SMILES N1(C(Cc2cc(C)cc(F)c2)=O)CCC(C)N(C(C2CC3C(C2)C3(F)F)=O)CC1 c1(C(=O)NC2C(CNC(C3N(C)CCC3)=O)CCC2)ccc2c(c1)CCC2 c1(OC)ccnc(C(=O)NCC2CC(C)N(C(=O)Cn3cc(CO)nn3)C2)c1C C1(OC)CN(C(=O)CN2CCC(C)CC2)CC1NC(C1CCCN(C(C)C)C1)=O Cc1nn(C)nc1C(=O)NC1COCC1CNC(=O)CC(C)c1ccccc1 C1(O)(C(C(=O)NC(C)Cc2cn[nH]c2)NC(CCCOC(C)C)=O)CCCCC1 C(=O)(N=c1[nH]c(Cl)ncc1C)c1c(C(=O)Nc2ccc(CC)cn2)scc1 C(=O)(CCCCCSC)N1CC(N(C(=O)C=C(C)C(C)(C)C)CC)C(O)C1 C(=O)(C(C(C)O)NC(c1cnn(CCNC(c2ccncn2)=O)c1)=O)OC c1(C(N2CCC(CO)CC2)C(=O)NCCSC2CCCCC2O)ccc(O)nn1 c1(C(C)C)cc(C(=O)NC2CCCC(NC(=O)CN(CC(C)(C)C)C)C2)nn1C Cc1cc(C(=O)NCC2CC2CC(=O)NCC2CCCC2C)ncc1F Cn1cnnc1CCCNC(=O)C#CCNC(c1nccn1C)=O N1(C(CS(=O)(=O)NC)=O)CC(C(=O)NC2(CO)CCC(C)C2)CC(C)C1 c1(C(N2CCCCC(Nc3c(C#N)c(Cl)ncn3)C2)=O)cc2cccc(F)c2o1 Cc1cc(-c2cncc(C(=O)Nc3nc(C4CC4)c(Br)s3)n2)cc(C)c1 C1(C)(C(=O)NCC2N(C(c3cc(C)sn3)=O)CC2)CC(C)OC(C)C1 CCC(CN=c1[nH]c(=NCC2=CCCC2)[nH]c2ccc(Cl)cc12)n1cccn1 c1(OC)cc(Cl)ccc1CNC(C1(C)CCCN1Cc1cccnc1OC)=O C1(O)(C(=O)NC2CN(C(c3c(OC)c(C)cs3)=O)CC2O)CCC(C)(C)CC1 c1(CC(=O)NC2CCN(C(C3C(CC)CCC3)=O)C(C)C2)nnc2n1CCOC2 N1(C(CCC=C=C)=O)CCn2ncc(CNC(c3nnc(O)nc3O)=O)c2C1 C(=O)(CC(O)C(C)C)N1CCC(C(C(=O)NCCc2ccn(CC)n2)C)C1 c1(CC)ncc(C(=O)NC(C)(C)CNC(C2CC2CF)=O)s1 c1(C(=O)NC23CN(C(c4c(CC)c(C)ccc4)=O)C(C2)C3)cc2ccccn2n1 C1(NC(Cc2c(C)nn(CC)c2C)=O)CN(C(c2ccncc2)=O)CC12CCC2 c1(CC)cncc(C(=O)N(C2(CCCCO)CC2)C)c1.C12COCC1C(=O)N2 c1(C(=O)NCCCC2CCN(C(C(OC)OC)=O)CC2)cn2ncccc2n1 Cc1csc2c(N3CC(CC(C)NC(=O)Cc4ccco4)C3)ncnc12 N1(C(CCC)=O)CCC(NC(c2nccnc2Cl)=O)C(F)C1 N1(C(C(CC)SC)=O)CCC2(CCCC2N2CCC3(CC2)CC(C)=NO3)CC1 O=C(CCCC1CCC1)NCC1CCC1NC(=O)C(C1CCCCC1)O CC1(C)CC(NC2CCC2)CN(Cc2cc(N)n(-c3ccccc3)n2)C1 N1(C(C2=C(C)OCCC2)=O)CC2CCCCC2(NC(=O)C=C(Cl)Cl)C1 c1(OC)ncc(F)c(N2CC(CNC(c3ccc(F)c(C)c3)=O)(OC)C2)n1 C1(C(N2CCCC(CC(=O)NCC(c3ncon3)C)C2)=O)CCCC1C1CC1 N1(C(C2(CC)CC2(F)F)=O)CCCN(C(=O)C(C)(F)CC)CC1 CCC(C)(COC)C(=O)NCC1CCC1NC(c1cc2n(n1)CCC2)=O c1(NC(CCN(C(=O)C(F)CC2CCC2)C)=O)cnc2ccnn2c1 C1(C(N(C2CCC2O)C)=O)CCCN(C(c2cnnc(O)c2)=O)C1 CS(=O)(=O)c1cncc(C(=O)NC2CCCN(C(C34COCC3C4)=O)C2)c1 N1(C(COC(CC)C)=O)CCC2CCN(C(c3c(O)cc(F)cc3F)=O)CC2C1 N1(CC)CCC(N(C(c2ccc(COC)s2)=O)CC)C1 c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC1CN(C(=O)CC(C)C2CC2)C1 C1(CNC(C2C=C(C)CS2)=O)CN(C(c2cc(C)nn2C)=O)CCC12CCC2 C1(C(N2CC3C(CNC(c4cc(C)sc4)=O)(C3)C2)=O)CC2(C1)CC(C)C2 c1(CNCc2cn(-c3c(C)ccnc3)nn2)ccc2nnnn2c1 N1(C(C(=O)NC(C)C)=O)CCC(NC(c2scnc2C(C)(C)C)=O)C(F)C1 Nc1cc(C(=O)NCC2(NC(=O)CC3(O)CCC3)CC2)cc(F)c1 C1(CC(=O)NCC2(O)CN(C(c3cc(N4CCC4)ccn3)=O)C2)CC(=O)NC1=O N1(C(CNS(NC)(=O)=O)=O)CC(CNC(=O)Cc2nonc2C)N2CCC1C2 c1(OC)ccc(Cl)c(C(N2CC(NCc3nc(C(N)=O)co3)C3(CC3)C2)=O)n1 c1(OC(F)F)cc(C)cc(F)c1NC(c1ccnc(OC)c1)=O.CO CC1(C)C(NC2CCC23CCCC3)CC1O N1(C(C2(CCC)CC(=O)C2)=O)CC2(CC(CC(=O)NCC(C)C3CC3)C2)C1 C(C(CC(=O)NCC1C2CCCC12)NC(=O)CN1CC(=O)NC1=O)OC CC1=NOC(C(N2CCCC2CN(C(=O)C=CCN2CC3CC3C2)C)=O)C1 C1(C(=O)NCCCNC(CP(C)(C)=O)=O)CC1C1(C)COC1 N1(CC(=O)NC(C(C)C)CNC(C2CC(C)(F)C2)=O)CCNC(=O)C1 S(=O)(=O)(c1cnc2ccoc2c1)N1CC(C)N(S(C)(=O)=O)CC1 C1(C(=O)Nc2c(C(=O)OC)[nH]nn2)CCN(C(=O)OC(C)(C)C)CC1(C)C N1(C(CC)=O)CCCC(C(N2CCC3C(NC(c4ncn(CC)n4)=O)C23)=O)C1 c1(C(=O)NCC(CC)NC(C2CC(C(F)F)C2)=O)cnn(-c2ccncc2)c1C CC1CC(NC(C2(C)CCN(C)C2=O)=O)CCN1C(=O)Cc1cc(Cl)cc(Cl)c1 C(=O)(C(CCCCN)CC(F)(F)F)CC=CCNC(c1cn(C2CC(N)C2)nc1)=O C(C(N=c1[nH]c(=N)[nH]c(=NCc2cccc(C(N)=O)c2)[nH]1)C(C)C)OCC N1(C(c2nn(CC)nc2C)=O)CCCC2(CCN(C(=O)CCNC(C)=O)C2)C1 C1(NC(C(C)(N(C(c2nc(OCC)oc2)=O)C)C2CC2)=O)CC2COCC2C1 c1(C(=O)NCC2CCCN(C(C(C)SCC)=O)C2)c(OC)cc(Cl)cc1F C(CCN=C(NCc1ccc(SC)o1)N1CCC(C(F)(F)F)(SC)C1)OC Cc1ccc(N2CCCC2C(=O)NCC(N2CC(N3CCNCC3)C2)=O)cc1 N1(C(=O)OC(C)(C)C)CC2CC(C1)C(CO)C2Nc1[nH]c2cnccc2c1Cl C(=O)(C(C#N)C(C)(C)C)NC(C)(C)CCNC(=O)Cc1cncc(O)c1 N1(C(C(=O)NC(C)C)=O)CC(C)(C)OCC1CNC(C1(C#N)CC1)=O C(C1=CCN(C(C2CC(C3CC3)=NO2)=O)CC1)NC(c1ccc(=O)oc1)=O c1(C(=O)NCCC(=C)CNC(C2(C)CNC(=O)C2)=O)ccncc1Br CC1CCN(C(c2csc(CNC(C3(N4CCCC4)CC3)=O)c2)=O)CCO1 C1(C2CCN(C(=O)C(C)(C)C(C)O)CC2)(NC(C(CCC)N(C)C)=O)CC1 N1(C(CC(n2c(CC)ncc2)C)=O)CC2CCN(C(=O)CCN(C)C(C)=O)CC12 C1(NC(C=CC)=O)CCSC12CN(C(C1CCCN(c3nccs3)C1)=O)C2 N1(Cc2c(C)nn(C)c2C)CCN(C(c2ccc(C#N)cc2)=O)C2(CC2)C1 N#CC1CN(Cc2cnn(C3CC3(F)F)c2)CC1NC(=O)C(N)=O C1(NC(c2c(Cl)cn(CC)n2)=O)CC(CNC(C2SCCS2)=O)C12CCC2 C#Cc1cc(C(N2CCC(CCNC(=O)C(C)CCC)C2)=O)cc(N)c1 C(=O)(CC(C)(C)C(=O)NCC1(NC(=O)CS(N)(=O)=O)CCOCC1)OCC c1(OCC)cc(C(=O)NC2CCCN(C(=O)COC3CC3)C2)cc([N+](=O)[O-])c1O C1(CC=C)(NC(c2ncccc2CC)=O)CCCN(C(C2CCOC2=O)=O)C1 C1(C(N2CC(O)(CNC(CC3C(C)CCO3)=O)C2)=O)CC(=O)NC(=O)C1 C1(NC(C2C(C(C)NC(C(CC)CN(C)C)=O)C2)=O)CC2(CCCCO2)C1 CCC(C)CCCC(=O)NC(C1CCCN1C(c1cccc(C#N)c1C)=O)C Cc1ccc2c(CCNC(N3CCC(O)(Cc4ccccc4)C3)=O)cn(C)c2c1 C=Cc1cc(C(=O)NC(C)C(C)NC(c2cc(CSCC)on2)=O)cc(F)c1 CC1CCCC(C)N(C(c2conc2CNC(=O)C(C)n2cccc2)=O)C1 C1(C(=O)NCC(=C2CN(C(CC3(CSC)CC3)=O)C2)F)CCCCN1C(C)C c1(C(N2C(CNC(c3c(C)csc3)=O)C(C)(C)CC2)=O)cccc2c1C(=O)CC2 c1(C(=O)NC(CC2CN(CC(c3ccc(CC)o3)=O)C2)C)cc(O)nc(O)n1 CC(O)C(=O)N=c1ccn(CC(N2CC(F)C(F)C2)=O)c(O)n1 C1(NC(C2N(C(C=NOC)=O)CCOCC2)=O)CCOCC12CCC2 N1(C(C(C(C)CC)N(C(CC=CC)=O)C)=O)C2CCC1CC1(CC1)C2 c1(NC(c2c(Cl)cnn2C)c2n(CC=C)nnn2)sc(Br)c2c1OCCO2 C1(CC(=O)NC(CNC(C2(SCC)CC2)=O)C(C)C)CCCCCO1 C1(NC(CCc2nc(C)sc2)=O)C2COCC1CN(C(c1cnncc1C)=O)C2 C=CC1CN(C(C2C3CC4C(C3)C24)=O)CC1NC(=O)C(C)CC(N)=O CC1(C(=O)NCc2ccnc(Oc3ccc(F)cc3)c2)CC=CCO1.C1CN1 CC(C)=C=CC(=O)NCCCN(C(=O)CC(C)C)C1CC1 C1(C(=O)OC)CCC(NC(C2CC(n3cc(CNC)nn3)C2)=O)CC1 CCC(CC)(CO)C(=O)NCCC1CN(C(c2cc(Br)n(C)c2)=O)C1 CC(C)(C)C1=NOC(C(N2CC=CC(NC(c3ccnc(Cl)c3F)=O)C2)=O)C1 C1(NC(c2cc(C3(C)CC3)n[nH]2)=O)CC(NC(=O)C(=O)C(C)(C)C)C12CCC2 N1(C(Cc2cc(C)sc2C)=O)CCN(C(=O)CNC(c2ccco2)=O)C2CCC12 C(=O)(C(C)CCCCCC)N1CC(C(N2CC(C#C)(F)C2)=O)C(C)(C)C1 c1(CNC(c2n(CCOC)nnn2)CCCSC)ccnc(Cl)c1Cl C1(C(N(C(CCCC)C)C)=O)CN(C(=O)Cc2c(C)cnn2C)CCN1C c1(OC)c(Cl)cc(C(=O)NC23CCCC2CN(C(c2cnccn2)=O)C3)nc1Cl Cn1cnc(C(N2CC(O)(C(F)C(=O)NCC3CCCS3)C2)=O)c1 CCCC(CCCNC(c1cc(C(C)(F)F)ccn1)=O)NC(C1(N(C)C)CC1)=O N1(C(C)=O)CCCC1(C)C(=O)NCC1(O)CCN(C(=O)CCCC2CC2)C1 C#Cc1c[nH]nc1C(=O)NCC1CC(F)CN1C(c1ccoc1Cl)=O c1(C(=O)NC(CC=C)CNC(C2CC(C(C)C)C2)=O)ccc(C2CC2)cc1C c1(CC)ccc(C(=O)NC2CCC(C)N(C(c3cc[nH]n3)=O)C2)cc1CC N1(C(c2nc(C(=O)OC)oc2)=O)C2CCC1CC(NC(C1(C#N)CC1)=O)C2 c1(NC(C2(C)CCC3(CC2)CC3)=O)nc2c(F)cc(Cl)cc2s1 C(CC(CC)C(=O)NCC(O)CC(=O)NC(C)C(C)C(=O)OC)=CC C(=O)(CCCC(C)(C)C(=O)N1CC2(CNC(=O)C(C)SC)CCC1C2)OC n1(CCOC)cc(C(=O)NC23CC(C2)N(C(=O)CCc2nc(O)n[nH]2)C3)c(C)n1 c1(C(=O)N(c2cnc(C3CCNC3)s2)C(c2ccco2)=O)ncc(Cl)cn1 C1(N(C(c2cc(CCO)on2)=O)CC)CCCN(C(=O)Cn2ncc(Cl)c2C)C1 c1(C(=O)NCC2C(C)CCN(C(=O)C(C)(C)CO)C2)ccc(S(N)(=O)=O)nc1 C(=O)(C(C(C)(C)C)NC(N)=O)NCC1(NC(C=Cc2cnc(C)s2)=O)CC1 CCCC(CCCNC(C1CCC(O)CC1)=O)NC(=O)CCF CC1(C)CCN(C(c2csc(Cl)n2)=O)C1C(=O)NC1C(=O)OCC1CO CCC(CC)C(c1nnnn1Cc1ccco1)NC1CC1CC(C)C CC1CCC(NC(=O)CC2(O)CCCOC2)CN1C(=O)Cc1ccon1 CN1C(C(N)=O)CCC1C(N1CCOC(CNC(C2(C(C)(C)C)CCC2)=O)C1)=O C1(CNC(CC(C)(C)NC(=O)CCNC(=O)CO)=O)CC2(CCCO2)C1 c1(C(N2c3ccoc3C2=O)=O)cc(F)c(Cl)c(Cl)c1.N1(CCO)CCN(C2COC2)CC1 C1(CC(=O)NC2CC(C#N)C2)CCC(C(=O)O)CC1 c1(C(N2CCC(NC(CC3C(C)(C)OCC3)=O)(CF)C2)=O)cncc2ccccc12 CC1CN(C(c2c[nH]c(=S)cn2)=O)CCN1C(c1cocn1)=O c1(CN2CC(OC)C(NC(c3cc(C)cc(C)n3)=O)CC2)ccc(S(N)(=O)=O)o1 c1(CC)nc(C)oc1C(=O)NCCOCC(=O)NCC(O)CO C1(C(=O)NCC(CCNC(C=CCCC)=O)OC)CCc2c[nH]nc2C1 c1(CCC)ccc(CC(C)C)cc1.C12CCN(C1)CC(O)COC2 c1(OC(CC)C)ccc(CN2CC3C(CNC(c4cscc4C)=O)C3C2)cc1 c1(C(=O)NC2C(NC(=O)CSC3CCCO3)C2)cc(C(F)(F)F)ccc1F C12(C(N3CC(CNC(CC4(C)CC4(F)Cl)=O)C3)=O)CC3CC(C1)CC(F)(C3)C2 C(CCCC(=O)NC(C1CC1)C1CC1)NC(CC(C)C)=O N1(Cc2ccc(C(=O)OC)cc2)CC2CN(C(c3cc(O)ccc3Br)=O)CC12 C(C(=O)NC1CN(C(c2ccncc2O)=O)CC1C)(C(C)C)NC(C)=O c1(OCC)cc(F)ccc1C(=O)N(C)CCn1cc(-c2cncs2)nn1 c1(C(N2CC3OCC(NC(CC4C(C)(C)C4)=O)C3C2)=O)cncc2ccccc12 C(CC(N)=O)(C(=O)N1CCC(C)(C)CC1)NC(c1c(OC)scc1)=O C1(N(C2CCOCC2)C(C(N)=O)=O)C2CC(n3cc(-c4ccncc4)nn3)C1C2 c1(OC)ncc(C(=O)OCC(n2cc(-c3cncc(N)c3)nn2)C)cc1C C(=O)(CS(=O)(=O)C(C)C)NC(CNC(CC(=O)NCC)=O)CC Cc1ccc(Br)cc1CC(=O)NCC1CCCN1Cc1ccc(Br)cc1Br N1(C(C2(F)CCN(C(C3(CCN(C)C)CC3)=O)C2)=O)CC(C#N)C2(CCC2)C1 C(=O)(C#CC1(C)COC1)N1CCC(N2CCN(C(C3C(C)OC(=O)N3)=O)CC2)C1 C1(CNC(C(F)=CCC)=O)CC2(CCC2)CN1C(c1ncc(C#N)cc1C)=O c1(C(N2C(CNC(C(C3CC3)OC)=O)CC(O)C2)=O)[nH]c2ccc(C)cc2c1C N1(C(C2C(=C)C2)=O)CCCC(C)(C(=O)C2=CCCC2)C1 C(=O)(C#CC1CC(F)(F)C1)NC(CNC(CC(CCCC)C)=O)(C)C C1(CCC)(NC(=O)CCc2cc(C)[nH]n2)CCCN(C(=O)CS(=O)(=O)CC)C1 c1(C(=O)Nc2c(SCCC(=O)OC)cccc2)cc(F)c(O)c(Cl)c1 C1(C(=O)NCC(CC=C)(C)C)CC(C)(C)CN1C(c1ccnc(O)c1F)=O c1(CNC(CN(CC)CC)C(=O)OC)ccc(C(O)C(F)(F)F)cc1 C1(NC(C2CCCC2)=O)COC2(CCCN(C(=O)COc3cncc(Cl)n3)C2)C1 CCCC(C)CC(C)Nc1cccc(-c2c(C(CN3CCCCC3)NC)c[nH]n2)c1 c1(CC(N2CCC(C)C(NC(c3cc(Cl)ccn3)=O)C2)=O)cccc2ccoc12 CCCCC(CNC(c1ccc(SC)cc1)=O)NC(c1n[nH]cc1C1CCC1)=O C1(CC(=O)NCC(C)(O)C2CC2)C2CN(C(c3csc(Cl)c3)=O)CC12 CC(C)CC(O)C(C)C(=O)N1CCC(N=[N+]=[N-])(C(=O)NC2CC(N3CCCC3)C2)C1 N1(C(C)C)CCCC1C(=O)NC1CCC1CNC(=O)Cn1cnnc1 c1(C(N2CCOCC(NC(C(CC)(C)C)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 c1(OCCC(=O)N(C(CNC(CN(CC)CC)=O)C)C)ccccc1F N=c1[nH]cnc2c(C(N3CCCC(NC(=O)C=CC4CC4)CCC3)=O)cnn12 c1(OC)cc(Br)ccc1CCC(=O)NC1CN(C(=O)CNC(C)=O)CC1C Cc1c(C(=O)NC(C)(CO)C(=O)NC2CCN(CCF)C2)ccn1C c1(N2CCC(CCNC(=O)CCN3CCCS3(=O)=O)CC2)ncc2ccnc-2[nH]1 N1(C(C2C(C)OC(=O)N2)=O)CCC(F)(C(=O)NCC2CCSC2)CC1 C(=O)(CCN=C(NCCc1cnn(C)c1)NCC1CCCC1OC)NC C#Cc1ccc(NC(C2CCC(CNC(c3coc(SC)c3)=O)O2)=O)cc1 c1(C(CC(=O)NCCn2ccc(C)n2)NC(=O)C(C)C#N)ccccc1Br CC(C)(CC(=O)NCC1CCC1NC(c1cc(F)ccc1F)=O)CC(F)(F)F C(CC(C)C)(C(=O)N1CCC(OC)CC1)ONC(c1c(CC)n[nH]c1)=O N1(C(c2c(C)ncs2)=O)CC(NC(=O)C(C)CC(C)(C)C)CC(C)(C)C1 CC(C)(C#CC(=O)OC(C)(C)C)CNC(=O)Nc1nc(-c2ccccc2)ns1 CC1CN(C(=O)CC2(CS(C)(=O)=O)CC2)CCC1NC(=O)CN1CCNC(=O)C1 c1(OC)c(C(=O)NC2(C)CN(C(c3cc(N)ccc3O)=O)C2)ccc2c1CCC2 N1(C(c2n(CCC)ncc2)=O)CCCC(NC(c2cncc(C(C)(C)C)c2)=O)C1 C1(CC(N2CC(C)(NC(c3c(C)cc(F)nc3)=O)C2)=O)CC(C)CC(C)(C)C1 C12(CNC(C3N(CC)CCCC3)=O)CCC(CC1)CN2C(=O)C(C#N)C(C)C CC1(C)CCC(NC2CC3C(C(=O)NC(=O)CCc4ccc[nH]4)C3C2)C1 C#CCCN=C(NCC(C(C)CC)OC)N1CCc2cc(Br)ccc2C1 C1(C(C)C)CC(C(N2CC3CC2C3NC(=O)Cn2cccnc2=O)=O)CCO1 C1(CNC(C2C(CC)CCC2)=O)CC(O)CN1C(=O)CCCc1ccsc1 C1(CC(C)NCCc2ccc(OC(F)(F)F)s2)CC(C)(C)NC1=O CC(C)(CNC(C1(C)CC2CCC1O2)=O)CC(=O)NCCc1ccnc(O)c1 C12(NC(C(CCCC)C)=O)CC(C)(C1)OC21CN(C(=O)CC(C)C)C1 CC1=C(CNC2CC(NC(=O)OC(C)(C)C)C(O)C2n2cccn2)C(C)(C)CCC1 C1(NC(c2ccncc2O)=O)CCCCN(C(c2cc(Br)cnc2Br)=O)C1 C1(N(C(=O)CCC2CCCOC2)CC)CCCN(C(C2CN(CC(C)C)C2)=O)C1 N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CCN(C(=O)Cc2occc2C)C(CO)C1 CC1(C)COC(C(=O)NCC(C2CCC2)NC(=O)CCN2CCOC2=O)C1 N1(C(c2c(CSC)n(C)nc2)=O)CCN(C(=O)C(=O)NC2CC2)C2CC12 c1(C(=O)NC(C2CCCCC2C)C)cc2c(cc1F)NCCC2 S(=O)(=O)(c1ccc(N2CC3CC2C3)cc1Br)N(C1C(C)C1)CCO N1(C(=O)NC2CC(n3cc(C4CC45CC5)nn3)C2)CC2C(C1)C2(F)F C1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)O)CNC(=O)C(C)(C)C1 C(=O)(C(C(C)CC)N(C(=O)Cc1cc(CC)no1)C)NCC(C#C)CC CCC(C#N)C(=O)NCC1CCCN1C(=O)CCCSC(C)(C)C N1(C(C(c2ccccc2)NC(Cn2ncc(C#N)c2)=O)=O)CC2COCC(C2)C1 C1(Cn2cc(CCCCCCC)nn2)CC(C)(C)CCN1C(=O)CC(F)(F)CC N1(C(=O)C(F)(F)CN2CCCC2)CCN(C(=O)CCc2cncnc2)C(CO)C1 CCC(C)CC(C(=O)NC1CCCCCC1)NC(=O)CC1(N(C)C)CCC1 C1(NC(C2(CSC)CC2)=O)CCOCC1C(=O)NCc1ncnn1C N1(C(c2c(C(N)=O)ccs2)=O)CCCC2(CCCN2C(c2ccncn2)=O)C1 N1(C(c2cnc(CC)o2)=O)CCC2CN(C(c3ccccc3)=O)CCC12 c1(C(=O)NC2CN(C(C=CCCC)=O)CC(O)C2)cc(F)c(F)cc1OC C1(C(=O)NCC(C)(CO)NC(c2cnn(C)c2C#N)=O)(OC)CCCC(C)(C)C1 C(=O)(C1CCc2c[nH]nc21)N1CC2C(CN3C(C)CCCC(C)C3)(CCC2)C1 c1(OCC)ccccc1NC(=O)CN(CC1CC1)CC(C1CC2C=CC1C2)=O CC1CN(C(c2nscc2I)=O)CCCN1C(=O)CCC1CC1 n12cnc(c1)C(=O)NCC2.C(C)(CCCO)NC(CCC)=O c1(C(N2CC(C(C(=O)NCc3ccco3)OC)C2)=O)cncc(F)c1C C(=O)(C1CCc2nnc(C)n21)NC(CC)CNC(c1csc(C(C)C)n1)=O C(C(O)C(C)(C)C)N(C)C(C1(C)CC=CCC1)=O.C1=CCNC1=O c1(C(CNC(C)=O)NC(CC(=C)I)=O)ccccc1F CC1CN(C(=O)CC2(O)CC2)CCN1C(c1ccc(-n2cccc2)cc1)=O C12(C(=O)NCC(C)N(C(=O)CC3OCCO3)CC)CC3CC(C1)CC(F)(C3)C2 C(C(C)(C(=O)NCC(C)(Cn1cccn1)NC(C1CCCN(C)C1)=O)OC)OC c1(OC)ccccc1-n1ncc(C(=O)N(c2cccc(F)c2)C)c1C C(CC(C(=O)N(C)CCc1ccccc1)NC(=O)C(CC)OC)OCC C1(CN(C(C2C(C(=O)OC)C2)=O)C)COCCN1C(c1ccoc1C(C)C)=O C1(F)(C(N(CC(C)O)C2CC2)=O)CCN(C(=O)CC2(N(C)C)CC2)CC1 Cc1cc(F)cnc1C(=O)NCC1CC(CNC(c2ccccc2CO)=O)CO1 CC12CN(C(c3cccc(-c4ccccc4)n3)=O)CC1(C)CS(=N)(=O)C2 C1(c2cccc(Cl)c2)CCN(CCC(=O)N(C2COC2)NC(=O)OC(C)(C)C)CC1 C=CC(CCC)CC(=O)N1CCC2(C(=O)NCCC3C=CCC3)CCCC12 N1(C(C(C2CC2)OC)=O)CC2(NC(=O)Cc3csc(Br)c3)CCC1CC2 C1(CNC(C#CC(C)C)=O)CC2CCC(C1)N2C(=O)CCC(=O)c1ccc[nH]1 N1(C(C(CC=C)CC)=O)CCC2(CC1)CC2C(=O)NCC1C=CCOC1 C1(CCOC)(NC(=O)C=Cc2ccoc2)CCN(C(=O)Cc2nnc(C)o2)C1 C1(CC(=O)NCC2CCC(C)CN2C(C2(F)CCCC2)=O)CCCC2(CCC2)O1 c1(C(N2CC(C)(C)C(NC(c3ccc(O)cc3)=O)C2)=O)ccc(P(C)(C)=O)cn1 S(=O)(=O)(c1cnc2sccc2c1)NCC1CC(c2cccc(C)c2)C1 C12(CNC(c3c(CC)n[nH]c3)=O)CCC(CC1)N(C(C1(C)CCC13CCC3)=O)C2 c1(CC(=O)N(C2CN(C)C2)C)ncccc1NC(=O)OC(C)(C)C C(C(=O)NCC(C)(O)CNC(c1ncnn1CC)=O)(C(C)C)OCC CC(C)CC(C(=O)NCC1C=CCOC1)NC(c1cnc(S)nc1)=O C1(N(C(C23CC(C2)C3)=O)CC)CCCN(C(=O)CC(=O)N(C)C)C1 CC1CCn2cc(C(=O)NC3CCN(C(C4(C#N)CCOC4)=O)CC3F)nc2C1 CN1C(=O)CCC1(C)CNC(C1(CO)CCN(C(C2CCCC2C2CC2)=O)C1)=O c1(CCNC(N(C2CCCN(c3ccccn3)C2)C)=O)cccc(C(F)(F)F)c1 C(=O)(CCCS(C)(=O)=O)NCCC(C)CCNC(=O)CN(c1ccnc(Cl)n1)C CCC(CC)CCCC(=O)NCC1(C)CCCN1C(=O)Cc1c[nH]ccc1=O c1(CC)nc[nH]c1C(=O)NCC(C)(C1CC1)NC(=O)CCc1ccc(C)s1 C1(O)(NC(C(CN(CC(=O)NC)CC)O)=O)CCOCC1 C12(CNC(CC(CC)OC)=O)CCN(CC1)CC2.C1(CO)C(=O)N1 C=CCC(C(=O)N1CCCCC1CCCO)NC(=O)C(C)SCCCC C(=O)(C1(C)CCc2ccccc21)NCC(CC)NC(C1(F)CCC1)=O N(C1CCCOc2ccc(Br)cc21)C(=O)NC1CN(C)CC1c1ccccc1 C1(C(C(=O)NC2C3CCN(C(c4ccnnc4)=O)C23)O)CCS(=O)(=O)CC1 C1(NC(CCC(N)=O)=O)CC2CC(C1)N(C(=O)CCC(=O)OC(C)(C)C)C2 C1(C(=O)NC(C(=O)NC(C(CCC)O)CO)CCOCCO)CCC2(CCC2)O1 C1(CC(=O)NCC(CC)NC(c2cc(O)ccc2N)=O)CCCC(C)(C)O1 c1(C(C)C)ccc(C(N2CC(O)(CNC(c3ccc(-c4ccco4)s3)=O)C2)=O)o1 CN1CCN(C(c2cccc(C(=O)NCc3cccs3)c2)=O)C(C(C)(C)C)C1 c1(C(=O)NCC2(C)C(C)CN(C(=O)C(C)(C)C(C)O)C2)c[nH]c2ccc(F)cc12 c1(OC)cc2c(cc1OC)CC(C(N1CCN(C(C)=O)CC1)=O)C2 c1(CC)ccc(CCC(=O)NCC23CC(NC(C4CC(=O)C4)=O)(C2)C3)cc1 N1(C(C(c2ccccc2)=O)=O)CCN(CCc2cccc(Cl)c2Cl)C2CC12 C1(C(=O)NCC(CC(C)C)NC(c2cc(O)cnc2Cl)=O)(OC)CCC(C)CC1 C(CN=C(NCc1cn(C)c(=O)n1C)NCC(C)CCC)COCC c1(OCC)cc2ccccc2cc1C(=O)NC1CC2(CCC2)CN1C(C)=O c1(C(=O)NCC2CC(C)C2)ccc(S(=O)(=O)N2CCC(C(F)(F)F)C2C)c(Cl)c1 C(=O)(CCCCCn1cnnn1)NC1(CNC(C2C(C)C2)=O)CCOCC1 c1(OC)ccc(C(N2CCCC(CO)(NC(C3CC3F)=O)C2)=O)cc1S(C)(=O)=O N1(C(C(C)CC2CC2)=O)CCN(C)CC1CNC(C1CCOC1C(N)=O)=O N1(CC(=O)NC2C(C)CCCC2)CCCC(C)(NC(=O)CNC(=O)C(C)(C)C)C1 CCCCC(CC(=O)O)N(C(C1CCCN1Cc1ccccc1)=O)C(C)C C1(C(=O)NC2(CNC(c3nc(OCC)oc3)=O)CC2)OC2CCC1C2 C(=O)(C1CC(=O)OCC1)OC.O(N(C)C(=O)CCC)C(=O)OC(C)(C)C c1(C(N2C(CNC(C(CC)(C)OC)=O)C=CC2)=O)cccc(S(=O)(=O)C2CC2)c1 c1(CC(N2CC(C)OC(CC3CCC3)C2)=O)cccc2occc12 C12(C(=O)OC)CC(C(=O)NC3(CN(C(=O)C(C)n4cccc4)C)CC3)(C1)C2 C1(CN(CC(C)NC(=O)CCn2cccn2)C)CCC1C(F)(F)F C(C(F)(C(=O)N1CC2CCC2(C)C1)C(C)C)NC(c1c(C)cc(CC)o1)=O C(C(CC(=O)NC(C)(CO)C1CCCC1)C1CCC1)NC(C(CC)OCC)=O N1(Cc2nc(C)on2)CCN(C2CCSC2)CC1.N1(C)C(=O)N1 C(C(C(C)(C)C)NC(c1cccnc1C(F)F)=O)NC(CC(C)OC)=O C1(C(C(=O)N(CC)Cc2ccco2)C)CCCN(C(=O)CCC(C)C)C1 C1(CNC(C(CC=C)CC)=O)CC2CCC1N(C(=O)CC(O)C(C)CC)C2 C1(NC(c2c(CC)cco2)=O)C2CCC1N(C(=O)Cc1cnc[nH]1)C2 C1(OCC(=O)NC(C)(C)CCNC(=O)Cc2nc[nH]n2)CCCCCC1 N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CNC(=O)CCC(C)C Cc1[nH]nc(C(N2CC3(NC(=O)CNC(N4CCCC4)=O)CC2C3)=O)c1C N1(C(C2(C)CCC2)=O)CCC(C2(NC(c3sc(Cl)cc3Br)=O)CC2)C1 C1(CC)CCN(C(=O)CC2COCC2NC(=O)CCc2nncs2)C1 O=S(Cc1ccccc1)CCNc1ccnn1Cc1ccccn1 c1(C(=O)NC(C(CO)NC(c2c(F)ccc(OC)c2)=O)C)cc2c(s1)CCCC2 C1(OC)CCCC1C(N1CC(NC(=O)Cc2ncc(C)s2)C1)=O c1(OC)n[nH]c(C(=O)NCCOCCNC(C2CCC(O)CC2)=O)c1Br C1(C(N(C)CC2(O)CN(C(=O)CC3=NNC(=O)C3)C2)=O)CCCc2ccccc2C1 C1(NC(C2CN(C)C(=O)N2)=O)CCC2CN(C(=O)COCC3CCCO3)CC2C1 c1(C(=O)NC(CNC(=O)C=Cc2ccccc2Cl)CO)c[nH]c2cccnc12 C1(C(=O)OCC)CCC(NC(=O)C(=O)NCc2nc(C)c(C)s2)CC1 N#Cc1c(NC(C2CC23CCOCC3)=O)ncnc1Cl C(=O)(CC(C)(O)CC(=O)O)N1CCCC(C(=O)NCc2ccnc(C)n2)CC1 C(=O)(C(C(C)(C)C)C1CCC1)N1CC(N(C(c2cnc(CC(C)C)s2)=O)C)C1 c1(C(=O)NCC2C(OCC)CN(C(c3cc(Cl)no3)=O)C2)c(Cl)ccc(C)c1O N1(C(C(C(CC)C)NC(C2CSC2)=O)=O)CCCC(N=[N+]=[N-])C1 N1(CCc2cn(C(C)(C)C)nc2)CC=CC2COCC12 c1(CC)cc(C(=O)NC(C)CNC(c2ncccc2SC)=O)sc1C c1(CNC(=O)OC(C2(CC3CC(=C)C3)CC2C(=O)O)=O)ccnn(CC)c1=O CCC(CCCC(=O)N1CC2C3CCC(C3)C12)NC(=O)Cc1ccn(CC)n1 c1(C(=O)OC)cccc(CNC(C)(C)CCCF)c1Br N1(C(C)C)CCCC(C(=O)NC2CNC(=O)C2)C1.C12CC(C1)CNC(=O)N2 N1(C(C2C(C)OC(=O)N2)=O)CC2CCCC2(CNC(=O)C(C)CC2CCC2)C1 C1(NC(C(C)C2CCC2)=O)CC2(CCN(C(=O)CCc3cocn3)C2)C1 c1(C(=O)NC2CC(C(=O)OCC)CC2O)cc(S(=O)(=O)CC#N)ccc1F CC(CC(F)(F)F)C(=O)NCCCOCCNC(=O)C(O)C1CCC1 N1(C(Cc2cn(C)nc2)=O)CCC2CCC(NC(C3CC34CCOC4)=O)C1C2 C(=O)(CCCC(F)(F)F)NCC(C)(Cn1cccn1)NC(c1occ(C)c1C)=O N1(C(C(CC(F)F)NC(COCC=C)=O)=O)CC2(COC(=O)C2)C1 Cc1cc(Cl)c(C(=O)NC2CC2NC(c2ccnc(CO)c2)=O)cc1N C(C(=O)N(C)CC1CCCC1)(C(C)O)NC(C(C)CO)=O CC(N=[N+]=[N-])C(=O)NC1CCCCC1C(N1CC(N2CC(O)C2)C1)=O n1(C2N(C(=O)OC(C)(C)C)CCC2)cc(CC=Cc2ccccc2)c(Br)n1 C(=O)(C1CCCn2nccc21)NCCCCNC(c1ccc(OC)c(F)c1N)=O C(=O)(CS(=O)(=O)CC(=O)NC1CCCCC1NC(c1cnc[nH]1)=O)OC C=CCC(CC(=O)NCC1(C)CCCCO1)NC(C1CCCCCN1C)=O C1(NC(Cn2ncn(C)c2=O)=O)CC2CC(C1)N(C(C1COC(=O)C1)=O)C2 O=C(CCCC1CC1)NC1(C(=O)NCCCc2ncco2)CC(CO)C1 N(C(=NCCCn1ccnn1)NCCc1ccccc1Br)CC(C)C C(=O)(C(C)n1cncn1)NCC(C1CC1)NC(C1(CC)CC1)=O CC1CN(C(=O)C(=O)NCCOc2cccnc2)CCC1C c1(NC(C2C(NCc3ccc(OC)c(O)c3)C2)=O)ccc(C(C)C)c([N+](=O)[O-])c1 N1(CCC)CCCC1C(N1CCCC1C(C)NC(=O)Cc1ccc(C)s1)=O N1(C(C)C)CC(C(=O)N(C)CCN(C(=O)CC2CC(O)C2(C)C)C)CC1=O c1(CC(c2cn(CCCC(=O)N(C)C)nn2)O)ccc(F)cc1.C12(CC1)C(=O)NC2 C1(CC(=O)NC(c2cccnc2)C)CCC(NC(c2cnc(C)cn2)=O)CC1 CCC(CC(C)C)C(=O)N1CCC(CCNC(c2ncncc2F)=O)C1 N1(C(c2cn(CCC)nc2C)=O)CCN(C(c2csc(C)c2OC)=O)C2CC12 C(=O)(C1=NN2CCCN=C2N1)N1C(CNC(C(C)SC)=O)CCC(C)(C)C1 c1(C(N2C(CN(C(C3(COC)CCC3)=O)C)COCC2)=O)ccc(C#N)c(Cl)c1 Cc1cc2cc(NC(C3CCN(C(c4ccncc4Br)=O)CC3O)=O)ccc2[nH]1 C(C(CO)(CO)NC(=O)Cc1nocc1C)N(C(C(COC)NC(C)=O)=O)C C(CCCCCCC(=O)N1CC(CNC(c2ncc[nH]c2=O)=O)C(C)(C)C1)SC N1(C(c2c(C)nn[nH]2)=O)CC2(CCCC2NC(C2CC(=O)N(CC3CC3)C2)=O)C1 C1(C(=O)NC(CNC(CCc2onc(CC)n2)=O)C2CC2)CCC(N(C)C)CC1 C1(CNC(C(CC)SC)=O)CN(C(C2(CCF)CCC2)=O)CCC1(C)C c1(CN(C(C2CC2NC(c2nocc2Br)=O)=O)CC)ccc(OC)cc1 n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CN(C(=O)COC(C)=O)CCN2C)n1 C(=O)(CC(O)CC(C)(C)C)NCC1C(C(N2C(C(N(C)C)=O)C=CC2)=O)CCO1 c1(C(N2CCN(CCCN(C(CCC)=O)C3CC3)CC2)=O)c(C)cc(Br)cc1F c1(C(N2CCC(NC(C(CCC)CC)=O)C(F)C2)=O)ccc(O)c2c1CCCC2 S(=O)(=O)(c1cccnc1CN(S(C)(=O)=O)C)NC(c1ccc(C)o1)C C1(NC(CN(C(C)=O)C)=O)CCCN(C(c2cc(C3(Cl)CC3)n(C)n2)=O)C1C C1(O)(CC)CCCN(C(c2ccc(CNC(=O)C(C)=C3CCC3)nc2)=O)C1 c1(C(N(CCCCNC(C2CC2F)=O)C)=O)c(O)nnc2c1CCCC2 C12(C(N3CC4C(C(N)=O)C(C4)C3)=O)C3C4C1C1C2C3C41Cc1cccs1 C1(C(=O)NC2CC(NC(CCc3cc(C)no3)=O)C2)CCC2C1C2(F)F C1(NC(C2C(CC)C2)=O)CC2CC1N(C(C1(F)CCC1)=O)C2 c1(-c2cn(CCC3CN(C(C4C(C)CC=CC4)=O)C3)nn2)ccc2ncsc2c1 N1(C(c2ccnc(OC)n2)C(=O)NC2CCC2)CC(C)CCC12CC2 c1(N2CCC(CNC(C3C(C)=C3)=O)C2)nc2c(cc1C#N)CCC2(C)C c1(CC(=O)NCc2nc(CNC(c3cnc(C)s3)=O)sc2)cccnc1Cl c1(OC)cccc(CC(N2CCCC(NC(=O)C(C)(C)C(N)=O)C2C)=O)c1Cl c1(CC(=O)NCC2(C)CCCN2C(=O)Cc2cc[nH]c2)ccc(F)c(Cl)c1 C(=O)(C(C)(CSC)NC(c1cnc(=N)[nH]c1)=O)NCCN(C)CC C(CCC(=O)NCC1CNC(=O)O1)(C(C)C)NC(C1C(C(=C)C)OCC1)=O c1(C(=O)NC2CC(O)(CNC(c3c(CC)nc[nH]3)=O)C2)oc(COC)cc1C c1(C(N(C(C)CCNC(=O)CCC(F)(F)F)C)=O)cc2c(cc1N)CCC2 C1(C(=O)NCC(C(C)C)NC(C2(C)CC=CC2)=O)CCOC(C(F)(F)F)C1 c1(OC)ccc(OC)c(C(O)CNC2(CO)CC2)c1 N1(C(CCCOCC=C)=O)CC(C)(C)OCC1CNC(=O)C(O)CCCC NCS(=O)(=O)Cc1cnn(CCc2nnnn2Cc2cc(Br)cs2)c1 C1(CNC(CCC)=O)CCN(C(=O)COCc2nc[nH]n2)C1(C)C c1(NC(=O)NC(Cc2c(C)noc2C)C)cccc([N+](=O)[O-])c1F c1(N2C(C(CC)N(C(=O)C=CC3CCCC3)CC)CCC2)ncnc2c1CCC2 CC1(C)CC(C(=O)NC2CC3(C2)CC3NC(c2ccc(C3CC3)o2)=O)CNC1=O Cc1[nH]c2c(CN3CCC(C(=O)OC(C)(C)C)CC3)cccc2c1C N1(C(c2ncc(F)cc2F)=O)CCC2C(C1)CN2C(c1ccn2nccc2c1)=O C1(NC(C(C)CN(C)C)=O)(CO)CCCN(C(=O)C(C)(C)C2CC2)C1 CN1CCCC(C(C2CC2)Nc2ncccc2F)C1.C1(C(C)(C)C)COc2nnnn21 C1(CC(=O)NC(=O)CN(C2CC2)CC2CC(N(C)C)C2)COCCO1 Cc1cccc2cc(C(C)(C)NC(=O)Cc3nc4cc(Cl)ccc4n3C)cnc12 N1(C(c2c(CC)c[nH]n2)=O)CCOC2CN(C(C3(C)CC=CCC3)=O)CC12 N1(C(C(n2c(C)ccn2)C)=O)CC(OC)CC1CNC(C12CSCC1C2)=O c1(C(=O)NC2CCN(C(CCOC(C)C)=O)CC2CO)cc(Cl)c(N)cc1F Cc1sc(N)c(C(=O)NC2CCCC(NC(C3(C)CC(C)(C)C3)=O)CC2)c1C C(C(=O)NCC(=O)OCC)(C(C)C)OCC.C1(C=O)CSCCN1C(=O)COC N1(C(CC2C(C)(C)C(O)C2)=O)CC2(C=C(C(=O)NOCCCF)CO2)C1 Cc1nc(NCC(c2ccsc2Cl)C)cc(N(C)Cc2ccco2)n1 C1(C(N(CC(CN(C)C)O)C)=O)CC=CCN1C(=O)C=C(C1CC1)C1CC1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(C(C)(C)NC(CC(C)(F)F)=O)C12CC2 Cc1cc(C)nc(-c2cccc(C(=O)NCC(c3cccc(C#N)c3)O)c2)n1 c1(OCC(=O)N(CC(N2CCC(OC)C2)=O)CCOC)ccccc1C C1(CC(N2CC(SCC(=O)NCC(C)NC(=O)OC(C)(C)C)C2)=O)CCCCC1 N1(C(c2ccc(CC)s2)=O)CCC(CNC(c2cc(N)nc(Cl)c2)=O)CC1C Cn1ncc(C(=O)NCC(C)(C)CNC(C2CC3C=CC2C3)=O)c1C#N CC1(C)C2CN(C(c3sccc3NC(c3ccsc3Br)=O)=O)CC12 c1(OC)cc(C(=O)NCC2C=CCN2C(C2CCCOC2)=O)ccc1C(F)F C(=O)(CCC(=O)C1CCc2ccccc21)NC1C(c2cc(F)c(F)c(F)c2)(C)C1 CCC(CC(=O)N1CC(C2(NC(=O)CCNC(c3cccs3)=O)CC2)C1)C(C)C c1(C(=O)NCC2N(C(c3c(SC)nn(C)c3)=O)CC2)nn(C)c(C)c1Br C(C(C)(C)CNC(C1(F)CCOC1)=O)N(C(=O)C(C)c1ncco1)CC C1(CNC(C(c2cnccn2)C)=O)CCN(C(C2CC2C2(C)COC2)=O)CC1(F)F Cc1cccc(C(F)C(=O)NC(CN(C)C(c2cncc(F)c2)=O)(CO)CO)c1 C12CC(C)CN(C1)C2=O.C(=O)(CS(=O)(=O)N1CCCCC1)NCC(C)C c1(C(N(C2CCS(=O)(=O)C2)CC)=O)ccccc1C(N)=O C=C1CCC(C(N2CCCC(CCNC(C3CC(O)CN3C)=O)C2)=O)CC1 C1(NC(C(=O)NC(C)C)=O)CCN(C(=O)CNc2ccccn2)CC1C(C)C c1(CC)conc1C(=O)NCc1cc(C(=O)N(CCO)CC2CC2)cs1 c1(C(=O)NCCCCCCNC(c2cncc(C)c2)=O)ccc(C)c2c1CCC2 C1(NC(C(C)=C(CC)C)=O)CCCC12CN(C(=O)C(c1c(F)cccc1F)C)C2 c1(C(=O)NC(CNC(C2COC3CC2C3)=O)C2CC2)cc(C2CC2)nc(O)c1 c1(C(N(CCN(C(C(COC)N(C)C)=O)C)C)=O)cnc2cc(C)nn2c1 c1(SCCC(=O)NCC2(C)CCCN2C(C2CCC(=O)N2)=O)ccc(C#N)cc1 c1(CCNC(Cc2c(NS(CC(C)C)(=O)=O)cccc2)=O)ccc(Cl)cc1Cl c1(C(=O)NCC2C3CN(c4nccc(C(C)C)n4)CC32)nccc2ccn(C)c12 c1(C(=O)NC2C(C)CN(C(=O)CCc3ccsc3Cl)CC2)ccnc2c1CCC2 N1(C(c2ncc(Cl)s2)C(=O)NCCSCc2ccncc2)CCC(CO)CC1 c1(C(=O)NC2(C)CN(C(C(C3CCCO3)OC)=O)C2)[nH]cnc1C#N c1(OC)n[nH]c(C(N2CCCC2c2ncon2)=O)c1Cl N1(C(C(C)CC2CC2)C(=O)NC(C)(C)C)CCc2cc(F)cc(Br)c2C1 c1(CNC(C2CC(F)(F)C2)(C#C)C)ccc(Br)c(Cl)c1 N1(C(N(C)CCO)=O)CC(CF)OCC12CNC(=O)OC2 c1(C(=O)NC(C)CNC(C2CN3CCCC3CO2)=O)ccc2c(O)ncnc2c1 CC(C)C(CC(=O)N(CC(C)C(F)(F)F)C)NC(c1cscn1)=O N1(C(C(CC=C)C2CC2)=O)CCC(=C(F)F)CC1.C12C(=C)C1C(=O)NC2=O Cc1cnc(NC(CO)CCO)c(S(=O)(=O)N2CCC(CS(C)(=O)=O)C2)c1 N1(C(C(COC)N)=O)CCOCC(n2cc(CC(=O)O)nn2)C1 N1(CCC(C)F)CCC(CC(=O)Nc2ccccc2CN2CCN(C)CC2)CC1 c1(C(=O)NCCNC(=O)CC2OCCCO2)cccc(=O)o1 C1(C)(C(C)O)CCCN1CCc1cccc(-c2nn[nH]n2)c1 c1(C(C(=O)NCC2(F)CN(C(c3cnc(O)o3)=O)C2)O)cccc(OC(F)F)c1 C(C(COC)C(=O)NC(CN(C)C)C(=O)N1CC(CC(C)C)C1)OC C#CC(CNC(=O)NCC(c1ccc(F)c(F)c1)(F)F)CC(C)(C)C n1(CC(=O)NC2(C(C)NC(=O)COC3CCCC3)CCC2)ncccc1=O c1(C(N2CCC(S(=O)(=O)N3CCCC3)C2)C(=O)NCC=C)c2c(nn1C)CCC2 c1(C(N2CCC(CCNC(CNS(NC)(=O)=O)=O)C2)=O)ccc(O)c(CO)c1 c1(C(N2CC(C)(NC(C(CCC)C)=O)C2)=O)cc2cc(N)ccc2[nH]1 C(CNC(C1C(C)CCN1C(=O)Cc1ccn(C)n1)=O)(CC(C)C)OC C1(C(N(C(c2ccccc2Cl)C(=O)O)C)=O)CCC2(CCOCC2)C1 C(=O)(N=c1ccc(C2CCOCC2)n[nH]1)N(C(c1ccncc1Cl)C)C1CC1 C1(C(=O)NCC(C)CNC(=O)CCOCC(F)F)CCN(C2CC2)C1=O c1(C(=O)OCC2(Br)CCCC2)ccc(OC(F)(F)Cl)cc1 N1(C(CNC(=O)NC)=O)CCN(C2CCCN(C(C3CCN3C)=O)C2)CC1 c1(SCCC(=O)NCC(C(C)C)NC(C2CN(C(N)=O)C2)=O)c(F)cccc1Cl C1(CC(=O)NCC=CCNC(=O)C(c2ccc(Cl)cn2)(F)F)CCC2(CC1)CC2 c1(NCC(=O)Cc2ccsc2)cccc(Cl)c1OC(F)(F)F C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(C1(C2CCCO2)CCC1)=O c1(NC)nc(C(N2C3CCC2CN(C(=O)CCF)C3)=O)ccc1[N+](=O)[O-] c1(OC)cc(C(N2CC(NC(=O)C=C(C)C(C)(C)C)C(O)C2)=O)c(O)c(Cl)c1 c1(CC(N2CC(NC(C(C(CC)C)O)=O)C2)=O)c(Br)sc2ccccc12 N1(C(c2nc(C)oc2C)=O)C2CCC1CC(N(C(=O)CCCCO)C)C2 C1(C(=O)NC(=O)C(Cl)(Cl)Cl)COCCC12CN(C(c1cc(F)cc(Cl)c1)=O)C2 c1(C(=O)OC)sc(N2CCNCC2)nc1CC1CCOC1 C1(C)(NC(CC2CC(C)(C)C2)=O)CCN(C(c2ccccc2N2CCCC2)=O)C1 N1(C(C2(CC=C)CCN(C(C3CCCN3CCC)=O)C2)=O)CCN(C)C2(CC2)C1 N1(C(C2C(C=C)CC2)=O)CC(F)(F)CC1CNC(=O)CCOc1ccc(C)cc1 N1(C(C(C(C)C)SC)=O)CCC2(C)CN(C(C3CCC(C(C)(C)C)O3)=O)CC12 c1(OC)ccc2oc(C(N3CCC4CCC34CNC(C3(C)CC3)=O)=O)cc2c1 CC1CN(C(=O)CNC(C2CCC(C)(O)CC2)=O)CC(=O)N1 Cc1cn2c(n1)C(C(=O)N(CCCCNC(=O)CC1(O)CCCOC1)C)CCC2 c1(N2CC3CC(NC(c4cc(CCC)[nH]n4)=O)C3C2)cc(C)c(C#N)cn1 N1(C(C(C)=CC)=O)CCN(C(C2CCC(=O)N(C(C)C)C2)=O)C(CC(F)F)C1 c1(C(=O)NCC2N(C(C(COCC)(C)C)=O)CCC2)cc2cccnc2[nH]1 c1(C(N2CC3C(NC(C(C)CN(C)C)=O)(C3)C2)=O)cnc2n(c1=O)CCS2 c1(C(=O)NCC(C)(O)CN2CCOCC2)nc2nc(O)c3ccccc3n2n1 c1(C(N2CC(c3onc(C)n3)C(N)C2)=O)nc2ccccc2nc1O N1(C(c2cn(C)nc2N)=O)CCN(C(=O)CCS(C)=O)C(CS(C)(=O)=O)C1 Cc1cc(C(N2CC(NC(C3CC4CCC(C3)O4)=O)C(C)C2)=O)n2nccc2n1 C1(NC(CNC(=O)COc2ccccc2[N+](=O)[O-])=O)CCS(=O)(=O)C12CCC2 CCCCS(=O)(=O)CC(=O)NC12CCCC(NC(c3ccns3)=O)(C1)C2 C1(F)(C(N(CCC(=O)NC(C)CCC2CCCO2)C)=O)CCCC1 Cc1nc(C)c(C(=O)N(C)CC2COCCN2C(=O)CN(c2ncccn2)C)[nH]1 c1(NCCCC(C)NC(c2ccnn2-c2ccncc2)=O)ncc(C#N)cc1F c1(CN=[N+]=[N-])ccc(CSc2ccnc(Cl)c2)cc1[N+](=O)[O-] CCC(O)C(C)(C)C(=O)NCC1C=CC(NC(=O)CC2CC(C)C2)C1 C12(NC(c3n(CC)ncn3)=O)CC3CC(C1)CC(N(CC(=O)NC)C)(C3)C2 C1(C(=O)NC(C2CSC2)C)CCN(C(C2CCCC(C#N)C2)=O)CC1(C)C C1(NC(CC)=O)CN(C(c2ccc(-c3sccc3C)s2)=O)C2(CCCOC2)C1 C1(Cn2c(C(C3(C)CCOC3)Nc3ccccc3)nnn2)CCS(=O)(=O)CC1 Cc1cc(NC(C2CCCN(C(c3nc[nH]n3)=O)C2)=O)n(C(C)C)n1 C1(C(=O)NCCCN(C(C2(C=C)CCC2)=O)C)CNC(=O)CC1C N1(C(c2cc(C)ns2)=O)CCCC2(CC(NC(c3cnn(C)c3Cl)=O)CO2)C1 CCC(F)(C(=O)OC)C(=O)N1CC2C(N(C)C(c3cc(F)cnc3O)=O)C2C1 Cc1cnc(C(=O)NCCCCCCNC(C2(C(C)(F)F)CC2)=O)c(O)c1 C(c1ccc(F)cc1)=C(C)C(=O)NCC1CC1NC(=O)C=Cc1ccsc1 c1(CC)oc(C)cc1C(=O)NC(CO)C(C)NC(=O)C(C1CCC1)OC Cc1nc(C(N2CCSCC2C(=O)NC2CCOCC2F)=O)c(C)s1 c1(C(=O)NCC(N2CCN(C(=O)Cc3cnns3)CC2)=O)ccc(O)nn1 c1(C(N2CCC(c3n(C)ncc3)C2)C(=O)NCC2CCOC2)ccc(Cl)cc1Cl C1(CNC(Cc2cn(CC)nc2)=O)CN(C(=O)CC2COCC2O)CC(C)(C)C1 C1(CO)CCCCN(C(C2CC2CNC(=O)Cc2csc(Br)c2)=O)C1 N1(C(c2c(C)ccnc2)=O)CC2(C1)CN(C(C1(C)CC1Br)=O)CC2CO N1(CCCN2CCSC(C)(C)C2Br)CC2(C(=O)OC(C)(C)C)CC1CO2 C1(C(=O)NCC2CCC(CO)CC2)CCN(C(=O)C2CCCSC2)O1 Cc1ncnc(C(=O)NCCC2CCCN(C(=O)CC(C)F)CC2)c1C c1(C(=O)NCc2ncc(C)c(C)c2)nccc2c(Cl)cccc12 c1(C(=O)NCc2c(C3CCN(C(CC=CC=C)=O)C3)n[nH]c2)cccn(C)c1=O C1(O)(CCNC(CCOCCOC)=O)CCCN(C(c2cnn3c2SCC3)=O)C1 c1(C(N(CC(C)NC(c2c(C)cns2)=O)C)=O)nccnc1N C(c1ccoc1)=CC(=O)NCCN(CCC)C(C1CC1OCC)=O Cc1oc(C(F)(F)F)nc1C(=O)NCC1CC1NC(=O)CC1C=NN(C)C1=O N1(C(CC)=O)CCC2(CCN(C(c3cccc(N(C)C)c3)=O)C2)C1 C1(CC(N2C3CN(CC(c4c(CC)nccc4)=O)C(C3)C2)=O)CN2CCC1CC2 c1(N2CCC(OC)(CNC)CC2)ncnc2ccc(Oc3ccccc3F)cc12 Cc1sccc1C(N1CCC(CNC(=O)C(C2CCOCC2)O)C1)=O Cc1cnc(C(=O)N(C)CCNC(c2csc(-c3ccccc3)n2)=O)cc1Cl C(=O)(CC(C)C(F)F)N1CCC(NC(CC2(C=C)N=N2)=O)C1C(C)C c1(N(C2CCC3(CC2)OCCO3)C)cc(S(=O)(=O)Nc2ccccc2)ccn1 CCCC(CC(C)C)C(=O)N1CCC(CNC(=O)C(C(C)(C)C)OC)C(C)C1 C1(NC)CCN(CC2CC(O)C2(C)C)CC1 C(=O)(CCCCC(N)=O)NC(CC)CN(C(=O)C=CC(c1ccccc1)=O)C C12(C(=O)NCC(c3ccccc3)CNC(CCOCC)=O)CC(F)C1C2 CCCCCC(O)C(=O)NC1(COC)CCCN(C(c2ncccc2Cl)=O)C1 c1(OC)ccnc(-c2nc(C3CC3C(F)F)n(CCCO)n2)c1 c1(C(=O)NCC2C(CNC(C(C)S(N)(=O)=O)=O)C2)cnc2c(c1)CCCO2 C=CCC(C)(CC)C(=O)NC1(CNC(=O)CC2CC3(CC3)C2)CCCCC1 C1CCC(=O)NOC(CC(C)C)C(=O)N1.C(CC(O)CO)N(C(C)=O)C N1(C(C(=C(C)C2CC2)F)=O)CCCCC1CNC(=O)CNS(C)(=O)=O N1(C(CNC(=O)OC)=O)CCC(OCCNC(=O)C(C)(CO)N(C)C)CC1 CC1CCCN(C(=O)Nc2ccccc2F)C1c1noc(-c2ccccc2)n1 c1(C(=O)N)conc1C1CC1.CC1C(=O)NC(C)CCN1C.N(C)C Cc1ccc([N+](=O)[O-])c(C(N2CC(NC(C3(O)CC3(C)C)=O)C(O)C2)=O)c1 c1(C(=O)NCC(CNC(CN(C)C2CC2)=O)F)cc2cccc(Br)c2s1 C1(NC(c2[nH]cc(C)c2)=O)CC2CC(NC(=O)Cn3ncn(C)c3=O)CC12 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C1(O)CCN(C(c2ccnnc2O)=O)CC1)C c1(C(N(C(C)CNC(=O)CCCC(F)F)CC)=O)sc2nccc(C)c2c1C C=CC(O)C(C)(C)C(=O)N1CCC2(CC1)CC2C(N1CCC(OCCC)CC1)=O C1(C(=O)NCC(CN(C(C=CCOC)=O)C)O)CC2(CC2)CN1C N1(C(C(CCC=C)NC(=O)COC2(C)CCCC2)=O)CCC2(CCCC2)CC1 C1(N(C(=O)CC2CC2)C)CN(C(c2ccccc2OCC(F)(F)F)=O)CC1F C1(OC)CN(C(=O)CNC(c2ccccn2)=O)CC1NC(=O)C=Cc1cocn1 c1(OCC)nc(C(=O)NC(C)CNC(c2nc(O)sc2C)=O)cc2ccccc12 c1(NCC2(C)CC2Br)[nH]c(=NCCc2cnc3n2CCCC3)nc2scnc12 Cn1nc(C(N2CC3CC3(CNC(C3CCCC3(F)F)=O)C2)=O)cc1C(C)(C)C C1(C)(C(=O)NC2CC(CNC(CC(=C)Br)=O)C2)CC(OC)CN1C N1(C(CCN(CC)CC)=O)CC(NC(C2COCC2C(N)=O)=O)C(C)C1 c1(OC)cc(C(=O)NCCC2CCC(NC(=O)Cc3cccs3)C2)cc(Cl)c1O N1(C(Cn2cc(-c3c(C)ccnn3)nn2)=O)CC(OCc2cccs2)CC(C)C1 n1(CC(C)(O)C(N2CC(=O)N(C(C(=O)O)C3CC3)C2=O)=O)cnc2ccccc12 CC1CCCC(CC(N2CCC(C)(NC(C3(NC4CC4)CCCC3)=O)C2)=O)C1 C12(C(=O)NC3(CNC(C4C(C)CN(C)C4)=O)CCC3)C3C4C1C1C2C3C41C Cc1[nH]cc(C(=O)NCC2CCN2C(=O)C=CCF)c(=O)c1Br c1(C(N2C(CCNC(C3C(C)(C)C3)=O)CCC2)=O)cccc2c1COCCN2 CC1CN(C(=O)COCC(F)F)CC(C)N(C(c2cc3c(s2)CC(C)(C)C3)=O)C1 C1(c2nnnn2C)(NCCC2(C(=O)OCC)CCCC2)COCC1C N1(C(C(C)CF)=O)CC(NC(c2ccc(C3CCCO3)[nH]2)=O)C(O)C1 C1(CC=C)CCCN(C(=O)C(C)(C2CC2)N(C(=O)CN(C)CCC)C)C1 N1(C(CCC(C)C)=O)CCC2(CCCN(C(=O)CCCc3nccs3)C2)C1 n1(CC(=O)OC(C)(C)C)ccc(=O)n(C)c1=O.C1(OC)CC2N(C1)C(=O)NC2 c1(OC)cc(CC(=O)NCC(O)CCNC(C2OCCO2)=O)cc(Cl)c1 c1(C(N2CCn3c(C)cnc3C2)=O)ccnc2cc(Cl)ccc12 Cc1cc(C(=O)NCCN(C(=O)CC(C)c2ccccc2)C)nn1C N1(C(c2ccnc(Br)c2)=O)CCC(C2CN(C(c3cc(Br)cnc3F)=O)C2)CC1 N#CC1(CNC(=O)CCC2CCCN2C(=O)CC2CCCC(O)C2)CCCC1 N1(C(c2ccnc(O)c2)=O)CCC2CCN(C(=O)COC3CC(F)(F)C3)C2C1 c1(CNC(C=CC(C)(C)SC)=O)cnn(C)c1C(N1CC(CO)C1)=O C#Cc1ccc(C(=O)NC(CNC(c2cccc(OC)c2OC)=O)C2CC2)cn1 c1(CN(C)C)ccoc1C(N1CCCC1C1CCN(C(=O)CCC2(C)CC2)C1)=O C1(OC)CC2CC(C(=O)NCC3(C)CCN(C(c4sc(F)cc4C)=O)CC3)CC12 Cc1ccc(C(=O)N(C)CC2CN(C(=O)C(F)C3CCC3)CC23CC3)c(N)c1 N1(C(C=CCCC(C)C)=O)CCC(NC(c2cnn3occc23)=O)CC(C)(C)C1 C(CCC(C(=O)NCCN=[N+]=[N-])NC(c1cc(F)ccc1O)=O)OC C(C1CCCCc2ccccc21)c1c(O)nccc1.c12nc(ccc1Cl)CN2 C#CC1(O)CCN(C(=O)CC2C3CN(C(C45CSCC4C5)=O)CC23)CC1 N1(C(C(CC=C)CC)=O)CCN(C(c2csc(C(C)C)n2)=O)C2CCC12 c1(-n2cc(C(CC)N(C(=O)CC3(C)CCC3)CC)nn2)cccc(C(F)(F)F)c1 C(C#CC(=O)NCC(CO)(CO)NC(c1oc(CC)cc1C)=O)(OCC)OCC c1(C(NNC(=O)NC(c2ccc(OCC)c(Br)c2)C)=O)nc2ccc(C)cc2[nH]1 C(=O)(C(O)C(C)(C)C)NCC1(CN(C(=O)C(c2ccccc2)O)C)CC1 C1(CNC(c2ccn(CCN(C)C)n2)=O)C2CN(CC3CCCCO3)CC12 C1(NC(c2cc(C)n(C)c2)=O)CCN(C(=O)CCc2cnn(C)n2)CC1CO N1(C(C=CC2(C)COC2)=O)CC(NC(c2cnncc2O)=O)C(O)C1 Cn1cnc(N2CCC(CCNC(c3cccc(F)n3)=O)C2)c(Br)c1=O c1(C(=O)NCc2ccc(Cl)cc2F)c(Cl)cc(Cl)cc1Cl.C12(CC1)C(=O)N2 O=C(C1=CCOC1)NCCOCCNC(=O)Cc1csc(Br)n1 C1(CNC(C2CCCS2(=O)=O)=O)CC12CCN(C(C1CCC(F)(F)CC1)=O)CC2 c1(OC)c(C(=O)NCC2(O)CCN(C(=O)C(F)C3CCOC3)CC2)ccnc1F C1(NC(=O)Cc2ccccc2F)CCCC2CN(C(=O)CCc3nc[nH]n3)CC12 c1(NC(=O)CN(C)CCOC)ccc(C(=O)N(CC)Cc2ccc(Cl)s2)c(Cl)c1 C(=O)(C1=CCC(NC(=O)C(C)(C)n2cnnn2)C1)NCC(CC(=O)OC)C N1(C(C2(CC)CC2)=O)CC2CN(C(C3CCC=CCC3)=O)CC(C1)O2 C1(OC)CN(C(C2(C)CCC(C)(C)C2)=O)CCC1NC(=O)CC1CCOC1 N1(C(COc2cccc(C)c2)=O)CCCCC(CNC(=O)CC2CCCC2C)C1 N1(C(C2CC(C)(O)C2)=O)CC2CC(C1)N(C(=O)CCC1CC1CC1CC1)C2 CC1CN2CCN1CC2C(=O)N(CCCNC(C12CCC(CC1)OC2)=O)C1CC1 N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(c3cnc(Cl)s3)=O)CC2C1 c1(OC)c(C(=O)NCC(CNC(=O)C=Cc2ccncc2)OC)cc(F)cc1F C1(C(=O)NCC(C)(CO)NC(CN(S(C)(=O)=O)C)=O)CCS(=O)(=O)N1 c1(OC(C(=O)NC2(CCNC(C=C(C)C)=O)CC2)C)ccc(C)cc1C C#Cc1cccc(CC(N2CC3CC2C3NC(=O)C(N2CCSCC2)C)=O)c1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)NC(C)CN(C(c1cncc(C)c1)=O)C C(=O)(C1COc2ccccc21)N1CC2C(NC(CCSCCCC)=O)C2C1 N1(C(C2CCC(=C)CC2)=O)CC=C(CC(=O)NC2CSCC2C)CC1 c1(-c2nnc(NC(N3CCC(C(F)(F)F)(CO)C3)=O)s2)ccc(F)cc1Cl CC(C)CC(C)(C)C(=O)NCC1CC1NC(=O)COc1ccc(C#N)cc1 c1(C(N)=O)ccc(C(=O)NC2CCCC2NC(C2CC3CC3C2)=O)cc1 N1(C(C2C(CC)OCC2)=O)CC2=C(C1)CN(C(=O)C(c1ccc(F)cc1F)=O)C2 C(=O)(C1=CC2CCCCCCC12)N(C1CCN(C(c2cc(Cl)nc(Cl)c2)=O)C1)C C(=O)(C(C)CC(=O)NCC1(C(=O)NCCC(C)N2CCCC2)CC=CC1)OC O=C1NCCOc2ccc(CNCC3CCCN(Cc4ccccc4)C3)cc21 Cc1ccc(C(=O)NC2CC(O)CN(C(c3ccc(O)cc3)=O)C2)cc1C c1(NC(C(C)(C)C)C2CC(F)(F)C2)cc(Cl)cc(Br)c1 C1(N(C(=O)CC2CCCOC2)CC)CCN(C(C2(c3occc3C)CC2)=O)CC1 c1(OCC)nc(Cl)ccc1C(N1CCCC(CNC(C23C=CC(CC2)C3)=O)C1)=O c1(CNC(CC2N(C(C3(N(C)C)CCC3)=O)CC2)=O)ncccc1O N1(C(CCC)=O)CCC(C2CCCCN2C(=O)Cn2cc(C(C)O)nn2)CC1 Cc1cc(NC(c2ccc3c(c2)CCO3)=O)c2cc(-c3ccco3)ccc2n1 C(=O)(C(CCC(N)=O)N(C)C)N1CC(C(C)C)N(C(=O)CCC(C)(C)C)CC1 c1(NC(C(=O)Nc2cccc(-c3ccncc3)c2)=O)ccc2c(c1)CCNCC2 N1(C(COC(CC2ON=C(C)C2)=O)=O)CCN(C(C(C)(C)C)=O)CC1 N1(C(COCCC=C)=O)CC2CN(C(c3cnc(OC)c(Cl)c3)=O)CC2(C)C1 C(=O)(CC(C)C(C)(C)NC(c1sc(C)cc1C)=O)NC1CC(C#C)C1 C=CC1(O)CC(C(=O)NC2(CC(N3CCC(SC(=O)OC)C3)=O)CCCCC2)C1 Cc1ccc(C(=O)N(C2CCCC(N(C(=O)COCC(F)F)C)C2)C)nn1 c1(C(=O)NCCCN(C(=O)C(C)C2CCC2)CC)cc2ccncc2s1 N1(C(c2cc(C)c(C)s2)C(=O)NCCOC)CCCc2ccc(C)cc21 Cc1ncc(CCC(=O)NC2(CNC(c3csc(-c4ncccn4)n3)=O)CC2)o1 C1(CC(=O)OC)CCCN1C(C1C=CC(NC(C2CCC(=O)N2)=O)C1)=O Cc1noc(C2CC2)c1C(=O)NCC1(C)CCCN1C(=O)CC1(C)CCCCC1 c1(C(=O)OCc2c(C)sc(-c3ccco3)n2)sccc1S(=O)(=O)N1CCOCC1 N1(C(COC)=O)CCC(CON(C2C3CCC23)C)CC1 N(C(=NCc1ccc(F)cc1)N1CCC(F)C1)C(c1cccs1)C(c1cc[nH]n1)O C1(CC(=O)NC(C(C)C)CCN(C(=O)C=CCO)C)NC(=O)CNC1=O N1(C(C(C)n2cccc2)=O)CC=CC1CNC(c1ccsc1C(F)(F)F)=O c1(C(=O)NCCC2(CNC(C3CC4CCC4C3)=O)CC2)ccnc2ccsc12 CC1CCCn2cc(C(N3CC(O)(CNC(=O)C(c4ccccc4)F)C3)=O)nc21 C1(C(=O)NCC(C2CC2)NC(c2cc(OC)ns2)=O)CCC2(CC1)CNC(=O)C2 CC(C)(CS(C)(=O)=O)C(=O)N1CC2CCCC2(NC(c2cnc3n2CCC3)=O)C1 C1(NC(c2c(OC)ccs2)=O)CCCCN(C(c2cc3ccccc3[nH]2)=O)CC1 CC1CCC(C(N2CCN(C(=O)CCF)CC2)=O)CN1C(=O)Cc1ccnn1C N1(C(CCOCC(C)(C)C)=O)CCN(CCNC(C2(CCF)CC2)=O)CC1 c1(C(=O)NCCC2C(C)(C)CCO2)ccc2c(=O)[nH]ccc2c1 Cc1noc2cc(C(N3CC4CC(NC(=O)CC(C)(F)F)CC4C3)=O)ccc12 C1(OC)CN(C(c2cccc(C)n2)C(=O)NC2CCOC2)CC1O c1(C(=O)NC2C(C)N(Cc3c(Cl)cccc3Cl)CCC2)cnc2cnccc2c1 c1(C(=O)NC2C3OCC(NC(c4occ(C)c4)=O)(C3)C2)cccc(O)c1[N+](=O)[O-] N1(c2cc(C)nc(N3CCOC(c4cn[nH]c4)C3)n2)CC(C)C(C2CCC2)C1 N1(C(CN(S(CC)(=O)=O)C)=O)CCC(NC(=O)C=Cc2ccc(C)o2)C12CCC2 c1(C(=O)NCCN(C(C=C(CC)C)=O)C2CC2)nccc(Cl)c1C c1(SC)nnc2n1CCC2.C1(C2CC2)CN2CC1C2=O.c12cn(nn1)C2 C(=O)(C1=COCCO1)N1C(CNC(CC2CC(OCC)C2)=O)C=CC1 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CC(CO)N(C(C23CC(O)C2C3)=O)C1 C(=O)(C1=CNC2=NCCCC2=C1)NCCN(C1CCCCCC1)C(C(CC)C)=O C1(C(N(C(C)CC(N)=O)C)=O)CC2CCC(C1)N2C(C1CC1C1CC1)=O C(=O)(C1=CCCCC1)N1C(C(C)NC(c2csc(O)n2)=O)CCCC1 N1(C(C(n2ccc(C3CC3)n2)C)=O)CCC(C(C)(C)NC(C2CC23CC3)=O)CC1 c1(CNC(C(=O)NC(C2CC(C)C2)C)=O)cccc(CO)n1 C(CN=c1[nH]c(N2CCC(=CBr)CC2)nc2c1CCCC2)N1C(=O)NCC1 C1(NCc2c(N(C(C(CC)CCOC)=O)C)nc(C)cc2)CCCCN(C)C1=O C(=O)(C(CN(C)C)CC(C)C)N(CCNC(COCC)=O)Cc1ccccc1 N1(C(c2ccc(CCC)[nH]2)=O)CCCCC(NC(c2ncc(F)c(OC)n2)=O)C1 CC1(C)C2CCC1(C(=O)NC13CC(CN1C(=O)C(=O)NCCOCCO)C3)C2 CC1=C(F)CN(C(=O)C(C(C)(C)O)NC(=O)C=CC(=O)N(C)C)CC1 C1(CCCC)CN(C(=O)CC(C)(C)OC)CCN1C(C1CCCNC1=O)=O C1(CCC(=O)NC)CCN(C(C)C)C1.c1(CCCNC(=O)CS)ccncc1 Cn1cnc(CCNC(C(CCCO)c2ccccc2)=O)c1 C1(NC(C(C)O)=O)CCN(C(C2CC3CCC2CC3)=O)CC(C)(C)C1 Cn1cccc1C(N1CC(CNC(=O)CCc2cnc(C3CCC3)o2)C1)=O CON(CCO)C(=O)C1(N(CC(CC(=O)OC)C)C2CC2)CCC1 C(=O)(CC(C)C(=O)NC(C(=O)Nc1cnn(CCF)c1)C1(C)CC1)OC N1(C(C2OCC(C)C2)=O)CC2(CCC2)CC1CNC(C1CC2CCC(C1)N2C)=O c1(SC)cccc(C(N2CCCC2C2(O)CN(C(C3(OC)CCC(C)C3)=O)C2)=O)n1 CC(C)(C)CN=C(N(C)CC1C=CCCCC1)NC1CC(OC(=O)N(C)C)C1 c1(C(N2C(C)C(NC(=O)CCC3CCC3)CCC2)=O)ccnc2ccnn12 C(=O)(C(CC(C)(C)C)OC)N(C(CC(=O)NC1CC(CC)OCC1)(C)C)C CCC(C)(C)CCCC(=O)N(C(C)C(N1CCC12CCCSC2)=O)CC C1(C(N2C(C)(CC)CCC2)=O)CC2(CC(NC(c3c[nH]nc3C3CC3)=O)C2)C1 O=C(CCC(=O)c1ccc(F)cc1)NC(=O)Cc1cn(CC2CC2NCCl)nn1 Nc1cc(F)c(C(=O)NC(CNC(=O)CCC2CC2)CO)cc1F c1(C(=O)NC(C(C)NC(=O)C(C)C(C)O)C)cncc2nnn(C)c12 C1(N(C(c2ccc(=O)oc2)=O)CC)CCCN(C(C2(COC)CCOC2)=O)C1 c1(C(N2CCC(N(C(=O)CN3CSCC3=O)CC#C)CC2)=O)ncc(F)cc1F C1(NC2CC(c3ccccc3)(CC(=O)OCC)C2)CCC(S(C)=O)C1 C(CCN1CCCC1)(C(=O)N1CCCC1)NC(=O)NCc1c(CC)occ1 C1(NC(CC(C=C)CC)=O)CN(C(c2cc(CC)[nH]n2)=O)CCC12CCC2 C1(CNC(c2cc(CO)on2)=O)CN(C(=O)CCc2cnc(O)[nH]2)CC1O c1(N2CCCC(C=C)C2)nc2c(c(=NCC3(N(C)C)CCSC3)[nH]1)SCC2 C=CCC(CNC(c1sccc1F)=O)NC(=O)C(n1ccc(C(F)(F)F)n1)C N1(C(CCc2ccc(C)cc2)=O)CCC(F)C(NC(=O)Nc2ccccn2)C1 N1(C(C2CN(C(c3n(C=C)ncc3)=O)CC2C=CC)=O)CCC(C)CC(C)C1 CC1(C)CC(NC(=O)C=C2CCC2)CN(c2ncc(C#N)cc2F)C1 c1(C(=O)NCC23CC2CN(C(=O)CCn2ccnn2)C3)cncc2nc(O)[nH]c12 n1(CCCC)nccc1C(N1CCC(N(C(C2CCCC2C(F)F)=O)CC)C1)=O C(=O)(C1=CC2CCCCCC12)N1CC2CCC(NC(=O)CCCC(F)F)CC2C1 C(=O)C(C)(O)C(C)C.C1(CC)CCCN(C(CC)C(=O)NCc2cnc(SC)[nH]2)C1 c1(C(=O)NC(CCN(C(Cc2cn(CC)nc2)=O)C)C)ccncc1C(F)F c1(C(=O)NC2C(NC(Cc3c(CC)cccc3)=O)CC2)cccc(Cl)c1O N1(C(C(c2ccc(Cl)s2)C)=O)CCC2C1CCCN2C(=O)Cc1nncn1C N1(C(C(C)(C)C2CC2)=O)CCN(C(C2C=CCC2)=O)C(C2CC2)C1 c1(C(=O)NCCCN(C(C(CCCC#C)C)=O)C)ccc2ncc(Br)n2c1 c1(OC)ccc(CC(N2CC(CNC(=O)CC3CCC(CN(C)C)O3)C2)=O)nc1 Cc1ccc(OCC(=O)NCC2(C)CN(C(=O)CCCC(C)F)CC2C)cc1C c1(CC)cccc(C(=O)NCC2CCCCN(C(=O)CC3OCCCO3)C2)c1F N1(C(C2C(CNC(Cc3cc(CC)no3)=O)CCO2)=O)CCCC(CN(C)C)C1 C(=O)(CCC(=O)C1CC1)NCCCN(C1CCCC1)C(c1nc(CC)sc1)=O CC(c1ccccc1F)=CC(=O)NC(C)(C)C(C)NC(c1c[nH]cc1Br)=O c1(C(N2CC(NC(CCCC=C)=O)C(C=C)C2)=O)oc2ccccc2c1Cl C12(NC(Cc3c(CSCC)cccc3)=O)CCCC1N(C(c1cocn1)=O)CC2 c1(C(=O)NCC2C(NC(C=C(COC)C)=O)CCC2)c[nH]c2cccc(C#N)c12 C1(C(=O)NCC(C)(F)F)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C(=O)NCC(C)N(C(C(CCC)OC)=O)C)cccc(C2=CCOCC2)c1 c1(C(=O)NC(c2ccc(C#N)cc2F)C)cn2cc(C(F)(F)F)ccc2n1 C1(C(=O)NCC(c2ncc[nH]2)C)CC(C)(C)CCN1C(=O)CCC1CCOCC1 c1(C(=O)NC2(CNC(c3ccc(O)nc3Cl)=O)CCC2)ccnc2ncnn12 Cn1ncnc1CNC(c1cn(CCNC(C2CCCC2)=O)cn1)=O C1(C)(CNC(CC2(COC)CCC2)=O)CCCN1C(=O)CCc1ccc(C)nc1 CCC(C)(CC)C(=O)NCc1ccoc1C(=O)Nc1cnc(Cl)nc1C c1(C(C(=O)NCCOCCNC(=O)C=Cc2ncco2)O)ccc(F)c(F)c1 N(C(=NCCc1ccn(CC)n1)N1CCC(c2ccccc2F)C1)C(CC)C c1(C(=O)NCCC2COCCN2C(c2nc(Cl)cs2)=O)c[nH]nc1[N+](=O)[O-] c1(OCOC)cc(F)c(CN(C)Cc2ccoc2C)cc1Cl C=CCCC(C)(C)C(=O)N1CC(NC(c2c(Cl)cccc2Cl)=O)C2(CC2)C1 CCCCCCn1nnnc1C1(NCc2cnc(C(C)C)s2)CC1(C)C Cc1nc(C(=O)NCC(C)(CO)NC(c2cscc2Cl)=O)nn1-c1ccccc1 c1(OC)ccc(CC(O)C(=O)NC(CO)C(C)NC(=O)Cc2conc2C)cc1 C(N=c1[nH]cncc1Br)C1(CNC(C(C)(C)c2cncnc2)=O)CCCC1 N1(C(CN(C(C)C)C(c2ccnc(N(C)C)c2)=O)=O)CCCCC1CO N12C3CCC1CC(C3)C2=O.Cc1c(NC(=O)C(F)C(C)(F)F)cccc1F c1(C(C)C)ccc(CC(=O)NCC2(O)CC(NC(C3COC(=O)C3)=O)C2)cc1 N1(C(c2c(C)nc(C(C)C)o2)=O)CCN(C)CC1CNC(C1CC12CC2)=O C#Cc1ccc(F)cc1NCC1C(NC(=O)NC(C)(C)C)CCC1 N1(C(c2nc(C)[nH]n2)=O)CCCC(C(=O)NCCCNN2CCN(C)CC2)C1 c1(CC)cc(C(=O)NC(C(N2CC3CC2C3C(N)=O)=O)c2cccs2)c(C)o1 N1(C(C(C2CCCC2)OC)=O)CCCCC1CNC(C1(N2CCCC2)CC1)=O c1(CC(=O)NC(C(C)(C)C)CNC(c2cncc(F)n2)=O)ccc(C#N)cc1F C1(NC(=O)CC(O)c2ccccc2)(CNC(=O)C(O)C2CC2)CCCCC1 Cc1cc(C(N2CCCC2(C)C(N2CCn3ncnc3C2)=O)=O)cc(C)c1O CCC(CC)(CO)C(=O)N1CCCOC(CNC(c2cn(C)nc2C)=O)C1 C1(C(=O)NC2CC3(CC(OC)C3)C2)CC12CCN(c1ccc(C(C)=O)cn1)CC2 CC(C)CC(CNC(=O)C(CC1CC1)CC1CC1)NC(=O)Cc1ccccc1Cl c1(NC(C2C(C(=O)NC(C)CO)C2)=O)onc2ccccc12 N1(C(c2scc(C(N)=O)c2)=O)CCN(C(C2CC2CF)=O)C(c2ccccn2)C1 c1(CNC(C2C(C3C(C)C3)C2)=O)cccc2c1CCN(C1CCN(C)C1=O)C2 N1(C(C(C)S(N)(=O)=O)=O)CC(NC(C2CC3(C2)CC(F)C3)=O)CC(C)(C)C1 C1(NC(C(CC)OCC)=O)CC2CN(C(c3ncc(Br)cc3O)=O)CC12 Cn1cc(Cl)cc1C(=O)NCC1CCCCC1NC(c1cnccc1Cl)=O c1(C(N2CCC(=CCNC(C(CSC)O)=O)CC2)=O)cnc(O)cc1F C1(C(N(CC(CN(C)C(c2ccc(F)cc2)=O)O)C)=O)CCC2(CCC2)CO1 C1(C(N2C(CC)CC(O)C2)=O)CCC2(CC2)N1C(c1cc[nH]c1)=O n1(CCC)nnnc1C(C1CC1C1CC1)NCCNC(=O)C(C)C C12(C(=O)NC(CNC(C(C(=O)OC)C)=O)(C)C(C)C)CCC(CC1)OC2 C12(C(=O)NC3C(NC(C4(OC)CCC4)=O)CCCC3)CCCN(CC1)S2(=O)=O C1(C(=O)NCC2CN(C(C(CCNC(=O)C3CC3)O)=O)C2)CCc2ncnn2C1 C(C(F)(F)C(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)C(SC)C1)SC CCC(CC)C(F)C(=O)N1CCCC(F)(C(=O)NCC(n2cccn2)C)C1 C1(C2CC2)(CNC(c2n(CC=C)ccn2)=O)CCN(C(=O)C=CS(=O)(=O)CC)C1 C1(CNC(=O)NCC(c2ccsc2)C)CCCC1N(C)C C(=O)(CC(C)CC(=O)OCC)NC1(CC=C)CCCN(C(=O)C=CC(F)(F)F)C1 N1(C(C(C)OCC=C)=O)CC(=O)NC(=O)C1 N1(C(C=NOC)=O)CCC(C)N(C(=O)CCOc2ccc(Cl)cc2F)CC1 Cc1cc(C(=O)NC2CCC(C)N(C(c3cc(C#N)c[nH]3)=O)C2)cnc1C C1(NC(Cc2ccc(C)c(C)c2)=O)CCC2CC1CN2C(=O)CCC(F)F N1(C(c2n(C)nc(C(F)F)c2)=O)CC(NC(c2ccc(F)s2)=O)C2(CC2)C1 C(=O)(N=c1ccc(C(F)(F)C(F)(F)F)n[nH]1)N(C1(OC)CCC(C)C1)C(=O)C1CC1 CCCCC(C)(CO)NC(=O)CCCCCNC(c1cc(C)nc(C)c1)=O C1(C(=O)Nc2ccc(CC(=O)OC)cc2)CC2(CCOCC2)CO1 c1(OCC)ccc(CCC(=O)NC(CNC(C2CCN(C)CC2)=O)C2CC2)cc1 CCN=c1ccc(C(N2CCCCC(NC(=O)C(C)OCC3CC3)C2)=O)c[nH]1 N(C(=NC(C)c1nncn1C)NCC1(SC)CC1)C(CC)CC Cc1nn(C(C)C)cc1COC(c1ccc(CC(=O)N(C)C)cc1)=O c1(C(=O)NC2(CNC(CCC)=O)CCCC2)cnncc1C C(N=c1[nH]c(=NCCC#N)[nH]c2c1CCCC2)c1ccnc2[nH]cc(C)c21 c1(C(N2C(CCN(C(COCC=C)=O)C)CCCC2)=O)ccc(Br)c(O)n1 N1(C(C(=O)N(C)CC2(OC)CCCCCC2)=O)CCC(C)CC(C)C1 n1(-c2ncc(C(=O)NCC(=O)N(C3CCC3)CC#C)s2)c(C)ccc1C C(=O)(C1CCc2nccn21)NC(C)C(C)C(=O)NCC1CN(C(N)=O)C1 C1(C(C)C)CN(C(C(=O)NCC2CCOC2)C2CC2Cl)CCO1 Cc1nccnc1C(=O)NC(C)CCN(C(=O)Cc1cncs1)C C(C(C)(C)CNC(=O)CC1(CO)CC1)N(C(C(C)=CC1CC1)=O)C CC1CN(C(C2(C#N)CC3(CC3)C2)=O)CCC1NC(C1(C2CC2)CCC1)=O CC1(C(=O)NCC#CCN(C)C)CC12CCN(C(c1ccon1)=O)CC2.C(=O)OC c1(CC)c(C(N2CCCC2C2(C(=O)OC)CC2)=O)cnn1-c1ccccc1 N1(C(CCC(C)OC)=O)CC(N(C)C(c2ccnc(C(F)(F)F)n2)=O)C2(CC2)C1 c1(OC)cc(C(N2CCOC3CC23)=O)c(NC(c2cccc(O)c2F)=O)cn1 C1(C#N)(CC)CC2CCC1CC2(C#N)NCCCC1CC1(Cl)Cl N#Cc1c(Br)ccc(C(=O)NC2Cc3ccccc3C2O)c1F N1(C(=O)NC2CCC(C)C2)CCN2CCCC2C1 C1(CC)CN(C(=O)C(C)Cn2ccnc2)CCN1C(c1cc(Cl)cnn1)=O CCCC(CC1CCCC1)C(=O)NCC(C)(C)OCCNC(=O)Cc1ccsc1 c1(SC)cccc(NC(=O)Cc2ccc(C3CCNCC3)cc2)c1 Cc1ccoc1C(=O)NC1COCC1CNC(=O)C(C)c1ccco1 c1(C(N2C(C)(CNC(C3C(CC)OCC3)=O)CCC2)=O)cc(O)cc(O)c1 CN1C(=O)CCc2cc(NCC3CCCC3C(C)(C)C)ccc21 C1(C(=O)NC2N(C(C(COC)N(C)C)=O)CC=CC2)CC(C)(C)OC1=O Cc1csc(=O)n1CC(=O)NCCN1CCN(C(=O)CCCc2cnn[nH]2)CC1 c1(OC2CC(NC(C(C)SCc3cccs3)=O)C2)cccc(Br)c1 N1(C(c2c(C)cc[nH]2)=O)CCC(C(N2CCC(C)(CCO)C2)=O)C1C C(=O)(C(C)C(C)c1ccccc1Cl)NCCCN(C(c1c(CC)noc1)=O)C c1(CCN)nccc(C(=O)N(CC2CC2)CC2CCCO2)n1 C1(NC(CC(C)F)=O)Cc2ccccc2C1NC(c1ccc(Cl)c2occc12)=O N1(C(=O)C=CCn2cncn2)CCC(C(C)CCNC(C(C)O)=O)CC1 c1(OC)nc(C)c(C(=O)NCC(=O)Nc2nc(Cl)cs2)s1 C(N=c1[nH]c(Cl)nc2c1SCC2)C1CN(C(C(C)NC(C)=O)=O)CC12COC2 CC(C)CCC(F)C(=O)NCCOCCOCCCNC(=O)C(C)C#N C1(CC=C)(C(=O)NC(C2CCCN2C(=O)CCC2CC(F)(F)C2)C)CCOC1 c1(OC)ccc2c(CC(=O)NCC(C3CCC3)NC(c3cnco3)=O)coc2c1 c1(C(N2CC(C)C(C(N3CCC(O)(C(F)F)C3)=O)C2)=O)cn(C)c(=O)n1C C1(CC(=O)NCCC2CC(NC(Cc3cn(C)nn3)=O)C2)CCCCCC1(F)F C1(C)(C(N2CC(C(C)NC(c3c(COC)cco3)=O)C2)=O)CCC(=O)N(C)C1 C(=O)(CCS(=O)(=O)Cc1ccccn1)NCCN(C)C(C12CCCN1CCC2)=O C1(C(C)NC(=O)CCCC(N)=O)COC(C)(C)CN1C(c1cnc(O)c(F)c1)=O CC(C)C(N=[N+]=[N-])C(=O)NC(C(N1CC2(CCCN2C)C1)=O)C1CCCO1 c1(CNC(c2coc(C3CC3)n2)=O)n[nH]c2c1CN(C(=O)Cn1cccn1)CC2 CCCCCC(C)(CC)C(=O)N1C2CCC1CC(NC(=O)C#CC1CC1)C2 c1(C(=O)NC(C)CNC(C2CC2C2CC2)=O)cc2ccccc2n1C C1(F)(CNC(c2cnc(C)n2C)=O)CCC(CNC(=O)CCCC2CC2)CC1 c1(C(=O)NCC2(O)CN(C(c3n(CCC)ncc3)=O)C2)nn(C(C)C)cc1Br C1(CC(C)C)(C(=O)NC2CC(CCNC(=O)C(CO)N(C)C)C2)CCCC1 c1(NC(=O)NCC2C(OC)(OC)CC2)ncoc1-c1cc(C)no1 C(CC(=O)N(C)C(c1cc(C)on1)C)(C(F)F)Nc1c(C(=O)OC)cccc1 c1(OC)ccc2cc(C(N3CC4CC(NC(=O)C(F)C(C)C)C3C4)=O)n(C)c2c1 N1(C(c2c(C)cc(C)o2)=O)CCC2CCN(C(c3ccc(CN(C)C)[nH]3)=O)C2C1 C=CC1OCCC1C(=O)NC(C1(O)CN(C(=O)CC2(C(F)(F)F)CC2)C1)C C(=O)(C(C)NCCN(C)C)NC(CCN(C(C)C)NC(=O)OC(C)(C)C)C N1(C(C=C(CC)CC)=O)CCCCC1C1CCN(C(=O)C2=C(Cl)CC2)C1 C1(CC(=O)NCC(n2cccn2)C)CCN(C(c2ccc(F)c(F)c2)=O)C1(C)C c1(CN2CCC(O)(C(=O)Nc3cccnc3Cl)C2)ccc(Cl)c(I)c1 C1(NC(C=C(C)CNC(=O)CC2C=NN(C)C2=O)=O)COC2(CCC2)C1 Cc1nn(C2CCCN(CC3CCC(CCC(=O)N(C)C)C3)C2)c(C)c1Cl C12(C(=O)NCC(CN(C(c3ccc(CC)[nH]3)=O)C)(C)C)CCC(C1)OC2 c1(C(N2C(CNC(C(C(C)C)F)=O)C(C)CCC2)=O)nccc2ncccc12 CC1C(NC(=O)C(=O)Nc2sccc2F)CCCN1C(=O)OCC(C)(C)C C#CCC(CC#C)C(=O)N1CCCCC(NC(=O)CC(C)C(F)(F)F)C1 Cc1cccc(N)c1C(=O)NCC#CCNC(=O)C(C(C)C)c1ccccc1 Cc1ccc(NC(C2CCN(C(c3c[nH]ccc3=O)=O)C2C)=O)c(O)n1 N1(C(c2c(CC)noc2)=O)CC2(CC(NC(=O)C(N3CCCC(C)C3)=O)CO2)C1 Cc1[nH]c2ccccc2c1C(=O)NC1CCCC1C(=O)NC(C1CCOC1)C c1(N2CC(CC)C3(C2)CCC3)[nH]c(=NC2CC(N)C2)nc2c1cnn2C(C)C.SC N1(C(COCCC#C)=O)CCCC1C1CCN(C(=O)CSCCN(C)C)C1 C(=O)(C(F)C(C)(C)O)NCC1C(C)CCN1C(=O)C=Cc1ccccn1 N1(C(C(C)NC(N)=O)=O)CCC=C(C(=O)NCC2CCCCS2)C1 c1(C(CNC(c2cc(C)[nH]n2)=O)NC(=O)C(F)(F)c2cscn2)ccc(F)cc1 C1(CC)(NC(=O)C(O)C2CCOC2)CCN(C(=O)Cc2cccc(C)c2F)CC1 C1(C2(NC(=O)CSn3cncn3)CC2)CCCN1C(c1cccnn1)=O CCCCCC(=O)N1CCOC(CNC(=O)CN2CCNC(=O)C2)C1 C1(CNC(Cn2ccc(C)n2)=O)CN(C)CCN1C(c1ccc(C(C)C)cn1)=O c1(C(=O)NC2CC(N(C(=O)CSC(F)(F)F)C)C2)cccn2ccnc12 C1(C(=O)NC(CNC(c2c(CC)n(C)nn2)=O)C2CC2)C2CCCCCC12 N1(C(C(COC)OC)=O)CC(NC(c2ccoc2)=O)CCC(O)C1 C1(C(n2cc(C3COCCN3Cc3ccncc3Br)nn2)C)CC2CCC1CC2 c1(C(N2CC(C)(NC(C3C(=C)C3)=O)C2)=O)ccc(-n2cccc2)cc1O NS(=O)(=O)c1ccc(C(=O)NCC(O)CNC(=O)CN2CC3CC3C2)cc1 C1(NC(=O)CCc2cnco2)CCN(C(=O)CC2CC2)C(c2ccccc2)C1 C1(C(N2C(CCNC(C3(C)CC=CCC3)=O)CCC2)=O)CCC2C(C1)C2(F)F C12(C(N(CCCNC(=O)Cc3cc[nH]n3)CCO)=O)CCC(F)(CC1)CC2 N1(C(C2(O)CC(C)(C)C2)=O)CCC(NC(c2cc[nH]c2)=O)C(CO)C1 Cc1cc(C(N2CC(N3CCN(C(=O)Cn4cnnc4O)CC3)C2)=O)c(O)nn1 CC(CC(=O)NCC(C)CN(C)C(C1CC(C)(C)C1)=O)c1ccco1 N1(C(Cc2c(C)nc[nH]2)=O)CCC2CN(C(=O)C(O)CC[S+](C)C)CC2C1 C1(c2ccccc2)(C(=O)NCCCC(c2cccnc2)=O)CCCCO1 CN1CCN(CC(=O)NCC23CC2CN(C(=O)COc2ccccc2)C3)CC1 c1(NC(CC)(CNC(C2CCC(C)CC2)=O)CC)ccc(C#N)c(C)n1 c1(C(N2C(C(=O)Nc3cc(OC)cc(F)c3)CC2)=O)c[nH]c2ccc(F)cc12 C1(NC(CC2N(C)CCCC2)=O)CCCCCCC1NC(=O)CC=CC(C)(C)C CS(C)(=O)=NCC(=O)NC1CCN(C(=O)Cc2cccnc2Br)C12CC2 c1(OC)ccc(C(N2CCN(C(=O)Cn3cnnc3O)C3CC23)=O)cc1Cl C(CCCC(C)NC(=O)C(CC1CC1)CC1CC1)NC(CCCSC)=O C(=O)(CC(C)CC(C)(C)C)NC1CN(C(c2cnc(C)n2C)=O)CC1O CC1CC(NC(=O)C(=O)Cc2ccccc2)CCN1C(=O)Cc1cocn1 CCC(CC)C(=O)N(C(CC)CC(=O)NCCC1(COC)CCC1)C c1(C(=O)NCC(CC)NC(c2cnc(C)[nH]2)=O)c(C)oc(C)c1Br c1(C(C(C)C)NC(C2(c3ncon3)CC2)=O)ccccc1Cl C(=O)(CCCNC(=O)COC)N(CC(C)NC(=O)CCOC(C)CC(C)C)CC C(CCCNC(=O)CCC1CCCOC1)(c1ccccc1)NC(C=C(C)Cl)=O CCCC(C(=O)OC)C(=O)NC1CC1NC(c1sc(O)nc1C)=O c1(CCC(=O)NCCN2CCN(C(C3C(=C)CC3)=O)CC2)ccc2ncsc2c1 C1(C(=O)Nc2cn(CC#C)nc2)CCN(C(=O)C2=C(C)OCCCS2)O1 C1(CC)(NC(=O)C(C)CC(F)F)CCN(C(c2ccncc2)=O)CC1 c1(CC)sc(C(=O)NCC2CCN(C(=O)CCC3CCOCC3)C2)cc1C c1(N(CC=C)C)ccc(Br)c(S(=O)(=O)NCCc2c(F)cncc2F)n1 c1(CC(=O)NCC)ccccn1.C1(C(F)F)CC1 C1(C(=O)NC2(CC)CCOC2)CC2CCC(C1)N2C(c1cc(C(C)=O)[nH]n1)=O N1(C(c2c(NC)c(F)ccc2)=O)CC2CCCC(C1)N2C(C1(SC)CCC1)=O Cc1cccc2[nH]c(C(N3CCC4CCC(C3)N4C(=O)CNC(N)=O)=O)cc12 C1(C)(NC(c2ncn(CC)c2)=O)CCN(C(c2cc(-c3csc(C)n3)c[nH]2)=O)C1 C(CN=c1nc(C#N)[nH]cc1C)C1N(C(Cc2cnc(C)s2)=O)CCCC1 C12(NC(c3nn(CC)c(C)c3)=O)CCCC1CN(C(c1cc(C)oc1C)=O)C2 C(=O)(C(C)(C)CC(C)C)NCC1OCCC(NC(c2c(Cl)cnc(CC)n2)=O)C1 C1(C(=O)NCC(C)N(C)CC2CC23CCOC3)COCCN1C1CCCC1 Cc1cc(Br)c(Cl)cc1NC(C1CC1NC(c1cc(=O)cco1)=O)=O C1(C)(NC(C(C)CCN(C)C)=O)CCCN(C(=O)CC2CCC(C)C(C)C2)C1 C1(CNC(C(COC)C)=O)CC2CCCCC2N1C(=O)CCn1cccnc1=O N1(C(C(F)OC)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C(C)C)=O)C(C)C1 c1(C(=O)NC2CC3CN(C(C4ON=C(C)C4)=O)C2C3)c(C)[nH]c2ccccc12 Cc1ccc(C(=O)NC(C2CCN(C(=O)CC3COCCO3)CC2)(C)C)c(C)c1 c1(OC)ccc(C(=O)NCCCNC(C2CS(=O)(=O)CC23CC3)=O)c(OC)c1Cl C(=O)(C#CC1CCCCO1)NCCCN(C(c1c(Br)ccc(C)n1)=O)C1CC1 Cc1cccc2oc(C(N3CCCC4(C3)CN(C(C3(C)CC3(F)Cl)=O)C4)=O)cc12 c1(C(C)C(=O)NCC2(F)CN(C(=O)CCN3CCCC3)C2)nc(F)ccc1Cl N1(C(CC2CN(CCN(C)C)CC2N)=O)CCc2cc(C(F)(F)F)ccc21 N1(C(CCC)=O)C2CCC1CC(CNC(c1ccc(OC(F)F)cc1)=O)C2 c1(C(=O)NCC2CC(NC(C(C)N(CC(F)(F)F)C)=O)C2)ccc(N)cc1Cl C(=O)(C(CNC(c1ccn2nccc2c1)=O)CC(C)C)NCCN(C(=O)OC)C C1(C(N2CCCC(OCC)C2)=O)CC2(CCN(C(=O)C(c3cccn3C)=O)C2)C1 CN1CC(C)(C)CC1C(N1CCCC1c1cn(-c2c(F)cccc2Cl)nn1)=O Cc1cc(C(N2CCCCC(NC(c3ccc(Cl)nc3O)=O)C2)=O)nc(C)c1 C(=O)(C1=NOCC1)N(CC(CC)NC(=O)Cc1cccc(OC(F)F)n1)CC N1(C(=O)CS(=O)(=O)N2CCOCC2)CCC2CCN(C(=O)C(F)C3CC3)C2C1 CN1N=CC(CC(=O)NCC2CN(C(C3CCS(=O)(=O)C3)=O)C2)C1=O CCC(C#N)C(=O)NC1(C)CC(NC(c2cc(C(F)(F)F)on2)=O)C1 c1(C(=O)NCCN(C(CC(C)n2ccnc2)=O)C)ccc(C(=O)N(C)C)c(F)c1 c1(CNC2(c3n(C(C(=O)OC)C)nnn3)CC(F)(F)C2)ccc(C)c(Br)c1 C1(CC(=O)NC2(COC)CN(C(=O)C(CO)N(C)C)C2)CC2(CC2)CO1 C(=O)(C1=CCc2ccccc21)NCC1C(NC(c2cc(C3C(C)C3)on2)=O)CCC1 c1(C(=O)NCC2C(NC(C(CC(C)C)O)=O)CCC2)ccc2c(c1)CC(C)O2 Cc1nn(CC(F)F)cc1-c1nc(-c2occc2C)nn1CCCN(C)C c1(C(=O)NCC2C(NC(C3CN(CC)C(=O)C3)=O)C2)cncc(Cl)c1C N1(C(C(COC)(C)O)=O)CCN(C)C(CNC(=O)Cn2nc(C)cc2C)C1 c1(OC)cc(C(N2CCC(CNC(C3CNC(=O)C3)=O)CC2)=O)cnc1Cl C#CC1CC2(CC2)CN1C(=O)NCC(C(C)C)c1ccccc1 N1(C(C(C)OCCOC)=O)CCC2CCCC12C(=O)NCC1CCC(C)(CO)O1 C(=O)(CCCCCCC(=O)NC(CO)C(C)NC(=O)C(F)OC(F)(F)F)OC N1(C(C2CC(O)CN2S(=O)(=O)CCc2ccccc2)=O)CC2(CC2)CC1CN C(=O)(CC1=NN(C)C(=O)C1)N1CC(CC)C(NC(c2cc(Cl)c(Cl)[nH]2)=O)CC1 CN1CC2CC1CN(C(=O)CCC1CCCCN1C(=O)COc1ccsc1)C2 C1(NC(C2CCCC(C)CC2)=O)CC2CCC1N(C(=O)C=Cc1cccnc1)C2 C1(CNC(c2c(CNC(CCC#C)=O)ocn2)=O)CCC(=O)NC1C C1(CNC(C(C)CCN(C)C)=O)CC2(CCN(C(C3(C)CCCN3C)=O)CC2)C1 c1(C(C)C)ncc(Br)c(=NC(CNC(C2CCC(=O)N(C(C)C)C2)=O)CO)[nH]1 C1(C)(CNC(c2cc(CCC)[nH]n2)=O)COCCN(C(=O)C(C)c2ccsc2)C1 c1(N(C)Cc2cc(Br)cs2)nc(N2CCN(CS(C)(=O)=O)CC2)c2c(n1)CCS2 N1(C(C2(CC#C)CCCO2)=O)CC(C(N2CC(F)(CF)C2)=O)CCC1(C)C C(C1CCCC1)=C(C)C(=O)NCC1CN(C(C2(n3cc(C(C)C)nn3)CC2)=O)C1 N1(C(C(CSC)O)=O)CC(NC(=O)Cc2csc(C)c2)C(C2CC2)C1 CCC(C)(C(=O)NCCOCCCNC(=O)Cc1ccoc1)OC N#Cc1cnn2ccc(N3CCCCC(NC(=O)Nc4ccccc4F)C3)nc12 C(=O)(CCCCC(C)C)N1CCCC(O)(CCNC(CC(C=C)C)=O)C1 C(C(O)C(C)(C)C)NC(c1scc(CNC(CC2C(CC)C2)=O)c1)=O c1(C(N(C(CNC(=O)C(C)(F)C(F)(F)F)C2CC2)C)=O)cc([N+](=O)[O-])ccc1Cl CCC(C)(C)C(O)C(=O)N(CCC(=O)NC(C)(CO)C1CC1)C C#Cc1ccnc(C(N2CCN(C(c3cc(O)cc(=O)o3)=O)C3CC23)=O)c1 c1(C(C)NC(c2c(C(=O)NC(CC=C)=O)ccs2)C)[nH]c(C)nc1C c1(C(=O)NC(CCC)CCCNC(=O)CC(CC)C2CC2)cn2cccnc2n1 Cc1noc(C)c1CC(=O)N(C)CCC1CCCCN1C(C1CC1C(C)(F)F)=O C1(C2CCC2)(C(=O)NCC(CO)NC(C2(c3cccc(F)c3)CC2)=O)CC1(F)F C1(NC(c2cc(C)cc(F)c2N)=O)CCCC2CN(C(=O)C3=CCOCC3)CC12 C#CCC(CC(=O)NC(c1nnnn1C)C)NC(C1(C)CCOCC1)=O C(=O)(C1CCc2nccn21)N(C)CC1CCN(C(C2CCCS2(=O)=O)=O)CC1 C(=O)(C(CC(C)C)N(C)C)NC(CCN(C(CC(C)SC)=O)C)C c1(C(=O)OCC)cc(N(C2CCN(C(c3ncoc3CC)=O)C2)C)nc(C)n1 N1(C(C(C=C)O)=O)CCCCC1CCC(=O)N1CC(N(S(C)(=O)=O)C)C1 C1(CO)CCCC2(CCN(c3nnc(-c4csc(CO)n4)s3)CC2)O1 C1(O)(CNC(=O)C(c2ccccc2)O)CN(C(=O)CCCC2CC2)C1 C1(C)(CNC(CN(CCOC)C)=O)CCC(NC(=O)C(C)=CC(C)C)C1 c1(OS(C2C(NCCOC)CC2)(=O)=O)ccc(S(=O)(=O)C2CC2)cc1F c1(OC)c(Br)ccc(F)c1CNC(c1ccc(F)cc1F)C1CC1 C(C(CC(=O)NC1CN(C(=O)CC2(C)CC2)CC(C)(C)C1)C(F)F)N(C)C C(=O)(C(C)CC(F)(F)F)NC1C(CCC)CN(C(C2C=CC=CC=C2)=O)C1 c1(C(N(C2CCN(C(C34CCC3C4)=O)C2)C)=O)cccc(C#N)c1 c1(C(N2CC(CC=C)(NC(c3nc(C)sc3C)=O)C2)=O)cc(C#N)ccc1O C(=O)(CCC(F)F)N1C(C(C)(C)CNC(=O)CCCc2ccccc2)CCC1 N(C(=NCCCF)NCC(C(=O)OC(C)(C)C)Nc1ccccc1)CC(=C)C C1(F)(CNC(c2c(C)onc2)=O)CC2CCC(C1)N2C(=O)Cc1ccsn1 CC1CN(C(c2cccc(C#N)c2)=O)CCC1N(C(=O)C1=CCOCC1)C c1(C(N(C)CC2CN(C(=O)C=Cc3cncnc3O)C2)=O)cc2ncccc2s1 c1(OCC)cc(Cl)ccc1C(=O)NC1CN(C(C2CCCC2(F)F)=O)C1 c1(C(N2C(C)CCC(NC(C3CC34CCOC4)=O)C2)=O)cccc2c1OCCN2 c1(OC)ccc(CN2CC3CC2CN3C(=O)C(C)NC(=O)C(C)(C)C)cc1F C1(NC(c2n(C)nc(CNC(=O)CCCCCF)c2)=O)CC2(C1)CC(C#N)C2 N1(C(COCC)=O)CCN(C(c2scnc2CC)=O)CC1COC CCCCC(C(=O)N1CC(C(N2CC(CC)(OC)C2)=O)CC12CCC2)C(C)C C(CC1CC1)(CC(=O)N1CCOCC1CCO)NC(c1ccn(COC)n1)=O S(=O)(=O)(c1cc(C(=O)Oc2ccc(C(=O)O)cc2Cl)c(Cl)cc1Cl)NC CCC(CCC(=O)N(C(C)CN(C)C(c1ccc(C(=O)OC)s1)=O)C)OC C(=O)(C1=CC2CCCC12)NC1(CNC(CNC(C(C)(C)C)=O)=O)CC1 C1(CC(=O)NC2(CCC)CC2)CCCN(C(C2CC(F)C(=O)N2)=O)C1 C12(CNC(C3CC(C#N)C3)=O)CCC(NC(=O)Cc3cccc(Cl)c3)(CC1)CO2 CC1=C(C(=O)Nc2ccc(-c3ccc(OC(C)(C)C)cc3F)nc2C)CCO1 N#CC1CN(Cc2ccc(N3CCCC3)nc2)CC1NC(c1cc(Cl)ncc1Br)=O N1(C(C2(S(C)(=O)=O)CC2)=O)CC2CCCC2(CNC(=O)Cc2ccc(O)cc2)C1 c1(NCc2c(CNC(CN(C)CC)=O)cccc2)ncc2ncnc-2[nH]1 CC1CN(C(c2cnnn2C)=O)CC1NC(C1(C)C=CCC1)=O N1(C(C2N(C(c3c(CC)nn(C)c3)=O)CC(C)C2)=O)CC2CC2C2CC12 C1(NC(C2CCSCC2)=O)CCCC(C(=O)NCC2C3CCCC23)C1 C1(CC(=O)NC(c2ccccc2)CNC(c2c[nH]c(=N)o2)=O)CCCN1C=O CC1CCCCC1CC(N1CCC(CF)(NC(=O)CNc2ncccn2)C1)=O N1(C(c2c(C)cnnc2)=O)CC2CCCC(C1)N2C(C12CCC(C)(CC1)CC2)=O c1(CC)cnccc1C(=O)NCC1C(C)CCN1C(=O)Cc1cnccc1C c1(C(=O)NCC2CC(C)N(C(c3cnnc(Cl)c3)=O)C2)cc(Cl)cc(F)c1N c1(C(N2CCC(N(C(=O)C3=NOCC3)CCC)CC2)=O)cn2c(n1)CCC(C)C2 C1(NC(N=S(CC#C)(C)=O)=O)CCOC2(CCC2)C1 C(C(CC1CCCC1)C(=O)NCCCN1CCC1)NC(CSCC=C)=O CC(C)CC(CC(=O)N1CCC(CCN(C)C)C1)NC(=O)CCC(C)(F)F Cc1cnn(C)c1C(N1CC(NC(c2ccc(OCF)cc2)=O)C(O)C1)=O C(=O)(C1c2c[nH]nc2CN1C(=O)CSC(F)F)NCc1cc(OC)ncn1 N1(C(c2cc(OC)ns2)=O)CCC(NC(=O)C=Cc2cccc(F)c2)C(C)(C)C1 c1(C(=O)OC)cc(F)ccc1NC1(CC(=O)NCC2(SC)CCCC2)CCC1 C1(C(=O)NC2(CC)CCN(C(C3SCCCS3)=O)CC2)CCC2CC(C)CN2C1 O=C1NCC2(CCN(c3nnc(-c4cccs4)n3CCCOC(F)F)CC2)N1 CC1(F)CCN(C(C2(C)CN(C(=O)CCn3cccc3)CC2C)=O)CC1 Cn1ccc(C(N2C3CCC(C3)C2CNC(C2CC2c2cccs2)=O)=O)cc1=O Cc1ccn(CC(C)C(=O)NCC2(NC(C3CC(=C4CC4)C3)=O)CCOC2)n1 C1(CC(=O)N(C2CCCC2)CCCNC(c2c(C)n[nH]c2)=O)CC(C)(C)CO1 C1(O)(CC)CCN(C(=O)CC2CC2CNC(=O)C(C2CCCCC2)F)C1 Cc1n[nH]c(C)c1CCC(=O)NCCC1COCCN1C(=O)CN(C)C1CC1 C(=O)(CCC(=O)c1ccc(F)cc1)NC1C(CNC(C(C)(F)F)=O)CCC1 C1(CC)C(NC(=O)CCN2CCCC2)CCCN1C(c1ccc(F)c(F)c1)=O C1(Cn2cc(C(C)(C)SC)nn2)N(C(C23CCCC2C3)=O)CC1(C)C c1(C(N2C3(C#C)CC(C2)C3)C(=O)Nc2cccc(Cl)c2C)c(Cl)cc(Cl)cc1Cl c1(N2C(C)CC(NC(C3CNC(=O)CC3C)=O)C2)c(C#N)c(=O)n(C)c(=O)n1C N1(C(CCNC(=O)OC)=O)CCN(C)C(CNC(c2cc(C3CC3)[nH]n2)=O)C1 C1(NC(c2cnc(C)nc2)=O)CC2CC(NC(C3(CCF)CC3)=O)C2C1 c1(C(=O)OCC)ncc(Br)cc1NC(C1(c2cccs2)CC1C)=O C1(C)(C(N2CC(F)(CC)C2)=O)CCN(C(=O)C#CC2CC2)CC1 N1(C(c2c(S(C)=O)cccc2)=O)CCC(C2CCCN(c3nnns3)C2)CC1 CC1(C)C2CCC1(C(=O)NCC(N1CCN(C(=O)CCn3ccnn3)CC1)=O)CC2 c1(OC)c[nH]c(C(=O)NCCCCCCC(c2cncn2C)C(=O)NC)cc1=O Cc1cccc(C(N2CC(O)CC2C(=O)NCCC(C)C(C)(C)C)=O)c1C C1(c2ccccc2F)(C(=O)NC(C)C(CO)NC(=O)C(C)CO)CCCCC1 C1(NC(C(C)Oc2cccnc2)=O)CC(N=c2nn[nH]n2-c2ccccc2)C1 C1(NC(C(CC)NC(N)=O)=O)CCN(C(=O)C(Cl)=CCl)CCC1(F)F C1(O)(CNC(C2CC(OC)C2)=O)CCCN(C(=O)CCCc2nncn2C)C1 c1(C(C(C)C)NC(C(=O)OC)COC(C)(C)C)ccc2c(c1)OCCO2 CN1CC(C)(C(=O)NCCCNC(=O)Cn2cc(CO)nn2)CCC1=O N1(C(C(C(C)C)O)=O)CCOC2(CCCCC2NC(C2CNC(=O)C2)=O)C1 C1(NC(c2c(C(C)C)ncnc2)=O)CC2CN(C(C3(C#N)CC3)=O)CC2C1 c1(C2C(CNCc3nc(CC)on3)C2)ccc(Br)cc1 C1(C(F)(F)F)(NC(N2CCN(CCOCCO)CC2)=O)CC2CCC1CC2 c1(C(=O)NCC2N(C(CCCc3nnc(C)n3C)=O)CCC2)cccc(O)c1C CCCC(C)CN=c1ccc(S(=O)(=O)N(CC(C)N(C)C)C)c[nH]1 c1(C(=O)NCC(CC)NC(=O)CCC=CBr)cc(N)cc([N+](=O)[O-])c1 CCC(CCC(=O)NCC1(CO)CCN(C(=O)CCCn2ccnc2)C1)OC c1(C(=O)NC23C(CN(C(c4cc(=N)[nH]c(=N)[nH]4)=O)C2)CC3)cccn2cnnc12 C1(CC)CN(C(=O)C(CC2CC2)NC(C2CC(O)CN2C)=O)CCN1C C1(NC(=O)OC(C)(C)C)CCCCC1CNC(C1CN(C(=O)C(N)=O)CCO1)=O N1(C(C2CC(C)N2C(C2CC(O)CN2C)=O)=O)CC2COCC2(C)C1 C(=O)(C(CCCC)C(C)C)NCC(C(=O)NC(C1CCCCC1)C#C)CC1CC1 N1(C(c2cn(CC=C)nn2)=O)CCOC2(CCN(C(C3(CC)CC3)=O)C2)C1 C(=O)(C(C)(C)CF)N(C)CC1C(NC(C(CC)OC)=O)CCC1 c1(C(N2CCC(NC(CCCC)=O)CC2C)=O)ccc(Cl)c(F)c1F CCC(CN=c1ccc(S(=O)(=O)NCCC2CCCS2(=O)=O)c[nH]1)N1CCCC1=O Cc1cccc2[nH]c(=NC3CC(CNC(=O)C4=CCCCO4)C3)sc12 N1(C(=O)NCCn2nnc(C)n2)CCC(OC)C1(C)C C1(C(N2C(C)CC(CNC(c3ccncc3)=O)C2)=O)CC2C=CC1C21CC1 CC1CSCCCN1N1CCCC1.C1(C=O)CCN(CC(F)F)CC1 C1(C(=O)NCCn2cc(C(N3CC(OCC)C3)=O)nn2)OCCC1(C)C N1(C(c2c(CCC)nco2)=O)CCC(F)(F)C(CNC(c2sc(F)cc2C)=O)C1 C1(C(=O)NCC=CC)CCN(C(=O)Cc2cccnc2)C1C N1(C(C)=O)CCCc2cccc(N3CCCC3)c21.Cc1cc(C(=O)C)c(C)[nH]1 N1(C(C2(c3cn(C4CC(COC(C)=O)C4)nn3)CC2)=O)CCOC(C)C1CO CC(C)CC(C)CC(=O)N1CCC(F)C(NC(=O)C(C)(C)c2cscn2)C1 c1(C(=O)NC2C(OC)CN(C(=O)CC(C)N(C)C)C2)cccc(C)c1O N1(C2(C)CC2)N=C(C(=O)NCC2CCN2C(c2cc(C3CC3)[nH]n2)=O)CCC1=O N1(C(C2(SC)CC(C)(C)C2)=O)CC(C(=O)NCC2(O)CCN(C)C2)CC(C)C1 C1(C(=O)NC(CC)CN(C(=O)C=Cc2nccs2)C)CN(C)C(=O)CCO1 CC1C(C(=O)NC2C3CC2N(C(C2(C)CCCC2)=O)C3)CCN1C CCCC(O)(CCC)CC(=O)NCC(C)CN(C(=O)CS(=O)(=O)CC)C c1(SC(C)C)ccccc1C(=O)N(CC(C)NC(c1ccc(COC)cc1)=O)C c1(C(=O)NCC2CN(C(C(=O)NCC)=O)CC23CC3)ccc2nnn(C)c2c1 C1(CC(C)C)(C(=O)NC2CCC(CNC(C3(C#N)CC3)=O)C2)CCNC1=O c1(CN2C(CNC(c3ccc(=NC)[nH]c3)=O)CCC2)cn(C)c2c(Cl)nccc12 c1(C(=O)NC2CCC(NC(COC3(C#C)COC3)=O)C2)cnc(CN(C)C)nc1 N1(C(C2(C=C)CCN(C(=O)CCOC3CCC3)C2)=O)CC(C)OCCC1C N1(C(c2nc(C)sc2)=O)CC2CC(C1)C2C(=O)CC1CCCC1C c1(C2(C)CC2)ccc(C(=O)NCC2CC(F)(F)CN2C(c2cnsn2)=O)cc1F C1(C)(SCc2cnc(C(C)(C)C#N)s2)CC2CC2C1 C(=O)(C(C(C)NC(c1ncccc1Cl)=O)C(C)C)Nc1c(OC)cc(F)cc1 C12(CNC(c3ncn(C)c3)=O)CC1CN(C(=O)CCCC1CCOCC1)C2 C1(c2n(CCOC(C)C)nc(-c3ccccc3)n2)CN2CCC1CC2 C(=O)(CCCC(C)(C)C)N(C1CC1)C.CC1CCCc2n[nH]nc21 c1(C(=O)NCC2CN(C(CC(=O)OC)=O)C2)oc(C2CC2)nc1C(F)F.C1CC1 C=C(C)c1cccc(NC(=O)C(CCC)NC(=O)CC2CC(F)(F)C2)c1 c1(CC)nc(N2CC3C(NC(=O)CC(C)(O)COCC)C3C2)c(F)c(Cl)n1 CC1(C)CCC1C(=O)NCC1(CCNC(c2ccn(C3CC3(F)F)n2)=O)CC1 N1(C(C(CC)SC)=O)C(C)C2CC1C2NC(=O)CNC(c1cnoc1C)=O C1(NC(C2(CC#C)CCCCC2)=O)CC2CCC(C1)N2C(=O)C1=C(C)CCCC1 C1(NC(C2OCCN(C(c3cnn(CC)c3C)=O)C2)=O)=CN=C(O)CN=C1C c1(CC)cccc(C(N2CCOC(CNC(=O)CSCC(C)C)C2)=O)n1 N1(C(c2ncc(OCC)nc2)=O)CCCCC(CNC(C2(F)CC=CC2)=O)C1 C1(NC(C=CC(C)(C)SC)=O)CN(C(=O)C=C2CCN(C)CC2)CC1CN(C)C c1(C(C)(C)C)scnc1C(=O)N(CCNC(C1CCCN1C1CC1)=O)C1CC1 C1(C(=O)NCCCN(C(CC=C)=O)C)CC2(C1)CC(F)C2 C1(OC)CC(NC(c2cncnc2)=O)CN(C(=O)Cn2ncc(Br)n2)C1 C1(N(C(c2c(C)nc[nH]2)=O)C)CCN(C(=O)C(C)Oc2ccc(F)cc2)CC1 C1(=O)CCN=C(NC2CCS(=O)(=O)C2)NCCN1.C1(SC)CC(=O)N(C2CC2)C1 CCCCC#CC(C)(C)NC(C1CC(C)N1C(C1CCC(=O)NC1)=O)=O Cc1cc(=NC(=O)C(=O)N2CC(CNC(c3cncc(F)c3)=O)C(O)C2)[nH]o1 C(CC(O)C(=O)NCC(CC1CCCC1)C(=O)NCC(c1ccccc1)C)SC C1(c2onc(CN(C)C)n2)CN(CC2(C)CSCCO2)CCO1 N1(C(c2cc(C)[nH]c2C)=O)CCCC(CO)(NC(C2CCSC(C)C2)=O)C1 C1(c2n(C)nc(-c3cccc(OC(C)(C)C)c3)n2)CCCC1S(C)(=O)=O C(=O)(C(C(C)C)NC(N)=O)NC(CC(C)NC(C(C1CCCC1)OC)=O)C c1(CN2CC(O)(CNC(C(C(C)C)c3ccccc3)=O)C2)c(F)cccc1F C(=O)(C(O)CCCNC(C1CCOC(C)(C)C1)=O)NCC(C=C)(C)C N1(C(c2cc(C)on2)=O)CCCC(C2CN(C(=O)C(C3CC(F)(F)C3)O)C2)C1 c1(OCC(=O)N(CC(CC)NC(=O)Cc2cncn2C)C)cncc(Br)c1 C1(C(N2CC(c3ccccc3)(NC(C(F)OC)=O)C2)=O)CCN(C)C(C)C1 C1(C(=O)NC2(C)CN(C(C3(CC#C)CCCO3)=O)C2)CC(c2ccccc2)=NO1 C1(C(=O)NCC(C#C)CC)C(C)CCN1C(=O)C=Cc1cocn1 N1(C(=O)Nc2csc(-c3ccc(Cl)cc3)n2)c2ccc(Cl)cc2N2CCC1C2 c1(CC(N2CCC(N(C)Cc3ccc(Cl)nc3)C2)=O)ccnc(O)c1 Cc1cncc(C(=O)NC2CCCC(NC(c3ccccc3Cl)=O)C2)c1 N1(CC)CC(C(N2CCC(C)(NC(=O)C(F)=CCCF)C2)=O)NC1=O c1(OC)ccccc1CCOC(=O)CC1CCCC(C)C1 c1(C(=O)NC2(C)CN(C)C(=O)CC2)cc2n(c1)CCCNC2=O c1(CC(=O)NCC(CNC(C2(CC=C)CCC2)=O)C)ccc(F)c(Br)c1 CC1CC=C(C(=O)NC2CCCCC2NC(=O)COc2ccc(Cl)nc2)CC1 N1(C(c2ccc(N(C)C)cn2)=O)CCCCCC(Nc2ccccc2[N+](=O)[O-])C1 c1(C(C(=O)NC2(c3cn(-c4ccc(OC)cn4)nn3)CC2)=O)ccc(Br)c(F)c1F O=C(N=c1[nH][nH]c2c1CCCC2)C1CCN(C(c2cc(Br)ccn2)=O)CC1 N1(CC(=O)NC2(C)CCN(C(c3c(C)cco3)=O)C2)CCSC2CCCCC12 CCCC(C)(CCC)C(=O)NC1C2CC3C(C2)C13C(=O)N(CC(=O)N(C)C)C C(CCCCC(=O)NCC(CO)NC(=O)CCN1CCC(F)C1)=CC N1(C(C2N(C(c3cc(C)c(C)nn3)=O)CC(O)C2)=O)CC2(CCC1CO)CC2 N1(C(CSCC#C)=O)CCCC(C(C)C(=O)NCC2(CC)CCC2)C1 N1(C(CC2OCCC(C)(C)C2)=O)Cc2ccccc2C(NC(=O)CC2CCC2)C1 c1(C(=O)NCC(CC=C)NC(=O)CC(C)(C)COC(C)=O)ccc2[nH]ccc2c1 N1(C(c2c(C=C)cncc2)=O)CC=C(C(C)(C)C(=O)NCC(C)(O)CC)C1 c1(OC)cc(CNC(Cn2cncn2)C(=O)O)cc(C#N)c1 CC(C)CC(O)C(=O)N1CCOCC1CNC(=O)CCN1CCCCCC1 c1(C(=O)NCCC2CC(OC)CN2C(C2CCOC2)=O)c(F)cc(Cl)cc1F C1(CNC(C(CC=C)C)=O)CC2(CCOCC2)CN1C(=O)C(F)=C1CCCC1 c1(C(N2CCC(C(C)NC(=O)Cn3cc(Cl)cn3)C2)=O)ccc2nc(O)oc2c1 C1(CNC(c2scnc2C(F)(F)F)=O)COCCN1C(=O)CC1(O)CCC1 C1(NC(c2ccn(CC(C)C)n2)=O)CC2(C1)CC2NC(=O)Cc1cccc(Cl)c1 S(=O)(=O)(c1ccc(NC2CCCC3CC23)cc1Br)N1C(C(N)=O)CC(F)C1 c1(C(=O)NC2CC3CN(C(Cc4cc(C)no4)=O)C2C3)ccc(P(C)(C)=O)nc1 N1(C(=O)CC2CCCCO2)CCOCC1NC(CC1CC(NS(C)(=O)=O)C1)=O Cc1cc(Cl)c(Cl)cc1CC(N1CC(NC(c2c(C)cccc2C)=O)C(F)C1)=O C1(C(=O)NC2C(C(=O)NCCCCC(=O)OC)CCC2)OCCCC1(C)C C1(CCOC)CN(C(C2CCCCC(=O)N2)=O)CCN1C(=O)CN1CC(C)C1 c1(C(=O)NC2CC(C)N(C(c3cnc4sccn34)=O)C2)c[nH]c(=N)nc1O C1(N2C(N3CC(C)(C)OC3=O)CCCC2)CCC2(CCNCC2)CO1 c1(CC)noc(C(N2CCOCC2CN(C)C(C2(COC)CCCC2)=O)=O)c1C Cc1cc(C)c(C(=O)NC(C2CC2C(=O)NCc2nn[nH]c2C2CC2)C)s1 CCCCCC(CC)C(=O)NCC(=O)NCC(=O)NC12CC1COC2(C)C C(=O)(C#CC1(C)CC1)NCCC(C)(C)OCCOC(C)C(=O)Nc1ccccc1 CCC(CN(C)C)CC(=O)NCC(C)CNC(c1cnc(OC)c(C)c1)=O C(CCCCC(=O)NC(C)CCN(C)C(c1cn(C2CC2)nn1)=O)=CC CC(C)CC(CC(=O)NC1(CNC(=O)CCc2cc[nH]n2)CCOC1)CC(N)=O C(=O)(C(C)CS(C)(=O)=O)NC1(CNC(c2cn(CC)nc2C(C)C)=O)CCOC1 N1(C(C(C)C#N)=O)CCC(C2(NC(c3cc(C4(C)CC4)ccc3F)=O)CC2)C1 N1(C(CCOCCOCC)=O)CCC2(CCN(C(c3ccc(C#N)[nH]3)=O)C2)C1 N1(c2nnc(CC)o2)C(CNC(=O)C=Cc2cocn2)CC2COCC12 c1(OC(=O)CCN(C(C2CCCO2)=O)C2CC2)ccccc1Cl c1(C(N2CCC(CC=C)(NC(c3cc(C)sc3C)=O)C2)=O)cccc(F)c1F c1(CC)noc(C)c1C(=O)NCC1(F)CC(CNC(C2CC2F)=O)C1 N1(C(c2c(C)nc[nH]2)=O)CC(N(C)C(c2ccnc(C3CC3)c2)=O)C2(CC2)C1 Cc1nc2ccccc2n1CC(=O)NC1CN(C(C2CCSC2)=O)CC1O CC1(C)CC(N=c2[nH]nc(C(F)F)o2)CN(Cc2nc[nH]c3nccc2-3)C1 C(C)(C(=O)N1CC(c2ncccn2)C1)(C1CCC1)NC(COCCN(C)C)=O c1(CNC(N2CCOC(C(C)C)C2)=O)cc(F)cc2c1CCC2 c1(C(=O)NC(C)C(C)NC(=O)C=Cc2ccccc2)ncc(Cl)cc1Cl c1(OC)ncnc(OC)c1C(N1CC(CN(C)C(C2CCCCC2(C)C)=O)C1)=O CP(C)(=O)CC(=O)NCCOCCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O CC1(C=O)CC(c2cc(Cl)cc(Cl)c2)=NO1.C12CCCN(C1=O)CN2 c1(C(=O)NC2CCCC(CNC(c3ccc(C)n3C)=O)C2)cc(F)cc(Cl)c1N c1(CC)cc(C(=O)NCC2CC2C(=O)NC2CC(CC)(CC)C2)on1 C=Cc1ccc(C(=O)NCCC2CC(C(N3CC(OC(=O)N(C)C)C3)=O)C2)cc1 c1(C(N(CC(CN(C(C2C(OC)CC2)=O)C)O)C)=O)cccc(C)c1[N+](=O)[O-] c1(N(CCCC)C(c2csc(-c3ccc(C)cc3)n2)=O)ccc(F)cc1 c1(CNc2c(NC)ccc(F)c2)cc(=O)n2c(n1)CCCC2 c1(OC)cc(C(=O)NC(C2CCN(C(=O)CC#N)CC2)C)cc2c(C)c(C)[nH]c12 CC(C)(C)CCCCNC1(c2nnnn2-c2ccccc2)CCCCCC1 n1(CC(=O)N(C2CCCC2)CCC2CCC(NC(=O)CNC=O)C2)nnc(=O)[nH]1 c1(C(=O)NCCCCCCN(C(=O)CC2CCC(=O)N2)C)ccc([N+](=O)[O-])s1 CC1CC(CC(=O)NC2CCOC2(C)C)CN1C(=O)CC=C(Cl)Cl O=C(NNc1cccc(Br)c1F)c1ccc(SCC(F)(F)F)nn1 C1(CC(=O)NCCNC(C2C=CCCC2)=O)COCCO1 C1(F)(CNC(C(C)O)=O)CCC(CNC(=O)Cn2cc(CO)nn2)C1 C1(CCN(C(=O)CC2(C)CCCO2)C)CCCCN1C(=O)CCCN1CCCC1 C1(C(=O)NC2(C)CC(NC(=O)CC3(O)CCOCC3)C2)CC2C(C1)C2(C)C C1(COC)CCC(NC(=O)CC2CCCN2C(=O)CC2CC(SC)C2)CC1 c1(C(=O)NC)cccc(NC(=O)C(N2CCNC(C)C2)=O)c1Br C1(NC(c2c(C)nc[nH]2)=O)CCCCC1NC(C1CCN(c2ccncc2)C1)=O O=C(NNc1cc(F)c(Br)c(F)c1)NCCc1ncc(C(F)(F)F)cc1Cl C1(CNC(=O)C(O)C2CCC2)CC2CCCCC2N1C(=O)CCC1CCCOC1 c1(C(N2CCCSCC2)=O)cccn2ncnc12 C1(CC=C)(NC(c2cccc(NC3CC3)c2)=O)CCCN(C(=O)C(C)O)C1 N1(C(c2n(CC)nnc2)=O)CCC2CCN(C(c3nnc(C(C)(C)C)s3)=O)C2C1 C1(C2CN(C(C3CC(C)(C)O3)=O)C2)(NC(c2c(C)nc(CC(C)C)o2)=O)CC1 CCCCC(=O)NC1CC(C(F)C(=O)N2CC(C3CCCCO3)C2)C1 C1(NC(C2(COC)CC(=C)C2)=O)CCN(C(=O)CSc2nncs2)CC1CO C1(CNC(CCC2CCN(C)CC2)=O)COC(C)(C)CN1C(=O)CC1CCCO1 C12(CNC(C3CCC4(CC4)C3)=O)CC1CN(C(=O)C=CCO)C2 c1(CC(C(=O)NC(C)CCN(C(=O)CCc2nncn2C)C)O)ccc(Cl)cc1 c1(C(=O)NC2CN(C(C3CCC(C)NC3=O)=O)C2)cn2cc(Cl)cnc2n1 C(=O)(C1CCc2c[nH]nc21)NC(CCC=C)C(=O)Nc1cc(Cl)ccc1O C1(CNC(=O)C(N2CCC(C3CC3)C2)=O)CCC2(CCCCCC2)O1 N1(C(c2c(C)[nH]nc2Cl)=O)CCCC(C)C1CNC(C1CC(=O)NC(=O)C1)=O Cc1cc2c(cc1C)C(C(=O)NCCCCC(C)NC(C1CCCSS1)=O)CO2 C1(C(=O)OC)CCC1(C)C(=O)N(CCCNC(=O)C(C)CC)C1CC1 C1(C(c2nnnn2C2CCC2)NC(c2ncc(C(C)C)s2)C)CCC(C)CC1 C(=O)(C(C)CN(C(=O)C=C(C)C)C)N(C1CCCOC1)CC N1(C(C(C)(C)CO)=O)CCN(c2ncc([N+](=O)[O-])cn2)CC(O)C1 CCCN(C1CC1)N(C)Cc1cnc2ccccc2c1 CC(C)CCCC(C)C(=O)NC(C)CNC(c1cccc2c1OCC2)=O N1(Cc2n(CC)ncn2)CC2CCN(C(=O)CS(=O)(=O)C(C)(C)C)CCC2C1 c1(C(N2CCC(CC)CC2C(N2CCC(C3CC3)C2)=O)=O)cccc2ccccc12 c1(-c2cc(C(=O)NC3CN(C(C(CN(C)CC)O)=O)C3)no2)ccc(OC)cc1 N1(C(C(C=C)CC)=O)CCCC(C)C1CCNC(c1nc(Cl)ccc1N)=O N1(C(c2cccc(C(C)C)n2)=O)CCCC12CCN(C(c1cncs1)=O)CC2 N1(C(C(C(C)(C)C)NC(C)=O)=O)CC2CC(C1)N(C(=O)CCC1OCCO1)C2 Cc1cc(N2CCN(C(C)C(=O)N3CCCC3)CC2)cnc1O N1(C(c2ncn(C(C)(C)C)c2)=O)CCCOC(CNC(C2(C)CC2)=O)C1 N1(C(C(C)CC(F)F)=O)CC2COCCC2(NC(c2ccc(Cl)cc2Cl)=O)C1 C(c1ccsc1)=CC(=O)NCC(CC)NC(C1(N2CCNC2=O)CC1)=O C1(OC)COCCC1CC(=O)Nc1cccc(NC(C2(CO)CCCC2)=O)c1 c1(C(N2CCN(C(C(=O)NC(C)C)=O)C(C)C2C)=O)nnc(O)c2ccccc12 c1(NC(C2CC(O)CCN2Cc2c(F)cccc2F)=O)ncc([N+](=O)[O-])cc1Br C(CN=c1ccc(C(=O)NC2(C(C)C)CCCC2)c[nH]1)NC(=O)OC(C)(C)C C1(NC(COCP(C)(C)=O)=O)CCC2(CCN(C(=O)C3Cc4ccccc43)C2)C1 c1(NC(c2n(CCC)nnn2)c2scnc2Cl)cccc(OC(C)CC)c1 c1(NC(C(=O)NC2CC(F)(CNC(C(C3CC3)OC)=O)C2)=O)cccc(C)c1 c1(N(CCCCN(C(C(CC)NC(N)=O)=O)C)C)ccnc(C(F)(F)F)n1 c1(CC)cccc(F)c1C(N1CCOCC1CCNC(=O)C=Cc1ncc[nH]1)=O N1(C(C(C#C)(C)C)=O)CCCC(C(=O)NCC2(CO)CC3CC3C2)CC1 N1(C(C(CN(C)C)(C)C)=O)CC2(NC(=O)C(C3CCCCCC3)O)CCC1CC2 C(=O)(CCCCCN(C)C(c1nccn1C)=O)NCC(COC)OCC O=C(C(F)CC1CCCC1)NCC=CC(=O)NCC1CCCCS1 c1(C(N2C(CN(C)C(C3CC3c3ccsc3)=O)CC(F)C2)=O)cc2ccncc2[nH]1 Cc1cc(Br)cnc1C(=O)NCCC1CCN(C(C23CC(N(C)C)C2C3)=O)C1 C(CCC1CCC1)(C(=O)NCc1cnn[nH]1)NC(c1ccc(SC)o1)=O CC(C)(C)C1=NOC(C(=O)NC(c2ccccc2F)CNC(=O)C(C)(Cl)Cl)C1 Cc1cccnc1C=CC(N1CCC(NC(=O)CCc2cn(C)cn2)CC1C)=O N1(C(c2c(C)con2)=O)CCn2ncc(-c3cn(CCCCCO)nn3)c2C1 N1(C(c2cc(Cl)cc(Cl)n2)C(=O)NC(CC)(C)C)CCC(C2CCCC2(C)C)C1 CC(C)C(C(=O)NC1(C)CN(C(=O)C(C)(C)O)C1)NS(C)(=O)=O N1(C(C2C=CC(NC(CC3(N(C)C)CC3)=O)C2)=O)CCOCC(CO)C1 C(CCCCC(=O)NC1CCN(C(c2cnc(OC)c(Cl)c2)=O)CC1C)OCC C(=O)(C1=CC2(CCOC2)C1)N1C(C)CC(NC(=O)CC2CC(=O)C2)CC1 C1(C)(CC)C=C(C(=O)NC(C(=O)N(C)CC)C2CCC2)C1 CC1(C#CC(=O)NCC23CC2CN(C(=O)C(c2cc(Cl)cc(Cl)c2)=O)C3)CC1 C1(C(=O)NC(C2CN(C(C(C3C(C)C3C)OC)=O)C2)C)CCCCC1 C1(CC(=O)NCC2(F)CN(C(=O)COCCc3ccccc3)C2)CC=CCC1 C(=O)(CC(CC)C(C)C)NCC(CCCC)NC(c1ccsc1Br)=O N1(C(COC2(C)CCC2)=O)CC2(CC(C(=O)NC3(CN(C)C)CC3)CO2)C1 N1(C(C)=O)CCCC(C)C1CNC(=O)CCc1ncc[nH]1 c1(NC(c2ccc(-c3cc(C)c(O)cc3)c(C)n2)=O)ccc([N+](=O)[O-])c(Cl)c1Cl C1(C(=O)NC2C=CC(CNC(=O)CNC3CCOC3)C2)CC2OC1C1CC21 N12CC3CC1CN3C(=O)C(O)c1cccc(c1)C2=O.c1(CC)nccnc1OC C1(C)(C(N2CCCC(CN(C(C(C(=O)NC)(C)C)=O)C)C2)=O)CCC(C)C1(C)C N1(C(C2C(C=C)CC2)=O)CCN(C(c2ccc(CSCC)cc2)=O)C2(CC2)C1 Cc1ccc(S(=O)(=O)NCc2ncc(CSc3ccccc3)o2)c(C#N)c1 C1(C(N2CCC(C(=O)Nc3cccc(OCC)c3)CC2)=O)CCS(=O)(=O)C(C)C1 N1(C(C2CC(C(=O)OC)C2)=O)CCCC(NC(=O)Cn2ncn(C)c2=O)C1 Cc1cccc2c(=NCCC(C(F)(F)F)Nc3ccccc3)[nH]cnc12 Cc1cccnc1-n1cc(-c2ncccc2C)nn1 C1(CC)CCN(CCNC(c2cn(Cc3csnc3NC)nn2)=O)CC1 N1(C(CC(C)(C)O)=O)CCC2(CCC2)C(NC(C2CCC(=O)NC2)=O)C1 N1(C(=O)Nc2nc(-c3ccc(F)cn3)cs2)CC2CCC(C1)O2 c1(C(N(CC(CN(C(C(CC)F)=O)C)O)C)=O)cc(OC)ccc1F c1(CNC(Cc2cc(C)ns2)=O)cccc(CNC(C2CCS(=O)(=O)N2)=O)c1 c1(C(=O)NC2CN(C(c3c(CC)n(C)nc3)=O)C2)cc(OC)c2c(c1)CC(C)O2 c1(C(=O)NC2C(CNC(CSC)=O)C2)cccnc1C1CC1 C1(C(C(=O)NCC(CC)CO)(C)C)CCCN(C(c2cscc2C)=O)C1 N1(CC(=O)NCCC(=C)CNC(=O)C(C)C(=O)OC)CCc2sccc2C1 C1(C(=O)NCC(COC)(C)CO)CCOCCN1C(=O)Cn1ncnn1 c1(CC(N2C(CCNC(=O)Cc3ccsc3)CCC2)=O)ccccc1O.C(C=C)=CC C(c1ccncc1)=C(C(=O)N(CCN(C(C1(OC)CCOC1)=O)C)C(C)C)C CCCC(C)(O)CC(=O)NC(CC(=O)NCCc1cnc(C)cn1)C1CC1 c1(C(=O)NCC2N(C(C(CC=C)C)=O)CCCC2)c[nH]c2cccc(F)c12 C1(C)(CNC(c2c(C)nn(C)c2)=O)CCC(NC(C2CC2c2cnc[nH]2)=O)CC1 C1(NC(Cc2c(CC)con2)=O)CCS(=O)(=O)C12CN(C(=O)CCC(=O)OC)C2 c1(N2CC(C)C(C)C2)nc(N2CCC3(CCCC3)CC2)nc2c1CSC2 c1(C(CC(=O)O)NC(c2ncc(C(C)=O)s2)=O)ccc(Br)c(C)c1 C12(CNC(CC=C=C)=O)COCCN1C(=O)CN(C(c1cccc(Cl)c1F)=O)C2 N1(C(C2(C)CC=CCC2)=O)CCCC(C(=O)N(C2CC2)C2CC2)CC1 C(=O)(CC(C)(C)F)NCC1C(NC(c2cc(OC)ns2)=O)CCC1 C1(NC(c2csc(Br)c2)=O)CCN(Cc2cc(Br)c[nH]2)CC1F C(=O)(C1CCCc2nc(C)[nH]c21)NC1(C)CN(C(c2cc(C)nn2C2CC2)=O)C1 O=C(CCC1=CCCCC1)NCC1COCC1NC(C1CCCN1C1CC1)=O C1(CNC(N2CCC(n3cc(C(N)=O)nn3)CC2)=O)COC2COCC12 c1(OC)cc(F)cc2[nH]c(NC(N3CC4CN(C5CCC5)CC4C3)=O)cc12 c1(CC(=O)N(CC(CN(C(Cc2nnc(C)o2)=O)C)O)C)ccc(C)c(C)c1 C1(C(N2CCCN(C(c3ccc(C)nc3C)=O)CC2)=O)CC2CSCC(C1)C2 C(=O)(C(O)CC(C)(C)C)NCC(CC=C)NC(=O)CC1CCC2(CC1)CC2 N1(C(c2c(C)nsc2)=O)CC2(C)CN(c3nc4cc(F)ccc4o3)CC2(C)C1 N1(CCCC)CCC(N=c2[nH]c(CCN3CCCC3)nc3c2CCC3)C(F)C1 c1(OC)ccc(CCC(N2CC(C(F)(F)F)C(CNC(=O)CC3CC3)C2)=O)cc1 C(C(C)C(=O)NC1COCC1NC(c1c[nH]nc1C(C)C)=O)OC(C)=O c1(OC)ccc(C(=O)NCC2CN(C(=O)C=CSC)CC2C(F)(F)F)c(C)c1 C12(CNC(COCC)=O)CC1CN(C(C1CCCC1(C)OC)=O)C2 N1(C(CCOC(CC(C)C)C)=O)CC(NC(=O)C=Cc2cc[nH]c2)C2(CCC2)C1 N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)C(C)(COC)COC)CC1C N1(C(c2nc(C)c(C)[nH]2)C)CCC(O)(Cc2cn(C3COCC3O)nn2)CC1 CC1CCCN(C(=O)C=Cc2cnn(C)c2)C1CNC(=O)CCCC#N C(=O)(C(O)CCC(C)C)NC(C(=O)NC(CC=C)CO)CN=[N+]=[N-] C(C(C)(C(=O)NCC1CC(O)CN1C(=O)CC=C(Cl)Cl)OC)OC c1(N2CCC(C=C)CC2)[nH]c(=NCc2c[nH]nc2C2CCCCC2)nc2scnc12 n1(C(N2CC(CC)N(C(=O)CCn3cncn3)CC2)=O)ccc2c(C)cccc12 c1(NC(N(CC(O)C2CC2)C)=O)ccc(N2CCOCC2)nc1C C(=O)(CCCCCCCC1CC1)Nc1cn(CCN(CCCN(C)C2CC2)C)nn1 C1(C2CCN(C(=O)Cn3ccnn3)C2)(NC(C(C)C(C)(F)F)=O)CC1 C1(C(=O)NCC2N(C(CC(n3c(C)cc(C)n3)C)=O)CC2)CCCC1S(C)(=O)=O c1(CC)nn(C)c(CC)c1C(=O)NCC1CCCN1C(=O)CN(C)C(C)C C1(NC(CCOC(C)C)=O)COCC1CNC(=O)CN(C1CCC1)C C1(C(=O)NCc2c(COC)noc2)CN(C(=O)CC(C)(F)F)CC12CC2 C(=O)(C(C)CC(F)F)NCC(CCC)NC(C1(C)CC2(CC2)C1)=O c1(N2CC(NC(CCC(C)SC)=O)(CO)C2)ccnc2ncnn12 CCCCCCCC(=O)NCC1(F)CN(C(=O)CC2CC(F)(F)C2(F)F)C1 CCC(CC(=O)NC1(C)CCN(C(=O)CCn2ccnc2C)C1)C(C)(C)C N1(Cc2ccc(C)o2)CC2CCN(S(=O)(=O)c3ccc(O)cc3)CC2C1 c1(SC)ccc(O)c(C(=O)NCC(CC)N(C)C(c2cccc(C)c2F)=O)c1 Cc1ccc(OCC(N2CCN(C(=O)CC3CC3)C3CC23)=O)c(Br)c1 C1(CC)C(N)CCCN1Cc1ccc(N2CCCC2)o1 CC1CN(C(C2CC(=O)NC(=O)N2)=O)CCCN1C(=O)Cn1cccn1 Cc1n[nH]c(C)c1CCC(=O)NCC1CCCN1C(C1CC1c1cccnc1)=O c1(C(=O)NC2C(NC(COCC(C)(C)C)=O)C2)ccc(OC(F)(F)F)cc1 c1(CNC(=O)NC2CC(CO)C3CC23)nccc(Cl)c1O C(=O)(CS(=O)(=O)C(C)(C)C)NCC1(O)CCN(C(c2ccc(COC)[nH]2)=O)CC1 C1(CC(N2C(C)CC(CNC(C3(C)C(C)CCC3)=O)C2)=O)CN2CCC1CC2 Cc1c(C(=O)NC2CN(C(C3COCC3(C)C)=O)CC2O)cnc2ccccc12 CCC(CNC(=O)CCCCCF)CC(=O)NC(C)CCC(C)(C)C CCCC(C(F)(F)F)NC(C1CCC(C2CC2)N1C(=O)C=CC(=O)OCC)=O Cc1n[nH]c(C)c1C(C)CC(=O)NCC(F)CNC(=O)COCc1ccco1 Cc1ccc(C(=O)NCCC2CN(C(=O)CCCC(C)(F)F)C2)c(N)c1C C12(C(=O)NCC(C)CNC(=O)C(c3ccc(Cl)s3)C)CC3CC1C2C3 Cc1ccc(CC(N2CCN(C)CC2CNC(=O)COCC(F)F)=O)c(F)c1F C(=O)(C(CCSC)N1CCC(F)(c2ccccc2)C1)NCCSC N1(C(C=C(C)Cl)=O)CC2CCC(C1)N(C(c1cncc(F)c1C(F)(F)F)=O)C2 C#CCCCCCCC(=O)N(CC(N1CCC2(CC1)CC2C#N)=O)CC#C C1(NC(COC2CCCC(C)C2)=O)CN(C(=O)CS(N)(=O)=O)C(C)(C)C1 C12CCCN(C1)C(=O)C1N(CC1)C2=O.C(CCCN(C)C)N(CCO)CC CC1(C)CC(CCNC(=O)CN(C(=O)Cc2cccn2C)C(C)(C)C)CO1 c1(C(N2CC(CC)N(C(=O)CCCCCSC)CC2)=O)ncnc2c(C)csc12 CC12CC(NC(C3CC4CCC(C3F)N4C(=O)COC(F)F)=O)(C1)C1(CCC1)O2 c1(C)cn2cccnc2n1.Cn1cnnc1Cn1cc(-c2cnc(C(=O)N)s2)nn1 N1(C(C(COC)(C)O)=O)CC2CC(NC(c3ccc(OC)nc3Cl)=O)CC2C1 N12CCOC(C13CCC3)CNC2=O.C1(C(N)=O)CCCC(C(N)=O)CC1 c1(C(C)C(=O)NCCOCCNC(C2CC2C(F)F)=O)ccc(Br)s1 c1(C(N2C(C)CC(CNC(c3ncc(C)nc3)=O)C2)=O)cc(N)cc(N)c1 C=CCC(CNC(=O)C(c1ccccc1)OC)NC(=O)C(C)(C)C c1(CNC(C(C)OC(C)=O)=O)ccc(C(N2CCC2(C)C(C)C)=O)s1 c1(OC)cnc(C(N2CCCCC2C(C)NC(c2cc(C#N)cs2)=O)=O)nc1 N1(C(c2cncc(Br)c2)C(=O)NCCCSC)CCn2[nH]c(=N)nc2C1 C1(C)(CC)C=C(C(=O)NC2COCC2NC(c2ccc(F)cc2)=O)C1 C1(C(=O)NCC(CC=C)NC(=O)C=C2CCCC2)CCN(c2nncs2)CC1 C(CCC(C)C(=O)NC1CCCC(NC(=O)CCCNS(C)(=O)=O)C1)OC CCC(COC(c1cnn(-c2ccc(C)cc2C)n1)=O)CC(F)F C1(C(N2CC(NC(C(C3CCCC3)OC)=O)C(SC)C2)=O)CS(=O)(=O)CC(=O)N1 S1(=O)(=O)c2ccc(nc2)NCC(C)N1CC.C1(C(=O)NC)CCC(C)CC1 Cc1cc(C(=O)NCC2CC3CC3N2C(=O)CC2(OC(C)C)CC2)n(C)n1 C1(C(=O)NCCCCCCO)(CNC(c2c(CC)ncs2)=O)CC2(CC2)C1 Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(c2sccc2C(F)F)=O)cc(O)n1 C1(C(=O)NCC(C)(CNC(=O)C2=C(C)CC2)OC)CC(C)(C)C(C)(C)C1 Cc1cc(NC(C23CC2CN(Cc2ncccc2F)C3)=O)cc(Br)c1 c1(C(=O)NCC2CC(C)N(C(=O)CCc3cn[nH]c3)C2)csc(N=S(C)(C)=O)n1 c1(-c2nc3nn2CC2(CC2)C3)n[nH]c2ccccc12.N1(OC)CC2C(C1)C2(F)F CP(C)(=O)c1cnc(C(=O)Nc2cc(Br)cc3c2OCCC3=O)nc1 C(C(C)N=c1cccc(S(=O)(=O)NCC(c2ccccc2)(C)C)[nH]1)N(C(C)C)C N1(C(CC(C=C)C)=O)CC2(C1)SCCC2NC(c1cc(C)cnc1OC)=O N1(C(C(C)Oc2ccccc2)=O)CC2CCCC(CNC(=O)CSC(F)F)(C2)C1 N1(C(C2CC(OCC)C2)C(=O)NCCCC2CC2)Cc2ncsc2C1 C1(NC(C2(C)CS(=O)(=O)C2)=O)CCC2(CCCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 C#Cc1cncc(NC(=O)C(CCF)NC(=O)Cc2cn(C)cn2)c1 c1(C(N2CC(C(C)NC(=O)Cn3cnnn3)C2)=O)cccn2c(O)nnc12 CC(C)C(F)C(=O)NCCCC1CCN(C(c2cnn(C(C)(C)C)c2)=O)CC1 c1(C(N(C(C)C(=O)NC(C)CCSC)CCC)=O)nccnc1C C1(NC(C(c2cn(C)nc2)(F)F)=O)CCN(C(=O)C2=CCSC2)C1CC1CC1 C(=O)(CC(O)CC(C)(C)C)N(CCCNC(=O)Cc1cc(C)on1)CCOC C1(NC(c2n(C)ncc2)=O)CCC2CN(c3ccnc(C4CC4)n3)CC2C1 C1(CNC(c2scc(OC)c2)=O)CCCCN(C(=O)Cc2cc(C)cc(F)c2)C1 c1(CC(=O)NCCC2N(C(CC(CC)SC)=O)CCC2)ccc(C2CC2)cc1F c1(C(=O)NC2CCN(C(C(CC)C#N)=O)C2(C)C)cc2c(Cl)ccc(Cl)c2[nH]1 C1(CNC(=O)CCc2ccncn2)COCCN1C(=O)Cc1cnccn1 C(=O)(C1Cc2ccccc21)N(C1CCN(C(c2c[nH]nc2S(N)(=O)=O)=O)C1)C C(=O)(CCC(F)(F)F)NCCC1(C)CCN(C(c2c(C(C)C)ncnc2)=O)C1 C1(NC(CCSC)=O)COC2(C1)CN(C(=O)C(C(F)(F)F)=Cc1ccccc1)C2 N1(C(Cc2ccc(C)o2)=O)CCC(C)N(C(c2n[nH]c3c2COCC3)=O)CC1 c1(C(=O)NCC2(NC(C(C3CCC3)OC)=O)CCC2)ccc(Cl)cc1 Cc1nc2ncc(C(=O)N(C(C)CNC(=O)C(C)Cc3ccccn3)C)cc2o1 c1(C(N2CCC(NC(C3(C)CC3)=O)CC(F)C2)=O)ccc2[nH]nc(Cl)c2c1 N(C(=NCCC1COC(C)(C)OC1)NCC1CC1)CC1C(C(=C)C)CNC1 C1(NC(Cc2ncc(CC)[nH]2)=O)CCCCC1CNC(=O)Cc1cccc(F)c1 c1(NC(N2CCC2C2CCOC2)=O)ccc(F)c(F)c1 C1(C(C(=O)NC2(C(C)NC(c3occc3C3CC3)=O)CCC2)C)CCOCC1 c1(N2CCC3(C(C(=O)NCC4(F)CCC4)C3)CC2)ncc2ccccc2n1 N1(C(c2c(C)n[nH]c2C)=O)CCCC(C(=O)NCc2cccc(Cl)c2)CC1 C1(C2(C=O)CC2)CCCN1C(=O)CC1CCC(C(F)(F)F)O1.N(CCO)(CC)CC c1(C(=O)NCC2N(C(CNC(=O)NC)=O)CC=C2)snc(O)c1Cl C1(OCCNC(CCCOCC)=O)(CNC(=O)Cn2ncnn2)CCOCC1 CN=c1[nH]nc(CC(=O)NC2CC2NC(c2ccc(SC)cc2)=O)s1 C1(O)(CNC(c2c(C)cco2)=O)CCCN(C(C2CCCN(C)C2)=O)C1 C(=O)(C(F)CC(C)C)NC1CCC(NC(c2ocnc2COCCOC)=O)CC1 N1(C(=O)OC(C)(C)C)CCC2(CCOC2)C1.C12COCC1SC2 N1(C(CCC2(C#N)CCC2)=O)CC2CCC2(C(=O)NC2CC(CF)C2)C1 c1(C(=O)NC2(C3CN(C(C4C(C(C)C)C4)=O)C3)CC2)ncccc1N=[N+]=[N-] C1(C(N2C(C(C)Nc3ncccn3)CCC2)=O)CN(C(=O)CC(C)(C)O)CC1C C1(CCNC(C(C)S(N)(=O)=O)=O)CCN(C(=O)Cc2ccn(C)n2)CC1(F)F c1(C(N2CCC(C)(CNC(c3cc(F)c[nH]3)=O)C2)=O)ccc(O)c2c1CCCC2 c1(C(N(C2CCCN(C(CC)=O)C2)C)=O)cccn2c(O)nnc12 C1(C(=O)NCC2(OC)CN(C(C3CC(C)(C)CN3C)=O)C2)CCS(=O)(=O)C(C)C1 C1(C(N2CCCC2(C)CO)=O)(NC(CC(=O)OCC)=O)CC(F)(F)C1 Cc1nc(N2CCOCC2)sc1CC(=O)NC1(CC(F)F)CC1 c1(C(N2CCC(N(C)C(C3CC3C(F)F)=O)CC2)=O)ccn2ccccc12 c1(C(N(C2CCN(C(c3cc(CCC)n(C)n3)=O)C2)C)=O)[nH]cc2c1CCCC2 c1(CC)cc2c(NCC3CCCC3NC(C3(O)CC(C)(C)C3)=O)nc(C)nc2s1 Cc1ccc(F)cc1C(=O)NC(c1nocc1C(=O)NC1CCCCCCC1)C CCCCCCCCCc1nc(CC(N2CCCC(F)(F)CC2)=O)no1 N1(C(CCCn2cc(-c3ccn(CC)n3)nn2)=O)CCC(CO)C1(C)C S(=O)(=O)(c1cc(C#N)ccc1F)NC(CNC1CN(C(=O)OC)C(C(C)C)C1)=O C1(C(=O)NC2C(CNC(C=CCC)=O)CC2)CCOC1(C)C Cc1nc(O)nc(S)c1C(N1CCCC1(C)CNC(=O)Cn1cccc1)=O C1(C(=O)NCC2N(C(CC3CCC(C)NC3=O)=O)CCC2)CC2C=CC1C21CC1 n1(COC)ncc(C)c1C(C(=O)NCC1CCOC1)N(C)Cc1cccc(C)c1 C(=O)(C1=C(Cl)CCC1)NCC1N(C(C2(C#C)CCCC2)=O)CCC1 CCCCC(C)C(=O)NCC(CNC(c1ccc(Br)cc1Cl)=O)CO C12(C(=O)NCC(CNC(C(C(C)C)n3cccc3)=O)C)CC(C)(C1)OC21CCC1 CC1(C)COCC1C(=O)NCc1ccc(C(=O)NCCCCS(C)=O)cc1 c1(N(C(=O)NC(C2CCSCC2)C(=O)OC)Cc2cnn(C)c2)cc(O)ccc1F C1(NC(c2nc(CNC(CCC=CC)=O)oc2C)=O)CCn2cnnc2C1 Cc1cc(F)ccc1S(=O)(=O)C(=O)NCC(C1OCCCO1)(C)C c1(C(=O)NCC(C)NC(C=C(C)c2ccsc2)=O)cc2c(ccn2C)[nH]1 N1(C(CSCC=C)=O)CC2CC2(CNC(C2CC(CC)C2)=O)C1 N1(C(CC#C)=O)CC2CCC2(CCNC(c2ccsc2Cl)=O)C1 C(=O)(C(CO)C(F)(F)F)N(C)CC1CCN(C(c2cncnc2C2CC2)=O)C1 C1(CC(=O)NCC2(CNC(CCc3ccn(C)n3)=O)CCC2)CCOC(C)(C)C1 C1(N(C(C2C(C)C2)=O)C)CCN(C(=O)COCc2nc(C3CC3)no2)C1 c1(C(N(CCC(=O)NCCN(OC)C)C2CC2)=O)cccc(Cl)c1 CCCCC(C)(F)C(=O)N1CC(CCNC(C2CC23CCCC3)=O)(OC)C1 Nc1cc2c(cc1C(=O)NCCCCCNC(=O)CCc1cncnc1)OCO2 N1(C(C2(CC)CCN(C(C3CCN(C)CC3)=O)C2)=O)CCOC2COCC12 C(=O)(C(C)(C)C(=O)N1CCC(CC(=O)NCC2CC3(CC3)C2)C1)OCC c1(C(=O)NCC(CNC(=O)CCC2OCCO2)OC)cccc(C(F)(F)F)c1O N1(C(=O)NC(c2scc(C(=O)OC)n2)C)CCOC(c2cccc(O)c2)C1 N1(C(C(C)(C)OC(C)C)=O)CCCC(CCC(=O)NCC(C)CC2CCC2)C1 C1(NC(CCCNC(=O)C=CC2CCOC2)=O)CCn2ncnc2C1 C(CNC(=O)CCc1nccs1)(C(C)C(C)C)NC(c1ccn(COC)n1)=O Cc1nc(CC(=O)N(CCC(C)NC(C2CCCO2)=O)C)c(Cl)s1 c1(CC)ccnc(C(=O)NC2CC2CNC(C2(C(C)(C)C)CCCCC2)=O)c1 c1(C(=O)NCC(CCC)NC(c2c(C)n[nH]c2C)=O)cc2ccnc(Cl)c2[nH]1 c1(CC(N2CC(C(C)NC(=O)CC3CCC4CC34)C2)=O)c[nH]c2ncccc12 C1(C(=O)NCCC2(O)CCN(C(c3cccnc3O)=O)C2)CN2CCCN1CC2 S(=O)(=O)(c1c(OC)cccc1F)NC1CC(C(N(CCOC)C)=O)C1 CC1CCN(C(c2ccon2)=O)CC1NC(=O)Cn1cc(Br)ccc1=O CCCCCCC(=O)NC(c1ccnn1C)C(N1CC([N+](=O)[O-])C1)=O N1(C(C2C(OCC)CC2)=O)CC2(CCN(C(c3cnc(O)n(C)c3=O)=O)C2)C1 c1(-c2ccc(NCC3CCC(CCCC)O3)s2)ccc2c(OC)cc(=O)oc2c1 C1C(C(=O)OC)NC(=O)N1C1CC1.c1(CCC(=O)NCCCOCC)scnc1C C1(C(=O)NC(c2ccccc2)COCC)CC2CC2N1C(=O)CSC C(=O)(CC1=CCCC1)NC1CCC(NC(C(CC)(O)c2cccc(Cl)c2)=O)CC1 C(=O)(C#CC1(C)COC1)N1CCCC(C)(C(N2CC(C(CC)C)C2)=O)C1 C1(C(C)C)Cc2cc(F)ccc2N(C(c2cc(Cl)ccc2C(F)F)=O)C1 c1(C(N(c2nc(OC)c(C)cn2)C2CNCC2F)=O)cc(F)cc(F)c1OC N1(C(CCOC)=O)CC(CNC(c2cncnc2)=O)(OC)C1 c1(C(=O)NCCC2(C(N(C3CC(OC)C3)C)=O)CC2)cccnc1 C(c1sc(Cl)nc1Cl)=CC(=O)NCC1C2CN(C(C3CN(C(N)=O)C3)=O)CC21 c1(C(N(CCCCNC(=O)C(F)CC2CC2)C)=O)cnc(O)cc1C(F)(F)F c1(OC)cc(O)ccc1NC(c1oc(CNC(=O)C2=CCCC2C)cc1C)=O C(=O)(C1=Cc2ccccc2C1)NC1CC(C(=O)NC2CN(c3ccncc3)C2)C1 Cc1c(C(=O)NC2CCN(C(C3CCC(C)CC3)=O)C2)cnn1CCN(C)C C1(CCNC(c2ncn(C(C)C)c2)=O)COCCN1C(C1CC(C(C)(C)C)C1)=O C12(NC(C3C(C)C3C)=O)CCC1CN(C(=O)CCc1cc(Br)ccc1F)C2 CC1CN(C(=O)CC2CN(Cc3cccc(-n4cncn4)c3)CCO2)CC(=O)N1 C(=O)(C(CC=C(Cl)Cl)c1ccccc1)NC1(C)CCC(O)CC1 C(C)(CC(=O)N1CCC(CC(=O)NCc2ncc(CO)o2)C1)OC C1(C(N2C(CN(C(c3c(C)occ3)=O)C3CC3)CCC2)=O)CCC12CCC2 C(CCCC(=O)N(C1CCN(C(c2cnccc2Br)=O)C1)C)OCC C12(CNC(Cc3cc(COC)on3)=O)CC1CN(C(=O)CCNC(C)=O)C2 c1(C(N2C(CN(C(C(CCC)(C)O)=O)C)CCCC2)=O)ccc([N+](=O)[O-])cc1F n1(CC=C)nnnc1C(CCOC)(C(C)CC)NCc1noc(C2CC2)n1 CCCC(CNC(=O)C(CC)CCOC)C(=O)N1CCC(NC(N)=O)CC1 C(=O)(CCn1cccn1)NCC(C1CCC1)N(C(=O)CNC(c1cc[nH]n1)=O)C c1(NC(c2cncc(NCc3nc(C)c(Br)cc3)c2)=O)cccnc1[N+](=O)[O-] C1(NC(Cc2c(CC)cc(F)cc2)=O)CN(C(=O)C=C2CC2)C2(CCC2)C1 N1(C(CCCNC(=O)OC)=O)CC2CC2(C(N2CCCC2CNC(C)=O)=O)C1 Cc1nn(C)cc1C(=O)NC(c1cn(CC(F)(F)F)nn1)C(=O)NCC1(C)CC1 c1(CC)ncncc1C(=O)NCC12CC1CN(C(=O)C(=Cc1cccs1)C)C2 C(=O)(CCCC(N)=O)NC1(C)CCN(C(Cc2c(C)cco2)=O)C1 C(=O)(C(C(=O)N1CC(CCCCNC(=O)C(F)C(C)C)C1)OC)OCC CC1(NC(C2CC(O)CN2C(=O)COC2CN(C(N)=O)C2)=O)CCC(O)CC1 CCCC(CC)CC(=O)NCCC(F)Cn1cc(-c2ccc(F)cn2)nn1 c1(C(=O)NC2CC(CNC(CC(=C)C)=O)C2(C)C)ccc2cc(O)ccc2n1 N1(C(c2c(CC)ocn2)=O)CCC(F)C(NC(C2(C)CCN(C)CC2)=O)C1 C1(CC=C)(NC(=O)C=Cc2cc[nH]n2)CCCN(C(C2CCC3CC2CO3)=O)C1 N1(C(C2CCCO2)=O)CCCC2CN(Cc3nnc(-c4ccccc4F)s3)CC12 C=CC1CN(C(=O)C(c2cncn2C)O)CC1NC(=O)CN1CCCCC1=O N1(C(c2c(C)nc(C)o2)=O)CCCC(C)(CNC(=O)C(c2ccccc2)F)C1 C1(N(C(=O)CN2CC3CC3C2)C)CN(C(c2cc(C(F)(F)F)nn2C)=O)CC1F CC(C(=O)NCCCCn1cc(COC(F)(F)F)nn1)C(=O)N1CCOCC1 c1(NC(C)=O)ccccc1CC(=O)NC1CC1NC(C1C(C)(C)C1(C)C)=O CCC(C)C(C(=O)N1CC(OC(F)F)C1)NC(=O)Cc1cnsc1 c1(C(=O)N(C2CC2)CC2CCC3CC23)ncccc1NC(=O)CC(C1CC1)C1CC1 c1(COC)cnc(OC)c(C(=O)NC2COCC2NC(C2C=CCCC2)=O)c1 c1(C(C2CCN(C(C=COCC)=O)C2)=O)ccc(O)c(O)c1O CC(C)(C(=O)NC(C1CC2(C1)CC(O)C2)=O)C(=O)N1CCOCC1 C12(C(=O)OC)CC(CC(=O)OCC3CC(O)C3)(C1)C2.C1(C=O)(CO)CCOC1 N1(C(CONC(c2c(C)ocn2)=O)=O)CC=CC1(C)CO CC(c1cccc(Cl)c1)=CC(=O)NC1CN(C(C2CCN(C)C2=O)=O)CC1(C)C C1(NC(c2c(SC)ccs2)=O)CCC2CC1CN2C(=O)CC1(O)CCCOC1 C=CCC(CC=C)C(=O)NC1CCN(C(C2CCOCC2)=O)C12CCC2 C(N=c1nc2ncn(C)c2c(NCCC(C)O)[nH]1)c1cccc(C)c1F C1(C(=O)NC2CC23CC(O)C3)(COC)CCCN1C(=O)C(C)=NOCC#N c1(OC)ccc(C2CSCCN2C(=O)CCCn2cccn2)cc1 C(=O)(CC(C)C(=O)N1CC(C(C)NC(=O)CCc2nc(C3CC3)no2)C1)OCC c1(C(=O)NCC2CC(NC(c3occc3C3CC3)=O)C2)ccc2[nH]nc(O)c2c1 C1(NC(CC(CC)C2CC2)=O)CN(C(c2nnn3c2CSCC3)=O)CC(C)(C)C1 CC1CN(C(c2sccc2Cl)=O)CCC1NC(=O)Cc1cnn(C(F)F)c1 N1(C(C=C(CCC)CCC)=O)CCN(C(c2[nH]ccc2C2CC2)=O)CC12CC2 C1(C)(COC)C=CCN1C(=O)CCC1CCN(C(C2CC=CC(O)C2)=O)C1 CCCCC(C)CCC(=O)NCC1C=CC(NC(c2ccoc2Br)=O)C1 c1(OCCN(C)C)cccc(F)c1.C12COCC1C(=O)NC2 c1(C(=O)NC(C2CCCN(C(c3cscc3C(F)F)=O)C2)C)ccc(=O)n(C)c1 N1(C(C=CCN(CC#C)C)=O)CCC2(CC1)CN(C(=O)C1=CCCC1)CC(C)O2 c1(CNC(C(N2CC(C)SCC2)c2nncn2C)=O)ccc2c(c1)OCCO2 N12CCC(C1)N(CCO)CC(=O)N(CCC)C(C)CC2=O.C(C)(C(=O)NC)OC(C)=O Cn1nnc2cc(C(N3CCCC3(C)CNC(=O)CC3CC4CC4C3)=O)ccc12 c1(C(C)C)ccc(C(N2CCCC(NC(=O)CCC(C)CN(C)C)C2C)=O)c(O)n1 N1(C(C(CN(C)CC)F)=O)CC(Cn2cc(CCC3CCOC3)nn2)CC1CO c1(C(=O)NC2CC(CCNC(CC3CC(=C)C3)=O)C2)conc1C(F)(F)F c1(C(=O)NCCC(C)(C)CNC(C2CCOC2)=O)ccc2ncnn2c1 CC1(CCC(=O)NCC(=O)NCC(=O)NC(N)=O)CN(C(=O)CO)C1 C1(C(=O)NC(c2ccccc2)CNC(C(C)NC(CC)(C)C)=O)CC(C2CC2)C1 C#Cc1cc(C(=O)NC2CCC(C)N(C(=O)C=Cc3nnn(C)n3)C2)ccc1Cl CCC(CC(=O)NCC1(C)CN(C(c2ccc(C)cn2)=O)CCO1)C(F)F C1(C(N(CC(=O)NC(c2cncnc2)C)CC)=O)CCCC(C#N)C1 CC(C)CC(CNC(c1cn[nH]c1)=O)C(=O)NCC1(F)CCOCC1 CC(C(=O)OCC(C)(C)C)C(=O)NNc1nc(Cl)c(C#N)[nH]1 c1(C(=O)NC(CCCC)CNC(=O)CC)[nH]cc2c1CCC2 C(=O)(C(C)(CCC)CCC)N1CCC(N(C(CCC)=O)C)C(C)C1 N1(C(CCC(C)(C)C)=O)CC2CCCN(C(C3CC4C=CCC(C3)C4)=O)C2C1 c1(OC)cccc2c1CN(C(c1cnn(C)c1Cl)C(=O)NC1CCCCC1)C2 C1(CNCC2CC(C(F)F)OC2)CC12CCCCC2 C(c1cnn(C)c1)=C(C(=O)NC1CCC(CNC(c2c(CCC)[nH]cc2)=O)C1)C c1(CCC(C)N(CC(C)C#N)C(=O)NCC(=O)OCC)nc(C)cs1 C(CC1=CCN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC1)NC(C1(C)ON=C(C)C1)=O c1(C(N2CC(C)(C(=O)Nc3c(C)cc(Br)cc3F)C2)=O)cccc2c1cnn2C C1(C(=O)NC2CC(O)(CNC(c3cc(C)[nH]c3C)=O)C2)CCCCC1(C)C C1(CC)CN(C(c2ccccn2)=O)CCC1NC(c1ccc(OC)s1)=O C=C(F)CN=C(NCc1ccnn1C)NC1CCC(F)(F)CC1 NS(=O)(=O)c1c[nH]c(C(=O)OC2CCCC2C#N)c1 c1(N2CCC(C(C)NC(=O)NCC3(C=C)CCC3)C2)ccccc1C c1(OC)ccc(C(=O)N(C2CCCC(NC(=O)CC3CCSCC3)C2)C)c(C)c1 C(C(C)(C)CC(=O)NCC#CC(=O)NCC1CCC2(CC2)CO1)OC C(=O)(C1CCc2c[nH]nc21)NC(CCNC(C(=Cc1ccccc1)CC)=O)C C1(NC(C=C(CNC(CN2CCC(OC)C2)=O)C)=O)CCC(F)(F)CC1 N1(C(c2c(NC(C(C)OCC)=O)cccc2F)=O)CCC2(C(=O)O)CCCC12 CC1CC(NC(=O)C(F)=CC2CC2)CN1C(C12CC(c3ccccc3)(C1)C2)=O C(=O)(N=c1cc(C)n(CCO)[nH]1)C1CCN(C(COC)=O)C1.c1(N)cc(C2CC2)[nH]n1 N1(C(Cc2n(C)nnc2)=O)CC2CCC2(CC(=O)NC2(CC(N)=O)CC2)C1 CC(C(=O)N(C)CCN(C)C(C1CC(N2CCCC2)C1)=O)c1ncco1 c1(C(=O)NCC2(F)CN(C(CCCCNC(N)=O)=O)C2)cc2cc[nH]c2cn1 c1(NC(C)=O)cccc(C(=O)NC(C2CCCCN2C(=O)C(C)C)C)c1 N1(C(C2N(C(C)C)CCC2)=O)CCC2C(C1)CN2C(=O)COc1cnc(Cl)cn1 C(=O)(C1CCc2ccccc21)NCCC1(NC(Cc2cc(C)sc2)=O)CCC1 c1(C(CC(=O)NC2CC(C)(NC(CC(C)SC)=O)C2)C)c[nH]c2ccccc12 c1(C(N(C2CN(C(c3c(CC)n[nH]c3)=O)CC2F)C)=O)cc2cccnc2cn1 C(CCC(O)C(=O)NCC(C)(C)CC(F)F)NC(C(C)c1cccs1)=O c1(C(=O)OCC2CC(C)CC(C)C2)c(F)cc(F)cc1Br Nc1ccc(=NCCOc2cnc3ccccc3c2)[nH]c1 N1(C(Cc2c(C)n(C)cn2)=O)CCCC(C)C1CNC(=O)CCN1CCCC1 c1(C(N(CC(CC)NC(C(C(CC)C)O)=O)C)=O)c(F)cc(C)cc1Br c1(C(=O)OC)cc(C(N2CCC2CNC(C23CCCC2C3(F)F)=O)=O)cc(C)c1 C1(CC)CCCCN1C(C1C(C)CN1C(=O)C=CC(F)F)=O C1(C(=O)NC(CCN(C(CC(C)NC(N)=O)=O)C)(C)C)CCC2CC1C2(C)C c1(C(C(C)C)C(=O)OCc2cnn[nH]2)ccccc1C#N Cc1c(F)ccc(C(N2CC(C3CN(C(C4CC4[N+](=O)[O-])=O)C3)C2)=O)c1C C1(CC=C)(NC(=O)Cn2ccc(C)n2)CCCN(C(c2cnc(O)c(F)c2)=O)C1 CCC(CC(=O)N1CCN(C(c2cc(C)ncn2)=O)C(CS(C)(=O)=O)C1)C(C)C C(=O)(CCCCCCNC(c1cccc(-c2cc(OC)ccn2)c1)=O)OCCC CCC(O)CC(=O)NCc1csc(C(N2CC=CC2)=O)c1 CCC(CNC(=O)CC(C(C)C)NC(=O)CC(C)CCO)(CC)CO C1(C(=O)Nc2ccc(NC(C(CC(C)C)O)=O)cc2)CCn2cnnc2C1 C1(C(N2CC(C)=C(C)CC2)=O)CCN(C(C2(C)CCCOC2)=O)CC1(C)C C=CCC(C(=O)NCCN(C(=O)C(CC)SC)CC(C)O)c1ccccc1 N1(C(C(CC(C)C)C)=O)CCCC(C2(NC(c3ccc(F)cc3)=O)CC2)C1 c1(CCC)c(C(=O)NC23CC2CN(C(c2[nH]c(=N)sc2CC)=O)C3)cnn1CCO c1(CC(F)(F)F)nc(CS(=O)(=O)Cc2ccccc2)n(-c2ccccc2)n1 C(C(CC(=O)N(C)Cc1cn[nH]c1)NC(=O)CN1CCCC1C)OC CC1CCCn2cc(C(=O)NCC3CC(NC(=O)CCCCCF)C3)nc21 C1(F)(C(N(CC(C)NC(=O)C(c2ccc(Cl)cc2)(C)O)C)=O)C(C)(C)C1(C)C C(CCC)(C(=O)NC1(CNC(=O)CC(C)c2cnn(C)c2)CC1)=CCC N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3COCCO3)=O)CC2)C1 c1(C(=O)NC2CCN(C(CSCCCC)=O)C(C)C2)cccc2cccnc12 Cc1nc(C(=O)N(CCC#N)CC2CCCC2(C)C)nn1-c1nc[nH]n1 C1(C(=O)NC23CC(C)(C2)C3)(CC)CCCN(C(=O)CC2CCCOC2)C1 C(CN=C(NCC(C)C#N)NCc1cncnc1)c1ccc(OC(C)C)cc1 C(=O)(CCCCCc1cccc(OC)c1)NCC(CCNC(CCCC)=O)OC c1(C(=O)NC(CC)(C)CNC(C2CCCCO2)=O)cc2c(cc1C)OCO2 C(C)(C)(CCC(=O)NCCN(CC(F)F)C)OC.c12cc(C)c(o1)c(=O)[nH]2 C(=O)(CC(F)(F)C(F)F)N(CCCNC(=O)CCC(F)(F)F)CC c1(OC)cccc(C(=O)N(CC(C)C(=O)N(C)C(c2nc(C)no2)C)C)c1 C(=O)(C1=CC2(CCN(C(C(=O)NCC(C)CC(F)(F)F)C(C)C)C2)C1)OC c1(CCC(=O)NC2CN(C(CSCC#C)=O)CC(O)C2)c(C)nc(SC)nc1O C1(SCCC(=O)NC2(O)COC2)CCCN(C(=O)C=CCn2cncn2)C1 c1(CN(CCN(C(CC2ON=C(CC)C2)=O)C)C)ccnc2ccccc12 CCC(CC(=O)N1CCC(C(=O)NCC(F)C(C)(C)O)(CC)C1)CC(C)C c1(N(C(c2nc(CCCC)sc2)C(=O)NCCSC)C)cccc(Cl)c1 N1(C(C2(C#C)CN(C(=O)C(O)CCSC)C2)=O)CCC(CO)C(O)C1 Cc1sc(Cl)cc1C(C(=O)NCCCOCC1CC1)N(CC(C)C#N)C c1(CC)ccc(O)c(C(=O)N(C)CC2CCCN(C(=O)C(=O)NCC(F)F)C2)c1 c1(C(=O)OC)cc(-c2cncc(-c3nccn3CCCCCO)c2)ccc1O c1(C(=O)NC2(CC(=O)Nc3ccc(Cl)nc3Cl)CCC2)ccc(F)c(Br)c1 C1(OC)CCN(C(=O)CCC(C)(C)C)C(c2cn(C3CCCC3)nn2)C1 C(=O)(CCC(F)(F)C(F)(F)F)NCC1N(C(=O)C(O)CC2CC2)CCN(C)C1 N1(C(c2nnc(C)s2)=O)C2CCC1CC(CNC(C1CCSCC1)=O)C2 C1(CN(C(C(CC)N(C)C)=O)C)CCCN(C(=O)C(CO)N(C)C)C1 C=CCCC(C(=O)NC1CCOC1)NC(=O)CC1(C)CC1 N1(C(CSC(C)C)=O)CC(C)CN(C(c2ccc(F)cc2Cl)=O)C(C)C1 C1(C(N2CC(F)(CNC(c3cc(CCCO)on3)=O)C2)=O)CN2CCC1CC2 C(=O)(CCCCC(C)C)NC1CCN(C(c2ccc(C)cc2Cl)=O)C1C(C)C C1(CC=C)(NC(c2cnc(N(C)C)cn2)=O)CCCN(C(c2cnc[nH]2)=O)C1 CC(C)CC(C)(C)NC(=O)C=CC(C)NC(C1CCCCO1)=O Cc1ccncc1-n1cc(C2CCN(C(C3CCC(C(N)=O)CC3)=O)C2)nn1 C1(NC(C(C2CCN(C(=O)C3=CCCOC3)CC2)C)=O)CC2(CCCO2)C1 Cc1cccc2nc(C(=O)NCC3COC(CNC(=O)C4=NOCC4)C3)cn12 C1(OC)CC(C(=O)N(C)C(c2cnn(C)c2)C)N(C(=O)C(CO)NC(N)=O)C1 C1(O)(C(C(=O)NCc2c(C(C)C)noc2)NC(=O)C(C)OC2CC2)CCCCC1 c1(CN(C(C(C)OCC(F)(F)F)=O)C)ccccc1CNC(=O)CCNC(N)=O C1(CC)(NC(C2C(C(=O)OCC)C2)=O)CCCN(C(=O)CCCN(C)C(C)=O)C1 Cc1cc(C)c(C(N2CCC3CC23C(=O)NCc2nccn2C(C)C)=O)cn1 c1(C(N2C(COC)(CNC(=O)CNS(N)(=O)=O)CCC2)=O)ccc(F)c(O)c1 c1(NC(=O)NC2CC3(C(=O)OC(C)(C)C)C2C3)cc(O)nn1-c1ccccc1 C1(C#CC(=O)N2CCC(CO)C(NC(c3ccc(F)c(Cl)c3)=O)C2)(CC)COC1 c1(C(N2CCCN(C(C=C(COC)C)=O)C(CO)C2)=O)ccc2nc(O)[nH]c2c1 c1(C(=O)NC2CC(CNC(c3cccs3)=O)C2)c(F)c(F)cc(F)c1F N1(C(C(C)NC(c2ccccc2)=O)=O)CC2(CCCO2)C1 N1(C(CC2(C)CCC(=O)C2)=O)CCCC(O)(c2cn(C3CC3)nn2)CC1 Cc1cc(C(N2CCCC2C(=O)Nc2cccc(F)c2O)=O)ccc1F c1(C(N2CCC(O)(C(C)NC(=O)C(O)C3CCC3)CC2)=O)ccn2c1CSCC2 c1(CN(C(=O)NC(C2(n3ccnn3)CC2)C)C)ccncc1Cl C(CC(=O)N1CC(C(=O)NC2(CN(C)C)CCC2)C1)N(C)CCO n1(CC)nc(C)c(C(N2CCOC(C)C2c2nc(C)no2)=O)c1C(F)(F)Cl C1(C#N)(C(=O)NC(CC)CNC(c2cnc(C3CC3)o2)=O)CCOCC1 N(C(=NCCC1(CCO)CCOCC1)NC(C)C1CC1)C1C(C)C1C C1(C(=O)OC)CC(C)N1C(=O)CC1(NC(=O)Cc2cnn(CO)c2)CCC1 C1(=O)CCCCCn2cc(nn2)-c2cccnc2N1.c1(CCN)ccccc1 N1(C(C(c2ccsc2)CCNC=O)=O)CCCCC1CNC(=O)CCC1(C)CC1 C1(C(C)NC(=O)C2=CCC2)CN(C(c2cc(C3CC3)cs2)=O)CCO1 c1(C(=O)N(C(C2COCCN2CCO)=O)CCc2ccccc2)cc(I)ccc1Cl C(=O)(C(F)CC(C)(C)NC(c1cn(C)c(C)n1)=O)NC(CC=C)CC C(CC(C(=O)Nc1cccc(Cl)c1)NC(c1n[nH]c(C)c1Cl)=O)=CC c1(CN2C(C)(C(=O)Nc3ncc(Br)nc3I)CC2)c(F)cc([N+](=O)[O-])cc1F c1(C(=O)NCC2CN(C(C3(CC)CCC3)=O)C2)ccc2nc(O)oc2c1 c1(C2C(C)CCO2)c(Oc2cccc(Cl)c2)ccc2ccccc12 c1(C(N(C)CCN(c2nccc(CO)n2)C)=O)ccc(C(=O)OC)c(F)c1 c1(CCC)c(C(N2CCCC2C(C)(C)CNC(=O)CC2CCOC2)=O)nnn1C CCCC(C(=O)N1CCOCC1)NC(C1(CC2CC2)CCC1)=O C1(CNC(C2C(C)CCN2C(=O)CC2CC3(CCC3)C2)=O)CC(C2CC2)=NO1 Cc1cccc(C(=O)Nc2ccsc2C(N2CCOCC2C(C)C)=O)c1C Cc1ccc(Br)cc1C(N1CCCC(C(=O)NCCc2cscn2)C1)=O C(=O)(C#CC(C)(C)O)NC(C(C)NC(c1cn(C(C)C)nc1)=O)C(C)C c1(C(=O)NC2(CC=C)CCN(C(C3CCN3CC)=O)C2)coc2c1CCCC2 N1(C(Cn2ccc(C)n2)=O)CCC2(CC1)CCN(c1ncnn3ccc(Br)c13)C2 c1(C(C(=O)NC2CN(C(c3occ(C)c3)=O)CC2F)C)ccc(F)c(F)c1 CCC(CC)C(C)C(=O)N(C)CCNC(c1cc2c(s1)COCC2)=O N1(C(C(C)(CO)NC(C)=O)=O)CCN(C(C2CC(O)CN2C)=O)CC(C)(C)C1 C(=O)(C(COC)NC)NCCN1CCC(C(=O)OCC)C1 c1(C(N(CCN(C(CC(COC)C)=O)C(C)C)C)=O)cc(Br)ccc1OC N1(C(=O)OC(C)(C)C)CCC(F)(CNC(C2CC(CCO)C2)=O)C1 N1(C(C2(C)CCCNS2(=O)=O)=O)CCn2c(CNCC3CC(OC)C3)nnc2C1 c1(C(=O)NC(CCN(C(C(CC)OC)=O)C)C)ccc(C#CC2CC2)cc1 CC1CN(C(=O)CCOC2CC2)CC1CNC(c1csc(C(F)F)n1)=O n1(CC(=O)OCC)c(N2CCC(C)C2)nnc1-c1cc(Br)no1 N1(C(CN(C)CC)=O)CCC2(CC1)CC(C)N(C(C1CC3C=CC1CC3)=O)C2 C(=O)(CCC(C)CCCC)N1CC(NC(CCCOCC=C)=O)C(C(F)(F)F)C1 c1(C(=O)NC2C(C)N(C(c3ccc[n+]([O-])c3)=O)CC2)cncc2c(O)nccc12 CN1C(=O)CC(NC(=O)NC2CCC23CCCC3)C1c1ccc(F)c(F)c1 CC1(C)CN(C(C2CCC(C(F)(F)F)C2)=O)C(C)(C)C1O N1(C(c2ccc(OC(C)C)cc2)=O)CC2(CCC2NC(=O)C=C2CCCCC2)C1 c1(C(N2CC(CNC(CCC(C)SC)=O)C(N(C)C)C2)=O)ccc(CO)c(F)c1 C#CCCCC(C)C(=O)NC(CCC1CCC1)C(=O)NCC(C#N)CC c1(C(=O)NC(CCNC(C(C)=C2CC2)=O)Cc2ccccc2)c(Br)ncn1C CC(CC(=O)NC1CN2CCC1CC2)C(C)(C)NC(C1C=CC=CC=C1)=O Cc1cc(C(N2CC(CNC(C3(C(F)F)CCOCC3)=O)C3CC23)=O)c(C)n1C Cn1cc(C(N2C3CCC2CN(C(=O)CCn2cnnn2)C3)=O)cc1S(N)(=O)=O c1(C(N2C(CNC(CCn3c(C(C)C)ncc3)=O)CC2)=O)nn(C)cc1N N1(C(C2(CC)CNC(=O)C2)=O)CC2(CC(C(N3CC(=O)NC(C)C3)=O)CO2)C1 c1(NC(=O)OC(C)(C)C)ccc2c(c1)C(=O)CC(NC(c1cnco1)=O)C2 C1(NC(C(c2nc(C)sc2)=O)=O)CN(C(=O)C(C)(C)C)CC(C)(C)C1.C1(C(=O)N)CC1 c1(OCC2CCN(C(C3C(OC)CCC3)=O)CC2)cccc(F)c1[N+](=O)[O-] C1(CNC(C(CCCC)=O)=O)CN(C(c2cc3sccc3s2)=O)CCC1(F)F C1(CC)C(C(=O)NC2(CO)CC(O)C2)CCCN1C(=O)C(C)COC c1(OCCC)ccc(C(=O)NCC2CCC(C)CN2C(=O)CS(N)(=O)=O)cc1N C1(CNC(c2cnc(SC)[nH]2)=O)CCN(C(=O)C(F)(F)CO)CC1C C(=O)(C(C)(O)C(F)(F)F)N1CCC(OC)(CNC(C23CCCC2C3)=O)CC1 CC(C)CCCCC(=O)N(C)CC1CN(C(C2CCC3CCC2O3)=O)CCO1 C1(C)(C(=O)NC(CC)CN(C)C(c2csc(C(C)C)n2)=O)CC2(CCC2)C1 N1(C(c2cncc(SC)c2)=O)CCC2(CCC2NC(=O)Cn2nnc(C)n2)CC1 c1(N2CCCN(Cc3cc(O)c(Cl)cc3)CC2)ncnc2[nH]ccc12 C#CC1(C(=O)NC2CC(=O)N(C)C2=O)CCN(C(c2c[nH]c(C)c2)=O)C1 C(=O)(C(C(C)C)N(CC(C)NC(C1(C)CCCC1)=O)CC)NCC N1(C(C23CC(COC)(OC2)C3)=O)CCCN(C(c2cnns2)=O)C(C)C1 C(=O)(C(CC(C)C)n1ccnc1)N(CCNC(c1c(C)nc(Br)o1)=O)C1CC1 c1(C(N2CCC(CNC(c3c(COC)ncs3)=O)C2)=O)cc([N+](=O)[O-])ccc1C c1(C(N(CC(CNC(C2CC=C(C)CC2)=O)C)C)=O)coc2c1COC2 C12(C(N3C(C(=O)NCCN(CCC)C(C)=O)CCC3)=O)CCCC1CCC2 C1(NCc2ccccc2)C(C)CCCN1C(CSc1cccc(C)c1)=O N1(C(C(c2cn(C)nn2)NC(C=C(C)C(C)(C)C)=O)=O)CCC2(C1)CN(C)C2 C1(C2CCC2)(C(N2CC(O)(CNC(C(c3ccccc3)OC)=O)C2)=O)CC1(F)F c1(OC)ccc(Cl)c(CC(=O)NCC(C2CCC2)NC(C2CC2F)=O)c1 Cc1cccc(CN(CC(=O)NC(C)C(C)NC(=O)COC2CCCC2)C)c1 C(=O)(C1=NOC(C)C1C)N1C(CC)C(NC(c2ccnn2C(C)C)=O)CC1 c1(-c2cccc(C)c2)cnc(Cl)c(C(N2CC(O)C(O)C2c2ccccc2)=O)c1 C1(CC(=O)NC(C2(O)CCN(C(C3CSCCS3)=O)C2)C)CCC(C)(C)CC1 C#CC(C(C)(C)C)NC(=O)CC1(NC(=O)CCOCC2CC2)CCCCC1 c1(NCC2(OCC)CCOC2)cc(=NCCc2nc[nH]c2Br)[nH]c(CC)n1 C#CCC(O)C(=O)NC1CC1CNC(=O)Cc1csc(-c2ccc(Cl)cc2)n1 CCC1=C(C(=O)NC2CCC(CCC(=O)NCC3CC(C)(O)C3)C2)CCCO1 c1(CC)c(N2CC(CCOC)(OC)C2)ncnc1Cl.c12cccc(c1)CNC2=O C#Cc1cc(C(=O)NCC2(C)CCCN2C(c2ccc(=O)n(C)c2)=O)cc(F)c1 Nc1cccn(CC(=O)NC2CCCC(NC(=O)C=CSCc3ccco3)C2)c1=O C1(CNC(C(C)OCCOCC)=O)CCC(C(N2CCC(F)(CF)C2)=O)CC1 N1(C(CC2CC(=C)C2)=O)CCC=C(C(=O)N2CCCC(N(C)C)CC2)C1 c1(C(=O)NC(CNC(C(CC)(C)OC)=O)C)ccc(C(F)(F)F)c(F)c1 C1(C(N(C(CNC(=O)CCCCO)C2CC2)C)=O)CC(=O)NC1(C)C N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)CC2CC3CCC2O3)C2(CCC2)C1 C1(C(=O)NCC(N(C(=O)CC2CS(=O)(=O)C2)C)C2CC2)Cc2n[nH]cc2C(=O)N1 C1(CC)CCC(N=c2nc(O)c3c(ncn3C)[nH]2)C1 CC1CN(C(=O)C(F)C(C)(C)O)CCCN1C(c1cc(Cl)ncc1N)=O CCCC(C)CC(=O)NCC(C1CCCCC1)NC(C12CC(C1)C(C)O2)=O N1(C(CSC)=O)CC2(CCC2CNC(=O)CSc2cccs2)C1 c1(OC)cncc(C(N2CC=CC2CNC(=O)CCOCC(F)(F)F)=O)c1 S(=O)(=O)(c1cccc2c1OCCCO2)NC(c1ccc(=NC)[nH]c1)=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC1CC1C(=O)NCC(COC)CO Cn1cc(C(=O)NC(CNC(C2(S(C)(=O)=O)CCC2)=O)CO)n(C)c1=O c1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)cc(S(N)(=O)=O)co1 c1(C(N2C(COC)C=CC2)=O)n[nH]c2cccc(-c3cnoc3C)c12 N1(C(c2c(C3(C)CC3)cccc2)=O)CCN(C(C23CCCC(C2)OC3)=O)C(CO)C1 CC1=NOC2(C1)CC(C(N1CCC(NC(=O)Cc3cncc(C)c3)C1(C)C)=O)C2 c1(C(=O)NCC(CC)NC(=O)C(F)(F)C2(O)CCC2)ccc(COC)s1 C1(NC(CCOC)=O)CCCC1NC(=O)COCC1CCC1 Cc1cc(C)c(C(=O)NCC(C2CCCN2C(=O)COC(F)(F)F)(C)C)c(O)n1 c1(C(=O)NC2C(NC(CCc3cc(C)on3)=O)COC2)cnc2[nH]ncc2c1 CCC(COC)C(=O)NC1CCCC1CC(=O)NCC1CC(C(C)C)C1 CC(C)(CO)CC(O)CNC(c1ccccc1N1CCCCC1)CCO Cc1cc(C(=O)N(C2CCCN(C(=O)C(N3CCNC3=O)C)C2)CCF)n(C)n1 Cc1ncc(C(=O)NC2CC(C(N3CCC(CC(N)=O)C3)=O)C2)cn1 N1(C(c2c(CC)nc(C)s2)=O)CCN(C(=O)C(COC)N(C)C)CC(C)(C)C1 CC(C)C(C(=O)NCC(C)CNC(c1ccon1)=O)NS(N)(=O)=O N1(C(Cn2c(C)ncc2)=O)CC(C)N(C(c2ns[nH]c2=O)=O)CC1C N1(C(C=CCCC)=O)CCN(C(=O)CCN(C(=O)C(CCOC)OC)CC)CC1 c1(CN2CC(C(=O)NCCn3c(C)ncc3)SCC2)cc(F)ccc1Br CC1(CNC(=O)CCN2CCOCC2)CCN(C(c2cnc(C3CC3)s2)=O)C1 c1(C(=O)NC(CNC(=O)OCC)C)cccc(NC(C2CC=CCC2)=O)c1 C1(N(C(=O)Cn2cc(Cl)cn2)C)CN(C(C2CCCCC2(C)C)=O)CCC1O N1(C(Cn2c(C)ccn2)=O)CC(NC(c2ccc(C3(C)CC3)cc2)=O)CC1C C(N=c1nc(N(C)CCc2nccs2)c2sccc2[nH]1)c1c(OC)c(Cl)ccc1 C(CC(=O)NCC1(C)CCN(C(c2ccc(SC)cc2)=O)C1)(C(C)C)OCC C1(C(C)C)CN(C(=O)CC(C)c2ccccc2)CCN1C(=O)C1=COCCO1 N1(C(CCc2cc(C)on2)=O)CCC(C)(CNC(=O)Cc2ccc(Br)cn2)C1 n1(CCC)ncc(C(=O)NCC2CN(C(c3cc(F)cs3)=O)C2)c1C C(=O)(C1=NN(C)C(=O)CC1)N1C(CC)C(NC(c2cncn(C)c2=O)=O)CCC1 c1(C(=O)NCCCNC(c2[nH]cc(C(=O)OC)c2)=O)cnnc2ccccc12 c1(COC)ccc(NCc2ccccc2)c(C2(C)CC2N2CCCC(CN)C2)c1 N1(C(c2c(N)cnc(Cl)c2)=O)CC2CCCN(C(c3cnn[nH]3)=O)C2C1 C1(CC(=O)NCC2=C(C)CCC2)N(C(C2CCN(C)C2C)=O)CCC1(C)C C1(C(=O)NC2CCCC2C(=O)NC2CCN(CCO)CC2)CCS(=O)CC1 N1(C(=O)NCC2(c3ccc(C#N)c(Cl)c3)CCCCC2)CCN2CCCC2C1 CC(Cc1ccccc1)C(=O)NCCC(C)(C)NC(c1cc(C(N)=O)no1)=O c1(C(N2CCC(C(=O)Nc3c(C)ccc(O)c3)C2(C)C)=O)c[nH]c2cccnc12 CC(F)(F)C(C)(C)CNC(=O)C(=O)N(CCO)CC1CCC(=O)N1c1ccccc1 CCCC(CCC)=CC(=O)N(CCNC(=O)Cn1nccn1)C1CC1 CC1(C)CCCN(S(=O)(=O)N2CCC(F)(F)CC2c2ccccc2)C1 CC1CCC(CNC(c2nccnc2-n2ccnc2)=O)N(C(=O)COC(F)F)C1 C1(c2n(C3(C)CC3)nnn2)(NCC23COC(CF)(C2)C3)CCOC2(CC2)C1 O=C(C#CC1CCCO1)NCC1CN(C(=O)C2=CCCS2)CC12CCC2 C(CCCCC(=O)NC(C1(O)CCN(C(C2CC(SC)C2)=O)C1)C)SC C(=O)(C(CC1CCOCC1)NC(=O)CC1CC1CC)N(CC=C)CC1CCCC1 C(=O)(CC(C(F)(F)F)N(C)C(c1csc(O)n1)=O)NCC(COC)OC N1(C(c2cc(Cl)ncc2Cl)=O)CCCC2C1CCN2c1ncnc2cc(Br)sc12 C1(C(C)C)CN(C(=O)CC2(C)CC(F)(F)C2)CCN1C(C1CC(=O)NC1(C)C)=O C1(NC(CSCCCC)=O)CCC12CN(C(c1ccco1)=O)C2 c1(NC(C2C(C)(NC(=O)OC(C)(C)C)CCCC2)=O)ccc2c(c1)C(O)CC2 c1(NC(C(CCC#C)NC(=O)Cc2nc(=N)[nH][nH]2)=O)cccc2c1CCO2 N1(C(c2ccc(F)cc2Cl)c2nn[nH]n2)C2CCCC1CC(O)C2 c1(NC(C(N2C(CC(=O)OC)CC(F)(F)C2)=O)=O)cnc2ccccc2c1Br Cc1cc2ncn(CC(=O)NCC(C)N(C(=O)C=CCCC(C)C)C)c2cc1C N1(C(c2c(C(C)C)nns2)=O)CC2CCC1CN2C(c1cnc2ncccn12)=O C1(C(=O)NC(CC#C)CC#C)CCN(C(=O)C(CC(=C)C)OC)C12CCC2 N1(C(c2cc(CNC(CCC(=O)NCC)=O)no2)=O)CCC(CO)C(C)C1 N1(C(C=NOC)=O)CCC12CN(C(C1CCN(C3CC3)CC1)=O)C2.c1(C)ccccc1 C#CC1CCN(C(=O)C(F)C2CC(NC(C3(N(C)C)CC3)=O)C2)C1 C(=O)(C(CCF)NC(C1C=CCN(C(c2oc(C)cc2C)=O)C1)=O)OC C(=O)(CC(C)C(C)C(C)C)N1CCC(CNC(c2c(OC)scc2)=O)C(C)C1 c1(C(CN(C(N2C(Cn3ccc(C)n3)CCCC2)=O)CCO)=O)c(C)nn(C)c1F C1(CNC(CN(c2ccncc2)C)=O)CC(F)(CNC(C23CCC2C3)=O)C1 c1(OC)ccc(C)c(C(=O)N(C(CNC(c2cc(O)no2)=O)C2CC2)C)c1 C(=O)(C1=CNC2=NCCCN12)N1CC(CN(C(=O)C=CC(F)(F)F)C)OCC1 c1(C(=O)NC(CN(C(=O)C(C)CC(N)=O)CC)C)cc(Br)c2c(c1)CCO2 CCC(CCCC(=O)NCCCC(C)(C)C)NC(c1cnn(C)c1OC)=O C1(O)(CNC(C=CC(C)C)=O)CCN(C(C2CCN(CC(C)C)C2)=O)C1 C1(OC)CC(NC(=O)CCc2cc(C)on2)CN(C(C2CC(C)(O)C2)=O)C1 N1(C(C=C(C)C2CC2)=O)CCOC2(CCC(N=c3nc(C(C)C)[nH]s3)CC2)C1 C(C(C(C)(C)C)NC(=O)CC(C)O)NC(C1N(CC)CCC1)=O C1(C(=O)NCC(C)=CC(=O)NCC2CCC(=O)O2)CC12CCCC2 Cc1ccc2cc(C(=O)NC(C)(C)CN(C(=O)C=Cc3cn(C)nn3)C)[nH]c2c1 n1(CC(=O)NC(CNC(c2cnc(CC(C)C)[nH]2)=O)C)ccc(O)nc1=O c1(C(=O)NCC(CC(C)C)NC(C=C(COC)C)=O)ccc2c(c1)CCCS2 c1(C(N(c2ccoc2)CCNC(c2n(C(CC)C)ncc2)=O)=O)ccc(Cl)nc1 C1(c2n(C)nnn2)(NCCCSCCO)CC2(CCCOC2)C1 CCCCC(CC)C(=O)NCc1occc1C(=O)NCC(CC)n1cccn1 c1(CC(N2CC3C(CNC(c4c(C)ncnc4)=O)C3C2)=O)cccc2c1OCO2 N1(C(Cc2ccc(SC)cc2)=O)CCN(C(=O)C2=C(Cl)CCOC2)CC(O)C1 C(=O)(C1CCCn2c(Br)cnc21)NCCCN(C(C(C)O)=O)C1CC1 N#CC1CN(C(c2cncc(F)c2)=O)CCN1C(c1c(I)ccnc1Cl)=O C=C1c2ccccc2C(=O)N1C(C)C(N1CCC(C)S(=O)(=O)CC1)=O N1(C(C=CCN(C)C)=O)CCN(C2CCN(C(c3csnn3)=O)C2)CC1 CCCCCCC(C)C(=O)NCC1CCC1NC(C1(CC)CCC1)=O C(=O)(C(F)C(C)(F)F)NCC1(COC)CCCN1C(c1cccc(C(C)C)n1)=O O=C(CC(C1CCCCC1)c1ccon1)N(C1CC1)CC1CCC(=O)NC1 c1(SC(CC)C(=O)NC(c2ccc(C(C)C)cc2)CO)ccc(Br)cc1 C1(NC(C(CC=CC)NC(c2ccn(C(F)F)n2)=O)=O)CCC(=O)NC1C C1(NC(C2(C(C)C)CCCN2C(C2CCCOCC2)=O)=O)CC2(C1)CC(C#N)C2 c1(C(=O)NCCn2cc(C(c3ccccc3)(C)C)nn2)cnc2c(Cl)cccn12 C1(NC(CSc2ccc(OCC)cc2)=O)CCN(C(=O)CC(=O)OC)CC1F C1(COC)(NC(c2ccc(OC)s2)=O)CCCN(C(=O)C(C)SC)C1 C1(NC(C(=O)NCc2c(Br)cc(OC)c(F)c2)=O)CC(C)(C)NC(C)(C)C1 c12cccc(c1)C2=O.C1(CC(=O)NCC(N)=O)COCCO1 N1(C(CC(c2c(C)noc2C)C)=O)CCC(NC(C2CSC2)=O)C(C)(C)C1 N1(C(c2nc(CC)sc2)=O)CC(CNC(=O)C(=O)NCCC(N)=O)CC1C C1(NC(CNC(CCC)=O)=O)CC(C)CN(C(c2cc(CCCO)on2)=O)C1 N1(C(=O)OC(C)(C)C)CC(C(=O)NC2CC23CCCC3)CC(F)C1 C1(C(C)C)CN(C(c2ncn(C)n2)=O)CCN1C(c1cc(Br)n(C)n1)=O n1(CC)nc(C(=O)NCC2CC(C)N(C(=O)Cc3ncoc3C)C2)cc1C Cc1ccc2cc(C(=O)NC(C)Cn3cc(-c4cocn4)nn3)sc2c1 c1(SC)cn(C)nc1C(=O)NC1C=CC(CNC(C2CC=CCO2)=O)C1 C(CC)(C(=O)NC(C1CC1)CC)=CC.C12CCCN1C(=O)CN(C)C(=O)C21CCC1 C1(C(=O)NC(c2nc(C)no2)C)(CC)CCCN1C(=O)C(c1ccn(C)c1)C C1(C(N(CCNC(=O)CSc2cccc(Cl)c2)CC)=O)CCCCC12CCC2 N1(C(=O)OC(C)(C)C)C2CCC1CC(NC1(CCC#N)CCS(=O)(=O)C1)C2 c1(C(=O)NCC(C)N(C(C(C)OCc2ccc(C)cc2)=O)C)ccc(C)nc1N CC1=NOC(C(=O)NC(CNC(=O)CNC(c2cccc(F)c2)=O)C2CC2)C1C N1(C(c2ncc(C)[nH]2)=O)CC2(CCOCC2)C1c1cn(C2CC2)nn1 c1(C(=O)NCC(=O)NCC(C2CC2)SC2CC(O)C2)cnccn1 c1(C2N(C(=O)Nc3[nH]c(=N)sc3)CCC2)cc(C(F)(F)F)cc(F)c1 N1(C(c2c(C)ncnc2)=O)CC2CCCC(NC(c3cnoc3)=O)C2C1 N1(C(CCC2C(C)C2)=O)CCC2(CCC(N(C(=O)CC3CCC(=O)N3)C)CC2)C1 C1(NC(CNC(C2C(C)C2)=O)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1O CC1(C2(C(=O)NCCCCC3CC3)CC2)CC1 C1(C(=O)NCCC(C)NC(=O)C(C)(C)C2CCCO2)CCC(N(C)C)CC1 n1(CCC(=O)NCC(CN(C(Cc2cc(C)n(C)n2)=O)C)O)ccc(O)nc1=O c1(C(NNC(=O)Nc2cn(CC(=O)N(C)C)nn2)=O)cccc2ccoc12 c1(C(N2C(CNC(C3C(C)C3C)=O)C(O)C(O)C2)=O)cc(=O)c2ccccc2[nH]1 C1(NC(c2cc(C(C)C)on2)=O)CC(O)CN(C(C2OCCCC2(C)C)=O)C1 c1(C(N(C(C(=O)NC)CO)C2CC2)=O)nc(C(=O)OC)co1 C1(C(N2CC(O)(CCNC(c3nocc3Cl)=O)C2)=O)CCC2(CC1)CC(O)C2 C=CCC(C)(C)CC(=O)NC1COCC1NC(C1CCCN(C(=O)N(C)C)C1)=O Cc1nn(C)c(C)c1C(=O)NCc1cc(C(=O)O)ccc1C(F)(F)F N1(CC)CCCC(C(N)=O)C1.C1(=O)C(C)(C)n2cc(nn2)CC(C)C(=O)O1 N1(C(c2c(CC)nn(C)c2)=O)CC(C)N(C(c2ccc(COC)o2)=O)CC1C C(C(=O)N1CC(C)(O)CO1)N(C(=O)CC1=CCCC1)C(C)C C1(C2C(CC(=O)NC(CCC)c3ccco3)C2)CC(C#N)C1.C(=O)C(F)OC(F)(F)F C(=O)(CCC(=O)N(C)C)NC(C)CNC(=O)C(C)C1CCCC1 N1(C(C(CC#C)NC(c2cccc(CO)c2)=O)=O)CCCC(C)(C#N)C1 Cc1ncnc2c1CC(C(=O)N(CCC(C(C)C)NC(c1ccoc1)=O)C)CC2 N1(C(C(C)NC(N)=O)=O)CCCC(C2CCCN(C(C3OCCC3(C)C)=O)C2)C1 C1(CC(=O)NC2C=CC(CNC(C(C)O)=O)C2)C(C)(C)C1(C)C S(=O)(=O)(c1cccc2cnccc12)N(C(C(F)(F)F)C12CC(C1)C2)C1(C)CCC1 C(CCCC(=O)N(CC(C)(C)CNC(C1CCC1c1nc[nH]n1)=O)C)(OC)OC c1(C(N2CCCC(N(C(=O)CC3CCC3)CC)C2)=O)c2c(nn1C)CCCC2 c1(NC(C2(C)CCCC2)=O)cnc(Cl)cc1C(=O)NCc1ccccc1F CCCC(C)(O)CNc1cccc(-n2cc(C(C)(C)CC)nn2)c1 N1(C(CN2CCC(C)(C)C2)=O)CC2ON=C(CNC(=O)CC(=O)N(C)C)C2C1 CCCCC(O)C(=O)NC1(C)CC(C(=O)NC2(C)CCOCC2)C1 n1(CC(=O)N(C(C)CCNC(c2nc(C3CC3)cs2)=O)C)nc(O)ccc1=O C(CCS(C)(=O)=O)(N(C)C(=O)OC(C)(C)C)NC1CC2C=CCC12 Cc1nc(C)c(C(=O)NC2CCN(C(=O)CC3CCN(C)C3=O)CC2O)c(C)n1 N1(C(c2cc(C(C)=O)oc2)=O)CC(N(C)C(c2c(C)ncn2C)=O)C(F)C1 c1(C(=O)NC2CCC(NC(C(CCC)O)=O)CC2)ccc(C)nc1O c1(OC)cc(C(N2CC3(CCN(C(=O)C(C)C(C)(F)F)C3)C2)=O)c(N)c(C)c1 C(=O)(C1COc2ccc(Cl)cc21)N1C(CNC(=O)Cc2nc[nH]n2)CC(O)C1 c1(C(=O)NCCC(=O)NC(CNC(C2C(C)CCO2)=O)C)ncccc1O C12(C(N3CC(CNC(C4(C)CC4)=O)OCCC3)=O)CCCCN1CCC2 CC(C(=O)N1CCCOC(CNC(=O)Cn2cnnn2)C1)C(F)(F)F C(C(=O)N(CCC(=O)N1CC(O)(C(=O)OC)C1)OC)N1CC2N(CC)C(CC2)C1 C1(COC(=O)CCC(C)SCCCC)CN(C)C(=O)CCN(CC(C)(C)C)CC1 Cc1cc(C(=O)NC2CC(=O)N(C3CN(C(c4cnc(C)s4)=O)C3)C2)ccn1 N1(C(CCCCCC)=O)CC2=C(C1)CN(C(C1CC3CCC1C3)=O)C2 c1(C(C(=O)O)NC(N(C)CC2CCCN2C)=O)ccccc1Br C(=O)(C(C)(F)C(=O)N(CC(C)NC(=O)CN1CCCC1)C)OCC N1(C(C(N2CCOCC2)C)=O)CCCC1CC(=O)NCC1(CC2CC2)CC1 C12(C(N3CC(C)C(CC(=O)NCC4CNC(=O)C4)C3)=O)CCCC1OCC2 C#CCC(C)(CC)C(=O)N1CCCC(CNC(c2scnc2C)=O)C1 Cc1ccccc1COCC(=O)NC(C)C(C)NC(c1ncccc1O)=O N1(C(CCn2c(C)csc2=O)=O)CCN(C(c2cncc(CO)c2)=O)C(CO)C1 N1(C(c2c(CC)c[nH]c2)=O)CC(O)CC1CNC(c1csc(=NC)[nH]1)=O N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)C(F)(F)C(O)C3CC3)CC2CC1 C1(C(=O)Nc2cn(CCN3CCCCC3)nn2)CCCCC1C1CC1 Cc1ccc2cc(C(N3CCC(NC(C4CCC(C)CC4)=O)C(C)C3)=O)cn2c1 C1(C(=O)NC(C(C)C)C2CCC2)CN(C(=O)NC2CC2)CC1C(C)C c1(C(N2CCC(NC(CC(C)(C)SC)=O)C2)=O)cccc(S(N)(=O)=O)c1 c1(C(=O)NC2CC(C)(NC(C(CC)C)=O)C2)cccn(C2CCSC2)c1=O C1(C(=O)NC2C(C)(C)CCN(C(C=NOC)=O)C2)COc2ccc(O)cc2O1 c1(C(=O)NCCCNC(c2c(CC)scc2)=O)cc(C)c(F)o1 C1(C(=O)NCc2c(C(=O)NC3COC(C(F)F)C3)c[nH]n2)CC12CCCC2 c1(C(C)NC(c2c(C)nn[nH]2)=O)cccc(N2CCOC2=O)c1 c1(Cc2cn(CCCNC(C(CN(CC)CC)F)=O)nn2)cccc(S(C)(=O)=O)c1 c1(C(=O)NCC2CC3CC3N2C(=O)CC2CC=CC2)[nH]nc2ncnc(O)c12 C(=O)(C1CCc2scnc21)NCC(C1CCCCN1C(=O)CC1CCSC1)(C)C c1(CC(N2CCCCC(NC(C3(Cl)C(C(C)=O)C3)=O)C2)=O)cnc2cccnn12 C1(C(C(=O)NCC2C(NC(c3c[nH]cc3-c3ccc(Cl)s3)=O)C2)F)CCOCC1 c1(OCC(=O)N(C(C)CNC(c2ccc(C(C)O)cc2)=O)C)cc(F)cc(F)c1 C1(CNC(c2cc(C)on2)=O)CCN(C(C2(C)CCC(O)CC2)=O)CC1(F)F C1(F)(CNC(c2cccc(OCC)c2)=O)CCN(C(=O)C(C(=O)OC)OC)CC1 c1(C(N(CCOC)CCNC(C23CC(C)C2C3)=O)=O)cccc(C(C)C)n1 c1(C(=O)NCC(CCNC(C(C2CCCCC2)C)=O)O)ccn2nccc2c1 N1(C(C(CC)COC)=O)Cc2ccccc2C(NC(=O)C2=CCCC2)C1 C12(CNC(C(CO)NC(C3(C)CC(C)C3)=O)=O)CC(C)(CCO1)C2 Cc1cc(N)cnc1C(N1CCC(F)C(NC(=O)CC(C)C)C1)=O N1(C(CCC(C)NC(CSCCC)=O)=O)CCCC(C)C1CO C(=O)(CC1=CCCC1)N1CC(C)C(CNC(=O)CCNC(N)=O)C1 c1(C(N(C)CC2N(C(C3(CC(C)C)CCCC3)=O)CCC2)=O)cccnc1O c1(OC)ccc(C(N2CCC(OC(c3ccnnc3)=O)CC2)=O)c(OC)c1Cl c1(C(N(C2CCC(NC(c3ccnnc3O)=O)C2)C)=O)nccn2ccnc12 N1(C(C2=CC(C)(CC)C2)=O)CCC2CCN(C(c3sc(C)cc3Cl)=O)CC12 c1(OC)ccc(OC)c(C(=O)NC(CCN(C)C(C2CC(F)C2)=O)C(C)C)c1N c1(N2CCC(C)(NC(C3CCCCS3)=O)C2)ncc(C#N)cc1F CCCCCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C=CC=C(Cl)Cl)C1 C1(CC(=O)NC(c2cccc(C)c2)C)CCCN(C(=O)C=CC2(C)COC2)CC1 c1(C(=O)NC2(CNC(COC)=O)CCC2)cc2c([nH]1)CCOC2 C=CCC(CC)C(=O)NC1(c2cn(CCSCCO)nn2)CCOC1 N1(C(c2c(CC)c(F)ccc2)C(=O)NC(C)CC)C(C)CS(=O)(=O)CC1C CC1CCC(C(=O)N2CC(n3cc(CNC(=O)OC(C)(C)C)nn3)CO2)CC1C n1(C(CC)C)nc(C)cc1C(=O)NCC1CN(C(=O)C=CCn2cncn2)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(O)C(F)(F)F)ccc2cc[nH]c2c1F C1(N(c2nnnn2C2CC(F)(F)C2)C(c2cc(C(F)(F)F)cs2)=O)CCCC12CC2 C1(NC(COCCC(C)C)=O)COCC1C(=O)NCC1(O)CC(CO)C1 C1(C(C)NC(C2CC2C2CCCO2)=O)CCN(C(=O)C(c2ccnn2C)C)CC1 N1(C(c2c(C)nn[nH]2)=O)CCCOC(CNC(C2(C)CCCO2)=O)C1 CC12CCC(CNC(=O)NOCCCCC3CC3)(CC1)CO2 C1(C(N2CCC(CNC(C(CC=C)C)=O)C(C)C2)=O)C2CCC1(C)C2(C)C N1(C(CCC(C)OC)=O)CC2CC2CC(NC(c2c[nH]cc2Br)=O)CC1 C(=O)(CCCOC(C)(C)C)NCCN(C)C(c1cc(-c2ccccc2)ns1)=O N1(C(c2ccc(C)cc2C)=O)CCC(NC(=O)C2=C(C)CCOC2)CC(C)(C)C1 C=C(C)C(O)CC(=O)NCC1CCC1NC(c1cc(-c2csc(C)n2)c[nH]1)=O N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(C12CCCC1C2Br)=O C(=O)(C1=CCC(F)(F)CC1)NC1(CNC(C(C(C)OCC)O)=O)CCOCC1 C1(C(=O)NCc2ccc(CNC(c3cscn3)=O)cc2)CCc2c[nH]nc2C1 c1(C(C)C)cc(=NC2CC3CCC(C2)N3C(C2CC3(C2)CC3F)=O)[nH]c(Cl)n1 c1(NC(C2N(Cc3ccc(OC)cc3)CCC2)=O)ccc2c(c1)C(C)(C)C(=O)N2 c1(OC)cc(C(=O)NCc2ccc(CNC(=O)C(=O)N(C)C)cc2F)cc(C)c1 Cc1ccc(Cl)c(O)c1C(=O)N(C)CC1CCCC(NC(=O)C2=CC(C)(C)C2)C1 c1(C(N2CCC3CCCC23C(=O)O)=O)ccc2cnccc2n1 N1(C(C#C)=O)CCCC2(CCCCN2C(=O)CCc2ncc[nH]2)C1 C1(C#N)(C(N2CC(CNC(C=CC)=O)C(O)C2)=O)CC2(CC2)C1 CC1(C)CN(C(=O)C(C)(C)C2CCC2)CC(CNC(=O)CCNC(=O)C2CC2)O1 N1(C(Cc2ccc(C)cc2)=O)CCN(C(=O)C(C)n2ccnc2)C2CC12 Cn1cc(C(=O)NC(CNC(=O)C=C2CCSCC2)CO)c(C2CCC2)n1 C1(CN2CC(C3OCCN(C(C#CC(=O)N(C)C)=O)C3)C2)CCn2cnnc2C1 c1(C(=O)NCCC(C)NC(C2CCC(C)CC2)=O)cc(=O)c2ccncc2o1 C(C(F)(C(=O)N1CCCC(C)(C#N)C1)C(C)C)NC(C1CC(OCC)C1)=O N1(C(CCc2n(C)c(S)nn2)=O)CC2CCN(C(C3(F)CCCOC3)=O)CC2C1 Cc1cc(=NC(=O)CNC(c2cnc(C3CC3)nc2)c2nnnn2C2CC2)[nH]o1 c1(C(=O)NC2(CC=C)CCC2)ccoc1CNC(=O)C(C)(C)OC C(=O)(C(C)C(C)(C)C)NCC(CNC(=O)C=Cc1ncc[nH]1)OC N1(C(C(C)n2cccc2)=O)CCCC(O)(CNC(=O)CCC2CC(F)(F)C2)CC1 O=C(C1=CC2(CCN(C(=O)CC(F)(F)F)C2)C1)NCCC1CCCCC1O C1(C(N2CC(OC)C(NC(C3CC4CCC3O4)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 N1(C(C2(C#C)CC2)=O)CCC2CCN(C(=O)Cc3cccc([N+](=O)[O-])c3C)C2C1 C1(C(=O)NCC(C)(C2CC2)NC(c2c(CC)occ2)=O)CCN(C)C1C N1(C(C(CC(N)=O)NCc2cccc(C(=O)OCC)c2)=O)C2CCC1CN(C)C2 C1(C(=O)N(C(C)CC(N)=O)C)(CC)CN(C(=O)CCNC(=O)NC)C1 c1(C(=O)NCC(C2CC2)NC(CCSC)=O)cc(C#N)c(F)cc1F CCC(C(=O)NCCOC1CCN(C(=O)Cn2ncnn2)C1)N(C)C C1(NC(CSc2c(OC)cccc2)=O)C2CCC1N(C(c1sccc1SC)=O)C2 C1(NC(C2C(NC(C(C(C)C)=O)=O)CCC2)=O)CCCC2(CC1)CC2 CN1C2CCC1CC(=CC(=O)NC13CC1CN(C(c1ccc[nH]1)=O)C3)C2 c1(SCC)ccc(CN2CCC(NC(=O)C(c3nc(CSC)no3)C)C2=O)cc1 CC1CC(C(N2CCC2(C)CCO)=O)CCN1C(c1csc(F)c1)=O C1(CNC(c2occ(C(N)=O)c2)=O)CCCCN(c2ccc(C#N)nc2)C1 N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CC1)CCN(C(C1CC(C)(O)C1)=O)C2 C1(C(N(C2CCOC2)C)=O)C2CN(C(C3(C(F)(F)F)CCC3)=O)CC12 N1(C(C(C)NS(C)(=O)=O)=O)CCC(NC(C2(S(C)(=O)=O)CCCC2)=O)C12CCC2 C1(C(=O)NC(CC)C(F)(F)F)CN(C(=O)Cn2ccnc2C)CCC1(F)F c1(C(=O)NC(CC=C)CNC(C2CC(O)CN2C)=O)ncc([N+](=O)[O-])cc1C C1(C(=O)NCc2n(CC)cnn2)CCN(C(c2snnc2C)=O)C1C C(=O)(CCCN=[N+]=[N-])N1C(CC(=O)NC(C=C)C2CCC2)CC1 CC(C)CCC(=O)NCCCC(c1ccccc1)NC(=O)CC12CC(C1)C2 CC(O)C(C)C(=O)N1CC(O)(C(C)OC2CCC2)C1.c12cccc(c1)C(=O)OCC2.OC C1(CC#C)(C(N2CC(N=[N+]=[N-])C2)=O)CCN(C(c2cc[nH]c2C)=O)C1 N1(C(C(CC)N(C)CC)=O)CCN(CCNC(C2CC(n3cnnc3)C2)=O)CC1 C12(NC(c3scc(C(N)=O)c3)=O)CCCC1CN(C(C13CCC(CC1=O)C3)=O)C2 C(=O)(C#CC(C)(C)CNC(c1nc(O)sc1C)=O)N(C(C)C(=O)NC)CC C1(CC(=O)NCC(C)N(C(CCC)=O)CC)CCOC1=O CC(C)C(O)CC(=O)N1CC=CC(C(N2CCC(F)(CO)C2)=O)C1 C(=O)(C1CSc2ccccc21)N1CCC(O)(C(C)NC(CCC(=O)NC)=O)CC1 N1(C(C(C(C)C)C#N)=O)CCC(C2CC2)C1C(=O)Nc1ccc2nncn2c1 CC1CC2CCN(C(C3CCN(CC4CN(C)CCO4)CC3)=O)CC12 c1(C(=O)NC2C(NC(c3c(OC)cc(O)nc3)=O)CC2)cc2cccn2cn1 C1(C)(C(N2CCC(CNC(C(CC#C)O)=O)CC2)=O)CC(C(C)(C)C)=NO1 N1(C(C(F)OC)=O)CCC2(CC1)CN(C(C1CCCC(F)(F)C1)=O)C2 c1(C(=O)NCC(CC)NC(C2(C(=O)OC)CCC2)=O)coc(C(C)OC)n1 c1(C(=O)NCCOC2CN(C(=O)Cn3cc(Cl)cn3)C2)cc(O)ccc1F c1(OCOCC)cc(OCl)cc2ccccc12.c1ccccc1 N1(C(c2nn(CC)c(O)c2)=O)CC2(CC2)CC1CC(=O)NCCCS(C)=O C1(NC(C2C(OC)CN(C(COCCCC#C)=O)C2)=O)COCCN(C)C1 C1(CN(C(C(CC=CC)C)=O)C)CN(C(c2cccc(C#N)c2)=O)CC12CC2 CC(C)C(C)CC(=O)NC1(CCNC(C2(F)CCCOC2)=O)CC1 N(C1CCOc2cc(F)cc(F)c21)C(=O)NC(C)C(C)(C)c1ccccc1 c1(N2CC(CCO)(N(c3ccc(C)cc3)C(C)=O)C2)ncc2c(ncn2C)n1 c1(OC)cc(OC)nc(N(c2ncc(C)cn2)C(C2CCNCC2O)=O)n1 N1(C(C(CC=CCC)C)=O)CCC(CNC(c2nn[nH]c2Cl)=O)C12CC2 N1(C(CC(CNC(COCC(=O)OC)=O)O)=O)CC(=O)NCC1C(C)C c1(NC(C2N(c3ncc(C)c(C)n3)CCCC2)=O)cc(Br)c([N+](=O)[O-])cn1 C1(CC)CC(c2nnnn2C2CC(F)(F)C2)(NC2CSC2)CCO1 C1(NC(C)=O)CC2(C1)CN(C(c1cccc(C(F)F)c1F)=O)C2 N1(C(CSCCC)=O)CCC2CN(C(=O)C(C)Oc3ccc(F)cc3)C2C1 c1(C(C(=O)N(C2CN(C(C(CC)SC)=O)C2)C)O)ccc(Br)cc1 CC(C)C1=NOC(C(N2CCCC2C(C)NC(c2c(SC)cccc2F)=O)=O)C1 N1(C(C(C=C)O)=O)CC(NC(c2cnccc2C(F)(F)F)=O)CC2(CCC2)C1 N1(c2n(CC(=C)C)c(-c3cnn4cc[nH]c34)nn2)CCCC(C2CCC2)C1 C1(C(N2C(C)CN(C)CC2)=O)CCN(C(=O)C(O)O)CC1(C)C C(=O)(C1=CC2CC=CCC12)NCC1CC(NC(c2cc(C)c(Cl)c(N)c2)=O)C1 C1(N(CC(N2CCCC2=O)C)C2CC2NC(=O)OC(C)(C)C)CC2CC1CN2 C1(NC(c2nn(C)c(O)c2)=O)CCN(C(c2cnc(C3CC3)s2)=O)CC12CCC2 C1(NC(C(CC)F)=O)CN(C(=O)CN(C)Cc2ccc(Cl)cc2)CC1C c1(C(=O)NCC(C2CCCC2)NC(C(C)(C)N(C)C)=O)cccc2c1CCN2 Cn1cc(-c2cccs2)cc(NC(=O)CC(=O)NCC(F)(F)F)c1=O C=CCCCCC(=O)N1CCOC(CNC(C2CC(Oc3ccccc3)C2)=O)C1 CC(C)(CC(F)(F)F)C(=O)NC(=O)NCCN1CCC2CCCCC2C1 CC(CC(=O)NCC(C)(O)CNC(=O)C1=CCCSC1)C(F)(F)F CCC(CCOC)C(=O)NC1(CC)CCCN(C(=O)Cn2cc(Br)cn2)C1 C(=O)(CC(C)(C)C(F)(F)F)NCCCN(C(=O)C(c1cccc(F)c1)(C)O)CC CC1=C(C(=O)NC2CN(C(C3CC4C=CC3CC4)=O)CC2N(C)C)CCCO1 c1(C(=O)NCCCC2(NC(CCCCC)=O)CC2)cc2n(n1)CCNC2=O C1(C)(C(N2C(CN(C(=O)COCC3CCCC3)C)CCC2)=O)CCCNC1=O Cn1c(C(N2CCC3(NC(=O)OC(C)(C)C)CC3C2)=O)cc(=O)c2ccccc12 c1(C2C(C(N(CCCNC(C(CC)(C)O)=O)C)=O)C2)c(Cl)cccc1Cl C(CC(C)C)(C(=O)NCC(CC(F)(F)F)NC(c1coc(C(=O)OC)n1)=O)OC C1(O)(CNC(C2(CCOC)CCC2)=O)CCCN(C(=O)CCn2ccc(C)n2)C1 c1(C(N2CC=CC(C(N(C3CCNC3=O)CC)=O)C2)=O)cc2ccncc2[nH]1 Cc1nn(C)c2nc(O)cc(C(=O)NC(C)CC(C)NC(=O)CCC3(C)CC3)c12 N1(C(C(n2c(C)ccn2)C)=O)CC2(C(=O)NCC(O)CO)CC1CO2 N1(C(CC)=O)CCN(C(c2ccc(CC)nc2)=O)CC(O)C1 C(C(C)(COC)CC)NC(C(C=CC)O)=O.C1C(=O)N1CC(C)C C1(C(=O)NCCN(CCOC)C(C2(C(C)(C)C)CCC2)=O)CCC(=O)N1.S(C)(=O)(=O)N C(C1CCc2cc(F)ccc21)NC(c1ccc(N2CCCS2(=O)=O)cc1)=O C1(C(=O)NCC(=O)NCC2(C)CC2)CN2CCC1C2 N1(C(c2c(NC)cncc2)=O)CC(CNC(=O)C(C)c2ccco2)CC1(C)C N1(C(C(C=C=C)C)=O)CCN(C(=O)Cc2nnn(C(C)(C)C)n2)C(CO)C1 FC(F)(F)C(CN=c1[nH]cnc2ccc(I)cc12)N1CCCCCC1 N1(C(C2CC(O)(CC#C)C2)=O)CC=CC1(C)C(N1CC(N(C)CC)C1)=O C(c1ccncc1)=CC(=O)NC1CC(CNC(c2nnc(C(F)(F)F)s2)=O)C1 C1(CNC(C=CC(CC)=CC)=O)CCN(C(c2ccncc2NC)=O)C(C)C1 N1(C(C2C(C)C2)=O)CCC(CNC(=O)C(C)Cc2ccccc2F)C1(C)C N1(C(CC(CC2CC2)NC(C2ON=C(C)C2)=O)=O)CC2CC1CS2=O C12(NC(CCOCCOC)=O)CCCC1N(C(=O)COCCCC(C)C)CCC2 N1(C(C23N(C(c4ccc(Cl)o4)=O)CCC2C3)=O)CCC([N+](=O)[O-])CC1 N1(C(c2c(N)nccn2)=O)CCCC(NC(c2nn[nH]c2Cl)=O)C(F)C1 C1(C(N(C)CC2N(C(C(C)C)=O)CCOC2)=O)CCN(c2ccncc2)CC1 C#CC1CCCN(C(=O)C(=O)NCc2cc(-c3csc(C)n3)ccn2)C1 c1(-c2cn(CCCN(CCOCC(=O)NOCO)C)nn2)ccc(F)cn1 N1(C(=O)Cn2ncnn2)CCC2CN(C(C3(n4cncn4)CC3)=O)CC2C1 CCC(C)(F)C(=O)N1CCC(NC(=O)C(O)Cc2[nH]cnc2C)CC1 CCC(CC)(C(=O)NC1CC(C)N(C(=O)Cc2cnsc2)C1)OC N1(C(=O)C=CCNC(C2CCN2Cc2ccccc2)=O)CCC12CCCOC2 Cc1ncc(N)cc1C(N1CC(CNC(=O)C(c2cccc(F)c2)O)C1)=O C1(C(C(=O)N(C2CCN(CC)C2)C)C)CCN(C)CC1 N1(C(C(C(CC)CC)C)=O)CCC(C(=O)NC2CC3CCC2C(O)C3O)=C(F)C1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(c2cnn(C3CC3)c2Cl)=O)CC1(C)C C1(COC(C2OCCCO2)=O)CCCCC1.C12CN(C1)C(=O)O2 C1(NC(NC(C=C)C)=NCC2CCCS2)CCn2c(CCOC)nnc2C1 C#Cc1ccnc(C(N2CC(NC(=O)CCc3ccc(F)cc3)CC2C)=O)c1 c1(N(CC(C)(C)O)C(N(CCCCO)C)=O)cnc(C(F)(F)F)cc1 N1(CCSc2scc(C)n2)CCOC(C)(CNC(=O)C(C)(C)C(F)F)C1 C1(NC(C(CN(C)C)O)=O)CCOCC1NC(C1(CO)CCCC1)=O CN=c1c(C(=O)NC(C)C(C)NC(=O)Cn2cncc2C)c[nH]c2ccccc12 C1(C(=O)NCC(CCC)OCC)C(C)OCCN1C(=O)C(C)N(C)C N1(C(C(C)SC)=O)CCC2C(NC(=O)CCOC3CC3)CC12 c1(CC)ccc(C(C)C(=O)NC(C)(C)CNC(=O)C(C)(C)C2CCCCC2)cc1 c1(-c2c(Cl)occ2)nc(-c2ccco2)nn1-c1ccnc(F)c1 C(c1ccc(C)cc1C)=CC(N1CC(CNC(CSCC(=O)OC)=O)C(C)C1)=O C1(C(=O)NC(C)CC(C)NC(=O)CC2CCC2)(OC)CCOCC1 c1(C(=O)NC(C2CCCN(C(C3C4COCC34)=O)C2)C)ccnc2c1OCO2 N1(C(C(CCC=C)NC(=O)CC(C)n2cccc2)=O)CC2(C1)NC(=O)NC2=O N1(Cc2cncc(C)c2)CCC2(CCN(c3cc(C)ncn3)C2)C1 CC(C)C(C(=O)N1CC(C(=O)Nc2ccc(C(C)C)nc2)C(C)C1)C1CCC1 C1(NC(c2n(CC)ncc2)=O)C2CCC1CC(NC(c1cc(C)ccc1N)=O)C2 C1(C(=O)NC(C(C)NC(c2c(OCC)csc2)=O)(C)C)CCc2nc[nH]c2C1 c1(C(=O)NC(CC)CNC(=O)C(c2ccc(C)cc2)O)cc(C(N)=O)ccc1C N1(C(CC2C(C)=NN(C)C2=O)=O)CCC(C2CC2)C1CNC(=O)C=CCF C(=O)(C1=NNC(=O)C1)NCCN1CCN(C(c2cc(C(=O)OC)ncc2)=O)CC1 C#CCCCC(=O)N(C1CCN(C(=O)C=C2CCCO2)CC1)CCOC Cc1n[nH]c(C)c1CCC(=O)N(C1CN(C(=O)CC2CCC(=O)N2)CC1O)C c1(C(N2C(CCC)CN(C(=O)COC)CC2)=O)c(OC)ccc(C)c1OC c1(CNc2c(CNc3c(Cl)cc(C)c(Br)n3)nccc2)cccc2cnccc12 C1(NC(c2n(C)nc(CC)c2Cl)=O)CC2CCC1N(C(=O)CC(C)C(C)C)C2 S(=O)(=O)(c1cc(Br)c(F)cc1F)NCC1N(Cc2n(CC)ncc2)CCOC1 c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCC#C)=O)cccc([N+](=O)[O-])c1 N1(C(C(C)OCCOCC)=O)CCCN(C(=O)C=CC(C)(C)C)CC1C CCCCC(CC(=O)NC1CC(C(F)F)C1)NC(C12CCCN1CCC2)=O C(=O)(CCCCCNC(=O)Cc1cc[nH]n1)N1C(CC)(CC)CC1 CC1C(C)N(C(c2cc3ccncc3o2)C(=O)Nc2ccc(F)cc2)CCS1=O C(=O)(CS(=O)(=O)CCO)N1CCC(NC(c2cc(CC)n(C)n2)=O)C(F)C1 C1(C(=O)NC2(C(=O)NC(c3cn[nH]c3)C)CC2C)CC2CCC(C1)C2 N1(C(c2c(CC)nnc(C)c2)=O)CCCCC2(CCN(C(=O)C(C)(C)OC)C2)C1 C(=O)(C(F)CCC(C)C)N(C)CC1CCN(C(=O)C(F)(F)CCn2ccnn2)C1 c1(NC)cccc(C(N2CC=CC(NC(=O)C=C3CCC(C)CC3)C2)=O)n1 c1(N2CCC(C)C(NC(c3c(C)onc3)=O)C2C)ncc2ncn(C)c2n1 c1(C(N2CC(NC(C(N3CCOCC3)C)=O)C2)=O)ccc(C2CCC2(C)C)cc1 Cc1ncccc1NC(C1CSCCN1Cc1cncc(-c2ccccc2)c1)=O C1(NC(CC=CC(C)(C)C)=O)CCCC(C(=O)NC2(CC(C)(C)C)CC2)C1 c1(C(=O)NCC2C(NC(=O)CCCC3CCC3)CC2)cc(O)nc2cnccc12 c1(OCC(=O)NC2C(C(=O)NC3CN(C(C)=O)C3)CCC2)cncc(C)n1 C1(C2CCOCC2)(C(=O)NC(CNC(c2c(Cl)ccc(C)c2)=O)C)CC1(F)F C1(C(=O)NCCSCCC=C)CCC(O)CN1C(c1ccn(C)c(=O)c1)=O N(C1CCCc2ccc(Br)cc21)CC(C)(C)C N1(C(CCC(=C)Br)=O)CCC(CO)(NC(=O)CC2CCCNC(=O)C2)CC1 c1(C(=O)NCC2(O)CC(CNC(CC=CCC)=O)C2)cc(F)cc([N+](=O)[O-])c1 c1(CNC(=NCC=C)NC(CO)CCF)ccc2c(n1)CCCC2 CCC(C)C(O)C(=O)N1CCCC(C(N2CC(c3nc(=O)o[nH]3)C2)=O)C1C c1(C(C(F)(F)F)NC(=O)C(N2CCCC2CN2CCCC2)=O)ccc(Br)cn1 C1(NC(c2cc(OCC)n[nH]2)=O)CN(C(=O)CC(C)CN(C)C)C(CC)(CC)C1 CC1CN(C(C2CC2CNC(=O)C(F)CC2CCC2)=O)C(C)(C)C1 N1(C(C2(SC)CC2)=O)CCC2CN(C(=O)CC3CNC(=O)O3)CCC2C1 C1(OC)CCC(C)(c2nc(-c3ccncc3)nn2CC(=O)O)CC1 C(CC(=O)N(C1CCC(NC(=O)CCCN(C)C)C1)C)(C(F)(F)F)OC N1(C(CC(CC)(C)C)=O)CC2(CNC(C3(CCOC)CCC3)=O)CCC1CC2 C1(C(=O)NC2CCN(C(c3ccn(CC)n3)=O)C2C2CC2)CS(=O)(=O)CC12CC2 C1(NC(c2cnco2)=O)CC(C(=O)NCC2(CO)CC23CCC3)=CC1O C1(CC(N2CC(CNC(C3C(C)C3)=O)N(C)CC2)=O)CC(C)CC(C)(C)C1 c1(N2CCC(CNC(C(C)OCCCCCC)=O)C2)cc(C)ncc1C#N N1(C(Cc2nccc(OC)n2)=O)CC(C)CN(C(=O)C=CC(=O)N(C)C)C(C)C1 c1(C(=O)NC(C(C)C)CNC(=O)CC2CCN(C)CC2)cc(C#N)c(N)cc1O N=c1[nH]c(=NCCN2CCCC2=O)[nH]c(=NC(CC2CC2)c2ccccc2)[nH]1 Cc1cc(N)c(C(N2CCCCC2CCNC(C2(C)CCCO2)=O)=O)cc1C c1(C(=O)NCCCN(C(C(C=C)(C)O)=O)CC)cnc(O)c(Br)c1 CC1(C)CN(C(C2CC3(C2)CC(F)C3)=O)CC(CNC(=O)CC2CC2(Cl)Cl)O1 C1(CC(=O)NC2CCCN(C(C=C(Cn3c(C)nnn3)C)=O)C2)CCCCC1(C)C C1(CCNC(c2c(C)coc2)=O)CN(C(=O)C=CC2CCCC2)CCO1 C1(C)(CNC(C(CCOC)(C)C)=O)COCCN(C(C2CC(C)C2)=O)C1 N1(C(c2n[nH]c(C)c2Br)=O)CCOCC(NC(=O)C=CCN2CCCC2)C1 N1(C(C2CCC(=O)C2)=O)CCC(C2(NC(C3(Sc4ccccc4)CC3)=O)CC2)C1 C1(C(=O)NCC2(O)CN(C(c3nn(C)c(F)c3)=O)C2)CC2OC(=O)OC2C1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCC(CNC(C(C)(C)OCC)=O)C(C)C1 C1(C(=O)NCCSCC(=O)NC(C=C)(C)CC)CCCC12CC2 C=CC(CC)CC(=O)NC1CCCN(C(c2cnc(OC)cc2C(F)F)=O)C1 N1(C(CN(C(C)=O)C)=O)CCC2(C1)CN(C(c1cn(C3CC3)nn1)=O)CC(C)O2 C1(C2CCN(C(=O)CNC(=O)NC3CC3)C2)(NC(=O)CC2COC(=O)C2)CC1 c1(C(N(CC(C2CCCN2C(=O)C2=CCCCO2)(C)C)C)=O)cnn2ccccc12 C=CCC(C)(C(=O)N1CC(C)(C)CC1CNC(c1ccncn1)=O)N(C)C C1(=CC(=O)NCCC2COCCN2C(c2ncccc2F)=O)CN2CCC1CC2 c1(C(N2CCCC(CCNC(=O)CCC[N+](=O)[O-])C2)=O)ccc2scnc2c1 C(CC(C)C)(C(=O)NC(C)C(C(C)C)NC(C1CCCC1)=O)NC(C)=O c1(CC)c(C(=O)NOC(C)C)cnn1-c1ccc(OC)cc1 C(=O)(CCCCC(C)C)N1C(CCCNC(CCSCCC)=O)CCC1 C1(CNC(C(C)CO)=O)CCC2CN(C(c3coc(O)n3)=O)CCC2C1 N1(C(C2CC(N(C)C)C2)=O)CCC2(CCC(NC(C3CSCC(=O)N3)=O)C2)CC1 C(=O)(CCCS(N)(=O)=O)NC1CCN(C(C(c2ccc(C)nc2)(F)F)=O)CC1C N1(C(c2nnc(C)s2)C)CCC(C)(NC(=O)CC2CC=CC2)C1 Cc1cc(N(C(=O)C(C)(C)C2(O)CCOC2)C(=O)C(F)(F)F)cnc1Br N1(C(=O)Nc2nccc(-c3ccc(Cl)cc3)n2)CCCC2(CCNC2=O)C1 Cc1ccc2[nH]c(C(N3CCN(C(=O)C(O)C4CC4)CC3)=O)c(Cl)c2c1 Cc1cc(=O)oc2ccc(OCC(=O)NCC(O)CCNC(=O)CN(C)C)cc12 c1(C(=O)NCCCC2(NC(C(C)OC(C)(C)C)=O)CC2)csc(C(F)F)n1 Cc1cc(=NCc2nc3ccccn3c2Cl)[nH]c(NC2CCN(C)C(=O)C2)n1 C1(C(N(CCCNC(CCC=CC(C)C)=O)C2CC2)=O)CC1C1CCCC1 c1(CCNC(C2C(C)CNC2)=O)ccccc1Oc1ccncn1 c1(C(=O)NCCC(O)C(=O)N2CC(N3CCC3)C2)ccn2nccc2c1 N1(C(C(C2CCCC2)OC)=O)CCCC1C(=O)N(C1CCN(CC2CC2)C1)C c1(OC)c(C(N2CCCCC2c2cccs2)C(=O)NCCC2CC2)cccc1F N1(C(C=CC=CC)=O)CC(CO)C2(CCN(C(=O)C(C)(C)CC3CC3)CC2)C1 N1(C(CCc2ncn(C)c2)=O)CCC(NC(=O)CCSC(F)(F)F)C(O)C1 Cc1c(C(=O)NCC2N(C(c3ccc[nH]3)=O)CCC2(C)C)c[nH]c1C#N c1(C(=O)NC(C2CCN(C(C3(OC)CCSC3)=O)C2)(C)C)ccccc1Cl C1(C(=O)NCC(=O)OC(c2cccc(Cl)c2)C)CC1C1CCCC1 C1(N(C(CC(OCC)OCC)=O)C)CCCN(C(=O)C(C)(C)C)CC1 c1(NC(C2CC(C(=O)OC)C2)=O)cnn(C2CCCC2)c1C.C12(O)CN(C1)CC2 C1(OC)CN(C(c2ccns2)=O)CCC1NC(=O)CN1CC2CC2C1 S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CC(C(=O)Nc2cccc(C#N)c2)OCC1 n1(CC(=O)NCC2CN(C(c3cscc3C(F)(F)F)=O)C2)nnc(SC(F)F)n1 C1(C(=O)NC(C2CCCN2C(c2cc[nH]n2)=O)C)(COC)CCOCC1 c1(C(C(=O)NC(C)CC)N(CCOCC=C)C)cccc(C2CCCC2)c1 c1(NC2C3CN(C(C4CCC(CC)CC4)=O)CC32)cc(CO)nc(C(F)(F)F)n1 C1(C(N2C(CC(C)C)CC2)=O)N(C(C2CCC(=O)CC2)=O)CC12CCCC2 C1(C(=O)NC(c2ccc(F)cc2)CNC(CCCOC(C)=O)=O)CCCC1(C)C N1(C(C(COCC)NC(c2cncnc2C)=O)=O)CC(N(C)C)C2(CCC2)C1 CCCCC(CCC)NC(=O)CC(C)(C)NC(C1CC(F)C(=O)N1)=O C12(CNC(CC)=O)CCCCC1N(c1ncc(I)cn1)CC2 N1(C(=O)C=CCN2CCOCC2)CCC2CC(C1)CN(C(=O)C(O)C1CCCC1)C2 c1(C(=O)NCCN(CCOC)CC2CCCO2)c(C2CC2)cnn1C.C1(=O)CN1 C(C(C)(C)C(=O)N(C1CC(C(=O)Nc2cnc(SC)nc2)C1)C)SC N1(Cc2c(C)coc2)CCCC1(C)C.c1(NC(c2nc(C)c(C)s2)=O)ccc(F)cc1 CC1(C)CC(CC(=O)NCCC2CCCC23CC3)CN1C(=O)Cn1cnc(=N)[nH]1 c1(SC(C)C(N)=O)nc(CC(=O)N(C2CC2)CC2CC(C)CO2)cs1 Cc1cc(C(N2CCCC(O)(CN(C(=O)CN3CC=CC3)C)C2)=O)c(C)cn1 c1(C(=O)NCC2(OC)CN(C(CC(=C)C)=O)C2)ncc(C)cc1OC c1(C(=O)NCC2N(C(CC3(C)CCCO3)=O)CCC2)ccc(Br)cc1F C1(NC(C(c2cnn(C)c2)C)=O)CCCCCC1NC(c1cnc(O)n1C)=O C1(CNC(c2c(C)c[nH]n2)=O)CN(C(=O)Cn2cc(C#N)cn2)CCC1C Cc1c(CC(=O)NC2CC(CC(=O)NC34CCC(CC3)C4)C2(C)C)ncn1C C12(NC(=O)Cn3cc(C4CC4)cn3)CC1CN(C(c1ccc(C(F)F)cc1)=O)C2 Cc1cnc(NC(c2ccccc2)CF)c(S(=O)(=O)NCCc2cn(C)cn2)c1 c1(C(=O)NC2CCCN(C(=O)C(F)OC(F)(F)F)C2)ccc2ccccc2c1F C1(C(=O)NC(CCNC(CCOCCOC)=O)C(C)(C)C)CC1C1CCOCC1 Cc1nc2sccn2c1C(=O)N(C)CCC(=O)CO.c1(OCCN)cnn(C)c1 c1(C(N(C(c2cccc(OC)c2)C)C)=O)cc(S(=O)(=O)NC(C)C)ccc1Cl C1(C(=O)NC(C(C)F)C)CCC(C2CC2)N1C(c1cnns1)=O N1(C(C(OC)OC)=O)CCC(CNC(=O)C(=O)NC2CC2)C(C)C1 N1(C(C(=O)NCC=C)C2CC(C(=O)OCC)C2)CCCC1CC C1(N(CC(=O)Nc2ccsc2)C)CCCCCC1n1cccn1 c1(OC)c[nH]c(C(=O)N(CCC(C(C)C)NC(c2cccc(C)c2)=O)C)cc1=O C1(c2cn(CC3(O)CCN(C(C)(C)C)C3)nn2)CC2(C1)OCCO2 C(=O)(C1=NOCC1)N1CCC(CN(C(C(c2ccc(F)cc2)OC)=O)C2CC2)C1 c1(CNC(C(=O)NC)C)cc([N+](=O)[O-])c(O)cc1F.C12CC(O)CCN1C2=O C1(NC(c2c(C)n[nH]c2)=O)CCN(C(=O)CC(=O)OC(C)(C)C)CC1F c12ccc(cc1)-c1nnc(o1)SC(C)C2=O.C(C(=O)NCCNCC)=CC=CC Cc1onc(C(N2CCC23CN(C(C2CCC(=O)N2C)=O)C3)=O)c1[N+](=O)[O-] C1(CNC(CCCOC)=O)CN(C(c2ccc(C(=O)NC(C)C)[nH]2)=O)CCO1 c1(OC)cc(F)ccc1C(=O)NC1(CNC(=O)C(C)CC2CCC2)CC1 N1(C(C2(N(C(c3c(C)nco3)=O)C3CC3)CCC2)=O)CC(C)(C)OCC1C N1(C2CN(C(C(COC)O)=O)C2)CCN(C(=O)C=CC(C)(C)C)CC1 N1(C(COCCOCC)=O)C2CCC1CC(O)(CNC(c1cc(C)ns1)=O)C2 c1(CC)cn2c(n1)CCC(C(=O)NCC1CC(F)CN1C(C1CC1C)=O)C2 N1(C(C2CC2F)=O)CC2CCC(C1)N2Cc1ccc(Br)nc1Br c1(C(N2C(CCC)(C(=O)NC)CCC2)=O)cc2c(F)c(F)cc(F)c2[nH]1 c1(C(=O)NCC2OCC(CNC(=O)CC3CCC3)C2)ccc2ncnn2c1 c1(C(=O)NC2(C)CN(C(=O)C(Cl)=CCl)C2)cnc(S)n1-c1ccccc1 c1(CC(N2CCC(N(C(C(C(C)C)C)=O)C)CC2)=O)cc(Cl)cc2ccccc12 C1(CC)CCN(C(=O)CCOC(C)C)C1C(=O)NCc1cnn(CC)c1C c1(N(C2CCN(C(=O)Nc3ncc(CN)s3)CC2)C)ccccc1[N+](=O)[O-] c1(Oc2ccccc2)cccc(OCCCCCNC(C2C(C)C2C)=O)c1 C1(CC(N2CCN(C(C(Cc3ccc(C)cc3)C)=O)CC2)=O)CCC(C)(O)CC1 N1(CC=C)CCCN(C(=O)C(CO)NC(=O)CC2COCC(C)O2)CC1 c1(N2CCCC(CSC)C2)nc(N2CCCOC(CCO)C2)c2ccccc2n1 C1(N(C(=O)C(C)O)CC)CCN(C(c2[nH]ccc2Cc2cccnc2)=O)C1 C1(NC(c2c(C)nccn2)=O)CN(C(=O)Cn2nnnc2C(C)C)C2(CCC2)C1 C1(C(=O)NC2CN(C(c3c(NC)cncc3)=O)C(C)(C)C2)CC(C)(C)OC1(C)C c1(SC)cccc(C(=O)NC2CCOCC2NC(=O)C(C)(C)C(N)=O)c1[N+](=O)[O-] c1(C(=O)O)ccc(CNCc2c(I)ccnc2Cl)cc1Br N1(C(Cc2ccc(OC)nc2)=O)CCC2CCCC(C1)N2C(=O)C1=CC(C)(C)C1 N1(C(C(CC)N(C)C(C2CC2C#N)=O)=O)CCc2c(cnn2C)C1 N1(C(c2cc3c(nc2O)CCCC3)=O)CC2(CCOCC2)C2CCCC12 N#Cc1cc(C(N2CC3=C(C2)CN(C(=O)CCF)C3)=O)ccc1F C(CN=c1[nH]c2c(F)cccc2n1C)c1scc(CC)n1 CC1(C)CC(NC(=O)C2=CSCCO2)CCN(C(C2CCn3cnnc3C2)=O)C1 c1(SC(C)C)ccccc1C(=O)NCC1CN(C(=O)CC2(C3CC3)CC2)CC1C c1(C(=O)NCCC2(CNC(c3c(C)nc[nH]3)=O)CC2)cccc(=O)o1 N1(C(CCC(C)C)=O)C2CC1CN(C(=O)CNC(=O)COc1ccccc1)C2 N1(C(CC(CCC)O)=O)CCN(C(=O)Cc2ccon2)CC(O)C1 N1(C(C(C(C)C)n2cnnc2)=O)CCC(C)N(C(C2CC(C)(C(=O)O)C2)=O)CC1 CCCCC(C)C(=O)NCC(O)CN(C(=O)CC(F)(F)Br)C c1(NCC(CSC)OC)nc(N(C)CC2CCCCCC2)c2ncsc2n1 N1(C(C2C(CCOC)C2)=O)CCCC(C)(C)C1C(=O)Nc1ccc(C)nc1C C(=O)(C(C)SC(F)(F)F)NC(CN(C(C)=O)C(C)C)C1CCC1 N1(C(C2(C)CCNC2=O)=O)CCC2(CC1)CC2CNC(=O)C(F)(F)C(F)(F)F c1(C(=O)NCC2(CNC(CCN(C)CC)=O)CCCC2)cccc(CO)c1N O=C(C1CCCc2n[nH]cc21)NC1CN(C(c2coc(Br)n2)=O)C2CCCCC12 S(=O)(=O)(c1ccc(NCCCC2CCOC2)cc1Cl)N1CCC(CCC)(CO)C1 CC1(NC(c2ccccc2)=O)CCN(C(=O)CC2(O)COC(C)(C)C2)CC1 N1(C(c2c(F)cc(OC)cc2Cl)=O)CCc2[nH]nc(CNC(=O)C(C)(C)F)c2C1 C1(CNC(C=COCC)=O)CC2(CCOCC2)CN1C(c1cc(O)n(CC)n1)=O C(=O)(C(CC(C)C)ONC(C1CC(=O)NC1(C)C)=O)NC(CCC)CO c1(CC)nnc(C)cc1C(=O)NC(c1ccccc1)CNC(C1CC(C)(O)C1)=O c1(CC)ccc(O)c(C(=O)NCC2CN(C(C3CCCC3(F)F)=O)CC23CC3)c1 C1(CNC(CC(CC)(C)C)=O)CN(C(=O)C(O)CCC(C)C)CCC12CCC2 CCC(N)CCC(=O)Nc1cccc(Oc2cccnn2)c1 Cc1cc(C)c(C(=O)NCC(C)CNC(c2cn(C(C)(C)C)nc2C)=O)[nH]1 C(=O)(C(C)CC(F)(F)F)N1CCC(C#C)(C(=O)Nc2ccccc2OC)C1 C1(O)(CNC(C(C(C)SC)O)=O)CCN(C(=O)CC(=O)OC(C)(C)C)CC1 C1(CN(C(=O)CSCC(F)(F)F)C)CN(C(=O)CC2OCCCO2)CCO1 C(=O)(C1NCc2n[nH]cc21)NCC(CC(=O)OCC)c1ccccc1 C12(NC(c3ccnc(CO)c3)=O)CCCC1CN(C(c1ccc(F)c(F)c1)=O)C2 C1(C(=O)NC(CCC)C(=O)NCCOCCCO)CCCCC1(C)C CN1CCCC(C(C)(C)C(N2CCC(F)(CNC(c3cc(C(F)F)cs3)=O)C2)=O)C1 c1(OC)ccc(C)nc1C(=O)NC1(CO)CN(C(c2cc(C(F)F)[nH]n2)=O)C1 c1(NC(C2C(OC)CCCC2)=O)ccc(NC(=O)C(C(C)O)N(C)C)c(C)c1 Cc1nc(N)cnc1C(=O)NCC(C1CCCC1)NC(C1CC(=C2CC2)C1)=O C1(NC(c2cc[nH]c2)=O)CCCC2CN(C(C3(n4cnnn4)CC3)=O)CC12 C1(NC(c2nc(-c3cccnc3)cs2)=O)CCNCC1CO N1(C(CC(CC2CC2)NC(C2C3CCC(F)C23)=O)=O)CC2CC(O)CC1C2 c1(CNC(C2C3CN(c4c(OC)c(C)ncn4)CC32)=O)ccc2oc(C)nc2c1 CC(CC(=O)NCC1CCC(NC(=O)CCc2nc[nH]n2)CC1)C(F)(F)F N1(C(CC=CC)=O)CCC2(CO)CN(C(=O)CSc3ccc(O)cc3)CC2C1 c1(C(CNC(=NC)NCC2CCCC(C)(C)C2)(C)OC)ccc(F)c(F)c1 c1(C(N2CCCC(C)C2CCNC(C2(O)CCC2)=O)=O)noc2cc(F)ccc12 C1(C#N)(C(=O)NCC(CNC(CC(C)OC)=O)OC)CC(=O)C1 c1(N2C(CC#N)CN(C(=O)Cc3cc[nH]n3)CC2)ncc2cc(Br)cc(F)c2n1 C(=O)(C1=CC2CCCC12)NCC1(CNC(c2[nH]c(=NC)sc2)=O)CC1 Cc1ccc(C(=O)NC2(CF)CN(C(c3cc(C(F)F)nn3C)=O)C2)nc1C CCCC(C(O)C(=O)NCC(C)(C)CO)NC(C1(C)CCOCC1)=O N1(C(c2c(CC)nco2)=O)CCC(Cc2nc(C3CCCC3)no2)CC1 C(C(C)(C)CC(=O)O)NC(c1cnn(CC)c1-c1ccccc1)=O C12(NC(c3ccnnc3O)=O)CCCC1N(C(=O)C=CBr)CCC2 C(=O)(C1=CS(=O)CCC1)NCC(CN(C(c1c(NC(CC)=O)cccc1)=O)C)C N1(C(C(CCSC)O)=O)CCN(C(=O)C(C(C)C)Sc2cccs2)CC12CCC2 N1(C(C2N(CC)CC2)=O)CCC2(CCCC2NC(C2CCCC3CC23)=O)CC1 C1(CNC(CSCC#C)=O)N(C(C2CCC(=O)N2CCC)=O)CCC1(C)C C1(C(=O)NC2CCN(C(C=CC(C)(C)SC)=O)CC2)Cc2nccn2C1 CC(CNC(=O)CC1CC1(Cl)Cl)CN(C(=O)Cc1cnco1)C CN1C(=O)C(=O)N(CC(=O)NCc2ccnc(N3CCNCC3)n2)C1=O C1(C(N(C2CCSC2)C)=O)(CNC(C2CCC2)=O)CC2(CC2)C1 N1(C(CNC(c2cnc(CC)o2)=O)=O)C(C(N)=O)CCC1C c1(C(=O)NC(C2CCN(C(CS(CC)=O)=O)CC2)C)ccnc(F)c1F C(CCCCCNC(=O)CCc1cnn(C)c1)NC(C1C(CC)CCC1)=O c1(NC(C2C(NC(C(F)OC)=O)CCCCC2)=O)cccc2cccnc12 C1(CNC(CC(C)OC)=O)CC2(CO1)CN(C(=O)C(C)(F)c1ccccc1)C2 N#Cc1c(NC2CC3CN(C(C4CCC(N=[N+]=[N-])CC4)=O)CC23)ncnc1Cl N1(C(C2(C)CC2)=O)CCC2CCCN(C(c3c[nH]c(=O)c4ccnn34)=O)C2C1 N1(C(COCCCCC)=O)CCC(N(CCC)C(C2(C)CCOC2C)=O)CC1 c1(C(C(=O)N(CCC)CCNC(=O)CC2(OC)CCC2)C)c[nH]c2ccccc12 Cc1ccc(O)c(C(N2CCC(NC(=O)Cc3ccco3)CC2)=O)c1 C1(CN(C)C(C2CCCN2C(=O)Cc2cncs2)=O)CCCC2CC12 C(C(C)(C)Cc1ccccc1)SCCNC(CN(C(COCC)=O)C)=O N1(C(CC2C(CNC(C3CN(C(C)=O)C3)=O)C2)=O)CCOCC(C)(C)C1 C(C(C)(C)CNC(=O)CC1CC1(Cl)Cl)N(C(=O)Cn1ccc(C(F)F)n1)C N#Cc1ccc(Br)c(C(=O)NC2CCCC2NC(c2cnco2)=O)c1 c1(Cc2cn(-c3c4ccc(OC)cc4ncc3)nn2)nc2c(cc1C#N)COCC2 N1(C(c2cc(OC)nn2C)=O)CC(C2(NC(=O)Cn3cc(C(C)O)nn3)CC2)C1 c1(CC)c(C(=O)N(C)CC2CCCC2NC(C2CSCCS2)=O)ccn1C CC1CCC(CCNC(C2(CNC(=O)C(N)=O)CC3(CC3)C2)=O)CC1 N1(C(CC2(C)CCCO2)=O)CCC(C2(NC(=O)C(F)=CCCF)CC2)CC1 c1(OC)cc(OC)c(NC(=O)CCC(C2CCC2)NC(=O)C(=O)N)c(OC)c1 N#CC1(O)CC(C(=O)NCC2(N3CCNCC3)CCCC2)C1 C1(C(=O)NCCNC(C2CN(C(C3C(C)(CC)C3)=O)C2)=O)CC2(CC2)C1 CCCCC(CNC(C1CC1C#N)=O)NC(c1ccoc1CC(N)=O)=O Cc1c(C(=O)N(CC(C)(C)NC(=O)CC(C)C(F)F)C)cc(C(C)C)n1C c1(NCCC(C)(C)N(C)C)cc(=NCc2ccc(S(C)=O)cc2)[nH]cn1 N12CC(C1)NC(=O)C1(CC1)CNC2=O.C(C(F)F)OC(C)=O Cc1oncc1C(=O)N(CCCNC(=O)CN1CCC1)C(C)C N1(C(c2c(CC)cnn2C)C(=O)NCc2cccs2)CCCNC(=O)C1CC(C)C N1(CCOC)CC2CC1CN2C(=O)CNC(c1ccco1)=O C(C(=O)NC(C)CCO)(C1(O)CCC1)NC(C=CC(C)C)=O N#Cc1ccc(C(N2CC3CCC(NC(=O)CC(F)(F)F)(C3)C2)=O)c(O)n1 C(=O)(C#CC1CCCCO1)NCC1C(NC(c2ncc(C)cc2F)=O)CCC1 C(=O)(C(O)C(C)(C)C)N1C(CN(C)C(c2ncc(Br)cc2F)=O)CCCC1 CC(C)(O)C#CC(=O)NC(CNC(=O)C(C)(C)CC1CCOC1)CO N1(C(c2nc(C)n(C)c2)=O)CCCC(C)C1CNC(=O)C(F)OC(F)(F)F C1(CC=C)(NC(=O)Cn2ncnn2)CCN(C(=O)CSc2ccc(C)cc2)CC1 C12CC=CCC1C(=O)N2CC(C)(C)C.C(C(C)C(=O)OC(C)(C)C)OCC CC(C)C(C(=O)NOCC(F)(F)F)NC(=O)CCCCC1CC1 N1(C(C=NOC)=O)CCC2(CC1)CN(C(c1conc1C1CC1C)=O)CCO2 CC1(C)CN(C(=O)C2=CCCO2)CCC1NC(=O)C(C)(C)C1CCOC1 C1(NC(=O)NCC(C(=O)OC)OCCOCCCOC2CC2)CCCNS1(=O)=O N#Cc1cc(Br)ccc1C(=O)NC1CCN(C(C23CCCC2C3)=O)C1 C(=O)(CC(C)(C)CC(=O)N1CCC2C1CCCN2C(=O)Cn1ccnc1C)OC N1(C(CNC(N)=O)=O)CCC2CCN(C(=O)Cn3c(-c4cccs4)nnc3S)C2C1 n1(CC(=O)N(CCOCC=C)C)ncc(C#N)c1N C(N=c1[nH]c2c(c(=NC(C)C3CCOCC3)[nH]1)COCC2)C1(CC(C)C)CC1 c1(CC)nc(C)c(C(=O)N(CCCNC(c2ccncc2C)=O)C2CC2)s1 N1(C(C(C(C)C)O)=O)CC2CC1CN2Cc1cccc(-c2cncnc2)c1 C#CC(C)(C)C(=O)NCC(C1CC1)N(C(=O)C(C1CCOCC1)O)C C1(N(C)C(c2cnn[nH]2)=O)CCN(S(=O)(=O)Cc2ccccc2)CC1 CC(C)(C)C(C(=O)NCN)NC(c1ccncc1-n1cccn1)=O C(=O)(C(C)(F)C(C)(C)F)N1CCN(C(CCCCC)=O)C(CC(=O)NC)C1 C1(C(N2CCC(C)(NC(=O)C(=O)N=S(C)(C)=O)C2)=O)CCCN(S(N)(=O)=O)C1 c1(C(=O)NC(C)CCCNC(C2(c3cccnc3)CCC2)=O)ccncc1F O=C(O)C(CNc1ccccc1Cl)C(=O)N1CCCC1CC(F)F CC1CN(C(=O)CCCNC(C2CC=CCC2)=O)CC1NC(=O)C(C)CO n1(CCNC(=NCC)NCC2CCS(=O)(=O)C(C)(C)C2)c(=O)oc2ccccc12 C1(CC(=O)NC(C(CC)C)=O)CN(C(=O)CN(CCO)CCO)CCS1 C1(C(=O)NC(C)CCN(C)C(c2cncc(N)c2)=O)CCS(=O)(=O)C1(C)C c1(C(N(CC(C)NC(=O)C(C)(c2ccccc2)N(C)C)C)=O)cncn1C C(C)(CCCCNC(=O)Cc1cn(C)nc1C)NC(COCC#C)=O CC1C(NC(=O)C(C)(C)CC(F)F)C2CCN1CC2 N1(C(CN(CC)CC)=O)CC(CC(=O)N(C)CC2CN(C)C2)C(C)C1 C1(CNC(=O)C2=CCCCCC2)CN(c2ccncc2C#N)CCC12CCOC2 O=C(CC1C2CCCC2N1C(=O)CC1CCCNC1=O)N1Cc2ccccc2CO1 CC(C)C(C#N)C(=O)NC1C=CC(CNC(c2cnn(CCO)c2)=O)C1 C(=O)(C(C)C(C)COC)NCc1c(C(N(CC(=C)C)CC(=C)C)=O)cccn1 CCC(C)C(C)C(=O)N1CCC(C)(CNC(c2cc(Cl)ccc2N)=O)CC1 C1(N)CC2CC(C1)N(C(=O)C=CC=C(Cl)Cl)C2.CCCCCC=CCC=O c1(CN(C)C(=O)NCC2CCN(c3nc(Cl)ncc3F)C2)ccc(F)c(F)c1 CCC(CCC(C)C)NCC(O)COc1ccccc1Br Cc1ccc(CCC(=O)NC23CC2CN(C(=O)Cc2cccnc2O)C3)cc1 O=C(C1CCCc2nnnn21)NC1CCOC2(CCC2)C1 C(=O)(C(C(C)(C)C)NC(c1cc(OC)cc(F)c1)=O)N1C(C)(C(=O)OC)CCC1 C(CC(C)C(=O)N1CCCC1(C)CCC(=O)NCC1(C)CCCC1)=CC CN1C(=O)CCCC1C(=O)NC1CCCCN(C(=O)C(C)(C)c2ccno2)C1 c1(C(=O)NC(CC)CNC(c2cccnc2O)=O)ccc2c(c1)CC(C)O2 c1(NC(CCN(C)Cc2cccc(NC)n2)=O)ccc(C#N)c(Cl)c1 C1(C)(C(=O)NCCC(C)N(C(c2cnc(OC)nc2)=O)C)CCCNC1=O C(C(C(C)C)NC(=O)C(F)(F)c1ccccc1)NC(CSCC#C)=O C1(C(C)C)COCCN1C(C1(CN(C)C)CCCN1)=O C1(NC(c2c(C)cco2)=O)CCCCC1NC(=O)C(=O)N(C)C c1(CCNC(C(=O)Nc2cccc(-c3ccsc3)c2)=O)ncc(F)cc1F CC1(C)CC(CO)CN(CC(=O)Nc2cnc(Cl)c(F)c2)C1 C1(CNC(C(CSC)C)=O)CC2(CC2)CN1C(c1c[nH]c(C)cc1=O)=O CCC(CNC(c1ccsn1)=O)(CC)NC(C1CCN(C2CCCC2)CC1)=O C1(F)(CNC(C(c2ccccc2)OC)=O)CCN(C(=O)C(C)(F)F)CC1 CCC(CC(=O)N1CCC1Cn1cc(C2CC23CC3)nn1)C(F)F N1(C(CCC)=O)CCC(OCCNC(=O)C(OC)OC2CC2)C1 C1(C(N(CC(=O)NOC(COC)COC)CC#C)=O)CCOC(C)C1 C=CCC(C(=O)NC1CCC(NC(=O)C(CO)NC(=O)CCC)C1)C(C)C C(=O)(C#CC(C)(C)C)N1CC(C(C)NC(c2csc(-c3ccccc3)n2)=O)C1 Cc1cc(=NCC(C)NC(=O)C(=O)Cc2cccs2)[nH]c(C(C)(C)C)n1 C(C)(C)(C(=O)NCc1cn(CC(C)NC(=O)C(=O)N(C)C)nn1)OC(C)C c1(CNC(C(=O)Nc2ccc(C)c(Cl)c2F)=O)sc(Br)c2c1OCCO2 n1(CCC=C)cc(C2CCCN2CCC2CCC2)nn1 C1(OC)CC(CNC(=O)C(C(C)C)n2cnnn2)N(C(=O)CC2CCOCC2)C1 c1(NC(CCCCCCn2cc(C(C)OC)nn2)=O)ccc(S(C)(=O)=O)c(C)c1 c1(C(N2CC(C)C(NC(C3(O)CC3(C)C)=O)C2)=O)coc2c1N(C)C(=O)CCC2 N1(C(CCC)=O)CC(O)C(O)C1CNC(=O)CC1CCN(C)C1=O C1(C(N(C)CC2CCN(C)C2)=O)C2CC1N(C(=O)CC1CCCN1C)C2 C(=O)(C1=Cc2ccccc2C1O)NCC1(NC(C2=CCC(C)CC2)=O)CCCC1 N1(C(=O)C=CSc2cccs2)CCOCC(CNC(C2CC(OC3CC3)C2)=O)C1 CCC(CO)C(=O)NCCCCC(C)NC(c1scnc1C1CCCC1)=O C1(NC(c2cscc2Br)=O)CN(C(=O)CCn2cccn2)C2(CCC2)C1 C1(CCOC)CN(C(c2sc(=N)[nH]c2C)=O)CCN1C(c1ccn(C)n1)=O C(CCF)(C(=O)NCCNC(=O)C(C)C)NC(c1c(CC)c[nH]c1)=O N1(C(C)=O)CCC2(C1)CN(C(=O)CC1COc3ccccc31)C2.C=O N1(C(C2C(=C)C2)=O)CCCC(C2(NC(C3CC(O)C3)=O)CC2)C1 N1(C(c2nocc2C)C(=O)NCCCCCC)CCc2c(Cl)cccc21 N1(C(C2(C)C(C(=O)OC)C2)=O)CCC2(CC1)CC(NC(=O)CCCC(C)C)C2 C(=O)(CCCCC(F)F)N1CCC(CCNC(=O)CSCC2CCCCO2)C1 CCC(CC(F)(F)F)C(=O)N(C(C)CNC(=O)C(F)C(C)(C)O)C N1(C(C(CC)CCc2ccccc2)=O)CC2CCC1CN2C(=O)C1=CC(C)(C)C1 N1(C(c2n(C)c(O)nc2)=O)CC2CN(C(C3CC3C#N)=O)CCC2(CO)C1 C1(C#N)(C(N(CCNC(=O)C(c2cccc(OC)c2)(F)F)CC)=O)CCCCC1 C(=O)(CC(C=C)CC)NC1(CC=C)CCN(C(c2nccnc2Cl)=O)C1 c1(CN=C(NC(C=C)C)NC2CC2C2CC2)cc(OCC)c(O)cc1C O=C(C1=CC2(CCN(C(=O)CCNC(N)=O)C2)C1)N1CCC(C2CC2)C1 CN1CCc2cc(C(=O)NCC3CC(NC(=O)C4=CCCC4)C3(C)C)ccc21 C1(CC)CC(O)(CNC(C2(NC(=O)CCOCC(C)(C)C)CCC2)=O)C1 C(=O)(CC(CNC(c1ccc(F)c(F)c1C)=O)C(C)C)OC C(=O)(C#CC1CCOC1)NCCC(C)NC(c1c(C)oc(Br)c1)=O N1(C(CC(C=C)(C)O)=O)CCC(O)(C2(NC(c3cnccn3)=O)CC2)CC1 C12(CNC(CN3C(C)CC3)=O)CCC(CC1)CN2C(=O)C(O)CCn1cncn1 c1(C(N2CC3(C2)CN(C(c2csc(-c4ncc[nH]4)n2)=O)C3)=O)ncc(Cl)cc1Cl C1(CNC(c2c(CC)occ2)=O)CC(NC(c2c(Br)cnn2CC)=O)CC1O c1(C(N2CCCC(C)(CNC(C(C)C3CC3)=O)C2)=O)cc(C#N)ccc1F c1(C(=O)NCC2C(NC(CCN(C)CC)=O)CC2)noc2ccc(OC)cc12 c1(CC)ccc(O)c(C(=O)NCCN(C(C2CCSC(C)C2)=O)CC)c1 C(c1c(Cl)cccc1Cl)=CC(=O)NC1C(F)CCN(C(CCOCCOC)=O)C1 c1(C(N(C2CCN(C(=O)CSC(F)(F)F)C2)C)=O)cc(C(N)=O)ccn1 C(N=c1[nH]c(N2CCOC(C(C)C)C2)nc2cc[nH]c12)C1CC(NC)C1 C(=O)(C(C)C(CC)CC)N1CCC(N(C(c2nc(CC)oc2)=O)CC)C1 c1(C2N(C(=O)NCCc3cc(=N)[nH]o3)CCC2)ccc(Br)cn1 N1(C(NOC(C)(C)C)=O)CCCC(C(=O)NC2(C)C(NC(=O)C3CC3)CC2)C1 N1(C(CCOC)=O)C2CCC1C(CNC(=O)Cc1cccc(NC(C)=O)c1)C2 c1(C(=O)NCCN(CCOC)C(C2CCOC2)=O)ccc(Cn2cccn2)cc1 N1(C(C(C2CC2)OC)=O)CCCC1C=CC(=O)NC(CC)C(C)CN(C)C C(=O)(C1c2c[nH]nc2CN1C(c1cnc(=N)[nH]c1)=O)NCC(C(=O)NC)(C)C c1(COC)nc(OC)cc(N2CCC(F)(C(=O)OC(C)(C)C)C2)n1 C1(NC(C(C)=CC2CC2)=O)CCSC12CN(C(C13CCC(F)C1CC3)=O)C2 C(CN=c1[nH]n(C)cc1[N+](=O)[O-])(C(C)(C)C)NC(CCc1cnn(C)n1)=O c1(C(=O)NCCC(C)(C)NC(c2occ(C)c2)=O)cc2n(n1)CC(F)C2 n1(C(C(=O)NCC)C)cc(CN(C)C(C2(NC(=O)C(CC)OC)CC2)=O)nn1 c1(C(N(CC(C)N(C(=O)CC(=O)c2cnn(C)c2)C)C)=O)ccc(O)cn1 N1(C(c2cc(SC)oc2)=O)CCSCC1CCNC(=O)CC1CCCO1 CN1CC(NC(C2(NC(c3cc(=N)[nH][nH]3)=O)CC2(C)C)=O)C(=O)N1 C1(OC)(NC(=O)Cc2cccc3c2OCO3)COC(C)(C)OC1 C1(C(C)O)CCCCN1C(C1C2CN(C(=O)CC3CCNC3=O)CC12)=O Cc1cc(C(C)C(=O)NCC2CN(C)CCN2C(C2CCCCS2)=O)cc(F)c1 C1(NC(CCOCCCOC)=O)CCCCC1C(=O)NCCCCC1CC1C c1(C(=O)NC2CCC(CNC(C3CCCOCC3)=O)C2)cc2cccnc2[nH]1 Cc1cc(Cl)cc(C(=O)NCCN2CCN(C(c3cc(=O)n(C)o3)=O)CC2)c1O CC(=O)CCCC(=O)NC1CC(F)CN(C(=O)CCN2CCN(C)CC2)C1 N12CCC(O)(CC1)C(=O)N1CCC(CC1)C2=O.N1(CC)CCCC(C(F)(F)F)C1 CCC(CC)C(C)C(=O)N1CC(O)CC1CNC(=O)C(C)=CC1CC1 N1(C(C2N(C(C3CCN(OC)CC3)=O)CC2)=O)CC2CCCC2C12CC2 N1(C(CC=CCC)=O)C(C(=O)NCc2ccns2)CC1C C1(NC(CSCC#C)=O)CCC(CCNC(=O)C(C)SCOC)C1 N1(C(C(c2ccccc2)=O)=O)CC(NC(c2nn[nH]c2Cl)=O)CC2(CCOCC2)C1 C1(NC(C(c2ccoc2)NC(C(CO)OC)=O)=O)CC(=O)N(C(C)C)C1 CCC(N=c1nc(N2CCC(C(=O)NC)C2)c2sccc2[nH]1)c1ccncc1 c1(C(=O)NC2(CN(C(CC3(CSC)CC3)=O)C)CC2)nccc(C)c1N N1(C(C(C)S(C)(=O)=O)=O)CC2CCN(C(=O)C(C)(Cl)Cl)CC(C2)C1 C1(NC(CCC(CC)C)=O)CCCC12CN(C(c1cc(O)ncn1)=O)C2 N1(C(CCSCC)=O)CCC(C)(C)C(C(=O)NC(c2ccco2)CO)C1 N1(C(=O)NC(c2cc(Cl)ccc2Cl)C)CCNCC2(C)CCCC12 C1(CN(C(=O)COC2CCC2)C)CCCCN1C(=O)C(F)(F)c1ccsc1Cl C1(CNC(C(=Cc2ccncc2)C)=O)CCN(C(=O)C(C)OC(C)(C)C)C(C)C1 CCCCCC(O)C(=O)NC12CC(C(=O)NC3CCCC4(C3)N=N4)(C1)C2 CC(CCNC(=O)C(C)c1ccsn1)NC(=O)CCn1cccn1 C1(C)(COC)CN(CC(C2CCC(F)(F)CC2)C)CCO1 c1(C(=O)NCC(CNC(C(C)n2cccn2)=O)O)cc2c(o1)CCCNC2=O c1(NC(c2c(NC(C(c3ccc(F)c(F)c3)C)=O)c[nH]n2)=O)ccc(Br)cc1Cl n1(CC=C)cc(CNC(=O)COC(C)(C)CNC(c2csnc2Cl)=O)nn1 c1(C(=O)NCCN(C(C(CC)F)=O)CCOCCO)oc(C)nc1C Cc1cc(N)ccc1C(=O)NCC(C)(C)CN(C)C(C1CCN1C)=O c1(C(N2CC(CCNC(=O)C(O)Cn3cncn3)(OC)C2)=O)cncc(N)n1 C12(C(N3CC(C)N(C(=O)CC45CNC(=O)C(C4)C5)CC3)=O)CCCCC1C2(F)F C(=O)(C(C(C)(C)C)C(=O)N1CC(O)CO1)N1CCC(C)CC1 C(=O)(C(C)CC(C)(C)C)NCCC(C)(C)NC(CSc1ccc(C)cc1)=O N1(C(c2scc(-c3ccc(C)cn3)n2)=O)CCc2nc[nH]c2C1 CC(N=c1ccnc(NC(c2cc(F)c(F)c(F)c2)CO)[nH]1)c1ccc(O)nc1 Cc1nc2oc1NC(=O)N1CCCC2C1.C1(C(N)=O)CN(C2CC2)CC1C CC(CC(=O)NC(=O)C(F)(F)F)NC(C1CSCN1C(=O)C(C)(C)C)=O C1(CCNC(c2c(OC)nsc2)=O)CCCN(C(C2CC(C#N)(OC)C2)=O)C1 N1(C(c2ccn(C)n2)=O)CCC(CNC(=O)C(F)CC2CCC2)CC1 C1(C(N2C3CN(C(CCC(C)SC)=O)C(C3)C2)=O)Cc2ccccc2C1 CC1CCCC1C(N1CC(CCNC(c2cnc(O)o2)=O)C1)=O C1(n2cccc2)(C(=O)NCC2C(NC(=O)Cc3ccco3)CCC2)CCCC1 N1(C(C23CC(C2)C3)=O)CC2CN(c3nnc(CO)s3)CC2C1 N1(C(C)C)CCN(C(=O)NCC(C2CCOCC2)F)CC1C C1(CC(N2CC(C(=O)NCC)C2)=O)CCCCC1NC(c1cn(C)c(C)n1)=O N1(C(c2c[nH]c(=N)s2)=O)CC2(CCCCN(C(c3cc4ncccc4s3)=O)C2)C1 C(=O)(C(=O)N=c1nc(CS(C)(=O)=O)[nH]o1)OC(Cc1ccc(OC)cc1)C C1(NC(c2c(C)nc[nH]2)=O)CN(C(c2ncccc2C2CC2)=O)CC1(C)C Cc1cc(-n2cc(C3CCCCN3C(=O)CN3CCOC3=O)nn2)cc(C)c1Br S(=O)(=O)(c1cccc2nsnc12)NC1CCN(CCN(C)Cc2cccnc2)C1 c1(C(C2CCC2)N(C(=O)CCn2cc(C3CC3)nn2)C)cc(P(C)(C)=O)cs1 c1(CC(=O)NCC(CNC(C2CCN(CCC)CC2)=O)O)nsc2ccccc12 N1(C(CN(C2CCC2)C)=O)CCC2(CC1)CC2C(=O)NCCC(O)C(F)(F)F c1(CN=C(NC(C=C)CC)NC2CC(=O)N(CCC)C2)cc(Cl)ccc1N(C)C N(C(=NCCc1cc(OC)ccc1C)NC1CCCC(F)(F)C1)C(COC)C c1(C(=O)NCC2CCCCN2C(=O)CCCCCF)ccn2cncc2c1 c1(NC(c2cnn(C)n2)=O)cncc(CNC2COCCO2)c1 N1(C(COCC(C)C)=O)CCCCC(N(C)C(C2CN(C(C)C)C2)=O)C1 C1(NC(c2cnc(C3CCCC3)s2)=O)CCCCN(CCCC2CCOC2)C1 N1(C(C(CSC)OC)=O)CC(C2CCCCN(C(c3ccc(Cl)c(F)c3)=O)C2)C1 CN1CCCC1(C)C(=O)NCC(c1ccccc1OCc1ccccc1)N(C)C C1(CNC(C2CCCCO2)=O)CC12CCN(C(c1cc(F)n[nH]1)=O)CC2 c1(C(=O)NCC2N(C(C(CC)Oc3ccccc3)=O)CCC2)cnc(N)cn1 c1(C(N(C)CC2(CNC(c3c(C)cccn3)=O)CC2)=O)ccc2nncn2c1 Cc1nc(C)c(CC(=O)NC2C=CCN(C(=O)CC3(O)CCOC3)C2)s1 CC1(C)CN(C(C2(O)CCCCCC2)=O)CC(C)(C)S1(=O)=O S(=O)(=O)(c1ccc(F)c(Cl)c1)N1CC(F)CC(Nc2ncc(N(C)C)cn2)C1 C1(CC(C)NC(CC=C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1 c1(C(N(CCN(C(=O)COC(F)(F)F)CC)CC)=O)ccc(C)c(O)n1 c1(C(=O)NC2CCc3n(C)ncc3C2)cc2cc3c(cc2[nH]1)OC(F)(F)O3 C(=O)(CC1C(=O)Nc2c(F)cccc21)NC(CN(C(c1csc(C)n1)=O)CC)C c1(C(=O)NC(CNC(c2c(C)coc2)=O)CO)ccc(-c2nnc(O)o2)cc1 C1(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CC2CCC(C1)N2c1ncnn2cccc12 C12(CNC(CCCCC)=O)CCCCC1N(C(c1cccnc1F)=O)CC2 Cc1csc2c(CC(N3CCCC3C(=O)N(C)C3CC3)=O)cccc12 N1(C(C(C)OCCCC)=O)CCC2CN(C(c3cc(C#N)ccc3F)=O)C(C)C12 c1(CC)ccc(OCC(=O)NCC(C)N(C(=O)CC2CCC23CCC3)C)cc1 C(=O)(CCCCCF)N1CC(CNC(c2ccc(CCCC)cc2)=O)C(O)C1 Cc1ccncc1C(N1CC(NC(c2cccnc2O)=O)C(C)C1)=O C1(CNC(C=CC)=O)COCC1NC(=O)CSc1nncn1C(C)C Cc1cc(C(=O)NC2CCN(C(=O)CCn3cccn3)C(C)C2)ncc1Br C1(F)(CN2CC(C)(OC)C2)CCC(NC(=O)CC(=O)N(C(=O)CCS(C)=O)C2CC2)C1 C1(NC(CNC(=O)OC)=O)CCOC(C(=O)NCC2CC(N(C)C)C2)C1 CC1CN(C(=O)CN(C)C2CC2)CCN(C(=O)C(c2ccccc2)C)C1 N1(C(Cc2c(OC)nccc2)=O)CCC(NC(=O)Cc2csc(C)n2)C(F)C1 N1(C(CCCCC)=O)CCCOC(CNC(c2n[nH]cc2Br)=O)C1 N1(c2nc(C)nc3c2cc[nH]3)CCC2(CN(C(C3CCCC3O)=O)CC(C)O2)C1 C(CN=C(NCC1CC1)NC1CCC(C)(C(C)C)CC1)C1CCC(OC)CC1 C(=O)(C1Cc2ccc(F)cc21)NC1(C2N(C(C3C(C)C3C)=O)CCC2)CC1 C1(NC(CCCN(C)C)=O)CN(C(c2c(Cl)ccc(O)c2N)=O)CC2(CCC2)C1 c1(C(N2C(CNC(c3cnc(Br)s3)=O)CCC2)=O)nc2ncccn2n1 c1(C(=O)NC(CC=C)CNC(=O)C(C)CN(C)C)cc2nccnc2[nH]1 c1(C(=O)NCC(CC)(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)ccc(C)c(Cl)c1F N1(C(CC(C)NC(c2ccn(CCC)n2)=O)=O)CC(=O)NC(=O)C1C c1(OC)ccc([N+](=O)[O-])c(C(N2CC3C(NC(=O)CCC#N)C3C2)=O)c1 CC1(C(=O)NC(CNC(C2CCCN2N=O)=O)C2CCC2)CS(=O)(=O)C1 C1(C(C(=O)N(CC=C)C)C)CCCN(C(C2CN(C(C)=O)C2)=O)C1 c1(CN2CC(NC(C3Cc4ccccc4O3)=O)C(F)C2)c[nH]c2ncc(Br)cc12 CC1CCC(CNC(=O)C(C)(C)C(F)F)CN1C(c1coc(C#N)c1)=O C1(NC(CC2(C)CC2(F)F)=O)CCN(C(c2ccncc2N)=O)C1C1CC1 C(=O)(C(C)CCC(C)(C)C)NCC1(CNC(CSCC#C)=O)CCC1 CC1CC(NC(C2CCC3(CC2)CC3)=O)CCN1C(=O)COC1(C)CCCC1 C1(CC=C)(C(=O)NC2CCC2NC(C)=O)CN(C(=O)CCCOC(C)=O)C1 Cc1cccc(C)c1C(=O)NC1CC2(C1)CC2NC(=O)CC1(C)CC(F)(F)C1 C1(N(C(C2(COC)CCCC2)=O)CC)CCCN(C(c2cc(F)ccc2F)=O)CC1 c1(OC)ccc(C(=O)NCCOCCS(C)(=O)=O)c(Br)c1F c1(N2CCC(CC=C)(NC(=O)CC3COC(C)(C)C3)C2)cc(C)nc(COC)n1 C1(NC(C2C(C(=O)OC)C=C2)=O)CC2(CCC2)C1OC C1(CN2CCC(NC(c3c(C(=O)OC)c(C)[nH]n3)=O)C2)CCC(F)(F)CC1 CC1(C)OCc2c1n[nH]c2C(=O)NC1CC(NC(c2cnc(S)nc2)=O)C1 N1(C(CCC2CC(C)C2)=O)CCC(CC(=O)Nc2cc(CO)cc(F)c2)C1(C)C C1(OC(C(CC)Oc2ccccc2)=O)CCCCC1n1cc(C(=O)O)nn1 C#Cc1ccnc(C(=O)NCCN(C(=O)CCc2nncs2)CC(C)O)c1 N1(C(c2c(C)csc2Cl)=O)CCOCC(NC(=O)C(C)(C)C)C1 C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)CN2C(=O)CCC2=O)C1 c1(C(=O)NCCc2c(CNC(CC3C(C)OCC3)=O)nco2)c(F)ccc(F)c1Cl C1(CNC(CC(CC)C2CC2)=O)CCC2(CN(C(c3cc(CC(C)C)c[nH]3)=O)C2)O1 CC1(C)CC=C(C(=O)NC23CCC2CN(C(c2ocnc2C2CC2)=O)C3)CC1 C(CCCCN(C)C(C12CCC1CC2)=O)NC(CC=CCC)=O CC(C)(O)CC(=O)NC(Cc1ccco1)C(N1CC2CCC1C2)=O C1(F)(C(N2CCC(OCC(C)C)C2)=O)CCCN(C(=O)CC2COCC(C)O2)C1 N1(C(C(c2cccc(C)c2)C)=O)CC2(CNC(c3c[nH]nc3C)=O)CC(F)(C1)C2 c1(OC)cc(C)cnc1C(N1CCCC(CNC(=O)C(O)CSC)CC1)=O C1(NC(C(C)N(C(=O)Cc2ccns2)CC)=O)CCCC2(CC1)CC2 N1(C(C2CCCCN2Cc2cccnc2)=O)CCC(C2CCOC2)CC1 C(=O)(C1=NN(c2ccccc2)C(C(=O)NCc2coc(C)n2)C1)OC C(=O)(C(C)(F)C(C)(C)F)N1CCC(C2NCCCC2)C1.c1(CC)c(F)ccnc1F C(=O)(C(C)CCCC(C)C)NC(C(C)OC)CC(N1CCOCC(C)(O)C1)=O Cc1ccc(CNC(=O)COC2CN(C(c3ncccc3N)=O)C2)c(F)c1 CCC(C)(CNC(=O)CCOCCOC)C(=O)NCc1cc(C)nn1C CCCC(C)(CC)C(=O)N1CC(C)C(C)(CNC(=O)CCCc2ccccc2)C1 N1(C(C=CC(=O)N(C)C)=O)CC(F)(F)CC1CO.c12cc(no1)C(=O)NC2 c1(C(=O)NCC=C)ccc(C(N2CC(NC(c3ccc(C)o3)=O)C(C)C2)=O)cc1 CN1CC=CCC1CC(=O)NCCN(C(C1(CF)CC1(F)F)=O)C1CC1 c1(C(N2CCC(CNC(C(COC)OC)=O)CC2C)=O)ccc2ccccc2c1 C=CCC(CC=C)NC(C)(COCc1cccc(Br)c1)c1nnnn1C1CC1 CCCC(C)(O)CC(=O)NC12CCCC1N(C(c1cnc(C(C)C)s1)=O)CC2 C(=O)(C1=COCCO1)NCCCN(C(=O)CCc1c(F)cccc1F)C C1(C(N2CC(OC)(CNC(C3(C)CCCN3C)=O)C2)=O)CCCCCC(=O)C1 C1(C(N2C(C)CCN(C(c3c(C)cc[nH]c3=N)=O)CC2)=O)CC2CCC(C1)N2C Cc1nnc(CC(=O)NC(C)(CNC(=O)C(F)(F)c2cnn(C)c2)CO)o1 c1(C(C)C)ccc(C(=O)NCC2CC2CNC(C2CC(n3cnnc3)C2)=O)s1 N1(C(CSC)=O)CCN(C(=O)C(=O)N(C)C)C(c2ccccc2)C1 C(CC(C)C(=O)NC(C1CCN(C(=O)CCc2cccnc2F)C1)(C)C)OC c1(C(N2CC3(CC(NC(C4CCC5(CCC5)C4)=O)C3)C2)=O)cnc2n1CCOC2 Cc1cc(O)c(C(N2CC(N(C(=O)CN3C(=O)CCC3=O)C)C2)=O)nn1 C1(=O)N=C2N=CN(N2)CCC(=O)N(Cc2ccccc2)C(C)CN1C.N(C)C.N(C)C c1(C(N(CCNC(=O)COCCSC)CC)=O)ccc(-n2ccnn2)cc1 C1(NC(CC(CC)(C)C)=O)CN(C(c2cc(C(F)F)ncn2)=O)CC12CCC2 C1(C(=O)N(C)CCNC(=O)Cc2ccc(NC(C)=O)cc2)(COC)CCC(=O)N1 C=C1CCN(C(=O)C(C)C(F)F)C(C(=O)N(C)Cc2nccs2)C1 c1(C(=O)NCC2N(C(C=C3CCN(C)CC3)=O)CC=C2)csc2nccn12 c1(CCC)nc(C)c(C(N2CCCC2C2(NC(c3cnn(C)n3)=O)CC2)=O)o1 c1(C(=O)NCC(C)CN(C)C(c2ncc(F)cn2)=O)ccc(N)c(Br)n1 C1(CNC2(C)CCOCC2)CN(CCSc2ccccc2)CCCO1 C(N=c1nc2sccc2c(NCC23CCCN2CCC3)[nH]1)C1COCC(C)(C)O1 C1(C(C)C)C(=O)N1.c1(OC)cc(C(=O)NC(CC2CCC2)CO)on1 c1(C(=O)NC(C(C)NC(c2c(C)con2)=O)CO)cnn(-c2ccccn2)c1C C1(NC(C2N(C)C(=O)CCC2)=O)CCC2CCN(C(C3(n4ccnn4)CC3)=O)C12 C1(NC(C(=O)NC2(c3cccc(C)c3)CCCC2)=O)CCCNCCC1(F)F N1(C(c2cccc(-c3cnco3)c2)C(=O)NC(CC)C)CCC2(CCCOC2)C1 CC1(C)CC(CNC(C2C=CCCN2C(=O)CCc2csnn2)=O)CC1 c1(C(N2C3CN(C(CC(C)=C(C)C)=O)C(C3)C2)=O)cc2ccc(N(C)C)cc2[nH]1 c1(OC)ccc(N)c(C(=O)NC2C3CC2CN(C(C2CC4CC4C2)=O)C3)c1 N1(C(=O)NCCC2C(C)C(=O)CC2)CCCC2(C1)OCCCO2 C(=O)(C(F)CC(C)(C)C)NCc1cc(C(N2CCCC(C=C)C2)=O)sc1 Cc1cc2ncnc(N3CC4C(CNC(c5ccccc5COC)=O)C4C3)c2[nH]1 c1(C(=O)NCCN(CCOC)C(C2CCCCC2OC)=O)c(C)cncc1C N1(C(c2c(NC)cnc(Cl)c2)=O)CCC(NC(=O)C(CCC)N(C)C)C12CCC2 c1(OC)nccc(C(=O)NCCCCN(C)C(c2sccc2CC#N)=O)c1F N#Cc1c(F)cc(C(=O)NCC2(NC(c3cnc(O)o3)=O)CC2)cc1F C1(C(=O)NCC(CC(C)C)OC)CCCN(C(C2C3CCC(F)C23)=O)CC1 c1(C(=O)NCC(CC)(C)NC(C2CC(C(=O)OC)C2)=O)ccc(Cl)cn1 C(C1(C)CCOCC1)=CC(=O)NCC(C)CNc1ncc(Br)cn1 c1(N2CCCC(C(C)NC(Cc3c(CC)cccc3)=O)C2)nc(C)ncc1F CN(C)S(=O)(=O)NCC(N1CC=CC(NC(C2CC2c2ccccc2)=O)C1)=O CCCCC(CNC(c1cc(C2CC2)ncn1)=O)NC(c1cc(CC)c[nH]1)=O C(=O)(C1CCCc2ccccc21)N1C(C)CCC(NC(c2c(CC)cco2)=O)C1 C1(CC=C)(NC(=O)C=CC(C)(C)C)CCN(C(=O)CCS(N)(=O)=O)CC1 c1(N(C)Cc2cccc(F)c2F)nc(N2CCCCCCCC2)c2c(n1)COC2 C1(NC(COCC=C)=O)CCN(C(=O)CN2CC(=O)NC2=O)C(C2CC2)C1 c1(N(C)CC2CCCN2C(=O)C#CC2(C(F)(F)F)CC2)ncc(C#N)cc1F N1(C(C2(COC)CC2(F)F)=O)CCC(F)(CNC(c2cccnc2C)=O)CC1 C1(NC(C(C)(N(C(c2c(C)cns2)=O)C)C2CC2)=O)CCCCC1(F)F Cc1cc(C(N2CCCC(CN(C)C(C3CCCSS3)=O)C2)=O)cc(C)c1 Cc1c(C(N2CC3(CCC3NC(c3sccc3F)=O)C2)=O)cncc1Br N1(C(c2cnc(C)o2)=O)CCC(NC(=O)C(C)(O)c2ccccc2)C(F)C1 Cc1cc(C(=O)NCC(Cc2ccccc2)NC(=O)C=CCO)cn1C(C)C C12(CCSCC1)n1nnnc1C2NCC1(CC)CC1.c1(C2CC2)ccc(F)cn1 Cc1cc(O)ccc1CC(N1CC2CC2(NC(=O)CC(C)NC(=O)C2CC2)C1)=O C1(C(=O)NC2(CO)CC2)CC2(CC2)CN1C(=O)CC1CCCOC1 N1(C(Cc2cnc(C)[nH]2)=O)CC(CNC(c2ccc(Cl)c(N)c2)=O)C(C)(C)C1 CCCCCCCCC(=O)N1CC=C(CNC(C2CN3CCCC2CC3)=O)CC1 N1(C(C(C)CN(C)C)=O)CCCCCC(NC(=O)COCC2CCCC2)C1 C1(CC(=O)OC)CCCN(C(N2CCC3(CC2)CC3)=O)CC1 c1(C(N(C2CCN(C(=O)CSc3cccs3)C2)CCCC)=O)ncccc1SC c1(C(=O)NC2CCN(C(C(CC)COC)=O)CC2)ccc(SC)cc1OC CCC1=C(C(=O)NCC2CCN2C(=O)CC(C)OC)CCCO1 C(=O)(CCCCC(C)(C)C)NC1CCCN(C(CSCCCC)=O)CCC1 N1(C(C2C(OC)C2)=O)CCC(OCCNC(=O)CN(n2nccn2)C)CC1 C1(CNC(CCC=C)=O)CN(C(c2ccncc2-c2ccccc2)=O)CC1(F)F N#Cc1ccc(C(=O)NCC2CCN(C(c3ccnnc3C3CC3)=O)C2)o1 N1(C(C2CN3CCC2C3)=O)CCC2(C1)CN(C(C1CCCCO1)=O)C2 C1(C2CCN(C(=O)CNC=O)CC2)(C(=O)NCC(CCC)O)CCOCC1 C12(NC(=O)CCCc3nccs3)CCCC1(F)CN(C(=O)CCn1cncn1)C2 c1(C(=O)NC2CCCC(CNC(=O)C=C3CCCCC3)C2)c(F)ccc(F)c1O c1(NC(C(CC)NC(=O)Cc2cc(C)cs2)=O)cc(C)c(C)cc1C C(=O)(C1Cc2ccccc21)N1C(C(=O)NCC(C(CC)C)CO)CCC12CC2 Cc1cccn2c(C(=O)NCC3CN(C(C4(C(C)C)COC4)=O)CCO3)cnc12 C1(CNC(C2CC(OC)C2)=O)CN(C(c2cc3ccsc3s2)=O)CC(C)(C)O1 c1(-c2nc(-c3c(OC)n(C)nc3)on2)c[nH]c2nccc-2c1 C(=O)(CS(=O)(=O)C1CC1)N1CC2C(CNC(c3ccc(CC(C)(C)O)s3)=O)(C2)C1 N1(C(c2c(CC)c(Cl)ccc2)=O)CCC2CN(C(=O)Cn3cncn3)C2C1 c1(OC)cc(F)c(CN2CCC(C(=O)Nc3sc(C)cc3C#N)C2)c(F)c1 C1(C(=O)NC(C)Cc2cccc(Cl)c2)CCC(=O)CC1C C1(C)(CN(C(C=C(COC)C)=O)C)CCCC1NC(=O)C=CSc1nc[nH]n1 c1(C(N2CC(CSC)OCC2)C(=O)NCC2CC2)ccc2ccc(F)c(F)c2n1 N1(C(C2CC(NC(CCC3CCC(=O)C3)=O)C2)=O)CCCC(c2ncc[nH]2)C1 Cc1cnn2ccc(C(N3CCCC3C3(NC(C4CCCC4O)=O)CC3)=O)nc12 c1(C(=O)NCC(CNC(C2C(C)OCCC2)=O)C(F)(F)F)[nH]nc2ncccc12 c1(OC)nc(=NCC2CCCN2C(=O)C(C)O)nc(OC)[nH]1 CC1COCC1(C(F)(F)F)NC(c1nnnn1C1CC1)C1CCC1 C(=O)(C(C)C(O)CC(C)C)N1C(CNC(c2c(C)c(F)cnc2)=O)CC2(CC2)C1 C(C(N=[N+]=[N-])C(=O)N(C)CC1CN(C(c2cc(C)cnc2C)=O)C1)OCC c1(C(N2CCC(C(C)NC(C3(C#N)CCC3)=O)CC2)=O)cc(C(F)(F)F)ccc1O c1(-c2nn(CC(=O)NC(C)C)c(CCC(F)(F)Cl)n2)cc(F)c(N)c(F)c1 CC1CCC(C(F)(F)F)CN1C(c1ccc(Br)cc1F)=O C1(C(=O)NC2CCC(NC(C3CC3c3cccs3)=O)C2)(CO)CC(F)(F)C1 C1(CNC(c2c(C)ccnc2)=O)CN(C(=O)Cc2ccoc2)CCC12CCC2 C(CCOCCO)(C(=O)NCCc1ccn(C)n1)NC(C(CN(C)C)O)=O c1(C(N2CC(CNC(CCC=C=C)=O)C3(C2)CCC3)=O)nc2nc(C)ccn2n1 c1(CC)ccc(C(N2CCC(C)C2CNC(c2cccc(C3CC3)n2)=O)=O)cn1 Cc1cccnc1C=CC(=O)NC1CCN(C(=O)Cc2ccnn2C)CC1F N1(C(CCC2(C(N3CC(OC)C3)=O)CC(=C)C2)=O)CC(F)(F)CC1C C#Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(C)(O)COC)ccc1C C1(C(=O)NC2(CCNC(c3cncn(C)c3=O)=O)CC2)CCC2(C1)CC2(F)F N1(C(c2cc(C)ncc2Cl)=O)C2CCC1CN(C(=O)C(C)(C)C1=CCCC1)C2 C12(NC(CCCOCCOCC)=O)CCCN(C(=O)C3=CCCOCC3)CC1C2 c1(NCC(CN(C)C)OC)ccc(S(=O)(=O)NC(c2cncs2)C)c(Cl)c1 Cn1c(C(N2CCC(NC(c3cncc(CO)c3)=O)C(O)C2)=O)ccc1[N+](=O)[O-] c1(C(=O)NC2C(O)CCN(C(C(COC)OC)=O)C2)ccc(OC)c(OC)c1C C(CCCC(C)NC(=O)Cn1ccsc1=N)NC(C=C(C)Cl)=O c1(C(N(CC(C)NC(=O)CCNC2CC2)CC)=O)csc(Cl)c1Cl C1(NCC2CCN(C(=O)NCc3c(CC)cccc3)C2)CC2(CCCC2)CO1 c1(OCC=C)ccc(Cl)c(C(N2CCCC(O)(CNC(c3ccc[nH]3)=O)C2)=O)n1 C1(C2CC2)(CNC(c2cc(OC)c(C)nc2)=O)CCN(C(c2c[nH]nc2C)=O)C1 N=c1ccc(C(=O)NC2C=CC(CNC(c3cn(CC(F)F)cn3)=O)C2)n[nH]1 c1(NC(C2CS(=O)(=O)CC2N2CCOCC2)=O)nc2cccc([N+](=O)[O-])c2s1 c1(C(C)NC(C(=O)NCCCC)CC)ccc(OC)cc1 c1(C(=O)NC(CNC(C(C=C)(C)C)=O)(C)CO)cc(C)cc2c1NCCC2 Cc1cccc(N)c1C(=O)NC1CC(O)CN(C(=O)CC2CSCCS2)C1 C1(C(=O)NCC2C(C(F)(F)F)CCN(C(CSC)=O)C2)CCc2nn[nH]c2C1 Cc1cc(C)c(C(=O)NCC2(C(=O)NC3(Cc4cnn[nH]4)CCCCC3)CC2)s1 c1(OCC(=O)NC2C(CNC(Cc3c(C)ccnc3)=O)C2)ccc(Cl)c(F)c1 N1(C(c2c(C)ncn2C)=O)CC2CC(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 c1(C(=O)NC2(CF)CCN(C(C(CC(=C)C)C)=O)C2)ccc2c(Cl)nccc2c1 CC(C(=O)OCc1nccnc1O)C(C)NC(=O)OC(C)(C)C c1(CC(=O)NCC2CN(C(CCCOCC)=O)C3C2C3)c(C)nn(C)c1C C1(C(N2CC(CCNC(CCC(=C)Br)=O)OCC2)=O)CCC(C)(O)CC1 c1(CN2C(C(=O)NC3(C(=O)OCC)CCC3)CC(O)C2)cc(I)ccc1F c1(CCC(=O)NCC(C2CCOC2)NC(COCCCOC)=O)ccnn1C C(=O)(C(C)CCOC)NC1(CCCNC(C2C(=C)CC2)=O)CC1 Cn1c(=O)ccn(CC(=O)NC23CCCC2N(Cc2csnn2)CC3)c1=O CCCCCC(C(=O)NC1CCCC(CNC(=O)C=CC2CCCC2)C1)C(C)C c1(CC(=O)N(CCN(C(C2CC2C)=O)CC)CC)ccon1 Cn1cc(S(N)(=O)=O)cc1CC(=O)Nc1ccc(OCCO)cc1 CC1CN(C)CC1(c1nnnn1CCCF)NC1(CCF)CC2(CSC2)C1 C1(NC(C2C(CCC)C2)=O)(CNC(=O)C(O)CN2CCCC2)CCCCC1 C1(NC(CCCC#CC)=O)CCOC12CCN(C(=O)CC1NC(=O)NC1=O)CC2 C1(CC)(OCCNC(C(C)C2CCOC2)=O)CCOCC1.C1(CC(=O)N)CC(F)(F)C1 C1(N(C(c2c(C)snc2)=O)C)CC2CC1N(C(c1cccn1C)=O)C2 N1(C(c2ccc(C#N)o2)=O)CCN(C(C2CCCC2(F)F)=O)CC(CO)C1 CCC(C)C(C)C(=O)N(C)CC1(O)CN(C(c2ccc(SC(F)F)cc2)=O)C1 Cn1cccc(C(=O)NC2(C3CCCN3C(=O)C(F)CC3CC3)CC2)c1=O N1(Cc2cnc(SC)nc2Cl)CCC2CN(C(c3ncc(C)s3)=O)CC12 N1(C(CCOCCCNC(Cc2c(C)scc2)=O)=O)CC(CO)C1(C)C CSC1=C(C(=O)NCCC2(O)CCCN(C(=O)Cc3cnnn3C)C2)CCCC1 c1(C(=O)NCCC(C)N(C)C(c2cscn2)=O)n[nH]c2c1CC1CC21.C1(=O)CN1 c1(NC(NC2C(C)CCN(CCc3ccccc3)C2)=S)c2c(nn1C)CCC2 c1(C(N2CCC(NC(c3cccc(C)c3Cl)=O)C2)=O)n[nH]c2c1CC(C)(C)C2 C1(NC(c2ccc(Cl)s2)=O)COC2(CCN(C(c3cnc(Cl)s3)=O)CC2)C1 c1(CC(=O)N(C(CNC(CC(CC)OC)=O)C2CC2)C)ccc(Br)c(C)c1 N1(C(C(c2cccnc2)C)=O)CCCCC(NC(c2ccccc2C2CC2)=O)C1 N1(C(c2cc(Br)co2)=O)CC2CCC(C1CO)N2C(C1CC1[N+](=O)[O-])=O CC1CC(NC(=O)C(c2ccc(F)c(F)c2)=O)CN(C(c2cc[n+]([O-])cc2)=O)C1 CCC(CCCC(=O)NC1CCCC1(C)O)NC(c1ncccc1F)=O N1(C(C(CCNC(=O)OC(C)(C)C)(C)C)=O)CC2(CCCO2)C1OC(C)(C)C C1(NC(c2ccc(Cl)cn2)=O)CCN(C(c2csc(Cl)n2)=O)C12CC2 c1(CC(N2CC3CC2CN3C(c2cnc(O)cc2O)=O)=O)c(Cl)cc(Cl)cc1Cl c1(C(=O)NC(CNC(C=C(CC)C)=O)CO)cc2cc(C)ccc2[nH]1 C(=O)(CC(C)C(=O)NCCCC(=O)NCc1cnccc1Cl)OCC C1(O)(CCNC(C(C)N2CCC2)=O)CCCN(C(c2cc(=O)c(O)c[nH]2)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)CCCc1cnn[nH]1)N1CC(C)(COC)C1 N1(C(CCCOCC)=O)CC(NC(=O)C2=C(Cl)CC2)CC(O)C1 CC1(F)CN(C(=O)CN2CCOCC2)CCN(C(C2(C(F)(F)F)CCCC2)=O)C1 C1(C2(NC(C3CCN(C(=O)c4occc4C)O3)=O)CC2)(OC)CCC1 N1(C(c2c(C)ccs2)=O)CCC(C)(C)C1CC(N1CCC(C)(CCO)C1)=O N1(C(CC(CC)NC(CCCC#C)=O)=O)C2CCC1COC2 CC1=CCCN(C(C2(F)CN(C(=O)CC3CCCC(C)O3)C2)=O)C1 c1(OC)ccccc1CC(C)(C)C(=O)NCC(CNC(C1CC1(F)F)=O)CO c1(CNC2(c3n(C(C(=O)OC)C)nnn3)CC(C)C2)c(Cl)c(C)nn1C Cn1ncc(C(=O)NC(CC2CCC2)C(=O)N2CCCC2C(N)=O)n1 C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(c2ccnc(C)c2Cl)=O)C1 C(=O)(C(C(C)(C)C)C1CC1)NCc1cn(CC(=O)Nc2cccc(OC)c2)nn1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCN(C(=O)CC(=O)NC)CCC1C C1(OC)NC(C(=O)N(C2CCCCC2)Cc2ccc(F)cc2)CCC1Br C(CN(C)C)(C(=O)N1CC(n2cnnc2)C1)NC(C1C(C(C)(F)F)C1)=O C1(C(N(C(COC)COC)C)=O)C=CCCN1C(=O)CC1CCC(C)(C)C1 C1(C)(C(=O)NC(C)C(=O)NCCC(Cl)Cl)C=CCCC1 CC1CC(C)C1C(=O)NC1(CNC(=O)CSCc2cccs2)CCCC1 N1(C(C2CC(C(C)C)OCC2)=O)CC=C(CCNC(C2(C)CCCOC2)=O)CC1 C1(NC(CCCSC(C)C)=O)CN(C(=O)C(O)CC(=O)OC(C)(C)C)C(C)(C)C1 C1(CN(C(C2(COC)CCC2)=O)C)CCN(Cc2ccccc2)C1 C1(CNC(CCOC)=O)C(C2CC2)CCN1C(c1nc(Cl)cs1)=O C=C1Cn2c(C(N3CC4CCC4(NC(=O)CC4CCCO4)C3)=O)nnc2S1 c1(CCC(=O)NC2CC(NC(COC(CC)C)=O)C2)ccc(F)cc1Br C1(NC(c2cc(C)n(C(C)(C)C)n2)=O)CC(C)CN(C(c2ccc(O)nc2)=O)C1 Cc1cc(C(=O)NC(C)CNC(c2cnc3[nH]ncc3c2)=O)cc(C)c1O c1(OCC=C)ccccc1CC(N1CCC(N(C(=O)C(C)CCC)CC)CC1)=O c1(C(N(CCOCCC(=O)NCC(CC)O)C)=O)nccnc1CC c1(C2(C(N3CC(CC=C)(NC(=O)CCF)C3)=O)CCCC2)cccc(C)c1 CC(C)C(C#N)C(=O)NCC(C)CNC(c1ccc(Cl)cn1)=O N1(C(c2cc(C)oc2C(F)(F)F)=O)CCN(C(=O)CC2CC(F)C2)CC(O)C1 c1(C(=O)NC2C(C)(C)N(C(=O)Cc3ccsn3)CC2)noc2c(F)cccc12 CC(C)CCCC(=O)NCC1CN(C(=O)C2=CCCCO2)CC1O C(=O)(C1CCC(=O)c2cccn21)N1CCN(C(C(C(C)C)NC=O)=O)CC1C C(CN=C(NCC1CCc2ccccc2CC1)N1CCOC(CF)C1)SCC#C Cc1nocc1CNC(=O)C(C1(O)CCC1)NC(=O)C(C1CC1)C1CC1 Cc1c(C(=O)NC2CCN(C(=O)C(C)C(C)C)C2)cc([N+](=O)[O-])cc1Br C=C(CNC(=O)CC(C)C(C)(C)NC(=O)Cc1cnc(C)s1)c1ccccc1 N1(C(c2cnc(C)s2)=O)CCC(C(CO)NCC2(c3ccncc3)CC2)CC1 C12(C(=O)NC3(C)CCN(C(c4nc(C)n(C)c4)=O)C3)CCC(CC1F)C2 C1(NC(C(CCCC)C)=O)CCC2(CC1)CN(C(=O)CNC(c1ccco1)=O)C2 C1(NC(C2(COC)CCC2)=O)CCN(C(=O)Cc2ccc(CO)cc2)CC1 C1(C(=O)NCCS(=O)(=O)NC)N(C(=O)CCCC#N)CC12CCCC2 c1(C(C)NC(c2nscc2Br)=O)nnn(C)c1N C1(CC(=O)NCCCN(C(C2CCCCO2)=O)C(C)C)(OC)CCOCC1 N1(C(C(=O)NCC(=C)C)C(C)C)CCCN(S(=O)(=O)C(F)(F)F)CC1 C(=O)(C1=CS(=O)(=O)CCC1)NCC1C(NC(C=Cc2n(C)ncc2)=O)CCC1 CCCCC(C)C(=O)N1CCCOC(CCNC(c2c(C)ccnc2O)=O)C1 C(=O)(C(C)C(C)C)NCC1C(NC(c2nc(C(C)C)oc2)=O)COC1 c1(C(N2CCC(CCNC(C(C#N)C3CC3)=O)CC2)=O)cnc(O)c(Cl)c1 CC1CN(C(C2CN(C(c3cc(CCO)on3)=O)CC2(C)C)=O)CC1(C)CO N1(c2cc(C)nc(CO)n2)CCC2(COC(CNC(=O)C=C3CCCCC3)C2)C1 C1(NC(N(C(c2c(C)nn(C(F)(F)F)c2C)C)C)=O)CCn2ccnc2C1 Cc1cnc2n1CCC(C(=O)NC1(c3ncon3)CCOCC1)C2 Cc1ccc(O)c(C(=O)NCCCCCCNC(c2cc(C)[nH]n2)=O)c1 c1(COC)nn(C)cc1C(=O)NCC1C=CCN1C(=O)C(O)CN(C)C N1(C(c2on(C)c(=O)c2)=O)CC2(CCN(C(C3(c4cccs4)CCCC3)=O)C2)C1 c1(C(N(CC(C)(C)NC(C23CCCC2C3)=O)C)=O)n[nH]c2c1CCC2 Cc1cc(C(=O)NC2CCOC(CNC(=O)CCCC3CCOCC3)C2)[nH]c1C CCC(C)(C)C(=O)C(=O)N1C(C(=O)NOC)CC1C C(C(O)C(=O)NCC(C1CC1)NC(=O)CSC)=CCCC N1(C(c2ccc(C3CC3)o2)=O)CCN(c2ccc(CCO)cn2)C(CCO)C1 c1(OC)c(Cl)ncnc1NNC(=O)NC1CC1(F)F C(=O)(CCC(C)(F)F)N1CCC(N(C(c2nn(CC)c(C3CC3)c2)=O)CCO)C1 c1(C(=O)OCC)ccc(C(=O)NC(C)(CNC(C2C=C2C)=O)C(C)C)cc1 c1(-c2sc(NCc3c(C)cccn3)c(C)n2)cccc(O)c1C C1(CC=C)(C(N2CC(CC(C)NC(=O)CNC(=O)C(F)(F)F)C2)=O)CC=CC1 CCCC(C(=O)NCCCOCCNC(C1(NC(C)C)CCC1)=O)OC C1(CC)C(C(=O)NCC23CC(NCC4(C(=O)N(C)C)CC4)(C2)C3)CCN1C c1(SCC(=O)NC(C2CCCC2)CNC(=O)CSC(F)F)cccnc1 N1(C(C2CC(OC)C2)=O)CCC(C)(NC(=O)Cc2cc(C(F)(F)F)nn2C)C1 C1(CNC(c2ccc(NC)cc2)=O)CN(C(=O)C(O)CC(N)=O)C2(CCC2)C1 c1(C(C(C)C)NC(C(=O)N(CCn2c(C)ncc2)C)=O)cccc(C2CC2)c1 N1(C(c2n(CCC)ncc2)=O)CC(NC(=O)Cc2nocc2C(C)C)C(SC)C1 C1(NC(CCc2n(C)ncn2)=O)CN(C(=O)CSc2ccccc2)CCC1F c1(OCC=C)ccc(Cl)c(C(=O)NCC2CCN2C(c2cc(CCC)[nH]n2)=O)n1 C(=O)(C(C)(C(F)F)c1ccccc1)NC(C)CC(C)NC(=O)COCC1CCC1 c1(C(N2C(C)(C)C(CNC(=O)Cn3ccnn3)CC2)=O)ccc(N)c(F)c1F Cc1[nH]c2ncccc2c1C(=O)NCC1CN(C(=O)C(C)CS(C)=O)CCCO1 c1(N2CCC(CC=C)C2)nc2c(c(=NCCS(=O)(=O)C3CC3)[nH]1)SCC2 N1(C(C2N(C(C)C)C(=O)CC2)=O)CCCC(O)(CCNC(c2ccnnc2)=O)C1 C#CCCCC(C)C(=O)NCCCCCC(=O)NCC1CC12CCC2 C12(C(=O)NCC(=O)NCc3ccc(F)cc3Cl)CC3CC(C1)CC(O)(C3)C2 c1(CNC(C2CC(CCC)C2)=O)nc(C(=O)N(C2CCCC2C)C)c(C)o1 CCC(CC)C(=O)NCC(=O)NC(CC1CC1)C(=O)NC(C)(C)CC(N)=O N1(C(C2N(C(=O)OC)CC2)=O)CCc2cc(NC(=O)C(=O)N=S(C)(C)=O)ccc21 N12CCCC(C1)C2=O.O=C1CCC(C(=O)NCc2cccnc2)O1 c1(C(=O)NCCC(C)N(C(=O)CSc2n[nH]c(O)n2)C)cc2cccc(F)c2s1 C1(CC(=O)NC2C(NC(c3c(COC)noc3)=O)CCC2)CCOCC1OC c1(OCC)cncc(C(=O)N(C(CNC(c2ccnn2CCF)=O)C2CC2)C)c1 C1(C(=O)NC2(COC)CCCCC2)COCCN(C(C2(C)CC2C)=O)C1 N1(C(C2C(C(=O)OC)C=C2)=O)CCC(C)(C)C(C(=O)N(C2CCCC2(C)O)C)C1 N1(C(c2cc(C)n(C)n2)=O)CCC(C)(C)C1C(=O)NCC1COC(C)(C)C1 N1(c2nc(C)cc(OC)n2)CC2(CCOCC2)CC1CNC(C1CCCOC1)=O CC1(NC(C2CC2F)=O)CCCN(C(C2CC(O)C2)=O)C1 c1(C(=O)NCCNC(=O)NCc2csc(Br)c2)cccc(OC2CCCC2)c1 C1(C(=O)NCC(C)CC(=O)NC(CC2CCCC2)CO)(OC)CCC(C)(C)C1 n1(CC(=O)OCC)cc(C(=O)NCC(O)CN(C(=O)C(C)n2ccnc2)C)nn1 N1(C(N(CCF)CC)=O)CCCC(CC2CC2(F)F)C1 N1(C(C2(C)CCCCO2)=O)CCCC(C2CCN(C(=O)CSS(C)(=O)=O)CC2)C1 C(=O)(C1=NOC2(CCNCC2)C1)N(CCN(CCC1CCC(C)O1)C)C C(CCCC(=O)NCc1ncnn1C)N(C(c1c(C(C)C)onc1)=O)C Cc1c(NC(=O)C(F)=C2CNC2)cccc1-c1nn[nH]n1 C(CC(F)F)(C(=O)N1CCC1CC1CCCC1)N(C)C(c1cc(CO)on1)=O c1(C(N2CC(C)(CC(=O)NCC(N3CCCC3)=O)C2)=O)nnc2ccc(Cl)nn12 C#CCC(O)C(=O)N(C1CCN(C(=O)Cc2coc(-c3ccccc3)n2)C1)C CC1(C(N2CCC(CNC(c3cc(F)ccc3Cl)=O)C2)=O)CCC(F)(F)C1 CC1CCC(NC(C2CCC3(CC3)C2)=O)CN1C(=O)CC12CCC(CC1)C2 C1(C(=O)NCC2CCCO2)CC(F)CN(Cc2ccc(F)nc2)C1 C12(NC(C3N(CCC)CCC3)=O)COC(C1)C(NC(=O)CCC(=O)OC)C2 C(=O)(C(C(C)(C)C)NC(=O)CC(F)(F)CC)N1CCC(O)(CCC)C1 N1(C(C(C(C)C)OC)=O)CC2(CCN(c3cc(O)nc(=O)n3C)CC2)CC1C CC(C)(CC(=O)NC1CC(NC(=O)C(C)(F)F)C1)C(F)F CCCCC(F)C(=O)NC1CC1NC(=O)CS(C)(=O)=O C1(CNC(NC(C#C)C)=NCCCOC(C)C)Cc2cc(C)cc(Br)c2O1 c1(C(N2C(C3(NC(C4CCOCC4)=O)CC3)CCC2)=O)cc2ccccc2[nH]1 c1(CNC(C(=O)OCC)Cc2ccncc2)cc(C)c(Cl)c(C)c1 N1(C(C(CC)C)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)CC1c1cn[nH]c1 O=S(=O)(c1cccnc1NC12CCCC1C2)NCCn1ncc2ccccc12 c1(C(=O)NCC(C(=O)OC)CC2CCCC2)ccnc2[nH]c(C(F)F)nc12 C(=O)(C=CS(C)=O)NCCNC(C1CN(C(C2C(C)OCC2)=O)C1)=O c1(C(N2CC3CC(NC(c4ccc(CC)s4)=O)C3C2)=O)c(C)ccc(F)c1N Cc1cccc(C(=O)NC2CCC(C(=O)N(C3CCCC3O)C)C2)c1O N1(C(C=Cc2n(C)ncc2)=O)CCC(CNC(=O)C(F)=CCCF)C(O)C1 C(=O)(C1CCCc2nn[nH]c21)N1C(C)CC(CNC(c2c(F)ccnc2F)=O)C1 c1(CC)ccc(CCCC(=O)NCC(O)CNC(c2coc(OC)n2)=O)cc1 c1(C(=O)Nc2nccc(-c3cn(C)nc3)c2)cc(S(C)(=O)=O)ccc1O C(=O)(CC(C)(O)C1CC1)N(C(C(=O)NC1CCN(S(C)(=O)=O)C1)C1CC1)C C1(NC(C=CCOC)=O)CCN(C(C2(C(=O)C3CC3)CC2)=O)CC1F CC1OCCC1C(=O)CN(C(=O)CC1CCCC1O)CCO.C(=O)(CS)O C1(C(N(CCC(=O)NC(C2CCCC2)C#C)CC#C)=O)COCCN1CC C(C(C(=O)NC1CCN(C)CC1C)C(C)C)NC(C1(CCOC)CCC1)=O c1(CC(=O)NC2C(CNC(c3cc(OCC)no3)=O)CCC2)cc(F)ccc1F C(C)(CC1CCCCC1)(C(=O)NC(C)CN(C(=O)Cn1nnnc1C)C)OC c1(C(=O)NCC2(OC)CN(C(C3(C)CCCN3C)=O)C2)ccc(F)c(C(F)F)n1 c1(C(=O)NC(C2(CNC(c3cn(CC)nc3)=O)CC2)C)ccc2c(c1)CNC2=O CC(C)C(O)CC(=O)NC1CCC(NC(C2OCCC2C)=O)CC1 c1(C(=O)NC2CC(NC(C3(C)CCC(C)C3)=O)C2)n[nH]c2cccnc12 c1(C(=O)NCC2CCCCC2C(c2cnc[nH]2)=O)cccc(CC2CCOC2)c1 CCC(C(=O)NCCC(C)NC(c1coc(C(C)(C)C)n1)=O)OC n1(CC(N2CC(OC)C(OC)C2CSc2ccccc2)=O)cnc2c1CCCC2 c1(C(N(C2CCN(C(=O)CC(C)(C)OC)C2)CCC)=O)c(C)nn(C)c1OC C=C=CCCC(=O)N(C1CCCN(C(=O)C(C)SC(F)(F)F)C1)CC CN1CCC(C)(C(=O)NC2(C)CCCN(C(c3nscc3N)=O)C2)C1=O N1(C(C(C)CC2CC2)=O)CC(C(=O)NC(C)(C)CC2CC2)C(F)C1 CC(CC(=O)NCC(C)NC(c1cnn(-c2ccccc2F)c1)=O)C(F)F C1(CC=C)(NC(c2c(COC)cc[nH]2)=O)CCN(C(=O)Cn2nc(C)cc2C)C1 C(=O)(CCC(C)CN(C)C)NC1(CNC(c2ccc(OC)cn2)=O)CC(F)(F)C1 C(=O)(CCCC(C)CC)NC(CC#C)CC(=O)NCCCN1CCOCC1=O N1(C(CCC#C)=O)CCC2(CC2C(=O)NOCC2CCCC2)C1 N1(C(c2c(Br)sc(C)c2C)=O)CC2CCC(C1)C(NC(C1CC1C)=O)C2 Cc1ccc(C(N2CCC(C)C2CNC(=O)Cc2cc(Cl)ccc2F)=O)cc1Cl C(=O)(C(C)N=c1cc[nH]cc1)NCC1CCN(C(c2c(OC)scc2)=O)CC1C C1(COC)(NC(=O)Cc2ccsc2)CCN(C(c2cn(C3CC3)cn2)=O)C1 C#Cc1cccc(C(=O)NCC(C2(O)CN(C(=O)C=CC3CC3)C2)(C)C)c1C c1(C(N2CCC(CN(C(c3cc(COC)oc3C)=O)C)C2)=O)[nH]c(=N)ccc1C CC1(CNC(c2cc(C3CC3)cs2)=O)CCC(NC(=O)Cc2cc[nH]n2)C1 c1(N(C2CNC2)C)nc(Cl)ncc1Br.C(=O)CCCn1ccnc1 CC1(C)CCN(C(C2CCC3(CC3)C2)=O)C1C(=O)NCC1=CCCCCC1 CCCCCC(F)C(=O)NC(CCCC)C(=O)NCc1cc(C(C)C)no1 c1(C(=O)NCC2C(CNC(C3(C)CC=CCO3)=O)C2)n[nH]c2c1CCC2 C1(C(=O)NCC(C)C(=O)NCC(c2ccncc2)C)CCCCNC1=O N1(C(C(c2n(C)cnn2)(C)C)=O)CCN(C(C2(CF)CC2(F)F)=O)CC12CCC2 Cc1nc(C(=O)NC2CCC2NC(=O)COC2(C)CCCC2)c(C(F)(F)F)[nH]1 CC(C(C)(C)Nc1cnn(CC2CCC2)c1)NC(=O)OC(C)(C)C C1(C2CCCCC2)(NC(C2CC(C(=O)N3CC4CC4(CO)C3)=NO2)=O)CC1 N1(C(C2(C)C(C)C2)=O)CC2COCC(C1)N2C(c1cc2cnccc2[nH]1)=O N1(CC(c2cccc(F)c2)C)CCN(CCCn2nccn2)CC1C C1(CC(=O)NCC2N(C(c3cncn(C)c3=O)=O)CC2)CCC2(CC1)COC2 C#Cc1ccc(C(N2CCC(NC(c3c(C)csc3Cl)=O)C(O)C2)=O)cc1Cl c1(-c2c(C(=O)NCc3cc(OC)cc(F)c3)nccc2)ccccc1[N+](=O)[O-] C1(C(N(CC#C)C)=O)CCC2CCC1N2C(c1ncn(C)c1C)=O O=C1NC(C(=O)O)C2=C1C(c1cc3c(cn1)COC3)NC(=O)N2CCC1CC1 N1(Cc2c(OCC)cco2)CCC2(CC1)CC2C(=O)Nc1c[nH]nc1Cl C1(NC(COC)=O)COCC1C(=O)NCCC(N1CCCC1C1CCOC1)=O Cc1cc(-c2cn(C3CCN(C(c4c(C)ccn4C)=O)CC3)nn2)ccc1F c1(C(N(C)CCN(C)C(C2CCc3nccn3C2)=O)=O)cc(F)cc2nc[nH]c12 C1(CCC)CCc2nc(N(C(=O)C(CC(C)(C)C)OC(C)=O)CC)sc2C1 Cc1cccnc1-n1ccnc1-c1c[nH]c(-c2ccccc2)c1.c1nccnc1N C(=O)(C(C)(C)CC(C)(C)C)NCC12OCC(NC(C3N(CC)CC3)=O)C(C1)C2 C1(C(=O)NCCCC(=O)NC)CCN(C(=O)C=C(C)C(C)(C)C)C(C)(C)C1 C=CCC(C(=O)NCC1CCC(C(=O)NC(c2cn[nH]c2)C)C1)C(C)C n1(CC)cnc2[nH]c(=NCC3CC(O)C3)nc(N3CCOCC(C)(F)C3)c12 c1(C(N2C(C)(CCC)CC2)C(=O)NC2CC(F)(F)C2)cccc(C2CC2)c1F CC(C(=O)OC(C)(C)C)C(=O)N1CC2C(CN(C(=O)CCC=CC(C)C)C)C2C1 C=CC1OCCC1C(=O)NCC1CC1CNC(c1ccc(SC)o1)=O N1(C(=O)NCc2ccc(Cl)cc2C(F)F)CCCC1C1CCCO1 c1(C(C)=O)cc(NCCCNC(C2CCC(=O)N2)=O)ncn1 c1(CC(=O)NC(CCCNC(CC=C)=O)C)coc2cc(Cl)ccc12 c1(N(C(C2CN(C(C(=O)NC(C)C)=O)CC23CC3)=O)C)ccn2nccc2n1 c1(C(=O)OCCc2ccccn2)ccc(NC(c2ccon2)=O)cc1 c1(NC2CCN(C(C(n3ncc(C)c3)C)=O)C2)cc(O)nc(C)n1 c1(C(N(C2CC(NC(C3C(C=C)C3)=O)C2)C)=O)cnc(O)c2cncn12 Cc1cccc(CC(=O)NC2CC2NC(=O)COc2cnc(Cl)cn2)c1 c1(C(N2C(Cc3cn(CCC=C=C)nn3)CCC2)=O)nn(C)c2ncccc12 C(=O)(C(CC(C)C)C(N)=O)NCC(CN(C(Cc1cc(C)nn1C)=O)C)C N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(=O)C(N2CCSCC2)C)CC(F)C1 N1(C(CNS(NC)(=O)=O)=O)CC2CCC1CN2C(=O)C(F)C(F)(F)F c1(CNC(CC)Cn2cncn2)cc(OC)c(C)cc1F CC1CN(C(c2c[nH]c(Br)c2)=O)CC2(CCN(Cc3cc(Cl)ccc3Cl)C2)O1 N1(C(c2n[nH]c(C)c2C)=O)C(C)CN(C(c2cnccn2)=O)CC1C CN1Cc2ccccc2CC1C(N1CC(NC(C23CC(C2)C3)=O)C(F)C1)=O C1(=CC(N2CC(C(C)NC(CC3N(CC)C(=O)CC3)=O)C2)=O)CN2CCC1CC2 C(=O)(C(O)CCCNC(=O)C(C)CC(C)C)NCCC(=O)NCC#C c1(CC)cc(C(=O)OCC2CC2c2ccc(Br)cn2)c(Br)s1 N1(C(C2C(NC(C34CC(C3)C4)=O)CCC2)=O)CC2CCC1CO2 C1(N(C)C)CN(C(C2C=CCCC2)=O)CCC1CNC(C1CC=CCC1)=O Cc1ncn2ccc(C(=O)NC(C)(C)CN(C(=O)C3=CCCC3)C)cc12 N1(C(CC(=O)OCC)=O)CCCCC1CN(C(=O)C(C)(C)COC)C c1(C(=O)NC2(CC=C)CN(C(=O)C(C)C3CC3)C2)ccn2c(C)cnc2c1 C1(C(N(CC(C)(C)CNC(c2ccnc(CO)c2)=O)C)=O)OCC2CCCC12 C1(OCCC)CCCN(C(=O)CCCCNC(c2ccnnc2O)=O)C1 N1(C(C(COC)C)=O)CCN(C)C(CNC(=O)C=C(C)c2ccco2)C1 C1(C(N(CC(O)CN(C)C(c2n[nH]cc2[N+](=O)[O-])=O)C)=O)CCCCC(F)(F)C1 C1(C(=O)NCC2(F)COC2)COCCN(C(c2ccnnc2O)=O)C1 N1(C(C(C(C)C)O)=O)CCC(C2CC2)C1CNC(c1cccc2nsnc12)=O CCCC(CNC(=O)C1=CCCC1)C(=O)Nc1cccc(F)c1F C(C(C(=O)NC1(c2ncc(C)s2)CC1)C(C)(C)C)NC(CCCSC)=O C(CCCCC(=O)N(C1CCOC(C)C1)C)N(C(c1c(C)noc1C)=O)C C(=O)(C#CC(C)(C)C)NC(C1(O)CCN(C(=O)CCc2nc[nH]n2)C1)C C(c1ccccc1C)=CC(=O)NC1CCC(N(C(C2CC(CC)(CC)C2)=O)C)C1 C12(C(=O)NCC(CC(C)C)(C)NC(=O)C#CC3CCOC3)CCCN(CCC1)C2 C(=O)(C1=NOC(C)C1C)NC(C1C(C(N2C(C(=O)NC)C=CC2)=O)C1)C C(=O)(C(=O)C(C)(C)C)N1CC2C(C(N(C)CCC3CCC3)=O)(C2)C1 C(=O)(C(C)CC(F)(F)F)NCC1C(NC(c2c(C)n(C(C)(C)C(C)C)nc2)=O)C1 N1(C(CC2(OC)CCOCC2)=O)CCC(O)(C(C)NC(C2CCCC2O)=O)CC1 c1(C(N(CCOCCN(C(C(CC)OC)=O)C)C)=O)ncc(OC(C)=O)cc1F c1(C(N2C(C)C(C)N(C(c3cscn3)=O)CC2)=O)cnc2ncccc2c1 O=C(C(C1=NOCC1)N1CCCC1C1CC1(F)F)NCc1ccc(Cl)cc1 C(=O)(N1CCC(C(N2CCCC2CCC(C)C)=O)O1)c1nc(C)oc1 C(=O)(C(CNC(c1nc(C)oc1C)=O)CC(C)C)NC(c1nc[nH]n1)CC CCC(C)(C(=O)N1CCN(C(=O)CCc2ccnc(Cl)c2)C(C)C1)C(N)=O CC(C)C(C)(CNC(C1(CS(N)(=O)=O)COC1)=O)NC(=O)Cn1nccn1 c1(C(C)NC(C2OCCC2CNC(=O)C(CO)N(C)C)=O)cccnc1O c1(C(=O)NCC2COCCN2C(=O)CC(F)(F)F)ccnnc1O CCCC(C)(C)C(=O)NCCN(C(=O)CCC=Cc1ccccc1)CC1CC1 CCC(C)C(O)C(C)C(=O)NC(C(N1CCC2(CCCC2)C1)=O)C1CCOC1 C1(C(N2CCC(CN(C(=O)C(C)(C)n3ccnn3)C)C2)=O)CCCC(C)(C)CC1 C=CCCCCNC(=O)C(C)(C1CCC1)NC(=O)C(C)N(C)C(C)=O N1(C(=O)C=CCF)CCC2(CCCN2C(C2SCCCS2)=O)C1 c1(C(=O)NC(C(=O)NC(c2nnc(O)n2C)C)C2CCOC2)ccnnc1O c1(C2(F)CN(C(C3C(c4n(CC)ccn4)OCC3)=O)C2)ccccc1Br C12(CNC(C3(CC)CC3(F)F)=O)CC1CN(C(C1(CO)CCCCC1)=O)C2 C1(NC(CN(C)C(=O)C2CC2)=O)CCC(F)(CNC(c2cc(O)ncn2)=O)C1 c1(NCc2c(Cl)ccc(N(C)C)c2)sc2c(c1C(=O)NC1CC(O)C1)CCC2 C1(NC(c2cscn2)=O)CN(c2ncc(OC(F)F)cn2)CCC1(F)F c1(C(N(CC(CNC(c2nccc(C)n2)=O)C)C)=O)cc(N)c(C)cc1C N(C1CCCn2ccnc21)C(=O)CC1COCCN1C(=O)CC(C)(C)C#N.CNC n1(CCOC)cc(C(=O)NCCC2CCCN2C(C2CC(CF)C2)=O)nn1 N1(C(C2(N(C)C)CC2)=O)CCC(F)(F)C(CNC(c2nc(Cl)sc2Cl)=O)C1 N1(C(c2c(C)c[nH]n2)=O)CC(C)CCC1CNC(c1ccc(F)c(CO)c1)=O N1(C(C2C(C=C)C2)=O)CC2CCC1CN2C(C1(C#N)CCOC1)=O n1(CC(=O)N(C(CCNC(C2N(CCC)CCC2)=O)C)C)cc(C#N)cn1 C(=O)(C(C(C)(C)O)NC=O)N(CCCF)C.C1CC(C)(C)C1 Nc1cc(C(=O)NCCC2CCN(C(C3(C(F)F)CCCO3)=O)C2)cc(O)c1Cl CC1(C)CC(C(=O)O)N(C(=O)CNC(=O)CCCC2CC2)C1 C(c1c(C)coc1C)=CC(N1CCC(N(C(=O)C(C)C2CCC2)CC)C1)=O Cc1cc(C(C(=O)NCc2ccco2)N(C)CC2(O)CCOCC2)cc(F)c1 c1(C(=O)NC2C(CNC(=O)Cn3cccc3)CCC2)cc2sccc2[nH]1 C1(C(=O)NCCNC(=O)CCc2nnc(-c3ccccc3)o2)CCCS(=O)(=O)C1 C1(NC(c2nc(CC)oc2C)=O)CC2CC1CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 CN=S1(=O)CCN(C(=O)C(c2ccc3c(c2)OCO3)=O)CC1 N1(C(C(N2CCN(C)CC2)C)=O)CC2CCN(C(c3cccc(=O)o3)=O)CC2C1 CCCCC(C)CCC(=O)NCCCOCCCNC(=O)CCc1ccccc1 N1(CC(CC)S)C(=O)CN(CCS(N)(=O)=O)C1=O.c1(N)ccccc1Cl C1(C(=O)NC2CCCC(OC)C2)CCOCCN1C(=O)Cc1cccs1 c1(C(=O)NCc2nc(CC(=O)OCC)on2)cnn(CC)c1C1CCCC1 c1(NC(C(n2ncc(C)c2)C)=O)ccc(C(N)=O)cc1 C1(C(=O)OCC)(CC)CCCN1C(C12CC(CCO1)C2)=O CCCC(CNC(=O)Cc1ccsc1C)C(=O)NCCOCCO C(=O)(C(CCNC(=O)C(C)OCC1CC1)OC)NCCC(=O)OCC c1(C(=O)NC2C(NC(c3cccc(C(C)C)c3)=O)C2)cccc2c1CNC2=O N1(C(C(CC)C)=O)CCCOC(CNC(c2cnc(CO)nc2C)=O)C1 C1(CNC(c2nc(Cl)sc2Cl)=O)CC(F)(F)CN1C(c1cnnc(Cl)c1)=O N1(C(C(COCC)O)=O)CC(OCC)CC1CF C1(C(=O)NC(C2(OC)CCC2)C2CC2)OCCCC1c1ccccc1 c1(OC)cc(CN)cc(N)c1O.N1(CCC(=O)N2CC(CO)C2)CCN(C(C)C)CC1 C1(C(=O)NCC2CCN(C(c3cc(C)on3)=O)C2)CCc2n[nH]cc2C1C C1(NC(=O)NCC2CNC(=O)C2)CC2C=CCC(C1)C2 C1(NC(c2coc(C3CC3)n2)=O)CCCN(C(C23CC(C(F)F)(CO2)C3)=O)C1 Cc1ccncc1CC(N1CC(OCCNC(=O)CC2CC=CCC2)C1)=O C(CN=c1ccn2ncc(I)c2[nH]1)NC(C1(C(C)C)N=N1)=O c1(C(=O)NCCCC(C)(C)NC(COCCN(C)C)=O)ccc(O)c(=O)cc1 c1(NC(c2csc(CNC(c3cccnc3F)=O)n2)=O)ncccc1[N+](=O)[O-] Cc1nc(C(=O)N(C2CCCC(N(C(=O)CCC(C)C)C)C2)C)c(C)n1C Cc1ccnc(NC(C)(CCCO)c2nnnn2CC2CCCO2)n1 C1(C(C)NC2CC2)CCCCN1C(c1cn(C2CCOC2)nn1)=O c1(C(N2CCC(CNC(CN(C(COC)=O)C)=O)C2)=O)c(C)oc2ccccc12 Cc1[nH]nc2c1CCC(C(=O)N(C1CN(C(C3CCN(C4CC4)C3=O)=O)C1)C)C2 C1(C(=O)OCC)CC(C)N(Cc2ccc(Br)cc2OCC)C(C)C1 C1(CC)CN(C(=O)C(F)C(C)CNC(C2(C#N)CC2)=O)CCN1C C1(NC(C(c2cn(C)nc2)(C)C)=O)CCCC(NC(=O)COC2CCC2)CC1 C1(O)(CNC(C2C(C(=O)OC)C2)=O)CCCN(C(=O)CC2(OC)CCC2)C1 CC1CC(NC(=O)CC(C)n2cccn2)CN(C(c2cc[nH]c2)=O)C1 CC1CN(C(c2ccns2)=O)CC(CCNC(c2cc(C3CC3)ncn2)=O)O1 C1(C(C)NC(=O)Cc2ccns2)CCN(C(=O)CCC2CCC2)C1 N1(CCOC(CN2C(=O)CCC2)=O)CCN(C(=O)CN2CCSCC2)C(=O)C1 Cc1cc(CCC(=O)NCC(C)CNC(C2CCC2(C)C)=O)on1 C1(NC(C=C(C)C2CC2)=O)CC2CCC1CN(C(=O)CC1CCS(=O)(=O)CC1)C2 C1(CCNC(C(C)Cn2ccnc2)=O)CN(C(c2c[nH]c(=N)s2)=O)CCO1 c1(C(=O)NCCCNC(C(CC)n2cccn2)=O)cc(C(F)(F)F)cc(F)c1 c1(C(=O)NCC2(F)CC(NC(C3(C#C)CCC3)=O)C2)c(C)c(C)c(C)c(C)c1C C(=O)(C(CC(C)(C)C)NC(=O)OC(C)(C)C)N(C1CCOCC1)CCC c1(C(=O)NCC2CCC(CNC(C)=O)CC2)nnc(C)cc1NC1CCCS1 C(CC(O)CNC(=O)C(C1CCCCC1)O)NC(=O)COCCF c1(C(N(CC(C)N(C)C(C2CCCC2C(C)(C)C)=O)C)=O)ncccc1Cl C1(CCNC(C2C(C=C)C2)=O)CN(C(=O)COCc2ccnn2C)CCS1(=O)=O N1(C(c2cnn(C)c2Cl)=O)CC(NC(c2nncs2)=O)CC1(C)C N1(C(C(COC)C)=O)CCOC(CC2(C(=O)NC3CCCC3)CCCC2)C1 C1(CC(C)NC(C(CC)(C)O)=O)CC2CCC(C1)N2C(C1(CCF)CCC1)=O N1(Cc2c(C)ocn2)CCCC(NC(=O)C(C)Cn2cccn2)C1 c1(C(N(CCC2CCN(C(CCNC(C)=O)=O)CC2)C)=O)cccc(F)c1C(F)F CCC(C)C(O)CC(=O)N1CCN(CC(C)NC(c2ccc(F)cc2F)=O)CC1 N1(C(COCCC)=O)CCN(C(=O)Cc2cccc(Br)c2C)CC1CO N1(C(CC2C(C)CCN(C(Cc3ccn(CC)n3)=O)C2)=O)CC2(COC(=O)C2)C1 C(C(C)(O)CC(=O)NC1CCCC(C(=O)NC2CCC3(CC2)N=N3)C1)OC C(=O)(C#CC1CCC1)N1CC(CCNC(C2(C)CC(C(F)(F)F)C2)=O)C1 Cc1ccoc1C(N1CCCC1CNC(=O)CCNC(=O)CC1CCCCC1)=O N1(C(CCN(CC)CC)=O)CCC2(CC2)CC1C(=O)NC(c1cncn1C)CO c1(C(=O)NCC2CCCN(C(C(CC)COC)=O)C2)cc(F)c(Cl)cc1Cl C1(CC(N2CC(N(C(=O)CCn3ccccc3=O)C)C2)=O)COC(C)(C)CO1 CC1COCCN(C(=O)C(C)(C)C)C1.S1(=O)(=O)CCN1C C(=O)(CCC(=O)c1ccc(Br)cc1)NC(CNC(=O)C(F)=CCCF)CO C(C(=O)NC1CC(F)(F)C1)(C1=CCSC1(C)C)N(CC(N1CCCC1)=O)CC n1(CC)ncc(I)c1NC(=O)Nc1cccc(OC)c1.C1CO1 C1(C(N(C)CC2CCCCC2)=O)CCCCCC1NC(C1CCC(O)CN1C)=O C(=O)(C(C)C(O)C(C)C)N(C1CCN(C(c2cc(CC)[nH]n2)=O)C1)CC C(=O)(CCN=c1ccc(C)c[nH]1)N1C(CCNC(CCCCC)=O)CC(OC)C1 c1(C(=O)NCC(C)CN(C(=O)C(O)C2CCC2)C)cccc(C(C)(C)C)n1 c1(CC)ccccc1C(CNC(=O)CNC1CCCC1)NC(=O)C(C)N1CCCC1 C1(CNC(C2(SC)CCC2)=O)CC2(CC2)CN1C(C1CCCC(CF)C1)=O c1(C(=O)NC2CCCC(NC(COCCCCOC)=O)C2)c([N+](=O)[O-])cnn1C C1(C(=O)NCC2(CO)CCCC2)CC2CC2N1C(=O)Cc1cnns1 c1(C(=O)Nc2cccc(C(=O)NCC3(C)CC3)c2)cc(Br)cc(Br)c1 CCC(CN(C)C)C(=O)N(CCCN(C)C(c1cnn(CCC#N)c1C)=O)C c1(C(N2CC(C)(C(N3CCC(C(C)(C)O)C3)=O)C2)=O)cnn2cccc(F)c12 CN1CC2CN(C(C3C(c4ccccc4)C3F)=O)CCN2C1=O N1(C(c2cnn(CC3CCCCC3)c2)C(=O)NC(C)C)CCOCC(C(C)C)C1 C1(C)(CC(C)C)CCCN1C(=O)CC(c1ccccc1C)N c1(-c2c(C)ccc(CO)c2)cc(C(N2CC(NS(C)(=O)=O)C2)=O)c2cc[nH]c2c1 c1(C(C)NC(c2ccc(C)cc2OCC(F)F)=O)ccc2c(c1)NC(=O)C2 N=c1nc(C(=O)NC2(C(=O)NCC3CCOC3=O)CCCC2)cc[nH]1 C1(NC(C(c2cccnc2)NC(CC(=O)NCC)=O)=O)CC(C)OC(C)C1 C1(CC)CN(C(=O)Cc2ccsc2)CCC1NC(C1(OC)CCCSC1)=O C1(NC(=O)OC)CC2CCC(C1)N2C(c1c(NCc2ccccn2)c[nH]c1C)=O c1(Cn2cc(C(C)NC(c3csc(=N)[nH]3)=O)nn2)c(F)cccc1F CCN=c1[nH]c(C(N2CCOC(CCNC(=O)COC3CC(F)(F)C3)C2)=O)cs1 N1(C(C(C2CCOC2)OC)=O)CC23CCCC2(C1)CN(C(=O)CCP(C)(C)=O)C3 c1(CN2CC(NC(C(CCC)N3CCNCC3)=O)C(C)C2)ccnc(F)c1Cl c1(CNC(C(C#C)(C)C)=O)cc(C#N)ccc1Cl C(CCC(=O)NCc1nc(Cl)oc1C)(C(C)C)NC(C(CSC)OC)=O C1(C(=O)NC2C(CNC(=O)C=Cc3cncc(F)c3)CC2)CCn2nncc2C1 CC(CCCC(=O)N(c1ccc(O)cc1)C)NC(=O)C=CCO c1(CNC2(CC(=O)OC3CCN(C(C)=O)C3)CCC2)cccc(F)c1C c1(CCC(=O)N(C2CCN(C(C=CC)=O)C2)CCC)ccc(O)cc1 c1(N2CCC(O)(C(C)NC(C(C)=C3CCC3)=O)C2)nccc(C)c1[N+](=O)[O-] N1(C(C2CC3(CCN(C(C4C(C)(C)C4)=O)C3)C2)=O)CCC2C(=O)NCC2C1 c1(C(N2CC(CCCCOC)C2)=O)nc(C2CC2)oc1C C1(NC(C2(CNC(C3CCC(=O)O3)=O)CC2)=O)C(CC2CC2)CCC12CCC2 c1(C(N(CCCn2cc(CCCN)nn2)C)=O)nc(=N)cc[nH]1.n1(CCC)ccnc1 C1(C(N(CC(=O)NC(C)Cc2cnc[nH]2)C2CC2)=O)CC2(CC2)C1 c1(C(CN(CC(=O)OC)CC)C(=O)OC)ccc([N+](=O)[O-])cc1 Cc1nccc(F)c1C(N1CCC1C(=O)Nc1sc(-c2ccccc2)cc1Br)=O N1(C(CCC(=C)Cl)=O)CCN(C(c2cn3c(n2)SCC3)=O)CC1C Cc1oc(=O)oc1CS(=O)(=O)CCc1ccc(OC(F)(F)F)nc1 CC1SCCCC1C(=O)NCCC1CC(C(=O)NOCC2(C)CCC2)C1 c1(C(N2CC3C(CNC(=O)Cc4ccsc4)C3C2)=O)c(Cl)ccc(Cl)c1O C1(CC(N2CC(O)(CN(C)C(c3ccn(C4CCC4)n3)=O)C2)=O)CCOC1(C)C N1(C(CSc2cccc(C)c2)=O)CCN(C(c2sc(C)nc2C)=O)C2CC12 c1(C(N2C3C(NC(C(CCOC)OC)=O)CC(C3)C2)=O)ccc2ccccc2c1 N1(C(CN2CCC(C)CC2)=O)CC(C)(C)OC2(C1)CN(C(C1OCC1(C)C)=O)C2 c1(C(=O)NCC(C)Sc2ccccc2)csc(=NC2CC2)[nH]1 C1(C(=O)NCc2cc(C)[nH]n2)CC(C)CN(C(c2occ3c2CCC3)=O)C1 CN1CC2CCN(C(c3csc4ccccc34)C(=O)NCC3CC3)C2C1 N1(C(c2nccc(OC)c2)=O)CC(CC(=O)NC2CC(N(C)C)C2)C2(CC2)C1 N1(C(C2(OC)CCSCC2)=O)C2CCCC1CC(NC(=O)CN1CC=CC1)C2 S(=O)(=O)(c1ccc(NCC23CCSCC2C3)c(F)c1)N(CCC)CC N1(C(C(CC2CC2)OC)=O)CC2CC1(C(=O)NC1(CCCCO)CC1)C2 N(C1c2ccccc2CC1NC(=O)CCc1ccc(F)nc1)C(C1(OC)CC1)=O N1(C(CC2(NC(C)=O)CC2)=O)CC(CN(C)C(C2(O)CCSC2)=O)C2(CC2)C1 C(=O)(NN1CCCCC1C)c1cccc(N(CC(F)F)CC)n1 C1(C)(CNC(C(COC)C)=O)CCCN1C(c1cnn(C2CCCC2)c1)=O c1(NC(c2ccc(F)cc2)C)ncccc1S(=O)(=O)NCc1nocc1C1CC1 N1(C(c2c[nH]c(=N)o2)=O)CCC2C(C1)CN2C(C1CCS1(=O)=O)=O c1(C(C(=O)NCC2CCCO2)N(C2CCCC2)CCC)cc(C)c(Br)c(Cl)n1 C=C(C)CCCC(=O)N1CC(NC(C2CCCN2N=O)=O)CCC1C N1(C(COC(CC2N(C(=O)OC(C)(C)C)CC(F)C2)=O)=O)CC2CC(O)C2C1 c1(C(N(C)CC2(CNC(c3c(COC)ccs3)=O)CC2)=O)cnn2c1OCC2 c1(-n2cc(SC)nn2)ccc2[nH]c(C(=O)N(CC(C)(C)C)C(C)C(C)C)c(C)c2c1 CC(CN(C)C)CCC(=O)NCC1CC2CCC1N2C(c1ccc(Cl)nc1O)=O c1(C(=O)N=c2cc[nH]c(CCCO)c2)cnc2cccc(Br)c2c1 C1(NC(c2c(C(C)(C)C)nsc2N)=O)CC2CC1CN(C(c1ccc[nH]1)=O)C2 c1(C(=O)NC2CN(C(c3c(C)cn(C)c3)=O)C(C)CC2)cn(C)c2ncccc12 C(CCCCC(=O)N1CCC1CNC(=O)C(F)(F)CCn1ccnn1)OCC C1(C(=O)NC2C(C)CN(C(C3CCOCC3)=O)C2)CCn2ccnc2C1 Cc1ccc2cc(C(=O)NC3CC(CCNC(=O)C(C)CS(C)(=O)=O)C3)[nH]c2c1 C(=O)(CCN(C(C1CC1F)=O)CC)N(CC#C)CC C(=O)(C(F)C1=CCCCC1)NCC1CCN(C(C2CCCCN(C)C2=O)=O)C1 C1(C(N2C(C=C)CC2)=O)CC(O)CN1C(c1c[nH]c(C#N)c1)=O c1(C(=O)NCC2C(NC(COCCC=C)=O)COC2)cc(N)ccc1F C1(C(=O)NC2C(SC)CN(C(c3coc(SC)c3)=O)C2)COc2ccccc2C1 c1(C(=O)NCC2(O)CCN(C(c3cnc(Cl)[nH]3)=O)C2)nc[nH]c2nccc1-2 C(=O)(C1CCc2ccccc21)NC(CNC(C(C1CC1)OCC)=O)CC(C)C C(c1nc2ccccc2o1)=CC(=O)NCC(CO)NC(=O)COCC1CC1 N1(C(CSCC#C)=O)CCN(C(=O)CNS(=O)(=O)CCCOCC)CC(C)(C)C1 N1(C(C(CC)OC(C)=O)=O)CC(C)(C)CC1CNC(=O)CCOC1CCCCC1 C1(C(C)(C)NC(CSCC#C)=O)CCN(C(C2CCCCO2)=O)CC1 C1(C(N2C(C(=O)OCC)C=CC2)=O)CN(C(=O)CC(C)CN(C)C)CC1F C1(CCNC(C2CC2c2cccnc2)=O)CCCN(C(C2CC2C(=O)O)=O)C1 N=c1[nH]c2c(s1)CCCC2C(=O)N1CC(CNC(C2(CN)CCCC2)=O)C1 c1(OC)ccc(C(C(=O)NC(C)C)N(CC(C)(CO)CO)C)nc1OC c1(NC(N2CCOC(C)C2)=O)cncc(-n2ccnc2)n1.C1(O)CC(F)(F)C1 N1(C(COCCOCCOC)=O)CCN(C(C2CC23CC(O)C3)=O)CC1CF c1(C(=O)NCC(=C)CCNC(C2CC2C(C)(C)C)=O)ccc(-c2cc[nH]n2)cc1 N1(C(c2c(OC)cc(OC)cc2)=O)CC(NC(=O)C(C)CN)CC2(CCC2)C1 C1(NC(=O)Nc2c(F)cc(C)c(F)c2)CCOC2(CCSCC2)C1 N1(C(C(C)(F)F)=O)CCC2(CC1)COC(CNC(C1CC13CCC3)=O)C2 c1(SC)ccc([N+](=O)[O-])cc1C(N1CC2NCC1(C)C2)C(=O)OC c1(C(C)C(=O)NCC2(NC(c3ccc(F)cc3)=O)CCOC2)nc(F)ccc1Cl O(CP(C)(C)=O)CC(=O)NC(C1CCCCC1)CNC(C1C(CCC)C1)=O c1(C(N(CCNC(c2scc(C(C)=O)c2)=O)C)=O)n[nH]c2c1CCCC2 c1(CC(C(N)=O)NC(C2C(NC(c3c(C)scc3)=O)CCC2)=O)ccc(O)cc1 C(=O)(C1=C(Cl)CCC1)NC(C(C)NC(=O)CN1CCC(C(N)=O)CC1)CO N1(C(CCc2onc(CCC)n2)=O)CCC(NC(c2snnc2C)=O)C(F)C1 c1(SCC(=O)NCC2C(C(=O)NC(CSCC(=O)OC)=O)C2)nc(C)cc(C)n1 C(=O)(C(C(C)(C)C)NC(N)=O)N1CC(c2cn(Cc3nc(C)sc3)nn2)(F)C1 C1(C(=O)NCC(=CC(N2C(CCC)COCC2)=O)C)CC(C)(C)CN1C c1(C(=O)NCC(CNC(CC(C=C)CC)=O)O)cc(Cl)c(C)cc1Br C1(N(C(c2cn(CCCC)nn2)=O)C)CCCN(C(C2(SC)CC2)=O)CC1 c1(OC)cc(C(N2CC3CC2C3C(=O)NC(CO)C(C)C)=O)c([N+](=O)[O-])cc1O C12(C(=O)NC3CN(C(c4c(C)sc(C(F)(F)F)n4)=O)CC3C)CC1COC2(C)C c1(NC(c2c(OC)c(F)ncc2)=O)nn(C)cc1C#C[Si](C)(C)C C(C)(CC(=O)NCC1CCCN1CC(=O)N(C)C(c1nc(C)no1)C)OC N1(C(C2CCN(CC)CC2)=O)CCN(C(c2coc(Cl)n2)=O)CC(CO)C1 N1(CC)CCOC(C(=O)NC2CC(CNC(c3c(C)cnn3C)=O)C2)C1 N1(C(CC2(C=C)CCC2)=O)CCC(C)(NC(=O)C(c2ccccn2)C)C1 c1(SCC(=O)NC2CC(NC(C=C3CCC(C)C3)=O)C2)ccc(F)cc1Br C(=O)(C1=CC2CCC(C1)N2)NC(C(=O)N(C1CC(CC)C1(C)C)C)=O c1(C(=O)NC2(C)CN(C(c3ccn4nccc4n3)=O)C2)cc(O)c2ccoc2c1 N1(C(C2N(C)C(=O)OC2)=O)CCS(=O)(=O)C(CCNC(c2ccc(O)nc2)=O)C1 CC(C)C(F)(CNC(C1C=CCS1)=O)C(=O)NCC1(c2ccon2)CC1 C1(C(N2CCC(CC(C)NC(C(=O)NCC)=O)CC2)=O)CS(=O)(=O)CC(=O)N1 C(CC(C)C(=O)NCC1CC1NC(c1cnc(C2CC2)o1)=O)=CCC Cc1ccc(C(C)CC(=O)NCC2(C)CCN(C(=O)C(F)(F)C3CC3)C2)cc1 C1(NC(C2c3nnc(CC)n3CCC2)C)CCCC(C2CCC2)C1 c1(CCC)cc(C(N2CCC(CN(C(=O)C3=CCCC3)C)C2)=O)sc1C c1(C(=O)NCC2C(NC(C=C(CCC)C)=O)CC2)cc2c(C)ccc(Cl)c2[nH]1 c1(NC(c2c(NC(C3(O)CCOCC3)=O)ccs2)=O)cc(Cl)cc2[nH]ncc12 N1(C(C2(CC)CCCN2C(c2nc3ccccc3[nH]2)=O)=O)CCCC(C)(C)CC1 c1(CC(C(=O)NC(=O)N)C2CC2)ccc(O)cc1.c1(C(C2CCC2)N)ccccc1 C(=O)(CCS(C)(=O)=O)NC1CC(N(C)C(c2n[nH]cc2Cl)=O)C1 C(=O)(C1=CC2(CN(C(c3csc(Cl)c3)=O)C2)OC1)N1CC(C)(C(F)(F)F)C1 C=CCC(CNC(=O)CCCC(OC)OC)C(=O)N1CC(COC23CC(C2)C3)C1 O=C(CCN=c1[nH]c(=NCCCF)[nH]c2c1CCCCC2)Nc1ccccc1 N1(C(CC=CCC)=O)CCC(NC(c2coc(S(C)(=O)=O)c2)=O)C12CCC2 Cc1nc(F)ccc1CNC(=O)CC1CCCC1NC(C1CC(O)C1)=O C1(CNC(C(c2ccc(Cl)cc2)OC)=O)CCC(C)(C)CN1C(c1ccoc1)=O c1(N2CCCC(CC)C2)nc(C)cc(=NC2CN(C(=O)C(F)C(C)(C)O)C2)[nH]1 N1(C(c2c(SCC)nccn2)=O)CCC2C1CCCN2C(=O)CCC(C)(F)F N1(C(c2c(C)occ2)=O)CC(NC(=O)C=Cc2ccc[nH]2)C(C2CC2)C1 CC(C)(F)CCC(=O)NC12CC(C(N3CC(CF)OC(CF)C3)=O)(C1)C2 N(C1CCOc2ccc(Br)cc21)S(=O)(=O)c1cccc(N2CC3CSCC3C2)n1 n1(C(C)(C)C)nccc1C(N1CCC(OCCNC(=O)Cc2csnn2)C1)=O C1(CNC(Cc2cccc(OC)c2)=O)C(C)CCCN1C(c1coc(Br)n1)=O C1(NC(CCC(C)(F)F)=O)CN(C(=O)CC2CCCCC23CC3)C2(CCCC2)C1 C1(NC(c2cccc(N)c2O)=O)CCCCCN(C(=O)CCCC2CCCC2)C1 N1(C(CN2CCCC(CC)C2)=O)CC(NC(c2cn(C)nn2)=O)CC(C)(C)C1 c1(C(C(N2CCCC(NC(CC)COC3CC3)C2)=O)=O)cccc2c1OCC2 Cc1oc(Br)cc1C(N1CCCC1C1(NC(C2CC2F)=O)CC1)=O C(=O)(CC(F)(F)C(F)F)NCCC(C)N(C)C(C1C(F)(F)C12CC2)=O C1(NC(=O)OC(CC(C)C)C)CC2(C1)CN(C(=O)CN1CCCC1)C2 N1(C(C(C)C#N)=O)CCC(NC(C23CC2C3)=O)C(C)(C)C1 C(=O)C1=CCC2(COC2)OC1.Cc1nc(C(C)N(C)CCN(C(C)=O)C(C)C)n[nH]1 N1(CCN(C(C2(CC)COC2)=O)C)CCN(C(=O)COCC(C)C)CC1 N1(C(c2cc(C)c(Cl)cc2)=O)CC2OCCN(C(=O)CC3CCCN(C)C3)C2C1 C1(C(=O)NC2CCCCC2CNC(=O)COCCC(C)C)(OC)CCOCC1 CC(CN(C)C)CCC(=O)NCCCN(C(C1(F)CCN(C)CC1)=O)C1CC1 C(=O)(CCCSc1ccccc1)N1C(CNC(c2ccsn2)=O)CC1 c1(C(N2CCN(C(C3C(F)(F)C34CC4)=O)CC2)=O)nnn(C2CC2)c1C(F)F c1(NCC2C(O)CCC(C)(C)C2)[nH]c(=NCc2nc[nH]c2Br)nc2sccc12 C1(CNC(CCC(CC)C)=O)CN(C(=O)Cc2ccnnc2O)CCC1(F)F c1(OC)cc(CC(=O)NC(C)(C)C(C)NC(=O)CCc2ccsc2)c(F)cc1O CP(C)(=O)C1CCC(NC(=NCCCOc2ccc(C#N)cc2Cl)NCC2CC2)C1 C(CCC(c1ccccc1)NC(=O)Cc1cnco1)NC(CSCC=C)=O C(C(=O)NC1CC1)(C1CCSC1)N(C)CC1(C)CC1 C=CCC(C)(C)C(=O)NCC1CN(C(=O)C(F)(F)CO)CC1(F)F C1(C(C)C(=O)NCF)CCCN(C(=O)C(C)(C)N(C)C)C1 C(=O)(CCCC(=O)NCC)NCCCC1OCCN(C(C(COCC)C)=O)C1 Cc1cc(C(=O)NC(CNC(=O)C(C)O)C2CCC2)c2cccc(C)c2n1 C1(NC(c2cc(Cl)c(Br)c(Cl)c2)=O)CCc2nc(NC(=O)C(F)F)sc2C1 CC1(C)CN(C(=O)C(c2ccc(Cl)s2)=O)CC1NC(=O)C1=NNC(C(F)(F)F)C1 c1(C(C=C)NC(c2cnc(Br)s2)=O)cc(Br)ccc1C N1(CCCNC(=O)C(O)Cc2cnc[nH]2)CCN(C(=O)CCC2CC2(F)F)CC1 CCCCS(=O)(=O)NCC(N1CCOC(C(C)NC(=O)C(F)(F)CO)C1)=O C1(CNC(c2n(CC)ncn2)=O)CCC(C)N(C(c2cncnc2)=O)C1 C1(N(C(CC=CC)=O)C)CCCCN(C(C2CC=C(C)CC2)=O)C1 C1(CC)C(NC(=O)C=Cc2ncc[nH]2)CCN1C(C1CCS(=O)CC1)=O Cc1nc(=NCC(C)(C2CC2)NC(=O)CCc2ccc(OC(F)F)nc2)s[nH]1 N1(C(C(CCC)C#N)=O)CCC2(CC1)CC2CNC(=O)CCn1cc(C)cn1 N1(C(CC2CC(C)(C)C2)=O)CC(F)(F)CC1CCNC(C1CC1CF)=O N1(C(=O)CC2CCCC23CC3)CC2(C1)CN(C(c1cnc(Cl)s1)=O)C2 C1(C(N2C(C(N(CCCCCC)C)=O)C(O)CC2)=O)CCC2(CC1)CC2 Cc1ccc(C(F)(F)F)cc1CN1CCC(C)(C(N2CCC(O)C2)=O)C1 C1(N(C(=O)C(C)=CC(C)(C)C)CC)CCCN(C(c2ccc(N)c(N)n2)=O)CC1 C1(CNC(CC2CC(OC)CN2C(=O)C#CC(=O)N(C)C)=O)CCC(C)(C)CC1 C1(C2CN(C(C34CCCN3CCC4)=O)C2)(NC(C(CC)N2CCCC2=O)=O)CC1 C1(N2CCN(CC(c3ccsc3)=O)CC2)CCCC2(CC1)CC2 c1(C(=O)NC2CCCN(C(=O)C(F)F)C2)ccc2nc(-c3ccccc3)sc2c1 N1(C(C2(C#N)CC(C)C2)=O)CCC(NC(C2(C)CCCC2)=O)C(C)(C)C1 C1(C(N2CCC(CC(=O)NC34CC(CCC)(C3)C4)C2)=O)CC(=O)N(CCOC)C1 C1(NC(=O)OC(C)(C)C)CN(C(=O)NCCc2cc(Cl)cc(Cl)c2)CC1C1CC1 C(=O)(CC(C(C)CC)NC(c1cncc(OC)n1)=O)Nc1cccc(CC)c1F c1(C(N2CC(CN(C)CC3CCSCC3)C2)=O)ccc(-c2cnco2)cc1 c1(C(N2CCC(CNC(C(C(C)C)N(C)C)=O)CC2)=O)cnn2c(=O)cc[nH]c12 C(N=c1[nH]nc(C(N)=O)s1)C1C(NC(C2(C)CNC(=O)C2)=O)CCCC1 N1(C(=O)C2=CCCCC2)CCC(C2CCCN(C(C3COCCO3)=O)C2)CC1 Cc1ncnc2c1CC(C(=O)NC1(CCNC(=O)C(CO)N(C)C)CC1)CC2 C1(C(=O)NC(C2CC2C(N2CCC=C(C)C2)=O)C)CCCCC(=O)N1 C(=O)(N=c1ccn(CC(F)(F)F)[nH]1)N1CCC(C(C)C)C1 N1(C(=O)Nc2nn[nH]n2)CCC(N2CCCC2)(C(F)F)CC1 C1(O)(C(C)NC(CCCc2scc(C)n2)=O)CCN(C(=O)CSC(F)(F)F)CC1 c1(OC)ccc(-n2nnnc2C(C(C)OC)NC2CCSCC2)cc1 S(=O)(=O)(C1CCOC1)NC(c1cc(C(C)(C)C)nn1-c1ccccn1)=O C1(c2nn[nH]n2)(C(C)C)CCN(C(c2cc(O)no2)=O)CC1.C12CCCN(C1)C2=O c1(OC)ccc2cc(C(N3CC(CNC(=O)C(Cl)=CCl)CC(C)C3)=O)n(C)c2c1 C=CCCC(C(=O)OC)NC(c1cc(OC)c(-c2cc(F)ncc2F)cn1)=O c1(C(C(=O)NCCN(C(CC2N(CC)CCC2)=O)C2CC2)C)ccc(C#N)cc1 N1(C(c2cc(C)[nH]c2)=O)CC2(CC2)CC1C(=O)NCCc1ccon1 CC1CC(C(=O)NCC2CN3CCC2C3)N(C(=O)COc2ccccc2)C1 Cc1ccc2nc(-c3nc(CC4CC4)nn3C(C3CCOCC3)C)cn2c1 CC1CCC2(CCC2)CN1C(=O)CSc1ccc2c(c1)CCC2 c1(OC)ncc(C(=O)NCC2CCCCCN2C(=O)CCNC(=O)CO)cc1C C1(CNC(C2(S(N)(=O)=O)CC2)C)CC2(C1)CC(F)C2 C1(NC(C(CC)NC(C)=O)=O)CC2CC(NC(C3(F)CCCCC3)=O)CC2C1 CCC(C)C(CC(=O)NCCC(C(C)C)OC)NC(=O)C(O)CC(N)=O n1(CC(N2C3CN(C(C(CC(C)C)F)=O)C(C3)C2)=O)ccc2ccc(F)cc12 C1(CNC(c2c(C)snc2)=O)CN(C(c2ccccc2)=O)CCN1C.C1(N)CC1 c1(NC(C2CCC2)C)ncccc1S(=O)(=O)N1CCCC1C1CC1 N1(C(c2c(N)nccn2)=O)CCOC2CN(C(=O)CNc3ncccn3)CC12 c1(C(N2C(CNC(=O)Cc3csc(-c4ccsc4)n3)CC2)=O)cccc(F)c1F Cc1nc(CC(C)C)c(C(=O)NC(C)C(CO)NC(=O)CSC(F)(F)F)s1 N1(C(C(C)=CC)=O)CC2CCN(C(=O)C(c3ccccc3S(N)(=O)=O)C)CC12 n1(CC)ccnc1C(=O)NCCCCCN(C(=O)CC1CC1(Cl)Cl)C c1(C(=O)NC2C(NC(C(C)C(C)O)=O)COCC2)c[nH]c2ccncc2c1=O C1(CC(=O)NCCCN(C(=O)CC(C)N2CCCC2=O)CC)CCCC(C)(C)O1 C(CC1=CCN(C(C2(C(F)F)CCCC2)=O)CC1)NC(C1C(OC)CCCC1)=O C(=O)(CC(=O)NCC(CNC(=O)CC1CCCOC1)CO)OCC c1(OC)cccc(C(C)=CC(N2CCN(C(c3ccc(C)s3)=O)C(C)C2C)=O)c1 CN1CCC12CN(C(C13CC(CN1C(C1CCCCC1(C)C)=O)C3)=O)C2 N1(C(=O)C2CC2)CCNC(c2ccc(Br)cc2)C1.C12CCCCC1N2CC(F)(F)F N1(C(CC2CCC(C)(C)CC2)=O)CCCC12CCCN(C(C1CC(CF)C1)=O)C2 c1(CC(=O)NC(CC2CN(C(C(C=C)(F)F)=O)C2)C)ccc(Cl)c(OC)c1 N1(C(C(C)OCC)=O)CCC(NC(c2cnc(F)c(Cl)c2)=O)C(CC)C1 c1(C(=O)NCCC(C)NC(C2CCOC2C(F)(F)F)=O)ncc(C(F)F)s1 N1(C(CC=CC(=O)N(C)C)=O)C(CNC(C2CC2(C)C)=O)CC2CCCC12 CC1CN(C(=O)Cc2cc(Br)ccc2O)CCN1C(c1cc(F)nc(F)c1)=O C(CCS(C)=O)(C(=O)N1CC2(C1)CN(C(C1(c3ccncc3)CC1)=O)C2)N(C)C c1(OC)ccnc(C(=O)NC(C)(C)CN(C(=O)C(O)CC(C)C)C)c1OC N1(C(c2c(CC)onc2C)=O)CCN(C(=O)C(C)CF)C(c2ccccn2)C1 N1(C(C2(OC)CCOCC2)=O)CCC(C(F)(F)F)C(NC(c2[nH]cnc2C)=O)C1 C1(C)(COC)CN(CCCc2cn(CC3CCCC3)nn2)CCO1 C1(NC(c2c(F)cncc2Br)=O)CN(C(=O)CC2CCC2)CCC1F C(C(CNC(=O)CCc1nnc(S)n1C)C(F)(F)F)NC(C1(N(C)C)CC1)=O c1(C(=O)NC(C)CN(C)C(C2CCC(=O)N2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NC(C)CN(C)C(C2CN(C3CCC3)C2)=O)ccc(CO)s1 c1(C(=O)NCC(C)(CO)NC(CC2(COC)CC2)=O)cccc2nc(C)nn12 c1(C(=O)NCCC(C)NC(c2cccc(C(C)C)n2)=O)ccc2c(c1)COCO2 Cc1ccc(Br)c(F)c1CNC1CCC(=O)N(C)CC1 c1(C(=O)NCc2nc(CNC(CCC#C)=O)sc2)cnn(C(C)CC)c1C Cc1ccc(C)c(C(=O)NC2(CNC(=O)C3=CCSC3)CCC2)c1 c1(CC(=O)NCC(=O)NC(CN(C(N2CCCC2)=O)CC)C)cnc(C)o1 C(C(=O)N(C)OCC)NC(c1nc(OCC)oc1)=O.N12CCC(C1)C(C)C2=O N1(C(C=NOC)=O)CC2CC(NC(C3(C4CCOCC4)CC3)=O)CC2C1 C=CC(C(=O)N(C1CCN(C(c2csnc2C)=O)C1)CCO)c1ccccc1 C1(C(=O)NCC(CO)NC(CCNC(C=CC=CC)=O)=O)C(CN(C)C)C1(C)C N1(C(CCSCC)=O)C(C(=O)NCC2CCCSC2)CC2CCCC12 c1(C(N2CCC(N(CCC)C(c3cn(C)nc3CC)=O)C2)=O)c(C)cncc1C c1(C(N(CC(C)N(C(=O)C(N2CCOCC2)C)C)C)=O)csc(S)n1 C1(C)(C(=O)NCC(C(C)C)NC(C=C(C)Cl)=O)CC(C)(C)C1 Cc1ccc(CC(C)NCC2CC(C(=O)OC(C)(C)C)C23CCC3)nc1O CC(C)C1=CCC(C(=O)NCCC2CC(NC(C3(C)CCCOC3)=O)C2)CC1 c1(CC)oc(C)cc1C(=O)NCc1nnn(C)c1C(=O)NCC1CCCSC1 Cc1cn2ccc(C(=O)NC3COCC3NC(C3(OC(C)C)CCC3)=O)cc2n1 c1(C(=O)NC(C(C)NC(c2c[nH]cc2-c2ccccc2)=O)C)ccc(Cl)cc1O C(=O)(CCCC(=O)NC1CCCC1)NC1C(NC(Cc2n[nH]c(=NC)s2)=O)CC1 C(CCCN=[N+]=[N-])NC(C1N(C(CC2CCC(C)O2)=O)CC1C)=O O=C(C#CC1CCOCC1)NCC1(NC(C2CCCC3(CCC3)O2)=O)CC1 C#CCC(C)(C(=O)N1CCCC1CNC(C)=O)NC(=O)CC1CCOC1(C)C c1(C(=O)NC(CC=C)CNC(=O)COC2CCC2)ccc2cc(Cl)ccc2c1 C(=O)(C(C(C)C)NC(=O)CC(C)C)NC1(C(=O)NC2C(OC)C(O)C2)CCC1 c1(C(=O)NCCN(C(c2cc(Cl)no2)=O)CC)cc(C(F)(F)F)ncc1N N1(C(C(c2cccc(Cl)c2)C)=O)CCC(NC(=O)Cc2n[nH]cc2Br)C1C c1(CC(=O)NCC(O)CCNC(c2ccc(C(F)F)nc2)=O)cncnc1O N1(C(C2(OC(C)=O)CC2)=O)CCC(F)(C(=O)NC2(C3CCCO3)CC2)C1 c1(NC(NCCCN(C2(c3ccccc3)CC2(F)F)C)=S)ncccc1O c1(C(=O)NCCCCCNC(C(C)Cn2cccn2)=O)cnc2c(ccn2C)c1 c1(C(=O)NCC(CC(C)C)NC(C2(C)CC=CCC2)=O)c(F)ccnc1Cl C(=O)(C#CC(C)(C)CNC(C1CCC(C2CC2)C1)=O)N1CC(C)C(C(N)=O)C1 N1(C(CN(CCOC)C)=O)C2CCC1CC(CC(C)NC(=O)C(C1CC1)SC)C2 CC(=O)CCC(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cnsc1)C C1(c2n(CC)ccn2)OCCCC1C(=O)NCC1COCCN1C(=O)CC1CC1 c1(OC)cccc(C2CC(O)CN2C(=O)C(N)Cc2cn[nH]c2)c1 N1(C(c2ccc(C#N)cc2)=O)CCC(C2CCCN(C(c3ccoc3Cl)=O)C2)C1 N1(C(c2ccc(CC)o2)=O)CCC(NC(c2cnn(C(C)(C)C)c2Cl)=O)C1C C1(CN(C(=O)CSCCC#N)C)CCCN1C(=O)CCc1ccncc1 c1(NC(C2SCCN(Cc3c(C)cc(Br)cc3C)C2)=O)ccc(Cl)c(C#N)c1Cl C(CC1CCCCC1)(C(=O)NC(C)(CNC(c1coc(C(N)=O)c1)=O)CO)OC Cc1cc(C(=O)NCC2CN(C(=O)C(c3ccn(C)n3)C)CC2(F)F)cc(F)c1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NCC1(F)CCC(NC(C(C)N(C)C)=O)C1 N1(C(=O)C(c2cc(F)ccc2F)=O)CCC(C)C(CNC(C2(CC)CCOC2)=O)C1 C#CC1(C(=O)NC(C)COC)CCN(C(c2ccc(C(C)C)o2)=O)C1 C(C(C(=O)N(C)C(c1nccs1)C1OCCO1)n1cc(CO)nn1)OCC C=C(C)CCC(=O)NCC(C)(C1CC1)NC(=O)CN(C(=O)OC(C)(C)C)C1CC1 C1(C(N2CCC(=CCNC(CCCN(C)C)=O)CC2)=O)CCc2ccnn2C1 N1(C(c2c(NC(C)C)cccn2)=O)CCN(C(c2ccco2)=O)C2CC12 c1(-n2cc(C(c3cc(C(=O)OC)cc(C(O)SC)c3)=O)nn2)cnn2c1OCCC2 c1(CC(=O)NCC(CC)NC(=O)CC2CC3CC3C2)cnn2ccccc12 C1(NC(CCc2onc(C)n2)=O)CC2CN(C(c3nc(Cl)oc3C)=O)CC12 C=C(CNC(c1csc(C(C)C)n1)=O)CCNC(=O)C(C)C1CCOC1 C(C1=Cc2ccccc2OC1)=CC(=O)NC1CN(C(C2CCC(F)(F)CO2)=O)C1 C1(CC(N2CC(O)(CN(C)C(C34CCC(CO3)C4)=O)C2)=O)CCC(=O)NC1=O C1(CN=C(NCC2(OC)CCC2)NCC(F)F)CCOC2(CCOC2)C1 c1(CC(=O)NC2C3CCN(C(C(C)SC(F)(F)F)=O)C32)ccnc(Cl)c1F N1(C(C(N)CCSC(F)(F)F)=O)CCCC(c2ccncc2)CC1 N1(CCC)CCC(C(=O)NC2CN(C(=O)CN(C)C(C)C)C3CC23)CC1 c1(CC)oc2ccccc2c1C(N1CCOC2(C1)CN(C(=O)C(C)(F)CC)C2)=O C#Cc1ccc(C(=O)NCC(C)(O)CNC(=O)CN2CC(=O)N(C)C2=O)cc1C CCCC(C(=O)OC)C(=O)N(CC(O)CN(C(=O)COCCF)C)C N1(C(CC2CN(C(C)=O)C2)=O)CCC2(CC2C(=O)N(C2CCCCCC2O)C)C1 CCC(C)C(O)CC(=O)NCCCCC1CN(C(c2cc(CCCO)on2)=O)C1 c1(C(=O)Nc2cncc(C(N3CCC(N(C)C)C3)=O)c2)ccc(Br)c(F)c1 Cc1ocnc1CCNC(=O)C(c1ccnn1C)NC(=O)COC1CC=CC1 c1(CC(=O)NCC(CC)NC(c2nocc2Cl)=O)csc(C2CCOCC2)n1 C1(N(C(CNC(CC)=O)=O)C)CCCN(C(c2cc(Br)c[nH]2)=O)C1 Cc1cc(F)cnc1NC(c1nc(C(=O)Nc2cnc(C)c(F)c2)cs1)=O c1(C(=O)OCC(=O)NC(C(=O)NC)C)cc(C)nn1CC(F)(F)F CC1CN(C(=O)CCF)CCN1C(C1CCCN1C(c1ccccn1)C1CC1)=O C(C)(CCNC(C1(OC)CC1)=O)N(C(C=C(CC)C)=O)C N1(C(C(C)S(N)(=O)=O)=O)CCC2C1CCCN2C(c1nccc2n[nH]cc12)=O C1(CNC(c2cc(OCC)ns2)=O)N(C(C2CC(C)=NO2)=O)CCCC1(C)C C(=O)(C1CCc2c[nH]nc21)NC1(C)CCN(C(CSCC(=O)OC(C)(C)C)=O)C1 CC1CC2(CO1)CN(C(c1ccc(CNC(=O)C(C)(C)CCF)o1)=O)C2 O=C1CSC(C(N2CCC2C(N2CCC(n3ccnc3)C2)=O)=O)C1 Cc1cc(Cl)ncc1S(=O)(=O)N1CCC2CN(C(=O)NC(C)(C)C)CC2C1.C(C#N)O CCC(CC(=O)NCc1ncnn1C1CC1)NC(=O)CC1OCCO1 CCCCS(=O)(=O)CC(=O)N(C)CC1(O)CCN(C(c2ccccc2CO)=O)C1 CC1(C)CN(C(=O)Cc2ccccc2O)CC1NC(=O)C(O)Cc1ccccc1 CC(C(=O)NC1CCN(C(=O)Cc2nc(C3CC3)nn2C)C1C1CC1)C(C)(C)C Cc1ccc(C(N2CC(CC(=O)NC3CC(C)OC(C)C3)C3(CC3)C2)=O)c(O)c1 Cc1nc(C(N2CC3CC2CC3N2CCCC(C(C)(C)O)C2)=O)ccc1Br N1(C(C(CSC)C)=O)CC(NC(=O)C(C2CCCCC2)O)C(CC(C)(C)C)C1 c1(C(N2Cc3cccnc3C2)C(=O)NCCCC2CC2)nc(Br)c2ccccn12 c1(C(N(C(CCNC(c2cc(CC)[nH]n2)=O)C)C)=O)ccc(C(C)=O)cc1 C(CC(=O)N)OCCOCCCC(F)(F)F.C(CCN(C(=O)C)C)OCCOC N1(C(c2cccc(OCC)c2)=O)CCC(C)N(C(c2c[nH]ccc2=O)=O)CC1 c1(NC)cnncc1C(=O)NCC1CCC1NC(C1(F)CC1)=O c1(C(=O)NC2CCC(C)N(C(=O)COc3cn[nH]c3)C2)cncc2ncn(C)c12 c1(C(N(C(CC)CO)C)=O)c[nH]nc1C1CCN(C(=O)C(C)C)C1 c1(C(=O)NC2CN(C(CCOC)=O)CC(O)C2)nn(C)c(=O)c2ccccc12 C(=O)(C(CNC(c1ccc(F)cn1)=O)CC1CCCC1)N(CCCF)CC C1(C(=O)N(CCC(C)(C)NC(=O)CSC(F)F)C)(OC)CCSC1 c1(C(=O)NC2CCC2NC(C2CCS(=O)(=O)C2)=O)cnc2nccnc2c1 C1(CC(=O)NCCC(C)(C)NC(c2cc(OC)n[nH]2)=O)CCCCN1C c1(C(=O)NCCOCCCNC(c2c(CC)noc2)=O)[nH]cc2c1CCCC2 N1(C(c2cncc(OCC)c2)=O)CCCC2(CCC(NC(=O)CC(F)(F)Cl)C2)C1 CCC(CC(=O)NC(C)C(C)NC(=O)COC1CN(C(C)=O)C1)SC C1(C(=O)NCC(C)CNC(=O)CCc2cn[nH]c2)C2CCN(C)CC12 c1(OCC(N2C(CNC(C(C)OC)=O)C3CC3C2)=O)cccc(F)c1F c1(C(N)=O)ccccc1-n1ccc(-c2cnc(C3CC3)nc2)n1 N1(C(c2cc(SC)oc2C)=O)CCC=C(CNC(=O)CC(C)(C)CN(C)C)C1 c1(C(N)=O)cccc(C(=O)NC2CN(C(c3csc(F)c3)=O)CC2C(F)F)n1 C1(C(=O)NC(C)CNC(=O)CCc2cnco2)CCC(=O)N1 CC1(C)CC(NC(C23CSCC2C3)=O)CCO1.C12(CCCCC1)C(=O)NO2 C1(CCC)(NC(c2nn(C)nc2Br)=O)CCNC1=O N1(C(c2c(C3(C)CC3)c[nH]c2)=O)CC(C)(C)C(NC(=O)C(Cl)=CCl)C(C)(C)C1 C(=O)(C(CNC(=O)CC1CC1(C)C)CC1CCCC1)NCCSC N1(C(C2CC(SC)C2)=O)CCCC(C)(C)C1CNC(c1cncn1C1CC1)=O C1(CCNC(C2(CCNC(c3n(C)nnc3)=O)CC2)=O)CCC(C)(C)O1 CN=S(=O)(c1ccc(C(=O)OC)cc1)N(C)C.C12CCC3(CC(C3)C(=O)NC1)O2 Cc1cccc(F)c1C(=O)NC1CN(C(=O)Cc2ccc(F)cc2)CC1CO c1(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)C(F)(F)F)cccc2c1COC2 c1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)N(C)C)C2)n[nH]c2c1CC1CC21 O=S(=O)(c1cnc(NCc2sncc2Br)c(Cl)c1)N1CCCC2(C1)OCCO2 CC1CCN(C(c2ccc(CCC(=O)Nc3cnn(C)c3)[nH]2)=O)CC1(F)F Cc1ccc(C(N2CCC(C)(NC(c3cc4sc(C)nc4[nH]3)=O)C2)=O)c(F)c1F c1(C(=O)NCC2N(C(c3cn(C)nn3)=O)CCC2)cncc(N)n1 C1(CNC(C(CC#C)C2CC2)=O)CCN(C(=O)CCCCC)CCC1(F)F C(=O)(CCCCCCNC(C1CC(=O)CC(=O)N1)=O)NC(C(CC)C)C(=O)NC n1(CCOCC)nc(-c2cccc(CC)c2)nc1-c1cnc(-c2ccco2)s1 c1(C(N2CC3CC(O)CC2C3)=O)cc(Br)c2nccnc2c1 N1(CC(=O)N(CCNC(C(C(C)SC)O)=O)C(C)C)C(=O)CCCC1=O N1(C(C2C(CC)CCO2)=O)CCCCC1CCC(C)(C)NC(=O)Cc1cnoc1 CCC(C)C(C(=O)N1CCCC1CNC(C1OCCC1C)=O)N(C)C N1(C(c2cc3n(n2)CCC3)C(=O)NCCOC)Cc2ccc(OC)cc2CC1C c1(C(=O)NCCC(C)N(C(C(CC)OC)=O)C)cc2cc(F)cc(F)c2[nH]1 N1(C(c2cccc(C)n2)=O)C2CCC1CC(NC(C13CCC1C3)=O)C2 c1(C(N2C(CN(C)C(c3nnsc3N)=O)CCC2)=O)ccc(O)nn1 C1(NC(c2cccnn2)=O)CCCC12CN(C(c1cc3nc[nH]c3cn1)=O)C2 C1(CNC(c2c(C)cns2)=O)CCCC(NC(c2ncnn2C2CCOCC2)=O)C1 C1(C(=O)NCC2(O)CN(C(C3C(OC)CCCC3)=O)C2)CCC(N=[N+]=[N-])C1 C(c1nc2ccccc2[nH]1)=CC(N1C(CNC(C(C(C)C)(C)O)=O)CC(F)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(CCC=C)=O)CC(F)(F)F Cc1cn2c(C(C3CCCC3)NC3CN(C(=O)C(C)CC(N)=O)C3)cnc2s1 c1(C(=O)NCCC2CN(C(C(CCC)C)=O)C2)ccnc2cc[nH]c12 C1(C(NOCCOCC)=O)CN(C(=O)C(C)(C)CF)CC(C)O1 c1(C(=O)NC2C(NC(CCCC)=O)CCC2)ccc(C(C)C)cn1 c1(OC)cccc2ccc(C(=O)NCC(C)NC(c3cc(=O)n(C)cn3)=O)nc12 CC1CN(C(=O)CCc2nncs2)CC1(C)CNC(=O)C(c1cccn1C)=O C1(CCc2ccncc2)(NC(N2CCCC2)=O)CN(C(=O)COC2CCOC2)C1 C1(CNC(CC(C)OC)=O)CC2(CCOCC2)CN1C(c1ncccn1)=O N1(C(CC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)C1Cc2c(Cl)cccc21 O=S(=O)(c1cc(Cl)c(I)s1)N1CCCC1c1cc(F)c(F)c(F)c1 C(CC(CC)C(=O)N(CCCCN(C(=O)CC(C(F)F)n1ccnc1)C)C)=CC C1(C(=O)NC(C)CCO)CCCN(C(c2cc(Cl)c(Cl)s2)=O)C1 Cc1cc(C(=O)NC2(C)CCC(NC(c3ccon3)=O)CC2)cnc1O C1(C(N2C(C(=O)NC3CC(C)(CC)C3)C3CC3C2)=O)CC2OC1C1CC21 c1(C(N(CCCNC(c2cnn(C(F)F)c2)=O)CCO)=O)ccc2c(c1)CCO2 N1(C(Cc2c(C)n[nH]c2C)=O)CC2CCN(C(C3C4CC5C(C4)C35)=O)CC12 C(=O)(C(C)CC(C)(C)C)N1C(CN(C(=O)CC(C)(C)C(F)F)CC)CCC1 C(CCC(=O)N(C)C)NCCNC(C)=O.n1(C)cc(-c2c[nH]nc2C(=O)OC)nn1 CCCC(O)CC(=O)NCCC(C)N(C)C(c1scnc1COC)=O N1(C(C(Cc2cn(C)nn2)NC(=O)OC(C)(C)C)=O)CCCC(c2cccc(F)c2)C1 N1(C(C2CC(C)CN2C(=O)C=Cc2ccccc2)=O)CCC(O)C(C)(CO)C1 Cn1cc(C=CC(=O)NCCCCCC(=O)NOCC2(C)CC2)nn1 c1(C(=O)NCC2(NC(c3cnc(C(C)(C)C)o3)=O)CCC2)cc2cn[nH]c2cn1 C(=O)(C(CC(C)C)NC(c1sc(C)cc1C)=O)N(CCC#C)CC N1(C(c2n(C)ccc2)=O)CCCC2(CCCN2C(C2CCc3c[nH]nc3C2)=O)C1 c1(C(C)NC(CC(C)n2cccc2)=O)ccc(CNC(=O)COC2CC2)cc1 CC(C(=O)N1CCCCC(NC(c2ccsc2C#N)=O)C1)C(F)(F)C(F)F c1(C(=O)NCC2OCCC(NC(C3CCN(C)C3)=O)C2)cc2c(Cl)nccc2o1 C1(CC=C)(C(=O)NCCP(C)(C)=O)CCN(C(=O)C(C)O)C1 C1(NCc2c(OC)nc(Cl)cc2)CC2(C1)CC1(CCCC1)C2 CC1(C)CCN(C(c2cccc(F)c2F)=O)C1CNC(C1(C)CCCS1(=O)=O)=O c1(C(N2CCC(c3c(F)cccc3F)(C)C2)=O)cnc2ccccn2c1=O c1(CC)ccccc1C(CNC(c1ncncc1Cl)=O)NC(c1cc(F)n[nH]1)=O C(C1=CCN(C(=O)CCCSC)CC1)NC(CCc1onc(C(C)OC)n1)=O O=C1CC2CCC1C(C(=O)Nc1cncc(-c3ccc4c(c3)CCO4)c1)C2 C(=O)(CCCCC(=O)NCC1CC1NC(=O)COCCc1cccs1)OC c1(N(C)CC2CN(S(=O)(=O)Cc3ccc(Cl)c(Cl)c3)C2)cccc(C#N)c1[N+](=O)[O-] CON1CCC(C(=O)NCC2C=CCN2C(c2cc(C3(C)CC3)n[nH]2)=O)CC1 N1(C(C=COCC)=O)CCC2C(CCN2C(C2C3COCC23)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC(C)CN(C)C(C1CCCCN1S(C)(=O)=O)=O C1(NC(C(c2ccccc2F)C)=O)CCN(C(=O)CC2CCCC23CC3)CC1 N1(C(c2cc(Cl)ccn2)=O)CCN(C(C2CCS(=O)CC2)=O)C2CS(=O)(=O)CC12 Cc1cnc(N2CCOC(CN(C)C(c3cc(Cl)nn3C)=O)C2)nc1 c1(OC)ccc(C(=O)NCCC(C)CCNC(c2cc(SC)oc2C)=O)c(F)c1 C(C(C(=O)NCc1ncn(C)n1)n1cc(CN2CCNC2=O)nn1)OCC Cc1nc(Cl)ccc1CC(=O)NCC1CCCCC1NC(=O)C(C)n1cccn1 N1(C(CNC(CC)=O)=O)CC2CCC1C(CNC(=O)C(C)CNC(=O)C(C)=O)C2 C1(SCC(=O)NCCC(Cn2cc(C(C)(C)S(C)(=O)=O)nn2)F)CCC(=O)NC1 C1(CC)CN(C(C2CC(c3cc(OC)ccc3Cl)C2)=O)CC(=O)N1 C(=O)(CCC(CC)CC)N1CCC2(C(C(NOCC=C(C)C)=O)C2)C1 N1(C(c2cc(F)ccc2Cl)C(=O)NCCCSC)CCC(O)CC12CC2 C1(CN(C(C2CC(SC)C2)=O)C)CCCN1C(=O)C(C)=C1CCCC1 N1(C(C2CC(OCC)C2)=O)CC2(CCC2)CCC1C(=O)NCC1(C)CCCCC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCc1cccc(CNC(CCCCOC)=O)c1 c1(C(=O)NC23CN(C(C(COC)(C)OC)=O)C(CC2)C3)cc(F)c2[nH]nnc2c1 C(=O)(CCCCCF)NCCn1ccc(C(=O)NCC(COC)C(C)C)c1 c1(C(=O)NCC(CC)NC(c2cccc(N)n2)=O)ccccc1NCCO c1(C(=O)NCCCN(C(=O)CCN(C)CCO)C(C)C)ccc2nc(O)[nH]c2n1 c1(-c2c(C3(C(N4CCCC5(C4)OCCO5)=O)CC3)cccc2)cccc([N+](=O)[O-])c1 N1(Cc2c(OCC)cccc2)CCC(=O)N(CCc2cnoc2)C1=O C1(CC(=O)N(C(C=C)C)C)CC(C)(C)CN1C(=O)Cn1nccn1 c1(C(=O)NC(C(C)NC(CCCC)=O)C)c[nH]c2cc(C(=O)OC)ccc12 N1(C(C(C)N(C(C2(CC)CCCC2)=O)C)=O)CC(F)(C2CC2)C1 c1(OC)ccc(C(C)C(=O)NC2CCCC2NC(C2(O)CC3CC2C3)=O)cc1 N1(C(C(C)N(C(=O)C2CC2)C(CSCC=C)=O)=O)CCC(C)(C)C1 C1(NC(C(C)c2cccs2)=O)CC2C(NC(=O)CCCn3cncn3)C2C1 c1(-c2cn(CCN(C(CC(=O)OCC)=O)C)nn2)cccc(S(C)(=O)=O)c1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C(C)NC(=O)CC2COC(C)(C)C2)CC1 N1(C(C2C(=C)C2)=O)CC(C(=O)NC2CNC(=O)C23CC3)CC(C)(C)C1 c1(CC(C(=O)NCC(C(C)(C)C)NC(CCC(=C)Cl)=O)C)ccc(C#N)cc1 CC1(C)CN(C(C23CCNCC2CNC3)=O)Cc2ccccc21 c1(C(CC(=O)OCC)NC(c2ccc(NS(C)(=O)=O)cc2)=O)ccc(Cl)c(F)c1 Cc1nc2ccc(Br)cc2c(NC2CCCn3cnnc32)c1C c1(C(CC)NC(=O)NC(c2ccccc2)CC)ccc(C)cn1 N1(C(C2(CC=C)CCCC2)=O)CCN(C)C(CNC(C2CC2COC)=O)C1 c1(-c2cccc(N)n2)cc(N2CCCC2=O)ccc1F.Cc1cc(C=O)on1 c1(C(N(CCC(C)NC(c2ccc(C3CC3)o2)=O)C)=O)snnc1C(C)(C)C C(C(C(C)C(C)C)NC(=O)CNC(c1ccccc1)=O)NC(CC(CC)OC)=O C1(C(=O)NCCOCCOCCNC(c2cn(C)nc2)=O)CCS(=O)(=O)N1.C1CC1 c1(OC)c(Cl)ccc(C(N2CC(NC(=O)CCC3(C)CC3)CC2C)=O)c1F C1(CNC(C2(C)CC2(F)F)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CCC12CCC2 c1(C(=O)NC2CCOC2)ccccc1.C1(=O)CCOCC(=O)NC2CC(C2)N1 C12(C(=O)NCC(=O)NCC(C)C)CC1CCN2C(=O)CC=C(Cl)Cl C#CC(C)(C1CCOC1)NC(=O)C=CC(C)NC(=O)CC=CCC C1(NC(=O)NCC(C)OCC)CSC(C)(C)C1 C1(CNC(=O)COCC2CC2)CC12CCN(C(c1ccsc1Br)=O)CC2 c1(NC(c2cncc(NCc3ccc(C)c(Cl)c3)c2)=O)cc(F)c(C#N)cc1Cl N1(C(CSC)=O)CCCC(C)(C)C1CNC(C1CN(C(N)=O)C1)=O CC(CN=c1ccc([N+](=O)[O-])c[nH]1)NC(C1CC2(CC2)C1)=O c1(C(=O)NCC(CN(C)C(c2cnn(C)n2)=O)(C)C)ccnc(S(N)(=O)=O)c1 N1(C(C2(OC)CCC(C)C2)=O)CCCC(CCNC(=O)CC2(N(C)C)CC2)CC1 C1(C(NNC(=O)NCC2(C)CCCCC2)=O)COC2(CCC2)C1 c1(N(CCCNC(C2CC3(CC(=O)N3)C2)=O)C)nc2cc(F)cc(F)c2o1 C1(CC(N)=O)(C(C)NC2CC(n3cc(C(C)C)nn3)C2)CCCCC1 C(C)(C)(CC(=O)NC1(CCOC)CCN(C(=O)C(C)OC2CCCC2)C1)OC N1(C(c2ccc(C3CC3)o2)C(=O)Nc2c(C)cccc2C)CCCC2CCCC12 CC1=C(C)CC(C)(C(=O)NC(C)CCNC(c2cc(C#N)[nH]c2C)=O)CC1 c1(-c2c(NC(C)=O)cccc2)cccc2[nH]c(C(=O)NCC(O)C(F)(F)F)cc12 C1(C)(C(N(CCCCCC)C)=O)CCN(c2ccnc(N(C)C)n2)C1 CCC(CC)CCC(=O)N1CCCC(CC)C1C(=O)NCC1(CC(C)C)CC1 c1(OC)cc(O)c(C(=O)NC2CCC(Nc3cc(C(F)(F)F)ncn3)C2)cc1Br N1(C(Cc2nc(C)oc2)=O)CCN(C(c2nc(C(F)(F)F)ccc2F)=O)CC1C C(=O)(CCCc1ccccn1)NCC(C)N(C)C(C1CCC1C)=O CCC(C)C(CC)(c1nnnn1C(C)C)NC(C)CCC(=O)OC C1(C(=O)NCC2COCCN2C(C23CCCC2C3(F)F)=O)CN2CCCN1CC2 CC(C)CCC(O)C(=O)NC(C)CCCC(N1CCCNC(=O)CC1)=O C1(NC(=O)CC2CCC(=O)N2)CCN(C(=O)CC2(N3CCCC3)CC2)CC1O N1(C(C(C(C=C)C)C)=O)CC2CCC1C(CNC(c1c(C)cccc1Cl)=O)C2 N1(C(COC2(C)CCC2)=O)CC(C)(C(=O)NCC2(C)CC(O)C2)CC1(C)C CCS(=O)CC(=O)NC(c1ccccc1CO)CNC(=O)C(C)OC(C)(C)C CC(C)CCC(O)C(=O)N(C)CC1CCN(C(=O)Cn2cnc(C#N)n2)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC(C2CCCN(C(C3(C)C=CCC3)=O)C2)C1 n1(CC)c(C)cc(C(N2CCCC2CN(C(=O)C=Cc2cocn2)CC)=O)c1C FC1(F)CC1C1CCCN(c2nc(N3CCCCCC3)c3ncsc3n2)C1 C1(CNC(c2cccnc2Cl)=O)CCN(c2ncc(I)cn2)CC1(F)F C1(C2CN(C(=O)Nc3cn[nH]c3)C2)CCCCC1=O N1(C(C=CSC)=O)CCN(C2COCC2NC(=O)Cc2ccns2)CC1 N1(CC(N2C(N(C3CCC3)C)CCC2)=O)CCN(CCc2ccno2)CC1 C1(CC#N)CC12CCN(S(=O)(=O)CCCN=[N+]=[N-])CC2 c1(CN2CCC(C#N)(c3ccccc3)CC2)ccc2nn(C)cc2c1 N1(C(C(C)(C)C)=O)CCC2(CCC2NC(C23CC(F)(C2)C3)=O)CC1 C1(CNC(c2cn(CCO)nn2)=O)CCN(C(C23CSCC2C3)=O)C1 c1(NC(C2(OC)CCSC2)=O)ccc(NC(=O)C(C)CC(C)C)cc1C C1(C=O)C(C)C1(C)C.c1(C(C)CCO)nnc(O)o1.C12CC(C1)C(=O)NC(=O)C2 C12(C(=O)NC3(CC=C)CN(C(C4CCCN4CCC)=O)C3)CC1COC2(C)C C1(NC(c2c(C)coc2)=O)CCC2(CCN(C(c3sc(O)nc3C)=O)C2)C1 C1(C(N(C)CC2CCCN2C(=O)CCc2cnoc2)=O)CCS(=O)(=O)C1 c1(C(=O)NC2C(CNC(C(C)SC)=O)C2)ccc([N+](=O)[O-])cc1-n1cnnn1 c1(C(=O)NC2C(OC)CN(C(=O)C(C3CCOCC3)C)C2)cc(S(N)(=O)=O)co1 C1(N(C)C(c2cnn(CF)c2)=O)CCCCN(C(C2CC(=O)C2C(C)(C)C)=O)C1 c1(C(N2CC(C)C(C(=O)NCC3CCC(C)CC3)C2)=O)cncc(C#N)c1 Cc1ccc(SC(C)C(=O)NCCC2CCCN2C(=O)CCCF)cc1 Cn1cnc2ccc(CN3CCOCC3CCN)cc12 C1(C(N2CCN(C(C=CC)=O)CC2)=O)Cc2nn[nH]c2C(C)C1 Cc1cccc2c(C(N3CCCC(F)(CNC(=O)C(F)C(C)C)C3)=O)n[nH]c12 CCC(C)C(C(=O)N(CC(C)COC)C)NC(C1CCCC1CC)=O c1(CC(=O)N(CCNC(=O)CSc2nncn2C)CC)cnc2cccnn12 C1(NC(c2cnoc2)=O)CCCCC12CCN(C(c1ccns1)=O)CC2 C1(C(=O)NC2CN(C(c3coc(O)n3)=O)C2)CCc2nnc(O)n2C1 N1(C(CN2C(=O)CCC2)=O)CC2CCN(C(c3ccccn3)=O)C2C1 CCC(CC)(CCOC)C(=O)N(CC(O)CN(C)C(C1CC2(CC2)CN1C)=O)C N(C(=NCC(c1ccccc1)N1CCCC1)NC1CCCC1)C(C#C)COC C1(C(=O)NCC2CN(C(C3C(C)(Br)C3)=O)C2)Cc2cc(F)ccc2C(=O)O1 c1(COC)cc(C(=O)NC2CCCC2NC(=O)C=Cc2cc[nH]c2)n(C)c1 C1(OC)C(OC)CNC1NS(=O)(=O)Cc1nc(-c2ccccc2)ns1 c1(C(=O)NC2CCC(NC(C(C)CF)=O)C2)noc2c1COCC2 C1(n2cccn2)(CNC(C(CSC)O)=O)CCN(C(C2(CCF)CCC2)=O)CC1 N1(C(C2(C)COC(=O)C2)=O)CCOC(C)(CNC(=O)CCS(C)(=O)=O)C1 c1(-c2nccc(NCc3nc(C)sc3)c2)ccc2c(c1)C(C)C(C)O2 n1(C(C)C)cc([N+](=O)[O-])c(=NCC2CCCN(C(C3CC=CCC3)=O)C2)[nH]1 C(C(CC(C)C)C(=O)NCC(C(=O)OCC)OC)NC(CCOCC#C)=O N1(C(CCC(C)N(C)C)=O)CCC(CO)(NC(c2cc(C(F)F)[nH]n2)=O)CC1 C1(C(=O)NC2COCC2NC(c2ncsc2C)=O)(OC)CCC(C(F)F)CC1 N1(C(COc2c(OC)cccc2)=O)CC(NC(c2ccncc2O)=O)C(C)(C)C1 N1(C(Cc2ccc(C)cc2)=O)CC(C(=O)NC(C(N)=O)C2CC2)OC(C)C1 c1(C(=O)NC(CNC(C(F)=CC)=O)CCOC)sc2cccc(Cl)c2c1Cl c1(N(C(=O)CCN(CCO)C2CC2)C(C2CC(F)C2)C)cccc2occc12 N1(C(=O)OC(C)(C)C)CCC2(CCC(CNCc3ccnc(Cl)c3)C2)CC1 C12(C(=O)NCC(C=C)(C)C)CC(CO)(CN1C(=O)CCNC(=O)OC)C2 C1(CC)CC(O)CN1C(C1CCOC1CNC(=O)C(C)OC(C)=O)=O C(CCCC(=O)NCCCC(C)NC(=O)CC(c1ccccc1C(F)(F)F)C)OC C1(CNC(c2ncn(CC)c2)=O)CN(C(c2cc(SC)ccc2C)=O)CCN1C CCC(C)(COC)C(=O)N1CCCCC(C(=O)NCC(C2CCC2)OC)C1 N1(C(c2cccc(Cl)c2Br)C(=O)NCCSC)CC(C)CCC12CC2 c1(CC)cc(C(=O)NC(C)(C)CNC(C2CC(OCCOC)C2)=O)c(F)cc1C C12(C(=O)NCC(C3CCN(C(C45CC4C5)=O)CC3)(C)C)CCC(F)(CC1)CC2 CC1(CNC(c2ncc(C(F)(F)F)s2)=O)CCN(C(=O)CCCCO)C1 C1(C(N2CCC(N(C(CC3CCC(C)CC3)=O)C)CC2)=O)CC2(C1)CC(O)C2 C=C(Cl)C(C)(C)C(=O)NCC1CCCCN(C(C2CCN(CCF)CC2)=O)C1 c1(C(C(N2CCC(O)(C(C)NC(C(C)CO)=O)C2)=O)C)nc(F)ccc1Cl C1(C(N2CCCC(N(C)C(c3cnn[nH]3)=O)CC2)=O)CC(=O)C12CCCC2 c1(NC(C(C)CC2CCCO2)=O)ccc2ccn(CC(=O)N(C)C)c2c1 C1(C)(C(N(C)CC2(CC(C)C)CC2)=O)CCCN1C(=O)CC(C)n1cccn1 N1(C(C(C)CC(C)(C)C)=O)CCC2CCN(C(=O)CCc3cnn(C)c3)CC2C1 N1(C(=O)NCCN2CCCC(OC)C2)CCc2cc(Br)cc(F)c2C1 N1(C(c2nc(C(C)=O)sc2)=O)CCC(C(C)C)C1CNC(=O)Nc1ccco1 Cc1c(CCC(=O)NC(C)CCN(C(=O)C=CC(F)(F)F)C(C)C)cnn1C N1(C(C=Cc2ccn(C)c2)=O)CC(C)(C)CCC1CNC(c1cnco1)=O c1(C(=O)NCC(CC)NC(C2C(OC)C2)=O)c(C(C)=O)sc2ccccc12 CCC(C)CCC(=O)NCc1ccc(CN(C)C(C2(F)CC=CCC2)=O)cc1 CC1CN(C(=O)C(Cl)Cl)CC1(C)C(=O)NCC1(C(C)O)CC1 CC1(C(=O)NCCC(O)CNC(C2(Br)CC2)=O)CC(F)(F)C1 C(C(C)C(C)C(=O)N(C)CC1CCN(C(C2CC(OC)C2)=O)CC1)OC N(C1CC2(CN(C(c3ccc(F)s3)=O)C2)n2ccnc21)C(c1ccc(C)nn1)=O c1(CC(=O)NC2(C3CN(C(C4C(C)(C)C4)=O)C3)CC2)cccc2sccc12 N1(C(C(CC)(F)F)=O)CCN(C(c2cc(CCCO)on2)=O)C(CC(F)F)C1 c1(OCC)cccc(CNC(C2CC(C)(C)O2)=O)n1 C1(NC(c2cnc(OC)nc2)=O)CC2CC(NC(C3COC3)=O)CC2C1 C1(C(N(CC#C)CCF)=O)CCCCC1NC(=O)C(CO)NC(N)=O C1(NC(CCc2nc(C)c(C)[nH]2)=O)CC2CCC(C1)N2c1ncncc1Cl N1(C(c2scc(C)c2C)C(=O)NCCCSCC)CCC(O)C(C)(C)C1 c1(CCC(=O)NCC2(CNC(c3c(C)scc3)=O)CC2)ccc(Cl)cc1Cl N1(C(c2c(CC)csc2)=O)CC2(C(=O)NCC(c3nccs3)C)CCC1CC2 N1(C(C(C)(C)OCC(F)(F)F)=O)CC2(CCC(CNC(=O)CC34CC(C3)C4)O2)C1 Cc1ncc(NC(=O)C(CO)NC(c2csc(=N)[nH]2)=O)c(C)c1C N1(C(C(=O)N)=O)CCOC(C(=O)OC)C1.C1(C)(NC(=O)NC)C(=O)C1CC N1(C(c2occ(OC)c(=O)c2)=O)CCCC2(CCC2NC(=O)CC2CC2)C1 C(=O)(C(CC(C)C)C(C)C)NCC1C2CN(C(c3c(C)csc3)=O)C1C2 N1(C(c2nn(C)cc2Cl)C(=O)Nc2c(C)cc(F)cc2)CCC(C)C(O)CC1 C(=O)(C#CC1CCC1)NC1CC(C(C)NC(C2CC(=O)N(C(C)C)C2)=O)C1 c1(C(=O)NCC2N(C(CCc3cc(OC)no3)=O)CC2)ccc(Br)cn1 CCCCC(CNC(C1(C)COC1)=O)NC(C1CC(C)N(C)C1)=O CC(Cc1ccccn1)C(=O)N(CCCNC(=O)CSc1nnnn1C)C C(=O)(C(C)(F)C(C)(C)F)NCC(C(C)(C)C)NC(c1ccc(C#N)cn1)=O c1(C(N2CC(CCOC)C2)=O)cnn(CCNC(=O)C(C)C2CCCO2)c1 c1(OC)cccn2ncc(C(=O)NCC3(C)CCCN(CC(C)O)C3)c12 CN1CC(C)(C(=O)NCC2CCCN2C(c2cc(C(F)(F)F)ncn2)=O)CC1=O C(=O)(CC(C)(O)COC)NCC1(OC)CN(C(c2nnn(CCC)n2)=O)C1 N1(C(C2N(C)CCOC2)=O)CCC(F)(CNC(=O)CCCCn2ccnn2)CC1 Cc1c(C(N2CCCC(CNC(=O)CS(C)(=O)=O)CC2)=O)ccnc1Cl CCC(CC(=O)N1CC(CNC(c2ccc(-c3cccs3)cn2)=O)C(O)C1)OC c1(C(=O)NC2(CO)CN(C(c3ccn(C4CC4)n3)=O)C2)nc2c(s1)COCC2 CC1CC(C)N(C(=O)CSc2ccccc2)CCN1C(c1cc(O)nc(Cl)c1)=O C1(CC=C)(NC(c2cnc(C3CC3)nc2)=O)CCN(C(=O)C(C)n2cncn2)C1 c1(CNCC(c2ccc(OC)cc2)O)cnc2c(Br)cccc2c1 N1(C(=O)OC)CSCC1C(=O)NCC1(F)CC(C(C)(C)C)C1 N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCCN2C(C)=O)=O)C1 C1(C(=O)NC2CC(C(C)O)C2)CCC(O)CN1C(c1cccc(F)c1)=O c1(OC)cc2ccccc2cc1C(N1CC(NC(=O)CC2CCC(=O)N2)C1)=O N1(C(C(CCCC)F)=O)CCC2(CC1)CC2NC(=O)C=Cc1ccc(C(F)F)o1 c1(NC(C(C2CCN(C(c3ccncn3)=O)CC2)C)=O)nc(Cl)ccc1I N1(C(C(C=C=C)C)=O)CCCCCC(NC(c2cc(C)cc(C)c2C)=O)C1 Cc1cncc(C(=O)NC2CCC(NC(C3CCC(C(N)=O)O3)=O)CC2)c1C CC1(C)CC(CNC(c2cccc(N)c2)=O)CN1C(=O)C=Cc1ccccn1 c1(OC)cc(C(=O)NC2CN(C(=O)CCc3cnn[nH]3)CC2OC)ccc1Cl C12(NC(CNC(CC)=O)=O)CC(NC(c3cnoc3C3CC3)=O)(C1)C2 N1(C(C(C)C2CCCC2)=O)CC(C2(NC(=O)CCN3CCC3)CC2)C1 c1(C(=O)CC)cc(=NCC2(O)CC(CN=c3[nH]cc(CC)s3)(OC)C2)[nH]c(C)n1.OC Cc1nccn2ncc(C(N3CC4CC(NC(=O)C(O)C5CC5)C3C4)=O)c12 N1(C(C2N(C(C(CC)n3cncn3)=O)C3(CC2)CC3)=O)CC(O)C(O)C12CCC2 C1(C)(C(=O)NCC(C)(F)CNC(C2CC3CC3C2)=O)CCC2CC2C1 Cc1cc(C)n(CC(=O)NCC2CCC(NC(=O)C(C)OC3CCCC3)C2)n1 c1(CC2C(C)(C)C(CO)O2)ncnc2c1ncn2C.c1(C(=O)O)nc2ccccc2s1 CC1CN2CCN1CC2C(N(CC(C)(C)NC(c1csc(C(F)F)n1)=O)C)=O c1(C(=O)NCC2C3CN(C(C4CC(=C)C4)=O)CC32)cc(F)c(C)cc1F N1(C(c2c(C)nn(C)n2)=O)CC(O)(C2(CNC(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)C1 c1(OC)ccc2c(c1Br)C(NC1(c3ncccn3)CC1)CC2 C(=O)(CC(=O)N1C(C(=O)NC(c2ccncc2)(C)C)CC1C)NCC n1(CC(=O)NCC(C(=O)N(CCC#C)CCOC)OC)cccnc1=O N1(C(c2c(CS(N)(=O)=O)n[nH]c2)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 c1(CNC(C2(CC#C)CCC2)=O)c[nH]nc1C1CCN(C(c2cscn2)=O)C1 c1(NC(C2(C)CN(C(C(C)OC)=O)C2)=O)cnc(Cl)nc1C c1(C(N2CCCC(C)(NC(CNC(=O)NC)=O)C2)=O)cccc2nc(C)nn12 C1(CC(=O)NCC(N(C)C)C2CC2)CCC(NC(=O)C=Cc2ccco2)C1 C=Cn1nccc1C(N1CC(NC(c2sc(C)cc2OCC)=O)CC1CO)=O C1(NC(c2c(C)noc2)=O)CC(F)CN(C(=O)C(C)Oc2ccc(Cl)cc2Cl)C1 CC(CC(=O)NC1CCC(NC(=O)CNC=O)C1)C1CCCC1 N1(C(C=C(C)C(C)(C)C)=O)CCSCC1C(=O)NCCc1ccc(C)cc1 C1(CC(=O)NC(CC)(C)CNC(c2cscc2F)=O)CC=CCN1C CC1CCC(NC(=O)CNC(=O)C(F)(F)F)CN1C(c1ccnc(CO)c1)=O C1(C(=O)NCCCn2cnnn2)CCCCC1NC(C1CCSC1)=O C1(CNC(c2c(CC)noc2)=O)CC2CC(C1)N(C(=O)CSC)C2.N1(C=O)CCCC1 c1(C(N(CCN(C(C2SCCCS2)=O)CC)CC)=O)cnn2c1N(C)CC2 C(=O)(C(C)N(C(C1CN(c2ncco2)C1)=O)C1CC1)NCC N1(C(C2CCC(=O)N2)=O)CCC2(CC1)CC(C(=O)O)CCO2 C1(c2cccc(OCC#C)c2)NC(=O)N(CC2CSCCS2)C1=O C=CCCCCCC(=O)NCc1ccc(CNC(C2(C)CCC(F)(F)C2)=O)cc1 n1(CC(=O)NC(c2oc(C)nc2C)c2ccc(C)o2)cc(C(N)=O)c2ccccc12 N1(C(C2C(COC)C2)=O)CC2CC1CN(C(c1cc3occc3n1C)=O)C2 C1(NC(CC2(C(=C)F)CCC2)=O)CC2(CCN(C(c3cccc(N)n3)=O)C2)C1 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)NC(C)C(C)NC(C12CCC(CC1)C2)=O C1(NC(C=CCC)=O)CN(C(=O)Cc2ccsc2Br)C2CC12 CC1(C)NC(=O)CC1C(=O)NC(C)(C(=O)NCc1ccc(Cl)nc1)C1CC1 c1(NC(c2c(OC)cccc2)C(=O)OC)nc(C)ncc1C(=O)N(C)OC CCCC(CC)CC(=O)N1CCCC(CNC(c2ncc(C(N)=O)cc2Cl)=O)C1 Cc1cn2nc(N3CC=C(CCNC(=O)C(O)C4CC4)CC3)sc2n1 C1(NC(c2c(OC)ccs2)=O)CN(C(c2cc(O)nc(Cl)c2)=O)C2(CCOC2)C1 CCCC(CC)CCC(=O)NC1CCN(C(=O)CNC(=O)CC(C)(C)C)C1C CN1CC(NC(=O)CC(C)(C)CNC(=O)CC(=O)NC2CC2)CC1(C)C C1(C(=O)NC2C(NC(c3ccc(C(=O)OC)[nH]3)=O)COC2)(CO)CCCC1O c1(C(=O)NCC(CC)(CC)NC(=O)Cc2cncs2)nccc2n[nH]cc12 C(c1cn(C)cn1)=CC(=O)N(C(C)CCNC(=O)CCN1CCCC1)C N1(C(C(C(C)C)F)=O)CCC(C2(NC(=O)C(C3CCC3)C3CCC3)CCC2)CC1 C=C(Cl)CC(C(=O)NC)NC(=O)C(C(C)(C)C)NC(=O)CCC(C)(C)F NS(=O)(=O)c1cc(C(N2CC(C3(NC(=O)Cc4ccco4)CC3)C2)=O)c(Cl)o1 N1(C(C(C)CC(N)=O)=O)CCS(=O)(=O)C(CCNC(=O)CC(C)C(F)(F)F)C1 CC(C(=O)NC1CC2(C1)CC(NC(C1OCCN(C)C1=O)=O)C2)C(C)(C)C c1(C(N(CC(C)(C)NC(Cc2ccc(C)c(Cl)c2)=O)C)=O)cc(Cl)cc(F)c1F Cc1cc(C(N2CCCC(C(=O)NC3(C)CCOCC3)CC2)=O)nnc1C C(CC(=O)N(CC(O)CN(C)C(c1sc(COC)nc1C)=O)C)(C(C)C)OCC C1(NC(C2(c3ccc(OC)cc3)CC2)=O)CN(C(=O)CC2CSC2)CCC1CO N1(C(c2ccc(OC)cc2F)=O)CCC2(CC1)CN(C(=O)CC1CCSCC1)C2 C1(NC(c2cc(CCC)[nH]n2)=O)CC(O)CN(C(C2(CC)COC2)=O)C1 c1(C(c2nnnn2Cc2nnn(C)n2)NCC2C(C)C2)csc(Cl)c1Cl C(C)(CCCCC#N)(c1n(-c2c(CC)cccc2)nnn1)NCCC(C)O CCC(C)C(O)C(=O)NCC1(C)CCN(C(c2ccc(=O)n(CCO)c2)=O)C1 c1(NC(C2N(C(c3cn(CCC)nc3)=O)CCC2C)=O)ccc(O)c(=O)cc1 N(C1CCCc2ncccc21)C(=O)NCCCS(=O)CC(F)(F)F C1(O)(CNC(Cc2scc(C)c2)=O)CCN(C(C2CC(CN(C)C)C2)=O)C1 c1(C(=O)NCCCCC)ccc2c(c1)OC1(CCCCN1C(=O)COC)CC2 C1(C(N2CCC(NC(Cc3c(C)n[nH]c3)=O)C(O)C2)=O)CCc2c(ncn2C)C1 S(=O)(=O)(c1ccc(C)cc1)N(C(c1c(CC)noc1C)=O)CC1CCNC1 C1(NC(CC2C(C)(C)C2)=O)CC2(CCN(C(=O)CCNC(C3CCC3)=O)CC2)C1 N(C1CC(C)(C)Oc2c(Br)cccc21)OC(N1CC(NC(C)(C)C)C2(CC2)C1)=O Cc1nc(Nc2ccc(C(=O)N(C)C)c(Br)c2)cc(C(C)C)n1 c12ccc(cc1)SCCCC(=O)N2.c1(C(=O)OC)nnc(C(C)C)s1 CS(=O)c1ccc(C(=O)N(C2CCN(C(=O)C(F)C(C)(C)O)CC2)CCO)cc1 C(=O)(CCCC(C)(F)F)NCC1N(C(C2CC(C)OC(C)C2)=O)CC(F)C1 N1(C(C(CC=C)CC)=O)CCOCC(C)(CNC(=O)CCc2cc(Cl)cs2)C1 N1(C(c2c(C)nc(CCO)nc2)=O)CC2CCCC1C2CNC(=O)CSC(C)C c1(C(=O)NCC2CCN(C(c3ccco3)=O)CC2)cccc2c1CCO2 CCCC(C)(C)CC(=O)N1CCC2CC2(NC(c2cn3ccnc3s2)=O)CC1 c1(CC(=O)N(C(C)CCNC(C2CC2c2cn[nH]c2)=O)C)ccc(Br)s1 C(CCC(C(=O)NCCOC1CCOC1)NC(=O)CC(=O)N(C)C)OC Cc1cc(C)c(CC(=O)NC2CCN(C(c3cn(C)c(O)n3)=O)CC2)s1 Cc1cncc(C(=O)NCC2(CO)CN(C(c3ccc(OC(F)F)cn3)=O)C2)n1 C(C)(CN=c1[nH]c(C)cc(=NCc2nc(C)ccc2Cl)[nH]1)OC N1(C(C(C)NC(CC)=O)=O)CCC2(CCCCN(C(C3CC3C3CC3)=O)C2)C1 C1(COC)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CC1(C)CC1 N1(C(c2csc(-c3cnc[nH]3)n2)=O)CCN(Cc2ccc(O)c(F)c2)C2CC12 c1(C(N(CCCNC(Cc2scc(C)n2)=O)C(C)C)=O)ccc(O)cn1 C1(CN(C(C(C)OC)=O)C)CC(F)CN1C(=O)C(C)Cc1cnco1 c1(C(=O)NCC2(C)CCN(C(=O)CC3CC3)C2)ncc(P(C)(C)=O)cn1 c1(C(N(C2CCN(C(C3CC3(C)CC)=O)CC2)CC)=O)cc(OC)ncc1F CC(C(=O)NCC1(CNC(=O)CNC(=O)NC2CC2)CC1)C(C)(F)F C1(NC(C2N(C)CC2)=O)CCN(C(N)=O)CC1.C1(n2ccnn2)CCN(C)C1 N1(C(c2ccc(COC)[nH]2)=O)CCOC(CCCNC(=O)CC=CC(C)(C)C)C1 C(C)(C)(CCCC(=O)NCC1CCCC(OC)C1)NC(C(C)=CCC)=O c1(C(N2CC(CNc3nc(C)nc(Cl)c3)C(C)C2)=O)cc2c([nH]1)CCCC2 CC1(C)CCOC1CCC(N1CCC(NC(c2cocn2)=O)C1)=O N1(C(C(C)OCC2CC2)=O)CC2(CC(NC(=O)CC(C)c3cccnc3)CO2)C1 c1(NC(=O)CN(C2CCCC2)C)ccc(F)cc1.C=C1CNCC=CC(=O)NCC1 c1(C(=O)NCC2(F)CCN(C(COC(C)C)=O)CC2)cccc(C#CC2CC2)c1 Cc1cn2c(C(N3CC=CC3CNC(=O)COCC(C)C)=O)cnc2s1 C1(NC(C=CC(CC)C)=O)CN(C(c2ncccc2O)=O)CC2(CC2)C1 N1(C(COC(CNC(CCC#C)=O)(C)C)=O)CC(CC)C(O)C1 C1(C(C)C)CCOCCN1C(C1CC2CCC1CC2)C(=O)NC1COC1 c1(C2(C)CC2)ncc2c(n1)CCN(N1CCN(C(=O)NC3CCCO3)CC1)C2 Cc1cc(F)ccc1NC(C1CC(O)CN1C(c1ccncc1F)=O)=O CCCC(C(=O)NCC1CC1CO)NC(=O)C(Cl)Cl C1(NC(C2CCC(C)N(C(c3cscn3)=O)C2)=O)CCC2(CC1)CC2(F)F S(=O)(=O)(c1cn(C)c(=O)n(C)c1=O)NCc1ccc(CSC)o1 C1(C(=O)NC(C(C)(C)C)CO)C(C2CC2)CCN1C(=O)Cc1ncccc1F C(c1c(Cl)nc2sccn12)=CC(N1CCC(NC(=O)CC2(O)CCOC2)C1)=O C(CC(O)CNC(=O)C(C)OC(C)=O)NC(C=C(COC)C)=O C(=O)(C(C)(C)CC(F)F)N1CC(OCCNC(C(C(C)C)c2cnc(C)s2)=O)C1 C1(CNC(C(C=C)OC)=O)CCN(C(c2ccccc2)=O)C1(C)C c1(CCC(=O)NCC(CCOC)NC(c2nc(C)nn2C)=O)ccccc1C C1(CC)CCCN(C(=O)COC2CCN(C(c3sccc3C)=O)C2)C1 Cc1nn(C)c(C(=O)NCC2(NC(=O)C(C)(C)n3cnnn3)CC2)c1[N+](=O)[O-] C1(C(=O)NC23CC(C)(C2)C3)CC2CN(C(=O)C(O)C(F)(F)F)CC2C1 C1(CC)CCN(C(=O)CC2(OC)CN(C(=O)C(O)C(C)SC)C2)CC1 N1(C(C(CC)COC)=O)CC2(CC2)CC1CNC(=O)Cc1ccccc1C(N)=O N1(C(CS(CC)=O)=O)CC2(C1)C(NC(c1nc(C)c(C)nc1O)=O)CCS2(=O)=O C(C)(C(=O)OC(C)(C)C)(C(=O)N1C(C)CN(C(=O)C=CC(C)C)CC1C)OC C1(NC(c2cc(COCC)c(F)cc2)=O)CC2CN(c3ncc(Br)cn3)CC2C1 Cc1cc(C)c(SCC2(N(C)C(=O)OC(C)(C)C)COC2)c(O)c1 C1(NC(CCC2(CCC#C)N=N2)=O)CC2CCCC(C1)N2C(C1(Cl)CC1(F)F)=O N1(C(CCC(CC)NC(c2nnsc2C)=O)=O)CCC(O)C(F)(F)C1 c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC(O)C2)cc2nccnc2cc1F N(C1CCCCc2ccc(Br)cc21)C(=O)NCc1nc(C)c(C)n1C CC1CN(C(c2coc(C#N)c2)=O)CCN(C(=O)CCCCC2CCCCC2)C1 C#Cc1cccc(C(N2CCN(C)C(CNC(C3CCS(=O)(=O)C3)=O)C2)=O)c1 C(C(C(=O)N(C(C)CSC)C)NC(=O)CC1CC=CCC1)OC C(CC(C(=O)N1CCC(C)(O)C1)NC(C1CC2(CC2)CO1)=O)N(C)C C=CC(F)(F)C(=O)NC1CC(C)N(C(c2cccnc2NC)=O)C1 c1(C(=O)NCC2CC3(CN(C(C4C(C)CCO4)=O)C3)C2)n[nH]c2ccc(Cl)cc12 c1(C(N(CCNC(C2C(C)C3CCC2C3)=O)C)=O)c(F)ccc(N)c1F CC1(C)C2CCC(C2)C1(C)C(N1CC2CC1C2CNC(=O)Cc1ccccc1)=O CN1CC(C(N2CCCC(CNC(=O)Cc3ccc(C4CC4)cc3)C2)=O)NC1=O C1(NC(c2nc(CNC(C(C)=NOCC#N)=O)oc2)=O)CNC(=O)CC1C c1(CNC(C(C=CC)O)=O)ccc2c(c1)CN(C(c1ccc(F)c(F)c1C)=O)C2 CCCC(C)(O)CC(=O)NC(CC(=O)N1CC2C(C1)C2(F)F)C(C)OC C(=O)(C(COC)CC(C)C)N1CCCC(CCNC(C2(C=C)CCC2)=O)CC1 N1(C(c2cccc(C)c2F)C(=O)N(C(CC)(C)C)CC)CC2CCC(C1)C2(F)F c1(C(=O)NCC(CC)NC(=O)C=Cc2ncc[nH]2)cc(C2CCCC2)[nH]n1 C(=O)(C(C)C1=CCCC1)N1CCN(C(c2ncn(C(C)C)c2)=O)CC1CF N1(C(Cc2cc(C)on2)=O)CCC2(NC(=O)OC(C)(C)C)CCCCC12 N1(CC(N)=O)CCCC(C(=O)N(c2ccccc2)CCC(=O)C(N)=O)C1.O CCC(CC)CC(C(=O)NCC(=O)Nc1ccco1)N1CCC1C1CCC1 N1(C(C(N2CCCC(O)C2)C)=O)CCCC1(C)CNC(c1ccoc1Cl)=O C1(C(=O)NCc2n(CC)ccn2)CCC2CCC1N2C(=O)Cn1[nH]cnc1=N c1(-c2nc(C(C)O)nn2CCN2CCOCC2)ccnc(Cl)c1Cl C1(C(=O)NC)C=CCN1C(c1conc1CNC(C1CC1OC(C)(C)C)=O)=O N1(C(CC(=C=C)C)=O)CCN(C(c2scnc2Cl)=O)CC1CC(F)F c1(CN(C)CC2CNC(C)(C)C2)cccc(OCC(F)(F)F)n1 C1(C(=O)NCCC2CCSC2)CCCN(C(C2(Cl)CC2(F)F)=O)CC1 c1(C(=O)NCCN(C(c2c(C)[nH][nH]c2=N)=O)C)cc2cccc(F)c2o1 CC1(C)OCc2cc(NC(=O)Nc3cnn(-c4ccccc4F)c3N)ccc21 c1(C2(C(=O)NC3(CNC(c4c(C)nc[nH]4)=O)CCOC3)CCC2)ccccc1Cl c1(C(N2C(CC)C(NC(=O)CC3CCCCC3)CC2)=O)ccc2c[nH]nc2c1 O=C(C1CCc2c(Cl)cccc21)N1CC2(C1)CN(C(C1CCCC3(CC3)C1)=O)C2 C(=O)(C(C)(COC)CC)NCCCN(C(c1c(CC)occ1)=O)C C(=O)(CC(C)CC(=O)N1CC2(C1)CN(C(C1(COC)CC=CC1)=O)C2)OC N1(C(=O)NCC2(O)CC(C)(C)OC2)C2CCC1CC(CO)C2 c1(CC(=O)NCC#CCNC(c2cc(C(C)(C)C)n[nH]2)=O)cnn2c1CCCC2 C12(C(=O)NCC3N(C(c4n(CC)nnc4)=O)CCOC3)CC1COC21CCC1 c1(C(=O)NC2CCN(C3CCC(C)CC3)CC2)ccnc2ncccc12 C1(CC)C(NC(c2cc(-c3cccc(F)c3)no2)=O)CCN1C(=O)CC(O)CC Cc1ncccc1-c1cn(CC2CCCC2NC(C2CS(=O)C2)=O)nn1 c1(CC(=O)N(C2CCCN(C(=O)Cc3cccs3)C2)CC)cc(F)c(F)cc1F C1(CNC(C=C(C)C(C)C)=O)OCC2CCC1C2.C12C(C1(C)C)NC2=O CCC(C(=O)NCC1CC(F)(CNC(=O)Cn2nnc(=O)[nH]2)C1)C(F)(F)F c1(C(=O)NC2CCC(CN(C)C(C3CC34CC4(F)F)=O)CC2)c[nH]nc1[N+](=O)[O-] c1(OC)cccc(C(C(=O)NCc2ccc(F)cc2)N(C2(C)CC(C)(C)C2)C)c1 c1(CC(=O)NC(C)CN(C)C(C2(C#N)CCC2)=O)nn(C)c2ccccc12 C12(C(=O)NC3C(NC(c4nc(COC)sc4)=O)CCCC3)CC3CC(CC1C3)C2 c1(C(N2C(C)C(C(=O)NC3COC3)CC2)C(=O)N(C)C)cc(Cl)c(Cl)c(Cl)c1 C1(NC(c2n(C)ncc2)=O)CCN(C(=O)CC2CCCC(=O)N2)C1(C)C C12CC(N(C(c3cccc(C4CC4)c3)=O)C1)N2.Cn1cc(OC(=O)C2CC2)cn1 C=CCC(C(=O)NC(CCC)C(O)C(=O)NCCN1CCCC(O)C1)C(C)C c1(CC(=O)NCC=CCNC(C2(C)CC=CCC2)=O)cc(F)ccc1Cl c1(CCC(=O)NCC(CNC(CCC(=C)Br)=O)F)ccc(O)c(Cl)c1 C1(CNC(CCC2(NC(C=C(C)C(C)C)=O)CCCC2)=O)CC2(CC2)C(=O)O1 C12(CC(=O)NCC(N(C(=O)C=Cc3cscn3)C)C3CC3)CCC(CC1)C2 c1(C(=O)NCC(C)N(C)C(c2cn(C)nc2Cl)=O)cccc2c1CNC2=O N1(C(c2c(C)con2)=O)CCC2(CCCC2NC(C2(F)CCCCC2)=O)C1 O=S(=O)(c1ccnn1C1CC1(F)F)Nc1cnn(-c2ccccc2)n1 CC(O)C(C)C(=O)NCCC1CCN(C(=O)CSC(F)F)C1 C(=O)(C1=Cc2ccccc2C1C)NC(CC)(CNC(=O)C(F)(F)C(C)O)CC C1(c2n(CCCCCCC)nnn2)(NCC(C)(C)C2CCC2)CC2CCC1CC2 c1(C(=O)NC(CN(C(=O)C=NOC)CC)C)ccc(-c2ccc(Cl)cc2)cc1 C1(SCC(=O)NCC)CC(O)CN1C(c1ccccc1)=O.N12CCC(C1)NC2=O C(N=c1[nH]c(=NCCCc2ncc[nH]2)[nH]c2c1CSC2)c1nc(C(F)F)sc1 N1(C(c2c(C)nco2)=O)CC(NC(C2(C)CC(C)(C)C2)=O)CC12CCOCC2 C1(NC(c2cc(C)sc2)=O)CC2(CCN(C(C3CC(=O)CO3)=O)C2)C1 c1(C(=O)O)cnc(Cl)c(F)c1.c12ccccc1C1(CC1)CN2.c1(OC)nccc(C)n1 CCC(C)CC(=O)C(=O)N1CC2CC(C1)N(C(=O)C=CCF)C2 CCCCCCCCCC(C)CC(=O)N1CC2CCC(C1)N2C(C1SCCS1)=O C1(=CCNC(C(COC)O)=O)CCN(C(=O)C(C2CCCCC2)=O)CC1 C(C1c2ccsc2CCN1C(C1CCCCC1)=O)NC(CC1(C)CCC1)=O C1(C(=O)NC2(C)CN(C(c3cnc(OC)s3)=O)C2)CC2CCCCN2C1 N1(C(=O)OC(C)(C)C)CC2CCC2(C(=O)NC(c2nn[nH]n2)C2CC2)C1 C1(CCC(C)=CC(=O)NCC(C)(C)C)CCOCC1.C1(C(=O)N)CC1C(C)C Cc1ccc2c(c1)CCC(C(=O)NCC1CCCN1C(c1cnnc(O)c1)=O)O2 N1(C(C2N(C(c3ccc(C)cc3)=O)CC(F)C2)=O)CCC(C)(C#N)C1 c1(C(N2CCCC(NC(c3c(C)nn[nH]3)=O)CC2)=O)cc(F)cc([N+](=O)[O-])c1Br Cc1c(C(=O)N(C)CC2CCCN(C(=O)C(C)c3ncco3)C2)ccc(F)c1F C1(N(C(c2c(C)sc(Cl)n2)=O)C)CCCN(CC2CC(C)(C)C2)CC1 C1(NC(c2cc(CC)n(CCO)n2)=O)CCCN(C(c2coc(C#N)c2)=O)CC1 c1(CC(=O)NCC(CC)NC(c2cnc(C3CCCO3)s2)=O)cc(C)cs1 CC1CCN(C(=O)C=CCN(C)C)CCN1C(C1CCCCC1)=O Cc1nn(C)c(C)c1C(=O)NCC1(C)CCCN(Cc2ccccc2C(C)C)C1 N1(C(=O)C(Cl)=CCl)CC2(C1)CN(C(c1ccc([N+](=O)[O-])s1)=O)C2 CC1CN(C(=O)CCCN2CCOCC2)CC1CNC(c1cccs1)=O N1(C(c2cccc(CCC)c2)=O)CCC(C)C(NC(=O)CN(C)C(C)=O)C1 N1(C(C2CC=CCN2C(c2cc(CO)[nH]n2)=O)=O)CCC(CO)C(O)C1 C(=O)(CC(Cc1ccccc1)CC(C)C)OCc1onc(-c2ccc(CC)nc2)n1 Cc1ccc(F)c(CNC(C2CCN(C(=O)CC3CCC(=O)N3C)CC2O)=O)c1 C(=O)(C1=CC2C=CC1C2)NCCCN(C(C1CC(SC)C1)=O)C1CC1 Cn1ncc(C(=O)NCCC2CCCN2C(C2CCCCO2)=O)c1C(F)F C12(N3CC(CCNC(COC(CC)(C)C)=O)C3)CC3CC(C1)CC(C)(C3)C2 c1(N2CCC(OCCOC)C2)nc(C)cc(=NC(C)CN2CCOCC2)[nH]1 N1(c2nnn(C)n2)CCn2ncc(CNC(C3CC(C)(C)C3C(F)(F)F)=O)c2C1 C1(CC(=O)Nc2c(C)nc(Cl)nc2)CC2(CCN(C(c3cn[nH]c3)=O)CC2)C1 N1(C(C(=O)N(C(C)C)C)C)CC2CCC1CN2C(c1c(Cl)nn(C)c1Cl)=O CC(C)CC(C)C(=O)N(C1CCN(C(c2coc(C3CCCC3)n2)=O)C1)C c1(CC)[nH]nc(Cl)c1C(=O)NC(C1CCN(C(c2csnc2C)=O)C1)C c1(C(N2CCC2Cc2c(-c3cn(CCC)nn3)n(C)nc2)=O)c(C)cccc1Cl c1(N2CCC(OC)CC2)nc(=NCCC(CSC)(CC)CC)[nH]c2ccccc12 c1(C(N(c2nc(Br)c(Br)cc2O)C)=O)ccc2c(c1)CN(C(=O)OC(C)(C)C)C2 c1(C(C(=O)NC(CC)CNC(=O)C=CC(=O)N(C)C)F)c(F)cccc1F C1(NC(c2c(CNC(=O)CN3CCOC3=O)ocn2)=O)CC2(CCC2)C1O C1(CC(=O)NCC(C)(C)C(N)=O)CCCN(C(=O)CCc2cn[nH]c2)CC1 c1(C(=O)NCCC2CN(C(C(C3CCCO3)OC)=O)C2)cc(C)nc(Cl)c1N c1(C(=O)NCCNC(=O)Cc2ccc(F)cc2C(F)(F)F)cnc2n1CCCC2 CC(C)C(CO)C(=O)NCC1CCC(NC(=O)CC2CCC(C)(C)CC2)C1 N1(CC(c2ccc(NC3CCC3)cc2)=O)CCCC(S(=O)(=O)OC(F)F)CC1 Cc1ncc(C(=O)NCC2CCCC2NC(=O)Cn2cccnc2=O)n1C N1(C(c2c(C)coc2)=O)CCCC(N(C(=O)Cc2nc(=N)[nH][nH]2)CCO)C1 CC(C(=O)NC1CC(NC(C2C(C)(C)C2(F)F)=O)C1)S(=O)(=O)c1ccc(F)cc1 c1(SCC2CC(C(=O)NCC(=O)NC(c3ccccc3)C)C2)ccccc1 N1(C(C2CCC(=C)CC2)=O)CCC2C(CCCN2C(C2CCC(O)CN2C)=O)C1 Cc1ccc(CCNC(C2CCC(C)N2c2ncncc2F)=O)cn1 CC1(C)CCCCC1CN1CCC(=CC(=O)NC(c2ccccc2)C#N)CC1 c1(C(=O)NC2C(OC)CN(C(C(CC)F)=O)C2)cc2n(n1)CCNC2=O O=C1NC2(CO1)CC(C(=O)NCC1CCN1C(=O)C1=COCCC1)C2 C1(C2CCCCN2C(C2CC(F)C2)=O)(CNC(C23CC(F)(C2)C3)=O)CCOCC1 C1(C)(C(=O)NCC2C(NC(CCOCC(C)C)=O)C2)CC2(C1)CC(F)(F)C2 C1(OC)CN(C)C(C)(C(=O)NCC2(NC(C3CC(C)(C)C3)=O)CC2)C1 C1(C)(C(=O)NC2CC(CCNC(c3c(C)cn(C)n3)=O)C2)CCOC12CC2(F)F Cc1onc(C(N2CC(NC(=O)CCc3ccccn3)C3CC23)=O)c1Br N1(C(C2(COC)CC=CC2)=O)CC2(C1)CN(C(=O)CCc1ccsc1)CCO2 C1(=O)CC(C(F)(F)F)O1.C(=O)(C(CC)CCC)N1CCC1.O(CP(C)(C)=O)C(CC)CC C1(CNC(C(CC)C2CCOCC2)=O)CN(C(=O)CNC(=O)C2CC2)CCO1 c1(C(N2CCNC(=O)C2C)C(=O)NCC)cc2cc(Br)ccc2o1 N1(C(COCCCC)=O)CCC(NC(=O)CC2CC2C2CC2)C1C1CC1 C1(NC(C(C)C(C)C)c2n(CCOC)nnn2)(CC2CC2)CCCCC1 C(CC(C)(C)C(=O)N1CCC(C(=O)NC(CO)C2CC2)C1)SC CCCC(C)(C)C(=O)N1CCN(C(=O)CCc2nncs2)C(c2ccccn2)C1 C1(C(=O)NCC(CC)C#N)CC(NC(c2nc(C)oc2C)=O)C1(C)C C1(NC(c2cn(CCN(C)C)nn2)=O)C2CCCN(C(C3(C4CC4)CC3)=O)C12 N1(C(CCN(C(=O)CCc2nc[nH]n2)C(=O)OC)=O)CC2CC(CC)CC2C1 N1(C(c2ccn(C(C)C)n2)C(=O)NCC2CCCO2)CC(C)CC1C c1(CNC(N(C(C)CC(N)=O)C)=O)ccccc1OC1CCC1 C(C(C)(CC)C(=O)Nc1cnc(C)nc1)NC(C(F)=C(C)C)=O N1(C(=O)CN2CCCC2)CCOC2(C1)CN(Cc1cc(O)ccc1Br)C2 C1(CNC(c2cnc(N(C)C)s2)=O)CCCCC1NC(=O)CSc1ccccc1 c1(C(=O)NC(C(=O)NCC(CC)SC)C2CCCO2)ncncc1OC N1(C(C(COCC)C)=O)CCC(NC(=O)CCC2CCC2)CC(O)C1 c1(CC)ccc(C(C)C(=O)N(C)CCNC(=O)Cn2ccnn2)cc1 CC(C)C(C(=O)N1CCC(C(=O)N(C2(CO)CC2)C)C1C)C1CCC1 c1(C(=O)NCCCC2N(C(c3cc(C)no3)=O)CCC2)c[nH]c2cccnc12 c1(OCCC(=O)NC(C)C(C)NC(=O)C=Cc2cn[nH]c2)cc(Cl)cc(Cl)c1 c1(CNC(C2CC(O)CN2Cc2c(Br)cccc2Br)=O)ccc2ccccc2n1 C1(Cn2cc(COC(COC3CCCN(C)C3)=O)nn2)CC2(C1)OCCO2 c1(OCC(=O)NCC2CCCN(C(c3c(C)coc3C)=O)C2)ccc(F)c(F)c1 C1(C(N(CCOC)CCNC(C2(S(C)(=O)=O)CC2)=O)=O)CCn2cc(C)nc2C1 C(C(C(=O)NC(C)CC(C)C)NC(=O)C(c1cnn(C)c1)=O)OC C1(COC)(CNC(C2CCOC(C)(C)C2)=O)CCN(C(=O)Cc2ccco2)CC1 c1(C(N2CCN(C(CC3CC(C(=O)OC)C3)=O)C3C2C3)=O)cccc2nccn12 c1(-c2ccc(OC)cc2OC)nc2c(s1)CN(C(=O)COc1ccccc1)CC2 c1(OC)c(C(=O)NC(CNC(=O)CSc2ccccc2)CO)cccc1Cl C(=O)(C1CCOc2ccc(Cl)cc21)N1CCC(CNC(Cc2n(C)ncc2)=O)C1 Cc1cc(C(=O)N(C)CC2CCCC(NC(C3CC(OC4CC4)C3)=O)C2)sc1Cl N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC(O)(C(C)CNC(C2CNC(=O)N2)=O)C1 C=CC(F)(F)C(=O)N1CCOC(CCNC(c2cn(C(F)F)cn2)=O)C1 N1(C(CN(C2CC2)CC)=O)CCCN(C(c2cncc(O)c2Cl)=O)C(C)C1 Cc1conc1CC(=O)NCC1CC(CNC(=O)C(C)n2ccnn2)CO1 C1(NC(c2cc(OC)nn2C)=O)CC2CN(C(c3cc(CSC)on3)=O)CC2C1 CC1(C)C(CNC(=O)CCC2CC(NC(=O)CN3CCC(F)CC3)C2)C1(F)F C1(O)(C(=O)NC2CC(C)(NC(CN3CCC(C)C3)=O)C2)CCCCC1 C1(CS(=O)(=O)NC(c2c(C)c(Br)ccc2)=O)CCCC2(CCC2)O1 C1(NC(c2c(C)[nH]cc2)=O)CCCCCC1NC(c1cc(O)cc(Br)c1)=O C1(C)(NC(CCC(C)SC)=O)CCCCC1C(=O)N.N12CCC1C2=O.C(C)C C1(CN(C(CCN(C)CC)=O)C)CN(C(c2cnnc(C)c2)=O)CCO1 C1(CC)CC(C(N2CCC(OCCNC(C3(C(F)(F)F)CC3)=O)CC2)=O)CCO1 CCC(C)(C)CC(=O)NN1CCCC1C(=O)NCC(C)(C)CO Cc1cc(CC(=O)NCC(C)SCC(=O)NCCN(C)C)cs1 N1(C(=O)CC(F)(F)F)CCC2C(C1)CN2C(c1cnn(CC(F)(F)F)n1)=O C(=O)(C1CCc2ccc(OC)cc21)N(C)CC1N(C(CSCC)=O)CCC1 c1(OC)cc(C(N2CCC(N(C(=O)Cc3cnsc3)C)C2)=O)ccc1C#N C1(NC(C=Cc2n(CC)ncc2)=O)CN(C(=O)CCOC2COC2)CC12CC2 O=C(C1Cc2ccc(Cl)cc21)NCC12CC1CN(C(=O)CCC(F)F)C2 c1(OC)cccc2ccc(C(=O)NCC3(F)CC(NC(C)=O)C3)nc12 C1(C)CCCCN1N1CC(NC(=O)CCc2nc[nH]n2)C1.N1(C=O)CCCCCC1 N1(C(C(C)C(C)(F)F)=O)CC2CCCC(NC(c3cnc(Cl)[nH]3)=O)C2C1 C#CCC(C(=O)N1CCCCC1CF)NC(c1oc(C)nc1CC)=O C1(COCC(C)O)CCCN1C(=O)CCCC1CC1 C1(CC)CN(C(=O)C=CC2CCCN2C(=O)C(=O)C(C)(C)C)C(C)CO1 c1(SC)nc(C)c(CCC(N2CCC(C(=O)N(c3ccccc3)C)C2)=O)c(O)n1 c1(OCC(C)C)cccc(C(=O)N(CC(C)N(C(=O)C=C(Cl)Cl)C)C)c1 C(C(C)C)(C(O)C(=O)NC1(CCNC(C2CC2(C)C(F)F)=O)CCC1)OC C12(NC(=O)CSc3nncs3)CCC(CC1)N(C(C1CC(O)C1)=O)C2 C1(NC(C2CC(OCC)C2)=O)CN(C(c2ccc(O)nc2)=O)CC2(CCC2)C1 C1(C(=O)NCc2c(C)ccc(C)n2)CC2(CCCC2)CO1 CCC(C)CCCCC(=O)N(CCCCCC(=O)NC1(C)CC(F)C1)C N1(Cc2cn(-c3ccc(C)nc3)nn2)CCCN(C(=O)C(F)OC(F)(F)F)CC1 C#CCC(C(=O)NCCCC(C)CO)NC(=O)C=COC c1(CC)ccoc1C(=O)NC(C1CCN(C(C2(OC(C)C)CCOC2)=O)C1)(C)C C(=O)(CCCC(C)(C)C)NC1C(C)CN(C(c2sc(Cl)cc2Br)=O)C1 N1(C(c2cncc(N)n2)=O)CCN(C(C2CC(F)(CO)C2)=O)C2CCC12 C1(C(N2CCC(O)C2)=O)(C)CCCO1.CC(C)(C)OCC(=O)O CC1C(NC(c2cccc(F)n2)=O)CCN1C(=O)C(c1ccccc1Cl)(F)F CCC(C)(CC)C(=O)NCC1(CNC(c2ccc(C)cc2SC)=O)CCCCC1 CC1CC(CNC(c2cnc(N)c(Cl)c2)=O)CCN1C(=O)Cc1cnoc1 C1(COC)(NC(=O)C(O)CC2CC2)CCCN(C(=O)C#CC(C)(C)C)C1 C1(N(C(CN(C(=O)C(C)N2CCCC2)CC(C)C)=O)C)CCOCC1C Cc1cc(NC(C2CCN(C(=O)C(C)CC(F)F)CC2O)=O)cc(F)c1 c1(C(=O)NC2(CC(=O)NCCn3c(CC)nnc3)CCC2)ccc(C#N)[nH]1 C(=O)(N1CC2COCC2O1)C1(NC(=O)CN2CC(=O)NC2=O)C(C)C1 c1(-n2cc(C(C)NC(C)(C)COC(F)(F)F)nn2)c(C(F)(F)F)cccc1C c1(C(=O)NCCCCNC(c2cn(CCC=C)nn2)=O)[nH]c2c(c1C)CCCC2 N1(C(C(CC)NC(C)=O)=O)CC2CCC(NC(c3ccc(C)nc3SC)=O)C2C1 C1(C(C(=O)NCC(C2CCCC2)NC(C2(SCC)CC2)=O)C)CCOCC1 N#Cc1ccc(C2(C(=O)NC3CC3NC(C3(C4CC4)CC3)=O)CCC2)cc1 C(C)(CNC(=O)CCc1cnc[nH]1)(C(C)C)NC(c1c(CC)c[nH]n1)=O N1(C(c2ccnc(OC)n2)=O)CCC(O)(C(C)NC(=O)C(C)c2ccco2)CC1 C1(CCC)(NC(c2cc(COC)cs2)=O)CN(C(c2conc2CC)=O)C1 N(C1CCCn2ncnc21)C(C(CC#C)NC(c1c[nH]c(C#N)c1)=O)=O c1(CCN2CCC(NC(Cc3ccn(C(C)C)n3)=O)C2)cccc(F)c1 c1(OC)cccc(F)c1C(=O)NCC1CCN(C(c2cc(O)ccc2C)=O)CC1 O=C1NCC2(CN(C(=O)NC3(c4ccc(F)cc4F)CC3)C2)O1 CCC(C)C(C(=O)NCC1CC(O)CN1C(c1cscc1C)=O)NC(C)=O c1(NC(c2c(NC(C3C(C(=O)OC)C3)=O)cc(C)cc2)=O)c(C)ccnc1C#N c1(C(=O)NCC(c2ccccc2)NC(C(C)(CO)OC)=O)ccc([N+](=O)[O-])[nH]1 c1(C(N(CCCNC(CSCC)=O)C)=O)nc(N(C)C)nc(=N)[nH]1 c1(N2CCN(C)C(C3CC3)C2)ccc(S(=O)(=O)N2CCc3ccccc3C2)cn1 C(=O)(C(CC)C(=O)N1CCCC1NC(c1cc(C2(C)CC2)on1)=O)OCC c1(C(=O)NCCCN(C(C=NOC)=O)C2CC2)cn(C(C)(C)C)nc1C CC1COCCN1C(C1CCOC(C)C1)C(=O)Nc1ccccc1 C(=O)(C(Cc1cscn1)NC(C1CC(CCC(=O)O)CO1)=O)OCC CCCCCC(=O)NCC(=O)NCC=CCNC(=O)CC1CCCC1(F)F N1(C(C(C)OCC)=O)CCC(C(N2CC(C#N)C2)=O)C1CC N1(C(c2ccc(CC)cc2)=O)CCC2CN(C(C3C4CC5C(C4=O)C35)=O)C2C1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)C(C)SCCN(C)C)C(CCO)C1 N1(C(c2c(C)c(Br)cnc2)=O)CC2(C1)CN(C(=O)C#CC1CC1)CC2CO CC(C)CC(O)C(=O)NCC(CO)NC(c1ccn(C)n1)=O C1(CC(=O)NCC2C=CC(NC(CC=C)=O)C2)CCCC(F)(F)C1 c1(C(=O)NCCCN(C(c2c(C)nc(C3CC3)o2)=O)C)coc2ccc(Cl)cc12 N1(C(COCC)=O)CC(CNC(=O)Cc2conc2C)C(c2cncn2C)C1 C1(NC(CS(N)(=O)=O)=O)COCCN(C(=O)C(F)(F)c2ccncc2)C1 c1(C(=O)NCC2C=CC(NC(c3c(C)nco3)=O)C2)ccc(F)c2[nH]ccc12 C1(C(=O)NC2CCN(C(C3(N(C)C)CCCC3)=O)C2)CCOCC12CCCCC2 c1(OC)cc(Cl)cc(CN2CCC(O)CC2C(N2CC(F)C(F)C2)=O)c1O CCN=C(NCCOc1ccc(Cl)cn1)NCc1csc(C)n1 CCC(CC(=O)NCC(C)N(C(=O)CCc1cscn1)C)C1CCC1 N1(CC)CC(C(=O)NCC2C(C)CCN2C(c2n[nH]c(C)n2)=O)CC1=O c1(CSC)ccc(OCC(F)(F)F)cc1.C1(C)(C)C(=O)N2CCC(C2)C(=O)N1 C1(OCC)(CO)CCN(C(=O)C(CC)n2ccnc2)CC1.C(=O)C(C)n1ccnc1 Cc1ccc(Br)c(C(=O)NCC2COCCN2C(C2CC2(C)C)=O)c1F c1(NC(C(CC)NC(=O)CC2CSC2)=O)ccc(F)cc1F c1(N(C)C)cccnc1C(=O)NC1CC1CNC(c1cnc(CC(C)(C)C)o1)=O c1(C(N(CC(CNC(c2c(COC)cco2)=O)C)C)=O)c(O)cccc1Cl C1(C(C)C)COCCN(C(=O)C(O)Cc2cn(-c3ccc(Cl)cc3C(N)=O)nn2)C1 N12CCC3CC(C3C1)C2=O.c1(C(=O)NC)ccc(CN(c2nncn2C)C)cc1 c1(SCC(N2CC(C)C(NC(=O)COC3CC3)C2)=O)nc2ccccc2s1 c1(CC)ccc(O)c(C(=O)NC2CC3CC(NC(=O)Cc4ccoc4C)CC23)c1 C1(NC(c2cc(C)ncn2)=O)CC2CN(C(c3cscn3)=O)CC12 C(CC(=O)N1CCC(C#N)(CC)CC1)(CC(C)C)NC(C(C)NC(CC)=O)=O C1(O)(CNC(CCC(N)=O)=O)CCN(C(c2ccsc2)=O)CC1 C1(CC(=O)NC(CCNC(CC(=C=C)C)=O)C(C)C)Oc2ccccc2NC1=O Cc1ncc(C(N2CCOC(C3CN(C(c4cnc(S)nc4)=O)C3)C2)=O)c(=N)[nH]1 [N-]=[N+]=NCCCCC(=O)NC(CC1CCC1)C(=O)N1CC(NC(N)=O)C1 c1(CC(=O)NC2CCN(C(CSCC=C)=O)C2C(C)C)c(C)nn(C)c1C C1(CNC(C2CC2c2cccc(Br)c2)=O)CCCN(CCCC2CCOC2)C1 c1(OCC(=O)NCCC2CN(C(C3C(C)(COC)C3)=O)C2)c(C)occc1=O c1(Cc2nc(C(C)NCC3C(COC)C3)sc2)ccc(C)cc1 C(CCC(=O)NC(C)C(C)NC(c1cnc(C2CC2)s1)=O)NC(=O)OCC C1(O)(CCNC(C2(C)CNC(=O)C2)=O)CCN(C(C2CCCCC2)=O)CC1 c1(CC2CN(C(CCCN(C(C)=O)C)=O)C2)ccc(N)cc1 C1(C(N(CCCF)CC)=O)CC(NC(=O)CCc2ncccn2)C(O)C1 N1(C(C(C(C)(C)C)OC(C)(C)C)=O)CC(C2CN(C(=O)C(Cl)=CCl)C2)C1 Oc1ncnc2scc(-c3nc(C(n4cccn4)C4CC4)nn3-c3ccc(Cl)cc3)c12 N1(c2ncc(C)cc2[N+](=O)[O-])CCC(C2CCN(C(=O)C(C)N3CCC3)CC2)C1 C(=O)(CC(C)CC(F)(F)F)N1C2CC(NC(C3(COC)CCCC3)=O)CC1CC2 c1(C(=O)NC(C)C(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)cccc2ncn(C)c12 c1(NC(=O)CCNC(=O)Cc2cn[nH]c2)c[nH]nc1Cl CCC(C)(C)C(O)C(=O)N1CC2(C1)CN(C(c1nnn(C)c1C)=O)C2 C(C)(C)(CC(F)C(=O)NCC(C)(C)CO)NC(C(CN(C)C)O)=O C#CC1(O)CCN(C(=O)C(C)(C)NC(=O)C(F)C(CC)CC)C1 C(=O)(C1=CCN(C(=O)CC2CC3CC3C2)CC1)NCC1(O)CCC(C)C1 C1(NC(CC2ON=C(CC)C2)=O)CCN(C(c2c[nH]cc2COC)=O)CC1F C(=O)(CC1=CCOCC1)NCCCC(C(=O)N(C1CC=CC1)C)O c1(C(N2C(CN(C(=O)C(CO)C(C)(C)C)C)COCC2)=O)c(F)ccc(N)c1F c1(COC(C2(CNC(C)=O)CCOCC2)=O)ncc(C)cc1Br C1(C(N(C(C(C)SC)C)C)=O)C(C2CC2)CCN1C(C1Cc2ccccc2C1)=O c1(C(N2CC(CCNC(C(C(=C)Cl)(C)C)=O)C2)=O)ccc2c(c1)CC(=O)NC2 C1(C(N(C(CCNC(Cc2cccc(C)c2)=O)C)C)=O)CC1C1CCCC1 N1(C(C(F)OC)=O)CCCC2(CCCCC2NC(=O)Cc2nc(C3CC3)cs2)C1 C1(CCC(=O)NC2CC(CNC(CN(C3CCC3)C)=O)C2)CCC(=O)N1 c1(NCCC(CCC)C)cc(=NCc2cnc(C3CC3)nc2)[nH]cn1 Cc1nc(N(C)C(c2ccc(Cn3cc(CC4(O)COC4)nn3)o2)=O)ccc1F CCCCC(O)CC(=O)N1CCC(C)(C(=O)NCCN(CCO)CCO)CC1 N1(C(CCC)=O)CCC2C(C1)NC(=O)CN2C(C1CCCN1Cc1cccs1)=O c1(C=O)cnncc1C.c1(COC)ccoc1C(N1CC(C2NCCC2)(O)C1)=O c1(CC(CNC(=O)NC2CC(C(C)(C)C)C2)N(C)C)nn[nH]n1 c1(N(C(C(=O)NCC2CCCCC2)C2CC2(C)Br)CCCC)ccc(F)c(C)c1 c1(C(=O)NCC2C(NC(c3c(C)scc3)=O)CCC2)sccc1C#N C#CC1CCCN(C(=O)C(C2CC=CCC2)NC(C2CCC2C#N)=O)CC1 c1(OCCCOCC)cnc(C(=O)NCCNC(C2CCCC(O)C2)=O)c(Cl)c1 C1(CC)CN(C(=O)CCN(C(=O)Cc2cn(C)cn2)C)CCN1C C(=O)(CC(O)CC(C)(C)C)N(C(CC(N1C2CN(CC)C(C2)C1)=O)(C)C)C C1(CNC(CCCNC(=O)NCC#C)=O)CN(C(=O)CCCN=[N+]=[N-])CCC1C c1(OC(CCC=C)C)ccc(CNCC(C2CCC(C)CC2)(C)O)c(OC)c1 CC1CC(NC(c2cc(C#N)cs2)=O)CCN1C(=O)C=Cc1ccc(Cl)s1 CC1(CO)CCC(N=c2[nH]c(=NCc3cncs3)[nH]c3c2SCC3)CC1 c1(C(=O)NCC2N(C(Cc3c(C)noc3)=O)CCCC2)ccc(C#N)nc1O C(=O)(C(CC=C)NC(c1cocc1C)=O)NCCCC=C c1(C(=O)NCC(CC(C)C)NC(=O)C(F)F)cc(C(F)(F)F)cc(O)n1 C1(NC(CC2CC(=O)C2)=O)CCN(C(c2csc(Cl)n2)=O)CC12CCC2 C(CNC(=O)Cc1csnn1)(CC(F)(F)F)NC(C(N1CC(C)C1)C)=O C1(C(=O)NCC2(C(=O)NC(CC)C3CCC3)CCCC2)CCN(C)CC1 N1(C(C2(C(N(C)C)=O)CC2)=O)CCN(C(c2cc(S(N)(=O)=O)cs2)=O)CC(O)C1 C(C(=O)NC1(CCNC(C2(N(C)C)CC2)=O)CCOC1)(C(F)(F)F)OC(C)=O C12(C(=O)NC3CC(NC(=O)C=CBr)C3)CC(c3ccccc3)(C1)C2(F)F c1(CC2(CC(=O)N(CC(C)(C)NC(COCC(=C)C)=O)C)CC2)ccccc1 N1(C(CC(C)F)=O)CCC2CN(C(c3csc(-c4cnc[nH]4)n3)=O)CC12 C1(NC(C2(COC)CC(F)(F)C2)=O)CN(C(c2cn(C)cc2C)=O)C2(CCC2)C1 N1(C(=O)CC2CCCN(C(c3ccc(O)cc3)=O)CC2)CCC2(CCCC2)C1 Cc1cc(CC(N2CCC(C(C)NC(C3CC(O)C3)=O)C2)=O)ccc1Cl C(=O)(C#CC1CCCCC1)NCC(CCOC)NC(c1cn(CC)nc1C1CC1)=O CC1CCOC(C(=O)NCc2csc(C(=O)NCCC3CCC(C)(C)O3)c2)C1 c1(C(N2CCC3(NC(c4nn(C)c(O)c4)=O)C(C2)C3)=O)ccc(Cl)c(N)c1Cl CCCC(O)C(CO)NC(=O)CNC(=O)CCn1cnnn1 c1(C(=O)NC2(CO)CCN(C(C3(C)CCCC3)=O)C2)ccc(NC(N)=O)cc1 c1(C(C(=O)NC(CC)C)N(CCC(N)=O)C2CC2)cc(C)c(C)c([N+](=O)[O-])c1C C(=O)(C1=CCCC1(C)C)N1CCN(C(c2nn(C)c(F)c2)=O)CC1CCO C(CCCC(=O)NC(CNC(=O)CNC(c1ccccc1C)=O)CC(C)C)OC CCN=c1ccc(C(N2CC(NC(c3nocc3C(C)C)=O)CC2(C)C)=O)c[nH]1 C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NCCN(C)C(C1CN(C)CC1C)=O CN1CCC2CC(NC(=O)CCc3cnc(C4CC4)o3)CCC12 Cc1cc(C(N2CC(O)(CCNC(=O)Cc3cnnn3C)C2)=O)c(C)cn1 c1(C(N2CC(OC)(CNC(C3CCSC(C)C3)=O)C2)=O)cc2ccccn2n1 C(=O)(C1CCc2nccn21)N1CC2(CC(NC(C(C)Cn3cccn3)=O)C2)C1 C1(C2CCN(C(=O)CC3CCC(=O)NC3=O)C2)(NC(c2c(C)coc2)=O)CC1 C12(C(N3CCC(NC(C(C)(C)OC(C)C)=O)C(F)C3)=O)CCOC1CCOC2 C1(N(C2(C(N(C)C)=O)CC2)C(C2CC=CCC2)=O)CCN(C(=O)C=CCF)O1 N1(C(CCCCCC)=O)CC2CCCC2C1C(=O)N(CC(F)(F)CO)C C(=O)(C1CCCn2nccc21)NC1CC(C(C)NC(=O)CS(=O)(=O)N(C)C)C1 N1(C(CCCCC#C)=O)CC2CCCC(C1)N2CCC1CCCCCC1 c1(OC)c(C(N2CCC2CNC(c2ccnc3[nH]ncc23)=O)=O)cc(Cl)cc1Cl c1(CNC(NC(C)C2CC2)=NCc2cn(C)nc2C(F)(F)F)ccccc1C#N N1(C(CN(C)C)=O)CCCC(C)(C(=O)N(C(CO)C(=O)O)CC(N2CCOCC2)=O)C1 C(CCC(=O)NC(C1(C(=O)NCC2(S(C)=O)CC2)CC1)C)OCC c1(C(N(CC#C)C2CC2)=O)ccn(CCNC(=O)Cc2ccc[nH]2)c1 CCCCC(O)C(=O)N1CCC(CNC(=O)CC(C)F)C1(C)C C1(NC(C(C)NC(=O)NC)=O)C=CCCC1C(=O)NCCC1OCCC1(C)C C1(N(C(C(C2CN(C(C(C=C)C)=O)C2)OC)=O)C)CCOC(C)C1 c1(C(C(=O)N(C2CN(C(C3CC4CC4C3)=O)C2)C)CO)ccc(Cl)cc1 CC(C)S(=O)(=O)CC(=O)N1CCCC1CNC(=O)C=CC c1(-n2ncc(C(=O)NC3CCC(CNC(C(C)OCC)=O)C3)c2)ccc(Cl)cc1 N1(C(c2ncn(C)c2)=O)CCC2(CCCN2C(c2c(F)ccc(F)c2Cl)=O)C1 Cn1cc(S(C)(=O)=NC(=O)c2cnc3cc(C(=O)O)ccn23)cn1 C1(C(N(C)CC2(CNC(C3(C(C)C)CCC3)=O)CC2)=O)CC2C(C1)C2(C)C C(=O)(C#CC1CCC2(CC1)OCCO2)N1CCC(N(C(C(C)C(F)F)=O)C)CC1 c1(N2CC(NC(C3(C(C)C)CCC3)=O)CC(F)(F)C2)ncnc2c(Br)c[nH]c12 C(=O)(C1Cc2ccc(F)cc21)N(CC(C)(C)NC(C1CCc2nncn2C1)=O)C c1(C(=O)OC)ccc(S(=O)(=O)NCC2(F)CC(NC(=O)OC(C)(C)C)C2)c(Br)c1 c1(CNC(C(=O)OCC)Cc2cscn2)n[nH]c2c1CCOC2 Cc1ccccc1C=CC(N1CCC(NC(C2(C)CC=CCO2)=O)C1)=O C12(CC(=O)NCc3ncsn3)CCC1CN(C(=O)C(O)CC1CCCO1)C2 c1(C(=O)NCCCN(C(=O)C(c2cnn(C)c2)C)CCC)cnc(O)cc1O c1(N(C(C(=O)NCC)C(C)C2CCCCC2)CCC)ccc(F)c(F)c1 C1(C(=O)NCC2(OC)CCN(C(=O)CCc3cnco3)C2)CCCC(C)(C)CC1 c1(CC(=O)NCCCNC(COc2c(C)c(Cl)ccc2)=O)cnc2n1CCOC2 c1(C(=O)NC2CCC(C)N(C(=O)CC3CCSCC3)C2)cc2cc(F)ccc2s1 CC1(CNC(=O)CC2CC3(CCO2)CC3)CCCN(C(c2ccncc2)=O)C1 C1(C(=O)Nc2ccccc2NC(c2cc(C)cs2)=O)C2CCC1CN(CC)C2 C1(NCC(C)O)CCN(C(C2(C)CC(Oc3ccncc3)C2)=O)CC1 c1(N2CCC(CC=C)C2)ccc(S(=O)(=O)NC(c2ccccc2)C2CC2)cc1F c1(C(OC(C(N2CCN(CC)CC2)=O)=O)NC2CCCC3CC23)c(F)cccc1Cl c1(COC)nccc(N2CC3C(NC(c4cnon4)=O)C3C2)n1 N1(C(C2(CC)COC2)=O)CCOCC12CCN(Cc1c[nH]c3ncccc13)C2 N1(C(c2ccc(C(C)C)cc2)=O)CCCC(C)(C(N2CCCC2C#N)=O)C1 CC1CC(NC(C23CC2CCN3C(=O)CN(C)C)=O)CCN1C(N)=O N1(C(CC=CC=C)=O)CCC2(CCOCC2)C(CNC(=O)Cn2[nH]cnc2=N)C1 C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)(OC)CCC12CCC2 C(CC1=CCCCCC1)NC(CC1OCCCN(C(C2=C(C)OCC2)=O)C1)=O C1(CC(=O)NCC(CC=C)NC(c2cnc(N(C)C)nc2)=O)COC(C)(C)C1 c1(CCC(=O)NCC2(F)CC(NC(=O)CC3CCC(=O)N3)C2)ccc(Cl)nc1 C1(C(=O)OC)CCCC1C(=O)N(CCCCNC(c1cnc(CC(C)C)[nH]1)=O)C c1(CC)c(C(=O)NCC2CC(COC)CN2C(=O)CC)nnn1CC.C(C)=O c1(OC)cc(C(=O)NCC(CC(C)C)NC(c2cc(C(C)C)no2)=O)ccn1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CC(C(=O)NCCC(C)C(C)C)CC12CCC2 C(N=c1[nH]nc(Cl)s1)c1ccc(CNC(c2ccccc2)=O)cc1 c1(C(=O)OC2CCCN2CCl)cncc(N2CCCC2)n1.C1C(C2CC2)O1 C1(NC(c2ccc(C)nc2C)=O)CCN(C(=O)Cc2cccnc2O)CC(O)C1 Cc1cc(Br)ccc1S(=O)(=O)NC12CC(C(=O)N=c3cc(Cl)cn[nH]3)(C1)C2 N(C(=NCc1ccc(C(F)(F)F)cn1)N1CCC(CN(C)C)C1)C(=O)OC(C)C c1(C(=O)NC2N(Cc3c(Br)ccc(OC)c3)CC(F)(F)C2)ccc2nc[nH]c2c1 C1(C(=O)NC2(CC(=O)NC(C(CC)C)CN(C)C)CCC2)CCC(=O)N(C)C1 c1(C(N2C(CCCNC(C3CC34CC4)=O)CCC2)=O)cc([N+](=O)[O-])cc(Cl)c1Cl Cn1c(S)nc2cc(C(=O)NCCCNC(C3CCC3CF)=O)ccc2c1=O CN1CCN(Cc2ccccc2)C(NC(=O)C(F)(F)Oc2cc(F)cc(F)c2)C1 N1(C(c2ccc(C)s2)=O)CC(NC(C2CCCO2)=O)C2(CCOCC2)C1 c1(CC)c(C(=O)NC2C3CN(C(C4(O)CC4)=O)CC23)cnc2ncnn12 C1(NC(CN2CC(CC)C2)=O)CC2CCC(C1)N2C(c1oc(C2CC2)nc1C)=O c1(C(N(CC(C)NC(C2(CC=C)CC2)=O)CC)=O)nc(C)[nH]c2nccc1-2 N(C1CN(C(c2cocn2)=O)Cc2ccccc21)C(c1cc(C)c(C)[nH]1)=O C1(CNC(CC(=C=C)C)=O)CN(C)CCN1C(=O)CCNc1ncccn1 c1(CC(=O)NCC(C)(C)Cn2cc(C3CC=CCC3)nn2)ccc2ncoc2c1 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)COCC3CC3)C2)=O)cc1)NC CC1CC(=O)NCC1C(N1CCN(C(=O)CCc2ccn(C)n2)C(C)C1)=O c1(C(=O)NC2CN(C(=O)C3=CCSC3)CC23CC3)cc(Cl)c(F)cc1F C1(CC)CN(C(=O)CN2CCCS2(=O)=O)CCN1C(=O)Cc1nnc(C)o1 C1(C)(C(N(CCCNC(CN(CCC)C)=O)C)=O)Cc2ccccc2NC1=O C(=O)(C1=CCCCCC1)NCCCC1N(C(C(C)(Cl)Cl)=O)CCCC1 N1(C(c2ccc(C(C)=O)cn2)=O)CCN(C(c2ccc(C(C)C)o2)=O)C2CCC12 C1(C(=O)NCc2cncc(C(=O)NC(CO)C3CCC3)c2)CCC(=O)NC1 C12(C(=O)NC3(CSC)CC3)C(=O)C3CC1C2C3.c1(C(=O)NC)ccnc(COC)c1 C1(NC(c2nn(C)c(O)c2)=O)CCCCN(Cc2ccc(O)c(C(=O)O)c2)C1 N1(C(c2c(C)ccnc2O)=O)CCC2(CC1)CC2NC(c1ccc(O)nc1Cl)=O N1(CCn2c(C)csc2=O)CCC2(CCCN(C(C3CCCC4CCCN34)=O)C2)C1 c1(CNC(C2(C=C)CCC2)=O)cnn2c1CN(C(c1cc(C)on1)=O)CC2 C(=O)(CCCCC(=O)OC)N(CC(CC=C)C(=O)NC1CC(=O)N(C)C1)C c1(CNC(CC(=C)C)=O)nnc2n1CCN(C(c1cnc3sccn13)=O)C2 Cc1coc(C)c1C=CC(N1CC(CNC(C2CC2C#N)=O)C(O)C1)=O CC(C)CC(C(=O)NCC1CCOC1)N(C(=O)CC1CC2(CC2)C1)C C(=O)(CC(C)C(C)(C)NC(=O)C(CC)C(=O)OCC)N(CCC#C)CCO N1(CC(=O)NC(c2ccccc2)C)CCCC(CCNC(=O)C(C)(C)CO)C1 c1(C(=O)NCC2C(NC(CC3(C)CC3(Cl)Cl)=O)CC2)nc(O)nc(O)c1F C1(C(N2CC(O)(CNC(=O)CC3CCCSC3)C2)=O)CCC(=O)N1C1CC1 C=C(C)CC(C(=O)NCCN(CCOC)C(c1cc(OC)n(C)n1)=O)NC(C)=O c1(-c2cccc(C3(C(N4CC(O)C(F)C4)=O)CC3)c2)c(F)ccc2[nH]ccc12 C(=O)(C(CC(F)F)C1CCC1)NCC12CC(CNC(c3c(C)cco3)=O)(C1)C2 N1(C(c2ncn(CC)n2)=O)CCN(C(C23CC2COC3(C)C)=O)CC(C)(F)C1 N1(c2snc(C(=O)OC)n2)CCC(NC(c2ccc3ncsc3c2)=O)C12CCC2 Cc1ccc2cc(-c3c(C)noc3-c3ccc(C(N)=O)cc3)cnc2c1 c1(C(N2CCC(C)(NC(c3ccncc3)=O)C2)=O)cnc(Cl)c(N)c1 c1(C(=O)NC2CC(C)N(C(=O)CN(CC(C)(C)C)C)CC2)c(O)cc(F)cc1F N1(c2nnc(CCOC)s2)CC2(CCC(NC(=O)CC3CCCS3(=O)=O)CC2)C1 c1(-n2ncc(C(=O)NCC3N(C(COC4(C)CCCC4)=O)CC3)c2)ncc(Cl)cn1 Cn1cnn(CC(=O)NCC2CC2CNC(=O)CN2CSCC2=O)c1=O C=CC(C)(CCOCC)C(=O)NCCC(O)Cc1cnn(C)c1-c1nn[nH]n1 C1(C)(C(=O)NC2CC(CNC(C3(OC)CCOCC3)=O)C2)CCC(=O)CC1 C1(N(C(C2CCN(C(c3c(OC)nn(C)c3)=O)C2)=O)C2CC2)CC2CCC(C1)C2O CC(C)=C=CC(=O)NC(C(=O)NC(c1n[nH]c(CO)n1)C)C1CCOC1 C1(C(=O)NCc2c(CNC(C3(C)COCCO3)=O)cccc2)CC12CCOCC2 C1(C(=O)OC)CC2(C1)CC(C(N1CC(C)(CNC(C3C4CNC(=O)C34)=O)C1)=O)C2 N1(C(CC(C)(C(F)F)N(C)C)=O)CCC2(CCCCN(C(c3ccsc3)=O)C2)C1 c1(C(N2CC(F)C(F)C2)=O)cn2c(n1)CCC2 c1(C(=O)NC(c2ccncc2)CC=C)cc(Cl)nc(Cl)n1 N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)NCC2CCCN2CC)=C(F)C1 C(=O)(C1=CS(=O)CCC1)NCCN(C(C(C)CN(C)C)=O)C c1(NC)ccc(C(=O)NC2CC(N(C)C(C3CC(C(F)(F)F)C3)=O)C2)c(Cl)c1 CCS(=O)(=O)c1ccc(-c2noc(Cc3c(F)cc(C(F)(F)F)cc3Br)n2)cn1 C1(NC(C(c2ccc(C)cc2)F)=O)CC(O)CN(C(=O)CCCN2CCCC2)C1 c1(-c2nc(CC(CCCN(C)C(=O)OC(C)(C)C)CO)on2)c2c(nn1C)CCC2 N1(C(c2ncn(CC)n2)=O)CCC2C(CCN2C(=O)C(N2CCN(C)CC2)C)C1 c1(CC)nc(C)sc1C(=O)N(C)CCOCCN(C(=O)Cc1ccccc1F)C c1(C(=O)NC(C)(CNC(C2CCNC2=O)=O)C2CC2)nc(C2CC2)n2ccccc12 c1(C(N(C2CCCC2)C(CN(C(C)C)C)=O)C)ccccc1F c1(C(=O)NC2CC(CNC(CCC(C)OC)=O)C2)ccc(Br)cc1N C1(CC)(NC(=O)CC(=O)NCCCCl)CCCN(C(=O)CC2(C)CCCCC2)C1 O(P(=O)(CCC1CCCCO1)OCC)CC c1(OCC(=O)N(C(C)CNC(=O)COC2CCCCC2)C)cc(Cl)cc(Cl)c1F C(=O)(C(O)CCNC(c1cc(C(=O)NC)[nH]n1)=O)NC1(CC)CC1 c1(CC(=O)OC)ccc(NNC(=O)C(C)NS(=O)(=O)c2ccc(F)cc2)cc1 N1(C(C(CC(F)F)NC(c2cc(C)ncn2)=O)=O)CCCCCCCC1 C1(NC(C2(C#C)CCCC2)=O)CC2(CCN(C(c3cccc(C)c3)=O)C2)C1 n1(CCC)nc(C)c(C(=O)NCC2CC(NC(=O)C3=CCCCO3)C2)c1C CC1CN(C(=O)CCC(=O)NCC(F)F)CC1(C)CNC(=O)CSc1nncs1 C(=O)(CC(C)(C)SC)N(CC=CC(=O)N(CC(CC)O)CC)C c1(C(N(C(CC)C=C)C)=O)nc(C(F)(F)F)n2c1CCCC2 c1(C(N2C(CNC(Cc3c(C)nccc3)=O)CC2)=O)ccc(O)c(Cl)n1 C(=O)(C(CO)C(C)(C)C)N1CC(N(C(CSCC)=O)CCC)C(O)C1 N1(C(c2cnc(CC)s2)=O)CCOC(C)(CNC(=O)CC2(N(C)C)COC2)C1 CC(CCNCc1ccccc1OCC(F)(F)F)C(F)F CC1(C)CCCCCC1NC(C1C2CCCC2CN1C(C1CCSC1)=O)=O c1(C(=O)OCC)[nH]cc(C)c1C(=O)NC1CN(C(C2(C)CS(=O)(=O)C2)=O)CC1C CC1=C(C(=O)N2CCOC(CCNC(c3cncc(Cl)c3Cl)=O)C2)CCCO1 c1(SC)cc(C(N2CC3CC(NC(=O)COCC(F)F)C2C3)=O)ccc1N C1(CNC(c2onc(C)n2)=O)CCC(NC(=O)C(C)CF)CC1 C(N=C(NC)N1CCC(Oc2ccc(C#N)cn2)C1)c1c(CCC)onc1C.CC Cc1cccn2cc(C(N3CCCC(F)(CNC(=O)CCCN=[N+]=[N-])C3)=O)nc12 C1(CNC(COC2CCC(C)CC2)=O)CC2(CC2)CN1C(=O)C(C)N(C)C C1(C(NOCC(=O)NCc2ccsn2)=O)CCC(CO)CC1 c1(C(=O)NC2CCC(NC(CC3C(C)(C)OCCO3)=O)C2)cc(F)c(F)cc1Cl C1(C(N(CCNC(CCC#CC)=O)CC2CC2)=O)CCC(O)(C(F)(F)F)CC1 N1(C(c2c(C)n(C)cc2)=O)CCC(C)C(CC(=O)NCC(C)(C)C2(O)CCC2)C1 Cc1cccn2ncc(C(=O)NC(C)CCN(C(=O)C=C3CC3)C)c12 C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(C(CC#C)CC#C)=O)CC=C1 n1(CC(=O)NC2CC(N3CCNCC3)C2)ccc(C(=O)O)n1 N1(C(C2C(=C)C2)=O)CCC(CNC(c2cscc2C2CC2)=O)CC1C c1(C(N2CC(N(C(C3C(C(C)C)C3)=O)C)C2)=O)cc2ccc(Br)c(F)c2[nH]1 C1(NC(C(C)n2cnnn2)=O)CCCC2CN(C(=O)C(O)CC(C)(C)C)CC12 c1(C(N2C(CN(C)C(c3c(N)cccc3F)=O)CCC2)=O)cncc(N=[N+]=[N-])c1 C1(CNC(C(C2CCCC2)OC)=O)C2CN(C(=O)C(=O)Nc3ncc[nH]3)CC12 c1(CC)cc2cc(c1)Cc1ccc(cc1)NC2=O.c1(COC)ccc(Cl)cc1 N1(C(c2c(C)nsc2C)=O)C2CCC1C(CNC(=O)Cc1cc(F)cc(F)c1)C2 c1(CN(CC(CC)(C)COC)C2CC2)cc(I)ccc1Br c1(C(=O)OCC)ccc(C(N2CC3C(C(=O)NCc4cn[nH]c4)C3C2)=O)cc1 N1(C(CC(CC=C)NC(C2CCCCC2(C)C)=O)=O)CC2(CCC(=O)O2)C1 N1(C(CCC(CC)C)=O)CCC2CN(C(=O)CCN(CC)CC)C2C1 C1(OCCNC(C2CC(CCC)C2)=O)CCN(C(C2(C(N)=O)CCC2)=O)C1 c1(C(N2CC(C)C(CCNC(C3CC3CF)=O)C2)=O)csc2c1CCC(C)(C)C2 N1(C(Cn2cnc(=N)[nH]2)=O)CCN(C(c2cnn(CCC(F)(F)F)c2)=O)C2CC12 C1(NC(=O)NC(Cc2cccnc2)CO)COCC1C(=O)O c1(SC)cncc(C(N2CCC(CN(C(=O)C(=C3CCCCC3)F)C)C2)=O)c1 Cc1cc(=O)n(CC(N2CC3CC(CNC(c4ccon4)=O)C3C2)=O)cn1 C(c1ccc2c(c1)NC(=O)CO2)=CC(=O)NCC(CC)NC(CSCCC)=O c1(CC(=O)NC(CC)(C)CNC(c2ccsc2OC)=O)ccc2c(c1)CCCO2 CCCC(C(=O)NC1CC(O)C1)NC(=O)CCCn1ccnn1 c1(CNC(C=CC(C)NC(C(C)NC(C)=O)=O)=O)nc(C)c(C)[nH]1 N1(C(=O)CC2CCCOC2)CC2CCC1CN2C(c1cc2ncccc2o1)=O C1(NC(COCC=C)=O)(COC)CCCN(C(=O)C(C)P(C)(C)=O)C1 C1(C(=O)NCCCc2ccc(CNC(=O)OC(C)(C)C)cc2)CCCCC12CC2 c1(C(N(C2CC(NC(CCCC#C)=O)C2)C)=O)sccc1S(=O)(=O)N(C)C c1(C(=O)NCCOCCCNC(C=CC=CCC)=O)ccc(C)cc1 C1(C(N(CCCCNC(Cn2c(C)cc(C(F)F)n2)=O)C)=O)CC(C)(C)CN1C N1(C(=O)C2CC2)CCCCC1NCc1cnc(C(C)C)s1 Cc1cccc2ncnc(N3CC(NC(=O)C(c4cncn4C)O)CC3C)c12 C(CC(=O)O)(c1cccnc1)NCC(CO)NC(=O)OC(C)(C)C c1(C(=O)NCC(CN(C(=O)CN2CCCNC2=O)C)O)cnn(C2CC2)c1N c1(CC)cc(Br)ccc1C(N1CC(NC(c2cc(I)ccc2F)=O)C(O)C1)=O C(=O)(CC(F)(F)C(F)(F)F)N1CCC(N(C(C(=O)N(C)C)=O)C)C2(C1)CC2 C1(NC(c2c(C)nn(C)n2)=O)CCC2CCN(C(c3cnsn3)=O)C1C2 c1(C(=O)NCC(CC=C)NC(C2CCN(C)CC2)=O)cc2n(c1)CCCC2 N1(C(COC(C)(C)C)=O)C2CCC1CN(C(c1cncc(OC(F)F)c1)=O)C2 CC1(C)CN(C(=O)Nc2ccc(Cl)cc2)C1Cn1cc(CCC[Si](C)(C)C)nn1 N1(C(C2C(C)CCO2)=O)CCC(C2CC2)C1C(=O)NCc1ccncc1 CC1CN(C(C2(C)CC2(F)Cl)=O)CC(C)N(C(c2n[nH]c(C3CC3)n2)=O)C1 c1(C(=O)NCCNC(CCNS(NC)(=O)=O)=O)ccc(C)cc1.C1(=O)CCOCN1 N1(C(C(CSC)O)=O)CC(C2CN(C(=O)C(C(C)O)NC(C)=O)C2)C1 N1(C(C(CC)N2CCCC2=O)=O)CCC(CN2CCC(F)(F)C2)CC1 CC1Cc2cc(S(N)(=O)=O)ccc2C1NCCc1cc(F)ccc1Br C1(C)(CC)CC(C(=O)NC(C)CNC(c2ccc(NC(=O)NC)s2)=O)CCO1 CC1CCN(C(c2ccc(OC(F)F)cn2)=O)CC1CNC(=O)Cn1cnnc1 C(C(C)(C)CC(=O)NC(C)(CN(C)C)C(C)C)NC(CCC(C)SC)=O N1(CC)CCOCC1CC(=O)NC(C)CNC(=O)CCc1ccc(C)s1 c1(C(=O)NCC(CNC(=O)C(C)(C)O)OC)cn(C)nc1C1CCCC1.C(C)=O N1(C(C(=O)Nc2ccc(OC)c(OCC(N)=O)c2)=O)C2CCCC1COC2 C1(CCNC(C23CC(C(C)C)(C2)C3)=O)(OC)CN(C(c2cnc(C(C)C)[nH]2)=O)C1 c1(C(=O)NCC2(C)CCN(C(C3CCOC3=O)=O)C2)cnn2c1OCCC2 N1(C(CCC=C=C)=O)CCCCC(C2CN(C(=O)COC(C)C)C2)C1 C(=O)(C(O)CC(C)(C)C)N1CCCCC(NC(COc2ccc(CC)cc2)=O)C1 C#Cc1ccc(C(N2CCN(C(=O)CC3CC4CC4C3)CC2CCO)=O)cc1 c1(OC)ccc2nccc(C(=O)NCC3CCN3C(c3cc(C(C)=O)c[nH]3)=O)c2n1 CC1CCC(NC(c2cn(C3CC3)nn2)=O)CC1.C12CC1NC2=O N1(C(Cc2c(C)scc2)=O)CCOC(C)(CNC(c2c(Cl)c(C)nn2C)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2CC3CCC2O3)=O)cc(Cl)c(Br)[nH]1 c1(OC)c(C(=O)NCC(O)CN(C)C(C23CCC(CC2O)C3)=O)cc(Cl)cc1Cl S(=O)(=O)(c1cc(Cl)ccc1F)N1CCC2(C(C(=O)NC(CC)C(=O)NC)C2)CC1 C1(C)(NC(c2ccc(-c3ccc(F)cc3)o2)C)CCC(O)CC1 N1(CC(C)C)CCC(C(=O)NC(C2CN(C(C3(CF)CCOCC3)=O)C2)C)CC1 C1(CNC(=O)COCCF)CC2CCCCC2N1C(=O)CC1CCS(=O)(=O)C1 c1(OC)ccc(C(=O)NCC2CC(C)N(C(c3ccccc3C)=O)C2)c(OC)c1 N1(C(C(C)N(C)C)=O)CCN(C(=O)CC2CCN(C)CC2)CC(CO)C1 c1(C(C)C)ccc2c(c1)C(NC(N1CC3CC(O)CC3C1)=O)CCC2 c1(C(N2CCC(O)(C(CNC(CC(=C)Br)=O)C)C2)=O)c(C)ccc(C)c1N C(=O)(CC(C)(C)C(=O)N(CC(C)NC(c1cncc(Cl)n1)=O)C)OC C1(CNC(CC(CN(C)C)(C)C)=O)CC2CCCCC2N1C(C1CCC1)=O c1(C(C(CC)=O)=O)cncc(NC(C2(C)CC2)=O)c1.C1(CC(=O)N)(CN)CC1.OC c1(C(=O)NCC(CNC(c2cccc(C3CC3(F)F)c2)=O)O)cc(F)ccc1O c1(C(N2CC3CC(C(=O)NCCCC(C)(C)CO)(C2)C3)=O)cncc2[nH]ccc12 c1(NCc2ncc(OC)nc2)nccc(=NCc2cccnc2Br)[nH]1 C1(OC)CCCC(CNC(=O)CN(CC(C)C)C(c2nc(C)oc2OC)=O)C1 Cc1nn(C)c(C)c1C(=O)C(=O)NCC(C)N(CC(=O)NC(c1cccs1)C)C c1(C(N(C2CC(NC(C3(C(F)F)CC(F)(F)C3)=O)C2)C)=O)cnc2n1CCC2 C1(C)(C(=O)NCc2nnc(C)s2)CCCN1C(=O)C=Cc1cc[nH]n1 CS(=O)(=O)c1cc(C(=O)NC2CCC(NC(c3ccsc3CN(C)C)=O)C2)cs1 C(=O)(CCN=C(NCc1ccc(Br)c(F)c1)NC1CC12CC2)N(C1CC1)CC CC1CN(C(C2CCCOCC2)=O)CC2(CCN(C(c3cnc(O)n3C)=O)C2)O1 C1(C(=O)NCC2(N(c3cncnc3)C3CC3)CCCC2)CC(F)CN1CC C(=O)(C(O)C(CCC)NC(C1CCS1(=O)=O)=O)NC1(C#C)CC(F)(F)C1 C=CC1CCN(C(C2(NC(C3CCCOCC3)=O)CCOCC2)=O)C1 C1(CNC(C(C)(C)C)=O)CN(C(C2CCCCCC2)=O)CCC1C(F)(F)F N(C1CCc2cccnc21)C(C12C(NC(c3c(C)ncs3)=O)C3CC1C2C3)=O N1(C(C2(n3cc(Cc4cccc(C)c4)nn3)CC2)=O)CCCC2C(O)C(C)(C)C12 Cc1c(C(N2C(C(=O)NCC(F)CO)CC2C)=O)cccc1C#N C1(NC(C2CCCCC2)=O)CCCC12CCN(C(c1cc(Br)cs1)=O)C2 c1(C(=O)NC2(CNC(c3sccc3-n3cnnn3)=O)CC2)csc([N+](=O)[O-])c1 Cc1ccc(CCC(=O)NC2CCC(NC(C3SCCCS3)=O)C2)cn1 C1(C(=O)NC(C)CO)CCCN(C(c2cn(C)cn2)=O)C1 N1(CCNC(C(C)(C)F)=O)CCCN(C(C2C(c3ccncc3)C2(C)C)=O)CC1 C1(N(C(C(C(C)O)N(C)C)=O)C)CCCCN(C(c2ccc(O)cc2)=O)C1 Cc1cc(Br)c(NC(=O)NCC2CCOCC2C)cc1[N+](=O)[O-] CC12CCCCC1(C(N1CCC(CC(=O)NCCN3CCC(CO)C3)C1)=O)C2 N1(C(CCN(C(C)=O)C)=O)CCC(C(C)NC(=O)Cc2c(C)n[nH]c2C)CC1 c1(OC)cc(C=CC(=O)NCc2ccc(C3CC3)cc2C)cc(Cl)c1O N1(C(C2ON=C(CC)C2)=O)CCC2C(CCCN2C(=O)C(C)CC2CCCC2)C1 c1(NC)ccc(C(N2CCCC2CNC(=O)C(O)C2CCCC2)=O)c(C)c1 C1(C(C(=O)NCc2cccs2)N(C)Cc2cn(CC)nc2)CCC2(CC1)CC2 N1(C(C=Cc2cc(C)no2)=O)CCC2CC1CN2C(c1ccc2cnoc2c1)=O C1(C(N2CCC(NC(c3cn(C)nc3C3CCCC3)=O)C2)=O)CCC2(CCC2)O1 c1(C(c2nnnn2C2COC2)NC(C)CCCCO)cc(Br)cc2c1OCC2 C1(C(=O)NC(C)CN2CCN(C)CC2)CC12CCN(C(c1cnns1)=O)CC2 N1(C(C=CC)=O)CCC(C2(NC(c3cccn3CCC)=O)CC2)C1 Cc1cc(NC(=O)NC2CCN(C(=O)CC(C)(C)F)C2)ccc1NC(C)C C1(CNC(C2C(C)COCC2)=O)CC2(C1)CC(N)CCO2 c1(OCCOC)cccc(CC(=O)NC2CC(CO)N(C(=O)CC(F)F)C2)c1 N1(C(CCc2nc(C)sc2)=O)CCCN(C(=O)C(C)CC2CCCO2)CC1CO CC1CCC(NC(c2cncc(-n3cnnn3)c2)=O)CN1C(=O)CCC(C)(C)C C1(NC(CCNC(C)=O)=O)CCSC12CN(C(C1CCC1c1nncn1C)=O)C2 C1(NC(c2cncc(CC)c2)=O)CCCN(C(=O)Cc2ccnn2C)CC1 c1(C(=O)NCC(O)CCNC(C2(F)CCC2)=O)cnc2ccc(F)cn12 N1(C(C(c2cncnc2)C)=O)CC(CNC(c2ncc(F)cc2N)=O)C(C)(C)C1 N1(C(c2cc(CC)c(C)cc2)=O)CCC2(C1)CN(C(=O)CC1(O)CC1)CC(C)O2 N1(C(C(c2cc(C)oc2C)C)=O)C2CCC1C(CNC(c1cc(F)n(C)n1)=O)C2 C1(C(=O)NCC2(CCNC(=O)C(O)c3ccsc3)CC2)CC12CCOCC2 CC(C)(C)C(CNC(C1CC2(CCC2O)C1)=O)C(=O)NCCc1ccc(O)cn1 c1(NC(C2CCC(CN)CC2)=O)cnn2c1CCCC2 N1(C(c2c(COC)cco2)=O)CC2(CCCC(CNC(=O)C(C)C3CCC3)O2)C1 C(=O)(CC(C)CN(C)C)NCC(CC)NC(=O)CCc1ccc(CO)cc1 C1(CNC(c2ccc(OCC#C)cc2)=O)CN(C(C2CCCN2C)=O)CC12CC2 c1(C2(N(C(C(=O)NCC(n3cccn3)C)=O)C3CCCC3)CC2)ccccc1 C1(OC)CN(C(=O)CCCN(C(=O)C(C)(C)n2cncn2)C)CC12CC2 S(=O)(=O)(c1c[nH]ccc1=NCC1COCC(=O)N1C)N1CCCC(F)(CC)C1 c1(C(N(C2CCCN(C(C3(C)CC=CCO3)=O)C2)C)=O)cnc(O)c(F)c1 C1(OC)(CNC(=O)Cc2cncn2C)CCN(C(=O)C(c2ccc(F)cc2)=O)C1 Cc1csc2ncc(C(N3CC4CCN(C(=O)CC5CCCO5)C4C3)=O)c(=O)n12 C1(NC(=O)Cc2cncs2)CC2CCC1(C(=O)NCCCC(F)(F)F)C2 N1(C(c2ccc(C)c(Cl)c2Cl)=O)CC2COCC(C1)C2NC(=O)C(Cl)=CCl C(=O)(CC(C)CC(C)(C)C)N1CC(O)(C(C)NC(C=C(C)C(F)F)=O)C1 C=CCCC(C(=O)NCCCNC(=O)NC)NC(=O)C=CCCC c1(CC(=O)NCCOC2N(C(CC(CC)C)=O)CCCC2)cccc(C#N)c1 C1(C(=O)NC(CC)CNC(c2cc(Cl)c(Cl)s2)=O)CCc2nncn2C1 Cc1cnc(CN2CC(C(N3CCCCC(C)C3)=O)CC(F)C2)c(F)c1 c1(C(N2C(C)CC(NC(c3cc(CCC)[nH]n3)=O)C2)=O)coc2c(C)cccc12 CN1CCN(C(C2(F)CCN(c3ccc(CN)cn3)C2)=O)CC1 c1(C(=O)OCC)c(C)sc(CNC(CC2CCCN2C)C2CC2)c1Cl N1(C(C2CC2C2CCCC2)=O)CC2CCCC(C1)N2C(C1CCC2CC2CC1)=O c1(CC)cc(C(N2CC=CC2CNC(C2CC(N(C)CC)C2)=O)=O)ns1 Cc1cc(OCC(=O)NC2(CNC(c3cc(Cl)cn3C)=O)CCCC2)cc(C)c1 c1(CN2CCN(C3CN(C(C4C5COCC45)=O)C3)CC2)ccc(O)cc1O O=S(=O)(c1cccc(CNc2cc(Br)ncc2Oc2ccccc2)c1)N1CC1 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CCC1NC(C1CC=CC1)=O C1(CNC(c2c(OC)ccs2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC2(CCC2)O1 C1(C(=O)NCC2C(NC(C(c3nc(C)sc3)=O)=O)CCC2)CCCCCC1 N#Cc1c(N2CC3CC(C2)C3NC(=O)Cc2ccc3c(c2)COC3)cccc1F Cc1sc(C(=O)NCC2CC(C(F)F)CN2C(=O)CSC(C)(C)C)c(C)c1C c1(OCCOC)ccc(C(=O)OC(C)CC(=O)O)cc1 C1(CCNC(C(C=C)O)=O)CSCCN1C(c1cc(Br)nn1C)=O N1(CCNC(C2CC(OCC3(COC)CCOC3)C2)=O)CCCC(C)C1 c1(NC(=O)NC(c2ccc(C)nc2)C)ccc2c(c1)C(F)(F)C(=O)N2 C1(C(=O)NCCSCC(=O)Nc2c(COC)ncnc2)CC(C(C)C)=NO1 Cc1nc(C(N2CCN(C3CN(C(=O)C(F)F)C3)CC2)=O)c2ccccn12 Cn1c(C(=O)NC2CCC(CNC(c3cc(N)cc(N)c3)=O)C2)cc(Cl)c1Cl C1(NC(COC)=O)(CO)CN(C(=O)CCc2nnc(C(F)F)o2)C1 CC1C(NC(c2cnc(Cl)c(C3CC3)c2)=O)CCCN1C(C1CC2(CCC2)C1)=O C1(C(=O)NC(COC)C)C2CCCC1CN(Cc1c(Br)cc(Br)c(O)c1Br)C2 S(=O)(=O)(CCCOC)NC(C(COC)C)=O c1(C(=O)NCCNC(C(CC)OC)=O)cc2nc(Cl)ccc2o1 CC(C)C(C(=O)NCCc1ocnc1CO)C(C)NC(=O)CNC(N)=O CC1(C)CC(CNC(c2ccccc2)=O)CN(C(c2nnn3ccccc23)=O)C1 Cc1ccc(C)c(S(=O)(=O)NC2CN(C(c3nc(CO)cs3)=O)CC2O)c1 C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCN(C(=O)C=C2CCCC2)C1 N1(C(C(C2CCCC2)NC(CC2ON=C(C)C2)=O)=O)CC(O)CC1C(N)=O c1(C(=O)OC)ccc(C(=O)NCC2CCCCCN2C(c2cnco2)=O)cc1Cl C(=O)(CCCCCCNC1(CF)CCC1)NCC1(C)CCOC1 c1(OCCC)ccccc1C(=O)NCC(O)CNC(=O)C#CC(C)C c1(NC(CSS(=NC)(C)=O)=O)n[nH]c2c1CCN(C(=O)CCCC(CC)OC)C2 N1(C(CC#N)=O)CC(C2(NC(C3(C(=O)NCCc4ccccc4)CC3)=O)CC2)C1 C(c1ccc(Br)cc1)=CCCNC(c1c(C)nccc1)=O c1(C(N2CCCC(NC(c3c(CC)nn[nH]3)=O)(CO)C2)=O)cccc2c1COC2 C#Cc1cccc(C(=O)NCCNC(c2cc(O)nc(OC)n2)=O)c1F C(=O)(CC(C)CNC(=O)CCc1cncnc1)NCC(C#C)CC CC1CCC(C(=O)NCCCN(C)C)CN1C(=O)CCc1nc(=N)[nH][nH]1 C1(COC)CCN(C(=O)CNC(=O)COC2CC2)CC1.C12CCC1CNC2=O C12(C(=O)NCc3nccc(C)c3)CC(CO)(CN1C(C1CC3COCC3C1)=O)C2 C1(C(=O)N)(CO)CCCC1.C1(CC(=O)NC(C(=O)OC)C2CCCO2)OCCC1C c1(NC2CC(C)N(C(C3(CN(C)C)CC3)=O)C2)cc2nncn2cn1 c1(OC)cccc(Cl)c1CNC(N1CCC(C)C(NC(=O)OC(C)(C)C)C1)=O C(=O)(CC(C)CN=C(NCC1(O)CCN(C)CC1)NC1CCS(=O)(=O)C1)OC C1(NC(CNC(CN2CCC(C)C2)=O)=O)(CO)CCN(C)C1 C1(C(N(C2COCC2O)CC)=O)CC2CN(C(=O)CCCC(C)(C)C)CC2C1 C1(CNC(C2(SC)CCC2)=O)CC(C(=O)Nc2cc(C)ccc2O)=NO1 C1(CNC(CC(C)C(F)F)=O)CN(C(=O)CCn2ccnc2)C2(CCOCC2)C1 Cc1nc(C(=O)NCCC2CC(NC(C3C(C)C3(F)F)=O)C2)c(C)n1C1CC1 c1(SCC)cncc(C(N2CC(CNC(c3c(C)cnn3CC)=O)(OC)C2)=O)n1 Cc1cc(C(=O)NNC(=S)NC2CCS(=O)(=O)C2)c(C)n1C C#Cc1ccc(C(N2CCCC2CN=[N+]=[N-])=O)cc1C N1(C(c2cnc(SC)n2C)=O)CCC(NC(C2CC2C)=O)C(F)C1 C1(NC(COCCOCC)=O)CN(C(C2CCC(O)CC2)=O)CC1C C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC(CCNC(c2ccccc2)=O)CC1 Cn1ncc(Cl)c1CC(=O)NCCCN1CCN(C(C2CC23CCC3)=O)CC1 C1(NC(C2COCCC2(F)F)=O)C2CC1CN(C(c1ccccn1)=O)C2 CN=c1[nH]cc(C(=O)NCc2c[nH]nc2C(=O)NC(C)C(C)n2cccn2)s1 c1(NC(N2CCCC2)=O)nc(Cl)nc2[nH]cnc12.c1(O)cc(OC(F)(F)F)ccc1C c1(OCN2C3(CCC(N)C2)CCC3)cccc2[nH]c3ccccc3c12 c1(C(=O)NCC(C)NC(=O)C2=CCCC2)cc2ccnn2cn1 c1(C(N2CC(C(N3CCC(OCC)C3)=O)(SC)C2)=O)cnncc1O c1(OC)ccc(C(=O)NC2CC(CC(N3CC4C(C3)C4(C)C)=O)C2)c([N+](=O)[O-])c1 Cc1cc(C(=O)NCC23CC2CN(C(=O)C#CC2CC2)C3)ccc1F C1(CCC)(NC(=O)C(C)CCCOC)CCCN(C(c2c(C#N)cnn2C)=O)C1 C1(C)(CNC(CC2CCCC(C)O2)=O)CC(F)(F)CN1C(c1cnn[nH]1)=O CCC(C)C(O)CC(=O)NC1CCOC1C(=O)NCC(C)(C)C1=CCCC1 C1(F)(C(N2CCC(C(C)NC(c3cnccc3Cl)=O)CC2)=O)CCCC=C1F Cc1ccc(S(=O)(=O)NC2CCCC2NC(N2CCCSCC2)=O)c(F)c1 C1(C(=O)NCCN(CCC)CC)CC(O)CCN1C(=O)CNC(=O)NC CCCC(CC)C(=O)NC1CCCCC1CNC(c1ccc(F)s1)=O N1(C(Cc2c(C)cco2)=O)CCC(c2ccccc2)(NC(C2CC23CC3)=O)CC1 C(CN(C(C(C)(C)C)c1ccccc1)C)(C(C)C)OC.C1CO1 c1(OCC)cc(NCC2CC(NC(C3CC3F)=O)C2)nc(C)n1 Cc1nc(Br)ccc1C(N1CC2CCC2(CNC(=O)Cc2cc(Br)cs2)C1)=O N1(C(c2c(C)snn2)=O)CC(NC(c2cn(C)cc2C(F)(F)F)=O)CC(O)C1 c1(CC(=O)NC(CNC(C2N(CC)CCC2)=O)(C)C2CC2)nc2ccccc2s1 Cc1cc(NC(C(C)NC(c2cccc(F)n2)=O)C(C)C)nc(S(C)(=O)=O)n1 C1(C(N2CC(CNC(c3cncc(SC)c3)=O)C(C)C2)=O)CCN(C)C(=O)C1.C1CC1 c1(C(N2CCN(C(CC(CCC)C)=O)CC2CCO)=O)cc(F)c(C#N)c(F)c1 C1(NC(C(C)=CC2CC2)=O)COC2(C1)CN(C(C1CCCC3(CC3)C1)=O)C2 CC(C)CCC(F)C(=O)N(CCCNC(=O)C(C)C1CCOC1)C(C)C c1(C(=O)NCC(C)CN(C(=O)Cc2cncn2C2CC2)C)n[nH]c2c1CCOC2 N1(C(c2c(CC)ccs2)=O)C2CCC1CC(NC(C1C=C1C)=O)C2 Cc1cccc2cc(C(=O)NCCCOCCNC(C3COC(=O)C3)=O)oc12 CC(C)CC(C)(C)C(=O)NC1CCCC1NC(c1ccccc1CO)=O C1(NC(CC(C)F)=O)CCC(NC(c2nccnc2N)=O)CC1 C(=O)(C(C)CO)N(C(C(=O)N(CCCOCC)C)C1CC1)C N1(C(c2cc(OC)c(Br)nc2)=O)CCC(C)(C)C(NC(C2CCC2)=O)C1 CCCC(CC1CCCC1)C(=O)NCC1CN(C(=O)C(COC)N=[N+]=[N-])C1 C1(NC(C(CC=C)OC)=O)COC2(C1)CN(C(=O)CC1OCCO1)C2 c1(CC(=O)NCC2C(C(=O)Nc3cccc(OCC)c3)C2)cc(C)ccc1F N1(C(C2CCC(C)O2)=O)CC2CC(C1)CN(C(=O)CN1CCCCC1)C2 c1(C(N2CC(NC(C3C(CCC)CCC3)=O)(CO)C2)=O)cnc2c(c1)COCC2 c1(OC)ccccc1CN(C(=O)CN(CCN(C)C)C(C1CCC1)=O)C Cc1ccc(C(N2CCCC(N(C(=O)CC3CCC(C)CO3)C)C2)=O)cc1C C1(C(N2CCCC(C=C)C2)C(=O)NCC(=C)C)Cc2ccccc2C1 c1(C(N2CCC(O)C(C(N3CC4COCC4C3)=O)C2)=O)ccc(F)c(I)c1 C1(NC(C(CC2CCC2)OC)=O)CCC(C)(CNC(C2CCC(=O)O2)=O)C1 Cc1cc(Cl)c(Cl)cc1C(=O)NC1CN(C(=O)C(O)CC(F)F)C2(CCC2)C1 N(C1CCCc2occc21)C(CCCNC(=O)C=CC1CCOCC1)=O C1(C2CCCN(C(=O)CN(C)C)C2)(NC(CN(C)C(c2ccncc2)=O)=O)CC1 c1(CNC(=O)NCC2CC23CCC3)ncc(Cl)cc1Cl C1(NC(CC(C)N(C)C)=O)CC=CCC1C(N1CC(N(C)C)CC1C)=O C=C1CCN(C(C2COCOC2)=O)C(C(N2CCC(OCCO)C2)=O)C1 N1(C(c2c(SC)ccs2)=O)CC2(CCC2)CC1CNC(=O)CN(C1CCC1)C c1(C(=O)NC(CC=C)CNC(=O)Cc2ccn(CC)n2)cc2c(s1)CCC2 N1(C(c2c(C)cccc2N)=O)CC(C)(CNC(C23CCC2C3)=O)CC1(C)C c1(C(=O)NCCN(C(C(n2c(C)ccn2)C)=O)C(C)C)cnc(=NCCF)[nH]c1 C1(NC(C(CC)OC)=O)CCSC12CN(C(c1cc(O)ncc1Br)=O)C2 c1(C(=O)NCC(C2CC2)NC(C=C(C)c2cnn(C)c2)=O)ccc(S(C)(=O)=O)[nH]1 c1(C(N2C(CNC(C3CC=C(C)CC3)=O)C(C)CCC2)=O)c([N+](=O)[O-])cnn1C C(=O)(C1=CS(=O)CCC1)N1CC(C)C(CNC(C2(C)CNC(=O)C2)=O)C1 C1(NC(CCC=C)=O)COC2(CCN(c3ncc4[nH]ccc4n3)CC2)C1 C1(C(=O)NCC(CC2CC2)CO)(CNC(C=C(C)C(F)F)=O)CCCC1 N1(C(Cc2ccn(C)n2)=O)CCOC(C)(CNc2ccccc2)C1 CCC(C)(C)CC(=O)N1CCOCC(CNC(c2c(Cl)csc2Cl)=O)C1 CCCC(CNC(c1cc(C)nn1C)=O)C(=O)NC1CC12CC(OC)C2 C1(CC=C)(CNC(=O)Cc2cnoc2)CCCN1C(=O)C(O)CCN(C)C Cc1nc(C(=O)NCC2(F)CC(CNC(=O)Cc3cnn(C)c3)C2)c(C)s1 c1(C(N2CC(NC(C3N(C)CCC3)=O)C(F)C2)=O)cc2nnn(C)c2s1 CN1N=C(C(=O)N2CCC3CC23C(=O)NC2CCCC2C#N)CCC1=O c1(C(N2N=C(C=O)CC(C)C2)=O)cnc2ccc(Br)cc2c1 C(CC(=O)N1CC(O)CCO1)NC(C(c1ccccn1)C)=O c1(C(N(C(=O)NCCN(C2C(F)(F)C23CC3)C)C)O)ccccc1Cl c1(N(C)C)ccc(S(=O)(=O)NCC2COCO2)cc1 Cc1ncc(S(N)(=O)=O)cc1C(=O)NC1CC1NC(C1CCC(C)(C)O1)=O c1(OC)ncc(-c2scc(C)c2C)cc1C(=O)Nc1scc(C)c1C(N)=O C(CCC(C(=O)N(C)Cc1cocn1)NC(c1cc(CCO)on1)=O)OC C(=O)(C1=CCN(C(=O)Cn2cncn2)CC1)NC(C)C CC1CC2CC2CC1C(N1CCCC1CN(C(=O)CCc1cccnc1Cl)C)=O S(=O)(=O)(c1ccc(Br)cc1)NC1C(C)(C)NC(=O)CC1 c1(C(N2CCC(NC(C3CCC(C#N)CC3)=O)C2)=O)ccn2cccc2c1 N1(CC(=O)N(C2CCN(C(COCC(=C)C)=O)C2)CC)CCN(C)C(=O)C1 C12(C(=O)NCc3c(C)noc3)C(NC(c3ncc(F)cc3C)=O)C3CC1C2C3 CCCC(F)(F)C(=O)NC1CCOC(C(=O)NCc2cn(C)nc2OC)C1 C1(CC(=O)N(C2CCN(C(=O)C(C)C(=O)OC)C2)CCC)(COC)CCCCC1 c1(C(=O)NCC(C)NC(C=Cc2ccc(SC)s2)=O)ccc2nc(O)n(C)c2c1 c1(C(=O)NCC(C)N(C(=O)C(C)OCC(C)C)CC)cnsc1C C#Cc1cc(C(=O)NCC(C)(O)CNC(=O)C(C)(C)N(C)C)cc(F)c1 C(=O)(C(C)CC(=O)c1ccc(F)cc1)NCC#CCNC(C(C)SCCCC)=O C1(C(=O)NCCC(C)NC(c2c(C(=O)OCC)c[nH]c2)=O)CCN(C)C1C c1(CC(=O)NC2(CNC(C(CC)O)=O)CCOCC2)cc(F)c(F)cc1F CC(C(=O)NCC(C1CC1)N(C)C(C1CC(=O)C1)=O)S(C)(=O)=O C1(=O)CCCCCN1C.C1(C(=O)NCC2(C(=O)OC)CC2)C2CCC(C2)C1C c1(CC(=O)NC2CC(CNC(c3cncc(F)c3)=O)C(O)C2)n[nH]c2c1CCCC2 C1(CC(=O)NCc2cnc(C)s2)CC(NC(C23CC(F)(C2)C3)=O)C1(C)C c1(-n2cc(CC3N(C(=O)NC4CC4c4cccs4)CCC3)nn2)ccccc1F c1(C(=O)NCCC(C)NC(C2CC23CCC3)=O)cncc(S(C)(=O)=O)c1 Cc1cc(C(=O)NC2CCC(C)(N3CCOCC3)CC2)nnc1O c1(C(N(CCCNC(c2nccc(OC)c2F)=O)C)=O)nc2n(c1Cl)CCCC2 C1(CNC(C2C(c3cn(C)nc3)CCO2)=O)CN(C(c2csc(Cl)n2)=O)CCO1 N1(C(C(c2cncnc2)C)=O)CCCC(C)(C)C1C(=O)NC1C(C)CCC1C Cc1nsc(N)c1C(N1CCC(C(C)NC(=O)C#CC2CC2)CC1)=O C(=O)(C(C)(C)CCCO)NCC(C)(C1CC1)NC(C1CN(C)C(=O)CC1)=O Cc1ccc(Cl)c(F)c1C(=O)NC1CC(C(=O)O)C2CC12 c1(C(=O)OC)cc(C(=O)NCC2(CNC(c3nc(=O)n(C)[nH]3)=O)CC2)cn1C c1(C(=O)NCCC2CN(C(CN(C)C)=O)C2)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 C=CCCCC(C(=O)N1CCCC(C#N)C1)NC(=O)C(C)C(O)C(C)C Cc1nc(O)c2cc(C(=O)NCC3CC3NC(C3CC4CCC3O4)=O)ccc2n1 C(C(CC(F)(F)F)NC(C1CCC1(C)C)=O)NC(C1(CC#C)CCC1)=O N1(C(CC2CC(=O)NC2=O)=O)CC2CCC1C(NC(c1ncc(Cl)s1)=O)C2 c1(C(N(C2CCN(C(=O)Cn3nccn3)CC2)C)=O)cc(C(F)(F)F)cc(O)c1 CCCCCC(O)CC(=O)N(CCC(C(C)C)NC(c1ccc(N)c(F)n1)=O)C n1(CC(=O)NCC2(NC(C3CC=C(C)CC3)=O)CCC2)nc(C)c2c1CCCC2 CCCCC(CC)CC(=O)NCCN(CCOC)C(c1cc(Cl)nn1C)=O Cc1ncsc1COCC(=O)NCC(C)(C1CC1)NC(C1CCC(C)S1)=O C(=O)(C(F)(Cc1ccccc1)C(C)C)OC.C1(=O)C(CO)(CO)N1 c1(N2CCC(C(C)NC(C(CCCC)C(C)C)=O)C2)nc(Cl)nc2[nH]c(O)nc12 C(CCCCCCC(=O)NC(CNC(=O)C(C1CC1)C1CC1)CO)SC C1(N(C(=O)NC(c2ccc(C(F)(F)F)cc2)CC)CC(C)(C)C)CCCCC1O c1(-n2cc(-c3cnc(C)s3)nn2)ccncc1C(=O)NC1NC(=O)C2CC12 C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(=O)C(C)(C)CF)C2(CCOCC2)C1 C1(NC(c2ccc(F)cc2Cl)=O)CC(C2CCN(C(=O)C3=C(Cl)CCCC3)C2)C1 CCCC(CC(=O)NC(C)COCC)NC(=O)CC1CCC(=O)NC1 CCCC(CCCNC(C1CC(C)OC1C)=O)N=c1nc(C)[nH]s1 C(=O)(C1CCc2c[nH]nc21)NCC(CCOC)NC(c1ccc(F)c(C)c1)=O N1(C(=O)NC(C)Cc2ccncc2)CCC(F)(C(c2ccccc2)O)C1 CC(CS(C)=O)C(=O)N(C)CC1(NC(c2cccc(N3CCOC3=O)c2)=O)CC1 c1(CC(=O)N(C)C)cn2ccccc2n1.C12CCCN(C1)CC(=O)NC2 c1(C(=O)NCC2CCC(NC(c3c(C)ncs3)=O)C2)nc(O)c(C)s1 N1(C(CNC(CCCCC)=O)=O)CCC(NC(c2ccoc2)=O)C2(CCC2)C1 C1(C#N)(C(N(CC(=O)NC2CCN(CC)C2)CC)=O)CCCO1 C(CC(C)C)(C(=O)NCC(C)(C)NC(=O)CCc1cccc(OC(F)F)c1)OC n1(CC(C)N(C2CCCNC2)C2CC2)cc(Cl)cn1 Cn1[nH]c(C(=O)NCC2CC(CNC(C3(C(F)F)CCCC3)=O)CO2)nc1=O N1(C(c2c(C)nc(O)cc2)=O)CCC2(NC(=O)Cc3ccco3)CCCC12 C1(NC(CCN(C)CCO)=O)(CNC(=O)CC2OCCO2)CCSC1 C1(C(=O)NCC2(NC(CN(C(C)C)C)=O)CCC2)CCC2(CC2)C1 CC1(C)C=C(C(=O)NCC2CCCC2NC(=O)CC2CCC(C)(O)CC2)C1 N1(C(c2c(OC)csc2)=O)CCC(O)C(C(N2CCCCC2C)=O)C1 c1(C(=O)NCC(c2ccccc2)CN(C)C)ccc2[nH]c3c(c2c1)CN(C)CC3 c1(-n2cc(CCCC(C)=O)nn2)cc(C(=O)NCCCSC(F)F)c(=O)n(C)c1 C1(C)(NC(C2CCC(C)O2)=O)CCN(C(=O)CC(C)F)CC1 C1(NC(c2c(C)onc2-c2ccccc2Cl)=O)CCN(C(=O)C(C)C)CC1F N1(C(C(F)=CCC)=O)Cc2ccccc2CC1CNC(=O)CC1CNC(=O)C1 C(=O)(C(C)S(N)(=O)=O)NC(C1(C(N2C(CSC)CCC2)=O)CC1)(C)C n1(CC(=O)NCC(c2ccccc2)NC(C=CCCC)=O)c(C)ccc1C c1(COC)ccc(C(=O)N(C2CCN(C(=O)CO)CC2)C)cc1OC C(=O)(C1=CCCSC1)NC(C(C)O)C(=O)N(C1(CCO)CC1)C C=CC(C)CC(=O)NCC(C1CCCCC1)NC(c1cc(C(C)(F)F)on1)=O C1(CN(C(C2CCCC2F)=O)CC)CCCCN1C(=O)CCSCC(N)=O C(=O)(C1=CCCC1C)NCC(C)N(C)C(c1cn(C)nc1C1CCOCC1)=O CC(F)(F)CC(=O)NCC1(CNC(C2CCNC(=O)C2)=O)CC1 S(=O)(=O)(c1cccc(S(=O)(=O)NC(C)(C)C)c1)NCC(=C)CC c1(C(N(C)CC2N(C(C(C)SCC)=O)CCCC2)=O)cc(O)cc(=O)o1 N1(CCNC(=O)CC2CCCO2)CCN(C(=O)C(O)Cn2cncn2)CC1 c1(C(=O)NCC=CCNC(C2CC(OC(C)(C)C)C2)=O)ccc2ncsc2c1 N1(N2C(C=O)C(C(=O)C3=C(Cl)CCOC3)CC2)CC2(CNC(=O)N2C)C1.CC(=O)NC c1(NC(C2N(S(CCC)(=O)=O)CCNC2)=O)cc(F)ccc1[N+](=O)[O-] c1(CNC(C2CCCCN2C(=O)NCCC)=O)cc(F)c2cc[nH]c2c1 C1(C(=O)NCC2(C(C)N(C(=O)CC(C)n3cccn3)C3CC3)CC2)C2CC(=O)CC12 N1(C(c2nc(C(C)OC)oc2)=O)CCCC(O)(CCNC(c2cnns2)=O)C1 N1(C(C2(C#C)CCCC2)=O)CCN(C(=O)CCC(C(=O)OC)OC)CC(CO)C1 N1(C(C=CC)=O)CC2CCC1CC2NC(=O)CC(C)(C)O N1(C(c2nc(CC)oc2)=O)CC(NC(C2CCC(=O)N2)=O)CC2(CC2)C1 c1(C(=O)NCCCC(C)NC(C2CC3C=CC2C3)=O)cnn2cc(C#N)cnc12 N1(C(c2cn(C)nc2)=O)CC(CNC(=O)Cc2cccc(OCC(F)F)n2)C(O)C1 C1(C(N(CC(C)C#N)C)=O)CC2CC1CC2NC(=O)CCC(N)=O n1(CC(=O)NCC2C(CNC(c3c(N)cn(C)n3)=O)C2)cc([N+](=O)[O-])cn1 C=CC(CC)C(=O)NC(C1CCN(C(C2CC(OC(C)(C)C)C2)=O)CC1)C C1(C(=O)NCC(C(=O)NC2C=CCC2)N(C)C)(OC)CCOC1 c1(C(N2CCCC(CNC(C(C)c3ncco3)=O)C2)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NCC(C)CNC(c2ccnn2CC(F)F)=O)cccc(Br)c1 N1(C(C(CN(C(=O)CN(C2CCC2)C)C)(C)C)=O)CCCN(C)C(=O)C1 N1(C(c2cc(O)ccc2O)=O)CCN(C(c2cc(Cl)ncc2Cl)=O)C2(CCC2)C1 N1(C(C2(CC=C)CCOC2)=O)CCCC2(CCCN2C(c2cnn(C)c2C)=O)C1 C(C)(CCC(=O)NCC1CCN(C(c2csnc2Br)=O)CC1)SC Cc1cccc(C)c1C(c1nc(-c2nccs2)nn1CCc1ccc(Cl)cc1)C Cc1ccc(C(=O)NC2CC(C)CN(C(c3ccnc(C)c3C)=O)C2)cc1Cl C1(C(N(C2CCCOC2)CC)=O)COC(CNC(=O)CCCOC(C)=O)C1 C#Cc1c[nH]nc1C(=O)N(Cc1cncc(C(N)=O)c1)CC C(=O)(CS(=O)(=O)C(C)C)NCC1C(CNC(C2(OC)CCCCC2)=O)C1 c1(C(=O)NC2COC3CN(C(CCOC(C)C)=O)CC32)cnc(O)c2cncn12 CC(C)C(C)CC(=O)NCCC1CN(C(=O)C(O)CN(C)C)C1 n1(CCC)nc(C)c(C(=O)NC(CNC(c2n[nH]c(Cl)c2Cl)=O)CO)c1C C(=O)(C(CC(F)(F)F)NC(=O)Nc1cccnc1OC)OCCCC C(=O)(CC(F)(F)F)N(C(Cc1ccccc1Br)C(=O)NC1CC(CCF)C1)C n1(COC(c2ncnc3c2ncn3CCl)=O)c2ccccc2c(=O)c2ccccc12 C(CCN=c1ccnc(SC)[nH]1)NC(C(CC)F)=O c1(C(N2C3CC(NC(CCCC(C)=O)=O)(C3)C2)=O)cnc2c(F)cc(C)cc2c1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC2(CNC(c2csc(C)n2)=O)C1 C1CCS(=O)(=O)C(C)(C)C1.c1(C(C)C)nn(C)c(Cl)c1CNc1nnnn1C C1(C(N(CCOCCNC(c2c(CC)c[nH]n2)=O)C)=O)C(O)C(=O)N(C)C1C C12(C(N(C(C)C3CC3)C)=O)CC(NC(=O)CC3OCCO3)(C1)C2 c1(CC(=O)NCCN(C(=O)C2=NOCC2)CC)cc(C(F)(F)F)cc(Cl)n1 CCCCC(C)C(=O)N1CCC(O)C(NC(=O)CCC(=O)NC)C1 N1(C(C2(CC)CC2)=O)CC2(CCC(CNC(c3cc(C4CCC4)on3)=O)O2)C1 c1(C(C)NC(C(C2CCC2)OC)=O)cnccc1C n1(CC(=O)N(C(CC)CSc2ccccc2)C)cc(C=O)c(C)n1 CCC(CNC(=O)C(C)CN(C(=O)CSCC(N)=O)C)CC(C)C C(=O)(C1CCCc2nc[nH]c21)NCc1nc(O)cc(CNC(C(C=CC)O)=O)n1 Cc1nc2ncnn2c(C)c1C(=O)NCC1CN(C)CCN1C(c1ccon1)=O c1(CC(N2CCC(OCCNC(c3c[nH]nc3F)=O)C2)=O)ccc2c(c1)OCO2 C1(NC(c2ccnnc2)=O)CN(C(=O)Cc2ccc(Br)s2)CCC1CO C1(CCO)(NC(c2cnc(-c3ncccn3)s2)=O)CCNCC1 c12cccnc1N2.c1(C(N(CC(CN(C)C)O)C)=O)ccc(C(N)=O)cc1 C(c1ccc(F)cc1)=CC(N1CCC(N(C(CC=C(C)C)=O)CCO)C1)=O N1(C(C2C(=C)C2)=O)CC2(CC(NC(c3cn(C4CC4)nn3)=O)c3nccn32)C1 C(=O)(C(F)CC(CC)CC)NCC1C(CC)CN(C(=O)C=CC=C(C)C)CC1 c1(C(N2CC(C)N(C(=O)CCC3CCCCO3)CC2)=O)nncc2c1CCCC2 C(C(O)CC(=O)NC1COCC1CO)NC(Cc1n(C)nnc1)=O N1(C(c2ncc(C(C)C)cn2)=O)CCN2C(=O)C(C)CC2C1 S(=O)(=O)(c1ccc(NC2CCN3CCCC23)c(Br)c1)N(CC(OCC)OC)CC C(=O)(C1=CCC(NC(C2CC(C3CC3)C2)=O)C1)N(CC)CC1CCOCC1 c1(C(=O)NC(CC)CNC(=O)C(CO)NC(=O)C(F)(F)F)cc2sc(C)cc2s1 N1(C(C(CCC)NC(C2CNC(=O)C2)=O)=O)CCC(=O)N(C)CC1 N1(C2(C#N)CCN(C(=O)NCc3cccs3)C2)CCC2(CC1)CC2CCCO C(CC(=O)NOC1CCCC1)NC(C=CC(C)N(C)C)=O c1(CNC(C2COCCN(Cc3cc(O)ccc3Cl)C2)=O)ccc2c(c1)OCCO2 C(=O)(CS(=O)(=O)CC(=O)N1CCCC(NC(=O)CC2CCC2)CC1)OC N1(C(C2CC(CC)C2)=O)CCC(NC(=O)Cc2ccc(CO)cc2)C(O)C1 C(=O)(C1=CCSC1)N1C(C(=O)NCC(C)OCCO)CCC1 c1(C(C)C)cnn(C)c1C(=O)N(CC(O)CNC(=O)C(C)(C)CO)C C1(NC(C2CCOC2)=O)CCN(C(=O)C(F)C2CCC2)CC1C(N)=O c1(C(C)CC(=O)N(CCNC(C2COC2)=O)C2CC2)ccccc1Br C1(C(=O)OC)CCC(NC(=O)OC(C)(C)C)CN1C(=O)OCc1cn(C)nc1I N1(C(Cc2c(CC)con2)=O)CCC2(CC2NC(C2CCCC(F)C2)=O)C1 S(=O)(=O)(CC#Cc1ccccc1)NC(CCC1CC(C)OC1=O)=O C1(NC(Cc2ccn(C(C)C)n2)=O)CCC2CN(C(c3cc(Cl)cs3)=O)CC2C1 C1(C(=O)NC(C)(C)C)CC2CC2N1C(=O)N.C(CCC=O)OCCOCCOC N1(C(c2[nH]c(=NCC)sc2)=O)CCC2(CCCN(C(C3CCOC3(C)C)=O)C2)C1 CCN=C1NCCOCCN1.C(CCC)NOC n1(CC(=O)NC2CC(NC(Cc3cc(C)nn3C)=O)C(O)C2)nc(O)ccc1=O Cc1ccc(C)c(NCC(N2CCN(C(=O)CSC(F)(F)F)CC2CCO)=O)c1 C1(SCC(=O)NCC(O)CNC(C2(c3cnsc3)CC2)=O)CCCCO1 CN1CC2CCN(C(=O)CCN(C)C(c3ccc(C#N)o3)=O)C2C1 c1(C(N2CC(NC(C3(C#N)CC4CC4C3)=O)C2)=O)cc2c([nH]1)CCCC2 CC(O)(CC(=O)NC1C2CCC1N(C(c1[nH]nnc1C1CC1)=O)C2)C(F)(F)F c1(COC)ccoc1C(=O)NC(C)C(C)NC(=O)CCc1ncccn1 n1(CC)ncn(NC(=O)c2cc(C)n(CNC(=O)C=CCO)n2)c1=O Cc1nc(NC(C2(C)CN(C(c3cccc(O)c3)=O)C2)=O)c2sccc2n1 C(=O)(C1=CCCOC1)N1CC(C)C(CCNC(=O)CCc2cccs2)C1 N1(C(Cc2c(C)non2)=O)CCOCC1CNC(=O)CSc1cn[nH]c1 CCC(CC)(CC)C(c1ccccc1)N(S(=O)(=O)CC(=O)OC)C C1(NC(CCCOC(C)C)=O)CCN(C(=O)CCC2CC2(C)C)C1C N1(C(c2ccnnc2)=O)CCC2(CC1)CC(NCc1ccnc(O)c1)C2 N1(C(C(C)NC(=O)C(C)(C)C)=O)CCCC(NC(c2cnc(C#N)s2)=O)CC1 Cc1oc(Cl)nc1C(=O)NC1CCN(C(=O)CSC2CCOC2=O)C1C1CC1 Cc1cc(C#N)cnc1N1C2CCC1CC(CC(C)NC(=O)C=CBr)C2 C1(OC)CC(CCNC(=O)CC2CCC(=O)N2)N(C(=O)Cc2nc[nH]n2)C1 C(C)(CNC(=O)C(C1(O)CCCC1)F)(CC(C)C)NC(Cn1c(C)cc(C)n1)=O C12(C(N(CCC(=O)N(C)CC3(C#N)CC3)CCO)=O)CCC(CC1F)C2 C1(C(N(CC(C)C)C)=O)(NC(C23CC(C#N)(C2)C3)=O)CCCC1C C1(C(=O)NCC2CN(C(=O)CC(O)C3CCCC3)C2)C2CC3C(C2=O)C13 c1(C(N2CCN(C(CCC(C)C#N)=O)C(C(F)F)C2)=O)ccc2sncc2c1 C1(CC(=O)NC2CC(C)(CNC(c3cnc(C)[nH]3)=O)C2)CCCCC1O c1(C(=O)NCCN(C(C(C=CC)O)=O)CCOC)c(C)[nH]cc([N+](=O)[O-])c1=O C1(C(=O)NCC2CCC(NC(c3ccno3)=O)CC2)CN2CCN1CC2 C(=O)(CC(=O)NCC(C1CC1)NC(=O)Cc1cncn1C)OC N1(C(C2C(=C)CC2)=O)CCC2(CCCN(C(=O)CCc3cnc(OC)s3)C2)C1 Cc1ncccc1CCC(N1CC(F)CC1CNC(=O)CCc1cncs1)=O C(CC(C)(C)C)N(C(C(C)N(C)C(C1CCCOC1)=O)=O)CCN(C)C CC(C)CC(C(=O)NCc1cccs1)ONC(=O)C(C)(O)C1CCCC1 C1(CNC(C(CC)C)=O)CCOCC1C.C12(CC1)CC(=O)N2 C(=O)(N=c1cc(C)o[nH]1)NC(C(=O)Nc1cccc(C)c1)CC1CCCC1 N1(C(C(CCSC)NC(C2CC(F)(F)C2)=O)=O)CCn2nc(C)cc2C1 N1(C(c2nc(C)oc2C)=O)CCCC(C2CCN(C(=O)C(C)(C)CO)CC2)C1 CC(C)C(C)C(=O)NC1CCCCC1CNC(=O)C=CI c1(C(=O)NC(CC2OCCO2)CO)cncc2c1CCCC2 c1(NCC2(CNC(c3cc(C)c(C)s3)=O)CCC2)ncnc2cnn(C)c12 C1(NC(c2cnn(CCF)c2)=O)CN(C(c2cccc(F)c2)=O)CC12CC2 N1(C(c2cc(C)cc(OC)c2O)=O)CCCC2C1CCCN2C(C)=O C1N=C2NC3=C(C(=NCCOC14CCCC4)N2)COCC3.C(=O)(N(C)C)NCC C(=O)(C1CCCCc2ccccc21)N(CCCNC(C(CSC)(C)C)=O)C(C)C C1(NC(COC)=O)CC2(CCN(C(C3CCC4CCC34)=O)CC2)C1 c1(C(=O)NCC2CN(C(C(CC)C(C)C)=O)CC2O)cc2cccnn2c1 c1(NC(C(c2cccc(Cl)c2)CC)=O)ccc2c(c1)oc(=O)n2C C1(NC(CCCC#CC)=O)CN(C(c2cc(Cl)ccc2OC)=O)C2(CCC2)C1 Cc1ccc(C(=O)NCCNC(N2CCCC(Cc3ccc(O)cc3)C2)=O)cc1 C1(C(=O)OCCn2c(NC(C(=O)NC)=O)ccn2)CCC2COCCC2C1 c1(C(N2CC(CCC=C)(C(=O)NC(CC)C(C)(F)F)C2)=O)c[nH]c2cnccc12 N1(CC2CC3(CCC3O)C2)CCC2CN(C(=O)CC3(C#N)CCCCC3)C2C1 C(=O)(C(CC)CCOC)N1C(CCNC(C(CC)CC)=O)CCC1 C1(C(=O)NC2C(C#C)CCC2)CC2CC1CC2NC(c1ccn(C(C)C)n1)=O C1(CNC(=O)C=CC2CCCO2)COCCN(C(c2ccc(Cl)nc2)=O)C1 C1(NC(C2C3(CN(C(=O)OC(C)(C)C)C3)C2)=O)CCC2(CC1)CC2C#N c1(NC(C2(C)CCN2C(=O)Cn2cc([N+](=O)[O-])cn2)=O)cc(Cl)nnc1Cl C(=O)(C1CCOc2c(F)cccc21)N1CCCCC(NC(C(=O)NC2CC2)=O)C1 N1(C(C2CC(C)(CC)C2)=O)CC2CCCC(N(C(=O)CC(C)C(F)F)C)C2C1 N1(C(C2N(C)CCCC2)=O)CCC2(CC(NC(=O)C=CCF)C2)C1 C1(CCC)CC(C(=O)N(C)CC2CCCN2C(=O)C(CC)n2cncn2)CCO1 C1(CNC(C(CC)(C)CC)=O)CCN(C(=O)Cc2nncn2C)CC1(F)F C1(C(=O)NC2C(NC(c3ccn(C)c3)=O)COC2)CCOC1(C)C c1(OC)cc(CN(C2CCCN(C(C3CC(C)C3)=O)C2)CCO)nn1C C12(C(=O)NC3C4CC(NC(CC(C)SC)=O)CC43)CC1COC21CCC1 c1(C(N(C)CP(C)(C)=O)=O)coc2c1CN(C(=O)Cn1ncn(C)c1=O)C2 c1(COC)cc[nH]c1C(=O)NCCn1cc(C(=O)NCC2CC3(CC3)C2)nn1 C(=O)(C(O)CCCNC(c1c(OC)noc1C)=O)N(C(CC)C)CCO N1(CC)OCC(NC(=O)CC(F)(F)c2cscn2)C1=O.n12cc(nn1)COCC2 N1(C(CNC=O)=O)CCCCC1C1CCCN1C(C1CCC(=C(F)F)CC1)=O CCS(=O)(=O)c1cccc(C(=O)NC2CC(n3cc(C4(O)CCC4)nn3)C2)c1 C(CC(C(=O)NCCn1ncnn1)NC(=O)C(c1cnn(C)c1)=O)=CC CC1(C)CC1(C(=O)O)NC(=O)Cc1nc(-c2cccs2)cs1 c1(N(C2CCNC2)C(c2ccn(Cc3ccccc3)n2)=O)ccnc2ccnn12 N1(C(CCCCCSC)=O)CC2CCCC(C1)N2C(=O)C1CCCc2cncn21 c1(C(=O)NCC(CNC(c2ncccn2)=O)F)c(Cl)sc2nnsc12 C1(C2CCC2)(C(=O)NCC2(C)CCCN(C(C(C3CCC3)OC)=O)C2)CC1(F)F C1(CCC)CC(C(N2CCC(OCCNC(=O)COC(C)CC)CC2)=O)CCO1 c1(CC)conc1CC(=O)NC(CNC(=O)CCc1ncnn1C)C1CC1 c1(C(N2C3C(NC(c4ccn(C(C)C)n4)=O)CC(C3)C2)=O)cnn2c1NCCC2 [N-]=[N+]=NC1CN(C(=O)CCn2cc(Cl)cn2)CC1NC(=O)CNc1ccccn1 c1(C(=O)NC(C(=O)NC(Cc2cc(C)[nH]n2)C)C2(O)CCC2)cccn(C)c1=O CCCCC(CC)C(=O)NCC1(NC(=O)C(C(C)(C)C)C2CCCC2)CCCC1 C1(N(C(C(CN(CC)CC)F)=O)CC2CC2)CCN(C(=O)C(C)C(F)F)CC1 C(=O)(C(F)CCC(C)C)N1CCCC(C(C(=O)Nc2c(C)nn(C)c2)C)C1 C1(c2ccc(CN=c3c(C)cnn[nH]3)cc2)CC(C2CCC2)=NO1 c1(OC)ccc(C(=O)NCCNC(C2CCN(C)C(=O)C2)=O)c(Cl)c1 c1(C(=O)NC2CC(F)(CNC(C3CCS3(=O)=O)=O)C2)c[nH]c2cc(F)ccc12 N1(C(C(CCC)O)=O)CC(C2CCCCN(C(C3CCC(=O)N3CC)=O)C2)C1 C(CN=c1[nH]c(=NCc2ccc(CO)c(F)c2)[nH]c2c1COCC2)(C1CC1)OC C1(NC(C(C)NC(c2ccco2)=O)=O)CCC(NC(=O)C(C)(F)F)C1 c1(C(N2CC(NC(C3(C=C)CCC3)=O)C(OC)C2)=O)c(Cl)nc2cc(Cl)ccn12 N1(C(=O)CC2C=CCC2)CC2CCN(C(c3c[nH]cc(F)c3=O)=O)C2C1 N1(C(=O)NC2CCN(C3CCN(C)C(=O)C3)CC2)CCOCC12COCCN(C)C2 CC(C)CC(C)C(=O)N1CCCC(C)(CNC(c2cc(C(C)C)cc(O)c2)=O)C1 CCC(CC(=O)N1CCC2C(NC(c3cccc(OC)n3)=O)C12)SC C1(C)(CNC(C2CC(NC(C3C(COC)CC3)=O)C2)=O)CCCO1 C1(C(=O)NCC2CN(C(=O)C3=COCC3)CC2(F)F)(OC)CCCCCC1 c1(C(=O)NCc2ccc(CNC(C(C)CN(C)C)=O)cc2)sccc1S(C)(=O)=O c1(C(N2CCN(C(C(CCC)NC(C)=O)=O)C(CO)C2)=O)cnn2ccn(C)c12 Cc1cnc(N(CC(C)NC(=O)CC2C(C)(C)C2(C)C)C)nc1S(C)(=O)=O C(=O)(C(C)(C)C(C)O)N1CC(OC)C(NC(=O)Cc2ncccc2C)C1 c1(CNC(C(Cn2ccnn2)NC(C2CC(CCC)C2)=O)=O)ccncc1C C1(NC(=O)NC2C(CCC(=O)OC)CCC2)CC(=O)N(c2ccccc2OC)C1 CC1CNc2c(C(=O)NCCc3nc(-c4ccccc4)ns3)cnn2C1 N1(C(CC=CCC)=O)CC2(CCCC2NC(c2ncn(C)c2C)=O)C1 n1(CCOC)cc(C(=O)NC2CCC2NC(c2ncc(C(F)F)s2)=O)cn1 N1(CCNC(c2c(CC)scn2)=O)CCCN(C(=O)CCC2CCOC2)CC1 N1(C(C2C3CCN2CC3)=O)CCCC(C(C)NC(c2nc(COCC)sc2)=O)C1 c1(C(=O)NCc2c(F)cc(C)c(F)c2)c(F)cncc1C1=CCN(C)CC1 C1(CC(=O)N(C(CN(C(c2ncn(CC)c2)=O)C)C)C)CC(C)(C)CCO1 C=C=C(C)CC(=O)N1CCC(C2CCCN2)C1.C12CSCN1C1CN(C1)C2=O N1(C(C(COCC)C)=O)CC(NC(c2cc(C)sc2C)=O)C(O)C1 N1(C(CCCCC#N)=O)CCC2(CC1)CC2(CO)CNC(C1CCCC(O)C1)=O CCC(CCC(=O)N1CCN(C(=O)CCN(C2CC2)CC)C(CO)C1)OC C1(NC(C2(C)CC2)=O)CCC2(CCN(C(=O)CCc3ncc[nH]3)CC2)C1 c1(C(N2CC(CC(=O)NC(C(=O)NC(C)C)C)OCC2)=O)ncc(F)cc1F C(=O)(CC1=CCCCC1)N1C(c2nnc(C3(C)C(C)CCCC3)o2)CC(F)(F)C1 C1(C(=O)NC(CCC)C(F)(F)F)C(C2CC2)CCN1C(=O)CN1CCNC(=O)C1 C1(N(C)C)(CNC(=O)NCC(c2nccs2)OCC)CCc2ccccc2O1 c1(C(=O)NCCOCCNC(C(C(=O)OC)C)=O)c(OC(C)C)ccnc1F c1(NCc2ccc(CC)cc2)cccc(S(=O)(=O)N(C)C)c1.C(C)(=O)O N1(C(C(Cc2ccccc2)OC)=O)CCCC(CNC(c2cc(CF)on2)=O)C1 C1(CN(C(C(C(=O)OC)SC)=O)C)CN(C(=O)C=C(C)C(C)C)CC12CC2 C12(C(=O)OC)CC(C(=O)NCC3CN(C(=O)C(c4cnccn4)C)C3)(C1)C2 N1(C(=O)OC)CCC(C(C)C(N2CCN(C(C3CCC3)=O)CC2)=O)CC1.C1CN1 C(=O)(C(O)CC(C)(C)C)N1CC(c2c(CNC(CCCCCOC)=O)nco2)C1 Cc1cc(C(=O)NC(C2CN(C(c3cc(C)[nH]c3C)=O)C2)C)n(C)n1 CCC(C(=O)NCC(F)CNC(=O)C=CSC)OC1CCCC1 CCCC(CN(C(=O)COC(=O)CC(C(C)C)c1nc[nH]n1)C(=O)CO)CCO N1(C(C2C(C)C2)=O)CC(C2CC2)(C(=O)NCC2CC(C#N)C2)C1 C1(NC(CSC)=O)CCC2(CCCN2C(=O)C(C(C)C)c2ccc(Cl)cc2)CC1 CC(COCc1ccco1)N=c1ccnc(NC2CCCC(C)(C)C2)[nH]1 C#Cc1cccc(OCC(=O)NCC=CCNC(=O)C(N2CCCCCC2)C)c1 CCC(C(=O)N1CCC(C(C)(C)NC(=O)Cc2sc(C3CC3)nc2C)C1)C(C)C C1(NC(=O)CCSC(F)(F)F)COCCN(C(=O)CC2CC3CC3C2)C1 N1(C(C(c2ccc(F)cc2)C)=O)CCC(C)C(NC(=O)Cc2ccc(F)cn2)C1 C=CC(C)CCNC(c1occc1CNC(=O)C(c1cnn(C)c1)O)=O N1(C(CN2CC(C)(C)C2)=O)CC2(CCC(CNC(C3CC=CCO3)=O)O2)C1 c1(N2C(c3ccccc3)C3CC3C2)ccc2nncn2n1 N1(C(CC(C=C)C)=O)C2CCC1(CNC(=O)C(C)CCCOC)CC2 c1(C(COC(=O)C(O)CN2CCCC2)NC(C2CSC2)=O)cc(F)ccc1Cl C1(NC(c2c(C)nn[nH]2)=O)CC(NC(=O)CSCCC(F)(F)F)C1(C)C CN=c1ccc(C(N2CCCC2C(C)NC(=O)C(=O)NOC)=O)c[nH]1 C12(NC(C=NOC)=O)CCC(CNC(C3CC3COC)=O)(CC1)OC2 c1(OC(C(=O)NCC(CC)NC(=O)CSC)(F)F)cc(Cl)cc(Cl)c1 c1(C(N(CCCCN(C(C2N(CC)CC2)=O)C)C)=O)ccc(S(=O)CC#N)cc1 C(=O)(C1=NNC(=O)CC1)NCC1(CNC(c2cccc(NC)n2)=O)CC12CCC2 c1(CN(C(C(CC)C)=O)C)cccc(CNC(C2(c3cc[nH]n3)CC2)=O)c1 CC(C)C1C(=O)N1.c1(C(COCCNC(=O)OC(C)(C)C)O)ccccc1.C=O c1(CSC2CCC(CC)CC2)cc(C#N)c2c(n1)CCCC2 C=CC1CCCN(C(c2cnccc2Br)=O)C1.c1(C(=O)OCC)cc[nH]c1 N1(C(C2(CNC(C3CCC(CC)O3)=O)CCC2)=O)CC2(CCCC2)C1 n1(CCC(=O)OC)cc(CC2(O)CN(C(C3(CCS(N)(=O)=O)CCC3)=O)C2)nn1 N1(C(C2CCC(C)(CC)O2)=O)CC(C)N(C(=O)Cc2cnn(C)c2C)C(C)C1 n1(CC)nc(C(=O)Nc2ccc(N3CCCC3)c(Br)c2)c2c1CCOC2 C(=O)(CC(C)(C)C#N)NC(C)C=CC(=O)NCc1ncccn1 c1(CC)cc(Cl)ccc1C(=O)NCc1ccnc(C(=O)O)c1 C(=O)(CS(C)(=O)=O)NC(C(=O)N1CC(CC(=O)OC)C1)COC C1(C(=O)NCCC2(CNC(C(CC)(C)C)=O)CC2)Cc2cccnc2C1 Cc1nc2c(s1)CCCC2C(=O)NCC1CN(C(C2(CO)COC2)=O)CCCO1 CCCC(C)C(CC)(c1nnnn1C1CCCCC1)NC1CCC(C)CC1 C1(C)(CNC(c2cn(CCC)nn2)=O)CCN(C(=O)CC(=O)N(C)C)CC1 c1(COCCNC(C(c2ccc(Cl)s2)N(CCC(C)C)C2CC2)=O)ccccc1 C1(C)(C)CC(=O)OCc2cn1nn2.C1(NC(=O)OC(C)(C)C)CC(CCO)C1 C1(CC)CCN(C(=O)CSCCF)C1NC(=O)COC C1(NC(c2c(C)cccn2)=O)CN(C(C2Cc3nnc(C)n3C2)=O)CC(F)(F)C1 C1(CC)CC(O)CN1C(C1CC1C(C)NC(=O)Cn1[nH]cnc1=N)=O C(=O)(C1=CCN(C)C1)NCCC(C)NC(c1cnc(CC)o1)=O CC1=C(C(=O)N2CCCC(NC(=O)C=C3CCN(C)CC3)C(F)C2)CCCO1 CC1CN(C(c2nncn2C2CC2)=O)CC1CNC(=O)C(F)=CC1CC1 C1(N(C(C(C)Nc2ccccc2F)=O)C)CCCN(C(=O)C2=COCCO2)CC1 N1(C(C(COCC)NC(=O)CC(O)C2CCCC2)=O)CCC2C(=O)NCC2C1 N(C1CCCc2c(Cl)ccc(Cl)c21)C(N1CCC2CNC1C2)=O N1(C(C2C3CN(C)CC32)=O)CCC(NC(=O)Cc2cnc[nH]2)C(F)C1 N12CCN(CC1)C2=O.c1(C(C)NC2CNCC2F)ncccn1 C1(C(C(=O)OC2C(C(=O)NC)C2)OC(C)(C)C)CCCCC1 C=CCC(CC(C)C)C(=O)N1CCCC(CC)(NC(=O)C(O)CC2CCCC2)C1 n1(C(CC)CC)nc(C)cc1C(N1CCCC1CNC(=O)CN1CCCC1C)=O c1(N2Cc3c(-c4c(OC)c(C)ccc4)n[nH]c3CC2)nc(C)nc2cccc(Br)c12 c1(CC(N2C(CCNC(CCC3C(C)C3)=O)CCC2)=O)ccc2c(c1)CCCC2 c1(C(CNC(c2n[nH]cc2Br)=O)NC(CC=C=C)=O)ccccc1F N1(C(C2CC(=O)NC2)=O)CCCC2(C1)CN(C(c1cc(Cl)nc(Cl)c1)=O)CCO2 C(=O)(C1CC=Cc2ccccc21)N1CCCC(F)(CNC(=O)Cc2cnns2)C1 c1(C(=O)NCC2(CC(=O)NC3(c4nccs4)CC3)CC2)cccn2ccnc12 c1(CC)oc(C(=O)O)cc1S(=O)(=O)NC(C)C(=O)Nc1ccc(F)cc1 C1(CC(CNC(C2(C(=O)OCC)CNC2)=O)O)(C(F)(F)F)CCCCC1 C1(C(N2CCN(CCN(C)C(c3c[nH]c(=N)s3)=O)CC2)=O)(OC)CC2CCC1C2 CC(CC(=O)NC1(CF)CCN(C(=O)CN2CCCCC2=O)C1)C(F)(F)F c1(CC)ccsc1C(=O)NC(C)CN(C(=O)CCc1ncc[nH]1)CC C1(C(C)NC(C2C(C)C2C)=O)CN(C(c2sccc2Cl)=O)CCO1 c1(CCCN2C(C)(C(=O)O)CCC2)ccc(F)c(F)c1 CC(O)CC(C)N=c1ccnc(NCCC23CCCN2CCC3)[nH]1 N1(C(C2OCCN(C(c3cc(OC)c(Cl)nc3)=O)C2)=O)Cc2ccc(F)cc2C1 N1(C(C(C2CC2)OCC)=O)CCOC2(C1)CN(C(C1CC1C(C)(F)F)=O)C2.C1(C)CC1 N1(C(c2c(CC)ccs2)=O)CCCC(NC(C23CC(C2)C(C)(C)O3)=O)CC1 C12(C(N3CCC(O)(CC)C3)=O)CCC(CC1)N(C(C1(NC(N)=O)CC1)=O)C2 O=C(CC1NC(=O)c2ccccc21)NCC1(NC(C2CCC3C2C3(F)F)=O)CC1 C1(C(=O)NCCC(=O)NC)CCN(C(C2CC(C(C)C)C2)=O)CC1 C#CCC(CC(F)(F)F)C(=O)NCC1COC(C(F)(F)F)CN1 CC1(C)CC(CNC(c2cnccn2)=O)CN(C(=O)CCCS(N)(=O)=O)C1 Cc1cc(C(=O)NC2CC2NC(c2ccn(C)c2C)=O)cc(S(N)(=O)=O)c1C c1(C(NCP(C)(C)=O)C)cc(OCNC2CC2)n(C)n1 CCN=c1[nH]c(C)c(C(N2CCCC2C(C)NC(C2CCCCC2(C)C)=O)=O)s1 N1(C(C2N(CC)CCCC2)=O)CCc2c(CNC(=O)C3=CCC3)cccc2C1 c1(OC)ccc(C(C)C(=O)NC(CNC(c2cn(C)cn2)=O)CO)cc1OC Cc1ccc2c(cnn2C)c1-c1csc(NC(C2CC23CCOC3)=O)n1 c1(CN(C(c2ccc(F)cc2)C(=O)NC2CC(F)(F)C2)C)cc(O)cc(Br)c1 CC(C)CC(=O)NCC(CC1CCNCC1)CO C1(c2n(CC(F)F)ncc2)NC(=S)N(C2CC2)C2=C1C(=O)NC2c1ccccc1 Cc1cccnc1C=CC(N1CC(n2ccnn2)C(C)C1)=O C(=O)(C(C(C)NC(c1cc(C)ccc1C)=O)C(C)C)NCCN1CCC=C(C)C1 c1(CC(=O)N(C2C3CN(C(CC4CN(C)C4)=O)CC32)C)c[nH]c2cc(F)ccc12 c1(C(=O)NCC2N(C(C=CC=CC)=O)CCCCC2)cc2cccnc2o1 N1(C(C(N)=O)=O)CC=CC(NC(C2(O)CCC2)=O)C1 c1(-c2cc(OC)cc(COC)c2)ccc2nnc(C(N3CCOCC3C)=O)n2c1 c1(C(=O)NCC(C)(CO)NC(C2C(C)CC2)=O)cc(C(C)(C)C)n(C)n1 C(CO)(CCCCNC(=O)C(F)=C1CCCC1)NC(=O)CCC1CCC(O)CC1 C(CC(C)C)(C(=O)N(CC(O)CO)C)N(C(C(C)=CC(F)(F)F)=O)C c1(C(CNC(CS)=O)NC(c2cnn(C)c2)=O)ccc(C)cc1.C1(CSC)CC1 CC(C)CC(O)C(=O)NCC(C1CCC1)NC(=O)CC1(O)CCCN(C)C1 C1(C(=O)NC23CC(NC(c4cnc(C)s4)=O)(C2)C3)CCCN2CCCCC12 C(=O)(C(O)C1=CCCCC1)NCC(CNC(c1ccn(CC(C)C)n1)=O)CO C(=O)(CC(C(F)(F)F)NC(=O)C(C1CCCCC1)F)NC1(CC=C)CCCCC1 c1(OC)cccc(F)c1CNC(=O)CC1CN(Cc2ncccc2OC)C1 c1(C(=O)NCC2CC(OC)CN2C(C2OCCC2C(C)C)=O)cc2occc2[nH]1 C1(CC(=O)NCC(CC)(C)C)CN(C(=O)C(C(C)C)C2CCC2)C(C)(C)C1 c1(C(=O)NCC(CC=C)NC(c2c(Cl)cnn2C)=O)ccccc1CC C(=O)(C#CC(C)(C)CNC(c1cnc(N)cn1)=O)NCC(C(=O)OC)OC C1(NC(c2cccc(F)c2O)=O)CCC2CCN(C(=O)C(F)(F)CO)C1C2 C(=O)(CC(C)(C)CCC)NC(C1(O)CCN(C(C2(CC=C)CCOC2)=O)CC1)C CC(C)CC(O)C(C)C(=O)N1CC2(CCC2NC(=O)Cc2cc(Cl)ccc2Cl)C1 N1(C(c2c(CC)c[nH]n2)=O)CC(CNC(=O)C(C#N)C(C)(C)C)C2(CCC2)C1 C1(C)(CC(=O)NCCC=CCCC)CCN1C(c1cnc(C)o1)=O C1(OC(C2CCC2(F)F)=O)CC(=O)N(CCOC(=O)C2CC2)C1 N1(C(CCC2N(C(c3c(C)cc[nH]3)=O)CCCC2)=O)CCOCC(O)C1 C1(NC(CN(C)C)=O)CN(C(=O)CCC2CCOC2)CC1Cc1ccccc1 Cc1cc(CN=c2[nH]cc(CCNC(c3nccs3)=O)s2)cc(Br)c1 CC1(C)CC(NC(c2c(F)cccc2Cl)=O)CN(C(=O)C(C)(O)C2CCC2)C1 Cc1cc(-c2ccc(O)c(Cl)c2)c(O)c(C=O)c1 N1(C(C(N2C(CC)Cc3ccccc3C2)=O)=O)Cc2cc(F)ccc2CC1C c1(N(C)C)nc(Cl)c(C(N2CCOCC2CNC(=O)CCc2cnc(O)[nH]2)=O)s1 C=CCC(C)(C)CC(=O)NCC(C)CN(C)C(C12COC(CO)(C1)C2)=O N1(C(C(=O)NCC)=O)CCCC(CCNC(=O)CN(c2ccncc2)C)C1 N1(C(CC(CC(C)C)CN)=O)CCC(OCCO)S(=O)(=O)CC1 CC1CC(C(=O)NC2CCC(NC(c3cc(O)nn3C)=O)C2)CCN1C C1(CCNC(CSCC(C)C)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1(F)F c1(N(C(C)C)C)ccccc1C(N1CCC(N(C)Cc2scnc2Cl)C1)=O C1(C(=O)OC)(SC)CN(C(C2CN(C(C)=O)C2)=O)C1.C1(Cc2cc[nH]n2)C(=O)N1 CC1(C)C=C(C(=O)NC2CCN(C(=O)CCCCCc3cccs3)C23CC3)C1 C=CC1CCCN(C(=O)C(CC(N)=O)NC(=O)C(CC)=CC)C1 C12(C(=O)NCC(=C)CCNC(C3(CO)CCCCC3)=O)CCCN1CC(OC)C2 C1(CC)CN(C(c2cnc(Cl)c(C)c2)=O)CCN1C(c1cc(I)ccc1C)=O C1(C(=O)O)COCCN1C(C12CC1CN(C(=O)CCc1ncccc1F)C2)=O C1(CC)CCC(C(=O)N(C)CC2COCCN2C(C2CCOC2)=O)CC1 c1(C(N2C(C)(CNC(=O)CN3CCOCC3)CCC2)=O)cc2ccccc2s1 c1(CC(=O)NC2(CNC(c3c(CC)onc3)=O)CC2)cn2cc(F)ccc2n1 CCCCC(O)C(C)C(=O)NC1CC(CC(N2CCC2(C)C(=O)NC)=O)C1 c1(C(N2C(CNC(C(C)NC(=O)CC(C)(C)C)=O)CC2)=O)cnn2c1OCC2 C(c1c(Cl)cccc1Cl)=C(C)C(=O)N(CCCNC(=O)CCc1cn(C)nn1)C C1(C(=O)NCC2C(NC(c3cccc4c3COC4)=O)C2)CCc2ccccc2C1 c1(-c2cncc(OC)c2)ccc(F)c(COCc2n[nH]cc2C(F)(F)F)c1 c1(CNc2ccc(C(C(F)F)F)cn2)cccc2ncnn12 N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(=O)C=CCN2CCOCC2)C(C)(C)C1 N1(C(C2C(C(=O)OC)CC2)=O)C(C(N2CCC(O)(COC)C2)=O)CCC12CC2 c1(NC(CC(c2cn(C)nc2)NC(=O)C=CC(F)(F)F)=O)cccc(C#N)c1 c1(-n2cc(C(C)NC(c3c(C)nc(Br)s3)=O)nn2)cccc2ncccc12 c1(C(N(CCCN(C(CC2C(C)C2)=O)C)C)=O)cn2c(n1)COCC2 N1(C(C2CN(C(C)=O)C2)=O)CCOCC(C(=O)Nc2ccc(C)c(O)c2)C1 C1(C)(C(N2C(CNC(C(C)=NOCC#N)=O)CCCC2)=O)CCN(C)C1=O c1(CNC(C2(CNC(C(C)OC)=O)CC2)=O)ncn(C(C)C)n1 c1(C(=O)NC2C3CC(CNC(CC(=C)C)=O)(C3)OC2)ccc2c(c1)CC(C)O2 C1(CNC(C(CC(=O)OC)C)=O)CC2CCC1N(C(=O)CC1COCC(C)O1)C2 Cc1[nH]c2ccccc2c1C(=O)NCC(CNC(C1CCS(=O)(=O)C1)=O)CO C1(CNC(CSCC=C)=O)CN(C(=O)COCC2CCCCO2)CC2(CCC2)O1 c1(C(=O)NC2C(NC(C3CC(C)C3)=O)CCCC2)cc(C2CC2)nc2ccnn12 C1(C(N(CCCNC(c2ccc(C)cn2)=O)CCO)=O)CCOC(C)(C)C1 c1(C(=O)NCC(=CCCC)C)c(CCCC)nn2c1CCC2 c1(C(N2CCCC(C(C)(O)CNC(=O)C(N)=O)C2)=O)cc2ccc(F)cc2o1 C1(NC(C(C=C=C)C)=O)CN(C(c2cccnc2SC(F)F)=O)CC12CC2 c1(CCC(=O)NCCCN(C2CCCC2)C(C2(CSC)CCC2)=O)ccc(F)cc1 C1(CNC(C(F)=CCC)=O)CC(C)N(C(c2cncnc2C)=O)C1 C1(NC(=O)CC2CCC3CC23)CC2(C1)CN(C(=O)C=Cc1cncc(O)c1)C2 CN1CCC(CC(N2CCC(CNC(=O)CN3CC(C)(C)C3)C2)=O)C1 c1(C(=O)NCCOCCNC(C(CC)(C)CO)=O)n[nH]c2ccc(C)cc12 N1(C(C(C(C)C)F)=O)CCC2(CCCC2CNC(=O)C=C2CCCC2)CC1 C(=O)(CC(O)C(C)(C)C)N1CCC(COC)(NC(C2OCCN(C)C2=O)=O)C1 Cn1c(O)nc2c(S(=O)(=O)NC3CCCCC3C)cccc12 Cc1nnc(NC2CCCCN(C(=O)C(C)CC3CCC3)C2)c(C#N)c1C c1(C(C(=O)NCCSC)N(CC#CC)C)ccc(F)c2c1CCC2 C1(C(=O)NC(C)CCCNC(=O)COCC(C)(C)C)CC2(C1)NC(=O)NC2=O CCCCCCC(F)C(=O)NC1CC(CCNC(=O)Cc2nonc2C)C1 C(c1c(F)cccc1F)=CC(N1C2C(N(C)C(c3ccoc3)=O)CC(C2)C1)=O C1(CC(=O)NC(CCC)CO)CCCN(C(=O)CN2CCNC2=O)C1 O=C(CNC1CC12CCCCC2)NNC(=O)N1CCC(c2ccccc2)CC1 O=C(CCC(F)(F)F)NC(C1(O)CCCCC1)C(=O)NC1CCCSC1 Cc1cc(Br)cc(CN2CCC(N(C)C(c3cnc(O)cc3O)=O)C2)c1O C1(NC(=O)Nc2c(C)n(CCN(C)C)nc2)CC(C(=O)OC(C)(C)C)C12CCC2 C1(C(=O)NC2(CC=C)CN(C(=O)Cc3n[nH]c(=NC)s3)C2)CCN(C)C(=O)C1 C1(C(=O)NCC(CC)N2CCCC2)CCCCCN1C(=O)C(CC1CC1)OCOC c1(C(=O)NCCOC2CCN(C(CCC3C(C)C3)=O)C2)ccc(C)cn1.C(CF)O N1(C(C2C(C)OCC2)=O)CC2(C1)C(NC(=O)Cc1cccc(F)c1)CCS2(=O)=O N#CC1(C(=O)NC(c2ccc(C#N)cc2)CC2CCCCC2)CCCCCC1 C1(CC=C)(NC(C2CC2(C)C(C)C)=O)CCN(C(=O)CSc2nncn2C)C1 c1(CC)nn(C)cc1CNC(c1ccccc1)CCc1c(C)noc1C C=CC1(C(=O)NC23CC4CC(CC2C4)C3)CCN(C(=O)C#CC2CC2)CC1 c1(-c2nnc(N3C(C)COCC3)n2CC2CCOC2)nnc2n1CCNC2=O c1(C(=O)NC2CCN(C(C3(C)CC=CC3)=O)C2)ccc(-c2cc(O)ns2)cc1 c1(CC(N2CCC(N(C)C(C3CCN3S(C)(=O)=O)=O)C2)=O)cc(F)cc(Cl)c1 c1(C(N2C(CNC(C(CC)(C)OC)=O)CCCC2)=O)cc(C)c(C)cc1Cl c1(C(=O)NC2CC(C)N(C(=O)CCc3ccn(C)c3)CC2)cnn2ncccc12 C1(CNC(C(N2C(C(N)=O)CC(OCC)C2)=O)=O)CCC2(CCOCC2)CN1 Cc1ccc(C(=O)NC(C)CN(C(=O)CCC(=O)c2cccnc2)C)cc1CO C1(C(N2CCC(Nc3ncnc(O)c3Br)C2)=O)CC2(C1)CS(=O)(=O)C2 Cc1scc(C(N2CCC(CF)(NC(c3cccc(C(C)C)c3)=O)C2)=O)c1C C12(NC(COCC(C)C)=O)CC(CNC(=O)COCC(c3ccccc3)C)(C1)C2 C(=O)(CCCN(C)N=O)NCCCN(C(=O)Cc1cnn(C)c1)CCC N1(C(CCSC2(C)CCC2)=O)CC(NC(=O)Cn2ccnn2)CC12CCOCC2 Cc1ccc(CC(=O)NCC(C2CCN(C(=O)CSc3nncs3)CC2)F)cn1 C1(C(N(CC(C)C)CC)=O)CCN(C(=O)CCOCCN(C)C)C1C Cc1ccc(C=CC(=O)NC2CCCC2NC(c2cc(Br)no2)=O)cc1C c1(C(=O)NC2CCCC(CNC(C3(Br)CC3)=O)C2)coc2c1COC2 C1(CNC(C(C)SC)=O)N(C(c2cccc3oncc23)=O)CCCC1(C)C c1(N(CCN)CC)ccc(S(=O)(=O)N(C)C)cc1.C1(C(C(CC)=O)=O)CC(CSC)C1 N1(C(c2c(C)cncc2)=O)CCC2CCC(C1)N2C(=O)CN1CC2CC2C1 CCCC(F)(F)C(=O)NCC(O)CN(C)C.c12cc(on1)C(=O)N2 c1(CNC(C(c2ccccc2)OC(C)C)=O)nc(C2CC2)sc1Br c1(CN(C(Cn2ccc(C)n2)C=O)C(C)(C)C)ccc2c(c1)OCCO2 c1(C(N2CC(NC(C3CCCO3)=O)CC(C)(C)C2)=O)ccc2c(O)n[nH]c2c1 C1(=CCNC(C(C)OCCC=C)=O)CN(C(c2cnc[nH]2)C2CC2)CCS1(=O)=O C=CCC(C)(C)CC(=O)NC1CCN(C(c2ccc(CC3CC3)cc2)=O)CC1F Cc1ccc(C(=O)NCC2CCC2c2ccccc2)nc1C1CC1 c1(OC)ccc(C(=O)NC2CC2CNC(=O)CN2CCC(C)C2)cc1O c1(C(N2C(CNC(c3c(C)cn(C)n3)=O)CC3(CC3)C2)=O)ccc2cccnn12 c1(C(N2CC3C(CC(=O)OC)(CC3)C2)=O)cc(Cl)nc(Br)c1N CCC(CC)(CN=c1nc(C(C)C)[nH]s1)NC(=O)C(C)Oc1ccccc1 C1(NC(c2c(C)nc(CC)o2)=O)CN(C(c2ccc(C)cc2O)=O)C2(CCC2)C1 c1(C(=O)NCCN2CCCC(CO)C2)cc2ccccc2c(I)c1O Cc1cc(C(N2CCN(C(c3c(C)cnn3C)=O)CC2C)=O)c(O)c(C)c1 C(=O)(C1=CC2(CN(C(C3CCC(F)C3)=O)C2)OC1)NCCc1n(C)cnc1 C(=O)(CC(C)CC(C)C)NCCC1N(C(CCCc2nnc(C)n2C)=O)CCC1 C(C(CCC)C(=O)OC)c1c(NC(C(=C)C(=O)OCC)=O)cccc1 N1(C(c2c(OC)ccc(OC)c2)=O)CC(C)CN(C(=O)CSCCSC)CC1C c1(CC(=O)NC2(C)CC(NC(c3cnc(Cl)c(N)c3)=O)C2)ccc([N+](=O)[O-])cc1 C1(NC(c2c(N)non2)=O)CC2CCC(C1)N2C(C12CC(C(F)F)(C1)C2)=O N1(C(c2c(C)sc(O)n2)=O)CCCN(C(c2cc(N)cc(O)c2)=O)CC1 N1(C(C(C)CCN(C)C)=O)CCOCC1C1CCCO1 N1(C(C=CCC)=O)CCC(C(=O)OC)C1CCSC.C1(CCOC)(NC)CCC1 c1(C(=O)NCCN(C(C2CC2(c2ccccc2)F)=O)CC)cc(C(C)C)nn1C CC1=C(C(=O)NC2CCN(C(=O)Cc3ccc(F)cn3)C(C)C2)CCS1(=O)=O C1(S(C)(=O)=O)(C(=O)NC2CC3CN(C(Cc4n(C)ncc4)=O)CC3C2)CCCC1 c1(NC(C2C3(CN(C(Cc4ccc(C)nc4)=O)C3)C2)=O)c(F)cc(Br)cc1Br C(=O)(C1CCc2nnc(C)n21)N1C(CC)CN(C(C2(CN(C)C)CC2)=O)CC1 c1(NC(C)C)cncc(C(=O)NCC2(C)CCN(C(c3cc(CF)on3)=O)C2)c1 c1(C(=O)NCCCCCNC(COC(CC)C)=O)cncc(C(C)=O)c1 O=C(CC(C(F)(F)F)N1CCOCC1)OCC(c1cc2ncccc2[nH]1)=O c1(SC)ccccc1Cl.C12CCN(C1)C(=O)C(Cc1ccsc1)N(C)CC(=O)N2 C12(C(N3CC(C)(NC(C4(C(=O)OC(C)(C)C)CC4)=O)C3)=O)CC=CCN1CCC2 CC1(C)CCCC(C(=O)NC2CC(C(N3CC(F)(F)CC3C(N)=O)=O)C2)C1 C1(NC(C2CC(OC)C2)=O)CN(C(=O)CC(C)c2ccccc2)CC12CC2 Cc1cc(C(N2CCC(C(C)NC(=O)COCC3CC3)C2)=O)ccc1O C(=O)(C(O)C(C)(C)CC)NC(CN1CCN(C(C(CC=C)(F)F)=O)CC1)C N1(C(C)C)CCc2c(NC(=O)CC(F)(F)c3ccccc3)cccc2C1 c1(C(=O)NCC(C)NC(c2[nH]cc(C)c2)=O)cccc(C#N)c1Br C1(C(C)NC(C(COC)O)=O)CN(C(=O)Cn2cnnc2O)CCO1 c1(C(N2CC(COC)(CNC(=O)C(CO)N(C)C)C2)=O)cc2n(n1)CCCO2 CC1(C(=O)NCC2(CNC(c3cc(Cl)cs3)=O)CC(F)(F)C2)COC(=O)C1 CCC(CC(=O)NC(c1n[nH]c(C)n1)C(=O)NC1CC(O)C1OC)OC C=CC1OCCCC1C(=O)N(CCCN(C)C(C1CN(C)C(=O)N1)=O)C Cc1sc(C(=O)NCC2COCC2NC(c2cc(O)n(C)n2)=O)nc1O N#Cc1cccc(CNC(=O)NCC2CC2C2CCOCC2)c1Br CCCC(O)CCN=c1ccnc(NC(c2nccn2CC)C)[nH]1 N1(C(C(CN(C(c2c(CC)cncc2)=O)C2CC2)C)=O)CCC2(CC1)CC2 Cc1cc(=O)n(C)nc1C(N1CC(Oc2ccc(Cl)c(F)c2)C1)=O C12(C(=O)NCCOC(C)=O)CC(C)(CN1C(=O)CCCC1CC1)C2 C1(NC(CCc2cc(C)[nH]n2)=O)CN(C(C2CC3CCC2CC3)=O)CC12CCC2 c1(C(C)C)cc(C(N2CCN(C(=O)C(F)C(C)(C)O)CC2C)=O)cc(F)c1 O(NC(=O)C(Cc1ccco1)NC(c1[nH]ccc1COC)=O)CC(CC)C C1(C(N2C(CNC(=O)C=Cc3cc[nH]n3)CC(F)(F)C2)=O)CCc2nn[nH]c2C1 CCCC(CNC(c1ccnc(C)n1)=O)C(=O)N(C)CC1(OCC)CCC1 Nc1cc(C(=O)NC2CCCC(NC(c3cc(F)c[nH]3)=O)C2)cc(F)c1 C(=O)(C1CCCc2sccc21)NC(C(C)NC(C(C)C)=O)CO C=C(C)CCC(=O)N1CCN(CC2CCCN(C(C3CC3C(C)C)=O)C2)CC1 N1(C(CN(C(C(COC)OC)=O)CC2CC2)=O)CC2(CCC(=O)O2)C1 CC(C)P(=O)(CC(=O)NCCC1CN(C(=O)CC2CCCC2(F)F)C1)C(C)C N1(C(C(=Cc2ccc(F)cc2)C)=O)CCC2(C1)CN(C(=O)Cn1nnc(=O)[nH]1)C2 N1(C(C(C)n2cnnn2)=O)CCC(C(C)NC(=O)C(c2cccc(O)c2)C)CC1 c1(NC(C2CCN(C(C(COC)OC)=O)C2(C)C)=O)cccc2cccnc12 C=C1CON(C(=O)C(c2c(C)cccc2Br)NC(c2cc(C(C)=O)cs2)=O)C1 C1(C(C(=O)NC(C2(NC(C3CCCC3C)=O)CC2)C)=O)CCCCC1 C1(NC(CC)=O)(CC)CCCN(C(c2cnn(C3CCC3)n2)=O)C1.C1C(=O)N1 C12CN(CCC1(F)F)C2=O.c1(NC(C(CC)(C)O)=O)cc(C)c(OC)cc1Br c1(C(N2CC(C(N)=O)(CNC(c3cnsn3)=O)C2)=O)ccc2c(c1)C(=O)NC2 N1(C(C(CSC)C)=O)CCCC2(C1)CN(C(C1(C#N)CCCOC1)=O)C2 CC(C)C(C#N)C(=O)NCCOCCN(C)C(C1CNC(=O)N1)=O c1(OC)ccc(CC(=O)NCC2CCN2C(=O)CC2CCOC2(C)C)cc1 Cc1ncc(C(=O)NC2(CCCCNC(c3ccc(=O)n(C)n3)=O)CC2)c(=N)[nH]1 N1(CC(N2C(C(C)NC(CN(C(=O)OC)C)=O)CCC2)=O)CCN(C)CC1 Cc1cc(O)c(Cl)cc1CN1CCC(O)(C(=O)NC(CC(=O)O)C(C)C)CC1 CCC(C)(C(=O)Nc1ccc(NC(C2CC3(CCCC3)CO2)=O)c(C)c1)C(F)F c1(C(N2CC(O)(C(C)NC(C(C)C3CCCC3)=O)C2)=O)ccc([N+](=O)[O-])cn1 C1(CNC(c2scnc2C2CC2)=O)CC2CCCC(C1)N2C(=O)Cc1cnsc1 c1(OC)cc(C(N2CC(CN(C(=O)C3=C(C)OCC3)C)C2)=O)c(C)cc1O C12(C(=O)NCCCCN(C(=O)CCc3ncc[nH]3)C)CSCC1C2(F)F CCCCCC(O)C(=O)N1CCCC1C(N1CCCC(C)(CC)C1)=O Cc1cn2ccnc(C(=O)NCCC(C)N(C(=O)CN3CCC3C)C)c2n1 C(CC(=O)NCC1COCCOC12CCC2)(C(C)(C)C)NC(=O)OC(C)(C)C N1(C(=O)CN2CCCCC2c2cccnc2O)Cc2ccccc2CC1CO c1(C(N2CC(CNC(C(CCC)OCC)=O)C(C)C2)=O)cc(Cl)c(Cl)cc1N N1(C(c2c(C)cccn2)=O)CCC(NC(c2cccs2)=O)C(C(C)C)C1 C(=O)(CC(C(F)(F)F)NC(C12CC(CO)(C1)C2)=O)N(C1CCOC1=O)C C1(NC(c2c(F)ncc(OC)c2)=O)CCCC12CN(C(=O)CCCSC)C2 c1(C(=O)NC(C2CCOC2)CNC(C(C)(C)C)=O)cc2c(Cl)ccnc2s1 O=C(O)CC(CC1CC1)NC(C12CC(c3ccc(C(F)(F)F)cc3)(C1)C2F)=O C1(C(=O)NC2(CC)CCOC2)C2CC3C(C2NC(=O)COCC2CC2)C13 c1(OC)cc(NC(C2CCC3(CCC3)C2)=O)c(C)cc1C c1(CCNC2N(c3ccnc(N(C)C)n3)CCC2)ccc(C#N)cc1 N1(C(N)=O)CCCC1C(=O)NC1CC(CNC(=O)C(c2ccccc2)O)C1 C1(C(N(C2(CCC(NOCCCOC)=O)CC2)C)=O)OCCCC1(C)C N1(C(C(CC)C)=O)CCOC(CNC(=O)CC2CC3(COC3)C2)C1 C12(C(=O)NCCCCC3CN(C(C4CC(C)OC4)=O)C3)CCC(O)(CC1)CC2 c1(CC)ccc(C(=O)NCC(CC)NC(=O)Cc2cc(C)cs2)s1 N1(C(C2(CSC)CC2)=O)CCCC2(CCN(C(=O)C#CC3CCCOC3)C2)C1 c1(CC(=O)NCCN(C(=O)C(C)C(F)(F)F)CC(C)O)cc(O)nc(O)n1 CCCCCCCCNC(=O)C(N1CC2(C1)CN(C(C1(CO)CCC1)=O)C2)=O c1(C(C(=O)NCCCOC)N(CC(C)OC)CC#N)cc(C)cc2c1CCC2 N1(C(C2CC(F)CN2Cc2cc(C(F)(F)F)ccc2Br)=O)Cc2ccncc2C1 c1(SCC)ccc(Cl)c(C(=O)NC2CCC(C(=O)NCCCO)CC2)c1 C(=O)(CS(=O)(=O)CC1CCCO1)N1CC=CC(NC(c2c(NCC)scn2)=O)C1 c1(C(=O)NC2C3CC2CN(C(C2C=CCC2)=O)C3)ccc2c[nH]nc2c1 CS(=O)CCC(O)C(=O)NCC1CN(C(=O)CC2CC2)C1 c1(C(N(C)CC2OCCN(C(C(CCC)O)=O)C2)=O)nn(C)c(=O)cc1C CN1N=C(CC(=O)NC(c2ccnn2C)C(=O)NCC2(C)CCOCC2)CC1=O C(=O)(C#CC1CCOCC1)N1CC(NC(C(F)OC)=O)C2(C1)CC2 C1(C(=O)NC(C=C)(C)CC)CCC(NC(=O)CC2(C)CCCCC2)CC1 Cc1ccc2c(c1)CN(C(C1CCC(NC(C3(C#N)CC3)=O)C1)=O)C2 C1(CC)CN(C(=O)CCc2ccc(F)cc2F)CCC1NC(c1csc(O)n1)=O C1(C(=O)NC(C#C)(C)C2CCCC2)CCC(CCNC(=O)CCc2nc[nH]n2)C1 c1(C(O)Cn2cc(-c3ncoc3-c3ccccc3)nn2)c(F)cccc1F C1(CC(=O)N(C)CCNC(=O)CCCN2CCCCC2)(OCC)CCCC1.OCC c1(NC(C2CCC(CC)CC2)=O)cc(NC(C)(C)C)ccc1P(C)(C)=O C(=O)(C(C)S(=O)(=O)Cc1ccc(Br)cc1)N1CCC(N(C)CC)CC1 c1(C(=O)NCCN(C(=O)C(C)(C)F)CC)cc(-c2ccccc2)oc1C CC1(C)CN(C(c2ccc(F)cn2)=O)C(CNC(C2CCO2)=O)CO1 c1(C(=O)NC2CC(C)(NC(=O)Cn3cnnc3O)C2)c(F)cc(Cl)cc1F C(=O)(C(C)(F)C(C)(C)F)NCC(CC)(CC)NC(=O)Cc1cccc(C)c1C C(=O)(C(CC(=C)C)NC(C1CCC(=O)N(C)C1)=O)NCC(C#C)CC C1(C(C)NC(c2ccnc(N(C)C)c2)=O)CCN(C(=O)C=CCO)CC1 c1(OC)cncc(Cl)n1.C12(COC1)C(=O)NCCOC1CN(C1)C2=O.CC N1(C(CCc2scc(C)n2)=O)CCCC1C1CCCN1C(=O)CCOCC1CC1 c1(CC(=O)NCC(C)NC(c2cc(-c3ccncc3)ccn2)=O)nn(C)cc1Cl C1(NC(C(C=C)C)=O)CCC(CC(=O)Nc2cnc(SC)nc2)CC1 C12(C(=O)NC3(CNC(c4c(N)cccc4F)=O)CCC3)CCCCC1C2(F)F c1(C(=O)NCC2CCC2C(=O)NCC2CCCO2)cccs1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC2C(NC(=O)CC3(CO)CC3)(C2)C1 c1(NC(N(C(CC)C)C)=O)cnn(CCOC)c1 C1(C)(CNC(C2(C(=O)OCC)CCC2)=O)CN(C(=O)C(O)C(C)CC)CC1C Cn1ncc(C(c2nnnn2-c2ccccc2)NCC2CCCS2)c1Br N1(C(C(COC)(C)C)=O)C2CCC1(CNC(C1CCC(F)CC1)=O)CC2 C1(CN(C(C2(COC)C=CCC2)=O)C)CC(F)CN1C(c1cc(C)c(Cl)s1)=O Cc1nc(C(=O)NC2CCN(C(c3c(C)nn(C)c3C)=O)C2)c2ccnc-2[nH]1 c1(C(=O)NCCCN2CCN(c3cc(OC)ncn3)CC2)cccc2nccn12 C1(C)(CNC(Cc2c(C(C)C)con2)=O)CCCN(C(C2(C)COC(=O)C2)=O)C1 C1(CC=C)(CNC(=O)C(=O)Nc2ccnn2CC2CCOC2)CCOCC1 C1(NC(CCc2nc(C3C(C)C3)sc2)=O)CCC(N=[N+]=[N-])CC1 CCC(C#N)C(=O)NC1CC(C(C)NC(=O)C=Cc2cnccn2)C1 C1(CC(=O)OC)C2CN(C(C3(N)CCC4CC34)=O)CC12 c1(C(N2CC(COC)(NC(=O)C(C)=O)C2)=O)ccccc1OC c1(C(N2CC(CNC(c3cncc(C)n3)=O)C2)=O)nc2n(c1Cl)CCCC2 C(=O)(C1CCCc2sccc21)NC1C(C)(C)CN(C(c2ccoc2)=O)C1 N1(C(c2cccc(N(C)C)n2)=O)CC(NC(C2(CCF)CCC2)=O)C(C2CC2)C1 C1(C(=O)NC(CC=C)C)CCC=CC1NC(=O)CC=O.OC N1(C(CC2CC(OCC)C2)=O)CCCN(C(=O)CC2SC(=N)NC2=O)CC1 N1(C(C(CC2CC2)OCC)=O)CCCCC(NC(c2cc(COC)on2)=O)C1 C1(CN(C(=O)C(O)c2cnc[nH]2)Cc2cnns2)CCOC1=O CC1CCN(C(=O)C(F)OC(F)(F)F)C1C(=O)NC(c1ccoc1)C C(=O)(C1CCCc2sccc21)N1CC(C)(NC(c2onc(C)n2)=O)C1 CC1CC(CO)CN(C(C2CCCN(Cc3ccnn3C)C2)=O)C1 C(=O)(CC(O)CC(C)C)N1CCC(C)(C(=O)NC(CCC)C(F)(F)F)CC1 Cc1cc(CCC(=O)NC2CCCC2CNC(c2n[nH]cc2Cl)=O)nn1C C(=O)(C(O)C1=CCCCC1)NCCC(CC)(C)NC(C1CC12CCOC2)=O C1(C)(C(=O)NC(CNC(c2cc(C(C)C)[nH]n2)=O)C2CC2)CCC(=O)N1 c1(C(=O)NC(C2N(C(c3c(SC)ccs3)=O)CCCC2)C)cc2cccnc2[nH]1 Cc1ccc(C(=O)NCC(C)(CO)NC(c2cccc[n+]2[O-])=O)cc1C C1(CNC(C(CCCOC)C)=O)CC2(CCC2)CN1C(C1CCCN1C=O)=O c1(OC)cscc1C(=O)NC(c1ccccc1)CNC(CCC(C)(C)C)=O c1(C(=O)NC2CN(C(CSCCC)=O)CC2C(F)F)cn2ccnc2s1 C(=O)(N1CCC(C(=O)NCCC(C)(O)COC)O1)c1c(CCC)n[nH]c1 N1(C(c2c(N)non2)=O)CCC(C2CCN(C(=O)C(=O)NCC(F)F)C2)C1 C(=O)(CC(C)(C)C#N)NCC=CC(=O)N(C)Cc1nnc(CC)o1 c1(C(=O)NCC(CC=C)NC(=O)CCC(C)(F)F)cc2c(s1)CCS(=O)(=O)C2 N1(C(c2ccc(C)s2)=O)CCC(C)(CCNC(=O)CC23COC(CF)(C2)C3)C1 Cc1oc(C(C)(C)C)cc1C(N1CCC(CCNC(=O)C(C)c2ccsc2)C1)=O C(=O)(CCC(=O)NC(C(C)NC(=O)C(=Cc1cccs1)C)C(C)C)N(CC)CC Cc1noc(NC(C2CN(C(c3cccc(=O)n3C)=O)CCN2)=O)c1C#N S(=O)(=O)(C=Cc1ccccc1)NC1CCC(NC(c2ccsc2Br)=O)C1 N1(C(c2c(C)occ2)=O)CC2(CCC2)CC1CNC(c1ccc(CCO)cc1)=O N1(CC)CCC(C(N2CC=CC2(C)C(N2CCOC(CC)C2)=O)=O)CC1 CC(CC(=O)NCCC(N)=O)NC(=O)Nc1ccccc1 C(=O)(C1=C(C)Oc2ccccc2C1)NC(CCNC(CCSCCCC)=O)(C)C C(=O)(CC(CN(C)C)C(F)F)N(C1(NC(CN(C(C)C)C)=O)CC1)C C(CC(CC)C(=O)N1CC=CCC1C(=O)NCC1CCC(C)C1)=CC C(C(=O)NC(CNC(c1cccc(SC)c1)=O)C1CCC1)(C(C)(C)C)OC N1(C(=O)C2=C(Cl)CC2)CCCC(C2CN(C(=O)COCCO)C2)C1 c1(CC(=O)NCCN(C(c2cnc(C3CC3)[nH]2)=O)C2CC2)ccc(F)cc1 N1(CCC)C(=O)CCC1C(=O)N(C)CC1CCCCN1C(c1coc(CO)c1)=O C1(CC)CCN(C(c2cnn(CC)c2)=O)C1C(=O)N(CCc1cc(C)[nH]n1)CC N1(C(COCC#C)=O)CCC2CCN(C(=O)CCCCCCCSC)CC2C1 C1(NC(C(C)NC(N)=O)=O)C2CC3CN(C(c4cc5occc5s4)=O)C1C3C2 CC1CN(C(C2(CNC(C3CC(O)C(F)C3)=O)CC3(CC3)C2)=O)CC(CO)O1 c1(CCC)cc(C(N2CC(CNC(=O)CCc3nncn3C)CC2C)=O)n(C)n1 c1(C(=O)NCCCN(C)C(C2(CF)CCC2)=O)cncc(C(F)F)c1 C(CC(F)F)(C(=O)NC(C)CN1CCOCC1)NC(Cc1c(C)nccc1)=O C(C)(c1ccccc1C)=CC(N1CC(OCC)(CNC(c2c[nH]cc2Br)=O)C1)=O N1(C(COCCCOC)=O)CCN(C2CCN(C(C3CCC(=O)N3)=O)CC2)CC1 c1(C(N2CC(CC(C)NC(C(CC)(C)F)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl C1(C(N2CCCC(CCNC(C(C)=C(C)C)=O)CC2)=O)CC2CSCC(C1)C2 C(Cc1ccco1)(C(=O)N1CCC1Cc1ccco1)NC(C(C1CC1)OC)=O C=CCN=C(NCC(C(C)(C)C)OC)N1CCC(OC)CC1.C1CC(=O)N1C1CC1 c1(C(N2CCC(NC(c3cnc(OC)c(Cl)c3)=O)C2)=O)c(Cl)cccc1[N+](=O)[O-] C1(CNC(C(=CC2CCCC2)C)=O)CC2(C1)CN(C(C1CCCC1(F)F)=O)C2 N1(C(C(C)OC)=O)CCC2(CCCCC2NC(c2cc(C)no2)=O)C1 C(CCCCCN=[N+]=[N-])NC(C(C(C)NC(C1CCCCN1C)=O)(C)C)=O C1(O)(C(C)NC(=O)CCc2cn[nH]c2)CCN(C(=O)C(N2CCC(O)CC2)C)C1 CCC(O)C(C)(C)C(=O)N1CCC(CNC(c2sccc2F)=O)(OC)C1 c1(CC)ncc(Cl)c(C(=O)NCC2CN(C(=O)CC3(C4CC4)CC3)CCN2C)n1 C(=O)(C1=NOC(CC(=O)N(CC(CC(C)C)NC(C2(CO)CCC2)=O)C)C1)OC c1(OC)ccccc1CC(=O)NCCCOCCNC(=O)C=C1CCSCC1 C1(OC)CCN(C(C2C=CCCN2C(=O)CC2(O)CCC2)=O)C1(C)C O=C1Cc2cc(C(N3CC(NC(c4cc(Br)c[nH]4)=O)C(F)C3)=O)c(Cl)cc2N1 N1(C(c2c(C)ccs2)=O)CCCC(CNC(c2c(C)cnn2C(C)C)=O)CC1 CCC(CC(=O)NCc1c[nH]nc1C(=O)NC12CC(C)(C1)C2)C1CCC1 C12(C(=O)NCCN(C(=O)Cc3cn(CC)nn3)CCC)CC(OC)C1C2 CC1N(C(=O)C(C2CN(C(c3ccc(F)c(O)c3)=O)C2)N(C)C)CCCC1(C)C CC12CC(NC(=O)C(C3CCCCC3)O)(C1)C1(CN(C(c3ccc(F)s3)=O)C1)O2 c1(C(=O)NCC(C)N(C)C(c2ccc(F)o2)=O)c(Cl)cc(Cl)cc1Cl N1(C(C2(C(=O)OC)CC2)=O)CCC(C)(CC(N2CC3CC3C2)=O)CC1 C(CCOCCO)(C(=O)NC1CC(O)(CO)C1)NC(C1CCC(F)(F)C1)=O C1(NC(C=COCC)=O)CC2CCC1(CNC(c1cnc(C3CC3)o1)=O)C2 c1(COC)cccc(C(N2CC(NC(=O)C(Cl)=CCl)CC2CO)=O)c1C c1(CC(=O)NCC2N(C(CNC(=O)NC)=O)CCC2)ccc2nc[nH]c2c1 c1(OC)cc(OC)c(OC)cc1CN(C)CC1(O)CN(c2ncncc2F)C1 N1(C(CN(C)CC)=O)CCN(C(=O)CN2CC(=O)NC2=O)C2CC12 Cc1cccc(C(=O)NC2CC2C(N2CCC(O)C2)=O)c1 Cc1ncnc(C)c1CC(=O)N(CC(C)O)CCNC(=O)CSC1CC1 C1(C2CCCCN2)(C(N(CC(C)CO)C)=O)CCOCC1 CC1(C)CN(C(=O)Cn2ccc(=O)c(O)c2)CC(CNC(C23CC(C2)C3)=O)O1 N1(C(C(C)OCc2cccnc2)=O)CCC2CN(C(C3(CF)COC3)=O)CC12 CC(CCC(=O)NC1CC(NC(=O)CC2CN(C)C2)C(O)C1)N(C)C C1(NC(=O)C2CC2)Cc2ccccc2N(C(c2cn(Cc3cccs3)nn2)=O)C1 CCCCC(C)C(=O)N1CC2(C1)CN(C(c1ccc(N(C)C)cc1OC)=O)C2 C1(C(N2C(CC(=O)NC3CCC(N(C)C)C3)CC(O)C2)=O)CCCC12CCC2 N1(C(=O)CC2CCC2)CCCC2(C1)CN(c1ccnc3cc(Br)nn13)CCO2 Cc1cc(NC(c2cc(Cl)cn2C)c2nnnn2C(C)(C)C)cc(C(F)(F)F)c1 C1(C(N2CC(COC)(NC(=O)CCc3cccs3)C2)=O)(OC)CCSCC1 C(=O)(CC(F)(F)C(F)F)N1CCC(C#C)(C(=O)NCCC2CC(C)=NO2)C1 N1(C(CC(=O)NCC#C)=O)CC2COCCC2(NC(c2ccc(F)cc2C)=O)C1 N1(CCC(NC2c3n(C)ncc3CCC2)=O)CC2(CCOCC2)CC1CC(=O)NC Cc1cnn(CC(=O)NC2CCC(NC(c3cscn3)=O)C2)c1 c1(C(=O)NC2C(NC(C=C(C)C(F)F)=O)CC2)ncnc2c1CCC2 C1(C(=O)NC(c2ccccc2)CNC(C2(CO)CCC2)=O)CN2CCN1CC2 CCCCC(C)CC(=O)N1CCCC1C(C)(C)C(=O)NCC(=O)N(C)CC c1(NCCCN(C(c2n(CC)ncc2)=O)C)nc(O)n(C)c(=O)c1[N+](=O)[O-] n1(-c2ccc(-n3c(C)ncc3)s2)ccc(=NC(=O)C2CC2C(=O)OC(C)(C)C)[nH]1 C=CC(C)(CC)C(=O)NCC1(F)CCN(C(c2ccc(C)c(F)c2)=O)C1 C=CCCCCC(c1nnnn1CCCC(=O)OCC)Nc1cccc(F)c1 C(=O)(CCCCC(F)(F)F)NCCN(C(=O)C(C(C)C)C1CC1)CCOC C12(C(N(CCCCO)CC)=O)CCN(C(c3nc(O)sc3C)=O)CCC1C2 c1(C(N2CC(CC=C)(NC(=O)CNS(=O)(=O)N(C)C)C2)=O)cccc(Cl)c1C c1(C(N2CCC(F)(CNC(Cc3cc(C)on3)=O)C2)=O)cccc2cnn(C)c12 c1(-n2c(C(C(C(C)C)N3CCOCC3)NCCOCC)nnn2)ccc(OC)cc1 C(C1=NOC2CCCC12)NC(C(C1CN(C(CCC=C)=O)C1)O)=O C1(C(=O)NCC2C(CNC(COc3cccc(CC)c3)=O)C2)OCCOC1(C)C C(=O)(C(C)(C)CCF)N1CC2C(C(=O)NCCC(C)N3CCC3)(C2)C1 c1(CN(CCOCC)C(C2CCN2CC)=O)ccccc1Cl.C1CC(=O)N1 C1(C(=O)NC(c2nc(C(N3CCC3CC(C)(C)C)=O)co2)C)(CO)CC=CC1 c1(OC)ccccc1-c1ncc(C(=O)NC2CCC2CNC(=O)C(C)N(C)C)s1 CC(C)(C)C(CNC(C1CC12CCOC2)=O)NC(=O)CSc1ccc(O)cc1 N1(C(C(c2ccc(Cl)cc2)C)=O)CC2(C1)CN(C(=O)C(C)(C)S(C)(=O)=O)CCO2 C#CC1(C(=O)NC2CCOC2=O)CCN(C(=O)COC)C1 c1(NCc2cn(CCCCCCNC(C(C)(CO)OC)=O)nn2)cnc2ccnn2c1 N1(C(CSCc2nc(C)sc2)=O)CCC(C)C1CNC(=O)CCc1cc(Cl)no1 CCCC(O)C(=O)N(C1CCC(NC(=O)C(C)(F)F)CC1)C CC1CCCC2CCCN(C(c3c(F)cc(F)cc3[N+](=O)[O-])=O)C12 c1(OC)cnc(Cl)[nH]c1=NC(=O)C1(SC)CN(S(=O)(=O)C(Cl)(Cl)Cl)C1 c1(NCC(CC)C)cc(NC2CC2c2ccc(OC(C)C)cc2)nc(C)n1 C12(C(N3CC(CCNC(CCNC(=O)NC)=O)C3)=O)CCCCC1CCCC2 CCC(C)CC(C)C(=O)N1CCC(C(=O)O)C(F)(F)CC1 c1(CC)nn(C)c(C(=O)NCC2CCCCN(C(=O)CCc3cnoc3)C2)c1Cl CCC(CCC(=O)N(C(C)CC(=O)Nc1ccc(OC)c(O)c1)C)OC CCCN(OC)C(=O)CC(CCC)NC(=O)C(N)CCCC(C)C C(=O)(C(C)(C)C(C)C)NC(C=CC(=O)NCC1CCN(CCC)C1)C Cc1c(C(N2CC=CC2CNC(=O)C(F)C(F)(F)F)=O)oc2ccc(F)cc12 C1(CC#C)(C(=O)NCC(=C)CCNC(=O)CCC2CCCOC2)CCOC1 Cc1n[nH]cc1CN(C)C(c1ccoc1CNC(C12CSCC1C2)=O)=O C1(NC(c2nc(C(C)OC)sc2)=O)CCN(C(C2(CSC)CC2)=O)CC12CCC2 c1(C(N(C(CC)C(=O)NC2CC2)C)=O)ccnc(OC)n1 C(CC(CC)C(=O)N1CC(CC(F)C(N2CC3C(C(C)C)C3C2)=O)C1)=CC C1(NC(CS(=O)(=O)N(CC)CC)=O)CC2CN(C(c3c(Cl)n[nH]c3C)=O)CC2C1 Cc1nc(C(N2CC=CC(NC(=O)CCCCNC(N)=O)C2)=O)nn1C c1(CC(C(C(=O)Nc2cncc(OC)c2)F)C)c[nH]c2ccccc12 c1(CC)ncc(C(N2CCC(NC(c3csc(C#N)c3)=O)CC2C)=O)c(C)n1 CC1CN(C(=O)C(c2cnn(C)c2)NC(c2ccc(F)cc2)=O)CCN(C)C1 N1(C(CC(C)c2ccco2)=O)CCSCC1C(=O)NCCC1(C)CC1(F)F C(C(CO)(CO)NC(C1OCCC1(C)C)=O)N(C(C1(CC)CC1)=O)C c1(OC)ccc2c(c1)CCC2(O)CNC(=NC)N1CCN(c2ccccn2)CC1 c1(CC)nc2sc(C)cn2c1C(=O)NC1CCC(CNC(C2C3COCC23)=O)C1 C1(NC(CSC)=O)CN(C(c2cc(O)nc3c2CCCC3)=O)CC12CCOCC2 CC(CC(N)=O)C(=O)N1C(CNC(=O)CCc2nnc(C(F)F)o2)CC2CC12 C(C)(CCCCNC(c1cccc(C2CC2)n1)=O)NC(C=CC=CC)=O N1(C(CCSC)=O)CC2CC(CNC(C3(c4ccnc(Cl)c4)CCC3)=O)CC1C2 N1(C(C(COC)O)=O)CCN(C(c2ccn(C3CC3)n2)=O)C(C(F)F)C1 C(CO)(C(=O)N1CCCC1CN(C(=O)CN(C1CC1)CC)C1CC1)OC c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1c(Cl)cnn1C)=O N#CC1CCC(CC(=O)NCC2(NC(c3cc(C4CC4)n[nH]3)=O)CC2)C1 N1(C(c2cncc(OC)c2)=O)CC(C)CN(C(C2CC(F)(CO)C2)=O)CC1C N1(C2(C)CC2)CCN(CCC(=O)NC2CCN(C(c3nn[nH]c3Cl)=O)CC2)CC1 c1(C(=O)NC(CC(C)NC(c2cnc(C(N)=O)s2)=O)C)ccc(C2CC2)cc1 C(=O)(C1=CC2CCCC12)NCC1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 C1(CCOC)CN(C(=O)C2=NOC(C(C)(C)C)C2)CCN1C(=O)CS(N)(=O)=O C1(NC(CC(C2(O)CCCCCC2)(C)C)=O)CC2CCC(C1F)N2C(=O)C1CC1 N1(CCC(=O)NC(CNC(C(CC)F)=O)(C)C2CC2)CCN(C)CC1 c1(C(N(C2CCN(C(C3CC3F)=O)C2)CCC)=O)cc2c(nn1)OCCS2 c1(OC(C)C)nc(N2CC3C(C(=O)Nc4ccc(CO)nc4)C3C2)ncc1Br C=CCC(C)(C)CCN(C(=O)C(c1cccs1)NC(C)=O)C Cc1ccc(C(=O)NCC2CC=CCC2)nn1 C1(C(N2C(C)C(NC(=O)C(F)Cc3ccccc3)CC2)=O)CC2(CCCCC2)C1 Cn1c(C(=O)NC2CC(NC(C3(CO)CCCO3)=O)C2)cnc1S CC(O)C(C(=O)NC1CCC1)NC(C1CC1C(N)=O)=O c1(OC)c(Cl)cc(C(=O)NC2CC2NC(=O)CCOc2cccnc2)nc1Cl C1(CCNC(c2ccc(Cl)s2)=O)CSCCN1C(C1(c2cccnc2)CC1)=O c1(C(=O)NC2C(NC(c3c(CC)nn[nH]3)=O)CCC2)c[nH]c2cccc(Cl)c12 C(=O)(C1=CNS(=O)(=O)N=C1C)NCCN(C(C(C)OCC#C)=O)CC(C)O C1(C(N2C(CNC(C3C(C)(C)C3C#N)=O)CCC2)=O)CC(=O)CC(=O)C1 C1(NC(CCCc2n(C)cnn2)=O)CN(C(C2(c3ccnn3C)CC2)=O)CC1F Cc1ccc(CC(=O)NC2CCN(C(c3cc(O)nc(Cl)c3)=O)CC2F)c(C)c1 c1(C(=O)NC(CC(C)C)(C)CNC(C2CC=CCO2)=O)ccc2cncn2c1 O=C(CC1CCc2ccccc21)NC1CCN(C(C2C3CC4C(C3)C24)=O)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CC)CC1(CNC(=O)C(C1CC1)OC)C2 N1(C(CSCC(C)C)=O)CCCC(CN(C)C(c2cc(C(N)=O)cn2C)=O)C1 c1(C(=O)NCCCN(C(=O)CC2CCC(C#N)C2)C)cn(C)nc1Br Cc1cc(C(=O)NC2CC(O)CN(C(c3ccccc3C(C)C)=O)C2)cc(C)c1 N1(C(C(C)=C(CC)C)=O)CC2(COC(CNC(c3nccn4ccnc34)=O)C2)C1 C1(C(N2C(C(=O)Nc3ccc(OC)nc3C)CC3CC32)=O)CCc2ccccc2C1 C1(CNC(CCC=C(C)C)=O)CCCCN(C(C2(C#N)CCCO2)=O)C1 c1(CC(=O)NCC2CCN(C(c3ccc(C(N)=O)s3)=O)C2)nnc2n1CCCC2 c1(N2CCCC(CC)CC2)nc2ccsc2c(=NCC2(CO)CCCOC2)[nH]1 C1(CNC(=O)CN2CCOC2=O)CC2(C1)CN(C(=O)CO)C2 c1(OCC(N2CC(NC(c3nc(CC)oc3)=O)C(C)C2)=O)c(C)cc(C)cc1C c1(C(N2C(C(CNC(C(C)(C)F)=O)(C)C)CCC2)=O)cnc2cc[nH]c2c1 CCCC(O)CC(=O)NCC12CC(CNC(c3n[nH]c(C)c3Cl)=O)(CO1)C2 CCN=C(NCc1cnc(Cl)cc1C)N1CCC(O)C1 C(CCC(C)NC(c1cccnc1)=O)NC(C(c1ccccc1)C)=O c1(CN(C)C)cc(C(=O)NCC2CCN2C(=O)CC2CCCO2)ns1 C1(CNC(CC(CC)C2CC2)=O)N(C(=O)C=CCOCCO)CCCC1(C)C C=Cn1nncc1C(=O)NC(COCC)C(=O)NCCC1COCCO1 N#CC1CCCC(C(N2CC(CC(F)C(=O)NCC(C)(C)NC=O)C2)=O)C1 c1(CC)ccc(Cl)nc1NC(C)Cc1ccccc1C.C(CC)(CC)n1c(=O)c1=O c1(NC(c2ccncc2-c2ccccc2)=O)ccc2oc(Cl)cc2c1 Cc1cc(C(N2CCC(C(C)NC(=O)CC(c3cccs3)C3CC3)C2)=O)c(C)s1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCOC(C(C)NC(C2(C(C)(F)F)CC2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC(C1(O)CN(C(C(Cc2ccccc2)OC)=O)C1)C C(CNC(=O)CC=CC(C)(C)C)(CC(F)(F)F)NC(C(C1CC1)OC)=O c1(CNC(C(=O)OC)(C)c2cccnc2)cc(Br)sc1Br C1(NC(c2cscn2)=O)CC2CCC(C1F)N2C(c1sccc1OC(F)F)=O c1(CC(=O)N(CC(O)CN(C)C(C2CC(O)C2)=O)C)cncnc1O N1(C(CC2CC(=C)C2)=O)CCC(C2CC2)C1CNC(C1C2C3CCC(C3)C12)=O C1(C)(C(=O)NC2C(NC(C(c3c(C)cncc3)C)=O)CCC2)C(C)(C)C1(C)C c1(C(CC)C)nc(C)c(CC(=O)NC(C)CCCNC(=O)C(C)CO)c(C)n1 C1(CC(=O)NC(C2CCN(C(C3CC(=C)C3)=O)CC2)C(C)C)CC(O)C12CCC2 O=Cc1cccc(-c2cncc(CN3CCC(Br)CC3)c2)c1Br C1(C(N2C(C)(C(=O)NCCCN(C)C)C=CC2)=O)CC2(CCC2O)C1 CCCC(C(=O)OC)C(=O)NCC(C(C)C)NC(=O)COc1cnc(Cl)cn1 c1(OCC(=O)NC2CN(C(C(C)(C)Cc3ccccc3)=O)C2)nc(O)nc(O)n1 C1(NC(c2c(C)nccc2)=O)CN(C(=O)CCc2ccncc2)C2CCCCC12 CC(C)CC(C(=O)NCCC1CC(NC(C2(CF)CC2(F)F)=O)C1)C(C)C c1(C2(OC)CCN(C(c3n(CC)ccn3)=O)C2)cc(Br)ccc1F C(=O)(CC(O)C(C)C)N1CCC(OCC(=O)NCc2nc(C)c(C)s2)C1 N1(C(C2CC(C)=C(C)CC2)=O)CC2(CCCC2NC(=O)CCOC(C)C)C1 N1(C(c2c(C)oc(C#N)c2)=O)CCC2(CC1)CCN(C(=O)C=CI)C2 CCC(O)C(C)(C)C(=O)NC1CC(CNC(c2ccoc2C2CC2)=O)C1 c1(C(=O)NC2C(C(N3CCC(OC(C)=O)C3)=O)COC2)nccc(C)c1N CCC1(CNC(C2CN(c3ccc(Br)cc3)C(=O)O2)=O)OCCc2ccccc21 C=CCC(C(=O)NCC(C)N(C(=O)Cn1nccc1C)CC)NC(C)=O N1(C(C(CC)(CC)OC)=O)CC(NC(=O)CCCCCOC)C(C2CC2)C1 Cc1cccc(C(c2ccccc2)SCCCNC(=O)CCC2CCCN2C)c1 N1(C(c2c(C)noc2)=O)CC2CC1CN(C(=O)C(C(C)C)n1ccnc1)C2 C(CCC(=O)NCC1CCCN1C(C1CC2CC2C1)=O)N(C(C)=O)C CC(C)(CCCNC(c1sccc1F)=O)NC(=O)COc1ccccc1C(N)=O c1(CC)nsc(CNC(=O)C(C)CN(C(=O)Cc2cc(C)cs2)C)n1 N#Cc1ccc(C(N2CCC2CC(=O)Nc2ccc(C3CC3)cc2)=O)nc1 C(=O)(C1Cc2ccc(Cl)cc21)NCC(CC)NC(=O)C=Cc1ccccn1 CCCCC(CNCc1cccc(C#N)c1F)CCC c1(C(=O)NCC(CNC(c2ccccc2F)=O)OC)cc(S(N)(=O)=O)oc1C C(=O)(C(C)(C)C(=O)NCC1CC(C)(C)CN1C(=O)C(CC(C)C)N(C)C)NC CN1C(=O)C2CN(C(=O)C(=O)N(C3CNCCC34CCC4)C)CC2C1=O Cn1nnc2cc(C(=O)NCCCC)cc(Br)c12.C1(C(=O)N)CC(C)(C)CCO1 C1(COC)(NC(c2cc(Cl)cnn2)=O)CCN(C(=O)CCCc2ccccn2)C1 C(=O)(C(=O)CCC(C)C)NC1C(CC)CN(C(=O)COC2CCOCC2)CC1 C1(CC)CN(C(c2cc(C)ccc2I)=O)CCN1C(c1cc(C)on1)=O c1(C(N2CCC(O)(CN(C)C(C3CCCO3)=O)C2)=O)cccc2c1CCC2=O c1(C(CNC(CSC)=O)NC(=O)C(O)CF)ccc2ccccc2c1 C(CCN(C1CCCCCC1)N1CC(C(=O)OC)C(c2cncn2C)C1)OCC c1(OC)cc(Br)ccc1CN1CC2CC1CN2Cc1ccc(C(=O)N(C)C)nc1 C#Cc1ccc(OC)c(C(=O)NC2COCC2NC(c2conc2C2CC2)=O)c1 C1(CC(=O)NCC(=O)NC(CN(C(c2cncnc2)=O)CC)C)CCOCC1 C1(NC(CC2(OC)CCC2)=O)CCC12CCN(C(c1nsnc1OC)=O)CC2 C#CCCCCC(=O)NC(c1cn(C)nn1)C(N1CCC(C)(O)C1)=O C1(C(F)(F)C(=O)NC2CC(NC(=O)Cc3cnsc3)C2)(OC)CCOCC1 C1(NC(Cc2cc(C)[nH]n2)=O)CN(c2ncnc3scnc23)CC2(CC2)C1 C12(CNC(CC3C=NN(C)C3=O)=O)CC(NC(=O)CCOC(C)C)(C1)C(C)(C)O2 CN=c1[nH]c(=NCC(C)c2ccsc2)[nH]c(=NC2CCCCC2CC(C)C)[nH]1 Cc1cc(C(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)ncc1F c1(C(C(N2CC(OCC)(CNC(c3cc(F)c[nH]3)=O)C2)=O)(F)F)cccc(C)n1 c1(C(N2CC(NC(C3(O)CCOCC3)=O)CC(O)C2)=O)cccc2ccccc12 C(=O)(C(C)CC(=O)OC)NCC(CC)NC(c1ccc(OC)nc1C)=O Cc1nc(S)nc(C)c1CCC(=O)NCCC(C)N(C)C(c1ncccc1Cl)=O N(C1CN(C(C23CC(F)(C2)C3)=O)CCc2ccccc21)C(C(CC)OC)=O C1(C(=O)NCC=CCNC(C(C2CCCC2)OCC)=O)CC(CC)CO1 N(C1CN(C(=O)C(C)N(C)C)Cc2ccccc21)C(C1(C(C)C)CCCCC1)=O c1(NC(=O)NC2CC(SCCCOC)C2)c(C)nn(-c2ncccc2Br)c1C C(c1cnc(C)nc1O)=CC(=O)NC1CCN(C(c2cn(CC)nn2)=O)C12CC2 C(=O)(C(=O)N=S(C)(C)=O)NCC1CC(C)N(C(=O)CCC(C)(F)F)C1 c1(OC)ncc(F)cc1C(=O)NC(C)(C)CNC(=O)C(C)c1cc[nH]n1 CN1CCC(CO)(CNC(=O)C(CCC2CC2)NC(c2coc(C(N)=O)c2)=O)C1 c1(C(N(CCNC(=O)CCc2cccnc2Cl)CC)=O)c(C)cccc1C c1(C(C)C)ccc(C(=O)NCc2cc(C(N3CCCC3CO)=O)on2)s1 C1(NC(c2ncoc2C2CC2)=O)CCCC(CNC(C2CC(O)C2)=O)C1 c1(C(=O)NC(C(=O)NCC2OCC(C)(C)C2)C2(O)CCC2)cc2ccccc2o1 c1(C(=O)NC2C3CN(C(=O)C=CC4CCOC4)CC23)cc2c[nH]cnc-2n1 N1(C(CC2(C)CCC2)=O)CCC(O)(CCNC(c2cccc(F)c2)=O)C1 C1(NC(C2C(C)C2C)=O)CCOCC1C(=O)NC1(CN(C)C)CCCCC1 C(=O)(C1=C(C)OCC1)NC1CC(C)(C(N2CC(C)(OC)C2)=O)C1 CCCCC(=O)C(=O)N1CC(N(C(=O)Cc2ccc(OC)cc2)C)C(O)C1 CC1CC(CO)CN1C(=O)C#CCNC(=O)CCCC1CCCO1 Cc1nn(C)cc1C(=O)N(C1CC2CNC1C2)CCc1cnc[nH]1 c1(CCC=C)ccc(C(=O)NCC(C)(O)CNC(C2CCCOC2)=O)cc1 C1(NC(c2ccc(COC)s2)=O)C2CN(C(C3C4CCC3(OC(C)=O)C4)=O)CC12 CCC(C)(CO)C(=O)NCCC1CCN(C(c2csc(=N)[nH]2)=O)C1 C(CCO)N(S(C)(=O)=O)CCN(C(CCC)=O)C.N c1(C(=O)NCC(CCOC)Nc2ncc(C#N)cc2F)sc2nccn2c1C N1(C(C(CCOC)C)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 c1(CN(C)C(=O)NCC2(Cl)CC2(F)F)nc2c(s1)CCCC2 c1(COC(C(C2CCCOC2)OC)=O)cccn1C(c1ccncc1)C C(=O)(C(C#N)(CC)CC)NC1CC2(C(C(N3CC(C#C)OCC3)=O)C2)C1 Cn1nc(C(=O)NCC(C)(Cn2cccn2)NC(=O)CC2CC23CC3)cc1O CC1=NOC(=O)C1CC(=O)NCCC(C)NC(=O)Cc1nc(C2CC2)cs1 C(CC(N)=O)(C(=O)NCc1cn(C)nc1O)NC(CCC=C=C)=O c1(CC(=O)NC2CC2CNC(C2(c3cccs3)CC2)=O)ccc(O)nc1 O(NC(=O)CCCC(C)(C)NC(C1CC(OCc2ccncc2)(OC)C1)=O)CC c12cccc(c1)O2.c1(CC)ccc(C(=O)NC(C)CNC(=O)COCC(C)C)s1 c1(C(=O)NCC2N(C(CCC3CC(OC)C3)=O)CC2)ncccc1O c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CCOC2)cc(=N)[nH]c(Cl)n1 c1(C(N2C(CNC(C3ON=C(C)C3)=O)CN(C)CC2)=O)cnc2[nH]cc(C)c2c1 Cc1cc(CN(C(=O)C(N2CCC(c3nncs3)C2)=O)C)cs1 c1(COC)cc(C(N2CCCC2C2CCN(C(=O)CC3CCSC3)C2)=O)n[nH]1 c1(C(N2CC(NC(C3CCCN3C=O)=O)CC(OC)C2)=O)ccc(C#N)c(C)c1 Cc1c(C(=O)NC(C)CCCCNC(=O)CCC(C)N(C)C)cnn1CCN(C)C N1(C(C2C(CNC(C(C)n3ccnn3)=O)CC2)=O)CCN(C(C)(C)C)CC1 N1(C(CCSC)=O)CC2CCCC1C2CNC(=O)CC1CCCCCC1 c1(C(=O)NC(C2CCCN(C(c3cc(F)n[nH]3)=O)C2)C)ccc2nsnc2c1 C(=O)(CS(=O)CCC(F)(F)F)N(C1CN(C(c2cc3cccnc3s2)=O)C1)C C1(NC(CCC)=O)CCC2(CCCN2C(c2cccn(C)c2=O)=O)CC1 N1(C(c2c(CC)c[nH]n2)=O)CCCC2(C1)CN(C(=O)CN1OC(C)(C)CC1=O)C2 C#CC1(C(=O)N(C2CCC2C)C)CCN(C(=O)C(F)CCC)C1 N1(C(C(c2n(C)ccc2)=O)=O)CCOC2(CCN(C(C3CC(F)(F)C3)=O)C2)C1 c1(C(=O)OC)cc(NC(=O)C(=O)Nc2ccc(SCC(C)C)cc2)c(C)cc1F c1(C(=O)NC(CN(C(CC(c2ccc(F)cc2)C)=O)C)C)ccc2ncnn2c1 c1(C(N2C(NC(C(c3c(C)cncc3)C)=O)CC2)=O)cc(Br)cc(N)c1C Cc1ncc(NC(C2CCCCC2CNC(=O)C(C)CN(C)C)=O)c(C)n1 c1(N(C2C(C)CCNCC2)C(c2ccc(F)cn2)=O)cc(Cl)c(I)cc1[N+](=O)[O-] c1(C(=O)NC(C2(CNC(C(C)Cn3cccn3)=O)CC2)C)ccsc1C#N CC1C(NC(c2ccc([N+](=O)[O-])s2)=O)C(C)CCN1C(=O)Cn1cccc1 CC1(C)CN(c2cc(Cl)c(O)nn2)CC(CNC(=O)CN2CCC(F)CC2)O1 N1(C(C2(NC(CC3CCN(C)C3=O)=O)CC(F)(F)C2)=O)CCN2CCC1C2 C(=O)(CC(F)(F)C(C)C)NC1CCC(CCNC(C2(OC)CCSC2)=O)C1 C1(NC(C(CC)(F)F)=O)CCC2CC1CN2C(=O)C=Cc1ccccn1 CC1CN(C(=O)CCC2CCCN(C)C2)CCCN1C(=O)Cn1cccnc1=O C(CC1=CCN(Cc2cncs2)CC1)NC(C(c1c(C)noc1C)C)=O c1(C(=O)NC(C2CCCCN2C(=O)C=Cc2ccncc2)C)ncccc1Cl CC1(CNC(C2(CCO)CC2)=O)CCCN1C(c1cccc(C(F)(F)F)c1)=O C1(CC(=O)NC23CC(NC(CC4CC(=C)C4)=O)(C2)C3)C=CS(=O)(=O)C1 c1(SCCC)ccc(C(=O)NCC2(NC(=O)CC34CCCC3C4)CCC2)cc1 C1(NC(CN(C(C2(CC=C)CC2)=O)CCC)=O)CCn2ccnc2C1 C(=O)(C(C)(C)C)N1CC(c2cn(C3C(S(C)(=O)=O)CCC3)nn2)(O)C1.c1ccccc1 C1(CCNC(C2(C(CC)=O)CC2)=O)C(C)CCCN1C(c1coc(O)n1)=O c1(CNC(N2CC3(C(C)(C)CC3)C2)=O)c(Cl)cccc1[N+](=O)[O-] c1(CC(N2C(CNC(C(C)Cc3ccc(Cl)cc3)=O)CC2)=O)c(O)ncnc1O c1(C(N(C2CCCCC2)CCC(=O)OCC)=O)cc2n(c(=O)c1)CCS2 n1(CC(C)N(C(c2coc(C)n2)=O)C2CC2)cc(CNC(C2CC(=C)C2)=O)nn1 c1(NCC(C)(Cn2cccn2)NC(C2N(C)CCOC2)=O)ncnc2c1COC2 N1(C(C(CO)N(C)C)=O)CC(F)(F)CC1CCNC(c1cc2n(c1)CCC2)=O c1(C(=O)NC2(C)CC(NC(c3c(CC)c[nH]c3)=O)C2)cc2c(Br)cccc2[nH]1 N1(C(CC(C)OC)=O)CCCC2(CNC(c3cccc4occc34)=O)CCCC12 CC(N=c1cc2n([nH]1)CCOC2)c1nc(Cl)ccc1Br C1(C(=O)NCC#CCOC)C=CCN(C(c2ccc(SC)o2)=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)N(C)CC2CCCN(C(=O)CCN3CCC3)C2)n1 C1(NC(C(=O)NCC)C)COc2ccc(Cl)cc2C1=O C(C1=CCN(C(c2scnc2Cl)=O)CC1)NC(C1C(C)C1C)=O c1(C(=O)OC)c[nH]c2ncnc(N3CCOCC3C(=O)CC3CCCC3)c12 C12(NC(C(CC(C)C)O)=O)CCCCC1CN(C(c1nc3cnccc3s1)=O)C2 c1(C(=O)NC(C(C)NC(=O)Cn2nccn2)C)cnc2sccn2c1=O N1(C(C(CCC#C)O)=O)CCC2CN(C(=O)C=Cc3nccs3)CCC12 C1(NC(c2n(C)c(S)nn2)=O)CC2CCC1N(C(c1ncc(F)cc1F)=O)C2 C1(NC(C(C(C)(C)C)OC)=O)CCCCCN(C(=O)C=C(Cl)Cl)C1 N1(C(C(c2cccc(O)c2)C)=O)CC2CCC(C1)N2C(C1CCC2(CCC2)C1)=O c1(C(N2CCC(CN(C(=O)CSCCC#N)C)C2)=O)c(O)nnc2c1CCC2 Cc1c(C(=O)NC2CC(C)(CNC(=O)CCCCN(C)C)C2)cccc1O C#CCCCCCC(=O)NC1(C)CCC(C(=O)NOCC(C)O)CC1 C1(C)(C(N2CCC(CC=C)(NC(=O)CC(=O)NCC)C2)=O)CCNC(=O)C1 C1(SCC)CCCCN1C(=O)C(O)CCn1cc(-c2ccnn2C2CCC2)nn1 CC(C)(C)C(O)C(N)C(=O)N1CCCC(O)(c2cnn[nH]2)C1 C(CC(CC)C(=O)N1CC(C(=O)NOCC(C)(C)C)CC(C)C1)=CC N1(C(C2C(O)CCN2C(C2CC2c2ccc(F)cc2)=O)=O)CC2CCCCC2C1 C12(Nc3nc(CC)cc(CC)n3)CCCC1CN(C(C1(COC)CC1)=O)C2 c1(C(N2C(C(=O)O)C(c3ccccc3)CC2)=O)cc(Br)cc([N+](=O)[O-])c1 c1(NC(N2CC(F)(F)CC2c2ccc(C(F)(F)F)cc2)=O)c(O)ncnc1O C1(CCC2(OC)CC2)CC(C)N(C(=O)OC)C(NC(=O)OC(C)(C)C)C1 C1(NC(C2OCCN(C(CCCOCCC)=O)C2)=O)CCCCC1C#N c1(C(N2CC(CNC(=O)CCCc3nccs3)C3C2C3)=O)ccc(O)c(Cl)n1 C(CCSC)(C(=O)NC(C)CCC=C)NC(CCC#C)=O c1(C(N2C(C(=O)NC(CSCC)CO)CCCCC2)=O)cccn2ccnc12 C1(CNC(c2c(CC)c[nH]n2)=O)C2CN(C(=O)CC3CCC(=O)CC3)CC12 S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1C(C(=O)Nc2cnc(I)cn2)CC(F)(F)C1 CC(C)S(=O)(=O)CC(=O)N(C1CCN(C(C2CCc3cncn3C2)=O)C1)C CCC(Cc1cccc(C)c1)C(=O)NCC(C)CNC(=O)CCn1ccc(C)n1 N1(C(CN(C(C)=O)C)=O)CCCC(CNC(=O)CCN(c2ccccc2)C)C1 C1(CNC(CN(CCC#C)C)=O)CN(C(=O)C(C)(C)CSC)CC1O c1(C(=O)NCC(C)NC(=O)CCCCN2CCOCC2)cc([N+](=O)[O-])cc(=O)n1C C(=O)(C(F)(F)CC(C)C)N1CC(OC)(CNC(c2ccc(CO)cc2)=O)C1 N1(C(c2ccc(C#C)cc2)=O)CCCC1C1CCCN1C(c1cc[nH]c1)=O C1(C(=O)NCc2cncn2C2CC2)CCC(O)CN1C(c1cnc(S)nc1)=O C1(C)(C(=O)NCc2ccc(SC)o2)CCCN1C(c1ccsc1C#N)=O CC1CC(NC(=O)C2=CCCCO2)CN(C(c2cc(=N)[nH]c(=N)[nH]2)=O)C1 c1(CN2C(C(N3CCC(SC)CC3)=O)CC(O)C2)nc(C)c(C)cc1Br N1(CCCN(C)CCO)CC2CN(C(c3cnn(C4CCC4)c3)=O)CC2C1 N1(C(C2C(CC(=O)OC)C2)=O)CC(NC(=O)CCSCc2ccccc2)C(O)C1 C1(NC(CS(=O)(=O)NCC)=O)CC2(CCN(C(=O)C(CC)N(C)C)C2)C1 C(C(CC(=O)NC1CCN(C(c2ccc3oncc3c2)=O)C1)C(F)(F)F)N(C)C c1(CC)ccc(C(C(=O)NCCCOC)N(C)CC2CCCCC2)o1 C=CCC(C(=O)NC(C)C)NC.C1(=O)C(C)N1C.C(C)(C)(C)OC(=O)N(C)C C1(N(C)C(C2COCCO2)=O)CCC(NC(c2sccc2C#N)=O)CC1 N1(C(c2ccc(=O)oc2)=O)CCC2CCN(C(n3nnc4ccccc34)=O)C2C1 N1(C(c2cc(C(=O)NCC)no2)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 c1(CC(=O)NCC(c2cccc(C)c2)OC)c(F)cccc1Cl C1(C(=O)NC2C3(CC(NC(C(CN(C)C)(C)C)=O)C3)C2)CCC(N=[N+]=[N-])CC1 C1(CNC(C2(C(C)NC(c3cnsn3)=O)CC2)=O)(CO)CCCC1 Cc1nc(O)ccc1C(=O)NC(C)CN(C)C(C1CCN(S(C)(=O)=O)C1)=O C1(CC(N2CC(NC(c3nc(C)oc3)=O)C(C)C2)=O)OCCCC1(C)C O=S(=O)(NCC(C1CC1)C1CC1)N1CCC(F)(F)C1.c1(C(C2CC2)N)ccccc1 C1(CN(C)C(c2cc(CCCO)on2)=O)CCCN1C(c1ccc(C(N)=O)[nH]1)=O c1(NC(C23C(CN(C(C4(Br)CC4)=O)C2)C3)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C2C(C)(C)COC2)=O)CC2(C=C(C(=O)NCCC34CCCC3C4)CO2)C1 C(=O)(CCCC(=O)NC1CC(F)(CNC(C2CCC3(CCC3)C2)=O)C1)N(C)C N1(C(c2cnc(C3CC3)nc2)C(=O)NC(CC)C)CC(N(C)C)C(C)C1 c12cc(ccn1)NC2=O.C12(CNC(CC3(OCC)CCC3)=O)CCCCC1C2 C1(C)(C(N2CCCC(CN(C(c3cc(C)on3)=O)C)C2)=O)COC(C)(C)CO1 Cc1ccc2nc(SCC(N3CC(CNC(=O)CC4CCCCO4)C3)=O)[nH]c2c1 C1(CNC(c2ccc(Cl)s2)=O)CCCN(c2ccnc(N3CCCC3)n2)C1 Cc1ncn(C)c1C(C(=O)NC1CCC1)N(Cc1nccs1)CC1CCCO1 C=CC1(C(N2CC(OC)CC2CNC(C2COCCO2)=O)=O)CCCCC1 Cc1cnc(N(C2CCCNCC2)C(c2ccc(CO)o2)=O)nc1 CCCCC(O)CC(=O)NCCC1(O)CCN(C(c2ncc([N+](=O)[O-])n2C)=O)C1 c1(C(=O)NCCN(C(c2cnoc2C2CCC2)=O)CC)ccnc(CO)c1 NS(=O)(=O)c1ccc(C(N2CCOCC2CC(=O)Nc2sncc2C#N)=O)c(Cl)c1 c1(CCC)cc(C(=O)NC2COCC2CNC(=O)C(C)(C)c2cscn2)no1 N(C1CCCOc2ccc(F)cc21)C1(c2n(CC)nnn2)CC2COCC2C1 C1(NC(c2cc(OC)nc(C)c2)=O)CN(C(C2(C)CCCS2)=O)CCC12CCC2 c1(C(CC)NC(=O)CC2CCN(c3cc(C(C)=O)cnn3)C2)ccc2c(c1)OCO2 CC1CC(C)(NC(=O)C=CCN(C)C(C2CNC(=O)N2)=O)C1 c1(OC)ccc(Cl)cc1C(=O)NCCC1CC(NC(C2CC23CCCOC3)=O)C1 C1(C2CCN(C(c3c(C)nc(C)o3)=O)C2)(NC(C2CC3CCC2O3)=O)CC1 C1(CC(=O)NC(C2CCN(CC3(C)CC4CC4C3)C2)(C)C)CCCC1C1CC1 c1(C(N(CCCNC(=O)C(C)C2CCOC2)CC)=O)scnc1Br c1(C(=O)NCC2N(C(C3C(C=C)CC3)=O)CC(O)C2)cc(Br)ccc1OC Cc1ccccc1CNC(c1nnnn1-c1cccc(Br)c1)CC1CCCCC1 N1(C(C23CC(OC(C)=O)(C2)C3)=O)CC2(CCC2)CC1C(N1CCn2ncnc2C1)=O C(=O)(CCC(CF)CF)N(CC(=O)NCCC1CCOCC1)CC#C C(=O)(CCCC(F)(F)F)Nc1c(CN2CC(C)(CC(=O)OC)C2)nc(Cl)cc1 CC(CC(=O)N1CC(C(c2cn(Cc3nocc3Cl)nn2)C)C1)c1ccccc1 c1(-c2nc(Cc3nc(C(CC)(O)CC)on3)on2)cn2ccsc2n1 c1(CN(CCC)Cc2cnc(-c3ccccn3)s2)cccnc1 c1(C(N(CCCN(C)C(C2CC3(C)CC2CO3)=O)C)=O)onc2ccccc12 C(=O)(C1=CC2C=CC1C2)NCC1(O)CC(C(N2CC(C3CC3)(OC)C2)=O)C1 C#CC1CN(C(=O)CSCC(=O)OC)CCN1C(c1ccc(OC)nc1)=O c1(C(N2CCC(C)C(NC(=O)CSc3cn[nH]c3)C2)=O)ccc2nccn2c1 c1(C(N(C(C(=O)NCCC(C)SC)=O)C)C)cc2ccccc2o1.N1CCOCC1 CC(C(CO)NC(=O)CCSCC(N)=O)NC(=O)CCCOc1cccnc1 N1(C(CN2C(=O)NC(C(C)C)C2=O)=O)CC2(C1)CN(Cc1ccccc1)CCO2 C1(CNC(C2(F)CC2(F)F)=O)CCCCN1C(CCNC(N)=O)=O c1(C(N2CCC(O)(CNC(CSC)=O)C2)=O)nc(C)ccc1F N1(C(CCC(C)c2ccccc2)=O)CC2(C1)CN(C(=O)C1=CCCOC1)C2 c1(C(N2CC(=C)C2)=O)oc(CNC(c2ccc(CC)s2)=O)cc1C N1(C(Cc2nc(C)sc2)=O)CCC(F)(CNC(=O)C(C(C)C)N(C2CC2)C(C)C)C1 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)Cn2cc(C)cn2)C(C(C)(C)C)C1 c1(NCc2c(C)nc(-c3ccccc3Cl)s2)nccc(=NC(C)C2CCOC2)[nH]1 N1(C(C(=O)NC2CC(N(C(c3ncc(OC)cn3)=O)C)C2)C)CCP(C)(=O)CC1 C(c1ccc(N(C)C)cc1)=CC(N1CC(O)(CN(C(c2scc(C)c2)=O)C)C1)=O C1(C)(NC(C(COCC)C)=O)CCN(C(C2CCCS2)=O)CC1 N1(C(CCC(C)=O)=O)CC2(CC(NC(C3CCCCN(C)C3=O)=O)CO2)C1 C1(NC(c2cc(COC)no2)=O)CN(C(=O)CC2CC3(CCC3)C2)C2CCCC12 C1(NC(C(CC)NC(c2ccccc2)=O)=O)CC2CCC1CN2 C1(C(CNC(COC(C)C)=O)C)CCN(C(=O)C(C2(O)CCCC2)F)CC1 C1(C(N2C(CNC(C3C(OCC)C3C)=O)CC2)=O)C2Cc3ccccc3C12 c1(C(=O)NCC(=O)NCC(=O)N(C(C)CO)C)ccc(C#N)o1 N1(Cc2cncc(CCC)c2)CC2CN(C)CC2C1 C(C1c2ccccc2CCN1C(C1(OC)CC1)=O)NC(C1CCC(CC)O1)=O c1(C(=O)NC2CC(C)CN(C(=O)C(F)CC3CCCC3)C2)ccc(N=[N+]=[N-])cc1 C1(O)(CC(N2CC3CC(O)C2C3)=O)CCN(Cc2cc(-c3cccs3)[nH]n2)CC1 Cc1nc(O)ccc1C(=O)NCC1CCN1C(C1(CO)CC1(F)F)=O C1(C(N2CCC(OCCNC(C3CCC(=O)O3)=O)CC2)=O)CCN2CCOCC12 C1(C(N2C(CC)CCC2)=O)CN(C(=O)CC(=O)O)CC1(F)F NS(=O)(=O)c1cc(C(=O)NC2CCC2NC(=O)C=CC2CCCC2)c(Cl)o1 N1(C(C(C)C2CCCC2)=O)CC(CC(N2CCC(C(C)(C)C)CC2)=O)C2(CC2)C1 Cn1cc(C(N2CCN(C(=O)C(C)(F)F)C3CCC23)=O)c2cccc(Cl)c12 C1(NC(c2ccc(CC)s2)=O)CCCC(NC(=O)C(C)(C)CN2CCCC2)CC1 C1(=CC(=O)NC2(C)CCN(C(C(Br)=C(C)C)=O)C2)CCCCCC1(F)F C(C(C(C)C)NC(=O)CC1CCN(C(=O)Cc2cc[nH]c2)C1)NC(C)=O N1(C(CC(CCC)C)=O)CCOC2(C1)CN(C(=O)C1=C(C)OCCS1)C2 C(=O)(C1Cc2ccccc21)NCCCN(C(c1c(C)nc2sc(C)cn12)=O)CC CC(C)C(O)C(=O)NC(C(=O)N1CCC(CN(C)C)C1)C(C)C C(=O)(C(C)CC(F)(F)F)NCC1(NC(C=Cc2c(C)n[nH]c2)=O)CCCC1 C1(CNC(C=CCCC)=O)CCC(C)CN1C(=O)C(C)=C1CC1 C1(CN(C(C2CC(=C)C2)=O)C)CCCC(NC(=O)CCCc2ccc(Cl)cc2)C1 N1(C(CCC=CC(C)C)=O)CC(F)(F)CC1CCNC(=O)C(F)C(C)(C)O n1(CC(=O)NC2CN(C(C34CC3C4)=O)CC2C2CC2)cnc2c1CCCC2 CC(O)(C(=O)NC1COCC1C(=O)NC1CCN(S(C)(=O)=O)C1)C(F)(F)F c1(CC(C)(C)C)nc2cc(NCC3(C)COCCO3)ccc2o1 c1(CCC(=O)NCC2CCN(C(C3CC34CC(F)(F)C4)=O)C2)ccc(F)c(F)c1 C1(C)(NC(C(CCC)O)=O)CCCN(C(=O)CCCOc2ccc(C)cc2)C1 C(=O)(C1CCCc2ncccc21)NC(C)CNC(=O)CCC(C)(C)F C1(=C(C(=O)OC(C)(C)C)F)CCN(C(C2CCC(C)CO2)=O)CC1.CC(=O)O Cc1nc(C)n(CC(=O)NCCC2(O)CCN(C(C3(C#N)CCCO3)=O)C2)n1 C12(NC(C3CC(=C)C3)=O)CCN(C(=O)Cc3cccc(OCCCC)c3)CC1C2 N1(C(c2c(C#C)cn(C)n2)=O)CC2=C(C1)CN(C(c1cc(Cl)cc(Cl)c1)=O)C2 c1(C(N(C2CCN(C(=O)Cc3sccc3C)CC2)CC#C)=O)ccc(C)cc1Cl c1(C(=O)NC2(C)CCC(NC(C(C=C=C)C)=O)CC2)cccc2cnsc12 C1(CNC(C2C(C(=O)OC)C2)=O)CC2(CCN(C(c3cccn3C)=O)C2)CO1 Cc1ccc([N+](=O)[O-])cc1C(=O)NCC(CO)NC(=O)C(C)SC(F)(F)F C(=O)(CC(C)C(F)(F)C(F)(F)F)NC1(CNC(CCC(C)OC)=O)CC1 c1(-c2ccc(C)o2)nn(C)cc1C(C)Sn1cc(CSC2CCCC(C)C2)nn1 N1(C(c2nccc(OC)c2)=O)CCCC(F)(CNC(=O)CCC(C)(C)F)C1 c1(-c2cn(CCCCNC(=O)C(C3CCOCC3)F)nn2)ccc2ncsc2c1 CC(CCCC(=O)NCCCCC1CC1C)NC(=O)Cc1cc[nH]c1 c1(C(=O)NCC(COC)NC(C2C(C)C2(F)F)=O)ccc(C)cc1 c1(OC)ccc(C=CC(=O)NCC2C(C)CCCN2C(=O)CC(C)(C)F)cc1 Cn1cnc2c(-c3nnc(N4CCc5ccccc54)o3)nc(Cl)nc12 C1(C)(NC(=O)NCc2cccc(NC(c3c(C)cccc3)=O)c2)CCC12CCC2 c1(CCC(N2C3C(NC(C=C(C)C)=O)C(C3)C2)=O)cc(Br)ccc1C C(=O)(CCC(C)(C)F)N(C1CCN(C(=O)C(c2ccc(OC)cc2C)C)C1)CC C1(C(C(N2CCCC2C2CC2)C(=O)NCC)OC)CCC(F)(F)CC1 C1(CC(C)CNC(=O)NC2COC2)CCC(F)(F)CC1 C=CC(CC)C(=O)NC1CC(CNC(C2(CCC)CCC2)=O)CC1O C(=O)(C(CCC1CC1)NC(C1C=CCS1)=O)NC1(C)CC(O)C1 Cc1cncnc1C(=O)NC1CCC1C(=O)NCC(C)(C)C(N)=O c1(NC(C(COC)NC(C)=O)=O)cc(C)n(C2CN(C(=O)C(C)(C)C)C2)c1C C1(N(C(C(=O)N(C)Cc2onc(C)n2)=O)C)CCN(C2CCCCC2)CC1 CC(CCC(C)(C)C)C(=O)NCCCN(CC(c1ccc(F)cc1Cl)O)C1CC1 Cc1c(C(=O)NCCC2CCCN(C(c3c[nH]nc3C(F)F)=O)C2)cncc1Cl CC1=C(CNC(c2cccc(C)c2)C(F)(F)F)C(C)(C)CCC1 C1(NC(c2nccn2-c2cccc(-c3nc[nH]n3)c2)=O)CCC(F)(F)CC1 c1(C(=O)NCc2scc(C)c2)cc(CNC(=O)C(C)(C)C2CCCC2)nn1C c1(-c2c(F)ccc(OC(C)C)c2)cccc2c(C(=O)NC3CC3C3CC3)c[nH]c12 N1(C(C2C(C=C)C2)=O)CCOCC1CCNC(c1ccccc1C(C)(F)F)=O c1(C(N2CCC(O)(CNC(C(CC)SC)=O)C2)=O)ccc2ncc(=O)[nH]c2c1 C1(CNC(C2(CCC)CCNC2=O)=O)CN(C)CCN1C(=O)Cc1nc[nH]n1 N1(C(c2c(CNC(C=CC(=O)N(C)C)=O)nnn2C)=O)CCCC(N=[N+]=[N-])C1 c1(CC(=O)NC(C(CO)NC(CCC=CC)=O)C)ccnc(C(N)=O)c1 N1(C(C2CCC(=C)CC2)=O)C2CCC1CN(C(C1CC1C1CCOCC1)=O)C2 CC1SCCC1N=c1nc(N2CCN(C(=O)C(N)=O)CC2)c2ncccc2[nH]1 c1(C(=O)OC)cc(C(=O)NCC(F)CNC(=O)CC2(C)CC2)cc([N+](=O)[O-])c1 C(CC(C(C)(C)C)NC(c1ccccc1Cl)=O)N(C(CCOC)=O)C C1(NC(C2=C(C)CCC2)=O)CCOC2(CCN(C(c3cc(CO)[nH]n3)=O)CC2)C1 N1(Cc2c(C)nc(C)s2)CCS(=O)(=O)C(CCNC(c2cc(C)n(C)n2)=O)C1 c1(NC(=O)NC2(C(F)(F)F)CC2)nccc(NC(CC(=O)O)c2ccncc2)n1 C1(C(C(=O)NCC2(CO)CCCC2)F)CCN(C(c2ccoc2)=O)C1 CC1CCCC(C)N1CCCCSC.N12CCC1(CC)CC2 c1(OC)cc2nc(NC3CCCN(Cc4cccs4)C3)nc(O)c2cc1OC CCC(CC(F)(F)F)NC(=O)CC(CNC(=O)Cc1cnoc1)C1CCC1 c1(C(=O)NCCC2CN(C(C(CC=C)(C)C)=O)CC2C)ccc2oc(=N)[nH]c2c1 c1(C(=O)NC2CC(NC(c3n(CC)nnc3)=O)C2)c(F)ccc(C#N)c1F c1(C2(C)COC2)cn(CCCC(=O)NC(C2CCC2)C2CC2)nn1 c1(C(N2CC(O)(CNC(c3ccc(OC)s3)=O)C2)=O)cnnc(C)c1 C1(CN(C)C(c2cncc(CN(C)C)c2)=O)COCCN1C(C1COCCN1C)=O C1(CNC(CCc2c(C)noc2Cl)=O)CN(C(=O)C(C)N(C)C)CC1(C)C c1(C(C(=O)NC(C)C(CO)NC(=O)CSCCN(C)C)OC)ccc(Cl)cc1 N1(C(C2C(CC)CN(C(c3ccc4cncn4c3)=O)C2)=O)CC2C=CCC(C2)C1 N1(C(c2c(CC(=O)OC)scc2)=O)CC2CCN(C(=O)CCC(C)N(C)C)C2C1 CCC(CCOC)C(=O)N(CC(N1CC2(CC2)C1)=O)C1CCC1 Cc1ccc(C(=O)NCc2cn(CCN3CCOCC3)nn2)c(Cl)c1 C1(NC(CCc2ccc(CC)cc2)=O)CCN(C(C2CC23CC3)=O)CC1F C12(C(=O)NCC3(F)CCN(C(=O)COc4ccsn4)CC3)CCCCN1CCC2 Cc1oc(C2CC2)nc1C(=O)NC1(CCO)CN(C(C2(F)CCOC2)=O)C1 N1(C(C(n2cc(Cl)cn2)C)=O)CC2CCCC(C1)N2C(=O)C(C#N)CC1CC1 C1(CCNC(C2CC(=O)OC2)=O)CN(C(C2(CF)CCOCC2)=O)CCO1 C1(NC(C2(C)CCCC2)=O)CCN(C(=O)Cc2cccc(N)c2N)CC1F CCC(CC(C)C)C(=O)N1CC(C(=O)NCC2CCC2CO)C(F)(F)C1 CCC(C)(CC)C(=O)N1CCOC(CNC(C2(C#N)CC3(CC3)C2)=O)C1 C(C(O)CS(=O)(=O)c1cccs1)NCC(c1c(F)cccc1F)C CCCCC(=O)C(=O)NC(C(=O)NCc1c(F)cccc1F)C1CCOC1 CC1CCC(=CC(=O)NCC2(CNc3cn(CC(=O)N(C)C)nn3)CC2)C1 Cc1cc(C(=O)NC2CC(NC(=O)CCOC3CC3)C(O)C2)ccc1O c1(SC)cc(O)ccc1NC(=O)CC1CCCN1C(=O)Cc1ccccc1O C(C)(C(C)C(=O)N1CC(OCCO)C1)NC(c1cc(OC)n[nH]1)=O C1(N(C)C)CCCC(C(=O)OCN2CCCC2NC(=O)C(c2ccccc2)F)C1 CCCC(C)C(=O)N1CC2C(N(C(=O)CCOC3CCCCC3)C)C2C1 C1(NC(C(N2C(CSC)CCCCC2)=O)=O)CC2(CCC2)C12CCC2 Cc1nc(N2CCCC(CNC(c3ccno3)=O)CC2)c(C)c(Cl)n1 C=CCCCCCCCC(=O)NC1CN(C(=O)Cn2ncn(C)c2=O)C(C)(C)C1 N1(C(C(c2ccc(F)cc2)=O)=O)CCCC2(NC(C3CCCCCC3)=O)CC2C1 N1(C(C=CC(C)NC(=O)C2=C(Cl)CCOC2)=O)C2CCCC1CN(C)C2 c12ccc(cc1)-c1n[nH]c(n1)C1CC21.C(c1cccnc1)=CCNC c1(-n2c(C(C)(C)CC#N)nc(CN3CCC(O)CC3)n2)ccc(F)cc1C(F)(F)F C=CCN(OC)C(=O)C(F)CC(C)(C)NC(c1ncccc1Cl)=O CCC(C)(COC)CNC(=O)CCCCNC(=O)C(C)NC(=O)OC C1(F)(C(=O)NCC(O)CC2CCCC2)CCCN(C(c2cc3n(n2)CCC3)=O)C1 N1(C(CC(C=C)CC)=O)CC(C)CN(C(c2cnn(CC(C)C)c2)=O)CC1C Cc1ccc2ncc(C(=O)NCCC3CN(C(c4ccnnc4O)=O)C3)cc2c1 CCCC(CNC(C1(C#N)CCC1)=O)C(=O)NC(C(C)C)C(C)C Cc1nn(C(C)C)cc1C(=O)NC1CC1NC(C1CC1C)=O c1(C(=O)NCCCC(C)(C)NC(C2CCCN(C)C2)=O)cc(N)c(F)c(F)c1Cl CC1C(NC(=O)C2=CCC2)CCN1C(c1cc(C2CC2)cs1)=O C1(NC(CC(CCC)C)=O)CC(C(=O)N(c2ccccn2)CC(C)C)=CC1O c1(C(C)O)cc2ccccc2[nH]1.C12(C)CN(C1)C(=O)C1CCN1C(=O)CC2 N1(c2ncnc(C)c2Br)CCC2CCC(C1)N2C(c1cn2c(n1)CCC2)=O C1(NC(c2cc(F)n[nH]2)=O)CN(C(=O)C(F)n2cccn2)CC1O c1(C(=O)OC)ccc(C(N2CCC(N(C(=O)C(C(C)(C)C)SC)C)C2)=O)cc1F c1(NC(N(CC(C)NC(=O)OC(C)(C)C)C)=O)ncccc1Cl C1(c2cn(C)nc2)CN(C(c2ccoc2)=O)CCN1C(c1cc(C(N)=O)co1)=O N1(C(CN(C(C)=O)C)=O)CCC(C2CC2)(NC(=O)CN2CCN(C3CC3)C2=O)C1 n1(CCCC)nc(C(N2CC(NC(C3CC(C)=NO3)=O)C3CC3C2)=O)ccc1=O N1(C(=O)NC2C(C(C)(C)C)C2)CCC2CC(O)CCC2C1 c1(C(C(=O)NCC=C)N(C)Cc2ccc(NC(C)=O)cc2)ccc(Cl)cn1 O=C(O)C1=CCC(NC(c2ccn(C3CC3(F)F)n2)=O)C1 C1(C(=O)NC(C=C)(C)CC)C2CC(O)C(C2)N1C(C1CC2CCCC2C1)=O C1(NC(c2cc(CC)no2)=O)CC(NC(C2(COC)CC(F)(F)C2)=O)C12CCC2 CC(c1cccc(Cl)c1)=CC(=O)NC1(C)CCN(C(=O)CS(N)(=O)=O)C1 C1(C(=O)NCC2(COC)CCC2)CN(C(c2c[nH]nc2C)=O)CCO1 C(CN=c1[nH]ncs1)OCCNC(CS(=O)(=O)NC)=O Cc1ccc(NC(=O)CC2CCCN2Cc2cnn(C)c2C)c(F)c1 N12CCC3(CC1)CC(C3)NC2=O.c1(Oc2cnoc2)ccccc1[N+](=O)[O-] CCCC(C)(C)CC(=O)N1CC(NC(=O)C(C2CCC2)C2CCC2)CCC(O)C1 C1(C(=O)NC2(CN(C)C(c3ccc(C(N)=O)cn3)=O)CC2)OCC2CCCC12 CC1=C(C(=O)NC2(C(N(CCC(C)N(C)C)C)=O)CCCCC2)CCC1 C=CCCCC(C(=O)NCC(C1CCCCC1)O)NC(C1CC(=O)N(C)C1)=O N1(C(CC2(OC)CCC2)=O)CCN(C(c2cc(C3CC3)ccn2)=O)C(CCO)C1 C1(O)(CC)CCCN(C(C2(CC)CCCN2C(C2CCCCCC2)=O)=O)C1 C(=O)(CCC=CBr)N(CC(C)NC(=O)Cn1ccc(C(F)F)n1)CC c1(C(=O)NCC(CO)NC(CNC(C)=O)=O)cc2c(ccn2C)s1 C1(NC(=O)NC2CCN(CP(C)(C)=O)C2)Oc2ccccc2NC1=O C1(C#N)(N(C(CCCC#C)=O)C(C)(C)C)CCN(C(c2cc(F)ccc2C)=O)C1 C=CC1(C2(C(=O)NC(C3CCN(C(c4c(C)cnn4C)=O)C3)C)CCC2)CCC1 CCCC(CCC)=CC(=O)NC1(CO)CCN(C(=O)C(C)(C)C2CCO2)C1 c1(CCC(=O)NC2(CF)CCN(C(CCC(C)C)=O)C2)nc2ccccc2[nH]1 c1(C(N2CC(CNC(=O)CN3CSCCSC3)C2)=O)cccc2occc12 C1(NC(CCCN(C(=O)CCC(F)(F)F)C)=O)CC2(C1)CC2(F)F N1(C(C(C)SC)=O)CCOC(CNC(=O)CC(c2c(C)n[nH]c2C)C)C1 c1(-c2cn(CC3CN(C(CN(C)C(N)=O)=O)C3)nn2)ccn(C)c(=O)c1 c1cc2c(NC3C4CCCCCC34)[nH]c(=NCCn3cncn3)nc2s1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC2(CNC(C2(C(N)=O)CC2)=O)C1 C(CCCCCC(=O)NC(c1ccccn1)CO)NC(c1ccc(SC)o1)=O c1(C(=O)NCC2(F)CC(NC(CC(C)C)=O)C2)cccc(C(C)C)c1F C(=O)(C(C)(C)CCS(C)(=O)=O)N(CCCN(C(C(=C(C)C1CC1)F)=O)C)C c1(OC)ccc(C(C)=CC(=O)NC2CCC(C)(NC(c3cnsn3)=O)CC2)cc1 CN(CC(O)CN1CCCC1)N1CC2CN(CC(F)(F)F)C2C1 N(C1CCCc2occc21)C(C1(n2cnnn2)CCOCC1)=O C(=O)(C(F)(F)CCC1CCC1)NCCN(C(C(c1ccccc1)OC)=O)C1CC1 c1(C(N2C(C)C(C(=O)NCC(C)(O)CCO)CCC2)=O)ccc2ccoc2c1 n1(NC2CC(C)(COCC3N(CC)CCCC3)C2)ncc(O)nc1=O c1(C(C(=O)NC(CNC(C2(CC(=O)OC)CC2)=O)CO)C)ccc(Br)s1 c1(CC(N2CC(N(C(C(CC)N(C)C)=O)C)C2)=O)nnc(O)c2ccccc12 CC(=NOCC#N)C(=O)N1CC(CNC(C2NC(=O)OC2C)=O)CC1C C1(OC)(CNC(c2ccnc(C3CC3)c2)=O)CCN(C(c2cnc(Cl)s2)=O)C1 C1(CNC(=O)CC2(O)CCC2)CC2(CCN(C(c3csc([N+](=O)[O-])c3)=O)C2)CO1 C(=O)(C(C)(F)C(F)(F)F)NCC1(O)CCCN(C(c2c(CC)ccs2)=O)C1 C12(C(N3CC(NC(c4scc(C)n4)C)OCC3)=O)CCC(CC1F)C2 N1(C(c2cc(Br)ccc2C)C(=O)NCCOC)CCC(F)(F)CC1C C#CCC(CC(=O)NCCCCCCCOC)NC(c1ccsc1Cl)=O C(=O)(C#CC1CCCO1)N1CC(O)CC(NC(c2cc(=O)cc[nH]2)=O)C1 Cc1nc(O)ccc1C(=O)NCC(CNC(c1ccc(C(C)C)c(F)c1)=O)CO c1(C(=O)NCC2CC(C(N3CC(COC)OCC3)=O)C2)ccc(C)c(C)n1 C1(C)(C(=O)NCCCCC(C)NC(c2c(C)nccc2)=O)CCC(=O)NC1 C1(CN(C(c2c(OC)ccs2)=O)C)CCCC(NC(=O)CCc2cnco2)C1 C1(C(C)NC(c2nocc2Cl)=O)CCCCN1C(=O)C(=O)N(CCC(N)=O)C1CC1 CC1(C)CCC(CNC(=O)CC2CCCCN2C(=O)COC2CCOC2)CC1 c1(CC(C)C)n[nH]c(=NCCC2CCN(C(=O)CCc3cc(F)ccc3F)C2)s1 C1(NC(CCc2n(C)ncc2)=O)CCN(C(c2ccoc2Br)=O)C12CC2 C(CC(C)C(=O)NCC1CC(O)CN1C(c1[nH]c(O)nc1C)=O)=CC C(=O)(C(C)C(C)NC(=O)OC(C)(C)C)OCCC(=O)NCCO.C(CC(C)C)=CC c1(NCc2n(C)c(-c3nn[nH]n3)cc2)cc(Cl)ccc1OCC(F)F c1(CC(=O)N(CCCNC(C(CCC)O)=O)CCO)ccc(OC)cc1Br CC(C)(C)CC(O)CC(=O)NC1CC(C)(NC(=O)COCc2nccs2)C1 C12(NC(c3ccc(C)s3)=O)CCC(CN(C(c3csc(C)c3C)=O)C1)C2 CC1CN(C(=O)Cc2ccon2)CCC1NC(c1cc(Cl)ccc1C(F)(F)F)=O C1(OC)CCCC(CC(=O)NCC(C)CNC(c2ccc(C3CC3)cc2)=O)C1 N1(C(C(CCCC)NC(N)=O)=O)CC2=C(C1)CN(C(=O)C=CBr)C2 c1(C(=O)NC2C(NC(c3c(C)nsc3)=O)CC2)cccc(-c2nnco2)c1 C(C(C(=O)NCC1CC1[N+](=O)[O-])NC(=O)CCOCC1CC1)N(C)C C1(C(=O)NCC2N(C(c3ncc(C(=O)OC)nc3)=O)CCC2)C(F)(F)C12CCC2 C12(C(=O)NCc3c(CC)nns3)CCCC1CN(C(=O)C(C)(C)C#N)C2 c1(OC)cc(Br)ccc1CC(=O)NC1C=CC(C(=O)Nc2ccc(Cl)cc2O)C1 C1(F)(CNC(=O)C=CC(=O)NC2CC2)COCCN(C(C2COC(=O)C2)=O)C1 c1(CC)cncc(-c2nc(CCCSC)n[nH]2)n1.c1(C2CC2)ccccc1 C12(NC(CCCN(C)C)=O)CC(CNC(=O)C(F)OC(F)(F)F)(C1)OC2(C)C C1(CNC(=O)CC2COCCO2)CC2CCC1N(C(c1ncnc(O)c1Cl)=O)C2 C1(NC(C(C)(C)OCC)=O)CC(CN(C)C)CC1O.c12conc1C(=O)NC2 c1(C(=O)OC)ccc(OC(c2c(C)nn(CC(C)C)c2Cl)=O)c(Br)c1 Cc1coc(C(F)(F)F)c1C(=O)NCC(CC(C)C)NC(=O)CN1CCOCC1 Cc1nn(C)c(C)c1CC(=O)NCC1(C)CCC(NC(=O)C(O)C2CCC2)CC1 N1(C(C2C(CC(C)C)C2)=O)CC(NC(c2coc(CS(C)(=O)=O)n2)=O)CC(F)C1 c1(C(=O)NC(C2CCN(C(C3CCCC3O)=O)CC2)C)snc2ccccc12 C(C1=NOC2CN(C(c3nnc(O)nc3O)=O)CC12)NC(C1(SC)CC1)=O c1(COC(C2(c3ccc(Cl)cc3)CCCC2)=O)c(F)ccc(F)c1F Cc1c(NC(c2c[nH]nc2CCNC(=O)C(C(C)O)N(C)C)=O)cnn1C c1(CC(N2CCC(NC(C(CC)C3CCOCC3)=O)(CF)C2)=O)c(F)cccc1Cl C1(C(=O)OC(CCC)CC)CCC(F)(C(=O)OC(C)(C)C)C1 C1(CC(C)NC(=O)CC2CC2(C)C)CCN(C(C2CC(N(C)C)C2)=O)CC1 C1(C(=O)NC(C(=O)NC)C2CC2)COC2(C1)CN(C(=O)C1=CCCSC1)C2 c1(NCC2N(C(=O)C=CI)CCC2)ccnc2ncnn12 N1(C(COC2(C)CCC2)=O)CCC(CCNC(C2OCC2(C)C)=O)CC1 C1(NC(c2nncc(C)c2)=O)CCC2CN(C(=O)CCc3cnn[nH]3)CC2C1 C1(C(=O)NCC2(CNC(c3ccc(C#C)o3)=O)CCOCC2)CC(=O)NC1(C)C N1(C(CNS(C)(=O)=O)=O)CCC(N2CCC(NC(=O)CCC(F)F)CC2)CC1 N1(CC(=O)N(C2CCC(NC(C3(CC)CC3)=O)C2)C)CCC(=O)NC1=O C(=O)(C1=C(C)CCCC1(C)C)N(CC(C)NC(C1CCCCC1SCC)=O)CC C1(CNC(CC(C)(C)OC)=O)CN(C(c2ccc(C)nc2O)=O)C2CCN1C2 c1(C(N2CCC(NC(C#CC(C)C)=O)C(O)C2)=O)ccc2c(=O)n(C)cnc2c1 C1(CC(=O)OCC)CCC(NC(C)=O)C1.n12nnnc1C1(CCC1)NCC2 C1(C)(C(N(CC(C)NC(C(CC)(C)F)=O)C)=O)CC2CCC1CC21OCCO1 C1(C(=O)NCCCN(C(=O)Cc2ccoc2)C)CC(c2cccc(Cl)c2F)=NO1 C1(C)(CNC(COCC)=O)CC(F)(F)CN1C(C1CCc2n[nH]cc2C1)=O c1(C(=O)NC2(C)CCCN(C(CNC(CC)=O)=O)C2)ccc(S(=O)(=O)CC)cc1 c1(C(N2CCC(C)(C(=O)OCC)C2)C(=O)NC(C)(C)CC)cc(Br)ccc1C c1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)O3)=O)C2)cc2ccccc2cn1 Cc1cccn2cc(C(N3CCC(C(C)NC(=O)C(F)n4ccnc4)C3)=O)nc12 C(=O)(CC(C)(C)C#N)N1CCC(C(C)(C)CN(C(=O)C(F)OC(F)(F)F)CC)CC1 Cc1cc(C(=O)N(C2CC2)CC2CCCN2C(c2ccc(C(C)C)o2)=O)nc(C)n1 c1(C(=O)NC2C=CCN(C(=O)CC3CCSC3)C2)occ2c1CCC2 c1(N(C(c2ncsc2Br)C(=O)NC)C)ccc(NC(=O)OC(C)(C)C)cc1 c1(C(C(=O)N(C)CC2CN(C(=O)CC3CSCCS3)C2)O)cc(F)cc(F)c1 Cc1c(C(=O)NC2CN(C(=O)CC3C=CCC3)CC2C)ncn1C N1(C(C2N(CC)CC2)=O)CC(CNC(=O)CC2CCC(C)(C)O2)C(C)C1 CCC(C)C(O)C(=O)NCC(CNC(C1CC=CC1)=O)S(C)(=O)=O c1(NC(=O)CCc2cccnc2)cnc(SCC)nc1.CC1CCC1N(C(=O)C)C c1(C(=O)NC2CCC(CNC(c3cc(Cl)c(Cl)[nH]3)=O)CC2)ccc2cccnn12 CS(=O)c1cccc(C(N2CC=C(CNC(C3(Br)CC34CCC4)=O)CC2)=O)c1 C1(CC)CCN(C(=O)CC(C)C2CC2)C(C(=O)NC2CC(CCF)C2)C1 C1(CNC(c2ccn(CC)c2C)=O)CN(C(=O)CNC(=O)C(C)(C)C)CCC1C c1(CNC(CCCCC#C)=O)nnc2n1CCN(C(=O)C(O)CCCC)C2 C1(C(N(C2CCN(C(=O)CCc3nc(C)no3)C2)CCC)=O)CCCC1C(C)C c1(C(N(CCCCNC(C2CCCCC2(C)C)=O)C)=O)c(F)ccc(O)c1F N1(C(C(C)NC(C)(C)C)=O)CCN(C(c2ccn(CC(F)F)n2)=O)CC1CO c1(C(=O)NCCC2CCCN(C(C(C)CN(C)C)=O)C2)cn(C)c(=O)n(C)c1=O N1(C(=O)CCN(CCO)Cc2ccccc2Br)CC2CNCC2(CO)C1 C#Cc1cn(C)nc1C(=O)N(C1CCCC(NC(c2cncs2)=O)C1)C CC(C)(C)C(O)CONC(=O)COC1CCN(C(c2ncc(F)cn2)=O)C1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C(C)NC(c2ccccc2F)=O)OCC1 N1(C(CC(CC=C)NC(c2ncc(F)cc2N)=O)=O)CCOCCCC1C C1(NC(c2nnc(CC)s2)=O)CCCN(C(=O)CCc2cc(C)[nH]n2)CC1 C1(NC(CN(C2CCC2)C)=O)CCOCC1NC(=O)CCn1cnccc1=O c1(Cn2ncc(C(=O)OCC)c2)nc(C)c(C(N2CC(F)CC2C(F)(F)F)=O)s1 c1(OCC)ncccc1C(=O)NC1CCCC(C(=O)NOCCCF)C1 C1(N(C(CCOCCOC)=O)Cc2cccnc2)CC(C#N)C1.C1(=O)CN1 C1(C(N2C(C)(C(C)C)CC2)=O)CCCCN(C(=O)C(C)S(C)(=O)=O)C1 N1(C(C(CCC#C)O)=O)C2CCCC1CN(C(C1(Cc3ccccc3)CC1)=O)C2 c1(C(=O)NCC(CNC(c2cc(C)[nH]n2)=O)(C)C)ccc2c(n1)CCC(C)(C)C2 c1(C(=O)Nc2cc(-c3ccc(C(F)(F)F)cc3)cs2)cncc2cnccc12 c1(CC)ncccc1C(=O)NC1CCCC1C(=O)NC(C(N)=O)C1CCCC1 c1(CN(C(=O)CC2(C(N(C3CCOCC3)C)=O)CC2)C)cccc(CO)c1 N1(C(c2cn(CC=C)nn2)=O)CCC(O)(CCNC(C2C=CCCC2)=O)C1 C1(C2CCN(C(=O)C(O)C3CCC3)CC2)(NC(=O)CNc2ccccc2Cl)CC1 C=CCC(CC(=O)N1CC2CC2C2CC12)NC(=O)COC1CCCC1 C=CCC(C(=O)N1CC(NC(c2ccc(N(C)C)cc2C)=O)C(O)C1)C(C)(C)C c1(CN(CCC#N)C)ccccc1.C12CN(C1)OC(=O)C2 N1(C(C(CC=CCC)C)=O)CCC2CN(C(=O)C(=CC3CCCC3)C)CC2CC1 c1(C(=O)OC)cccc(CSCCC2CCOC2)c1O C(CCCCC(=O)NC1(C(=O)NCCc2csnn2)CC1(C)C)OCC Cc1nc(C2CC2)ccc1C(N1CCOCC1CN(C(=O)Cc1nc[nH]n1)C)=O c1(C(=O)NC(C(N2CC3COCC3C2)=O)C2(C)CC2)c[nH]c2nccc-2c1 CC1(C(N2CCC(C)(NC(=O)CC3COC(=O)C3)C2)=O)CNC(=O)C1 c1(NC(c2ccoc2)C)nccc(NC(CCO)c2nccs2)n1 C1(NC(c2nnn(C)c2N)=O)C2CC1CN(C(=O)Cc1cc(F)ccc1Br)C2 C1(NC(c2ccc(C)c(O)n2)=O)CC2CC(C1)N(C(C1C=CCS1)=O)C2 c1(N(CC(C)NC(c2coc(C(F)F)c2)=O)C)ncnc2c1ncn2CC1CC1 C1(CC)CN(C(=O)CNC(C2CCCN2C(C)=O)=O)CCN1C(=O)CCC(C)C c1(OC)ccccc1C1(C(=O)NC2CCC(NC(=O)CSC)CC2)CCCC1 Cc1cccc(C(=O)NC2CN(C(=O)CC3SC(=N)NC3=O)CC2O)c1Cl C(CN=c1[nH]c(=N)[nH]c(=NCC(C)c2nccs2)[nH]1)NC(=O)OCC Cn1cc(C(=O)NCCNC(C2CCCC3(C2)CC3(F)F)=O)c(=O)n(C)c1=O C1(C(=O)NC2(C)CCCN(C(=O)COCCF)C2)OCC2CCCC1C2 c1(C(=O)NC2CN(C(CCN(CCCCC)CCC)=O)C2)nc(O)nc(O)c1F CC1(C)CCCN(c2nnnn2C2(c3ccccc3Br)CCC2)C1C(N)=O C1(C(=O)NCCCN(C(=O)Cn2cnnc2O)C2CC2)CN2CC3CC2(CO1)C3 C(CC#CCO)NC(C(N(C(=O)C(C)(C)C1CC1)C)C1CC1)=O Cc1cc(C(=O)NC2CC3(C2)CC(NC(c2cccn(C)c2=O)=O)C3)cc(O)n1 N1(C(C2(CNC(=O)Cn3ccnn3)CC2)=O)CCCC2(COC2)C1 Cn1nc(C(=O)NCC2CC23CCN(C(=O)CNC(N)=O)CC3)c2c1CCC2 N1(C(C(C(C)C)NC(Cc2c(C)n[nH]c2C)=O)=O)CC2CCCCC2C1 S(=O)(=O)(c1ccc(F)cc1F)N(C)CCNC1CCC1(F)F c1(C(=O)NCCC2(NC(C(C3CCCCC3)OC)=O)CC2)ccc([N+](=O)[O-])cc1 N1(C(c2nnc(-c3cccc(F)c3F)o2)=O)CCCc2cncc(Cl)c21 N1(C(c2sc(C)c(O)n2)=O)CCCC2C(NC(=O)CCC(C)(C)F)C(C)(C)C12 CC1(C)CC1(C)C(=O)NCC1(CNC(c2cc(Br)n[nH]2)=O)CCC1 c12ccc(s1)S(=O)(=O)NC2.C1(NC(c2cccs2)C)CN2CCC1(F)CC2 N1(C(C(n2cc(Cc3ccccc3F)nn2)C)=O)CCC(C(=O)O)CC1(C)C C(=O)(C(O)C(C)(C)C)NCc1cn(CC(=O)NCC(C)CC2CC2)nn1 c1(OC)nccc(Br)c1C(=O)NC1(CO)CN(C(c2cncc(C3CC3)c2)=O)C1 C#CCC(C)(C(=O)NCCOCC(F)(F)F)N(C(=O)C(C)C1CC1)C1CC1 Cc1nn(C)c(C)c1COC(=O)C(O)Cn1cncn1 c1(Cn2c(C)cc(C)n2)c(Cl)cccc1Cl.c12cn(nn1)C(C)C(=O)N(C)C2 Nc1nc(Cl)ccc1C(N1CC2CC1C2NC(c1ccc(Br)o1)=O)=O Cc1ccc(C(=O)NC2CCCCC2NC2CN(c3ncncc3F)C2)nc1O C1(CNC(=O)C=C2CCC2)CC(C(F)(F)F)CCN1C(C1CC2(CCC2)CO1)=O CC1CN(C(=O)CC2CCCC2NC(c2ccncn2)=O)CC(C)(C)O1 c1(C(=O)NC(C2(O)CN(C(C(C)c3cc[nH]n3)=O)C2)C)cn2c(n1)COCC2 N1(C(C(C)OCCC=C)=O)CCCC1CNC(C1CCC(F)C1)=O C1(C(=O)NCCCN(C(=O)CSCC(C)C)CC)C2CCCOC12.CCOC C1(C(=O)Nc2c(C)cccn2)CN(C(c2cc(F)c(F)cc2I)=O)CCC1(F)F C(=O)(C1CCCc2sccc21)NCCN1CCN(C(C2C(C)C2C)=O)CC1 Cc1cc2c(o1)CC(C)(C)CC2NCCNS(=O)(=O)CC1(CC#N)CC1 CCCC(O)(CN1CCC(C(CO)CO)C1)C(F)(F)F CC(C)C(F)C(=O)N1CCC(NC(=O)C(c2ccc(F)cn2)(F)F)C1C n1(CC)nc(C(=O)NC2CCCCC2CC(=O)NCc2cc(C)nn2C)cc1O C1(NC(c2ncc(OC(C)C)nc2)=O)CCN(C(=O)CC#N)C(C2CC2)C1 C1(C(=O)NC(C)CN(c2cc(Cl)nc(C3(C)CC3)n2)C)CNC(=O)CC1C N1(CC(=O)NCC2CC(NC(C3(COC)CCC3)=O)C2)CCCNC1=O C1(NC(C2C(NC(Cn3c(C)nc(C)n3)=O)CCOC2)=O)CC2(C1)CN(C)C2 C(=O)(CC(C)C(F)(F)F)NCCC1CC(OC)CN1C(c1cnc(C)s1)=O CC(CC(F)(F)F)C(=O)NCCC(O)CNC(=O)C(F)(F)C(C)(C)O Cc1c(C(=O)NCC23CCC(CC2)N3C(=O)C(O)C2CC2)c(C(F)(F)F)nn1C Cc1nc(Cl)ccc1CCC(N1CCC(C(C)NC(C2(O)CC2)=O)CC1)=O c1(CC)cc(C(=O)NCc2csc(CNC(C3CCC(OC)C3)=O)n2)nn1C N1(C(c2c(CC)cco2)=O)CCC2(CC1)CC2NC(=O)CN1CC=CC1 C12CCN(CC1CC)C2=O.c1(NC(C(CC=CC)C)=O)c(CO)cccc1C N1(C(CC2(C)CC2(F)F)=O)CCCC(N(C(=O)CN2CCCCC2)CCO)CC1 c1(NC(C)(C)CC(=O)N2CCCCC2)ccc(S(C)(=O)=O)cn1 C(=O)(C1=CC(O)C(NC(=O)CNC(=O)CNC(C)=O)C1)NCCS(CC)=O C=CC1CCN(C(=O)C(C2(O)CCCCC2)NC(c2cc(C)oc2CC)=O)C1 c1(OC)ccc([N+](=O)[O-])c(C(N2CCC(NC(c3cnns3)=O)C(CO)C2)=O)c1 C12(C(N3CCC(CNC(CC(C=C)(C)C)=O)C3)=O)CCC(CC1)C2(C)C C(=O)(CC(C)CC(C)(C)C)NCCC(C)N(C(c1ccc(C#C)cc1)=O)C C1(NC(C2(CC(=O)OC)CC2)=O)(COC)CCN(C(C2(F)CCCCC2)=O)CC1 CCCCCC(CC)C(=O)N1CCCC(NC(C2CN3CCC2CC3)=O)CC1CC C12(CNC(c3ccncn3)=O)CCCCC1N(C(c1ccc(F)nc1)=O)CC2 C#CCCCC(C)C(=O)NC(C1CCCC1)CNC(=O)C=Cc1cncn1C C1(C(=O)NOC2CCOC2)CCN(C(=O)c2cnc(S)nc2)O1 c1(CNC(C(C)C)=O)nnc2n1CCN(C(=O)Cc1ccc(Br)cc1)C2 c1(C(=O)NCC2(NC(C3CCCN3C3CCCC3)=O)CC2)ccncc1Br c1(NC(C2CN(Cc3cc(B(O)O)co3)C2)=O)nc2cc(Cl)ccc2s1 C=CC(C)(O)CC(=O)N1CC(N(C(=O)CS(=O)(=O)N2CCCCC2)C)C(O)C1 Cc1cc(-c2cn(CCC(=O)NCC3OC(=O)NC3(C)C)nn2)cc(C)n1 C12(CC)CCC(C(N3CCC(CNC(c4ccncc4F)=O)(OC)C3)=O)(CO1)C2 C#Cc1ccc(NC(=O)Nc2n[nH]cc2C(=O)NC2CC2)cc1 C(=O)(C(F)(F)C(F)(F)F)NCC1CCCC(NC(c2ccc(N(C)C)cn2)=O)C1 c1(OCCC)ccccc1CN1CC2C(C1)N2C(C1CCC(F)(F)C1)=O C1(C(=O)NCC(C)(C)n2ccnc2)CC2(CC2)CN1C(C1CC2(CC2)C1)=O C(=O)(C(F)CCC(C)C)N1C(CN(C(c2cc(C)cc(C)c2)=O)C)CC(F)C1 c1(C(=O)NC(C)CN(C)C(C2(C#N)CC2)=O)ccc(Cl)c(Br)c1F C1(C(=O)NCC(CC)NC(c2cc(C)c(C)o2)=O)CCCN(S(N)(=O)=O)C1 CC1(CCNC(c2ccns2)=O)CCN(C(C2CCC(=O)N2C2CC2)=O)CC1 N1(C(C=CCC)=O)CCCCCC1CNC(c1c(Cl)cncc1Br)=O C1(NC(C)=O)COCCC1NC(c1ccc(-c2ccccn2)nc1)=O C1(NC(COCc2ccc(C)s2)=O)CCOCC1NC(=O)Cc1cncnc1O C1(N(C(CN(C)C)=O)CC2CC2)CCN(C(=O)C(COC(C)(C)C)N(C)C)C1 C#Cc1cccc(CCCC(=O)NCCNC(C2CC3(C)CC2CO3)=O)c1 N1(C(C=CCOC)=O)CCN(C(c2csc(Br)n2)=O)C(C(C)C)C1 Cc1cnc(Cl)cc1NC(C1(C)CCN(C(c2ccc(F)c(O)c2)=O)CC1)=O CC(CC(C)(C)O)N1CCC(CNC(C2(c3ccc(F)cc3)CCCC2)=O)C1 C(CCCC(=O)N1CCC(O)C1C(C)(C)C)NC(C(C)SC(C)C)=O C=CCCCCN=c1nc2ncn(CC)c2c(NCC(C)C(=O)N(C)C)[nH]1 Cc1cc(C(=O)NC2(CNC(=O)CNC(=O)CC(F)(F)F)CC2)nc(O)n1 c1(C(=O)NCC2(NC(C(CCOC)C)=O)CCC2)ccc2[nH]c(=N)oc2c1 N1(C(C2CCCC(C)CC2)=O)CCCN(C(c2ncccc2N)=O)CCC1 C(=O)(C1=CCCCCC1)NCC1N(C(C2CC(C)OC(C)C2)=O)CC=C1 N1(C(C2C(CNC(C(C(C)C)OC)=O)CCC2)=O)CCC2(CC1)CN(C)C2 C=CC(CCC)CC(=O)N1CCOC(CCNC(c2ccc3c(c2)COC3)=O)C1 c1(C(=O)NC2CC3CN(C(C(CC)C#N)=O)CC(C2)C3)cnc(O)c([N+](=O)[O-])c1 CC(F)CN=c1nc2c(cnn2C)c(NCC2CCCC2N2CCCS2(=O)=O)[nH]1 C1(CC)CN(C)CCCN1C(C1CC(O)CN1C(=O)C(Cl)Cl)=O C=CC1CCN(C(=O)CC2CC3(C2)CN(C(c2cc(C)ccc2OC)=O)C3)CC1 CCC(CNC(=O)C(n1nccc1C)C)(CC)NC(c1n[nH]c(C)c1Br)=O C1(OC)CCC(n2nc(-c3ccncc3)nc2C(C)OCc2ccccc2)CC1 C1(CNC(=O)NCCCc2[nH]nc(C(C)C)n2)CC12CCOc1ccccc12 C(C(=O)NC1CCC1NC(c1c[nH]cc1Br)=O)(C(C)C)SC c1(CC(C)NC(Cc2c(OC)ccnc2)=O)cc(C)ccc1C C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(=O)C(CO)OC)C12CCC2 CC(C)(C)C#CCCNC(=O)C(CNC(c1cc(F)c[nH]1)=O)CC1CC1 N1(C(C2C(NC(c3c(CC)onc3C)=O)CCOC2)=O)C2CCC1CC(OC)C2 c1(C(=O)NCC(N2CCN(C(C3CCCCS3)=O)CC2)C)cc(O)ccc1F C12(CNC(CCCCSC)=O)CCC(C1)N(C(=O)Cc1cc(F)ccc1F)C2 c1(C(N2CCC(C)C2CNC(c2nocc2Br)=O)=O)cc(F)ccc1O c1(C(=O)NC2CC(C)N(C(c3csc(=N)[nH]3)=O)C2)cccc([N+](=O)[O-])c1 c1(C(N(C(C)CO)C(C)C)=O)c[nH]c2ccc(-c3cccc(N(C)C)c3)cc12 n1(CC)nc(C)c([N+](=O)[O-])c1NC1CC(CCNC(=O)Cn2ncc(Cl)c2C)C1 c1(-c2cncc(CNC(CS(CC)(=O)=O)=O)c2)cc(F)c(C#N)c(F)c1 C1(n2cccn2)(C(=O)NC(C(=O)NCC)C)CCN(C(=O)CCCCCF)CC1 C(=O)(C=C1SCC(=O)N1C)N1CCCC(CCC)(NC(c2nc(Cl)oc2C)=O)C1 CC(C(=O)NCC1CN(C(=O)C(C)(C)n2cccn2)C1)C(F)(F)F c1(OC)c(CC(=O)NC2(O)CCCC(C)C2)cc(Cl)cc1Cl c1(C(=O)NC(C(CCC)C)C)coc2c1CN(C(=O)C(=O)NCC(F)F)C2 N1(C(c2c(C)cc(=O)n(C)n2)=O)CCCC2CN(C(=O)C=CC3CCC3)CCC12 c1(C(=O)Nc2cccc(CNC(CC(=C)C)=O)c2)cc2c(ncn2C)[nH]1 C1(C)(CNC(CCSC)=O)COCCN(C(c2c(C)noc2C2CC2)=O)C1 C(CC(F)(F)F)N(C(c1cn(CCO)nn1)=O)CC1CCCN1 c1(OC)cncc(-c2nc(CCOC(C)C)nn2CCn2cc(Br)cn2)n1 c1(OCC(=O)NCC2CC(NC(c3c(C)nsc3)=O)C2)cccc(Cl)c1 C1(NC(c2cc(C)nnc2O)=O)CCCCN(C(=O)C(C)(Cl)Cl)CC1 N1(C(CC2CCCN(C(C(C)CC3CCC3)=O)CC2)=O)CC2(CCCCC2)C1 C1(C(N2CC(C(N)=O)(CNC(C3(C)CCCCC3)=O)C2)=O)Cc2ccccc2O1 C1(NC(C2CCCN2C(=O)C2CC2)=O)CCOC12CCN(C(=O)CCC(F)F)CC2 c1(C(N(CCCCCNC(=O)CC2CCCO2)C)=O)nn(C)cc1Br c1(C(N(CCCN(C)C(C2(N(C)C)CC2)=O)C)=O)cc(O)cc(Cl)c1 CCCCC(CNC(c1occc1Cl)=O)NC(C1CCC(C)(C)C1)=O n1(CC)nc(C(=O)N(C)Cc2ccccc2CNC(=O)CS(=O)(=O)NC)c(C)n1 C(=O)(C(C1=CCC2CC2C1)NC(=O)N)OC.c1(C(C2CCC2)C)ccccc1Cl CCCC(CNC(=O)CCOC(C)C)NC(c1cc(=N)[nH][nH]1)=O CCC(CC(=O)N1CC(CC(C)NC(c2sccc2S(N)(=O)=O)=O)C1)C(F)F c1(OC)ccc(N)c(C(N2CC(C3(NC(c4ccc(Cl)[nH]4)=O)CC3)C2)=O)c1 c1(C(=O)OC)sccc1C(=O)NCC1(O)CN(C(C2(CN(C)C)CC2)=O)C1 C(C(C(=O)N1CCCC1CCCNC(c1cn(CCO)nn1)=O)NC(C)=O)OC N1(C(=O)NCC(C2CCC(F)(F)CC2)CO)CC2(CO)CC1CC2O C1(C(=O)NC2C(C)OCC2)CCC2CN(C(=O)C(C)(C)C)CC2O1 CC1(C)CN(C(=O)C(c2ccoc2)NC(c2ncc[nH]2)=O)C2CCCC12 Cc1cc(F)cnc1C(=O)NCCCCC(C)NC(C1CC2(CCC2O)C1)=O c1(C(N2CCCC(CNC(C(C3CCCC3)OCC)=O)C2)C)ccc(C#N)cc1 C1(N(C(=O)Cn2cc(CO)nn2)C)CCC(NC(c2cnc(OC)nc2)=O)CC1 c1(C(=O)NCC2CC(NC(CCC(C)(C)C)=O)C23CCC3)scc2c1CCCC2 CC1(C)CC(NC(C2CN(C(=O)CC3OCCCO3)CC2C2CC2)=O)C(C)(C)O1 C(=O)(C1CCCn2cncc21)NCC(CCCC)NC(=O)CCOC C1(C(=O)NCCCCC2CN(C(c3cc(C)no3)=O)C2)CCCCC12CCC2 N1(c2cc(C)[nH]n2)CCN(C(C2CCCC(NCc3ccoc3)C2)=O)CC1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CC2CC(C1)CN(C(C1CCC3CCC13)=O)C2 C1(CC(=O)NCC(CN(C(=O)C(C)(O)C2CC2)C)(C)C)CCCC(F)(F)C1 C1(CNC(=O)COc2ccccc2[N+](=O)[O-])CCC2(CCC2)C1NC(=O)C1CC1 Cc1cc(N2Cc3c[nH]nc3C2)nc(N2CCCC(n3ccnn3)CC2)n1 Cc1ccc(Cl)c(OCC(=O)NCC2(F)CC(NC(=O)C(=O)N(C)C)C2)c1 C12(CNC(C(C=CCCC)O)=O)CC1CN(C(c1cnn(CC)c1Cl)=O)C2 C1(C(=O)NCC2CC(NC(Cc3c(C)cco3)=O)C2)CC(C)(C)CO1 c1(NC(c2n(C(CC)C)nnn2)c2coc(C)n2)cccc(C#N)c1C c1(C(N(CC)CC2CCCN2C(=O)COC2CCCC2)=O)cc(=O)n(C)o1 C1(C#N)(CC(=O)N(C)CCOCCN(C)C(c2cccc(Cl)c2)=O)CCOCC1 CC1CC(C(=O)Nc2ccc(C(C)(C)C)nc2)N(Cc2ccc(F)nc2)C1 Cn1ncc(CNC(C2(C)C=CCCC2)=O)c1C(=O)NCC(c1cccnc1)O C(=O)(CCC(C)(F)F)N1CCN(CC(C)NC(c2c(CC)cncc2)=O)CC1 Cc1cc(Cl)ccc1-n1nc(CCn2ccccc2=O)nc1C1CCCN1C=O c1(C(=O)NC2CCN(C(c3ccc(CSC)o3)=O)C2)ccc2cnccc2n1 c1(C(N2CCC(OC)(CNC(c3ncccc3Cl)=O)C2)=O)ncc(C)cc1C CC(C)C(O)CC(=O)N(CCNC(c1csc(NC(N)=O)n1)=O)C(C)C N1(C(C(=O)NCC)=O)CCc2cc(NCC3CC3C)ccc21 c1(C(=O)NC(C(=O)NCCC)C)ccnc(CNC(=O)CN2CCCCC2)c1 N1(C(C2Cn3c(C)nnc3C2)=O)CCCn2nncc2C1 c1(C(N2CCC(NC(CCCCCN(C)C)=O)C(F)C2)=O)ccc2c(n1)CCO2 Cc1cccc(CNC(=O)CC2(C)CN(C(c3c(C)n[nH]c3C)=O)C2)c1 c1(CN2CCC(F)(C(N3CC(C)(C)C3)=O)C2)ccc(Cl)c(F)c1 CCS(=O)(=O)NCCC(=O)NC1(CNC(=O)CN(C)C(C)=O)CCC1 CN1CNC(=O)C12CCN(C(c1ccc3c(n1)COCC3)=O)CC2 N1(C(c2ccc(C(C)=O)cc2)=O)CCC2CCC12CNC(c1cc(F)c[nH]1)=O C=CCCCC(=O)NC1(C)CN(C(C2(c3ccccc3)CC(C)C2)=O)C1 N1(C(C)=O)CC=C(C(C)(C)C(=O)N2CCN(c3cc4cccnn4n3)CC2)C1 N1(C(C2C(C)=C2)=O)CCC(CF)(NC(c2ccc(C3CCOC3)s2)=O)C1 C1(F)(CNC(C(C)SCC)=O)CCN(C(c2cc(C3CCCCC3)n(C)n2)=O)C1 C(C)(C(O)C(C)C)NC(c1nc(CNC(c2c(C)snc2)=O)oc1)=O C1(=O)C(CC(F)F)c2ccc(cc2)C2C3CN1C2C3.Cc1cc(CC2CC2)c(C)s1 c1(C(=O)NCCN(CCCCCC)C(C2CC2CC)=O)nccc2ncccc12 CC1CC(NC(c2cc(O)cc(O)n2)=O)CN(C(C2(C)CC2Br)=O)C1 c1(OCC(=O)NC2C(NC(CC(CC)SC)=O)C2)c(F)cccc1F N1(S(CC#N)(=O)=O)CCC(O)C(NC(=O)Cc2ccnc(Br)c2)C1 Cc1cc(COC(=O)CCN2CCCC(OC(C)(C)C)C2)cc(C)n1 Cc1ccc(F)cc1C(N1CCC(C)C(C)C1)C(=O)NC1(C)CC1 c1(C(C)C)ccc(C(N2CC(F)(CNC(C3CCC3C)=O)C2)=O)c(F)c1 N1(C(c2n(C=C)nnc2)=O)CCC(C)C(CNC(c2cn(CC)cn2)=O)C1 c1(N2CC(=O)NCC2)ccc(NC(C2C(F)(F)C23CCC3)=O)cc1Cl N1(C(CCOCCOCC)=O)CC(NC(=O)CC2CSCCS2)CC(C)C1 C1(C(N2CCC(F)(C(N3CCOC4CC34)=O)C2)=O)CC2CCC1O2 C1(NC(C(CSC)OC)=O)CCCC(NC(c2cncc(C(F)F)c2)=O)C1 C1(C(N2CCC(N(C(=O)C(F)=C(C)C)CC)C2)=O)C(C)(C)C1(F)F C(=O)(C(C)CCC(C)(C)C)NC(C(C(=O)Nc1c(OC)cc(C)cc1)(C)C)C N1(C(C(CO)OC)=O)CC2CC1CN2C(=O)CC1(OC)CCOCC1 C1(CNC(c2ccc(OC)nn2)=O)CC2(CC2)CN1C(=O)C(C)(F)F c1(OC)ccc(OC)c(C(=O)NC2CC(CO)CN(C(c3cnn[nH]3)=O)C2)n1 N1(C(c2c(C)nco2)=O)CC2CN(C(=O)CCCC3CC3)CC2C(F)(F)C1 c1(OC)ccc(O)cc1NC(C1(F)CN(C(c2[nH]cc(C)c2C)=O)C1)=O c1(N(C(=O)NC(C)C)C)nnc(C2CCOC2)n1CC(C)SC(C)C C(c1cccc(F)c1)=CC(=O)NCCCCCCN(C(=O)CCCCC1CC1)C C=CC(CCC)CC(=O)NCc1cccc(NC(=O)C(=O)NCC2CC2)c1 c1(C(N(C(C(=O)OCC)C)C)=O)csc(CNC(C2(C#N)CC2)=O)c1 C1(NC(C(COC)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCCCCC1(F)F C(C(CN=c1[nH]n(C(C)C)cc1[N+](=O)[O-])C(F)(F)F)NC(c1c(C)ocn1)=O C1(O)(CC(=O)NC(C2CCCCC2)CNC(=O)C=CCN2CCCCC2)CCCC1 C1(C(=O)NCc2cncs2)CN(C(=O)CC2CCCC3CC23)CCO1 C1(O)(CNC(CCSc2n(C)ccn2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)C1 N1(C(CC=C=C)=O)CCCCCC1C(=O)NC1CCC(N(C)C)C1 CC1CN(C(=O)C=CC2CC2)CC(C)C1NC(c1ccc(Br)cn1)=O C1(C)(NC(C2(CCNC(c3cn(CC)nc3)=O)CC2)=O)CCC(=O)N(C)C1 c1(CN(C)Cc2n(CC)ccn2)nc(N2CCOCC2)[nH]c(=N)n1 N1(C(C(C#C)(C)C)=O)CCN(C(=O)Cc2cc[nH]n2)C2(CC2)C1 CC1CCC2(CCN(C(=O)CN(C(=O)CCc3ncccn3)C)C2)C1 C1(CNC(c2nccc(C)c2F)=O)CN(C(=O)CSc2cn[nH]c2)C2(CCC2)C1 C1(OCCC)CCC(NC(c2noc(C)n2)c2nnnn2C(C)(C)C)CC1 c1(N(C2CCOC2C)C(=O)NC(CC(=O)OCC)C2CC2)ccc(C)cc1C c1(C(N2CC(CN(C(C(Cc3ccc(C)cc3)C)=O)C)C2)=O)cnn(C)c1C#N C(=O)(C(CC(C)C)NC(c1ccc(F)c(C)c1)=O)N1CCC(SC)C1 c1(CN(C(C2CC2NC(=O)Cc2cc[nH]n2)=O)CC)ccc(Br)cc1 C1(NC(c2ccc(I)c(Cl)c2)=O)CC12CCN(C(C13CC(C1)C3)=O)CC2 C=C1CCN(C(C2CC(C)N(C)C2)=O)C(C(=O)NCc2[nH]ccc(=O)c2O)C1 N1(C2CCN(C(C(C)CF)=O)CC2)CCN(C(=O)C=CC2CC2)CC1=O c1(C(=O)NCC(C)N(C)C(c2nnc(S)n2C)=O)cc2cc(Cl)ccc2o1 N1(C(c2nc(O)cc(CC)n2)(C)C)COC2CCCCC2C1 N1(C(CC2(OC)CCOCC2)=O)CCCC(O)(CNC(c2nn[nH]c2Cl)=O)CC1 C(=O)(C(CC)CC(C)C)NC(CCCC(=O)N(CC)Cc1cnn(C)c1)C c1(C(=O)NCCC2CC(NC(CC(CN(C)C)O)=O)C2)ccn2cc(C)nc2c1 c1(OCC=C)ccc(CC(=O)NCC2(F)CC(NC(C3CCCC3C)=O)C2)cc1 N1(C(COC(C)(C)C)=O)CC2CCC1C1CN(C(=O)C=Cc3ncco3)CC21 CC1(C)CC(CNC(C2(C3CC3)CCC2)=O)N(C(=O)CCCn2ccnc2)C1 c1(CNC(C(COCC)NC(CC=CC=C)=O)=O)ccc(O)cn1 c1(NC(C(=O)NCCC(=O)OC)=O)ccc(NCc2cccc(I)c2)cc1 Cc1nncc(CN2CC(C)C2C(=O)NOCC(F)F)c1C c1(C(=O)NCC2(CCNC(c3ccc[nH]3)=O)CC2)nccc2c(F)cccc12 c1(C(C)(C)C(=O)NCC2CCN(C(=O)CS(=O)(=O)N(C)C)C2)ccc(F)c(F)c1 c1(C(=O)NC(C2CCN(C(c3c(CC)occ3C)=O)C2)C)cc(C)ccc1C C1(C(=O)NCC(CC)NC(c2sncc2Br)=O)COCCN1CC Cc1cc(O)c(Cl)cc1C(=O)NCC(C)CNC(c1ccc(Cl)[nH]1)=O N1(C(CCOCC)=O)CCC(F)(CNC(C2CC(O)(CC)C2)=O)C1 C1(C(=O)NCCCN(C(c2nc3cnccc3s2)=O)CC)CCc2nnnn2C1 CC1(C)CC(CNC(=O)Cc2cc[nH]c2)CN(C(=O)CC2COCC2(C)C)C1 C1(c2nn[nH]n2)(C(=O)NCC2(C(=O)NC)CC2)CCOCC1 C(=O)(C(C)(C)C(O)C(C)C)NCC(CC(=O)NCC(C(=O)OC)O)C1CCC1 C1(CC(N2C(C=C)CCC2)=O)CCCCN(C(=O)CCc2nc[nH]n2)C1 c1(NS(=O)(=O)C2CC2)csc(=NCC2C3CCOCC23)[nH]1 c1(CNC(C(=O)NC(c2nc3c(s2)CCC3)C)=O)cc2occc2n1C Cc1cc(C(=O)NC(C)CC(=O)NC2CCCC2)nn1-c1ccccc1 C1(NC(C(C)N(C)C)=O)CCN(C(c2cc(-n3cccn3)ccn2)=O)C1(C)C N1(C(CC2C(C(=O)NC3CC(CO)C3)CCCC2)=O)CC=CC(O)C1 C1(CC(=O)NC2CCCC2NC(C2CCC(=O)O2)=O)(COC)CCCC1 CCCCN=C(NCC1CCNC(=O)C1)N1CCN(CC(F)(F)C(F)F)CC1 C1(C(=O)NCC(C)CNC(C2(CO)CC2)=O)CC(=O)N(C(c2ccccn2)C)C1 c1(NC(C2CCCN(Cc3ccc(CCC)cc3)C2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(C(CO)OC)=O)CC(F)(F)CC1(C)CNC(=O)C(c1ccccc1)C c1(N2CC(C(C)NC(=O)C=Cc3cn[nH]c3)C2)nccc(-c2ccccc2F)n1 C(=O)(C1=CCCCCC1)NCC(C)CN(C(=O)CCc1cccc([N+](=O)[O-])c1)C CCCC(F)C(=O)N1CC(CC(C)NC(c2cnccn2)=O)C1 C1(NC(c2ccc(C)n2C)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC1(C)C C1(OCCCC)CC(NC(=O)N(CCC)Cc2ccco2)C1(C)C C1(CC=C)(NC(=O)C(O)C(C)C)CCN(C(c2cn(CC(F)(F)F)nn2)=O)CC1 C1(S(N)(=O)=O)(C(=O)NC2CCCN(C(C(F)OC)=O)C2)CCC1 c1(C(=O)NCCOCCNC(C2(CC(=O)OC)CCCC2)=O)nnc(O)cc1C N1(C(C(C)OCCN(C)C)=O)CCCC(CNC(=O)CC2C=CCCC2)CC1 C#Cc1cnn(C)c1C(=O)NC1CC2C(NC(=O)COCCCOC)C2C1 C1(C(N(C2CCN(C(C(C)OCCN(C)C)=O)CC2)C)=O)Cc2ccccc2S1 C1(CC)CN(C(=O)Cn2nccn2)CCC1CNC(c1c[nH]c(=N)o1)=O N1(C(c2c[nH]nc2[N+](=O)[O-])=O)CCC2(CCC2)C(NC(C23CC2C3)=O)C1 Cc1cc(C(=O)NC2CCC(CNC(=O)CC(C)(C)O)C2)nn1C N#CC1(C(=O)NS(=O)(=O)Cc2ccc(F)cc2Br)CCc2ccccc21 c1(C(=O)NC2CN(C(C(CC=CC)CC)=O)C(C)C2)cc(Br)c([N+](=O)[O-])[nH]1 N1(C(C)=O)CCC(CC(=O)NC2COCC2NCc2cnnn2C)CC1 C=CCCCC(C)NC(=O)C(COCC)NC(c1ccco1)=O C(=O)(C1=C(c2c(F)nnn2C)N(C)C(=O)N(C)C1c1cnn(C2CC2)c1)CC C1(C(N2CCC(COC)C2)=O)CC(CO)CCN1C(=O)Cc1n[nH]c(C)n1 Cc1cc(C(N2CC3C(NC(C4(Cl)CC45CCOCC5)=O)C3C2)=O)c(O)c(C)n1 C=CC(O)C(=O)N(C1CCC(NC(c2ccc(C(=O)OC)[nH]2)=O)C1)C C(=O)(C1=Cc2cc(F)ccc2OC1)NC1CCN(C(C=C2CCN(C)C2)=O)CC1 C1(C(=O)NCC2CCN(C(C3(CC=C)CCCCC3)=O)C2)CCCC2(CCC2)O1 c1(C(=O)NC2CC3(CC(C)C3)C2)nc(Cl)c(=O)[nH]c1N C1(C(=O)NCC=CC(=O)NCCC(CC)O)OCC2CCCC12 Cc1nccc(C(C(=O)NC2COC2)NC(C2CC(OC(C)(C)C)C2(C)C)=O)n1 C=C(C)C1OCCC1C(N1CC2(COC(CNC(=O)CCOC3COC3)C2)C1)=O N1(C(=O)N(C(CN(C(C)C)C)C)C2CC2)CCOCC1C1CCOCC1 Cc1cc(C(=O)N(C2CC(C#N)C2)CC(=O)NCCN2CCCC2=O)c(C)s1 C1(CCC)CN(C(C2CCCN2Cc2cn(Cc3csc(Br)n3)nn2)=O)CCO1 Cc1c(C(=O)NCCCCCCNC(c2cc(C(C)C)[nH]n2)=O)noc1C1CC1 Cc1nc2cc(C(N3CCN(C(=O)CCC(C)(C)C)CC3CF)=O)cc(O)c2o1 c1(CNC(C2C=CCC2)=O)c[nH]nc1C1CCN(C(c2cc(C3CC3)on2)=O)C1 C1(C(N2C(C)(CC)CC2)=O)CCCC(NC(=O)CC23CCCC2C3)C1 N1(C(CC(CCC)O)=O)CCC(C)N(C(=O)C(O)CN(C)C)CC1 CC1SCCCC1C(N1CC=CC1(C)C(=O)NC1CCC(C(N)=O)C1)=O c1(N(C)Cc2nnnn2C)[nH]c(=NCc2coc(CO)c2)nc2c1ncn2C C1(=O)C(C)(C)C(=O)O1.C1(c2nc(CC(=O)OC)no2)(C(=O)OCC)CCOCC1 C#CC1CCN(C(=O)C(c2ccnn2C)NC(c2scnc2Cl)=O)C1 C(=O)(CC1NC(=O)c2ccccc21)N1CC(NC(C(CSC)(C)C)=O)C(O)C1 Cc1nc2c([nH]1)C(C(=O)N1CC3CN(C(=O)C(=O)NC(C)C)CC3C1)CCC2 C(=O)(C(C#N)C(C)(C)C)NC1C(NC(CC2(OC)CCC2)=O)C1 C1(C(N2C(CNC(C3(COC)CC3(F)F)=O)CCC2)=O)CC(C)CCO1 C(CCC(C)NC(c1cnc(-c2ccncc2)s1)=O)NC(COC)=O C1(CNC(c2nc(CC)sc2)c2nnnn2CCCSC)CCCC(F)C1 Cc1nn(C)c(C)c1CC(N1CC2(CC2)CC1CNC(C1COCC1(C)C)=O)=O c1(C(=O)NC(CNC(CCCCCCC)=O)CO)cc2cccc(OC)c2o1 C(=O)(CS(=O)(=O)c1ccccc1C)NC1CCN(C(c2c(C)ccc(C)n2)=O)C1 C(N=c1nc(C2CC2)[nH]s1)C1C(CNC(=O)COCC2CCCC2)C1(F)F Cc1ccc(C)c(OCCC(=O)NC2CCCN(C(=O)CCF)CC2)c1 c1(C(=O)NC(C(CO)NC(c2oc(CC)c(C)c2)=O)C)coc2c1COC2 c1(CC(C)NC(CCN(C(CCN(CC)CC)=O)C2CC2)=O)cccnc1 N1(C(CCCc2onc(CCC)n2)=O)CCCN(C(c2cnc(S)[nH]2)=O)CCC1 C1(COC)CCCCN1C(=O)CC1COCCN1C(c1cc(C)ccn1)=O C=C=CC(C)C(=O)NCCC1CCCN1C(=O)C(C1CC(F)(F)C1)OC CC1CC(CC(=O)NCCCC2CCCCC2)CN1C(=O)Cc1cncn1C N1(C(=O)OC(C)(C)C)CCC(CF)(CNCC2CC2(F)F)C1 Cc1cc(C(F)(F)C(=O)NCC(O)CCNC(C2CCCN2N=O)=O)cnc1Cl C(=O)(CC(C)C(=O)OC)NCc1c(CC)n[nH]c1.c12cccnc1CNC2=O C(=O)(C1=NN(C)C(=O)CC1)N1CC(CCNC(=O)C=Cc2csc(C)n2)(OC)C1 CC(C)C(CCNC(C1CCCC1O)=O)NC(=O)CSCC1CCCO1 C1(c2ccc(C(=O)OC)cc2)CCCN(Cc2nnc(-c3ccccc3)o2)C1 N1(C(C(c2ccnn2C)NC(CCC=CC(C)C)=O)=O)CCCC2(C=CCO2)C1 C1(CNC(c2c(CCC)nsc2N)=O)CC2CCC1N(C(C1CC1(F)F)=O)C2 c1(C(N2CC(CNC(C3N(C)C(=O)CC3)=O)C2)=O)nnc2ccccn12 C1(CC(=O)NC2CCC(F)(CNC(c3c(C)ncn3O)=O)C2)(OC)CCOCC1 N1(C(C2N(C(CC3(OCC)CCC3)=O)CC=C2)=O)CCCC(C)(C)CC1 C1(OC)CC2(CCC(C(=O)NCCCNC(c3n[nH]cc3C(F)(F)F)=O)CC2)C1 N1(C(C2=CC(C)CC2)=O)CCCC2CN(C(=O)CCn3cc([N+](=O)[O-])cn3)CC12 Cc1occc1CC(=O)NCCOCCCNC(=O)C(c1ccccc1)O C12(CC(=O)NC3CCCOC3)CC1CN(Cc1cscc1Br)C2 c1(C(N2CCCN(C(CC(CC)C)=O)CCC2)=O)cc(O)c(OC)c(C#N)c1 Cc1ccsc1C(=O)NCC1CC(F)(CNC(C2CC2(c2ccccc2)C)=O)C1 N(C(=NCCCCl)N1CCN(C(c2ccco2)=O)CC1)CC(CC)C(C)C C(CN=C(NCCF)N1CCC2CCCOC2C1)N(C)C(=O)OCCSC.C(C)(C)(C)O C1(C(CC(=O)O)NC(=O)COC2CCCCC2)CCCC(=O)N1 CC1CCCN(C(=O)C(C2CC2)NC(=O)CS(C)(=O)=O)CC1 C1(NC(CC2CC(SC)C2)=O)C2CC(NC(c3ccc(Cl)cn3)=O)CC12 C(C1CCC(C)CC1)=C(C)C(=O)N1CC(NC(c2ccc(F)c(C(F)F)n2)=O)C1 C1(CCC=C)(C(=O)NCCOCCNC(=O)Cn2cc(Br)cn2)CCCC1 C1(NC(C(CC(C)C)F)=O)CN(C(c2cocn2)=O)C2(CCCCC2)C1 Cc1ccc(CCCNC(=O)CCn2cc(CNc3ccccn3)nn2)cc1 C#CCCC(=O)N(CC(C)C(=O)NCC1(C(C)C)CCCC1)C N1(CC(=O)NC(=O)CNC(N2Cc3ccccc3C2)=O)CCC2(COC(=O)N2)C1 c1(CNC(C2N(C(C(CC)n3cncn3)=O)CC2)=O)nnc(O)n1C CC1CC(NC(C2CCCCCC2)=O)CCN1C(c1cc(F)c[nH]1)=O Cn1nc(C(N2CCC(C3CCC3)(NC(=O)CC(=O)N(C)C)C2)=O)cc1Br c1(-c2scc(CNc3n(C(C)C)nc(Br)c3)n2)cc(F)ccc1F C1(C(N(CCOCCNC(C(CC)OC)=O)C)=O)CC(=O)c2ccccc2C1 c1(C(NNC(=O)NC(c2sccc2Cl)C)=O)cccc2ccccc12 S(=O)(=O)(CCC(F)(F)F)N1CCC(F)(C(=O)Nc2ncc(C)s2)C1 c1(OCC=C)cccc(CCC(F)F)c1.c1(C2C(=O)NN2C)csc(C(F)F)c1 C1(CCCOC)CCCCN1C(C1C2CN(c3cc(OC)ncn3)CC12)=O c1(C(N2CCN(c3nccc(OC)n3)CC2)=O)ccc(F)c2[nH]ccc12 N1(C(Cc2cc(C)sc2)=O)CC2CC(C1)CN(C(c1sc(N(C)C)nc1Cl)=O)C2 c1(C(=O)Nc2c(C)nsc2)nc2ccc(C(F)(F)F)cn2c1C1=CCC(C#N)CC1 C1(CNC(COCC#C)=O)OCCCC1(C)C.C12(CSC1)C(=O)N2 c1(NC(=O)NCCc2ccc(OCCCC)cc2)cnnc(O)c1Cl C1(C(=O)NCCN(C(Cc2cn(CC)nc2)=O)C)CCCCC1(F)F c1(N(C)C)nc2cccc(C(=O)NCCC3CN(C(C4CC45CC5)=O)C3)c2o1 C1(C)(NC(C(Br)=C(C)C)=O)CCN(C(=O)C(F)=CC2CC2)CC1 c1(C(=O)NCC(C2CC2)NC(C2COC2)=O)cc(Cl)c(Cl)s1 C1(c2ccn(C)n2)CCN(CC2CCN2C2CCNCC2)CC1 Cc1occ(-c2ccccc2)c1C(N1CCC(N(C(=O)CC2CC23CC3)C)C1)=O CC(C)(CNC(N1CCC(CCO)C1)=O)Cn1cc(CCCC#N)nn1 Cc1c(C(=O)N(C(C)CCNC(C2CCC2)=O)C)csc1Br N1(C(c2ccc(SC)s2)=O)CCC2CN(C(c3ccc(F)c(C)c3)=O)CCC12 c1(C(N2CCCCC2(C)C)C(=O)Nc2c(CC)cccc2)ccc(Br)cc1[N+](=O)[O-] CC1CC(C(=O)N2CCC(C)(CC(=O)NC3CCCCC3(C)C)C2)=NO1 C(C(=O)N=c1cc[nH]cc1N1CCOCC1)(C(C)C)c1c(O)ccc(C)c1 CC(O)(CNC(=O)CC1CCCC1NC(=O)C=CC(F)(F)F)CCO C(=O)(CCC(C)CN(C)C)NCCC(CCNC(c1nn(CC)c(C)c1)=O)C C(=O)(C(C#N)C(C)(C)C)N1C(C)CC(CNC(CC2(CSC)CC2)=O)C1 N1(C(C2OCC(C)C2)=O)CCC(CNC(=O)C(C)(C)N(C)C)C(F)(F)CC1 c1(C(=O)NCC2OCC(CNC(C(C)SC)=O)C2)oc2ccc(C)cc2c1C CC1CN(C(c2ccsc2)=O)CC1(C)CNC(=O)C(C)(C)Oc1ccccc1 N1(C(C2C(OC)CCCC2)=O)CCN(C(c2nn(C)cc2SC)=O)CC12CC2 c1(CNC(CC(C)SC)=O)cccc(NC(c2ccns2)=O)c1 N1(C(c2nc(C)[nH]n2)=O)CCCCC1CN(C)C(C1(c2ccncc2)CCC1)=O CC1OCC2(CCC(CNC(=O)C(=O)N(CC(F)(F)Cl)C)O2)C1C N1(C(CC2(COC)CC2)=O)CCC(NC(=O)CC23COC(C)(C2)C3)C(C)(C)C1 C1(C)(C(N(C)CC2(O)CN(C(C(c3cccc(F)c3)C)=O)C2)=O)CCSCC1 N1(CCOC)CCC(NC(=O)C=CC(C)(C)NC(=O)C=CC2CCOC2)C1 N1(C(C(COC)(C)OC)=O)CC2(CC(CNC(=O)CCc3ccn(C)n3)C2)C1 CCC(CC)C(=O)NCC(=O)NCC1CCCC1NC(=O)CSc1ccoc1 N1(C(C(C)OCCOC)=O)CC(O)(CNC(C2CC2F)=O)C1 c1(C(=O)NC(CNC(CC(CCCC)CC)=O)CO)ccc2c(c1)COC(=O)N2 N1(C(c2ccc(F)cc2)=O)CCC2CCCN(C(c3cc4[nH]ccc4s3)=O)C2C1 C1(OC)CCCCC1C(=O)NC12CC(C1)N(C(c1ccc(C(N)=O)nc1)=O)C2 n1(CC#C)cccc1C(=O)NC(C1CCCN1C(c1cnc(C2CC2)s1)=O)C N1(C(C2(CC)CC2)=O)CCC(C(=O)NC2(C(N)=O)CC2)CC1 C1(C(N(C(CCO)C(F)F)C)=O)C(C2CC2)CCN1C(=O)C(O)CN(C)C C(CCCCNC(=O)C(F)F)N(C)C(c1sccc1NS(C)(=O)=O)=O C1(OC)CC(CNC(c2[nH]c(C)cc2C)=O)N(C(=O)CCN(C)C(=O)OC)C1 C12(NC(C3CCC(OC)C3)=O)COC(CNC(=O)CCc3cccc(F)c3)(C1)C2 C1(CC(=O)NCC2(OC)CN(C(=O)C(F)=C(C)C)C2)CCCC(O)C1 N1(C(c2c(C)n(C)cn2)=O)CCC(NC(c2ccccc2F)=O)C(O)C1 C1(NC(=O)Nc2ccc(CC(=O)OC)cc2)C2Cc3c(Br)cccc3C12 C1(CCNC(c2n(C)nnn2)CC(C2CCCCC2)OC)CC(O)CCO1 c1(OC)cc(CN2CCC(NC(=O)Cn3ccnn3)C(F)C2)c(OC)cc1Br c1(C(N2CCC(NC(C3CCSCC3)=O)CC2)=O)ccc2cnnc(O)c2c1 S(=O)(=O)(c1cc(Cl)ccc1CS(C)(=O)=O)Nc1ccn(C2CN(C(C)=O)C2)n1 CC1(C(=O)NCC23CC2CN(C(=O)C=Cc2cccc(F)c2)C3)CC2(CCC2)C1 C(=O)(C(F)(CNC(=O)C=Cc1cn(C)nn1)C(C)C)N1CC(CCCCC)C1 Cc1cnc2cccc(C(N3CC(NC(=O)Cn4cncn4)CCC3C)=O)n12 c1(C(=O)NC(C2CCCN(C(CCC(=O)NC)=O)C2)C)ccc(F)c(F)c1F c1(NC(=O)N=c2ccn(C3CCCCC3)[nH]2)cccc(C#Cc2ccccn2)c1 N1(C(C(COC)O)=O)CCN(C(c2c(C)ccn2C)=O)CC1CF N1(C2C(NC(C(C=C)O)=O)CCC2)CCN(C(C2(C3CC3)CCC2)=O)CC1 N1(C(CN2CCN(CC)CC2)=O)CCC(C)(NC(c2ccc(C#N)s2)=O)CC1 c1(C(C)C(=O)NCCC2COCCN2C(=O)C2=C(Cl)CC2)c(Cl)cccc1Cl N1(C(Cc2cc(COC)on2)=O)CC(NC(C2CC(C)=NO2)=O)C(C(F)(F)F)C1 n1(CC)ccc(C(=O)NC2CCCCC2NC(=O)CC2(n3cccn3)CC2)c1C CC1=C(C)CC(C(=O)NC2CC(C)(C(=O)NCCC3CCSC3)C2)CC1 C1(C(=O)NCC2C(NC(c3cccc(C(=O)NC)c3)=O)C2)CCN(C)C(C)C1 c1(CC(=O)NCC(CC=C)NC(=O)Cc2cncs2)c(C)nc2ncnn2c1C CN1CCN(C(=O)CCOCC2CC2)C(NC(C2CC2c2ccccc2)=O)C1 C(=O)(CC(O)CC(C)(C)C)N1CC(OCCNC(C(CCC=C)(C)C)=O)C1 c1(-c2c(CC(=O)OC(C3CCCO3)C)ccnc2)cc(F)c(OC(C)C)cc1Cl NC(CC(=O)N1CCCC(CCC(=O)O)C1)C(F)F C(CC(C)(C)C)(C(=O)NCc1nc(=O)o[nH]1)NC(COCCCOC)=O N1(CC(=O)NC(C)CCCNC(C2CC(CC(C)(C)C)C2)=O)CCCCS1(=O)=O C1(CNC(CCC)=O)CC(NC(=O)C=C(C)c2ccco2)CCO1 C1(C(N(CCCNC(c2c[nH]nc2Br)=O)C(C)C)=O)CCC=CCCC1 Cc1ncnc(NC2CCN(C(=O)Cc3ccc(F)cc3)CC2)c1Br Cc1ccc(O)cc1C(=O)NC1CCC(CNC(=O)C#CC(C)C)CC1 Cc1csc(C=CC(=O)NCC(C(C)C)NC(=O)COc2ccon2)n1 c1(C(=O)NCC(CC)NC(=O)CCNC(C2CCC2)=O)cc(Br)n[nH]1 Cc1cc(C)c(C(N2CC(O)(CCNC(C3(C)CCCC3)=O)C2)=O)c(Cl)n1 c1(C(=O)NCCCN(C(C(C)=C2CC2)=O)CC2CCCC2)c(Cl)cc(Cl)nc1N C(C(F)(F)CNC(=O)C(CC1CC1)OC)OC.C1(=O)C(CO)N1 c1(C(=O)OCC)cc(C(=O)NCCC2CN(C(c3ccon3)=O)C2)no1 c1(C(=O)NC23CC(CNCc4ccc(Br)s4)(C2)C3)cccc2nc[nH]c12 C1(NC(c2noc(CC)c2C)=O)CCCC12CN(C(=O)CC1COC(=O)C1)C2 CON(CCC(=O)NCC1CC2(CC2)CO1)C(=O)CCC1CCCCO1 C1(c2cn(C(CNC(COCCCOC)=O)C)nn2)CN(C(C)=O)CC(C)(C)C1 C1(NC(COCCC#C)=O)CN(C(=O)CCCNC(N)=O)CC1O Cc1cc(F)cnc1C(=O)NCCCCCCNC(=O)CC(C)(C)O N1(C(c2ncc(C(C)C)s2)C(=O)NCCCF)CCCC2(CCCCC2O)C1 CC(C)CC(C(=O)NC(C)CNC(=O)Cc1coc(C(F)F)n1)N1CCCC1=O c1(NC2CC2)ncc(C(C)NC(C2(C(=O)NC3CCC(SC)C3)CC2)=O)cn1 c1(C(=O)NC2CCCCN(C(c3c(OCC)scc3)=O)C2)cnn2ccccc12 c1(C(=O)NC(CN2CCN(C(C=CC=CCC)=O)CC2)C)cc2cn[nH]c2cn1 c1(NC)cncc(C(=O)NCC2CC(F)CN2C(c2cc(COC)[nH]n2)=O)c1 N1(C(C(CCC)(C)CCC)=O)CCCC2(CCN(C(=O)C#CC(=O)N(C)C)C2)C1 c1(CC)nnc(N2CC3CC(NC(C4(CC)CCCO4)=O)C3C2)nc1CC C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)C(F)(F)c2ccncc2)C1 C1(NC(Cc2c(CC)cccc2)=O)CCC2CN(C(=O)CCOC(C)C)CC2C1 N1(C(C2CN(C(C)C)C2)=O)CCC(C(=O)N2CCC(C)C(C)C2)=C(F)C1 c1(OCC)ccc2cccnc2c1.N12CCCCCC1C(=O)NC1CC(C1)C2=O C1(C(=O)NC(c2ncc(C)[nH]2)CC)CCCN(C(C2CC3(CSC3)C2)=O)CC1 CCCC(C(=O)N1CCN(CCC)CC1)NC(c1cccc(C)n1)=O CC(CSC)CC(=O)NCC1CCN1C(C1(c2ncccc2F)CCC1)=O.C(N)(=O)N C1(NC(C(CC)(C)O)=O)CCCCN(C(=O)COc2c(C)nc(C)nc2O)CC1 c1(NCC2C(CCC)C2)ncccc1S(=O)(=O)N(C1CS(=O)(=O)C1)C c1(CCC(=O)NC(CNC(C(C)(CO)OC)=O)C)c[nH]c2cc(Cl)ccc12 S(=O)(=O)(c1cc(C)ccc1C)CN1CC(NC(CCSC)=O)C(C#N)C1 C1(C)(C(N2CCCC(N(C(C=CC(C)(C)C)=O)CCO)C2)=O)CCC(F)(F)C1 c1(NCC(=O)N(C)CCN(C)C(c2cc(Cl)nc(=N)[nH]2)=O)ccc(C#N)cc1F CCCCC(C)C(=O)NC1(COC)CN(C(=O)CC2CCC(C)O2)C1 c1(OCC(=O)OC)cccc(OC(=O)COCc2cn[nH]c2)c1 C(=O)(C(CC(N)=O)NC(C1CC12CCC2)=O)N1C(C)(CCO)CC1 C1(CC(=O)NCCOCCNC(C(C(CC)O)(F)F)=O)CCC2(CC1)OCCO2 C1(C(c2n(CC)nnn2)Nc2cccc3c2OCO3)CC(C)(C)OC(C)(C)C1 N1(C(Cn2ncc(CC)c2)=O)CCC(N(C(=O)CC2CC3(CCC3)C2)CC)CC1 N12CCC(C)(C)C(C1)NC(=O)c1c(cccc1F)OCC2=O.C12(CC)CC(C1)C2 CC1=C(C(=O)N2CCCC(NC(=O)C3=CCC3)CC2)Cn2nnnc2N1C c1(C(N2CCC(CC=C)C2)C(=O)NCC)ccc2nc(C)ccc2c1 CCC(C(=O)NC(c1cn(C2COC2)nn1)C)C(F)(F)F C#CCCCCC(=O)NCCN(CCCCCC)C(=O)C(c1ccsc1)N(C)C C1(NC(=O)C=CBr)COCCN(C(=O)CCc2cccc(F)c2Cl)C1 c1(C(=O)NC(CC)CN(C)C(c2cc(C)no2)=O)cncc(C(=O)OC)c1 c1(NC2CC(NC(C(c3c(C)noc3C)C)=O)C2)nccc(C#N)n1 c1(CC)ccc(C(=O)NCCC(O)C(=O)NCc2nn(C)cc2CO)cc1 C(=O)(C(CC)C(F)(F)F)NCC1(C#N)CN(C(C2CCC(C#C)CC2)=O)C1 C1(CC(=O)NC(c2nc(C(=O)NCC3CCCC(C)C3)co2)C)C(C)(C)C1(C)C c1(Cc2cn(C3CN(C(C(CC)CO)=O)C(C)C3)nn2)c(Cl)c(C)nn1C Cc1cc(C(C)C(=O)NC2CN(C(=O)C(C)CCO)C2)cc(C)c1 c1(CC)cncc(C(=O)NCC2CC2CNC(C2CC2C(F)F)=O)n1 C(C)(CC(=O)NCC1CCC(NC(=O)Cc2cccnc2)C1)OC C1(NC(CSc2n(C)cnn2)=O)CCOCC1C(=O)NCc1ccc(F)cn1 c1(C(N2C(C(C)NC(C3(CN(C)C)CC3)=O)CCC2)=O)cn2ccsc2n1 N1(C(C(C(C)C)F)=O)CCN(C(=O)CCCC2CCCC2)C(C(F)(F)F)C1 c1(C(=O)OC)c(Br)ccc(-c2ccc(-c3nc(C(F)(F)F)n[nH]3)cc2)c1F N1(CC(C)(C)NC(C2C(=C)C2)=O)CCN(C(=O)CC2OCCOC2C)CC1 c1(C(N(CC(C)NC(CCC=C)=O)CC)=O)ccc2c(Br)cnn2c1 C(=O)(C(C(C)C)N(C)C)NCCN(C(C(C)OCCOC)=O)CC C1(OC)CCCC1C(N1CCCC1CNC(=O)C=CC1CCCO1)=O N1(C(CCc2n(C)cnn2)=O)CCC2CC2(NC(=O)C(Cl)=CCl)CC1 c1(C(=O)NC(CCOC)CNC(=O)CCCc2nccs2)cccnc1Cl c1(C(=O)NC2C(NC(c3n(C)c(S)nn3)=O)C2)cnc(O)c2cccnc12 C1(n2cccc2)(CNC(C(C)CF)=O)CCN(C(c2sc(F)cc2Cl)=O)CC1 CC1(CNC(=O)Cc2cscn2)CCCN(C(=O)CCC2NC(=O)NC2=O)C1 c1(C(=O)NCC2C(C)(C)C(=O)N2)cccc(S(=O)(=O)N2CCSC23CCC3)c1 c1(C(N2C(CC)CN(C(C3(C(N)=O)CCC3)=O)CC2)=O)cc(=O)n2ccsc2n1 Cc1c(C(N2CC3(CCN3C(=O)CC3C=CCC3)C2)=O)sc2nnc(S)n12 C1(NC(Cn2ncc(C)c2)=O)C(C)CCN(C(c2cc(O)cc(N)c2Cl)=O)C1C c1(N(C(C(CC#C)O)=O)C2CC2N2CCOCC2=O)ccc(C)c(OCC)c1 Cc1ccc(C(=O)NC(C(=O)N(C2CCOC2)CCO)C2CC2)o1 C=CCC(CC)N=c1nc(N(C)Cc2nonc2C)c2cnn(C)c2[nH]1 c1(CCNC(c2n(CCSC)nnn2)c2ccoc2C2CC2)ccccc1Br c1(C(=O)NC(CNC(C=CCCC)=O)CO)cc2sc(C)c(C(=O)OC)c2[nH]1 c1(CC(=O)NC(CCOC)CNC(C)=O)sc(C2CCC2)nc1C Cc1cc(=NC(=O)C2CCCC23CCN(C(=O)CCc2ccsc2)C3)[nH][nH]1 N1(C(CC2N(C)CCCC2)=O)CC(CNC(c2cc(C(F)F)no2)=O)CC1(C)C C1(C)(C(=O)NCCn2cc(CNC(CC)=O)nn2)CCC(=O)C1 N1(C(CC2C(C)OC(C)C2)=O)CCCC(N(C)C(c2ccc([N+](=O)[O-])s2)=O)CC1 C1(NC(Cc2ncc(CC)[nH]2)=O)CN(C(c2cc(O)nc(O)n2)=O)CC(C)(C)C1 C12(CNC(C(C3CCOCC3)OC)=O)CC(CCO1)N(C(c1cc(C)cs1)=O)C2 c1(NC(C(N)=O)=O)cccc2c1C1CN(C(=O)COc3ccccc3)CC1O2 C1(OC)CC2CC(C(=O)NCCN(C)C(C3(C(=O)OC)CC3C)=O)CC12 C1(CNC(C(CCOC)C)=O)CC(NC(=O)C(=O)NC2CC2)C12CCC2 N1(C(c2cncc(OC)c2)=O)CCC(C2CC2)C1CNC(C1CCCC(F)C1)=O c1(OC)cnncc1C(=O)N(CCCNC(c1ccoc1)=O)C1CC1 CN1C(=O)CCCC1C(=O)NC1CC2CC(NC(=O)C(O)(C3CC3)C3CC3)C2C1 CCCC(C(=O)OC)C(=O)NCC1CC1CNC(=O)CC1CCC1 C1(C(=O)NCCC2(C)OCCO2)(CC)CCN(C(=O)C=C=C(C)C)C1 C1(N(C(c2cnsc2)=O)CC)CCCN(C(C2CC23CCSCC3)=O)CC1 c1(C(=O)NC2CC3CC(NC(CC(CN(C)C)O)=O)C2C3)ccc2nncn2c1 C(C(C)(CC)C(=O)NCCn1cccnc1=O)NC(CCC(=O)NCC)=O N1(C(c2cc(SC)oc2)=O)CCC(CF)(NC(=O)CCC(=O)OC(C)(C)C)C1 C(CCC(=O)NC(C)(CNC(=O)CCn1ccnc1)C1CC1)OCCOC c1(C(=O)NCC2(F)CCCN(C(c3nc(=N)[nH]cc3)=O)C2)ccnc2cc[nH]c12 N1(C(c2nc(COC)oc2)=O)CC(C)CN(C(c2cc(Cl)no2)=O)CC1C C1(C(=O)NCC(C)NC(=O)C(C)c2ccsn2)CC(F)(F)C1 c1(SCCC(N2C(CCCNC(C(CC)F)=O)CCC2)=O)ccccc1C C(=O)(C1CCCn2ncnc21)NCC1CN(C(C(C)C)=O)C1 C1(C(N2CCC(CCNC(c3cccc(OC(F)F)c3)=O)C2)=O)CC2CC1CO2 N1(C(c2cccc(Cl)c2OC)C(=O)NCCCCCC)CC2OC(=O)N(C)C2C1 N1(C(c2cnn(CCC)c2C)=O)CC(NC(c2cc(C)nnc2O)=O)CC(C)C1 N1(C(c2nc(COC)oc2)=O)C2CCC1CN(C(=O)CCC=CBr)C2 C12(CNC(C(=O)N(C)C)=O)CCC(CN1C(=O)C(C(C)(C)C)n1ccnn1)C2 C(=O)(C(C)(C)C(=O)N1CCCC1)N1CC(C(C)NC(CNS(NC)(=O)=O)=O)C1 C=CC(C)(CCOC)C(=O)N1CC2(CNC(C3(C)CC3C(=O)OC)=O)CC1CO2 C1(C(C)C)CCCN(C(C23CC2CN(C(=O)C(C)N2CCCC2)C3)=O)CC1 c1(C(=O)NC(C2CCCC2)CNC(C2C=CCC2)=O)ccc(C(F)(F)F)cc1 c1(C(=O)NC2CCCN(C(c3c(C#C)c[nH]n3)=O)C2)cnc(C)cc1Cl Cc1ccc(CC(=O)NC2CCC2CNC(C2CCCSC2)=O)cc1 C1(F)(CNC(C2CCCO2)=O)COCCN(C(=O)C=CCN2CCOCC2)C1 C1(COC)CC(CNC(C2CC23CC(O)C3)=O)N(C(c2ccoc2Cl)=O)C1 c1(NC(C(c2nc(C)sc2C)N(C(C)COC)CC=C)=O)ccc(OC)c(C)c1 Cc1ccc(CSCC(C)C)c(I)c1.C1(CC(C)C)C(=O)N1 C(CC(C(=O)N(C)Cc1nc(C)ns1)NC(c1nn(C)cc1C)=O)=CC c1(C(C(=O)N(CCNC(=O)CN(C)C(N)=O)CC)C)c(F)cccc1F N1(C(C(CC)C)=O)CC(NC(c2ccc3nncn3c2)=O)CC(F)(F)C1 C(=O)(C(C)CC=CC)N(CC(=O)NC(CC=C)CC)CCC O=C(CCCCSc1ccccc1)NCCC(O)CNC(=O)CCn1cccn1 CC(CC(C)(c1nnnn1C1CC(F)(F)C1)CC(=O)OC(C)(C)C)C(F)F CC1CCN(C(=O)Cc2ccnc(O)c2)CCN1C(=O)COc1ccsc1 c1(C(=O)NC(C)CNC(C2COC(=O)O2)=O)ccc(C(=O)N(C)C)cc1 c1(C(=O)NCC2C(NC(c3noc(CC)c3C)=O)CC2)cc(C)cc2ccoc12 Cc1cccc(C(O)C(=O)NCCCOCCCCCNC(=O)C=CC(C)C)c1 Cc1cc(C(N2CC3(CC(CNC(=O)CCC(C)N(C)C)C3)C2)=O)ccc1O N1(C(c2cccc(C)c2C)=O)CCC(C(=O)NCc2nn(C)c(=O)n2C)=C(F)C1 Cc1ccc(CN(CCCc2nnco2)C=O)c(OC2CCCCC2)c1 C1(C2CN(C(=O)C=C(C)Cl)C2)(NC(C2CC(C(F)(F)F)(OC)C2)=O)CC1 N(C1CCCCc2ccc(Br)cc21)CC12CN(C)C(CC1)CC2 c1(N2CCC(N(C)CC)CC2)nc2c(c(=NCC3CC(O)CCO3)[nH]1)CCC2 C=CCC(C)(O)C(=O)NC(CC1CCC1)C(=O)NCCC(O)C(F)F C1(C(N(CC(C)NC(c2coc(O)n2)=O)C)=O)COCOC1 CCC(C(=O)N1CCN(C(c2ccn3cccc3c2)=O)C(CO)C1)C(C)(C)CC C(CN1C(=O)COc2cc(Br)ccc21)NC(=O)NCc1cncc(C)c1 c1(N2CC(C(=O)NCC(CNC(C(CSC)OC)=O)F)C2)ccc(Cl)c(Cl)c1 CCC(CC)C(C(=O)N(C(CC)CC(N1CCC(O)C(CO)C1)=O)C)OC C12(C(=O)OC)CC(NC(N3CCCC3CN(C3CCNC3=O)C)=O)(C1)C2 Cc1c(C(N2CCC(NC(=O)C(Cl)(Cl)Cl)C(F)C2)=O)ccnc1Cl Cc1cc(F)cnc1C(=O)N(C1CCN(C(C2CC(C)(F)C2)=O)CC1)C C1(C(=O)NCCC2CCCCN2C(=O)C=Cc2cscn2)CCOCC12CCC2 Cc1cccn2nc(C(=O)N(C(c3ccccc3)CNC(C34CC3C4)=O)C)cc12 c1(NCC2C(CC)(NC(=O)COC(=O)OC)CC2)oc2ccccc2c1CCCO Cc1nc(N(C)CC23CCNCC2C3)cc(-c2ccco2)n1 N1(C(C2N(C(c3c(NC)cccc3)=O)CCCC2)=O)CCN2CCCCC2C1 c1(C(=O)NC(C2CCN(C(=O)C=CC3CCCC3)C2)C)ccc(Br)cc1O c1(OC)cc(C)c(C(=O)NC(CNC(=O)C2=CCCS2)C2CCC2)cc1OC CC(C)(CCCNC(=O)CSC1CC1)NC(=O)OC(C)(C)C.C12CCN(C1)C2=O C1(O)(C(C)NC(C(CC=C)C)=O)CCN(C(=O)COc2cncc(Cl)n2)CC1 c1(C(N2CCCC(CN(C(=O)CC3CCCO3)C)C2)=O)ccc(C2CC2)nc1O c1(C(N2CCC(C)C2CNC(c2coc(C(N)=O)c2)=O)=O)cc(O)cc(F)c1 C1(CNC(C(CC)c2cccnc2)=O)CCC(C)(C)CN1CCC1CCCCC1 c1(C(N2CC3=C(CN(C(C(CCSC)O)=O)C3)C2)=O)ccc(F)c(C)c1C#N S(=O)(=O)(c1ccc(NCCCF)cc1Br)N(C(Cc1cccc(C)c1)C)C CCC(CCC(=O)NC(C)(C)CCCOC)NC(c1cc(C)ns1)=O c1(C(=O)NCC(CC=C)NC(=O)Cc2ncc(C)o2)cc(C)c2[nH]cnc2c1 C12(C(N3CC(NC(C(C)OC)=O)(CO)C3)=O)CC(C)(C1)OC2C N1(C(c2c(C)ccs2)=O)CC(C(N2CCSCC2C2CC2)=O)C2(CCC2)C1 O=C(C1=CC2CCCCC12)NCCN(C(=O)COCCF)Cc1ccccc1 c1(C(=O)NCCC(CNC(=O)CC2CC(F)(F)C2)O)cc(Cl)ccn1 Cc1cc(C(N2CC(NC(c3ccc(C)s3)=O)CC(C)C2)=O)n2ncnc2n1 N1(Cc2cc(C(=O)OCC)no2)CCOC(CN(C)Cc2ccccc2)C1 C1(CNC(c2c(CC)scn2)=O)CN(C(=O)C(C)=C2CCC2)C2(CCOCC2)C1 C1(C(=O)NC2C(C)N(C(c3cc(F)c(F)cc3Cl)=O)CC2)CCC2CCCCN12 C(=O)(C1=CCN(C(C2CCCOCC2)=O)C1)NCC1CC(C(C)(C)C)C1 c1(N(CC(C)NC(=O)CN2CC3CC3C2)C)ccnc(C2CCCC2)n1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2cscn2)=O)ns1 CCCCC(C(=O)N(C)CCOCCNC(=O)Cc1cncn1C)C(C)C N1(C(C2(CC)COC2)=O)CCN(C(=O)CN2CCCC2)C(COC)C1 c1(C(=O)NCCN(CC(C)O)C(c2cc(C(C)C)nn2C)=O)cnn2c1OCC2 C1(CC(C)NC(=O)CC2(O)CCC2)CN(C(=O)COC2CCC2)C1 CC(C)C(C)(O)C(=O)NCCn1cc(CNC(=O)C=Cc2cc[nH]n2)nn1 N1(C(CCC(C)OCC)=O)C2CCC1CC(N(C(=O)C(=CC1CCCC1)C)C)C2 N(C(=NCc1ccccc1)NCC(c1cn(C)cn1)(C)C)CCOCC=C Cc1ncc(F)c(N2CC3CC3(NC(=O)Cc3ccc(F)c(F)c3)C2)n1 Cn1c(C(=O)NC2CC2NC(C2CC=CCC2)=O)nnc1S c1(CC(=O)NC2(C)CC(NC(CC(C)(C)O)=O)C2)c(F)cccc1F c1(N2CC(CNC(CC(C)n3cccn3)=O)OCC2)ncnc2[nH]ccc12 C(=O)(CCC(CF)CF)NC1C2CC(C(=O)NC(C)(CO)C3CC3)C(C2)C1 C#CCCCCCCC(=O)NC1C=CC(CNC(=O)CC(C)C(C)C)C1 C(C(O)CC(=O)NC1CCC(=O)NC1)NC(C=C(CC)CC)=O c1(C(N2CC(COC)(CNC(C3(O)CCSCC3)=O)C2)=O)cc(N)ccc1C C(N=c1[nH]c(=N)[nH]c(=NCC(F)(F)CC2CC2)[nH]1)C1N(C)CC(O)C1 c1(C(=O)NC(C2CCCCC2)C(C)NC(=O)C2CC2)nc2cncnc2nc1O CC(C)C(C)C(=O)NC1CCOC1C1CCN(C(C2(O)CC(F)(F)C2)=O)CC1 c1(C(=O)NCC2N(C(C=CC=CC)=O)CCOC2)ccc(F)c(Br)c1 C12(CNC(C3CC34CCOCC4)=O)CCCC1CN(C(c1sccc1Cl)=O)C2 S(=O)(=O)(c1ccc(F)cc1)N(C)CCNC1CN(C(=O)CC(F)(F)F)CCN1 N1(C(C(C)C2CCOC2)=O)CCOCC(NC(=O)CCOC2CCOCC2)C1 C1(c2n(COCC)nnn2)(NCC(c2ccc(F)cc2F)=O)COCC(C)(C)C1 Cc1cc(=NC(=O)C2c3ccccc3CN2C(=O)C(C)CCC(C)(C)C)[nH]n1C N1(C(c2cc(CCOC)on2)=O)CC(NC(=O)CC#N)CCC1C CCC(C)C(C(=O)NCC1(C(N2CC3C=CC3C2)=O)CCC1)N(C)C c1(C(=O)NC(C(C)NC(C2C(CC(C)C)C2)=O)CO)ccc(N2CCCC2)c(F)c1 c1(OCC#C)ccccc1CNCc1ccnnc1 N1(CCCC)CCCC1C(=O)NCC1(NC(=O)CN(C)C)CC(OC)C1 N1(C(C(F)OC)=O)CCN(C(=O)CCSC(F)(F)F)C(C(F)F)C1 C(=O)(C1=CCOCC1)N(C(C)CN(C(=O)Cn1nccn1)C)C Cc1ccc(NC(C2OCCC2CNC(c2ccccc2)=O)=O)cc1F Cc1ccc(C(=O)N(C)CC2CCCC(NC(c3nccnc3N)=O)C2)nc1O N1(C(CCC(=O)NC)=O)CC(CO)C2(C1)CN(C(=O)CCCCCl)C2 c1(C(=O)NC(CCSC)C(=O)NCCC(O)CO)cccc2cc[nH]c12 N#Cc1c(NC(C2CCN2C(=O)C(CO)c2ccccc2)=O)cccc1Cl C1(NC(C2C3CCCC23)=O)COC2(C1)CN(C(C1CN3CCN1CC3)=O)C2 C(C(F)C(=O)NC(C1CCCCC1)CNC(=O)C(C)CN(C)C)N(CC)CC CCCCC(CC)C(=O)N1CC(CCCCNC(c2ccc(F)o2)=O)C1 C(CC(=O)N1CC2CCC1CC2)(C(F)(F)F)NC(C(C(=O)OC)C)=O c1(OCC(=O)N(C2CCN(C(c3cc(CC)no3)=O)C2)C)ccc(Cl)cc1Cl N1(C(C2CC(C)OC2)=O)CC2(CCN(Cc3cnon3)CC2)C1 C1(C(=O)NCCC2OCCN(C(C3(C)CS(=O)(=O)C3)=O)C2)CCC2(CCC2)CO1 c1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCCC2C)ccc([N+](=O)[O-])cc1Cl C(=O)(C1=CS(=O)CCC1)NC1CCCN(C(C2C(C)CCO2)=O)CC1 Cc1ccc(NC(C2CN(C(C3CCCC34CCC4)=O)CC2F)=O)c(O)n1 c1(NC(CC(C)NC(c2cnc(O)n2C)=O)C)cc(C(F)(F)F)ncc1[N+](=O)[O-] c1(NS(=O)(=O)CCc2cn[nH]c2)cccc2c1OCCC2 C1(N(C(=O)CCNC(N)=O)CC)CCN(C(=O)C(N2CCOCC2)C)C1 N1(C(C=CC)=O)CCN(C(c2conc2Cc2ccccc2)=O)CCC1C N1(C(C2C(C)C2)=O)CCN(C(=O)CC2CN(C)C2)C(C2CCC2)C1 C12(CCNC(c3c(C)nc(CCC)o3)=O)CCC(C1)N(C(C1(SCC)CC1)=O)C2 C1(CC(=O)NC(c2ccc(C)s2)CO)CCn2cncc2C1 CCCCC(CCC)C(=O)NCCCOCC(=O)O CC1CN(C)CCC1NC(C1CCC(CNC(=O)CC(F)(F)F)O1)=O c1(OC)ccc(NC(=O)CN(C)CC23CC2CCN3)cc1NC(C)=O C1(NC(CC(=O)NCC)=O)COCCN(C(c2ccnc(OC)n2)=O)C1 N1(C(c2c(CC)nc[nH]2)=O)CCCC(N(C)C(C2(C)CCC(F)(F)C2)=O)CC1 CC(C)(C(=O)NCC1CCC(NC(C2CC3(CCOC3)C2)=O)CC1)S(C)(=O)=O C#CC1CCCN(C(C2(C)CCCN(C(c3cc(=O)cco3)=O)C2)=O)C1 C=C=C(C)CC(=O)N1CCC(N(C(C2(N3CC4CC4C3)CC2)=O)CC2CC2)CC1 Nc1cnc(C(=O)NC2C3CCC2N(C(=O)CC2(C(F)(F)F)CC2)C3)c(Cl)c1 C1(COC)CN(C(=O)C(C2CCOCC2)F)CCN1C(c1nc(Cl)cs1)=O C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC2=C(CN(C(c3c(C#N)csc3)=O)C2)C1 C1(C(N(CC(CN(C)C(c2[nH]nnc2C(F)F)=O)O)C)=O)CC2(CCO1)CC2 c1(OCCC(C)C)ccc(CNC(=O)NC2CCCC(F)C2)cc1 Cc1cc(=NCCc2ccc(C#N)cc2)[nH]cc1S(=O)(=O)NCC1CC12CCOC2 Cc1cc(C(N2CC(NC(=O)CCCc3ccc(Br)cc3)C(F)C2)=O)c(C)o1 CC1(C)CCC(CO)N(C(C2CN(C(=O)Cn3cnc(=N)[nH]3)CC2(C)C)=O)C1 C1(C(N(C)Cc2cc(C#N)ccn2)=O)CC12CCN(Cc1cccnc1)CC2 CC1(C)OCCC1CNC(c1ccc(Cc2cccc(O)c2)cc1)=O N1(C(C=C(C)CNC(c2cnn(C)c2C#N)=O)=O)CCN(C)C2CC12 N1(C(C(C)OCCC=C)=O)CCOCC(F)(CNC(c2cc(C(F)F)cs2)=O)C1 C1(CNC(=O)NC2CCN(C(C3(C#C)CCCC3)=O)C2)CC2(CC(OCC)C2)C1 C1(NC(C2(COC)CC(F)(F)C2)=O)CCN(C(c2sccc2F)=O)CC1O C(=O)(C(O)CCCc1ccccc1)N(CCCNC(C1N(CC)CC1)=O)C N1(C(C(CC=C)C)=O)CC2OCCN(C(c3scnc3C3CC3)=O)C2C1 C=CC(CC(=O)N1CC(NC(c2occc2Br)=O)C(O)C1)c1ccccc1 c1(C(=O)NCC(CNC(C2(C)CC2Br)=O)O)cccnc1OCCO C1(NC(C2CCCC23CC3)=O)CN(C(c2ccoc2Cl)=O)CC1O C#CCCCC(C)C(=O)N1CCCC1C(=O)NCCc1ncc(C)o1 c1(OC)ncc(Cl)cc1C(=O)NC1CC(CNC(=O)C(C)c2ccco2)CC1O c1(C2(C(N3C4C(NC(CCSC)=O)C(C4)C3)=O)CCC2)ccc([N+](=O)[O-])c(C)c1 O=C(CC1=CCOCC1)N1CC(O)CC1C(N1CCCC(CO)CC1)=O C1(NC(c2cc(SC)oc2C)=O)CCSC12CN(C(=O)C(c1ccccc1)F)C2 N1(C(CC(C)C)=O)CCN(C(=O)C(CC(C)C)N(c2ccccc2)C)C(CO)C1 C1(C(N2C(C)CCCC2)=O)CC(c2ccccn2)=NO1 N1(C(C=CC)=O)CCCC(C2CCN(C(=O)C(CC3CC3)CC3CC3)C2)C1 c1(C(=O)NC(CC(C)C)c2nc[nH]n2)ccc(OCC2CC2)c(F)c1 C1(CN(C(C2CCC2(F)F)=O)CC)CCN(C(c2ccc(C3CC3)o2)=O)C1 C(C(C(C)(C)C)NC(c1ncccc1Cl)=O)NC(C1C(OCC)C1)=O CCC(C(=O)N1CC2CCC2(NC(c2nnc(O)cc2O)=O)C1)C(C)C CC1OC2(C)CC1(C(N1CCC(CNC(c3ccnc(F)c3Cl)=O)C1(C)C)=O)C2 C1(NC(C(CC=C)OC)=O)CCN(C(c2ncn3c2CCC3)=O)C12CCC2 c1(C(N(CCC(C(C)C)NC(C(C2CC2)OCC)=O)C)=O)ccnc(F)c1OC c1(OC)ccc(C(N2CCC(C)C2CNC(c2nc(C)nn2C)=O)=O)cc1O c1(NCc2cccc(C(N3C(C(CC)O)CCC3)=O)c2)ccc(S(C)(=O)=O)cn1 c1(CC)nc(O)c(C(=O)NCC(CC)(CC)NC(=O)C#CC2CCC2)cc1C N1(C(CCCSC)=O)CCC(NC(c2cnccc2C(C)(C)C)=O)C(F)C1 C1(CNC(C(C)SC)=O)CCN(C(=O)CCNC(=O)CO)CCC1(F)F C(C(O)CC(=O)N1CC(F)CC1CNC(c1cc(C(F)F)cs1)=O)N(C)C C1(NC(=O)CC(F)F)CC2(CCN(C(C3C(F)(F)C34CC4)=O)C2)C1 N1(Cc2cn(CC)nc2)CCN(C(c2cc(Cl)ccc2OC)=O)CC1C(C)C C1(C(=O)NCC(CN(C)C)(C)O)CCCC(NC(=O)C=Cc2ccncc2)CC1 c1(CC)cc(C(N2CC(NC(c3cc(F)c[nH]3)=O)C(F)C2)=O)cc(C)c1 c1(C(=O)NC2C(NC(c3nc(C(C)C)sc3)=O)COC2)ccnc2ccccc12 O=C(C(F)C(F)(F)F)Nc1cn(-c2ccc(CC3CCCOC3=O)cc2)nn1 N1(C(C(C)C(C)(C)C)=O)CC(NC(=O)Cc2ccccc2[N+](=O)[O-])CC(C)(C)C1 c1(CCC(=O)NCC(CC=C)NC(c2conc2C(C)C)=O)nnc(C)n1C c1(OC)c(Cl)ccc(C(N2CCCN(C(=O)CC3C=CCC3)C(CO)C2)=O)c1F C1(NC(C(C)OC)=O)CC2C(NC(=O)CNC(c3cc(C)oc3C)=O)C2C1 c1(C(=O)NC2CC(NC(C(CC)n3cccn3)=O)C2)nn(C(C)C)cc1Br c1(CC)cccc(C)c1C(=O)Nc1ccc(Cl)nc1NS(=O)(=O)C(C)C C(=O)(CCCCCC(C)O)NCC1CC(O)(CNC(c2cc(CC)nn2C)=O)C1 C1(C(=O)NCC(CCOC)NC(=O)Cc2n[nH]c(=N)s2)CNC(=O)N1 C1(F)(C(=O)NCC2C(C)(C)C2CO)CCCN(C(=O)CC2CCC(=O)N2)C1 c1(C(=O)NC2CCN(C(CCC(CC)C)=O)C2)ccc2nnc(C)c(C)c2c1 c1(C(=O)NCC(C)NC(=O)CCN2CCC2)ccc(-n2ccnc2)nc1 c1(C(C)(C)C)ccccc1C(=O)NC1CN(C(C2CC2c2nnsc2Cl)=O)C1 N1(C(=O)OC(C)(C)C)CCCC(C(=O)NCC#CCN(C(=O)C=CS(C)=O)CC)C1 CCC1=C(C(=O)NCC2(O)CC(NC(=O)C(C)(C)CC#N)C2)CCCO1 C1(C)(NC(C2(COC)CN(C(=O)C(C)N=[N+]=[N-])C2)=O)CCC(=O)N(C)C1 C(=O)(C(CN(C)C)C(C)C)NC(C(N1C(CC)(CC)CC1)=O)Cc1ccco1 c1(C(c2nnnn2CC2CC2)NCC(CC)Oc2ccncc2)c(Cl)ncn1C c1(C(N2CC3CCN(C(C4C(OC)C4)=O)CC32)=O)cccc2cccc(OC)c12 N1(C(c2c(CC)nco2)=O)CCOC(C(C)NC(c2ccccc2C2CC2)=O)C1 CC#CC1CCN(C(=O)CCN(C(c2cc(C#N)cn2C)=O)CC2CC2)C1 c1(C(=O)NC(CNC(c2cnn(CCC)c2Cl)=O)(C)CO)ncnc2c1CCC2 C1(C)(C(=O)NCCC(=C)C)CCN(C(=O)C=C(C)c2ccccc2)CC1 CC1OC2(C(N3CC4CC(NC(c5cnnc(O)c5)=O)C3C4)=O)CCC1CC2 C(c1nc2ccccc2o1)=CC(=O)NC1CCN(C(C=C(CC)C)=O)CC1CO c1(SCC(CC)N(C)C)nnc(-c2ccc(OC)cc2)n1CCC#N N1(C(c2c(SC)scc2)=O)C2CCC1C(CNC(=O)C(C)CC(F)F)C2 Cc1ccc(C23CC(C(=O)NCCc4cc(C)n(C)n4)(C2)C3F)cc1 n1(C(C)C)ncc(F)c1C(N1CCOC(C(C)NC(=O)C=Cc2ccco2)C1)=O c1(C(N2C(CNC(C3CCCO3)=O)CC(C)(C)C2)=O)cc(Br)c2c(c1)OCO2 C12(C(=O)NCC3N(C(CCC(C)(F)F)=O)CC3)CCOC1CCOC2 N1(C(CCOCCCOC)=O)CC2CCC(C1)N2Cc1ccc(C)cc1F N1(C(c2cnc(C(C)O)s2)=O)CCC(C)(NC(c2n[nH]cc2CC2CCC2)=O)C1 N1(C(CCC(C)OC)=O)CCN(C(c2ccc(C)cc2N)=O)CC1C1CC1 c1(CNC(C(C(C)SC)O)=O)c(C)nn2c1CN(C(=O)CCCSC)CC2 c1(C(=O)NCC2CCC(NC(Cc3cc(C)[nH]n3)=O)C2)c(Cl)ccc(F)c1C N1(C(C=C(C)Cl)=O)CCC(CNC(=O)C(C(C)C)OCC(C)C)C12CCC2 N1(C(c2c(C)nccn2)=O)CCCC12CCCN(C(=O)Cc1ccc(Cl)cc1)C2 C1(CC)(NC(=O)CCOCC(F)F)CCN(C(c2occc2C)=O)CC1 CCC(C(=O)N(C1CCN(C(C2(C)CCCCC2)=O)C1)CCO)C(C)(F)F C1(CC(=O)NC(CC#C)C)CC(C)N(C(=O)CSCCCC)C1 C1(C(N(CCNC(C2C(C=C)C2)=O)C(C)C)=O)CC(F)C(=O)N1C C1(CC)CCCN(CC(=O)N(C)CC2CCCN(C(c3cn(C)c(O)n3)=O)C2)C1 C12(NC(c3nc(CNC(C)=O)sc3)=O)CC1CN(C(=O)CC(O)CN(C)C)C2 C1(F)(C(=O)NC2(CC)CCOCC2)CCCN(C(c2cc(C)c(C)o2)=O)C1 CC(C)CN=C(NCc1ccccc1CS(C)(=O)=O)NC1CCCC1(F)F C=Cn1nccc1C(=O)NC1CC(OCC)CN1C(=O)COCCCC C1(O)(c2cn(CCNC(C(CCC)F)=O)nn2)CCC(C)(C)CC1 C1(C(N2CCCC(CC)C2)=O)CN(C(c2cc(O)cc(=O)o2)=O)CCN1C C1(C(N(CC(c2ccccc2)N(C)C)C)=O)CCCC2(CC2)C1.N12CC(O)(C1)C2 C1(NC(Cc2cc(C)on2)=O)CCN(C(=O)CC2CCC=CCC2)CCC1CO c1(CC(=O)NC2(CN(C)C(C3CCCC(F)(F)C3)=O)CC2)cc(Cl)cc(Cl)c1 c1(C(=O)NCC2CC(NC(=O)CCF)C(O)C2)cccc2c1COC2 C1(C(C)(O)CNC(=O)CCc2ccc[nH]2)CCCN(C(=O)CP(C)(C)=O)C1 c1(NC(CC2N(C(c3ccc(OC)s3)=O)CCOC2)=O)c(C)ccc2c[nH]nc12 CC1CCC(NC(=O)CCC2CC(C)(C)CO2)CN1C(=O)CCn1cncn1 c1(C(=O)NC(CNC(c2c(C)occ2)=O)C2CCC2)ccc(F)c(C)c1N C1(NC(Cc2cn(C)nc2)=O)CC2(C1)CC2C(=O)NC1CN(CC(F)F)C1 N1(C(C(CSC)O)=O)CC(NC(c2csc(C(F)F)n2)=O)C(O)C1 CC(C)CC(CNC(=O)C(C1(O)CCCC1)F)NC(c1cc(Br)cs1)=O c1(OC)ccc(O)cc1C(=O)NC1(C)CCCCC1O C1(C2CC2)(CNC(C(CCCC)N(C)C)=O)CCN(C(c2cc(C)c(C)[nH]2)=O)C1 OC1CC2(CC(NC(c3sccc3Br)c3nnnn3C3COC3)C2)C1 N1(C(C2(C)CCC(=O)N2)=O)CC23CCCCC2(C1)CN(C(=O)CCCF)C3 c1(SC)ccc(Cc2cc(-c3ccccc3)cs2)cc1.N12CC(F)CC1C2=O c1(NC2C(NC(c3c(CC)nc[nH]3)=O)CS(=O)(=O)C2)cc(C#N)nc(C)n1 CC(CCCNC(c1cc(Cl)cs1)=O)NC(=O)Cc1nc(C(F)(F)F)n[nH]1 C1(NC(CC(CCC)CC)=O)CC2CCCC(C1)N2C(C1CCS(=O)(=O)N1)=O C(c1ccccc1C)=CC(=O)NC(C1CCCC1)CNC(c1c(C)cn(C)c1)=O C1(NC(CCOCC#C)=O)CCC(C)(NC(=O)C(F)Cc2ccccc2)CC1 N1(C(CCC2CCN(C(C(CC(=O)OCC)C)=O)C2)=O)CCc2ncn(C)c2C1 CCCC(C)(CC)C(=O)N1CC2CC1(CNC(c1cccnc1)=O)C2 C=C1Cn2c(C(N3CCN(C(c4c(C)ccn4C)=O)CC3CC)=O)nnc2S1 c1(CC(N2CCCC(C)(NC(C(C)NS(C)(=O)=O)=O)C2)=O)ccc2nsnc2c1 C1(CNC(=O)CCCCCCn2cc(CO)nn2)CCCC2(CCOCC2)O1 c1(CC(=O)NC(CCNC(C(CN(C)C)N(C)C)=O)C)ccc2c(c1)COC2 C12(C(=O)NCc3ccc[nH]3)CC(c3cccc(C(F)F)c3)(C1)C2F C1(NC(C(C)=C(C)C)=O)CC2(CCN(C(c3cccc(C4(C)CCO4)c3)=O)C2)C1 C1(C(=O)NC(c2c(C)n[nH]c2C)C)CN(C(c2cocn2)=O)CC(C)O1 C1(C(N2C(CN(C(c3snc(C)c3N)=O)CC)CCC2)=O)C2CN(C)CC12 C12(CNC(Cc3ccc(OC)cc3)=O)CC(C1)C(NC(c1cnc[nH]1)=O)CO2 c1(CC(=O)NCC=CC(=O)NCC(C)(C)O)cccnc1O C1(C(C)C)CN(C(c2nc(Cl)cs2)=O)CCCN1C(c1cc(C(C)(C)C)c[nH]1)=O N1(C(CC2(N(C)C)CCCC2)=O)CCC(CCCNC(C2CCOC2)=O)CC1 c1(C(=O)NC2CC(C)NC2)ccc(S(=O)(=O)NC(C2CCCCN2C)C)cc1 C1(c2onc(C)n2)CC(F)CN1C(C1COC(C)C1)C(=O)NCC(F)F Cc1nnc2n1CC(C(=O)NC(C)CCNC(=O)CNC(c1ccoc1)=O)C2 c1(C(C)NC(=O)C(=O)NCC2CS(=O)(=O)CCO2)nc2ccccc2[nH]1 CC1CCOC(C(=O)NC(C)(C(=O)NCC(c2cnc[nH]2)C)C2CCC2)C1 C1(CC=C)(C(=O)N(CC(O)COC)C)CCN(C(=O)CCOCC)C1 n1(CC)cc2ccc(C(=O)NCC=CCNC(c3ccc(F)o3)=O)cc2n1 c1(CNC(=O)NCC)ccc(S(=O)(=O)NCC2(CC(F)(F)F)CC2)cc1 C1(CC(=O)NCC(CCC)C)CN(C(c2cccc(CC#N)c2)=O)CC12CC2 CC(C)C(O)C(C)(C)C(=O)NC1CCC(C(=O)NCc2cncc(Cl)c2)C1 Cc1cc(-n2ccc(C(=O)NCCC(C)(C)O)n2)ccc1Cl CC1(C)CCC=C1C(=O)N1CC2CCN(C(=O)CC=C(Cl)Cl)C2C1 N1(C(C(C2CCOCC2)OC)=O)CCN(C(=O)CCCN=[N+]=[N-])C(C2CCC2)C1 C(=O)(C1CS(=O)(=O)c2ccccc21)N(C1CCCC1)CCNC(c1csnn1)=O C12(CN(C(C=CCN(C)C)=O)CC3CC3)CN(C(=O)C3=CCC3)CC1CS(=O)(=O)C2 CN1CC(O)CC1C(N1CCC(N2CCN(C(=O)CC(F)(F)F)CC2)C1)=O.c12cccn1c2=O c1(C(=O)NC(CC)CNC(=O)C(C)CC2CC2)noc2cc(F)ccc12 c1(C(=O)NCC2(OC)CN(C(C(CC)F)=O)C2)cccc(Cl)c1O N1(C(C(C)OCc2ccccc2Cl)=O)CC2CCCC(C1)N2C(C1(CF)CC1)=O CCCC(C(=O)NC(Cn1ccnn1)C(=O)NCCCCS(C)=O)OC c1(NCC(=O)NC(c2ccc(F)cc2)C)cn2c(n1)CCCC2C(=O)O N1(C(C(CC)SC)=O)CCc2c(ncn2C)C12CCN(C1CCCNC1=O)C2 N1(C(c2occ(C)c2)=O)CCN(C(=O)CCC2OCCO2)CC1CC(F)F C1(NC(CCCC(C)O)=O)CC2CN(C(c3ccc(NC=O)cc3)=O)CC2C1 C(=O)(CC(C)CC(C)(C)C)NCC12OCC(NC(C(C)OCC(C)C)=O)(C1)C2 C#CCC(CC(=O)NC(C1CSC1)C)NC(=O)CC1(COC)CC1 c1(C(=O)NC2CC(N(C(C(C(C)C)F)=O)C)C2)c[nH]c2ncc(Br)cc12 Cn1nc2c(c1C=CCSc1ccccc1)CCC2 N1(C(C(C)O)=O)CC(F)(F)CC1CCNC(c1scnc1C(C)(C)C)=O c1(CC(=O)NCC2(NC(C3CC3F)=O)CCC2)ccccc1Br c1(OC)cc(C(=O)NC2CN(C(C3CCCC3)=O)C2)cc(Br)c1OC(C)C c1(C(N(CCCNC(C2(C)CCCN2C)=O)C)=O)cnc(S(C)(=O)=O)s1 c1(C(=O)NC(CNC(C(C)N2CCCC2)=O)(C)C2CC2)cc(C(N)=O)co1 c1(C(=O)NCC2CC(CNC(c3c(C)cnn3C)=O)OC2)cc(Cl)cnc1C C1(CNC(c2cc(C(C)C)no2)=O)CC(NC(c2cn[nH]c2)=O)C1(C)C C(=O)(C1Cc2ccc(F)cc21)N1CCN(C(CN(C)CC)=O)CC12CCC2 C1(C#CC(=O)N(C(C)CNC(=O)CCc2c(F)cccc2Cl)C)(CC)CC1 C1(CNC(C(=O)NC2(CCC)CC2)=O)CC(C)(C)CN1 C1(OC)CC2CC(C(c3nnnn3C3(C)CC3)NCCCCF)CC12 c1(C(N2CC(O)(CNC(Cc3scc(C)n3)=O)C2)=O)cc2c(F)ccc(F)c2[nH]1 C1(NC(CCOc2ccc(C)cc2)=O)CCN(C(c2ncc(F)cn2)=O)CC1C C1(CC)CCC(C(=O)N(CCCCCNC(=O)CCCc2csc(=N)[nH]2)C)O1 C(=O)(C1CCc2c[nH]nc21)NC(CC=CC)C(=O)O C1(NC(=O)CC2CC=CCC2)CC(F)CN(C(c2cc(Cl)ccc2O)=O)C1 N1(C(C(CC2CN(C(C=C(CC)CC)=O)C2)F)=O)CC(O)CC(C)(C)C1 c1(C(N(CC(CC)NC(c2n[nH]c(C)c2Cl)=O)C)=O)cnc(C)c(C)c1 N1(C(C(=O)N(CC(C)NC(C=C(CC)CC)=O)C)C)CCCCC1=O c1(C(=O)NCC2N(C(c3ccc(OCC)c(OC)c3)=O)CC2)n[nH]c(C)c1[N+](=O)[O-] Cc1ccnc2c(NC3COc4ccccc43)ccnc12 c1(OC)cc(CN2CCC2Cc2cc(Cl)ccn2)ncn1 CC1CCC(CNC(=O)C=C2CCC2)N(C(=O)CN(c2ccncc2)C)C1 c1(C(=O)NC(CC(C)C)C(F)F)c2ccccc2nn1C CCCC(C(=O)OC)C(=O)N1CC(NC(c2cc(C(C)C)[nH]n2)=O)C(N=[N+]=[N-])C1 N1(C(C2ON=C(CC)C2)=O)CC(N(C(=O)C(c2ccccc2)=O)C)C2(CC2)C1 CN1CCOC(C(=O)N(CCCNC(C2CNC(=O)N2)=O)CC2CCCC2)C1 c1(C2(NCc3nc(-c4ccc(OC)cc4)oc3C)CC2)cc(Br)cc(Cl)c1F CC(C)C(CNC(=O)CCn1ccnc1)C(=O)N1CCC(N(C)C)(CF)C1 N1(C(CNS(C)(=O)=O)=O)CCC2CCN(C(=O)CSc3ccc(Cl)cc3)CC12 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)(CNC(c2cscc2Cl)=O)C1 C(c1ccc(C(N)=O)o1)=CC(=O)N(CCN(C(C1C(C=C)C1)=O)C(C)C)C N1(C(COC2(CCCC)CC2)=O)CCC(n2cc(-c3csc(C)n3)nn2)C1 C(CCC(C(=O)NCC(C)CO)N(CC(=O)OC)CC)OCC C1(c2nc(CC3(N(C)C)CCCC3)[nH]n2)CCN(CC2CCCS2(=O)=O)CC1 CCC(C(=O)NCCCC(C)NC(C1(C(N)=O)CC1)=O)C(C)C O=C(C=CSc1nc[nH]n1)NC(c1cc(C(F)(F)F)on1)C1CCCN1 N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(c2cc(C)ns2)=O)C1 C1(NC(C)=O)CC2CN(C(=O)C(C)(C)Oc3ccc(F)c(F)c3)CCN2C1=O c1(C(=O)NCCCCN(C(CS(=O)(=O)NC)=O)C)cc(F)ccc1C(F)F c1(C(=O)NCC(C2CCCC2)NC(=O)CCc2ncco2)cc(Cl)ccn1 c1(C(N(CC(CNC(C(F)OC)=O)O)C)=O)cnc(C2CCC2)cc1C C1(NC(=O)NC(C)C(C)(C)F)CCN(c2ccccc2C(F)(F)F)C1=O c1(OC)ccc2cnn(CC(N3CCC(C4(C(=O)O)CC4)CC3)=O)c(=O)c2c1 N1(C(C(CCC)OC)=O)CC(NC(c2c(OC)ncnc2C)=O)CC2(CCC2)C1 C(=O)(C(O)CCC(C)C)NCC(CC(=O)N(CC)CC1CCOC1)C1CC1 c1(C(N2CCC(NC(C(C)n3cnnn3)=O)C2C)=O)cccc2c1CCCCC2 c1(CC(=O)NC(C)C(N2CCOCC2CC2CCCC2)=O)ccc(Br)cc1 C1(NC(C2(C=C)CCC2)=O)CCCCC1NC(=O)CCN(C(CC)CC)C C1(C)(C(=O)NCCC2OCCN(C(CC(C)(C)OC)=O)C2)COCC1(F)F C(N=c1nc2[nH][nH]cc-2c(O)n1)C12CC(NC(Cn3c(C)ccn3)=O)(C1)C2 N(C1CCc2cc(CNC(C3(C#N)CC(=O)C3)=O)ccc21)C(C1(C)CC1(Cl)Cl)=O C=CC1(C(=O)NCCC2(O)CN(C(c3ccc(CCC)[nH]3)=O)C2)CCC1 N1(C(CC=CC)=O)C2CCC1CC(NC(c1cn(CC(=O)N(C)C)nn1)=O)C2 N1(C(C2CCCS2(=O)=O)=O)CCCC2(CCCCN2C(C2CCC(O)CC2)=O)C1 c1(C(=O)NC2CN(C(c3[nH]cc(CC)c3)=O)CC2C(F)F)cccc2[nH]ccc12 C1(CC)C(=O)N(C)CCN1C(C1CN(C(c2ccc[nH]2)=O)CCC1O)=O CCCCC(C)CCC(=O)N1CCC2C(C1)CN2C(=O)CCn1ccnc1 N1(C(c2ncn(C)c2)=O)CCCC(Nc2cnncn2)C1 c1(C(=O)NCC(CNC(C2(CC=C)CC2)=O)F)cc(Cl)ccc1Cl C1(NC(C23CC(C)(C2)OC3C)=O)CC2CCC2C1.N1(C(=O)NC)CC(NC=O)C1 C#CCC(CC(=O)NCC1CC2(CC2)C(=O)O1)NC(c1cc(Cl)c[nH]1)=O CCC(C)(C#N)C(=O)NC(CC(=O)N(CC(C)C(C)C)C)C(C)OC N1(C(C=Cc2cnc(-n3cc(CCN(C)OC)nn3)o2)=O)CCN(C(C)C)CC1 c1(C(N2C(C)(CNC(C3C(C)(C)C3)=O)CCC2)=O)cc(Br)cnc1N c1(CC)[nH]nc(C(=O)NC2CC3CC2CN(C(=O)C(CSC)OC)C3)c1[N+](=O)[O-] c1(COCc2cn(C3CN(C(C(C(=O)OC)OC)=O)C3)nn2)cc(C)cc(F)c1 C1(NC(CCCCOCC)=O)CC=C(C(=O)NC2(C)CCC(C)(C)C2)C1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(CCNC(=O)Cc2cccs2)CC1 C1(NC(C2CCCCO2)=O)CCN(C(C2CCCCC2(F)F)=O)C12CCCC2 Cc1cc(=NCCCCC#N)[nH]c(=NCCOCCS(N)(=O)=O)[nH]1 c1(C(=O)NC2(CO)CN(C(COCc3cc(C)no3)=O)C2)cc(Cl)c(C)cn1 C1(C(=O)NC2CCN(C(CCCC(C)O)=O)CC2F)CS(=O)(=O)CC(=O)N1 C(=O)(C1=CCc2ccccc21)NCCCC(C)NC(C(CC(C)C)NC(C)=O)=O C(=O)(C(CO)C(C)(C)C)NC1(C(N2CCC(C(C)(C)O)C2)=O)CCCC1 Nc1nccnc1C(=O)NOCc1cn(C2CCCCC2)nn1 N1(C(CNCCC)=O)CC(NC(=O)C=CC(=O)OC(C)(C)C)C(C(F)(F)F)C1 C1(C)(CN(CCN2CCN(C(=O)OCC)CC2)CC)CNCCC1(F)F Cc1cc(N(C(C)CNC(=O)COCc2cc(C)on2)C)n2nc(C)cc2n1 N1(C(CN(C(C(CC)C)=O)C)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 CC1CC=C(C(=O)N2CCC2CNC(=O)Cn2ccc(Br)n2)CC1 C1(NC(=O)COC2CC2)CCN(C(c2cccc(Br)c2Cl)=O)CC1O C(C)(C)(CC(F)C(=O)N1CCCC(N2CCC2)C1)NC(C(C(C)C)SCC)=O C1(C(=O)NCCC(C)(C)NC(CCc2ccn(C)n2)=O)CC2CCC1O2 c1(OC)ccc(CC(=O)NCC2CC(NC(=O)CC=C(C)C)C2(C)C)c(F)c1 C12(CN(C(CN(C(CN(C3CC3)CC)=O)C)=O)C)CCC(CC1)CC2 Cc1cc(C(C)C(=O)NCCCCN(C)C(C2C3CCC(F)(F)C23)=O)cc(F)c1 c1(CC(=O)NC2CCN(C(C=CC)=O)CC2O)nnc(O)c2ccccc12 Cc1cc(CN2CC3CC3(C(=O)NCc3cccc(C4CC4)c3)C2)cc(C)c1Br C1(CNC(C(COC)C)=O)CCCC2(CN(C(c3cc(N)c(Cl)c(O)c3)=O)C2)O1 N1(C(C(CC)COC)=O)CCCC(C)(C)C1C(=O)NC1CCC2CCC12 C12(C(N3CCC(N(C)C(C4C(C)(C)OC4(C)C)=O)C3)=O)CC=CCN1CCC2 N1(Cc2ccc(OC)c(SC)c2)CCC2(CCC(O)C2)C1 CCCCC(O)C(=O)N(CCC(C(C)C)NC(=O)C(C)Sc1ncccn1)C C1(NC(C(C(C)C)O)=O)CCCCN(Cc2ccc(Cl)cc2Cl)C1 C(=O)(C(CCCOC)NC(c1c[nH]nc1C(C)C)=O)NCC1CN(C(C)=O)C1 c1(C(N(C2CCN(C(=O)CCC(C)(C)O)CC2)CC)=O)ccc2c(c1)OCCO2 Cc1ccnn1C(C)C(=O)NC1CC(CNC(c2csc(C(C)(C)C)n2)=O)C1 Cc1cc(C(N2CC3CC2CN3C(=O)C(C)NC=O)=O)nc2nccn12 O=C(CCCCCn1cc(-c2ccc(Cl)cn2)nn1)NC1(C(=O)O)CCS(=O)(=O)C1 C1(NC(CC2CN(C(C=CCN(CC)CC)=O)C2)=O)CCCN(C)C1C c1(C(N2CCC(CNC(CCC(=O)NC)=O)C2)=O)sc(C#N)cc1Cl C(CCCCCC(C)C)n1cc(C2N(C(CC(C)(C)OCC)=O)CCCC2)nn1 N1(C(Cn2ncc(C)c2)=O)CC2CCN(C(C3COCC3C(F)F)=O)CCC2C1 c1(C(N(CC(CC)NC(C(CCCC#C)C)=O)C)=O)cc([N+](=O)[O-])c(C)cc1Cl c1(C(=O)NC2CC3CC2N(C(C2CC2F)=O)C3)cc2c(nc1O)CCCCC2 C1(NC(Cn2nc(C)c(C)c2C)=O)CC12CCC(NC(c1cccnn1)=O)CC2 n1(CC(N2CC(CC(C)NC(=O)Cc3cnoc3)C2)=O)nnc(C2CC2)n1 C=CC(C)(CCOC)C(=O)NC(C)C(=O)NC(C)CCC1CC1 C(=O)(CC(C)(C(F)F)N(C)C)N1CCC(C)(NC(C(CCOC)(C)C)=O)C1 C1(NC(C(C)OC2CCCC2)=O)CN(C(=O)Cc2c(F)cncc2Cl)CCC1F c1(C(N2CCC(CCC(=O)N(CCC)C3CC3)C2)=O)ccccc1C1CC1 N1(C(N2CC(C)N(c3ccccc3)CC2)=O)CC(CCO)C2CCCC12 c1(-c2nn(CC)c(C(F)(F)F)c2)ccc(N(C)C)cc1F C(c1ccc(C)cc1)=C(C(=O)NC(CN(C(c1ccc(CC)nc1)=O)CC)C)C CCCC(C)(O)C(=O)NCCCCN(C)C(C1(C)CCN(C(C)=O)C1)=O c1(OCC)ccc(C(=O)NC2CCC(C(=O)Nc3cnc(OC)cn3)C2)nc1 C1(NC(=O)Nc2c(OCCOCC)cccc2)CCOC2(CCS(=O)(=O)CC2)C1 C1(OC)CN(C(=O)C(C)(O)C2CCC2)CCC1NC(c1cc(Cl)cs1)=O C(=O)(CC(C(C)(C)C)NC(=O)CC1(N(C)C)CC1)NC1(CC)CC(C)(C)C1 CCN=c1[nH]c(C)c(C(=O)NCC(O)CN(C(=O)C(S(C)(=O)=O)C2CC2)C)s1 Cc1ncc(C(=O)NCC2CCN(C)C2)c(Cl)c1Br c1(C(=O)NCCOCCCNC(C(CCSC)O)=O)ccc(S(C)=O)cc1 C1(C)(NC(c2n(CCN(C)C)ncc2)=O)CCN(C(=O)CCC2CC(F)(F)C2)C1 N1(C(Cc2c(C)noc2)=O)CC(NC(=O)C=Cc2cscn2)C(O)C1 c1(-c2nc(CC(C)C)nn2-c2ccnc3ccsc23)ccc(F)c(S(C)(=O)=O)c1 CC1CC(NC(c2cnc(C3CC3)o2)=O)CCN1C(=O)CSc1nnc(S)s1 N1(C(C2(CCC)CC(=O)C2)=O)CCCC(CNC(C2CC(=O)NC2=O)=O)CC1 CC1(C(=O)NCC2(O)CC(NC(=O)CN3CCCC3CO)C2)CC=CCC1 c1(C(=O)NCCC(C)N(C(=O)CCc2ccoc2)C)ccn2ccccc12 c1(OC)ccc(CN2C(C(=O)Nc3cc(C4CCC4)no3)CC3CC23)cc1F c1(C(=O)NCC(C2CC2)NC(C#CC2(C)CC2)=O)ncn2cc(Cl)ccc12 c1(-c2ccc(C(N3CC(C(=O)OC)N(C)CC3)=O)cc2)nccn2nccc12 C1(CCS(=O)(=O)NC)NC(=O)CCN(CC(c2cccc(C)c2)(F)F)C1=O c1(OC)ccc(F)c(C(N2CCCC(C(=O)Nc3ccnc(Br)c3)C2)=O)c1 C1(CN(C)C)CCCN1C(=O)C(C1(O)CN(C(C2(Br)CC2(C)C)=O)C1)F C1(C(N2CC(NC(CC(C)C3CCCC3)=O)(CF)C2)=O)CC(F)(F)CS1 CCC(C(=O)N1CCOCC1CNC(c1c[nH]nc1C(C)(F)F)=O)C(C)C N1(C(c2cc(OC)no2)=O)CC(C(N2CCC3C(C(N)=O)C3C2)=O)C2(CC2)C1 c1(NCC(=O)NC)nccc(=NC(C)c2nc(O)n[nH]2)[nH]1 N1(C(C(=Cc2cnc[nH]2)C)=O)CCC2CN(C(=O)CCCN3CCCCC3)C2C1 N1(C(c2c(Cl)cc(C)c(C)c2)=O)Cc2ccccc2CC1CNC(=O)CC(C)F Cc1c(O)ccc(C(=O)NCC2CCN(C(c3ccc(Cl)nc3)=O)C2)c1C C1(CNC(C(C(C)C)OC)=O)CC2CCC1N(C(=O)CN1CCCC1=O)C2 N1(C(c2c(CNC(CC(C(C)C)C)=O)cc[nH]2)=O)CCC(O)CC(C)(C)C1 CP(C)(=O)C(CC(=O)NC12CCCCCC1N(C(=O)CCC#N)CC2)C(F)(F)F N1(C(CCCCC)=O)CCCCC(C(=O)NCC2CC2OC(C)=O)C1.OCC C(CC(=O)N1C2CCC1CC2)(C(F)F)NC(C1CCC(OC)CC1)=O C1(C(CC)NC(=O)NCCOCC(C)(C)OC)CN(C)CCO1 C1(C(=O)NC2CCC(CNC(C(CC)(F)F)=O)CC2)CCc2nccn2CC1 Cc1cc(C(=O)N(C)CCOCCCN(C(=O)C(F)n2cccn2)C)ccn1 c1(SC)ccc(OCCOC(=O)NC2C=CCC2)cc1 C1(NC(C2CC(CCC)C2)=O)CCC(NC(C2CC3C=CC2O3)=O)CC1 C1(NC(COCCN(C)C)=O)CS(=O)(=O)CC1NC(=O)C=CC1(C)CCOCC1 N1(C(CC2ON=C(C)C2)=O)CC(C)CC1C(=O)NC(c1cccnc1O)C CN1CCC(C(=O)NCCCn2cccn2)(NC(=O)C(F)=CC2CC2)C1 C1(CCOC)CN(C(=O)CSCCN(C)C)CCN1C(C1CC12CC(O)C2)=O C1(N(C2CCOCC2N(C)C)C(C2C3CN(C(C)=O)CC32)=O)CCCCC1(C)C N1(C(C2(C)C=CCC2)=O)CCC(C(F)CNC(c2cc(Cl)no2)=O)CC1 C(=O)(CCC(=O)NCc1cc(C(N2CCC(OCC(N)=O)C2)=O)n[nH]1)NC c1(OC)cc(Br)ccc1CNCCCCCN N1(C(C(C=C)O)=O)CCCC2CN(C(c3[nH]nnc3COC)=O)CCC12 C1(NC(CCN(CC)CC)=O)CC(OC)CN(C(C2CCC(C(C)C)CC2)=O)C1 c1(NC(C2C(NC(c3c(C)n[nH]c3)=O)C2)=O)ccc(I)c(C(F)(F)F)c1 C1(C(N)=O)CC1C(=O)NCCSCC(=O)NCCCOCF Cc1oc(C2CC2)nc1C(=O)NC1(C2CCCCN2c2nnc(C(F)F)s2)CC1 c1(COCC)cn(CC(C)(C)CNC(C2(CSC3CC3c3nccs3)CC2)=O)nn1 c1(C(=O)NC2C(CNC(c3cn(C)nn3)=O)C2)ccnc(-n2cncn2)c1 C1(C(=O)NC2C(C(=O)NCCCCC#N)CCC2)CCNC(=O)C1 c1(C(=O)OC)nc(NC2CCN(C(=O)CC3CC4(CC4)C3)CC2C)ncc1Cl N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2C(CCN2Cc2ncc[nH]2)C1 C1(C(=O)NC2CN(C(c3c(OC)nn(C)c3)=O)CC2C)CCn2c(cnc2C)C1 CC1(C)Cc2cccc(CNC34CCCC(CC3CO)C4)c2O1 N1(C(C)=O)CCC(C)(NC(=O)C(O)CN2CCCC2)C1.N12CCC(C1)C2=O c1(C(N2CC(NC(c3n(CCCC)ncc3)=O)C(C)C2)=O)cc(F)cc(C)c1N CCCCC(CC(=O)NCC(c1cccnc1)O)NC(C1CC1C(F)(F)F)=O C1(N(C(c2c(C)scn2)=O)C)CCCC(N(C(=O)Cn2cc(C(F)F)cn2)C)C1 c1(C)ccc(F)cc1.C1(C)(C(=O)OCC)CC1C(=O)N.C1C(=O)N(CC)CCCO1 CC1CCN(C(C23CC(C)(CO2)C3)=O)CC1NC(c1cccc(=S)n1O)=O C1(CNC(C(C)=CC)=O)CC2COCC2N1C(=O)C(O)Cc1ccccc1 N1(C(C2C(C)C2)=O)CCN(C(=O)C(c2cc(Cl)ccc2Cl)(C)C)CC1CCO N(C1CN(c2ncnc(Cl)c2F)CCc2ccccc21)C(C1C(=O)NCCC1)=O c1(CC)cccnc1C(=O)NCC(C1CCCN1C(=O)CN1CCCC1=O)(C)C Cc1cn2c(C(=O)NCC3(NC(C4C5CCN4CC5)=O)CCCC3)c(C)nc2s1 CCS(=O)(=O)CC(=O)NCCCCCN(C(=O)C(C)(C)C1CCCO1)C c1(C(=O)NC2(C(N(OC)CCO)=O)CCC(C)(C)C2)cccc2cncn12 CC1=NOC2(C1)CC(C(N1CCC(C)(C)C(NC(=O)CSCCN(C)C)C1)=O)C2 c1(-c2nnc(N3C(c4n(C)cnn4)CCCCC3)o2)nccc(Br)c1Br CC1CN2CCN1C(C(=O)NCC1CCN(C(=O)CCCC(N)=O)C1)C2 N1CCC2(CCCC2Nc2ncc(C#N)cc2F)CC1.c1(C=O)coc(Br)n1 c1(C(=O)NC2CN(C(C3C(C(C)C)CCO3)=O)CC(C)C2)c(F)cc(F)cc1F C1(NC(=O)NCc2c(NCCC)cccc2)CCN2CCCC12 C1(CNC(C(CCC)NC(C)=O)=O)(CO)CC12CCN(C(=O)C(C)NC=O)CC2 C1(NC(c2cc(C)ncn2)=O)CC2CCC1(NC(=O)CC1(N(C)C)CCC1)C2 C1(C(N2CC(CN(C(CC3(OC)CCC3)=O)C)C2)=O)CCCC2CC12 N1(C(Cc2cc(C)sc2)=O)CCN(C(C2CC3CCCC3C2)=O)CC1C1CC1.C1CC1 CCCC(C)C(=O)NCC1(CNC(=O)C(F)CN(CC)CC)CCOCC1 C1(C(=O)NC(C(=O)O)C2CC2)CN(C(c2ccc(-c3nccs3)cc2)=O)CCO1 O=C(N=c1ccn(C2CCSCC2)[nH]1)Nc1ccc(O)c(Cl)c1 C1(CC)CN(C)CCCN1C(C1CCN(C(=O)C(C)(C)O)CC1)=O Cc1cc(C)c(C(=O)NCC2(NC(=O)C=Cc3cc[nH]n3)CC2)c(S)n1 C#CC1CCC(C(=O)NC2COCCC2NC(c2[nH]nnc2C)=O)CC1 N1(C(CN(CC#C)C(c2ccn3ccccc23)=O)=O)CCC2CCC(C2)C1 CC(C)(C)CCC(F)C(=O)NC(CC1CCC1)C(N1Cc2cc(F)ccc2C1)=O N1(C(C(=O)Nc2ncc[nH]2)=O)CC(CNC(c2ccccc2F)=O)N2CCC1C2 C1(C(=O)NCC#CCC)CCCCCCN1C(c1ncc2ccccn12)=O c1(C(C(=O)NC2CCCN(C(c3cnc(C)[nH]3)=O)C2)C(C)C)ccc(C#N)cc1 c1(C(C)C)nc(NCC2CCCS2)cc(N2CCC(c3cc[nH]n3)CC2)n1 N1(C(C(N2CC(C)OCC2)=O)=O)CCCC2CCC(C)CC12 c1(C(=O)NC2CN(C(c3nc(C)c(C)s3)=O)CC2C)cc2oc(Br)cc2[nH]1 c1(C(=O)NC(CCN(C)C(C2CC2F)=O)C(C)(C)C)cc2ccc(F)cc2s1 c1(C(N2CCCCC(NC(CC(COC)(C)O)=O)C2)=O)ccc2c(c1)C(=O)OC2 C1(NC(CC(CCSC)O)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC1(C)C Cc1ncncc1C(=O)NC1CC2(C1)CC2NC(c1n[nH]cc1F)=O C1(CN2CCC(C(=O)NCCc3cn(C)nc3)C2)COC(C)(C)O1 c1(CNc2ccc(NC(c3ccccc3)CNC(C)=O)nc2)ccc(Cl)c(F)c1 CCC(C)(C)C(O)C(=O)N1CCC(C)C(NC(c2cc(C(C)C)oc2C)=O)C1C Cc1cn2cc(CC(=O)NCCC3CCCN3C(=O)CN3CCNC3=O)nc2s1 C(C(C)(C)C(=O)NCCCN1CCOCC1)N(C)C(c1cc[n+]([O-])cc1)=O c1(CC)ccc(S(=O)(=O)NC2CN(Cc3cccc(OC)c3)CC2(F)F)cc1 CC1CCCN(C(=O)C(=O)N(CCCCNC(C2CCCN2N=O)=O)C)C1 N1(C(C2(C)CC2(F)Cl)=O)CCC(NC(c2c[nH]cc2Br)=O)C(CO)CC1 C1(CNC(c2cc(CCC)oc2C)=O)CCCN(C(=O)C(C(C)C)OC)CC1 C(=O)(CC(C)CC(C)C)N1CCC(NC(c2n(COC)ncc2)=O)C(CO)C1 C12(CNC(CC(C=C)C)=O)CCCC(CN1C(=O)COc1cccc(C)c1C)C2 c1(C(C)C)ccc(CC(=O)NCC2CN(C(=O)CCCC3CCC3)CC2O)cc1 C(=O)(C1Cc2ccc(F)cc21)NC(CC=C)CNC(c1ccc(C)nc1C)=O c1(C(=O)NC2CN(C(C3(C#C)CCCC3)=O)CC2C)ccc(S(N)(=O)=O)cc1 c1(C(=O)Nc2n(C)nnc2)ncn2cc(-c3ccc(-c4cccnc4)cc3)sc12 Cc1ncc(Br)cc1NC(=O)C(O)C(F)F C(=O)(C(=O)N=S(C)(C)=O)NCC1CCCC(NC(c2c(CC)nc(C)nc2)=O)C1 CCCCC(C)C(=O)N1CCC(COC)(NC(c2c(C)cnn2C)=O)C1 C1(CNC(C2C(OCC)C2)=O)CC2(C1)CN(C(c1ccsc1C(F)(F)F)=O)C2 Cc1c[nH]c(CC(N)=O)c1C(=O)NCC(C)NC(=O)C(C)Cc1ccc(F)cc1 c1(OC)nc(NC(C2CN(C(C3CCCCN3C)=O)CCN2)=O)c(Br)cc1Br C1(CCN(C)C(C2CCCNC2=O)=O)CCCCN1C(=O)C(C)(F)F c1(NC(=O)COc2ccc(SC(F)(F)F)cc2)ccc2c(c1)OCO2 C1(C(=O)NCC(CC)(CC)NC(CC)=O)CCCC1C1CC1 c1(CC(=O)NCCN(CC(C)O)C(c2cnns2)=O)nccn1C CCS(=O)CC(=O)NC1CN(C(=O)Cc2c[nH]nc2O)CC1C C(N=c1[nH]c(N2CCC(c3nncs3)C2)nc2c1SCC2)c1cccc(CC)n1 C(C(C)(C(C)C)NC(C1CCN(C(C)=O)C1)=O)NC(C(C)(C)OC)=O C(=O)(C(C)(C)c1cscn1)N(C(CNC(c1cnc(C(F)F)s1)=O)C1CC1)C C1(NC(c2c(C#C)c[nH]n2)=O)CC1C1CCN(C(=O)CCOCCCOC)CC1 Cn1nc(C(N2CCC(CCC(=O)N3CC(n4cccn4)C3)C2)=O)cc1O C(=O)(C#CC1(C)CCCO1)NCC(CC(=O)NCCn1c(C)cc(C)n1)C C1(c2nnnn2CC2CCOC2)(NCCC=CC=C)CC1CCCC c1(N2C(CNC(C(C)=C(C)C)=O)C(C)CC2)ccc2c(n1)CC(C)(C)CC2=O N1(C(CCCCOCC)=O)CCC(NC(=O)CCSCC(N)=O)C(F)C1 C1(NC(CSCCCC)=O)COCCN(C(=O)CCC2COC(C)(C)O2)C1 N1(C(CC(=O)OC)=O)CCC(NC(c2ccc(C)c(C3CC3)c2)=O)C(F)C1 c1(NC2(C)CC(NC(C3CC(F)(F)C3)=O)C2)nc(C2CC2)nc2[nH]ccc12 C=CCC(CC)C(=O)NC(C1(O)CN(C(c2ccc(C(F)(F)CF)cc2)=O)C1)C N1(C(C(CC)C)=O)CC(CNC(c2cn(CCC3CC3)nn2)=O)C(O)C1 C1(CNC(c2cc(C)ns2)=O)CC(C)(C)CN1C(c1nn(C)c(Cl)c1Cl)=O C1(C(=O)NCC(C(N)=O)O)CCC=CC1NC(=O)CCCn1ccnn1 CC1CN(C(=O)CC(c2ccc(F)cc2)C)CC1CCNC(=O)C(C)(C)CF Cn1cc(Br)c(CS(N2CC(C(=O)O)C(C(F)(F)F)C2)(=O)=O)n1 CC1CCCC(C(N2CCCC2CC(=O)NCCOc2cccnc2)=O)C1 CN1CCn2cc(C(N3CCOC(CNC(=O)CCP(C)(C)=O)C3)=O)nc2C1=O N1(CC)C(=O)CCC1CC(=O)NCCC1(NC(c2n[nH]cc2C(F)(F)F)=O)CC1 c1(-c2n(C)nc(CCC(C)(C)C)n2)cc2ccccc2n1C(F)F c1(N2CCC(CC)(CO)C2)nc(NCC(C2CC2)OC)c2ccsc2n1 N1(C(c2c(CCC)n[nH]c2)=O)CCOC(C(=O)Nc2ccccc2)CC1 Cn1cc(C(=O)NCC(CNC(C2(n3nccn3)CC2)=O)CO)n(C)c1=O C1(C(=O)N(C2CCN(CC(C)C)C2)C)(COC)CCCN1C(=O)C(Cl)=CCl C1(NC(C(C2CCN(C(c3c(OC)n[nH]c3)=O)C2)C)=O)CCc2ncnn2C1 n1(CC(=O)NC2(CN(C(C(CC)(C)O)=O)C)CC2)c(C(N)=O)nc2ccccc12 CCCS(=O)(=O)C(C)C(=O)NCCN(C(=O)C1=C(C)OCCS1)C(C)C c1(C(N2CC(C)(CNC(CSCC#C)=O)OCC2)=O)cn2c(Cl)cccc2n1 N1(C(C(C)(C)C)=O)CCC(NC(=O)C(F)(F)Oc2ccc(F)cc2)CC1C1CC1 C1(C(=O)NCC(C)(C)NC(C=C(CC)CC)=O)CCc2c(cnn2C)C1 Cc1cc(C(=O)NCC2(F)CCN(C(=O)CC3NC(=O)NC3=O)CC2)nc(C)n1 c1(C(=O)NCC(Cn2cc(C(CC)O)nn2)(C)C)cc2c(C)n[nH]c2cn1 C12(CNC(Cc3cc(C)no3)=O)CN(C(C3CCCCS3)=O)CC1CCO2 N1(C(Cc2ccc(OCC)cc2)=O)CC2(CCCCN2C(=O)C(C)CF)C1 N1(C(C(C)(C)F)=O)CC(CC(=O)NC2COCC2CO)C2(CC2)C1 Cc1cccc(SCC(=O)NCC2CCN(C(C3CCCCS3)=O)C2)c1 C(C(CC(C)C)C(=O)NCC1CCCN1C)NC(c1cncc(C)n1)=O C1(CNC(CCOC)=O)CCC2(CCC2)C1NC(c1cccc(O)c1C)=O CCCC(O)C(=O)N1CCC1C(=O)NCCC(F)(F)CO C=CCC(C)(CC)C(=O)NCC(CO)NC(=O)CSC C1(CNC(C(CC)OC)=O)CCN(C(C2C=CCS2)=O)C12CC2 C1(C(=O)NCC(CC(=O)OC)C)CCC2CCC1N2C(=O)C(F)(F)C1CC1 C1(C(N2CCC(C3CCCCN3C(=O)CCF)CC2)=O)CC2CCC2C1 Cc1c(C(N2CCCC(CC(=O)NOCC(F)F)C2)=O)cccc1Cl c1(N2CC3C(C(=O)Nc4cn(CCOC)nc4C)(C3)C2)ncc2[nH]ncc2n1 C(C(C)(O)CC(=O)N1CCC(CNC(=O)C(C)(C)c2ccccn2)C1(C)C)OC N1(C(CCNC(=O)CO)=O)CCCC12CCN(C(c1ccoc1Cl)=O)C2 C1(C(=O)NCC2CN(CC)C(=O)O2)CC2CCC(C1)N2C(=O)CC(C)(C)C CC(CC(=O)NCC(=O)NCc1nncn1C1CC1)c1ccco1 NC(=O)CC(N=c1[nH]c2c(c(=NCC34CCC(CC3)O4)[nH]1)SCC2)C1CCCC1 CC1C(NC(=O)C=CCN(C)C)CC2CCC1N2C(=O)C(N)=O CC(C)CC(CC(C)C)(c1nnnn1C1(C)CC1)NC(c1cccc(Cl)c1F)C c1(C(N2C(C(N)=O)CCC2C(=O)O)=O)cccc2[nH]ccc12 Cc1ccc2c(=NC(C)c3ccc(Br)cn3)[nH]c(=NCC(C)CO)[nH]c2c1 CC1CN(C)C(=O)CN1C(=O)CCC(C)NC(c1cncc(F)c1)=O N1(C(CCN(C(C2CC(C)(O)C2)=O)C2CC2)=O)CC2(COC(=O)C2)C1 C=CC(C)CC(=O)NC1CCC(N2CCN(C(C3COC3)=O)CC2)CC1 c1(-c2c(OC)cccc2)nc(=NCC2CCCN2C(c2cscc2C)=O)s[nH]1 C1(C(N(C(C)C2CC2)CC)=O)CC(NC(=O)C(C)NC(C2CCC2)=O)C1 c1(OC)cccc(C(=O)NCCN(C(C2CC(Cl)(Cl)C2)=O)C(C)C)c1C C1(CC)(NC(=O)CC(F)(F)F)CCCN(C(=O)Nc2ccccc2C(C)(C)C)C1 C(CC)(CCC(=O)N(CC(O)CF)C)NC(c1[nH]cc(C(C)=O)c1)=O C1(C(N2CC(O)(CCNC(=O)C(CC3CCC3)OC)C2)=O)(SC)CC(=O)C1 N1(C(C2(C)CCNC2=O)=O)CC2(C1)CN(C(=O)C=Cc1cn[nH]c1)CCO2 c1(C(N2CCN(C(C3CCCCC3)=O)C3CC23)=O)ccc2c(O)nnc(O)c2c1 c1(C(=O)NCCC(CCC)C)ccnc2c1nnn2C CC(C)CC(O)CC(=O)NCc1ccc(C(=O)NC2CC3C=CC2C3)c(F)c1 C1(C(N2C(CC(=O)N(CCn3c(C)ncc3)C)CCC2)=O)CC2C=CC1C2 C1(NC(c2cc(SCC)ncc2)=O)CC2(CCCN(C(c3occc3Br)=O)C2)C1 Cc1cc(C(=O)NC(CNC(C2CCCC2O)=O)C(C)(C)C)nn1CCO CC1CCN(C(c2c(Cl)nsc2Cl)=O)CC1NC(c1occ2c1CCC2)=O n1(CCC(=O)NC2CN(C(C=CCC)=O)CC2(C)C)c(C)nc2ccccc12 c1(C(N(C2CC(=O)N(CCNC(c3ccccc3)=O)C2)C)=O)ccc(C(=O)O)nc1 CC(C)(Cc1ccc(Br)cc1)C(=O)NC1CC1NC(C1CC(C)(C)CO1)=O C1(C2CN(C(=O)CCCC3CCCO3)C2)(NC(Cc2c(C)cc(C)s2)=O)CC1 N1(C(c2c(CC)noc2)=O)CC(NC(=O)C(CC(N)=O)NC(C)=O)C(C)(C)C1 c1(C(=O)NC(CNC(Cc2cc(C)sc2)=O)C(C)(C)C)cnc2ncnn2c1C C12(NC(CC3(NC(C)=O)CC3)=O)CC(C1)N(C(c1scc(C)c1C)=O)C2 c1(C(N2CC3CC(C2)N(C(=O)CSCC(F)F)C3)=O)ccc2cncn2c1 C1(C(=O)NCCCC(C)NC(=O)CO)CC2(CCC2)C1 C(=O)(CC(C)C(=O)NCC(C)(F)CNC(C1CN(C)CCO1)=O)OC C1(COC(C2CC(C(=O)OC)C2)=O)CCCOC1.C1CC(=O)NC(=O)N1 N1(C(CC=CC)=O)CCCC1C1CCCN1C(=O)COc1cccc(Cl)c1C C1(OC)CN2CCCC2(C(=O)NC(c2cc(Cl)ccc2C)C)C1 C(c1ccc(Cl)cc1)=CC(N1CCC(CCNC(C2(Cl)C(C)(C)C2)=O)C1)=O c1(C(N(CCCCN(C)C(C2C3CCC(=O)C23)=O)C)=O)n[nH]cc1[N+](=O)[O-] C#CC1(C(N2CC3CC3(CO)C2)=O)CCN(C(c2cc(OC(C)=O)ccn2)=O)C1 C1(C(N2CC(COC)OCC2)=O)CC2CCC1N(C(=O)CCCN=[N+]=[N-])C2 C1(CCNC(=O)Cn2nccn2)CCCCN1C(c1ncncc1Cl)=O C(CCCCC(=O)N1C2CCC(C2)C1C(N1CCC(n2ccnc2)C1)=O)N(C)C C(CNC(C1CCCCO1)=O)(CC(=O)N1CC(F)(CO)C1)OC c1(C(=O)NC(CC)CN(C)C(C2CCCN(C)C2)=O)cc2cc(OC)ccc2o1 c1(C(=O)NC(CNC(C2(CCOC)CCC2)=O)(C)CC)ccc(F)cc1[N+](=O)[O-] C1(NC(=O)C=Cc2ncc[nH]2)C=CCN(C(C2CCC(=O)N2)=O)C1 c1(C(COC(C2C(C)(C(C)C)C2)=O)=O)ccc2ccccc2c1 c1(C(=O)NCCN(CCC)C(C2(F)CCOC2C)=O)cc(C)nn1C(C)(C)C c1(CCNC(C2(C)CSC2)=O)ccc(CNC(=O)CC2CCC(=O)N2)cc1 C1(C(=O)NC2CC3(C(NC(C4(C)COC4)=O)C3)C2)CC(F)(F)CCC1(C)C c1(C(N2CC(C)N(C(=O)Cn3ncnn3)CCC2)=O)cnc2sccn2c1=O CC(C)=C=CC(=O)N(CCNC(C1CCC(C)(C)C1)=O)CCOCCO C(=O)(CCN=c1ccc(C)c[nH]1)NC1C(NC(c2nn(CC)nc2C)=O)COC1 C1(C(=O)NCCN(C)C(C2CC3(CCC3)CO2)=O)CC(C)(C)CCO1 C1(CC(=O)NCC(CCNC(=O)CSc2ccncc2)O)CC2(CCC2)CO1 C=CCC(C(=O)N1CCC(CC)C1C(N1CCC1(CC)CC)=O)NC(C)=O C(=O)(CC(O)CC1CC1)N1CCC(OCC)C1 N1(C(CN(CC)CC)=O)CCC(NC(c2c(SC)cccc2F)=O)C1(C)C c1(C(N(CC(CNC(C(C)(CO)OC)=O)C)C)=O)cnc2cc(Br)ccn12 C(C(C)(O)CC(=O)NC1(C)CC(NC(=O)Cc2ccc(SC3CC3)cc2)C1)OC c1(-c2cn(CCN(C(C34COCC3C4(F)F)=O)CC)nn2)ccccc1[N+](=O)[O-] CC1(C)CCCC(C(C)(O)CNC(C2CC3CCC(C2)S3)=O)C1 c1(C(=O)NC2C(CNC(C(C=C)(C)CC)=O)CC2)c[nH]c2c(Br)cccc12 c1(OC)c(Br)cc(C(N2CCC(C)(c3ccccc3Br)C2)=O)cc1Br C1(C(N(CCCCCO)C)=O)CC12CN(C(C1CC(O)CN1)=O)C2 CC1C(C)N(C(=O)OC(=O)Cc2ccco2)CCN1C(=O)CN(C1CCC1)C C1(C)(CNC(CCOC)=O)CCN(C(=O)C(C)Cc2ccc(N)cc2)C1 c1(C(N2CCC(N(C)C(c3coc(O)n3)=O)C2)=O)cccc(C2CC2(F)F)c1 C1(CCOC)(NC(C2CCC3(CC3)C2)=O)CCN(C(=O)CCOCC2CC2)C1 C1(OC)CC(NC(c2cscn2)=O)CN(C(=O)C(C)(O)c2ccccc2)C1 c1(OC)cccc(-n2cc(CC3CCCN3CC3CC3)nn2)n1 C1(CC)CC(C(=O)NCC2C=CCN2C(=O)CCc2csc(C)n2)CC(=O)N1 C1(NC(C(C)CN2CCCCC2)=O)CCN(CCF)C12CCC2 Cc1ncc(C(=O)NC(C2CCCN(C(C3(S(C)(=O)=O)CC3)=O)C2)C)cc1N CC1(C)CCC=C(C(=O)NC2CCCC2Cn2cc(C3CCCCC3)nn2)C1 C12(CNC(C=Cc3nc(C)c(C)[nH]3)=O)CCCC(CN1C(=O)CC(C)C(C)C)C2 C1(CN(C2C(C)(C)CO2)CCO)CCN(C(=O)C(c2ccccc2F)O)CC1 C1(C(=O)NCC(C2CCN(C(CC3(C=C)CC3)=O)CC2)C)CN2CCC1CC2 C(CC(C(=O)NC(c1ccco1)C)NC(c1cc(Br)cs1)=O)SC N1(C(CCC#CC)=O)CC2(CC(CNC(c3ccc(OC(C)CC)cc3)=O)C2)C1 C1(c2n(CC)nnn2)(Nc2cc(COC)cc(C#N)c2)CCC2C3C=CC(C3)C12 C1(C(=O)OCc2cccc(OCC(=O)OCC=C)c2)CC2(CCO1)CC(F)(F)C2 C(CC1=CCOCC1)NC(C(CCC)NC(=O)CCOC(C)C)=O C(CC(C)(Cc1ccccc1)NC(C12CC3CC1C2C3)=O)NC(CC(=C)C)=O C(CCCCCNC(C1C2CCCC12)=O)N(C)C(C1CC(=O)N(C)C1)=O c1(CNC2C(C(=O)NCCc3ccccc3O)C2)cc2ccccc2cc1O C1(CCC(=O)N(C2(CCO)CC2)C)CCCCN(C(=O)CCCF)C1 C12(C(=O)NC3(CNC(C4CSC4)=O)CCCCC3)CCCC1CC(F)(F)CC2 C#Cc1cc(C(N2CCC(NC(=O)COCCCF)C(C)C2)=O)cc(Br)c1 Cc1cc2c(cc1Br)N(Cc1cc(C(=O)O)c(O)c(I)c1)CCO2 c1(C(=O)NC(C(C)NC(=O)CC(F)(F)Cl)C)cc(C(F)(F)F)cc(N)c1 c1(C(N(C2CN(C(c3ccc(Cl)[nH]3)=O)C2)C)=O)ccn2cccc2c1 CC1CC2(CC(C(=O)NCCCCC(=O)N3CCOCC3)C2)C1 C(=O)(CCC(C)(F)F)N1C2(C(=O)NCCOCC=C)CC2CC1 CC(C)CCC(O)C(=O)N1CCCC(CCC(=O)NCCN=S(C)(C)=O)C1 c1(N2CCC(CN(c3cncc(F)c3C)CC)CC2)ncc(C(F)(F)F)cc1Cl N1(C(CC)=O)CCC(CNC(=O)CCNC(c2ccccc2OC)=O)(OC)C1 CC1(C)CN(Cc2cc(C(=O)O)cs2)C(C)(C)C1O N1(C(C2C(C)(C)CC2)=O)CCn2c(CNC(C3(C)C=CCCC3)=O)nnc2C1 c1(OC)ccc(CN2CCC(O)(C(=O)NCc3cnn(C)c3)C2)c2ccccc12 c1(N(CCCS(C)=O)C)cc(S(=O)(=O)N2CCCCC2CCCO)ccc1C#N C1(C(=O)NC2CC(CNC(CN(CCC#C)C)=O)C2)CN2CCN1C(C)C2 N1(C(c2nn(CC)c(C)c2)=O)CCC12CN(C(c1cc(C(F)(F)F)n[nH]1)=O)C2 C1(COC)CN(C(c2cc(-c3ccn(C)n3)on2)=O)CCN1C(=O)CP(C)(C)=O c1(OCC)oc(C)nc1C(N1CC(CNC(=O)C=CC2(C)COC2)C(O)C1)=O C1(NC(C(C2(O)CCC2)NC(C=C(CC)CC)=O)=O)CN(C)C2(CCC2)C1 c1(CC(CNC(=O)NCCC2CC3C=CC2C3)CO)ccccc1F c1(C(N2CC(C(C)NC(C(C#C)(C)C)=O)OCC2)=O)cc(F)c(Br)cc1N C#CCCC(C(=O)N(C(C)C(=O)OC)C)NC(C1CN(C)C(=O)N1)=O c1(C(N2C(CCCC)CN(C(=O)C(C)O)CC2)=O)ccc(Cl)c(Cl)c1OC c1(OCC)cccc(NC(=O)C(C)N(C(c2cc(C)sc2N)=O)CC)c1 c1(CC)cscc1C(=O)NC1(CNC(c2cnsc2C)=O)CCOC1 CC(C)CCC(F)C(=O)N1CC(NC(C2CCNC(=O)C2)=O)CC(C)C1 C(C)(CNC(=O)CSc1nncn1C(C)(C)C)(C(C)C)NC(C(CC)F)=O C(CC(=O)NCCC(C(C)C)NC(C1CCC1)=O)(C(N)=O)NC(C)=O c1(OC)cccc(NC(N2CCN(c3cncc(OC)n3)CC2)=O)c1C#N O=C1CC(CNC2CCC(CCO)C2)CN1CCO O=C(NOC1CCCC1)C1(F)CCCC2(C1)OCCO2 C=CC1(CC(=O)NC2CC(NC(=O)C(C)c3ccco3)C2)CCOCC1 Cc1ccccc1C(=O)NC1CCC(CC(=O)NOCCOCCF)C1 Cc1ccc(C(N2CC(C(C)NC(C3C=CC=CC=C3)=O)C2)=O)cn1 C1(C(N2CCC(N(C(=O)Cc3csc(NC=O)n3)C)C2)=O)CC2CC1CO2 C(c1ccccc1OC)=CC(N1C(CNC(c2ccc(OC)s2)=O)CCC1)=O Cc1c(O)c(=O)ccn1CC(=O)NC1CCN(C(=O)CN2CCCCS2(=O)=O)C1 C1(N(C(=O)C(C)CC(N)=O)C(=O)OC(C)(C)C)CC2C(C1)C2(F)F c1(C(=O)OC)ccn2c1CN(S(=O)(=O)N1CCC1C(=O)OC)CC2 c1(NC2CCN(C(Cn3ccc(C)n3)=O)C(C)C2)ncnc2c1nnn2C(C)C c1(CNC(c2scc(CNC(=O)CC3CC(=O)NC3=O)c2)=O)cccc(C#N)n1 CCCCCC(C)(C)C(=O)NC(C)CNC(=O)CCc1cccnc1F Cc1ccnc(Cl)c1NC(N1CC2CC(NCC(c3ccccc3Br)F)C1C2)=O C1(NC(C)=O)CCN(C(=O)CC2CCC2C)CC1.C1(=O)CN1C c1(C(N(C)CC2CCCN2C(=O)CCF)=O)cc2cccc(Br)c2[nH]1 CCC(CC(=O)N1CC(NC(c2nnsc2C(F)F)=O)C(C)C1)c1ccccc1 N1(C(C2C(C)=C2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)C2(CCC2)C1 Cc1ccc(NCCC(N2CC(NC(c3cnncc3O)=O)CC2C)=O)cc1 c1(N2CCC(NC(C(CCC)N(C)C)=O)C(F)C2)ncc([N+](=O)[O-])cc1C N1(C(c2cc(CNC(C=CCCC)=O)sn2)=O)CC(C2CC2)C1C1CC1 C(C(N)=O)(C(F)(F)F)NC(C1N(C(c2c(C)cnnc2)=O)C(C)C1)=O c1(OCCOCC(=O)N(CC(CC)NC(=O)CC2C=CCC2)C)cccc(C)c1 C1(NC(C2C3CCC2(c2ccco2)C3)=O)CCCCN(C(C2C3CCCC23)=O)C1 C1(NC(CC23CC(C)(OC2)C3)=O)CCC2CCN(C(C3CC3(F)F)=O)C1C2 S(=O)(=O)(c1ccc(C)cc1C)NC(CC)C(=O)NC1CCCCC12CCNCC2 c1(CCC(=O)NCC2C3CC2N(C(=O)C=Cc2ccoc2)C3)ccc(F)cc1F N1(C(c2cnc(N3CCOCC3)nc2)C(=O)NC)CC(CCN)CC1(C)C c1(NC(CNC(CCNC)C)=O)cc(Br)c2c(c1)OCCO2 c1(OCCOC)ccccc1NC(N1CCC(c2ccn(C)n2)CC1)=O C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(CCC(=C)Cl)=O)(CC)CC1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCO3)=O)C2)ccccc1O N1(C(c2ccc(C(C)=O)nn2)=O)CCC(NC(c2cnc(C)nc2)=O)C(F)C1 C1(OCC(=O)NC2(CC#C)CC2)CC(NC(C2CC2(C)CC)=O)C1 c1(N2CCCC(CCC)CC2)nc2c(c(=NC(C)C3CC3)[nH]1)SCC2 C1(CNC(C(C(C)C)N(C)C)=O)CC2CN(C(c3cc(O)cc(Cl)c3)=O)CC12 c1(C(=O)NC(CNC(c2cccc(SCC)c2)=O)C)ccc(C(F)(F)F)cc1N c1(CNC(C2C(C=C)OCC2)=O)ccc2c(c1)CCOC2.C12CCCCN1C2=O c1(C(N2C(CCNC(C(C)C3(O)CCC3)=O)CCC2)=O)coc2c1CS(=O)(=O)C2 n1(C(C)C)cc(Br)c(=NC(=O)c2cnn(C)c2)[nH]1 N1(C(C(C)n2cccn2)=O)CCCC(CC(=O)Nc2ccccc2Br)C1 C1(NC(c2cc(OCC)n[nH]2)=O)CC2CCC1N2C(=O)CC1CCCC1(F)F N1(C(C(CC)N2CCCC2=O)=O)CC2(CCC(NC(=O)C=CC(F)(F)F)CC2)C1 C(C)(CCCCCO)NC(C1(C2N(C(c3nc(C)oc3C)=O)CCC2)CC1)=O C(CN=c1[nH]c(=N)[nH]c(=NCCCC2(C)CC2)[nH]1)c1nc(C)nc(O)c1 C1(OC)CC(C(N2CCSCC2)=O)N(C(c2cc(-c3ccnn3C)cs2)=O)C1 c1(C(N)=O)cccc(C(=O)NC2CC(NC(C3OC4CCC3C4)=O)C2)c1F c1(C(=O)NC2C(CNC(CC=C)=O)C2)nn(C(C)C)nc1Br CCC(C#N)(CC)C(=O)N1CCCCC(CNC(=O)Cn2nc(C)n(C)c2=O)C1 c1(SC)cccc(F)c1C(N1CC(NC(C2CCCCN2C)=O)C(O)C1)=O N1(C(Cc2ccn(CC)n2)=O)C2CCCC1CN(C(c1cc(C)cc(F)c1)=O)C2 Clc1nsc(NCCn2ccc(Br)n2)n1 N1(CC(CN(c2ccc(OCC(C)N)cc2)C)O)CCN(C)CC1.C(=O)O c1(NC2C(C)CCC2)cc(C(F)(F)F)nc2c(Br)cccc12 C1(NC(C2(C)CC=CC2)=O)CCCCN(C(=O)CN2CCCC2=O)CC1 C(=O)(CCC(=O)N(C)C)NC(C1CCCN(C(=O)C(C2CC(F)(F)C2)O)C1)C CCC(CNC(C1CCN(C)C1)=O)(CC)NC(c1ccc(C(N)=O)nc1)=O N1(C(CN(C(=O)C(C2CCOCC2)F)C)=O)CCC(C2CC2)(NC(N)=O)C1 c1(C(=O)NC(C)CNC(=O)Cc2nc(C(F)(F)F)n[nH]2)cnn(C)c1N CCC(CC)C(C(=O)N1CC2CC2(NC(=O)C(C)c2cc[nH]n2)C1)OC C=CC1CCCCN1C(c1c(Cl)ncn1C)C(=O)NCC(C)C C1(CNC(c2cc(CC(C)C)[nH]n2)=O)(NC(=O)CC(C)(F)F)CC(F)(F)C1 c1(CSCC(=O)Nc2ncc(-c3ccccc3F)o2)ccccc1Br CCS(=O)(=O)CCn1c(N(C2CCCC2)Cc2nccs2)nnc1CC(C)C C(CCCCN(C(=O)C(C1CCCC1)C1CCCC1)C)NC(CN(C)CC)=O Cc1cc(C(=O)NCC2N(C(=O)CS(N)(=O)=O)CCCC2(C)C)c(N)c(Cl)n1 c1(OC)cc(C(=O)NC2CC(C)N(C(C3CCC(C)CC3)=O)C2)cc(N)c1N C1(NC(C2CC(OC)C2)=O)CCN(C(=O)CCSC2CCCC2)C(C)C1 C#Cc1ccc(C(N2CC(CNC(=O)C(F)(F)C(F)(F)F)OC(C)C2)=O)cc1C C12(NC(CC)=O)CC(C)(C1)OC21CN(C(c2ccc3nc(=N)[nH]n3c2)=O)C1 n1(CC(=O)NC2C(C)(C)CN(C(=O)C3=COCCC3)C2)ncn2cccc2c1=O O=C1CCc2cccc(C(=O)NC34CC(C3)N(C(=O)CNS(N)(=O)=O)C4)c2N1 C1(NC(C2ON=C(C)C2)=O)CCN(C(c2ccccc2C)=O)CC1 CN1CCN(C(=O)CCc2cncnc2)CC1NC(=O)COCC(C)(C)C c1(C(=O)NC2COCC2CNC(C2CC23CCCC3)=O)sc2ncccc2c1Cl N1(C(CC(CC)C)=O)CCC2(CC1)CN(C(C1CCN(c3nncs3)CC1)=O)C2 C1(c2ccc(C(c3ccccc3)=O)c(F)c2)CN(N2CC3CCCCCC3C2)C1 CC(C)C(O)C(=O)NC(C1CCCCN1S(C)(=O)=O)=O.C1CN(C2CC2)N1.NC c1(C(N(C(CN(C(c2c(CC)nco2)=O)C)C)C)=O)cc2nc(C)[nH]c2cc1F N1(C(C(=O)N(C2CCCNC2)CC(C)C)=O)CCC(CCCF)CC1 c1(C(c2n(C(CC)Nc3cccnc3)nnn2)(C)C)cc(Br)cc(C)c1F C1(COC)CCN(C(=NCCc2ccc(F)cc2)NCC(c2nc(C)cs2)C)C1 C(=O)(C(CN=[N+]=[N-])NC(=O)C(C(=O)OC)OC)Nc1cnc(CC)nc1 c1(C(=O)NC2CCCN(C(=O)Cn3nccn3)C2C)cnc(OC)c(N)c1.COCBr c1(OC)ccc(CC(=O)N(CC(CO)(CO)NC(=O)C(C)CSC)C)c(C)c1 N1(C(c2cnn(C)c2C#N)=O)CC2CC(NC(C3CC34CCOC4)=O)CC1C2 C1(OCC)CC2CN(Cc3cc(C(=O)O)ccc3OCC)CC12 C(CCC(=O)O)(C(N)=O)NCC1CCN(C(=O)OC(C)(C)C)C12CC2 n1(CC)cc2ccc(NC(=O)NC3(C4CCC4)CCCC3)cc2n1 N1(C(C2CC(NC(COCC(=O)NCC)=O)C2)=O)CC(O)(c2ccccc2)C1 O=S(=O)(c1ccc(Br)s1)N1CCCC(Oc2ccccc2OC(F)(F)F)C1 c1(C(=O)NC(CC)CNC(c2cnccc2C)=O)ccc2c(C)cc(Cl)nc2c1 C1(C(=O)NC2(C(N(CC)CC)=O)CC2)COC(=O)C1 c1(CC(=O)NCC(CN(C)C(C2CC2c2ccco2)=O)O)nc2c([nH]1)CCCC2 C1(C(N2CC(O)(CC=C)C2)=O)CNC(=O)CN1C(=O)CSCC(N)=O C1(CC(=O)N(CC(CC)NC(c2cnc(C(N)=O)cn2)=O)C)CCCCC(=O)N1 n1(CC)ncc(C(=O)N(CCCn2cc(COCCN(C)C)nn2)C)n1 c1(C(=O)OC)cnc(C(=O)N(C(C2CC2NC(=O)C2CC2)C)C)o1 c1(C(C2CCC2)NC(c2n(CC)nnn2)c2coc(C)n2)ccc(F)cc1 Cc1ccc(Cl)c(NC(N2CCCN(CC(=O)Nc3ccccc3)CC2)=O)c1 CCC(C)(C)C(O)C(=O)NC(c1ccccc1)CNC(c1cccc(OC)n1)=O C(=O)(NNC(=O)C(C)(C)CCCCNC(c1cnc(CC)[nH]1)=O)C1CSC(C)=N1 Cc1ncnc(C(N2CCN(C(c3cc(C4CC4)[nH]n3)=O)C(C(F)F)C2)=O)c1C c1(NC(C2CN(C(C3(F)CCC3)=O)CCO2)=O)ccc(I)c(Br)c1 C(=O)(C1Cc2ccccc21)NCCCCCNC(C(CNC(C)=O)(C)C)=O C(C1=CCN(C(c2ccc(C(F)F)cc2)=O)CC1)NC(C1CC12CC(O)C2)=O Cc1ccc(F)c2[nH]c(C(=O)NCCN(C(c3ccnc(S)c3)=O)C3CC3)cc12 c1(C(=O)NCCn2cc(C(N3CC=CC3)=O)nn2)ccc(O)cc1 C=CC(C)C(=O)NC1CC(CNC(=O)CN(C)CCOC)C1 c1(C(N2CCCC(NC(C(CC)(C)OC)=O)CC2)=O)cc(C)c(C)c(F)c1 C12(NC(C3CC(N(C)C)C3)=O)CCCC1CN(C(=O)CC1CCCCC(=O)N1)C2 c1(NC2CN(C)C2)[nH]c(=NCc2c(Br)cccc2Br)nc2scnc12 C#CCCN=C(NCC(C1CC1)Sc1ccc(Br)cc1)N1CCC(NC(C)=O)C1 N1(C(C2(NC(=O)CC(=O)N(C)C)C(C)CCC2)=O)CC2CCC(C1)C(=O)O2 c1(CC)cccc(C(=O)NC(C2CCN(C(c3[nH]ccc3C)=O)C2)C)c1 C1(C(N2CC(OCC(=O)NCc3n(CCC)ccn3)C2)=O)CC2(CC(=O)C2)C1 c1(CC(=O)NCCCNC(c2cc3cc[nH]c3cn2)=O)ccc2c(c1)CCOC2 N(C)(C(=NCc1ccccc1)NC1CCC(c2cc(F)cc(Cl)c2)C1)CC.CC=O c1(N2CCC(CCNC(C(CC)N(C)C)=O)C2)ncnc2cc(Br)ccc12 Cc1cc(=N)[nH]cc1C(=O)NCC(C)(C1CCC1)NC(c1cccs1)=O c1(C(=O)NC2CC3(C(NC(C(CC(C)(C)C)O)=O)C3)C2)cc2ccoc2cc1F N1(C(C2(C(C)NC(=O)CCCF)CC2)=O)CC(=O)NC2(CC2)C1 CCC(CO)CCNCc1cc(C(F)F)nn1C C1(C(N2C3CC(=C)C(C3)C2)=O)C(C2CC2)CCN1C(=O)CCC=C(C)C Cc1cc(S(N)(=O)=O)ccc1CNC(=O)NCCc1cnnn1C c1(C(N2CCC(NC(c3nnn(CC)c3C)=O)C2)=O)cncc2ccc(F)cc12 Cc1cc(Br)cc(C(N2CC(NC(C3OCCN(C)C3=O)=O)C2)=O)c1F C1(CNC(C(CC)O)=O)C(CC)CCN1C(=O)C=NOC C1(C(N(C2CCN(C(c3cc(C)c(C)nn3)=O)C2)CC)=O)CCC(F)(F)CC1 c1(C(N2CC(CC(C(=O)N3CC(C=C)C3)F)C2)=O)ccc(C)nc1C C(CN=C(NCC1(F)CCCCC1)NC1CC1)=C(C)C1CC1 N1(C(CC(CN(C)C)O)=O)CCc2[nH]nc(CNC(C3(C)CC=CCO3)=O)c2C1 CC(C)CCCCC(=O)N1CCCC(CNC(=O)C(C)CCn2cccn2)CC1 CCC(O)C(C)C(=O)NCC1C2CC1N(C(c1cc(F)ccc1C(F)(F)F)=O)C2 C1(N=[N+]=[N-])(C(=O)NCc2nc(C)c(C)o2)CCN(C(C2CN3CCC2C3)=O)C1 C12(NC(C3CC4(C3)CC(F)C4)=O)CCCC1N(C(c1ccc(O)cc1)=O)CC2 c1(C(CNC(=O)CC2CCNC2=O)NC(=O)CCCC2CC2)ccc(Br)cc1 Cc1cncc(CC(=O)NC(C)(CNC(C2CC2(C)C)=O)CO)c1 N1(CCC(C(C)C)N)CCC(O)(C2CCC2)CC1 C1(C2CC2)(NC(Cc2n(C)ccn2)=O)CCN(C(=O)COc2cccnc2)C1 N1(C(C(COC)O)=O)CC2CC(NC(c3occ4c3CCC4)=O)C(C2)C1 C12(NC(=O)CCn3cnccc3=O)CCCC1N(C(C1CSC1)=O)CC2 c1(C(=O)NC2(C)CC(NC(CSCC(C)C)=O)C2)ccc(F)c(C(F)(F)F)n1 CC(C)C(O)CC(=O)NC1CN(C(=O)C(O)C(C)C)CC1O N1(C(CCC=C(C)C)=O)CCCCC2(C1)CN(C(c1cncn1C)=O)C2 c1(C(=O)NC(COC)C(=O)NCc2ncco2)ccnc2cc[nH]c12 C=C(C)CC(C)C(=O)NCC(C)(CO)NC(=O)CC1(O)CCOCC1 c1(C(=O)NCCCN(CCO)C(C2C3CCCOC23)=O)cn2ccnc2cn1 C1(N(CC(=O)NCC(C2CC=CCC2)NC(CSC)=O)C)CCCC1O c1(CN2CC(c3n(C)ccn3)C3(C2)COC3)cc(CN)cc2c1CCC2(C)C N=c1cc(C(N2CCC(NC(=O)C(Cl)=CCl)C23CC3)=O)c(Br)c[nH]1 C(=O)(C(C)(C)CC(F)F)N(CC(CNC(CC1CCC(C)C1)=O)C)C CC1CC(N=c2ccc3c([nH]2)CCCC3=O)c2ncnn21.C12(CCC1)C(=O)N2 C1(C(N)=O)CCC(NC(C2CCCCC2c2ccccc2)=O)CC1 Cc1[nH]c2ccccc2c1CC(=O)NC1COCCN(C(=O)CCS(N)(=O)=O)C1 C1(NC(C2(CCNC(=O)CCn3cccc3)CC2)=O)CC(C2CCCC2)C1 C1(NC(Cc2c(C)ncs2)=O)CCC(S(C)=O)C1 c1(C(N2CCCC(N(C(c3ocnc3C)=O)CC)C2)=O)ccc(N)c(N)c1 N1(C(C(C)n2ccnc2)=O)CCC2C1CCCN2C(c1cc(Cl)cc(F)c1Cl)=O c1(C(=O)NC2C3(CC(NC(COCC=C)=O)C3)C2)ccc(N)cc1C Cn1ccc(=O)c(CC(=O)NCc2nc(C3CCC3)no2)c1 CCCC(C)(CCC)C(=O)N1CC2CCC2(CNC(c2cnccc2OC)=O)C1 C1(C(=O)NCc2cncc(CC)c2)CN(C(c2cc(F)n(C)n2)=O)CC12CCC2 CC1CN(C(c2c(F)cccc2Cl)=O)CCCN1C(C1CCCC1(F)F)=O CCCCCC(C)(C)C(=O)N1CCC(N(C(=O)CCCN(C)C)C)C1 c1(-c2cc(C)[nH]n2)ccc2ncc(C(N3CCC(CF)CC3)=O)c(Cl)c2c1 C1(CNC(c2nc(C(C)=O)sc2)=O)CC(C)(C)CCC1NC(c1ccc(C)s1)=O C12(C(N(CC(N3CCCC(CC=C)C3)=O)CCC)=O)CCC(CC1)CC2 C(C(=O)NOC(CC(C)C)C(=O)NCC(c1ccccc1)O)(C(C)C)SC N1(C(C(CCC)NC(=O)CC2CC2C2CC2)=O)CC(C)OCC1C N=c1[nH]cncc1C(N1CC(C)(OCC(N2CCOC(C(N)=O)C2)=O)C1)=O C12(CNC(c3c(C(N)=O)csc3)=O)CCC1CCN2C(c1ccsc1)=O C(=O)(C(C)(CC)C(=O)NCC1(O)CN(C(=O)COc2ncc(F)cn2)C1)OCC c1(CC(CCOC)NC(CC)CC2CCOCC2)ccc(F)cc1F CC1(C)CCCCC1C(N1CCC(=CC(N2CC3CC2CO3)=O)CC1)=O c1(CCC(=O)N(C(C)CCNC(C2COC2)=O)C)ccccc1Cl n1(CC)nc(C(=O)N(C)CCNC(=O)C=Cc2nccs2)cc1C C1(CNC(C2(COC)CC2)=O)CCC2(CN(C(c3nnc(O)nc3O)=O)C2)O1 c1(C(N2Cc3c(C(=O)OCC)ncn3CC2)=O)cc(F)cc2cc[nH]c12 N1(C(c2ccc(CN(C)C)o2)=O)CCN(C(C2(C)CCCCC2)=O)CC(C)(C)C1 C(=O)(CCCCCS(N)(=O)=O)NCC(CN(C(=O)CCn1cnnn1)C)O Cc1cccc2c1OC(C(=O)NCCCN(C)C(C1C(C)(C)OC1(C)C)=O)C2 c1(CC)ccccc1OCC(N1CC(NC(=O)CC2CCC(=O)N2C)C(C)C1)=O Cc1nc(O)ccc1C(=O)N1CCC(C(=O)NC2CC3(CCCC3)C2)O1 c1(CC(=O)NC2(CO)CCN(C(c3cc(OC)ns3)=O)C2)cccc(Cl)c1F CC1CC(C(=O)NCC2CN(C(c3snc(Cl)c3Cl)=O)C2)Cc2nn[nH]c21 N1(C(COCCC=C)=O)CCC(C)(CNC(=O)C(c2ccc(C)o2)C)CC1 N1(C(CC(=C=C)C)=O)CC(NC(=O)C=Cc2nccs2)CC2(CC2)C1 Cc1c(Cl)ccnc1C(=O)NCC1(CNC(=O)CC2CCN(C)C2)CCCC1 C(=O)(CCC[N+](=O)[O-])N(CC(CNC(C(c1ccncc1)C)=O)C)C C1(CO)CCCCCC1OCCn1cc(C2(COCCO)CCC2)nn1 C1(N=c2[nH]c(=NCC3CCCO3)c3c(F)cccc3[nH]2)(CCOC)CCC1 N1(C(c2cncc(C)c2Cl)=O)CCC2CN(C(=O)CC3CCCC34CC4)C2C1 C1(S(N)(=O)=O)(C(=O)NC2C(CNC(c3n(CCC)ncc3)=O)CCCC2)CCC1 CN1CCN(C(C2CC3CCC3C2)=O)C(C(N2CC(C3CCCO3)C2)=O)C1 c1(C(=O)NCC2CCCN2C(=O)CCc2cccc(CO)c2)ccc([N+](=O)[O-])o1 C12(SCCNC(CC(CCC)O)=O)CC3CCC(C1C2)N3C(=O)OC(C)(C)C N1(C(C(CCC)N(C)C)=O)CCC(NC(=O)CC(C)(C)O)CC(C)(C)C1 c1(OC(C)C)cncc(=NC(=O)C(=O)NC2CCC(=O)N(C)C2)[nH]1 C1(C(N2C(C)(COC)CC2)=O)CCCCCC1NC(c1sccc1C)=O c1(C(N2C(C)C(C)N(C(c3cscn3)=O)CC2)=O)cnn2c1OCC(C)(C)C2 S(=O)(=O)(c1ccc(NCCOC2CC2)nc1)NC1CC(C)SCC1 C1(C(C)NC(=O)CC2CC(C(F)F)C2)CN(C(c2nccnc2N)=O)CCO1 C(=O)(C(C)C(O)CC(C)C)NCC1CCCN(CC(=O)OCC)C1 C(CC(CNC(c1cnoc1-c1ccoc1)=O)NC(C12CC(F)(C1)C2)=O)OC C1(CC)CCN(C(C2CNC(=O)N2)=O)C1C(=O)NC(C(C)C)c1ncc[nH]1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nccn2)cncc(P(C)(C)=O)c1 C=C1CC2CC1CN2C(c1ccc(C(F)F)o1)C(=O)NCCCF C(C)(C)(C(C)NC(=O)Cc1ccc(Cl)s1)NC(CCC1C(C)C1)=O Cc1cccc2sc(NC(C3CCN3Cc3ccc(O)c([N+](=O)[O-])c3)=O)nc12 c1(CC(=O)NC(CN(C)C(C2CCCC(C)(C)C2)=O)(C)C)cc(F)c(F)cc1F Cc1c(C(=O)N(C(C)(C)CC(=O)NCCC2CCC(C)O2)C)cncc1F N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(C2CCCCC2)=O)C(C)C1 Cc1nn(C)c2c(NCC3C4CCCC34)nc(=NCc3cscn3)[nH]c12 N1(C(C(c2ccc(C)cn2)(F)F)=O)CC2CCCC(C1)N2C(=O)CC1CC1C n1(CC(=O)NCCC2CC(NC(c3c(C)noc3)=O)C2)ccc(=O)c([N+](=O)[O-])c1 Cc1cc(C(F)(F)F)c(C#N)c(=NCCSCCc2ncnc3ccccc23)[nH]1 C(=O)(CC(CC)c1ccccc1)N1CCC(N(C(=O)Cc2cnoc2)CCC)C1 c1(C(C)C)ncncc1C(N1CC(CNC(=O)CC2(O)CCOC2)CC1C)=O C1(CC(C)NC(C2(C(=O)C3CC3)CC2)=O)CCN(C(=O)CCS(C)=O)CC1 c1(C(N2CCC(C(C)NC(=O)CCCN3CCCCC3)C2)=O)cncc(F)c1Cl c1(C(=O)NCCN(C(Cc2c(CC)con2)=O)CC(C)O)cccc(OC)c1F c1(CC(=O)NC23CCN(C(c4ccnc(O)c4)=O)CC2C3)ccc(Cl)cc1F C1(CC)(NC(c2ccc(O)c(N)n2)=O)CCN(C(c2[nH]c(O)nc2C)=O)CC1 Cc1ncc(C)c(=NCCC2CCN(C(c3cnn(CC(F)(F)F)c3)=O)C2)[nH]1 C1(CNC(CC2(C)CC2(Cl)Cl)=O)CCCN(C(c2cccc(Cl)c2N)=O)CC1 c1(C(N2CC(NCc3ncn(C)c3)C2)=O)ccccc1S(=O)(=O)N1CCCCC1 c1(CCCc2cc(C)[nH]n2)nc(-c2ccco2)nn1C1CCOC1 Cc1cc(O)cc(O)c1CNC1CC(C(N2C3COCC2C3)=O)C1 c1(C(=O)NCCC2CCCCN2CCC(C=C)C)ccc(Br)cc1N1CCOCC1 C(=O)(C(C)(CCC)CCC)NC1C2CN(C(C3(CC=C)CCOCC3)=O)C1CC2 C1(C(=O)NC2(CCCCNC(CCOCC(C)C)=O)CC2)CC(O)C(F)C1 C1(C(N2C(C3CCN(C(CNC(N)=O)=O)CC3)CCC2)=O)Cc2cccnc2C1 N1(C(C2(C(=O)OC)CCCC2)=O)CC2CN(C(=O)CC3CC(C)(C)C3)CC2C1 C(=O)(C(F)(F)C(C)(C)O)NCC1C2N(c3cc(C(=O)OC)nc(Cl)n3)C(CC2)C1 C1(NC(CCCCCCCC)=O)CCOC12CCN(C(C1(OC)CC1)=O)CC2 C1(NC(c2c(C)ccnc2)=O)CCCC(NC(c2ccc(C#N)s2)=O)CC1 C1(CC)(NC(=O)Cn2cc(CN3CCC(O)CC3)nn2)CCSCC1 c1(C(=O)NC2(c3ccccc3)CCN(C(C)=O)C2)ccc2c(c1)B(O)OC2 C1(CCNC(=O)CC2CCC(=O)O2)CCCCN1C(c1cc(C2CCC2)no1)=O C=CCC(C)(C)CC(=O)NC1CN(C(c2cncc3n[nH]cc23)=O)CC1O N1(C(C(COCC)c2ccccc2)=O)CCC(c2ccc(C)cc2)CC1C c1(CC(=O)NCCn2cc(C(=O)NC3(C#C)CC3)nc2)ncccc1C c1(C(=O)OC)c[nH]c(=NCC2CCCCN2C(=O)C(=O)NC2CC2)s1 C(C(C)(C)CNC(=O)CC1(O)CCOC1)N(C(=O)COC(F)F)C N1(C(Cn2c(C)nnn2)=O)CC(C(N2CCN3CCCC3C2)=O)C2(CCC2)C1 Cc1ccc(C(=O)C(N2CC(NC(=O)CN3CCSCC3)CC2C)=O)cc1 N1(C(C2(C)C(CC)CCC2)=O)C(CNC(=O)CCC=CC(C)C)CC2CCCC12 CC(C(=O)N1CCC(n2cc(C3CC3)nn2)C1)S(N)(=O)=O CC(C)(C(=O)N1CCC(C)(NC(c2ccc(N)cc2Cl)=O)C1)C1=CCSCC1 c1(C(=O)NC2CC(C)N(C(C3CC(=O)CCO3)=O)CC2)cn2cccnc2n1 c1(OCC)ccc(C)c(F)c1-c1ccc(C(=O)NCC2(O)COC2)nn1 N1(C(C2CCC(C)O2)=O)CCCC12CCN(C(c1cc(C3(C)CC3)on1)=O)C2 c1(CCC(=O)NCC(O)CNC(=O)C(=O)Nc2ncc[nH]2)ccncn1 c1(OC)c(C(=O)NC2COCCN(C(=O)C(C)c3ccco3)C2)c(C)nn1C CCC(C)(C)C(=O)N(C)Cc1ccc(CNC(C2(n3nccn3)CC2)=O)cc1 C(=O)(C(CCF)NC(=O)CCCn1cncn1)N(CC(=O)NC(C)C)C C1(NC(c2cccc(NC(C)=O)n2)=O)CCN(C(=O)Cn2cccc2)CC12CC2 c1(C(N2CCC2C(N2CCC(c3ccc(Cl)cc3)C2)=O)=O)n[nH]c2cccc(F)c12 C(C(C)(CC(C)C)NC(=O)C#CC1CC1)NC(c1c(CC)nco1)=O c1(NC(=O)NCCC)cccc(NC(=O)CCNC(c2nn(C)cc2Br)C)c1 C(=O)(C1=NOC(C)(C)C1)NCCC(C(C)C)NC(c1cc(C)c(Cl)s1)=O CC1CN(C(c2cc(Cl)sc2Cl)=O)CC2(CCN(C(C3CCC(=O)NC3)=O)C2)O1 C1(CCC(=O)NC(C)C(CO)NC(c2cnc(S)n2C)=O)CCC(=O)NC1 CC(C)CCN=C(NCc1ccc(Br)s1)NC1CC1c1c(Cl)cccc1Cl c1(C(=O)NCC(CC)NC(C2(F)CCCC2)=O)ccccc1CCn1ccnn1 CCCCC(CNC(c1ccc(C(F)F)nc1)=O)NC(C1CCCOC1)=O c1(NC(C2C(NC(C(CC)COC)=O)CC=CC2)=O)c(C)nc(C)nc1C Cc1cc(C)c(O)c(C(N2CC(S(C)(=O)=O)C2)=O)n1 C12(C(=O)NCCCCNC(c3cnc(OCC)s3)=O)CC3CC1C2C3 C#CCC(C)C(=O)NCC1CCC1NC(C1CCCC1C(C)C)=O c1(Oc2ccc(-n3c(C)nc(C)n3)cn2)c(C)cc(Br)cc1C N#Cc1ccc(S(=O)(=O)N2CCCc3n[nH]cc3C2)cc1F C1(C(N(C(CCNC(c2ccc(NC)cc2)=O)C)C)=O)CN2CCN1CC2 C(=O)(C(CC(C)C)C(N)=O)NCC#CC(N1C2CC(CC)CC1CC2)=O C1(CNC(c2nc(C(=O)OC)sc2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC12CC2 CCC(C)(C)C(O)C(=O)NC(C)CCC(=O)NCC(c1ccsc1)C c1(C(=O)NC(C(C)C)C(=O)NCc2nccn2C(C)C)cc2n(n1)CCC2 C1(C(=O)NC2CC(C(N(CC(C)C)C(C)C)=O)C2)CCCCCN1C N1(C(c2cnc(S(C)(=O)=O)s2)=O)CCCC12CCN(C(=O)Cc1cscn1)CC2 Cc1cccc(C(N2CCCCCC2CNC(c2cn(C)c(=O)cn2)=O)=O)c1N C(=O)(CCCC(F)(F)F)NCC12C(CN(C(c3c(OC)ncc(Cl)c3)=O)C1)C2 N1(C(c2cc(Cl)cc(Cl)n2)C(=O)NCC=C)CCC2(C1)NC(=O)NC2=O N1(C(c2nc(CC)on2)C)CCC(CC)CC1.c12nc(cs1)CCNC2=O c1(OCC)ccc(C(=O)NC(C)C(C)NC(c2cc(C3CC3)no2)=O)cc1 c1(C(=O)NCC(C)NC(c2ccc(OC)cc2Cl)=O)nn(C)cc1[N+](=O)[O-] C1(NC(C(c2c(C)n[nH]c2C)C)=O)CCN(C(c2ccc(C#N)cn2)=O)CC1F c1(C(N(C2CCCN(C(=O)CC(C)C)CC2)CCC)=O)cnc2cc(Cl)ccn12 C(CC(=O)NC1CCN(C(c2coc(C(N)=O)c2)=O)CC1O)(C(N)=O)NC(C)=O N#Cc1cccc(CN2CCOCC(C(=O)Nc3cc(Cl)ccc3O)C2)n1 C(CCCCCC(=O)N1CC(C2CC2(F)F)C1)NC(C1(CC)CCCC1)=O N1(C(C2C(C)N(C)CC2)=O)CC2CN(C(c3ccccc3Cl)=O)CC2(C)C1 c1(C(N2CC(C)(C)C2COC)C(=O)NCCCCCC)nc(C)n(C)n1 C#CCC(C(=O)Nc1cnc(CCC)nc1)NC(C1CC1Cl)=O CCCC(CC)C(=O)NC1CCCCC1CNC(=O)Cc1c(C)noc1Cl N1(C(C(n2c(C)ccn2)C)=O)CCN(C(=O)C=C(Cl)Cl)C(CC2CC2)C1 C1(CCNC(c2cc(Br)no2)=O)(NC(C2C(=C)CC2)=O)CCCC1 c1(OC)cc[n+]([O-])c(C(=O)NCCC2CC(NC(c3cc(Cl)c(C)cn3)=O)C2)c1 c1(CC(=O)N(CC(CC)(C)NC(c2cnc(OC)cn2)=O)CC)nc(C)c(C)s1 C1(CNC(c2cc(CC)n(C)n2)=O)CCC2CN(C(=O)C(O)CSC)CC12 C#Cc1cnn(C)c1C(=O)NCC1CCCCN1C(=O)C(COC)N(C)C c1(CC(=O)N(CC2CCN(C(CC3C(CC)C3)=O)CC2)CC)ccc(F)c(Cl)c1 c1(C(N)=O)ccc(CNC(=O)NCC2(N3CCCC3)CCOC2)o1 c1(OCC)c(C)cc(C(=O)NC2CC(NCc3ccccc3F)C2)cc1C C1(CNC(CCc2cncc(OC)c2)=O)CC(NC(=O)C(=O)N(C)C)C12CCC2 CCCC(C#N)C(=O)N1CCCC(C(C)C(=O)NCC2CC3(CCC3)C2)C1 CC1(C)CCCC1(O)CNC(=O)Cn1cc(CNC(C2CCNC2=O)=O)nn1 N1(CCCC(C)C)CCC(CC(C)NC(=O)C(F)CN(CCO)CCOC)CC1 CC(C)CCC(C(=O)NCC(C)CC1CCC1)NC(C12CCC(C1)C2(C)C)=O c1(C(=O)NCCN(C2CCCC2)C(COC(CC)(C)C)=O)cc(Cl)c(Cl)n1C C=CC(C(F)(F)F)NC(C1CCCN(C(=O)C(C)C(=O)OC)C1)=O C(=O)(CCS(=O)(=O)C1CCCC1)NCC1CC(OC)CN1C(C1CCCN1C)=O c1(C(=O)NCCC(C)N(c2ncnc(C(C)(C)C)n2)C)ccc(O)nc1 C(C(C(C)C(C)C)NC(c1cn(CCO)nn1)=O)NC(CCN(C)CC)=O C1(O)(C(C)NC(=O)COCC(C)(C)C)CCN(C(=O)CC2CC3CC3C2)C1 C1(C(=O)NCC2(C)CC2)CCN(C(=O)C2C3CC(=O)CC23)O1 C(CCN=c1cc[nH]c(=NCCCCc2ncc[nH]2)[nH]1)c1cccc(C)n1 C1(NC(c2c(C)n(CCO)cc2)=O)CCN(C(=O)CC(C)(F)F)CC1C(C)C C1(NC(c2ccccc2O)=O)(CNC(C2(CN(C)C)CC2)=O)CC2CCC1CC2 C(=O)(C(C)(C)C1=CCSCC1)NC1CCN(C(CCC(CCC)CC)=O)CC1F N1(C(CCC(CC)C)=O)CC2CN(C(=O)CCc3ccc(Cl)c(F)c3)CC2C1 C1(C)(CNC(C(CC)C(C)C)=O)COCCN(C(c2ccnc(OC)n2)=O)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CC2CCCC2(NC(c2ccn(C)c2C)=O)C1 N1(CC)CCC(n2nc(COC)nc2-c2cnn(CC3CCOCC3)c2)CC1 c1(C(=O)NC2(COC)CN(C(CC3CC(CC)C3)=O)C2)cnc2ccncc2c1 C(=O)(C1c2c[nH]nc2CN1C(=O)C1=C(Cl)CCCC1)Nc1cncc(C(N)=O)c1 CC1(C)OCCOC1c1nnc(N2CCCCC2)n1CC1CC12CCCCC2 C1(CNC(C2CCCN(C(C(CC)CC)=O)C2)=O)CC(=O)NC(C)C1 c1(NC(=O)OC)cccc(CC(=O)NCCS(=O)C(F)F)c1 c1(C(N2CCC(n3cccc3)C2)=O)csc(-c2ccoc2)n1 C(CCC(C(=O)NCC(=O)NCCOC)N(c1ccccc1OC)C)OC c1(C(N(CC(=O)OCCNC(=O)COC2CC2)C)=O)cc2c(nn1)CCC2 N1(C(=O)OC(C(C)(C)C)=O)CC2CC2(N(C(=O)CC=C(Cl)Cl)CCO)C1 Nc1ccc(Cl)cc1C(=O)NC1COCC1CNC(C1CCNC1=O)=O C1(C(=O)NCCC(C)(C)NC(c2c(CCC)n(C)nn2)=O)C2CCC(F)(F)C12 c1(C(N2CC(CCNC(CC=CC)=O)C(C)C2)=O)[nH]c2ccccc2c1Cl c1(CC)nccnc1C(=O)NCCC(O)C(=O)NC1CCCC(CO)C1 C(=O)(C(CCc1ccncc1)NC(=O)C(C#N)C=Cc1ccccc1)OCC C1(NC(C(C)n2cncn2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)O)C2 Cn1nc2cc(Br)ccc2c1C(N1CCC(NC(=O)CN=S(C)(C)=O)C1)=O c1(NC(=O)NC(Cc2ccoc2)CO)csc2c1CCCC2 Cc1ccc2c(=NC(C)c3nccn3C(C)C)[nH]c(N3CCC4(CC4)C3)nc2c1 Cc1cc(C(C)(C)NC(=O)CN(C(=O)CNC(=O)C(C)CF)C)cc(C)c1 C(=O)(CC(C(C)CC)NC(C1CC(CC)C1)=O)NC(CCC=C)C1CC1 c1(CC)nocc1CN(C)CC1CCC(=O)N1 c1(CCC)ccc(C(N2CCC(O)(CCNC(=O)C3CC3)C2)=O)cc1[N+](=O)[O-] C=CC(C)(C)C(=O)N(C)CC1CCCN(C(=O)CCCN2C(=O)CNC2=O)C1 O=C(C1COc2ccccc21)NC1(C2CCN(C(C3CC34CCOC4)=O)C2)CC1 c1(C(N(CCC)CCNC(C2CCC(C)(C)CO2)=O)=O)ccnc(S(N)(=O)=O)c1 c1(N(CCCC)C)nnc(-c2ccco2)n1CC(n1cccn1)C CC1CCCC1(C)C(=O)NCc1cn(CCN(CCCF)C)nn1 C1(CCCC)CN(C(=O)CNC(=O)CNC(c2ccoc2C)=O)CCN1C(C)=O C1(CC(=O)NCc2c(C)cns2)CN(C(=O)Cc2ccccn2)CCC1C n1(CC(=O)NCC(CC=C)NC(c2cncnc2)=O)cc(C)c(O)nc1=O N1(C(CNS(CC)(=O)=O)=O)CC2CC(CNC(=O)CC3OCCCO3)C2C1 c1(C(N2CC(O)(CCNC(C3CC=C(C)CC3)=O)C2)=O)cc(N)c(C)c(N)c1 N1(C(C=NOC)=O)CCC(CCNC(c2scc3c2CCCC3)=O)C(F)(F)CC1 C(=O)(C1SCCc2sccc21)N1CC(N(C(=O)CCc2cnoc2)C)C1 C1(CNC(c2cnc3ncccn23)=O)CCN(C(=O)C(F)F)CC1(F)F C1(C(=O)NC2C(NC(c3c(N)c(Cl)ccc3)=O)CC2)CCOCC12CCC2 c1(C(N2CC(NC(c3ccc(C(C)N)cc3)=O)C(F)C2)=O)cc(O)cc(O)c1 C1(C(=O)NCCN(C2CC2)CC)C(C)OCCN1C(=O)CC1CCC(C)CO1 N1(C(CC=CC=C)=O)CCN(C(=O)Cc2cc(OC)cc(C(F)(F)F)c2)C2CC12 Cc1ccc(C(C)C(N2CCC(CF)(NC(C3CC(C)(C)C3)=O)C2)=O)cc1 Clc1ccc(C2(NCCC3CC=CC3)CCCC2)cc1Cl c1(N2CC(CNC(C(CC)NC(C)=O)=O)C(C)(C)CC2)nc2cc(C)ccc2o1 CCC(CC(=O)NCCC1(O)CN(C(c2nc(=N)cc[nH]2)=O)C1)C(F)F CC(N=c1cc[nH]cc1S(=O)(=O)NC1(C)CCCC(C)(C)C1)C12CCCC1C2 N1(CCc2cn(C)nc2)CCC(NC(c2cc(=O)cc[nH]2)=O)C(O)C1 C(=O)(C1=CCCCCC1)NCC1CN(C(=O)CC2COCC2O)CCC1CO Cc1ccccc1-n1cc(C(N2CCN(C(C3(CF)CC3)=O)CC2)C)nn1 C1(C(=O)NC2CC(CCNC(=O)Cn3ccnn3)C2)CC(c2ccccc2)=NO1 C1(CC(N2CCCC(C)C2)=O)N(C(c2ccn(C3CC3)n2)=O)CCC1(C)C C(CC1CCC1)(C(=O)NOCCC1(C)N=N1)NC(c1cccc(CC)n1)=O C(C(=O)NC1C=CC(C(=O)NCc2scnc2C)C1)(C(C)C)SC C(=O)(C1CCCc2nnn(C)c21)NC1CN(C(c2c(CC)n[nH]c2)=O)CC(F)C1 C1(C(N2C(CC)CCC2)=O)Cc2c(C)cccc2O1 c1(C(=O)NC(CNC(C(C#N)C2CC2)=O)C2CCC2)ccc(-n2cccn2)cc1 Cc1c(Cl)ccnc1C(=O)NC(C1CCCCN1C(=O)CCCSC(C)(C)C)C N1(C(c2scc(C)c2C)=O)CCN(C(C2CC2[N+](=O)[O-])=O)CC12CCC2 C(=O)(C1=Cc2ccccc2C1O)NCCN(C)C(c1cccc2nc(O)oc12)=O C=CC1(CO)CCN(C(C2C=CCCN2C(c2cc(Cl)ns2)=O)=O)CC1 N1(C(C(C)OCCOC)=O)CCC2(C1)CN(C(=O)CCNC(C1CCCO1)=O)C2 Cc1nc(CO)ncc1C(=O)NCC(C1CCC1)NC(=O)C(Cl)=CCl c1(C2(C)CC2)cccc(C(=O)NC2(CNC(C3CCCS3)=O)CCCCC2)c1 N1(C(C=C(C)C(F)F)=O)CC2C(CN(C(=O)CC(C)N(C)C)C)C2C1 C1(C(=O)NCC(C)(C(C)C)NC(C=C(CCC)C)=O)CCN(C)S1(=O)=O C(CCCCF)NC(CCN(C)CCn1cc(CCO)nn1)=O N1(C(C(CCC)CCC)=O)CC2CCCCC2(NC(C2COC(=O)N2C)=O)C1 C1(NC(C(CO)N(C)C)=O)CN(C(c2cnc(C(N)=O)s2)=O)CCC1CO Cc1n[nH]c(=NC(=O)c2ncnc3c2cnn3-c2ccc(Cl)c(F)c2)n1C C1(CNC(C(C)OCCCC)=O)CCN(C(c2ccnnc2)=O)C12CC2 CCN=C(NCCC1CCCCC1)NC(C)CCN1OC(C)CC1 CC1OC2(CN(C(N3CCOC(c4cccc(F)c4)C3)=O)C3CC3)CCC1C2 c1(C(N2CCCC(N(C(C=COCC)=O)CC)C2)=O)cn2ccn(C)c(=O)c2n1 N1(C(c2ccc(CC)o2)C(=O)NCC2CC2)C2C=CCC1CCC2 c1(C(=O)NCCCCC(C)NC(C2CCS(=O)(=O)C2)=O)c(N)nn2ccccc12 CN=c1ccc(C(N2CCSC3CCC23)=O)c[nH]1 C1(NC(C2(C)CC3CC3C2)=O)CN(C(=O)Cc2ccsc2)C2(CCCC2)C1 c1(NC)cncc(C(=O)NCc2cc(C(N3CCC(N(C)C)C3)=O)n(C)n2)c1 C1(O)(CNC(C=CC=CCCCCC)=O)CCN(C(=O)CC2CNC(=O)C2)C1 C1(NC(C2(C3CCC3)CC2)=O)CC2CN(C(c3ccc(C)nc3)=O)CC12 C1(C(C)OC)CCN(C(=O)C=CC2CCCN2C(c2n[nH]c(=N)[nH]2)=O)CC1 N1(C(c2ccc(C#C)o2)=O)CCC(C2CC2)C1C(N1CCCOC(C)C1)=O C1(C(=O)OC)(C(N2CC3C(CNC(=O)OC(C)(C)C)C3C2)=O)CCS(=O)(=O)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(NC(c2nn(C)c(O)c2)=O)C(C(N)=O)C1 N1(C(C2N(C(COCCC#C)=O)CC=C2)=O)CCC(F)(C#N)C1 C1(c2cc(CNC(c3c(CC)non3)=O)on2)CCN(C(=O)C2=CCC2)CC1 C=C1CC(C(F)(F)F)(C(N2CC(O)(CNC(C3CCCCS3)=O)C2)=O)C1 C1(O)(C(=O)NCc2c(CC)ocn2)CC2(CCCN(C(=O)OC(C)(C)C)C2)C1 c1(CN(C(C2(CC)CN(C(c3ccsc3C)=O)C2)=O)C)cccc(C)c1 c1(C(N(CC(C)NC(C2(c3nccs3)CC2)=O)C)=O)cnccc1N(C)C Cc1ccc(C)c(C(N2CCN(C(c3cn(CCO)nn3)=O)C3CC23)=O)n1 N1(C(CC=CC)=O)CCC(c2ccccc2)(NC(=O)C(CC)OCC)C1 C1(CC#C)CCN(C(=O)C(CCC)NC(=O)Cc2cc(C)cs2)CC1 c1(C(=O)NC(CCNC(CN(C)CC)=O)C(C)C)c(F)ccnc1Cl Cc1nn(C)c(C)c1C(=O)NC1CCCCC1C(N1CCCC(C(F)(F)F)C1)=O C(=O)(C(F)CCC(C)C)NCC1CCN(C(C2CC(CC)OCC2)=O)CC1 O=C1CC(C(=O)N2CC3(C2)CN(C(c2cc4c[nH]nc4s2)=O)C3)c2ccccc21 Cc1nc(N2CCC(NC(c3cc[n+]([O-])cc3)=O)C23CCC3)ccc1C#N Cc1ccc2c(CCC(N3CC(F)(CNC(C4CC4(C)CF)=O)C3)=O)c[nH]c2c1 CC(O)C(C)C(=O)N(CC(C)(C)CNC(c1csnc1C1CC1)=O)C CC#CCC(C(=O)NCC1CC2CCCC2C1)NC(c1ccccn1)=O C1(C(C)(C)C)CC(CNC(C2(F)CCCC2)=O)CN(C(=O)Cc2ccsn2)C1 C(=O)(CCC1=CCCCC1)NC(CC(=O)NCC1(C)ON=C(C)C1)C C1(NC(C(CO)OC)=O)COC2CN(C(=O)CC3CCSC3)CC12 C1(CNC(C2(SCC)CC2)=O)CCCCCN1C(=O)CCc1cn(C)cn1 N1(CC(COCC(C)C)O)CCC(C)(NC(c2cnc(Cl)c(Cl)c2)=O)CC1 C1(C(=O)NCCC2(NC(C(=O)NCCOC)=O)CC2)CS(=O)(=O)CC12CC2 CC(N=c1[nH]c2cc(Cl)ccc2s1)C1CCCCN1C(=O)C1=COCC1 Cc1ccc(C(N2CC(NC(c3c[nH]c(=N)o3)=O)C3(CC3)C2)=O)c(C)c1 CC1CCN(C(=O)CCc2ncccn2)CC1NC(c1cscn1)=O CCC(C)(C)CCCC(=O)N1CC(C)N(C(=O)C(C)OC2CCCCC2)CC1C CC1CCC(OC(c2c(O)ncc(Br)c2C)=O)C=C1C(N)=O Cc1ccc(C)c(C(N2CCCCC(N(C)C(C3CCCCC3C)=O)C2)=O)c1C N1(C(CC=C(C)C)=O)CCN(C(c2ccnc(C3CCC3)c2)=O)C(C2CCC2)C1 C1(O)(C(=O)NCCOCCN(C(C2CCC(C)S2)=O)C)CC(C)(C)C1 c1(C(C)NC(c2c(C)n(CC(F)(F)F)nc2)=O)ccc2c(c1)CC(=O)N2C c1(COC)ncc(C(N2CCCC(CN(C)C(C3CCOC3C)=O)C2)=O)c(O)n1 c1(NC(C2CCCCN2S(=O)(=O)C(Cl)(Cl)Cl)=O)cc(O)c(Br)c(O)c1 CC1CN(C(=O)C(F)CC2CCOC2)CC1NC(C1CCNC(=O)C1)=O Cc1nc(C=CC(N2CCCC2(C)CNC(c2ccncc2)=O)=O)cs1 C(=O)(CC(C)n1ccc(C)n1)NC1(CCCNC(COCCCCC)=O)CC1 c1(C(=O)NCC2OCCCN(C(C3C(C)CCO3)=O)C2)cccn2[nH]c(=N)nc12 c1(NC2CC(NCCC(F)(F)F)C2)cc2cccc(Br)c2nc1Cl C1(C(N2CC(C)(NC(C(C)OC(C)(C)C)=O)C2)=O)(N(C)C)CCOCC1 C=C(C)CCCC(=O)NCCOCCNC(=O)C(C)(C1CCOCC1)OC Cc1cnc(NC(c2cccc(Cl)c2)C)c(S(=O)(=O)N2CCC(CCO)CC2)c1 c1(C(=O)NC2CCN(C(C3(C(=O)OC)C=CCC3)=O)C2)cccc2ncsc12 C(=O)(C(F)(F)CC(C)C)N1CC2C(NC(Cc3c(CC)cccc3)=O)(C2)C1 N1(C(C2C(C)=C2)=O)CCC2(CC1)CCN(C(C1(CC3CC3)CC1)=O)CC2 N1(C(Cc2c(C)snc2)=O)CCc2cc(-c3cn(C4(C)CC4)nn3)ccc21 c1(COCC)n[nH]c(=NC(CO)C(C)C(O)c2nc(CC)no2)o1 C(CCC(C(=O)NOC(C)CC)NC(=O)C1CC1)OCC C1(C)(C(=O)NC(CC)CN(C(=O)C(F)=C2CCCC2)C)CS(=O)(=O)C1 C1(NC(C2CCN(CC#C)CC2)=O)COCCN(C(C2CC3CCC2O3)=O)C1 c1(C(C(=O)NCC=C)N(C2CCS(=O)(=O)C2)C)cc(C(F)(F)F)cc(Br)n1 c1(CC)noc(C(=O)NCCCC2CCCN2C(=O)CC(=O)OC)n1 C(=O)(CC1NC(=O)c2ccccc21)N1CCC(NC(CNS(NC)(=O)=O)=O)CC1 Nc1ccc(C(N2CCCC2CCNC(C2CCCC(C(N)=O)C2)=O)=O)cc1O N1(C(C(CCC=C)NC(=O)CCSCC)=O)CC2CC(C1)N(C)C2 c1(C(N2C(C(C)NC(=O)CC3CCC34CCC4)CCC2)=O)cnn2ncccc12 CC1C(=O)OCC(C)(C)N1C(c1ccc(C#N)n1C)=O N1(CC)CCC(NC(c2ncoc2CNC(=O)C(C)(O)C2CCC2)=O)C1 N1(C(C2CN(C(=O)Cn3ccnn3)CCO2)=O)CC(F)(F)CC1CO CCC(C)C(O)C(=O)NC1CCC(NC(c2ccco2)=O)C1 CCC(C)(C)CC(=O)NC1CCC1NC(=O)C(C)CCCC CCC(C)C(C(=O)NC1CCC(CNC(C2(CC(C)C)CCCC2)=O)CC1)OC c1(OC)cc(C(=O)N(CC(O)CN(C(=O)C2=CSCS2)C)C)n(C)n1 C1(C(N2CCCC2c2ccco2)=O)CN(Cc2cnccc2C(F)(F)F)CCO1 C(C)(C(C)(C)C(=O)N1CCCC(OC)C1C)NC(c1n(CC)nnc1)=O c1(C(=O)Nc2scc(CC)n2)cc(Br)ccc1CC(=O)N(C)CCN(C)C N1(C(COC(C)=O)=O)CCC(NC(c2cc3c(cn2)CCCC3)=O)C12CCCC2 C1NCCCC12CCC2.c1(C2C(C)(C)CCNC2)c(N)cc(Cl)cc1F Cn1nc(C(=O)NCCC2CCCN2C(=O)CC2(C)CC2(F)F)cc1C(F)(F)F c1(C(=O)NC2CCC(N(C(=O)CCc3ccsc3)C)C2)ccc(Cl)c(F)c1O c1(C(=O)NCC(C2(O)CCN(C(c3nn(C)cc3N)=O)C2)C)ccc[n+]([O-])c1 C1(NC(C2C(=C)C2)=O)CN(C(=O)CCOc2ccccc2C(=O)OC)CC1C1CC1 C(CO)(C(=O)NCC1CCC1C(=O)NCC1CCCO1)N(C)C C=CC(C)(C)CC(=O)N1CCC(NC(C2CC23CCSCC3)=O)CC1C N#Cc1ccc(C(=O)NC2CCCCC2NC(C2CCOCC2)=O)nc1 C1(C(=O)NCC(CNC(C(C)(F)F)=O)(C)O)CC2(CC2)CN1 c1(C(N2CC(CNC(C3(OC)CCC3)=O)OCC2)=O)cccc(C(C)(C)C)c1N Cc1nc2cccc(C(=O)N(CC(C)NC(=O)C=Cc3cncnc3O)C)c2[nH]1 N1(C(c2c(C)oc(Cl)n2)=O)CCCOC(CCNC(C2CCCN2C=O)=O)C1 C1(C(N2CC(=C(CNC(c3cc(C(F)(F)F)cs3)=O)F)C2)=O)C(F)(F)C12CC2 C1(CC)CCCN(C(=O)CC2CN(C(=O)C=CC=C(C)C)CC2C)C1 Cc1c(C=CC(=O)NC2(CCCNC(C3COC(C)C3)=O)CC2)cnn1C C1(CNC(CCN(CCCCC)CC)=O)CCN(C(=O)CS(C)(=O)=O)C1(C)C c1(C(=O)NCC=CCNC(Cc2cncc(C#N)c2)=O)cc2c(nc1O)CCOC2 CCC(C)CCC(=O)N1CCN(C(=O)CCCC(=O)NC)C(C(C)C)C1 N1(C(c2cnc(O)[nH]2)=O)CCc2ccc(-c3ccc4c(O)ncnc4c3)cc2C1 C#CC1CCCN(C(C2CCC=CC2NC(C2CC(=O)C2(C)C)=O)=O)CC1 C(CCF)(C(=O)NCCCNC(=O)OC)NC(C(CC)=CCCC)=O N1(C(CCc2cccc(OC)c2)=O)CC2(C1)CN(S(=O)(=O)c1cccs1)C2 C1(C2CC2)(CNC(C(C=C)C)=O)CCN(C(c2cc(CC)nnc2C)=O)C1 C(=O)(C(C(C)C)C(C)C)NC12CC(CNC(CCCCOCC)=O)(OC1)C2 CC(C(=O)N1CCC(CNC(c2ccnn2CCF)=O)C1)P(C)(C)=O C1(NC(CC(C=C)C)=O)CN(C(=O)CC2CCC=CCC2)C2CCCCC12 C1(C(N(C2CCN(C(=O)C3=CCCCC3)CC2)C)=O)CC2CCCC2C1 N1(C(c2cnc(OC)nc2C)=O)CC(NC(=O)CCCCCF)C(C2CC2)C1 c1(CCC)cc(C(N2CCCC(N(C)C(C3CC4CC4C3)=O)C2)=O)cc(O)n1 c1(C(=O)NCCNC(c2sc(Br)cc2F)=O)cc2c(cn1)COCC2 C1(C(N2CCC(C(C)C)C2)=O)CCCN(C(=O)CC2C=NN(C)C2=O)CC1 C1(C(N2C(CN(C(CNC(CC)=O)=O)C)CCC2)=O)CCCN1N=O c1(CC(C)(C)C)noc2ncc(C(N3CCN(C(=O)C(N)=O)C(CO)C3)=O)cc12 C1(C(N2CCC3(CCC3)C2)=O)CCN(C(=O)C2(Cl)CCC2)O1 C1(C(N2CCC(N(C)CC)C2)=O)CC(NC(C2CCCC2O)=O)C(O)C1 c1(OC)cccc(C(N2CCC3(CC3C(=O)NC3CS(=O)(=O)C3)C2)=O)c1OC c1(C(N(CCC(C)NC(c2cn(CCC)nc2)=O)C)=O)sc2ccsc2c1C CC(C)(CN=c1[nH]ncs1)NC(=O)C(CCc1ccsc1)Nc1ccccc1Cl N1(C(C2(C)CC(F)C2)=O)CCCCC(CNC(c2ccc(SC(F)(F)F)o2)=O)C1 N1(C(CCC#CC)=O)CCC(C)(C(=O)NCC(C)COCC)CC1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(CCc2cn(C(C)C)nn2)OCC1 C1(OC(C)C)CCC(c2ccccc2)CC1.C12CCCN1C2=O C1(C(N2CC(C)C(C)(C)CC2)=O)CCCN1NC(=O)C=Cc1ccn(C)c1 C1(NC(COC(CC)C)=O)CC(O)CN(C(C2(OC(C)=O)CC2C)=O)C1 c1(OC(C)(C)C)ccnc(CNCC23CC(CCO2)C3)c1 c1(C(=O)Nc2ccc(-n3ccnn3)cc2)ccc2c(c1)CNCCN2 C1(CC)CCCCC1C(=O)N(C1CCN(c2nnc(C(=O)OC)o2)CC1)C C(=O)(CCCNC(=O)OC)N(C1CCN(C(=O)C(Br)=C(C)C)C1)CC C(CC(C)C(=O)NC(CNC(C1(c2ccn(C)n2)CC1)=O)CC)=CC N1(C(C(c2c(F)cccc2F)C)=O)CC(O)(C2CCN(C(C3CCC3)=O)CC2)C1 c1(C(=O)NCCN(C(=O)CCOCCCOC)C)ncccc1O C1(C(=O)NN2CCN(C(C(C)O)=O)CC2)CC2COCC(C1)C2.c12cn(nn1)C2 CC1CCN(C(=O)CCC2CC2)C1CNC(C1CCCC1O)=O c1(OC)ccc(S(=O)(=O)N2CCC3(CC2)CC3(C)C(=O)NC(C)CO)c([N+](=O)[O-])c1 C=CC(C)CC(=O)N1CC(C(=O)NCc2cccc(Cl)c2)C(C)C1 N1(C(CCCCOCC)=O)CC2(CC1CNC(c1ccncn1)=O)CC2(F)F CC(C(=O)NC1CC(O)CN(C(=O)Cc2cnccc2Cl)C1)S(N)(=O)=O c12cccc3nc([nH]c13)C1C(CC)(C1)CNC2=O.c1(SC(C)(C)C)ccccc1 S(=O)(=O)(c1cccc(Br)n1)N1C(C(=O)Nc2nc(Br)cs2)C=CC1 C1(C(=O)OCC)CCN(C(=O)C(Cc2ccc(C)cc2)NC(C)=O)C1C N#Cc1cnn2cc(C(=O)NC3CCCN(C(c4ccccn4)=O)C3)cnc12 C1(C2CC2)(C(N2C(C)(C(=O)NC)CC2)=O)CN(C(=O)CNC(=O)OC)C1 c1(C(=O)NC(CNC(C23OC(C)(C)C(C2)C3)=O)(C)C2CC2)cnn2ncccc12 N1(C(C(CC)OC)=O)CCOC2(C1)CN(CCN=c1cc(C)nc[nH]1)C2 CC(C)CC(CNC=O)CC(=O)N1CC2C(CNC(c3cnncc3O)=O)C2C1 C(=O)(CCCCC(C)=O)N1CC(C)(COC)C1 C1(NC(CC(C=C)CC)=O)CN(C(=O)CCC2CCCC2)CCC12CCOCC2 CC(O)(CC(=O)N1CC(NC(c2cccc(OC(F)F)c2)=O)C1)C1CC1 c1(NC(N(C)C)=O)ccnc2ccc(C(N3CCCCC3C(O)C(F)(F)F)=O)cc12 c1(C(=O)NCC(C2CCCOC2)OC)c(O)cc(=O)n2c1CCCC2 C=CCC(CNC(=O)C(F)CCCC)C(=O)NC(c1cc(C)no1)(C)C CC(C)C(F)(CNC(C1C=CCS1)=O)C(=O)N1CC(C)(O)C1 CC(C)(CCC(=O)NCC1CC2CCCC2N1C(c1cc(CO)[nH]n1)=O)[N+](=O)[O-] c1(C(C(=O)NC2CC(NC(c3ccc(OC)nn3)=O)C2)O)cc(F)c(F)c(F)c1 CC1(C)CN(C(=O)COC2CCC2)CC(C)(C)C1NC(C1CN2CCC1CC2)=O c1(OCCC(=O)N(C)CC2CCCN(C(C(CC#C)C)=O)C2)ccc(F)cc1Cl C(=O)(C1OCCc2ccccc21)N1CC=CC(NC(C(C)(C)n2cccn2)=O)C1 C1(O)(CCNC(C=CCN(C)CC)=O)CCCN(C(=O)C(C)C2(O)CCC2)C1 C1(C(CC)C(=O)N2CC(CO)(NC(=O)Cc3nncs3)C2)CCC(C)CC1 C=CCCCCCCC(=O)NCCCCNC(C1(c2ccnc(OC)c2)CC1)=O CC1(C)CC(C(=O)CC2C(F)(F)C23CC3)CC(C)(C)C1.C12CCCN(C1)C2=O C(C(C)(C)C(=O)NCC1(CO)CCN(C(C2CC=CCO2)=O)C1)OC CCC(C)CCC(=O)NCCn1cnc(C(N2CC(O)(COC)C2)=O)c1 N1(C(CC(=O)NC)=O)CCC(C2CCCN2C(=O)C(C2CCOC2)OC)CC1 N1(C(COCC)=O)CCC2(CCCC2C(N2CCC(C)(C)C2)=O)C1 C1(NC(=O)COCC2CCCCO2)CC2CC(C1)N(C(=O)Cn1ncnn1)C2 C1(Cc2cn(CC(=O)NCCCS(C)=O)nn2)CCC(C)(C)CC1 c1(C(N(C2CCCCC2NC(=O)Cn2cc(Br)cn2)C)=O)cnncc1O N1(C(CC)=O)CCCC1C(=O)NC1CC(N(C(=O)C(C)C2CCOC2)C)C1 N1(CCC)C(=S)NC(c2c(Br)n[nH]c2Br)C(C(=O)OC)=C1c1cnn(C)c1 C(=O)(C(C(C)NC(C1CC2C=CC1O2)=O)C(C)C)NCc1c(C)ccs1 C1(NC(CCCCC(CC)C)=O)CCOC12CCN(C(=O)CC(C)C(F)F)CC2 C(=O)(CS(=O)(=O)C1CC1)N1CC(CNC(c2ccc(C)nc2N)=O)CC1(C)C C1(C)(CNC(c2cc(OC)ncc2)=O)CCCN(C(C2CC(=O)C2(C)C)=O)C1 N1(C(C2N(C(c3ccnc(C)c3N)=O)CCC2(C)C)=O)CCOC2COCC2C1 N1(C(c2ccc(C)n2C)=O)CCC(NC(=O)CC2CCOC2)C(F)(F)CC1 N1(C(C(C)(c2ccccc2)OC)=O)CC2CCCC(CNc3nccc(C)n3)C2C1 N1(C(C2(C)CC(F)C2)=O)CCCC(CO)(NC(=O)C(F)(F)c2cscn2)C1 C(=O)(CCCCCN(C(=O)CC(C)(C)C)C)N(C)CC1CC1c1ccco1 CC(C)CC(C(=O)N1CCC(CN2CCCCC2)CC1)NC(c1nn(C)cc1Br)=O C1(NC(COC(CC)C)=O)CCCCN(CCc2ccccc2)C1 N1(C(CC2C(C)C2)=O)CC(O)(CN(C)C(c2csc(-c3cnc[nH]3)n2)=O)C1 Cc1c(C(N2CC(NC(c3n[nH]cc3Br)=O)C(O)C2)=O)ccn1C(C)C Cc1nn(C)c2c(NCC3(Br)CC3(F)F)nc(NCc3cc(Cl)ccc3Cl)nc12 N1(C(c2n(CCC)ncc2)=O)C2CCC1CN(C(C1CCOCC1)=O)CC2 C(=O)(C(C)CCCCCC)NC(CC#C)C(=O)NCC=CCl N1(C(c2ncn(CC)n2)=O)C2CCC1C(F)C(NC(c1coc(C(C)C)n1)=O)C2 Cc1cc(=NC(=O)C(CN(C)C)NC(c2ccc(=O)n(C)n2)=O)[nH]n1C(C)C C(C(C)(C(=O)N1CC2C(NC(c3coc(Br)c3)=O)C2C1)OC)OC c1(C2C(C(N(CCN(C)C)CC)=O)C3CCC2O3)cccc2c1CCCC2=O Cc1cccc2c1CCC2NC(c1ccc(OC(F)(F)F)cc1Cl)=O c1(CN2CCN(C(c3cc(F)ccc3Br)=O)C(CO)C2)c[nH]c2c(F)cccc12 N1(C(C)=O)CCC(N(C(=O)C(C)CC2CC2)C(=O)CC2(CN(C)C)CCC2)C1 C1(NC(CNC(=O)OCC=C)=O)CCN(C(C2CCN(C)C2C)=O)CC1 c1(C(=O)NCC2C(NC(c3ccc(CSCCOC)o3)=O)C2)nc(O)c(C)s1 C1(C)(CC(=O)NC(C(C)C)CNC(C2CCOC2)=O)CC(F)(F)C1 Cc1cc(C(N2CCC(c3nc(C)ns3)CC2)=O)nc(C(F)F)n1 C(CCC(=O)NC1CCCC1CNC(C1CC1C(N)=O)=O)=CC c1(C(N(CC(C)NC(=O)CCc2ncccn2)CC)=O)cccc([N+](=O)[O-])c1Cl C1(CNC(=O)C(F)n2ccnc2)C2CC1N(C(c1cccc(C(F)(F)F)c1)=O)C2 c1(N2CCC(N(C(=O)CN3CCOCC3=O)C)C2)c(C)cncc1[N+](=O)[O-].CN c1(C(=O)NCC(C)CNC(C2(F)CC2C)=O)ccc(CC(C)(C)C)cc1 c1(C(C)NCC(c2cccnc2)OC)ccc(Br)c(Cl)c1 c1(CN(C)C(c2conc2CNC(=O)CCC2(C)CC2)=O)ncccn1 c1(N2CCCC(CNC(c3cn4c(n3)CCC4)=O)CC2)nc2ccccc2s1 Cc1cc(C(N2CCN(C(=O)C(C)C(C)(C)C)C3CC23)=O)n2nc(C)c(C)c2n1 c1(C(=O)NCC(CC)NC(c2cc(C)ncc2C)=O)ccn2c1CSCC2 N1(C(C(CCC)=CCC)=O)CCC2(NC(=O)C(Cl)=CCl)CCCC12 C1(C)(C(=O)NCCCCN(C)C(c2ccc(N3CCCC3)cc2)=O)CCCOC1 N1(C(c2cc(Cl)cc(C)c2N)=O)CCN(C(c2nccnc2C)=O)CC(C)(C)C1 C1(C(CC)=O)CCC(C(=O)N(C2CC2)Cc2cn(Cc3cnnn3C)nn2)CC1 c1(C(=O)NC(C2CCN(C(c3cncc(SC)c3)=O)C2)(C)C)cnc(C)cc1C Nc1cccc(C2CCN(Cc3cn(C4CC(C5COCCO5)C4)nn3)C2)c1N CCCCCCCCCC(=O)NC1C2CCN(C(=O)C(=O)C(C)(C)C)C12 C1(NC(Cc2ccc(C(C)C)cc2)=O)CC2CC1N(C(C1CCCN(C)C1)=O)C2 C1(CNC(COCCCN=[N+]=[N-])=O)CCC(NC(=O)C2=CCCS2)CC1 C1(CNC(=O)CCOc2cccc(Cl)c2)CN(C(=O)C=Cc2ccoc2)CCCO1 c1(COC)nc(Cl)cc(=NC2CN(C(C3CCCN3C=O)=O)CC3(CCC3)C2)[nH]1 O=C(C1=CCCN(C(C2C3CCC(F)C23)=O)C1)NC(CCC1CC1)C1CC1 N#Cc1cc(S(=O)(=O)NC2CCOCC2)ccc1NCC(C1CCCC1)O Cc1[nH]c(=N)nc(O)c1CC(=O)NCC(C)CNC(=O)CC1CCC(F)(F)CC1 C1(C(C(=O)N(CC=C)CCOC)C)CCN(C(c2n[nH]cc2Cl)=O)CC1 c1(CSC)ccc(C)cc1OCCc1cccc(NC(=O)NCC(=O)N(C)C)c1 c1(C(=O)NC2C(C=C)CN(C(C3(C)CCCO3)=O)C2)nccn2cc(C)nc12 C1(C(=O)NC(CCC)C2CCCC2)CCN(C(=O)C(C)CC#N)C(C)(C)C1 CCCC(CC)CC(=O)NC1CN(C(=O)Cc2coc3ccccc23)CCC1O C#CCC(CC(F)F)NC(=O)CCN(C(=O)Cc1ccc(O)cc1)C1CC1 c1(N2CC(C(=O)OC)C(OC)C2)ncnc(N(CC)CC)c1N.C1CC1 c1(C2(C(C)NC(N3CC4C(C3)C4(C)C)=O)CC2)cccc(F)c1F c1(C(N2CCN(C(=O)CCCn3ccnn3)C3C2C3)=O)cncc2nc[nH]c12 c1(C(N(CC)CC2CCCN2C(=O)CCSC2CCCOC2)=O)cc(C)nn1C c1(CNC(c2c(C)scn2)c2nnnn2C2CC2)cccc(N(C)C)c1 C1(OC)CC(NC(=O)CCc2cc(C)[nH]n2)CN(C(C2(n3nccn3)CC2)=O)C1 N1(C(C(n2c(C)ccn2)C)=O)CCOC(CN(C)C(C2(F)CC=CCC2)=O)C1 C1(CNC(=O)NCC2CCC(C)(C)O2)CCCC(F)(F)C(=O)N1 c1(NC(C2CC(NCc3c(C)cc(O)cc3)C2)=O)cc(F)c(F)c(Br)c1 C(C)(CCC(=O)N1CCOC(CCNC(c2cnn(C3CCC3)c2)=O)C1)SC c1(CCNC(c2n(CCOC)nnn2)c2cc(C3CC3)[nH]n2)cncc(C)n1 c1(C(=O)NCCOCCCNC(C(C)c2cccs2)=O)ccc2c(n1)OCCO2 c1(N(C)CC2CC(=C)C2)cc(NCCC2CCCCC2C)ncn1 N1(C(C2(COC)CC2)=O)CCCC(CN(C2CC(=O)N(c3cnn(C)c3)C2)C)C1 c1(CC)ccc(C(=O)NCC2(C(=O)NC3CCOCC3)CCC2)[nH]1 N1(C(C(c2ccccc2O)OC)=O)C2CCC1C(NC(=O)CN(C)C(C)C)C2 C1(C(N(CC(=O)NCc2occ(C)n2)C2CC2)=O)COCC(C)O1 N1(C(C(=O)Nc2cc(C3C(C)C3)oc2)=O)CCCN(CC(F)F)CC1 C(=O)(C(CC(C)C)N(C)C(C1OCCCO1)=O)N(C)Cc1ccc(C)cc1 CC1(C(=O)NCCC2CCCCN2C(c2ncc(Cl)s2)=O)CNC(=O)C1 Cc1cc(=NC(CCO)C2CC2)[nH]c(C)c1C#N CCC(C)C(=O)NC(c1ccccc1)C(=O)NCCC1(C)CCOC1 c1(N2CC(CC=C)(NC(C3CCCCC3O)=O)C2)nc2c(cc1C#N)CCC2 C#CCCCCC(=O)NCC1C2CN(C(C3CCC3c3nnc(S)n3C)=O)CC12 C=C(C)C1CN(C(C2CC3(CCN(C(c4nnn(CC)c4C)=O)C3)C2)=O)CCO1 C1(C)(C(N2CC(CSC)C2)=O)CN(C(C2(SC)CCC2)=O)C1 N1(C(C(C)N(C(C)=O)C)=O)CC2(CC2)CC1CC(N1CCCC(CN=[N+]=[N-])C1)=O Cc1ccc(C)c(NC(C2(NC(c3cc(C)c(C)[nH]3)=O)CC(CO)C2)=O)c1 C(=O)(NNc1cc(C)nc(F)c1)N1CCC2(CCC(CC(=O)OC)C2)C1 C1(OCC#C)CCN(C(=O)CN(C(=O)CCC=C(C)C)C2CCC2)C1 N1(C(c2c(C)nc[nH]2)=O)CCCCC1CCC(C)(C)NC(C1CC(C)CCO1)=O C12(NC(CC)=O)CCC(CC1)N2C(=O)C(=O)NCC(=O)Nc1ccc(C)cc1 C1(C)(CC(=O)NCC(C(C)(C)C)NC(=O)CCc2csc(=N)[nH]2)CCS(=O)(=O)N1 C=C(Cl)CCC(=O)NC1CCCN(C(=O)C(O)CN(C)C)C1 C1(C(=O)NC2CC(CCNC(CCOCC(C)C)=O)C2)CCc2nncn2C1 N1(C(C(C2CC(F)(F)C2)OC)=O)CCCN(C(c2c(C)noc2C)=O)CC1C Cc1cn(CC(N2CCC2(C)C(N2CCOC3CC23)=O)=O)c(=O)nc1O Cc1nc(C(=O)NC2C3CN(C(c4cc(C)c(Br)s4)=O)CC23)c(C)o1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC(CNC(C(CC)CC)=O)C(O)C1 CN1C(=O)Cc2cc(S(=O)(=O)N3CCCC3CCC(=O)N3CCC3)ccc21 CCC(C)CC(=O)NCc1cc(C(=O)NC(C)Cc2cn[nH]c2)co1 c1(NC(=O)NC2CC(C(F)(F)F)CN(C(=O)CO)C2)cccc2c1CNC2=O c1(NC)nc(C)ccc1C(=O)NCC1CCCN(C(=O)CCOCC(F)F)C1 C1(C(N(C(CC(=O)OC)C)C)=O)CCN(C(C23CCC(C2)C3)=O)C12CC2 c1(C(=O)NC(CNC(C2(C#C)CCCC2)=O)(C)CO)cncc2[nH]ccc12 N1(C(CC(C)C)=O)CC2CCCC2(CNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(=O)Nc2cccc(OC)n2)[nH]c2ccccc2c1-c1ccnc2[nH]ccc12 C1(C(=O)NC(C)(C)C)C2CC(CC2F)N1C(C1CC1C1(C2CCCCO2)CC1)=O C1(C(=O)NC2CC(C)(NC(CCc3cn(C)nc3)=O)C2)CCC(C)(C)OC1 N1(C(C(c2ccccc2)C)=O)CC2N(C(c3ncsc3C(C)C)=O)CCC2(C)C1 Cc1cccc(C(N2CCC(NC(=O)CC3CC(C(F)F)C3)C(F)C2)=O)c1Cl c1(SCC(N2CCCC(NC(C3CC4CC4C3)=O)C2)=O)ccc(F)cc1 C(CC)(CCCC(=O)Nc1ccc(F)nc1C)NC(C=CCCC)=O N1(C(C(C(C)C(=O)NC)C)=O)CCC2(COCC(CC(=O)OC)O2)C1 Cc1cc2c(C(N3CCCN(C(c4oc(C)cc4C)=O)CC3C)=O)nccn2n1 c1(C(N(C2CCN(C(c3csc(C(=O)OC)n3)=O)C2)CC#C)=O)coc(C2CC2)n1 N1(C(C(C)S)=O)Cc2ccccc2CC1C(=O)Nc1ccc(OC(F)F)nc1 N1(C(CCSCCCC)=O)C2CCCC1CC(NC(=O)CC1CCC3CC3C1)C2 S(=O)(=O)(c1c(C(F)(F)F)cccc1Cl)NC(C#C)C(C)(C)C c1(CC(=O)NC2C3CN(C(C4(C#N)CCCC4)=O)C(C3)C2)ccc2c[nH]nc2c1 C(=O)(CCCC(=O)OC(C)(C)C)NCC1CC(NC(CC(C)N(C)C)=O)C1 C1(C(=O)NC(C2CCCN2C(c2ccc(CCC#N)cc2)=O)C)CCCCNC1=O C1(O)(NC(CNC2C(NC(C(C3CCOCC3)OC)=O)C2)=O)CCOC1C c1(C(c2nnnn2CC(F)F)NC(c2ccnn2C)C)cc(Br)ccc1Cl c1(OCC(C)N(C(=O)C=Cc2ccco2)CC)ccccc1F c1(C(N(C2CCN(C(=O)C=CC(C)C)CC2)CC(C)C)=O)nnn2c1CCCC2 c1(C(N2CC(C)C(NC(c3nc(O)nc(O)c3F)=O)C2)=O)cc(Cl)cc(Cl)c1O N1CCCN(C(=O)C=C(Cl)Cl)C(C)C1.Cc1nc[nH]c1-c1cn(CCCC=O)nn1 CC(F)CC(=O)NCC(C)CN(C)C(C1(C(=O)OC(C)(C)C)CC1)=O c1(OC)ccc(Cl)cc1C(=O)NCCN(C(=O)C(Cc1ccsc1)NC=O)C(C)C C1(NC(C2C(C)C2)=O)CCCC12CN(c1cc(Cl)nc(CS(C)(=O)=O)n1)C2 c1(C(N2CCC(C(=O)OC)(CO)C2)=O)cc([N+](=O)[O-])n[nH]1 Cc1cc([N+](=O)[O-])cnc1NC1CCCC(CNC(c2cncn(C)c2=O)=O)C1 C1(OC)CCCC(OCCC(c2nccn2C)Oc2nc(-c3ccccc3)ns2)C1 c1(CSCC(C)C)ccccc1OC1(C)CC1.C1CC(=O)NN1CCCN(C)C CCCC(CC)C(=O)NCC(C)(CC(C)C)NC(=O)Cc1ccc2c(c1)CC2 c1(C(N(C)CCNC(c2cn(-c3ncccn3)cn2)=O)=O)ccnc(C2CC2)n1 c1(C(C(=O)NCC(CN(C(C=CC)=O)C)O)C)ccc(C(F)F)cc1 c1(C(=O)NC23CC(NC(C(C)NC(C)=O)=O)(C2)C3)ncnc2[nH]c(C(F)(F)F)nc12 c1(OCC)cc(OC(=O)N(C)Cc2c(Cl)cccc2Cl)ccc1Br N1(C(c2cnc(CC)s2)=O)CCOCC1CNC(=O)C(C1CC1)C1CC1 C1(C(=O)NC(C)CCN(C(=O)CCc2cncc(O)c2)C)CCC2(CCC2)O1 C(c1c(F)cccc1F)=CC(=O)NCC(CN(C(=O)CC1CCOC1)C)O N1(C(CN2CCC(C)C2)=O)C2CC=C(C(=O)NCCc3cscn3)C1CC2 CC1CON(C(=O)c2cccc(C3SCCS3)c2)C1 C1(C(C)C)(C(=O)NC(CNC(=O)C(C)(C)OC(C)(C)C)C2CC2)CCCO1 Cc1ccc(C(C)(C)C(=O)NCCC2(NC(C3CCC4CCC34)=O)CCC2)cc1 C12(C(=O)NCCC(C)NC(C3CCCN3CC(C)C)=O)CCC(N=[N+]=[N-])(CC1)C2 Cn1c(C(=O)NC(CNC(C2CCCC(O)C2)=O)CO)cc2sccc12 c1(C(=O)NCC(CO)NC(C(=O)NCCOC)=O)cnc(O)n1C N1(C(C=CC=CC)=O)CC2(CNC(c3occc3-c3ccccc3)=O)CCC1C2 c1(OCCCNC(c2c(SC(CC)C)ccnc2)=O)cc(C)cc(C)c1 CC(N=c1[nH]c2ccc(O)cc2s1)c1ccc(N2CCCC(C)C2)cc1 C#CCC(CC(=O)Nc1cc(CO)cc(F)c1)NC(c1ncoc1CC)=O C(=O)(CCCC(C)(C)C)NC1CCN(C(c2ccc(CC)c(C)c2)=O)C(C)C1 C(=O)(C(CNC(=O)Cc1cc(C)on1)CC1CCCC1)NCC(CC)C c1(C(N2CC(F)(CNC(C3(C)C(CC)CCC3)=O)C2)=O)cc(C)nnc1O C(CC(=O)N1CCC(CNC(CCOC)=O)(OC)C1)(C(C)(C)C)OC C=C1Cn2c(C(N3CCN(C(=O)C(C)CSC)C(C4CCCC4)C3)=O)nnc2S1 c1(CC(=O)NCC(CNC(C23CCCC2C3(F)F)=O)OC)ccc(C)c(Cl)c1 N1(C(CSCCC#N)=O)CCC(CF)(NC(C2CCCOC2)=O)C1 N#CC1CCCC(C(=O)NCCCOCCC(=O)NCC2CCS(=O)(=O)C2)C1 CCCCC(C)C(=O)NC1CN(C(c2cccc(C3CC3)n2)=O)CC1C CC(CCNC(=O)CC1CCCOC1)CCNC(c1cc(=O)n(C)o1)=O c1(C(=O)NCC2(C)CCCN2C(=O)CCF)ccc2c(Br)cccc2n1 c1(C(C(N2CCC(CN3C(=O)CCC3)C2)=O)=O)c(F)ccnc1F Cc1nn(C)c(C)c1CC(C)C(=O)NC(C)CC(C)NC(C1(C)C=CCCC1)=O Cc1nc(C)c(C(C)NC(=O)COC2CC(NC(=O)CCC3CCC(C)O3)C2)[nH]1 C(=O)(N=c1[nH]nc(-c2ccc(C)o2)s1)N(CC1CC(=C)C1)CC N1(C(c2ccc(OC)s2)=O)CCC(O)(CCNC(c2sc(C)cc2Cl)=O)CC1 c1(C(N2C(CNC(CCC(=O)N(C)C)=O)CC2)=O)cc2c(F)cc(F)cc2[nH]1 C1(CNC(CN(C)C(c2cccs2)=O)=O)CCC(NC(=O)CC2(C)OCCO2)C1 c1(C(=O)NC(C(C#C)(C)C)C)cccc(S(=O)(=O)N(CC)CC)c1 N1(C(C(NOC)=O)=O)CCN(C(C23COCC2C3)=O)CC(C)C1 C1(n2cc(C(C=C)(C)O)nn2)CCCN(C(=O)COCCN(C)C)CC1 CCCC(C)(O)CC(=O)N1CCC(CNC(C2CN3CCN2CC3)=O)C(O)C1 Cc1cccc([N+](=O)[O-])c1NC1CC(CNC(=O)CC2CC3(CCC3)C2)C1 c1(OC)nc(N2CC3CC2CN3Cc2nc(Br)cs2)ncc1F C1(CCC(=O)NCC2CCC2NC(=O)Cc2ccccc2)CCCC(=O)N1 c1(CC)cc(C(=O)NCCOCCNC(=O)CCC(C)c2ccccc2)ccn1 c1(C(=O)NC2CC2NC(=O)C(O)Cc2ccc(F)cc2)cccc2ncccc12 c1(N2CCC3(CC(NC(C(C)OCCC=C)=O)C3)C2)nc(C)cc(C)c1C#N C(CC(C)N=c1nc(N2CCC3(CC2)CC3C#N)c2ncccc2[nH]1)OC C1(C)(CNC(C2C(C=C)OCC2)=O)CCN(C(c2nocc2CC)=O)CC1 CN1CC(C(=O)NCC2CCCC(NC(c3cc(F)c[nH]3)=O)C2)CCC1=O C1(Cc2cn(CCCCCC)nn2)CCCN(C(=O)Cn2nc(C)nc2C)C1 C(=O)(CCCCCNC(=O)CC12CCCC1C2)NCC(C)(C)N(C)C C#Cc1ccc(OCC(=O)NC2CC(F)(CNC(=O)CCC3CC3=C)C2)cc1.CC c1(CC(=O)NCC(C)NC(CC2C(C)CCC2)=O)cccc(F)c1F C1(NC(CC2N(CC)CCC2)=O)COC2(CCN(C(=O)CNC(C)=O)C2)C1 c1(C(N2CCC(CNC(c3ccc(F)cc3)=O)C23CC3)=O)ccc2c(n1)CCO2 c1(C(N2CC(NC(C3CC(C)(C)C3)=O)C2)=O)cc(C(=O)CBr)ccc1O C1(C(CNC(c2c(C)ocn2)=O)F)CCN(C(c2c[nH]ccc2=O)=O)CC1 Cc1cc(C(=O)NC2CCN(C(=O)C(=O)NC3CC3)CC2C)c2c(O)n[nH]c2n1 N1(CC)CC(C(=O)NCC2(OC)CN(C(=O)C(C)(C)CC3CC3)C2)CCC1=O Cc1nsc(C)c1C(=O)NCC1CCN1C(=O)CC1CSCCS1 C1(CC(=O)NC(CC)CC(=O)NC2(C3CCCCO3)CC2)CCC2(CC2)CO1 c1(C(N2C(CNC(C(C)OC)=O)CC2)=O)nn(C(F)F)cc1Cl N1(C(c2ccc(C)nc2)=O)CCCOC(CCNC(C2C3CCCCCC23)=O)C1 c1(CNC(C2CCC(NC(c3csc(C)c3C)=O)C2)=O)nnc2n1CCC2 C(=O)(C(F)C(C)(F)F)NCC(C)(CO)OC.C12CC13CC(C3)NC2=O N12CCC3(CCN(C3)N(C)CC1=O)C2.c1(CN)cccc(Cl)c1.n1(CC)cccn1 [N-]=[N+]=Nc1ccnc(NC(C2CCN2C2CCCC2)=O)c1 c1(C(CNC(C2CNCC2O)=O)N(C)C)ccccc1Cl C1(C(=O)NCC(C2CCC2)NC(c2cncc(C)n2)=O)CCC(F)(F)CC1 N1(C(C(c2ccc(C)cc2)C2CC2)=O)CC2CC1CN2C(C1SCCS1)=O C1(CNC(c2c(C(=O)OC)scc2)=O)CCN(C(=O)CC(C)F)CC1C C1(C(=O)NC(CNC(C=NOC)=O)(C)CO)CC(C)(C)CCO1 Cc1cc(C2CC2)ccc1C(=O)NCC1CC(C)CCN1C(C1CCS1(=O)=O)=O C(CCCN=c1[nH]c2ccc(C(=O)OC)cc2s1)NC(C=CC=CCC)=O c1(CC)ccc(C(=O)NCCCCCCNC(C2CC2(F)Cl)=O)cc1Br Cc1cc(C)c(OCC(=O)NCC(CO)NC(C2(C)CCNC2=O)=O)c(C)c1 C1(COC)CC(CNC(=O)CCc2cc[nH]n2)N(C(c2cc(C(F)F)[nH]n2)=O)C1 Cc1csnc1C(=O)NCC(CO)NC(c1ccn(C2CC2)n1)=O C1(C(=O)NC(C=C)C2CCC2)CC=CCN1C(=O)C(C(C)OC)N(C)C C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)C(=O)N(C)C)C2(CCCOC2)C1 C(C(C)C)(C(O)C(=O)NCC(C)(C)CNC(c1cc(Cl)ccc1O)=O)OC c1(C(=O)NC2CC(CCNC(CNC(C3C(C)C3)=O)=O)C2)ncc(N)cc1Cl c1(C(=O)NCC(C)NC(CCNC(CC(C)C)=O)=O)cnc(Cl)c(F)c1N N1(C(C2N(C(Cc3c(C)n(C)nc3)=O)CC(=O)C2)=O)CC2CC1CS2=O C1(F)(C(=O)NCC(C=C)O)CCN(C(=O)CC(C)n2cccn2)CC1 C1(NC(c2n(CCOCC)nnn2)c2nocc2Br)CCOCC1OCC O=C(C1CCCc2nccn21)NC1CC12CCN(C(=O)CCOCC(F)F)CC2 c1(C(=O)NCCCCC(C)NC(=O)CC2COCCO2)ccc(Cl)c(Cl)c1N c1(OC)ccc(-c2nc(-c3nccn3N3CCOC3=O)c(C)o2)cc1OC C1(CNC(c2cc(C(F)(F)F)ccc2C(F)(F)F)C)CC(C)NC(=S)N1 Cc1csc(=NCC(=O)NCC(C)(C)CNC(c2cc[nH]n2)=O)[nH]1 C(C1=NOC2COCC12)CNC(COC1CCN(C(C(CCCC)O)=O)C1)=O C1(NC(C2N(C(=O)COCC3CCCC3)CC=C2)=O)CCCCC12CCC2 c1(CC)ccc(F)cc1C(=O)NC1CN(C(=O)C(C)C(C)CC)CC1CO C(=O)(C1CCCCc2ccccc21)NCC1(O)CN(C(Cc2cc(C)no2)=O)C1 c1(C(=O)NCC2CCN(C(C(c3ccc(F)cc3)CC)=O)C2)cccc(N)c1C C1(C(N2CC(N(C(c3cn(CC=C)nn3)=O)C)C2)=O)CN2CCN1C(C)C2 N1(C(C2C(=C)CC2)=O)CC2CC2(CNC(c2cncc(C(F)F)c2)=O)C1 c1(OC)ccc(CNC2CC2C(=O)NCc2cc(Br)ccc2F)c(F)c1F Cc1cc2ccc(C(=O)NC(CO)CCCCNC(=O)CCC3CC3C)cn2c1 c1(CC)oc(C(=O)NC2CC(CCNC(=O)C(c3ccccc3)C)C2)cc1C c1(C(N(C2(CC(=O)NC3CCNC3=O)CC2)C)=O)cc(O)ncn1 C(CCCC(=O)NC1CCC1NC(c1ccn(C(C)C)c1C)=O)SC c1(NC)cc(C(N2CCC(NC(c3nc(C)cs3)=O)C(C)C2)=O)cc(Cl)n1 C(C(CNC(C1(NC(=O)CCc2ccccn2)CC1(C)C)=O)C(C)C)OC c1(C(=O)NCC(C#C)CC)cccc2ccc(O)nc12 C1(NC(COC(CC)C)=O)CCC(CNC(c2nc(C(C)(F)F)cs2)=O)C1 C(CCC(=O)NC(C)CCNC(C)=O)N(C(=O)OC)C.C1(CCC(=O)N)CC(F)(F)C1 N1(C(C(C)NC=O)=O)CCC(C2(C(=O)N(CC(N)=O)C3CC3)CCOCC2)CC1 N(C(=NCCC(C)=O)NCc1cc(F)c(F)c(F)c1)C1CC(C)(CC)C1 C1(NC(C(C)n2cnnn2)=O)CCC(O)CN(C(=O)C=CC(F)(F)F)C1 N1(C(c2cc(C)nc(O)n2)=O)CC2CC1CCC2NC(c1cc(Cl)cc(Cl)c1)=O CC(C)C(C(=O)NCC(C)(C)CN(C(=O)C(O)C1CCC1)C)N(C)C c1(SC)cncc(C(=O)NC2COCC2NC(c2c[nH]c(=N)o2)=O)c1 N1(C(C(C)OC2CCOC2)=O)CCC(NC(=O)C2=CC(C)(C)C2)C2(CCC2)C1 C(=O)(CN(CSc1ccc(Br)cc1)N(C)Cc1ccco1)OC N1(C(C(n2ncc(C)c2)C)=O)CC2CC(O)C1C2NC(c1cccc(Cl)c1O)=O c1(CC(=O)NC(CC=C)CNC(=O)C(n2cc(Cl)cn2)C)n[nH]c2ccccc12 N1(C(C2C3COCC23)=O)Cc2ccc(F)cc2C1.CC12CCCN(C1)C2=O c1(C(=O)NC2C(CNC(c3c(OC)scc3)=O)CCC2)ccccc1C(N)=O c1(C(=O)NCC(CC)NC(C2CCCCC2(F)F)=O)cc(Br)c2occc2c1 c1(C(N2CCC(CC(C)NC(C(CC)OC)=O)CC2)=O)cc(N)c(Cl)cn1 c1(C(C(=O)NC)N(c2ccc(C(F)(F)F)c(C)c2)CC)ccc2nonc2c1 N1(C(C(CC(C)C)OC)=O)C2CCC1CC(CNC(c1cc(C(F)F)no1)=O)C2 C(=O)(C(CCOC)NC(=O)OC)NC(CC)CN(C)C CC1CN(C(C2CCS(=O)(=O)CC2)=O)CCN1C(=O)CN1CSCC1=O N1(C(Cc2c(C)occ2)=O)CCC(NC(=O)C=C2CCOCC2)C1(C)C CC(C)C1=NOC(C(=O)NCCCCC2CN(C(C3CC4C=CC3C4)=O)C2)C1 c1(OC(C(=O)N(c2c(OC)ccc(F)c2)C)C)ccc2c(c1)CCC2 C1(C(CO)NC(c2cccc(Cl)n2)=O)CCN(C(C2CC(O)C2)=O)CC1 C1(C(=O)NCC)CCC2CCCCN12.C123CC(C1)(C2)C1(CCC1)OC3=O CC(C)CC(C)CC(=O)NCC(C)(C)CCNC(=O)C=CC(C)(C)SC C1(C(N(C(CCNC(c2cnn(CCOC)c2C)=O)C)C)=O)CCC(C)(C)CO1 CC(C(=O)N1CCCC1CNC(c1cncc(O)c1)=O)P(C)(C)=O C1(NC(c2ccc(C)cc2O)=O)CC2CC1CN(C(=O)CS(=O)(=O)CC1CC1)C2 CCC(CC(=O)NCC1CN(C(c2ccsc2C#N)=O)C(C)(C)C1)C(F)F N1(C(=O)CCCc2ccc(O)cc2)CCC2C(CCCN2c2ccncn2)C1 C(c1cccc2ccccc12)=CC(=O)NC1CN(C(c2c(C)occ2)=O)C2C1C2 c1(NC(C(C)NCc2cn(CCOC)nc2)=O)ccc(Cl)nc1 N1(C(C(CCC)OC)=O)CCCC(NC(c2cnn(CCN(C)C)c2C)=O)C1C C1(NC(C(Cc2c(C)noc2C)C)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 S(=O)(=O)(CCC(=O)NC(CNC(=O)CN1CC=CC1)C1CC1)NC CS(=O)(=O)CC(=O)NC1CC(F)(CNC(=O)CC(c2cccs2)NC(N)=O)C1 Cc1nnc2n1CC(C(=O)NC1(CNC(c3cc[nH]c(=N)n3)=O)CCC1)C2 n1(CC=C)c(N(C(C)CCOC)Cc2csc(C)n2)nnc1COC c1(C(N2CC(F)(CNC(C(CC)=CCCC)=O)C2)=O)ccnc(Br)c1N C1(NC(C(c2ccc(Cl)s2)C)=O)CCC(C)(CNC(=O)C=Cc2ccoc2)C1 CCC(C(=O)N1CC(O)(C2CCCN2C(=O)COCc2ccncc2)C1)SC c1(OC)cc(C#N)ccc1-c1noc(-c2cc3scnc3[nH]2)n1 C1(C(N(CC)CC2CCCO2)=O)CCC(CNC(C2OCCC2C)=O)O1 C(C)(C)(CC(=O)NC(C1CCCN1C(=O)CC1(N2CCCC2=O)CC1)(C)C)OC N1(C(c2n(CC)nc(C)c2)=O)CCC2(CCC(NC(=O)CCCN(C)C)CC2)C1 N1(C(C2(SC)CCC2)=O)CCN(C(c2nn(C)cc2N)=O)C(C)C1 CC(C)C(CCNC(=O)C(C1CC1)N(C)C)NC(=O)CN1CC=CC1 C=Cc1ccc(NC(C2CCN(C(c3cc(C(C)C)n[nH]3)=O)C2C(C)C)=O)cc1 C(C(C)(C)C(=O)N(C(C)CC(N1CCCC(CC(C)(C)C)C1)=O)C)OCC CCCCC(CNC(=O)CCc1cccnc1C)NC(C1(C)CSC1)=O CC(CC(=O)NC1CCNC(=O)C1)C(C)(C)NC(c1cccc2cncn12)=O c1(-n2ccc(CC(=O)NC(C)C(CO)N(C)C)n2)ccc(F)c(F)c1 C1(O)(CC(=O)N(C(CNC(c2cncc(C)n2)=O)C)C)CCCN(C)C1 c1(NC2CCC(N(C)C(=O)Nc3ccc(Cl)cc3)C2)cc(F)ccc1N1CCCC1 C1(C#CC(=O)N2CCC(N(C(=O)CC(C)F)CC3CC3)CC2)(CC)CC1 c1(CN(C)C(C2CCCCCC2)=O)cccc(CNC(c2cc(Cl)on2)=O)c1 Cc1ccc(C=CC(N2CCN(C(=O)CCc3cn(C)cn3)CC2CO)=O)cn1 c1(OC)ccc(C(=O)NOCC(CCNC(C(=O)O)C(=O)O)OC)cn1 c1(C(=O)NC(c2ccc(CNC(C(CC)COC)=O)cc2)C)ccc(Cl)c(C)c1 C(=O)(C(=O)N=c1ccn(CCC(C)C)[nH]1)NC(c1nc(CC)[nH]n1)C C(CN=c1ncc(F)c[nH]1)C1(CO)CCN(C(=O)C(F)OC(F)(F)F)CC1 c1(NC(c2ccccc2)COC)[nH]c(=NC2CCCCCCC2)nc2scnc12 N1(C(c2c(CC)oc(C)c2)=O)CCC(OC)C(C)(C)C1.C1=CC=CCNC1=O c1(C(=O)NC(CNC(C2CCCN2C2CC2)=O)CO)cc(F)cc2ccncc12 C(=O)(CC1=CCOCC1)NCC1(F)CCC(NC(C(C(C)(C)C)OC)=O)C1 n1(CCC(=O)NC2CC(C)(NC(=O)CCC3CC3)C2)cc(C#N)c(O)nc1=O C(CC1=CCN(C(C2(CC3CC3)CCCO2)=O)CC1)NC(C=C1CCN(C)C1)=O C1(OC)CC2CC(NC(=O)C(CO)NC(=O)CCc3nncn3C)CC12 C1(CCN(C(C(F)=CCC)=O)C)CCCCN1C(=O)CC1CCC(=O)N1C c1(C(N2CC(NC(C3(C(F)(F)F)CCCCC3)=O)C(F)C2)=O)cc[n+]([O-])cc1 C1(NC(CC2CC(C)(C)N(C(C3C4CC(=O)CC34)=O)C2)=O)CCCCC12CCC2 c1(C(N(CC(C)NC(C2CCS(=O)(=O)N2)=O)CC)=O)noc2c1CCCC2 C1(NC(CC2CC(NC(C(C)SC)=O)C2)=O)CCc2n[nH]cc2C1 C1(C(N2CC(CNC(COC(CC)(C)C)=O)C2)=O)CCCCN1CC1CCCC1 C1(C(=O)NC(C(N)=O)CO)(NC(c2ncncc2Cl)=O)CC(F)(F)C1 CCCCS(=O)(=O)CC(=O)N1CC2CC1CN2C(c1[nH]nc([N+](=O)[O-])c1Cl)=O Cc1cccnc1C=CC(=O)NCC1CCN(C(=O)C=Cc2ncco2)C1 c1(CCC(=O)NCC(CC)NC(COC(CC)CC)=O)nc(C)c(C)[nH]1 N1(CC(=O)OC)CCN(C(C)=O)C(C)C1.c1(C(N2CC2)=O)ccc(C)cc1F c1(CC(=O)NCCCNC(CC2CCC(C)(C)CO2)=O)ncn2c1COCC2 C1(C2CCOCC2)(C(N2CC(c3cn(Cc4nc(C)sc4)nn3)C2)=O)CC1(F)F C(=O)(C1CCc2ccccc21)N1C(C=CC(NOCC2(C)CC2)=O)CCC1 C1(NC(=O)CC2CCCSC2)CCC2(CC1)CN(C(C1CN3CCN1CC3)=O)C2 c1(CC(=O)NC(CC=C)CNC(=O)C(C)O)cc(OC)ccc1OC Cn1nc(Br)cc1CC(=O)NC12CC(CNC(=O)COCC(F)F)(C1)C2 c1(NC(CN(CCNC(C2(O)CC2)=O)CC)=O)c(C)nc2ccc(F)cn12 CC1CCC(C)(C(N2CC(CN(C(=O)CCCC#N)C)C2)=O)C1 C1(C)(CC)CN(C(C(=O)Nc2ccccc2OC)C2CCOC2)CCO1 c1(SC(C)(C)C)ncc(C(=O)O)cn1.C123CC(C1)(C2)CNC3=O N1(C(c2cc(CCC)c(C)s2)=O)CC(NC(C2CC=CCO2)=O)C(C)(C)C1 N1(C(C(CC=C)N(C)C)=O)CCC2(CC1)CC2N(C(=O)C=C1CCC(C)C1)CC CC(C)C(F)C(=O)NCCC1CC(NC(c2csc(Br)c2Cl)=O)C1 N1(C(CC)C(N)=O)CCN(C(=O)CCC=CC(=O)N(C)C(C)C)CC1 C1(CNC(CCSCC)=O)(NC(=O)CN2CCCCC2C)CCCCC1 c1(C(N(C2CCN(C(C3C(C)C3C)=O)C2)CC)=O)cc(F)c(C)cc1Cl N1(C(c2ccc(OC)o2)=O)CC(NC(=O)CCc2ccc(C)nc2)CCC1C C1(C(N(C2CN(C(CC3(OC)CCC3)=O)C2)C)=O)CC(=O)CO1 c1(OC(C)C)nc(C(N2CC(CCNC(=O)COCP(C)(C)=O)C2)=O)cc(O)n1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)CC2C)csc2c(F)cccc12 C1(C#CC(=O)NC2CC(O)(CNC(=O)C3=CCCCC3)C2)(CC)CC1 N1(C(c2cc(C)n(C)c2)=O)CC2CCC(C1)N2C(=O)CSC1CCS(=O)(=O)C1 c1(C(N2CCN(C(c3cnsc3)=O)C(CC(F)(F)F)C2)=O)cc(Cl)c(F)cc1F N1(C(C=Cc2c(C)cccc2)=O)CCC2CN(C(c3cc4c(s3)COCC4)=O)C2C1 c1(NC(C2CCCC(N3CCCS3(=O)=O)C2)=O)ccc(CCN2CCCC2)cc1 c1(C(=O)NCC(CNC(c2n(CC)ccn2)=O)CO)ccc2ccsc2c1 C(=O)(C(CC)C(=O)N1CCCC1CNC(=O)C(C(C)C)N1CCCCC1)OCC C=C1CC(C(N2CCC2)=O)(CNC(=O)CNC(=O)OC(C)(C)C)C1.C1(Cl)(C)CCC1 C1(C(=O)NCC2(C(F)F)CCN(C(COCCC)=O)C2)CC2CCC(C1)O2 Cc1cnc(NC(c2cc(Cl)sc2Cl)C)c(S(=O)(=O)NCCN2CCCCC2)c1 c1(-c2n(CCC#C)c(N(C)Cc3ncc(C)s3)nn2)ccc(OCC=C)c(C)c1 n1(C(C)C)ccc2cc(C(=O)NC3CCN(CC4CC4(F)F)CC3)ccc12 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC(NC(C2CC3(CCC3)C2)=O)C(O)C1 Cc1cccc(-c2cc(C(=O)NCC(C)(C)CNC(=O)C(C3CC3)N(C)C)on2)c1 C12(C(=O)NCCCCCNC(C(C)O)=O)CC3(F)CC(F)(C1)CC(F)(C2)C3 c1(CC)cscc1C(=O)NCCC(C)N(C)C(c1cnc(-c2ccsc2)s1)=O CC1(C)OCCOC1C(=O)NCC1CCCCN1C(=O)C(c1ccc(Cl)cc1)=O C1(NC(C(C)=C2CCCC2)=O)C=CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(=O)NC(C2CCN(C(c3nc(COCC)sc3)=O)C2)C)c[nH]ccc1=N c1(C(N(C(C)CNC(C2(C(F)F)CC2)=O)CC)=O)ccc(Cl)cc1Cl C(C(C)CC(=O)NNC(=O)C(C)(C)CCCCNC(c1cc(C)n(C)n1)=O)OC c1(C(N2CC(CCNC(=O)Cc3ccsn3)OCC2)=O)ccc2n[nH]cc2c1Cl c1(OC)ccccc1NC(=O)C(C)N(C1CCN(CC2CC(O)C2)CC1)C C1(CC(=O)N(CCN(C(C)C)C(c2cnn(CCF)c2)=O)C)CN2CCN1CC2 N1(C(C2(OC)CCN(C(CC(CCC)C)=O)C2)=O)CCCCCCC1C C(C)(CCCN=c1cc[nH]cc1[N+](=O)[O-])NC(C1CC(CCC)OCC1)=O C1(C(N2CC(CCNC(=O)C(C)n3ccnc3)(OC)C2)=O)(CO)CCCCO1 C1(OC)CC(C(=O)NCc2ncsc2C)N(C(=O)C(C)COC(C)C)C1 c1(OC)ccccc1CCC(=O)NCC1CC(NC(C2CC(OC)C2)=O)CC1O Cc1c(C(=O)NCCN(C2CCC(CCC(=O)N(CCCO)C)C2)C)nnn1C N1(C(c2c[nH]c(=NC)o2)=O)CCC(NC(C2CN(C(=O)NC)C2)=O)CC(O)C1 C1(C(=O)OC)CCOC1C(=O)NC12CC(NC(c3cc(C4CC4)[nH]n3)=O)(C1)C2 c1(NC(CCNC)c2cccs2)cc(NCCc2cnn(C)c2)ncn1 CC1CCCCC1CC(=O)N(CC(O)CN(C(=O)CN(C1CCSC1)C)C)C CC1CCNCCN1C(c1cncc(O)c1Cl)=O.C(c1ccsc1)=CC=O c1(C(N(C2CCN(C(C=CCCC)=O)C2)CCC)=O)ccc(=O)n(O)c1 N1(C(CCC#C)=O)CCC2(CC2NC(=O)CN(C)CCO)C1 N1(C(c2c(N(C)C)nccc2)=O)CC2=C(C1)CN(C(=O)CCC1CCOC1)C2 C1(CC#C)(C(=O)NCCC2CN(C(=O)C(C)(C)N3CCCC3)C2)CCCO1 C1(CNC(c2n(CC)ncc2)=O)CN(C(C2(OC)CCC(C)(C)C2)=O)CCCO1 c1(OC)c(Cl)cc(C(=O)NC2CCCN(C(=O)CN3CC=CC3)C2)nc1Cl C1(NC(C(C)OCC)=O)(CF)CN(C(=O)COCC2CCC2)C1 c1(CC(=O)NCCNC(C2(C)CC=CCO2)=O)ccc([N+](=O)[O-])cc1Cl C1(CNC(COCCCC)=O)C(C2CC2)CCN1C(c1cc(Cl)ccc1C)=O c1(C(=O)NC(CC=C)CNC(C2CCCCS2)=O)cccc(N2CCOCC2)n1 C#CCCCC(C(=O)NC(C)(C)CC)N1CCC(OCCN(C)C)C1 c1(NC(C(=O)NC(CC)Cc2ccc(Br)cc2)=O)ccc2c(c1)CCCN2C N1(C(=O)CCc2ccc[nH]2)CC2CCCC2(C(N2CC(F)(C3CC3)C2)=O)C1 Cc1nc(NC2CCCc3n[nH]cc32)c(Cl)cc1C#N.C(=O)(C(F)(F)F)NCCC(=O)O N(C1CCc2cccnc21)C(C(CC(C)(C)C)NC(=O)CC1CC(F)C1)=O C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(c2cocn2)=O)C1 c1(C(CNC(c2c(CC)ncs2)=O)NC2(CO)CCCC2)cccc(OC)c1.OC C1(O)(C(=O)NCCOCCNC(Cc2nc(C)oc2)=O)CCC(C)CC1 N1(C(c2cc(C)sc2C)=O)CC(C2CC2)(C(=O)NCCc2ccncc2)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C)CCN(C(C(COC)C)=O)C1 CC1(CC(=O)NCCC2CCCCC2)CCN(C(C2CCCO2)=O)CC1 C(=O)(C(CCC1CC=CCC1)N1CCN(c2ccc(OC)nn2)CC1)NCC=C C1(NC(C(C2CCC2)OC)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC1 c1(CC(=O)NC2C(CNC(CCSCCCC)=O)CC2)c[nH]c2ccc(F)cc12 C=CC(CC)CC(=O)NCc1nc(CNC(C23CC(OC)C2C3)=O)cc(O)n1 C1(N(C(=O)CCNC(=O)CO)C)COCCN(C(C2CC(=O)NC2(C)C)=O)C1 C1(NC(COCCC#C)=O)CC2CC(C1)N(C(=O)C=CC(c1ccccc1)=O)C2 c1(C(=O)NC2CN(C(C=CC(=O)OCC)=O)CC2O)cc2scc(Cl)c2[nH]1 c1(C(=O)NCC(CO)NC(c2c(C(C)(C)C)con2)=O)ccc(F)c(Cl)c1F C1(C(=O)NC(CN(C(c2c(OC)ccc(C)n2)=O)C)(C)C)CCC2(C1)CC2(F)F c1(C2N(c3nnc(CCC)n3CC)CCC2)cccc(F)c1 C1(NC(C2(OC)CCSCC2)=O)CCN(C(=O)CC2CCC3CC23)CC1(C)C CC(C)S(=O)(=O)CC(=O)N1CCC1c1cn(-c2cncc(OC(C)(C)C)c2)nn1 CN(C1CCc2c(F)cccc21)C(C1CC(=O)N(C2CCCC2)C1)=O C1(CNC(CNC(CC)=O)=O)CC(C)(C)CCC1NC(=O)CN(CC)CC C=C(C)CC(C(=O)NC1COCC1C(=O)NC1CCC1(C)C)OC CC(C)C(F)(CNC(C1C2CC(=O)CC12)=O)C(=O)NCc1cccnc1O c1(C(N2CC(C)(C)C(NC(C3CCOC3)=O)C2)=O)cc2cc(Br)cn2cn1 C1(NC(C(C)SC)=O)CN(C(c2c(C)nc(C)n2O)=O)CC2(CCC2)C1 C1(C(=O)NC(C)CCCNC(=O)Cc2cc[nH]c2)CCCN(CCC2CC2)C1 C(=O)(C1=CCSC1)ONC(C1(C)CC(NC(c2ccccc2)C)C1)=O N1(C(c2cnc(-c3c(F)cccc3F)s2)=O)CCc2cc(O)ccc2C1 C1(O)(CCNC(C2CC(=O)NC2)=O)CCCN(C(c2cncc(O)c2)=O)C1 CCC(CC(=O)NCC1(C(=O)NCC(=C2CCCCC2)F)CCCO1)OC(C)=O C1(C(N(C)CC2CCC2)=O)CCC(n2cc(Cc3cnc(C(C)(F)F)s3)nn2)C1 C1(NC(CC(C)(C)C)=O)CCC(C)(NC(=O)Cn2ccnn2)CC1 CCCC(CCC)CC(=O)N1CCC(NC(=O)CCN2CCCS2(=O)=O)C1 c1(OC)cc(C(=O)Nc2cnc(Cl)c(CO)c2)c(-c2cncn2C)cn1 N1(C(c2cnn(CC)n2)=O)CC(NC(c2cncn2C(C)C)=O)CC(F)C1 C1(C(=O)NCCC2CCN(C(C(CSC)(C)C)=O)C2)CCCC1C1CC1 N#Cc1ccc(F)c(NC(C2CCCC2NC(=O)CCc2ncc[nH]2)=O)c1 N1(C(C(CCOCCO)NC(C(CSC)(C)C)=O)=O)CCCN(C)CC1C c1(C(=O)NC2CN(C(CC3C(C)(C)C(O)C3)=O)C2)nncc2c1CCCC2 C1(CNC(C(C)SC)=O)CCCN(C(=O)C=Cc2ccsc2C(F)(F)F)C1 C(=O)(CCCC(O)c1ccccc1)NC(C1CCCN1CC1CCOC(=O)N1)C C(=O)(CC(C)(C)C(F)F)N1CCC(N(C)C(C2C(=O)NCC2(C)C)=O)CC1 C(C(C)CC(=O)N1CCC(C(=O)NCCc2n[nH]cc2C(=O)OC)C1)OC c1(NC(CCN(C)Cc2ccncc2)=O)cc(C#N)ccc1F c1(CCC=C)ccc(C(=O)NCC=CCNC(C2CN(C)CC2C)=O)cc1 c1(C(=O)NCc2cc(C(N3CCC(O)(CC)C3)=O)sc2)ccc(C)c(O)n1 C(=O)(C1CCCn2c(C)nnc21)N1CCC(C)(NC(c2nn(CC)c(O)c2)=O)C1 CC12CN(C(=O)CN3CCOC3=O)C(C(=O)NC3(C(=O)C4CC4)CC3)(C1)C2 c1(C(=O)NC(C)CC(=O)NCCC2CCCC2)cc([N+](=O)[O-])c[nH]1 N1(c2nc(N3CC(C)C(N(C)C)C3)nc3c2ncs3)CCC(C)(O)C(C)(O)C1 N1(C(C(CSC)O)=O)CCCCC1C1(NC(c2cccc(F)n2)=O)CC1 Cc1ccc(Br)c(C(=O)NCCCC(C)NC(=O)COCCC(C)C)c1 N1(C(c2cnnc(Cl)c2)=O)CCCC(C2CCN(C(c3cc(Cl)on3)=O)C2)C1 C1(NC(c2ccnc3cc[nH]c23)=O)CN(C(=O)CC2=CCOCC2)CC2(CC2)C1 C(=O)(C(C)(C)C(C)(F)F)NCCC(C)N(C(C(C)OCCC=C)=O)C C1(NC(c2cc(C)c(Br)o2)=O)C2CC1CN(C(C1CCSCC1)=O)C2 c1(C(=O)OC)csc(C(N2CC(C)C(F)C2)C(=O)NCCCSC)c1Cl Cc1ccccc1CC(C)C(=O)NCC#CCNC(C1(C(=O)NC2CC2)CC1)=O C1(NC(C(C(C)C)NC(C)=O)=O)CCN(C(=O)Cc2cc(C)cc(C)c2)C(C)C1 C1(NC(c2nc(COC)sc2)=O)CC2CN(C(=O)C(F)(F)C3(O)CCCC3)CC12 CCCC(CNC(=O)CCc1csnn1)NC(C1CCN1C)=O Cc1ncc(CNC(=O)C(C)CN(C(=O)C(=C2CCCCC2)F)C)o1 N1(C(CC2CCCC(NC(C=CC(CC)C)=O)C2)=O)CCCC2(CCC2)C1 C1(CNC(C2C(C)=C2)=O)(NC(=O)Cc2cnco2)CCC1 C1(NC(c2ccc(OC)s2)=O)CC(NC(=O)C=CSC)C12CCC2 Nc1c(C(N2CC(CNC(=O)Cn3cnc4ccccc34)C2)=O)cc(F)cc1Cl C12(N(C(C3CN(C(C4C(C)(C(C)C)C4)=O)C3)=O)Cc3ccccc3)CC(F)(C1)C2 c1(C(N2CC(CC)N(C(c3ncnc(O)c3Cl)=O)CC2)=O)ccc2snnc2c1 CCC(C)CCCCC(=O)NCC1CCC2(CN(C(c3c(Cl)cnn3C)=O)C2)O1 C=CC1CCN(C(=O)CC2CC(F)CN2C(=O)C(C)NC(=O)NC)C1 C=CCCCCC(=O)N(CC(CC)NC(=O)COc1ccccc1C(C)C)C C1(C(N(CCSC)C)=O)CSCCN1S(=O)(=O)Cc1cccc(C)c1 C1(C(=O)NCC2(F)CC(NC(c3c[nH]c(=N)o3)=O)C2)CS(=O)(=O)CC(=O)N1 C1(C(N(C2CN(C(c3cccc(OCC(F)(F)F)c3)=O)C2)C)=O)CCC(C)(C)C1 CC(C)CC(C(=O)N(C(C)C(=O)NOC1CCOC1)C)C(N)=O n1(C(C)C)ncc(Br)c1CC1CC1.[nH]1nnn(C2CCCC(CC3CC3)C2)c1=O C#Cc1ccc(Br)c(C(=O)NCC(C)NC(C2CCN(C)S2(=O)=O)=O)c1 C1(CC)(NC(=O)CC(C)(C)C)CCCN(C(C2CC2c2sccc2C)=O)C1 C(=O)(N=c1cc[nH]cc1F)C1CCCC(NC(c2cccc(O)c2O)=O)C1 N1(C(CC(C)C(F)F)=O)CC(CNC(c2cn3c(n2)CCC3)=O)CC12CCC2 N1(C(C(C)=CC)=O)CC2CCOCC2(NC(=O)CCCc2ccsc2)C1 CCCC(C)(O)CNC(C1(CCNC(=O)Cc2coc(C)n2)CCC1)=O c1(N2CC(c3c(NCC4CC(OC)C4(C)C)nco3)C2)ncc(C#N)cc1Cl c1(C(N2CC(C(C)NC(C3CS(=O)(=O)C3)=O)OCC2)=O)ccc2nc[nH]c2n1 N1(C(CC2(C)CCCC2)=O)CCCC(C)(CNC(C2CC23CCCC3)=O)C1 c1(C(N2CC(NC(CC(C)n3cccc3)=O)CC2(C)C)=O)ccc2occc2c1 c1(C(=O)NC2CC(CNC(C3(COC)CC=CCC3)=O)C2)c(N)ccc(C)c1F NC(=O)CCCCC(=O)NC1CCC(C(=O)NCCCNC(=O)C2CC2)CC1 N1(C(C(CC2CC2)OC)=O)CCC2C(NC(c3cc(C(C)C)no3)=O)C2C1 S(=O)(=O)(c1c[nH]ccc1=NCCC1CCCC1(F)F)NCCN=S(C)(C)=O Cc1cnc(C(N2CC(C(=O)NCC(F)Cl)C(C)C2)=O)c[n+]1[O-] c1(CNC(CC2OCCN(C(c3c(CC)cns3)=O)C2)=O)cnc2n1CCC2 C(=O)(C#CC1CCOC1)Nc1c(C)cc(NC(C2C3CC4C(C3=O)C24)=O)cc1 C1(C)(N(C(CC(C)n2cccn2)=O)CC(=O)OCCC2(O)CCCC2)CCSCC1 CN1CCCC12CCN(C(=O)CCC(C)(C)NC(=O)COC1CC1)C2 C(=O)(C1=NOC(C)(C)C1)NCC1CC(C)N(C(c2ccsc2Cl)=O)C1 n1(CC(=O)NC2C(NC(C3(C)CCC3)=O)CCC2)cc([N+](=O)[O-])cn1 N1(C(c2cn(C)nc2)=O)CCC(NC(=O)CCc2nc(O)n[nH]2)C12CCCC2 c1(C(=O)NCCN(C(=O)CC2CC(C)(C)OC2=O)C(C)C)ccc2cnoc2c1 C(=O)(CCCCCS(N)(=O)=O)N1CC2(CN(C(c3c(C)c(N)ccn3)=O)C2)C1 CC(C)CCCC(=O)N1CCCC1CC(=O)N(CCO)CC1CC1 C=C(F)C1(CC(=O)NCC2CCC(N(C(=O)C(F)=CCCF)C)CC2)CCC1 CC(c1cnn(C)c1)=CC(=O)NCC1CC2(CC2)CN1C(C1CCCS1(=O)=O)=O N1(C(C(C(=C)C)(C)C)=O)CCCC2(C1)C(NC(=O)Cc1occc1C)CCN2C C1(C(=O)NC(C=C)COC)CCCN(S(=O)(=O)CC2CC2)C1 C1(NC(C2CCC(C)O2)=O)COC2(C1)CN(C(c1cc(Cl)on1)=O)C2 C1(NC(C2(F)CCN(C(C3(C#N)CCCO3)=O)C2)=O)CC12CCOCC2 c1(C(=O)NC2(CC=C)CCN(C(=O)COCC(C)C)C2)cncc2cccnc12 CC(C)(C)CC(O)C(=O)NCC1(F)CC(NC(=O)CC2CCCC2(F)F)C1 C1(=O)C(CC(C)C)NC(=O)CC2CCN12.c1(CC)onc(C)c1CC CC1CN(C(=O)CN(C)CCO)CC(C)C1NC(c1cc2sccc2s1)=O Nc1ccc(-c2noc(-c3cnc(-c4cccs4)o3)n2)c(Br)c1F c1(C(N2C3CC(CNC(c4c(C)ccs4)=O)(OC3)C2)=O)cnn2c1OCC(C)C2 CCC(C)(C)CCCC(=O)OCC(N=[N+]=[N-])C(=O)OC(C)(C)C N1(C(=O)NCCCc2ccc(F)cc2)CC2CC(O)CC(C2)C1 C=CC1(CC(=O)NCC2(F)CC(NC(=O)CNC(=O)CNC(=O)OC)C2)CCC1 C(=O)(CCC(CF)CF)N1CCCCC(C(N(C)Cc2cncs2)=O)C1 c1(C(N2CCC(O)C(CO)C2)C(=O)NCCCC)ccc2cccnc2c1 C1(NC(C2(NC(C(C(C)C)C3CCC3)=O)CC(F)C2)=O)CCC(C2CC2)C1 C(N(C)N1CCN(S(C)(=O)=O)C2(CCCC2)C1)c1ccc(SC)cc1 C(CC(C)C)(C(C(=O)NC1CCOC1)N(c1ccco1)Cc1nc(C)no1)OC CCCC(C(O)C(=O)NCCN(C(C)C)C(C)C)NC(=O)C(F)OC(F)(F)F C=CCC(C)(C)C(=O)NCCC1(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1 c1(C(CC2(OC)CCC2)=O)ccc(S(=O)(=O)Nc2ccn3nccc3n2)cn1 c1(C(=O)NC(C2(O)CN(C(c3c(C)nsc3N)=O)C2)C)csc2cc(Cl)cnc12 C1(N(c2cnn(C)c2)CC)CCCN(C(=O)C(N)=O)CC1 c1(C(N2C(CNC(=O)Cc3ccc(F)cc3C(F)F)CC2)=O)n[nH]c2c1COCC2 C1(C(=O)OC)CC2(CCCC2)CN1C(c1cc(Cl)cc([N+](=O)[O-])c1)=O C12(CNC(c3ccc[nH]3)=O)CC(C1)C(NC(C1CCCC(F)(F)C1)=O)CO2 CCC(N=c1cc(C)c(C#N)c(C)[nH]1)C1CCOC1.c12ccccc1NS(=O)(=O)C2 CN1CCC(=CC(=O)NCCC(O)CNC(c2ccccc2C(F)(F)F)=O)CC1 c1(C(=O)NCCC(C)(C)NC(c2cccnn2)=O)ccc2sncc2c1 N1(C(C2(OC(C)C)CCC2)=O)CC(NC(c2scnc2Cl)=O)CC(O)C1 c1ccc(F)cc1[N+](=O)[O-].N1(c2nc(=N)s[nH]2)CCNC(CC(F)(F)F)C1 CC1S(=O)(=O)CC1C(N1CCC(N(C(=O)CCc2cnc[nH]2)CCO)CC1)=O C1(NC(COCC)=O)CCC(N(C)C(c2c[nH]c(C(=O)OC)c2)=O)C1 C1(CNC(=O)CSC(F)F)CC(C(=O)NCCCc2cnccn2)=NO1 C(CC(C)C)(C(=O)NC(C)C(=O)NCC(C)(C)C(N)=O)OC C1(C(=O)OC)CN(C(C2CCCCC(c3ccccc3)C2)=O)CC(C)O1 c1(N2CCCC(NC(c3cscc3Cl)=O)CC2)ncnc2cccc(F)c12 N#Cc1ccc(CC(=O)NCC2CCN(C(=O)C3=CCCC3)CC2)c(F)c1 c1(N2CC(N(C(C=C(C)c3cccs3)=O)C)C2)cc(C)nc(CC2CC2)n1 CC(=O)n1cc(CN2CCSC(C(=O)Nc3nnc(C)o3)C2)c2cccnc12 n1(CCCC)nc(C(=O)NC2CC2CSc2ccccc2)c2ccccc2c1=O N1(C(CN2CCC(OC)C2)=O)CCOC(C)(CNC(c2ncc(C)cc2F)=O)C1 Cc1ccnc(C(=O)N(C2CCC(NC(=O)COCC3CCCC3)C2)C)n1 c1(C(=O)NC(C(=O)NCC(=C)CC)COC)cncc(F)c1C CC1(C)C(CNC(C23CCC(C2)C3)=O)CCN1C(c1cc(O)cc(F)c1)=O C(=O)(CC(C)(C)CC(=O)N1CCN(C(=O)CCCCCF)CC1CCO)OCC C1(C(=O)NCCCN(C(=O)CC2COCC(C)O2)C(C)C)C2(CC2)C12CC2 Cc1ncnc(O)c1C(=O)NCC1CC(C)(C)CN1C(c1ccoc1)=O C1(NC(=O)Nc2cc(C(C)C)no2)CC(=O)N(C(c2ccccc2)C)C1 N12CC(C)(C1)OCC2=O.C1(CC(=O)N(C2C(N(C)C)CC2)C)COCC1O N1(C(C(C)C)=O)CC(NC(=O)C(C)CC2CC2)C(C)C1 C1(NC(C2CNCCN2Cc2ccc(F)c(Cl)c2)=O)CCc2ccccc2C1 O=C(C1=C(Cl)CCCC1)NCC1(CNC(=O)C2CC2)CCCCC1 CCC(CC)CC(=O)NCCCOCCNC(=O)C(C)C(C)c1ccc(Cl)cc1 C(=O)(CC(F)(F)CC)N1C(C(=O)NCCOCC=C)CSCC1 N1(C(C2CN(C(N(C)C)=O)C2)=O)CC2CC1CCC2NC(c1ncc[nH]c1=O)=O CC(CCC(=O)N(C)CCN(C(=O)Cn1cnnc1O)C)N(C)C CC(CS(C)=O)C(=O)N(C)CCNC(C1(CCF)CCOCC1)=O Cc1c[nH]cc([N+](=O)[O-])c1=NC1CCN(C(c2cnn(CC(F)(F)F)c2)=O)C1 N1(C(C=CC)=O)CC=C(C(C)(C)C(=O)N2CC(CSC)C2)C1 CC12CCC(n3cc(CNC4(N)CC4)nn3)(CO1)C2 C(CN=c1cc(Cl)nc(CS(C)(=O)=O)[nH]1)(N(C(C1C(C)OCC1)=O)C)C1CC1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC(C1)C2NC(=O)C(C(C)C)n1cnnn1 c1(C(=O)OC)ccc(S(=O)(=O)NC(C)Cc2ccccc2Cl)c([N+](=O)[O-])c1 c1(OC)cc(C(=O)NC(C)CCNC(=O)C(C2CCCCC2)O)cc(N)c1O N1(C(c2scc(COC)c2)=O)CCC(NC(=O)CCCSC)C(F)(F)CC1 N1(C(CC2C(C)C2(F)F)=O)C2CCC1CC(CNC(c1nnc(S)n1C)=O)C2 C1(C(=O)NC2COCCN(C(C(C(CC)C)OC)=O)C2)CN2CCN1C(C)C2 C1(C(CCC)NC(=O)C(O)Cc2[nH]cnc2C)CCN(C(=O)COC(C)=O)CC1 C1(NC(C(CC)SC)=O)CCCC1(C)NC(=O)CCn1nc(C)nc1C c1(-c2nc(NCC(=O)Nc3nnc(CCCC)s3)sc2)ccccc1F n1(CC(N2CC=CC(NC(CCC(C)OC)=O)C2)=O)cc([N+](=O)[O-])nc1C C1(NC(CSCCC)=O)C(C)(C)CN(C(c2cn3ccccc3n2)=O)CC1(C)C C1(C(C)C)CC(C(=O)N(C2CN(C(=O)CC(O)Cc3ccccc3)C2)C)CCO1 N1(C(C=Cc2ccc(C)s2)=O)CC2CCN(C(C3CC3c3ccnn3C)=O)CC12 N1(C(c2cc(C)n(CCO)n2)=O)CCN(C(c2ccsc2)=O)CC1CS(C)(=O)=O C1(F)(C(=O)NCc2cnc(CNC(=O)OC(C)(C)C)s2)CCCOC1 Cc1nn(C)cc1CCC(=O)NCC1C2CN(C(C3CCCN3C(C)C)=O)CC12 N1(C(CC2(C=C)CC2)=O)CC(C)CN(C(c2ccc(C)nc2OC)=O)CC1C CCCCC(C)C(=O)N1CC(C(=O)N(CC(C)C)CCOC)C2(CC2)C1 N12CCC(CC1)N(C(N)=O)C1(CC1)C2=O.C1(CC2CC2)CCN(C2CC2)C1.CC=O CC1CN(C(=O)C(O)C(C)(C)C)CCCN1C(C1CCN(C2CC2)CC1)=O Cn1cc(NC(=O)CC2(CNC(c3cccc4c[nH]nc34)=O)CC2)c(O)nc1=O C(=O)(C(CCC(C)C)NC(=O)C(F)C1CCC1)NCc1cccc(CC)c1 C1(O)(CCNC(=O)COc2ccccc2)CCCN(C(c2cccc(=O)o2)=O)C1 N1(C(C2(CC)CCCC2)=O)CCCC(CCNC(=O)C(c2cnn(C)c2)OC)C1 C1(C)(CN(C2(C3CCCO3)CCC2)C(C)=O)COCCN(C(C2CCOCC2)=O)C1 C1(CNC(C=CSC)=O)CCCC2(CN(C(c3n[nH]c4c(C)cccc34)=O)C2)O1 N1(C(CC(CC)C)=O)CCC2(CCC2NC(c2ccc3n[nH]cc3c2Cl)=O)CC1 c1(C(N2C3C(NC(CCCc4c(C)ccs4)=O)C(C3)C2)=O)cc(C)c(N)cn1 CC1(CNC(c2cccc(C3(O)COC3)c2)=O)CCCN1C(=O)Cc1ccsc1 c1(NC(C2N(C(c3c(CC)ncs3)=O)CCC2O)=O)ccc(Br)cc1I c1(C(=O)NCC(CNC(c2nc(C)oc2)=O)(C)C)cc(S(=O)(=O)N(C)C)c[nH]1 N1(C(Cc2c(C)cccc2)=O)CCCCC(NC(c2c(O)cccc2Cl)=O)C1 c1(C(=O)NC2CC(CC)NC2)cc(-c2cccc(F)c2)n(C)n1 CCC(C)(CC)C(=O)N(C)CC1CCCN1C(c1ccc(O)c(C(C)C)c1)=O N1(C(c2c(CC)scc2)=O)CCCC2(NC(c3cn(C4CC4)nn3)=O)CC2C1 C1(C)(C(=O)NC(CCC)CO)C=CCN1C(c1cccnc1C)=O c1(CNC(=O)C=CC2CC2)ccc2c(c1)CCC2NC(=O)C1CCc2c[nH]nc21 c1(OC)ccccc1-c1ncsc1C(=O)Nc1nc(-c2ccoc2)nn1C C1CCCCCN1C(C1(N(C)C)CCC1)=O.C1(CC(=O)OC)(N(C)C)COC1 N1(C(CCC(C)OC)=O)CCC(C)(C)C(C(=O)NC(C)(CO)CO)C1 c1(C(=O)NCC(N2CC(COC)C2(C)C)=O)ncnc(O)c1F c1(C(=O)NC)cccc(C(N2CC=CC(NC(=O)C3=COCC3)C2)=O)c1 C1(CC(N2CC(C)C(NC(C3(O)CCOC3)=O)C2)=O)CCC2(CC1)CC2 N1(C(C(CCC)C)=O)CCC(CNC(C2CC2C(F)(F)F)=O)C12CCC2 N1(CCNC(C)=O)CCC2(CN(C(=O)Cc3ccnn3C)CC(C)O2)C1 CC(C)C(F)C(=O)N1CCOCC1CC(=O)NCCCC(C)(F)F Cc1cc(Br)cc2cc(CN3CCC(C)(C(=O)O)C3C)oc12 C1(C(=O)OC2CCN(C(=O)OC(C)(C)C)CC2)(OC)CC2(CN(C(C)=O)C2)C1 Cc1ncn(C)c(=O)c1C(=O)NCCC(C)CCNC(c1cc(O)cs1)=O N1(C(c2c(C)nco2)=O)CCC(O)(CCNC(=O)CCC2CCCN(C)C2)C1 C1(CN(C(COCC(=C)C)=O)C)CCCN(C(=O)COC2CCN(C)CC2)C1 N1(C(C(CC)C#N)=O)CC2CCN(C(C34CC(C(F)F)(CO3)C4)=O)CCC2C1 c1(-c2scc(CC(=O)NC(C3CN(C(C=CSC)=O)C3)C)n2)ccc(F)c(F)c1 C1(CNC(C(F)OC)=O)CCC2CN(C(=O)Cc3cnn(C)n3)CCC2C1 n1(CC(=O)N(C2CCN(C(=O)Cc3c[nH]nc3C)C2)CCC)cc(F)ccc1=O N1(C(c2[nH]c(C)cc2C)C(=O)NCc2ccc(OC)cc2)CCN(C)C(=O)C1 C1(C(N2CCN(S(C)(=O)=O)CC2)=O)CN(C(=O)Nc2ccncc2)CC(F)(F)C1 c1(N(C)C)ncccc1CNC(N1CCCC1c1ccc(Cl)cc1)=O CC(C)CC(Cc1ccccc1)C(=O)NCCCC(c1nnnn1C)NC1CC1 c1(C(N2C(CCNC(=O)CCc3cccc(F)c3)CCC2)=O)ccnc(CO)c1 C12(C(N3CC(CNC(c4ccc(-c5ccc(C)s5)s4)=O)C3)=O)CC3CC1C2C3 C1(NC(c2cnn(C)c2N)=O)CC2(C1)CN(C(C1CCC1C(C)(C)C)=O)C2 C1(O)(CC(=O)N(CC(CC)NC(=O)CSCCCN(C)C)C)CCCN(C)C1 CCCCC(C(=O)NC1CCCC(O)C1)NC(=O)COCCC1CC1 C1(C(N(C2CC(NC(C3(CO)COC3)=O)C2)C)=O)CN(S(=O)(=O)N(C)C)CCO1 C1(CNC(c2cncc(C(F)F)c2)=O)C2CN(C(=O)COC3CCCOC3)CC12 C(=O)(CC(C)(C)CC)Nc1ccc(CC)nc1.C12CCOCC1Cc1cn2nn1 N1(C(c2c(C)nc[nH]2)=O)CC(C)CCC1CNC(C1(C2(O)CCC2)CC1)=O CCCC(C)(C)C(=O)NCC1CN(C(C2C3CCC23)=O)CC1C C1(NC(CN2C(=O)C(F)(F)C23CCC3)=O)CCCC1SC.C(c1ccco1)=CC CCCC(F)C(=O)NCC(F)CC(=O)N(C(C)CO)C C(C)(CNC(C1CCOC1C(C)C)=O)(CC(C)C)NC(c1c(CC)csc1)=O C(CCNC(c1cccc(=O)o1)=O)(C(=O)NCC1COCCO1)OC c1(C(=O)NCC(CNC(c2ccc(CC)s2)=O)F)cc(C)nc2c1CCCC2 C=CCCC(C)(C)C(=O)NCc1nc(C(=O)NC(CN2CCCC2)CC)co1 C(=O)(C(F)C(=O)NCCCC1CCCCN1C(c1c[nH]c(Br)c1)=O)OCC C(C(=O)N)(C(C)CC(C)(C)C)N(CC(=O)C(C)=O)C.C(C)(C(=O)OC)CN c1(C(N(CCNC(C(COC)O)=O)C(C)C)=O)cnn(-c2ccc(F)cc2)c1C c1(C(N2CCN(C(c3cc(C)c(C)[nH]3)=O)C(C)C2)=O)nn2cccnc2c1Cl c1(C(C(=O)NC2(CN(C)C(C3CC34CC4)=O)CC2)C)ccc(Cl)c(Cl)c1 c1(N2CCCC(CCNC(c3cc(F)cnc3O)=O)CC2)ncnc2c1COC2 N(C1CCCn2ccnc21)C(C(CC=C)CNC(=O)C(C(C)C)NC(C)=O)=O N1(CCC(N2CCC(C(=O)NCCCO)CC2)=O)CCCS1(=O)=O c1(C(=O)NCC(CC)(CC)NC(=O)CC2CC2(Cl)Cl)ccc(NC)c(F)c1 CC(C(=O)NC(CC1CC1)C(=O)N(CC(C)(C)C)C)S(C)(=O)=O Cc1c(C(=O)NC(CNC(=O)CCC2CCOC2)C2CC2)ccc(Br)c1F C(C(=O)N1CC(NC(=O)CCCN(C)C(=O)OC)C1)(C(C)C)OC c1(CCNC(C(CSCC)NC(c2cnccn2)=O)=O)ccc(F)cc1 CCCCC(C(=O)NCC1(CNC(=O)C(n2cc(C)cn2)C)CCC1)C(C)C c1(C(N2CC(C=C)C(NC(=O)C(C)(C)C(F)F)C2)=O)ccc(S(N)(=O)=O)c(C)c1 c1(NC(C2C(NCc3c(OC)ccc(Br)c3)C2)=O)ccc2c(c1)COC2=O c1(OC)ccc(C=CC(=O)NCCOCCNC(C2C3CC4C(C3)C24)=O)cc1 c1(N2CC(CO)CC(CC)C2)nc2cccnc2c(=NC2CC(=O)N(C)C2)[nH]1 c1(C(=O)NCCN(C(=O)C2=CC(O)CCC2)CCC)cc(Cl)c(Cl)c(Cl)c1 N1(C(C=COCC)=O)CCN(C(C2CN(C3(C(F)F)CCOCC3)C2)=O)CC1 CC1(C)CC(N=c2nc(N3CC=CCC3)c3cc(F)ccc3[nH]2)CCS1(=O)=O c1(C(CO)NC(=O)NC(C)C(C)F)ccccc1Cl N1(C(CC2(COC)CC2)=O)CCC2(CC1)CN(C(c1sc(COC)nc1C)=O)C2 C(CC(=O)NCC(C)C(C)(F)F)(C(F)(F)F)NC(c1c(OC)ccnc1)=O c1(CNC(C2CC(NC(Cc3cccc(OCC)n3)=O)C2)=O)ccc(F)c(C)c1 c1(N2C(C(N(C3CCCC4CC34)C(C)=O)=O)CCC2)ncc([N+](=O)[O-])c(C)n1 C=CC(C)(O)CC(=O)NCCC1(OC)CN(C(=O)CC2CC3CCC2C3)C1 C1(C(N(C(C)CNC(=O)Cc2ccc(C(N)=O)cc2)C)=O)CC(C2CC2)=NO1 c1(CCC)ccc(S(=O)(=O)N2CC3(CC3C(=O)Nc3cccc(O)c3C)C2)cc1 C(CCC(=O)NC(CCO)C(F)(F)F)(C(C)C)NC(c1cc(SC)oc1)=O C12(NC(CS(C)(=O)=O)=O)CCN(C(=O)Cc3cnccn3)CC1C2 C1(C(=O)NC2CN(C(C(N3CCNC3=O)C)=O)C2)CCc2nc[nH]c2C1 N1(C(C(C)=C2CCC2)=O)CC2(C1)CN(C(=O)CC1CSC1)CC2CO N1(c2n(CC(C)C)c(-c3oc(O)nc3Br)nn2)CCC(O)C(F)C1 N1(C(c2cc(C)nc(O)c2)=O)CCN(C(c2oc(CO)nc2C)=O)C2CCCC12 c1(C(N2C3CC(NC(Cc4n(C)ncc4)=O)C(C3)C2)=O)cnn2cccc(Cl)c12 c1(-c2cn(CCN(C(=O)CN(c3ccncc3)C)C)nn2)cc(F)cc(F)c1 N1(C(CCN(C(=O)C(C2CC2)OC)CC)=O)CCC(O)CC1 C1(CCNC(c2ccsc2)=O)COCCN1C(C1CCOC1C1CC1)=O C(=O)(C(C)(C)C(C)(C)C)NCC(C(C)C)NC(c1cc(F)cnc1O)=O Cc1cc(C(=O)NC(C(=O)NCCC(F)F)C2CCCO2)oc1C Cc1cc(CNC2(C)CCC(C(N3CCC(O)C(F)C3)=O)C2)cc(C)n1 CN(C)S(=N)(=O)N1CCCC1C(=O)NCC1C2CN(C(=O)Cc3nc[nH]n3)CC12 C1(C(N2C(CNC(C(C)SC(C)C)=O)CC(F)C2)=O)CC2(C1)CC(F)C2 c1(C(N2CCOCC(CNCCCC3CC4(CCC4)C3)C2)=O)cnc(O)cc1O c1(C(N2C3CCCC2COC3)=O)ccc(=NCc2cccc([N+](=O)[O-])c2)[nH]c1 c1(C(C2CCN(C(c3cnc[nH]3)C)CC2)=O)cccc2cnccc12 c1(OC)ccccc1OCCC(=O)NCC=CCNC(=O)CCC1CC1C1CC1 C(CCN=c1nccc[nH]1)N(C(=O)CC1CCCC(O)C1)C COn1cnc(C)c1C(=O)NCC1CN(C(=O)C(C2CCOCC2)C)CCN1C N1(C(C2CCCN2C(c2c[nH]c(=S)cn2)=O)=O)CCC2(CCOC2=O)C1 C1(C(N(C)CC2CC(F)CN2C(=O)CCc2c[nH]c(=N)[nH]2)=O)CCCC2(CC2)C1 c1(CC(=O)N(C(c2ccccc2)CSC)CC)ccc2nc(Cl)sc2c1 C1CCN=C2NC(=NC=C2Br)O1.C#CCCC(=O)NCCOCCN C1(NC(C2C(C)(C)C2)=O)CC2(NC(=O)C=C3CCSCC3)COC1C2 CC1CN(C(C(=O)NC2COC2)C(C2CC2)C2CC2)Cc2c[nH]nc21 c1(C(=O)NCC2(NC(C3CC(CC)OCC3)=O)CC2)c2c(c[nH]c1=N)CCC2 c1(NC(N2CCC(O)(C(F)(F)F)C2)=O)ccc(C(O)C(F)F)cc1 C1(CC)(NC(=O)C(C)SC)CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1 N1(C(C=Cc2ccc(C)o2)=O)CCC(C)N(C(=O)CCc2ccn(C)n2)CC1 Cc1cc(OCC(=O)NC2C3CN(C(C4CNC(=O)CC4C)=O)CC23)ccc1Cl C1(C(=O)NCC2OCCN(C(C)=O)C2)CC2CC(CN2)O1 C(=O)(C(O)C1=CCCCC1)N1CC(C)(CNC(C2(OC)CCCC2)=O)CC1(C)C c1(C(CC(=O)NCCN(C(=O)Cc2ccns2)C)C)c[nH]c2ccccc12 N1(C(c2cc(C)sn2)=O)CCC(C(C)(C)CNC(C2(O)CCCC2)=O)CC1 Cc1cc(O)ncc1C(N1C2CC1CN(C(=O)Cn1cnc(=N)[nH]1)C2)=O C1(C(=O)NC(C)C(=O)N(C)C)CC2(CC(NC(=O)C(C)C3(O)CCC3)C2)C1 c1(NC(C2CC(C(N)=O)C2)=O)ccccc1CNCc1ccncc1 CCC(CC(=O)NC1CN(C(c2ns[nH]c2=O)=O)CC1N=[N+]=[N-])C(F)F C1(NC(=O)C(c2ccccc2)O)CCN(C(C2CC=CCO2)=O)CC1F c1(CC(=O)NC2CCN(C(=O)Cc3cscn3)CC2F)cc(Cl)c2c(c1)OCO2 N1(C(C(C(C)C)OCC)=O)CC2(CCNC(=O)Cn3nc(C)cc3C)CCC1C2 Cc1cn(C)nc1C(=O)NCC1CC1NC(=O)C(C)CN(C)C C1(S(N)(=O)=O)(C(N(CCC)CCNC(=O)CCOc2ccccc2O)=O)CCC1 C1(C(=O)NC2(c3ccc(F)cc3)COC2)CC2CC2N1C(=O)Cc1cc(Br)cs1 c1(C(N2CC(O)CC(NC(COCCC#C)=O)C2)=O)cnc2ccccc2n1 Cn1nnnc1C(C)(CCC1CCCC1)NCCCOc1nncs1 C(=O)(C1c2c[nH]nc2CN1C(=O)Nc1nc(-c2ccc(C)cc2)c(C)s1)NC CC(C)(C)C(CC(=O)N1CCC(CCCNC(=O)Cc2cc[nH]n2)CC1)C(F)F c1(C(N(CCNC(C(C)OCC#C)=O)CC2CC2)=O)cncc2nc(C)[nH]c12 N1(C(CCSC)=O)CCCC(c2nc(-c3ccncc3)nn2-c2nccn2C)C1 Fc1ccc(CN2CCN(Cc3ccsc3)CC2)cc1Cl N1(C(c2cc(C(C)=O)sc2)=O)CCC(NC(=O)CC2CCN(C)C2)C(F)C1 N1(C(c2ccn(CC)n2)=O)CC(OC)CC(NC(c2cnn(CC(C)C)c2)=O)C1 c1(CCC(=O)NC(CNC(c2cn(C)nc2)=O)C2CCC2)ccc(N(C)C)cc1 C(=O)(CC(F)(F)F)N(CC(C)N(C(=O)C(C1CCOCC1)O)C)C C=C=CCC(=O)NCCN(CCCN(C)C)C(c1cc(-c2ccn(C)n2)on1)=O C#CCC(CC#C)C(=O)NCC1CC(CNC(c2cc(N)cc(F)c2)=O)C1 c1(CCCCC=C=C)cccc(F)c1.C1(c2nnnn2C(C)(C)C)CCCN1 c1(C(=O)NC(c2ccc(Cl)cc2)C)ccc(CNC(=O)C(N)=O)cn1 CN1Cc2ccc(C(N3CCOCC(CNC(=O)Cc4cccs4)C3)=O)cc2C1 CC(CCNC(C1CC1c1ccncc1)=O)CCNC(C1CC(F)(CO)C1)=O c1(OC)cccc2c1CC(C(N1CCC(N3CCCNC3=O)CC1)=O)N2 N1(C(C(=O)N(C)CC2CC(F)C(C#N)C2)=O)CCC2(CCCO2)CC1 n1(C(C(=O)NC(CNC(C=C(CC)C2CC2)=O)CC)C)ccnc1C CC(CS(C)(=O)=O)C(=O)NCC1CCN(C(=O)CCCCCF)C1 C1(CC(=O)NCCSCC#C)CCCC1NC(c1sccc1COC)=O N1(C(C(C)SCC)=O)CCN(C(c2cn(CC)nn2)=O)C2CCCC12 Nc1c(C(=O)NCC2(NC(=O)COC3CCOC3)CCC2)cccc1F c1(CC2CCC(C(=O)NC(=O)NCC3OCCN(C)C3)OC2)ccc([N+](=O)[O-])cc1 C(=O)(C1=CCCOC1)NC1C(C)CN(C(=O)COCCF)C1 C=CCCC(C)(C)C(=O)N(C)CCN(CC(=O)O)C CC(C)CC(C)(C)C(=O)NC(C)C(C)NC(C1(CCN(C)C)CC1)=O C(=O)(CCC(=O)Nc1nccs1)NCC(C1CCC1)NC(c1ccc(CC)s1)=O CS(=O)(=O)CCC(=O)N1CC2CCC2(CNC(C2(F)CCC=CCC2)=O)C1 N1(C(C)=O)CSCC1CNC1(CNC(=O)Cc2ncc(C)s2)CC1 N1(C(C2(C=C)CCC2)=O)CC(N(C)C(c2cc(C)cc(F)c2)=O)C(C)(C)C1 CC1(C)CC(CNC(=O)Cc2cccs2)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 C1(F)(CNC(COC(C)=O)=O)CCN(C(c2cnncc2C)=O)CC1 C1(CC#C)(C(=O)N(C2CSC2)C)CCN(C(c2ccncc2Cl)=O)C1 N1(CCC(=O)NCC(C2N(C(C=CC=CC)=O)CCC2)(C)C)CCN(C)CC1 c1(C(=O)NCc2ccn(CC(C)C)n2)ncc(C(F)(F)F)cc1Cl N1(C(CCOCC#C)=O)CCCC(CCNC(=O)C2=CCCO2)C1 CCC(CC)(CC)C(=O)NCC(C(=O)NC(c1csnn1)C)N(C)C C1(C(N(CCCO)C)=O)CCCN1C(C1CC1C(=O)C1CC1)=O Cc1cccc(CCNC(=O)C(C)NC(c2c(C)nsc2C)=O)c1 CCC(F)(F)CC(=O)NCCCCN(CCCNC(=O)Cn1ccc(C)n1)C c1(CC(=O)NC2CC2C(=O)Nc2nc(Cl)ccc2I)c(F)cccc1F CC(C)CC(C)CC(=O)NC(C)(C)CN1CCN(C(c2cnc(Cl)s2)=O)CC1 O(NC(=O)CN(C)CCOCCNC(=O)C(C)CN(C)C)CC(=C)C C1(C(=O)NCCC(C)NC(c2c[nH]c(C#N)c2)=O)CCCC1P(C)(C)=O C1(NC(c2cncnc2C2CC2)=O)C2CN(C(c3csc(C(F)(F)F)n3)=O)CC12 c1(NC(C2(F)CCN(C3CCCC3)C2)=O)cc(NCCN2CCC(O)CC2)ncn1 Cc1ncc2n1CCN(C(=O)CCNC(C1CC(=O)CCO1)=O)C2 C1(C(N2CCCC(NC(=O)Cn3cnnn3)CC2)=O)CCc2nc(O)[nH]c2C1 CCCC(F)C(=O)N1CCCC1CNC(C1(OCC)CCCCC1)=O N1(C(C(C=C)(C)CC)=O)CCC2C(C1)NC(=O)CN2C(=O)CCc1cccs1 N1(C(C(CC)COC)=O)CCC(CNC(=O)CCCC2CCC2)C(F)(F)C1 CC(C)(CCSc1c(F)cccc1Br)CC(=O)NC(C)(C)C N1(C(CC(C=C)(C)O)=O)CC(CNC(c2ccoc2C2CC2)=O)OC2COCC12 c1(N2CC(CCNC(C(CC)C)=O)C2)ncnc2ccc(OC(C)C)cc12 C1(NC(c2c(OC)nccc2)=O)CC2CCC1N2C(=O)Cc1csc(C)n1 N1(C(CNC(C)=O)=O)CC2CC(NC(c3cc(C(F)(F)F)ccc3Cl)=O)C1C2 C(CCN=c1ccnc(NCCNCCCN2CCOCC2)[nH]1)OC C1(CNC(CCOCCN(C)C)=O)CCC(C)(C)CN1C(C1CCNC1=O)=O Cc1cc(Br)cc(C(=O)NC(CNC(=O)CC(C)c2cnn(C)c2)CO)c1N c1(SCC(=O)N(C2CN(C(=O)CC3CCCCO3)CC2F)C)cccc(F)c1 N1(C(C(C2CC2)OCC)=O)CCC2(C1)CN(C(=O)C#CC1(C)COC1)CCO2 C1(C(N(C(C(=O)N(CCF)CC)C)CC)=O)CC(C)CC(=O)N1 Cc1nc2ccccc2c(C)c1C(=O)OCC(C12CC(c3ccccc3)(C1)C2)=O c1(C(=O)NCC(CC(C)C)(C)NC(=O)COCCCF)occ2c1CCOC2 CC1CC(C(=O)NCC2=CCN(C(=O)COCC3CCOCC3)CC2)CC(C)C1 C1(O)(C(=O)NCCC2(CNC(CNS(N)(=O)=O)=O)CC2)CCSCC1 C1(NC(C(CCF)NC(COCCCCC)=O)=O)CCC(C2CC2)C1 c1(CC)conc1CC(=O)NC1(CNC(=O)C(C)Cc2cnco2)CCOC1 c1(NC(C2C(C(=O)OC)C2)=O)cc(=NC(=O)c2cc3c(C)cccc3[nH]2)[nH][nH]1 N1(C(CCCSC)=O)CCN(C(c2c(C)nc(C3CC3)nc2O)=O)CC1C#N CN1CCC(O)(NCC2(F)CCN(C(=O)OC(C)(C)C)C2)C1 CC(C)(C)C(CO)C(=O)NC1CCCC1NC(c1c(Br)cnn1C1CC1)=O c1(NC(N(C(C2CCCO2)CC2CCCC2)C)=O)c(CCC(N)=O)c[nH]c1C C1(NC(CCOCCCOC)=O)CCN(C(c2csnc2OC)=O)C1C(C)C CC12CC(CCNc3nccc(N4CCC(C)(C(F)(F)F)C4)n3)(CO1)C2 c1(OC)cc(C(=O)NCC2CCCC2NC(c2cc(C)ns2)=O)sn1 C1(NC(C2N(C(C)=O)CCC2)=O)CC(F)CN(C(c2cnn(C(C)C)n2)=O)C1 C1(C(=O)NC(CC#C)C(=O)NCCC)CC2C=CC1CC2.C1CCCC1N(C)C C=C1CCC(C(=O)NC(C(=O)NCc2cccc(Cl)c2)C2CC2)CC1 c1(CC)ncncc1C(N1CC2CC2(CNC(=O)Cc2csnn2)C1)=O C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(C(CC)CC(F)F)=O)C(O)C(O)C1 C(=O)(C(S(N)(=O)=O)c1ccccc1)NCCCCN(C(c1sc(C)c(O)n1)=O)C CCC(CC)CCCNC(C1(COC)C=CCN1C(C1CC2C=CC1O2)=O)=O N1(C(CC2(N(C)C)CC2)=O)CCCC1C=CC(N1CCOCC1C(C)(C)C)=O c1(OC)cc(OC)c(C(=O)NC2CCC(NC(C3CNC(=O)C3)=O)CC2)c(N)c1 C1(C(=O)NC(CC)CNC(=O)Cc2cnn(C(C)C)c2)CN2CCCCC2CO1 c1(C(=O)NCC(CN(C(C2=C(C)OCC2)=O)C)(C)C)cc2c(C)c(Cl)ccc2[nH]1 c1(CN(C)C(=O)NC2CCN(c3ccncn3)CC2)ccc(F)cc1Br C1(C(=O)NC(CC(C)NC(C(CC)=CCCC)=O)C)CCCOC1C c1(C(N2C(CNC(=O)CC3CCC3)(CSC)CCC2)=O)ccc(OC)c(Cl)c1F c1(CC)nc(=N)[nH]cc1C(N1CC(NC(c2ccncc2F)=O)C2CC12)=O C(C)(CC(=O)N(NC(=O)OC(C)(C)C)C(C)C)c1c(C)ncs1 c1(C2(CNC(c3cnc(C4(C)CC4)[nH]3)=O)CCCO2)ccc(Br)cc1 Cc1cc(C(=O)NCC2CCN2C(c2ccnc(N(C)C)c2)=O)ncc1Cl Cc1ccc(C(CN2CCCCC2)Nc2ccc(-n3cnnn3)cc2)cc1 Cc1cc(CC(N2CC(N(C)C(c3cnc(N(C)C)o3)=O)C(F)C2)=O)ccn1 O(S(=O)(=O)c1ccccc1F)C1C(c2nc3cccc(CCC(=O)OC)c3s2)C1 c1(OC)cc(CN=c2[nH]c(CN3CCC(CO)C(O)C3)cs2)cc(O)c1O C1(NC(c2c(C(=O)OC)scc2)=O)CCCC2CN(C(c3ccn(C)n3)=O)CC12 N1(C(CC2C(C)CCO2)=O)CCC(CO)(CNC(c2csc([N+](=O)[O-])c2)=O)CC1 c1(NC(C2CC(CC(=O)NCC3(OCCO)CCC3)C2)=O)ccc(Br)nc1 C(=O)(C(C)(C)C1CCCCC1)N(CCNC(=O)CC1CCCO1)CC c1(C(N(CCOC)CCNC(=O)C2=NOC(C)C2)=O)cc2c(s1)CCCCC2 c1(C(=O)NCCN(C(C(CCSCC)NC(N)=O)=O)C)ccc(S(N)(=O)=O)o1 CC1(C)CN(Cc2nn[nH]c2Cl)CC1NC(C1CCN(c2nncs2)CC1)=O C1(NC(CN(CCC#C)C)=O)CC2(CCCN(C(=O)CCCc3ncco3)C2)C1 c1(C(=O)NC2CC(C)(NC(C(CCCCC)O)=O)C2)cccc2nc(C)[nH]c12 c1(OC)ccc(C(=O)C(=O)NCc2ccc(Cl)cc2)cc1F C=CCCCCC(=O)N1C2CCC1C(CNC(=O)CS(=O)(=O)N1CCCCC1)C2 c1(C(=O)NC(CNC(C2CS(=O)(=O)C2)=O)CO)c(C(F)(F)F)cccc1Cl CC1(C)CCCN(C(C2(C#N)CCC2)=O)C1CNC(c1cccnc1O)=O N(C(=NCCCN(C)C(C)C)NCc1c(F)cccc1Br)C(CC)C c1(C(N2CCC(O)(CN(C(=O)C=C3CCC3)C)C2)=O)cnn2ccc(O)nc12 C1(CC)C(NC(=O)COC2CCOC2)CCCN1C(=O)CCCCOC CC1(CNC(C2(CC(F)(F)F)CC2)=O)CCN(C(=O)C=CC(F)(F)F)C1 CC1CN(C(=O)Cc2cc[nH]c2)CC(C(=O)NCCN(CCCF)C)O1 Cc1ccc(C=CC(=O)NC2(C3CCCCN3C(C3CCC3(C)C)=O)CC2)o1 Cc1cc(O)c(F)cc1NC(C1CCN(C(c2ccc3cc[nH]c3c2)=O)O1)=O C(=O)(C(C#N)C(C)C)NC(C(=O)N(C1CC(OCC)C1)C)CCF N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(C)(C)C(CNC(C2CCN(C)CC2)=O)C1 c1(C(N2C(CCC(=O)N(CC(N)=O)C)CCC2)=O)ccnc(Br)c1F CCC(CC)C(F)C(=O)NCc1c[nH]nc1C(=O)NC1CCC([N+](=O)[O-])CC1 N#Cc1cc(CNC(=O)CC2CC3(C2)CN(Cc2cc(C#N)cs2)C3)ccc1F N1(C(C2C(=C)C2C(=O)OC)=O)CCC(CCNc2ncc(CC)s2)C1 Cc1cc(Br)c(NC(C2CN(Cc3ccc(O)c(F)c3F)CCC2O)=O)nc1C C(C(C)(C)C(=O)N(C1CCOC1)C)NC(C(CC)SC)=O c1(C(=O)NCC(C2CC2)NC(C=Cc2c(C)cccc2)=O)ncc(C#N)cc1Cl C(=O)(CC1OC(=O)c2ccccc21)N(CCC(C)NC(c1scnc1Cl)=O)C N1(C(c2cn[nH]c2)=O)CCC2(CCCC2NC(=O)C(O)(C2CC2)C2CC2)CC1 CCCCCCC(C)C(=O)NCCC1(CNC(=O)CC2CC(=O)NC2=O)CC1 N1(C(c2c(CC)nns2)=O)CCCN(C(C2CC3CCC(C2)C3=O)=O)CC1C c1(C(=O)NCCCC(CCC)NC(c2ccco2)=O)cnn2ccc(OC)cc12 CCC(C)CCCC(=O)NCCCN(C(=O)C(C(C)O)N(C)C)CC c1(C(N2CCCC2CSC2CC2)C(=O)NCCCOC)ccc(C#N)c(C)c1 c1(CC(C)C)ccccc1C(=O)NC(C12CCC(CC1)C2)C c1(N2CCC(NC(CC(CCC)C)=O)C(F)C2)ccc2c(n1)CCC2=O C#Cc1ccc(F)cc1C(=O)NC1(C)CC(NC(=O)CCc2cccn2C)C1 c1(NC(c2c[nH]n3c2nc(=O)c2ccccc32)=O)nc2ccc(Cl)c(Cl)c2s1 c1(CC(C)(CSC)NC(=O)CS)ccc(C(F)(F)F)cc1.CCC(O)C=O c1(C(=O)NC(CO)C2CCC2)ccc(F)c(O)c1 N1(C2CCCN(C(C3C(C(N)=O)C3)=O)C2)CCN(C(=O)C(O)C2CCC2)CC1=O c1(N2CCC(CC=C)(NC(=O)C(c3ccccc3Cl)C)C2)ccncc1[N+](=O)[O-] Cc1nn(-c2ccc(F)cc2)cc1C(=O)NCCNC(c1cnc(C2CC2)s1)=O CCCC(O)C(=O)NCC(c1ccccc1)CNC(=O)C=CC(C)(C)SC CC1(C)CC(CNC(C2NC(=O)OC2(C)C)=O)N(C(C2C(C)(C)C2(C)C)=O)C1 c1(CC(=O)NC2(C)CCN(C(c3ccccc3)=O)C2)c(F)cccc1Cl CC(C)CC(C(=O)NCC1CC(C)C1)ONC(c1cc(Cl)cn1C)=O N1(C(C)C)CCOC(C(=O)NC(C2CCN(C(=O)COc3ccsc3)CC2)C)C1 c1(OC)ccc(Br)c(CC(=O)NC2CCCC2NC(C2CCOC2)=O)c1 C1(C=C)(C(=O)NCCC2(OC)CN(c3nc(C)ncc3F)C2)CCOCC1 c1(OC)ccc(CO)cc1C(=O)NCCC1CCN(C(=O)Cc2ccsc2C)C1 C1(O)(C(C)NC(C(=O)NCC)=O)CCCN(C(C2(CC)CCCC2)=O)C1 C12(C(N3C(CNC(C4N(CCC)CCC4)=O)CC3)=O)CC3CC(C1)CC(O)(C3)C2 CC1CC(C(=O)NC2(C)CC(C(=O)NCCc3cccnc3F)C2)CCS1 N1(C(Cn2cc(C)c(O)nc2=O)=O)CC2CN(C(=O)CC3CC34CC4)CCC12 c1(C(=O)NC2C(CCC)CN(C(c3cc(CC)oc3C)=O)C2)ccc(O)c(F)c1 c1(NC(=O)CC2CCCCCN2C(C2CC=CCO2)=O)cccc2[nH]ccc12 C1(NC(c2cccc(Br)c2F)=O)CN(C(C2CC23CCC3)=O)CC2CC12 N1(C(CCCCN(C)C)=O)CCN(C(=O)C(=O)C2CCCC2)CC1CO C1(OCCNC(CCCSC)=O)CCN(C(=O)CCN2CCOCC2)CC1.C=O C1(N(C(=O)Cc2csc(S)n2)C)CCCN(C(=O)CN2CSCC2=O)CC1 c1(C(=O)NC2(CC(=O)N(C(C)C3CC3)CC)CCC2)cc2ccccc2[nH]1 N1(C(=O)CC2COCCN2C(C2CC3C=CC2C3)=O)CCN2CCOCC2C1 CCC(C(O)C(C)C)NC(C1(CC)CCN(C(=O)CCCC(C)=O)CC1)=O C=CCC(C(=O)N1CCC(CF)(NC(C2CC2C2CCCO2)=O)C1)c1ccccc1 C1(C(=O)OC)CC(OC)CN(C(=O)NCc2nc[nH]c2C2CC2)C1 N1(C(CC)=O)CC2CC(C(=O)NCCS(C)(=N)=O)(C2)C1 O(C=C(C#N)C(=O)NC1C2CCC(C2)C1NC(=O)COC)CC C#CC1CCCC(C(=O)NC2(C3CCCN3C(c3ccc(F)cc3C)=O)CC2)C1 C(=O)(C(F)CC(C)(C)C)NC1CC=C(C(=O)NCC(c2ncn(C)c2)O)C1 Cc1ccn2cnc(C(=O)N(C)CCN(C)C(c3cncnc3C3CC3)=O)c2c1 C(=O)(CCCCCNC(c1cc(CO)n(C)n1)=O)NCC(CC(C)C)N(C)C CC(C)CCC(C(=O)NCC(F)C(C)(C)O)NC(C1(C)CC(C)C1)=O C1(C(=O)NC(C(=O)NCC2C(=C)C2)CCOCCO)CC2(C1)CC(C)C2 c1(C(=O)NC2CC(CCNC(CC(C=C)(C)C)=O)C2)c[nH]c2cc(Cl)ccc12 C(=O)(CCS(C)(=O)=O)N(CCNC(c1nc(COCC)sc1)=O)C C1(C(=O)NCC(C)(CO)NC(c2c(OC)nsc2)=O)CC(C)OC(C)C1 C1(CNC(c2cccc(NC(C)=O)n2)=O)CC2(CO1)CN(C(c1cnoc1)=O)C2 CC1(C)C2CN(C(C3CN(Cc4cccc(C(C)(C)C)c4)CCS3)=O)CC12 Cc1cnc(C(=O)N(C2CCN(C(=O)COc3cccnc3Cl)C2)C)cn1 c1(C(N2C(CCNC(c3n(C)nnc3)=O)CCCC2)=O)ccc2c(c1)NCC2 c1(N(C)Cc2nnc3n2CCOC3)nc(=NCC2SCCS2)[nH]c2ccsc12 C1(N2N3C(CC(O)C3)C2=O)COCCC1(F)F.C(CCC)N(CC=C)CC=C.C=O N1(C(c2ncc(OC)cn2)=O)CC(N(C)C(C2NC(=O)OC2C)=O)C(C)(C)C1 N1(C(c2ccc(C)[nH]2)=O)CCCC12CCN(C(=O)C(F)CC1CC1)C2 C(C(C)(O)CC(=O)NC(CNC(=O)CN(c1ccc(Cl)nn1)C)C(C)C)OC N1(C(c2c(C#C)cn(C)n2)=O)CC2(C)CN(C(C3CC(CC)=NO3)=O)CC2(C)C1 C1(C(=O)NC2C(NC(CN(c3ccncc3)C)=O)CCCC2)CCCC12CCC2 Cc1nn2c(C(=O)N(CC(O)CNC(c3ccc(N)cc3C)=O)C)c(C)nc2s1 CCC(CNC(=O)C(CC1CCC1)NC(c1c[n+]([O-])c(C)cn1)=O)C(C)(F)F N1(C=O)CC(=O)N(C)C1C(C)C.C1(N2CCCC(C)C2)(CCC=C)CCNCC1 C1(CN(C(c2cnc(C(C)C)[nH]2)=O)C)CCCN(C(=O)C(=O)NCC(F)F)C1 N1(C(c2cc(C)no2)=O)CC2(CCC2)CC1C(=O)NC(c1cnn(C)c1)CO C1(N(C(CCCC#C)=O)C)CCN(C(=O)CCCC(C)C)CC12CC2 C1(NC(C(COC)CC(C)C)=O)CCN(C(c2n[nH]cc2Cl)=O)CCC1(F)F Cc1c(C(=O)NC(CNC(=O)C(C)(C)C2CCCO2)C2CCC2)cnn1CCO N1(C(CCCC(CC)CC)=O)CCC2(C=C(C(=O)NC(C)Cn3cnnc3)C2)C1 N1(C(Cc2c(C)ocn2)=O)CCOC(C(N2CCN(CCO)CC2C)=O)CC1 c1(C(=O)NCCC2N(C(CC(C)C(F)F)=O)CCSC2)cccc2nn[nH]c12 N1(C(c2ccnc3cc[nH]c23)=O)CCC2CN(C(C3CC3(F)Cl)=O)CC2CC1 C1(NC(C2CCN(C(=O)OC)CC2)=O)CN(C(=O)CCC(C)(C)OC)CC12CC2 c1(C(=O)NCC(CCCC)NC(=O)Cc2cccc(C)c2F)cccc(O)c1F Cc1ccc(Br)c(C(N2CC(CNC(c3nnn(C)c3N)=O)C(C)(C)C2)=O)c1 S(=O)(=O)(c1ccc(N2CCCCC2)nc1)N.CC1OCCC1C(N1CCCC1)=O C(c1ccc(O)cc1)=CC(N1C(CCNC(c2c(C)csc2)=O)CCCC1)=O c1(CC(=O)NC2C(NC(C3N(C)CCC3)=O)CCOC2)ccc2ncsc2c1 c1(OC)ncc(C)c(C(=O)NC(C)C(C)NC(=O)Cc2ccc(F)c(F)c2)c1Cl c1(C(=O)NC2CC3(C2)CC3C(=O)NCC2CCCC23CC3)occ2c1CCC2 c1(C(N2CCN(C(C(C=CC)O)=O)CC(O)C2)=O)ccc2nc(C)[nH]c2c1 C1(C(=O)NCC(NOC)=O)C(C)CCN1C(c1nonc1C)=O CC(C#N)CCC(=O)N1CCOC(C)(CNC(c2ncc[nH]c2=N)=O)C1 CCCCC(O)C(=O)N1C(CC(N2CCCCC2CCOC)=O)C2CCCC12 CN1C(=O)C(NC(=O)NC2OC3CCC2CC3)c2cc(Br)ccc21 C=CCC(CC)C(=O)NCCC(C(C)C)NC(C1(OC)CCOC1)=O c1(C(N(CC(C)NC(C=CC(C)(C)SC)=O)C)=O)cnn2c1CN(C)CC2 C1(N(C)Cc2ccc(C(=O)OC)[nH]2)Cc2ccccc2C1OC C1(CCNC(=O)C(F)CC2CC2)CCN(C(C2(Cl)CCC2)=O)CC1 C=CCCC(F)(F)C(=O)N1CC2CC1C2CNC(C12CC(CO1)C2)=O C(CC(O)C(=O)N(CCNC(C1CC12CC(O)C2)=O)CCc1ccccc1)SC C12(C)CCCN(C1)C2=O.C12(CN(CCN(C)C)C)CC(c3ccccc3)(C1)C2 C1(NC(CN(C(c2cnccc2C)C(=O)NC)CC(C)C)=O)CCS(=O)(=O)C1 C12(NC(C(C)(F)F)=O)CCN(C(c3ccc(OCC(F)(F)F)o3)=O)CC1C2 c1(CCBr)cc(F)c(F)c(F)c1.c12ccc(cc1)NC(=O)C(=O)N1CCCC21 O=C1Nc2ccc(C(=O)NC3COCC3NC(=O)CCOCC3CC3)cc2C1=O c1(C(N2CCC(O)(c3cn(CC(=O)OCC)nn3)C2)=O)cc(F)cc2c1CCC2 C(C)(CCC(C)(C)C)NC(CSCCNC(CCCCOC)=O)=O Cc1nc(CSC(CNC(=O)OC(C)(C)C)CO)c(C)c(O)n1 c1(C(c2ccccc2)NC(C2C(C)=C2)=O)nc(C)ccc1F C1(C(=O)NC)C2CN(C(=O)NC3CCN(C4CCCCC4)C3)CC12 C1(NC(CSCCC)=O)CC(C(=O)N(CC(C)C)CC2CC2)C1 C(CNC(=O)CN1CC2CC2C1)(C(=O)NC1CC2(CC2)C1)N(C)C(N)=O C1(c2ccccc2)(C(=O)NC2C(CNC(C(n3cc(Cl)cn3)C)=O)C2)CCCC1 C=CC(CC)CC(=O)N1CCC(N=[N+]=[N-])(C(=O)NC(C)CN(CCCC)C)C1 N1(C(CCCC#N)=O)CCCC(CC(=O)NCC2CC3(CCC3)C2)CC1 c1(C(=O)Nc2ncn(C)c2)csc(=NCc2c(I)ccnc2F)[nH]1 C(=O)(C(C)CC(C)CC)NCC1(OCC)CN(C(=O)C2=COCC2)C1 c1(C(=O)NC2CC(F)(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)ccc2cccnn12 c1(OC)cc(C#N)ccc1NC(=O)Cc1cc(F)c(C)cc1F C1(NC(C(c2c[nH]c3ccccc23)C)=O)CC2CCC1N(C(=O)CC1CC1)C2 c1(C(N2CCC(C(C)NC(Cc3cc(C)sc3)=O)C2)=O)cc([N+](=O)[O-])cnc1C c1(N2CCC(OCCOC)CC2)nc(=NCC2CCCC2OC)[nH]c2c1COC2 Cc1oc(Cl)nc1C(=O)N(CC(N1CCCC(C)C1)=O)CC(C)C N(C1CCOc2ccccc21)C(c1cccnn1)C(=O)NC1CCOC1 c1(C(=O)NCCCCCN(C(=O)CCCC(N)=O)C)ncc(C#N)cc1Cl Cc1ccc(-n2nnnc2C(C2CC2)Nc2nc(C)c(C)[nH]2)cc1 C1(NC(CC2C(C)CCC2)=O)CC2CC(C1)N(C(=O)CCS(=O)(=O)N(C)C)C2 C(=O)(C(C)S(=O)(=O)C1CCOCC1)N(CC(C)N(C(CCCCCOC)=O)C)C C(c1cncc(OC)c1)=CC(=O)NC(CNC(CNC(=O)OC)=O)(C)C1CC1 C1(NC(CC=CC(C)(C)C)=O)CC(F)CN(C(C2CC3C=CC2C3)=O)C1 c1(C(N2CCCC(CN(C(C(CC(=C)C)C)=O)C)C2)=O)cc2c(nn1)CCOC2 c1(CC(=O)NCCN(C(=O)C(c2cc(Br)co2)=O)C)cnn(C(C)(C)C)c1 N1(C(C2CCN(c3ccc(OC)cc3)C2)=O)CC2C=C(Br)C2C1 c1(OC)ccc(NC(=O)C(C2CCCCC2)NC(c2ccco2)=O)nc1 Cc1nc(S(=O)(=O)NC(C)C(c2ccc(Cl)cc2)C)c(-c2ccccc2)o1 C(=O)(C1CNC(=O)c2ccnn21)NC1CC(NC(c2c(OC)ccc(C)n2)=O)C1 c1(CC)c(C(=O)NC(CNC(=O)CCC2CC2C)CCOC)[nH]c(C)c1C(N)=O C1(CNC(NC(COC)C)=NCCc2cccs2)COc2ccccc2C1 Cc1c(C=CC(N2CCC(CNC(c3sccc3Br)=O)C2(C)C)=O)cnn1C C1(C)(C(=O)NC(CNC(C2(C(=O)OCC)CCC2)=O)CO)CC=CCC1 C(=O)(CS(=O)(=O)c1ccccc1C)N(CC(CNC(C(CC)(CC)CO)=O)C)C c1(C(N2C(CCNC(c3ccc(CO)o3)=O)CCCC2)=O)cc2sccc2s1 CC1=NOC(C)(C(=O)NCC2(C(N)=O)CN(C(C3(C(F)F)CCCO3)=O)C2)C1 C1(F)(CNC(C2(CCC)CC2)=O)CCCN(C(=O)C2=C(Cl)CCC2)C1 Cc1cccc(C(F)C(N2CCSCC2CCNC(=O)C=CBr)=O)c1 Cc1[nH]nc(C(C)C)c1C(N1CCC(N(C(=O)C(C)n2ccnn2)CCO)C1)=O OCCC(N=c1nc2sccc2c(N2CC3COCC3C2)[nH]1)C1CCC1 Nc1ccc(Br)cc1C(=O)NCC1CCCC(NC(=O)Cc2cccnc2)C1 c1(CNC(c2cnn(C3CC3)c2)=O)ncccc1O.C1CC(=O)N1 N1(C(CC(COC)C)=O)CCOCC(CNC(=O)C=C(C)c2ccco2)C1 N1(C(CC(C)(C)n2cc(-c3ccncc3F)nn2)=O)CC(F)(F)C(F)(F)C1.CCO C1(CNC(C2CCc3c[nH]nc3C2)=O)CN(C(=O)C2=CCCC2)CCC12CCC2 N(C(=NCCC)NCCC(O)(C(F)(F)F)c1ncco1)CCCCCCC#C CC1(CNC(=O)CN2CCCOC2=O)CCCN1C(=O)C=C1CCC1 C1(NC(=O)CCCN2CCCC2)CC2(CCCCN2C(c2ccc(Cl)nc2)=O)C1 CCC(O)C(C)C(=O)NC12CC(NC(c3cccc(OCCOC)c3)=O)(C1)C2 CC(C)C(C(=O)N1CCCN(C)C(=O)C1)C(C)NC(=O)CN1CCC(C)C1 CC(C)C(C)(O)C(=O)NCc1nc(C(=O)NCC(C)(C)n2ccnc2)co1 Cc1cc(C(C)NCC2(O)CCC(O)CC2)ccc1C#N C(=O)(CS(=O)(=O)CC(C)C)NCC(CC=C)C(=O)N1CCOCC1 N1(C(CSCC#C)=O)CC(F)CC1CN(C(=O)CC(N1CCCCC1=O)C)C Cc1cc(C#N)ccc1NC(C1CCC(NCc2cnc(Cl)s2)CO1)=O c1(CC(=O)NCC2(CNC(CN(S(C)(=O)=O)C)=O)CCCC2)cccc(C)c1 CN1C(=O)CCC1C(=O)NCC(O)CNC(=O)Cc1cccc(C(F)F)c1 Cc1ccc(O)cc1NC(C1(CNC(=O)C=CC(F)(F)F)CCCC1)=O c1(C(N2CCC(c3ccc(C)s3)CC2)C(=O)NCCC#N)ccc2c(c1)CCC2 Cc1ccc(C)n1CCC(=O)NCCC1CCN(C(C2CCCCCC2)=O)CC1 C(=O)(C(F)(F)CCC1CC1)N(CCCNC(c1scc(C)c1C)=O)CC C(=O)(C1=NOC(C)C1C)NCC(C(=O)NC(CC)(C)C)O C1(C(=O)NCCCC(=O)N(C)CC2(OC)CCCC2)(OC)CCCCC1 C1(C(N2C3C(NC(c4ccc(CN(C)C)[nH]4)=O)C(C3)C2)=O)CC2(C1)CC1(CC1)C2 c1(SC)ccc(Cl)c(C(=O)NC2CC(F)(CNC(=O)CC3CCCS3(=O)=O)C2)c1 CCC(C)C(O)C(=O)NC(C)CN(C)C(c1conc1C1CCC1)=O N1(C(C(F)OC)=O)CC=CC1CNC(=O)C(O)CC1CCCCC1 C(C(=O)Nc1ccc(Cl)cc1F)(C1=NOCC1)N1CC(C)OC(C)C1 c1(CCC(C)NC2CC(=O)N(CC3C(O)C(O)CN3C)C2)cc(Br)ccc1F C1(NC(c2cnc(C)s2)=O)CCN(C(c2cc(C#N)co2)=O)C1(C)C CN1CC(C(=O)NCC(CO)NC(c2cc(O)cc(O)n2)=O)CCC1=O CCCCCC(O)C(=O)NC(C)(C)C(=O)NC1CCN(S(C)(=O)=O)C1 CCC(CC)(C(=O)N1CC2CCC(C(=O)NC3(C)CCSC3)(C2)C1)C(C)C C(=O)(C1=CC2CC(C1)CC2O)N1C2(CNC(C(CCC)CC)=O)CCC1CC2 C1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)CCC(F)(F)CO1 N1(C(=O)OC(C)(C)C)CCC(CC(=O)Nc2ccc(F)c(F)c2)C(F)(F)CC1 c1(SC)cccc(NNC(=O)Nc2cncc(NC(=O)OC(C)(C)C)c2)c1 CC(C)C(C)(O)C(=O)NC1CCN(C(C2CCCN2C2CCOCC2)=O)CC1 CCCCC(F)C(=O)N1C(C(=O)NC)CC1C.C12(CC1)C(=O)NC2 CCC(CC(=O)N1CC2(CCN(C(C3COC4(C)CC3C4)=O)C2)C1)C(C)C C1(O)(C(C(=O)NCCOCCCNC(=O)C)F)CCCC1.n1(CF)cc(C2CC2)cn1 C(=O)(C1CCc2c(Cl)cccc21)NC1CC2(C(NC(C3CC4CCC3O4)=O)C2)C1 N1(C(c2cnn(-c3cccc(Cl)c3)c2)C(=O)NCC(=C)C)CCS(=O)C(C)C1C C12(C(=O)OCC)CC(CN(CC3CCCS3(=O)=O)C1)C2 N1(C(C23CC(C)C2C3)=O)C2CCC1CN(C(=O)Cc1sccc1Cl)CC2 C(=O)(C(=O)CCC(C)C)N1C(CNC(C2=CC(C)(CC)C2)=O)C(C)(C)CC1 C(=O)(C(CC)CCCC)N1CCC(C(N(CCCSC)C)=O)(C(C)C)C1 N#Cc1ccc2c(C(=O)NC3CN(C(c4coc5c4CSC5)=O)C3)c[nH]c2c1 C(=O)(C(C)S(N)(=O)=O)NCCC1CN(C(c2n(CC=C)ccc2)=O)CC1C CN1CCN(C2CCCC2NC(=O)Nc2cnn(CCF)c2)CC1 Cc1nc2c(N3CC(CC(C)NC(C4CCSC4)=O)C3)ncnc2s1 C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(O)(CNC(COC(CC)(C)C)=O)C1 C1(NC(C(c2cnn(C)c2)OC)=O)CCC(NC(=O)CCc2ccccc2)CC1 c1(OC)csc(C(=O)NC2CCC(CNC(=O)CCn3cc(Cl)cn3)C2)c1 c1(OC)cc(Cl)c(C(N2CCCC2C(=O)Nc2nccc(OC)n2)=O)cn1 CC(C)C#CC(=O)NC1(C)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)C1 S(=O)(=O)(c1c(Cl)cccc1Cl)NC1CN(C(c2ccc(F)c3ccoc23)=O)C1 c1(OC)cccc(COC(C)C(=O)N(CC(C)NC(c2cnccc2Cl)=O)C)c1 c1(C(CC)(C)C)ccc(C(=O)NC2CN(C(c3cnsn3)=O)CC2F)cc1 C1(C(=O)NC2CCC(N(C(=O)CNC=O)C)CC2)OCC2COCCC12 CN1N=C(CC(=O)N2CC(CNC(=O)CC3(O)CCOC3)CC(C)(C)C2)CC1=O N1(C(C2CN(C(C)(C)C)C(=O)C2)=O)CCCC(C)(CNC(C2CCS2(=O)=O)=O)C1 C1(C(=O)NCC2C(NC(CCc3scc(C)n3)=O)C2)CC2C=CC1C21CC1 c1(C(=O)NC2CN(C(C(n3cnc(C#N)n3)C)=O)C2)ccc(F)c(C(C)(C)F)c1 N1(C(C(C)N2CCCC2)=O)CCC(O)(Cc2ccc(Br)o2)CC1 C(=O)(C(CC(C)C)N(C)C(c1cc(C(N)=O)co1)=O)NCC(C#C)C(C)C Cc1ccn(CC(=O)N(C)CC2CCN(C(C3C4COCC34)=O)CC2)c(=O)c1 N1(CC(c2ccccn2)(C)C)CCC2(CC(=O)NC2=O)C1 C(=O)(CCCC(C)(F)F)N1C(CCCNC(Cc2c(C)ncs2)=O)CCCC1 N1(C(c2nccc(C)n2)=O)CCCC(NC(=O)CN(C)C(=O)C2CC2)C1C C1(NC(c2ccc(N(C)C)nn2)=O)COCCN(C(C2(C)CCOC(=O)N2)=O)C1 N#Cc1ccc(=NCC(=O)NCCCCCNC(=O)CCCS(N)(=O)=O)[nH]c1 C=CCCCCCCCC(=O)NC(C)C(C(C)C)NC(c1ccc(C)c(N)c1)=O C1(NC(CSCCCC)=O)(CCSCC(=O)NC(c2ccco2)=O)CCC1 c1(N2C(C)CC(CNC(C3(COCC)CCC3)=O)C2)ncnc(Cl)c1[N+](=O)[O-] C(c1cnc[nH]1)=C(C)C(=O)NC(C1CCOC1)CNC(c1occc1Br)=O N1(C(CC(CC)O)=O)CC(C)(C)OC2(C1)CN(C(c1csc(COC)c1)=O)C2 c1(NCC2(C)CCCN(C(=O)COc3cccnc3)C2)ccnc2[nH]cnc12 Cc1ccc(C(=O)NCc2ccoc2C(=O)NCC2CCC3CC23)c(F)c1 CC1CN(C(=O)CC2CCCC2O)CC1CC(=O)N(C)Cc1cn[nH]c1 c1(NC(C2CCN(C(=O)C=CC3CCOC3)C2)=O)cnccc1CO C1(C2CN(C(c3cccc(C)c3N)=O)C2)(NC(C2CC(CC)C2)=O)CC1 C(CCCCC(=O)N1CC2CC(NC(c3cnn(C4CC4)c3Cl)=O)C1C2)OC CC1=C(C(=O)NCCC2(NC(=O)COc3c(C)cccc3Cl)CCC2)CCO1 C1(CC)CC(NC(=O)C(=O)N(C(C)COc2ccc(OC)cc2)C)CCN1 C1(OC)CCCN(C(c2cccc(COc3nc(C)cs3)c2)=O)C1C C(=O)(C1=C(Cl)CCC(C)C1)NCC1N(C(CCCC#C)=O)CC(C)(C)C1 C1(NC(=O)Nc2ncc(CCO)s2)CC2CC1(c1ccnn1C1CC1(F)F)C2 c1(CNC(C(=O)OCC)CO)cc2c(Cl)cccc2s1 C1(NC(C2(C#N)CCCC2)=O)CN(C(c2ccnnc2)=O)CC2(CCC2)C1 C#CCC(C)(C(=O)NCC1(CC)CCOC1)NC(C)=O Cc1ccc(F)c(C(=O)NCCC2(CNC(c3ccc(C)c(O)c3)=O)CC2)c1 c1(OC)cc(C(N2CCCN(C(c3cc(Br)oc3C)=O)CC2)=O)cc(C)n1 N1(C(C(C)(C)CO)=O)CCN(C(c2ccc(O)nc2Cl)=O)C2CCCCC2C1 C(=O)(CCCC(=O)NC(C)CCCNC(=O)CCN(C1CCCCC1)C)OC Cc1cc(N2CCCC2CN(C(=O)C(C)Oc2ccccc2)C)nc(C)n1 c1(OC)nccnc1C(N1CC(O)CC1C(=O)Nc1ccno1)=O N1(CCC)CCCC1C(N1CC(CN(C(=O)C(F)=C2CCCC2)C2CC2)C1)=O C1(CNC(COCC(=O)OC)=O)CCCCC1NC(=O)COCc1nc(C)no1 C(CC(=O)NCC1CN(C(c2cc(C)n(C(C)C)c2C)=O)C1)(C(N)=O)NC(C)=O C(CC(=O)NC1CC(N(C(=O)CC2C=CCC2)C)C1)N(CCC)C N1(C(C(C)(C)NC(C(C)Nc2ccc(C)cc2)=O)=O)CCOCC(C)(C)C1 CCN=c1cc(C(=O)NCCC2CCC(NC(=O)C3=NNC(=O)CC3)C2)cc[nH]1 c1(NCCNC(C(c2cccc(F)c2)C)=O)ccc(C(C2CC(CF)C2)=O)cn1 C1(C(NOC(N2CCCC(Nc3ncccn3)C2)=O)=O)CCC2(CC2)C1 N1(C(c2c(OC)ccc(C)c2)=O)CCOCC(F)(CNC(=O)C(C)C(C)(C)C)C1 N1(C(c2c(C)ccnc2)=O)CC(CC(=O)NCC(C)C(C)(F)F)CC1(C)C c1(CCC)nc(C(=O)N(CCC(C)NC(C2CCCOC2)=O)C)cs1 N1(C(c2cc(Cl)sc2C)C(=O)N(C(CC)(C)C)C(C)(C)C)CC(C)SC(C)C1 C12(CCCC(C)(C)C1)c1nnnn1CCCN2.c1(CC=CCCC)ccc(F)cc1 N1(C(CCC(=C)Br)=O)CCCN(C(c2cccc(C(=O)OC)c2)=O)C(C)C1 C(=O)(CC(C)P(C)(C)=O)NCCC1(O)CCN(C(c2c(NC)cnc(Cl)c2)=O)C1 C#CCCCC(=O)NC(CNC(c1ccnc(Nc2ccccc2)n1)=O)CC=C N1(C(Cn2c(=O)ccc(C)n2)=O)CC(NC(=O)C(C)C(F)F)C2(CCC2)C1 C1(NC(c2c(C)csc2)=O)CCC2(CC1)CN(C(c1cnnn1C)=O)C2 N1(C(C(CC=C)N)=O)CC=C(c2cccc(Cl)c2)CC1 Cc1ccc(CC(=O)NCCC(C)N(C)C(c2ccc(CO)c(F)c2)=O)cc1Cl N1(C(C=CSC)=O)C2CCCC1CC(NC(C1CCCC3(CC3)C1)=O)C2 C1(CCOC)(NC(=O)C(C)c2ncco2)CCN(C(=O)CCCN(C)C(C)=O)C1 C1(C)(C(=O)NC2CN(C(C(CCC)(C)O)=O)CC2F)Cc2ccccc2C1 c1(OCC(N2CC(C)C(NC(=O)CC3CNC(=O)C3)C2)=O)cc(Cl)cc(Cl)c1 c1(C(N2CCC(O)(C(C)NC(C3CCC3)=O)C2)=O)nnn2ccccc12 C1(C(=O)NCCC2(NC(=O)C3=CCCCO3)CCC2)CCn2c(O)nnc2C1 C#CC1(C(=O)N(C2CC(C)CC(C)C2)C)CCN(C(=O)Cc2ccccn2)CC1 c1(CCC(=O)N(C2CCN(C(c3ccco3)=O)C2)CCO)ccc2c(c1)CCO2 N1(C(C2(CC=C)CC=CC2)=O)CCC2(NC(c3cc(O)nc(OC)n3)=O)CC2C1 C1(C(N)=O)(OCC2OCCC2C(=O)NCCOCC(=O)NC)CC(C)(C)C1 c1(C(=O)NC2(C(=O)NCC)CC2)cnn2c(C)cc(C)nc12 N1(C(CCC(C)(C)C)=O)CC2CC(O)C1C2NC(c1cnc2[nH]cncc1-2)=O CC1(C(=O)NC2CCC3COCCC3C2)CC2CCC1CC21OCCO1 C(=O)(C(CCC(C)C)NC(C)=O)NCCC1(OC)CN(C(c2cnco2)=O)C1 c1(OC)cccc(C2(C(=O)NCC(C)(C(C)C)NC(C3CC3OC)=O)CC2)c1 c1(NC(C)=O)cccc(C(=O)NC2CN(C(=O)C(C)C3CC3)CCC2F)c1C c1(C(=O)NCC(c2ccccc2)NC(CC=C=C)=O)ncc(F)c2ccccc12 c1(C(=O)NC2C(CNC(C(=O)NCCC(N)=O)=O)C2)n[nH]c2c1CCCCC2 CC1C(=O)CCC(C(N2CC(CO)(NC(c3nccnc3Cl)=O)C2)=O)C1(C)C C1(N(C(C2(NC(c3nc(C)sc3)=O)CC(CO)C2)=O)C)CCCC1(C)O C1(CNC(c2cnc(NC(C3(COC)CC(=C)C3)=O)s2)=O)CCCC1(C)O N1(C(c2cn(CC=C)nn2)=O)CCC(F)(C(=O)NCC(CO)OC)CC1 C(=O)(C1CCc2scnc21)NC1CCC(NC(C(C=C)O)=O)C1 CCC(C)CC(C)C(=O)N(CCCNC(c1ccc([N+](=O)[O-])cc1)=O)C N1(C(COCC(C)(C)C)=O)CC(=O)NCC1C(N1CCSC2(CC2)C1)=O C1(NC(c2cc(C)[nH]c2)=O)CN(C(=O)C(C)OCCC(C)C)C2(CCC2)C1 c1(C(N(C2CCN(C(=O)CCC(=O)N3CCOCC3)C2)CC)=O)c(C)nsc1N c1(C(=O)NC2CN(C(CC(CCOC)(C)C)=O)CC2F)cccc(C#CCO)c1 N1(C(c2cn(C(C)C)nc2)=O)CCC2(CNC(c3ccoc3)=O)CCCCC12 c1(C(N2CCC(C)C2C(=O)NC2CCCC(O)C2)=O)cc(=O)n(C)cn1 CCC(O)C(C)(C)C(=O)N1CC2(CC(NC(=O)CC(C)(C)COC)C2)C1 Cc1cc(C(N2CC(C(C)NC(C3(CO)CCOCC3)=O)C2)=O)cnc1CC#N C1(F)(CNC(C2(C(=O)NC)CC2)=O)CCCN(C(=O)CCCCCC#N)CC1 C(=O)(C#CC1CCCC1)N1CC(C=C)(CC(=O)N(CC(F)Cl)C)C1 C1(C(=O)NC2C(CNC(C(C(=C)C)(C)C)=O)CCC2)CC2(CCOCC2)C1 c1(C(N2CCC(c3ccon3)C2)C(=O)NC)ccc(-n2cccn2)c(F)c1 C1(CC=C)(NC(c2cc(C3(C)COC3)no2)=O)CCN(C(=O)C(F)C2CCC2)C1 c1(C(=O)NCC2OCCCN(C(C(CC(=C)C)C)=O)C2)cc(C#N)ccc1O CC(C)(C)CC(O)CC(=O)NCCNC(c1ccc([N+](=O)[O-])c(C(N)=O)c1)=O FC(F)(Br)CN=c1[nH]c(=NCC2CC3CCCC(C2)C3(F)F)[nH]c2c(F)cccc12 Cc1cn(CC(=O)NCC2CC(O)(CNC(=O)C(Cl)=CCl)C2)c2ccccc12 S(=O)(=O)(c1ccc(NC2CN(C)C2)c(Br)c1)N1CC(CC)OCC1C N1(C(CC(C)NC(C2CC(O)C2)=O)=O)CC2(C)CC1CCO2 c1(C(C)NCC2(NC(C)=O)C(C#C)C2)cc(OC)cc(OCC)c1 C(=O)(C1=CCCOC1)N(CC(=O)NCC1CC(C)CO1)CCOC N1(C(c2ccc(OCC=C)cc2)=O)CC(NC(c2coc(OC)n2)=O)CC1(C)C CC(O)(CNC(c1cn(CCO)nn1)=O)CNC(c1cn(C2CC2)cn1)=O C1(C)(NC(CCN2CCN(C)CC2)=O)CCN(C(C2COCCO2)=O)CC1 n1(CC(=O)NCC2CN(C(c3c(C)c[nH]n3)=O)CC23CC3)nc2c(n1)CCCC2 CC1(C)CC(CNC(=O)C(O)C2CCC2)CN(C(=O)C(c2ccc(F)cc2)=O)C1 c1(-c2cn(C(C)CNC(N)=O)nn2)ccc(C(F)(F)F)cc1 C1(C(=O)Nc2ccc(C)nc2O)C2C(CN1C(c1cc(O)cc(O)c1)=O)C2(C)C c1(CNC(CSCC)=O)ccc([N+](=O)[O-])cc1C#N CC1CCCC1(C(N1CCC1(C)C)=O)NC(c1ccsc1C#N)=O C(C(C)(CO)NC(=O)Cc1cn[nH]c1)NC(C=C(COC)C)=O c1(CC(=O)NC2CC(N(C(c3ccn(CCOC)n3)=O)C)C2)nnc(S)n1C CCC(CC)CCCC(=O)NC12CC(C(=O)NC(C)C(C)(C)CN(C)C)(C1)C2 c1(C(=O)NCC(CC)(CC)NC(CSCC=C)=O)ccc2nc(C)n(C)c2c1 c1(C(=O)NCC(CC=C)NC(C2(C)CC2C)=O)cc(OC)cc(Br)c1O N1(C(C(CC)CCOC)=O)CCCCC2(CCN(C(C3CCOC3)=O)C2)C1 CC1(C)CCN(C(c2cccc(Br)c2F)C(=O)Nc2ccc(Cl)cc2)CCS1 c1(N2CCC(C(=O)NCCN)C2)cc(=O)c(O)co1 Cc1ccc(CONC(=O)CC2CN(C(C3CCC4CC34)=O)CC2C)cc1 c1(C(=O)NC(C)CNC(=O)CCOCC(F)F)cc(C(C)(F)F)n[nH]1 C=C(Cl)CCC(=O)N(CCC(C(C)C)NC(=O)C(c1cscc1Br)=O)C C1(NC(CCOCC)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CC2(CC2)C1 C1(C)(CC)CCC(C(N2CC=CC2C(=O)NC2COCC2N(C)C)=O)O1 c1(C(N2CCCC(NC(CC(=C)Br)=O)CC2)=O)ccc2c(c1O)CCC2 N1(C(C2COCC3(CCC3)O2)=O)CCOCC12CCC2 N1(C(CC(C=C)C)=O)CCCC(N(C)C(c2ccc(CCO)cc2)=O)CC1 c1(C(N2CC(CC=C)(NC(C3CC4C=CC3O4)=O)C2)=O)ccc(Br)c(C)c1 N1(C(C=Cc2nnc(C(C)C)o2)=O)CC2CCN(C(C3OCCC3C)=O)C2C1 C(CCN=c1[nH]c(=NC(C)C(C)C)[nH]c2cccc(F)c12)c1c(C)n[nH]c1 C(C1CCCCC1)=CC(=O)NCCCN(C(=O)Cc1cocn1)C(C)C N1(C(C(CC(C)C)C)=O)CC23CCCC2(C1)CN(C(c1occc1Br)=O)C3 C1(NC(C2OCCC(=O)C2)=O)CN(C(=O)CCc2ccoc2)C2CCCC12 N1(C(c2cn(C)c(O)n2)=O)CC2CCN(C(=O)CCCCCF)CC12 c1(C(N2CCC(NC(C3(CCC)CC3)=O)C(C)C2)=O)n[nH]c2c1CCSC2 C(=O)(C=CS(=O)(=O)CC)NC1(C2OCC2(C)C)CC1.C12CCCCN1C(=O)CC2 N1(C(C2(CNC(c3ccc(CO)o3)=O)CCCO2)=O)CCOC(CCF)C1 Cn1cc(CC(=O)NCC2CCCC2NC(=O)Cn2cnnn2)cn1 N1(C(CCCNC(=O)C2CC2)=O)CC2CCN(C(=O)CC34CCCC3C4)C(C2)C1 CC1ON=C(C(=O)N2CC(NC(c3c(F)ccc(O)c3F)=O)C3CC3C2)C1C CCCC(CCC)C(=O)NC1CCN(CCCOc2ccc(F)cc2)CC1 N1(C(Cc2c(C)con2)=O)CCC2CCN(C(=O)C3=CCSC3)C2C1 c1(CCc2ccc(C)o2)nc(-c2ccc(Cl)cn2)nn1-c1nc(Br)nn1C N1(C(c2cc(C(=O)OC)on2)=O)CC2CC(NC(C3CCOC(C)C3)=O)CC1C2 Cc1ccc(Cl)c(C(N2CCC(C(C)(C)CNC(C3COC(C)C3)=O)CC2)=O)c1 N1(C(c2n(CCC)ccc2)=O)CC(NC(C2CCCCCS2(=O)=O)=O)C2(CC2)C1 Cc1cccc2c1CN(C(=O)Cc1ccccc1NCc1c(F)cccc1Br)C2 c1(C(=O)NCC2(NC(=O)CN3CCc4ccccc43)CC2)n[nH]c2ccc(F)cc12 c1(C(=O)NCC2N(C(CC=C(C)C)=O)CCCC2C)cc2ncccc2[nH]1 N1(C(C2(C(=O)NC)CCC2)=O)CCOCCC1C(=O)NC1CCC=CCC1 N1(C(C(F)=CCC)=O)CCCC(C2CN(C(c3ccn(CC4CC4)c3C)=O)C2)C1 c1(OC)cccc(C(N2CCN(C(c3ccc(C)c(F)c3)=O)CC2CF)=O)c1N Cc1ccc(F)c(C(=O)NCC#CCNC(=O)CC2=CCCC2)c1O c1(C(N2CC(C#N)C(NC(C3CCCO3)=O)C2)=O)cccc2nc[nH]c12 c1(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)ccn2nccc2c1 c12c(C)nc(nc1O)SC2.c1(CC(COC)C(C)C)ccc(F)c(F)c1 C1(NC(C2OCC(C)C2)=O)CC2CCC1(N=c1[nH]nc(C3CC3)o1)C2 C1(C(N2CCC(N(C(c3cccc(C)c3O)=O)C)CC2)=O)CC2CCCCC2O1 C1(NC(C(CCC)C)=O)CC(O)CN(C(=O)CCc2cccnc2F)C1 C1(NC(c2cn(CC)nc2C)=O)CCN(Cc2cccc(F)c2F)CC1(C)C C(C)(N=c1[nH]c2cc(C)cnc2s1)c1cc(O)cc(OC)c1.N1(CC)CCCCC1 C1(N(C(CCNS(C)(=O)=O)=O)CC2CC2)CCN(C(=O)C(C)(C)C#N)CC1 C(=O)(C(O)C(C)(C)CC)N1C(C(=O)NC2(C=C)CCCC2)(C(C)C)CCC1 C1(C(=O)NCC2CCN(C(c3n(C(C)C)ncc3)=O)C2)CCS(=O)(=O)C1(C)C CC1C(NC(=O)Cn2nccn2)CC2CCC1N2C(=O)CN1CC(=O)N(C)C1=O CC1(C)CCCC(C(=O)NC2CC(C)(NC(=O)CNS(=O)(=O)C3CC3)C2)O1 C1(C(CNC(=O)C(F)=CC2CC2)F)CCN(C(C2CC3C=CC2C3)=O)CC1 c1(C(N2CC(C(C)NC(COC)=O)OCC2)=O)cc2nc(=O)ccn2[nH]1 N1(C(C2(SCC)CC2)=O)CCN(C(c2cc(CC)ccn2)=O)CC1CC CCC1(CNC(=NCC(C)CC)NCc2cccs2)OCCc2ccccc21 C1(CC(=O)NCCC(C(C)C)CC(=O)NC(C2CCOC2)=O)CCC(C)(C)CO1 Cc1cc(=NCC2(F)COCCOC2)[nH]c(N2CCN(C3CCOCC3)C(=O)C2)n1 Cc1cccc(CNC(C2CCC(n3cc(CCOC(=N)O)nn3)C2)=O)c1F CCCCCCCCCCCC(=O)N(C1(C(=O)N(CCO)CCO)CC1)C C(C(=O)NCC=CCNC(c1ccsc1C#N)=O)(C(C)C)SC N1(C(C(C(CC)O)C)=O)CCC2CN(C(c3cc4nc(C)sc4[nH]3)=O)CC2CC1 c1(C(N(C(C)C(N2CCC(OCCN(C)C)C2)=O)C)=O)cc2ccccc2cn1 CCC(CCCC(=O)Nc1cnccc1C)NC(C1(C)CCCCC1)=O CCC(CC(F)(F)F)C(=O)N1CC(CNC(c2c[nH]nc2C2CCC2)=O)C(C)C1 C(=O)(C(CNC(C1CCC(=O)N(C)C1)=O)C(C)C)NC(C(CC)C)CO c1(C(C)NC(N)=O)cn(CC(N2CCCC2CNC(=O)CC2(O)CCC2)=O)nn1 c1(OC)ccc(F)c(C(N2CCCCC23CC3)C(=O)Nc2ccccc2Cl)c1OC N1(C(c2c(OC)ccnc2)=O)CCC(CC(=O)NCC(O)C(N)=O)C1(C)C c1(CC(N2CC(O)(CCc3cn(CCC(C)C)nn3)C2)=O)ccc(Cl)nc1 C1(C(N(C(C)CCNC(=O)CCc2c[nH]c(=N)[nH]2)C)=O)CC2C=CC1C2 CCC(C)C(C(=O)N1CC2(C)CC1(C(=O)N(C)Cc1ccoc1C)C2)OC CCCCCC(CC)C(=O)N1CCC(C)(NC(c2ccc(OC)nc2F)=O)C1 N1(C(CC2CCC(=O)C2)=O)CC2(C=C(C(=O)NC3CCC(O)C(O)C3)CO2)C1 C(=O)(C(F)C(C)C)NCC1(C(N)=O)CN(C(c2n(COC)ncc2)=O)C1 C(=O)(C1CCCn2cnnc21)N1C(CC)CN(C(=O)CCN(CC)CC)CC1 C(CCCCCC(=O)N1CC(C(=O)O)C2(COC2)C1)S.N(C)CC C(=O)(C(=O)C(C)(C)C)N.C1(CN(CC)CC)CCCCN1C(=O)C(F)n1cccn1 C12(C(=O)NCC3CC(NC(CN(c4ccccc4)CC)=O)C3)CC=CC(C1)OC2 C1(C(N2CCC(N3CCC(CN4CCOCC4)C3)C2)C)OC(=O)CC12CNC2 C12(NC(C3CN(C)c4c3cccc4)=O)CN(C(=O)CCC3CC3)CC1CS(=O)(=O)C2 N1(C(CN2C(C)CC2)=O)CC2CC2(NC(c2ccc(CNC(N)=O)cc2)=O)C1 C(C)(c1ccccc1C)=NC1(CC2CC(COC)CN2C=O)C(C(=O)OC)C1.C1(C)CC1 C1(NC(C2CCC(CNC(c3c(C)nns3)=O)O2)=O)CC(=O)N(C(C)C)C1 c1(-c2[nH]nc(C(C)Nc3cn(C(c4ccccc4)C)nn3)n2)ccc(F)cc1F CCCCCCC(C)C(=O)NCC1=CCCN(C(=O)CN(C)C)C1 Cc1cnn(C(C)C(=O)NCC2(O)CN(C(=O)C(C)(C)c3cnco3)C2)c1 c1(NC(C2(O)CCN(C(C(C=CC)O)=O)C2)=O)cc(OC)ccc1C C1(C(N2CC(C)N(C(=O)CC3NC(=O)NC3=O)CC2)=O)CCc2nc(O)[nH]c2C1 N1(C(c2cnc(COC)s2)=O)CC2CC1CN2C(=O)C=Cc1cc(F)c[nH]1 N1(C(C2CC(N(C)CC)C2)=O)CCCOC(CNC(=O)C(C2CCCCC2)O)C1 C1(CC(=O)N(C2CN(C(=O)Cn3cc(Cl)cn3)C2)C)C=CCCC1 N1(C(Cc2cc(COC)on2)=O)CC(NC(c2csc(O)n2)=O)C(SC)C1 c1(SCC)cccc(CC(N2CCN(C(=O)C(C)C(=O)OC(C)(C)C)CC2)=O)c1 CP(C)(=O)c1ccc(C(=O)NC2CCN(C(C3OCCCO3)=O)C2)cc1 C(=O)(C1CCc2c(Cl)cccc21)NC1(C2CN(C(CC(=O)OC)=O)C2)CC1 CC(C)(C)S(=O)CCCN=C(NCC1CCCCO1)NCC1C=CCC1 c1(OC)c(C(=O)NC23CC(C2)N(C(=O)CC2(CO)CC2)C3)cccc1F N1(C(CC(C=C)c2ccccc2)=O)CC2(CCN(C(C3(C#N)CC(C)C3)=O)C2)C1 C(CCC(C)C)(C(=O)NCC1C(=O)NCCC1C)NC(C)=O C1(NC(C2CCN(C(c3cc(=N)[nH][nH]3)=O)C23CC3)=O)CCc2nn[nH]c2C1 C(CC(CC)C(=O)N1CC(O)(CNC(=O)COc2cn[nH]c2)C1)=CC c1(OC)cc(C(C(=O)NCC(CO)NC(c2occc2C)=O)SC)c(F)cc1O Cc1cc(C)c(C(=O)NC2CCN(c3ccccc3F)CC2)c(O)c1 C=CC1(C(=O)NC2CCCC2)CCN(C(C2CCOC(C)(C)C2)=O)C1 c1(C(C)NC(CCCOC)c2nnnn2CC(F)F)ccc(OC)c(C)c1 N1(C(C(CC)SC)=O)CCCC(F)(CNC(=O)C=NOC)C1 N1(C(CC2CC(C)C2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 c1(C(=O)NCC(C)(CC)NC(C(COCC)C)=O)cncc(C(=O)OC)c1C C1(C(=O)NCC2CCN(C(Cc3nnc(C)o3)=O)CC2)CCCNS1(=O)=O C(=O)(C(C)(F)C(C)(C)F)N1CC(CNC(=O)CCC(C)(C)F)CC(C)C1 C1(C(=O)NCC(CNC(C(C)NC(CC)(C)C)=O)C)CCS(=O)(=O)CC1 C1(CNC2(C)CN(CC(=O)OC(C)(C)C)C2)CCC(c2ccccc2)CC1 Cc1nccnc1C(=O)NCC1CCCN1CC(=O)NC1CCCC1 C12(CNC(c3ncn(C(C)C)n3)=O)CC(CO1)N(C(c1cccc(=S)n1O)=O)C2 c1(N2C(C(=O)Nc3ncc(C)nc3Br)CC3(CC3)C2)nc(Cl)c2c(ccn2C)n1 CC1(C)OCC2CC12C(=O)NCC(C1CC1)NC(C1C2CCCCC12)=O CC(CC(=O)N1CCCC1CNC(c1ccnn1CC#N)=O)CC(C)(C)C C1(CNC(c2cnc(C(C)C)[nH]2)=O)CN(C(=O)C(c2ccccc2)F)CC1(F)F C(=O)(C(C(C)C)c1ccc(Cl)cc1)N1CC(CC(=O)OC)(C(F)(F)F)C1 Cc1c(C(N2CCC(OCCNC(C3CCCN3C(C)C)=O)C2)=O)ccn1C Cc1cnc2c(C(=O)NCC(C)(C)CNC(=O)CSC(F)(F)F)cccn12 CCC(CC(F)F)C(=O)NCCCN1CCN(c2nsc(NC(C)=O)n2)CC1 C(=O)(C(C)(C)C(C)(C)O)NC1CC(CCNC(C(C)OCC)=O)C1 c1(SC)ccnc(N2C3CN(C(c4cc(I)c[nH]4)=O)CC23)n1 c1(NC(C(N2CC3C(C)C3C2)C2C(CC)C2)=O)ccccc1C c1(OCC)cccc(C(=O)N)c1.c1(C(=O)N)n[nH]c(C)n1.C1CCOCCOCC1 C(C)(C)(CCCNC(c1cc(-n2cccc2)ccn1)=O)NC(COCC)=O C=CC(C)(CCOC)C(=O)NC1CCC(CCC(N2CCC(C(N)=O)C2)=O)C1 c1(C(C(=O)OCC)OC(c2c[nH]nc2CC)=O)ccccc1Cl C(=O)(C1=C(Cl)CCC(C)C1)NC1COCCN(C(c2c(NC)cncc2)=O)C1 c1(N2CCN(C(COC)COC)CC2)nccc2oc(Br)cc12 c1(C(C)(C)C)cnn(C)c1C(=O)NC1CC(CNC(=O)C=Cc2ccc(Cl)s2)C1 C1(C(N(CC(C)(C)CNC(=O)CC2CCCO2)C)=O)CCCC2(CCC2)O1 c1(CC(=O)N(CCCNC(=O)Cc2cc(Cl)ccc2O)C)nc2ncccn2n1 CCC(CC)C(C)C(=O)NCC1(CN(C)C(c2ccnn2C2CC2)=O)CC1 N1(C(C(C)C(C)(C)C)=O)CCC(C2(NC(=O)COCC3CCCO3)CC2)CC1 c1(CC(=O)NCCCN(C(c2ocnc2C)=O)CC)cccc2c1OC(C)(C)C2 S(=O)(=O)(c1cc(C)ccc1C)NCC(=O)NC(C(F)=CC)=O.C12CCC(CC1)C2 N1(CCc2c(OC)cccc2)CCC(NC(C2CCC(=O)N2)=O)CC(C)(C)C1 C1(OC)CN(C)C(C)(C(=O)NC2CN(C(=O)CCc3cncs3)C2)C1 CCCC(C)(O)CC(=O)NC1CCN(C(=O)C(=O)NC2CC2)C1 C(=O)(C1CCCc2ncnn21)N(CC(=O)N(C1CCCCC1S(C)(=O)=O)CCO)C C=CCC(CC(C)C)C(=O)Nc1cccc(NC(C2CCCNC2=O)=O)c1 Cc1cc(OCC(N2CCC(CN(C)C(c3cc(C(C)(C)C)no3)=O)C2)=O)no1 C(=O)(C(O)C(F)(F)F)NC1C(CNC(=O)CCCNc2ccccc2)CCCC1 N1(C(C(CC(CC)C)NC(c2ccc(C(C)C)o2)=O)=O)CCCC(C2(C)CC2)C1 N(C(=NCCNS(C)(=O)=O)NCc1cc(Br)cc(I)c1)C(C=C)C C1(C(N(CC(F)Cl)C)=O)CN(C(=O)C(C)(C)C2CCOC2)CC12CC2 C(CCC(F)(F)F)N(C(=O)CCCN(C)C(C1CCCOC1)=O)C C1(C(N2CCC3(C2)CN(C(C2(C4(O)CCC4)CC2)=O)C3)=O)CCC2(CCOC2)O1 C1(OC)CC(NC(=O)CC2CCSC2)CN(C(C2(C)CC2C)=O)C1 c1(C(N(C2CCN(C(C34CC(C)C3C4)=O)C2)C)=O)cccc2c1CCC2=O C1(C(NOCC(C(C)C)O)=O)CCC2CCC1N2C(=O)CCc1cnco1 CC1CCCn2ncc(C(=O)NCC3CC(NC(C4C(C)C4C)=O)C3)c21 CC1Oc2cc(C(N3CC(NC(=O)C(N)=O)C(C(F)F)C3)=O)ccc2NC1=O C(CN=c1[nH]c(=N)[nH]c(=NCC(C)Cn2ccnc2)[nH]1)c1c(OC)cccc1C C1(CN)CN(C(=O)Cn2cn[nH]c2=N)CC1C.Cc1occc1CC(=O)N1CCC1 C1(CC=C)(NC(C2CC23CCCC3)=O)CCN(C(=O)CS(=O)(=O)NC)CC1 C1(NC(C2(C#N)CCC2)=O)CN(C(c2ccc3c(c2)OCC3)=O)C2(CCOC2)C1 C1(NC(CC(C)(C)N(C)C(C2CCCC(C#N)C2)=O)=O)CCOC12CCCC2 c1(SCC)ccc(C(=O)NC2CCCN(C(C)=O)C2)c(F)c1 C1(C)(C(=O)NC2(C)CC(NC(c3ccn(CC(C)C)n3)=O)C2)CC2CC2C1 c1(-c2ccc(CCCC)s2)ccc(C(N2C(C(=O)O)CC2C(C)C)=O)cc1 C1(NC(CC(C)(C)O)=O)CC(C2CCN(C(=O)Cc3cc(F)ccc3Cl)C2)C1 CC(C)CCCCC(=O)NCCN(C(=O)CCC1CC1(F)F)C1CCCC1 C1(CCNC(=O)CSc2cncs2)COCCN1C(=O)C(F)=C1CCCC1 N1(C(C(CSC)O)=O)CCCCC1CCC(N1CC(F)(F)C1C1CC1)=O CC1CCN(C(=O)CN2CC3CC3C2)CC1NC(c1ccc(Cl)cc1N)=O C(=O)(CC1NC(=O)c2ccccc21)NCCNC(=O)NCCON CCC(CC(=O)NCCN(C(=O)CC1CC(F)(F)C1)CC1CC1)C1CC1 c1(C(N(CC(C)N(C(CCSCCCC)=O)C)C)=O)[nH]c2ccc(C)cc2c1C c1(C(=O)NC2C(NC(C3(CC#C)CCCC3)=O)CCC2)cncnc1C1CC1 C1(C(N(C(C)CNC(c2cnc(SC)s2)=O)CC)=O)CC(C)=NO1 c1(-c2n(C(COC)C)nc(C(C)C)n2)cc(Br)c2cccnn12 CC(C(=O)NCC1CC1C(=O)NCCN1CCC1)C(C)(C)C CC1CN(C(C2CC3(CCO2)CC3)=O)CCC1NC(c1cnc[nH]1)=O c1(C(N2CCC(N(C)C(C3CC4CC4C3)=O)C2)=O)ccc2c(c1)COC2 N1(CCNC(CCN(CC#C)C(C2CC2Cl)=O)=O)CCCC1=O C1(NC(C2(C=C)CC2)=O)C2CCC(C2)C1NC(=O)Nc1c(C)cccc1C N1(C(CC2(C)CCOC2)=O)CC2(CCN(C(=O)CCn3ccnc3)CC2)C1 CC(C)(C)CC(C(=O)NCC1CCCCO1)NC(c1cccn2ccnc12)=O c1(C(C(=O)NCCCOC)N(C2CCOC2C)CC)cc(F)ccc1C c1(C(N(C)CCC2CCCCN2C(=O)COC2CCCC2)=O)nnc(O)nc1O C1(C(=O)NC(c2cc(C)on2)C)CC2CCCC2N1C(=O)C=CC1CCCC1 Cc1ncccc1CC(=O)NCC1(NC(C2CCCN2N=O)=O)CC1 C(CN=c1[nH]c(N2CCn3cnnc3C2)nc2cccc(F)c12)OC(C)C CC1CN(C(Cn2cc(Sc3ccncc3)nn2)=O)CC(C)O1 CCCCCC(C)CC(=O)N1CC2(CCC2NC(c2cnn(C)c2SC)=O)C1 C=CCCCC(=O)N1CCCC1(CC=C)C(=O)Nc1cncc(C)c1 C1(C(N)=O)(NC(CC2C(NC(CC(C)O)=O)CC2)=O)CCCCC1 C(=O)(C(C)C(CC)CC)N1C(C(=O)NC(C#C)C2CC2)CCCCC1.C1(C)CCCC1 C(C(C)(C)CC(=O)NC1CN(C(=O)CSC)CCC1F)SC C1(N(C)C(C2CC2c2cnn(C)c2)=O)CCCN(C(C2(C)CC(F)(F)C2)=O)CC1 N1(C(CCC=C)=O)CC2(CC(NC(=O)COc3cnn(C)c3)CO2)C1 N1(C(CCOCCNC(c2c(COCC)nn(C)c2)=O)=O)CC(O)CC1(C)C c1(C(C(=O)NC2C3CN(C(C(C(C)C)SC)=O)C2C3)C)cc(C)cc(C)c1 c1(C2(C(C=C)N(C(C)CCC(=O)OCC)C3CC3)CC2)ccc(Cl)cc1 C1(NC(C2C(C)N(C)CC2)=O)CN(C(C2CC(N(C)C)C2)=O)Cc2ccnn2C1 N1(CCn2cc(CCCNC(CCc3n(CC)ccn3)=O)nn2)CCC(F)(F)CC1 c1(NC(C(C)C2CCOC2)=O)cnc(O)c(F)c1 N1(C(C2N(C)CCOC2)=O)CCC(C2(O)CN(C(C3CC4(C3)CC4F)=O)C2)CC1 c1(-c2cccc(NC(CC(CCC)NC(C)=O)=O)c2)ccc2cnoc2c1 CON1CCC(C(=O)NCCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CCO2)CC1 N1(C(C(COC(C)C)(C)C)=O)CC2CC(NC(c3ccc(C(N)=O)nc3)=O)C1C2 N1(C(CCSCC(C)C)=O)CCC(CNC(C2(N(C)C)CCCCC2)=O)CC1C C1(CC(N2CC(CC(C)CNC(C(N3CC(C)C3)C)=O)C2)=O)CCC(=O)C1 c1(C(=O)NCC23C(CN(C(c4scc(COC)c4)=O)C2)C3)cnc(Cl)c(N)c1 c1(C(=O)NCC#C)cc(OCC)nc(C)n1.C1CC(=O)NC2C(CC2)N1 C(=O)(C1=C(Cl)CCCC1)NCC(CCC)NC(c1ccn(CC)c(=O)c1)=O c1(OC)cc(OCc2ccccc2N2C(=O)C(C)C(C)C2=O)c2c(n1)CCCC2 N1(C(=O)Cc2cccc3c2OCO3)CC2CN(C(c3coc(CO)c3)=O)CC2C1 N1(C(C2CC2F)=O)CC2CN(Cc3ccc(C(F)(F)F)cc3Cl)CC2C1 C1(CC)CCC(C(=O)NCC(C)(C)NC(c2cc(C)ns2)=O)C1 C(CCCC(CO)NC(=O)CSc1n[nH]c(=N)s1)NC(C(CSC)C)=O C(CN=c1cc[nH]c(=NCCCC2(NS(N)(=O)=O)CCC2)[nH]1)N1S(=O)(=O)CCC1 c1(C(=O)OC)cc(N2CCC(C)(NC(c3ccc(Cl)s3)=O)C2)nc(C)n1 c1(C(N2CC(O)CC2C(=O)OC)=O)cc2ncccc2[nH]1.C12CC3(CC13)C(=O)N2 CC1CC(C(=O)N(CC(=O)N(C)C)C)N1C(=O)COc1cn[nH]c1 c1(N(CC(=O)NCC)CC)nnc(CC2COCCO2)n1CC N1(C(c2n(C)cnc2)=O)CCN(C(c2ccc(C(C)(C)C)s2)=O)C2CCC12 C12C=CCCN1C(=O)CC=CCNC2=O.n1(C(C)C)cnnc1C(C)C N1(C(CNS(C)(=O)=O)=O)CCC2(CCOC2)C(CNC(c2csnn2)=O)C1 c1(C(C(=O)NCCCC2CC2)NC(C(C)N(C)CC)=O)ccc(CO)o1 C1(C2CC2)(COC)CN(C(=O)C(C(C)C)NC(C2(O)CC2)=O)C1 C1(NC(C2(CC#C)CCN(C(=O)CC3CC(=O)C3)C2)=O)CCCCC1N=[N+]=[N-] N1(C(c2ccc(OCOC)cc2)=O)CCCC12CCS(=N)(=O)CC2 c1(C(=O)NC(CNC(C(C)(C)SC)=O)CO)cnc(C(F)F)nc1 Cc1nn(C)c(C)c1C(N1CCCC(CNC(=O)CN2CCC(C)(C)C2)C1)=O N1(CCCCC)CCOC2(CCN(C(=O)Cn3nc(C)c(C)c3C)CC2)C1 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CC(NC(C34CCCC(CCC3)C4)=O)CC1C2 N1(C(C(C)CC2CCCCC2)=O)CCC2(CCC2CNC(c2ccns2)=O)CC1 C1(C(N(CCC)CC)=O)CC(=O)CN1C(c1cc(CC)sn1)=O C1(C(N2CC(C(C)NC(C3CCC(=C)CC3)=O)C2)=O)CCOC2(CCOCC2)C1 c1(C(=O)NC2CN(Cc3c(F)cccc3F)CC2O)c(F)cc(F)cc1Cl Cc1nnc(O)c(C(=O)NCC2CN(c3nnc(C(F)F)o3)CC2C)c1C N=c1[nH][nH]c2ccc(C(N3CCC(O)C3C(=O)NC3CSC3)=O)cc12 C1(O)(C(N(C)CC2CCCN2C(C2CC3CCC2C3)=O)=O)CCCCCC1 S(=O)(=O)(c1c[nH]ccc1=NCC(CO)C1CCC1)N(CCC(O)C(C)(C)C)C C#CC1(C)CCCN(C(c2csc(C(=O)OC)c2)C(=O)Nc2ccccc2Cl)C1 CC1(C#N)CN(C(=O)C(Cc2ccoc2)NC(c2cnn[nH]2)=O)C1 Nc1[nH]c(=O)c(Cl)nc1C(=O)NCC1CCCCC1NC(c1cnns1)=O c1(C(=O)NCCCOCCNC(C2(C(=O)NC)CCC2)=O)c(Cl)ccc(C)c1O N1(c2cc(C)nc(NC3CC(C)C4=CCC3C4)n2)CCc2cc(F)cc(F)c2C1 n1(C(C)(C)C(=O)NC2CCC(CNC(C3CC(C#N)C3)=O)C2)cc([N+](=O)[O-])cn1 C(C)(CC(C)NC(=O)C(F)(F)C1CCCC1)NC(C1(CCCC)CC1)=O C1(NC(CSCC(=O)NCCCOC2CCC2)=O)C2CCC(=O)C12 N1(C(CC(C=C)c2ccccc2)=O)CC2(CNC(=O)CC(C)(C)C)CC1CO2 c1(CC(N2C(CNC(C3N(C)CCOC3)=O)CC2)=O)cccc(C(F)(F)F)c1Cl c1(C(=O)NC2C(C(=O)NCCC(=O)Nc3ccc(Cl)cc3)C2)cc(F)ccc1Cl C1(NC(c2ncc(Cl)cc2Br)c2n(CC)nnn2)CCOC2(CCCC2)C1 C1(NC(CCNC(C)=O)=O)CCCN(C(=O)Cc2ccccc2C)CC1F c1(C(=O)OC(C)CNC(c2cnn(C)c2)C(=O)OC(C)(C)C)ncc(F)cc1F C1(CC(=O)NCC(C)NC(C2(c3ccc(F)cc3)CC2)=O)CCOC(C)(C)C1 C(=O)(CC(C(N)=O)NCCCOCCC(C)C)OCC c1(OC)cc(N)ccc1C(=O)N(C)CCNC(=O)C(Cc1ccccc1)N(C)C N1C2CCc3c(cccc32)OC(C=C)(C)c2nnc1n2CCOC.C1(OC)CCCC1 C=CC(C)CC(=O)N(C)CCN(C)C(C1C(c2ccncc2)C1(C)C)=O C1(O)(CNC(c2n(C)c(S)nc2)=O)CCCN(C(C2CN3CCN2CC3)=O)C1 C1(O)(C(C(=O)NCC2C(CN(C)C)C2)F)CN(C(=O)Cc2cncs2)C1 C(CCC(=O)N1C(=O)CCCn2ccnc21)n1cc(CC(C(C)(C)O)O)nn1 N1(C(CSCC(=O)OC)=O)CCCCC1CCC(N1CCCC1C(C)(C)OC)=O C(=O)(C(C)CC(F)(F)F)NC1CN(C(C2CC(C(C)C)C2)=O)C(CO)C1 c1(C(N(CC(CNC(C(c2ccc(Cl)s2)C)=O)O)C)=O)ccnnc1S CC(C)(C#N)CC(=O)N1CCC(O)(CCNC(=O)CS(=O)(=O)NC2CC2)CC1 C1(ONC(C2(NC(C=CC(=O)N(C)C)=O)CCC2)=O)CCCC1C n1(CC)c(C(=O)NCC(C)(CO)NC(=O)CCCn2cccn2)cnc1O c1(CC(=O)N(C2CCN(C(C3(O)CC3(C)C)=O)CC2)C)ccc2c(c1)CCC2 C12(C(=O)OC)CCC(C(=O)NCCC3(O)CN(C(C4CCCO4)=O)C3)(C1)C2 c1(CCC(N2CCC(CNC(=O)CC3CC3)C2)=O)ccc(Br)c(F)c1 c1(C(=O)NCCC2CN(C(C3COCC(C)O3)=O)C2)ccc(F)c(Cl)c1F C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCOC(C)C1C(=O)O Cc1cc(C(=O)OCCOC2CC(OC(=O)OC(C)(C)C)C2)nc(Br)c1 N1(C(CC2(OCC)CCC2)=O)CCC(C)CC1C(=O)Nc1cccc(C(C)C)c1 N1(Cc2n(C)nc(-c3ccsc3)n2)Cc2ccc(F)cc2C1 c1(OC)cccc(C(F)(F)C(=O)NC2CCCC2NC(=O)Cn2nnnc2C)n1 C1(NC(CCOCCC)=O)CN(C(C2CCC(C)(C)O2)=O)CC2CCCC12 N1(C(C2C(C)C2)=O)CC(CNC(=O)CC2=NNC(=O)C2)C2(CCOCC2)C1 N1(CCN2CCOCC2)CCCc2cc(C(c3ccc(OC)nc3)O)ccc2C1 c1(OCC)ccc(F)cc1COC(=O)C(N1CCCC(c2nc(C)nn2C)C1)=O C#CCC(CC(F)F)C(=O)N1CCC(CCOC)(NC(C2CN3CCC2C3)=O)C1 N12CC(C(CS(C)(=O)=O)C1)C2=O.c1(NC(COC(C)=O)=O)cccc(F)n1 c1(COC)ccc(C(=O)NCC(O)CNC(=O)Cc2cccnc2OC)cc1C c1(C(N(CCNC(C(CO)N(C)C)=O)CC2CC2)=O)cc(O)nc(N(C)C)n1 Cc1c(CCC(N2CCC(C)(NC(=O)CC3C=CCCC3)C2)=O)cnn1C CC1CN(C(C2(CCF)CCC2)=O)CC1(C)CNC(c1cc(Br)sn1)=O N1(C(C2C(C(C)C)C2)=O)CC(NC(c2cccc(OCC3CC3)c2)=O)C(F)C1 C#CC1(CNC(=O)CCC2CN(C(=O)Cc3ccccc3O)CCO2)CCOCC1 N(C(=NCCCCCCSC)NCC1COC1)CC1C(OC)CCC1 C(=O)(CCCCCC(C)O)NCC(C(C)(C)C)NC(c1c(CC)[nH]c(=N)s1)=O C1(NC(C=CC)=O)CN(C(=O)CSc2ccc(C)c(C)c2)Cc2nccn2C1 N1(C(C2(COC)C=CCN2C(=O)Cc2ccsc2C)=O)CC=C(CO)CC1 CCCCCCCCC(=O)N(CC(C)CNC(c1nc(O)c(C)s1)=O)C C1(C(N(CC)CC2CCCCO2)=O)CCC(NC(=O)Cn2cnnn2)CC1 C1N=C(NC2CC=CCC2)NCC2CCCC12.N1(S(C)(=O)=O)CCCC1 C1(C)(CNC(C2CC(C)OCC2)=O)CCCN(C(C2(F)CC2)=O)C1 C=CCC(CC)C(=O)NCC1CC(OC)CN1C(c1cc(Br)sn1)=O c1(NC(N2CCCC(NC(=O)CN3CCOC3=O)CC2)=O)ccc(Cl)c(F)c1F CC1CC(NC(C2(C(F)(F)F)CCC2)=O)CCN1C(=O)CCC1CC1 C(=O)(C(CC(=C)Cl)NC(C1CCC(F)C1)=O)NC(C#C)(C)C O=C1OC2CC(C(N3CCCN(C(C4CC(CCO)C4)=O)CC3)=O)CC2O1 c1(OC)ccnc(F)c1C(N1CCCC(C(C)NC(c2cc(CF)on2)=O)C1)=O CN1CC(O)CC1(C)C(=O)NCc1cc(C(=O)NC2(CCF)CCC2)on1 C1(N(C(CC(C)OCC2CCCCO2)=O)c2ccccc2)C2CN(C3CC3)CC12 N1(C(CC2(NC(C(n3ncc(C)c3)C)=O)CC2)=O)CCCC2(CCOC2)C1 C1(C(=O)NC(CNC(c2c(C)nn(C(C)(C)C)c2)=O)C2CC2)CC(C)(C)CN1C c1(C(N(CC(CNC(C(c2ccnn2C)C)=O)O)C)=O)cc2c(nn1)CCCC2 C1(C(=O)NC(CCCC=C)C2CC2)CC12CCN(C(=O)C1=CCSC1)C2 C1(C(=O)NCCCNC(C(C2CCCCC2)N(C)C)=O)C(C#N)C1(C)C c1(C(N2CCCC(N(C(COCCCC)=O)CCF)C2)=O)cnn2ncccc12 CC1CN(C)C(C)CC1NC(C1C(CNC(C2(C)C=CCCC2)=O)C1(C)C)=O Cc1ccc(Br)cc1CC(=O)NC12CC1CN(C(=O)C(C)Cc1ccco1)C2 N1(C(CC2(OCC)CC2)=O)CC(NC(c2ccn(C)c2)=O)CC(O)C1 C=CCCC(CC(C)C)C(=O)N1CC(CNC(c2ccnc3nccnc23)=O)C1 c1(CC(=O)NCC(CC)NC(=O)CCc2nc(SCC)no2)cccc(C)c1C C1(C(N(CCCO)CC)=O)CCOC1CNC(=O)CCCc1cnn[nH]1 c1(C(C)C)nnc2cc(N3CC(NC(C4CCC4(C)C)=O)CC4(CC4)C3)ncn12 N1(C(C(CCC)OC)=O)CCN(C(C2CCCC2OC)=O)CC1C1CCCC1 C=Cc1ccc(C(=O)NC2COCC2NC(=O)C(CC(C)C)NC(N)=O)cc1 CC(C(=O)NCC1(C)CCN(C(C2(c3cc[nH]n3)CC2)=O)CC1)C(C)(F)F c1(N2CC(CNC(CNC(CCC(C)C)=O)=O)C2)ncnc2sc([N+](=O)[O-])cc12 C1(C2CC2)(C(N2CCC(COC)C2)=O)CN(C(=O)C(C)N=[N+]=[N-])C1 CCCCS(=O)(=O)NCC(=O)N(C)CCN(C(=O)C(c1cnn(C)c1)OC)C c1(C(N2CCC(CNC(C(CC)(CC)CC)=O)C2)=O)cnc2ccc(C)cc2c1 C(c1ccccc1C)=CC(N1CCC(N(C(CSC)=O)CC(C)C)CC1)=O N#Cc1cc([N+](=O)[O-])ccc1C1CCCN1C(=O)NCCCc1cccnc1 c1(C(=O)NC2C3C(C)N(C(=O)CO)C2C3)cc2c(cc1Br)OCCO2 c1(N(CC(C)CNC(=O)C(C)(C)C(F)F)C)nc2ccccc2cc1[N+](=O)[O-] C1(N(C(COC(CC)C)=O)CC)C2CN(C(c3cnoc3C3CCC3)=O)CC12 Cc1ccc2c(C(=O)NCC3CCN(C(C4(F)C(C)(C)C4(C)C)=O)C3)onc2c1 c1(OC)ccc(Br)cn1.c1(C2C(=O)OC2COC(C)(C)C)cnn(C2CC2)c1 CC1CN(C(=O)COCCCF)CC1C(N1CCC(C(C)(C)C)CC1)=O N1(C(C=C(C)C(F)F)=O)CCC(N(C(=O)CC2CCC(C(F)(F)F)O2)CCO)C1 c1(C(=O)NCC2CC(c3cc(Cl)cc(Cl)c3)C2)[nH]cc2c1CCCC2 C(=O)(C1=CC2(CCOC2)C1)NC(CC(C)NC(c1c(C)nc(CC)nc1C)=O)C C1(C(N2CCCCC(NC(CS(N)(=O)=O)=O)C2)=O)CCc2[nH]nc(O)c2C1 c1(C(N2CCC(N(C(c3c(SC)n(C)nc3)=O)C)C2)=O)cccc2ncnn12 CCCCC(C)C(=O)NCC1CC(O)(CNC(c2cnc(C(C)C)nc2C)=O)C1 N1(C(c2cc(COC)sc2)=O)CCCCC(NC(=O)C(C)(C)c2cccnc2)C1 c1(C(=O)NC2C(NC(C(C)SC)=O)CC2)ccc(O)cc1[N+](=O)[O-] CCCC(CNC(C1CC(=O)C1(C)C)=O)C(=O)NCc1cn(C(C)C)nn1 C1(NC(C2C(C)(C)C2c2ccccc2)=O)CCCN(S(N)(=O)=O)C1 C(CC1CC1)(C(=O)NC1CCSC1)NC(=O)CCC1CC1 C1(CC)CN(C(c2ccc(CNC(=O)C(=O)NC(C)C)o2)=O)C(CC)CO1 N1(C(CCCC(C)C)=O)CCCN(C(=O)COCC(C)(C)C)C(C)C1 C1(CC(=O)NCC(C)(C2CC2)NC(CC(C)c2ccncc2)=O)CC(C)(C)CO1 C(CC(CNC(=O)CCN(C)C(C)=O)NC(=O)C(CO)c1ccccc1)OC C(CCCOC)(C(=O)N(CCO)CCOC)NC(C(C=C)CC)=O C12(NC(=O)Nc3cc(Cl)ccc3Cl)CCC(CC1)N(C(=O)CCC(F)(F)F)C2 Cc1c(C(=O)NCCC(C)NC(c2sccc2F)=O)nn2c1CCCC2 C(CC1C(=O)N1)N(C)C(C1CC2(CSC2)C1)=O.c1(CN)cccc(C)n1.CO c1(C(N2CCC(CC(=O)NC(C34CCC(CC3)C4)C)C2)=O)ccc(O)nn1 CC(C)CC(CC(=O)NCc1nncn1C1CC1)NC(=O)C(C)(O)CC(C)C N1(C(C2(C3CCCCO3)CCC2)C)C(=O)CCN(Cc2csc(C(F)(F)F)c2)C1=O C1(CC(=O)N(C(CC)CO)C)CCCN(C(C2CCN(C)C2C)=O)CC1 N1(C(COC(CC)CC)=O)CC=CC(C(=O)NCC2(O)CC2)C1 C=CCCC(=O)NCC(CNC(c1cn(C2CCCC2O)nn1)=O)CO C=CCCC(O)Cc1ccc(NC(N2CC(C(=O)NC)C2)=O)cc1 c1(C(=O)NC)c(NC(C2CC3CC3N2Cc2cncc(CC)c2)=O)cccc1Br Cc1ccc(CC(=O)NCCC2(C(=O)NCC3CCN(C)C3)CCCC2)o1 C1(C(=O)N(O)Cc2cn(CC3CCOCC3)nn2)NCCC12CCC2 c1(CNC(n2ccc3ccccc23)CC)cccc([N+](=O)[O-])c1 c1(C(N(C2CCN(C(c3cn(CC(C)C)nc3)=O)C2)C)=O)cc[n+]([O-])cc1 C1(NC(C(CC#C)O)=O)CCCCN(C(=O)CC2CSCCO2)C1 C1(NC(CCCOC)=O)CCN(c2cc(-c3ccco3)nc(C3CC3)n2)C1(C)C C(=O)(CC(C(F)F)NC(c1ccnnc1O)=O)N1C(CC)CC(C)C1 C1(O)(CC=O)COC(C)(C)C1.C1(SCC)CCC(NC(C2CCN(CC)C2)=O)CC1 CC1CN(C(=O)CCCC2CCC2)CC(C)N(C(c2cc(N)cc(F)c2)=O)C1 N1(C(C(C2CCOC2)OC)=O)CC2(CCN(CC3CCCCCC3)CC2)C1 c1(C(=O)NC(C(=O)NCC(CO)NC(C)=O)C2CCCO2)cc(CO)oc1C C1(N)CCN(C(=O)CC(C)(C)N(C(=O)CCC2CC(OC)C2)CC)CCO1 C(C)(C)(CC(=O)N1CCOC(C2CN(C(=O)C(C)SC(C)C)C2)C1)SC C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NCC1C(NC(COC(C)=O)=O)CCCC1 C(=O)(CCC(F)(F)C(F)F)N1CC(NC(C(C(=O)OC)(C)F)=O)C1 N1(C(C(CCC)OC)=O)CC2CCC(C(=O)NCC3C(C)(C)C3(C)C)(C2)C1 C1(C(=O)NCC(CN(C)C(c2cnccc2Br)=O)O)C(F)(F)C12CC2 C1(C)(C(N(CCOC)CCNC(=O)Cc2nocc2C)=O)CC=CCC1 C1(NC(C(C)(C)OCC)=O)CC2CC(NC(c3ccccc3SC(F)F)=O)CC12 CN1CCN(C(=O)C2=CCSC2)CC1C(=O)NCC12CCC(CC1)CC2 C(=O)(C1=NOC2(CCOC2)C1)NCC12C(CN(C(CNC=O)=O)C1)C2 C1(C(=O)NOC2CCCC2)C2CN(C(=O)CC3CC4CC4C3)CC12 CCC(C)(CC)C(=O)NC12CC(CNC(c3cnn(C)c3N)=O)(C1)OC2C CCC(C(=O)NC(C)CC1CN(C(=O)CNC(=O)CCC(C)C)C1)C(C)C N1(C(c2sccc2Br)C(=O)Nc2ccc(OC)cc2)CC2CCC1C(O)C2O N1(C(CCC(C)SC)=O)CC(C)CN(C(=O)Cc2c[nH]c(=N)nc2O)CC1C C1(NC(C=CCNC(c2cnn(CC)c2C)=O)=O)CCC2(CCC2)C1 N1(C(CCCOC(C)C)=O)CCC2(CC1)CCN(C(C1CCCN1C)=O)CC2 C1(C)(CC(=O)N(CCOCCN(C(=O)C(C2CC2)C2CC2)C)C)CCCO1 CCCCC(C)(F)C(=O)N1CCC1Cn1cc(CN2CCS(=O)CC2)nn1 CCC(C(=O)NC1CC(NC(c2cc(O)nn2C)=O)C1)C(C)(F)F N1(C(CC(C)C)=O)CCC(CNC(C2CC2c2ccsc2)=O)C1(C)C c1(C(N2CCC(NC(Cn3nnc(C)n3)=O)C2(C)C)=O)nn2cccnc2c1Cl c1(C(=O)OCC(=O)Nc2ccc(F)cn2)ccccc1-c1nc(C2CC2)no1 S(=O)(=O)(c1ccc(Br)c(C(=O)OC)c1)N1CC=C(CNC)CC1 C1(C)(NC(c2c(C)cco2)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 C12(CNC(Cc3cccc(SC)c3)=O)CCCOC1CCN(C(=O)C(C)S)C2 N(C(=NCCF)N1CCC(c2cccnc2)C1)Cc1nc(COC)on1 Cc1cc(C(=O)NC2CCCN(C(C3(CO)CCCO3)=O)C2)c(Br)cn1 c1(NC)cc(C(=O)NCC=CCNC(c2occc(=O)c2OC)=O)cc(Cl)n1 C1(NC(=O)NC23C(C)(C)OCC2C3)CCc2c[nH]nc2C1 c1(C(C(=O)NC2COC2)N(C)Cc2ccncc2)cc(F)nc(F)c1F c1(C(N2CC=CC(NC(Cc3ccc(C)nc3)=O)C2)=O)c(C)oc(C)c1C c1(C(=O)NCCC(C)(C)NC(Cc2c(C)ncs2)=O)[nH]cc2c1CCCC2 N1(C(c2cc(C(C)(C)C)on2)=O)CCC2CN(C(N3CCC(O)CC3)=O)CCC12 c1(C2(NC(=O)NC3C(SCC)COC3)CC2)ccccc1F Cn1ccc2cc(C(=O)NCC3CN(C(C4CC4CN(C)C)=O)C3)cnc12 c1(C(C(=O)N(CC(C)C)CC(=O)NCC2SCCS2)=O)cccn1C C1(NC(C2C(C)C2)=O)CC2CC1N(C(C1(c3ccc(F)cc3)CCCCC1)=O)C2 c1(CC(=O)OCC(=O)N(CCC#N)CC)ccc(F)cc1CC c1(NC(C2(CNC(CC(C=C)c3ccccc3)=O)CCC2)=O)ccc(N)c(O)c1 c1(C(N(C2CN(C(C3CCC(C)(CC)O3)=O)C2)C)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(C(COCC)C)=O)Cc2[nH]nc(C(N3CC(CC)OC(C)C3)=O)c2C1 CC1(CNC(=O)Cc2ccc(CO)cc2)CCCN1C(c1ccsc1Cl)=O Cc1cc(C(=O)NCC(C)NC(=O)CC(C)(C)C#N)cc(C)c1F C1(CCN(c2ncc(Br)s2)C)CC2CC1C1CCCC21 c1(C(=O)NCC2C(NC(c3c(CCC)nco3)=O)CC2)cc2cccc(C)c2[nH]1 C1(NCC(=O)NC(C(=O)N(c2cccnc2)CC)c2ccoc2)CCC(C)C1 C1(NC(=O)NCCSC)COCCC12CN(C(=O)OC(C)(C)C)C2 N1(C(CCC=CC(C)C)=O)CCC(C(=O)NCCc2ocnc2CO)C1C CC(C)(C)CCCCC(=O)N1CC=C(CCNC(C2CN3CCC2C3)=O)CC1 C1(CNC(CNC(C)=O)=O)CC(NC(=O)CSc2ccc(Cl)cc2)C1(C)C c1(C(N2CC(C(C(=O)NCC#CCCO)OC)C2)=O)ccc(C#N)n1C c1(N2C(C)(C)CC(C(=O)O)CCC2)ncnc2c([N+](=O)[O-])cccc12 c1(OC)cccc2sc(NC(CN(C)C)CC(C)C)nc12 C1(NC(C)=O)CCN(c2cc(C)nc(CC3(O)CCCC3)n2)C12CCCC2 C(=O)(C(C)CCCCCC)NCCC1CC(C(=O)NC(CC(=C)Cl)CO)C1 c1(C(=O)NCCC(C)(CC)NC(C(CC)OC)=O)cnc(OC)nc1C(F)F c1(OC)ccc(-c2ccc3c(c2NC(=O)CCS(C)(=O)=O)OCO3)c2cn[nH]c12 N1(C(c2ccc(CC)cc2)C(=O)NC(C)C)CCCN(c2ccccc2C)CC1 Cc1[nH]nc(C(=O)NC2CCC2CNC(c2ccc(CO)c(Cl)c2)=O)c1[N+](=O)[O-] C1(NS(CC)(=O)=O)CC2(C1)CN(C(c1ccnc(Oc3cccc(Cl)c3)c1)=O)C2 CCCCCCCCC(=O)N1CCN(C(C2CC3(C2)CC(CO)C3)=O)CC(C)C1 c1(OC)n[nH]cc1C(=O)N(CCCNC(C1CCC1C(C)(C)C)=O)C N1(C(c2onc(COC)n2)=O)CC2(C1)SCCC2NC(c1csc(O)n1)=O N1(CC(CCC(=O)OCC)CC)CCn2c(C(F)(F)Cl)nnc2C1 n1(CC)cc(CNC(=O)NC(C(F)(F)F)c2ccccc2)c(C)n1 C=Cc1cncc(C(=O)NC(C2CCN(C(C3CCC(C)(C)CO3)=O)CC2)C)c1 c1(CC(=O)N(CC(C)NC(c2ccnc(F)c2F)=O)C)cc(F)cc(F)c1 S(=O)(=O)(c1nc(NC2CCc3c(n[nH]c3C)C2)ccc1Br)NC(C(CC)CC)C C1(C(=O)NCCCCCNC(c2c(C(=O)OC)n[nH]c2)=O)CCCN(C(C)=O)C1 c1(C(=O)NC2C(C)(C)C(CNC(=O)Cc3cnccc3Cl)C2)cc2sccc2[nH]1 c1(C(=O)NCC(CCNC(Cc2cc(C)sc2)=O)O)cc2c(Cl)cccn2n1 C(=O)(CCCCCC#N)NC(c1cccnc1)C(=O)NCc1ccc(OC)nc1 C1(O)(CCNC(C2COCCO2)=O)CN(C(C2CC2c2ccc(Cl)s2)=O)C1 CC(C)CC(O)C(=O)NCC1CC2CC2N1C(c1cc(C(C)C)nn1C)=O C1(CNC(=O)NC(COC)C)CCC=CN1C(=O)OC(=O)CN(C)C N1(C(c2cn(C)nc2)=O)CCCCC(NC(=O)CNC(C2CCC2)=O)CC1 C1(CC)CN(C(C2(c3c(C)cccc3Cl)CC2)=O)CCN1C(=O)C(C)CC(N)=O C(CNC(c1cc(Cl)nnc1O)=O)(CC(F)(F)F)NC(C1(CC#C)CC1)=O C1(C(C(=O)OC)F)CCN(C(c2cnn(CCN)c2)=O)C1 C(=O)(C(F)(F)C(C)(C)O)N1CC(CCC)N(C(=O)CSCc2cccnc2)CC1 C1(C(=O)NC(C)C(C)(C)CO)CCCCCN1C(=O)CCCN(C)C C1(NC(c2n(CC)ncc2)=O)COCCN(C(=O)C(C)S)C1 c1(C2C(C(=O)NC(=O)C(=O)NC3CN(CC(F)F)C3)C2)ccc(Br)c(Cl)c1 N1(CCC(=O)NC(CCN(C(C2N(CCC)CCC2)=O)C)C)CCNC(=O)C1 C1(C(=O)NC2CC(=O)N(C)C2=O)COc2ccc(F)cc2C1 N1(C(c2c(C)nc(C3CC3)o2)=O)CCCC(C2CC2NC(c2ccn(C)c2)=O)C1 Cc1c[nH]c(C(=O)NCCC2(C(=O)NCC(C)(C)CO)CC2)c1C C(=O)(C1=CC(O)C(NC(=O)CC2CC(C)(C)CO2)C1)N(C(C)CO)CC C1(C(=O)NC2CCCC2CNC(c2cnc(Cl)s2)=O)(COC)CC1(F)F c1(N(C2CCC(C)(C)CC2)C)nc(=N)[nH]c(=NC(CF)c2ccccc2)[nH]1 C1(NC(C2C(CCC)CN(C(=O)C=CCF)C2)=O)(CO)CCN(C)CC1 Cc1nc2ncnn2cc1C(N1CC(CCCCNC(c2cscc2Cl)=O)C1)=O Cc1oc2cc(C(=O)N=S(C)(=O)CCC3(C)CNC3)[nH]c2c1C N1(C(Cc2ccc(C)s2)=O)CC(N=c2[nH]cnc3cnn(C)c23)CC2(CCC2)C1 C(=O)(CC(C(C)=O)OC(c1cccc(-c2nnc(C)o2)c1)=O)OCC C1(C(N(CC(CC)C)C)=O)(CCOC)CCN(C(c2ncc(C)cc2C)=O)CC1 C1(NC(c2c(CC)n[nH]c2)=O)CCCCC1NC(c1cnn(C)c1CC)=O c1(NC(C(N2CCC(NC(=O)OC(C)C)CC2)=O)=O)cc(Cl)c2nncn2c1 CCC(C)(COC)C(=O)N1CCC(CNC(=O)C(C2CC2)N(C)C)C1 C(CC1CCCC1)(C(=O)N=c1ccn(CCO)[nH]1)NC(c1cc(CC2CC2)on1)=O C1(NC(c2c(C)nc(C)[nH]2)=O)CCCC(NC(=O)CC2CC=CC2)CC1 C1(C(=O)NC(C(C)C)C(C)NC(=O)C=Cc2ccnn2C)CCC2(CC1)CC2 CCN=c1[nH]c(C(N2CCCC(C)(CNC(C3CC3CCOC)=O)C2)=O)cs1 N1(C(C(CC)CC)=O)CCC2C(CCCN2C(c2c[nH]c3cc(Cl)ccc23)=O)C1 C(=O)(CCC(N)CO)Nc1cc(C(=O)NC)ncc1 Cn1ncc2ncc(-c3nc(CCN(C)C)nn3Cc3ccccc3F)cc12 C(=O)(C(C)(C)CC(C)C)N1CC(CC(C(=O)NCCC(C(C)C)OC)F)C1 C(c1ccc(C(F)F)o1)=CC(=O)NC(C1CCN(C(C2CCCC2)=O)C1)C C1(C(=O)NCc2cn(C3CCN(C(CN(C)C)=O)CC3)nn2)CCC2(CCC2)C1 c1(CC(N2CCCC(N(C(Cc3ccc(C)s3)=O)CCO)C2)=O)cc(Cl)ccc1O c1(C(C(=O)NCC(C)CN(C(=O)Cc2cscn2)C)C)cncnc1 C1(C(=O)NCc2c(CC)nco2)CN(C(=O)CC2CN(C(C)=O)C2)CCC1(C)C c1(NC(=O)Nc2ccccc2)c(C#N)nc(Cl)c(Cl)c1Cl.C12CC1CN(C)C2=O C1(CNC(=O)Cn2cc(CC3(O)CCOCC3)nn2)CCC2(CCC2)CO1 C(=O)(C(CCc1ccsc1)NC(c1c[nH]cc1CC#N)=O)OC c1(C(N(CCOC)CCNC(c2c(C)ccn2C)=O)=O)cc(C)nc(O)n1 C1(CNC(c2cc(C)no2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1C c1(C(=O)NC2C3(CCN(C(CCCCC#C)=O)C3)C2)sc2[nH]cnc(=O)c2c1C Oc1ncnc2c1CCN(N1CCCC(c3ccc(O)cc3)C1)C2 N1(C(CCC(C)C)=O)CCN(C(C2(c3cccs3)CC2C)=O)CC2(CC2)C1 Cc1cc(CC(=O)NC2CC2NC(=O)Nc2ccccc2C(F)(F)F)ccn1 c1(C(N(C2CCCN(C(=O)CC3CCCCO3)C2)CC)=O)cnn2c(C)cccc12 n1(CC)ncc(Cl)c1C(=O)NC1CCC(N2CCN(C(=O)C3=CCC3)CC2)CC1 C(=O)(C(CC)C(=O)NC1CCCN(C(=O)CSCc2cccs2)C1)OCC C(C(C)(C)C(=O)Nc1cccc(C(=O)NC2COCC2COC)c1)SC CCCC(CC)C(=O)NN(C(C1(NC2(F)CCCC2)CC(CO)C1)=O)C C#CCC(C(=O)NCCC1CCCN(C(c2nnccc2C)=O)C1)C1CC1 C1(C(=O)NC(CC#C)C(=O)NC)C2CC3C(C2NC(C2CCS2(=O)=O)=O)C13 N1(C(C(=O)NCCCC)C2CC2Cl)CCOc2c(C(=O)OC)cccc2C1 N1(C(C2N(C(C)=O)CCC2)=O)CCC(NC(c2nnccc2C)=O)C2(CCC2)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CCCC2CN(C(c3sccc3F)=O)CCC12 c1(C2(C(=O)NC3C(OC(CC)C(=O)OC)CCCC3)CC2)ccc(N=S(C)(C)=O)s1 c1(CNC(C(N2CCCC(C(=O)OCC)C2)=O)=O)oc2ccccc2c1Cl CCCCC(CC(=O)NC(C1(O)CCCC1)(C)C)NC(c1cc(Cl)no1)=O c1(C(=O)NCC2N(C(C34CC(OC)C3C4)=O)CC2)ccc(O)c2c1CCCC2 C1(CC(=O)NC2CCN(C(c3c(CCC)n[nH]c3)=O)C2)(OC)CCCCC1 c1(C2(C(=O)OC)CC2)cccc(NC(=O)Nc2nc(-c3cccc(Cl)n3)cs2)c1 C(C(CCCC)NC(C1CN(C2CCOCC2)C1)=O)N(CC=C)C(C)C C12(OC)CCC(C(N3CCC(C(C)NC(=O)CC4CC(=O)NC4=O)C3)=O)(CC1)C2 c1(C(N2C(CC(=O)Nc3cc(N(C)C)ncn3)COCC2)=O)cc(Cl)ccc1Br C1(NC(c2cc(-c3ccc(Cl)cc3)ns2)=O)C2CN(C(=O)CC3CCCO3)CC12 N1(C(COCC)=O)CCCC(C2CN(C(=O)C=C(C)c3cccs3)C2)C1 C(=O)(C(O)CC(C)(C)C)N1CC(CCCC)N(C(=O)Cn2ncnn2)CC1 N1(C(=O)CC2CCC2)CC(C2CN(C(C3CC34CC(F)(F)C4)=O)C2)C1 N1(CC(=O)N(CC(CC)NC(C2CCS2(=O)=O)=O)CC)CCC(=O)NC1=O C1(Cc2cn(CCC=C=C)nn2)CN(C(c2cnc(C)cn2)=O)CCO1 N1(C(CCCN(C(C)=O)C)=O)CCCCC1CCN(C)C(C1CC1CN(C)C)=O N1(C(C2(C#N)CC3CC3C2)=O)CC2COCC(C1)C2NC(=O)C(F)=C1CCCC1 C(=O)(C(CCC)CCC(=O)OC)NCC(CNC(CCCCCSC)=O)(C)OC c1(C(=O)NC(CNC(C(C)C2CC2)=O)C2CCC2)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NCCN(C(c2cccc(O)c2)=O)CC)csc(N=S(C)(C)=O)n1 N1(C(C(C)O)=O)CCCC(C(=O)NCCc2cnn(C)c2)CC1 C1(C(N2CCCCC2CO)=O)CSc2ccccc2O1 CC1CCCN(C(=O)CC2CN(C(C3CCO3)=O)C(C)(C)C2)CC1 Cc1nc2c([nH]1)CC(C(=O)NCCC1CCCN1C(=O)C(C)OCC(C)C)CC2 CCC(O)C(F)(F)C(=O)NCC1CN(C(=O)CC(COC)COC)CC1(C)C C1(C(N(C)CC2CCN(C(c3coc4c3COC4)=O)C2)=O)OCC2COCCC12 c1(C(=O)NCCC(=C)CNC(C2CC2CC(C)C)=O)ccc2nonc2c1 c1(C(N(CC(C)CNC(=O)C(=O)NCC2CC2)C)=O)cn2c(n1)CCC2 c1(C(=O)NC2CC(C(C)NC(Cn3ncc(CC)c3)=O)C2)n[nH]cc1[N+](=O)[O-] c1(C(N(CC(C)N(C)C(c2ccc(N)cn2)=O)C)=O)cccn2nnnc12 C1(CNC(C2(CC=C)CC=CC2)=O)CN(C(=O)CSCC)C2CCN1C2 c1(C(N(CCCNC(C2C3CC4C(C3=O)C24)=O)C)=O)ccc2cnnn2c1 N1(C(=O)Cc2ccccc2)CC2(C1)CN(C(C1(Cc3cccc(F)c3)CC1)=O)C2 c1(CCC(=O)N(C)CC2(O)CN(C(C3C4CNC(=O)C34)=O)C2)cc(F)cc(F)c1 Cc1nn(C)cc1-c1ccc(C(N2CCN(C(C)(C)CO)CC2)=O)cc1 Cc1cc(C)c(C(=O)NC2CC(CNC(=O)CCn3ncn(C)c3=O)C2)cc1C C1(C(=O)NCC=O)CC12CN(C(=O)NC)C2.c1(C2CC2)ccn(C2CCCCO2)n1 N1(C(CCN(CCCCC)C)=O)CCC(C2(NC(=O)CCCNC(C)=O)CC2)C1 Cc1cc(C(=O)NCC2CCC2NC(c2ccnn2CCF)=O)ncc1N C1(CCCC)CN(C(C2CC2C2CC2)=O)CCN1C(=O)Cc1csc(Cl)n1 C1(C(=O)NC(C(CO)NC(c2nc(C)sc2)=O)C)CCC(C)(C)OC1 c1(C(N2CCCC2c2cc(C)nn2C)C(=O)NCCC)sc2ccccc2c1C N1(C(CN(C(=O)CN2CCC(OC)C2)CC#C)=O)CCC2(CCOC2)CC1 Cn1ncc2c1CC(C(=O)NCC(C1CCC1)NC(C1C3COCC13)=O)CC2 N1(C(c2c(C)n(C)nn2)=O)CCN(C(=O)CCOCc2ccccc2)C(C)C1 c1(C(=O)NC(C(C)NC(c2ccc(CC)[nH]2)=O)C)ccccc1CC#N c1(C(=O)NC2C(NC(c3cccc(SCC#N)c3)=O)C2)cc(O)cc(=O)o1 Cc1ccc(C=CC(=O)NC2CC2NC(C2CCC(OC(C)C)CC2)=O)c(C)c1 CC1(C)CC(C(=O)NC2CCN(CC3CC=CCC3)CC2)N(c2ncccn2)C1 CCC(CN1CCC1C(=O)NCCn1cc(C2CCN(C)C2)nn1)CC N1(C(C=NOC)=O)CCN(C(c2cc3c(s2)CCC3)=O)C(C(F)F)C1 Cc1nc2ccccn2c1C(N1CCNC(CO)C1)=O N1(C(c2cnn(C)c2F)=O)CCN(C(C2CCN(CCF)CC2)=O)C2CC12 N1(C(C(CC=C)C(C)C)=O)CC=C(C(C)(C)C(=O)N2CC3CC(C2)C3(C)C)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CCCN(C(=O)Cn2cncn2)CC1 c1(CNC(C2CCC(n3cc(CC4CCC(=O)C4)nn3)C2)=O)cc(F)ccc1Cl C(=O)(CC(C(C)C)NC(=O)CCc1ccco1)NCC(C=C)O CCC(CCC(=O)NCC1CC(NC(=O)Cc2cccc(O)c2F)C1)OC c1(C(=O)NCC2CC(F)(CNC(C3CCN(C)C3=O)=O)C2)cccc2sncc12 C1(CNC(CS(CC)(=O)=O)=O)CC2OCCC2N1C(c1ccc(C)c(C)c1)=O N1(C(CS(C)(=O)=O)=O)CC(NC(=O)CCCCc2ccccc2)C(C2CC2)C1 CCCC(O)C(=O)N(C)CC1CCN(C(C2(C)CCSCC2)=O)C1 c1(C(=O)OC)nc(=NCC2(C)CCCN(C(=O)C3=C(Cl)CC3)C2)c2c([nH]1)CCC2 C12(CCNC(C(C)(C)NC(C)=O)=O)CCC1CN(C(c1c[nH]c(=N)nc1C)=O)C2 N1(C(CC2CCC(C)C2)=O)CCC2(CC1)C(NC(=O)CC1CN(C)C1)CS2(=O)=O Cn1c(CCC(=O)NC(CC2CC2)C(=O)NC(c2ccccc2)CF)nnc1S c1(C(C)=O)cn(C)nc1C(=O)NCC1CC1CNC(=O)C=Cc1cocn1 C1(C(C)(C)O)CCN(S(=O)(=O)N2CCC(CC3(O)CCOCC3)C2)CC1 c1(C(=O)NCC2CC(NC(CC3C(C)OCC3)=O)C2)ccc2oncc2c1 C(=O)(CCN(CCO)C(C1CN(C2COC2)C1)=O)N(CCOC)C c1(CN2C(C(=O)Nc3cccc(C(=O)OC)c3C)C=CC2)c(O)ccc(Br)c1O C1(CNC(CCc2cc(C)[nH]n2)=O)CC(NC(=O)C=Cc2scnc2C)C1(C)C c1(OCC)ccccc1C(=O)NC(C)(C)CCCNC(=O)C(CC)OC c1(C(=O)NC23CCC(NC(CCCC#C)=O)(CC2)C3)ccc(F)c(S(C)(=O)=O)c1 c1(C(=O)NCCCCNC(c2cnncc2C(F)(F)F)=O)ccc(O)c(Cl)c1 C1(O)(CNC(=O)C=C2CCCC2)CC(CNC(c2ocnc2C(F)(F)F)=O)C1 N1(C(C2C(CC(C)(C)C)C2)=O)CCCCCC(NC(=O)CC2CCC(=O)O2)C1 C#CCC(CC#C)C(=O)NC1CN(C(C2(SC)CCC2)=O)CC1N1CCCC1 C(C(COC)CC(=O)NC1CC(O)CN(C(=O)CCCc2cnccn2)C1)OC c1(C(=O)NC2CN(C(c3ccnc(C)c3O)=O)CC(O)C2)ccnc2c1CCC2 c1(CNC(c2cc3cc(Cl)ccc3o2)C)c(Cl)c[nH]c2nccc1-2 C(=O)(C1=C(Cl)CCOC1)NCC12N(C(CCOCCN(C)C)=O)C(CC1)CC2 N1(CC)CCC(N(C(=O)CCCn2cc(C(=O)OC)nn2)C)C(C)C1 c1(C(N2CCN(C(c3ccn(C(C)(C)C)n3)=O)CC2)=O)cc2[nH]ccc2s1 C(=O)(C(F)(F)CC1CC1)N(C1CCN(C(C2CCCCC2C)=O)CC1)CC C#CCCCCC(=O)NC(C)CNC(C1(OC)CS(=O)(=O)C1)=O C1(CC(=O)NCCCC2CCC(NC(C3(CC#C)CC3)=O)C2)CCC(C)(C)CO1 c1(NC(C2N(C(C)=O)CCC2)=O)ccc(F)c(NC(C2OCCOC2(C)C)=O)c1 C1(CNC(C=CCOC)=O)(NC(=O)C(c2ccccc2F)C)CCCCC1C CC1CN(C(=O)CCc2cncs2)CC(C)N1C(=O)CC1CCCCCCC1 S(=O)(=O)(c1cnc(NCCOC(F)F)c(Cl)c1)NCC1CCCC(C)C1 N1(C(COC(C)C)=O)CCOCC(CNC(=O)CCc2ccc(Cl)c(F)c2)C1 Cc1ccc(CS(=O)(=O)NC(=O)Cc2cccc(N3CCCC3=O)c2)c(C)c1 C12(NC(c3cn(CCNC(CC4CC(OCC)C4)=O)nn3)=O)CCC(SC)C1C2 c1(SCC=C)ccccc1C(N1CC(NC(c2cnccc2NC)=O)C(O)C1)=O Cc1oc(CCC(C)C)nc1C(N1CCOC(CNC(=O)C=CC2CCC2)C1)=O N1(C(CC(C)C2CCCO2)=O)CC(C)(C)OC2(C1)CN(C(c1cc[nH]c1)=O)C2 CCC(C)CC(C)N=c1[nH]c(N2CCC3(CCC3)C2)nc2c1CCCCC2 C1(CC(=O)NCC(c2nccs2)C)CCCN(C(C2(C)CCOCC2)=O)C1 c1(C(=O)NC(CN(C(C(CC)N(C)C)=O)CC)C)sc(C)nc1C(F)(F)F Cn1cncc1C(=O)NC1CC(CNC(=O)Cc2csc(N3CCCC3=O)n2)C1 Cc1noc(C)c1-c1cn(CC2COCCN2C(C2(C)CC(C#N)C2)=O)nn1 Cn1ncc(C(=O)NC2CN(C(C3(O)CCC3)=O)CC3(CC3)C2)c1S(C)(=O)=O c1(C(N2CCCC(NC(COCCCCOC)=O)C2C)=O)ccn2nccc2n1 C1(NC(Cc2c(C)ocn2)=O)C(C)(C)C(NC(=O)C(O)CC2CCCC2)C1(C)C c1(OCCCOC)ccc(C(=O)NC(C)CCNC(=O)CCC=C(C)C)cn1 C(C1=CCN(C(=O)CCc2nc(C)c(C)o2)CC1)NC(c1c(SC)cccc1)=O C1(NC(C(CCC)O)=O)COC2C(NC(=O)C=CSc3nc[nH]n3)COC12 C(c1ccccc1C(F)(F)F)=CC(=O)NC(CSCC)C(=O)NC C1(NC(C(CC#C)NC(c2nn(C)cc2C)=O)=O)CC(C)N(C)CC1C C(=O)(C1Cc2ccc(Cl)cc21)NC(C(C)NC(=O)CCCCc1cnn[nH]1)CO C#CC1(C(=O)NC2CCC(C3CC3)C2)CCN(C(c2cnc(N(C)C)nc2)=O)C1 Cc1cc(C(=O)NCC(CNC(c2cscc2Cl)=O)CO)nc(O)n1 C1(NC(C(C)OCC2CC2)=O)CN(C(c2cc(F)cc(F)c2O)=O)CC(F)(F)C1 C(=O)(C(O)P(C)(C)=O)NCC(C)(C1CC1)NC(CCC(C)C)=O C1(NC(C(C)C2CC2)=O)Cc2ccccc2C1NC(c1cnsn1)=O C(=O)(CCC(C(=O)OC)NC(=O)CSCCn1cc(C)cn1)OCC c1(C(=O)NCCCNC(CCC2(C(C)(C)C)CCCO2)=O)cccc(CCO)c1 n1(C(C)C)cnc(C(=O)NC2CC(CNC(=O)OC(C)(C)C)C2)n1 c1(OC)cc(-n2nc(CO)nc2C2CCCN(CC(F)(F)F)C2)ccc1F C1(CC(N2CCC(CF)C2)=O)(NC(=O)C(O)CC2CCCC2)CCCCC1 C(=O)(CC1=NNC(=O)C1)NCC1CN(C(c2nc(CC)sc2)=O)C(C)CC1 C=CC1(C(=O)NC2(CCCC(=O)NC3CCC(F)C3)CCC2)CCC1 c1(C(=O)NC2C(CNC(c3ccc(C(N)=O)[nH]3)=O)CC2)[nH]cc2c1CCCC2 c1(OC)ccc2oc(C(=O)O)cc2c1.C1(COCC2CC2)CC12CCOC2 N1(C(c2scc(C)c2C)=O)CCC=C(C(=O)N(C)OC2CCCC2)C1 CC(C)(C)CC(O)CC(=O)NCCCN(C(=O)CC(F)(F)F)Cc1ccccc1 C1(C(=O)NC(C)CN(C(=O)CSC(F)(F)F)C)CN2CCCCC2CO1 C1(C(=O)NC2(C(C)C)CCC2)C2CCC(C2)N1C(=O)CC(C)F c1(C(=O)NC2C(CNC(C(C(=C)Cl)(C)C)=O)C2)ccc(S(=O)CC#N)cc1 C(=O)(C#CC1CCCCC1)N1CCC(CC(=O)NCC(N2CCCC2)=O)C1 C1(C(=O)NCC23CC(NC(c4scc(OC)c4OC)=O)(C2)C3)CC2CC2CC1C C12(NC(CSCC(C)C)=O)CCN(C(c3ccccc3C#N)=O)CC1C2 N1(C(COCC#C)=O)CCC(C2CCN(C(=O)CCC(C)(C)C)C2)C1 N(C1CCCn2nccc21)C(Cn1c(C(C)OCC)ncc1)=O CC(O)CCCC(=O)NC(C)CCNC(=O)C1=NNC(=O)C1 C(=O)(CC(=O)NC1COCC1CN(C)C)NCCC1C(C(=O)OC)C1 Cn1cc(CC(=O)NC2(CCCNC(C3(C)CC=CC3)=O)CC2)nn1 Cc1cc(N2CCC(C(C)NC(=O)CC(C)C(F)(F)F)C2)ccc1[N+](=O)[O-] c1(NC(C2CCN2C(=O)CSc2ccc(Br)cn2)=O)nc2ccccc2s1 C=C(Cl)CC(C(=O)NCCN=[N+]=[N-])NC(=O)CCNC(N)=O c1(OCC)ncc(NC(C2CC(OC)CN2C(c2c[nH]c(=N)s2)=O)=O)cc1C Cn1ncc2c(N3CC4(CC4)CC3CNC(C3(C(F)F)CC3)=O)ncnc12 c1(OC)cc(C(=O)N(C)CCOCCNC(c2sccc2OC2CC2)=O)ccn1 c1(C(=O)NCc2cccc(NC(C3C(C)COCC3)=O)c2)ccc(F)c(N)c1 c1(CN(CCNC(C2CC2c2ccccc2)=O)CC)nc2cnccc2s1 N1(C(C(c2ccccc2Cl)C)=O)CCC(C(C2CC2)NC(=O)C=CC2CCC2)CC1 N1(C(CC2N(CC)CCOC2)=O)CC(O)(C2(CNC(=O)CNC(C)=O)CC2)C1 C1(NC(C(COC)COC)=O)CN(C(=O)COc2ccn(C)n2)C(C)(COC)C1 N1(C(c2cc(OC)ns2)C(=O)NCCCSC)CCS(=O)(=O)C2(CCCCC2)C1 O=C(CCCS(=O)(=O)N1CCCC1)NCC=CCNC(=O)CC1CCOC1 n1(C(CC)C)nc(C(N2CCC(CNC(=O)CC(C)(O)C3CC3)CC2)=O)cc1C CC1CN(C(C2CCC2C)=O)CCCN1C(c1ccc(-n2ccnn2)cc1)=O O=C(CC1=CCOCC1)NCC1CN(C(=O)CCc2ccncc2)CCO1 CC1CCCn2ncc(C(=O)NC3CCCCN(C(=O)CCc4ccco4)C3)c21 N1(C(c2c(C)cccc2)=O)CCC2(CC(C(=O)NCCCCCO)=NO2)C1 C(=O)(C(C)(C)Cn1cc(-c2nccnc2CO)nn1)NC(CC)COC N1(C(Cc2ncn(C)c2)=O)CCCCC1CCNC(=O)CCC1CCCOC1 Cn1ncc(CNC(=O)Cn2ccnn2)c1C(=O)NCc1cn[nH]c1 Cc1ccc(CCNc2ncccn2)c(Br)c1 c1(CNC(=O)NCC2(C(F)(F)F)CCC2)cccc(F)c1Sc1ccccc1 N1(C(CCOCC)=O)CCC(NC(c2cc(C(=O)OC(C)(C)C)c(C)o2)=O)CC1 C1(C(N2CCC(=C)CC2)=O)CC2OCCC2N(C(C2CCC(F)(F)C2)=O)C1 Cc1ccc(C(=O)NC(C)CCCNC(C2CC2c2cnc[nH]2)=O)c(N)c1 Cc1onc(C(=O)NCC(C2CCC2)NC(=O)CC(F)(F)F)c1[N+](=O)[O-] C1(N(C(C(C)OCC)=O)CC)CCCN(C(c2ccnn(C)c2=O)=O)CC1 N1(C(N2C(C)(CC)COCC2)=O)CCc2nnnn2CC1 C(CC(=O)NC(C(=O)N(CC(O)COC)C)c1cccs1)OCC C(CC(F)F)(C(=O)N1CCC2(CCO2)C1)NC(C1CC(CC2CC2)C1)=O C1(C(=O)NC(CN(C(c2cnn(C3CCC3)c2)=O)CC)C)CCCN1C c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)Cc2ccco2)cc2ccccc2o1 O(NC(=O)CS(=O)CC)CC(=O)NC1CN(CC)CC1C c1(CC(=O)NCCC2CN(C(CC3C(C)OCC3)=O)C2)ccn2cncc2c1 c1(C(=O)NCCC2(O)CCN(C(CC=C(C)C)=O)CC2)cc(O)ccc1[N+](=O)[O-] n1(C(C)C(=O)NC(C)(CNC(=O)Cn2cccn2)C2CC2)cnc(C#N)n1 C1(O)(C(C)NC(c2ccc(SC)s2)=O)CCN(C(=O)C=CC(C)(C)SC)CC1 c1(C(=O)NC(C2CCCN2C(=O)C=C(Cl)Cl)(C)C)cccn(C2CCSC2)c1=O N1(C(C2CN(C(=O)NC)C2)=O)CC2CC(N3CCCC(C)(O)C3)C1C2 c1(OC)ccc(CCC(N2CCCCC2C(=O)NCC#N)=O)cn1 c1(C(=O)NC(CNC(C(CC)(C)CO)=O)C)ccc(NC(=O)OC)c(C#N)c1 CCCCCC(O)C(=O)N1CCCC(C)(C(=O)NCC2CCS(=O)(=O)CC2)C1 C1(C(=O)NC2C(NC(=O)COCc3ccncc3)CCC2)Cc2cscc2C1 C1(NC(c2c(OC)scc2)=O)C2CCN(C(=O)C=Cc3nc(C)cs3)CC12 C1(C(=O)NCC(C)(O)CNC(=O)CCCN2CCCC2)CCOC2(CCCC2)C1 c1(-c2cc(NC(c3cnc(OC)c(C)c3)=O)ncc2)cccc(C#N)c1F c1(NC(Cc2ccc(OC)cc2C(F)(F)F)=O)cc([N+](=O)[O-])c(N(C)C)cc1F C1(C2CCC2)(C(=O)NC2CN(C(C(c3cn(CC)nc3)=O)=O)C(C)C2)CC1(F)F c1(C(=O)NC(C)CC2CN(C(c3c[nH]c(C(C)(C)C)n3)=O)C2)ccc(Cl)nn1 C1(NC(=O)C(c2cc(Br)c(Cl)s2)N2CCCC2Cc2ccsc2)CCC(F)(F)CC1 N1(C(CSCCC(C)C)=O)CC(C(=O)N(CC2=CCCOC2)C)C(CO)C1 c1(NCC(N(C(c2c(C)scn2)=O)C)C2CC2)nc2c(cc1C#N)CCCC2 CC1CCN(C(=O)CN(C)S(N)(=O)=O)C1CNC(=O)CCC=CBr Cc1nnc2n1CC(C(N1CC(CNC(=O)C3=C(C#N)CCC3)C(C)C1)=O)CC2 C1(C(N(CCC(N2CCC(C)(N(C)CC)C2)=O)C(C)C)=O)CC2(CCO1)CC2 Cc1ccc(C(=O)NCC2CCCC(NC(c3coc(C4CC4)n3)=O)C2)nc1 C1(C(=O)NC(CC)CN2CCCC2)CN(C(C2(CC)CCCCO2)=O)CC1(F)F C1(CC(=O)N(CCCOC)C)CN(C(C2CCC2)=O)C(C)(C)C1 C(CC(=O)NC1C(C)(C)C(NC(C2(C)COC2)=O)C1(C)C)(C(F)(F)F)OC C1(c2ccno2)(C(=O)NCC(C)N(C(C(CC)SC)=O)CC)CCOCC1 c1(NC(C2C(CC)CCN2C(=O)C(C)OCCOC)=O)ccc(O)c(Cl)c1 C(=O)(C(C)C1=CCCC1)NCC(F)(F)F.c12c[nH]nc1NC(=O)C1CC(C1)C2C c1(C(N2CCC(C(=O)NCCCc3ccccc3Cl)C2)=O)n[nH]c2c1CCC2 C(CCC(=O)NCC1CC1CNC(=O)CCc1cnn[nH]1)SC c1(OC)cc(C=CC(=O)NC(C)CNC(c2cncc(C(F)(F)F)n2)=O)ccc1O c1(C(=O)NCC=CCNC(CC2ON=C(C)C2)=O)ncc(Br)cn1 N1(C(C(CC)C)=O)CC2CCCC2(CNC(C2(CO)CCC2)=O)C1 CC1CCCCC1(CO)NC(C12CC(CN1C(=O)CN1CCC(F)CC1)C2)=O Cc1nc2ncccn2c1C(=O)NCC1CN(C(c2ccc(Br)c(O)c2)=O)C1 n1(CC)nnc(C)c1CN1CCC1CNC(=O)Nc1cnn(C(C)(C)C)c1 C1(CNC(c2cccc(C(N)=O)c2)=O)CN(Cc2ccc(F)cn2)CCCO1 c1(SC)cc2ccc1N1CC2C1.c1(C(=O)Nc2ncsc2Br)nnnn1C1(C)CC1 c1(C(=O)NCC(CNC(c2cc(C)sc2)=O)C)ccc(Cn2cncn2)cc1 C(=O)(CS(=O)(=O)C1CCCC1)NCC1N(C(CC(CC)CN(C)C)=O)CCC1 C(=O)(C1CCc2nccn21)NCC1(F)CCN(C(CC(=C=C)C)=O)C1 C#Cc1cccc(C(=O)NC2(CNC(c3ccsn3)=O)CCC(C)(C)CC2)c1F c1(C(=O)NC2(C)CN(C(c3cnn4c3OCCC4)=O)C2)cc2sc(F)cc2[nH]1 CC(F)(C(=O)N1CCC(CNC(=O)C=CCO)C1)C(F)(F)F N1(C(c2cc(OCC)n[nH]2)=O)CC(NC(C2CC2F)=O)C(CC)C1 C(=O)(C(C#N)C(C)(C)C)NCc1occ(C(N2CCC(CC=C)C2)=O)c1 Cc1cccc(C(=O)NC2CCCN(C(=O)COc3ccc(F)c(Cl)c3)C2)c1F C=CC1CN(C(=O)CNC(=O)CC2CCCC2)CC1NC(=O)CCC(C)OCC C1(C(N2C(C)CS(=O)CC2)=O)CC2(CCC2)CN1C(C1CC(=O)N(C)C1)=O N#CCCCC(=O)N1CCOCC1CCNC(C1(c2ccno2)CC1)=O c1(C(=O)NC(CN2CCN(C(C(C)C3CC3)=O)CC2)C)nccn2nccc12 C#CC1CC(NC(=O)C(C2CCC2)NC(=O)CSCCC)C1 Cc1ccc(C#N)cc1C(=O)NCC(C)C(=O)NCCCC(=O)NC1CC1 C(=O)(CN=c1ccc(Cl)n[nH]1)N1C(CNC(c2n3c(nn2)SC(=C)C3)=O)CCC1 C1(NC(CC(C)(C)C)=O)C2CCC(C2)C1C(=O)N(C1CS(=O)(=O)C1(C)C)C CCC(CC)(CC)C(C(=O)OC)NC(c1nc2ccccc2n1CCOC)=O c1(C(=O)NC(CNC(c2ccc(C(=O)OC)[nH]2)=O)C)cccc(C(C)(F)F)c1 N1(C(COC)=O)CCC(C(=O)Nc2cc(C)ccc2OC)C(C)(C)C1 N1(C(C(CCC=C)(C)C)=O)CCOC2(CCN(C(C34CCC3C4)=O)C2)C1 N1(C(C=CCN(C)CC)=O)CCSCC1CCNC(=O)C(=Cc1ccccc1)C c1(C(=O)NC(C2CCCN2C(c2ns[nH]c2=O)=O)C)ccc(C(F)(F)CF)cc1 CCCCCC(=O)NCC(C)N(C(=O)C(CCSC)NC(N)=O)CC C(=O)(C1CCCc2ccccc21)N1C(CC)CN(C(=O)CCC(F)F)CC1 c1(C(=O)OC)ncc[nH]c1=NC1CC(NC(=O)CC2C=CCCC2)C1 c1(C(N(C(CNC(C(CC=C)C)=O)C)C)=O)c(F)cccc1[N+](=O)[O-] C(=O)(CC(C(F)F)n1ccnc1)N(CCCN(C)C(c1ccc(Cl)cn1)=O)C c1(C(N2CCC(C)(C(=O)NOC3CCNC3=O)C2)=O)nccc2cc[nH]c12 CC1CC2(CCN(C(C3CC3(Cl)Cl)=O)CC2)CN1C(C1CCCSC1)=O CC1(C)CC(NC(C2CCC(=C(F)F)CC2)=O)CN(C(C2CCCC23CC3)=O)C1 N1(C(c2c(C)nsc2)=O)CCCCC1CNC(c1ccc(Cn2cccc2)cc1)=O c1(CC)ccc(-c2nc(Cc3ccccc3F)nn2CCOc2nncs2)cc1 C1(C(=O)NCc2ccc(N(C)C)c(F)c2)CCOCC12CCCC2 C1(C(=O)NC2(CF)CCN(C(C(C(C)C)F)=O)C2)CC2CCCC(C1)C2 C1(C=O)(C(F)F)CCCC1.c1(N2CC(C(N3CCC3C)=O)C2)nnc(O)s1 CC12CCC(=O)N1CCCN2C(=O)C(c1cccnc1)O C(C(CO)C(C)(C)C)NC(c1c(C)cc(CNC(c2ccnc(CO)c2)=O)o1)=O c1(CN=C(NC(C(COC)C)C)NC(C)C)ccc(C#N)c(F)c1 C1(CCC(=O)NCC=CCNC(Cc2c(C)noc2)=O)CC(C)(C)CO1 N1(C(c2cc(C(=O)OCC)[nH]c2)=O)CC2CCCC2(C(C)NC(=O)C(C)OC)C1 C1(NC(c2c(C)cccc2C)=O)CN(C(c2cn(CCO)nn2)=O)CC(F)(F)C1 c1(C(=O)NC2C(NC(C3(SC)CCC3)=O)C2)c(O)nnc2c1CCCC2 Cc1cc([N+](=O)[O-])nn1CC(=O)NCC#CCNC(C1CCN(C)C1C)=O c1(CN(C(C2CCN(CCC)C2)=O)C)nn(C)cc1Br c1(OC)ncc(Br)cc1CC(=O)NCCCCC1(N)CC1.c1(=O)c(=O)[nH]1 C1(SC)CN(C(c2cc(F)n(C)n2)=O)CC1NC(C1(CO)CCOC1)=O C(CNC(C1CC1C1CCCC1)=O)(CC(=O)NOC1CCOCC1)OC C1(CNC(C2(C=C)CCC2)=O)CCCCC1NC(=O)C(c1ccc(OC)cc1)C c1(C(=O)OC)ccccc1C(=O)N(C1CCN(C(=O)CC(F)(F)F)C1)C c1(OC)cc(NC(C2C(O)CCN2C(c2sccc2Br)=O)=O)nc(Cl)c1 c1(CN(C)CC2CN(C(=O)C(=O)NC3CCCC3)CCO2)cc(Br)ccc1I c1(CCCC)ccc(C(C)C(=O)NCC(c2ccccc2)O)cc1 N1(C(COCCC#C)=O)CC(F)(F)CC1CCNC(c1ocnc1C(F)(F)F)=O CC(CCC(C)(C)C)NC(=NCc1ccccc1Br)NCc1ccnn1C c1(C(N2CC3C(CNC(=O)CC4CC4C(F)(F)F)C3C2)=O)n[nH]c2c1CCCC2 C12(NC(CC3CC(OC)C3)=O)CCCC1N(C(C1CC3CCC1C31CC1)=O)CC2 N1(C(c2cc(C)sc2)C(=O)NC2CCC2)CCS(=O)(=O)CC1C1CC1 CC(CC(=O)N1CC2CC1C2C(N1CCc2nn(C)cc2C1)=O)CC(C)(C)C CC1(C(=O)NC2CCC(C(N)=O)C2)CN(Cc2c[nH]c(C(N)=O)c2)C1 N1(C(C(C)(C)CO)=O)CCC2C(CCCN2C(c2csc3cncn23)=O)C1 c1(CN(C(=O)NCC2CCN(CC)C2)C2CC2)ccc(C)cc1 c1(C(=O)OC)cc2cccnc2nc1NC(N1CCOC2(CCSC2)CC1)=O C(C(CC(C)C)NC(=O)C(C)CCc1ccc(F)cc1)NC(C)=O.c1(=O)c(=O)[nH]1 c1(C2C(C(=O)NC3CCN(C(c4ccsn4)=O)C3)C2)ccc2oc(O)nc2c1 C1(CNC(CCC2(C)CC2)=O)C2CCCC1N(C(=O)CC1C=CS(=O)(=O)C1)C2 C1(CC=C)CCCN(C(=O)CC(COC)NC(=O)C(C)C2(O)CCC2)C1 N1(C(CN(CC)CC)=O)CC2C3CCC(C2C1)N(C(c1cccc(CO)c1)=O)C3.CC c1(CN2CC(CNC(c3ccc(C)s3)=O)OCC2)c[nH]c2cnccc12 c1(C(=O)OC(C(C)=O)C2CC2)ccn2ncc(Cl)c2n1 CCCCC(=O)C(=O)N(CC(C)(C)CNC(C1CCOC(CCC)C1)=O)C N1(C(c2cn(CC)nn2)=O)CCC2(CCCCN(C(=O)Cc3nncs3)C2)C1 C1(NC(C2(CC#C)CCCO2)=O)CN(c2nnc(CO)s2)C2(CCOCC2)C1 c1(OC)cc(-n2nc(C3CCCC3)nc2Cn2c(C)csc2=O)ccc1Cl Cc1cccc(F)c1CC(N1CCC(F)C(NC(=O)CC2CCSCC2)C1)=O c1(COC)nc(NCc2cc(Br)ccc2C)cc(=NCCC2CCCN(C)C2)[nH]1 c1(C(=O)NC(CN(C(c2ccc(OC(C)C)cc2)=O)C)C)cccc(S(C)=O)c1 N1(C(C(=O)NCC(C=C)C)=O)CCN(C)C(Cc2ccc(OC)nc2)C1 N1(C(C=C(CC)CC)=O)CC2CC(CNC(c3ccc4occc4c3)=O)CC1C2 N1(C(C2C(=C)C2)=O)CC(C)(C)C(NC(=O)CCSCCCC)C(C)(C)C1 S(=O)(=O)(c1cccc(C(=O)O)n1)NC1C(OC)C2(C1)CCC2 Cc1ccc2[nH]c(C(=O)NCC(C)CNC(C34COC(CCO3)C4)=O)cc2c1 c1(C(C(C)C)O)cn(CC2CCC(C(=O)O)C2)nn1 CCCC(C)C(=O)N(C1CCC(NC(c2ccc(C(C)C)o2)=O)CC1)C C1(CC(N2CCCC(CCNC(c3n(CC)ccn3)=O)C2)=O)CCCS(=O)(=O)C1 C12(C(=O)NC3C4(CC(NC(C5C(C)(C)OC(=O)C5)=O)C4)C3)CCC(CC1)C2(C)C CC(C)CC(=O)NC(C)CC(C)NC(c1csc(C(F)F)c1)=O c1(C(C(=O)NC(C2CN(C(=O)CC=CC(C)(C)C)CCO2)C)(C)O)ccc(F)cc1 C1(CNC(C(COCC)C)=O)CC2(CO1)CN(C(=O)CCCCNC(N)=O)C2 N1(C(C2C(C)OCCO2)=O)CCCC12CCCN(C(C1(C)CCN(C)CC1)=O)C2 C1(NC(C2CCCN(C(C)=O)C2)=O)CC1C1CCCC1.c1(CC(C)O)cn(CO)nn1 CC1COC2(C1)CN(C(=O)C(CCN(C)C)NC(=O)CN1CCCNC1=O)C2 n1(CC(=O)CCC2N(C(C3(C)CC3)=O)CCC2)nnn(-c2cccs2)c1=O N1(C(CCNC(C(=CC2CCCC2)C)=O)=O)CCCC(C)C1C(=O)O C1(NC(C(C2CC2)OCC)=O)CN(C(=O)CN(C)CCO)CCC1F C12(C(=O)NC(C(=O)OC)C3CC3)C(NC(=O)C(C)N3CCCC3)C3CC1C2C3 N1(CC(C2(OC)CCCC2)=O)CCC(C(C)C)CC1C(C)(C)O C1(CN(c2nnc(CC)o2)CC)CCCN(C(=O)CSc2cnn(C)c2)C1 C1(NC(c2c(C)cco2)=O)CCCC(NC(c2ccc(F)c(N)c2)=O)CC1 N(C(=NCCOC)NC1CCOc2ccccc21)CC(c1ccco1)OCC C(CCCCC(=O)N1CC(N(C)C)C1)N(C(c1cccc(NC)n1)=O)C c1(CC)nc(C(=O)NC(C)(CNC(=O)C(C)c2cncs2)C2CC2)co1 C12(C(N(CC(C)CO)C)=O)CC1CN(C(c1ccc(F)cc1)=O)C2 c1(-n2ccc(C(=O)NCCC(C)NC(c3cncnc3)=O)n2)ccc(Cl)c(F)c1 Cc1cnc(Cl)c(NC(C2CSCCN2C(c2noc(C)c2C)=O)=O)c1 CC1C(NC(=O)CC2CCC(=O)NC2)CCCN1C(c1ccc(C(N)=O)cn1)=O c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(c2c(C)ncn2O)=O)CC1C C1(NC(CNC(C2C(C)C2)=O)=O)CCOCC1C(N1CCC(C(C)C)(CO)C1)=O C(=O)(C(C(C)C)C1CCC1)NC(C(=O)NC1C(C(=O)NC)CCC1)C1CCCC1 CCCC(O)CC(=O)N1CC(=C(F)CNC(c2nncn2C)=O)C1 c1(C(=O)NC2C(CNC(C(C3CCCCC3)C)=O)C2)cn(C)nc1C(F)F C(=O)(CCCCCCC(=O)N1CCC1NC(c1c(C)nc2sccn12)=O)OC c1(C(=O)Nc2c(C)ccc(Br)n2)nc(-c2cccc3ncnn23)c2ccccn12 C1(NC(C(CSC)OC)=O)(CNC(c2csc(C)c2)=O)CC2CCC1CC2 CCC(CC)C(O)CNC(=O)C1=CCC(NC(C2CC(O)C2)=O)C1 N1(C(CN(C)CC)=O)CC2CN(C(c3nc(Cl)sc3C)=O)CC2C1 c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cn(C3CCOC3)cn2)=O)C1)=O Cc1cc(C(=O)NC(C2CCCN(C(=O)Cc3cn[nH]c3)C2)C)cc(C)c1F N1(C(C=CCCC)=O)CCC2(C=C(C(=O)NCC3CCCC34CCC4)C2)C1 c1(C(N2CC3C(CN=c4[nH]ccnc4F)C3C2)=O)cc2ccccc2s1 C1(C(N(C2CCCC2)CCNC(C2(C)CC2(Cl)Cl)=O)=O)CCn2cncc2C1 S(=O)(=O)(c1ccccn1)N(c1nc(OC)c(Br)cn1)C1CCCNCC1 c1(NC(C23C(CN(C(c4ccc(Br)s4)=O)C2)C3)=O)cccc2cccnc12 c1(OC)ccc(Cl)c(CC(=O)NC2CC(F)CN2C(=O)CNCC(C)(C)C)c1F N1(C(CSCC#C)=O)CCC2(NC(=O)C(=O)N(C)C)CC12 c1(CC(=O)NC2(CNC(=O)CC34CC(C3)C4)CCC2)ccc2ccccc2c1 C#CC1CCN(C(=O)C(CNC(=O)C(C)SCCCC)CC2CCCC2)C1 C(=O)(CCCC(F)(F)CO)N1C2C(CNC(C3(F)C(C)OCC3)=O)C(C2)C1 C(=O)(CC1COc2ccccc21)N1CC(OCCNC(c2cn(C)nc2)=O)C1 C12(C(=O)OC)CC3CC(CC(C3)C1NC(c1cc(C)nc(C)c1O)=O)C2 N1(C(C(C)c2cccs2)=O)CC2CCC1CC2NC(=O)CCC(N)=O C1(CNC(C2C3CC4C(C3=O)C24)=O)C2CCCC1N(C(c1c[nH]cc1Br)=O)C2 S(=O)(=O)(c1ccc(Cl)cc1F)NCC(=O)NCC(C)NC(=O)C1=NOC(C)(C)C1 C12(NC(C(CC)SC)=O)CN(C(c3cnccc3Cl)=O)CC1CS(=O)(=O)C2 c1(C(c2n(CCCC)nnn2)NCc2ccoc2C)cnc(C(F)(F)F)nc1 CC1CN(C(C23CC(C#N)(C2)C3)=O)CC1(C)CNC(C1COCCO1)=O CN(S(=O)(=O)N1CC(O)C1)Cc1cc(F)cc(Br)c1 C(C1CCCc2nc[nH]c21)NC(=O)C(c1ccc(Cl)cc1F)O C(=O)(C1CCc2nccn21)NC(C)(CNC(c1cnn[nH]1)=O)C1CCC1 Cc1cccn(CC(N2CC3(CC3)CC2CNC(=O)CN2CC=CC2)=O)c1=O CS(=O)(=O)c1cc(C(=O)NCC2CCC2NC(=O)Cc2ccccc2)ccc1F C1(OC)CN(C(=O)Cn2nccn2)C(C)(CNC(=O)CSCCN(C)C)C1 N1(C(C(CC)SC)=O)CCC2(CC1)CCN(c1cc(-n3ccnc3)ncn1)CC2 C12(CNC(c3nc(CC(C)C)sc3)=O)CC1CN(C(=O)CCCc1ccsc1)C2 C12CCCN(C1)C(=O)c1cnccc1N(C)C2=O.n1(CC)ccc(CN(C)C)n1.NC Cc1cccc(C(n2cc(-c3cccs3)nn2)C)n1 CCCCCC(O)C(=O)NC1(C(N2CC3(CCC(=O)N3)C2)=O)CC(O)C1 C(C(C(=O)N(CC(O)CNC(c1ccc(Cl)cn1)=O)C)C(C)(C)C)OCC=C C1(C(N2C3CN(C(c4c(CC)non4)=O)C(CC3)C2)=O)COc2ccccc2C1 C1(C(=O)NCC(CO)NC(CCC)=O)(COC)CCCCCC1 CC(CN(C)N1CCOCC2(CCOCC2)C1)c1cccc(Cl)c1 C1(C(=O)NCC(O)CNC(C2CCC(C(=O)OC)O2)=O)(COCC)CC=CC1 c1(C2(C(=O)NCC#CCNC(Cc3cn(C)nc3)=O)CC2)ccc(Cl)cc1Cl C(=O)(C(C)CC(F)(F)F)NC1C(O)CCN(C(CCc2scc(C)c2)=O)C1 N#Cc1ccc(OCC(=O)Nc2cc(N3CCCC3)nc(Cl)c2)nc1 C1(c2n(C)ncc2)CCCCC1NCc1ccc(O)nn1 C1(NC(c2cc(C)n(C)n2)=O)CCCC2CN(C(c3nncs3)=O)CC12 N1(C(c2c(C)c(N)ccc2)=O)CCC2CC(NC(c3ccncc3)=O)CCC2C1 c1(N(C)C)cc(C(=O)NCC2OC3(C)CC2(O)C3)c2ccccc2n1 C(=O)(C1=C(Cl)CCC(C)C1)NCCCN(C(CCN1CCC(C)CC1)=O)C c1(C(N2C(C)(c3cn(CC(N)=O)nn3)COCC2)=O)cc2ccncc2cc1F N1(C(C(C2CCC(=O)N2)C)=O)CC(NC(=O)C(=O)NC2CC2)C(CO)C1 C1(C(CO)NC(C(C=C)C)=O)CCN(C(=O)CCCC2CCCO2)CC1 C1(NC(c2ccccc2)=O)CCC12CCN(C(=O)CCN1CCCCC1)CC2 c1(C(N2C(CCNC(c3cc(C4CC4)no3)=O)COCC2)=O)cc(F)ccc1O c1(C(=O)NC(C2CCN(C(c3cnccc3C#N)=O)C2)C)ncc2cc(Cl)ccn12 C1(C(N2CC(NC(c3ccc(C)c(Cl)c3)=O)C(F)C2)=O)CCC2C(C1)C2(F)F N1(C(CC2CCCC(=O)C2)=O)CC(=O)NCC1C(=O)NCCCc1cncnc1 CCCC(C(O)C(=O)NOC(C)C)NC(=O)Cn1ccnc1CC C1(O)(C(=O)NCC(c2ccccc2-c2ccccc2F)=O)CC2(CCNC2)C1 c1(C(=O)NCC(C)(C)NC(C(C)c2ncco2)=O)cc(Cl)cc2cccnc12 c1(N(C)CC)ccc(C(=O)NCCN(CC(C)O)C(c2scnc2C)=O)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC(C1CCCCC1)(C)C C1(C(N(CCC(C)NC(c2scc(OC)c2OC)=O)C)=O)CCCNS1(=O)=O C1(NC(CCCOCC)=O)CC(CNC(=O)C(c2ccccc2)C)CC1O C(C(O)CC(F)(F)F)NC(CC1N(C(C2CCN(C)CC2)=O)CCCC1)=O N1(C(C=CC(C)(C)SC)=O)CC(NC(=O)Cn2ccc(=O)cc2)C2CCCC12 c1(OC(C)C(N2CCC(N(C)C(c3ns[nH]c3=O)=O)C2)=O)ccc(Cl)cc1 N1(C(CC(CN(C)C)O)=O)CCC(NC(c2ccnc(C(C)C)n2)=O)C12CCC2 Cc1cc(F)ccc1NC(=O)C(c1nocc1Br)N(C(C)C)C1CC1 c1(C(N2CCC(C)(NC(C3CC4(F)CC3C4)=O)C2)=O)cccc2occc12 CC1CCc2ncc(C(N3CC4C(CNC(c5ccc(Br)o5)=O)C4C3)=O)n2C1 C(CC(C)C(=O)NC1(C)CN(C(C2(C)CC2(Br)Br)=O)C1)OC CCC(O)CC(=O)N1CC(O)CC1c1cn(-c2ccc(Br)nc2)nn1 N1(C(CCCC#C)=O)CC(=O)NCC1C(=O)NCC(C)(C)CC(C)C N1(C(C=C)=O)CCCC(CN(C(=O)C(CC)c2ccccc2)CC)C1 N1(C(C(c2cccs2)SC)=O)CCC(C2CC2)(NC(c2cc(C)cs2)=O)C1 C(CC(C)(C)C(=O)NCC1CCOC1C(=O)NCCC(C)(C)N(C)C)SC c1(NCCC(C)OC)[nH]c(=NCc2cc(C)nn2C)nc2c1ncn2C(C)C c1(C(N=c2[nH]n(C)c(C(=O)OC(C)(C)C)c2)=O)ccc2ncccc2c1Cl c1(C(N2CCC(CC=C)C2)C(=O)NCCSC(=O)CC)cc([N+](=O)[O-])sn1 CCC(c1ccccc1)=CC(N1CCCC1c1ccc(Br)c(F)c1)=O c1(SCC2(CN(C(C)C)C3CC3)CC2)ccc(C(=O)N(C)C)s1 C1(NC(C(CCSC)O)=O)CN(C(=O)CC2(C)CCN2C(C)=O)CCC1O c1(CC(N2C(C)(CC)CC(NC(C3CSC3)=O)C2)=O)c[nH]c2c(C)cccc12 C=CC1(COC)CCN(Cc2nnnn2C)CC1 C12(C(N(CC(CC)NC(C34CCC(C3)C4)=O)CC)=O)CC3CC1C2C3 C1(S(C)(=O)=O)(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2F)CCCC1 C=C=CCCC(=O)NC(c1nocc1C(=O)N(C1CCN(C)C1)CC)C C12(C(N3CCC(C)(NC(c4c[nH]cc(F)c4=O)=O)CC3)=O)CCCCC1C2(F)F C#CC1(N(C)C)CN(C(C2CCCC2CNC(c2ccc(OC)o2)=O)=O)C1 C1(C(=O)NCC2(CC)CCCCO2)CC(O)C(O)CC1CNC(=O)C(C)C1CC1 C1(C(N2CCCC(CCNC(C(CC)CC)=O)CC2)=O)CC2(CCC2)CCO1 c1(C(N2C(C(=O)NC(N3CCCCC3)CC)CC2)=O)cc(C)nc(C)n1 c1(C(=O)NC(C2CC2C(N2CC(O)C(O)C2CO)=O)C)ccc([N+](=O)[O-])o1 c1(OC)ccc2c(n1)N(C)CCN2C(=O)CN1CCC(C(N)=O)CC1 S(=O)(=O)(c1cccnc1NCC1CC(O)CN1C)NCc1n(CC)c(C)nc1 C=CCC(C(=O)NCC1(CNC(=O)C=Cc2cnn(C)c2)CC12CCC2)C(C)C C(=O)(C1CCCc2nncn21)Nc1c(CNC(=O)C2=CC(O)CCC2)cccc1 N1(C(C(C)NC(=O)OC)=O)CCC(OCCNC(=O)CC2CCC2)CC1 N1(C(c2cc(C(C)=O)oc2)=O)CC(CNC(C2(N(C)C)CC2)=O)CC(C)(C)C1 CCCC(C#N)C(=O)NC1CCCC(NC(c2cc(O)nc(Br)c2)=O)C1 CCCCC(CC)C(=O)N1CCC(COC)(NC(C2CN3CCN2CC3C)=O)C1 N1(C(c2cn(C)nc2C2CCC2)=O)CC(NC(c2ccon2)=O)CC2(CCC2)C1 c1(OC)ccc(Cl)c(Cl)c1C(N1CC2CCC1C(NC(=O)C(F)=C1CCC1)C2)=O CCCCCCCCC(=O)N1CC2CCN(C(c3cc(C(N)=O)co3)=O)CC12 N1(C(C(COC)N(C)C)=O)CC(C)N(C(=O)C(n2ccnc2C)C)C(C)C1 n1(CCNC(C2C(C)(C)C2)=O)cc(C(=O)NCCCC2CCCCC2)cn1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(NC(C(C)Cc2cccc(F)c2)=O)C1 N1(C(CC2CCC(=O)O2)=O)CCC(CNC(C23CC(F)(C2)C3)=O)C(F)(F)C1 C1(C(=O)NCCCCNC(C2C(C)C2C)=O)CCCCN1Cc1cccc(F)c1 Cc1ccnc(C)c1C(=O)NC1CCOCC1C(=O)NCc1ncsc1C c1(-c2ncc(N(C)CC3C(C(=O)OC)CN(C)C3)cn2)ccc(C(=O)O)c(F)c1 C1(C(=O)NCCCN(C(c2cnc(N(C)C)o2)=O)CC)Cc2c[nH]cc2S1(=O)=O Cc1nc(NC(c2nc(C(=O)NC(CO)C3CC3)cs2)=O)nc(Cl)c1Br Cc1cc(C(F)(F)F)nn1CC(=O)N(CCCNC(=O)C=C1CCC1)C1CC1 c1(OC)ccc(C(=O)NC2CCN2S(C)(=O)=O)c(NC(c2ccncc2Br)=O)c1 S(=O)(=O)(c1cccc(N2Cc3cnc(Cl)cc3C2)n1)N1C(C)C(O)CCC1 C(=O)(C1=CCC(C)(C)CC1)NC(CNC(C1CN(C(=O)NC)C1)=O)(C)C1CC1 C#CC1CCC(C(N2CCC(C(C)NC(=O)COc3ccccc3C)C2)=O)CC1 c1(NC(C2CCC(CNC(CC=CCCCCC)=O)C2)=O)cc(Cl)nc(C)n1 C1(C(=O)NCC(F)C(C)(C)O)(CC)CCCN1C(=O)C(CN(C)C)CC CC1(C)CC(=O)NCC1C(=O)NC1CCN(C(c2ccsc2)=O)CC1 Cc1ccc(C(=O)C(=O)NCC2CCN2C(=O)Cc2nc[nH]n2)s1 CC(C)(C)CC(C)(C)C(=O)NCC1(C)COCCN(C(C2(F)CC=CCC2)=O)C1 c1(N)ccc2cc(Br)cnc2c1.n12nnnc1C(CC1CC1)C(=O)C1CC2C1.CO C(C(CC(C)C)C(=O)NCC1(CCNC(c2nn(C)c(N)c2C)=O)CC1)OC C1(CNC(C(CNC(C2CN(C)C(=O)N2)=O)(C)C)=O)CC12CCOCC2 C(=O)(CCC1=CCCCC1)N1C(C(=O)NC(C(=O)OC)C2CCC2)CN(C)CC1 Cc1nc(O)[nH]c1C(=O)NCC(C1CCC1)NC(C1(c2cc[nH]n2)CCC1)=O C(CCCC(=O)N1CCC(C)(CO)C1)N(C(C(C)=CCC)=O)C c1(OC)c(NC(=O)CSC(c2ccc(F)c(Cl)c2)C)cccc1F c1(C(N2CCC(C)(C(=O)NCCc3ccsc3)C2)=O)ccc2cc(O)ccc2n1 N1(C(C=C2C(C)(C)CCCC2)=O)CC2CC(NC(c3cncc(F)c3)=O)CC2C1 N1(C(c2c(C)con2)=O)CCC(C(C)(C)C)(CNC(=O)CC2COCCO2)C1 C1(C(=O)Nc2ccc(OCC)nc2)CCCCN(C(c2ncccc2Br)=O)C1 CC1=C(C(=O)NC2CN(C(c3snc(Cl)c3Cl)=O)CC2F)SCCO1 c1(NC(C2CCOCC2)COC)ncccc1S(=O)(=O)N1CCC2(CCCC2)C1 c1(NC(c2n(CC=C)nnn2)C2(SC)CC2)ccc(-n2nccc2C)cc1 C1(OC)(OC)CCC1C(=O)NC(CNC(c1ccc(SC)o1)=O)CO C1(NC(=O)Cc2csnn2)CCC2CCN(C(c3cnns3)=O)C12 N1(C(C(COC)NC(C)=O)=O)CC(NC(=O)C(C)C(F)F)CCC1C CC1CNC(=O)C1.c1(C(C)C(=O)OC(C)(C)C)nc(-c2ccccn2)cs1 C1(NC(c2cc(C)nn2C(C)(C)C)=O)CN(C(=O)Cn2cnnn2)CC2CC12 C1(C(=O)NCCOC(CNC(C=CC)=O)(C)C)CC2C=CCC(C1)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCCC2(C1)CN(C(C1CC3CC3C1)=O)CCO2 Cc1cccc(C(O)C(=O)NCC(C2CCC2)NC(c2cc(C#N)on2)=O)c1 C1(OC)CC(CCNC(C2CCSC(C)C2)=O)N(C(C2(OC)CCC2)=O)C1 CC1CCN(CCC(=O)NCC2(C(N)=O)CN(C(=O)CC(F)(F)F)C2)CC1 N1(C(CCn2ncc(C)c2)=O)CCC(CNC(c2nnc(O)cc2C)=O)C(C)C1 CN1C(=O)OCC1C(=O)NCC1CCN(C(c2c[nH]nc2C(F)F)=O)CC1 CCCCCCCC(=O)N1CC2CCC2(C(=O)Nc2nccc(Cl)c2I)C1 c1(C(N2CCC(C)(CNC(=O)C(F)(F)CO)C2)=O)c[nH]c2ccccc2c1=O N1(C(CCCOCCC)=O)CC(O)CCC1C(=O)Nc1cccc(OCF)c1 c1(C(=O)NCC(CO)NC(C(C)CC2CC2)=O)ccccc1OCC(N)=O C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CCCC(NC(C2(C)CCCCCC2)=O)C1 C(C(C(=O)N1CC2COCC2O1)C(C)C)NC(c1n(CC)nnc1)=O N1(C(C2(CC#C)CCCO2)=O)CC(OC)CC(NC(c2ccc([N+](=O)[O-])o2)=O)C1 C#Cc1cc(C(=O)N(C)CC2CCN(C(=O)CC3(CC)CCC3)C2)ccc1C CC1CC(=O)NC1C(=O)NCc1cccc(NC(=O)CCC2CCCCC2)c1 C(C(C)(C)CC(=O)N1CCCC(C(C)(C)C)C1)N(C)CC1(C(=O)OC)CCC1 C=C(F)C1(CC(N2CC3(CCC3)CC2CNC(=O)CC(C)F)=O)CCOCC1 Cc1ccnc(NC(C2CCN(C(=O)CC3(O)CCCOC3)C2)C)n1 N1(C(C=C(CC)C)=O)CCC(N(C)C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CC(N2CCCC(C)(NC(=O)CCc3nccs3)C2)=O)CCCC2(CCC2)O1 c1(C(C(=O)NC(C)C)N(CCC(C)C)C(N)=O)cccc(NC2CCOC2)c1 C=C(C)CCCC(=O)NC1CC(O)(CNC(=O)C(c2cc(F)ccc2F)OC)C1 C1(CNC(Cn2cc(C)c3c2cccc3)=O)CC2CCC(C1)N2C(C1CC1C)=O Cc1cc([N+](=O)[O-])cnc1N1C2CCC1C(CNC(C1(O)CCOCC1)=O)C2 n1(CC(=O)N(C2CCC(NC(=O)C3CC3)C2)C)nc2n(c1=O)CCOC2 C(C(=O)NCC(c1ccsc1)C)(C1CCCC1)NC(C=CCOC)=O C(CN=c1[nH]c(=NC)[nH]c(=NC2CCC(CC3CCCN3C)CC2)[nH]1)SCC Cc1nc2cc(NC(C34CC3CN(Cc3ccccc3)C4)=O)ccc2o1 c1(N2CCCC(CCCNC(=O)C(=O)OC)(OC)C2)nc2c(C)c(C)ccc2s1 c1(OC)ccc(CC(=O)NCC2(NC(=O)Cc3cncnc3)CC2)nn1 Cc1c(C(=O)NC(C(=O)NCC(C)F)C2(C)CC2)ccn1C c1(C(=O)OCC)cnc(Cl)cc1NC(C1CC12CCN(C(=O)CC(=O)OC)C2)=O c1(CC(=O)NC2CCCN(CCCCCOC)C2C)cc2ccccc2nc1O N1(C(C(C2CCCOC2)OC)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC1C N1(C(C(CCOC)NC(C2CCC(C)CC2)=O)=O)Cc2cccc(C)c2CC1 CCS(=O)CC(=O)N1CCC(NC(=O)C=Cc2ccc(C3CC3C)o2)C1 C#CCC(CC(=O)N(CCNC(c1ccnc(C)c1)=O)C(C)C)c1ccccc1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CC(NC(=O)CC3CCCC3O)C1C2 n1(CC)c(C(=O)NCC2(C)CC(NC(=O)C3=NOC(C)C3)C2)cc2ccccc12 C(=O)(C(C)P(C)(C)=O)N(C1CCN(C(C(CCC)c2cccc(Cl)c2)=O)CC1)C Cc1cc(C(=O)NCC2(O)CCN(C(=O)C(C)CC3CC3)C2)c(Br)c(C)c1 C(=O)(C(CNC(c1cc(C2CC2)no1)=O)C(C)(C)C)NCCC(C(C)C)OC c1(C(=O)NCC(CNC(C(C2CC2)SC)=O)O)ccc(CS(N)(=O)=O)cc1 N1(C(C(C2CN(C(C3CCOC3)=O)C2)OC)=O)CC(=O)NCC1C(C)C C(C)(CNC(=O)C=CC(C)(C)C)(CO)NC(C1C(C(=O)OC)CC1)=O c1(OC)cc(N(C)CCNC(=O)C(C(C)O)N(C)C)ccc1NC(C)=O n1(CC(=O)NC2CCC(NC(c3csnn3)=O)C2)cc(Br)ccc1=O C1(NCC)CCCCN(CCc2nccs2)C1.C1(C2CCCC2)C(=O)O1 N1(C(c2c(CC)ncs2)=O)CCC2(C1)CN(C(c1cc(C(C)=O)on1)=O)CCO2 Cc1cc(OCCC(=O)N(C)CC2CCN(C(=O)C(C)CC(C)C)C2)cc(C)c1 C=CC(C)CC(=O)N1CC(C)(CC(=O)NCCC(C)(O)C2CC2)C1 c1(C(N2CC(C)C(CNC(C3SCCS3)=O)CC2)=O)ccc(F)c(S(N)(=O)=O)c1 N1(C(C(C=CC)O)=O)CC2CCCC2C1C(N1C2CCC1CC(CCO)C2)=O Cc1cccc(CC(=O)NCC2CCC2CNC(=O)CC2CCCOC2)c1Cl c1(NCC(c2cccc(Br)c2)C(=O)OC)cc(Br)ncc1[N+](=O)[O-] C(=O)(C(C)CCCC(C)C)N(CCN(C(c1nc(C(C)OC)oc1)=O)C)C(C)C S(=O)(=O)(c1cccc(C(N2CC(CO)CC(C)C2)=O)c1)N(CC)CC1CCOCC1 C1(CC(=O)NCCN(C)C(C2CCC(=C3CCC3)CC2)=O)CC(O)C12CCC2 N1(C(C2(COC)CCCC2)=O)CCCCC(NC(=O)C(c2ccc(Cl)cc2)O)C1 C1(C)(NC(CN(C)Cc2ccccc2)=O)CCN(Cc2cc[nH]n2)C1 n1(CCN(C(C2N(C)CC2)=O)C)cc(-c2csc(NC(C)(C)C)c2)nn1 N1(C(C=CCOCCOC)=O)CCC(NC(=O)Cc2ccccc2O)C(O)C1 c1(C(C)C)nc(NC2C3CC2CN(C(=O)CCC2CCCCO2)C3)cc(Cl)n1 c1(OC)ccc(CC(N2CCC(NC(C3C(C)C3C)=O)C2C(C)C)=O)c(OC)c1 c1(CC)cccc(C)c1C(N1CCC(CN(CCCNC(C)=O)C(C)C)C1)=O c1(CCC(=O)N(CC(C)NC(C2(C)ON=C(C)C2)=O)C)cccc([N+](=O)[O-])c1 N1(Cc2ccn(CC)n2)CCC2(CC1)CN(C(C1CCCCC1OC)=O)C2 C1(O)(CN(C)C(C2CC(F)C2)=O)CCN(C(=O)CSc2cn[nH]c2)C1 n1(CCOC)nc(C(=O)NCC2C=CCN2C(=O)Cc2cnn(C)c2)ccc1=O N1(C(CC(CC)C(F)F)=O)CCCC2(CCN(C(=O)C=CC3CCCC3)C2)C1 C1(F)(CNC(c2cncc(C)n2)=O)CCCN(C(=O)C2=CCCCC2)C1 C1(NC(=O)NCC2CCC(C)(CC)O2)CCOC2(CCSCC2)C1 C1(NC(c2cn(C)c(=O)cn2)=O)CC2CCC(C1)N2C(C1C2CCCCCC12)=O C1(CNC(C2CCC2c2ccncn2)=O)CCCCN1C(C1(F)CC=CC1)=O C(=O)(C(F)Cc1ccccc1)N1CC(CC(=O)NC2CCN2C2CCCC2)C1 C(=O)(C1=COCCC1)NCC(C)C(=O)NC1CC(CN(C)C)C1 c1(OC)c[nH]nc1C(=O)NC1(C)CC(NC(=O)C(c2ccccc2)C)C1 C12(C(N3CCCC(CCC(=O)NCc4nc(C)c(C)[nH]4)C3)=O)CCCC1OCC2 N1(C(c2cc(C)[nH]c2C)=O)CCC(CN)CC1C.C1(C)(C=O)CCN(C)C1 N1(C(CCN(CC(C(C)C)C)C)=O)CC(NC(c2nsnc2O)=O)C(N=[N+]=[N-])C1 C1(C(N2CC(CC)N(C(=O)CCc3nccn3C)CC2)=O)OCCOC12CCC2 n1(C2(C(=O)NCC3C(CNC(CCCSC)=O)C3)CC2)cnc2ccccc12 C1(CNC(C2(OC)CC2)=O)CCN(C(=O)CC2CCCCC2(F)F)C12CC2 C(CN=C(NCc1cnc(-c2ccccc2)o1)NC(CC)C1CCC1)OCC c1(C(N2CC(C)(CNC(C3CN(C(C)=O)C3)=O)OCC2)=O)ccc(C#N)c(C)n1 N1(C(c2ccc(=O)oc2)=O)CCC(NC2CC(C(=O)OCC=C)OCC2)CC1 Cc1nccnc1C(=O)NC1CC(NC(c2ccnc(OC3CCOC3)c2)=O)C1 CC(CC(=O)NCCC1CC(NC(=O)Cn2cnc([N+](=O)[O-])n2)C1)C(F)F N1(C(c2ccc(OC)s2)=O)CCCC(C(=O)Nc2ccnc(Cl)c2)C1 c1(CC(N2CCC3C2CCN3C(c2ccc(Br)nc2)=O)=O)ccc2nonc2c1 C1(NC(Cn2cc(-c3ccc(OC)nc3)nn2)=O)CCCC(C(C)(C)C)CC1 N1(CC2(NC(C34CC(C(C)C)(C3)C4)=O)CC2)CCN(C(=O)CN2CCCC2)CC1 c1(C(=O)NC2CC(NC(C3CCC(C)C(C)C3)=O)C2)cnc2ccc(C#N)cn12 N1(C(C(C#N)CC2CC2)=O)CCCC(CNC(=O)C=Cc2cnccn2)CC1 CC(CCCc1ccccc1)C(=O)NC1(c2nc[nH]n2)CCCC1 C1(C(N2C(C)(CC(=O)NCCCC#C)CC2)=O)(C(N)=O)CCCCC1 N1(C(c2c(OC)ccnc2)=O)CCOCC(NC(=O)C(C(C)C)C2CCC2)C1 C(CC(C(C)(C)C)NC(c1ccc(C#N)o1)=O)N(C)C(c1cccc(F)c1Cl)=O N1(C(C(C(CC)O)C)=O)CCCC2(CCN(C(c3nc(=O)n(C)[nH]3)=O)C2)C1 N1(C(c2c(C(C)C)occ2)=O)CCC(C(C)NC(=O)CC2CCC(C)O2)CC1 CC1COCCN(C(C23COC(C2)C(NC(C2CC2Cl)=O)C3)=O)C1 Cc1ccc(C(F)C(=O)NCCCN(C(=O)Cc2cnccn2)C(C)C)cc1 c1(C(N2C(C)CN(C(=O)Cc3c[nH]ccc3=O)CC2)=O)cc(F)c(Cl)cc1F N1(C(c2cn(C)nc2O)=O)CC2CN(C(c3cc(C#N)ccc3N)=O)CC2C1 CC(C(=O)NCC(C)(O)CNC(C1CCC(O)CC1)=O)C(C)(C)C C1(CNC(C(C2CCCCC2)NC(=O)CCCC2CCCO2)=O)C2CCCCC12 c1(Cn2cc(CC(C=C)O)nn2)cccc(CNC(C2C3COCC23)=O)c1OC Cc1cnc(C(=O)NC(CC(F)F)C(=O)NCC(F)C(C)(C)O)c(F)c1 CCCCC(C)(F)C(=O)NCc1ccc(C(=O)NC(C(=O)OC)C2CC2)s1 Cc1cc(Cl)c2c(c1)CCN(C(c1cccc(N3CCCNC3=O)c1)=O)C2 CCC(CO)(C(=O)NC1(CCCC(=O)N(C)CCC2CCCO2)CCC1)OC C1(C(N2CC(C(C)(C)O)(CNC(=O)Cc3ccsn3)C2)=O)CC(=O)C1(C)C c1(C(N(CCN(C(=O)CC=Cc2ccccc2)C(C)C)C)=O)cc2cscc2s1 CC1CN(C(c2cncc3cccnc23)=O)CC(C)N(C(C2COCCO2)=O)C1 N1(C(c2cc(C)c(O)cc2)=O)CC2CCC1CN2C(c1ccc2snnc2c1)=O C12(C(=O)NC3C(C)(C)OCC3)CCCC1CN(C(c1cnc(=N)[nH]c1)=O)C2 CCC(C)CC(=O)N1CC(NC(c2ccc(C3CC3)s2)=O)C(CC)C1 Cc1cc(C(=O)NCCCN(C2CCCC2)C(c2csc(C#N)c2)=O)c(C)cn1 N1(C(C(C)OCC)=O)CC(NC(c2nc3cccnc3s2)=O)C2(CCC2)C1 C1(C(N2CC(NC(c3c(C)cns3)=O)C(C)(C)C2)=O)CCCC2(CCC2)C1 C1(NC(=O)CC2CC2)CN(CCc2cn(-c3cccc(F)c3)nn2)C2CCCC12 N1(C(c2cccc(C)c2Br)=O)CCC(C)(C(=O)NCC2CN(C(C)=O)C2)CC1 N1(C(c2cc[nH]c2)=O)CCN(C(=O)C(O)Cc2cccc(Cl)c2)C2CCC12 c1(CC)ccc(C(N2CC3CC2C3NC(C2(C3CC3)CC2)=O)=O)cc1Br C1(NC(=O)Oc2cc(COC)oc2-c2ccccc2)Cc2cc(OC)ccc2O1 C1(CNC(c2c(C)ncnc2O)=O)C2CCCC1N(C(C1CC(C)OC1C)=O)C2 C(=O)(CC(CC)C(C)(C)C)NC1CCCC1.CCCCN(CCO)C(=O)C1CC1 C1(n2c(-c3cnn(CCO)c3)nc(C(C)C)n2)CCC(F)(F)CC1 C1(C)(C(N2CCN(CC3CN(C(CCC#CC)=O)C3)CC2)=O)COC(=O)OC1 C1(F)(C(=O)NC2CC(C)(NC(=O)CCN3CCOC3=O)C2)C2CCCCC12 c1(C(=O)OC)cc(O)cc(S(=O)(=O)N2CCC(C)C(c3ccccc3)C2)c1 c1(C(=O)OCC2CCCO2)ccccc1.C1CO1 c1(C(=O)N(c2ccccn2)O)ccc(SCCCNC(c2cn[nH]c2)=O)cc1 C1(C2CC2)(CNC(c2cc(CC(C)C)on2)=O)CCN(C(C2CNC(=O)C2)=O)C1 c1(C(C)=O)cc(C(=O)NC2CCCCC2n2cc(COC(C)C)nn2)cc(F)c1 Cc1cc(Cl)cc(Cl)c1OCC(=O)NC(C)CNC(=O)Cc1cccn1C C1(N(C)C)(CC)CCN(C(C2C3CC2N(C(=O)C(C)=C2CCCC2)C3)=O)C1 CC1(C)CCCC(O)(C(=O)NC2CCC2NC(c2cccc3nccn23)=O)CC1 CC1CN(C(c2cc[n+]([O-])cc2)=O)CCN1C(=O)CCc1cnccn1 c1(C(N2CCC(CNC(C3(OC)CCC3)=O)C23CC3)=O)cc2occc2n1C c1(C(=O)NC2CC(CCNC(C(C)(C)SC)=O)C2)n[nH]c(C)c1Br C1(NC(c2c(C)csc2)=O)CCN(C(c2cc(Cl)ns2)=O)CCC1CO C(C(=O)NCC1C=CCN1C(c1cc(C(N)=O)no1)=O)(C(C)(C)C)SC c1(OC)ccc2c(c1)CC(C(=O)NC(C1CCCCC1)C(C)NC(=O)CC#N)O2 c1(C(=O)NCCNC(C23OCCCC2C3(F)F)=O)c(O)nc2ccccc2c1Cl c1(CC)ccc(F)cc1C(=O)NC1CC1NC(c1c[nH]nc1Br)=O Cc1noc(C)c1CC(=O)N(C1CC1)CC1CN(C(=O)CO)C1.C1(=O)CCN1 N1(C(Cc2ncc(C)s2)=O)CC2C3CCC(C2C1)N(CC1CCOC(C)C1)C3 Cc1ccc(C(C(=O)NCCCC2CC2)N(CC(=O)N(C)C)C)c2ccccc12 c1(C(N2CC(CNC(C3(OC)CCC3)=O)(OC)C2)=O)cn(C(C)(C)C)nc1C Nc1ccc(C(N2CC3CC2C3NC(c2cnn(CC3CCC3)c2)=O)=O)c(Cl)c1 N1(c2nc(=N)nc(N(C)Cc3cccnc3)[nH]2)CCC(C2CCN(C)C2)CC1 C1(CC(=O)NC(C#C)C2CCC2)CCN(C(=O)C(O)C=CCCC)CC1 C12(C(N3CCC(N(C(=O)Cc4cscc4C#N)C)C3)=O)CCC(CO)(CC1)CC2 Cc1cc(=O)ccn1CC(=O)NCC1(O)CCN(C(=O)CCc2cn(C)cn2)C1 c1(N2CCC(NC(C(C)NS(CC)(=O)=O)=O)C23CCC3)ncnc2c1nnn2C C1(C#N)(C(=O)NC(CCOC)CNC(C2CC(C)=NO2)=O)CCCCC1 N1(C(C=CC(C)NC(c2ccc(C(C)C)o2)=O)=O)CCN2C(=O)OCC2C1 C(C(C)(C)CC(=O)NCc1cc(C(C)C)n[nH]1)NC(C1C(C)OCCO1)=O C1(NC(c2ccc(C)nc2O)=O)CN(C(=O)C(C)(C)CF)Cc2nccn2C1 NC(=O)C(O)CCCNC(C1CC(O)CN1C(=O)Cc1ncccc1F)=O N1(C(C2CCCN(c3cc(C)nn3C)C2)=O)CC(C)(C)CC1CO c1(CNC(C)C(=O)OC)ccc(C2N=N2)cc1.S(S(C)(=O)=O)CC(=O)NC(C)(C)C N1(C(c2c(CC)nn[nH]2)=O)CC(NC(=O)Cc2csc(S)n2)C(SC)C1 c1(CNC(=O)NCC2(O)C3(c4ccn(C)n4)CCC2C3)c[nH]c2ccc(Br)cc12 N1(N2CCC2)CCN(C(=O)C=CC(=O)OC(C)(C)C)CC1.C(=O)(C(Cl)=CCl)OC.CC Cc1ccnc(Oc2ccc(NC(c3cnc(C)[nH]3)=O)cn2)c1 c1(CC(=O)NCC2(O)CN(C(=O)NC3(O)CCC3)C2)ccc(C2CC2)o1 c1(C(c2cn(C3CCN(C(=O)Cc4cocn4)C3)nn2)(C)C)cccc(Cl)c1 C[S+](C)CCC(O)C(=O)NCC1CCN(C(C2(C)CCC3(CC2)CC3)=O)C1 C1(C(N2CC(NC(c3c(C(=O)OC)cccn3)=O)C2)=O)CCC2C1C2(F)F n1(CC(=O)NCC2CC(NC(c3cnoc3-c3cccs3)=O)C2)cc(C2CC2)cn1 C=CC1OCCC1C(C)(C)NCc1nc(C)cs1 CC(C)CC(O)C(=O)NC1CC(NC(=O)C(C(C)C)c2ccccc2)C1 c1(C(=O)NC2C(C(N(C(CC)C)C)=O)OCC2)ncccc1Cl CCCC(C#N)C(=O)N1CC(CNC(c2cnc(C3CC3)nc2)=O)C(O)C1 CCC(CC)C(C)C(=O)N(C(C)C(=O)N(C)CC1CCCCC1O)C CC1(C)CCCOC1C(N1CC(CNC(c2cc(C#N)c[nH]2)=O)CC1(C)C)=O c1(N2CCC(F)(C(=O)Nc3c(C)cc(Cl)nc3)C2)ccn2ncc(I)c2n1 c1(C(=O)NCC(C(=O)OCC)CC)cc2cc(C)cc(C)c2[nH]1 CC1CC=C(C(=O)N2CCCC2CC(=O)NCC(O)CC(C)C)CC1 C1(C2CCC2)(CNC(CN2C(C)CC2)=O)CCN(C(=O)Cc2nc[nH]n2)CC1 N1(C(CCC)=O)CCCC(C(N2CCC(N(C)C(c3cc(Cl)n(C)n3)=O)C2)=O)C1 CC(C)C(C(=O)NC1CC(CCNC(=O)Cc2ccc(Cl)cn2)C1)N(C)C N1(C(c2ccc(C(F)(F)CF)cn2)=O)CC2CC1CN2Cc1ccccc1 c1(CN(C)CC2CCCCCCN2)cc2ccccc2nc1O N1(C(CC(C)N(C(CSCC)=O)C)=O)CC(C)C(C)C1C Cc1cc2c(C(=O)NCC(C)N(C)C(C3CCC4(CCC4)C3)=O)cccc2o1 c1(C(=O)NCC(C)NC(=O)C(C)Cc2ccccc2)ccc(F)c2cnccc12 c1(C(=O)NCC2CN(C(c3c(C)onc3)=O)C2)cccnc1CC(C)C c1(CC#N)cccc(S(=O)(=O)N2CCCC3(CCOC3)C2)c1 C1(F)(CNC(c2cccc(F)c2F)=O)CCCN(C(=O)CCC2CCCOC2)C1 C(=O)(CC(C(C)(C)C)NC(C1CCC2CC1CO2)=O)Nc1cccc(CC)c1 C12(NC(c3ccc(O)nn3)=O)CCC(C1)N(C(=O)Cc1nc(C3CC3)cs1)C2 c1(C(CC)(C)C)ccc(CCCNC23CC4CC2C3C4)cc1 c1(C(N2CC(CNC(C=CS(C)=O)=O)C(C)(C)C2)=O)cnc2ccccc2c1 c1(C(N2CC(O)CCC(NC(C(C)(C)C(F)F)=O)C2)=O)cn2cccc(Cl)c2n1 C1(NC(C2CCSC2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC2(CC2)C1 C1(C)(C(=O)NC(CCC)CCCNC(c2ccc(C)o2)=O)CCS(=O)(=O)CC1 C1(NC(CN(CCCCCC)C)=O)CC2(C1)CN(C(C1CCOC1C)=O)C2 c1(C(N2C3CN(C(=O)CC4CC4(Cl)Cl)CC2CC3)=O)ccc2c(c1)OC(F)(F)O2 CCC(CCOC)NC(=O)CCCC1(NC(c2c[nH]nc2OC)=O)CCC1 C1(C(=O)NCC2C(NC(Cn3nnc(C)n3)=O)C2)CCc2ccccc2O1 N1(C(C(CC)N(C(=O)C2CC2)C)=O)CC(NCc2ncnn2C)CC(C)C1 c1(C(=O)NCC2CN(C(C=CS(C)=O)=O)CC2O)cc(F)c(Br)cc1F c1(C(=O)NC2CCC(N(C(CCC=C)=O)C)C2)c(C)ccnc1C C(=O)(C1CCCc2n[nH]cc21)NCC1C(C)CCN1C(=O)CCc1cnoc1 c1(C(=O)NC2(CNC(=O)C=CC3CCCCCC3)CC2)cc2cc(O)ccc2[nH]1 c1(C(=O)NCCCN(C)C(C2CCC(=O)N2C2CC2)=O)cc2cnccc2o1 CC1(C#CC(=O)NC(CCCC=C(C)C)=O)CCCO1.c1(C)cnc2n1CCC2 CC1CC2CCC(C(=O)NCC3=CCN(C(=O)C(=O)C(C)(C)C)CC3)CN2C1 c1(C(=O)NCC2CCCN2C(=O)CCCc2ccncc2)ccc(O)nc1 c1(C(N2C(C(N(C)Cc3ccc(Br)cc3)=O)CC(F)C2)=O)c(Br)ccc(F)c1F c1(NCCNC(=NCCCC2(OC)CCC2)NC(C)CC)ncnc2[nH]cnc12 N1(C(c2c(C)onc2)=O)C2CCC1C(CNC(=O)Cc1csc(Cl)c1)C2 Nc1cc(C(=O)NCC(CNC(=O)C(O)C2CCCC2)S(C)(=O)=O)cnc1Cl CCCCCCC(C)C(=O)NC1COCC1CNC(=O)CC1(SC)CCC1 c1(C(=O)NCCCN(C(CC(CC)OC)=O)C)cn2cccc(Br)c2n1 c1(-c2n(-c3c(C(C)C)cccc3)nc(-c3ccc(N)cc3)n2)ncc(F)cc1N c1(C(N2C(CNC(=O)CC3CC3C3CC3)C=CC2)=O)ccccc1C(F)F CC1CCC(CNC(=O)CCc2ccc(F)cc2)N(C(=O)COCCF)C1 C1(CCCC)CN(C(C2NC(=O)C3CC23)=O)CCN1C(=O)C1=CCCC1 CCCC(CC)CC(=O)N1CCC(OC2CN(C(c3cnn(C)c3N)=O)C2)CC1 c1(SC)ccccc1C(=O)NC1(C)CCN(C(=O)CC2CC(C(C)(C)C)C2)C1 c1(COC)cc(C(=O)NCCCCC2CC2)no1.N12CC(C1)CNC2=O c1(C(=O)NC23CC(C(=O)NC(c4ncc[nH]4)CC)(C2)C3)ncc(F)cc1F C1(NC(CSCCNC(CCc2cc(C)[nH]n2)=O)=O)CC(O)CC1O Cc1cnccc1C(C)C(=O)NC1CCCCC1N(C)C(c1cccs1)=O C1(C(N2C(CNC(c3c(N)csn3)=O)CC3CCCC32)=O)CCOC2(CCC2)C1 c1(CC)cc(NC(c2ccc(Oc3ccc(C)nn3)cc2)=O)cnc1C n1(CCC(=O)NC(CC=C)CNC(c2c[nH]nc2C(C)C)=O)cnc(C)cc1=O C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(NC(=O)CC(C)(C)CN(C)C)CC(C)C1 c1(CNC2CCCC(CC(=O)O)(C(F)(F)F)C2)c(OC(F)F)ccc2ccccc12 C12(C(=O)NC(C(=O)OCC)CCc3ccccc3)CCC(CC)(C1)OC2 Cc1cc(C#N)nc(NC23CCCC2CN(C(=O)C(C)N(C)C)C3)n1 c1(CC(N2CC(NC(C(C)(C)SC)=O)C(C)(C)C2)=O)ccc(S(=O)(=O)N(C)C)o1 c1(C(C)OCC)cn(CCOCCNC(=O)CCn2ccnn2)nn1 c1(C(=O)NC2C(CC(=O)O)CC2)cncc(-n2cc(C3CC3)nn2)c1 c1(CC)ccc(C(=O)NCCCC(C)(C)NC(c2ccc(C)c(F)c2)=O)c(C)n1 c1(OC)ccc2c(c1)C(CCN(CC(F)(F)F)Cc1cccc(C)c1)=CC2 N1(C(CN(c2ccccn2)C)=O)CCC(O)(CCNC(=O)C(C)(C)N(C)C)C1 CCCN=C(NCC1CC1Cl)N1CCC(F)(c2cc(OC)cc(OC)c2)CC1 c1(C(=O)NCCOCCOCCNC(C2CC2Cl)=O)ccc2c(c1)CCN2 C#CCC(O)C(=O)NC1CC(NC(=O)C(F)(F)c2ccsc2Cl)C1 N1(C(c2cc(OC)n(C)n2)=O)CCOCCC1C(=O)NC1C(C)C1C C(=O)(C#CC1CCC1)NC1C(CNC(c2c(COC)cccc2)=O)CCCC1 C1(C(N2CC3C(NC(C=C(COC)C)=O)(C3)C2)=O)CC2(CC(C)=NO2)C1 N1(Cc2ccc(C)o2)CC2CCC1CN(c1ncc(I)cn1)C2 O=C(C(C1=CCCSC1)N1CCSCC1CCSc1ccccc1Br)NCCO N1(CC(N2CC(CNC(C(COC)OC)=O)C2)=O)C(=O)c2ccccc2S1(=O)=O c1(OC)c(C(N2CC=CC(NC(=O)CSC(F)(F)F)C2)=O)[nH]c2ccccc12 [N-]=[N+]=NC1CN(C(=O)CC2OCCO2)CC1NC(C1CNC(=O)N1)=O c1(C(=O)NCC2C3CN(C(c4ccc(OC)cn4)=O)CC32)cc2ccsc2cn1 c1(CCNC(Cc2c(I)ccc(C)c2)=O)cc(Br)c2c(c1)CCO2 c1(OC)ccc(CN2CCNCC2C(=O)NCc2ccc(Br)cc2)c(Br)n1 N1(C(CC=CCC)=O)CC2CCC(C1)N2C(=O)Cc1nnc(S)n1C c1(CC)c(C(N2CC(CC(C)NC(=O)COC)C2)=O)oc2ccccc12 N1(C(Cc2ccn(CC)n2)=O)CCCN(C(C2CC3CCC3C2)=O)CCC1 N(C(=NCCCF)NCC(=C1CCSCC1)F)Cc1ccc(C(C)C)c(F)c1 C12(CCNC(COC(C)=O)=O)CCC(C1)N(C(=O)CCOC1CCCCCC1)C2 C1(C(=O)NC2CCN(CCC)CC2)C2CC(O)C(C2)N1C(=O)C=CCO c1(OCCCC(=O)N2CC(N(C(=O)C(C3CC3)OC)CC)C2)cccc(C)c1C c1(NC(c2ccnc(C)n2)=O)ccc(NC(c2scnc2C)=O)c(F)c1 c1(SC)cc(NC(c2cc(-c3ccn(C(C)C)n3)ccn2)=O)ccn1 C(CC(C(C)(C)C)NC(=O)C1=C(Cl)CC1)N(C(CCCN(C(C)C)C)=O)C C1(CNC(C(C)NC(CC)=O)=O)CN(C(=O)C(O)C(C)C)CCC1C(F)(F)F C1(CC(F)F)(C(=O)NCCCC(C)NC(C2CCC(C)(C)O2)=O)CCOCC1 C1(C)(CNC(c2cc(CC)nn2C)=O)CCN(C(C2CC2(F)Cl)=O)CC1 N1(C(C=CC=CC)=O)CCCCC1C1CCN(C(=O)C(C)n2cnnn2)CC1 N1(C(C(C2CCCC2)OC)=O)CCN(C(=O)C=CSCc2ccco2)CC(C)(F)C1 C#CC1(CNC(=O)C(CC(N)=O)NC(=O)CCSCCC)CCOCC1 c1(N2CCN(CC3(C#N)C(C)(C)C3)CC2)cc2occc2[nH]1 C1(CNC(CC2CC(CN(C)C)C2)=O)CN(C(=O)C(C)(C)CC2CCC2)CCO1 C1(CNC(=O)COC(F)(F)C(F)(F)F)CCCCC1NC(=O)CN1CCOCC1 Cc1cc(C(N2CC3(NC(c4cc(C(C)C)[nH]n4)=O)CCC2C3)=O)cc(C)c1N C1(CNC(c2c(CC)ccs2)=O)CCC2(CN(C(c3[nH]ncc3C#N)=O)C2)O1 C1(NC(C=CC(=O)N(C)C)=O)(CF)CCN(C(C2COC(=O)O2)=O)C1 CN1CC(O)CCC1C(=O)NC1CC(Cn2cc(COc3ncccn3)nn2)C1 N1(C(C(C)OC)=O)CCCCCC1CNC(c1ccc(Br)nc1O)=O N1(C(c2cc(C)sc2)=O)CCC(F)C(NC(c2nc(C)oc2C)=O)C1 c1(C(C(=O)NCC(C2CCCC2)NC(C2(C)CC2(F)F)=O)(C)O)ccccc1F c1(C(=O)NC(CN(C(=O)CC(C)SC)CC)C)nnn(C)c1N Cc1ccc(CNC(C23COCC2C3(F)F)c2nnnn2C)nc1C C(=O)(CCCNC(=O)NC1CC1)N(C(CO)C1C(Cc2cscn2)C1)C C(=O)(C1COc2ccccc21)N1CCCN(C(c2c(O)cccc2Cl)=O)CC1 C(CCCCNC(c1cnc(C(C)OC)s1)=O)NC(C1C(=C)CC1)=O CCC(S(=O)(=O)NCC1CCC(N)CC1)c1ccccc1 C1(C(=O)NC2C(CC=C)CCCC2)CN(C(C2(C)CCCO2)=O)CC1(F)F C(=O)(C1=C(C)CCCC1)N(CC)CC1CCCCN1C(=O)CCc1cc[nH]n1 C1(CCNC(CS)=O)(C)CC1(F)F.C1(c2cc[nH]n2)(NC(CC(C)=O)=O)CCC1 N1(C(c2n(CC)ccn2)=O)C2CCCC1CC(N=c1[nH]c(Cl)ncc1C1CC1)C2 N1(C(CC2CN(C)C2)=O)CC2CCCN(C(C34COC(CF)(C3)C4)=O)C2C1 N1(Cc2cnc(N3CC4CC4C3)s2)CCOC2(CCCNC2)C1 c12ccc(O)c(c1)C(=O)NCC(=O)OC2.N1(C(C)=O)CCOC(CNC(C)=O)C1 c1(SCc2cn(CCCNC(CNC(CC)=O)=O)nn2)cc(C)cc(F)c1 c1(NC(C2CCN(C(=O)CNCCC(F)(F)F)C2)=O)cccc2c(O)nccc12 c1(CN2C(C)(C(=O)NCc3cc(OC)ncc3)CC2)cccc(OC)c1OC N1(C(C2=CCN(C)C2)=O)CCC2(CCN(C(=O)Cc3ccc(F)cc3)C2)C1 CC(CCNC(=O)CSc1ccccc1)CCNC(=O)CC(C)c1cnn(C)c1 C1(CN(C(c2cnccc2Cl)=O)CC)CCN(C(=O)Cc2ccc(F)cn2)CC1 N1(C(CC(CC)O)=O)CCCC2(CCCN(c3ncnc4[nH]cc(I)c34)C2)C1 N1(c2nc(COC)nc(C)c2)CC2CCC1C1CN(C(C3CC3(C)Br)=O)CC21 C1(C)(CNC(C2CCN(C)CC2)=O)CCCN(C(=O)CCCNC(=O)C=CCl)C1 N1(C(CC(CNC(c2c(C)ccnc2)=O)O)=O)CCC(C)(C)C1CO C1(NC(C=CC(CC)C)=O)CCN(C(=O)Cn2nc(C(F)(F)F)cc2C)CC1O CC(C)(CCNC(=O)CSc1nncs1)C(=O)NCC1CCC(CO)O1 C12(NC(C(CCSC)O)=O)CCCC(NC(=O)CCc3ccc(N)cn3)(C1)C2 c1(C(N2C(C)CC(CNC(CN(C)CC)=O)C2)=O)cc(Br)cc2c1OCO2 C(=O)(C1=CCCCC1C)N(CCOC)CCNC(=O)Cc1ccc(OC)cc1 C(Cc1ccccc1)(Cc1ccccc1)(c1nnnn1C)N(C1CCCO1)C N1(C(COCC=C)=O)CCC(C)C(CNC(=O)Cn2cccn2)C1 CC(=Cn1ccnn1)C(=O)N(CC(C)N(C(=O)CC1C=CS(=O)(=O)C1)C)C C(=O)(C(CC1CCCC1)NC(=O)C1CC1)N(C1CCCCC1)CC(=O)OC CC1(C)C(=O)CC1(P(C)(C)=O)C(=O)NC1CCN(C(=O)Cc2csnn2)CC1 C(=O)(C#CC1CCOC1)N(CCCCCNC(C1CCCCN1S(C)(=O)=O)=O)C c1(OC)ccc(=NC(=O)Cc2cc(-c3c(OC)cccc3F)cs2)[nH]n1 N1(N2CCC(CN3CCN(Cc4ccc(SC)o4)CC3)C2)CCOC2COCC12 c1(C(=O)NC2C(OC)CN(C(C3N(CC)C(=O)CC3)=O)C2)cnc2[nH]ccc2n1 C=C(C)CC(C)C(=O)NCC(CC(C)C)NC(c1ccc(OC)c(N)c1)=O CCS(=O)(=O)c1cccc(S(=O)(=O)N2CCCC(CO)CC2)c1 N1(C(Cc2nc(NC=O)sc2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C2CC12 c1(C(N(C)CC2CCN(C(C3(C#N)CCC3)=O)C2)=O)csc2ccncc12 c1(C(=O)NC(C)CCCNC(C2CC23CCCC3)=O)ccc2nnc(S)n2c1 Cc1cc(=NC(=O)C(C)OC(=O)CCc2ccc(Cl)cc2Cl)[nH]o1 C(C(C)CC(=O)N1CCCCC1C(=O)N(CCS(C)(=O)=O)C)OC N1(C(C(CC)CN(C)C)=O)CCC(NC(c2cc(C(N)=O)[nH]n2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc(NC(C2CCN(C)C2)C)cc1Br)NCc1nnc(COC)s1 C1(N(C(C2C(=C)C2)=O)CC)CCCN(C(c2cc(OC)cc(C)c2)=O)CC1 CC(C)(CCN=c1ncc2ccccc2[nH]1)NC(C1(c2ccc(F)cc2)CC1)=O CCC1=C(C)CC(COC)N1Cc1cnn(C(C)(C)C)c1C1CC1 N1(C(CCCC(=O)NCC)=O)C2CCC1CN(C(=O)C(C)C(O)CC)C2 C1(C(=O)NCc2cc(C)no2)C(C)OCCN1C(=O)C(C)CC(N)=O N1(CC)OCC(NC(=O)CC2(C)CCN(C(C3SCC=C3C)=O)C2)C1=O CC1COCC(CC(=O)NC(C(=O)NCCC2CC=CC2)C(C)O)O1 N1(C(CC(=O)NCC)=O)CCC(C)C(NC(=O)CCNC(C)C)C1 c1(C(=O)NCC(=O)NC2CC(CNC(=O)CC3CSCCS3)C2)cccc(O)c1 c1(C(N(C2CN(C(C(C)OCC#C)=O)CC2(C)C)C)=O)cccc2nn(C)nc12 CC(C)(CCC#N)C(=O)NC1CCC(NC(c2ccc([N+](=O)[O-])cn2)=O)CC1 c1(C(=O)NCC2(C)N(C(C(C=C)O)=O)CC(F)(F)C2)ccc2cnc(C)n2c1 c1(CC)onc(C(=O)NCCCCCn2cc(C3(O)CCCC3)nn2)c1C C1(NC(CC(CCC)C)=O)CN(C(=O)CCc2cc(C)[nH]n2)Cc2ccnn2C1 C(=O)(C(C)(C)CC(=O)NC(C)(C)CNC(=O)CCN1CCC(F)C1)OC N1(C(C2(F)CC(C(=O)OCC)C2)=O)CCC(NC(=O)CS(N)(=O)=O)C12CCC2 C(CC(C)CCS(=O)(=O)N1C(NC(=O)OC(C)(C)C)CC2OCCC12)OC S(=O)(=O)(c1cnc(Cl)c(Cl)c1)NC1(C#C)CCC(C(C)(C)C)CC1 C1(CNC(C(N2CCSCC2)C)=O)CCCN(C(c2ccc(F)cn2)=O)CC1 c1(CNC(C2CN(C(=O)OC(C)(C)C)C2)C(=O)NCC(=O)O)cncc2c1CCC2 c1(C(N2CC(CNC(c3cc(CCC)nn3C)=O)(OC)C2)=O)cc(C)c(O)nn1 C1(NC(c2[nH]cc(C)c2)=O)CCOC12CCN(C(C1CCCC13CC3)=O)CC2 c1(CNC2(CNC(c3c(C)ccc(Cl)c3)=O)COC2)ccc2cc(F)ccc2n1 C1(C(=O)O)CCCCC1C1CCN(CC(N2CCCCCCCCC2)=O)CC1 Cc1ccc2c(c1)CCC(C(=O)OCc1cn(C(c3ccccc3)(C)C)nn1)O2 N1(C(C(CC#C)C2CC2)=O)CCOC2(C1)CN(C(C1CC3CC3C1)=O)C2 N1(C(C23CC(OC)C2C3)=O)CCC(N(C)C(c2cc(C(C)(C)C)n[nH]2)=O)CC1 CCC(C)CC(=O)NCC1(c2ccccc2)CC(NC(=O)CCN2CCC2)C1 C(=O)(C1Cc2ccccc21)NC1CCCN(C(c2ccnc(C)n2)=O)C1 c1(C(=O)NCCCC(C)NC(=O)Cc2ccon2)cccc(C2(F)CC2(F)F)c1 c1(OC)cc(CC(N2CCC(O)C(NC(C3CCCN3C=O)=O)C2)=O)ccc1C Nc1cc(Br)ccc1C(N1CCCC1CCCNC(=O)C(O)C(F)F)=O C1(NC(c2ccc(Br)cc2)=O)CN(C(=O)Cc2cncs2)CCC12CCC2 N1(C(CC(=C)Br)=O)CC(CNC(c2ccc(OC)nn2)=O)CC12CCC2 C(CN=c1nc(N2CCC(CN(C)C)C2)c2ncccc2[nH]1)c1ccc(C)cn1 C1(C(N(c2cccnc2)C(C)C)=O)CCN(c2ccnc(C3CC3)n2)CC1 C1(C2C(NC(C=CC(=O)N(C)C)=O)CCO2)CCN(C(=O)CC2CCSC2)CC1 C(=O)(C1SCc2cccnc21)NCC1C(NC(C2(CC)CCC2)=O)CC1 c1(OC)cc(CC(=O)NC(C(C)NC(C23CC(F)(C2)C3)=O)C(C)C)ccc1Cl N1(CCC)CCCCC1C(N1CCC(F)(CNC(c2coc(C)n2)=O)C1)=O C(=O)(CCC(=O)NC1(COC)CN(C(C2CCCN(C)C2)=O)C1)NC c1(C(N2CC3C(CNC(CC=CC)=O)C3C2)=O)c(C)oc(C)c1Br C12(C(N(CC(CC)(O)CC)C)=O)COCC1CN(C(C1CCCC(C#N)C1)=O)C2 C(=O)(C(C(C)CC)NC(C12CCCC1CCC2)=O)NC N1(C(C(C)OCC#C)=O)CCN(CC(=O)NC(C2(OC)CCC2)CC)CC1 C1(C(C)NC(C(CC)Nc2ccccc2)=O)CCN(C(=O)C(C)(C)COC)CC1 Cc1cc(Cl)ccc1C(=O)Nc1cc(-c2ccccc2NS(C)(=O)=O)ccn1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nccn2)cc(F)ccc1Cl C(=O)(C(F)C(C)(C)O)N(C1CCN(C(C(CC)O)=O)CC1)CC C1(C(C)(C)C)(CNC(C2(CC#C)CC2)=O)CCN(C(c2ccc(F)cn2)=O)C1 c1(NC(C2CCC(C(C)C)N2C(=O)C=CCF)=O)cc(F)c(O)cc1C n1(CC(=O)NC2C(NC(CC3(C)CCCCC3)=O)C2)ccc(O)nc1=O Fc1ccc2c(c1)C(c1nc(-c3cccs3)nn1C13CC(C1)C3)CO2 n1(CCC(=O)NCC2(F)CC(CNC(C(C=C)O)=O)C2)cc(Br)ccc1=O c1(C(=O)NCC(CC)NC(C2CC2c2ccccc2)=O)ncccc1O C(=O)(C(C(C)(C)C)NC(N)=O)NCC(CNC(C(C)CC1CCCC1)=O)C C(=O)(C1CCCc2cncn21)N1CCCC2(CN(C(C3C(=C)C3)=O)C2)C1 N1(C(CC2(C=C)CCOCC2)=O)CC(NC(C2OCCO2)=O)C(C2CC2)C1 c1(C(N2CCCN(C(C3CCCN3C3CC3)=O)CCC2)=O)ncc2ccccn12 O=C1CCN(C(c2cncnc2C2CC2)=O)CCCN1 c1(CC(=O)C(=O)OC)ccc(O)c(C)c1.C12CCN(CC1)C2.C1(SC)CC1C(C)C c1(C(=O)NC2C(NC(c3cc(C)c(O)cc3)=O)CC2)cc(P(C)(C)=O)cs1 C1(C(C(=O)NC2(CC(N)=O)CCC2)NC(c2cn[nH]c2)=O)CCCCC1 c1(NC(=O)NC(c2n(CC)cnn2)C)ccccc1OC(c1ccccc1)C c1(CC)ccccc1C1CN(C(c2sc(C3(C)OCCO3)cc2Br)=O)CCO1 O=C(CCCCCF)NCC1C2CCC(C2)N1C(C1CCCOCC1)=O N1(C(=O)CCC2CCCN2C(=O)CCC2CCCO2)CCCC2(CC(O)C2)C1 c1(NC(C2CN(C(C3CC3c3ccccc3)=O)CCN2)=O)nc(F)c(Br)cc1Br Cc1cccc2c(C(=O)NC3CN(C(=O)CC(C)(C)C#N)CC3N=[N+]=[N-])c[nH]c12 c1(C(=O)NCCN(C(c2ccc(F)cn2)=O)CC)cccc(C)c1[N+](=O)[O-] c1(CN(C(=O)CNC(=O)CC2CC2)CC)cccnc1 C1(NC(CCC2(NC(CSC)=O)CCCC2)=O)CCN2CCC1C2 Cc1c[nH]c2ncc(C(=O)NCC3C4CN(C(=O)CCCN(C)C)CC34)cc12 C1(NC(c2cnc(OC)nc2)=O)CCN(C(c2sc(C)cc2C)=O)CC(C)(C)C1 Cc1ccc(OCCC(=O)N(CC(C)NC(C2CC(N(C)C)C2)=O)C)c(C)c1 C#CCCC(=O)NCc1ncoc1CCNC(=O)CSCc1csc(=N)[nH]1 C1(SC)CCC(N=c2nc(N3CCC4(CCNC4=O)CC3)c3sccc3[nH]2)C1 C1(NC(COC(C)=O)=O)CCC(N(C)C(c2sc(Cl)cc2Cl)=O)CC1 c1(OC)cc(N(C)C)ccc1C(=O)NCCC(O)CNC(=O)C#CC1(C)CC1 Cc1cccc2c(=O)c(C(=O)NCC3CN(C(=O)C(C)CC(C)(C)C)C3)c[nH]c12 Cc1ccc(Cl)c(C(=O)NC(C2(O)CCN(C(=O)C(C)C3CCOC3)C2)C)c1 c1(C(=O)NC)cc([N+](=O)[O-])ccc1N1CC2(CN(C(=O)CC(C)SC)C2)C1 C1(NC(C(C(C)C)CN(C)C)=O)C2CCC1CN(C(c1cc[nH]c(=N)n1)=O)C2 N1(C(CCC#C)=O)CCC(NC(=O)CCN(C)Cc2ccccc2)CC1C1CC1 N1(c2n(CCC#C)c(-c3ccc(Br)c(C)c3)nn2)CCc2c(I)n[nH]c2C1 C1(NC(C2(NC(=O)OC)CC2)=O)C2CCC(C2)C1C(=O)NC1CCCC1N=[N+]=[N-] C1(CC#C)(C(N2CC(OCCNC(=O)CCc3cccnc3)C2)=O)CCCCO1 c1(CC(=O)NC2N(C3CCN(C(C(N)=O)=O)C3)CCCC2)nsc2ccccc12 C(=O)(C#CC1CCOC1)N1CCC(C)(NC(c2c(C)ccc(SC)c2)=O)CC1 c1(CCCC(=O)N(CC(C)(C)NC(C(C)C(C)(C)C)=O)C)nc2ccccc2[nH]1 C1(O)(C(C)NC(=O)Cn2cnnc2O)CCN(C(=O)CNC(=O)C(F)(F)F)C1 CCCC(CC(=O)NC(C)C(N)=O)NC(C1C=CCC1)=O N1(C(c2cc(C)[nH]n2)=O)CCC(C)(C)C1CNC(=O)CCN1CCCC1 Cc1cc(Br)ccc1CNc1c[nH]nc1C(=O)NCc1ccco1 CC1=CC(C)CN(C(=O)C(C)CNC(c2cccnc2N(C)C)=O)C1 c1(OC)cc(C(N2CCOCC(CNC(c3nnc(S)n3C)=O)C2)=O)cc(F)c1 N1(C(C=COCC)=O)CCN(C2CCN(C(C34CCC3CC4)=O)CC2)CC1 C(=O)(C(C)(C)C#C)N1CCC(CC(=O)N(CC#C)CC=C)C1.C1(=O)CN1C1CCC1 C1(N(C(C(CCC)NC(C)=O)=O)CCC)CCCN(C(=O)CCF)CC1 N1(C(CC=C)=O)C2CCC1CN(C(=O)C(C1CCOC1)NC(C)=O)C2 C12CC(C)N(C1)CN(C(=O)OC(C)(C)C)C2.C(C(=O)C1CCC1)(N(C)C)CC CC1CCCCC1(C)C(N1CCC(C(=O)Nc2ccccc2)C(C)C1)=O C1(C(N2CCC(C)C2CN(C(=O)C(C)CF)C2CC2)=O)CCc2cnn(C)c2C1 c1(C(N(CC(CC)NC(C2CN3CCN2CC3)=O)C)=O)ccc2c(c1)ncn2C C(=O)(CCCCC#N)N(CCCOCCN(C(CN1C(C)CCC1)=O)C)C c1(CC)nc(N(C2CCCN2C(=O)Cc2ncccc2C)CCOC)[nH]c(=N)n1 C12(NC(C3C(NC(Cc4cccc(C)c4)=O)CCOC3)=O)CC3CC(CC1C3)C2 C1(NC(N(CC(CCC)C)C)=O)CC(=O)N(C(=O)OC)C1c1ccccc1 C(=O)(N=c1cnn(C2CCOC2)[nH]1)N(CCC#N)CC C(=O)(C(O)CC[S+](C)C)NCC(CC1CN(C(CC(C(C)C)O)=O)C1)(C)C c1(NC(C2CCCC2c2ccccc2)CC)ccc(O)c(C)c1 C1(C(=O)NCC(C(=O)OCC)C)CCN(C(=O)C(CO)C(C)(C)C)O1 Cc1nccc(C(=O)NCC2CCC(NC(c3ccnnc3Cl)=O)C2)n1 N1(C(CCC(C)OC)=O)CC2CCC(C1)C2CNC(c1ccc(N)c(SC)c1)=O C(CCCCC(=O)NCC1CC1CNC(c1cccc(F)c1N)=O)OC c1(C(=O)NC(C)C(C)(C)NC(=O)CC2C=CS(=O)(=O)C2)ccc2nn[nH]c2c1 c1(C(=O)NCC(C2CCCCC2)NC(CC(C(C)C)O)=O)cc(F)cc(Cl)c1N CC(C)CC(C(=O)OCc1ccc(C(C)C(F)(F)F)cc1)C(C)C C1(C(N2CC(NC(=O)CC(=O)N(C)C)CC(C)(C)C2)=O)CC2OC(C)(C)OC2C1 c1(C(c2n(CCCC)nnn2)NCCn2ccc(Br)n2)cnc(N(C)C)cn1 C1(NC(CC2CC(C)N(C(C3CC=CC(O)C3)=O)C2)=O)CCOC2(CCC2)C1 N1(C(COCC)=O)CCC(=C(c2ccco2)C(C)C)C1 Cc1c(C(=O)NCC(C2CCCC2)NC(=O)CCC2NC(=O)NC2=O)ccn1C c1(C(N(CCCNC(C(C)C(F)F)=O)C2CC2)=O)n[nH]c2c1CC(F)(F)CC2 N1(C(Cn2nc(C)oc2=O)=O)CC2(CCN2C(=O)C(c2ccc(Cl)cc2)CO)C1 c1(CC(=O)NC2CCC(NC(c3c(C)ccc(N)c3)=O)C2)ccc([N+](=O)[O-])cc1 N1(C(c2cc(C)oc2)=O)CCCN(C(C2CCN(CCO)C(=O)C2)=O)CC1CO C1(C(=O)NCCN(C(=O)CC2=CCN(C)CC2)C(C)C)CCCN1S(=N)(=O)N(C)C c1(C(=O)NCC(CC=C)NC(=O)CC(C)(CC)CO)cc2ccncc2cc1F C1(NC(C(CO)OC)=O)CN(C(=O)C(c2ccccc2F)F)C2CCCC12 CCC(CNCC1(c2cccc(F)c2F)CCCC1)(CC)CO Cc1ccc(C)c(CC(=O)NCCNC(=O)C(c2cccc(Br)c2)C)c1 C12(C(=O)NCC3C(NC(c4c(CC)occ4C)=O)C3)CCC(CC1)C(C)(C)O2 C1(C)(CNC(C2N(CCC)C(=O)CC2)=O)CCN(C(C2(CC)CC2)=O)CC1 C(=O)(C1=C(CC)OCCS1)NCC(CC)(CC)NC(=O)CC(C)(F)F N1(C(c2cc(C(C)C)on2)=O)CC2CCC(C(N3CCC(F)(C(N)=O)C3)=O)(C2)C1 n1(CC)nc(C)c(C(=O)NC2CC(CC(N3CCCC(C)CC3)=O)C2)c1C C(=O)(CCCCCNC(=O)C(C)(C)C)N1CCC(C(C)O)C1 C12(CNC3(c4nnnn4CCOCCO)CCCC(C)C3)CCC(CC1(F)F)C2 c1(CNC(C2(NC(Cc3ncn(C)c3)=O)CCC2)=O)cc(F)ccc1O CCCC(C(=O)NCCCOCCCNC(c1ccoc1Cl)=O)c1ccccc1 CC1Oc2ccccc2N(CCC(=O)Nc2cn(C)nc2Cl)C1=O C=CCC(CNC(=O)CCn1cccc1)NC(c1ccc(C2CCOC2)s1)=O c1(C(=O)NC(C)CNC(=O)Cn2ncc(Br)n2)cc2c(Cl)cccn2n1 c1(C(N2CCCC(N(C)C(C3CCC(F)(F)CO3)=O)C2)=O)ccn2ccccc12 N1(C(C2(OC)CCSC2)=O)CC2(CCCC(CNC(=O)CCCOC(C)C)O2)C1 N1(C(c2scc(OC)c2)=O)CC(C)(C)CC1CNC(c1cc(C)sc1C)=O c1(C(N2CCN(C(C(CCC)C(C)C)=O)C(C)CC2)=O)cccc2c1C(=O)CC2 N1(C(C(C2CC(NC(C(CCC)C#N)=O)C2)F)=O)CCN(C)C(C)(C)C1 CC1(C)CC(=O)NC1CNC(c1nnnn1C1CC1)CCC1CCCC(=O)N1 CC(C)CC(O)C(C)C(=O)NCCOCCNC(c1ccc2cncnc2c1)=O C1(CCNC(C2CC2F)=O)CC(F)(F)CN1C(c1ccc(F)s1)=O N1(C(CC(C)C)=O)CCN(C(C2CCC(CC(F)(F)F)CC2)=O)CC(C)(C)C1 C(=O)(C#CC1CCOCC1)NC(CNC(C(c1cccc(C(F)(F)F)c1)CC)=O)C c1(C(N2C(C(=O)NC3CCCN(C)CC3)CC3CC32)=O)ncc2ccccn12 C1(CNC(C(C)CF)=O)CCC(NC(=O)CC2(NS(C)(=O)=O)CCCCC2)CC1 c1(-n2cc(C(=O)CCSCCOC3CCC3)nn2)cccc(C(C)(C)OC)c1 N1(C(CCc2cc(C)no2)=O)CCC2CCC(C1)N2C(=O)C=CCF N1(C2(C(=O)NC3C(CNC(=O)CSCC4CCCO4)C3)CC2)CCNC1=O C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1C)N2C(=O)CC(C)n1ccnc1 c1(C(=O)NC2CCN(C(C3C(C)CC3)=O)CC2)ccc(F)cc1O C(C(=O)NCc1cc(OC)ns1)(C(C)O)NC(c1cnc(OC)s1)=O c1(C(=O)NCCC(CC)(C)NC(c2ccc(OC)cc2F)=O)cc(C)ccc1C C(=O)(C1CCCc2nn[nH]c21)N(C1(CNC(=O)CN2CC3CC3C2)CCCC1)C Cc1scc(CNC(=O)COC2CN(C(C3(C#N)CC=CC3)=O)C2)c1C C1(OC)CN(C(=O)C(=Cc2cn[nH]c2)C)CC1C(=O)NC1CCC(=O)NC1 C1(NC(=O)Cc2c(CN(CC)CC)csc2)CC(NC2(C3CCC3)CC2)CCO1 C(=O)(CS(=O)(=O)CC(F)(F)F)NC(CN(C(C(c1c(C)nn(C)c1)O)=O)C)C CC(C)CCCC(C)C(=O)NC(C)CNC(=O)Cc1ccc(F)cn1 C1(CNC(c2nc(C3CC3)cs2)=O)CN(C(c2cnoc2)=O)CCO1 C1(C)(NC(c2c(C)occ2)=O)CCCN(C(=O)CC2CCCOC2)C1 C(CN=c1cccc(S(=O)(=O)NCCn2ccnn2)[nH]1)NC(COC)=O Cc1nc(C(N2CCCC(CN3CCOCC3)C2)C(=O)N(C)C)nn1C CC(CNC(=O)CCC1CCOCC1)CN=c1[nH]cc(C#N)c2ccsc12 C(=O)(CC(O)C(Cl)(Cl)Cl)NCCN1CCCN(C(CC)=O)CC1 N1(C(COCCCC#C)=O)CCCC(CCCCNC(C2CCN(C)C2)=O)C1 CCCCC(CC)CCC(=O)NCCC(C)(C)NC(C1CC(=O)NC(=O)N1)=O N1(C(C(c2ccnn2C)NC(Cc2cn(CC)nn2)=O)=O)CC(CO)CC1CO c1(C(=O)NC2CN(C(C(C3CCCCC3)C)=O)CC2F)cc([N+](=O)[O-])ccc1Cl C(N=c1[nH]c2cc(Cl)ccc2s1)C1(CNC(c2n[nH]c(O)n2)=O)CC12CCC2 C1(C(N(CCNC(Cc2ccn(CC)n2)=O)C2CC2)=O)CC=C(C)CC1 C1(CCNC(CC2(C)CCN2C(c2cc(Cl)c[nH]2)=O)=O)CCCC2CC12 C1(CC(=O)N(C2CCN(C(=O)Cc3cc(F)ccc3O)C2)C)CC(C)(C)CCO1 N1(C(C2N(C(C(C)NC(N)=O)=O)CCCCC2)=O)CCn2cnnc2C1 Cc1cn2ccc(C(=O)NC(C)CCNC(c3cc(C)n(C)c3C)=O)cc2n1 C(=O)(CC1=CCN(C)CC1)NC(CCOC)CNC(=O)C(F)(F)c1ccccc1 c1(C(=O)NC(CNC(C2C(COC)C2)=O)C(C)(C)C)nc2ccc(C)cn2c1N Cc1nccc(C(=O)NCC(C)(C(C)C)NC(c2cccc(OCF)c2)=O)c1C C1(NC(C(C)N(CC(F)(F)F)C)=O)CCCCCN(C(c2cnc(O)n2C)=O)C1 C(C(=O)NCC(C)CNC(c1ncn(C)n1)=O)(C(C)C)NC(=O)OCC C1(C(=O)NCC(C)NC(c2c(C(F)(F)F)cnn2C)=O)CC12CC(C)(C)C2 C=CCC(CC)C(=O)NCC1CN(C)CCN1C(c1cnc(C2CC2)s1)=O C=CC(C)(CC)C(=O)N1CC2CC(NC(=O)C(C)Cc3cccc(F)c3)C2C1 C(=O)(C(CN(C(=O)Cn1ccnc1)C1CC1)C(C)C)N(CC(N)=O)CC C1(CNS(CC(N2C(c3c(C)cccc3)C(O)CC2)=O)(=O)=O)COCC(C)(C)O1 CN1C(=O)CCCC1C(=O)NC1CCN(C(=O)C(=O)NCC(F)F)CC1CO N1(C(c2c(C)n[nH]c2C)=O)C(C)CC2CN(C(c3ccc4ccnn4c3)=O)CC12 C=CCC(CNC(=O)COCC1CCC1)C(=O)N1CCC12CC(O)C2 c1(C(N(CC(=O)NCCCCSc2nc[nH]n2)C2CC2)=O)cscc1F c1(C(=O)NC(CNC(C2(CC)CCC2)=O)C2CC2)cccc(C2CC2)n1 c1(NC(Cc2cccc(NC(Cc3ccc(C)nc3)=O)c2)=O)cnc(Cl)c(C)c1 N1(C(C2C(=C)C2)=O)CCOC2(CCN(C(=O)Cc3cccc(OCC)c3)C2)C1 Cc1cc(C(N2CC(C(C(=O)NCCN3CCOCC3)N(C)C)C2)=O)c(C)nn1 C1(NC(C(CCF)NC(c2cn(CC)nc2C)=O)=O)CCC(=O)N(C)C1=O CC1(C)CN(C(c2cc(C(N)=O)no2)=O)CC1NC(=O)Cn1cnccc1=O c1(C(N2CC3C(NC(CC(c4c(C)noc4C)C)=O)(C3)C2)=O)cc2n(c1)CCC2 N1(C(c2c(CC)nc[nH]2)=O)CC(NC(c2cc3scnc3[nH]2)=O)CC2(CC2)C1 C(=O)(CC(C(F)(F)F)N(C)C)N(CC1(F)CC(C)C(N(CC)CC)C(=O)NC1)C C(C(CC(=O)N1CCC(C)(N(C)C)C1)NC(C1CC(F)(F)C1)=O)OC c1(CC(N2CCC(C(C)NC(c3c(SC)nn(C)c3)=O)C2)=O)cc(Cl)ccc1Cl C=CC(CC)CC(=O)NC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)C1C(CC)C1 Cc1nc(Br)cnc1NC(=O)CC1CCN(Cc2cc(CO)ccc2O)CC1 C1(NC(CCN(C)CC)=O)CN(C(c2cc(Cl)cnn2)=O)C2(CCCOC2)C1 C1(C(=O)OC)CCN(C(=O)CNc2cccc(OC(C)(C)C)n2)C2COCC12 c1(C(=O)NCC(CCNC(C=C(C)C)=O)O)cc(Cl)ccc1OC(F)(F)F c1(SC)cc(C)c(C(=O)NC(C2CCN(C(=O)Cc3cn[nH]c3)C2)C)o1 c1(C(=O)NCC2(CCNC(C(C)SCCCC)=O)CC2)ncc(F)cc1C N1(C(C(F)=C(C)C)=O)CC(F)(F)CC1CCNC(c1ncoc1C1CC1)=O Cc1ccc(NC(c2ccn(C(F)F)n2)c2nnnn2CC(F)F)c(F)c1 C1(O)(CNC(C2(NC(N)=O)CC2)=O)CCCN(C(c2ccon2)=O)C1 Cc1nc(C(=O)NC2CC(F)CN(C(C3CCC(O)CC3)=O)C2)c2n1CCCC2 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(OC)C(NC(c2cc(Cl)n(C)n2)=O)CC1 c1(N(C)C)nc(F)ccc1CNC1CC(CC(N2CCCC2CC#N)=O)C1 c1(NC(C2CCC(C)N2C(c2c(O)ccc(Br)c2O)=O)=O)cc(Cl)c(Br)cc1Cl N1(C(c2ccc(C(F)(F)F)cc2Cl)=O)CCC2(CCN(C(C3CCSC3)=O)C2)C1 C#CC1(NC(C2(CNC(=O)C(O)CCSC)CC3(CC3)C2)=O)CCC(C)CC1 N1(C(c2c(OC)n[nH]c2)=O)CCOCC1C(=O)NCC(C)C(C)(C)C c1(C(=O)NCCN(c2nnc(CO)s2)CC)c(C)oc(C)c1C C1(NC(CCN(C)CC)=O)CC2CC(NC(=O)C(C)Cc3ccccc3F)CC12 c1(C(=O)NCC(C)CNC(=O)CC2CC2)nc(C(F)(F)F)oc1Br c1(C(=O)NCC(C(C)C)NC(=O)CCc2ccc[nH]2)cccc2occ(Br)c12 C1(CC(=O)NCC2CCN(C(CC3CCC(C)C3)=O)C2)NC(=O)NC1=O C1(NC(C2CC(=O)C2)=O)CC(O)CN(NC(C2CC(Cc3ccccc3)C2)=O)C1 N1(C(C(c2c(C)noc2C)C)=O)CC2CC(NC(c3cn[nH]c3)=O)C1C2 Cc1ccccc1C=CC(=O)NC1CCOC1C(=O)Nc1cncnc1O CC1CC(CNC(C2(c3cccc(F)c3)CCCCC2)=O)CN1C(=O)CN(C)C n1(CCC(=O)NCC(CNC(=O)C(O)CSC)OC)ncn(C)c1=O C1(C)(C(=O)NCC(CN(C(=O)CNc2ccccn2)C)O)CC1(F)F C1(CNC(=O)C=C2CC2)COC(CNC(=O)CCc2ccon2)C1 c1(C(N2CC(O)(CNC(C(n3cncn3)OC)=O)C2)=O)nccnc1C(F)(F)F Cc1ncc(C=CC(=O)NC2(CNC(c3cnc[nH]3)=O)CCCC2)c(O)n1 N1(C(=O)N(CC2(C)CCC2)C2CC2)CCCCC1c1cccc(O)c1 CC(C)CS(=O)(=O)NC1CC2(CCO2)C1 C1(CC(N2CCC(C(C)(C)NC(=O)Cc3cnco3)C2)=O)CCCC(F)(F)C1 Cn1cnc(C=CC(=O)NC2CC23CC(NC(C2(C(N)=O)CCC2)=O)C3)c1 Cn1nc(CN2CCC(C)(C)C2)cc1C(C1CCCCO1)=O.C1(=O)CO1 C=C(C)CC(C(=O)NC1CC2CC(NCc3ccc(=O)n(C)c3)C2C1)NC(C)=O N1(c2n(CCC#C)c(C3CC3c3ccccc3Br)nn2)CC2(C1)CC(C)(O)C2 C1(C(N2CCC(C(=O)NC)C2)C(=O)NCC)CCC2COCCC2C1 C1(c2n(C)ncc2)COCCN1.c1(Cc2ncon2)cn(C)nc1Br C(CNc1ccc(N2CCC(C)CC2)c(Cl)c1)(CCS(C)(=O)=O)OC CC1CN(C(c2ccnc(C(C)(F)F)c2)=O)CCC1NC(=O)CCN(C)CCO C1(OC)CC2(C1)CC(C(=O)NC(C)CCNC(=O)CC(CC)OC)C2 C1(F)(CNC(C(c2cccs2)SC)=O)CC(NC(c2cnccn2)=O)C1 C1(C(C)C)CN(C(C2CCCCS2)=O)CCN1C(=O)CC1CCC(C)CC1 c1(-c2cc(C(=O)NC(C)CNC(C3CCCS3)=O)sn2)ccc(Cl)cc1 C1(Nc2cc(OCC)ncn2)CC2(CCN(C(c3cc(Cl)ccc3C)=O)C2)C1 c1(CC(=O)NC23CC2CN(C(=O)C=Cc2cnccn2)C3)ccccc1C(F)(F)F c1(C(C)C)nc(Cl)sc1C(=O)NC(CNC(c1ccncc1F)=O)C1CC1 C=C(Cl)C(C)(C)C(=O)NCC(CC(C)C)NC(c1ccc(OCCOC)nc1)=O C1(O)(c2n(CC)c(N(Cc3ccccc3)CC3CCC3)nn2)CCC(C)(C)CC1 CN1CCCC(C(N2CCCC2C(C)(C)C(=O)NCCC2CCCOC2)=O)C1 C1(NC(=O)CC(F)(F)F)CN(C(=O)C=Cc2cccc(Cl)c2)CC2CCCC12 c1(SCC)ccc(C(N2CC(OC)CC2CNC(C2CCC(C)O2)=O)=O)cn1 c1(CCC)n[nH]cc1C(=O)NCC(CC)NC(=O)CC(C)N(C)C C1(C(=O)NCC(C)(C)NC(=O)C(F)=C2CCC2)CCCN1C=O c1(OC)ncc(C(=O)NCC2CC(OC)CN2C(=O)Cc2cccc(C)c2)cn1 C1(CNC(C(C)OC(C)(C)C)=O)CCCC2CN(C(=O)CC3CC3(F)F)CC12 C1(C)(CC)CN(C(=O)C(C)(O)CN(C)C)CCO1 c1(C(N(CC(CN(C(COCCC(C)C)=O)C)O)C)=O)n[nH]c2ccc(Cl)cc12 C(=O)(C(CC(F)F)NC(C1CC(C)(C)C1)=O)NC1(C)CS(=O)(=O)C1 C1(NC(CC2C(C)C(=O)CC2)=O)CN(C(c2snc(O)c2Cl)=O)CC12CC2 C1(CNC(C(=O)NCC)=O)CC2CC1CN2C(c1cc(C)nn1C(C)(C)C)=O C1(N(C(=O)C=C2CC2)CC)CCCN(C(=O)C(C)OC)C1 C1(C(N2CCC(=C)CC2)=O)CN(C(=O)C(CO)N(C)C)CC(C)(C)C1 N1(C(CC(=C)Br)=O)CC(CNC(=O)COC2CCOC2)C2(CCC2)C1 c1(C(=O)OC)cnccc1N1CC2C(CNC(c3nccnc3C)=O)C2C1 N1(C(=O)CCOCC(F)F)CC2CC1CN2C(c1nccc(Br)c1O)=O N1(C(C2C(NC(c3nc(C)sc3)=O)CC2)=O)CCCC2NC(=O)CC12 c1(C(C)N(C(=O)CCc2cnn(C)c2)CCNC(=O)CC2(O)CC2)ccc(Cl)nc1 N1(C(C(C(C)C)(C)O)=O)CC2C3CCC(C2C1)N(C(c1cccc(F)c1O)=O)C3 C1(CCNC(C2C(C)C2C)=O)CN(C(c2n[nH]cc2Cl)=O)CCS1(=O)=O C(c1ccc(C(N)=O)o1)=CC(=O)N(C1CC(NC(CC(C)F)=O)C1)C C1(CNC(c2cc(=O)n(Cc3ccccc3)[nH]2)=O)CC(F)CN1C(CNC)=O.CO CCC(C)(C)CC(=O)NC(C)C(C)NC(c1ncoc1-c1cnn(C)c1)=O C1(NC(c2ccc(SCC3CC3)cc2)=O)CCCCN(C(=O)CCCC2CC2)C1 N1(C(C(C)N(C(c2ccc(C(C)C)o2)=O)CC)=O)CCCC(C(C)C)CC1 c1(C(N2CC3CN(C(C(C)(C)F)=O)CC(C2)O3)=O)cc2c(nc1O)CCCCC2 N1(C(c2c(C)ncs2)=O)CCOC(CC(=O)NC(C)CC(=O)NC(C)C)C1 C1(NC(CN(CC)CC)=O)CCCN(C(=O)CCCOC(C)(C)C)C1C N1(C(=O)Cn2nnc(C3CC3)n2)CC(NC(C23CC(F)(C2)C3)=O)CC(O)C1 N1(C(CC(=C)C)=O)CCC2(CCN(C(=O)C(C)C(F)F)CC2)C1 C#CC1CCN(C(=O)OCC)C1.c12nc(C)c(s1)C(C)N2C N1(C(c2c(OC)cccc2OC)=O)CC2(C1)SCCC2NC(=O)CSC1CC1 Cc1ccc(O)c(C(N2CCCCC2c2nc[nH]n2)=O)n1 c1(C(=O)NC(C2CCN(C(C(C)=C3CC3)=O)C2)(C)C)ccc(C(C)=O)cn1 Cc1oc2ccccc2c1C(C)N(C)C.C12(S(=O)(=O)Oc3cnn(c3)CCS1)CC2 N1(C(C2CC=C(C)CC2)=O)CCC(C2CC2)(CNC(=O)Cc2ccoc2)C1 c1(N2CCC(NC(c3cc4ccc(Br)cc4s3)=O)C2)ncc2cccc(O)c2n1 C1(C(=O)NC2CC(CNC(=O)C3=CCCOC3)C2)CCn2c(O)nnc2C1 N1(C(C2(C)N(C(c3nc(C)sc3C)=O)CC=C2)=O)CCC2(CC(CO)C2)C1 c1(OC)ccc(-c2cnc(CNC(c3ccc(N(C)C)nc3)=O)nc2)c(C)n1 N1(C(C2C(C)(C(F)F)C2)=O)CC(CNC(c2cnoc2C2CC2)=O)C2(CCC2)C1 O=S(=O)(c1cc(OC(F)F)cc(F)c1)NCC1(O)CCCCCC1 N1(C(c2ccc(C(N)=S)cc2)=O)CCC(C2(O)CCC2)CC1 c1(C(N2CC(c3cn(CCOC)nn3)OCC2)=O)cc(N)cnc1Br CC1CCC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)C(C)CO)C1 c1(C(=O)NC2C(CNC(C3(C)CC3(F)Cl)=O)CCCC2)c(F)cccc1[N+](=O)[O-] C1(CNC(CNC(=O)OCC)=O)C(C)CCCN1C(=O)Cc1sccc1C C1(C(N(C2CCN(C(CC(=C)Br)=O)C2)C)=O)CC2OC(=O)OC2C1 CCCCCC(=O)NCC1C(C)CCN1C(=O)Cc1nocc1C(C)C c1(N2C3CC(=C)CC2CC3)nc(=NCSC2(OCC)CCC2)[nH]c2c(F)cccc12 CC1COC(C)(C)CN1C(Cc1ccccc1)C(=O)NCCC#N Cn1ccc(C(N2CC(NC(c3cn(C4CC4)cn3)=O)CC3(CC3)C2)=O)c(O)c1=O c1(NC(C2(CSC)CN(C(=O)C(O)C(F)(F)F)C2)=O)ccc(F)c(Cl)c1 Cc1[nH][nH]c(=NC(=O)C2CN(C(c3ccc4n[nH]cc4c3)=O)C2)c1Br C1(CNC(c2cccc(SC)c2)=O)C(C)CCCN1C(=O)CCC1CCC1 N1(CC(=O)NC2CC(F)(CNC(C3(CC4CC4)CCC3)=O)C2)CCC(CO)CC1 C1(C(NOCCC(C)C)=O)CN(C(=O)CCc2cccnc2)CCC1(C)C C1(CCOC)(C(=O)NCC2CC2Cl)CCN(C(C2CCCCN2C)=O)CC1 S(=O)(=O)(c1ccc(NC2CC(CF)C2)cc1Br)NC(CC#CC)C C1(NC(C(C(C)O)(F)F)=O)CC2(CCCCN2C(c2cnncc2O)=O)C1 c1(OC)ncccc1CC(N1CCC(NC(c2cccc(C(C)(F)F)n2)=O)C1)=O c1(C(=O)NCCCN(C)C(C2OCCC2c2cnn(C)c2)=O)ccccc1Cl c1(NC(=O)NC(c2cc(OCC)c(OC(F)F)cc2)C)ccc(S(C)=O)cc1 Cc1nccc(C(=O)NC2(C(=O)N(C(C)CN(C)C)C)CCN(C)C2)c1C N1(C(C2N(C(C)=O)CSC2)=O)CCCCC1CCCNC(=O)CC1COCCO1 C1(COC)CN(C(c2cccc(SC)c2)=O)CCN1C(=O)C(C)C(F)F c1(N(C(=O)C(CC)C2CCC(=O)N2)CCC)cccc(N(C)C)c1 c1(CN(c2cccs2)CCOC)ccc(OC)c(-c2cccc(C)c2C)c1 C1(=O)CCO1.C(C(=O)OCC)OCCOCC N1(C(C=C(C)CN2CCOCC2)=O)C2CCC1C(NC(=O)COCCCF)C2 C(=O)(C1=CCCN(C(=O)CSCC=C)C1)NCCC(CC#C)C C(C)(C)(CCCCC(=O)NC1C2CN(C(c3nnc4ccccn34)=O)CC12)OC c1(Cn2c(N3C(C)CC(C4CC4)C3)nnc2-c2ccc[nH]2)occ2c1CCOC2 N1(C(C2CCCC(=O)N2)=O)CC2(CCC2NC(=O)C(=C2CCCCC2)F)C1 N1(C(CC(CC)(F)F)=O)CCOCC12COCCN(C(=O)CCC(C)O)C2 C1(NC(C(CC)C#N)=O)CCN(C(C2CN(CP(C)(C)=O)C2)=O)CCC1(F)F c1(C(N(CCNC(c2nnn(COCC)c2N)=O)C)=O)ccc2c(c1)CN(C)C2 CN1CCCCC1COC(C1CCCN1C(c1cc(Br)cn1C)=O)=O N1(C(CCCC#CC)=O)CCC2(CC1)CC2CNC(C1CC1OCC)=O O=C(N1OC2C=CC1CC2)C1CCN1C(C1(F)CC=CCC1)=O N1(C(=O)CSCCN2CCOC2=O)CCC(CO)C1c1ccccc1 Cc1ncc(Cl)cc1CC(N1CCC(NC(=O)CC2CNC(=O)C2)C(O)C1)=O c1(NC(C(CN(C)C)NC(c2n(CC)c(O)nc2)=O)=O)c(C)cc(C)cc1C c1(CC(=O)NC(C2CN(C(=O)C=Cc3cn[nH]c3)CCO2)C)cc(F)ccc1O c1(C(N2CCCC(c3c(C(=O)OCC)con3)C2)=O)cnc2c(Br)cccc2c1 Cc1cc(C(=O)NCCC2(NC(=O)CCC3CCC(=O)N3)CCC2)c(C)cc1Cl c1(N2CC3C(C)C3C2)ccc(Br)c(S(=O)(=O)N2CCOCC2C2CCCO2)n1 C1(CC(N2CC(NC(C(C)CSCc3ccccc3)=O)C2)=O)CCCS1(=O)=O CC1(C(=O)NCC2(CCNC(c3cncnc3)=O)CC2)CCC(=O)NC1 C1(C(=O)NC2CCCC2NC(=O)CCS(C)=O)(NC(C)=O)CCCCC1 C(=O)(C1=CCCOCC1)NCC12CN(C1)C2.c1(OOC)c[nH]c2nccc-2c1 N12CCCN(CC1)C(=O)c1cc2ncn1.C1(OC)CC(c2ccccc2)CO1 CC1CC(N=c2[nH]c(-c3ccccc3)nc(=NCC3CC3)[nH]2)CN1C1CC1 c1(C(=O)NCC2N(C(C=CC=CC)=O)CC2)ccc(N)cc1Cl Cc1ccc2c(c1CO)CCCN2CC(c1cccc(C#N)c1)O c1(N2CCC(NC(C3CC3C(=O)OC)=O)C23CCC3)nc2ccc(N)cc2s1 c1(C(=O)NCCCNC(c2cc(-c3cccnc3)on2)=O)sccc1F C1(C(=O)NC(CN(CC)CC)C)CC2CC1CC2NC(c1ncnc(C)c1C)=O c1(CC)nccnc1NC(C1(SC)CN(C(=O)CC2CCC3CC23)C1)=O C1(NC(C(CC)(C)OC)=O)CC2CC(NC(c3[nH]ccc3C3CC3)=O)C2C1 N1(C(CC(C)N2CCCC2=O)=O)CCN(C(=O)COCC(F)(F)F)CC12CC2 c1(C(=O)NCC(C)CN(C)C(C2CCS(=O)(=O)C(C)C2)=O)ccc2nn[nH]c2c1 c1(CN(CCNCc2ccnc(-c3ccccn3)c2)CC)cnc(Cl)c(F)c1 N1(C(C(CC(C)C)ONC(=O)C2CC=CC2)=O)CCC2(CCOC2)C1 C1(NC(c2n(CC)ccn2)=O)CCC(N(C)C(c2cocc2C(N)=O)=O)CC1 c1(OCCNC(c2ncc(C(N3CC(NC(C)=O)C3)=O)o2)=O)ccc(F)nc1 N1(C(C=CCC)=O)CC2CC(NC(c3cc(Br)n(C)c3)=O)C(C2)C1 O=C(C#CC1CCCOC1)NCCC1CN(c2ncnc(Cl)c2F)C1 CC1CCCCCC1NC(=O)CCOCCCNC(=O)CC1OC(C)(C)OC1=O C1(CCOC)CN(C(c2cc(O)nc(C)n2)=O)CCN1C(C1CC(C)(F)C1)=O c1(C(C)C)n[nH]c(=NCC2CC(NC(c3ccc(NC(N)=O)cc3)=O)C2)o1 C1(C(=O)NCC=C(C(=O)N(C(CC)C)CCO)C)CC=CCC1C C1(CC(=O)NCC(C)CNC(=O)C=Cc2ccc[nH]2)COC2CC1C2 c1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)cc(C)ccc1N N1(C(C2C(C)C2)=O)CC2CN(C(=O)C(C)(C)C(F)(F)F)CCC12 N1(C(N2CCCC2c2cc[nH]n2)=O)CCOCC1CCc1ccccn1 N1(C(C(CC)C)=O)CCN(C(=O)CCc2nc(C(C)C)no2)C(COC)C1 C(=O)(C1=NOC2(CCC2)C1)N(CCCCNC(=O)Cc1cc(F)ccc1F)C c1(C(=O)O)nn(-c2ccccc2)cc1C(N1CC(C(=O)O)CC1C(F)(F)F)=O Cc1cc(=O)ccn1CC(=O)NCCC1CN(C(=O)CC2(O)CCC2)CCO1 O=C(CCCCCNC(C1(O)CCSC1)=O)NC1CC(CSC)C1 c1(C(=O)NC2CC(CO)N(C(=O)Cc3cc(Cl)ccc3Cl)C2)csc2nnsc12 C1(CC(N2CC(CNC(C3(CC)CC(C)(C)C3)=O)C2)=O)CCCCC1(F)F C1(C(N2CC(C(C)NC(c3c(C(C)C)noc3)=O)C2)=O)CC12CCC(F)(F)CC2 CCCC(C(=O)N(C)CC1CC1(C)C)NC(=O)C(C)OC(C)=O C(C1=CCN(C(=O)C(C2CCCN(C)C2)(C)C)CC1)NC(Cc1c(C)noc1Cl)=O c1(C(=O)NC2(C)CC(NC(C3COCCC3(F)F)=O)C2)ccc(=N)[nH]c1Cl N#Cc1ccc(C(=O)NCC#CCNC(c2cc3c(s2)CCC3)=O)c(F)c1 C(=O)(CCS(C)(=O)=O)NCC(=O)NC1CCC(NC(C(CCC)C)=O)C1 C1(C(=O)NCc2c(C(=O)NOCc3ccccc3)cccn2)CCCC(F)C1 C1(CNC(CC(=C)Br)=O)CCN(C(c2nc(CC3CC3)cs2)=O)CC1C N1(C(C(CO)NC(C2C(C)N(C)CC2)=O)=O)CC(CO)C(C2CC2)C1 N1(C(C(C)SCC)=O)CC2(C)CC1(C(=O)NC(CC)CC(F)(F)F)C2 Cc1oc(CO)cc1C(=O)NC1(CC(=O)NC2CCN(CCCO)C2)CC1 N1(C(C=C(C)Cl)=O)CCCCC(NC(c2cc(Cl)c(Cl)cc2O)=O)CC1 C1(CNC(N2C(C)CC(C(=O)OC)C2)=O)CCCCCC1C1CC1 c1(C(N(C(C)CNC(c2cn(C)nn2)=O)CC)=O)cc(Cl)ccc1C c1(C(N2CC(NCc3ccncc3Br)C3(CC3)C2)=O)ccc2ccccc2c1Br N1(C(C(CCSC)O)=O)C2CCC1C(CNC(c1oc(C)nc1C(F)(F)F)=O)C2 c1(OC)cncc(C(=O)NC2COCC2NC(=O)CSc2c(C)n[nH]c2C)c1C C1(NC(C2CC(C)NC(=O)C2)=O)CN(C(=O)C(C)(C)c2ncco2)CC12CCC2 C1(NC(CCNC(=O)NC)=O)CC2CC(NC(C3CC34CC(C)(C)C4)=O)CC2C1 c1(C(=O)NCC2C3CN(C(C4CC(C)OC4)=O)CC32)c(Cl)nc2ccccn12 CCC(C(=O)NC1CCCC(NC(=O)Cc2ccc(F)c(F)c2)C1)C(C)(C)CC C1(C2CCCN(C(=O)Cn3cnnc3)C2)(NC(c2cnn(C)n2)=O)CC1 Cc1cc(NC(c2nn(C)c(C)c2Cl)=O)ccc1NC(c1[nH]nnc1C)=O C1(CNC(c2c(SC)snn2)=O)CC12CCN(C(=O)C(=Cc1cccs1)C)CC2 N1(C(c2ccc(OC)c(Cl)n2)=O)CCC2(C1)CN(C(c1ocnc1C)=O)C2 C1(CCC)(CNC(C2(C(C)(F)F)CCC2)=O)CCCN1C(=O)C(CCOC)OC n1(CC(=O)N(CCCN(C(CC(COC)(C)O)=O)C)C)ccc2ccc(F)cc12 C1(NC(C(C)NC(=O)C(N2CCOCC2)C)=O)C2CCCC1COC2 C(CC(C)CC(C)(C)C)NC(c1c(CNC(c2ccc(C)c(C)c2)=O)n[nH]c1)=O c1(CCCC)nc(C)c(CC(N2CCC2CNC(=O)C(C)=C(C)C)=O)s1 c1(C(=O)NC2CN(C(c3n(C)ncc3)=O)CC2F)nccn2ccnc12 N1(C(C2CC(SC)C2)=O)CCCC2(C1)CN(Cc1ccsc1)CCO2 C=C(C)C(C)(C)C(=O)NC1C2CC(NC(C3CCC(F)C3)=O)CC12 c1(CC)cc(C(N2CCC(C)C2CNC(c2ncoc2C)=O)=O)c(C)nn1 CCC(C(=O)NC12CCCC1N(C(c1ccc3nncn3c1)=O)CC2)C(C)(F)F c1(C(=O)NCCCCNC(c2cnn(C)c2N)=O)cc(Br)cnc1O N1(C(C(SC)SC)=O)Cc2occ(C(N3CCC(C(C)(C)C)C3)=O)c2C1 c1(C(=O)NC(CN(C(CNC(=O)NC)=O)CC)C)cncc2ccccc12 CC(C)CC(C)C(=O)N(CC(C)(C)C(=O)N(C(C)C(C)C)C1CC1)C N1(C(C#CC)=O)CCN(C(=O)C(c2cncc(C)n2)N2CCOCC2)C(CC)C1 c1(CNC(C2(CNC(=O)CCn3ccc(C)n3)CC(=C)C2)=O)c(C)cnn1C c1(OC)cc(C(=O)NCC2CC2NC(C23CC2COC3(C)C)=O)cc(C)n1 c1(N(CC(C)NC(C2CS(=O)(=O)CC(=O)N2)=O)C)ncc([N+](=O)[O-])cc1Cl C1(C(=O)NC2CC(CC3CC3)C2)CCCN(CC2CC2)C1.c12nnnn1C2 c1(C(=O)NCc2ccc(C(=O)N(CCCl)C3CC3)cc2)cc([N+](=O)[O-])c(O)cc1F Cc1cc(F)cc(NC(C2CC(CNC(=O)CC3CC4(CCC4)C3)CO2)=O)c1O C1(F)(C(=O)NCC=CC(=O)NC(C2CCCO2)CO)CCCCC1 CC(F)(F)CCC(=O)NCC1CCCC1NC(=O)C(O)CC1CCCC1 C(CCC(C)C(=O)NCC=CCC(N1CC(=O)NCC1C)=O)OC c1(C(=O)NC(CCCC)CNC(C2CCC(C)(C)C2)=O)ccc(C2CC2)c(F)c1 CCC(CC)C(C(=O)NC1CC(O)(CNC(=O)CC2C(C)(C)C2(C)C)C1)OC CC1=C(C(=O)NC2CCN(C(=O)C=CC3CCCO3)C2(C)C)CCC1 c1(C(C)C(=O)NC(C2CCN(C(C3CN(C)C3)=O)CC2)C)noc2ccccc12 Cc1cn(CC(=O)NC2CC2CNC(c2nnsc2C2CC2)=O)c2ccccc12 C1(NC(CCCOCCC)=O)CCCN(C(c2ccc(C)c(C)c2)=O)C1C c1(CC)oc(C)cc1C(=O)NC1CCC(CNC(=O)C(CCO)N(C)C)C1 CC1SCCN(C(=O)CC2(NC(c3cc(C4CC4)nn3C)=O)CCC2)C1C C1(NC(C(CC)C)=O)CC1C1CCN(C(c2cc(NC(C)=O)ccc2F)=O)CC1 C(=O)(C(C)(C)CSC)NCC(CC=C)NC(C1C(CCC)C1)=O Cc1nccc(C(N2CCN(C(=O)C(O)CC3CCCC3)C3CC23)=O)c1O O=C(CCCCCCCO)NCCc1nc(-c2cc3cc(Cl)ccc3o2)no1 C1(C)(CNC(c2cc(SC)oc2)=O)CCN(C(=O)CCC2CCCCO2)C1 C(=O)(C(C)CC(C)CC)N(c1cccc(C(NOCCOCC)=O)c1)CC C(CC(C)C)(C(=O)NCc1ncccc1C(=O)N(C)CC1(O)CCC1)OC C=CCC(CC(C)C)C(=O)N(CC)CC1CCCN(C(c2cnncc2C)=O)C1 c1(CN2CCC(O)(C(=O)Nc3cccc(OC)c3Br)C2)ccc2cc[nH]c2c1 C(C(=O)Nc1cccc(Cl)c1C)(C(C)C(C)(C)C)N1CCC(CC(C)O)CC1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CCCC1CF c1(NC(C)=O)ccc(CNC(C2(c3ccc(C)cc3Br)CC2)=O)cc1O C(=O)(C1=C(Cl)CCC1)N1C(C(N2CCCC(N3CCC3)C2)=O)(COC)C=CC1 C1(CNC(=O)C=Cc2nccs2)CN(C(c2ccn(CCF)n2)=O)CCCO1 c1(C(N2CCN(C(C(CC(C)C)F)=O)CC2)=O)ccc2c(c1)N(C)CCO2 CC(C)CC(C)CN1CCC(NC(=O)C(C(C)C)NC(=O)Cn2cccn2)CC1 N1(C(C(CCC)=CCC)=O)CCN(C(=O)CC(O)CC(C)C)CC(O)C1 c1(CC(=O)Nc2nc(C(=O)OCC)c(C(F)(F)F)s2)ccc2ccc(O)nc2c1 Cc1cccc(Cl)c1C(=O)NCCOCCN(C)C(c1nscc1N)=O Cc1[nH]nc(C(=O)NCc2csc(CNC(C3CCCC(=O)O3)=O)n2)c1C N1(C(C2(CC#C)CCCO2)=O)CCCC(N(C(=O)C=CC=C(Cl)Cl)CCO)C1 c1(C(N2CC3C(CNC(c4cccc(SC)c4)=O)(C3)C2)=O)cnn2c1N(C)CC2 C(CN=c1[nH]nc(-c2ccon2)s1)NC(C(N1CC(C)OC(C)C1)(C)C)=O C1(C(=O)OC)CN(C(=O)CNC(=O)CSCC#N)CC1C N1(C(c2n(CC=C)ccc2)=O)CCCN(C(c2cc(OC)nc(F)c2)=O)CC1C C1(CNC(C=C(C)C2CCC2)=O)CCN(C(=O)CC2CCOC2)CCC1(F)F C1(C(=O)NCCOCCN(C)C(c2nsnc2O)=O)CCC(C)(C)C1 CC1c2c[nH]nc2CCC1C(N1CC(CNC(c2ccc(C#N)nc2O)=O)C1)=O N1(C(CSC(C)C)=O)CC2(CC2)CC1CC(=O)NC1CCOC1C Cc1noc(C(=O)NCCCCCNC(=O)C(F)(F)c2csc(C)c2)n1 C(=O)(C#CC1(CC)COC1)NC(C1(C(=O)NC(CCC)C2CCC2)CC1)C C=CCC(CNC(C1CC(C)N(C)C1)=O)C(=O)N1CCC(O)(C(C)C#N)C1 C1(C(=O)NC2CC(O)(c3ccccc3)C2)CCCC2(CC2)C1 C1(C(N2ON=C(C(C)NC(CSCCCC)=O)C2)=O)CCC(N=[N+]=[N-])C1 C1(NC(c2ccn(COC)n2)=O)CN(C(c2ccc[nH]2)=O)CC1n1ccnn1 C(C(C)(O)CO)N(C(CC)CNC(C(=O)O)=O)C.C(C)(C)(C)O CC1CCN(C(=O)N(CCS(C)(=N)=O)C(C)C)C1c1cn(-c2ccc(C(=O)O)o2)nn1 c1(CC(=O)NCC(=O)NCC(COC)C)ccn(C)c1 C1(F)(CNC(C2CCCO2)=O)CCN(C(c2cccc(-c3ccoc3)c2)=O)C1 C1(CN(C(=O)CCS(C)=O)C)CCCCN1C(c1ccc(C(F)(F)F)cc1)=O C1(CO)CCN(C(C2(CNC(=O)CN3CCCC3C(F)(F)F)CCOC2)=O)CC1 CC1=NNC(=O)C1CN(C)C.N12CCOC(CO)(C1)Cc1cccc(c1)C2=O Cc1cc(Cl)c(C(N2CCS(=O)(=O)C(CCNC(=O)CC=CC(C)C)C2)=O)cc1C CN1CCOC(C(=O)NCCCOCCCNC(c2cnn(C)c(=O)c2)=O)C1=O C(C(=O)N1C(CO)CC1CO)(C(C)(C)C)NC(c1c(CC)noc1)=O c1(C(N2CC3(CN(C(CC(C)OC)=O)C3)C2)=O)cc(Br)cc2c1CCN2 CC(C)CCCCCC(=O)N1CC2CCC2(CNC(c2ncc(Cl)cc2F)=O)C1 N1(C(CC(C)SC)=O)CC(F)CC1CC(=O)NCC1CCCCCC1 c1(C(N2CCC(CNC(C3(C)CC(=C)C3)=O)C2)C)ccccc1Br C1(NC(c2ccc(C(C)C)nc2)=O)CCC2(C1)CN(C(C1(C)CC1C)=O)C2 c1(CN(CC)Cc2coc(COCC)n2)cccc(C(F)(F)F)c1F c1(C(N2CC=C(CN(C)C)CC2)C(=O)NC(C(=O)OCC)C)ccnc(F)c1F C=CCC(F)(F)C(=O)N1CC(C(C)(C)O)(COC)C1.C12(CCC1)C(=O)N2 C(=O)(C(C)(F)C(C)(C)F)N1CCN(CCCNC(C(C)c2cccs2)=O)CC1 N1(C(c2scc(C)c2)=O)CC2CCOC2(CNC(=O)C(C)(C)c2cscn2)C1 S(=O)(=O)(c1ccc(NC(CF)CF)c(Cl)c1)NCCc1cc(C)no1 CCC(CC(=O)NC1(C)CCN(C(=O)COc2cc(F)cc(F)c2)CC1)C(F)F CC1CN(C(C2(C)CC2(F)F)=O)CCCN1C(=O)Cc1csnn1 C(CCCOC(N(CCOCCOC(C)(C)C)C)=O)NC(=O)O.C=CC C1(N(C(c2c(C)cno2)=O)C)CC2CCC(C1)N2C(=O)CCS(C)=O Cc1[nH]c2ccc(C(N3CC(NC(=O)C4CC4)C4CC34)=O)cc2c1C C1(NC(COCC)=O)CCCC12CN(C(=O)CCn1ccnc1)C2 C1(NC(c2cn(C)nn2)=O)CC2CC(C1)N(C(c1ccccn1)=O)C2 C(=O)(C1=Cc2ccccc2C1)N1C(C(=O)Nc2cnn3c2CCC3)CC=CC1 c1(OC)ccc(OCCC(C)(C)CC(=O)N(CC(c2nn[nH]n2)C)C)cc1 C(=O)(CCCCC1CC1)N1CC(CC)(NC(C2(CCOC)CCCC2)=O)C1 N1(C(C2(NC(C3CC4CCC3O4)=O)CCCC2)=O)CC2CC(O)CC1C2 c1(C(N2CC3(C(NC(CC(C(C)C)O)=O)CCC3)C2)=O)c[nH]c(=O)c2ccnn12 c1(C(=O)NC2(C)CCCN(C(C(C(=O)OCC)CC)=O)C2)cn(C)c(=O)nc1O Nc1ccc(F)c(C(N2CCN(C(=O)CN3CCS(=O)(=O)CC3)C3CC23)=O)c1 C(=O)(CCCN(C(=O)C(n1ccnc1C)C)C)NCC(=CCCC)C C1(C)(CNC(CCCCC=C)=O)CN(C(C2CSCCS2)=O)C(C)(C)C1 c1(OCOC)cc(-c2cnn(C)c2C(F)F)cc(OC)c1OC Cc1cc(C(=O)NCCCN(C(=O)CCc2csc(Br)c2)C)nc(O)c1 c1(OC)cc(OC)nc(C(=O)NCC2(C)CCN(C(C3NC(=O)CC3C)=O)C2)n1 Cc1ccc(Cl)c(OC(C)C(N2CCC(CNC(c3cc(C#N)cs3)=O)C2)=O)c1 c1(C(=O)NCCC2(O)CCCN(C(=O)CC(F)(F)F)C2)cnnc2ccccc12 c1(C(=O)NCC2N(C(c3c(C)nc(Br)o3)=O)CC2)ccc2c(c1)C=CCC2 c1(C(=O)NCC2CCN(C(c3scnc3C3CC3)=O)C2)cc(Cl)cc(Cl)c1O c1(CC)ncc(Cl)c(C(=O)NCC2CCCN2C(=O)C2=CC(C)CC2)n1 N1(C(=O)C(F)F)CCOC2(CCCN(c3ncc4c(Br)cccc4n3)C2)C1 c1(C(=O)NC(C(=O)NC2CCC(=O)NC2=O)CO)ccn2ccnc2c1 C1(CNC(C=CCCC(C)C)=O)CN(C(C2(F)CCC2)=O)CCC1C(F)(F)F CC1(C)CC(Nc2cc(F)ncn2)CN(C(=O)CC2CC(=O)NC2=O)C1 C(=O)(C(CC)CCc1ccccc1)NCCC1(NC(CS(=O)(=O)NC)=O)CCC1 N1(C(c2c(CC)ccs2)=O)CC(C(=O)NOCc2ccc(F)cc2)C(C)C1 CC1(C)CC(C(N2CCC(C(=O)NCC3CCCC(=O)N3)CC2)=O)CCO1 N1(C(C(C)SCC)=O)CC(C(N2CCCC(F)(F)C2)=O)C2(CC2)C1 C(CC(=O)Nc1cncc(C)c1)(CC(C)C)NC(C12CCC(OC)C1C2)=O C(c1cccc2ccccc12)=CC(N1CCCCC(NC(=O)C=CC2CC2)C1)=O N1(CC(=O)N(C(c2cn(C3C(OC)CCC3)nn2)(C)C)C)CCNC(=O)C1 CC(C)C1=NOC(C)(C(N2CC3CCC2C3NC(c2cnn[nH]2)=O)=O)C1 O=C1CCC(C(=O)NCC(C(F)(F)F)N2CCN(C(=O)C#CC3CC3)CC2)CN1 N1(C(CCCC(=O)N(C)C)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 c1(CNC2CCCC(C(=O)NCc3cn[nH]c3)C2)cc(Cl)cnc1F O=C1NC2(C(=O)NC3CC(NC(C4(n5ccnn5)CC4)=O)C3)CC3CC1C2C3 C(=O)(C1(C)CCOc2ccccc21)N(C)CCNC(C1CC2C=CC1O2)=O c1(CC)nn(C)c(CC)c1C(=O)NCC(C)(O)CNC(=O)CC1=CCCC1 C(=O)(CCCCN1CCCC1)N(C1CCN(C(C2(F)CCCCC2)=O)C1)CC#C CCC(CC(=O)N1CCC(C(=O)NCC(C)(C)CSC)C(C)(C)C1)C(F)F C123CC(C)(CN1C(=O)N2)C3.CC(C)(C)CN.CNC c1(C2C(=O)N2)ccnc(Cl)c1Cl.C1(C(C#N)N(CCCSC)C)CCC(C)CC1 Cc1ccc2c(CN3CCCC3CCC(=O)Nc3ccc(I)nc3)c[nH]c2c1 C(=O)(C(COC)CC(C)C)NCCCC(=O)N(C(=O)CC(C)O)C.CN N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(c2ccsc2Cl)=O)C(C)(C)C1 C1(OC)CCn2cc(C(=O)NCC3C(C)CCN3C(=O)CN3CC=CC3)nc2C1 C(CC(C(=O)NCC1CCN(C(=O)C(C)N(C)C)C1)NC(C)=O)SC N1(C(C(CSC)C)=O)CC(N(C)C(c2cncc(C#N)c2)=O)C2(CC2)C1 c1(C(N(C(CN(C(C(CC(C)C)O)=O)C)C)C)=O)cc2ccsc2n1C Cc1cc(C(N2CCC(CNC(c3csc(Br)c3Cl)=O)C2)=O)nn1C N1(C(c2c(COC)cccc2)=O)CC2(C1)CN(C(C1CC(C(C)=O)C1(C)C)=O)C2 CC(CCO)CCN=c1nc(N(C)Cc2ccno2)c2cc(Cl)ccc2[nH]1 C(=O)(C(O)C(C)(C)SCC)NCCN(C(C(C)(C)NC(=O)NCCC)=O)CC CC1CCCN(C(N2CCCC(Cc3csc(Nc4ccnnc4O)n3)C2)=O)C1 Cc1cc(F)c(C(=O)NC2CCN(C(c3cccc(F)c3Br)=O)CC2O)cc1F c1(NC(=O)OCC)cc(-c2cccc(NC(=O)CCc3cnn[nH]3)c2)ccc1Cl C1(C(C)C)CCC(C(=O)NC2CCCC2NC(C2(c3ccno3)CCC2)=O)CC1 N1(C(CCCC(=C)C)=O)CCC2(C1)CN(C(c1cnsc1C)=O)CC(C)O2 C(=O)(C(CCCCO)NC(=O)CC1CC=CCN1C)NCC1CC(COC)C1 c1(CC)ccc(C(N2CCC(CCNC(c3cc(CO)[nH]n3)=O)C2)=O)c(OC)c1 c1(C(=O)NC2CN(Cc3c(O)cccc3Br)CC2O)c(F)ccc(O)c1F c1(CC(=O)NCC(CC)NC(=O)Cc2cc(C3(C)CC3)on2)cnn(C(C)C)c1 C(CC(=O)N1CCN(C)C2(CC2)C1)(C(C)(C)C)NC(C(C)=C1CC1)=O N1(C(c2nc(C)c(Br)cc2)=O)C2CCCC1CC(n1ccnn1)C2 c1(NC)ccccc1C(=O)NCCC(O)CNC(=O)C=CC1CC1 N1(C(CC2ON=C(C)C2)=O)C(C(=O)NC2(CO)CC(O)C2)CCC1C1CC1 C#CCCCCCC(=O)NCC1C(OC)C(OC)CN1C(c1nncs1)=O c1(CC(=O)NCCCn2cc(-c3c(OC)nccc3)nn2)cnc(O)nc1O C1(NC(c2scc(C)c2)=O)C2CCN(C(=O)CCn3cnnn3)CCC12 c1(C(=O)NC(CC)(CC)CCNC(C2CC2Cl)=O)ccc2ccccc2c1 C1(NCc2c(OCCOC)ccc(Cl)c2)CCC12CCCCC2 c1(C(=O)NCCNC(C23CCCCC2C3Br)=O)sc([N+](=O)[O-])cc1Cl C(N=c1[nH]c2cc(Cl)ccc2s1)CC1(CCNC(C2CC(C)(C)OC2)=O)CC1 c1(C(N2CC(NC(c3cc(C)sc3C)=O)C2)=O)ccnc2ccc(F)nc12 C12(C(=O)OC)C3C4C1C1C2C3C41NC(=O)N(C)CC1CCCCN1 C(=O)(C(Cc1cn(-c2ccncc2)nn1)NC(C1CCN1S(C)(=O)=O)=O)OC C1(C(N2CCCC(CCC)(NC(c3csnn3)=O)C2)=O)Cc2cc(F)ccc2O1 c1(C(N(CC(CC)NC(=O)CC2CCC(=O)O2)C)=O)cc([N+](=O)[O-])ccc1C NS(=O)(=O)c1ccc(S(=O)(=O)NC2CCc3ccccc32)cc1 N#Cc1ccc(Br)c(F)c1NC(C1CC2CC2N1C(C1CCN(CCO)CC1)=O)=O C1(CC)(NC(=O)CCn2c(C)csc2=O)CCCN(C(C2(C#N)CC=CC2)=O)C1 CCCCC(C)C(C(=O)NCCO)N1CCc2cc(C(C)(C)C)ccc21 CCC(c1ccc(C)cc1)=CC(=O)NCCCN(C)C(C1CCC12CCCO2)=O C1(CCNC(CN(CC)CC)=O)CCCN(C(c2c(C)oc(C)c2C)=O)CC1 c1(OCC)ccc(CN2CCC(CC(=O)NCc3c(F)cccc3Br)C2)cc1Br N1(c2c(C#N)cnc(N3C(C)(C(N4CCCC4)=O)CC3)n2)CCc2sc(Br)cc2C1 Cc1ccc(C(=O)NCC(=O)NCCC(C)NC(=O)CC(C)N2CCCC2=O)s1 C12(NC(CONC(=O)C(CO)OC(F)(F)F)=O)CCC(C1)N(C(=O)C(F)(F)F)C2 N1(C(C2(OCC)CCC2)=O)CCC2(CC1)CCN(C(=O)C(C#N)CC)C2 C1(NC(c2cccs2)=O)CC2CC1N(C(c1cc(Br)c[nH]1)=O)C2 N1(C(CC=CCC)=O)CCC(OCC(=O)OCC)C1 Cc1cc(C)c(C(N2CCC(N(C)C(C3CC(C(F)F)C3)=O)C2)=O)cc1C CCC(CC)C(F)C(=O)N1CC(C)CCC1CNC(c1cc2n(n1)CCCN2)=O N1(CC(=O)NC(Cn2cc(-c3cnc(C(C)C)o3)nn2)C)CCOCC1=O C1(C(=O)NC(C(C)C)(C)CO)CN(C(C2CCC(C(N)=O)C2)=O)CC1(F)F C1(C(=O)Nc2nc(C)c(C)s2)C2CCC(C2)C1NC(c1cnnc(Cl)c1)=O CCCC(C(=O)N(CC(C)CNC(=O)CCc1cc(Cl)no1)C)C1CCC1 c1(SCC(=O)NCCC(C)(C)NC(CCC=C=C)=O)cc(=O)n2ccsc2n1 C1(CC(=O)N(C)CCC2CCCC2)CC(F)CN1C(c1ccc[nH]1)=O C(C)(C(=O)NCCC1(O)CN(C(=O)CCCSC)C1)(C1(C)CC1)OC C(=O)(C(O)CC(F)(F)F)N(CC(C)(C)NC(c1ccc(N2CCOCC2)nc1)=O)C N1(C(=O)Nc2cc(C(F)(F)F)cc(Cl)c2)CCN(C)CC1Cc1ccc(C)cc1 c1(C(C(=O)NC(CNC(C2CC(OCC)C2)=O)C)(F)F)ccc(Cl)cc1 Cc1cccc(O)c1C(N1CC2CN(C(c3ccc(I)c(F)c3)=O)C2C1)=O CCCC(C)(C)C(=O)NCC(O)CCNC(C1CC(C(F)(F)F)(OC)C1)=O c1(C(=O)NC(C)(C)CCNC(C2CC23CC3(F)F)=O)nccc2cccnc12 C(=O)(CC(C)C(=O)NC(C)(C(=O)NC1CC(C)OC1=O)C1CCC1)OC(C)=O N1(C(C(C)(C)NC(=O)OC)=O)C2CCC1C(F)C(NC(=O)CC(F)(F)C(F)F)C2 c1(CN(C(c2cc(C(C)C)on2)C(=O)NC2COC2)CC)ccccc1F N1(C(C(n2ncc(C)c2)C)=O)CCC(O)C(NC(c2ccon2)=O)C1 CS(=O)(=O)c1ccnc(NC2CN(C(=O)Cc3ccc(Br)cc3Cl)CC2C#N)n1 Cn1cc(C(=O)C(N2CCC(NC(=O)CC(O)c3ccccc3)C2)=O)cn1 c1(NCC2(C)CCCN(C(C(C=C)(C)CC)=O)C2)cc(C#N)nc(C)n1 C1(CC(=O)NC(CC)CN(C(=O)CCc2nc(C)cs2)CCOC)OCCC1(C)C C1(C)(C(=O)Nc2cc(OCC)ncn2)CCCN(C(=O)C(O)C(C)C)C1 CC(C)CCCC(=O)N1CCCCC1C1(NC(=O)COCCF)CC1 C12CCC(CC1)N2.N1(CC)CCC(CCC2CCCNC2)C1 C1(C(=O)NC(C23CCC(CC2)C3)CNC(C(=O)NCCOC)=O)OCCC1(C)C c1(C(N2CC(C)(C(=O)NC(CCC)c3ccco3)C2)=O)[nH]cc(C)c1C Cc1cc(C=CC(=O)NCC2CCN2C(=O)C(c2cnn(C)c2)C)ccc1F c1(C(N2CC(NC(Cc3n(C)ncc3Br)=O)C2)=O)cc2ccccc2cn1 NS(=O)(=O)CCCC(=O)N1CC(O)C(O)C1CNC(C1CC2CC2C1)=O c1(CN(C)C(C2CC2c2cc(Br)cc(Br)c2)=O)noc2c1CCCCC2 C1(NCCNC(C2C(CC)C2)=O)(C)CCOCC1.c1(N)nc(C)cs1.C1(=O)C(C)N1 c1(C(=O)NC2CC(CNC(C3(CC=C)CCCC3)=O)C2)ccc(S(N)(=O)=O)nc1 N1(C(CNC(=O)NC)=O)CCC2(CC1)CC2(CO)CNC(c1ncccc1C)=O C1(C(=O)NCCC(C)NC(c2ccc(C(C)C)o2)=O)COC(C)(C)O1 C#CCCCCCCCNC(c1ccc(C)nc1O)=O.C1=CC(=O)N2CC1C2 c1(C(=O)NC2(C(=O)NC3CCN(C(=O)NC)C3)CCSC2)cnc(N)cn1 C1(c2n(CCCSCC)nnn2)(NC(C2CCC2)C)CCCC(OC)C1.OC C1(C(=O)NCC2(C#N)CCC2)(COC)CN(C(c2ccc(C)o2)=O)C1 CCC(C)(C)CCCC(=O)NC(C)(C)CNC(c1cc([N+](=O)[O-])ccc1OC)=O N1(C(C2(OCC)CC2)=O)CCC2(COCC(C(=O)NC3(NC(N)=O)CCC3)O2)C1 c1(OCC)nc(C)ccc1C(=O)NC1CCC1NC(=O)C=Cc1cscn1 Cc1ccc2scc(C(N3CCOCC3CNC(C3CC(F)C3)=O)=O)c2c1 c1(C2(CN(C(C(N3CCC(CC)C3)=O)=O)CCCO)CC2)ccc(Cl)c(Cl)c1 Cc1cc(F)cc(C)c1C(=O)NCC#CCNC(C1(C(C)C)CCC1)=O C1(NC(C2C(c3cc(C)sc3)C2)=O)CC2CCC(C1)N2C(=O)C(N1CCSCC1)C C#CC1CN(C(=O)CC2C(=O)N(C)N=C2C)CCN1C(=O)COc1cc(C)on1 CC1CCCC=C1C(=O)NCCCCCNC(=O)Cn1ccc([N+](=O)[O-])n1 Cc1ccc(C#N)cc1S(=O)(=O)N1CCC2C(CCN2Cc2cc(C)nn2C)C1 C12(C(N3CC4C(NC(C(C(CC)CC)C)=O)C4C3)=O)CC3CC(C1)CC(F)(C3)C2 c1(COC)nnc2ccc(=NCC3CCC(C(F)(F)F)O3)[nH]n12 C1(CNC(C2OCCN(C(C(C#C)(C)C)=O)C2)=O)CCC2(CCC2)O1 C#CC1(F)CCN(C(=O)C(c2ccoc2)NC(=O)C(C)=C(C)CC)CC1 CCCCC(C)(F)C(=O)NC(CC(=O)N(C)CCc1ccccc1)C(F)(F)F C1(C(N2C(C3(NC(C(C4CCC(=O)N4)C)=O)CC3)CCCC2)=O)CN2CCN1CC2 S(=O)(=O)(c1ccc2[nH]c(=NCC(CO)OC)sc2c1)N(CCCC(=O)NC)C N1(C(c2ccc(CC)nc2)=O)CCOC(C(=O)NCC(c2ccccn2)O)CC1 C1(C(N2C(C(C)C)CN(C(=O)CCSC(F)(F)F)CC2)=O)CCc2ccnn2C1 c1(C(=O)NC2C(NC(CC3(OC)CCC3)=O)COC2)ccc(C2CC2)c(F)c1 CCC(CCC(=O)N1CCC(NC(=O)CSc2ccc(Cl)cc2O)C1(C)C)OC CCC(C)C(C(=O)NC(c1ncc(C)cn1)C)N(C(=O)C=C(C)C(C)C)C C#CC1(NC(C2CN(C(c3c[nH]nc3OC)=O)C(C)(C)C2)=O)CCC(C)(C)C1 c1(COC)ccc(O)cn1.C12C=CCN1C(=O)CONC2=O C1(NC(Cc2ncc(C)s2)=O)CC2CC1N(C(c1cc(Cl)cnn1)=O)C2 c1(CC)noc(CN(C(C2CCN(C3CNC3)C2)=O)C(C)C)n1 C1(C(N2CC(SC)C2)=O)COCCN(C(=O)CC(N)CO)C1 n1(C(C(=O)NCC2(F)CC(NC(C3(C#C)CC3)=O)C2)C)nc(C)c([N+](=O)[O-])c1C N1(CCC(N2CCN(c3ccc(Cl)cc3)CC2)=O)CCC(F)C(O)C1 C1(NC(c2ccc(CN=[N+]=[N-])s2)=O)C2CN(C(c3cccs3)=O)CC12 Cc1ncc(C(=O)N(CCCNC(=O)Cc2ccc(C(F)(F)F)nc2)CCO)n1C c1(NC(c2c(Cl)n[nH]c2C)c2n(CC)nnn2)ccc2c(c1)CN(C)C2 CC(C)CC(C)(C)C(=O)N1CC(O)CC1Cn1cc(C2(C(=O)OC)CCC2)nn1.N(C)C c1(NC2C(CC)CN(C(C3CCCCS3(=O)=O)=O)CC2)ncccc1[N+](=O)[O-] c1(C(=O)NCC2(CCNC(C34CCC(C3)C4)=O)CC2)coc2c1COC2 c1(C(=O)NCC(C)NC(C(c2cccc(C)c2F)O)=O)cc2n(c1)CCOC2 c1(SC)cc(C(=O)N(C(C)CNC(=O)C=Cc2ccc(C)s2)C)cc(Cl)c1 n1(CCC(=O)NCC2(OC)CN(C(c3cc(C)c(C)o3)=O)C2)cc[nH]c(=O)c1=O c1(OC)cc(CO)ccc1C(=O)NC1CCN(C(=O)Cc2cccnc2)C(C)C1 N1(Cc2ccc(C)cc2)C2CCCC1CC(NC(c1cc(O)ccc1Br)=O)C2 C(=O)(CCCCCC(C)O)NCCCN(C(C(CC)c1cccnc1)=O)CC c1(NC(C(=O)NCc2n(CCC)ccn2)=O)ncc(C)cc1F C(=O)(CC(C)C(C)(C)C)NC1C(CC(=O)N(CC(C)OC)C)C(O)C1 N1(C(c2c(C)c[nH]n2)=O)CCC2(CC1)CN(C(C1C3CCC(=O)C13)=O)C2 c1(CSC)cc(C(N2CC3(CCC3NC(=O)C(F)C(C)(C)O)C2)=O)ccc1F N1(C(c2c(C)nn3c2NCCC3)=O)CCc2cc(Br)cc(F)c21 c1(NC(C2CN(c3ncnc4cc[nH]c34)CCS2)=O)cc2[nH]ccc2cc1Cl CCCC(C(=O)N1CCCC1C1(O)CN(C(c2ncn(C)c2C)=O)C1)OCC N1(C(CC(=O)NC)=O)C(CNC(c2c(F)cc(C)cc2F)=O)CC2COCC12 Cc1cnc(C(N2CC(CNC(=O)CCn3cc(C)cn3)C2)=O)c(F)c1 N1(CC(N2CCN(C(C3CCN(C)CC3)=O)CC2)=O)CC(=O)Nc2ccccc21 N1(C(C=COCC)=O)Cc2occ(C(N3CCC(O)C(C)(CO)C3)=O)c2C1 C(=O)(C(C)(C)C(C)NC(C1CC1(F)Cl)=O)NCCC(C)F C=CCC(CNC(=O)C1CC1c1ccccc1)NC(=O)C(C)=C(C)CC O=C(CS(=O)(=O)CCO)NCC1CCCCN1C(C1CC(OC(F)(F)F)C1)=O N1(C(C(N2CCCCC2)C)=O)CC(C2CC2C(N2CC(S(C)(=N)=O)C2)=O)C1 c1(C(N)=O)ccccc1C(=O)NCC1CC1CC(N1CC(F)CC1CO)=O N1(C(c2c(C)snn2)=O)CCCC(CCNC(=O)C(N2CCN(C)CC2)C)C1 c1(C(=O)NC2(C)CCN(C(c3c(C)cnn3C)=O)CC2)cnc2c(c1)NCC2 C1(c2n(C(C)(C)N(C(=O)CC(C)C)C(C)(C)C)nnn2)(OC)CN(CCCl)CC1C C(C(=O)NCC12CCCC1OCC2)(C(C)(C)C)NC(c1n(CCC)ccc1)=O C1(O)(N(C(C(F)OC)=O)C)CCN(C(C2(c3cccs3)CCCC2)=O)CC1 C1(C(=O)NC2CN(C(CNc3nccc(OC)n3)=O)C(CO)C2)CC2C(C1)C2(F)F CC(C)CCCC(C)C(=O)NC(C1(O)CCN(C(C2CCCC2(C)C)=O)CC1)C Cc1nc2ccc(NC(=O)NCc3cncc(Cl)c3Cl)cc2nc1C N1(C(CSCC)=O)CCOCC1C(=O)NC(Cc1cccc(Br)c1)CC(=O)NC c1(C(=O)NC2C(CNC(CCC=C)=O)C2)ccc2nccc(Br)c2c1 S(=O)(=O)(c1cccc(=NC(C)CCO)[nH]1)NCC(N1CCC(C)CC1)C C1(C(=O)NCC(C)(C)NC(=O)CSc2nc[nH]n2)CCCCC1C1CC1 C(=O)(CCCS(N)(=O)=O)N1CCC(N(CCC)C(c2cc(F)cc(F)c2)=O)CC1 C12(C(=O)NC(C)CS(C)=O)CC(c3ccccc3F)(C1)C2(F)F N1(c2nccc(OC)n2)CC2C3CCC(C2C1)N(C(=O)CCN1CCOC1=O)C3 N1(C(C(c2ccc(C)s2)C)=O)CCOC(CCCNC(=O)Cc2cncn2C)C1 N1(C(c2n(C)ncc2)=O)CC2CC1CN(C(=O)Cc1cc(O)cc(Br)c1)C2 C12(NC(C(C)C3CCC3)=O)CC(C1)N(C(=O)COCc1cccnc1)C2 Cc1cc(F)cc(C)c1C(N1CC(CC(C)NC(c2nnn3c2CCC3)=O)C1)=O C(CC1=CCN(C(=O)CC2CCC2OC)CC1)NC(CC1(OC)CCOCC1)=O N1(C(C(C(C)O)(F)F)=O)CC(C2CN(C(c3ccc(C4CC4)cc3Cl)=O)C2)C1 C1(F)(C(=O)NCC(C)N(C)C)CCN(C(C2CCC(C)(C)C2)=O)CC1 C(=O)(C(C)CCOC)NCC(=O)NCC(=O)N(C(CC)C1CC1)C C1(C(N2CC(NC(=O)Cc3cncn3C3CC3)(CO)C2)=O)OCC2CCCC12 C(=O)(C(=O)CC(C)C)NCC(C1CCCC1)NC(c1cc(C)no1)=O N1(C(c2cc(CC)nn2C)=O)C(CNC(c2sc(C)nc2C)=O)CC2CCCC12 C(c1ccc(C(N)=O)cc1)=CC(=O)NC1CC(NC(c2nc(C)sc2)=O)C1 N1(C(C(CCC)F)=O)CCC(C)C(CC(=O)Nc2cn(C)nc2C2CC2)C1 N1(C(C2CN(C)C(=O)CC2)=O)CC2CCC1C(NC(C1CN(C)C1)=O)C2 c1(OC)cc(CCC(C)NC2CCCC(n3cccn3)C2)cc(F)c1 n1(CN2C(c3ccccc3)C3CC3C2)nc(C)c(N2CCN(c3ccc(F)cc3F)CC2)c1C C#CCC(C)(C(=O)NCc1nc(C)sc1C)NC(=O)C(O)C(F)(F)F C(C(CC(C)C)C(=O)N1CC(C)C(C)(CNC(=O)C(C)(CO)OC)C1)OC Cc1cc(C(=O)NC2CC(CNC(=O)C(C)C3CC3)C2)c(Br)cc1F C1(NC(C2(CC=C)CCC2)=O)CS(=O)(=O)CC1NC(=O)CN1C(=O)CNC1=O Cc1cccc2[nH]c(C(N3CCN(C(c4ccc(F)cc4N)=O)C4CC34)=O)cc12 CC(O)CCCNC(c1coc(C(C)NC(=O)CCC2CC2(F)F)n1)=O C1(NC(CC(C)SC)=O)CCC2CN(C(=O)C=Cc3ncc[nH]3)CC2C1 c1(SCCNC(N2CC(=O)NC(C(F)(F)F)C2)=O)cnc2n1CCOC2 C1(C(=O)NC(C(C)C)CNC(=O)C(C)CC2CCCC2)CCc2cnnn2C1 c1(C(N(CC(C)CNC(c2coc(C(N)=O)c2)=O)C)=O)ccc(F)c2occc12 c1(CCN(C(CSC(C)(C)C)=O)C(c2sc(Br)cc2F)=O)nc2ccccc2s1 c1(C(CCC(=O)N(C(CCNC(C(C(C)C)O)=O)C)C)=O)ccc2c(c1)CCC2 C1(COC)CN(Cc2csc(C3CC3)n2)CC(C)(C)O1 N1(C(=O)Cc2cccs2)CC2CN(C(c3cc4scnc4[nH]3)=O)CCC2(CO)C1 CC1(C)CCCN(c2nnc(C(F)F)o2)C1CNC(=O)CCc1nc[nH]n1 Cc1[nH]c(=NC2CCN(C(c3ncc(Cl)nc3Cl)=O)C2)ccc1C#N C1(C(=O)NC2C(NC(c3cc(OC)ncn3)=O)C2)CCN(C)C(=O)C1 Cc1ccc(COCCNC(=O)CSCCC)cc1F.C1C(=O)CO1.C1(N)CC1 c1(OCC)nc(NC(c2ccccc2)CC2CCCCN2)ncc1C c1(C(=O)Nc2ncc(OCC)nc2)ccc2ncc(-c3cc(O)ccc3F)n2c1 C1(C(=O)NC2(C)CCN(C(c3cc(OC)n(C)n3)=O)C2)CCC2(CC1)CC(O)C2 c1(C(C(=O)NC(C(=O)OC)(C)C2CCC2)=O)cc(O)cc(F)c1 N1(C(Cn2c(C)cc(C)n2)=O)CC(C)CCC1CNC(C1(CO)CCOCC1)=O c1(C(N2CCC(C(C)NC(C3CC(O)C3)=O)C2)=O)cc(N)cc([N+](=O)[O-])c1 N1(C(CCC=CC)=O)CC(C)(C)OCC1CNC(C1CCC(=O)N(C(C)C)C1)=O N1(C(C=CC(CC)C)=O)CCOC2(C1)CN(C(c1cc3ncccc3s1)=O)C2 c1(C(C)=O)cc(C(=O)NC2(CCNC(=O)C(F)C3CCCC3)CCCC2)oc1C c1(C)nc2ccccc2o1.c1(C(=O)OO)c(F)cc(F)cc1Br CN=c1[nH]c(C(=O)NC2CCCN(C(c3cccc(Cl)c3)=O)C2)cs1 N1(C(CS(CCOC)(=O)=O)=O)CCC(C2(NC(=O)CN(C)C(=O)C3CC3)CC2)C1 C(CCN=c1nc(N2CCC(CC3CC3)CC2)c2sccc2[nH]1)c1nnc(C)s1 CC1OC(C)CC1CC(=O)NCCOCCN(C)C(C1(CO)CC(F)(F)C1)=O N(C1CCCn2nccc21)C(CCN(C(c1c(NC)cnnc1)=O)C)=O CCC(CCCC(=O)NC1CCN(C)CC1C)NC(C1(n2cccn2)CC1)=O C(CNC(c1c(C)nsc1NC)=O)(C(C)(C)C)NC(COCCOC)=O c1(C(=O)NC2(CF)CCN(C(CC(C=C)C)=O)C2)cc(OC)cc(Br)c1 c1(OC)cccc(C(CF)NC(=O)C(C2CCCCO2)OC)c1 C(=O)(C1=CS(=O)CCC1)N1CCC(=CCNC(C2ON=C(C)C2)=O)CC1 N1(C(CNC(=N)N)=O)CCOC2(C1)CN(C(c1ccc(SC3CC3)cc1)=O)C2 c1(C(N2CC(N(C(C(CCC)c3ccccc3)=O)C)C2)=O)cc(C)c(F)cc1N C(CC(=O)NC1(c2nc[nH]n2)CC1)(C(F)(F)F)NC(C(CC)(C)NC(C)=O)=O C12CCN(CC1O)C2=O.c1(C(=O)NC)cccc(NC(C2(O)CCCOC2)=O)c1 C(=O)(CC(C)(C)C(=O)N1CC(CCCCNC(=O)C(C)CSC)C1)OCC CCCCC(C(=O)N1CC(S(C)(=N)=O)C1)NC(=O)CN1C(=O)CCCC1=O c1(CCn2c(N3CCC(c4cncc(C)c4)CC3)nnn2)ccc(Cl)cc1F N1(C(CC2CCCN(C(CC(C)O)=O)CC2)=O)CC2CCCN2CC1C c1(CNC(C2(C)CC(C)OCC2)=O)nc2c(s1)CN(C(=O)C(C)(F)F)CC2 n1(C(CC)C)cc(Cn2nccc2C(N2CC(COC(C)=O)C2)=O)nn1 CC(C)(F)CCC(=O)NC12CCOC(CNC(C3CS(=O)(=O)CCO3)=O)(C1)C2 CC(CC(=O)NCCNC(=O)CN(C)C(=O)C1CC1)n1ccnc1 CC1=C(C(=O)Nc2nccc3c(Br)nccc23)C(C)(C)CCC1 Cc1nn(C)c2ccc(C(=O)NC3CC(NC(C4CCC(F)(F)C4)=O)C3)cc12 C1(C(N(C(CC)C)CCOC)=O)C(C)OCCN1C(=O)CN(C1CCC1)C N1(C(c2ccc(SC(C)C)cc2)=O)CC(NC(C2CCC(=O)C2)=O)CC12CCC2 C1(CNC(C(C(C)OC)N(C)C)=O)(NC(=O)C(O)CCN(C)C)CCCCC1 C1(CNC(C(c2ccnn2C)C)=O)CCC(NC(C2(F)CC2)=O)CC1 C1(C2CCCO2)(C(=O)NC(c2nc(C)c(Br)s2)CC)CCN(C)C1 c1(NC(=O)NC2CC(C)CN(CC3CC3)C2)c2c(nn1-c1ccccc1)CCCC2 n1(CC(=O)NC(CC)(C)CNC(=O)C2=C(Cl)CC2)cc([N+](=O)[O-])cn1 C1(C(N2CCC(O)(Cc3cn(CCC=C)nn3)C2)=O)CC12CCOC(C)C2 N1(C(C(CC)C(C)C)=O)CCCC2(C1)CN(C(c1ccc(C)c(F)c1F)=O)C2 C(=O)(CCCCC(C)=O)N(CCn1cc(Cc2c(CC)cncc2)nn1)C C1(NC(CCSCCCC)=O)CCCC12CN(C(c1cc[nH]c3nccc1-3)=O)C2 C1CN=C2N=c3ncn(C)c3=C(N2)N1.N1(C(COCCOC)(C)C)CCCC1=O Cc1ccc(C(=O)NCC2CC(NC(C3(C)C=CCC3)=O)C2)cc1F N1(C(CN(C)CC)=O)CCC(C(N2CCCC(Nc3nccnc3C)C2)=O)CC1 c1(CC)cc(C(=O)NC2CC(NC(C3CC34CCCC4)=O)C2)nn1C c1(C(=O)NC(CN(C(CCC)=O)CC)C)ccc(Oc2ccccc2)cn1 C(=O)(CC(CC1CC1)NC(=O)COCCCN=[N+]=[N-])N(C(CO)CO)C C12(C(=O)NCCN(C(c3cn(C)[nH]c3=N)=O)C3CC3)CCN(CC1)CC2 C(C)(CCC(=O)N1CC(C)CC1C(N1CCC(C)(C(N)=O)C1)=O)OCC c1(NC(=O)CCC2CCOC2)cc(CC(=O)NCc2cnsc2)no1 N1(C(c2c(C)cccc2)=O)CCCN(C(c2coc(Br)c2)=O)C(CO)C1 CCCC(C(=O)OC)C(=O)NC(c1ccccc1)C(N1CCC(C(=O)OC)C1)=O C12(CNC(C(C)(N(C(C3C(C)CCO3)=O)C)C3CC3)=O)CCC(CO1)C2 C1(CNC(CSC(C)C2CC2)=O)CN(C(c2cc(CC3CCC3)c[nH]2)=O)CCO1 C1(CC(C)C)CCN(C(=O)CSCCNC(=O)Cc2ccc[nH]2)C1 Cc1c(C(=O)NC(C)(CNC(c2sc(F)cc2Cl)=O)CO)ccn1CC1CC1 CC(C)C(CCNC(C1CC1Cl)=O)NC(C12CC3CC1C2C3)=O C1(NC(C(C=CC)O)=O)CCC2CN(C(=O)Cn3cnnn3)CC2C1 C1(COC)(SC2COC(C)(C)C2)CCS(=O)(=O)CC1 C1(C(=O)NC(C(C)C)C(C)(C)O)CN(C(c2ccccn2)=O)CCN1C Cn1cc(C(N2C3CCC2C(C(=O)NC2CCN(CCF)C2)C3)=O)ncc1=O CC(C)C(C)C(C)CC(=O)NCCCCN(C(=O)C(C)(C)c1ccnn1C)C c1(C(=O)NCC2(CNC(C(C)(C)N(C)C)=O)CCOCC2)cc2n(n1)CCCC2=O c1(C(C(=O)NC2(CNC(=O)OC(C)(C)C)CC(COC)C2)=O)cc(F)cc(Br)c1 C1(C)(C(=O)NCc2c(C(N(C(CCSC)C)C)=O)c[nH]n2)COC(=O)N1 N1(C(C2(O)CCC2)=O)CCCC(F)(C(N2C3CSCC2C3)=O)C1 C(=O)(CCCc1nc(C2CC2)no1)N(C(C)CNC(C1CC1C(C)C)=O)CC CN1CC(C)(C)CC1C(N1CCC(F)CC1C(N1C2CCC(C2)C1COC)=O)=O Cc1nc(=NC(=O)c2ccc(-c3cn(Cc4ccccc4)nn3)s2)o[nH]1 CC1=C(C(=O)N2CC(C)N(C(=O)CCCc3cnn[nH]3)CC2C)CCCC1 c1(C(=O)NC(CC(C)Nc2cc(CC)nc(CC)n2)C)nccc2ccccc12 C12(NC(c3ncc(OC)cn3)=O)CCC(C1)N(C(C1(n3cccn3)CC1)=O)C2 c1(-c2ccc(C3C(C(=O)OC)=C(CC)NC(=S)N3)cc2)ccc2oc(O)nc2c1 N1(CC2CCC(c3ccccc3)CC2)CC(c2c(C(=O)OC)cc[nH]2)C(C)(C)C1 c1(C(=O)NC2(CC=C)CN(C(c3snc(C)c3N)=O)C2)cc(F)c(F)c(Cl)c1F N1(C(c2c(CCC)nns2)=O)CCCN(C(=O)CNS(N)(=O)=O)C(CO)C1 N1(C(c2cn(CCC)nn2)=O)C(C(N2CCNC(=O)C2C)=O)CCC12CC2 C12(CNC(CCOCCC)=O)CN(C(=O)C(O)C3CC3)CC1(C(F)(F)F)C2 N1(CC(=O)NCC2N(C(C(CCC#C)O)=O)CCC2)C(=O)c2cccnc2C1=O C1(NC(C2C(CCC)C2)=O)COC2(CCN(C(c3cccs3)=O)CC2)C1 c1(CC)ocnc1C(=O)NCC1(F)CC(NC(=O)C(C)OCCC(C)C)C1 c1(OC)ncc(-c2cn(CC(=O)NCC3CCCCC3(F)F)nn2)cc1C N1(C(c2cn(C)nc2)=O)CCC=C(C(=O)Nc2cc(F)c(F)c(F)c2)C1 N1(C(C23C(CN(C(C(C)N(C)C)=O)C2)COC3)=O)CCC2(CCCOC2)C1 CCC(CCCC(=O)NC1CCC(C)(C)CC1)NC(=O)C(CC)CC C(=O)(C(C#N)(CC)CC)N1CC2(CN(C(c3c(CCCCC)cc(Cl)s3)=O)C2)C1 C1(NC(=O)CCc2ncc[nH]2)CN(C(c2ccon2)=O)CCC1C(F)(F)F C1(C(=O)NC(C=C)CO)(CC=C)CN(C(C2CCCO2)=O)C1 N1(C(C(COC)C)=O)CC(C)(C)CC1CC(=O)NCC(F)Cl C1(CC(=O)OCC)CN(c2ncccc2C(F)(F)F)CC(C)O1 c1(C(=O)NCCC(C)NC(c2nnc(O)nc2O)=O)ccc(CO)c(F)c1 C1(CNC(CC=CC=C)=O)CCCC(NC(c2nncn2C(C)C)=O)C1 CCC(CC)C(C)C(=O)NCCOCCCNC(=O)CCc1nc(C)cs1 C12(COC)CN(C(c3cnc(C(C)C)nc3)=O)C(CNC(=O)CC(C)SC)(C1)C2 CC(C)C(CO)C(=O)NC(C1CCCCC1)CNC(c1cnc(F)c(Cl)c1)=O CCCC(O)CC(=O)NC(CO)C(C)NC(=O)CCCc1cncs1 C1(CC(=O)NCCC2(NC(C3CC(=O)NC3=O)=O)CC2)C2CC3CC(C2)CC1C3 C(=O)(C1CCCc2n[nH]cc21)NC(CNC(c1cc(C)nc(C)c1O)=O)(C)C c1(CC(C(=O)OC)NCc2cn(CC(CC)C)nn2)cccc(F)c1 C=C1CCC(C(N2CC(OC)CC2CNC(=O)CNC(=O)CC)=O)CC1 c1(-c2n(CC=C)nc(C3CC3C)n2)ccc2nc(O)n(C3CCCC3)c2c1 c1(CC)ccc(NC(=O)CCC(C)NC(C2CCN(OC)CC2)=O)cc1C c1(C(=O)NC(C)CN(C(=O)C=CCN(C)C)C)cn(CCO)nn1 C=CC1CCN1C(=O)CCNC(c1cc(C2CC2)[nH]n1)=O C1(C(N2CCCC(NC(CCCC#CC)=O)(CO)C2)=O)CCC2(CC1)CC2(F)F C1(CC(N2CC(CN(C(=O)CCC(F)F)C)OCC2)=O)CCCCC1(C)C C1(C2CCN(C(=O)CC(c3cccs3)N(C)C)C2)(NC(CCC(=C)C)=O)CC1 C=CC(C)(C)CC(=O)N1CCC(=C)CC1C(=O)NC(C(C)(C)O)C1CC1 N1(C(CCOC)=O)CCC2CCC(C1)N2C(C1CCCCCCN1C)=O C1(C(N(CC(C)N(C)C(c2cocn2)=O)C)=O)CCc2n[nH]c(C)c2C1 N1(C(c2cc(C(N)=O)[nH]n2)=O)CC(CNC(=O)C(F)=CC2CC2)OC2CCCC12 Cc1ccccc1C=NOCc1sc(C2CC2(F)F)nc1C C(=O)(CCCCC(F)(F)F)NCC1CCC(C)(C)CN1C(C1CC12CCC2)=O Cc1cccc2c1CC(C(=O)NC(CNC(=O)CCCC1CCCC1)C(C)C)O2 C(=O)(C(F)CCC(C)(C)C)NCC1CC(NC(C(C)=C(CC)C)=O)C1 c1(CC)ccc(C=CC(=O)NC2CN(C(=O)CCn3ccccc3=O)C3CC23)o1 C1(N(C(=O)CN2CCSCC2)C)CC2CC1N(C(=O)C=Cc1cn(C)nn1)C2 C1(N(C(CCN(C(C)=O)C)=O)C)CCN(C(=O)C(C)OC2CCCC2)C1 N1(c2cccc(C(C)O)c2)CCCc2ccc(P(C)(C)=O)cc21 CC(C)C(C)C(=O)NCC(C(=O)NCc1ccc(OCCO)nc1)N(C)C N1(C(CCC2CC(OC)C2)=O)CC(NC(c2conc2C)=O)C2CCCC2C1 N1(C(C(C)O)=O)CC2CC1CCN2C(=O)CCc1cc(Cl)no1 C(CC(=O)NCC1(C)CCOCC1)(C(F)(F)F)NC(Cc1c(C)cnn1C)=O c1(C(N2CCC(C3N(C(C=CC=CC)=O)CCCC3)C2)=O)cc(F)c(Cl)cc1Cl N1(C(C(Cc2ccco2)NC(c2cc(CC)[nH]n2)=O)=O)C2CCCC1COC2 c1(C(N2C(C(=O)NCCN3CCN(CC)CC3)CSCC2)=O)c[nH]nc1[N+](=O)[O-] c1(-c2c(F)cccc2)nccc(=NCC2Cc3ccccc3O2)[nH]1 Cc1cc(O)c(Cl)cc1C(=O)NCC1CCN1C(C12CC1COC2(C)C)=O C1(C(=O)OC)CCC(C2CCCC2)CN1C(c1cc2occ(Br)c2[nH]1)=O C1(C(=O)NC(CN(CCCC)C)C)CN(C(c2cnns2)=O)C(C)(C)C1 N1(C(CSCC)=O)CC2CCN(CN(C)C)CC2C1.C12(CC1)N(C(C)C)C2=O N1(C(Cn2c(=O)ccc(C)n2)=O)CCC2(CCN(C(C3NC(=O)OC3C)=O)C2)C1 N1(C(c2scc(C(=O)OC)c2)=O)CC(C2CN(C(=O)C(C)CC(N)=O)C2)C1 C#Cc1ccc(CCCC(=O)Nc2cnn(CCN3CCNC3=O)c2)cc1 C#CC1CCCCN1C(c1ccc(CNC(=O)C(O)C(C)C)nc1)=O Clc1cc(CCCn2cc(CCC3CCOCC3)nn2)on1 C(=O)(C(O)CCC(C)C)N1C(CNC(Cc2nc(CC)sc2)=O)CCCCC1 C1(NC(c2c(C)nco2)=O)CCCC12CCN(c1ccncn1)C2 C(=O)(CCS(=O)(=O)NC)N1CC(CCC)C(NC(=O)C(C)CN(C)C)C1 c1(C(N(CCNC(c2cnnc(C3CC3)c2)=O)CC)=O)cc2cccnc2cc1F n1(CC)nc(C(=O)NCC(C2CCCC2)NC(=O)C(C)CN(C)C)ccc1=O CCCC(C(=O)N(C)CCC1CCN(C(=O)C(C)(O)C(C)C)CC1)S(N)(=O)=O C(CCN=c1[nH]c(=NCCC(OC)OC)[nH]c2c1COC2)n1c(CCC)ncc1 Cc1ccc(NC(C2(C)CCCN2C(c2cc(F)ccc2Br)=O)=O)c(C(N)=O)c1 c1(SC)cc(C(N2C(C(c3ccccc3)=O)CC2C(=O)OC)=O)c(C)o1 c1(C(N2C(CNC(C(C3CCCC3)OCC)=O)CCC2)=O)ccc(C(F)F)cc1 CN1CCN(C(=O)CCCNC(C23CCCN2CCC3)=O)CC1(C)C C(=O)(CC(C)C(C)(C)C)NC1C(NC(Cc2nc(C(C)C)sc2)=O)C1 Cc1cccc(CCC(=O)N(C(C)CCNC(C2CCC2)=O)C)c1Cl c1(CNC(=O)N(CCc2cccs2)CC2CC2)nnc2n1CCCC2C(F)(F)F C1(CN(C(C(CC)O)=O)C)CN(C(=O)CCn2ccnn2)CC12CC2 N1(C(C2CC(C)(F)C2)=O)CCC2C(CCCN2C(=O)C=CSCc2ccco2)C1 C=CC1(C(=O)NC2CN(C(c3ccnnc3O)=O)CCC2CO)CCCCC1 C1(NC(=O)CC2CCCOC2)CC2CN(C(c3ccc4cncn4c3)=O)CC2C1 N1(C(c2scc(CC)n2)=O)CCC(O)C(C(=O)Nc2cc(Cl)cnc2OC)C1 CN1C2(CCN(CC3CCCCC3)CC2)C(NC(c2ncccn2)=O)CS1(=O)=O N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)CCCCCC(C)O)C2CCCC12 CCC(C)CCC(=O)N1CCN(C(C2COCCOC2)=O)C(C(C)C)C1 N#Cc1ccc(C(=O)NC2C3CN(C(c4coc(Cl)n4)=O)CC23)c(O)n1 Cc1cc([N+](=O)[O-])cnc1N1CC2(CN(C(c3ccc4c(c3)OCC4)=O)C2)C1 c1(C(N2C3C(NC(c4ccccn4)=O)CC(C3)C2)=O)cc2cn[nH]c2cn1 C1(C(N(CCNC(CCCNC(C)=O)=O)C)=O)COCCN1C=O N1(C(C2N(C)C(=O)NC2)=O)CCC(C2CCN(C(=O)C(C)(C)CCC#N)CC2)C1 c1(C(=O)NC2(C3CN(C(Cc4ncc(C)s4)=O)C3)CC2)noc2c(F)cccc12 C1(C(N(C)Cc2nc(C)sc2)=O)CN(C(=O)C=CC2CC2)C2(CCC2)C1 c1(NC(=O)NCCN(C)C(=O)OC(C)(C)C)ccc(Br)cc1-n1cncn1 c1(C(=O)NCCN(C(CCOC)=O)CC(C)O)ccc2n[nH]c(C)c2c1 C(CCCCC(=O)NC1CCN(C(c2cc(C)c(C(F)F)cn2)=O)C1(C)C)=CC CCCCCS(=O)(=O)CC(=O)Nc1ccc2c(c1)N2C.c1(NC)ccc(F)cc1 c1(SC)ccc(Cl)c(C(=O)Nc2ncc(CN3CC(C(=O)OC)C(O)CC3)nc2)c1 C1(CC(=O)NCC2(C)CCC2)C2CCCC2N1C(C1(N)CCC1)=O.C(N)=O Cc1onc(Cl)c1C(=O)NC(C)CCCNC(=O)CCCOc1ccc(F)cc1 C(CCC(=O)NCC1CCCC1C(=O)NCc1cnns1)OCC C1(C(=O)NCC(C(C)C)NC(CCc2onc(CCC)n2)=O)CCCCC1(F)F C12(C(=O)NCC3N(C(C(C(=O)OC)OC)=O)CCCC3)CCCC(C1)OC2 C=CC1(NC(C2CC(CCNC(=O)C=C3CCOCC3)C2)=O)CCOCC1 C1(C(=O)NC2C3CC2CN(C(=O)CNS(=O)(=O)C2CC2)C3)CCCN2CCCC12 C=C(CNC(=O)Cc1ccccc1)CCNC(C1(C=C)CC1)=O c1(OC)ccc(CNC(C2CC2NC(=O)C2CC2)=O)c(C)c1 c1(NC(c2ccc(Cl)nc2F)=O)ccc(NC(C2COCCO2)=O)cc1F c1(C(=O)NCC(C)CNC(=O)CN(C)C(c2cccs2)=O)cc2sccc2n1C C1(CC)C(C(=O)N(CC(O)CN(C)C(c2cc(Br)ccn2)=O)C)CCN1C C(=O)(CC1OCc2cc(Cl)ccc21)NC1CN(C(CNS(C)(=O)=O)=O)C(CO)C1 c1(C(=O)NCC2(F)CC(NC(C(C)O)=O)C2)c(Cl)cc(Cl)nc1N C(N=c1[nH]c2ccc(Cl)cc2s1)C1CCCC(NC(C2CC(C)OC2)=O)C1 c1(C(=O)NC(CNC(C(CC)OC)=O)CO)ccc(OCC(N)=O)cc1 C1(CC(=O)N(C2CCCC2)CC#C)C2CCCC2N1C(C1CC(CC2CC2)C1)=O N1(C(CC(C)(C)C(F)(F)F)=O)CCC2CC(NC(=O)CS(N)(=O)=O)CCC2C1 C(CC1=CCCCC1)NC(C1C(NC(C(CCSC)O)=O)CC=CC1)=O c1(CC(C)(C)C)nc(-c2cc(CO)[nH]n2)n(C2(C)CCCCC2)n1 Cc1cccc(C)c1C(O)C(=O)NCC(C)(C)NC(c1cc(Br)n[nH]1)=O C1(C)(C(=O)OC)CC(NC(=O)C(C)N(C(=O)COCC(C)SC)C)C1.N1CCCC1 N1(C(CC)=O)CCCCC1C(N1CC(CCNC(=O)CCC2CCCN2C)C1)=O C1(CNC(C(C)CO)=O)CCCC2CN(C(=O)CC3(N(C)C)CCCC3)CC12 CCCCCC(C(=O)N(C)CC1CN(C(=O)CCCOCCOC)CCO1)C(C)C C12(CNC(C(CC#C)C)=O)CCC1CN(C(c1ccc(Br)cc1O)=O)C2 C1(C(=O)NC2(C)CC(NC(COCC)=O)C2)Cc2cc(C)ccc2S1(=O)=O c1(C2CN(Cc3c(OC)cc(F)cc3F)C2)nnc2ccc(SC)nn12 c1(C(=O)NCC23C(CN(C(C(CCC)OCC)=O)C2)C3)cc(F)ccc1C C1(NC(=O)NCc2cc(C(=O)OC)cc(F)c2)CCC2=NN=NN(C2)C1 C1(CNC(=O)CCn2cnnn2)CCC2(CO1)CC(NC(c1csc(Cl)n1)=O)C2 c1(C(=O)NC(c2n(C)ncc2)C(N2CCCC(CC3CC3)C2)=O)ccc(O)cc1 C1(c2nnnn2C2CC2)(Nc2cncc(NC(C)=O)c2)CCN(C)C(C)C1 N1(C(C(C2CCC2)OC)=O)CCCCC(CNC(c2cc3n(n2)CCO3)=O)C1 CCC1C(=O)Nc2ccc(C(=O)N(CCCOCCNC(C3CC3F)=O)C)cc21 C(C(C(C)C(C)C)NC(C1(CCF)CCC1)=O)NC(CCNC(C)=O)=O c1(C(=O)OC)sc(NC(c2ccc(NC(c3cn(C)cn3)=O)cn2)=O)nc1C N1(C(C=COCC)=O)CCC(CNC(c2cn(C)c(=O)nc2O)=O)C12CCC2 C1(C(N2C(CNC(=O)Cc3ccon3)CCCCC2)=O)CC1C1CCCCC1 CCCCCCCC(F)C(=O)NCCC1CN(C(=O)C=NOC)C1 Cc1ccc(O)c(CC(N2CC(NC(C3(C)CCCCCC3)=O)CC2(C)C)=O)c1 Cc1nc(CNC(C2CC3CCC2C3)=O)oc1C(=O)N(C)Cc1cnnn1C c1(OC)ccc(C(=O)NCC(C2CCC2)NC(=O)C(=Cc2cnn(C)c2)C)nc1 C12(C(c3n(CCCC)nnn3)NCC3(CC4CC4)CCC3)CCCC1C2(F)F c1(N2CC(CNC(C(COC)O)=O)N(C)CC2)cc2c(cn1)C(=O)CCC2 c1(CCC(=O)N(C(C)C)CC2CN(C(=O)COCCF)C2)ccccc1[N+](=O)[O-] C(=O)(C1SCCc2sccc21)N(C)CC1CN(C(C2CC(O)C2)=O)CCO1 C1(CC(=O)N(CCC(=O)N(CC(C)C#N)CC)CC)COCC(C)O1 C(=O)(CC(F)(F)Br)N(C)CC1N(C(c2cc(C)ns2)=O)CCC1 c1(CNC(C2N(CC)CCOC2)=O)ccc(CNC(C2CC2F)=O)c(F)c1 CC1CN(C(C2CC3C(C2)C3(F)F)=O)CCN1C(=O)Cc1ccc(Cl)s1 C1(N(C(CNC(C(CC)C)=O)=O)C)C2CN(C(c3csc(COC)c3)=O)CC12 C(=O)(C(C)C(O)CC(C)C)N1CCC(COC)(CNC(C2CC(C#N)C2)=O)CC1 CC(C)CC(C)CC(=O)N1CC2(CCCC2)C1C(=O)NCC1CCCCO1 c1(C(=O)NCC(C)N(C)CC2CCC3CC3C2)ccc2sccc2c1 N1(C(C#CCNC(Cn2c(C)nnn2)=O)=O)CC(C#N)(N(C)C)C1 C(=O)(CCCC(CC)NC(C1Cc2nccn2C1)=O)Nc1ccc(CC)nc1 C(CCN=c1nc2scnc2c(N2CCC(S(C)(=O)=O)C2)[nH]1)C1(C)CC1 N1(C(C(C(C)NC(c2c(C)non2)=O)C)=O)CC2OC(=O)N(C)C2C1 N1(C(C(C2CCOC2)NC(CC(CC)C(C)C)=O)=O)CC2CCOC(=O)C2C1 c1(OC)ccc(F)c(C(=O)NCC(O)COCC(C)C)c1F Cn1ncc(C(N)=O)c1C(=O)N(C1CCCCC1NC(C1(C)CC1(F)F)=O)C C1(NC(c2n(CC=C)nnn2)c2occc2Br)CCOC(c2cccc(Cl)c2)C1 CC1(C)OC(C)(C)C1C(=O)NCC1CCCCC1NC(=O)CCn1cnnn1 C(=O)(C1=NOC2COCC12)N1C2CCC(NC(C3CCC(CC)CC3)=O)C(C2)C1 C1(C(c2cn(CCCC(=O)O)nn2)NC(c2cc(OCC)n[nH]2)=O)CCCCCC1 CCCC(C)(O)CC(=O)NCC(C)=CC(=O)NCC(N1CCCC1)=O C(=O)(C(C)(C)CCC(=O)NCC1CCCC2(CN(C(=O)CCCF)C2)O1)OC N1(C(c2cn(CC=C)nc2)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)CC1CF C1(C(=O)Nc2ncn(C)n2)CN(Cc2c(Br)cncc2Br)CCC1O N1(C(C2(C#N)C(C)(C)C2)=O)CC2(C1)CN(C(C1C3CC4C(C3=O)C14)=O)C2 C(N=c1[nH]cnc(Cl)c1C(=O)OC)C1CC(NC(C=COCC)=O)C1 c1(C(N(C2CCCN(C(=O)C(C)CO)C2)CC)=O)cc(C(F)(F)F)cc(F)c1 N1(CC(=O)NC(=O)C2CC2)CCC2C(CCCN2C(c2sccc2Cl)=O)C1 N1(C(CCC2CCN(C(C(C=C)O)=O)C2)=O)C2CCCC1CC(=C)C2 C(=O)(CC(C)C(=O)OC)NC1CCN(CCNC(C=COCC)=O)CC1 c1(C(N(CCN(C(C2CCC(CCC)CC2)=O)C)C)=O)ccc2nn[nH]c2c1O N1(C(C2CSCCN2Cc2cscc2F)=O)CC(c2ccccc2)C2(COC2)C1 c1(C(=O)NC(C2CCCC2)CNC(C2(C)C(C)C2)=O)cc2n(n1)CCCO2 N1(C(C2N(C(C3CC(OC)(OC)C3)=O)C(C)C2)=O)CCC(F)C(F)C1 c1(-n2c(C(C3(CCl)CCC3)NC(CCC=C)(C)C)nnn2)ccc2c(c1)CCC2 CN1C(=O)NCC1C(=O)NC1CC(CNC(=O)CC2(O)CCCCC2)C(O)C1 C1(CCN(C)C)CCOCC1.c1(C2CN2)ccccc1 N1(C(c2c(C)con2)=O)CC2CC(C1)CN(C(c1cc3ccnn3cn1)=O)C2 N1(C(C23C(C)OC(C)(C2)C3)=O)CCC(C2CC2)(CNC(c2ccc[nH]2)=O)C1 N1(C(c2ccc(SC)o2)=O)CCC2(CCN(C(=O)C(C)C3CCC3)C2)C1 N1(C(CC(CC)C)=O)CC2C3CCC(C2C1)N(C(C1CCC2(CCOC2)O1)=O)C3 C1(C(=O)NCC2CCN2C(=O)CCc2ccccc2F)CC12CCSCC2 S(=O)(=O)(c1ccc(Br)c(F)c1)N1CC(C(=O)Nc2nccnc2Br)C(O)CC1 N1(C(CC=CCC)=O)CCOC(CCNC(C2(C#N)CCOC2)=O)C1 C12(C(=O)NC3CCC(NS(CC(=O)OCC)(=O)=O)CC3)COCC(C1)OC2 CCCC(C(=O)N(C)CCOCCOC)NC(=O)C(N1CCSCC1)C c1(C(=O)NCC(C)NC(=O)C(c2ncc(Cl)n2C)(F)F)cc2cc(Cl)ccc2o1 N1(C(CC2C(NC(CNC(=O)OCC=C)=O)CCC2)=O)CCCC(N=[N+]=[N-])C1 c1(CC)cc(CNC(=O)CN(C2CCC2)C(c2scnc2Cl)=O)n[nH]1 C1(CS(Cc2c(CC)occ2)=O)CCS(=O)(=O)C1.c1(C2C(=O)N2)ccccc1 c1(OC)cc(NC(C2CC(F)CN(C(c3c[nH]cc3C)=O)C2)=O)nc(Br)c1 c1(C(N(CCCNC(CC(C)OC)=O)C(C)C)=O)cc(C2CC2)cc(F)c1 C12(C(=O)NCC(=C)CCNC(c3cncc(C)c3)=O)CCCC1NC(=O)C2 C1(C(=O)NCCCCNC(CC)=O)CCC(=O)N(CC)C1 c12n[nH]cc1C(=O)N2.C(C(=O)NCCCC1(C)CC1)SCCC CCCC(C)CC(=O)N(CC(CO)(CO)NC(c1cnc(C2CC2)[nH]1)=O)C N1(C(c2c(C(C)NC(c3cnc(O)o3)=O)noc2)=O)Cc2ncsc2C1 N1(C(C(CC)COC)=O)CCc2ccc(C(=O)NC3CC3C3CC3C)nc2C1 c1(CNC(=O)C=C2CCCCC2)ccc(CCNC(C2CC23CCOC3)=O)cc1 C=CCCCC(C(=O)NCCCO)NC(=O)Cc1ccc(C#N)cc1 N1(C(C(COC)O)=O)CC2CN(C(c3ccnc(OCCO)c3)=O)CC2C1 C1(F)(C(N2CC3C(CNC(COCCCC#C)=O)C3C2)=O)C(C)(C)C1(C)C C1(NC(CCC2CC(OC)C2)=O)CN(C(C2(C#N)CC3(CC3)C2)=O)CCC1CO c1(Cc2n(CC)c(CN(C3CCC(C)C3)C)nn2)c(F)cccc1F c1(C(=O)NC2C(CC)CN(C(c3csc(O)n3)=O)CC2)noc2cc(F)ccc12 C1(CNC(CCC(=O)OC)=O)(NC(=O)CCC2NC(=O)NC2=O)CCCCC1C N1(CC(=O)NC2C(C)(C)CCC2)CCN(C(C2(N)CCC2)=O)CC1=O Cc1nc(NC(C)(CNC(=O)C(C)C(C)O)Cn2cccn2)ccc1[N+](=O)[O-] c1(CNC(=O)NC2CCNC2)ccc(-c2ccc(C(F)(F)F)c(F)c2)cc1F c1(NC(Cn2cc(CNC(C3C(C)CCC3)=O)nn2)=O)ccc(O)c(F)c1 C1(NC(c2c(C(C)=O)ccs2)=O)CCOCC1NC(c1ccc(C(F)F)cn1)=O c1(OC)ncc(C)cc1C(N1CC2(NC(=O)C(C)N(C)C)CC1C2)=O CC1OC(C)C(C)N(C(=O)NC(c2nccn2C)C)C1C c1(C(=O)NCC2CC(C)N(C(C3CC3(Cl)Cl)=O)C2)cnc2[nH]nnc2c1 c1(C(N2CCC(CCCNC(CC3C(C)C3)=O)CC2)=O)ccnc(Cl)c1N c1(N(C(C(=O)Nc2c(C)cccc2)CC2CC2)C)ccc(SC(F)(F)F)cc1Cl c1(OC)ccnc(O)c1C(N1CC=CC(NC(c2nccc(C)n2)=O)C1)=O C1(N(C(C(C2CCC2)OCC)=O)C)CCCN(C(=O)Cn2ncc(Cl)c2C)C1 N1(C(c2c(C)nns2)=O)CCC(C)(CCNC(c2cn(CCCC#N)nn2)=O)C1 c1(C(=O)NC(C)C(C2CCCC2)NC(=O)C(C2CCOCC2)=O)ccc(CO)nc1 c1(N(CCN(C(=O)Cc2nn(C)cc2Br)C)C(=O)C2CC2)cc2occc2[nH]1 N1(C(C2CCCC23CC3)=O)CC2CCCC(C1)N2C(c1c(F)ccc(F)c1O)=O C1(CNC(C2C(CC)CCC2)=O)CCCC12CCN(C(C1C=C1C)=O)CC2 c1(C(=O)OC)nccnc1C(=O)NC(C)CC(C)NC(=O)C(c1cnn(C)c1)O c1(C(C)=O)ccc2c(c1)CN(Cc1ccc(-c3ccc(N)cc3Br)o1)CC2 Cc1nnc2n1CC(C(N1CCC1CNC(=O)CCc1ccc(C(F)F)o1)=O)C2 N1(C(C2C(=C)C2)=O)CCN(c2ncnc(Cl)c2CO)C(C)C1 C1(C(C)C(=O)NCC=CBr)CCN(C(=O)CCc2cccn2C)C1 c1(C(c2nnnn2CCCF)NC(c2ccc(C)o2)CC)ccc(OC)nc1 c1(C(=O)NCC2(OC)CCN(C(C(CC)SC)=O)C2)cc2ccc(OC)nc2[nH]1 c1(C(=O)N)c[nH]c2ncccc12.C1(OC)CC(CO)(NC(c2ccc(C(N)=O)o2)=O)C1 C1(=CCNC(C(C)=CC)=O)CCN(C(=O)Cc2ccc(-c3ccsc3)cc2)CC1 c1(CC)cc(C(N2CCCCC2c2cn(Cc3cnn(C)c3)nn2)=O)c(C)o1 CC1COC2(C1)CN(C(=O)C#CCNC(c1csnc1Cl)=O)C2 C1(C(=O)NCC(=O)OCC=C)CSCN1C(C1CC(OC2CC2)C1)=O CC1(CCNC(c2csnn2)=O)CCN(C(C2CC3CC(=O)C2O3)=O)CC1 N#CC1(C(=O)NC2COCCC2NC(C2(C3CCC3)CC2)=O)CCCC1 CCCCC(C(=O)NCCN(C)CC)NC(c1cc(C)cc(O)n1)=O N1(C(c2n(C(C)C)ncc2)=O)CC2ON=C(CNC(c3ccsc3)=O)C2C1 c1(CC)cc(C(N2CC(CC(C)NC(=O)C=CBr)C2)=O)ccc1F c1(C2(C)CC2)cc(C(=O)NC2COCC2NC(=O)CC2CCOCC2)no1 c1(CNC(c2ccccc2OC)C(=O)OCC)nc2c(s1)CCCC2 C1(C(=O)NCC(CO)NC(c2cnc(N(C)C)s2)=O)CCOC(=O)N1 C(=O)(C(C)CCCC(C)C)NC1CC2CN(C(c3ncc(C)nc3)=O)C(C1)C2 CC1CN(C(C2CCCC(F)C2)=O)CCC1CNC(c1c(O)cccc1Cl)=O N1(C(c2c(OC)c(C)cs2)=O)CC(NC(=O)C(C)=C2CCCC2)C(C)(C)C1 C(=O)(C1=CCCCO1)NC1CCC(CCNC(=O)Cc2nc[nH]n2)C1 C1(CC(=O)NCC(N(OC)C)=O)CCN(C(=O)C(C)CC#N)C1(C)C c1(CN2CC(CC(=O)N(C)CC3CCC(=O)N3)OCC2)ccc2occc2c1 c1(C(=O)NC2(COC)CCC2)n[nH]c2c1CN(C(C1(C)CCN(C)C1)=O)C2 Cc1cc([N+](=O)[O-])cc(Cl)c1NC(=O)CC1CN(Cc2cc(C#N)ccc2Cl)C1 Cc1cncc(C)c1C(=O)NCCCCC(=O)NC(c1ccccc1O)C C1(CC(N2CC(C)(OCC(=O)N(CCCOC)CCO)C2)=O)CCCC(C)O1 C1(C(=O)NCC2(CO)CC2)(CNC(c2c(C)noc2)=O)CC12CCC2 c1(OC)cccc(C(C)C(=O)NC(C)C(C)NC(=O)CSC)c1 C(=O)(C1CCCc2nn[nH]c21)N(CCOCCCNC(C1C(C)C1C)=O)C N1(C(c2c(CC)cc(Cl)cc2)=O)CC2(CC(NC(=O)C(C)(Cl)Cl)CO2)C1 N(C(=NCCC1CC1)NCc1cncnc1)CCC1CCCC(C)C1 C1(C(=O)NCC(C)NC(c2cocn2)=O)CCCCC1P(C)(C)=O C(CCCCC(=O)N1CC(O)CC1(C)C)N(C(C1C(CC)CCO1)=O)C c1(OC)ccc(C2CC2C(=O)NC2(C)CCCN(c3cc(C)nc(Cl)n3)C2)c(C)c1 C(=O)(C(C(C)C)NS(C)(=O)=O)NC(C1CCCCC1)CNC(c1c(C)occ1)=O N1(C(COCCC)=O)CC(O)C(O)C1CNC(=O)CC1OC(C)(C)OC1=O c1(CNC(=O)NC2(C3CC3)CC2)cc(Cl)ccc1[N+](=O)[O-] S(=O)(=O)(c1ccccc1Br)N1CCC(CN(C(C(C)(C)C)=O)O)CC1 C(CC(C)C)(C(=O)N(C1CC=CC1)C)ONC(c1ccc(N(C)C)cn1)=O C1(C(N(CC(C)NC(CN(S(CC)(=O)=O)C)=O)C)=O)(OC)CCSCC1 C1(C(=O)OC)Cc2ccsc2CN1C(=O)C(=O)NCCc1ccc(C)cc1[N+](=O)[O-] C1(NC(COCC(=C)C)=O)CCN(C(C23CCCC2C3(F)F)=O)C12CCC2 c1(C(=O)NCC2CCN(C(C(CN(CC)CC)F)=O)C2)c(F)cc(F)cc1Cl c1(CCC(=O)N(CCN(C)CC2CCN(CC)C2)C)ccc(O)nc1 c1(C2(C(=O)NC3CC(CCNC(=O)Cn4ccnn4)C3)CC2)ccc(Cl)c(F)c1 N1(C(C(C=C)OC)=O)CC(C(=O)NC2(COC)CCC2)C(C2CC2)C1 N1(C(C(C(C)C)NC(N)=O)=O)CCCOC(CNC(C2COCCO2)=O)C1 CC1CCCC=C1C(=O)NC1CC(C(C)NC(c2c(F)cc(F)cc2F)=O)C1 CCC(C)C(O)CC(=O)NC(C(=O)NCCC(F)(F)CO)c1ccoc1 N1(C(C(CC=C)C)=O)CC2CCCC(C1)N2C(C1CCN(CC(F)(F)F)CC1)=O C1(C(C)C)C(=O)NCCN1C(C1CCN(C(c2n[nH]c(C(F)(F)F)c2F)=O)C1)=O N1(C(C(CC)=CC)=O)CC(CNC(c2cc(-c3ccccc3)ns2)=O)CC1C C=CCC(C)C(=O)NC(C)C(C1CCCCC1)NC(=O)CCCNC(=O)C1CC1 N1(C(c2c(C)ccs2)=O)CCC2(C1)CN(C(=O)CCc1ccc(C(C)C)cc1)C2 N1(C(CN(CC(=O)NC(C)C)C)=O)CCN(C(C2(C)C=CCC2)=O)CC(C)(F)C1 CC#CCC(CO)NC(C1(NC(=O)CCc2ncccn2)CCCC1)=O C1(NC(c2ccc(CC)nc2)=O)CCC12CN(C(=O)C=CC(=O)NC1CC1)C2 c1(C(=O)OC)cccc(C2CC2)c1.C1C(C2(C)CC2)N(C)C(=O)N1.C1(C)CC1 c1(C(=O)NC2CC(NC(=O)COCc3nc[nH]n3)C2)cc(C2CC2)cc(F)c1 c1(CNC(C(c2ccsn2)N(C2CC(F)(F)C2)CC=C)=O)cccc([N+](=O)[O-])c1 C(CCCC(C)NC(=O)CCCOc1ccc(C)cc1)NC(CC(=O)OCC)=O C1(C(N2CCCN(CC(N3CCOCC3)=O)CC2)=O)CC2(CCC2)CCO1 O=C(N=c1c(Br)c[nH]cc1I)C1CCN(S(=O)(=O)C2CCCCC2)C1 c1(C(=O)NC2CCC3CC2CN3C(C2CC=CC2)=O)coc2ccc(F)cc12 C1(NC(C2(CC)CC2)=O)CN(C(=O)C(c2cccc(Br)n2)C)C(C)(C)C1 c1(CNCCCCCC(C)(C)C)cccc(S(=O)(=O)NC2CC2)c1 C12(CNC(COCCOCC)=O)CC1CN(C(=O)COc1nc(C)no1)C2 N1(C(C(C)(C)SCCC)=O)CC2CN(C(=O)C3CC3)CC2C1.C1(=O)CCCCN1 Cc1nc(N(C)C)sc1C(=O)N(CCCCN(C)C(C1CCCC1C)=O)C Cc1ccc(F)c(C(=O)N(C(CC(C)C)C(=O)NC2CCN(C(C)(C)C)C2)C)c1 C=C(C)CC(C(=O)NCCc1cnn(C)c1C)NC(=O)CNc1ccccn1 c1(C(=O)NCC(CNC(CCC#C)=O)F)cc(F)ccc1-n1ccnc1 c1(C(=O)NC(CNC(CC(CC)C)=O)(C)CC)ccc(C)c(N)c1 CC1(C)CCCCC1NC(=O)CC1C2CC1N(C(C1CN3CCC1CC3)=O)C2 C(CCCC(=O)N1CCC(CCNC(=O)CCc2cncs2)CC1)NC(N)=O N1(C(CC(=O)NCC#C)=O)CC2(CC(CC(=O)NC3(CC=C)CCOC3)C2)C1 C1(F)(CNC(C(=Cc2cn[nH]c2)C)=O)CCC(NC(=O)CC2CC2(Cl)Cl)C1 CC(O)C(F)(F)C(=O)NCC(C)(C1CCC1)NC(=O)CN1CCCCC1=O N1(C(C2C(C)CCC2)=O)CCC(C)(CCNC(C23CCC(C2)C3)=O)C1 C1(NC(C)=O)CCCN(Cc2cnn(C)c2CCO)C1 c1(C(N2CC(NC(C3CCCC3)=O)CC(C)(C)C2)=O)cc(F)c(C#N)c(F)c1 C1(N)(C(=O)NC(C(=O)OCC)CSC)CCOCC1(C)C C#Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(C)(C)C2)=O)ccc1C Cc1ccc(C(N2CCC(C(F)(F)F)C2C)=O)cc1S(=O)(=O)N(C)C C12(C(=O)NCc3c(C)non3)CC(C)(CN1C(c1sccc1C#N)=O)C2 c1(CC)cc(C(c2nnnn2C(C)C)NCCO)ccc1NC1NC(=O)NC1=O N1(CC(=O)NC(=O)NC(C(=O)NC)Cc2ccncc2)CCC(C(=O)OC)CC1 CC(C)C(C(=O)NC1CCN(C(C2(C)CCC2)=O)CC1F)C(C)C C(=O)(C1COc2ccccc21)N1CC2CCN(C(c3n(C=C)nnc3)=O)C2CC1 C1(CNC(CC(C=C)CC)=O)CN(C(C2CC(CC(F)F)C2)=O)CCC12CCC2 N1(CC)CCCC(C(=O)NC2CC(O)(CNC(c3csc(C(F)(F)F)n3)=O)C2)C1 C(=O)(C1CCc2nccn21)N1CCCC(C(=O)NCCn2cncn2)C1 N1(C(CSCCSC)=O)CCC(C(CO)NC(=O)CCc2ccon2)CC1 CS(=O)(=NC(=O)CCn1cc(Br)cn1)c1ccccc1Cl CC1CC(CNC(=O)NC2(C(F)(F)F)CC=CC2)CC(C)O1 c1(NC(C=CC(C)NC(c2ccc(CO)nc2)=O)=O)ccc(O)cc1Cl CC1COCC(C(=O)NC2CC(O)(CNC(c3ccnn3C3CCC3)=O)C2)O1 C1(C(C)(C)C)CCN(C(C2CCCOCC2)=O)C(CNC(c2cc[nH]n2)=O)C1 N1(C(C(CCO)N(C)C)=O)CC2CS(=O)(=O)CC2(CNC(c2cnco2)=O)C1 Nc1ncc(C(=O)NCCOC2CCN(C(=O)C=CC3CCC3)C2)cc1Br c1(NC)cnccc1C(=O)N(CC(N1CC(N2CCOCC2)C1)=O)C1CCC1 CC(Cc1cnn(C)c1)C(=O)NC1CN(C(=O)COc2ccsn2)C1 N1(C(CNC(C(C)(C)OC(C)C)=O)=O)CCC(O)C(C)(C)C1 C1(O)(C(=O)NC2C3(CC(NC(c4scc(C)c4)=O)C3)C2)CCCC(C)(C)C1 N1(CC(=O)NC2CC(CNC(=O)CC3CCC4CC34)C2)CCCS1(=O)=O C1(CCNC(c2ncn(CC)c2)=O)C(C)CCCN1C(=O)C1=COCCC1 c1(NC(=O)NC2CC(Nc3ccccn3)C2)ccccc1CC1CCOCC1 c1(C(=O)NC(C2CCCCC2)CO)cncc(NC(c2ccc(Br)cc2)=O)c1 c1(C(N2CCCC3(C2)CN(C(C2CC=CC2)=O)C3)=O)ccc2cc[nH]c2c1F c1(N2CCN(CC(C)(C)NC(=O)C(N)=O)CC2)nc(Cl)nc2c1CCOC2 C1(NC(C(CC=C)CC=C)=O)CN(C(=O)Cc2[nH]cnc2C)CCC12CCC2 N(C1CCc2c(Br)cccc21)C(=O)NC1C(c2c(C)cccc2)(C)C1 C(=O)(CC(F)(F)C(F)F)N1CC(CC=C)(NC(c2nonc2CC)=O)C1 C1(CNC(CC=CCNC(CCCOC)=O)=O)COCC(C)O1 Cc1cc(CC(=O)NC(C)CNC(=O)C(F)CC2CCCCC2)on1 C1(NC(CN(CC)CC)=O)CCC(CN(C(=O)CNS(N)(=O)=O)C)CC1 O(N=C1CCCCCC1)CC(N1CC(OC)(CNC(=O)C(O)CN(C)C)C1)=O C1(C(N2C(C(N(C)Cc3cnc[nH]3)=O)CC(O)C2)=O)CCCC2(CC2)C1 C1(C(=O)OC)CN(C(=O)C(=O)NCC(c2c(Cl)cccc2Cl)(C)C)CCN1C N1(C(C(C)Oc2ccccn2)=O)CCc2[nH]nc(CNC(c3cnco3)=O)c2C1 N1(C(c2c(C)c[nH]n2)=O)CC(NC(=O)Cn2nnc(=N)[nH]2)C2(CCC2)C1 N1(C(C=Cc2ncn(C)c2)=O)CC2CC(C1)N2C(c1nocc1C1CC1)=O N1(C(c2c(OC)csc2)=O)CC(NC(C2(O)CCSC2)=O)CC(O)C1 C(=O)(C(=O)C(F)(F)F)NCC1CCCC(NC(c2c(CC#N)ccs2)=O)C1 c1(NC(C2(NC(C(C)CCN(C)C)=O)CC(F)C2)=O)cnc2[nH]ncc2c1 C12(NC(C(c3ccc(CC)s3)=O)=O)CC1CN(C(C1CCC(C)CC1)=O)C2 C1(CC2(C(=O)N)CC2)COCC1NC(C1CN(C2CCOC2)C1)=O.CO Cc1nc2ccc(C(=O)NC3CC4CC3N(C(=O)CC35CCCC3C5)C4)cc2o1 c1(CCC)nc(NC2CCCN(C(=O)CC)C2)c(C)c(Cl)n1 N1(C(C(C(CC)C)c2ccccc2)=O)CCC(C#N)(C(C)(C)O)CC1 N1(C(c2c(C(C)N)noc2)=O)CC(=O)N2CCCCC2C1 c1(C(N(C(CN(C(C(C)SCC)=O)C)C)C)=O)cc2c(cn1)OCCO2 Cc1c(C(=O)CNC(=O)C(c2ccc(Cl)cc2)C2CC2)sc2ccccc12 N1(C(C2N(CC)CCC2)=O)CCN(C)C(C(=O)NOC(CO)CO)C1 c1(NC(N2CCC(N(c3ccccc3)C)C2)=O)ncnc2c1ncn2C c1(C(=O)NC(CCOC)CNC(=O)CC(F)(F)Cl)ccc(N=[N+]=[N-])cn1 CC(CS(C)(=O)=O)C(=O)N1CC2(CCCN2C(=O)CC(Cl)Cl)C1 Cc1ccc(C(=O)NCC2(C(=O)NCCC3NC(=O)NC3=O)CCCC2)nc1 Cc1nncc(C(=O)NCC23CC(C2)C(NC(=O)C(O)C2CC2)CO3)c1C N1(C(C(=O)NCCCCc2ccccc2)=O)CCn2c(cc3c(Cl)cccc23)C1 c1(OC)ccc(C(=O)NCC2C(C)CCN2C(c2coc(C(C)(C)C)n2)=O)nn1 C1(C(N2CC(CC(=O)NCC3CC(OCC)C3)(OC)C2)=O)CC12CCCC2 c1(S)cccc(O)c1.C1(C(N2CC(n3cc(C(=O)OC)nn3)C2)=O)CCC(C#N)C1 Cc1nc(C(F)(F)F)ccc1C(=O)NC1CN(C(=O)Cc2cscn2)CCC1F c1(C(C(=O)NCCC(=C)CNC(C2C3CCC23)=O)(F)F)ccc(C)cc1 N1(C(C(=O)NCCOc2cc(O)nc(O)n2)=O)CCS(=O)(=O)CC1CCO C1(C(N2CCCC(NC(CSCC#C)=O)C2)=O)CCCC2(C1)CC2(F)F c1(OCC)cccc(NCCC(C(C)C)NC(c2cnc[nH]2)=O)c1[N+](=O)[O-] N1(C(C(C)(C)C#N)=O)CC2CC1CC2NC(=O)CNC(c1cccs1)C1CC1 c1(C(=O)NC(CC=C)CNC(c2cc(OC)n[nH]2)=O)cc(O)ccc1OC(F)F C(C(F)(F)C(C)(C)O)NC(C1(CNC(CCC2N(C)CCC2)=O)CC12CCC2)=O c1(CN2CCC(O)(C(=O)Nc3c(C(=O)O)cc[nH]3)C2)cccc(F)c1Br C1(C(=O)OCC)CC(C)(C)CN1C(c1nccc(Cl)c1C)C(=O)NC1(C)CC1 N1(C(c2sccc2Cl)=O)CC(CO)C2(C1)CN(C(c1csc(O)n1)=O)C2 C(=O)(C(CCC)S(N)(=O)=O)N1CC(OC)CC(NC(C=CC=CC)=O)C1 Cc1ccccc1C(=O)NCC(N1CCN(C(=O)CC23CCC(CC2)C3)CC1)=O CC1CN(C(c2cc[nH]c(=N)c2)=O)CCC1NC(c1nccnc1Cl)=O Cc1csc2ncc(C(=O)NCCC3CCCN3C(=O)Cc3cccc(N)c3)n12 C12(NC(CSCC)=O)COCCC1CN(C(c1cnoc1C1CCC1)=O)C2 c1(C(C(=O)N(CC(C)O)CCNC(CC(=O)OC)=O)C)cc2ccccc2o1 N1(C(C2(NC(c3ccn(CC)n3)=O)CC2)=O)CC(CNC(=O)COC(C)=O)CC1C c1(C(N2CCCN(C(C(C)C3CC3)=O)C(C)C2)=O)cc2c(n1C)CCOC2 C1(CC(=O)NCC2CC(NC(=O)CCn3cccn3)C2)CCCCCO1 C(=O)(C1=C(C#N)CCC1)NC(C(=O)N(C)Cc1ccoc1)CCF N1(C(c2c(C)noc2N)=O)C2CCC1CC(NC(C1CCC3(CCC3)CC1)=O)C2 N#CC1(C(N2CCC(F)(CNC(c3cncn3C3CC3)=O)C2)=O)CC2(CC2)C1 Cc1cc(NC(=O)CCC2CCN(C(C3CC3C#N)=O)C2)cc(C)c1C Nc1ccnc(C(N2C3CCC2C(NC(=O)Cn2nccn2)C3)=O)c1Cl Cc1nc2c(C(=O)NC3CC3CNC(c3ccc(C)c(C#N)c3)=O)ccnc2[nH]1 CC1=NOC(=O)C1CC(=O)NC1CCC1NC(c1ccncc1OCC(F)(F)F)=O c1(C(=O)NC(CCN(C)C(C2CCC3CC23)=O)C(C)(C)C)cc(Cl)ccc1CO N1(C(c2cnc(CC)nc2)=O)CCC2(CCCN2C(C2OCCC2(C)C)=O)C1 CC(C)C(O)C(=O)NCC12CC1CN(C(c1ccc(CO)cn1)=O)C2 C1(C(=O)NCC2CCCN(C(=O)Cn3cncn3)CC2)Cc2cccc(F)c2O1 C1(CCNC(CC=CCC)=O)CC(F)(F)CN1C(C1CC2OC1C1CC21)=O CC(C(O)C(F)F)NC(=O)CC1CCN(C(=O)C#CC2CC2)C1 N1(C(CN(C2CCC2)C)=O)CCCCCCC1C(N1CC=CC1CF)=O c1(C(N2CC(NC(C(CC)(C)CO)=O)C(O)CC2)=O)c[nH]c2cc(F)c(F)cc12 C12(C(N3CC(=C(CNC(C(n4ncc(C)c4)C)=O)F)C3)=O)CCCC(CO1)C2 Cc1ccn(CC(=O)NC2(CCCCNC(C3CCOC3C(F)(F)F)=O)CC2)n1 CCC(CC(=O)N(CCN(C)C(C1(O)CC(F)(F)C1)=O)C(C)C)C(C)(C)C c1(C(=O)NCC(CC)NC(C(C2CCC2)OCC)=O)oc(Br)cc1C CC1(CNC(=O)C(CC#N)NC(N)=O)CCCN(C(=O)CC23COCC(C2)C3)C1 C1(O)(C(N2CC(F)(CNC(CNS(NC)(=O)=O)=O)C2)=O)CN2CCC1CC2 c1(C(COC(c2cc(NC)n(C)n2)=O)=O)cccc(F)c1Br c1(OCC(=O)NC2CCC(CNC(CCSCCC)=O)C2)ccc(F)nc1 C(C)(C)(CC(=O)NCC(C)(O)CSC)NC(C(CC)SC)=O C1(NC(c2ncc(CC)s2)=O)CCC(C)N(C(=O)CN2CCCS2(=O)=O)C1 C1(CNC(CC(=C)C)=O)CC2(CO1)CN(C(=O)CC1CCC13CCC3)C2 C1(CNC(C(Cc2cc[nH]n2)NC(=O)C=CC(F)(F)F)=O)C2CCCCC12 c1(N2CCC(NCC(C(C)C)NC(=O)C3=CCOC3)C2)ncccc1C(F)(F)F N1(C(COCCCOC)=O)CCCC12CCCN(C(c1cc(C)oc1C)=O)C2 c1(OCC)nc(NC(C)(CNC(C2C(C)OC(C)C2C)=O)C2CC2)ncc1C N1(C(C2(COCC)CC(=C)C2)=O)CCCCC1c1nn[nH]n1 c1(C(=O)NCCOC2CCN(C(CC=CCC)=O)C2)cc2ncccc2cc1Cl N1(C(C(c2ccco2)NC(CCC2(C#N)CCC2)=O)=O)CCC2CCCC12 Cn1cc(C(F)(F)C(=O)NC2CCC2NC(=O)CC2CC=CC2)cn1 C#CCC(CC#C)C(=O)NC1CN(C(=O)C(n2ccc(C)n2)C)CC1C1CC1 C1(C(=O)NCC(C)NC(c2c(C)noc2C(C)C)=O)CC(c2ccncc2)=NO1 c1(C(N2C(C3CCN(C(CCc4cc(C)no4)=O)C3)CCC2)=O)c[nH]c(=O)cn1 C1(CNC(C(=O)NCCCC(C)=O)=O)CCC(F)(F)CO1 Cc1cc(N)c(C(N2CCN(C(=O)Cn3cnnc3O)CC2C(F)F)=O)cc1C C1(NC(c2ccc(SC)o2)=O)CC(F)CN(C(=O)CC2CC2(Cl)Cl)C1 C1(NCCn2cc(C(=O)NCC3CC(C(C)C)C3)nc2)CC(=O)N(C)C1 C(CC1CCC1)(C(=O)NC1CCC2CC12)NC(C(C)=C1CCC1)=O c1(OC)ccc(-c2nc(-c3ccccc3CCCC)no2)cc1.N1(C(c2ccc(Cl)cc2)=O)CCN(c2ccccc2)CC1 n1(CC)ccnc1C(=O)N(CCC(=O)NCC(Cl)C(C)(F)F)C1CC1 C1(C(CC)NCc2cncn2C(C)C)Cc2ccccc2C1 C1(NC(c2c(C)cc(F)c(Cl)c2)=O)CC1C1CCN(C(=O)Cc2cnc[nH]2)CC1 C(=O)(C#CC1CCCOC1)NC1(CO)CCN(C(c2nn(C)c(Cl)c2)=O)CC1 N1(C(C2CC(OC)C2)=O)CCN(C(=O)C(C)C(=O)N2CCCC2)C(C)C1 N1(C(=O)C=Cc2cccs2)CC2CCN(C(C3COC4(CO)CC3C4)=O)C2C1 C1(C(=O)NCC(CC)O)C2CCCC2CN1C(C1CCC1C)=O CC(C)C(C)CC(=O)NCC(C)C(=O)N1CCCC1 C1(CC(=O)N(CCC)CCNC(c2ccc(CN(C)C)o2)=O)CCOCC1 C1(C(N2C(CC#C)CCCC2)=O)CN(C(=O)CC2CCOC2(C)C)CCC1(C)C N1(C(c2oc(C)c(CO)c2)=O)CCN(C(C2OCCC2C(F)(F)F)=O)CC1C CCC(CC(=O)N(C1CCN(C(c2ccn3nnnc3c2)=O)C1)CC)C(F)F c1(C(N(CCCCNC(Cn2c(C)cc(C(F)F)n2)=O)C)=O)ccc(Cl)cc1N Cc1cc(C(C)C)nc(=NCC(CC(C)C)NC(=O)CN2CCCCCC2)[nH]1 c1(OC)ccccc1OCC(=O)NC1CCN(C(c2ccnnc2Cl)=O)C1 c1(CCC(=O)N(c2cccnc2)C2CCCC2)nc2cnccc2[nH]1 N1(c2nccc(OC)n2)CCCC(C2(NC(C3CCCC4(CC4)C3)=O)CC2)C1 C1(CNC(C2(NC(C3C=C(C)CS3)=O)CC2C)=O)CC12CCOCC2 Cn1cc(-c2cc(C(=O)NCC3CCCC3NC(=O)CSC(F)F)on2)cn1 N1(C(=O)CCc2ccccn2)CCOC2(CCN(C(=O)Cn3ccnn3)C2)C1 C1(NC(c2c(CC)nc(=N)[nH]c2)=O)COC2(C1)CN(C(=O)C1=C(Cl)CCCC1)C2 CCCC(C)C(=O)NC1(C)CN(C(C23CCC2C3)=O)C1 N1(C(C(C)n2cccn2)=O)CCC=CC1C(=O)Nc1cnc(N(C)C)nc1 N1(C(c2cn(CCC=C)nn2)=O)CCC2(CC1)CC(C)N(C(=O)CO)C2 Cc1cccnc1C(=O)NCCC(C(C)C)NC(c1ncnn1C)=O CC1CC(C)N(C(c2cnc(O)n(C)c2=O)=O)CCN1C(c1c[nH]c(=N)o1)=O C(CC(C)C)(CS(=O)(=O)N1CCOCC1CC1CCCO1)OC CCCCCCCN(C)C(C1(CNC(=O)CC2CC3(CC3)CO2)CC2(CC2)C1)=O c1(OC)ccc(C(N2CC(N(C(=O)CCC3CCCO3)C)C2)=O)c(F)c1 N1(C(CC(C)C)=O)CCCC(NC(c2cccc3ccsc23)=O)CCC1 c1(C(N2CCOC(c3nc(C(=O)OC)cs3)C2)C(=O)NCC)cccc(CC)c1 c1(C(N2CCC(N(C(C(CCCCC)O)=O)C)C2)=O)cnc2ccccc2c1 N1(C(C2CC23CCC3)=O)CC(CO)C2(C1)CN(C(c1ccccc1CCBr)=O)C2 C1(CC)CCN(C(c2ccc(Cl)s2)=O)C(C(=O)NCCOCCN=[N+]=[N-])C1 Cc1cnn(CC(=O)NCC2CN(C(c3cnc(C(F)(F)F)s3)=O)C2)c1 c1(C(N2C(CN(C(=O)Cc3ccoc3)C)CCC2)=O)cnccc1Br C1(CCC(=O)NCC2(C)C(C)(C)C2)CCCCN(C(=O)Cc2cccs2)C1 N1(C(C=NOC)=O)CCC(C)(C)C(NC(=O)C(C)Oc2ccc(Br)cc2)C1 N1(C(C2(COC)CC2)=O)CCC(C2CCCN(C(=O)Cc3sccc3C)C2)C1 C1(CNC(C(F)=C(C)C)=O)CCN(C(=O)CCn2ccc(C)n2)CC1CO c1(CC(=O)NCC2(F)CCCN(C(c3c(C)c[nH]c3)=O)C2)ccc2ncsc2c1 n1(CC(=O)NCC(N(C(=O)CC2CC2)C)C2CC2)ncnn1 CN1N=C(CC(=O)N2CCCC(NC(C3(n4nccn4)CC3)=O)C(F)C2)CC1=O C1(CC(=O)NC(C(=O)OC)C2CCC2)CN(C(=O)CC2CCCN2C)CCO1 c1(OC)ccc(CN=C(NCC2(C)COC(=O)N2)NC2CC(C)(CC)C2)cc1 N1(C(=O)NC2CC3CC(Cc4ccccc4)C2C3)CCC2(CCCNC2=O)CC1 C(CN=C(NCc1ccc(C)n1C)NC1CCCC(F)(F)C1)SC Cc1nn(-c2ccccc2)cc1CNC1CCOC1C c1(C(N2CCC3(C(NC(C4CC(=C)C4)=O)C3)CC2)=O)ccc(N)c2ccncc12 c1(C(=O)NC2C(C)CCN(C(=O)C(C)(C)C)C2)cc(F)cc2c1C(=O)CC2 N1(C(C2CCC(CC)O2)=O)CCC(C2CCN(C(=O)CC(C)(C)O)CC2)C1 CCC(CC)C(F)C(=O)NCC1CC(COC)CN1C(=O)Cc1cccnc1O C(CC1=CCN(C(C2CN(C)CC2C)=O)CC1)NC(C(C)(C)OC)=O CC1C(NC(c2cn(CC(F)F)cn2)=O)CCN1C(C1CCOCC1)=O N1(C(C(CC)(F)F)=O)CCC2(CC1)CN(C(C1CCCC(C(C)(C)C)CC1)=O)C2 c1(C(N(C(CC(=O)N(CC#C)CCF)CC)C2CC2)=O)c[nH]c2cnccc12 S(=O)(=O)(c1ccc(N2CCN(C)CCC(C)C2)c(Br)c1)NC1CCC(CC)CC1 C1(O)(CC(N2CC=CC2CNC(=O)C(N2CCCC2)C2CCCC2)=O)CCCC1 Nc1c(C(N2CCC(CNC(C3(C(N)=O)CC3)=O)C2)=O)sc2ccccc12 C1(C(N(CC(CC)NC(=O)Cc2c(C)cnn2C)C)=O)CC(C)CC(=O)N1 C1(N(C(=O)COc2ccn(C)n2)C)CCCCC1NC(c1nc(C2CC2)cs1)=O c1(C(=O)NC(C(=O)NC2CC(OC)C2)Cc2ccccc2)cc(F)ccc1O N1(C(C(=O)NCC2C(C)CCS2)=O)CCn2ncnc2C1 c1(C(=O)NC(C2CN(C(=O)CN3CCCC3=O)C2)C)cc(-c2ccccc2)cs1 O=C1CCC(CNC(=O)CCNC(=O)CN(C2CCCC2)C)CN1 c1(CC)cccc(C(N2CCCC2COc2ncccc2Cl)=O)n1 C1(NC(=O)CCSC(F)(F)F)CC12CC(NC(c1c[nH]nc1F)=O)C2 N1(C(c2ccn(C)n2)=O)CC2C3CCC(C2C1)N(C(c1ccc(S)cc1)=O)C3 C1(C(=O)NCC2C(CNC(C(OCC)OCC)=O)C2)(CF)CC(F)(F)C1 [N-]=[N+]=Nc1cc(NC(N2CCS(=O)(=O)C(CO)C2)=O)ccn1 N1(C(COCCOCC)=O)CCN(C(=O)C(c2cnn(C)c2)C)C(CC)C1 C1(CC(=O)NC(C)CNC(=O)Cc2nc(=N)[nH][nH]2)CCCCC1F c1(C(CNC(=O)CC#N)N(C)C(C2(CF)CCC2)=O)ccc2ccccc2c1 C(=O)(CCCS(C)(=O)=O)NCC(C)(CNC(C1CCCCS1)=O)OC O=C1CCc2nc(N3CC4CCC3C(NC(C3CCCC5(CC5)C3)=O)C4)ccc21 C(C(C)C(=O)NCC1CCC(=O)O1)N(C(C1CC(C(=O)OC)C1)=O)C C=CCCC(CC(C)C)C(=O)NC1(CCNC(C2CCN(CC(C)C)C2)=O)CC1 C12(C(=O)NCCCOC(N(C)C)=O)CCCC1NCC2 C(=O)(C1CNC(=O)c2ccnn21)N1CCC(CNC(=O)Cc2ccsn2)CC1 Cc1ncc(Cl)cc1C(=O)NCC(F)CNC(c1cnn(-c2ccncc2)c1)=O N1(CCNC(C(n2ccc(C)n2)C)=O)CCN(C(C2(n3cncn3)CC2)=O)CC1 c1(C(=O)NC(C2(O)CN(C(C3CCCC(C)C3)=O)C2)C)cnc2c(c1)CCCO2 C1(C#N)(C(=O)NCc2ccc(C)cc2)CC12CCCC2 c1(OC)cccc(SCC(N2CCOCC2CN(C)C(C2CCCOC2)=O)=O)c1 c1(C(=O)NC2(COC)CCN(C(=O)CCOC(C)C)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NC2(C)CCN(C(CC=CC=C)=O)C2)cc2c(Br)cccn2n1 c1(CSc2cccc(Cl)c2)cccc(I)c1.n12cc(nn1)CN(C)C(=O)C2 c1(OC(C(=O)N(CCN(C(C=CC(CC)=CC)=O)C)C)C)ccc(Cl)c(C)c1 CCC(CC)(CCOC)C(=O)N1CCC1CNC(c1ncc2[nH]ncc2n1)=O N1(C(=O)Cc2ccoc2)CC(NC(C2(C(F)(F)F)CCCC2)=O)C2CCCCC12 CC1=C(C(=O)NC2CC2NC(C2(CC3CC3)CCCC2)=O)C(C)(C)CCC1 C1(CC(N2CCC(N(C(=O)Cc3nnc(C)o3)CC)C2)=O)OCCOC1(C)C CCCC(C)CC(=O)N1CC2CC2C1CNC(=O)Cc1ccccc1OCC c1(C(=O)NC(CCCC)CNC(=O)C#CC2CC2)cnc(OCC(F)F)c(Cl)c1 c1(NC(C2N(C(c3n(C)ncc3Br)=O)CC(F)C2)=O)nc(Br)cn2ccnc12 N1(C(c2c(C)[nH]cc2)=O)CCc2ccccc2C(NC(=O)C2=CC3CCC2C3)C1 Nc1[nH]c(=NCCn2ccnc2-c2ccccc2)[nH]c2ncnc1-2 C1(CNC(NC(CC)CC)=NCC2CCC3(CCC3)OC2)CC2(CO1)CC(F)(F)C2 C1(CNC(C2CC(SC)C2)=O)CC2CCCCC2N1C(C1CNC(=O)C1)=O C(CN=c1nc(C)c([N+](=O)[O-])c[nH]1)NC(C1(C)C(CC)CCC1)=O c1(C(N2CCCCC(CO)C2)=O)cn2ccccc2n1 c1(C(c2n(CC)nnn2)NCCc2cc(C)no2)cncc(C(F)(F)F)c1 c1(OC)cc(C(=O)NCC(CO)NC(C2(C)CCCNC2=O)=O)cc(Cl)c1 CN1CCN(C(c2cccnc2N)=O)CC1CNC(=O)C#CC1(C)CC1 CCCC(C)(C)C(=O)N1CCCCC(CNC(=O)CC2CCCN2C)C1 c1(OC)nc(N2CCOC(CNC(c3sccc3CC(C)(C)O)=O)C2)cc(C)n1 CCCC(CCCO)C(=O)N1CCC2(NC(C3CCC(C)O3)=O)CCCC12 n1(CC(=O)N(CC(C)C)CC(=O)N(C)CCN(C)C)ncnn1 c1(NC(C2CN(C(c3cc(Br)ccc3F)=O)CCS2)=O)c[nH]c2ncc(Br)cc12 c1(NC(CN(C2CCCN(C(=O)C(C)(C)C)C2)C)=O)ccc(N(C)S(N)(=O)=O)cc1 N1(C(c2cnc(Cl)s2)=O)CC2CC(C1)N2C(c1cnn2ccsc12)=O c1(C(=O)NCCC2CCC(NC(C(CSC)(C)C)=O)C2)n[nH]c2c(C)cccc12 C1(C(=O)OC(C)(C)C)CC(C)(C)CCN1C(C1CC(S(N)(=O)=O)C1)=O N1(C(C2CN(C)C(=O)N2)=O)CCC2(CCN(C(C3CC(Cl)(Cl)C3)=O)C2)C1 C1(C(=O)NC2C(NC(CSCC#C)=O)CCC2)CCCCN(C)C1=O CN1CCC(C)(C(N2CC(CCCCNC(=O)C(F)CC3CC3)C2)=O)C1=O N1(C(C2CC(C)(NC(C3CC4C=CC3O4)=O)C2)=O)CCCN2CCCC2C1 C(CCC1CCC1)(C(=O)NCCCSC)N(c1cccc(C)n1)C(C#C)C Cc1ccc(S(=O)(=O)N(c2ccc(O)cc2)C(C2CCCC2)=O)cc1C Cc1[nH]c(C#N)cc1C(=O)NC(C)CCC(=O)NCCCc1cc[nH]n1 CCC(C)CC(=O)NC1CC(C)CN1CC(=O)Nc1nnc(-c2ccccc2)o1 N1(C(C=CC(CC)C)=O)CCCC(O)(CNC(c2ccsc2)=O)CC1 c1(C(N2CCC(F)(CNC(c3c(C)cco3)=O)CC2)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(CCS(=O)(=O)c1ccccc1)NC1(CNC(C2(C)CC(C#N)C2)=O)CCC1 C=C(C)C1OCCCC1C(=O)NCC1CN(C(c2cnsc2C)=O)CCC1(C)C Cc1oncc1C(=O)NCC(=O)NC1CC1CNC(C1CCNC1=O)=O c1(C(=O)NCCCCCN(C(c2c(C)coc2C)=O)C)ccn2cnnc2c1 C1(CC(=O)NCCOC)CCCN1C(c1ccsc1Cl)=O c1(C(N2CCC(N(C)C)(CC)C2)C(=O)NC(CC)C)cc(Cl)ncc1Cl c1(CN(C(=O)CCn2cc(-c3ccsc3)nn2)C)cccnc1Cl Cc1cc(Br)cc2cc(C(N3CCCC3CNC(C3(N(C)C)CC3)=O)=O)oc12 CCN=c1[nH]cc(C(=O)N(C)CC2CCN(C(C3CC3F)=O)C2)s1 Cc1coc(C)c1C(N1CCN(CCCNC(c2ccc(C(F)F)o2)=O)CC1)=O C(C(C)(O)CNC(c1csnc1C(F)F)=O)NC(C(c1ccccc1)C)=O CCC(F)(F)CC(=O)NCCCNC(C1COCC1C(F)(F)F)=O C1(CNC(=NCC)NCCN2CCOCC2)CCC2(CCC2)C1O N1(CCc2cn(CC(N3CCC(c4nc[nH]n4)C3)=O)nn2)CCC(F)(F)CC1 Cc1cc(Cl)c(C(N2CC(NC(c3coc(C(F)F)n3)=O)CC2C)=O)cn1 c1(OC)ccc(C=CC(=O)NC2CN(C(=O)C(C)CC3CCC3)CC2O)cc1F c1(C(N(C)CC2CCN(C(C3(C)C(C(=O)OC)C3)=O)C2)=O)scc2c1CCCC2 C1(CNC(c2n[nH]c(C)c2O)=O)CC2(C1)CN(C(=O)CCCc1ccccn1)C2 c1(CNC(=O)CONC(=O)c2ccsc2)nccc2[nH]ccc12 OCCC(N=c1nc2scnc2c(N2CC3CCC3C2)[nH]1)c1cccnc1 c1(OC)ccc(CN2CC3C(C(N4CC(C)CCC4C)=O)C3C2)c(Cl)n1 Cc1nnccc1C(=O)NCC(C(=O)NC1COC(C)(C)C1)N(C)C C1(NC(c2ccc(F)c(F)c2)=O)CC2CC1CN(C(=O)C(F)(F)CO)C2 C#CCC(CC(=O)N1CCCCC1CCCO)NC(=O)CCc1ccsc1 N1(C(c2c(C)ocn2)=O)CC2CCC2(NC(=O)Cc2ccc(OCC#N)cc2)C1 CC1NC(=O)CCC1CNC(=O)C(N1CCC(Cc2nccs2)C1)=O c1(C(=O)NCC(CN(C(C(CC)C#N)=O)C)C)ncn2cc(Br)sc12 c1(C(N2CCC(C)(NC(C(C)CSC(F)(F)F)=O)C2)=O)cccc2c1ccn2C N1(C(c2c(CC)cno2)=O)CCC2(CCN(C(C3CCCC(O)C3)=O)CC2)C1 C1(C(=O)NC(C)C(C)NC(=O)Cc2csc(CCn3cncn3)n2)CC=CCO1 C(CCCCCNC(=O)C=CCCC(C)C)NC(Cc1c(C)ocn1)=O CC1COCC(C(=O)NCCn2cc(CNC(=O)CCN(C)C)nn2)O1 c1(N(CCNC(=O)C2CC2)CC)cc(Cl)nc(C(C)(C)C)n1 c1(C(CC(=O)NC2(C)CN(C(Cc3ccc(C)s3)=O)C2)C)c(C)noc1C Cc1n[nH]c2cc(C(=O)NCC3CN(C(C4CCCCO4)=O)CCN3C)ncc12 N1(C(c2c(C(C)(C)C)cccc2)=O)CCC(NC(C2CC3CCC2O3)=O)C12CC2 c1(C(=O)NC(CCOC)CNC(C23CC(C#N)(C2)C3)=O)ccc(F)c(O)c1 C1(N(C)C(=O)OC(C)(C)C)CC2CC1N(NC(C1CCC(C(F)F)CC1)=O)C2 N1(C(C(=O)NC2(C)CCCO2)=O)CCn2ncc(S(C)(=O)=O)c2C1 C1(CCC2N(C(=O)OCC)CCC2)CCCCC1CC c1(OC)ccc(-c2nc(CCNC(=O)C(N3CCCCCC3)=O)cs2)cc1 C1(CNC(CCc2ncc(C)[nH]2)=O)CN(C(c2cnc(CC3CC3)s2)=O)CC12CC2 C1(CC(N2CCCC(OCC#C)C2)=O)CC(C)(C)CN1C(=O)CCc1cnco1 N1(C(c2cccc(-n3cccn3)n2)=O)CC2CCC1CN2CCn1ccnn1 CC1OC2(C(=O)NCC3CC(NC(=O)Cc4csc(NC=O)n4)CCO3)CC1C2 C(=O)(C(C(C)C)C(C)C)N1CCC(C(C)NC(CCc2cc(C)nn2C)=O)CC1 N1(C(c2c(OC)scc2)=O)CCCC(NC(=O)CCC(=O)NC2CCCC2)C1C c1(C(N2CCC(N(C(=O)Cc3nc[nH]n3)CC)C2)=O)ccc(S(=O)(=O)CC#N)cc1 c1(C(=O)OCC)cc(Br)c(C)cc1NC(C1CC(=O)N(CCOC)C1)=O C1(CC(=O)NC)CN(C(C2CCC(F)C2)=O)CCN1C(=O)CCS(C)(=O)=O C1(CNC(C(C)OCC)=O)CCCC2(CN(C(=O)CCc3cncs3)C2)O1 C1(CNC(=O)C(O)C(F)F)CN(C(=O)C=C(Cl)Cl)CCC12CCOCC2 C1(CC)CN(CC)CC1C.C1CC(=O)NC(C2CC2)C(=O)N1CC C=C1CC(C(=O)NCc2cscn2)(CNC(c2cnn(C(C)C)c2)=O)C1 c1(CC(=O)NCC(CN(C(=O)C2=C(C)CCC2)CC)(C)C)cnn2c1CCCC2 S(=O)(=O)(c1cc(C(=O)NCC2CCN2C(C2(C)CC=CC2)=O)ccc1OC)NC Cc1cnc2c(C(N3CCN(C(C4CC=CCO4)=O)CC3CF)=O)cnn2c1 Cc1nc2cc(C(=O)NCC(C3CCC(F)(F)CC3)C)cnc2[nH]1 CC1(C)C2CCC1(C(=O)O)C(NC(c1c[nH]nc1Cl)=O)C2 CC1CCOC(C(=O)NCC=CC(=O)N(C2CC2)Cc2nc[nH]n2)C1 C1(NC(c2c(C)nns2)=O)CC12CCN(C(=O)CC(=O)N(C)C)C2 CC(C(=O)NC(C)CC1CN(C(c2cccc(CF)c2)=O)C1)C(C)O c1(C(=O)OCCC(N2CCC(CCOCC)C2)=O)ccc(F)cc1 Cc1ncccc1CC(=O)NCCCC1CCCN1C(=O)C(C)C1(O)CCC1 C1(NC(C=CC=CC)=O)CN(C(c2ccc(Br)c(F)c2)=O)C2(CCOC2)C1 C=CC1(CC(=O)NCC(C)(CC)OC)CN(C(=O)C=CC2CCOC2)C1 O=C(C1=NOC2(CCN(c3ncncc3I)C2)C1)Nc1cc(Br)c(F)cc1[N+](=O)[O-] n1(CC)nnc(C)c1CNC(=O)C(C)(C1CC1)N(C(=O)CC1CC1(C)C)C Cc1noc(C)c1S(=O)(=O)N1CCCC1.C1(N)CC2CN(C(=O)CCCF)CC2C1 C(=O)(C#CC1(CC)COC1)N1CCC(NC(c2c(Cl)cn(CCC)n2)=O)C1 c1(C(N2CC(NC(C=CC(=O)OCC)=O)C3C(C2)C3)=O)csc(S(N)(=O)=O)c1 Cc1cccc2c1OC(C(=O)NCC(O)CNC(C1CCC(N=[N+]=[N-])C1)=O)C2 Fc1ccc(-n2ccnc2-c2cc(Br)cc(Cl)c2)cc1-c1ccc(F)cc1F N1(C(=O)CN2CCC2)CC2(C1)CN(C(c1cc(O)ccc1[N+](=O)[O-])=O)CC2CO Cc1ccc(CCC(=O)NC2CC2CNC(C2(F)CC2)=O)o1 C1(CN(c2ccccc2F)C(=O)C(C2CCOCC2)F)COC2(CCNCC2)C1 c1(COC)cccc(CC(=O)N(CCCNC(C2CC2C(C)(C)C)=O)C)c1 N1(C(c2c(OCC)ccc(C)n2)=O)CCC2CC2(NC(=O)Cn2cccn2)CC1 C1(CNC(c2cnc(OC)s2)=O)CCN(C(C2(C)CNC(=O)N2)=O)CC1O C1(CC)(NC(=O)C(C)S(N)(=O)=O)CCN(C(=O)CCc2nc(C)cs2)CC1 c1(OC)ccc(CCC(N2CCOC(C(C)NC(=O)COCCCF)C2)=O)cc1 c1(C(=O)NCCC(C(=O)N(CC(O)CO)C)OC)ccc(O)c(F)c1 C(C(C)C)(C(C(=O)Nc1cccc(Cl)c1C)N1CCCC1C(C)(C)OC)OC c1(-c2scc(C(C)NC(=O)NC3CCC(C4CCNCC4)N3)n2)ccc(Cl)cc1 CCCCC(C(=O)N1CCC1C(C)O)NC(c1cccc(F)c1O)=O C(=O)(C(C)(O)CCC)NC1CN(C(C(C(=O)OCC)F)=O)C(CO)C1 C(CC(=O)N1CCSCC1C1CC1)(C(F)F)NC(=O)COC1CCC1 C(C1CCOCC1)=CC(=O)NCCC(F)(F)Cn1cc(C(C2CC2)C2CC2)nn1 c1(C(CNC(NC(c2ccc(Cl)cc2)CF)=NCC2CCC2)F)cccc(F)c1 CN1CCN(C(=O)CCc2cscn2)C(C(=O)NC2CN3CCCC2C3)C1 C(=O)(C(O)C(C)CC)NCCCN(C(c1c(OCC#C)nccc1)=O)CCO Cn1cncc1C(=O)C(=O)NCCCCCNC(=O)CC1(C2CC2)CC1 c1(OC)cncc(C=CC(=O)NC2CC2(C)C(C)C)c1 CC1(CNC(C2SC3C=CC2CC3)=O)CCN(C(C2CCOCC2)=O)CC1 Nc1c(F)ccc(Cl)c1C(=O)NC1CCN(C(=O)Cn2cnnc2O)CC1 CCCC(C(=O)NCC1CCCN1C(=O)C(c1ccc(F)cc1)F)NC(N)=O c1(COC)cccnc1C(N1CCCC1CN(C)C(c1cn(C2CC2)nn1)=O)=O C1(NC(c2c(COC)cc[nH]2)=O)CN(C(c2cc(C)c(C)nn2)=O)C(C)(C)C1 N1(C(c2c(C)cccc2Br)=O)CCN(C(C2CC(C)C2)=O)C2(CCC2)C1 C1(CC=C)(NC(=O)Cc2cc(C)no2)CCN(C(C2CNC(=O)N2C)=O)CC1 c1(C(N(C2CCN(C(CCCCSC)=O)CC2)CCO)=O)cc(C#N)c(O)nc1N CC1CC(NC(c2cnncc2O)=O)CN1C(=O)CC1CCC2CC12 c1(C(=O)O)cc2ncc(CN3CC4CC4C3CO)cc2[nH]1 C1(NC(Cc2n(C)ccc2)=O)CCC2(CCN(C(C3(C)C=CCCC3)=O)C2)C1 c1(OC)nc(Br)ccc1S(=O)(=O)NC1CCCc2c1cnn2C(C)(C)C c1(-c2ccc(CNCc3c(OC)csc3)cn2)ccc(Br)c(C)c1 C=CC1(CC(=O)NC2CCCN(C(=O)CCC=CC)C2C)CCOCC1 C(=O)(C(CCC(N)=O)N(C)C)NCCC(C)CCNC(C1CC1c1cccs1)=O C(=O)(C(C)CC(N)=O)N1CC(c2oc(C)c(NC(C3CCC(N(C)C)C3)=O)n2)C1 c1(C(N2CC(CNC(C(CC(C)C)O)=O)OCC2)=O)cc(O)nc2ncn(C)c12 c1(-c2cccc(OC)c2C)cccc2c(C(=O)NCc3noc(CO)n3)n[nH]c12 C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C(CN(CC(C)(C)C)C)=O)C(CO)C1 C#Cc1cccc(CC(N2CCOC(C3CC3)C2)=O)c1.C1(CC(C)C)C(=O)N1C c1(OC)cc(CN2CCOCC2C(C)N=c2ccnc[nH]2)c(OC)cc1C c1(C(C)C)ccc(C(=O)N(C)CC2CN(C(C3COC(=O)C3)=O)CCO2)c(F)c1 c1(C(=O)NC2C(C(N3CCC(C(=O)NC)C3)=O)CC2)cccc2c1CCC2 N1(C(Cc2n(C)nnc2)=O)CCC(C)(C)CC1C(N1CC(CC(N)=O)C1)=O CC(C)(O)C(F)C(=O)NCC1(F)CC(NC(C2CC3CCC(C2)O3)=O)C1 C(=O)(C(C#N)C1CC1)NC(C1CCCN1C(=O)CSS(C)(=O)=O)C C#Cc1cc(C(=O)NC2(C)CCN(C(=O)COCc3nc[nH]n3)CC2)cc(F)c1 C1(C(=O)NCCc2ccc(CC)cc2)CCCCN(C(C2CCCN(C)C2)=O)C1 N1(C(C(CCOC)(C)C)=O)CCC2(CC1)COC(CNC(=O)C(F)(F)CSC)C2 Cc1nc(C2CC2)sc1CC(=O)NCCCC(C)(C)NC(C1CC2(CSC2)C1)=O c1(C(N2CC(CCCNC(C=CC)=O)OCC2)=O)ccc2oc(C)nc2c1 c1(NC(C2CC2C(=O)Nc2ccnn2-c2ccccc2)=O)ncccc1OC(F)F C1(CCNC(CCCOCCC)=O)CCCN(C(=O)CCC2CC(F)(F)C2)CC1 C1(NC(c2c(C)snc2)=O)CCC2(CC1)CN(C(c1ccc(CF)cc1)=O)C2 N1(C(c2cccc(OC)c2)C(=O)NC(CC)C)CC(C)(C)OCC1CC(=O)OC CC(O)(CC(=O)N1CCC(NC(=O)CCn2ccnc2)CC(O)C1)C(F)(F)F Cn1nc(CC(N2CCCC2C2(C(=O)NC3C(O)CC3O)CC2)=O)cc1Cl C1(C(C)NC(c2cc(CN(CCC)C)on2)=O)CN(C(=O)C=C(C)C)CCO1 C1(O)(CNC(c2c(CCCC)ocn2)=O)CCN(C(=O)C=CC2(C)COC2)CC1 C(C(C)(C(=O)NC1C=CCN(C(C2C=CCS2)=O)C1)OC)OC C(CN=c1[nH]cncc1I)(CC(C)C)NC(c1c2ccc(OC)cn2nc1)=O c1(C(=O)NC(C)(C)C(N2CC3(CCNC3=O)C2)=O)cc2ccccn2c1 c1(OCC)oc(C)nc1C(=O)NC1CCCC1NC(c1ccon1)=O c1(OC)cc(C)c(C(c2nnnn2CCC2(C)CC2)Nc2cn[nH]c2)cn1 N1(C(CC(COC)C)=O)CC2(C(=O)NCc3nc(CO)n[nH]3)CC1CCO2 C(=O)(C1CCOc2ccccc21)NCC1(C)CC(NC(c2cc(C)c(C)s2)=O)C1 c1(OC)cncnc1C(=O)NCCC(=O)NCc1cn[nH]c1 C(=O)(CC(C)(C1CCC1)N(C)C)NC(C)CC(C)NC(=O)C(N1CCOCC1)C Cc1ccc2c(NC(C3CC3NC(c3cc(C)c(Br)cc3C)=O)=O)cccc2n1 N(C1c2ccccc2CCC1C)C(=O)Nc1c(C)n(C(C)C(C)(C)O)nc1 C1(C)(NC(C=C2CCC(C)C2)=O)CCCN(C(=O)C2=COCCC2)C1 Cn1nc2ccccc2c1-c1nc(C2CCC(O)C2)n(C2CC2)n1 CCC(C)(C)C(C(=O)NC1CC(CCNC(c2ccc(F)c(C)c2N)=O)C1)OC C(CC(=O)NCCC(=O)NCCC1(C(=O)NC)CC1)SCC#C c1(CN2C(C(N(C)CCO)=O)CSCC2)cc(Cl)cnc1Br C1(C)(CNC(=O)NC(C(C)c2ccccc2)C#N)CC=CCO1 CCC(CC(=O)N1CC(C)(C)CC1CNC(C1(C)CC1)=O)C(C)(C)C C1(C(=O)OC)CCC(C)(C)N(C(=O)CCc2cn(C(C)CO)nn2)C1 O=C(C1=CCCN(C(C2CC3CC(=O)C2O3)=O)C1)NCCN1CC2CC2C1 N1(C(CC(CCC)C)=O)CC(NC(=O)Cc2c(Cl)c(CC)nn2C)CC2(CC2)C1 Cc1ncc(C(=O)NCC(C(C)(C)C)NC(=O)CN2CC3CC3C2)n1C c1(CNC(=O)C(=O)NCc2ncco2)ccc(C2CCOCC2)cc1 CN1CCC(CN(C(=O)C(CC2CCOCC2)NC(=O)CCC2CCOC2)C)C1 c1(CNC(CC(COC)NC(=O)Cc2cnnn2C)=O)ccc(F)nc1F C(=O)(C1=NN(c2ccc(C)cc2C)C(=O)C1)N(C(=O)CNC)CCC c1(C(c2nnnn2C)NCc2occ(C)c2)cccc(C(C)C)c1 N1(CCC)CCN(C(=O)CCC2CCCN(C(C3CCCS3)=O)C2)CC1 c1(C(=O)NC(CN(C(C(C)=CC)=O)CC)C)c[nH]c2cc([N+](=O)[O-])ccc12 c12ccc3c(c1)CN(C3)C2=O.C1(N(C(C)(C)C)C)CCN(Cc2cccnc2)C1 C(=O)(C(CC(C)(C)C)NC(=O)CCCNC(C)=O)N1C(C(=O)OC)C=CCC1 c1(CN(C(C)C)C)cn(C(C)C(=O)NC2CC(CCO)C2)nn1 c1(N2CCC(C(N(CC=C)OC)=O)CC2)ncnc2c1ncn2CCS N1(C(c2ccc(CC(C)C)nc2)=O)CC(N(C(=O)C=CBr)CCO)C(C)(C)C1 C1(N(C(C(C=C)O)=O)C)CCN(C(c2cc(Cl)cc(Cl)c2F)=O)CC12CC2 N1(C(c2cnc(O)c(F)c2)=O)CC(NC(C2CC(F)C2)=O)CC2(CC2)C1 C(=O)(CS(=O)CCC(F)(F)F)NC1(C2CCN(C(c3ccn(CC)n3)=O)C2)CC1 N1(C(c2c(CC)onc2C)=O)C(CNC(C2CC2(F)F)=O)CC2COCC12 N1(C(c2c(C)ccs2)=O)CC(=O)CC1C(=O)NCC1CCCOCC1 C#CCCCCCC(=O)N1CCCCC1C(C)NC(c1c(C)ncn(C)c1=O)=O C(=O)(C(F)(F)C(O)C(C)C)N1CCC(NC(c2[nH]cc(S(=O)(=O)NC)c2)=O)C1 Cc1c[nH]nc1C(N1CCC1CC(=O)NCC1(N(C)C)CCSC1)=O CCC(CC1CCCC1)C(=O)NCCCOCCCNC(C1CNC(=O)N1C)=O c1(NC(C2N(C(c3n(CC)ccc3)=O)CCC2(C)C)=O)ccc2occc2c1 c1(OCC)cccc(C(C)(C)C(=O)N2CCC(N(C)Cc3ncc(CC)o3)C2)c1 c1(C(=O)OC)ccc(C(=O)OC)c(NCCN2CCOC3(CCSC3)C2)c1Cl CC1(O)CCC(CC(N2CCC(CF)(NC(c3cc4n(n3)CCO4)=O)C2)=O)CC1 c1(C(=O)NC(C2CCN(c3nnc(C(F)F)s3)C2)C)cnc2c(c1)CCCO2 C1(NC2(c3cc(F)cc(F)c3)C(=C)CC2)CC1C1CCN(C(=O)OC(C)(C)C)CC1 N1(C(CCc2c(C)noc2)=O)CCCCC(C(=O)NCCCCN=[N+]=[N-])C1 Cn1nccc1C(C)(C)C(=O)NCCSCc1cn(CC2CCCO2)nn1 N1(C(C2(CC=C)CC2)=O)CCCCC(C(N2CCCC(OCC)C2)=O)C1 C(=O)(C1=COCCC1)NCC(CC(=O)NC1(C)CC(O)C1)OC C(=O)(C(CO)C(C)(C)C)NCCCNC(CC(c1cccs1)NC(C)=O)=O N1(C(c2cc(C)c(Cl)cc2)=O)CCCC2CN(C(=O)C#CC3CC3)CC12 c1(C(=O)O)ccc(CN2CC(C(=O)O)CCC2CO)c(Cl)c1 C1(CNC(=NCC(C)C2CCOCC2)NCCF)CCCOC1(C)C N1(C(CCOC)=O)C(C(=O)NCCn2cc(CO)nn2)CC1C c1(C(N(CCCNC(C2C3CCCC23)=O)C)=O)cccc(S(=O)(=O)C2CC2)c1 c1(C(N2CCC(CN(C(C(CCOC)C)=O)C)C2)=O)ncc2ccccc2c1O CC1(C(N2CCC2CNC(=O)C2=CCCSC2)=O)COC(=O)OC1 N1(C(CCCOCC)=O)CCOC2(CCCN(C(=O)C3=C(CC)OCCS3)C2)C1 C=C1CCN2C(C1)c1nnc2n1CC(N1CCN(C)CC1)CC.C(C)(=O)OC C#CCC(C)(C(=O)N(C)CC1CCCN1CC)NC(C1CCC(=O)N1)=O C1(CNC(C2CC(=O)N(O)C2)=O)CN(C(=O)CCN2CCCC2)CC1(F)F C1(C)(C(N2CCCC(N(C(CCOCCOC)=O)C)C2)=O)CCCCC1(F)F c1(CC(N2C(CNC(=O)CCC3CCOC3)C=CC2)=O)ccc2c[nH]nc2c1 C1(C(c2cn(CCN3CCSCC3)nn2)C(=O)Nc2cccnc2)CCCCO1 N1(C(c2c(C)snn2)=O)CCOC2(CCN(C(C3(C)CCC(F)(F)C3)=O)CC2)C1 N1(CCCCCC#C)CCCc2occc2C1 Cc1ccc(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C2)c([N+](=O)[O-])c1 c1(OC(C2N(C)C(NC(=O)OC(C)(C)C)CC2)=O)cc2oc(O)nc2cc1F C(N=c1[nH]c2c(c(=NC3COC4(CCC4)C3)[nH]1)CSC2)C1(C(C)C)CCOCC1 N1(C(C2C(NCc3ccc(OC)c(I)c3)C2)=O)CC2OCCOC2C1 c1(C(C)=O)cnc2n1CCN(C(c1ccn(C3CC3)c1C)=O)C2 N1(C(CN(C(=O)OCC)C)=O)CCC2(CC2NC(c2cccnc2CC)=O)C1 c1(C(N2CCCCC(N(C(C(CC)C)=O)C)C2)=O)ncc([N+](=O)[O-])n1C Cc1cc(C(N2CC(O)(C3CCCCN3)C2)=O)c(N)s1 c1(CN2CC(NC(c3cnc(C)[nH]3)=O)C(F)C2)cc(Cl)c(C)cc1O N1(C(C#CC2(C)COC2)=O)CCC2(CNC(=O)COC3CCCC3)CCCCC12 c1(C(N(CCNC(=O)C(C)(O)CC(C)C)CC)=O)nccc2ncccc12 N1(C(c2ccc(CC)[nH]2)=O)CCC(O)(C(C)NC(=O)Cn2ccnn2)C1 c1(CC(C)C(=O)NCC(F)CNC(=O)C2=CCSC2)ccccc1Br c1(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CC2)cc(O)c(O)c(O)c1 c1(C(=O)NCC(CC)N(C(c2c(CC)nns2)=O)C)ccc2nc(O)cn2c1 C1(CNC(C2(CCCC)CCCC2)=O)CCN(C(=O)Cn2cnnc2)C12CC2 Cc1coc(C)c1C=CC(=O)NC1CC1NC(=O)Cn1cnc([N+](=O)[O-])c1 C1(CC(=O)OC)CCC2(CCN(C(=O)CC3(CC4CC4c4ccccc4)CC3)C2)C1 N1(C(Cn2c(C)cc(C(F)F)n2)=O)CCCC2(C1)CN(c1nnnn1C)CCO2 Cc1coc(C(N2CCCC2CCNC(=O)CCc2c(C)noc2Cl)=O)c1C c1(C(N2C(CNC(CC(C)C)=O)COC(C)(C)C2)=O)cc2cc(F)c(F)cc2[nH]1 N1(C(c2cnn(CC)c2Cl)=O)CC(NC(=O)COCC(C)C)C2(CCC2)C1 C(=O)CS(=O)(=O)CC(C)C.N1CCC(C)C1Cc1cn(C2C(OC)COC2)nn1 N1(C(C2CCCC23CC3)=O)CC2CC(C1)N(C(C1CCCCS1)=O)C2 CN=c1nc(C(=O)NC2CC(CNC(=O)C(C)(F)F)C23CCC3)cc(C)[nH]1 N1(C(C(Cc2ccco2)NC(c2c(C)c(O)ccc2)=O)=O)CCC(F)(F)C(O)C1 c1(CCC(=O)O)ccc(CNC2CCCCC2n2ccnc2)nc1 C1(CCNC(C2CCCC2O)=O)CC2CCC(C1)N2C(c1cc(CCO)on1)=O c1(C(=O)NC(CNC(Cn2cc(C(=O)NC)nn2)=O)(C)C)cc(C)c(C)s1 c1(C(N(CCN(C(c2cc(C)sc2)=O)C(C)C)C)=O)[nH]ncc1C#N N1(C(CCN(CC)CC)=O)CC(C(N2CC3CCC3(C)C2)=O)CC(C)C1 N1(C(c2c(C)cnnc2)=O)CC(=O)NCC1C(N1CCCC(CC(N)=O)C1)=O C1(C(=O)NCC(=C)CCNC(c2ccc(SC(F)F)cc2)=O)CCC(C)(C)CC1 C(CC1=CCN(C(C2CCN(C)C(=O)C2)=O)CC1)NC(C1(CC)CCNC1=O)=O N1(C(CN(C)C(N)=O)=O)CCC(F)(CNC(c2ncccc2N(C)C)=O)CC1 c1(C(N2CC(CCNC(c3c(C)nsc3)=O)OCC2)=O)cc(C)c(C#N)c(C)c1 C(C)(CCC(=O)NC1(NS(C)(=O)=O)CC=CC1)NC(CC=CC=C)=O C1(CN(C(c2c(C)onc2)=O)C)CCCN(C(c2cccnc2C(F)F)=O)C1 C1(CN(C(C=CCC)=O)C)CCCN(C(=O)C=Cc2cncn2C)C1 N1(C(c2ccc(Cn3cc(CCC(=O)CCO)nn3)o2)=O)CCC2(CCCOC2)C1 N1(C(c2cccc(C)n2)=O)CCC2(CC1)CCN2C(=O)CSC1CCCCO1 Cc1cnn(C)c1S(=O)(=O)NC(CCC(=O)N(C)C)c1ccccc1 N1(C(C(CC)C)=O)CC2OCCN(Cc3cccc(OC4COCCO4)c3)C2C1 CC1C(C(=O)N2CCC3(CCCN3C(=O)C#CC3(C)CC3)C2)=Cc2ccccc21 N1(C(CC(C=C)CC)=O)CCCC2(CCN(C(=O)CCOC)CC2)C1 CC(=O)CC(C)(C)CC(=O)NCC1CC(NC(c2cnoc2)=O)C1 c1(CCN2CCC(CN3C(CC)CCCC3)CC2)oc2ccc(Cl)cc2c1C N12CC3CC(C1)N3C(=O)C1C(CCCC1)OC2=O.CC(C)(C)C(=O)CNC=O O=C(CC(F)(F)Cl)NCCNC(c1ccc(-c2nc[nH]n2)nc1)=O c1(C(=O)NC(C(N2C(CC)CC(O)C2)=O)C2CCCO2)ncn2c1CCC2 CC(C)(CCC#N)C(=O)NCC1CCC(NC(c2ccc(CF)cc2)=O)C1 c1(C(=O)NC(CC)CN(C)C(c2ncccc2OC)=O)cnc(OC)c(Cl)c1 CON(C)C1CN(C(c2nc(CNC(=O)Cc3ccccn3)oc2C)=O)C1 c1(C(N2CCC(CNC(c3cnoc3-c3ccco3)=O)C2)=O)csc2cncn12 C1(CNC(C=CCC)=O)CCN(C(=O)CCc2cncn2C)C12CC2 C1(NC(c2sccc2C(F)F)=O)CN(C(=O)CN2CCOCC2)C2CCCCC12 c1(C(=O)NCC2C(CNC(c3cn(CCC)nn3)=O)C2)ccc(O)c(C(N)=O)c1 N1(C(C=CC(C)NC(C2(C)CCCC2)=O)=O)CCC2(CCCCO2)C1 CC(C)CC(C)CC(=O)NC1(C(=O)NC2CC3CCCC3C2)CCCC1 Cc1ccc(-c2cn(C(C)C(=O)O)nn2)c(Cl)c1.C1=C(C(=O)O)CONC(=O)C1 C1(COC)CCN(C(C2CC(NC(C3CC=CCC3)=O)C(O)C2)=O)C1(C)C C1(CC(C)C)CC(C(N2CCC23CN(C(=O)C2=COCC2)C3)=O)CC(=O)N1 CCCC(C(=O)NCc1c[nH]nc1C(=O)NC1CNC(=O)C1)OCC C1(CN(C(c2n(CC)ncn2)=O)C)CCN(C(=O)C(N2C(=O)CCC2=O)C)CC1 N1(C(C(CCOC)C)=O)CCCCC2(CCN(C(=O)C(=O)NCC(F)F)C2)C1 C#CCCCCCC(=O)NCCC1CC(C(=O)NCC2CCN(C(N)=O)C2)C1 C1(NC(=O)Cc2ccccc2O)CN(C(c2[nH]ccc2C2CC2)=O)C2(CCC2)C1 n1(CC)nnc(-c2nc(-c3ccc(OC)cn3)nn2-c2cnnn2C)c1C CCCC(CCC)C(=O)NC12CCC(NC(C3(C#N)CCCCC3)=O)(CC1)C2 c1(OC)ccn2cc(C(=O)NCCCN(C(c3csc(C)c3)=O)C(C)C)nc2c1 c1(C(=O)NC2CN(C(c3c(COC)cco3)=O)C2)ccc(C(C)(C)OC)cc1 CC1(C#N)CCCN(C(=O)C(=O)NCc2ccc3c(c2)OCC3)C1 c1(NC(=O)NCc2nccc(OC)n2)cc(C)ccc1Br N1(C(CC2CCCC(C)O2)=O)CC2(CCN(C(=O)CN(S(C)(=O)=O)C)CC2)C1 C(=O)(C(C(C)C)NC(c1ncc(F)cn1)=O)NC(C(=O)OCC)C C=CCC(C)(CC=C)NC(=O)C1=CCC(NC(=O)CC(CC)C2CCC2)C1 CC(C)C(CCN(C(=O)CCc1cn[nH]c1)C)NC(c1cn(C)nc1Cl)=O N1(C(C(CC)OCC2CC2)=O)CCOC(C(=O)NOCC(O)C(C)C)C1 c1(C(N2CCC(NC(C3C(C(=O)OC)C3)=O)C(C)C2)=O)cnn2c1NCCC2 c1(CC(=O)NC(CNC(C(C=C=C)C)=O)C(C)C)ccc(OC)cc1Cl C=CCCCC(=O)N1CCC1(C)CC(N1CCCC1C1CCOC1)=O C1(C(N(CC#CC)CC#C)=O)CCCCCCN1C(=O)C(C)OCC=C N1(C(c2scc(C)c2)=O)CCCCC(C(=O)NCC2OC(=O)CC2(C)C)C1 c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)ccc(N2CCCCCC2)cc1 C(=O)(C(C(=O)N1CC(CNC(C2(C)CCN(C)CC2)=O)(OC)C1)C(C)C)OCC C(CCC(C(=O)N1CCC(c2nc[nH]n2)C1)NC(=O)CCC(F)(F)F)OC c1(N2CCCCC(NC(c3c(C(C)C)nn(C)c3)=O)C2)ccncc1[N+](=O)[O-] c1(C(=O)NCC(CCCC)NC(c2cocc2C)=O)cnc2c(cnn2C)c1 c1(-c2c(C)c[nH]n2)nc(-c2ccsc2)nn1-c1ccn(C)n1 CCCCCC(=O)NCC1CN(C(=O)CCOCCCC)C2CC12 c1(C(N(CC(C)(C)NC(=O)CCc2nccn2C)C)=O)c(F)ccc2c1OCC2 C#CCC(C)(CC)C(=O)NC1CN(C(=O)Cc2nc(C3CC3)nn2C)CC1SC O(NC(=O)C(CNC(C1(C)CCCC1O)=O)CC1CC1)CC(=C)Cl c1(NC(C2CCN(C(C3=NOC(C)C3)=O)C2C2CC2)=O)ccc2ccncc2c1 c1(C(N2CCC(OC3CCCCC3)CC2)C(=O)NCC(=C)C)cc(Cl)sc1C N1(C(C2CCCN(Cc3cn(CC(C)(C)C)nn3)C2)=O)CCCC(B(O)O)C1 CC1=C(C)CN(c2nccc(N(C)Cc3nccn3C(C)C)n2)CC1 c1(C(N2CCC(N(C(COCC(=O)NC)=O)C)C2)=O)cc(OC)cc(Cl)c1 C1(N(C(=O)CCn2cnnn2)C)CCC(NC(c2cnc(S)[nH]2)=O)C1 C(C)(C(=O)N1CC(O)CO1)N(C(C(COC)OC)=O)C1CC1 N1(C(C(COCC)C)=O)CCCC(N(C(=O)C=Cc2ccncc2)C)C1 c1(CNCC2N(C(c3nc(CCCCC)sc3)=O)CCC2)cncc(C)c1 C1(CNC(=O)CSCC(F)F)(NC(C2CC(=C3CC3)C2)=O)CCCCCC1 O=C(C(Cn1cccn1)NC(=O)Cc1ccon1)NC(c1ccncc1)C1CC1 N1(C(=O)NC2CCCC(C(N)=O)C2)CC2CCC1C(O)C2O Cc1nc2ccc3cc(C(=O)NC4CCN(CCC5CCCC5)C4)ccc3n2n1 c1(CC)cc(F)ccc1CC(=O)N(C1CCCN(C(C2(Cl)CC2(C)C)=O)C1)C c1(NC(C2(CC#C)CCCO2)=O)cccn(-c2ccccn2)c1=O Cc1nc(C(=O)NCC(C)(C)NC(c2nc(=N)cc[nH]2)=O)c(C)o1 c1(C(=O)NC2C=CCN(C(=O)Cc3ccccc3CO)C2)cn2cnnc2cn1 CCCCC(C(=O)NC1CCN(C(c2ccc(CC)nc2)=O)C1)ON=C(C)C N(C(=NCc1ccccc1)N(C)CC1CCC1)C1CCC(CC)CC1.S(C)(=O)(=O)N C1(CNC(C2CCN(CCCC)C2)=O)(CNC(=O)C(C)(C)SCC)CC12CCC2 c1(C(N(CCCN(C(C(C(C)C)O)=O)C)C)=O)cc(C(F)(F)F)cnc1N Cn1cc(C(N2CC3CC3(CO)C2)=O)c(CNC(C2(CC3CC3)CCCO2)=O)n1 N#CC1(C(=O)NC2CC(NC(C3CCCCC3)=O)C23CCC3)CC2CCC1CC2 c1(C(=O)NC2N(Cc3c(COC)cccc3)CC(O)C2)ccc(CC#N)c(F)c1 N1(C(C=C(C)C)=O)CC(NC(=O)CCCc2ccsc2)CC(C)C1 c1(C(=O)NC2CC(C)CN(C(C3(O)CC3)=O)C2)cc(Br)cn2ncnc12 C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(SC)C(NC(=O)COC(C)(C)C)C1 c1(CC#N)ccc(C(=O)NC2(CCNC(c3cn(C4COC4)nn3)=O)CC2)cc1 c1(C(=O)OC)nc(C)c(C(N2CCC(C(=O)NC3(C)CCCC3C)C2)=O)s1 c1(C(N2CCCC(O)C2O)=O)cc(F)ccc1OC(F)(F)F CC1(C)CCOC(C(=O)NCC#CC(=O)NC(c2ccccc2)(C)C)C1 C1(C(=O)NCC2CCN(C(=O)Cn3cnc(Br)c3)C2)CCCS(=O)(=O)C1 c1(C(=O)NCC2(NC(C=CCC)=O)CC2)cccn2ncnc12 c1(COC)ccccc1C(=O)N(C1CCCC(C(=O)OC(=O)C2CC2)C1)C c1(C(=O)NCC2(NC(c3nc(CCC)sc3)=O)CCC2)nc(OC)ccc1Cl C#Cc1ccc(F)c(C(=O)NCC2CC2NC(C2(Cl)CC2(C)C)=O)c1 c1(C(N2CC(CNC(c3c(C)noc3C)=O)N(C)CC2)=O)cc(F)c(F)cc1O C1(CNC(c2ccn(C(C)C)n2)=O)CC2COCC2N1C(=O)CSc1nncs1 C1(CC)CCOCCN1C(C1CCCN(CCOCc2ccc(Cl)cc2)C1)=O C1(CNC(=O)NC2(C(=O)OC)CC(O)C2)CC(OC)(OC)CO1 CC1C(NC(=O)Cc2cc(Cl)ccc2Cl)CCCN1C(=O)Cn1cccnc1=O Cc1ccc2c(c1)CCC2Nc1conc1C1CCNCC1 C1(CNC(C(C(COC)C)C)=O)C(C2CC2)CCN1C(=O)C(CCOC)OC C(=O)(N=S(C)(=O)C1CCNCC1)C1(NC(N)=O)C(C)(C)NC1 C1(CC(N2CCC(CC)CC2)=O)CCC2CN(C(=O)C(C(CC)CC)OC)CC12 C(C(=O)NC1CC(CCNC(=O)C=Cc2ccccc2)C1)(C(C)C)OCC CCS(=O)(=O)C=CC(=O)N1CCC(C)C(NC(=O)CCOCc2ccccc2)C1 c1(SCC(=O)N(C2CCC(NC(c3cnn[nH]3)=O)C2)C)ccc(F)cc1 N1(C(C(=O)NCC(C(C)C)c2ccnn2C)=O)CCCC(O)(C2CC2)C1 c1(NC(C(CC)SC)=O)cc(CCO)ccc1C c1(COC)ccoc1C(=O)NCc1cc(C(=O)NC2COC(C(C)C)C2)on1 CC(=NO)C1CC(C(=O)NCC2(NC(=O)CCCCO)CCC2)C1(C)C S(=O)(=O)(c1ccnc(NC(=O)Cc2ccc3c(c2)CN(C)C3)c1)NC N1(C(C=C(COC)C)=O)CC2C(NC(=O)Cn3cc(-c4ccccc4)nn3)C2C1 C1(NC(c2cc(C)ncn2)=O)CCSC12CN(C(c1cccnc1C1CC1)=O)C2 C1(CCC)(NC(C)=O)CCCN(C(c2cnn(C3CCOCC3)c2)=O)C1 N1(C(C2OCCN(C(C3(CC=C)CCOC3)=O)CC2)=O)CCC(O)C12CCCC2 C(C(C)C(=O)N1CCC2CC12)NC(COCC#C)=O N1(C(C=NOC)=O)CCN(C(C2(n3cccc(O)c3=O)CC2)=O)C2CCCCC12 N1(C(CC2CC(CC)C2)=O)CCC(C)(CN(C)C)C1.C12(CCC1)C(=O)NC2 c1(SC)nc(C)c(C(=O)NCC2C3CN(C(c4c(C)nsc4C)=O)CC23)s1 c1(-c2c(CC)ncnc2)cc(NC2(CC)CC=CCC2)c(O)c(C(N)=O)c1 c1(-n2c(CC3CC3)nc(-c3c(OC)nccn3)n2)cccn(C(F)F)c1=O N1(C(C2CCN(C)CC2)=O)CCCCC2(CCN(C(=O)CC3(C4CC4)CC3)C2)C1 c1(C(N(CCCCNC(C2(C)CCCO2)=O)C)=O)c(Cl)cccc1[N+](=O)[O-] C(=O)(CCN=c1ccc(C)c[nH]1)NCCC1OCCN(C(C(CC)(C)CO)=O)C1 CCCCCCC(=O)NC(CC(=O)NC1CCOC(CC)C1)C(F)F C12(C(=O)NCC3(CC(=O)NC4COCC4CO)CC3)CCN(CC1)CC2 N1(C(c2c(OC)c(C)sc2)=O)CC2CC(NC(c3c(C)nn(C)c3Cl)=O)CC1C2 C1(CC=C)(NC(=O)CC(C)O)CCN(C(=O)NCc2ccccc2)CC1 C=CC(C)CC(=O)NC(C(=O)NCCC(C)(C)F)C1CC1 c1(C(=O)NCC(C)(C2CC2)NC(C2N(CC)CCOC2)=O)cc(C)cc(Cl)n1 N1(C(COC(C)C)=O)CCN(CCCCCNC(c2scnc2C2CC2)=O)CC1 N1(C(c2c(C)c(Br)cs2)=O)CC(C)(C)CC1CNC(=O)C(C)CO c1(C(C(=O)CSCC=CCN)=O)csc2cnccc12.c1(NC=O)ccc(Cl)s1 CC1(C(=O)NC2CC(NC(=O)CCC3(c4ccccc4)CC3)C2)CCCO1 N1(C(CN(C)CC)=O)CCC2(CCC2CNC(c2ccc(C(C)C)cn2)=O)CC1 C1(NC(C2(COC)CC=CC2)=O)COC2C(NC(=O)CSC3CC3)COC12 c1(CNC(c2cc[nH]c2)=O)ccsc1C(N1CCC(c2cnco2)C1)=O C12(CNCc3cccc(OC)c3N(C)C)CC3CC(CC(C3)C1N)C2 C12(NC(C3CN(C)C(=O)C3)=O)CCC(NCc3ccc(CC(=O)O)cc3)(CC1)C2 N1(CC)CCN(C(=O)C(C)N(C(c2cn3c(n2)CCC3)=O)CC)CC1C N1(C(C2CCCC3(CCOCC3)O2)=O)CCOC2(CCCN(C(=O)CCF)C2)C1 c1(OC(C)C)ncncc1C(=O)Nc1ccsc1CO c1(C(Cn2cc(-c3c(OC)ccc(C#N)c3)nn2)=O)cccc2c1S(=O)(=O)CC2 N1(C(c2cc(NC)oc2)=O)CCC2(CC1)CN(C(=O)CC13CC(C1)C3)CC(C)O2 Cc1cccnc1CNC(=O)C(C)N(C(c1c[nH]c(C)c1)=O)C1CC1 CC(CC(F)(F)F)C(=O)N(CCCN(C)C(C1CC2(CCCC2)CO1)=O)C CC1CCCC=C1C(=O)N1CCOCC(CNC(c2cccc3c[nH]nc23)=O)C1 CS(=O)(=O)c1cnc2cc(C(=O)NC(c3cc(F)ccc3F)C(=O)O)sc2c1 c1(OC)ccc(C)c(C(=O)NCCC23CCC(C2)N(C(=O)CNC(C)=O)C3)c1 c1(C(N(CC(CC)NC(C(CCC)OC)=O)CC)=O)cc2cc(C)ccc2o1 C1(C(=O)NC2(C(O)CO)CC2)CC(O)CCN1C(C1CCC2CC1CO2)=O Nc1ccc(C(=O)NCC2CCCCC2NC(C2(F)CCCCC2)=O)cc1 C1(N(C)C(c2cncs2)=O)CC2CC1N(C(=O)C(c1ccccc1F)(C)F)C2 CC(C)(C(=O)NC(CNC(=O)Cn1cc(C(C)=O)nn1)C1CC1)c1cnsc1 N1(C(C2(C#N)CCC2)=O)CCOC2(CCN(C(=O)CCCc3cnn[nH]3)CC2)C1 c1(C(N2C(CCNC(C(C(C)C)O)=O)CC(F)(F)C2)=O)cccc2ccoc12 N1(CCCCNC(C(CSC)C)=O)CCCN(C(c2ccc(=N)[nH]c2Cl)=O)CC1 N1(C(C(C)N(C)C)=O)CCC(CCN(C)C(C2CC=CCC2)=O)CC1 c1(OC(COC)C(=O)NCC(C)(C)NC(=O)CN(C)CCO)cc(C)ccc1Cl C1(CNC(C2CCN(C)CC2)=O)CCN(C(C2CCCC2F)=O)CC1O CN=c1nc(C(=O)NC2CN(C(C3CCCN3C=O)=O)CC2C)cc(C)[nH]1 N1(C(C2(c3cc(F)c(Cl)cc3Cl)CC2)=O)CCCC(O)(c2ccccc2)CC1 C1(CNC(CCOC(C)=O)=O)CCCCN1C(=O)C=CC1CC1 C1(NC(c2c(CCC)n(C)nc2)=O)CCC2(CCN(C(c3cn(C)cn3)=O)C2)C1 c1(OC)cccc2cc(C(=O)NC3CCC3CNC(=O)Cc3cc(C)cs3)[nH]c12 N1(C(Cc2n(C)cnn2)=O)CCCCC(NC(=O)CCn2ncn(C)c2=O)C1 C(=O)(C1=CNC2=NCCC2=C1)N1C(C)C(NC(=O)CC2CC2(Cl)Cl)CCC1 CC(N=c1[nH]c(=NCC2CC(F)C2)c2c(F)cccc2[nH]1)c1cc(Br)ccc1F N1(C(c2c(CC)ncs2)=O)Cc2n[nH]cc2C1C(=O)N1CCC(CCN(C)C)C1 C(C(F)C(C)(C)O)NC(C1CC(C)(NC(CC(C)F)=O)C1)=O CC1(C)CN(C(c2cnc[nH]2)=O)CCN(C(c2ncoc2Br)=O)C1 c1(C(N2C(CC(=O)NCCC(C)F)CC(O)C2)=O)ccc2cccnc2n1 c1(NC(CC2(OC)CN(C(C3CCCN3C(N)=O)=O)C2)=O)ccc(F)cc1O c1(C(N2CCC(CN(C(CC=CCC)=O)C)C2)=O)ccc(C(F)(F)F)nc1 C(CCN=C(NCC1CC2(CCOCC2)O1)N1CCCC(CC(F)(F)CF)C1)OC N1(C(C2CCCC2NC(C23CCCC2C3)=O)=O)CCc2ncccc2C1 C1(NC(c2n(CC(C)C)ncc2)=O)CCCCN(C(=O)CC2COC(C)(C)C2)C1 Cn1cc(C(N2CCC(CCNC(c3ccc(O)cn3)=O)CC2)=O)c(O)nc1=O N1(C(C(CCC)OCC2CCCCC2)C)CC2C(C1)C2(F)F C1(NC(c2ccc(SCC)cc2)=O)CCN(C(c2cnc(C)[nH]c2=N)=O)C1(C)C c1(COC)cccc(C(N2CCCC2C(N2CC[Si](C)(C)C2)=O)=O)c1 c1(CCC(=O)NCCC(C)N(C(=O)C2=NNC(=O)CC2)C)ccc(C#N)cc1F CC1CCC(Cl)=C(C(=O)NCC(O)CCNC(=O)COc2cccc(F)c2)C1 CCC(C(=O)OC)C(=O)NCC1CCCCN1C(c1cc(Cl)ccc1F)=O c1(S)ccc(F)cc1.C1(C(CNC(C=C(CC)C)=O)(C)O)CCN(C(=O)CCF)CC1 N12CC3C(CS(=O)(=O)C3C1)C2=O.CC1CC(C)(CSC(C)(C)C)C1 c1(C(C)NC(C(=O)N(C)Cc2nnc(C(=O)OCC)s2)=O)ccc(C)cc1F c1(CC(=O)NCC(C)CNC(C2(C3CC3)CCOCC2)=O)cccc2sccc12 Cc1noc(C)c1C(=O)Nc1ccccc1NC(C1CC1Cl)=O Cc1ccsc1NC(=O)NC1(c2ncccn2)CCOC1 C#Cc1ccc(C(=O)NCC2CN(C(=O)Cc3ccnc(Br)c3)C2)cc1Cl c1(CN(CC)Cc2cccc(O)c2)ccc(-c2ccc(C(=O)N(C)C)nc2)cc1 c1(C(=O)NCC(CC)NC(=O)CC2CC(C)=NO2)c(C)nn(C)c1N C1(CNC(C(C)(F)F)=O)COC(C(F)(F)F)CN1C(C1CCCC1)=O c1(C(C)NC(=O)NC2C(C(CC)(C)C)CCC2)ccc2c(c1)CC(C)O2 N1(c2nnc(C3CCC(CO)O3)n2CC2CC2)CCOC2(CCCC2)C1 c1(C(N(C2CCN(C(c3cccc(NC(C)=O)c3)=O)C2)C)=O)nc(C)ccc1C c1(-c2cn(CCCCCCNC(CC3C=NN(C)C3=O)=O)nn2)cc(Cl)ccc1F C(CCN=C(NCc1nnn(C)n1)NCC(O)Cc1ccccc1)OC(C)C N1(C(C2CCC(C)(CC)O2)=O)CC2(CC(CNC(c3cnc(C)[nH]3)=O)C2)C1 Cn1c(C(N2CCCCC2CCNC(C2CC(=O)NC2(C)C)=O)=O)cccc1=O C1(NC(C2(C)C(C)CCC2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 C1(C(N2CCCC(CNC(CCCOC(C)=O)=O)C2)=O)Cc2nn(C)cc2C(=O)N1 Cc1cccn2ncc(C(N3CCC4C(C3)CN4C(=O)C(=O)NCC3CC3)=O)c12 c1(C(=O)OC(C2(O)CN(C(=O)OC(C)(C)C)C2)C)cc(C(C)(F)F)ccc1C C(=O)(C1CO1)N(CCCC)CCCC.c1(C(=O)OCC)ccccc1 C1(c2ccccc2)(C(=O)NC(CN(C(COCC)=O)CC)C)CCOC1 C(=O)(CCCCCNC(=O)CC1CCSC1)N1CC(C)(C(N)=O)C1 N1(C(c2cn(CC)nc2C)=O)CC2CC1CN2C(=O)CCC1CCOC1 C(=O)(C(C)(C)C(F)F)N(CCCCNC(c1cc(OC)no1)=O)C C(CCCN=C(NCc1ccccc1)NCC1CC12CCSCC2)OC(C)C C1(CNC(=O)CC2(C(F)(F)F)CCC2)CCCCN(C(C2C=CC=CC=C2)=O)C1 c1(C(N(C2CC2)CC2CCCN(C(C=CSC)=O)C2)=O)cc(C)ccc1O CC1=CC(C)=NS(=O)(=O)N1CC(=O)NC1CCN(C(=O)Cn2cccc2)CC1C C1(C(=O)OC)(CCNC2CCC2N(C)C)CCN(C(=O)CCc2csnn2)CC1 C1(CCC)CCCC1C(=O)NCCC1(CNC(=O)Cc2csc(=N)[nH]2)CC1 c1(OC)cc(OC)nc(C(N2CCC(C(C)NC(=O)CC(C)C3CC3)CC2)=O)n1 c1(OC)cc(CC(=O)OCC(=O)C2(C(F)(F)F)CC2)ccc1C C1(C(=O)NCCNc2c(C)ccnc2)CCC(C)C(C)C1 C12(C(=O)NCC(CC)(C)C)CCC(CC1)N(C(=O)C(C)C1CCC1)C2 C1(NC(CC2CCCN(C)C2)=O)CCS(=O)(=O)C12CN(C(C1(CO)CC1)=O)C2 Cc1nn(C)c(Cl)c1CC(=O)NC1CCCCC1CNC(=O)CCC1CCOC1 c1(OC)cc(C(N2C(C)CN(C(=O)C(O)CSC)CC2C)=O)c2occc2c1 C12(CNC(C3CCS3(=O)=O)=O)CCCC1N(C(=O)CSCCC(F)(F)F)CCC2 c1(C(=O)OCC)nccc(C)c1NC(C1(C)CC1(Cl)Cl)=O C1(CN(C(=O)C(CO)c2ccccc2)C)C2CN(C(c3ncn(C)n3)=O)CC12 Cc1cc(N2CCC(C(F)(F)F)(CO)C2)nc(=NCC(C)CC2CCC2)[nH]1 N1(C(c2cnoc2C2CC2)=O)CCN(C(=O)CCc2cocn2)C(c2cccs2)C1 N1(C(C2(C)CC=CCO2)=O)CCN(C(C2COC(=O)N2)=O)CC2(CC2)C1 c1(CCCOC)ccc(-c2nc(-c3cc(Cl)ccn3)nn2C(C)C(C)(C)C)cc1 c1(C(=O)NCC(C(=O)N(C(C)C(N)=O)C)CC2CC2)cc2n(n1)CCO2 c1(C(N2CC(CNC(CCCOC)=O)C(C(F)(F)F)C2)=O)c(F)ccc(F)c1F C(=O)(CC(C)C(C)(C)NC(c1ncoc1CC)=O)NC(C=C)C1CCC1 c1(CCCC)nc(CN2CC(NS(C)(=O)=O)C2)c(Cl)[nH]1.N12CC(F)CC1C2=O Cc1nc2cncc(CC(=O)NCC(C(C)C)NC(=O)C(=O)N(C)C)c2[nH]1 c1(C(N2CCC(CN(C(C(C)S(C)(=O)=O)=O)C)C2)=O)c2ccccc2nn1C c1(C(=O)NC2(CC=C)CN(C(=O)CSCC3CCCCO3)C2)cc(C)sc1C O=C1CCC(C(=O)N(c2ncnc3occc23)C2CC3(C2)CC(N)C3)=NN1 C12(C(N3CC(NC(C45CCCCC4C5(F)F)=O)C3)=O)CCCN(CCC1)C2 C1(NC(=O)C(F)OC(F)(F)F)CC(O)(C(N(C(CC#C)C)C)=O)C1 C(CCCCC(=O)N1CCCC1C(C)NC(C1(N(C)C)CC1)=O)OC c1(C(=O)NC(C2OCCN(C(c3cc(COC)no3)=O)C2)C)cc(O)ccc1Cl c1(C(C(=O)NCC=C)N(C(C)C(=O)OC)CC(C)C)nn(CC)cc1Br Cn1nccc1C(F)=CC(=O)NCC1CC(NC(c2cccc(C(F)F)c2)=O)C1 N1(C(C=C2CCC(C)C2)=O)CCC(C(N2CC3C=CC3C2)=O)C1C(C)C C=C1CCC(C(=O)NCCCCN(C)C(C2(C(F)F)CCCO2)=O)CC1 C(=O)(CCCC(C)(C)C)NCCC1CN(C(C2(CC)CC(C)(C)C2)=O)C1 c1(COCC(=O)N(C2CCN(C(=O)C(F)=CC3CC3)C2)C)cccc(C(N)=O)c1 Cn1ncc(C(=O)NC2CC3C(NC(C4CCC(CC#N)CC4)=O)C3C2)c1Cl C1(C(N)=O)CCCC(SCC(=O)Nc2ncccc2F)C1 C(c1ccc(Cl)cc1)=CC(=O)NCC(C1CC1)NC(CCNC(C1C(C)C1)=O)=O C12(CCNC(=O)NC(c3ccc(NS(C)(=O)=O)cc3)C)COC(C)(C1)C2 C1(C(=O)NC(CNC(=O)C=Cc2ncc[nH]2)C2CCC2)CCc2nnnn2C1 C1(C(=O)NCC(CC)NC(c2cc(OCC)n[nH]2)=O)CCCNC1=O C1(=O)C(O)COCC(=O)N1.c1(N(C(C)C)C(c2ccccc2)F)ccccc1 N1(C(C2(CC=C)CC2)=O)CC2CC(C1)N(C(=O)C(C)CC(C)(C)C)C2 C(=O)(CCC(C)C)N(CC(=O)N(C)CCC1CCCN1C)CCOC C1(CN(C(CNS(CC)(=O)=O)=O)C)CCCN(C(c2cnn(C3CC3)c2Cl)=O)C1 N1(C(c2c(CC)cc(N)cc2)=O)CCN(C(C2CC(CF)C2)=O)CCC1C C1(CC(N2CC(CC=C)(NC(=O)Cc3cc(C)cs3)C2)=O)CCN(OC)CC1 CCC(CC)C(C)C(=O)NCC1(C2CC2)CCN(C(C2CCOC2)=O)C1 C(C(C)(C)C#CC(=O)N1CCC(CO)C(O)C1)NC(COC(CC)(C)C)=O C(=O)(C1=CCCCCC1)N1CCCC(NC(=O)CCn2ccnc2)C1 c1(CC)nc2c(C(=O)Nc3cc4c(cn3)C(=O)CCC4)ccnc2[nH]1 C1(CC)C(NC(c2ccc(SC)s2)=O)CCCN1C(=O)C=CC1CCOC1 C(=O)(CCCCCCSC)NC(C(=O)NC(CC=C)C(=O)OC)CO C1(C(C)C)(C(N2CC(O)(c3cnn[nH]3)C2)=O)CCCN1C(=O)C=C1CCOCC1 N1(C(c2c(OC)nccn2)=O)CC2(C1)CN(c1ncc(C)cn1)C2 N1(CC#C)CC2CN(C(c3c(Br)cncc3Br)=O)CC2C1 c1(CC(=O)NCC2N(C(C(C)SC)=O)CC2)ccnn1C C1(C2CC2)(CNC(c2c(C(C)C)n[nH]c2)=O)CCN(C(=O)C(=O)C(C)(C)C)C1 N1(C(c2nccc(CNC(C(C)CC3CC3)=O)c2)=O)CCOC(C)CC1 c1(OC)cccc(O)c1NC(C1CC1C(C)NC(=O)C(O)CC(C)C)=O C(=O)(CCC(C(C)C)NC(=O)CC1CC=CCN1C)NCC(CCC)CCC C#CCC(C)(C)C(=O)N(CCN(C(C1C2CCC1CC2)=O)CC)CC CC1(NC(=O)C2CC2)CCN(C(C23CCC(CO2)C3)=O)CC1 c1(C(N2CCC(COCCO)C2)C(=O)NCC=C)nc(Cl)cc(Cl)c1C c1(C(N2CCC(O)(C(C)NC(c3cc(C)[nH]n3)=O)C2)=O)cccc2sncc12 C1(CCN(C2CCCC2)C(CN(C)CC2CCCCN2)=O)CCS(=O)(=O)C1 CCC(O)(CC)CCNC(C1CC(C)(NC(C2OCCCO2)=O)C1)=O C1(C2CCOCC2)(NC(C(COC)C)=O)CC1.c1(C2C(=O)N2)cnn(C)c1 c1(C(N(C)CCN(C)C(C2(O)CCSCC2)=O)=O)c(F)ccc2cnn(C)c12 CCC(CNC(=O)CC=CC(C)(C)C)(CC)NC(c1cc(CSC)n(C)n1)=O C(C(C(C)C)NC(c1conc1C1CCCO1)=O)NC(C1(COC)CC1)=O C1(NC(c2nnnn2C(C)(C)C)C2(SC)CCC2)C2CCCOC12 C1(NC(C2CCC(=C)CC2)=O)CN(C(c2ccsc2C#N)=O)CC1N=[N+]=[N-] C(=O)(CCCS(N)(=O)=O)NCC(C1CCN(C(C(C(C)C)F)=O)CC1)(C)C n1(C2CN(C(c3cc(C)on3)=O)C2)cnc(=N)[nH]1.C(CS(C)(=N)=O)NC(=O)C c1(C(N2CC3(CN(C(C=C(C)C(C)C)=O)C3)C2)=O)cc(C)c(C)c2ncccc12 C1(C(=O)OC(C)(C)C)(COC)CCCN(N2CC(OC)C3(CC3)C2)C1 N1(C(COC)=O)CCC(CNC(c2cc(C)sc2S(N)(=O)=O)=O)C(C)(C)C1 C#CCC(C(=O)NCc1cncn1C(C)C)NC(=O)Cc1ccc(C)o1 C#CC1(O)CC(C(=O)NCCC(C)(C)CNC(=O)CNC(c2ccncc2)=O)C1 c1(C(=O)NC(C(C(C)C)NC(COCCC)=O)C)ccn2ncnc2c1 c1(C(N(CC(CNC(COC)=O)C)C)=O)c(C(F)(F)Cl)n[nH]c1C C1(NC(C(C2CC2)SC)=O)C2CC1N(C(=O)CCCc1nc(C)no1)C2C c1(C(=O)NCC2CC(OCC)C2)cc(Br)c2[nH]c(C)nc2c1 C1(C(C(=O)NC2CC2)OCCOCCCC#C)CCN(C(=O)CC(C)(C)C)C1 C1(CNC(c2cnc(S)nc2)=O)CC2(CCC2)CN1C(c1cc(F)ccc1Cl)=O C12(C(N3CC(O)(C(C)NC(=O)CN4C(=O)CCC4=O)C3)=O)CCCC1CCN2 n1(CCC)cc(CNC(=O)Cc2ocnc2CNC(=O)CC(=O)OC)nn1 Cn1cc(C=CC(=O)NC(Cn2cncn2)C(=O)NCCc2ncccn2)nn1 C1(CNC(c2c(C)sc(O)n2)=O)(NC(c2nc(=N)cc[nH]2)=O)CC2CCC1CC2 c1(C(=O)NCC(CC)NC(=O)C(C)(C)COCC(F)F)cnc(SC)n1C CC1(C)CC=C(C(=O)N2CCOC(C(=O)NCc3ccnc(F)c3F)CC2)CC1 C(=O)(CC(C)(C)C(C)(F)F)N1CCC(CNC(CCc2c(C)ncs2)=O)C(C)C1 N1(C(C2(C#C)CC2)=O)CC2(C1)CN(C(C1CCN(C)C1)=O)CC(C)(C)O2 C1(OC)CC(C(=O)NC2CCN(C(c3cnnc(C)c3)=O)CC2)N(C(C)=O)C1 C1(=CCNC(C(c2cccnc2)C)=O)CCN(C(C23CC(C#N)(C2)C3)=O)CC1 C1(Cc2ccc(F)cc2)(OCCO)CCSCC1.C12CCCC1NC(=O)NC2 C1(OCc2ccc(Oc3cccc(SCC)c3)cc2)CCC2(CCOCC2)C1=O C1(NC(C2(C=C)CCC2)=O)CN(C(c2ccnc(SCC)c2)=O)CCC1CO Cc1ccc(C(=O)Nc2ccccc2-c2ccc(O)c(F)c2)c(O)c1 C(CCCCCNC(C1SCCC1C)=O)NC(c1c(CC)scn1)=O N1(C(C(CC)N(C)C)=O)CC2(CNC(=O)C=Cc3scnc3C)CCC1CC2 N1(c2cccc(S(=O)(=O)N3C(C)SCCC3)n2)CCc2c(C)cc(Br)cc2C1 C(CC(C)(C)C(=O)NC1CCCN(C(c2ccc(F)c(O)c2)=O)CC1)OC C1(C(N2C(CC)CC2)=O)CC(C)N1Cc1coc(C(N)=O)c1 Cc1cc(NCCCN(C(=O)C(C)CSc2ccccc2)CCO)nn1C N1(C(C(CC)SC)=O)CCOC(CCNC(=O)CC2(O)CC2)C1 N1(CC(C)C)CCCC1C(=O)NCC1(CNC(=O)C=Cc2cscn2)CC1(F)F C12(CNC(C3CC(=C)C3)=O)CCCCC1N(C(=O)C(C)CCOC)CCC2 C(=O)(N=c1[nH]nc2[nH]ccnc1-2)C12C(CN(C(CCc3c(C)nccc3)=O)C1)C2 C1(C)(C(=O)NC(C2CCN(C(Cc3ncn(C)c3)=O)C2)(C)C)CNC(=O)C1 CC#CC1CN(C(=O)C(C)N(C(=O)C=CC(=O)N(C)C)C2CC2)C1 C(c1cccc(Cl)c1Cl)=CC(=O)NCCCNC(C1CC2C=CC1O2)=O N1(C(=O)C=Cc2cccnc2)CCC2(CCN(Cc3cccc4nc[nH]c34)C2)C1 C12(NC(C3C4CCCCCCC34)=O)CCCC1N(c1cc(C3CC3)ncn1)CC2 Cc1cnc(N2CCCN(C)C(=O)C2)c(S(=O)(=O)NC2(C)CC(C)OC(C)C2)c1 C1(C(=O)NC(c2cccc(C)c2)CNC(CCC=C(C)C)=O)CCC12CCCO2 c1(C(N2CC3CC(NC(=O)Cn4ncnn4)CC3C2)=O)cc2ccc(Cl)cc2o1 Cc1cccc2oc(N(C)CC3CCCN(C(=O)C4=C(Cl)CCOC4)C3)nc12 C(Cc1ccccc1)(C(=O)NCCN(CC(C)O)C(=O)CC1OCCCO1)OC C(=O)(C(C)(C)C(F)(F)F)NC(CNC(c1cn(CC(CC)O)nn1)=O)CO C1(C(=O)NCC2(OC)CC2)CCC(CNC(=O)CNC(=O)C2CC2)CC1 C1(NC(c2ccc(C(C)C)nc2)=O)CCC(O)CN(C(=O)CCn2cccn2)C1 N1(C(CC2(C)CCCC2)=O)CC(NC(C2CCCC(O)C2)=O)CC2(CC2)C1 c1(CCC(N2C(C)(CNC(CN(C3CC3)CC)=O)CCC2)=O)c(F)cccc1Cl c1(C(=O)NCC2C(NC(C3CCC(=C)CC3)=O)C2)ccc(F)cc1C(F)(F)F N1(C(=O)CC2CC3CC3C2)CCCC(CNC(C2(Cl)CC2)=O)C1 c1(C(=O)NC2CCN(C(C3CCCC3)=O)C2)cc(C(F)(F)F)ccn1 c1(N2C(CCCNC(c3cnn(CC4CCCC4)c3)=O)CCC2)ncc(I)cn1 N#Cc1cc(C(=O)Oc2cccc(C(=O)NC34CCCC(C3)OC4)c2)cc(O)c1 CC(C)(C#N)CCCC(=O)NCC1CCCC(NC(c2ccc[nH]2)=O)C1 N1(C(C2CC(CC)C2)=O)CCC2CCN(C(=O)C=C(C)c3ccccc3Cl)C2C1 Cc1nn(C2CCCC2)c(Cl)c1C(N1CCC(CO)(NC(=O)NC(C)(C)C)C1)=O C(C1=CCN(C(C2CN(C3CCC3)C2)=O)CC1)NC(CC1C(=O)NC(=O)N1)=O C#Cc1cccc(C(=O)NC(CN2CCN(C(=O)CN(C)C(N)=O)CC2)C)c1 N1(C(C(CC)O)=O)CCn2nc(C)c(CNC(c3cc(=O)n(C)o3)=O)c2C1 C12(CNC(COC3(C)CCC3)=O)CCC(CNC(c3ccnnc3O)=O)(CC1)CO2 N1(C(C=NOC)=O)CCC2CCC(NC(c3cc4c(C)cccn4n3)=O)C1C2 CC(C)CC(C(=O)NCC(O)CN(C)C(C1CC(C(N)=O)(CO)C1)=O)C(N)=O Cc1nc(NCC(C)(F)F)cc(=NCc2cc(F)cc3c2CCC3)[nH]1 N1(C(C2OCCN(C(CCCC#C)=O)C2)=O)CC2(CCC2)OCC1C CC1CN(C(=O)C(O)C(C)c2ccccc2F)CCN1C(c1cc(CF)on1)=O Cc1cc(CC(N2CCC(C)(NC(C3CC4(C3)OCCO4)=O)CC2)=O)ccc1F C1(NC(c2cnc(C)[nH]2)=O)CN(C(=O)CCc2cn(C)nn2)CCC1(C)C c1(C(=O)NCCCN(C(CSCCC#N)=O)C2CC2)cc2[nH]ccc2cc1Cl C1(NC(=O)CNC(=O)C2CC2)CCN(C(c2occ3c2CCC3)=O)CC1CO N1(C(CC2CC(CC)OCC2)=O)CC2CC(C1)N2C(=O)C(C)(C)CN(C)C Cc1cc(C(=O)NC(c2cn(C3CCN(C)C3=O)nn2)C)c2n[nH]cc2c1 N1CCC(C=O)C12CCC2.C1(COCCNC(=O)OC(C)(C)C)CCCO1 C=C1CC(C)(C(=O)NC2COCC2C(=O)NC2(c3nc[nH]n3)CC2)C1 C1(C2CCN(C(=O)CCc3nncs3)C2)(NC(=O)CCCc2cnn[nH]2)CC1 c1(OC)ccc(CC(N2CCC(C(F)C(N3CCNCC3)=O)CC2)=O)c(Br)c1 C(=O)(C1=CCCC1(C)C)NCC1(F)CC(NC(C2CN(C(C)C)C(=O)C2)=O)C1 Cc1scnc1C(=O)N(C(C)(C(=O)N1CCC1C1CCCC1)C1CC1)C c1(C(=O)NC2CN(C(c3c(C)c(=O)cc[nH]3)=O)C(C)(C)C2)cc2nnn(C)c2s1 C1(CNC(C2(C)CC(=C)C2)=O)CC(O)CN1C(c1ccc(C(=O)N(C)C)cc1)=O C(CC(C(=O)NC(c1cccc(Cl)c1)CNC(=O)CCC1CCC1)N(C)C)SC C1(CCC)CN(C(c2cccc(C3CCCOC3)c2)=O)CCN1C(=O)C1CC1 C1(C(N(C(CCNC(CN(C(C)C)C)=O)C)C)=O)CCc2cc(F)ccc2O1 N1(C(CC(CNC(=O)CC(COC)COC)OC)=O)CCn2c(C)nnc2C1 O=C1CC(C(=O)NC2COCC2NC(C2(CCF)CC2)=O)c2cccnc2N1 C(C(CC(F)(F)F)NC(=O)C(=O)N(C)C)NC1CN(CCCC)C(=O)C1 O=C1NC(=O)C2(CCC(C(=O)Nc3ccc(OC4CCCCC4)cc3)CC2)N1 C(CC(=O)NC1(C)CSC1)(C(F)(F)F)NC(C(C)CC(F)F)=O CC1CN(C(C2C3CN(C(=O)CCc4cccc(O)c4)CC23)=O)CCC1=O N1(C(CNC(CC)=O)=O)CCC2(CC1)C(OC)CC2NC(c1ncn(C)c1C)=O Clc1ccccc1-c1ccc(-c2ccc(NC3CC3)s2)cn1 Cc1ccc2occ(CC(=O)NC(C3CN(C(=O)CSC(F)(F)F)C3)C)c2c1 C(CN=c1nc(C#N)[nH]cc1C)=CCNC(C(CC)C(C)O)=O c1(C(=O)NC(C2CN(C(C3COC(=O)N3)=O)CCO2)C)ccn2cccc2c1 c1(N2CC(COC)N(c3ncc(C(F)(F)F)cn3)CC2)ncnc2n[nH]c(Br)c12 N1(C(COc2ccc(OC)cc2)=O)CCC(CNC(=O)C(C)C(C)C)C12CC2 N#Cc1ccccc1CNC(C12CCN(C(=O)CC34CCCC3C4)CC1C2)=O c12cccc(c1Br)C(=O)N2.c1(N(C(C)=O)C)ccc(-c2ccccn2)s1 C1(C(=O)N(C2CC(O)C2(C)C)CC)CCC2(CC1)CC2.c1(CC)ncccc1C=O CN1C(=O)CC2CN(C(C3CCCN3C(C3CCCC3)=O)=O)CCC12 CCCCC(O)C(=O)N1CC(NC(=O)C(F)F)C(C(F)F)C1 C#CCC(C)(C(=O)Nc1ccc(F)c(CC)c1)NC(C1CCOC1(C)C)=O C1(C#N)(CC)CCN(C(C2(C)CCC(C)C2(C)C)=O)CC1 N1(C(C2C(CC)CN(C(=O)CC3(C)CCCCC3)C2)=O)CCC(C2CCCC2)C1 Cc1ccc2cc(CC(=O)NCC=C3CCN(C(=O)C(C)N(C)C)CC3)ccc2n1 c1(C(N2CC(O)(CNC(CC3C(C)C3)=O)C2)=O)ccc2ncsc2c1 C(=O)(CCCC(=O)NC1(C(C)NC(C2CCOC2C(C)C)=O)CC1)NCC Cc1cc(CC(N2CC(CN(C)C(c3ccn(C4CCOCC4)n3)=O)C2)=O)no1 Cc1cc2[nH]c(C(N3CCC(n4cc(-c5cc[nH]n5)nn4)C3)=O)cc2o1 c1(C(=O)NCCNC(CC(C)C2CCCO2)=O)cc(Cl)cc(Br)c1 C1(NC)CCCC1C(=O)NCCCF.C1(C)(C)C=CC(=O)NCCOC1 c1(OCCn2cc(-c3nc[nH]n3)nn2)cnn2c1OCCCC2 C1(CNC(C(C)(C)OC(C)=O)=O)CCCC(CNC(c2ccns2)=O)C1 CCCC(C)(CCC)C(=O)N(CCCCCCNC(=O)C(C)(O)C(F)(F)F)C C=C(C)CCCC(=O)NC1CC(C(=O)NCC(CC(C)C)OC)CC1O C(=O)(C1=CC2(CCOCC2)C1)NC1CC(NC(C(C)OCCC#C)=O)C1 CCC(C)C(C)CNC(C1(C)CN(C(C2(n3cccn3)CC2)=O)C1)=O C1(O)(CNC(=O)NCCC(C)(C)c2ccccc2)CCCC1(C)C N1(C(c2c(C)nc(C)s2)=O)CC(=O)NCC1C(N1CC=CC(O)C1)=O C12(CNC(CCNC(=O)OC)=O)CCC(CN1C(c1ccc(OC)nc1)=O)C2 N1(C(c2cccc(SC)c2)=O)CCC(NC(C2CC(CCO)C2)=O)CC1C N1(C(=O)OC)CC(C(=O)NC(C)CNC(=O)CN(C(C)=O)C2CC2)S(=O)(=O)CC1 C(=O)(C(F)C(C)CNC(c1sccc1F)=O)NCc1cc(OC)ncn1 N1(C(COCC#C)=O)CC(NC(=O)C(F)C(F)(F)F)CC12CCC2 CN1CCCCC1C(=O)NCCC1CCN(C(C2(C(=O)NC3CC3)CC2)=O)CC1 C1(NC(CCNC(=O)NC)=O)CCN(C(=O)COC)C12CC2 c1(-c2n(CCOC)c(N3CCC(F)(c4ccccc4Cl)C3)nn2)ncc(C)cc1Br c1(C(=O)NCC2(CN(C(C3(CC=C)CCOC3)=O)C)CC2)cc(N)c(F)cc1F N1(C(N2C(CC)CN(C(=O)CC3CCCC(C)O3)CC2)=O)C(=O)NC(C)(C)C1=O CC1CCOC1C(N1CCCC1CCCNC(=O)C=CSCc1ccco1)=O c1(C(=O)NC2(CNC(=O)CCC3CCCN3C)CC(OC)C2)cccc(C)c1C C1(C(=O)NC(C#C)CC2CCC2)(CNC(=O)CCC2CCCO2)CC12CCC2 C1(N(C)C)CCCN(C(=O)C(C)(C)C2CCCC2)C1.C1(CNC(C)=O)CCN1 C1(CN(C(=O)Cc2ccncc2)C)CCCN(C(=O)CC2CCCC(=O)N2)C1 N1(C(C(CC)N(C(=O)C(C)CC2CCC2)C)=O)CC(C2=NOC(C)C2)C1 c1(C(=O)NC(C)CC2CN(C(=O)COC3CCCOC3)C2)ccnc2[nH]nnc12 C1(COC)CN(C(=O)CSCC(=O)OC)CCN1C(=O)CC1CCS(=O)(=O)C1 N1(CC)CC(C(=O)NCc2cc(C(N3CC(CCO)C3)=O)cs2)CC1=O c1(CC)ncc(CNC(=O)C(C2(C)CC2)NC(C2CC(C)=NO2)=O)[nH]1 c1(-c2onc(C(N(CCOC)CCOC)C)n2)coc2ccc(OC)cc12 N1(C(C(C)CO)=O)CCOC(C(C)NC(c2ccccc2C2CCCC2)=O)C1 C(N=c1[nH]cnc2c(OC)cccc12)C1(C)CCCN(C(C(OC)OC)=O)C1 N1(C(C2(C)CC(=C)C2)=O)CC(N(C)C)C(CNC(=O)C(C)c2ccsc2)C1 C12(C(=O)NC3CN(C(=O)CCCn4cccn4)CC3O)CCCCC1CCCC2 C1(N(C)C)(CSC)CC2CCC1CC2.C1(=O)CCC(=O)NCC2CCC(C2)N1 C1(C)(COC)CC(NC(c2cn[nH]c2)=O)CN1C(C1CC(F)(CF)C1)=O N1(C(CCCOCCOC)=O)CCN(C)C(CNC(=O)C(O)CC(N)=O)C1 C1(CNC(C(CC#C)C)=O)CCN(C(=O)CCSCc2ccccc2)CC1(F)F C12(NC(c3csc(-c4ccccc4)c3)=O)CC1CN(C(C1(CO)COC1)=O)C2 C1(C(C)C)(C(=O)N(C)CC=CC(=O)N(C)CCN2CCCC2)COC1 c1(CNC(C2C(NC(C=Cc3cc(C)no3)=O)CCO2)=O)ccc(C)c(C)n1 C(CCCC(=O)NCC=Cc1cccnc1)N(C)C(c1ccnnc1O)=O c1(C(=O)OC)ccccc1CC(=O)NCCCN(C(=O)CCC(F)F)CCO C1(C(N2C(C)(C(=O)NC)CC2)=O)C2CCCC2CN1C(=O)CC1C=CCCC1 C1(C(N2C(C(=O)NCC)CCC2)=O)(NC(=O)C2=C(Cl)CC2)CCCCC1 Cn1c(NCC2(C)CCCN(C(=O)CC3CCC(=O)N3)C2)cc(O)nc1=O c1(C(=O)NCC(CN(C(=O)C(C)(C)n2cncn2)C)O)n[nH]cc1C1CC1 N1(C(C)=O)CCC(C)(C(=O)NCC2CCCN2C(c2cnoc2)=O)CC1 C(=O)(C1=CCOCC1)NCCC1CCC(NC(C=C2CCN(C)CC2)=O)C1 C1(C(N(C2(C)CN(C(=O)CCn3ccnc3)C2)C)=O)CCCC1C1CC1 C1(C(N(C2CN(C(=O)CCCc3ccncc3)C2)C)=O)CCS(=O)(=O)N1 C(N=c1[nH]c(N(C)Cc2ccccc2Br)nc2c1CCCC2)c1ncc(C)cn1 N1(c2ncc(C)c(SC(C)C)n2)CC2CC1CCC2NC(c1ccncc1)=O N1(C(c2c(OC)ccc(C)n2)=O)CC2CCCN(C(C3CC3C)=O)C2C1 CC1CCC(C(=O)NC(c2cccc(O)c2)C(N2CCCC2(CO)CO)=O)CC1 Clc1ccc2c(c1)OCC2NC(=S)NCC(F)(F)F CN=c1[nH]cc(C(=O)NC(C)CNC(C2CC2(c2ccccc2)C)=O)o1 C1(NC(=O)NCCC2N(CC(=O)N(CC)CC)CCC2)CN(C)CCO1 C1(C(=O)Nc2cnc(Cl)c(Cl)c2)CCc2nc(-c3cccc(O)n3)sc2C1 C12(C(N(CC(C)(C)NC(C3CCCNC3=O)=O)C)=O)CCCC1CC(=O)C2 N1(C(c2cccc3ccccc23)C(=O)OC)Cc2ccc([N+](=O)[O-])cc2C1 C(C)(C)(CC(C)(C)C)NC(C1C(C(C)C)OCC1)=O.C12CCC(CC1)CC(=O)N2 c1(C(=O)NCC2CN(C(C3CC(CC)C3)=O)CC2C)cc(=O)c2ccncc2o1 c1(COC)cccc(C)c1N(C)CCC1CCSC1 C1(CNC(CCN2C(C)CCCC2C)=O)CN(CCC2CCCC2)CCC1(F)F C(CC1=CCN(C(C2CC2C)=O)CC1)NC(C1N(C(C)=O)CC(O)C1)=O C(C(O)C(=O)N(C(C)CN(C(=O)C1CN1)C)C)SC.N1(C(C)C)CCCC1.C(C)(=O)N C(CC(CC)C(=O)NC(C)C(CO)NC(c1ccccc1SCC)=O)=CC C1(C(=O)Nc2nc(O)cc(C(=O)OC)n2)CCCC2CCCCC12 C(=O)(CCCC(=O)NC1CS(=O)(=O)CC1NC(=O)C(F)(F)c1cnccn1)NC C1(C(N2C(CC)CN(C(=O)Cc3cccn3C)CC2)=O)CCc2nnnn2CC1 CC1CCN(C(=O)CCc2cccc(Cl)c2)C1CNC(=O)Cc1cc(Cl)n(C)n1 O=C(C#CC1CCC1)NCC12CC1CN(C(=O)CCC1CCC(C(F)(F)F)O1)C2 N1(C(c2cccc(CCC)c2)=O)CC2(CNC(=O)C(C)(C)CF)CC1CO2 c1(C(NOCCCC)=O)occc1CNC(=O)C(C1CCCC1)OCC C(=O)(C(N=[N+]=[N-])C(C)C)NC12C(CN(C(C(COC)OC)=O)C1)C2 C1(OCC)CC2(C1)CC2C(=O)NCC1CC(O)CN1C(=O)C(C1CCCCC1)C N1(C(C(=O)NCCCC2CC2)C2C(CC)C2)CCC2CC12 N1(C(C2C(=C)C2)=O)CCC2C(C1)CN2C(=O)C(=O)N=S(C)(C)=O C1(CNC(C=COCC)=O)CCCC(CNC(c2cnn(C3CCC3)c2)=O)C1 CC1(NC(C2CC3CC3C2)=O)CC(NC(c2ccsc2-n2cnnn2)=O)C1 Cc1nc2c(C)cc(C(N3CCOC(CN(C(=O)C(C)CO)C)C3)=O)cn2n1 N1(C(CCCC2(C)N=N2)=O)CCC(C2CC2)C1CNC(=O)CN1CC(=O)NC1=O CC(C)S(=O)(=O)CC(=O)N(C)CC1(CNC(C2CCC(=O)O2)=O)CC1 CCCC(CCC)CN=c1cc(C)[nH]c(=NCc2ccnc(C)c2)[nH]1 C1(NC(c2scc(C)c2)=O)CCCC12CN(C(=O)CC1CCC(C)(C)O1)C2 Cc1ccc(C(=O)NC(C2CCOC2)CNC(CCNC(=O)N)=O)c(C)c1.C1(NC)CC1 c1(C(N(CCNC(C(CC=C)Cc2ccccc2)=O)CC)=O)ccc(N)c(Cl)c1O N1(C(C=Cc2ncn(C)c2)=O)CCN(C(c2n[nH]cc2Br)=O)C2CC12 C(=O)(C1=CCC(C)CC1)NCC#CCNC(c1ccc(C(C)=O)cc1F)=O c1(CC)ccc(C(N2CCC3C(CCN3C(=O)CNC=O)C2)=O)c2ccccc12 C(=O)(C1=C(C)CCC1)N1C(CNC(C2CC(O)CN2OC)=O)(CO)CCC1.C(N)=O CCC(=O)NNC(=O)C(C)(C)CCCCNC(C1CCCCC1(F)F)=O C1(C(C(=O)NCCOC)N(C)Cc2ncnn2C)CCCOC1 c1(C(=O)NCCCNC(c2cncc(N3CCCC3)n2)=O)ccn2c1CCCC2 Cc1nnn(CC(=O)N(CCC(C)NC(C2(CO)COC2)=O)C)n1 c1(CC(=O)NCC(C)N(C(c2cc(C3CC3)nn2C)=O)CC)sc(O)nc1O C1(CC(=O)NCC(O)CNC(=O)CC(F)(F)F)NC(=O)CNC1=O c1(OC(C)C(N2CC3CCN(C(=O)COC4CC4)C3C2)=O)c(F)cccc1F N1(C(CCSCCC)=O)CC(CNC(C2(OC)CCC2)=O)C(C)C1 S(=O)(=O)(c1ccc2oc(=O)ccc2c1)N(C)CC1(F)CCOC1 C1(C(=O)NCC2(NC(C34CC(COC)(OC3)C4)=O)CCOC2)CCN(C)C(=O)C1 C1(NC(c2nc(C)nn2C)=O)CCC2(CC1)CN(C(C1CC1F)=O)CCO2 C1(NC(N2CCC(C(C)C)C2)=O)CCC(C)(C)CC1c1ccccc1 Cc1cc(C)c(CC(=O)NCC(C(C)(C)C)NC(C2CCCC23CC3)=O)s1 C1(C(N(C(CC)CO)CC)=O)CC2CN(C(c3ncc[nH]3)=O)CC2C1 n1(-c2c(C)cc(Cl)cc2)nc(-c2ccsc2)nc1C1=NOCC1 N1(C(CNC(C)=O)=O)CCCC(NC(=O)CC2CCCCC23CC3)CC1 N1(CC)CCN(C(=O)C(C)(CNC(C2CC2C2CCCC2)=O)CC)CC1=O c1(C(N2CCCC(N(C(=O)CN(C)C(C)=O)CC)CC2)=O)cc2ccncc2s1 c1(OC)ncc(C(=O)NCC2CN(C(=O)CNC(=O)N(C)C)CCO2)cn1 N1(C(c2cc(-c3ccc(C(F)(F)F)cc3)no2)=O)CCC(N2CC(F)(F)C2)CC1 C=C(C)c1cn(CC(C2CN(C(=O)CCNC(=O)NC3CC3)C2)F)nn1 CCCS(=O)(=O)C1CCCC1C(c1nnnn1C1CCC2(CC1)CNC(=O)C2)NCC N1(c2nc(N3CCC(c4cccc(C)c4)C3)nc(C)c2)CCC2(CCCOC2)C1 c1(C(N(CC(C)N(C(c2c(C)cc(SC)o2)=O)C)C)=O)cc(C)cc(C)c1 C1(CNC(CC=CC=C)=O)(NC(=O)C(C2CCCOC2)OC)CCC(F)(F)CC1 CCC(F)(F)CC(=O)NC1(CNC(=O)Cc2cc(F)cc(Cl)c2)CC2CCC1C2 C(CCF)(C(=O)NC(C)CCO)NC(c1c(COC)cc[nH]1)=O N1(C(C(CSC)OC)=O)CC2COCC2(C(=O)NCc2cccc(F)n2)C1 c1(CC)c(N2CC3CCC2C(NC(=O)C(CSC)OC)C3)nc(C)nc1Cl c1(OC)cc(C(N2CCC(NC(=O)C3=CCOCC3)C(O)C2)=O)c(Cl)cn1 N1(C(C2(C(=O)OCC)CC2)=O)CC2CN(Cc3ccc(C(F)F)cc3)C2C1 CC(CCN(C)C(C1CN(C)C1)=O)NC(=O)OC(C)(C)C CC1(C)CN(C(C2CCC2)=O)CC(CNC(C23CCCCC2C3)=O)O1 C(C(C(=O)NCC1CN(CC)C(=O)O1)C(C)C)NC(CC=CCC)=O N1(C(C(=O)NCC2C(COC(=O)NC)CCC2)=O)CCC(OC(C)(C)C)CC1 n1(CC)nc(C(C)C)cc1C(=O)NCC(O)CN(C)C(C1(c2cccs2)CC1)=O c1(CN2C(c3cc(CC)c(C)o3)CCC2)cc(Cl)cc(Br)c1F C(=O)(C1(C)CCn2c(C)nnc21)NCC1C(NC(CCc2c(C)cccn2)=O)C1 C1C(C2CCC2)CC(=O)N1C1CC1.C(C(C)(C)C)NC(C1(OCC)CC1)=O C(=O)(CS(=O)(=O)C1CC1)N1CC(CC)N(C(=O)Cn2nc(O)ccc2=O)CC1 c1(C(=O)NCC(CN(C(=O)CC2COCCO2)CC)O)csc(CC(F)(F)F)n1 c1(OC)n[nH]c(=NC(C)C2CC2)cc1-c1ccc(C(F)(F)F)c(Cl)c1 CCCC(C(=O)NC)NC(=O)CCCCNC(C1(CC(=O)OC)CC1)=O N1(Cc2nc(C)oc2)C2CCCC1CN(C(=O)C(c1cnn(C)c1)C)C2 N1(C(C)=O)CC(C2CCCN(C(c3cncc(-c4c(OC)ccc(C)c4)c3)=O)C2)C1 C1(OC)CN(C(c2ccnc(CN(C)C)c2)=O)CC1NC(=O)Cc1cccs1 N1(CC#C)CCC(C(=O)NC2(CNC(=O)C(=C3CCCCC3)F)CCOC2)CC1 CC1(CNC(=O)COCC(F)(F)F)COCCN(C(C2(C)CCCCOC2)=O)C1 N1(C(C(C)C)=O)CCN(C)CC1n1cccn1.N12CCC(CC1)NC2=O c1(OC)ncc(F)cc1C(=O)NC1CC1CNC(=O)CCc1ccc(C)cc1 N1(C(C(C2CCC2)OCC)=O)CCC(C)(CNC(c2c[nH]nc2C(F)(F)F)=O)C1 N1(C(C(CC)CCOC)=O)CC23CCCC2(C1)CN(C(=O)Cc1scnc1C)C3 N1(CCC)CCCC(C(N2CCC(O)(CNC(c3ccoc3C(C)C)=O)C2)=O)C1 N1(C(CCC(=C)Cl)=O)CC(C(N2CCC(OCC)C2(C)C)=O)CCC1(C)C C1(CCC)(NC(=O)CNC(=O)NC)CCCN(C(c2cc(OC)ccc2Cl)=O)C1 C12(C(=O)NCC(C)NC(=O)CC3CC(C)(C)CO3)CCC(C)(CC1)OC2(C)C Cc1[nH]nc(C(=O)NCC(C)(C2CC2)NC(C2CCCC2C(C)C)=O)c1C CCC(C)CCC(=O)N1CC(NC(=O)CCC2(C)CC2(F)F)C(O)C1 C(CCC(C)C)(C(=O)NCCCC1CCOCC1)NC(CC1(C(=C)F)CCC1)=O N1(C(c2c(OC)cnc(F)c2)=O)CCC2(CC1)CC2CNC(c1cc(F)n[nH]1)=O CC1(C)CCCC1C(=O)NC1CCCC1NC(c1ccon1)=O C1(CC)CCCCCC1(c1nnnn1CCCF)NCC(c1cn(C)nn1)(C)C Cc1ncc(C(=O)NC2CN(C(c3cn(C)nn3)=O)CC2C)n1-c1ccccc1 C1(NC(C(C)NC(C=C(C)C(C)C)=O)=O)CCCCN1C(C)C.C1C(C)(C)NS1 C1(C(=O)NCC2CCC(NC(c3ncn(C(C)(C)C)n3)=O)C2)CC(S(N)(=O)=O)C1 N1(C(C=CSC)=O)CC2(CC2)CC1CNC(=O)Cc1sccc1Cl C(C(C)(C)CC(=O)NCCCNC(C1CC1(C)C(F)F)=O)OC(C)=O N1(C(C(C)OCCC=C)=O)CCC(C2CC2)(CNC(=O)COc2ccn(C)n2)C1 c1(CN)sc(C(C)NC(C(=O)NCc2c(C(=O)OC)non2)=O)cc1C C(=O)(CCCC(=O)C(C)(C)C)NCC1CCN(C(C(C)CCC(C)(C)C)=O)CC1 C(C(C)(O)CC(=O)N1CCC(Cn2cc(-c3ccc(Cl)cc3)nn2)C1)SC C1(C)(CNC(CC=CC=C)=O)CCCC1NC(=O)Cc1cccnc1F C=CCCCCCCCC(=O)N1CCCN(Cc2cn(CCOCC)nn2)CC1 CC1=CCC(C(=O)NCC2(C)CCCN2C(=O)C=Cc2cc(C)no2)CC1 c1(CC)nc(NC(CCN(C(=O)C2=CCS(=O)(=O)C2)C)C(C)C)c(C#N)cc1C N1(C(C=CC(CC)C)=O)CCC2(CC(C(N3CCCC(F)C3)=O)C2)C1 c1(C(N(C(C(N2CCCC2C2CCCC2)=O)C2CC2)C)=O)nnc(O)nc1O C1(OC)CC(CNC(=O)CC2CCCC23CC3)N(C(=O)C#CC2CC2)C1 C#CCC(C(=O)N1CCC(NC(c2cncc(C)n2)=O)C1C1CC1)C1CC1 N1(C(c2nc(CC)oc2)=O)CC=C(CCNC(c2cc(Cl)ncc2OC)=O)CC1 N1(C(CCCOCC)C(=O)NCCC2(C)CC2)CCC(C(=O)OC)C2(CCC2)C1 C(C)(C)(CC(C)(N=c1ccn(CCOC(C)C)[nH]1)c1nnnn1C)SC C1(N2CCC(C)CC2)(CNC(C)(C(=O)OCC)c2ccccc2)CCCCC1C C#CCC(C)(CC)C(=O)NCCC1CCCN1C(=O)CCc1cc[nH]n1 C=CC(CC)CC(=O)NCC=C1CCN(C(=O)CC2CC(C)(C)CO2)CC1 CN(C)S(=N)(=O)N1CCCC1C(=O)NC1CN(C(=O)C=Cc2cnc[nH]2)CC1O c1(C(=O)NC2CC(C)N(C(=O)Cc3cn[nH]c3)C2)cc(O)c2sccc2c1 Cc1ccc(Cl)c(C(N2CC(NC(c3n[nH]cc3C3CCC3)=O)CC2(C)C)=O)c1 C1(C(N(C2CCN(C(=O)COCC(=O)OC)C2)CCC)=O)OCCN(C)C1=O C1(C(=O)NCC2CC(NC(C(c3ccccc3)OC)=O)C2)CCC([N+](=O)[O-])CC1 C1(C)(CC)CCCN(C(=O)C(C)(CO)NC(C2CCCC(=O)CC2)=O)C1 N1(C(C2N(C(c3c(OC)ccc(I)c3)=O)CCOC2)=O)CCNCC12CCC2 CC(C(=O)NCC1(CC(=O)NCCOC(=N)O)CC1)n1cncn1 CC(CC(=O)N1C(C(=O)NCCOCF)CCC1C1CC1)C(C)(C)C C1(C(N(CC(C)NC(=O)C2=COCCO2)C)=O)CCCCC(=O)C1 N1(C(C)=O)CCN(C(c2cncc([N+](=O)[O-])c2)=O)CC12CCCC2 c1(CCC(=O)NC2CCCC2NC(c2ccc(Br)o2)=O)nnc(O)nc1O c1(C(N(C2CN(C(c3cn(C(F)F)cn3)=O)C2)C)=O)ccn(C)c1 c1(C(C(=O)N(CCCNC(=O)C(C)Cc2ccncc2)CC)C)ccc(C)cc1 C1(CNC(C23CC(F)(C2)C3)=O)CC2CC2N1C(C1(F)CCCCC1)=O Cc1ncc(CC(=O)NC(C2CN(C(c3ccncc3F)=O)CCO2)C)c(O)n1 C(C(O)CC(=O)N1CC(O)(c2cc[nH]n2)C1)C(=O)Cc1ccsc1 C#CCC(CC(F)F)C(=O)N1CCOCC(C(=O)NC(C)CC(C)(C)C)C1 CC1(C)C(=O)CC1C(=O)NC(C)(C)C=CC(=O)NCC1(C)CCCS1 C1(CNCC(C2CCC(F)(F)CC2)C)C(=O)Nc2ccccc2S1(=O)=O CC(CN(C)C)CCC(=O)N1CCC2C(C(=O)NCCC(=O)NC3CC3)C2C1 C1(NC(C=CCOC)=O)CCOC(C(=O)NCc2nonc2C)C1 Cc1[nH]c(C)c(C(N2CC(CNC(C3CCCOC3c3cn[nH]c3)=O)C2)=O)c1C CN=S(C)(=O)c1cccc(C(=O)NCCNC(=O)CC2OCCCC2(C)C)c1 c1(OC)ccc(CC(=O)NC2CCC2NC(c2cn(C)nc2C(C)C)=O)c(Cl)c1 N1(C(C2ON=C(C)C2)=O)CCCC(NC(C2(S(N)(=O)=O)CC2)=O)C1C C#Cc1cccc(C(=O)NCC2CC(C(=O)N(C3(CO)CC3)C)CO2)c1C C(CC(C(C)C)NC(=O)CS(=O)(=O)CC)N(C(COCC(=O)OC)=O)C C1(C(N(C)CC2CC2(C)C)=O)CC=CCN1C(c1cccnc1)=O C1(CC=CC)CCCN(C(=O)C(C2CCN(C(=O)C(C)c3ccsc3)CC2)C)C1 c1(C(C(=O)NCC=C)NC)cc(C)cc(C)c1O.C1CCCC(N2CCCC2)C1 C1(CNC(CC2(CC)CCCC2)=O)CN(C(c2nc(Cl)sc2C)=O)CCC1(F)F C1(C(=O)NC(C(=O)NC)CC2CCC2)CCC2(CC2)N1C(=O)C(C)CSC N#Cc1ncc(C(F)(F)F)cc1NC(C12CC1CN(C(=O)Cc1cc(Br)cs1)C2)=O c1(CC)cc(C(=O)NCCN(C2CCCC2)C(c2nnn(C)c2C)=O)c(C)o1 C(=O)(C(O)C1=CCCCC1)NCCCC(C(=O)NCCCc1n(C)ncc1)(C)C c1(NC(CNC(C2COCCO2)=O)C2CC2)ccn2ccnc2n1 c1(C(c2n(C)nnn2)NCC2CNCC(C)(C)O2)cc2ccc(Cl)cc2o1 C1(CC(=O)N(CCNC(=O)C(c2ccccc2)C2CC2)CC)COCC(C)(C)O1 C(C(N=[N+]=[N-])C(=O)NC1CCC(NC(c2ccnn2CC(F)F)=O)CC1)OCC c1(N(CCCC)C)ccc(C(=O)NC(CO)C(C)NC(=O)CCOCCC)cc1 c1(CC)nc(C)c(C(N2CCCC2CN(C)C(c2cc(CF)on2)=O)=O)s1 CCC(O)C(=O)NCC1CC(CNC(=O)C(C)Cc2cccnc2)C1 Cc1nc(NCC(C2CC2)N(C)C(C2CC3CCCC23)=O)cc2nncn12 C1(C2CCCCC2)(C(N(C2CC(NC(=O)CCNC(C3CCC3)=O)C2)C)=O)CC1 C1(OC)CN(C(=O)Cn2ncn(C)c2=O)CC1NC(c1ccc(Cl)o1)=O C1(n2cccn2)(NC(CCOCC)=O)CCN(C(=O)C(CCSC)OC)CC1 c1(CC)onc(C)c1SCC.C1CCC(C(F)(F)F)O1 C(C)(CCCCCO)NC(CC(CNC(c1cccc(CO)n1)=O)OC)=O c1(SCC(=O)NCCC(CNC(=O)CC2CCOC2C)OC)ccc(C)cc1C N1(C(C(C)N2CCCC2)=O)CCC(C(O)CNC(=O)CCCNC(N)=O)CC1 C12(C(=O)NCCC3N(C(c4cc(C(C)=O)oc4)=O)CCSC3)COC(CCO1)C2 c1(C(N(C(CCNC(CC(C)C)=O)C)C)=O)cncc(-n2cccn2)n1 C(C)(C)(C(=O)N1CC(c2ocnc2CNC(C2CCC(=O)N2)=O)C1)NC(=O)OC N1(C(c2c(C)cco2)=O)CCN(C(=O)C2CC2)C(c2cn[nH]c2)C1 C1(C(=O)NCc2n(C)ncc2)CCC2CCC1N2C(=O)Cn1ccccc1=O c1(C(=O)NCC(CNC(C(C)OCC#C)=O)(C)C)cnc(S)n1C C1(C)(C(=O)NCCSCC)CCCN(C(=O)CNC(=O)C(C)(C)C)C1 C(C)(CN=c1[nH]cnc(Cl)c1Br)N(C(C(C)CCN(C)C)=O)C N1(C(C2C(CC)OCC2)=O)CCN(C(c2ccc(COC)s2)=O)CC12CCC2 N1(C(C2(OC)CCC2)=O)CCC(CCNC(=O)C(F)=C(C)C2CC2)C1 C1(C(=O)NCc2n(C(C)C)ccn2)CCCC(NC(=O)C(C)c2cc[nH]n2)C1 c1(NC(C2CCNC23CCC3)=O)cccc(S(=O)(=O)NCC(F)(F)F)c1 c1(C(N2CCC3(NC(c4conc4C4CC4)=O)C(C2)C3)=O)cnc2ccccn12 S(=O)(=O)(C1CCN(C(c2cc(C)ncn2)C(=O)NCC2CC2)C1)NC C(C(CC(=O)N(CC(C)(C)O)C)NC(c1csc(F)c1)=O)OC c1(N2CCC(C)(OCC)C2)nc(N2CCC(N(C)CC)C2)c2ccc(C)cc2n1 Cc1sc(O)nc1C(=O)NC(C(=O)NCCc1cc[nH]n1)c1ccoc1 N1(C(C23CC(CN(C(C(CC4CC4)OC)=O)C2)C3)=O)CCC2(CCCCO2)C1 C(=O)(C1SCCc2ccccc21)N(CCn1cc(-c2nccc(OC)c2)nn1)C c1(OC)cc(F)ccc1N1CCN(C(=O)NC(c2cccnc2)CN(C)C)CC1 c1(OC)ncnc(C(=O)NCC(F)CNC(c2cn(CCO)nc2C)=O)c1F c1(C(=O)NCC(CC)NC(c2conc2C2CC2)=O)cnc2c(cnn2CC)c1 N1(C(C(C)Oc2cccc(C)c2)=O)CCC(NC(=O)C#CC2CC2)CC(O)C1 C12(C(=O)NC(CCC(C)C)C)CC(CO1)N(C(=O)CC(=O)N(C)C)C2 C1(C)(CNC(C2CN(C(C)C)C2)=O)CCN(C(c2c[nH]nc2-n2cnnn2)=O)C1 Cc1ccc(CN2CC(C(=O)Nc3csc(Br)c3)CC(F)C2)c(F)c1 Cn1cc(S(=O)(=O)NCC2(F)CCCN(C(=O)Nc3ccc(F)c(F)c3)C2)cn1 C1(C(N2CC(C)(CNC(c3cccnc3O)=O)OCC2)=O)CN2CCCN1CC2 C(=O)(C(C)OC1CCCC1)NCC1(CN(C(COC(C)C)=O)C)CC1 C12(CNC(c3c(C)nc[nH]3)=O)CN(C(C3(C)CCCCC3)=O)CC1CCO2 C(=O)(C(O)CC(F)(F)F)NCCOCCNC(C1CCCOCC1)=O c1(C(N(C(CNC(=O)CCC2CC(F)(F)C2)C2CC2)C)=O)ccc(O)c(F)c1F c1(C(N2C(CNC(C3CCNC(=O)C3)=O)CC(OC)C2)=O)ccc2c(c1)CCN2 Cc1ncc(CC(C)C)cc1-c1nc(C2(C)CC2)nn1CCCC(C)C Cc1ccc(=N)[nH]c1C(N1CCC(C)(CNC(C2(C)CC(C)C2)=O)C1)=O c1(CN(CC(C)(C)O)C(=O)NCCN2CCCCC2)ccc(F)cc1F C=C(C)C(CC(=O)NC1CCC(N(C)C(C2CCC(F)(F)CC2)=O)CC1)OCC N1(C(c2n(C=C)nnc2)=O)CCC2CN(C(C3(C)CC(C)(C)C3)=O)CCC2C1 CC(C)(C)C(CNC(c1cn[nH]c1)=O)C(=O)NCC1CCCC12CC2 C1(C(N2CC(N(C(C3CC(OCC)C3)=O)C)C2)=O)COCCO1 C1(C(C)C)CN(C(c2ccc(-c3cn[nH]c3)cn2)=O)CCN1C(=O)C(C)C1CC1 C1(C(N2CCC(CNC(=O)Cn3cccnc3=O)CC2)=O)(OC)CCCOC1 Cn1c(C(N2CCC(C)(O)C(C(=O)O)C2)=O)nc2cc(Br)ccc12 N1(C(C=Cc2ccc(C)cn2)=O)CCC2(NC(=O)CS(N)(=O)=O)CCCCCC12 n1(C(C)C)ncc(CNC(C2CN(C(=O)OC(C)(C)C)CC2CO)=O)c1F c1(C(N2CCC(C)(CNC(C3CC(=O)C3)=O)C2)=O)c(Cl)oc2ccccc12 CC1(NC(=O)CCc2nnc(C(F)F)o2)CCCN(C(C2CC2F)=O)C1 C1(OC)CC(CNC(=O)C(C)(C)c2ccn(C)n2)N(C(c2cnc(C#N)s2)=O)C1 N1(C(C(C2CC=CCC2)NC(CN2C(C)CCC2)=O)=O)CC2CCCC2C1 N1(C(C(=O)OC)=O)CCn2ncc(CNC(c3csc(C)c3)=O)c2C1 N1(C(c2c(SC)ccc(N)c2)=O)CC2CC(NC(c3c[nH]nc3C)=O)CC1C2 N(C(=NCCc1ccccn1)NCC1CCOC1)C(CC)C C=CC(CCC)CC(=O)NCC1(CNC(C2Cc3ccccc3O2)=O)CC1 c1(C(C)C)conc1C(c1nnnn1C)NCCn1cnnn1 N1(C(C2C(C(C)C)CCC2)=O)CCN(C(C23CC=CCN2CCC3)=O)CCC1C C1(O)(CNC(C2(C)CC2(F)F)=O)CCCN(C(c2cncn2C2CC2)=O)CC1 N1(C(C2N(C)CC2)=O)CCCC1CC(N1CCC(CC2CC2)C1)=O C(=O)(C(=O)N=S(C)(C)=O)N(CC(C)NC(=O)C(c1ccc(F)c(F)c1)O)C C(C)(CC(=O)NCCC1CCN(C(c2cnc(S)n2C)=O)C1)(C(F)F)N(C)C C1(NC(c2cnc(O)s2)=O)CC2(C1)CC(NC(C1(CC3CC3)CC1)=O)C2 C1(C2CCCCC2)(C(C)(C)C)CC1.c12ccnc(n1)NC(=O)NCCO2 c1(C(=O)NCC2C(OCC)CN(C(c3n[nH]cc3CC)=O)C2)cc(C#N)cn1C c1(C(N(C2COCC2CNC(C2CCC(C)(F)CC2)=O)C)=O)ccc(F)cc1F c1(OC)ccc2[nH]cc(C(=O)NC3CN(C(=O)Cc4coc(C)n4)C4CC34)c2c1 c1(OC)ccc(Br)cc1C1(C(=O)NCC(C)NC(=O)C2=CCSC2)CC1 c1(C(N2CCOC2)COC)ccc(Br)nc1[N+](=O)[O-] N1(C(C(C(C)C)C2(C)CC2)=O)CCCCC2(C1)CN(C(c1cnc(O)n1C)=O)C2 S(=O)(=O)(c1nccs1)NCC1CCC(C(=O)NCCc2ccc(Br)s2)CC1 N1(C(C(C)=CC=C)=O)C(C(=O)NC2(C(C)C)CCC2)CCC1C(C)C c1(C(=O)OC)ccc(NCC2CCC(OC)CC2)c(C#N)c1 CN1CCc2[nH]nc(C(N3CC(CNC(c4ccc[nH]4)=O)C4CC34)=O)c2C1 c1(CC(=O)NC2CC3C(NC(C(C=CC)O)=O)C3C2)ccc(F)c(F)c1 C(=O)(C(=O)C(C)(C)CC)N1CC(CC=C)(NC(C2CC(N=[N+]=[N-])C2)=O)C1 N1(CC2CCC(C(=O)OC)C2)C(=O)NC(C)(c2ccc(F)cc2)C1=O N1(C(CC)=O)CC(C2CCCN(C(=O)C=CCN(C)C)C2)C1 N(C(=NCCCF)NCCC=C=CC)C(c1cccc(Cl)c1)C#C c1(C(C)NC(=O)NCC2(c3ccccc3Cl)CC2)ccc2c(c1)CC(C)O2 C1(C(N(CC(=O)OCC)C)=O)CCN(C(=O)CCOCC(F)F)C(C)(C)C1 c1(CNC(C2(O)CCN(C(c3ccc(OC)nc3)=O)C2)=O)ccc(F)cc1Cl Cc1nccc(N2CC3CC2C3C(N2CCC2c2ccccc2)=O)n1 CC1(NC(C2(CF)CC2)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)C1 C1(NC(C(C)OCC=C)=O)C2COCC1CN(C(C1CC3CC(=O)C1C3)=O)C2 c1(OC)ccc(NC(=O)C(=O)NCc2ccc(Cl)cc2)c(C)c1 c1(OC)ccc2ccc(NC(C3CC(C4CC4)=NO3)=O)cc2n1 C1(NC(c2c(SCC)cc(Br)cc2)=O)CC2(CCC(C)(C)CC2)C1 C(=O)(C1CNC(=O)c2ccccc21)NCC1CCC(NC(C2C(=C)CC2)=O)CC1 CCC(CNC(=O)C(C(C)C)NC(=O)Cn1ccnn1)C(C)(F)F c1(OC)ccc(Cl)c(C)c1C(=O)NC1CC(N(C(=O)CN(C)C2CC2)C)C1 c1(C(=O)NCC2C(C)CN(C(c3cscn3)=O)CC2)ccc(C#CC2CC2)cc1 C1(NC(CC(=O)NCC2CC2)=O)CCOC12CCN(C(=O)C=CBr)CC2 c1(C(=O)NC2CCC(C)(NC(C(CC)O)=O)CC2)cn2cccc(F)c2n1 C1(CNC(C=CSC)=O)CCN(C(=O)CC23CCCC2C3)C12CC2 C1(CNC(C2(O)CCN(C(=O)CC(F)(F)F)CC2)=O)CC1C1CCCCC1 N1(C(C(C)C(F)F)=O)CCCCC2(C1)CN(C(=O)Cc1sccc1Cl)C2 C1(NC(CC(=O)NCC#C)=O)CCCN(Cc2nc(CCC(C)C)no2)C1C c1(CNC(N2C(CN(C)C)C(C)(C)C2)=O)ccnc2c1ncn2C C1(NC(c2c(CC)[nH]nc2Cl)=O)CCCCCN(C(C2CC(C)(CC)C2)=O)C1 C1(N(C(=O)COCC(F)(F)F)C)CCC2(CC1)CCN(C(=O)CC1C=CCC1)C2 C(=O)(C1=CCC(C(F)(F)F)OC1)NCCN(C(c1n(CC)ccc1)=O)C1CC1 C(CCC(=O)NC(c1cnn(C)c1)C(=O)NC(c1nc[nH]n1)C)OC(C)C c1(C(=O)NC2CCCC(CNC(CN(C)C)=O)C2)cncc2c1CCC2 Cc1c(C(=O)NC2CCN(C(c3cnncc3O)=O)C(C3CC3)C2)cncc1Cl C1(CNC(CC=C)=O)CC2(CO1)CN(C(=O)CCCC(OC)c1ccccc1)C2 c1(C(n2cc(CN(CCO)C(C3CCCN3C)=O)nn2)C)ncccn1 c1(C(C(=O)NCC2(NC(=O)CCCc3cncs3)CCC2)SC)cccc(Cl)c1 Cc1cc(C(C(F)(F)F)OC(c2ccc(N3N=CCC3=O)cc2)=O)cc(C)c1 C(CCCCCNC(C1C2CCCCC12)=O)N(C(C1OCC(C)C1)=O)C C1(C(=O)NC2(CNC(C3CC(C)(O)C3)=O)CC(OC)C2)CC2CCC1C2 C1(C(=O)OC)CCC2C(=O)N(c3c(CCC(=O)N(C)C)ncn3C)C(=O)N2C1 CC(C)C(C(C)NC(C1CC(N(C)C)C1)=O)NC(c1cncc(O)c1)=O c1(C(=O)NCC(CCOC)NC(=O)C(C)(F)C(=O)OC)c(F)ccc(C)c1Cl C#CC1CN(C(C2CCCN2C=O)=O)CCN1C(=O)C=CCOCCOC c1(C(N2CCN(C(C=C3CCC(C)(C)CC3)=O)CC2)=O)noc2c1CCCCC2 c1(C(=O)NC2C3CN(C(C(CC)(F)F)=O)CC32)cnc(CC(C)C)nc1O C(=O)(C(CO)C(C)(C)C)NC1C(C)(CN(C(CC(=C=C)C)=O)C)CCC1 C1(OC)CCCC1N=c1cc(C)[nH]c(=NCc2c(N)cccc2F)[nH]1 c1(CC(=O)NCC(CC(C)C)NC(=O)C(C)CC(C)(F)F)cc2ccccc2o1 N1(C(C2C(C)(C)C2(F)F)=O)CCC(C2CN(C(c3ccnc(O)c3)=O)C2)CC1 C(CC(C(C)(C)C)NC(c1cnc(O)o1)=O)N(C(=O)CC1(O)CCCCC1)C c1(C(=O)NC2CN(C(=O)C(=O)Nc3ncc[nH]3)C3CC23)coc2c1CCCC2 c1(CC(=O)Nc2c(C(=O)OC)cc(F)c(F)c2)cccc(F)c1[N+](=O)[O-] C12(NC(C(CC)OC3CCCCC3)=O)CC(CNC(C3(C#N)CC3)=O)(C1)OC2C C(C)(CCCCO)NC(C1CC(C)(NC(CCNC(COC)=O)=O)C1)=O S(=O)(=O)(c1cncc(C(F)(F)F)c1)NCC1CCC(NS(C)(=O)=O)CC1 c1(SCCC(=O)N(C2CCN(C(=O)C(C)Cn3ccnc3)C2)C)ccccn1 c1(C(C(=O)NCCNC(C(CC)=CCCC)=O)C)ccc(Cl)nc1 N1(C(=O)NCC)CCN(Cc2ccc(-c3onc(-c4scc(C)c4)n3)cc2)C2CC12 C1(C(=O)NCC2C(C)(C)CCCO2)CCCN1NC(=O)C(=O)NC1CC1 N1(C(C(C(CC)C)O)=O)CC(C)OC2(CCN(C(=O)CC3CC4CC4C3)C2)C1 N1(CC(C)NC(=O)C(O)CNC(=O)CC2CCN(C3CC3)C2)CCCC1=O c1(C(=O)NC(C)CCCNC(=O)C(O)CC(F)(F)F)ccc2ccccc2c1 c1(C(=O)NCCCCCN(C(=O)CC(C)(C)C(F)F)C)ccc2c(n1)CCOC2 c1(CCC)ccc(C(C(=O)NCC)N(C2CC(F)(F)C2)C)s1 Cc1c(C(N2CC(NC(C34CC(F)(C3)C4)=O)C2)=O)cc(S(N)(=O)=O)cc1[N+](=O)[O-] c1(OC)ccc(C=CC(=O)NC(C)CNC(C2(F)CCC2)=O)cc1Cl CCC(CNC(=O)C(O)Cn1cncn1)(CC)C(=O)NCc1nccn1C(C)C N1(C(Cn2ccc(C)n2)=O)CCC(C(=O)NC(=O)CSc2cn[nH]c2)C1C CC1CN(C)C(C)CN1.c1(C(=O)C(F)(F)F)csc(=NCc2cc(Br)cnc2F)[nH]1 c1(C(N2CC(CNC(c3cc(C)[nH]n3)=O)C(C)CC2)=O)ccc(C)c2c1CCC2 C1(C(=O)OC)(CN2C(CN(C(=O)Cc3n[nH]c(C)n3)CC)CCC2)CCCCC1 N1(C(C(=O)NCCCC)CCC2CCOCC2)CC(C2(O)CCC2)C12CCC2 CC1(C(N2CC(C(N)=O)(CNC(c3cccnc3)=O)C2)=O)CCCS1 c1(OC)cnc(C(=O)NC2CN(C(=O)CCCc3cccs3)CCC2O)c(F)c1 N1(C(CC)CC)CC(C(=O)NC23CC(C2)N(C(c2cc(=O)n(C)o2)=O)C3)CC1=O c1(N(C)CC2CC=C(C)CC2)ncc(C)cc1S(=O)(=O)N1CCC1 C1(CNC(CC(CCC)C)=O)CN(C(=O)CC2CC=CCC2)CC(C)(C)O1 c1(N2CC(CN(C)C(C3CC34CC(O)C4)=O)OCC2)ncnc(Cl)c1C(C)=O C1(CNC(CCC(=C)C)=O)(NC(=O)C(C)CC(C)C)CCC(F)(F)CC1 C1(NC(C(CNC(C)=O)(C)C)=O)CCCN(C(=O)CC2C=CCC2)CC1 n1(CCC)ncnc1CNC(=O)C=CC(C)NC(C1CC2CC2C1)=O c1(C(=O)NC2CC(OC)CN(C(CCC(C)OC)=O)C2)ccc2c(c1)CCCO2 CCCCCCC(C)C(=O)N1CCC2CCC(C1)N2C(=O)C(C)CCO C1(CN(C(C=CC(CC)=CC)=O)C)CCCN1C(c1cc(C)[nH]n1)=O CC1CCS(=O)CCN1C(=O)Cc1cccc(C(F)F)c1 N1(C(C2(OC)CCN(C(CCCCCC)=O)C2)=O)CCC2(COC(=O)N2)C1 C(=O)(C#CC(C)(C)C)N1CCC(c2c(CNC(C3(CCC)CC3)=O)c[nH]n2)C1 C1(NC(c2c(Cl)cc(C)nc2)=O)CCN(C(c2ncc(Cl)s2)=O)C12CCCC2 CCC(C)CC(CO)NC(=O)CCC1(NC(c2cnsc2)=O)CCCC1 C1(N(C(C2CN(C)C(=O)N2)=O)C)CN(C(=O)COc2cccc(O)c2)CC12CC2 c1(CC(=O)NC2CC(CCNC(CC(CC)C3CCC3)=O)C2)ccc(F)cc1F c1(CC(=O)NC(C)CNC(=O)C(C)(C)Cc2cnn[nH]2)ccc(-n2cccc2)cc1 N1(C(c2occ(C)c2)=O)CCC(F)(CNC(C2CCCCN2C(N)=O)=O)CC1 C(=O)(C(O)C(C)(C)C)N(CCCNCC(=O)NC(C(CC)C#N)=O)C1CC1 c1(OC(C)(C)C)ccc(OCC(=O)NCCNC(C2(C)CC2(F)Cl)=O)cc1 C(c1ccc2c(c1)CCO2)=CC(=O)NC1C(OC)CC(F)(F)C1 N1(C(C(CC=C=C)NC(=O)CN(C)C(=O)OCCOC)=O)CCC(O)C(F)(F)C1 C12(C(=O)NCCC3CC(NC(=O)C(O)CC(F)(F)F)C3)C3CCC(CC13)C2(F)F C(=O)(CCC(CC)OC)N1CC(CCC)C(NC(C(Cn2cncn2)CC)=O)C1 CC1(C)CCC=C(C(=O)NC23CC(CNC(=O)C#CC4(C)CCCO4)(C2)C3)C1 c1(C(=O)NC(CNC(CC2C(C)CCC2)=O)C)c(F)c(F)cc(F)c1F c1(NCC(C)S(N)(=O)=O)cc(S(=O)(=O)NCC2(N(C)C)CCCC2)ccc1C#N C(c1cc(F)c(F)c(F)c1)=CC(=O)N(c1ccc(NC(=O)OC(C)(C)C)cc1)C1CC1 c1(C(=O)OCC)ccc(C(=O)NCCCCC(C)NC(=O)CN(C)CC)nc1 C#CCCC(O)C(=O)N1CCOC(CCNC(=O)CCNC(=O)C(C)(C)C)C1 C#CC1(C(N2CCC(CCN(C)Cc3cn(C)nc3CC)CC2)=O)CCCC1 C(=O)(C(C)CC(C)C)N(C(C(NOC(COC)COC)=O)C)C c1(CNC(C2CC(=O)NC2)=O)cccc(CNC(c2ncc(Cl)s2)=O)c1 c1(NC2(C)CC(NC(CCCN(CCC)C(C)C)=O)C2)ncc2c(ncn2C)n1 N1(C(C(C(C)(C)C)O)=O)C2CCC1CN(C(=O)CC1OCCCO1)CC2 C1(CNC(=O)COc2cn[nH]c2)CC2(CCC2)CN1C(C1C=CCCC1)=O Cc1cnn(CCC(=O)NC2CC(NC(C3CC34CCC4)=O)C2)c1 N1(C(CC(C=C)(C)C)=O)CCC2CCN(C(c3cc4c(cn3)OCCC4)=O)CC12 C12(NC(CCC(=O)N(C(C)C)C)=O)CC(CNC(C3(C)CC3(Cl)Cl)=O)(C1)OC2C c1(C(N2CCC(CN(C(C(C)c3ccco3)=O)C)CC2)=O)cc2n(n1)CCCN2 Cn1ncc2ncnc(N3CC(F)CC3C(=O)Nc3ccc(F)cc3[N+](=O)[O-])c12 CCCC(CCNC(=O)C(CC1CCCC1)NC(=O)C(C)N1CC(C)C1)CCC C1(CCCC(=O)NC(C)CC2CN(C(=O)C(=O)N(C)C)C2)CCCC(=O)N1 C1(O)(C(=O)NC(C=CC(=O)N(C2(C#C)CC2)C)C)CCCC1 n1(CCC(=O)NC(CC)CN(C)C(C2COC2)=O)sc2ccccc2c1=O C1(N(C(=O)CC2CC2C2CC2)CC)CCN(C(=O)C=CC(=O)OC(C)(C)C)CC1 c1(CCSC)nc(-c2cncc(-n3cccc3)c2)n(-c2cccnc2)n1 N1(C(c2cc(C)sc2C)=O)CCCCCC1CNC(=O)CCc1cn(C)nc1C c1(CC)cccc2sc(NC(=O)NC(c3ncc(-c4ccc(F)cc4)o3)C)nc12 C1(NC(Cc2c(C)noc2)=O)CCN(C(=O)COc2ccc(Cl)nc2)CC(O)C1 CC(C(F)(F)C(F)(F)F)=CC(=O)NCCCOCCNC(=O)CSC(F)F C1(C(=O)NCC(CNC(CC(C)OC)=O)(C)C)CCS(=O)(=O)N1C N1(C(C=CCC(C)(C)NC(C(C)OCC=C)=O)=O)CCN(C)CC1CCO N1(C(C(C2CCCCC2)OC)=O)CCN(C(=O)CC2(O)CCC2)C(COC)C1 N1(C(CN(c2ccccc2)C)=O)CCC2CCC(C1)N2C(=O)CCCC1CC1 C1(CNC(c2cc(C(=O)OC)sc2)=O)CC(C)N(C(c2cc(C(N)=O)no2)=O)C1 Cc1nc(N(C)C)sc1C(N1CC(C)(NC(=O)CC2CC(N(C)C)C2)C1)=O Cc1ccc(N)c(C(N2CCC(NC(=O)C(C)(C)C)C2c2ccccc2)=O)c1 c1(C(=O)NC2C(NC(CCC(N)=O)=O)CCOC2)cncc2cccnc12 N1(C(CCc2c(C)noc2Cl)=O)CC2=C(C1)CN(C(=O)C(C)C(O)C(C)C)C2 c1(NC(C2(CN)CCO2)=O)ccc(-c2cnco2)cc1 c1(C(=O)NCCCNC(Cc2cncc(C)c2)=O)ccc2cnccc2c1 c1(C(=O)NCCCCNC(COc2ccc(C)cc2)=O)nn(C)c2c1CCC2 C=CC1(C(=O)NCC2CC(NC(=O)C(CC(C)C)OC)C2)CCCCC1 c1(CC)nc(C)[nH]c1C(N1CCC(F)(CNC(=O)COCC2CCC2)C1)=O C=C(C)C1OCCC1C(N1CCC(F)(C(=O)N(CC)Cc2ccccn2)CC1)=O c1(OC)ncc(Cl)cc1C(N1CCC(CCNC(=O)CC2CCCCN2C)C1)=O c1(OCC(=O)NCC(C)N(C)C(c2csc(CC3CC3)n2)=O)ccc(O)cc1 C1(C(=O)NCC(C)(CO)NC(=O)Cc2n[nH]c(C)n2)(CC)CNC(=O)C1 c1(OCC)cc(C(N2CCCN(C(=O)CN3CCS(=O)CC3)CC2)=O)oc(=O)c1 c1(C(N2CC(C)C(CNC(C3COC(=O)O3)=O)CC2)=O)n[nH]c2c1CCSC2 CCC(C(=O)OC)C(=O)NCCCN1CCN(C(C2CNC(=O)O2)=O)CC1 N1(C(C=CC=CC)=O)CCCC(NC(C2CCCC2(C)C)=O)C1C N1(C(C2(COC)CCCO2)=O)CCOC2CN(C(C3(C#N)CCCC3)=O)CC12 Cn1cnc2[nH]c(C(N3C4CCC3CC(NC(=O)CCC(F)(F)F)C4)=O)cc12 C(=O)(CC(C)C(F)F)NCCN(CC(C)O)C(c1nc(C2CC2)ncc1Cl)=O S(=O)(=O)(c1ccc2nc(N3CCS(=O)C(C)(C)C3)cnc2c1)NCC(CCC)C C(CCC(C)(C)NC(c1cnc(OC)s1)=O)NC(CC=C)=O C1(C(=O)NCC2(C(=O)NC(C)Cc3ccnn3C)CC2)(N)CCCC1.C1CC1 C1(C(=O)NCCCCn2cc(C3CC=CCC3)nn2)CC2CCC(C1)O2 C1(C(=O)OC)C2CN(C(c3cnn(-c4ccc(F)cn4)c3)=O)CC12 CCCCC(C(=O)NC)NC(C1COCCN1C(=O)C(c1ccn(C)c1)C)=O c1(C(N2C(CNC(c3ccc(C)cc3)=O)C3CC3C2)=O)cc2sccc2n1C c1(C(=O)NCC2CC(NC(C(C)=C(CC)C)=O)C(O)C2)ccc([N+](=O)[O-])[nH]1 c1(CNC(=O)NC(C(c2ccccc2Br)OC)C)ccc(C)nc1O c1(NC(C2(C)CCN2C(=O)CCCCCBr)=O)cccc2c1CC(=O)N2 C1(NC(c2cc(CC)oc2C)=O)CCN(C(C2CCN2CC)=O)C(C)C1 N1(Cc2cn(CC(C)O)nn2)CCCC(NC(C2(C)CC2(Cl)Cl)=O)C1 CC1(C)CCC(CNC(c2cccnn2)=O)N(C(c2cnns2)=O)C1 c1(C(=O)NCC2CCCN2C(C2(c3cccnc3)CC2)=O)ccc2cc[nH]c2c1 Cc1ccc(C(N2CCC(N(C(=O)C#CC(C)(C)C)CCO)C2)=O)c(=O)n1C C1(CNC(C2(C)CC2(Br)Br)=O)CC(NC(=O)CNC=O)CC1O C1(C(=O)NC2(CC=C)CC2)CC(O)CN1C(=O)CC(C)SCC C1(C)(C(=O)NCC(CCOC)NC(=O)Cc2ccc(C)cc2C)CC2CCC1O2 c1(C(C)C2CC2)ncc2c(n1)CC1CCC2N1S(=O)(=O)C1CCN(C2CC2)C1 Cc1ccc(C(CNC(C2(F)CC=CC2)=O)NC(C2COCCO2)=O)cc1 Cc1nc(O)[nH]c1C(=O)NC1(C2CCCCN2C(=O)CC2C(C)(C)C2(C)C)CC1 C=CC(CC)C(=O)N1CCC(CN(C(=O)Cn2c(C)ccc2C)CC)CC1 C(=O)(C1=CCC2(COC2)OC1)N1CCOCC(CNC(CCCNC(C)=O)=O)C1 CC1CCCCC1C(=O)N(C1CCN(C(=O)CC(=O)Nc2nccs2)CC1)CC N1(C(c2c(C)n[nH]c2)=O)CC(NC(c2cccc(C(F)(F)F)c2C)=O)C(C)(C)C1 c1(C(=O)NCC(CNC(C2CCSC2)=O)C(F)(F)F)cnnc2ccccc12 c1(C(c2nc(-c3ccccc3)no2)N(C(COC2(C=C)COC2)=O)C)ccc(F)cc1 N1(C(C(c2cn(C)nc2)O)=O)CCN(CCNC(c2coc(CO)c2)=O)CC1 c1(NC(CC2(C)CC2)=O)cccc(SCC2CC2CNC(=O)COC(F)F)c1 c1(C(=O)NCCCNC(c2cnc(Cl)[nH]2)=O)cnnc(-c2ccccc2)c1 c1(C(N(C(c2ccccc2OC)C(=O)OCC)C)=O)ccc(SC)c([N+](=O)[O-])c1 C1(CC)(NC(=O)Cc2occc2C)CCN(C(C2(C(F)F)CCOCC2)=O)CC1 C=C(C)CCCNC(C1CCN(C(C2CC2NC(C)=O)=O)C1)=O N1(C(C2(OC)CC2)=O)CCCC(C2CCN(c3c(C#N)ccc(C)c3[N+](=O)[O-])C2)C1 c1cccc(C2COC2)c1.c1(C2(C(N3CC(CN(C)C)C3)=O)CC2)cn(C)nn1 C1(NC(c2c(C)ccn2C)=O)CN(C(=O)C2=COCCO2)CC1N=[N+]=[N-] c1(C(C(C)C)N(C(c2cc(CO)[nH]n2)C(=O)NCC2CCC2)C)cccc(Cl)c1 N1(C(=O)NCc2cc3n(c2)CCCC3)CC2CC3CC(C2)CC1C3 c1(CC)onc(C(=O)NCCc2cn(CCCCC(=O)O)nn2)c1C N1(C(C(C)(C)C(F)(F)F)=O)CCCC(C2CC2NC(=O)C2=CCCCO2)C1 c1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CC2)nc2sc(C)cn2c1C Cc1cncc(C(N2CCN(CCNc3ccc(C)[nH]3)CC2)=O)c1 c1(NC(C2(C)N(C(Cc3cccc(C)n3)=O)CC2)=O)ccc2c(Br)nn(C)c2c1 Cc1ccc(N)c(C(=O)N(CCCCNC(c2cnn3ncccc23)=O)C)c1F N(C1CCOc2ccccc21)C(C(C)OCCN=c1[nH]cc(C#N)o1)=O c1(C(N2CC3C(N(c4nccc(C(=O)OC)n4)C)C3C2)=O)ccc2ccnn2c1 C=C1CC2CC1CN2C(C12CN(C1)C2=O)=O.C1(C)(COC)CC(F)(F)C1 C12(CNC(c3ccn(CC)c3C)=O)CC(NC(=O)C3=CCSC3)(C1)C(C)O2 c1(C(=O)NCC(CN(C(CC(CCC)O)=O)C)O)c(F)ccc(Br)c1C Cc1ccc(C(CNC(=O)C(C)O)NC(=O)C(C)(C)c2ccno2)cc1 CCC(C)C(CC(=O)NCCc1ccnc(O)c1)NC(C1CC(=O)CS1)=O c1(C2C(=O)N2)ccc(Br)c(OC)c1.C(=O)(C(C)N(C1CCCC1)C)OC c1(C(=O)NC2(CO)CCN(C(CC(CC)C)=O)C2)ncc(C#N)cc1Cl C1(C(=O)NC(CC)C)C=CCN(C(c2cc(Cl)cn2C)=O)C1 Cc1ccc2c(c1)CCC(C(=O)NC(C)CNC(C13CC(F)(C1)C3)=O)O2 N1(C(C(C)(O)C2CC2)=O)CCN(C(=O)Cc2cccc(F)c2F)CC1CF C(C(CC(C)C)C(=O)O)NC(=O)NCc1c(OC)cc(F)cc1 N1(C(c2c(C)n(CC(C)C)nc2)=O)CCCCC12CN(C(=O)COCCCF)C2 C1(C(=O)NCCC2CN(C(c3cncc(C)n3)=O)C2)Cc2nccn2C1 C(CCCCCC(=O)NC(C)(C)CCF)NC(c1cc(C(C)C)[nH]n1)=O CC1(C(=O)NCC2CC2)CS(=O)(=O)C1.C12COCCN1C1CCCC1CNC2=O c1(-c2ccc(C(=O)NCC(C)N(C(C(CC)N(C)C)=O)CC)o2)ccccc1F C(=O)(C1=CC2CCCCCC12)N1CCC(CCNC(c2cccnn2)=O)CC1 C1(O)(C(=O)NC2CCC(NC(C3(CO)CC3)=O)CC2)CCCCCC1 CN1CCC(CN(C(=O)C(c2cnn(C)c2)NC(c2cc(CCO)on2)=O)C)C1 Cc1ncc(CC(=O)NCC2C(C)CCN2C(=O)CC2(C)CC(F)(F)C2)c(O)n1 C1(C#N)(C(=O)NCC(CC(C)C)NC(=O)C(C)C(C)O)CCCOC1 CC1CN(C(C2CCN(C)CC2)=O)CC1CNC(c1ccc(-c2cccs2)o1)=O N1(C(c2c(C)[nH][nH]c2=N)=O)CCC2(C1)CN(C(c1ncsc1C1CC1)=O)C2 N1(C(C(CC(=C)C)C)=O)CCC2(CCC2NC(=O)CC2=CCCCC2)CC1 S(=O)(=O)(c1ccc(NCC(C)OC(C)(C)C)c(C#N)c1)N1CC(C)SC1 c1(C(=O)NCCOC2CN(C(CCC(C)OC)=O)C2)cc(C)cc2ccncc12 c1(C(=O)NC2CC(CNC(C3(C)CCCC3(F)F)=O)C2)ccc2c(c1)CNC2=O S(=O)(=O)(c1ccccn1)N1CC(CNC(c2cc(OC)c(O)cc2)=O)OCC1 Cc1cc(C)c(CN(C=O)C(c2ccc3nnnn3c2)=O)c(C)c1 CCC(C)(C)COC.N12CCC1C2NC(C1CN(C(=O)OC(C)(C)C)C1)=O c1(C(N(CC(C)NC(C)=O)C)=O)c(Cl)ccc(Cl)c1O C1(O)(CNC(CSCCC)=O)CCN(C(=O)C(n2ccc(C3CC3)n2)C)C1 c1(CCC)ccc(NC(=O)C(c2ccco2)NC(C2CC3CC3C2)=O)cc1 c1(CC(=O)NC(CNC(c2c(OCC)ccc(C)c2)=O)C)cn2c(C)csc2n1 C1(CC(=O)NCCC2CCN(C(=O)Cc3cc[nH]n3)CC2)CCCC2(CCC2)O1 c1(NC(CN(CCCNC(C2CC(OC)(OC)C2)=O)C)=O)ccccc1CO C1(NC(C(CCNC(c2ccn(C(C)C)n2)=O)OC)=O)CN(C)CCN(C)C1 CC#CCC(C(=O)NCC1CC[Si](C)(C)C1)NC(=O)C=Cc1cc[nH]n1 C1(C(N2CC(COC)C2)=O)C2CC3C(C2NC(C2(C(C)(F)F)CC2)=O)C13 C1(CC(N2CC(C)(CC(=O)NCC(C(C)C)O)C2)=O)CCCOCC1 Cc1cc(Cl)c(Cl)cc1C(N1CCN(C(=O)Cc2ccc(F)c(Br)c2)C2CC12)=O Cn1nc(C(=O)NCCC(O)CNC(C2(F)CCCOC2)=O)cc1Cl N=c1nc(O)cc(C2CCN(C(C3CC3C(=O)Nn3cccn3)=O)CC2)[nH]1 N1(C(c2occ(C)c2C)=O)C(CNC(c2coc(Cl)n2)=O)CC2CCCC12 N1(C(Cn2nc(C)c(Cl)c2)=O)CC23CCCCC2(C1)CN(C(C1CC12CC2)=O)C3 N#Cc1cccc(CCNCC(c2ccccc2Cl)O)n1 c1(CNC(CCNC(CCCC#N)=O)=O)ccc([N+](=O)[O-])o1 C1(C(=O)NCC2N(C(CC3CCC(OC)CC3)=O)CC2)Cc2cscc2C1 C1(NC(C(C)OCCC#C)=O)CC(C)(CNC(c2ccccn2)=O)C1 C1(C(C)C)CN(C(c2ccoc2C2CC2)=O)CCC1NC(=O)C(=O)C(F)(F)F Cn1c(C(=O)NC2CCC2NC(=O)C(F)n2ccnc2)ccc1C#N C=CCCC(C(=O)N1CCN(C(C)=O)CC1)NC(C1CC(F)(F)C1)=O C1(CCN(C)C)CN(Cc2nnc(-c3cccc(-n4cccn4)c3)o2)CCCO1 C1(CCC)CN(C(=O)CCC2CC2(F)F)CCN1C(=O)Cc1nnc(C)o1 CC(C(=O)NC1CN(C(c2cc(-c3cccnc3)n(C)n2)=O)CC1O)C(F)F Cc1nn(C)c(Cl)c1C=CC(=O)NCC1CCN(C(c2ccccn2)=O)C1(C)C c1(C(N(C2CN(C(C(C)OCCC=C)=O)CC2(C)C)C)=O)ccnc2[nH]nnc12 N1(C(=O)CC2CCN(C(C3CCCC(C4CC4)O3)=O)C2)CCOC2(CC2)C1 N1(C(C(C)NC(=O)NC)=O)CCCC(NC(=O)CC2CCOCC2)CC1 c1(NCc2ccc(C(=O)O)cc2F)cnc2cccnn12.N12CC3CC3(C1)C2=O N1(C(CC2CCN(C)CC2)=O)CCCC2(CCCCN2C(C2CCN(C)C2)=O)C1 C1(C(=O)OC)CCCCN1CCNC(C(C)(C)NC(=O)OC(C)(C)C)=O N1(C(C(C)N(C(C(CCC)OCC)=O)CCC)=O)CCC(C)(CSC)CC1 Cc1cccc(C)c1CN(CC(C)C#N)C(c1cccc(I)c1)=O C1(NCCN2CCC(C(=O)NC(c3ccccc3Cl)C)C2)CC(=O)N(CCN)C1 c1(C(=O)OCC)cc(CNCCCN2CCCCC2C2CC2)nn1C C1(C(=O)OC)CC(F)(F)CC1C(=O)N(C1CCCN(C(=O)C=C2CCCC2)C1)C CC(CN(C)C(c1coc(C(C)NC(c2ccnnc2)=O)n1)=O)C(C)(C)C C=Cn1ncc(C(N2C(C(=O)OC)CC2C)=O)c1N.C12(CC1)CC(=O)NC2 Cc1ccc(CC(=O)NC(C)C(C)NC(=O)C(C(C)C)N2CCCC2=O)c(C)c1 c1(C(=O)NCCCC)cc(-c2csc(NC(=O)CC3CCCC3C)c2)ccc1F C1(S(C)(=O)=O)(C(=O)NC(CCCNC(CC(C)C)=O)C)CCCCC1 C12(NC(c3[nH]cc(C(C)=O)c3)=O)CCCC1CN(C(=O)CC1CNC(=O)O1)C2 C1(O)(C(C)NC(=O)CSc2n[nH]c(O)n2)CCN(C(=O)CC2COC(=O)C2)C1 C1(NC(C2C(NC(c3c(NCC)scn3)=O)C2)=O)CCCC(F)(F)C1 C1(C(C)C)CCN(C(=O)CN(C)C)C(CNC(=O)CCc2ccc(F)nc2)C1 c1(NC(C2OCCN(Cc3scc(C)c3)C2)=O)ccc(C(N)=O)c(F)c1 N1(C(C(COC)(F)F)=O)CCC(CO)(CNC(=O)CCc2nncs2)CC1 c1(-n2c(C(F)Cc3ccccc3)nc(C(CC)O)n2)ccc(S(N)(=O)=O)cc1 c1(CC)cc(CC)nc(NC2(CNC(=O)C(CC)OC)CCCCC2)n1 N#CC1(C(=O)NCc2cc(C(=O)NCc3ccsc3)co2)CC(=O)C1 C1(OC)CN(C(c2cncs2)=O)C(C)(CNC(=O)CC#N)C1 CN1CCC2(CN(C(c3cnn(CC(F)F)c3)C(=O)NC3CC3)CCO2)C1 C1(O)(C(C)C)CCC(NC(c2cnn(C3CC3)c2Cl)=O)C1 C(C(=O)N1CCCC(CNC(=O)Cn2ccccc2=O)C1)(C(C)C)OC C1(NC(C(C2CC(N=[N+]=[N-])C2)N2C(C(C)(C)C(C)CCl)CCC2)=O)CN2CCC1(C)CC2 C1(CC)CN(C(=O)Cc2c(Cl)cnn2C)CCN1C(=O)C(CO)c1ccccc1 N1(C(C2(C)CC2(F)F)=O)CCC(NC(=O)Cc2cc[nH]n2)C(O)C1 C(=O)(C#CC1CCOC1)NCc1c(C2CN(C(C3(SC)CC3)=O)C2)ocn1 C(=O)(C(C)(C)C1CCC1)NS(CC)(=O)=O.C(=O)(CC1(CO)CC1)NCCN C1(NC(C2CCN(CC#C)CC2)=O)CC(O)CN(C(=O)C(COC)NC(C)=O)C1 C1(C(N2CCC(N(C(c3nnc(O)cc3C)=O)CC)C2)=O)CN2CCCC2CO1 CCC(CC)C(F)C(=O)N1CCC(F)(C(N2CC(CO)CC(C)(C)C2)=O)CC1 c1(CCC(=O)NCCCCCCNC(C=C(C)C(C)C)=O)ccc2[nH]ccc2c1 C=CC1COCCN1C(=O)CC1CCCC1NC(C1CCCC1)=O CCC(C)C(O)C(=O)NCc1ccc(C(=O)N(C)CCC2CCCN2C)o1 Cc1cc(C(N2CC(CNC(c3cncnc3)=O)C2)=O)c(Br)cc1F c1(C(C)(C)CSC2CCCC2NCCn2cc(C34CC(C3)C4)nn2)ccccc1F Cc1cnc(C=CC(=O)NC2CC(N(C(=O)CCN3CCC3)C)C2)[nH]1 N1(C(c2ccon2)=O)CC(F)(F)CC1CNC(C1(c2ccccc2)CCOC1)=O C1(NC(c2ccc(OC)nc2)=O)CC2CC(CN3CCCCC3)CC12 C(CCC(C(=O)N(c1csnc1OCC)C)NC(c1cnn(C2CC2)c1)=O)OC CCC(CC(=O)NC(C12CCC(CC1)C2)CNC(=O)CN(C)C)NC(=O)CSC N1(C(c2cc(CC)no2)=O)CC(CNC(=O)CCc2cnc(O)[nH]2)C(C)C1 C(CNC(=O)CCC1CCCCCC1)(CC(F)(F)F)NC(CN(C)C(N)=O)=O CC(CCNC(=O)CC1(C)CCCO1)CCNC(c1coc(Br)n1)=O C1(CN(C(=O)C(CCC2CCC2)NC(=O)OC(C)(C)C)C)CCC2(CCC2)O1 N1(C(CSc2n(C)cnn2)=O)CCC(NC(c2csc(CO)n2)=O)C(F)C1 N1(C(C2CC(OCC)C2)=O)CCC(N(C(=O)CCN2CCC2)CC(C)C)CC1 CCC(C)N=c1[nH]c2c(c(=NCc3ccccc3-c3cnn(C)c3)[nH]1)CCC2 c1(NC(C)=O)cc(C(=O)NC23CCN(C(C4CC45CC5)=O)CC2C3)ccc1C C1(NC(=O)NCC2=NOC(C)C2)CCCN(Cc2ccccc2)C1C C1(CC(=O)OC(C)(C)C)(NC(C)CCC2CCCO2)CCOC1 c1(C(N2CCCC(C)(NC(C(C(C)(C)C)SC)=O)C2)=O)cnn2c1NCC(C)C2 C1(NC(c2ccc(OCOC)cc2)c2nnnn2C(C)(C)C)COCC(C)(C)O1 C1(NC(CC(C)N(C)C)=O)CCCCC1NC(=O)Cc1cnco1 C=C(Cl)CC(C(=O)NCC1(COC)CCCC1)NC(=O)C(C)CO N1(C(CC(=C)C)=O)C2CCCC1CN(C(c1cccnc1NC(C)C)=O)C2 C1(N(C)C(c2cccnc2O)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1 N=C1NC(=O)C(CC(N2CC3C(CNC(=O)CC4(c5ccon5)CC4)C3C2)=O)S1 C1(N(C(Cc2cnc(C)o2)=O)C)CCCCN(C(C2CN3CCC2CC3)=O)C1 c1(C(=O)NCC(C)(CNC(c2cnn3ccsc23)=O)OC)nc2ccccc2[nH]1 N1(C(CSC)=O)CC2(CC(C(N3CCC4C(C(N)=O)C4C3)=O)CO2)C1 C1(C(=O)NC(C2CCN(C(C(CC=C)(F)F)=O)C2)(C)C)CCc2ncncc2C1 N1(C(C2C(CCOC)C2)=O)CCC2C(C(=O)N(C3CC3C)C)C2C1 C1(OC)CCn2cc(C(=O)NC(CNC(=O)C=Cc3nccs3)C(C)C)nc2C1 CC1CCCC(C)N1C(=O)COC(C1CCCN1C)=O N1(C(c2c(CC)n(C)cc2)=O)CC2CC(C1)N2C(C1(CC2CC2)CCC1)=O c1(C(C)(C)NC(CC2CC(NC(=O)OC)C2)=O)nnc(N)o1 C(CCCCNC(=O)Cc1cnc[nH]1)N(C(=O)CSCc1ccccc1)C O=C(CS(=O)(=O)C1CC1)N1CCC2(NC(=O)CNC(C3CCC3)=O)CC2C1 C1(NC(C2C(CNC(C)=O)CCC2)=O)CCC(NC(=O)CC(O)CC2CC2)CC1 N1(C(c2c(OC)cncc2)=O)C2CCC1C(CNC(c1cc(C)nc(O)n1)=O)C2 Cc1cc(-c2ccccc2F)nnc1N1CC(CCO)C(CCO)C1 c1(OC)ccc2c(n1)NC(C(N1CCC(CNC(c3ccc(F)cn3)=O)C1)=O)C2 C1(CN(C)C(c2ccccn2)=O)C2CC(CC2F)N1C(=O)C(c1cccn1C)=O C(CC(C)(C)CC(=O)NCC(N1CC1CO)=O)OC C1(C(=O)NC(CN(C)C(c2cccc(O)n2)=O)(C)C)CCCCN1CC(F)F C(C(C)(C)CC(=O)N(C(CO)C(C)C)C)NC(C(COC)OC)=O C#Cc1ccc(C(N2CC(N(C(=O)Cc3ccc(F)cn3)C)C(F)C2)=O)cc1F C1(COC)CN(C(C2CCCC2NC(=O)C=NOC)=O)CCO1 C1(C(=O)NCC)CC2CCC1N(C(=O)CCc1ccccc1C#N)C2 c1(CC)ccc(CC(=O)N(CC(O)CN(C(=O)C(C(C)OC)N(C)C)C)C)cc1 C1(C(=O)NC2CC(C)(NC(c3ccncc3C(F)F)=O)C2)CCc2nc[nH]c2C1 C(=O)(CCCC(C)(C)C)NC12C(CN(C(C(C)(c3ccccc3)N(C)C)=O)C1)C2 N1(C(C(CCC)C)=O)CCC2(CCOCC2)C(NC(=O)C(CC(C)C)OC)C1 N(C(=NCCC(=O)N(C)C)N1CCC(CS(C)(=O)=O)C1)C(CC)C c1(C(=O)NCC23C(CN(C(CC(C)C)=O)C2)C3)cc([N+](=O)[O-])c(Cl)cc1F C(=O)(C1=NOC(CNC(c2cccc[n+]2[O-])=O)C1)N(CC(C)(C)O)CC N1(C(C(C=C)OC)=O)CCC12CN(C(=O)CC1CCCN1C)C2 CCCS(=O)(=O)CC(=O)N1CC2CCOC2(CNC(C2CC2(C)C)=O)C1 C(c1ccncc1)=C(C)C(=O)NCC1CN(C(c2oncc2C)=O)C2CC12 N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(C2C3CCN2CC3)=O)CC(C)(C)C1 C[Si](C)(C)c1cccc(-c2ccc(C(=O)Nc3cc4sccn4c3)c(F)c2)c1 c1(CC(=O)NCC2CCC(NC(=O)C(F)=C3CCCC3)C2)ccc(F)c(Cl)c1F c1(NC(=O)Nc2c(N3CCN(C)CC3)ccc(F)c2)cc2ccc(O)nc2s1 O=C(C1=CCCCCC1)NC1CC12CCCN(C(=O)C(Cl)=CCl)C2 c1(C(=O)NCC(C)CNC(=O)CCCCCF)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCC2C(C)CCN2C(C2C3(CC3)C23CC3)=O)nc2cc(O)ccc2[nH]1 c1(C(N(CCC(C)NC(c2cn(CC)nn2)=O)C)=O)cccc(N)n1 C1(NC(c2ccc(CC)cc2)=O)CCN(C(c2csc(CC)n2)=O)CC1O CCC(C(F)(F)F)NC(CC(C)C1CCCC1)c1nnnn1C1CCCCC1 c1(NC(=O)NCC(CC)(C)c2ccccc2)ccc(F)c(OCCN(C)C)c1 C(C1=CCCN(C(=O)C(=Cc2ccccc2)C)C1)NC(CN(C(C)=O)C)=O C1(CNc2[nH]cc(C(C)(C)C)n2)CN(C(=O)CCCCn2ccnn2)CCO1 c1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CCC2)cnc(OC)cn1 Cc1cnccc1C(C)C(=O)NC(CNC(c1ccc(CSC)o1)=O)C1CC1 C1(C(=O)Nc2n(C)nnn2)COc2ccc(-c3ccc4c(c3)NCCO4)cc2C1 c1(C(N2C3(CNC(CN=S(C)(C)=O)=O)CCCC(C2)C3)=O)ccnc2ccccc12 C1(CC)CCC(C)N(C(C23CC(N)(C2)C(C)O3)=O)C1 C1(C(=O)NC(C=C)(C)C)CN(C(C2CC23CCOCC3)=O)CC12CCC2 c1(OC)ccc2cc(NC(=O)NC(C)Cc3cnccn3)ccc2c1 C=CC(C)(O)C(=O)NC1CCCC(NC(=O)C(F)(F)C2CC2)C1 C(c1cccc(O)c1)=CC(=O)NCC1(O)CCN(C(=O)C(F)=CC2CC2)C1 C1(NC(CC(=O)NCC)=O)(CO)CCCN(C(C2CSCCS2)=O)C1 C(=O)(C#CC1CCCO1)N1CCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 c1(C(=O)NC2CN(C(C(CNC(C)=O)(C)C)=O)CC2(C)C)ccc2cncn2c1 c1(CC(N2C(CNC(CN(CC)CC)=O)CC(C)(C)C2)=O)noc2ccccc12 c1(C(N(C2CCCC2)CCCNC(C=CCCC)=O)=O)cc(CSC)on1 N#CC1=C(C(=O)NCCOCCNC(c2cnc(O)c(Cl)c2)=O)CCC1 C1(NC(C2(C(C)(F)F)CC2)=O)COCC1n1cc(C(C2CC2)C2CC2)nn1 c1(C(=O)NC(N2CC(CO)CC(C)C2)=O)ccc2cccnc2c1 C1(CC#C)(C(=O)N(C)CCN(C)C(C2CN(C3CCC3)C2)=O)CCOC1 N1(C(=O)OC(C)(C)C)CC2C(COC(C3CC(O)(c4ccncc4)C3)=O)C2C1 CCC(CC(=O)N1CC=CC1(C)C(=O)NCC1(O)CC(C)(C)C1)C(C)C n1(CCOC)nc(-c2ccc(F)cc2)nc1-c1ccc(CC(C)C)cn1 C1(NC(c2c(OCC)ccs2)=O)CC(NC(C2CC=CCC2)=O)CC1O N1(C(C2(C(C)C)CCN(C(=O)C(C3CC3)C3CC3)C2)=O)CC(CO)OCC1C CCCN=C(NCC(C)CNS(C)(=O)=O)NCc1cc(C)on1 N1(C(C23CN(C(CCC(C)SC)=O)C(C2)CO3)=O)CC2(CCC(O)CC2)C1 Cc1cc(C(=O)NCC2CN(C(C3CCCCS3)=O)CCO2)c(C)nc1C c1(C(=O)NCCC(C)N(C(=O)C(C)CC(F)F)C)cnc2sccn12 CCCCCCCC(=O)N1CC(O)CCC1C(=O)NCc1nnc(O)n1CC c1(CC)cc(C(=O)NC(Cc2cn[nH]c2)C(N2CCOC(C)C2)=O)nn1C C=CCCCC(=O)NCCC1CCCN1C(c1cc(Cc2ccccc2)c[nH]1)=O N1(C(C2CCCN(C(C)=O)C2)=O)CCOCC(C)(CNC(=O)Cc2ccco2)C1 N1(C(C2C(=C)C2)=O)CCCC(CNC(c2ccc(CC(C)C)cc2)=O)C1 C1(NC(=O)CONC(=O)C2CC(OC3CCC3)C2)CC2CCCC2C1 N1(C(C(CC=C)CC)=O)CCC2C1CCCN2C(=O)CNC(=O)NC C(=O)(C1CCCc2ncnn21)N1CCC(NC(C)=O)CC1 C1(C(C)C)(C(=O)NC(CCO)C(C)C)CCCN1C(c1csnn1)=O N1(C(C2C(C)C2)=O)CC=C(CNC(=O)C(CN2CCCC2)c2ccccc2)CC1 c1(C(=O)NC(C2OCCN(C(c3scc(OC)c3)=O)C2)C)ccc(S(N)(=O)=O)o1 C1(NC(c2cn(CCO)nn2)=O)CC2(CCN(C(=O)C=C3CCSCC3)CC2)C1 CC(C)(CC1CCOC1)C(=O)NCCC1(O)CCN(C(=O)C=Cc2cc[nH]n2)C1 C1(F)(NC(=O)OCC)CCN(N2CCn3c(cnc3-c3ccccc3)C2)CC1 C12(CC)CN(C1)C2=O.c1(CNC(C(CC2CC2)NC(=O)OC)=O)ccccc1 c1(NCc2ccc(CNC(c3cc(CC)n(C)n3)=O)cc2)ncnc2scnc12 N1(C(c2cc(C)oc2C)=O)CCc2ccccc2C1CNC(c1cn[nH]c1)=O C(C)(C(=O)NCC1(NC(=O)CCc2ncccc2C)CCCCC1)(C(C)C)OC Cc1nn(C)c(Cl)c1C(=O)COCCSc1ccc(Br)cc1 CC1CCC(NC(N2CCC(Cc3ccnn3C)CC2)=O)c2ccccc21 N1(C(c2c(C)nccc2)=O)CC2ON=C(CNC(C3(CC4CC4)CC3)=O)C2C1 C(c1cccc(Br)c1)=CC(=O)OC1C(SCCOCC)CCC(C)C1 Cc1cc(C)c(C(=O)NC2(C(=O)NC(CO)CC(C)(C)C)CC(F)C2)cn1 c1(C(C2CC2)NC(C2N(C(C(CC)C)=O)CSC2)=O)ccccc1COC c1(C(=O)NCCN(C)C(c2cc[nH]c2)=O)n[nH]c(C2CC2)c1Cl Cc1ccc(COC(C)C(N2CCC(n3cc(C(O)C4CC4)nn3)C2)=O)cc1 c1(CNC(Cn2c(C)cc(C)n2)=O)cc(O)nc(CNC(=O)C(C)NC(N)=O)n1 C1(CNC(C2(N)C(C)(C)C2)=O)CS(=O)(=O)CCO1 CC(C)CC(O)C(C)C(=O)NCCC1(C(N2CCC(O)C(C)(O)C2)=O)CCCC1 c1(C(N2C(CNC(CN(C(C)=O)C)=O)CCC2)=O)cnc(C(C)(C)C)nc1C N1(C(COC)=O)CC(C)CN(C(c2ccc3nc[nH]c3c2)=O)CC1C N1(C(CC(=O)OC)=O)CC2CC2(C(=O)N(C(C)CO)C2CC2)C1 c1(C(N2CCN(C(C(C=CC)O)=O)CC2COC)=O)cnc(O)c2ccccc12 CC1CN(C2CCC2)CC1(c1nnnn1C1CCCC1)Nc1c(Cl)nsc1Cl c1(C(=O)NCC=CCNC(C(CC)n2nccc2C)=O)cc(SC)ccc1C C(=O)(C(O)CCCC)N1C(C(N2C(CC#C)COCC2)=O)CSCC1 c1(C(=O)NC2CCN(CC(=O)NCC(C)(C)OC)CC2)ccc(C)nc1C C1(NC(c2ccc(SC3C(C)C3)cc2)=O)CC2CC1CN(C(c1cccs1)=O)C2 N1(C(C(C(C)C)NC(C2N(CCC)CCC2)=O)=O)CCCCCCC1CC Cc1c(NC(C)CS(N)(=O)=O)ncnc1N1CCN2C(=O)CC12 c1(OC)cc(CC(N2CCC(C)(CNC(=O)CS(C)(=O)=O)C2)=O)cc(OC)c1O C(=O)(C1=CCC2(COC2)OC1)N(CCCN(C)C(c1ccnn1C(F)F)=O)C c1(CNC(c2cc(CC)oc2C)=O)ccc(CNC(C2(C)CC(C)C2)=O)c(F)c1 CC#CCC(C)N=c1nc(N2CC3C(C2)C3(F)F)c2c([nH]1)CCC(C)C2 C12(CCNC(c3ccc(CC)s3)=O)CCC(C1)N(C(C1CCOC(C)(C)C1)=O)C2 C(C)(CNC(=O)C1=CCOC1)(CC(C)C)NC(C(CCSC)NC(C)=O)=O C1(CNC(=O)Cn2cccn2)CC2CCC1N(C(c1ccc(CO)o1)=O)C2 N1(C(COCCCCC)=O)CCC2CN(C(C3CCOC(C)C3)=O)C(C)C12 C1(CC(N2C3C(CNC(Cn4nc(C)oc4=O)=O)C(C3)C2)=O)CCC(C)(C)CO1 C1(NC(c2cnc(Cl)c(Cl)c2)=O)CN(Cc2cc(O)c(F)c(F)c2)CCC1(F)F c1(NCC2(NC(C3CC4C=CC3C4)=O)C(C)CCCC2)ncnc(Cl)c1[N+](=O)[O-] n1(CCC)nccc1C(=O)N(CCC(=O)N(CC(C)C(C)C)C)C1CC1 C(=O)(C(C)CC1CC1)N(CC(=O)NC(c1ncc[nH]1)CC)CC1CC1 C1(NC(C2CC(NC(c3cc[n+]([O-])cc3)=O)C2)=O)CC2CC3C(C2)C13 C1(CC)CN(C(C2(C)CCCS2(=O)=O)=O)CC(C)N1 C1(C#N)(c2nc(NC(c3ccnc(SC(C)(C)C)n3)=O)sc2)CCOCC1 O=C1CCC(CC(N2CCCC2CN(C(=O)C2=NOCC2)C2CC2)=O)CN1 C(CC1CC1)(C(=O)N1CCCC1CC1CC1)NC(CC1CC(=C)C1)=O CC1CCc2[nH]c(C(=O)NC(C)CNC(=O)COCC3CCCO3)cc2C1 Cc1ccc(O)c(C(N2C3CCC2C(C(=O)NC2(C)CCC(C)C2)C3)=O)c1 N1(C(C2CCC(C3CC3)CC2)=O)CCC2OCCN(C(=O)COCC3CC3)C2C1 n1(CCCC)ncc(C(=O)NCCN(CC(C)O)C(c2occ(C)c2C)=O)c1C N1(C(C)=O)CCCC(NC(=O)C(Cn2ccnn2)NC(c2coc(C(N)=O)c2)=O)C1 C1(CC)(NC(=O)CC2CCCCN2C(c2cnn(C(C)C)c2)=O)CCCCC1 CCCCC(CC(=O)N1CCC(C)(CC)CC1)NC(c1coc(C)n1)=O C(CC(C)(C)C(=O)Nc1ccccc1F)NC(C(C)n1cccn1)=O C12CCN(CC1O)C(=O)CCc1nc(no1)CC(=O)N2.C1(O)(C(C)C)CCC1 N1(C(C2CN(CCC)C(=O)C2)=O)CC(CO)C2(C1)CN(C(=O)Cn1ccnn1)C2 C=CC1CCCN(C(c2cccc(C(c3ccccc3)=O)c2)=O)C1 C(=O)(C(C)CCCC)NC(CNC(C1(C=C)CCC1)=O)C1CC1 C#CC(CC(C)(C)C)NC(=O)CC(C(C)C)NC(C1(O)CCCCCC1)=O N1(C(C(C)S(N)(=O)=O)=O)CCC(CNC(=O)CCC(F)F)C(F)(F)CC1 Cc1cc(C(=O)NCC2CCCCC2NC(C2(F)CCS(=O)(=O)C2)=O)ccc1N c1(C(=O)NCC=CCNC(C2C(CC)C2)=O)ccc([N+](=O)[O-])cc1C(F)(F)F c1(CC(=O)Nc2cccc(-c3ccco3)n2)cn2cc(-c3cccs3)ccc2n1 C1(NC(=O)C=CI)CC(N=c2[nH]nc(-c3ccccc3)s2)C12CCOCC2 N1(C(C(CC)CC)=O)CCN(C(=O)Cn2[nH]cnc2=N)CC2CCCCC12 CC(c1ccccc1C)=CC(=O)N(C1CC(NC(=O)CCc2nncs2)C1)C c1(SCCC(=O)NC(C(C)NC(CCCC)=O)CO)ccc(F)cc1F Cn1ncc2cc(CN3CCC(NC(=O)C(=O)NCC(F)F)C3)cnc12 N1(C(=O)CC2CCN(c3c(F)cnc(C)n3)CCC2CO)Cc2ccccc2C1 c1(NCC2CCC(C)C2)ccc(S(=O)(=O)N(C)Cc2ccnn2C)cn1 N1(C(c2c(CC)csc2)=O)CCN(C(=O)CC2CCN(C)CC2)CC1CC(F)F C1(C2CCN(C)CC2)(C(=O)NCCCN(C(=O)CCCC(C)(C)C)C)CC1 N1(C(C(CC=C)CC)=O)CCC(C)(C)C(C=O)C1.N1(CC)CCC1 c1(CC)cc(C(=O)NCC2CCCN2C(C2CC23CCOC3)=O)c2c(c1)CCO2 C(CCC(C)C)(C(=O)N1CC2(CCC2)CC1CNC(=O)C(F)(F)CO)NC(C)=O N1(C(c2cn(C3C(OCC)COC3)nn2)=O)CCN(CCC(Cl)Cl)CC1 CCC(CC(=O)NCC1(NC(C2(CO)CCCCC2)=O)CCC1)OC C(=O)(CC(=O)NC(C(=O)NCC(F)C1CCC1)c1cccs1)OC c1(OC)ccc(C(=O)NCC2(O)CCCN(C(=O)C(C)n3ccnc3)C2)c(Cl)c1 C(CCC(=O)N(C)CC=CC(N1CCC(CC2CC2)C1)=O)=C(C)C C1(C#CC(=O)N(CCC(C)NC(c2cc[n+]([O-])cc2)=O)C)(CC)COC1 c1(N(C(=O)C2=CCC2)C)ccnc(-n2cncn2)c1.C12CCCN1C2=O c1(C(C(N2CCCC(c3cn(CC(=O)OC)nn3)C2)=O)C)ccc(F)c(OC)c1 c1(C(=O)OC)cc(CCC(=O)NC(C(C)(C)C)c2cccs2)c[nH]1 c1(C(=O)NC(CC(C)NC(c2cccc(OC)c2N)=O)C)ccc2c(n1)CCC2 Cn1nc(CC(=O)NC2CCC(NC(c3csc(C#N)c3)=O)C2)cc1Cl N1(C(c2cnn(CC)c2Cl)=O)CCN(C(=O)CC(C)(C)C#N)CC2CCCCC12 C(=O)(C(CC(C)CC)NC(=O)Cn1nc(C)cc1C)N1CCC(C=C)C1 C1(NC(c2scnc2Cl)=O)CC(F)CN(C(=O)CCc2cnc[nH]2)C1 C1(C(=O)NC(c2cccs2)C)CC(C)(C)CCN1C(c1cnn[nH]1)=O c1(OC)cc(F)c(CC(N2CC(NC(C3CCCCC3)=O)C(O)C2)=O)c(F)c1 CC1C(NC(c2cccnc2N2CCCC2)=O)CCN1C(=O)C(=O)NCC(F)F C(=O)(C1=CC(C)CC1)NC(CNC(C(c1ccccc1O)OC)=O)(C)C c1(C(=O)NCC2CN(C(CCc3cnc(C)o3)=O)C2)cncnc1C1CC1 CC1(C)C(CO)CN1C(=O)CSCCNC(C1CC(F)C1)=O CC1CC(NC(c2cc(N3CCCC3)ccn2)=O)CN(Cc2ccccc2F)C1 CC(C(=O)NC1(CCC(=O)N(CC(Cl)Cl)C)CCC1)NC(=O)C1CC1 C1(NC(c2c(C)cns2)=O)CCN(C(C2CCSC2)=O)C1(C)C N1(C(CS(CC)=O)=O)CCN(C(=O)CCCOc2ccc(Cl)c(C)c2)C(CO)C1 c1(C(=O)NC2CC(NC(C3CC(C)C3)=O)C2)c[nH]c2ccc(Br)cc12 N1(C(c2cncc(N(C)C)n2)=O)CC2(C1)CN(C(C1CC1c1ccc(Cl)s1)=O)C2 CCCC(C(=O)NC1C=CC(CNC(c2nccnc2C(F)(F)F)=O)C1)OC N1(C(CC(CCC)O)=O)C2CCCC1CN(C(c1c[nH]nc1C(F)F)=O)C2 C1(C(N(CCCSC)C)=O)CC12CCN(C(c1ccc(C)nc1C)=O)C2 C1(C2CC2)(CNC(c2cc(OC)nn2C)=O)CCN(C(=O)CC(C)C2CC2)C1 c1(C(N2CCC(C)(NC(C(CC)SC)=O)C2)=O)cc(C)c2c(O)nc(O)nc2n1 C1(CCNC(=O)CC2CCCO2)CCCN(C(=O)C=Cc2ncc[nH]2)CC1 C1(NC(c2cnc3sccn23)c2n(CCOC)nnn2)CCCCC12CCC2 C(=O)(CCC(=O)NCC(C)(F)CNC(c1nnc(S)n1C)=O)N(C)C N1(C(c2cc(C(C)C)no2)=O)CCN(C(C2(C)C=CCCC2)=O)CC(O)C1 Oc1nnc2n1CCN(CC(c1cccc(F)c1)NCc1ccccc1)C2 C1(N(C(c2ncc(C)nc2)=O)C)CCCN(C(=O)Cc2nc(C)c(C)s2)CC1 N1(C(C2(CC#C)CCCCC2)=O)CCCC2(NC(c3cncc(C)c3)=O)CC2C1 c1(NC2CN(C(C3(COC)CC=CC3)=O)CC2C)nc(C)nc2n[nH]cc12 Cc1cc(C(=O)NC2C3CN(C(=O)CN4CCCCC4)CC23)c2ncccc2c1 CC1CCC(C(=O)O)N(C(C2CN(c3ccc(C#N)cn3)C2)=O)C1 Cc1ccc(CC(=O)N(C)CC2CCN(C(c3nscc3C)=O)CC2)c(F)c1 O=C1CC(NC(=O)CCCCc2cn(C3CCS(=O)(=O)C3)nn2)CCCN1 NC(=O)CCC(=O)N1CCC(NC(=O)C=CCOC2CCOCC2)C1 c1(C(N(C2CCCC(NC(c3ccc(CC)[nH]3)=O)C2)C)=O)cc(N)nc(Br)c1 C(=O)(CCCCCC(=O)NC1C=CC(CNC(=O)C(C(C)O)N(C)C)C1)OCC C(C1CCOCC1)=CC(=O)N(CC(C(=O)NC(CCC)c1ccco1)C)C1CC1 CC1CC(CNC(=O)Cc2ccc(CO)cc2)CN1C(c1cccc(Cl)c1)=O S(=O)(=O)(c1c[nH]ccc1=NC1CC(N)CC1(C)C)N(CCN(CCN(C)C)C)C c1(OC)cc(Cl)c(C(N2CC3CCC(C2)N3C(C2CC2C2CC2)=O)=O)cc1OC N1(C(CC2CC(C)(C)C2)=O)CC(NC(=O)CC2CC(=O)NC(=O)C2)CC12CCC2 C1(C)(C(=O)NC2CCC(CNC(C(C)OC3COC3)=O)C2)CC(F)(F)C1 Cc1ncnc(C)c1CC(=O)NCC(=O)NCC1C=CCOC1 C1(O)(COC)CCN(C(c2n[nH]c(C)n2)C(=O)NCC2CCCO2)C1 c1(OC)ccc(OCC(=O)NC2(C3CCCN3C(=O)C(C)CN(C)C)CC2)cc1 CC1(CNC(C2(C)CC2Br)=O)CCCN(C(C2CC(=O)N2)=O)C1 c1(C(=O)NC2C(CNC(c3cc(C)cc(Cl)c3)=O)CCC2)c[nH]c2nccc-2c1.C C1(NC(C(C(CC)O)C)=O)CN(C(c2cc(C3CC3)ncn2)=O)CC(C)(C)C1 N1(CC)CC(NC(c2conc2CNC(=O)CC2CCCC(=O)C2)=O)CCC1=O c1(OC)ccc(=NC(=O)C2(C)CCCN2C(=O)C=Cc2ccccc2OC)[nH]n1 CC(O)CCCCCC(=O)N1CC(NC(=O)Cn2cnnc2O)C2(CCC2)C1 c1(C(=O)NC(CNC(c2c(SC)ccs2)=O)C)ccc2c(c1)CCCO2 C1(C(=O)NC2C(CC)C2)CCC(NC(c2ccnn2C2CC2)=O)CC1 Cc1sc(C)c2sc(C(=O)NCC3CCCCC3NC(=O)CC(F)F)cc12 c1(C(N2CCC(NC(c3cnc(-n4cccn4)s3)=O)C2)=O)ccc(C(F)F)nc1 C(C(C)(C)CNC(=O)Cn1ccnn1)N(C)C(c1cnn(-c2ccccn2)c1)=O N1(C(CCC2CC(SC)C2)=O)CCc2ccccc2C(O)C1 CC(C)CCC(=O)N1CC(CF)(NC(=O)C(N2CCCCC2=O)C)C1 c1(CC)[nH]c(Cl)nc(=NC(C)CNC(C2(C)CCOC2)=O)c1C#N C1(NC(CS(=O)(=O)NCC)=O)CN(C(=O)C=Cc2cc[nH]c2)CCC1O c1(NC(=O)CC(c2ccc(O)cc2)NC(COC(C)C)=O)cn(C)c(C(=O)O)n1 N1(C(c2c(COC)scc2)=O)CCOCC(NC(=O)Cc2ccns2)C1 CCC(CC)CC(F)C(=O)NC(c1cn(C)nn1)C(N1CCC(F)(C(N)=O)C1)=O CC(CC(=O)N1CCN(C(=O)C(F)=CC2CC2)C2CCC12)C(F)(F)F c1(NC)c(C(N2CC(COC)(NC(c3cc(C)cc(C)c3)=O)C2)=O)cccc1F c1(C(N2CC(CCO)(NC(c3nc(C)n(C)c3)=O)C2)=O)cc2cnccc2[nH]1 N1(C(CCc2c(C)nccc2)=O)CCN(C(=O)C(=O)Nc2ncc[nH]2)CC1CF C1(N(C(CCOCC)=O)C)CCN(C(c2csc(COC)n2)=O)CC1C C(N=c1nc(N2CC3CC2CS3(=O)=O)c2ccccc2[nH]1)c1n(C)cnn1 N1(C(=O)NC2C(C)CCCC2)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CCC1C N1(C(C=C(C)c2ccco2)=O)CC2CCC(N(C(=O)C(C)n3cccn3)C)C2C1 C1(CC(=O)NCc2c(C)noc2C)N(C(=O)CC2CC(F)(F)C2)CCC1(C)C CC(CNC(c1cccnc1-c1ccccn1)=O)(C(F)(F)F)C1OCCO1 N#Cc1ccc(S(=O)(=O)N2CCC3(CC2)CC3COC(F)F)cc1NCCO O=C(C1=COCCC1)NCCn1cc(C(=O)NC2C=CCC2)nn1 N(C(=NCCCC1CCCCO1)NCC1(C)CCCCC1)C(c1cccs1)C Cc1nc(-c2nc[nH]n2)sc1C(=O)N(CCCCNC(C1CC12CCCC2)=O)C C1(C(=O)NCC(C)NC(=O)C(c2ccccc2F)C)(OC)CCCCC1 CCS(=O)CC(=O)NC(C)(C)C=CC(=O)NC(c1n[nH]c(C)n1)C C#Cc1cncc(C(=O)NC(CCNC(c2cnc(N(C)C)o2)=O)C(C)C)c1 N1(C(CCOCCC)=O)CCC(N(C(=O)CCc2cscn2)C)C2(CC2)C1 O(NC(=O)C(C)N1CCOCC1)c1c(C(C)C)nsc1 c1(C(c2nnnn2CC2CCOC2)NCc2c(I)c[nH]n2)cc(F)c(Cl)c(F)c1 CCC(C)C(C(=O)NCc1cnco1)N(C)C(c1cccc[n+]1[O-])=O C(=O)(C(CC(F)F)N(C(=O)C1=COCCC1)C)NCP(OCC)(C)=O N1(C(CC2(OC)CN(C(C3CCCC4(CC4)C3)=O)C2)=O)CCC2(CCCCO2)C1 N1(C(C(CC)CO)=O)CCN(C(=O)C2=CCSC2)CC1CCOC N1(C(c2nn(CC)nc2C)=O)CC(C(N2CCC2(C)CCO)=O)CC12CCC2 N1(C(c2cnc(SC)s2)=O)CCN(C(C2CCOC2(C)C)=O)C(CCO)C1 CN1CCN(C(c2cc(CCNC(=O)CCc3cnco3)on2)=O)CCC1=O CC1CCCc2cc(C(N3CCC(CC(C)NC(=O)C4CC4)CC3)=O)nn21 C(=O)(CC(C)CC(=O)OC)N1CCCC(CN(C(=O)C(C)(C)C(N)=O)CC)C1 c1(OC)cc(NC(c2cccc(NCc3ccc(F)nc3)c2)=O)ccc1Br CCC(O)C(C)(C)C(=O)NC(C)CC(=O)Nc1ccccc1C c1(C(N2C3CC(C(N4CCCC(C#N)C4)=O)C2CC3)=O)cc2ncccc2[nH]1 Cc1cc(Cl)c(C(=O)NC2CC3CC2N(C(=O)CCc2cn[nH]c2)C3)cc1F Cc1cc(C(=O)NC2CCCCC2CNC(c2cc(C)n(C)n2)=O)ccc1F C1(NC(C2CC2F)=O)(CO)CCCN(C(=O)CCC2CCCCO2)C1 c1(C(N2CC(C(C)(C)O)(CNC(c3nc(C)c(C)s3)=O)C2)=O)ccc(Cl)nc1N N1(C(C2CCN(C)C(=O)C2)=O)C2CCCC1CC(NC(=O)CCc1nccs1)C2 c1(C(N2CC(SC)C(NC(C3C=CCC3)=O)C2)=O)cnc(C)cc1C C12(CNC(c3cc(=O)cc(Cl)[nH]3)=O)CCC(C1)N(C(=O)CCc1ccncn1)C2 C1(C)(C(=O)NC(CCCNC(c2c(CCC)n[nH]c2)=O)C)CCC(C)=C(C)C1 CC1CC(C(=O)NCC2CN(C(c3occc3-c3ccccc3)=O)C2)CO1 C1(CNC(c2[nH]cc(C#N)c2)=O)CN(C(C2CC3CCC3C2)=O)CC12CC2 Cc1cc(OCC(=O)NCCCOCCNC(=O)Cc2csc(C)c2)no1 CC(C(N)C(=O)NC1CCC1NC(c1ccccc1)=O)C1CCCCC1 c1(C(=O)NC2CCC(NC(C3(COC)CCCO3)=O)CC2)cc(=O)c(O)c[nH]1 c1(OC)cc(NC(C2CCCC2NC(c2cccnc2)=O)=O)c(F)cn1 Cc1oc2ccccc2c1C(=O)NC1CC1NC(=O)CCc1cc[nH]n1 N1(C(CCCCC)=O)CCC(C2CCN(C(=O)C(c3cnn(C)c3)O)CC2)C1 Cc1cc2ncc(C(N3CCC4(CCCN4C(=O)Cc4cnc[nH]4)C3)=O)cn2n1 C1(CNC(C(COc2ccc(CC)cc2)C)=O)CCCCN(C(=O)C(=O)NC)C1 c1(OC)ccc2[nH]cc(C(N3CCC(CNC(=O)C(C)OCC4CC4)C3)=O)c2c1 C1(C(=O)NCc2n(C)cnn2)CC(O)CN1C(=O)CC1CC(C)(C)CO1 C=CC(C)(C)C(=O)NCCC1(NC(c2cnn(CCC)c2C)=O)CC1 C(C(=O)N1CCCC1C(C)(C)NC(=O)Cc1cc(C)no1)(C(C)C)SCC C1(C)(C(N(CCC(C)NC(c2csc(C)c2C)=O)C)=O)COC(C)(C)CO1 C(=O)(CCS(C)=O)N1C(Cc2cn(CNC(CCN(C)CCO)=O)nn2)CCC1 c1(C(=O)NC2C3(CNC(C=CCOC)=O)CCC(C2)C3)cccc2nc[nH]c12 CCCC(C(=O)NCCCc1cc(C)no1)NC(c1ccc(C#N)o1)=O c1(C(N2CCC(C(C)NC(=O)Cc3cc[nH]c3)C2)=O)c(F)cc(C#N)cc1F C1(NC(c2c(C)cn(C)c2)=O)CC2CCC(C1C)N2C(c1ccoc1)=O c1(OC)ccc(CC(N2CC3CC3(CNC(C)C)C2)=O)cc1C(F)(F)F c1(C(N2C(COC)(CNC(=O)Cn3cc(C)cn3)CCC2)=O)cn(C)ccc1=O C1(C)(OC)CN(CC(=O)N(CCC(=O)N(CCCCOC)C)C)C1 N1(c2nnc(C(C)C)o2)CCN(C2CCCN(C(C3CC=CCC3)=O)C2)C(=O)C1 C(Cc1ccccc1)(C(=O)N1CCC(CCNC(=O)CCc2nc[nH]n2)C1)OC c1(C(=O)NCC2C(NC(CSCC#C)=O)CCC2)ccccc1S(C)=O CC1CN(C(C2CS(=O)C2)=O)CCC1NC(=O)C1=CSCS1 CC1(C(=O)NC2CC3C=CC2C3)CCCN1C(=O)CN1CCCC1=O CC1CN(C(C2(C)CC(=O)C2)=O)CC(C(=O)N(CC(O)CF)C)O1 N1(C(c2cnc(OCC)c(Cl)c2)=O)C2CCC1CN(C(c1cccs1)=O)CC2 N1(C(CC2CC(=O)NC2)=O)CC(NC(=O)COc2cccc(F)c2F)C2(CC2)C1 C1(NC(C(C)NS(C)(=O)=O)=O)CCCOC12CCN(C(c1cscn1)=O)CC2 CC1(C)CCC(C(N2CCOC3CC23)=O)CN1C(C1C2CC3C(C2=O)C13)=O C1(C)(C(=O)NC(C)CCCNC(=O)Cn2ccnn2)COC(=O)OC1 c1(CCNC(c2n(CC=C)nnn2)c2ocnc2C2CC2)ccc(OCC)cc1 C1(CNC(c2cc[nH]c2)=O)COCCN1C(C1(c2ccc(Cl)nc2)CC1)=O C(=O)(C(CC)C(=O)N1CCC(C)(C(=O)NCC(O)CO)CC1)OCC C1(C2CC2)(C(=O)NCC(CC)NC(c2cnn(C)c2F)=O)CC=CC1 C1(CNC(CN(CCC)C)=O)CC2(CCN(c3cc(C)ccc3[N+](=O)[O-])C2)CO1 N1(C(C(CSC)OC)=O)CCN(C(C2CCC(OC(C)C)CC2)=O)C2(CCC2)C1 N1(C(c2cc(CCNC(=O)C(O)CC(F)(F)F)on2)=O)CC2CCCC2C12CC2 c1(C2(C(=O)NC(C3CN(Cc4sncc4Br)C3)C)CCC2)ccccc1 C1(C(=O)NCC2(C(C)(C)O)CN(C(c3n(CC)nnc3)=O)C2)CCCN1N=O N1(C(CC(CC=C)NC(=O)CCCN(C)C)=O)CCC(O)CC12CC2 N1(C(CNC(CCC)=O)=O)CC(C)N(C(=O)CCc2ncccc2OC)CC1C C1(C(=O)NCC2N(C)CCN(C(=O)CCc3cc[nH]n3)C2)C2CCCCCCC12 CC(CN1CCCC1)CN=c1[nH]c(=NCC2C3CCCCCC23)[nH]c2c1SCC2 C1(CNC(C2CN(C(C)=O)C2)=O)CCC(NC(c2ccoc2Br)=O)C1 C1(CNC(c2c(CC)ncs2)=O)CC(F)(F)CN1C(C1CCCC(C2CC2)O1)=O Cn1nc(C2CC2)c(Br)c1CNC(c1cncc(-c2ccoc2)c1)=O O=C(CC1=CCOCC1)NC1COCCN(C(C2C3CCN2CC3)=O)C1 C1(C(N(C2(CC)CC2)C)=O)CC2C=CC1N(C(=O)CN(C(=O)COC)C)C2 CC(O)CC(C(=O)O)N(c1ccc(C(F)(F)F)cc1)C(=O)CCN1CCCCCC1 Cc1cc(C(=O)NCC2COCC2NC(=O)CCF)c(O)c(C)n1 c1(C(N2CCCN(CC(C)O)CC2)=O)ccc2ncc(=O)n(C)c2c1 CC(O)C(F)(F)C(=O)N1CCOC(CN(C)C(c2cncs2)=O)C1 c1(C(N2CCN(C(C#CC(C)(C)O)=O)C(CN(C)C)C2)=O)ccn2cccc2c1 N1(C(c2n[nH]c(O)n2)=O)CCCC(CNC(=O)C(c2ccc(F)cc2)(F)F)C1 c1(C(=O)NCC2(CO)CCCNC2)cnn2c1NCCC2C(F)(F)F N1(C(c2ccc(-c3ccc(C)s3)s2)=O)CCN(C(C)C(=O)O)C(=O)C1 N(C(=NCCCC(F)F)NCc1cc(C)ccc1Br)CCOCC Cc1nc(Br)sc1C(N1CCC(C)(C(F)(F)F)C1)C(=O)NCCC1CC1 C(=O)(C1=CCCC1)N1CC(CCC=C)(C(=O)N(C)Cc2ccn(CC)n2)C1 C1(NC(CCSCCCC)=O)CC(CNC(=O)CCCc2cncs2)C12CCC2 c1(C(N2C(CNC(C3(OC)CC3)=O)CC2)=O)cccn(CC(=O)N(C)C)c1=O C#Cc1cccc(CC(=O)NC(CCC2CC2)C(=O)NC2(C)CC2(C)C)c1 Cc1oc(CO)cc1C(N1CSCC1C(N1CCSCC1C)=O)=O c1(CC(=O)NC(C)CNC(C2CCOC2=O)=O)ccc2nc[nH]c2c1 C(=O)(C1CCCc2nncn21)NCC(CC(C)C)NC(CN1CCC(C)C1)=O C(C(C)(C(=O)N1CC(c2nncn2C)C1)NC=O)OC.C(C)(C)C c1(C(=O)NC(CNC(c2cc(C)c(C)nc2)=O)(C)C)cc(F)cc2c1NCCC2 N1(C(C(C)c2ccsc2)=O)CCN(C(=O)C=CSc2ccccc2)CC1C(F)F N1(C(CNC(=O)OC)=O)CCN(C(=O)C(CC(C)C)OC)CCC1C N1(C(C2CN(C)C2)=O)C2CCC1CC(N(C)C(C1(O)CC(C)(C)C1)=O)C2 c1(OC)ccc(C(=O)NCCC2CCCN(C(=O)CCCC3CCCC3)C2)nn1 N1(C(C(C)CS(C)(=O)=O)=O)CC2(CCCN(C(=O)CCOC3CCCOC3)C2)C1 C=CCCC(C)(C)C(=O)N1CCC=C(C(=O)NC(c2snnc2C)C)C1 C1(CCC(=O)NC2CCCC2(F)F)CCN(C(C2CCC(F)(F)C2)=O)CC1 N1(C(CCOCCNC(C(C)(C)C)=O)=O)CCCc2cccc(F)c21 N1(C(c2nc(C)oc2)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)CCO2 Brc1cc2ncnc(N3CCC(c4ncc[nH]4)CC3)c2s1 c1(C(=O)NC2CN(C(c3ccc(OC)cc3)=O)CC(O)C2)c(F)ccc(C)c1F N1(CC2(NC(c3c(C)onc3)=O)CC2)CCN(C(C2CCC(F)C2)=O)CC1 N12CCC(CC1)COC1CC(C1)C2=O.C1(C(=O)NC(C)(C)C)OC2CCC1C2 c1(C(N2CC(CC(N3CCOC4CC34)=O)C2)=O)cc(Br)cc2[nH]ccc12 CN1CC=C(CC(=O)N2CC3CCCC(C2)N3C(=O)Cc2ccc(O)nc2)CC1 c1(OCC)cc(NC(=O)NC(C)CS(N)(=O)=O)c(Cl)cc1Br CC(C)(CNC(=O)C(O)C1CCC1)CNC(C1CCN(S(C)(=O)=O)C1)=O c1(OC)cc(C(=O)N(C)CC2CCCN2C(=O)CCC2CC2(C)C)n(C)n1 C1(CNC(C(CC)F)=O)CCCCN(C(=O)Cn2ccc(O)nc2=O)C1 C(CC)(CC)(CCNC(=O)C(C)C(F)F)NC(c1cccc(SCCCC)c1)=O C1(O)(C(CC)C(=O)NC2CCC2CNC(C2(C(=O)NC)CC2)=O)CCCCC1 c1(C(=O)NC(C(C)C)CCNC(c2cccnc2CO)=O)cccc2c[nH]nc12 CC(=NOCC#N)C(=O)NCCC(O)C(=O)NCC(Cl)C(C)(F)F c1(C(N(C)CC2CN(C(=O)C3=CCCS3)CCO2)=O)nccc2cc[nH]c12 C1(CCC=C)(C(=O)NCc2ccc(C)nc2)CCN(C(=O)C(C)OCCOC)C1 C1(C(N2CC(O)(CNC(C3(NC(C)=O)CCCC3)=O)C2)=O)CCOC2(CCC2)C1 C(=O)(C(C)(C)C(F)F)N1CCC(C(CNC(C(C=C)OC)=O)O)CC1 C(=O)(CC(C)(C)C(F)F)NC1C(OC)CCN(C(c2cc(OC)c(O)cc2)=O)C1 C1(C(=O)NCc2ncc(OCC)nc2)CN(C(=O)C(C(C)O)N(C)C)CCCO1 C(=O)(CC(F)(F)C(F)(F)F)NCCCC(c1ccco1)NC(CC(=O)NC1CC1)=O c1(C(N2C3CC(NC(CCC#N)=O)CC2CC3)=O)ccc(F)c2occc12 N1(c2cc(NCc3scc(C)c3)nc(C)n2)CC(C)CC(C)(C)C1 C#CC1CC2(CC(C(N3CC(NC(=O)Cc4cccc(F)c4)C(O)C3)=O)C2)C1 Cn1nc(Br)nc1C(c1nnnn1CC(F)F)NCCc1cc(Br)no1 C1(O)(CC(=O)OC)CCN(C(=O)NC2CCC(C)CC2)C1 c1(CN2C(C(=O)Nc3c(C)occ3)CCCC2)ccc2cc[nH]c2n1 c1(NC(c2cncc(NCc3c(N)cccc3F)c2)=O)ccc2c(c1)OCCO2 c1(NCC)ccc(C)cc1C(N1CCC(CN(C)C(C2C3CCCC23)=O)C1)=O N1(C(C(CC)CC2CCCC2)=O)CCN(C(=O)C(C)(F)F)C(C(C)C)C1 c1(NC(C(C#N)c2ccccn2)=O)ccnc(O)c1 N1(C(CSCCCC)=O)CC2C(CNC(=O)CCn3ccnc3C(C)C)C2C1 c1(N(C)CC2N(C(CN(S(CC)(=O)=O)C)=O)CCC2)cc(Cl)ncn1 CC#CCC(C(=O)N(C1CC(C)CC(C)C1)C)NC(C1CCCCC(=O)C1)=O CCCCC(CC)CC(=O)NCCC(O)CNC(C1CC(n2cnnc2)C1)=O Cc1ccc(C(=O)N(C(C)CCNC(=O)CC2CC(CN(C)C)C2)C)cc1 Cc1cc(C)c(CC(=O)NCC(C)N(C)C(c2cnc3[nH]cnc3c2)=O)c(O)n1 C(C)(CCCCNC(C1(CS(C)(=O)=O)COC1)=O)NC(CC(C)OC)=O N1(C(CCNC(C)=O)=O)CC2CCOC2(CNC(=O)C(C)(C)CC(F)F)C1 N1(C(C(=O)Nc2cccc(NC3CCC3)c2)=O)CC2CCC1C(CO)C2 c1(OC)cccc(C(=O)NC(C)C(C)(C)NC(=O)C(C2CC(F)(F)C2)O)n1 c1(C(N2CC(O)(CN(C)C(C3CC3F)=O)C2)=O)ccccc1-c1cncnc1 N1(C(c2c(C)snc2)=O)CC(C)C(NC(C2CC(C)(O)C2)=O)C(C)C1 c1(C(N(C)CCOCCCNC(=O)CC2CCCC2)=O)cccn2cnnc12 Cc1cc(C(=O)N(C2CCC(NC(=O)CCN(S(C)(=O)=O)C)C2)C)nn1C1CC1 CC1(C)CN(C(c2cc(Cl)c(F)c(Cl)c2)=O)CC(C)(C)C1NC(=O)C1=CCCS1 Cc1cc(C(N2CC(CC(=O)Nc3ncc(Br)c(O)n3)C2)=O)cc(O)n1 C=CCC(CNC(C1CCSCC1)=O)NC(c1cc(C(F)(F)F)ns1)=O Cc1nc(O)[nH]c1C(=O)NC(C1CCN(C(c2cc(O)nn2C)=O)C1)(C)C c1(C(=O)NC2C(NC(CCc3scc(C)n3)=O)CC2)ccc2c(c1)C(=O)CCC2 C1(CC(=O)NCC(CNC(C=CCN(C)CC)=O)F)CCCN1C(C)=O C1(NC(c2n(C=C)nnc2)=O)CCN(C(c2ccccc2)=O)CC1C c1(CC)cc(C(=O)NC(Cn2cccn2)C(=O)N(CC(C)(C)C#N)C)no1 CCCCC(C(=O)NCCOCC(F)F)NC(=O)C(C(C)C)NC(C)=O C(C(C)(O)CNC(=O)C(Cc1cn[nH]c1)NC(=O)CCCNC(C)=O)OC C1(C(=O)NC2CN(C(CCCCSC)=O)C2)CC(C)(C)CCO1 C#Cc1ccc(C(=O)NC2CCC2C(=O)N(C(CO)CO)CC)cc1C C=C(C)C(C)(C)C(=O)N1CCC(C=CC(=O)NC2CC(C)OC2=O)CC1 N1(C(C2(C=C)CC2)=O)CCCC(C2CCN(C(=O)C3=CCC3)C2)C1 C1(CC)CCc2nc(NC(=O)NCc3c(F)cncc3Br)ncc2C1 N1(CC(=O)NCC2(CN(C(=O)C(N3CCCC3)C3CC3)C)CC2)CC(=O)N(C)C1=O N1(C(c2c(OC)cccc2C)=O)CC2CCCC2(CNC(C2CC(SC)C2)=O)C1 C(C1=CCN(C(=O)CC2CCCC(C(C)C)O2)CC1)NC(c1cnn(CC)n1)=O CON=CC(=O)NC(CNC(C1CC1(F)F)=O)C1CCC1 Cn1ncc(C(=O)OC2CCC(OC3CCC3)CC2)c1C(F)(F)F c1(C(=O)NC2(CNC(=O)C(F)(F)c3ncc[nH]3)CCOC2)cccc(OCF)c1 C(CCN=C(NC(C)C)N1CCC(F)(c2ccccc2Cl)C1)=CC Cc1ccoc1S(=O)(=O)NCC(c1cccnc1)C C(=O)(C(C)(O)CNC(c1nnsc1C)=O)OC.C12CCC1C(=O)N2 C(=O)(C(CC(F)(F)F)c1ccccc1)N1CC2C(COC(C)(C)C)C2C1 c1(CC(=O)NC(CC)(C)CNC(c2nc(Cl)sc2C)=O)c(C)cc(C)cc1C C1(NC(C23C(NC(Cn4c(C)nc(C)n4)=O)C4CC2C3C4)=O)CCC(=O)N(C)C1=O c1(OC)cc(C(=O)NC2CCCCN(C(c3ccsc3)=O)C2)c([N+](=O)[O-])cc1F CON(C(=O)c1c[nH]nc1CCNC(c1cc(C2CC2)on1)=O)C1CCCC1 C1(NC(c2ccc(C(C)(C)C)[nH]2)=O)CCC(NC(C2CC2C(F)F)=O)CC1 N1(Cc2cn(CC(CNC(c3cc[nH]c3)=O)(F)F)nn2)CC=C(CO)CC1 c1(-c2c(C(C)(F)F)cccc2)ncnc2[nH]cnc12 c1(C(=O)NCCC(=O)NC2CC3CCCC3C2)ccc2ccccc2c1 C12(C(N3C(C4(NC(CCC#C)=O)CC4)CCC3)=O)CCC(N(C)C)(CC1)CC2 C1(CC(=O)NCCNC(c2ccc(C(C)(C)C)cc2)=O)Cn2ccnc2NC1=O c1(CC(N2C(CCCNC(C3CC=CCO3)=O)CCC2)=O)ccc(O)c(F)c1 c1(C(=O)NCCCN(C(CC(CC)CN(C)C)=O)CC)cc2scc(C)c2[nH]1 C1(NC(c2c(C(C)C)n[nH]c2)=O)CC(C)CN(C(c2cn(C)nc2Br)=O)C1 c1(C(=O)NC2CC(CC(=O)NCCCn3cncn3)C2)c[nH]c2ccccc12 c1(CC(N2CC(OCC)C2)=O)nc([N+](=O)[O-])n[nH]1 C(=O)(CC1=CCOCC1)N1C(CN(C(=O)CC2CCCS(=O)(=O)C2)CC)CCC1 C1(OC)CC(C)CN(C(=O)C=CC(C)NC(C2C3CCCC(=O)C23)=O)C1 c1(C(=O)NC2CC(CNC(C(C=C=C)C)=O)C(O)C2)ccc(Cl)cc1C N1(C(c2cc(C)[nH]n2)=O)CCC(C(=O)NC(C2CCCC2)C)(C(C)C)C1 c1(OC)cc(F)ccc1C(N1C2CCC(C2)C1C(=O)NCc1nc(Cl)cs1)=O C1(CNC(CS(=O)(=O)N(C)C)=O)CCC2(CN(C(c3cccc(F)c3N)=O)C2)O1 C1(NC(CN2CCC(OC)C2)=O)CN(C(=O)CCCN=[N+]=[N-])C2(CCCC2)C1 C1(CNC(C#CC(C)C)=O)(NC(=O)CN(C)S(N)(=O)=O)CC2CCC1CC2 C1(CC=C)(NC(=O)CCCCCCN)CCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CNC(CCN(CCC(C)(C)C)C)=O)CCC(NC(c2cnc(Cl)s2)=O)CC1 c1(NC(Cc2c(C(C)=O)cccc2)=O)ccc(NC(c2ccco2)=O)cc1Br C1(NC(c2ccc(C(=O)OC)o2)C)CC2(CCCN(C(=O)CN(C)NC(C)=O)C2)C1 N1(C(C(C(CC)CC)C)=O)CC2(NC(c3cncc(N)n3)=O)CCCC2(F)C1 CC(CC(=O)NC12CC(CNC(=O)C(O)Cc3ccccc3)(C1)C2)CC(C)(C)C C(=O)(C(F)CC(C)(C)C)NCCN(CCNC(c1cccc(CO)c1)=O)CC c1(C(=O)NCC(F)(F)C(F)(F)F)ccc(F)c(Br)c1F C1(C(=O)NC(C)CNC(=O)CCCCN2CCOC2=O)Cc2cccc(F)c2O1 c1(SC)nc(Cl)cc(=NCCC2CCN(C(c3cc(C)nc4ncnn34)=O)C2)[nH]1 c1(OC)nc(C(N2CCCC2CNC(C2CCCCC2C(N)=O)=O)=O)sc1C c1(-c2nc(C3C(C)CCN3)on2)c[nH]c2cc(OC(F)(F)F)ccc12 c1(C(=O)NCCNC(c2ccc(C)c(O)c2)=O)ccc2cnnc(O)c2c1 C1(CNC(C(CC)C)=O)CC2CCC(C1)N2C(C1CCS1(=O)=O)=O C1(C)(N(C)C)CC=CC1.C12CC(C1)CN(CC1CCCO1)C(=O)CONC2=O c1(C(N(C)CC)=O)ccc(C(=O)NC(C)CNC(C2(N=[N+]=[N-])CC2)=O)cc1 CN1CC(C(=O)NCC23CC(NC(c4csc(Cl)n4)=O)(C2)C3)CC1=O C(c1nc(C)co1)=CC(=O)NC1CCC(CNC(Cc2c(C)con2)=O)C1 Cc1noc2cc(C(N3CC(NC(c4cccc(N)c4)=O)C3)=O)ccc12 C(=O)(C(O)CC(F)F)NCC12OCC(CNC(c3ccc(NC(C)=O)s3)=O)(C1)C2 C1(C(=O)NCc2cc(C(=O)NC(COC)C(=O)OC)n[nH]2)CN2CCC1C2 C=CC(C)(O)CC(=O)NC(CO)C(C)NC(C1(C(F)F)CC(=C)C1)=O N1(C(c2cn(C)c(O)n2)=O)CC2(C1)CN(C(C1CC(S(C)(=O)=O)C1)=O)C2 Nc1cc(C(=O)NCCC2CCN(C(=O)CN(c3ccncc3)C)C2)ccc1F CC(C)(C)C(=O)C1(C(N2CC(c3cn(Cc4cccnc4)nn3)C2)=O)CCC1 CCC(C)(C)C(C)CC(=O)NC1CCCC(CNC(=O)CCC(C)C)C1 c1(-c2n(CC(=C)C)nc(C(C)O)n2)cn2cc(C)nc2s1 c1(C(CCC)NC(=O)C(C)N(C(=O)C(C)C)C)ccc(Cl)cc1 CCC(O)C(C)C(=O)NCC1CC1CNC(c1n[nH]cc1Br)=O N1(C(c2c(C(C)C)occ2)=O)CCC(F)C(NC(=O)C=C2CCCCC2)C1 CC(CC(F)F)C(=O)NCC1CC(F)CN1C(c1coc(CO)c1)=O c1(C(N2CCC(NC(CCOCCC)=O)C2(C)C)=O)cc(Cl)cc2c1CCC2 CN1CC2CCC(C1)N2C(C1CC=CCC1NC(C1(F)CC=CC1)=O)=O N1(C(CCNC(=O)OCC)=O)CCCC(N(C(=O)C(C)(COC)OC)C)C1 C1(NC(CCC=CCC=C)=O)(CF)CCN(C(c2snnc2C2CC2)=O)C1 C1(C(=O)NC2(CC=C)CN(C(c3ccc(C#N)o3)=O)C2)CC2C(C1)C2(F)F N1(C(COCCOC)=O)CCC(CCNC(c2ccc(OC)cc2Cl)=O)CC1C CCC(CC(=O)NCC1COCCN1C(=O)C=Cc1cc(C)no1)C1CCC1 C(C#Cc1cccc(C(=O)OC(C)(C)C)c1)NC(C1C(C)(COC)C1)=O C1(NC(Cc2ccc(C)c(F)c2)=O)CN(C(=O)C(C)C(C)O)C2(CCC2)C1 c1(C(N2CCCN(C(c3c(C)n(C)nc3)=O)CC2)=O)csc2ccccc12 Cc1[nH]c(C(=O)NCCOc2ccc(Br)nc2F)c(C)c1C(=O)OC(C)(C)C c1(CC(=O)NCC2(NC(C(C=C=C)C)=O)CC2)cnn2c1CCCC2 C12(C(=O)NCC#CCNC(C(C(C)C)NC(C)=O)=O)CCCN1CCC2 N1(C(CCN(CC)CC)=O)CC(N(C)C(c2ccc(C)cn2)=O)C(O)C1 c1(C(=O)NCCCN(C(C2CCN(C)CC2)=O)C)c(O)ccc(Cl)c1F c1(OC)ccc(C(=O)NC(C)(C)CC(=O)NCC=CCl)cn1 c1(NC(CCCOC)C)ncc(S(=O)(=O)NC(C)CCCC(F)(F)F)cc1Cl c1(C(=O)NC(CC(C)NC(c2n(CCC)ncc2)=O)C)cc(F)cc(F)c1 N1(C(C(=O)NC2(CO)CCS(=O)(=O)CC2)=O)CCC(C2(O)CNC2)CC1 N1(C(c2c(C)coc2)=O)CCC(C(=O)NC2CCCSCC2)CC1 C1(C(=O)NC(C2CCCC2)C)CCN1C(c1cc[nH]c1)=O C1(C2CCCN(c3nccc(C#N)n3)C2)(NC(c2ncc(OCC)nc2)=O)CC1 CC1(C)CN(C2CC2)CCC1NC(=O)C=Cc1nc[nH]n1 c1(C(=O)NC2CCCC(CNC(C3CCCCC3)=O)C2)cc2occc2[nH]1 C#CCCCC(C)C(=O)N1CCC(C)(C)C(C(N2CC(=O)NC(CC)C2)=O)C1 C=CC1(CC(=O)NC2CCC(O)C2)CN(C(=O)Cc2ccc(C)nc2)C1 c1(C(=O)NC2C(OC)CN(C(=O)COCP(C)(C)=O)C2)nc(Cl)ccc1N c1(CN2CCOCC2)cccc(C2(O)CCC2OC(F)(F)F)c1 c1(C(=O)NCC2CCCC(CNC(=O)CCCCCF)C2)cc2n(c1)CCCC2 CN1CC(C)(C)CC1C(N1CCCC(O)(CNC(=O)CC2(N(C)C)CCC2)C1)=O C1(Nc2c(C3c4nnnn4CCCO3)ccnc2)CC(C)(C)C12CCC2.CC.SC c1(C(=O)NCC2C(NC(c3[nH]cc(CS(C)(=O)=O)c3)=O)COC2)cc(O)nc(O)n1 C1(C(=O)NCCN(C(C(C)(C2CC2)OC)=O)C)CCC(CCC(C)C)CC1 C(CC(=O)Nn1cccn1)C1CCN(C(c2c(CC)ccs2)=O)C1 C1(NC(c2c(C)noc2C(C)C)=O)CN(C(C2CN(C(C)C)C2)=O)CC1(C)C C1(C(C(=O)NCCSC)N2CCC2C(C)C)CCC(CC2CC2)CC1 CC1C(NC(=O)CC2CCCCCCC2)CCCN1C(=O)Cc1ccsc1 c1(C(N2CC(NC(C(C)=C3CC3)=O)CC2(C)C)=O)sc(S(N)(=O)=O)c(C)c1Cl N(C(=NCc1ccnn1C)NCC1(C)CCCOC1)CC1(SCC)CC1 C1(NC(CC(=C)C)=O)CCCCC12CCN(C(=O)C(F)CC)C2 N1(C(c2c(Cl)ncc(OC)c2)=O)CCN(c2nnc(C3CC3)o2)CC(O)C1 c1(C(N2CCC(CCNC(C(C)C#N)=O)C2)=O)ccnc(CSCC(F)(F)F)c1 C1(C(=O)NC2(CNC(c3c(C)nc(CC(C)C)s3)=O)CC2)CC2CCC1CC2 C1(NC(C(N2CCCCC2)C)=O)COCC1C(=O)NCCn1cnnc1 C1(CNC(C(C=C)OC)=O)CN(C(=O)Cc2cnn(C)c2)CC1(F)CO CCCC(C(=O)NCC1CCCCN1C(c1oc(C)nc1CC)=O)OCC C1(CNC(C(CC=C)C)=O)CCC(C)(C)CN1C(=O)C(C)C(C)COC c1(C(N2CCCC(c3cc[nH]c(=N)n3)C2)C)cc(I)cc(I)c1 c12nc3ccc(nc3s1)O2.C1(NC(COC)=O)(CO)CCN(CC2CC2)CC1 CC(CO)CCN=c1[nH]c(=NC2CCCC2C(N)=O)[nH]c2c1COCC2 C=Cn1nccc1C(N1CCCC(C2CCCN2C(c2cnc(O)o2)=O)C1)=O C(=O)(CCCCC(=O)NCC1CCC2(CN(C(c3c(C)n[nH]c3C)=O)C2)O1)NC c1(C(=O)NC2CCN(C(c3ccncc3Br)=O)CC2O)ccn2ccnc2c1 N1(C(CCNC(C)=O)=O)CC(NC(c2nccnc2N)=O)CC(C)C1 N1(CC(=O)NC(CNC(C(C(C)C)O)=O)C2CC2)CCP(C)(=O)CC1 C1(C)(NC(C(CNC(C2C(C)=CCS2)=O)N(C)C)=O)CCCCCC1 CC1(C)CN(CCC(=O)NCCC(O)CNC(C23CCCC2C3)=O)CCS1 c1(CC(=O)N(CC(CC)NC(=O)C=CC(C)C)CC)ccc2nsnc2c1 c1(C(=O)NCCCN(C(=O)Cc2cncnc2)C)nccc2ccn(C)c12 C1(C(=O)NC(C=C)(C)C)CCCN(C(C2Cc3nccn3C2)=O)CC1 c1(C(c2nnnn2-c2ccccc2)(C2CCOC2)NCCCOC)ncc(Cl)cc1Cl c1(CCOCC)nc(C(=O)NCC(C)CNC(C2CCN(CC(C)C)C2)=O)co1 C1(CC(=O)N(c2c(C)nsc2)C)CCCN(C(=O)CC(C)C)C1 c1(C(=O)NCC(CNC(c2ncc(C)nc2)=O)O)ccc2c(C)cc(O)nc2c1 c1(C(N(CC)Cc2cc(C)on2)=O)cn2c(n1)CCN(CC1(CO)COC1)CC2 C(=O)(CS(=O)CCC(F)(F)F)NCC1CN(C(C2C(OC)(OC)CC2)=O)C1 N1(C(c2c(CC)ocn2)=O)CCCC2CN(c3cnc(C#N)c(C#N)n3)CCC12 C1(NC(C2C(CC)CCC2)=O)CCCC12CCN(C(=O)C(C1CC1)SC)CC2 c1(C(=O)NC(CN(C(C2C(C)C2C)=O)CC)C)cc(C(F)(F)F)ccc1Cl N1(C(C2N(C(c3c(C)ncs3)=O)CCOC2)=O)CCCC(C)(O)C1 c1(C(=O)NC(CCCNC(CC=C=C)=O)C)c(OC)ncnc1C Cc1oc(-c2ccsc2)nc1CC(=O)NCC(C)CNC(C1COCCO1)=O C1(NC(C2(N(C)C)CC2)=O)CN(C(=O)CCn2cccc2)CC2(CCC2)C1 c1(C(=O)NCC(CCCC)NC(C2C(=C)CC2)=O)cnc2onc(C)c2c1 N1(C(C2(C3CCCO3)CCOCC2)=O)CC2COCCC2(N)C1 C1(C(=O)NCC(CCOC)NC(c2occc2CN(C)C)=O)CCN(OC)CC1 Cc1ccc2nonc2c1C(=O)NC1(CO)CCN(C(C2CCOC2)=O)C1 C1(CC)CN(C(=O)CC2CC=CC2)CCC1NC(c1c(Cl)c(C)nn1C)=O c1(C(=O)NCC(C(C)C)(C)NC(=O)C(O)CN(C)C)ccc(=O)n(C)c1 N1(C(c2c(C(C)C)ncs2)=O)CCC(C(F)(F)F)C(CNC(C2(F)CC2)=O)C1 Cc1cccc(-n2cc(C(c3nnnn3C)NC(C3(C)CC=CC3)=O)cn2)c1 N1(C(CC2C(OC)(OC)CC2)=O)CCC(N(C(=O)COc2ccsn2)C)C1 CC1CCCCN1CCC(=O)NC1CCC1CNC(=O)Cc1ccsc1Cl c1(C(=O)OC)ccc(Br)cc1S(=O)(=O)N1CC(c2cccc(F)c2)C1 c1(CC(N2C(CCNC(C(C(CC)O)C)=O)CCC2)=O)noc2ccccc12 CCCC(CCCNC(c1nc(Br)sc1C)=O)NC(C12CCC(C1)C2)=O C(CC(C(=O)NCCc1ccccc1O)NC(C1COCCN1C)=O)SC N1(C(c2nn(C)c(F)c2)=O)CC(C2CN(C(C3CC3c3ccnn3C)=O)C2)C1 c1(C(N2C(CNC(=O)Cn3cccc3)CCCC2)=O)ccc(OC(F)F)c(F)c1 c1(C(C)C)c(C(=O)NC2CN(C(=O)Cc3ccns3)CC2F)cnn1C N1(C(C(CCC)F)=O)CCC(CNC(=O)C2=C(C)CC2)C12CC2 C1(CC(=O)NCCCC(C)O)CCN(C(C2CC2C2(C)COC2)=O)C1(C)C c1(CCCNC(CCN(C(C2CCC(F)C2)=O)CC)=O)nc(C)no1 c1(OC)ccc(F)cc1C1CCCN1CCCNS(C)(=O)=O c1(NC(=O)CC2COCCO2)cccnc1CC(N1CCOCC1C1CC1)=O C(C(C(=O)NCCCCCN(C)C)C(C)(C)C)NC(C(COC)COC)=O Cc1sc(Br)cc1C(=O)NCCC1CCN(C(C2CC(N(C)C)C2)=O)C1 N1(C(C(=O)NC(c2ccc(Cl)s2)COC)=O)CCC(CC(=O)N(C)C)CC1 c1(C(N(C2CN(C(CC(COC)C)=O)CC23CC3)C)=O)ccc([N+](=O)[O-])n1C N1(C(c2ccnc(Cl)c2Cl)C(=O)NCc2cccnc2)CCOCC(C2CC2)C1 C(=O)(C#CC1CCOCC1)N(CCCCC(=O)NCC1(O)CCCOC1)C c1(CNC(C2(CC)COC2)=O)cnn2c1CN(c1ccc(C(N)=O)cn1)CC2 C1(NC(c2cnc(C(C)C)o2)=O)CN(C(C2CC=CCO2)=O)CC1(C)C c1(C(=O)NCC2CC(C)(C)N(C(c3ccncc3)=O)C2)ccc2c(c1)COC2 CC(C)CCC(F)C(=O)N1CC(N(C(=O)CCc2ccncn2)C)C(F)C1 c1(C(=O)NCCCC(C)NC(C=C(C)c2ccsc2)=O)cccc2nsnc12 N1(C(=O)CC2(CO)CC2)CCN(C(c2csc(-c3ccccn3)n2)=O)CC(O)C1 c1(C(N2CC(CC(N3CCOCC3C3CC3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 C1(NC(c2ccnc(C)n2)=O)CCN(C(=O)CC2CCC(=O)N2)C12CCC2 n1(CC(N2CC(N(C(c3c(COC)noc3)=O)C)C2)=O)cnc2ccc(C)cc12 N1(CCCCNCC(c2ccccc2C)OC)CCN(CCO)CC1 c1(C(=O)NCC2(CCNC(CSCC(=O)OC)=O)CC2)cc2c(F)cccc2[nH]1 C#CCC(C)(CC)C(=O)NC1CC1NC(=O)CCCC#CC C1(C(=O)NC(C)CCO)C2CC(CC2F)N1C(c1ccc(C(F)(F)F)cc1)=O C=CCCCCC(=O)NC(C)CN(C(=O)Cc1n[nH]cc1Br)CC c1(NCC(C)CC2CC2)nc(N(C)Cc2c(F)cccc2Br)c2c(n1)CCC2 c1(C(=O)NCC2C(NC(C=CCOC)=O)CCCC2)ccc(F)c(C#N)c1 C1(C(=O)NC(CC)(C)C)CN(C(C2CCC(F)CC2)=O)CC1CC(C)(C)C C1(COCC)CCCN(C(C2CCC3(c4ccc(COC)cc4)CC23)=O)C1 Cc1ccnnc1C(=O)N(CC(CO)(CO)NC(C1CCSC(C)C1)=O)C C1(NC(C(COC)O)=O)CCN(C(=O)Cc2cccc(F)c2)CC1F N1(C(Cc2c(C)noc2C)=O)CCOCC(C(=O)NC(C)CCO)C1 C(C(C(CS)(C)CC)CCCCC)NC(CC)COC N1(C(=O)NCc2cn(C(c3ccn(C)n3)=O)nn2)CCCS1(=O)=O c1(NC(c2csc(NC(c3ccc(Br)nc3)=O)n2)=O)cccc2ncsc12 c1(C(=O)NCC(CC(=O)N(C)CCN(C)CCO)OC)ccc(=O)n(C)n1 c1(C(N2CC(N(C(=O)C(C)(F)c3ccccc3)C)C2)=O)ccccc1OC(F)F CC(C)C(O)C(C)C(=O)NC(C)CN(C(=O)CCc1cnc(C2CC2)o1)C C(=O)(C(CNC(=O)CC(C)C)CC1CN(C(C2CC2(F)Cl)=O)C1)OC C(=O)(CCCN=[N+]=[N-])N1CC2C(CN(C(CN(CCOC)C)=O)C)C2C1 c1(C(N2C3(CCN(C(C4C(C=C)C4)=O)C3)CCC2)=O)ccnc2cc(F)cnc12 N1(C(Cc2c(C)nc[nH]2)=O)CC2CCOC2(CNC(=O)Cc2ccsc2)C1 C1(CC(N2CCC3(CCCN3C(=O)CCBr)C2)=O)COc2ccccc2O1 CCS(=O)(=O)CC(=O)NC1CCN(Cc2ccc(Br)c(C)n2)CC1C C1(C(=O)NC(CC)C(C)(F)F)CC1C1CN(C(=O)C(C)c2ccco2)C1 C(=O)(CC1=Cc2ccccc2C1)N(C)CCN(C)C(C1CCCCC(F)(F)C1)=O C1(OC)CCC(NC(C2(NC(c3nccn3C)=O)CCSC2)=O)CC1 C1(C(=O)NCc2ccc(OC(C)C)nc2)CCCN(C(=O)CNC=O)CC1 c1(C(=O)OC)ccc2c(c1)CN(C(C1(C#N)CCC1)=O)CC2 C1(C2CN(C(C3Cc4cscc4C3)=O)C2)(NC(c2cc(C3CC3)ns2)=O)CC1 c1(C(N2CC(=C(CNC(c3cc(C)sn3)=O)F)C2)=O)c(C(F)F)nn(C)c1C c1(C(N2C3CN(C(=O)CCCCBr)CC32)=O)cccc2c1CCC2 c1(C(=O)NCCCNC(Cc2cc(C)on2)=O)cnccc1N1CCCC1 C(=O)(C1CSc2ccccc21)NCCC1(O)CCN(C(C#CC(C)(C)C)=O)CC1 n1(CC)nc(C(N2CC3C(N(C4(C)CCC4)C)C3C2)=O)cc1C(=O)OCC N1(C(C2(CC=C)CC=CC2)=O)CC2(CC(C(=O)Nc3cncc(OC)c3)CO2)C1 C=CCCCC(C(=O)NCCC(F)(F)CO)NC(c1csc(Cl)n1)=O C12CCC3(CCC3)N(C1)C2=O.O=C1NCCN1CCC1CC1 c1(CNC(NCC(=O)NCC#C)=NCCCCl)noc2c1CC(C)CC2 c1(CC)c(C(=O)NC2CN(C(=O)C=C3CCC3)CC2(C)C)cccc1C C(=O)(CC(F)(F)F)NCc1cccc(CN(C)C(c2nnn(C)n2)=O)c1 C(=O)(C(C)C(C)NC(=O)C(C)c1ccco1)NCc1cn(CC)nc1 C(CCCCC(=O)NC(C(=O)NC(C)Cc1cccnc1)C1CCOC1)OC C1(CC=C)(NC(C2CC(n3ccnn3)C2)=O)CCN(C(=O)C(C)SCCCC)CC1 N1(C(C23N(C(c4n(CCC)ncc4)=O)CCC2C3)=O)CC2(CCNC(=O)O2)C1 C1(NC(C(c2cnn(C)c2)NC(C(C)c2ccsc2)=O)=O)CCCC(O)C1O C=CC(C(=O)N(C)CCOCCNC(c1n[nH]cc1F)=O)c1ccccc1 c1(C(N2CC(C(=O)NC(CC#C)C(N)=O)C(CC)C2)=O)ccc(C=C)cc1 C1(NC(CC=CCC)=O)CN(C(=O)CC(C)F)C2(CCCCCC2)C1 N1(C(c2c(C)cco2)=O)CCC2CCN(C(=O)CCCc3cccnc3)CC2C1 OC1c2ccccc2CC1CCCCN1CCN(c2ncnc(C(F)F)c2Br)CC1 C12(CNC(C(C)NC(C)(C)C)=O)CN(C(c3ccc(N)cc3F)=O)CC1CCO2 c1(CC)cc(OCC(=O)NC2(C)CCN(C(=O)CC=C(C)C)C2)ccc1Cl CC1C(=O)CCC1CC(N1CCC(C2CCCN2C(c2ccn(C)c2)=O)CC1)=O Cc1ccc(CC(=O)NCC2CCN(C(=O)CN(c3ccccc3)C)CC2)cc1 Cc1nc(C)c(CC(=O)NCC2C=CC(NC(=O)Cc3cncc(F)c3)C2)s1 c1(C(=O)NCC2CCC(C)N(C(c3ccoc3)=O)C2)cc2sccc2cn1 C(=O)(N1CC2COCC2O1)C1N(C(CC(C)F)=O)CCCCC1 C(=O)(C(F)C(C)(C)O)N(C(CNC(c1c(OC)n(C)nc1)=O)C)C C(=O)(N=c1ncn(Cc2cccc(F)c2)[nH]1)c1ccc(N(CC#N)C)cc1 c1(C(N(C2C3CCOC3C2(C)C)C)=O)ccc(S(N)(=O)=O)c(N)c1 C(=O)(CN=c1ccnc[nH]1)NC(CCCC)CNC(=O)Cc1ccc(OC)nc1 N1(C(C(=O)Nc2nc(CSC)c(C3CC3)s2)=O)CC2CC(C1)C2(F)F c1(C(N(C(c2ccccc2)CNC(C(F)=CC)=O)C)=O)cc(C)c(C)[nH]1 C1(C(=O)NC2(C(F)(F)F)CCC2)C2CCC(C2)N1C(c1cccc(Cl)c1F)=O c1(C(N2CC(C(=O)NCC)C2)=O)ccnc2c1CCC2 c1(C(N2CCC3CCN(C(c4ccco4)=O)CC32)=O)cc2ncccc2cc1Cl N1(C(Cc2c(OC)noc2C)=O)C(C)C2CC1C2NC(c1c[nH]c(Br)c1)=O C1(C(N2C(C)CN(C(=O)CC3CCC(O)C3)CCC2)=O)CC(C)(C)OC(C)(C)C1 C1(C(=O)NCCOCC(N2C(C)(COC)CCC2)=O)CC2CC1CC2O N1(C(CCC=CC)=O)CCC(CCF)(C(=O)O)C1 C1C(C(C)(C)C)C(=O)N1C1CC1.C1(C)(C(C)C)CC1C(=O)NCCC(C)C C(CN=c1[nH]c(=NC2COC(C(C)C)C2)[nH]c2cccnc12)SCC C1(CNC(C(C)C(F)F)=O)CCC2(CCC2)C1NC(c1ccc2occc2n1)=O C1(CNC(C(C#N)C2CC2)=O)CC2CCC1N(C(C1CCC(=O)N1)=O)C2 C1(CC(C(=O)NCCCSC)N(CC(C)C(=O)OC)C)CCCCN1C(C)=O c1(C(N2CC(NC(c3cnncc3O)=O)C(CO)CC2)=O)nc2cnccc2s1 c1(N(CC(=O)OCC)CC2CC2)cc(C(N)=O)nc2ccc(Br)cc12 CCC(CCC(=O)N1C(CO)CC1C)NC(c1ccncc1)=O C1(NC(C(C)n2cccn2)=O)CC2CC1N(C(c1ccn(C)c1)=O)C2 c1(CC)c(C(=O)NCC(C)CNC(c2c(Cl)c(C)nn2C)=O)cccc1C C(=O)(CC(C(CC)CC)C(COCCOC)=O)NCC(C)(C)N.C(=O)(N)NC(C)C C1(CNC(CCC#CC)=O)CCCCCN1C(=O)CNC(=O)Nc1ccccc1 C1(CC(=O)NCC(CC)N(C)C)CC(C)(C)CN1C(=O)CC1CNC(=O)O1 C1(C(=O)NCC(CN(C(CCOCC#C)=O)C)C)CCCCC1n1cccc1 C1(CCOC)CN(C(=O)C(C)OCC(C)C)CCN1C(c1cc(=N)[nH]n1C)=O C1(C(=O)NCc2cn(C3CN(C(c4ccno4)=O)C3)nn2)CC2CCC1O2 CC1(C)COCC(C(=O)NC2CN(C(=O)CCC3CC3(C)C)CC2(C)C)O1 C1(OC)CC2CC(OC)C2C1.N1(C(Cc2cn(CC)nn2)=O)CC2CC1(CO)C2 c1(C(N)=O)cc(C(=O)NC2CCC2NC(c2cc(-c3ccco3)[nH]n2)=O)co1 N1(C(c2c(I)ccc(C)c2)=O)CCc2cc(-c3ccnc(C)c3)ccc2C1 c1(C(=O)NC2C(CNC(c3cc(C)on3)=O)CCC2)csc2c1CCCC2 N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)COCP(C)(C)=O)CC1CC(F)F c1(OC)ccc(-n2nnnc2C(c2occc2Br)NCC(C)C2CCC2)c(C)c1 N1(C(c2c(=N)[nH][nH]c2)=O)CCC2(CCC2)C(NC(C2CCCC(F)(F)C2)=O)C1 c1(C(=O)NCC2=CCN(C(c3c(C)nc(N)cn3)=O)CC2)cccc2nn[nH]c12 N1(C(CC=C=C)=O)CCCC2CN(C(C3(OCC)CCSCC3)=O)CCC12 Cc1cnnc(O)c1C(N1CC2(NC(C3CCC(N(C)C)C3)=O)CC1C2)=O C1(COC)C=CCCN1C(C1(NC(=O)CNC(=O)NC)CCCC1C)=O S(=O)(=O)(c1cc(CN=c2ccc(OC3CCCCC3)n[nH]2)ccc1Cl)CC(=O)O CC(C(=O)NCCN(C)C(C1CC1c1cnn(C)c1)=O)C(C)(F)F c1(CC)ccc(C(=O)NC2CC(C)N(C(=O)CCC(C)CN(C)C)C2)c(C)c1 NCCCC(=O)NCc1cc(C(F)(F)F)cs1 CCC(C(=O)NCCCOCCC(=O)N(C)CCOCCO)C(C)(C)CC CC(C)(C(=O)NCC(CNC(C1CC2C=CC1C2)=O)C(F)(F)F)C1=CCSCC1 N1(C(COCC#C)=O)CC(CNC(=O)C(C=C)c2ccccc2)CC1(C)C C1(O)(CC)CCCN(C(=O)CC2COCCN2C(c2ccncc2O)=O)C1 CCC(CC(=O)NCCC(O)C(C)C)NC(c1ccn(CCF)n1)=O c1(C(N(C(C)CNC(=O)CNC(=O)NCCCCCC)CC)=O)ccc(CO)s1 C(CC(=O)NC1CCC(C(N)=O)CC1)(C(C)(C)C)NC(c1cn(CC=C)nn1)=O C1(NC(Cc2c(C)ncs2)=O)CCCC(N(C)C(c2ccc(C(F)F)cc2)=O)C1 CC1(C)CCc2onc(C(=O)NCCC3CN(C(=O)C=Cc4ccsc4)C3)c2C1 Cc1sc(C(N2CCC(C)(NC(c3cc4occc4[nH]3)=O)C2)=O)c(C)c1C CN1CCCC1CCNC(C1CC(N(C(=O)CC2CC2C2CC2)C)C1)=O C1(NC(Cc2cccc(OCC)n2)=O)CCCN(C(C2CSC2)=O)C1CC C1(C(=O)NCCCc2ccco2)(CC)CCCN1C(c1cn(C)c(C)n1)=O C(C)(C)(CC(F)C(=O)N1CCN(C(C)(C)C)CC1)NC(C(C(COC)C)C)=O C1(c2cn(CCCC(C)(F)CNC(c3c(C)nns3)=O)nn2)CCCNC1=O N1(C(C(C(C)(C)C)O)=O)CCC(C2CN(C(=O)CCCNC(=O)C3CC3)C2)CC1 N1(C(c2cccc(C#C)c2)=O)CC2CC(C1)CN(C(c1cnn3ccsc13)=O)C2 N1(C(c2c(C)ccs2)=O)CC2CCN(C(c3cnn4c3CCC4)=O)CC2C1 n1(CC(=O)NCC(CNC(C2(CC)CCC2)=O)(C)C)nnc2c1CCCC2 Cc1ccc(C(N2CC=CC2CNC(C2(C)CCC(=O)N(C)C2)=O)=O)c(N)c1C N1(C(C2CCC(C)(C)C2)=O)CCOC(C)(CNC(=O)Cc2csnn2)C1 C1(C2CN(C(=O)CCF)C2)(NC(=O)CC2CCCCC2F)CC1 c1(C(N2CC(OC)(CNC(=O)CNC(=O)CN(C)C)C2)=O)ccc(Cl)cn1 N1(C(CCS(N)(=O)=O)=O)CC2CCN(C(c3cnc4[nH]ncc4c3)=O)CC12 C1(C(=O)NC(CC(=O)NCc2c(C)cncc2)C2CC2)CCOC(=O)CC1 CCC(C)(COC)C(=O)NCCOCC(N1CCCC(O)C1)=O Cc1cc(C)c(C(=O)NC2CCN(C(c3ccc(F)c(N)c3)=O)CC2F)c(O)n1 N1(C(CCC=C)=O)CC(C)CCC1C(=O)Nc1cccc(C(C)=O)c1 c1(C(C(=O)NCC(=C)C)N(C2CCC2)CC)cnn2c1CCC2 c1(C(N2CCC(NC(=O)C(O)C3CC3)C2)=O)ccc(-c2ccncc2)cc1F c1(C(=O)NC2CC2)occ2c1CCC2.C12CN(C1)C(=O)CN2CC#C Cc1cc(C(=O)N(C2CC(C(=O)NC3CC(O)C(F)C3)C2)C)cc(C)n1 Cc1cc(C(=O)NCCCNC(=O)CC(=O)OC(C)(C)C)c(S(N)(=O)=O)s1 N1(CC(=O)N(C2CCN(CC(=O)C3CC3)CC2)CC)CCC(C)(C#N)C1 C(N=c1cc(NCc2nc(-c3ccc(Cl)cc3)no2)nc[nH]1)c1n(CC)cnc1 c1(C(N2CC(NC(C3(C(F)(F)F)CC(=C)C3)=O)C(OC)C2)=O)ccc(F)c(C)c1 C1(N(C(C)(C)C)C)CCn2cncc2C1.c1c2cn(c(=O)c1)CC2 CC1=C(C(=O)NCC2CC(C)N(C(c3cnccn3)=O)C2)CCCC1 C12(CNC(CC3(C)CC3)=O)CCC(CC1)N(C(c1cn(C3CCOC3)nn1)=O)C2 CC1=C(C)CC(C)(C(N2C3CCC2CC(NC(c2cnc(C)cn2)=O)C3)=O)CC1 C1(CC=C)(NC(c2ccc(OCC)cc2C)=O)CCCN(C(c2cn[nH]c2)=O)C1 Cc1nn(C)c(Cl)c1CC(=O)NC1(CNC(c2cccc(OCF)c2)=O)CCC1 C(=O)(CS(=O)(=O)CC(C)C)NCC1C(NC(CSCC#C)=O)CCC(C)(C)C1 N1(C(Cc2n[nH]c(=N)s2)=O)CCCCC(CNC(=O)C(c2ccccc2)F)C1 c1(CCNC(=O)NC2N(CC(CCC)C)CC2)noc(=O)n1C Cc1c(NC(=O)NC(C)C(C)(C)CO)cnc(F)c1Br C(=O)(C(O)C(C)(C)C)N(CCCNC(=O)CC1CCCOCC1)CCC N1(C(C(C)(C)CC2CC2)=O)CC2CCC1CC2NC(c1ccnn1C1CCC1)=O c1(C(N2CC(NC(=O)C(O)c3ccco3)C3(C2)CC3)=O)cccc2nc(O)[nH]c12 C1(C(=O)NCCCNC(c2ccnc(N3CCCC3)c2)=O)CCN(C2CC2)C1=O C1(O)(CC(C)N(C2CC3(C(=O)O)CC23)C)CN(C(=O)OC(C)(C)C)C1 C1(CNC(Cc2c(C)ocn2)=O)C(O)C(O)CN1C(c1cncc(Br)c1)=O n1(CC(=O)NC(CNC(c2ccnnc2)=O)C2CCC2)cc(Cl)c(O)nc1=O c1(C(=O)NCC2CC(NC(CC(CC)C)=O)C2)cccc2[nH]c(=N)oc12 C(=O)(C1=CCC(C)(C)CC1)N(CCC(=O)N(C12CC(C1)C2)C1CC1)C(C)C c1(C(=O)NCC(C2CCCCC2)C)cc(C2CC2)nn1-c1ccc(Br)cc1 Cc1c[nH]c2cc(C(=O)NC3CCN(Cc4c(F)cccc4Br)CC3F)ccc12 C1(C(N(C2CCCN(C(C(F)=C(C)C)=O)C2)CCO)=O)CCc2c[nH]nc2C1 C1(O)(NC(N)=O)CCN(C(=O)C(O)C2CN(C(C3CN(C4COC4)C3)=O)C2)C1 c1(C(N2C(CNC(=O)COCC3CCOC3)CC2)=O)c[nH]nc1[N+](=O)[O-] CCCCCCCCCC=CC(=O)NCCCN(C(=O)Cc1cnns1)C C12(CC(=O)N(CCC)CC3CC3)CC(CO1)N(C(=O)CC(=O)OC)C2 CC1CCC=C1C(=O)NC1CN(C(c2cc(Br)cs2)=O)C(C)(C)C1 C1(C(=O)NCc2c(C)coc2C)CN(C(c2cnsc2)=O)C2(CCC2)C1 CC(C)(C(=O)N1CC2CC2(CNC(c2c[nH]nc2C(C)(C)C)=O)C1)C(N)=O C1(C)(NC(COCC#C)=O)CCN(C(C2CC2c2ccccc2)=O)C1 C=CC(CCC)CC(=O)NC(CNC(c1ccc(CC)[nH]1)=O)CC(C)C c1(OC)ccc2cc(C(=O)NC(C)CNC(c3cccc(F)c3)=O)c(=O)oc2c1 c1(C(N2C(c3ccc(C)cc3)CCCC2)C(=O)NCC2CC2)cccc(Cl)c1C c1(NCC(CC)(C)CO)ncnc(N2CCN(C(=O)NC)CC2)c1C C1(NC(C(=O)NCC(C)C)C)CCC(NC(=O)CCNC(=O)CO)C1 c1(C(N2CC(C(C)NC(c3n(C=C)nnc3)=O)OCC2)=O)ncn2ccccc12 c1(OCC)ccc(C(=O)NC2CSCCN2C(=O)C(O)CC)cc1[N+](=O)[O-] Nc1c(C(N2CCNC(C(F)(F)F)C2)=O)ccc(F)c1Br Cc1ccc(C(=O)NC2CCC(NC(=O)CN3CCCCCC3)CC2)c(F)c1F Cc1ccc(N(C(=O)CN(C)C2CC2)Cc2ccc(C)s2)cc1 N1(C(c2cc(CC)on2)=O)CCCN(C(=O)C(N2CCCC2CC)=O)CCC1 C(=O)(CCC(C(N)=O)NC(N1CCN(C(C)C)CC1C)=O)OC(C)C C1(C(=O)NCC2(F)CN(C(c3cnc(C)nc3C)=O)C2)C2CCC(C2)S1(=O)=O c1(NC(c2c(C3CC3)ccc(OC)c2)=O)cccc(S(C)=O)c1 C1(O)(C(=O)NC2C(NC(C3(C)CC4CCC3O4)=O)CCC2)CC2(CCOCC2)C1 C1(C(=O)NC2(CC(N)=O)CCN(C(c3ccc(C4CC4)o3)=O)C2)CCCCC(=O)N1 c1(C(=O)NCC2N(C(c3cn(C)c(=O)n3C)=O)CC=C2)cnc2c(n1)CCCC2 C(=O)(CCCCCC(C)C)NC(CC#C)(C)C(=O)N(C)CC1CCN(C)C1 n1(CC(=O)NCCC2CCC(NC(C3(CC)CC3)=O)C2)ccc2cc(F)ccc12 C1(C(N(CC(CC)NC(c2cnn(CC)c2C)=O)C)=O)C=CC=CC=C1 C1(C)(C(N2CC(C)N(C(C3CCOC(C)C3)=O)CC2)=O)Cc2ccccc2C1 c1(N2CCC(NCC3(OC)CCSCC3)C2)c(OC(C)C)cccc1Cl C(=O)(CC1=CCCCC1)N1C(C2(NC(C(c3cccc(C)c3)C)=O)CC2)CCC1 c1(C(C)C)ccc(C(=O)NC2CCCCC2NC(=O)CC(C)(C)C)cc1Cl C12(C(N(CCCOC)C)=O)CCC(CN1C(c1cccnc1OC(C)(C)C)=O)C2 O=C1CCc2cc(C(N3CC4CC3CN4C(C3CC3(Cl)Cl)=O)=O)ccc21 c1(C(=O)NCC(N2CC(CNC(CC(C=C)C)=O)(OC)C2)=O)ccc(F)cc1F Cc1ccc2cc(C(=O)NCC(N3CCC(O)CC3)c3ccccc3)ncn12 C1(NC(c2ccc(CSCC)cc2)=O)CCCN(C(c2conc2C)=O)CC1F N1(C(c2c(CC)occ2)=O)CC2CCN(C(c3ccc(C(F)F)cc3F)=O)CC12 CCC(F)(F)C(C)(C)NC(=O)CC1C=CC(NC(=O)C(C)OC(C)(C)C)C1 c1(CN(CCCP(C)(C)=O)C(C)(C)C)ccc(F)cc1Cl C(=O)(CC(F)(F)CC(=O)OC)N1C(C)(C(=O)Nc2cc(OC)cc(Cl)n2)CC1 C1(NC(C=CC=C)=O)CCCN(C(c2cncn2C(F)(F)F)=O)C1 C(N=c1[nH]c(Cl)ncc1Cl)C1CCN(C(C2ON=C(C)C2)=O)CC1C c1(NC(C(C)N(C(CC#C)C(=O)OCC)C)=O)cccc2ccoc12 Cc1ccc2c(=NCC3CC4(C3)CC43CCC3)[nH]c(=NC(C)CN(C)C)[nH]c2c1 C1(NC(c2ccc(C(=O)NCC3CC3)cc2)=O)CC(O)C(O)CO1 c1(C(=O)NC2CCC2)cccnc1CNC(C1CCCCC1F)=O CCC(C)(C(=O)N(C)C(C1CN(C(=O)C(C)C2(O)CCC2)C1)C1CC1)OC C1(CN(C(C)(C)C)CC=CC(=O)OC)CC(NC(=O)C(F)CC2CCC2)C1(C)C c1(CC(=O)NC2CC(NC(c3cccc4nncn34)=O)C2)ccc2c(c1)COC2 c1(C(N2CC(NC(CCCN(C)C)=O)C(F)(F)C2)=O)cc([N+](=O)[O-])c(F)cc1F c1(CNc2cncc(-c3c(C#N)nccc3)c2)c(Cl)ccc(F)c1F C1(CNC(Cn2c(C)nnn2)=O)CC2(CCC2)CN1C(c1ccc(F)c(N)c1)=O C=Cc1ccc(C(=O)NC2CN(C(c3csc(Br)n3)=O)CC2OC)cc1 CC1=CC(C)=NS(=O)(=O)N1CC(N1CC2C(NC(=O)C(C#N)C(C)(C)C)C2C1)=O c1(C(C(=O)NC2CC(NC(=O)Nc3cc(OC)ncn3)C2)OC)c(Cl)cccc1Cl n1(CC(=O)N(C(C)CNC(=O)C(C)(C)CCOC)CC)nc(Cl)ccc1=O c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccc(F)cc1OC N1(C(C(C)=C(CC)C)=O)CCC(NC(=O)Cc2ccc(F)cc2)CC1C N1(C(C=C2CCN(C)C2)=O)CCOC2(C1)CN(C(=O)CCn1cnnn1)C2 N(C(=NCc1ncc(Br)cn1)NC(C)Cc1ccccc1)Cc1c(C)ccs1 N1(C(CN(CCCC)C)=O)CCCC1C(O)CO C1(C)(CNC(c2cnc(OC)s2)=O)CC(F)(F)CN1C(=O)CN(C1CCSC1)C C(C(O)CC(F)(F)F)NC(C(CNC(c1cc(CO)on1)=O)N(C)C)=O N1(C(CC(CC)C)=O)CCCC2C1CCN2C(=O)CCCCCl C(=O)(N=c1[nH]n(C)cc1P(C)(C)=O)NC1C(CC)CN(S(C)(=O)=O)CC1 Cc1csc2c(CC(=O)NC3(C4CN(C(=O)C(C)(Cl)Cl)C4)CC3)cccc12 N1(C(C2C(CC)CN(C(=O)C=Cc3ccoc3)C2)=O)CCCSCC1C c1(C(=O)NCCC(CNC(c2csc(S)n2)=O)O)c[nH]c(=O)c2ccnn12 C1(C(=O)NCC(CC(C)C)NC(=O)CCc2cncnc2)CN2CCC1CC2 C1(NC(C(c2ccccc2Cl)C)=O)CC2(C1)CC(CNC(=O)CC1CC(F)C1)C2 S(=O)(=O)(c1ccc(C)c(C)c1)NCC(N1CCCC(CNC(CSCC)=O)C1)=O C(c1cncc2ccccc12)=CC(N1CC2NCCOC2C1)=O c1(OC)cnnc(C(N2CCCCC2C(N2CCCC2CN=[N+]=[N-])=O)=O)c1 C#CC1CN(C(=O)NC(c2cc(C)on2)C)CCN1C(=O)OC(C)(C)C C1(=O)CCCC(=O)N2CCCC(CC2)N1.C(=O)(C(C)(C)C)N(C)C C1(CNC(c2c(OC)csc2)=O)CC(NC(=O)C=C(C)Cl)C1(C)C Cc1ccc(C)c(C(N2CC(CNC(=O)Cc3csc(Cl)n3)CCC2C)=O)n1 c1(CC(N2CC(F)(CNC(C3C(C)CCC3)=O)C2)=O)ccc(Br)c(Cl)c1 C1(NC(CC(C)SC)=O)CC2(C1)CC(NC(=O)Cc1c(Cl)cccc1Cl)C2 c1(C(N2CC(CNC(c3c(C)nc(C4CC4)s3)=O)C2)=O)ccc(S(C)(=O)=O)cc1 c1(C(=O)NC2CCN(C(CSCC)=O)C(C)C2)ccc(C)c(Cl)c1Cl N1(C(c2ccc(C(C)=O)cc2)=O)CCC2C(NC(c3ncn(C)n3)=O)C2CC1 c1(C(N(C)CCN(C)C(c2cnc(C3CCCO3)s2)=O)=O)cc(=O)cc(Cl)[nH]1 N1(C(CNC(CCC)=O)=O)CCCC1C(C)(C)CNC(=O)Cc1ncc(Br)s1 N1(C(=O)OC(C)(C)C)CC(O)CC1C(N1CCC(NC(c2cc[nH]n2)=O)CC1)=O C1(C(N2CCC(C(=O)OC)CC2)=O)CNC(=O)CN1C(c1cc(C2CC2)cs1)=O Cc1nn(C)c(F)c1C(=O)NCc1ccccc1CNC(C1COCC(C)O1)=O N1(C(c2cc(OC)c(Br)s2)=O)CCC(C)(c2cn(-c3cncc(Cl)c3)nn2)CC1 c1(C(C)O)cn(CC(=O)NCC2(NC(c3cc(Cl)no3)=O)CCCC2)nn1 CC(Cc1ccccn1)C(=O)NCCCNC(=O)CNS(=O)(=O)CCOC1CC1 N1(C(C(C=CCCC)O)=O)C2CCC1CN(C(c1cccc(CC#N)c1)=O)C2 C(CNC(c1cnn(C2CCC2)n1)=O)(C(C)(C)C)NC(CCC1C(C)C1)=O C1(C(=O)NC2C(OC)CN(C(c3cc[nH]n3)=O)C2)CC(=O)NC(=O)N1 C(=O)(C1CCc2c(Cl)cccc21)N1CC(O)(CNC(C(C(C)(C)F)(C)F)=O)C1 c1(CCC(=O)NCC2CCC(NC(=O)CNC(=O)C3CC3)C2)cccnc1Cl C1(F)(C(=O)NC2CCN(C(Cn3c(C)c(Cl)cn3)=O)C2)CCC2(CCC2)C1 C1(CNC(CC(C)SC)=O)CC(C)(C)CN1C(c1coc(N(C)C)n1)=O C1(CC(=O)NCCOC2CCN(C(=O)CC3CC3)C2)CCCOCC1 C(C(=O)N1CC=CC(C(=O)NCC2(N(C)C)CCCC2)C1)(C(C)(C)C)OC c1(OC)cc2c3c([nH]c2cc1Cl)CCN(C(=O)NCC1CCOCC12CCC2)C3 N1(C(c2nccc(OC)c2)=O)CCC2CN(C(=O)CCCCCC(C)C)CCC12 N1(C(c2cc(CC)on2)=O)CCCOC(CNC(=O)Cc2ccco2)C1 C1(C2N(C(CCOC(C)=O)=O)CCC2)CCCN(C(c2ccn(C)n2)=O)C1 C(=O)(C1CCc2snnc21)NC(CCCNC(CC(CC)(C)C)=O)CO c1(C(=O)NC(CNC(COC(C)C)=O)(C)C)coc(C(N)=O)c1 C(=O)(C1=CC2CC=CCC12)NCCC1(NC(c2c(CCC)nco2)=O)CC1 c1(OC)cc(C(=O)NC2CC(F)CN(C(=O)CCOC(C)=O)C2)c(Cl)cc1Cl CC1CN2CCN1C(C(N1CC(CNC(C3CCS(=O)(=O)N3)=O)CC1(C)C)=O)C2 N#CCCCCCC(=O)N1CC(F)CC1CNC(=O)C=Cc1cccc(Cl)c1 c1(C(=O)NC2C(NC(C3N(C(C)C)C(=O)CC3)=O)CCC2)ccccc1[N+](=O)[O-] C1(C(N2CC(COC)C2)=O)COC(CNC(=O)C(C)CO)C1 C(=O)(CCCCC(F)F)N1C2CC(CNC(=O)C3=CCCCO3)(OC2)C1 Cc1ccc(C(N2CCC(C)(NC(c3cccc(O)c3C)=O)C2)=O)cc1C N1(c2nc(SC)c(C)cn2)CCOCC12COCCN(C(C1CCCOC1)=O)C2 CC(C)C(C#N)C(=O)N1CCC(CNC(=O)CCc2nncn2C)CC1C c1(C(=O)NC(CN(C(c2cc(C(C)C)ccc2F)=O)CC)C)cnc(N)c(N)c1 C=CC(CC)CC(=O)NC1CCN(C(c2ncsc2C)=O)CC1CC N1(c2cc(N(C)CC3CC=CCC3)nc(COC)n2)CCCC2(C1)CC2(F)F CC1COCCC1CN(C=O)Cc1ccc(C(F)(F)F)cc1 C(=O)(C(C(=O)NCC1CCCC1C(=O)NC1(c2ccccc2)CC1)OC)OC N1(C(CCCn2c(C)ncc2)=O)CCN(C(=O)CC2(C(F)(F)F)CC2)C(C)C1C S(=O)(=O)(c1sc(Cl)nc1-c1ccccc1)N(C(C)C)C(C)C CC(C(=O)NC(CCF)C(=O)NC(CCO)C1CCCC1)C(F)(F)F N1(C(c2ccc(OC)o2)=O)CC2(CC1CNC(c1occ(C)c1C)=O)CC2(F)F C1(N(C(C2CC3(CC3)C2)=O)CCF)CCCN(C(c2csc(C(F)F)c2)=O)C1 N1(C(=O)Nc2cnc(C)s2)CC2CN(C(=O)CCC(C)(C)NC(C)(C)C)CC2C1 CC#CCCC(=O)N(CCNC(=O)Cc1cc(C)sc1C)Cc1ccccc1 N1(C(CNc2n(C)c(S)nc2)=O)CC2CC(NC(C3CC4COCC4C3)=O)C1C2 Cc1nn(Cc2ccccc2)cc1C(=O)Nc1cnn(C2CC2)c1 C1(C(=O)NC2CC(C(C)(C)C)C2)CCN(C(c2cnc(O)o2)=O)CC1O C1(C(=O)NCC(CC)(C)NC(=O)CCc2ccnc(C)n2)CSCC(=O)N1 C=CC1CN(C(=O)CN(C)CCC)CC1NC(c1ccc(-n2ccnc2)nc1)=O C1(CC=C)(NC(=O)C=CCF)CN(C(=O)C(CC)n2ccc(C3CC3)n2)C1 C1(CNC(C2CC2(Cl)Cl)=O)CCN(C(c2csc3nnsc23)=O)C12CC2 CCC(C(=O)NC1(C(=O)NCC2CC2Cl)CCCC1)n1ccnc1 C(CC(F)F)(C(=O)N(CCCCCO)C)NC(C(C=C)C)=O C12(CNC(C(N)=O)=O)CN(C(c3ccc4cnoc4c3)=O)CC1CCO2 C1(NC(C2C(C)C2)=O)CCN(C(=O)Cc2coc3cc(F)ccc23)CC(C)(C)C1 C1(NC(CCCCN(C)C)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1F C1(C(=O)O)(C(=O)O)CC=CCC1.CC(C=O)OC1CN(C)C1 c1(CCCC(=O)NCC(CN(C)C(C2CC3CCC3C2)=O)O)ccc(Cl)cc1 C1(C(=O)NCC2CCN(CCCC(F)(F)F)C2)C2CCN1CC2 C(C(C(C)C)NC(=O)COCC(=O)NC(=O)C(C)=C(C)C)OC c1(C(=O)NCCOC2CCN(C(C3C(CC(C)C)C3)=O)C2)ccc[n+]([O-])c1 CCCCCCCC(=O)N1CCCCC(NC(=O)CN2CCOCC2)CC1 c1(OCC)ccccc1OCC(=O)NCC1CCN(C(c2nn(C)cc2Cl)=O)C1 C1(NC(=O)CC2OCCCO2)CCCC(NC(c2cc(C(F)(F)F)cs2)=O)C1 c1(C(=O)NC2CCN(C(c3cc(C)ncc3)=O)C(C)C2)c[nH]nc1S(N)(=O)=O c1(C(=O)NCC(C)(C2CC2)NC(C2N(CC)CCC2)=O)cc(N)c(F)cn1 N1(Cc2cn(C(COCC)C(=O)NC)nn2)CCN(C)CC1c1ccccc1 c1(C(N2CCC(CNC(CCCC(=C)C)=O)C2)=O)ccc(N)c(F)c1Br c1(C(=O)NCCC(CNC(COCCCC#C)=O)O)cnn2cccc(Cl)c12 C(=O)(C(O)CCN(C)C)NC(CC)CN(C(=O)CCc1ccncc1)C C1(O)(c2cn(CCC(C)C)nn2)CCN(C(C2COC(C)(C)CO2)=O)CC1 c1(C(=O)NCC2CN(C(C(C)SC)=O)CC(C)(C)C2)ccc(S(C)(=O)=O)cc1Cl C1(NC(c2cc(OC)ncc2F)=O)COC2(C1)CN(C(c1ccc[nH]1)=O)C2 N1(C(C(CCC#C)O)=O)CC2CCC(C1)N2C(=O)C(CCC)NC(N)=O c1(C(=O)NCC2C(NC(c3c(C)onc3)=O)CCC2)c(C)nc2ccnn2c1C C(=O)(CCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(C(F)F)CCC2)=O)C1)OC Cc1ccc(C(N2CC(N(C)C(C3CC34CCC4)=O)C2)=O)nc1 c1(OC)cccc(NC(=O)C(c2ccc(Cl)nc2)N(C2(C)CC2)C)c1 C1(CC)(NC(c2sccc2OC)=O)CCCN(C(c2ccns2)=O)C1 CCC(CNC(=O)C(C)CSC)(CC)NC(C1OCCOC1C)=O CC1CC(CCNC(c2cc(O)cc(Cl)c2)=O)CCN1C(=O)Cn1cnnn1 N1(C(c2onc(C)n2)C)CCC(NC(C2(C)CCCC2C)=O)C(C)(C)C1 N1(C(C(CC)C(C)C)=O)CCN(C(c2cc(C)n(CCO)n2)=O)CC(O)C1 O=C1COc2cc(C(=O)NC3CCN(C(c4ccc(Cl)nc4O)=O)C3)ncc2N1 C=CCCC(C(=O)NCC(Cl)=CCl)NC(C1CC(C)CC(=O)N1)=O C1(CN(C(C2CCCOCC2)=O)CC)CCN(C(=O)C#CC(=O)N(C)C)CC1 C1(NC(c2nc(COC)oc2)=O)CC2CC1CC2C(N1CCCC(C#N)C1)=O C1(C(=O)NCCN(C(=O)C(c2c(C)noc2C)CC)CCC)CCOC(C)(C)C1 Cc1nn2c(c1C(N1CCC1CNC(=O)CC1(CO)CCCO1)=O)NCCC2 N1(C(C2OCCN(C)C2)=O)CCN(C(=O)COc2ccccc2O)C2COCC12 C(=O)(C(C1CCCC1)NC(=O)C(=O)NC1CC1)NC(c1ccns1)C C12(CC)CN(C(=O)C(O)COc3ccc(OC)cc3)C(CNC(=O)C(C)O)(C1)C2 N1(C(C(C)=C2CCC2)=O)CCCC1(C)CNC(c1ccnc(C(N)=O)c1)=O C(C(C)(C)CC(=O)N1CC(O)(C(F)C(N2CCOC(COC)C2)=O)C1)OC N1(C(CCC#CC)=O)CC2CCCC2(NC(c2cc(OC)ns2)=O)C1 C1(NC(c2c(C)ccs2)=O)CC(O)CN(C(=O)CC2CCC2)C1 C(C1=CCCOC1)NC(C1CCC(NC(C(C)(C)n2cnnn2)=O)C1)=O c1(CC)ccoc1C(=O)NC(c1cn(C)nn1)C(=O)NCCC1(C)CCCO1 c1(CC)cc(C(=O)NC(C(=O)NCCc2nccc(C)n2)C2(O)CCC2)c(C)o1 c1(CC(=O)N(CCOCCNC(C2(CN(C)C)CC2)=O)C)ccc[nH]1 N1(C(CCC)=O)CC(NC(=O)C(C)NC(=O)Cc2ccccc2)CC(C)(C)C1 CC1C(C)N(C(=O)CN(C)S(=O)(=O)N(C)C)CCN1C(C1CC(O)C1)=O CCC(C)(C)C(C)CC(=O)N(CCCNC(=O)C(Cl)=CCl)C1CC1 c1(CC(=O)NCCCCNC(c2cn(C)nc2Cl)=O)coc2cc(O)ccc12 CC1CCCC(C(N2CC(CCNC(C3(CO)CCCCC3)=O)C2)=O)C1 N1(C(C2C(CC)OCC2)=O)CCC2(CCCN2c2ncc(F)cn2)C1 c1(OC)ccc(C(=O)O)c(C(F)(F)F)c1.c12ccc(cc1)CC(=O)N1CCC2C1 N1(C(C(C2CCC2)OCC)=O)CCC(C(C)(C)NC(=O)C(C)n2ccnc2)CC1 c1(OC(C)C)cc(C(N2CCC(CNC(C3CCC(C)S3)=O)CC2)=O)ccn1 CC(C)(C(F)(F)F)OCC(=O)NCC1CC1NC(=O)CCc1cccc(Cl)c1 c1(C(=O)NCC(C)(C2CC2)NC(C(C)CC(N)=O)=O)cc(Br)c2[nH]nnc2c1 CC(C)CC(CC(C)C)C(=O)N(C1C2CN(C(=O)C(C)N3CCC3)CC12)C N1(C(C2(CC)CCOC2)=O)CCCCCC1CNC(c1cc(C)cc(Cl)c1)=O Cc1cc(C(=O)NCC2CCN2C(=O)C=CCOc2ccccc2)cnc1O C1(CNC(C2(CC(C)C)COC2)=O)(NC(C2CCCCO2)=O)CCCCCC1 C1(C(=O)NCCc2cc(C)n(C)n2)CCN(C(c2cncc(Cl)c2)=O)CC1O c1(C(N2CCC(NC(Cc3c(C)ccc(Br)c3)=O)C2)=O)cc2cccc(C)c2[nH]1 c1(CC)cncc(C(=O)NC(CNC(c2cnn(C)c2)=O)(CC)CC)c1 Cc1ncc(S(N)(=O)=O)cc1C(=O)NC1C=CCN(C(=O)COC2CCOC2)C1 Cc1cccc(C)c1C(=O)NC1CN(C)CC1C.n12cc(nn1)C(=O)NOCC2 C1(C(N)=O)CCN(C(=O)CC2CC(NC(=O)CCCc3ccc(O)cc3)C2)CC1 C=CC(C(F)(F)F)NC(C1CC(O)CN1C(=O)CCC1CCCCO1)=O N1(C(C=CC(CC)=CC)=O)CCN(C(c2cc(C)n(C)n2)=O)CC1CC(F)F c1(OC)cc(C)cc(C(=O)NCC(C)CNC(c2ccnc(C(C)C)n2)=O)c1N Cc1cc(O)ccc1C(=O)NCC1CCN1C(=O)C(F)n1cccn1 c1(C(N2CC(CNC(C(C(=O)OC)C)=O)C2)=O)csc2ccc(F)cc12 c1(C(=O)OC)nn(C)c2ncc(S(=O)(=O)NC(CCCCCO)C(=O)O)cc12 c1(C(=O)NCC(CNC(C(C=C)O)=O)F)sc2cccc(F)c2c1COCC c1(C(N2CC(C)CC(NC(c3c(OC)cccc3)=O)C2)=O)ccc2c[nH]nc2c1 c1(Oc2c(Cl)ccc(C)c2)ccc(C#N)cc1Cl C(=O)(C1CCCn2ncnc21)NCC1CN(C(CCCSC)=O)CC1C(F)(F)F Cc1ccn(C)c(=NC(=O)N2CCC(C3CCCO3)CC2)n1 CC#CCC(C(=O)NC1CC2CC1CC2COC)NC(=O)CN(C)C(C)=O N1(C(c2c(CCC)n(C)nc2)=O)CCCC(NC(c2occc2C)=O)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)NCC(CC)NC(c1cccc(Cl)c1C)=O N1(C(c2cc(C)cc(C)c2N)=O)CCN(C(=O)CC(=O)NC2CC2)CC2(CC2)C1 C1(CNc2cccc(NC(C)(C)C)c2C)CC2C=CC1N(CC)C2.C(=O)(OO)SC C1(NC(COC(CC)C)=O)CCCCCC1NC(c1nc[nH]c1C(C)(C)C)=O c1(C(=O)NC(CC)(CNC(=O)CCCC2CCCC2)CC)ccc2ccnn2c1 c1(N(C(N(CCC)CCc2nc[nH]n2)=O)C)ccc(C)cc1Cl N1(C(C2(C(=O)OCC)CC2(F)F)=O)CCC(N(C)C(c2cc(Cl)ccn2)=O)CC1 C1(NC(C(COCC)NC(c2n(C=C)nnc2)=O)=O)CCn2cnnc2C1 C(C(=O)NCCOC1CN(C(=O)C(c2ccccc2)O)C1)(C(C)C)NC(=O)OC CC1CN(C(=O)CC23CCC(CC2)OC3)CC(C)N(C(=O)CC(O)C(C)(C)C)C1 N1(C(C(F)OC)=O)CCC2(CCOC2)C(CNC(=O)COc2ccc(F)nc2)C1 C(C(=O)N=c1cc2n([nH]1)CCCC2)C1CCN(Cc2n(C)cc([N+](=O)[O-])c2)C1 c1(C(N2CCC(NC(C(C)=C3CC3)=O)C2C(C)(C)C)=O)ccc(C)c(C)c1N C#Cc1cn(C)nc1C(=O)N(CC(C)O)CCNC(=O)C=CC1CCCC1 CC1(O)CCN(CC(N2CC=CC(NC(=O)CCN3CCCS3(=O)=O)C2)=O)C1 N1(C(C(C)Oc2ccccc2)=O)CC(CN(C(=O)Cn2nccn2)CC)C(F)(F)C1 CCN(Cc1nccs1)N1CCN(c2cc(Cl)ccn2)CC1 C1(CNC(C(C)(C)OCC)=O)CCC2CN(C(c3cc(C)ns3)=O)CC12 c1(-c2nc(C)on2)ccn2ccccc12.c12ccc(n1C)C1CCCN1C2=O.c1(CC)ccccc1 C1(CNC(C(CCCC)C)=O)CCN(C(=O)CSCC(N)=O)CCC1(F)F C1(C(=O)NC(C2(O)CCN(C(=O)CN3CCOCC3=O)C2)C)CC2(C1)CC2F c1(NC(C(COC)N(C)C)=O)cc(C)ccc1F CC(C)C(CO)ONC(=O)C=CCC1CC1.C1(C)(N(C)C=O)CC1C c1(C(=O)OCC)c(NCC(c2ccc(F)cc2)N)oc2c1COCC2 C1(C(C)(C)F)CCN(C(c2cc(Br)sc2Cl)=O)CC1 N1(C(CCN(C(=O)Cc2nnc(C)o2)CC=C)=O)CCN(C)CC1C C1(C(=O)NCC(CC)(CC)NC(=O)CC2SC(=N)NC2=O)CC(C)(C)CN1C CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1ccccc1C(F)(F)F)=O Cc1cc(CNC(=O)CC2CCSCC2)oc1C S(=O)(=O)(CC(=O)NCCC(C)CCO)N.C(CC(=O)N)NS(C)(=O)=O C1(C(=O)NCC2CC(NC(C=CC(C)C)=O)CC2O)Cc2c(F)cccc2O1 Cc1nc(CC(=O)NCC#CCNC(=O)CSC(F)F)c(C)s1 N1(C(C=C(C)Cl)=O)CCCC2CN(C(C3COc4ccccc4C3)=O)CC12 C(CC(=O)N1CC2(CC(N(C)C)C2)C1)(C(F)F)NC(C(CC#C)O)=O C1(CS(C)(=O)=O)(CN(CC(=O)O)C(=O)Cn2cc(CN(C)C)nn2)CC(F)(F)C1 C1(C(=O)NC2CN(C(c3nc(Cl)c(Cl)s3)=O)CC2O)CC2COCC2C1 c12cccc(n1)C(=O)N2.N1(C(C2CCC(C(=O)OC)C2)=O)CCCC(F)C1 Cn1nnc(=NS(=O)(=O)c2cccc(NC(=O)C3CCCn4cnnc43)c2)[nH]1 Cc1ncc(Cl)cc1C(=O)OCC1CCCCC1(C)C C1(C(C)=O)CC(C)CN(C(c2cnc(Cl)c(F)c2)=O)C1.c12n[nH]cc1NC2=O C12CCC(C=CC(=O)N1)C2.c1(C2C(N(C)C)CCC2)ccc(C(F)(F)F)cc1 C1(C(C)NC(=O)CC2CC(=O)C2)CCN(C(C2(CF)CC2)=O)C1 C1(NC(C=CCNC(CSC(C)(C)C)=O)=O)CCNC(=O)CC1 C1(CC(=O)NCC2N(C(C(c3ccccc3)OC)=O)CC2)CCCNC(=O)C1 c1(C(N(CCCn2cc(CN(C)CC)nn2)C)=O)cnc2scnc2c1 C1(OC)(CNC(=O)C(CO)N(C)C)CCN(C(=O)C(c2cncn2C)O)C1 C1(NC(Cc2c(C)noc2)=O)CCCN(C(=O)Cn2cnnc2)CC1 C#Cc1ccccc1CNC(=O)C(C)N(C(C1CN2CCN1CC2)=O)C1CC1 C1(NC(CCCC#C)=O)CN(C(C2CCCC(C)(C)O2)=O)CC2(CCOCC2)C1 CC(C)C(C(C)NC(c1coc(Cl)n1)=O)NC(c1cn(CCC2CC2)nn1)=O C1(C(=O)NCC2(CN(C(C(CC)OC3CCCC3)=O)C)CC2)CCCC12CC2 c1(N2CC3C(C(=O)NCC(C(C)C)(F)F)C3C2)ncc2ccccc2c1N N1(C(CCSCC)=O)CCCC(O)(CNC(C2CC2C)=O)C1 CCCC(C(=O)N1CCC(NC(c2nc(O)sc2C)=O)C1)NC(C)=O N1(C(c2c(C)nco2)=O)CC(NC(c2ncnc(O)c2Cl)=O)CC(C)(C)C1 c1(C(N(C2CC(NC(C3(F)CC3C)=O)C2)C)=O)nsc2cc(Br)ccc12 c1(Sc2ccccc2)ccc(Cl)cc1CN(CC=C)C1CC1.OC C#Cc1cc(F)c(C(N2CCC(NC(c3ccsc3Cl)=O)C(C)C2)=O)cc1F c1(NC(c2ccccc2)CC)cccc(N(Cc2cnn(C)c2)CC)c1 C12(NC(CCC)=O)COCCC1CN(C(=O)CCc1cn(C)nn1)C2 N1(C(C(=O)NCCOCCCC)=O)CCC(C)(NC(=O)C2=COCC2)C1 c1(OC)ncnc(N2CCCC(CO)(NC(C3CCCC3O)=O)C2)c1OC N1(C(C2C(C=C(C)C)C2(C)C)=O)CCN(C(c2ccsc2C)=O)C2(CCC2)C1 N(C(=NCC1CCCN1Cc1cnccn1)NC1CCCC1)C1CCN(CC)C1 C1(NC(C2C(C(C)O)C2)=O)CCC2CC1CN2C(C12CCCC1C2(F)F)=O c1(C(=O)NC2C(C)N(C(c3[nH]nc4ncccc34)=O)CC2)nnn2ccccc12 C#Cc1ccc(Cl)c(C(=O)NCCN(C(=O)C(O)CC(C)(C)C)CCOC)c1 c1(NC(C2CC(NC(CSc3nc(C)[nH]n3)=O)C2)=O)n[nH]c(C)c1F Cc1ncnc2c1CC(C(N1CCN(C(=O)CP(C)(C)=O)C(CCO)C1)=O)CC2 N1(Cc2c(OC)cc(Br)cn2)CCc2c(C(=O)Nc3cccc(C)n3)n[nH]c2C1 C(CCCCCNC(C1(C2CC2)CCCO1)=O)N(C)C(c1cn[nH]c1)=O Cc1ccc(-c2n[nH]cc2C(=O)NCCOCCN(C(=O)CC(C)(C)F)C)cc1 c1(CN2C(CC(=O)Nc3cc(C)c(Br)cc3F)COCC2)ccc(O)c(C#N)c1 c1(CC(=O)NC2C(NC(CC(CCC)O)=O)CC2)cc(F)c(C)cc1F C1(C(N2CCCC(NC(c3nn(C)c(Cl)c3)=O)C2)=O)CCCOC1(C)C CCCC(CCCNC(c1c[nH]nc1CC)=O)NC(C1ON=C(C)C1C)=O Cc1cccc(-c2cn(C3CC(NC(=O)CCCF)C3)nn2)c1N(C)C Cc1cc(F)ncc1NC(=O)CC1CCN(C(=O)CNC(C)C)C1 N1(C(C2N(C(C)C)C(=O)CC2)=O)CC2CCN(C(c3cc(Br)n[nH]3)=O)C2C1 CCCC(CC)C(=O)NC(C)(CNC(C1(CF)CC1)=O)CC(C)C N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)Cn2nc(C)cc2C)C1(C)C N1(C(CC)=O)CCCC(C2CN(C(=O)COc3ccc(C)cc3)C2)C1 C1(C(N2CC(C)(CCC(=O)NCCCCCN=[N+]=[N-])C2)=O)OCC2CCCC12 c1(C(=O)NC2CC(CNC(CC3CCC(=O)C3)=O)C2)ccc2ncsc2c1 c1(C(=O)NCC(C2CCOC2)NC(c2n(CC#C)ccc2)=O)csc(C)c1C c1(C(=O)NC(C)CN(C)C(C2(C)CCSCC2)=O)cc2cccc(F)c2s1 c1(C(N2C(C(C)NC(=O)C=C3CCC3)CCC2)=O)cncc2[nH]ccc12 c1(CNC(C23CC(Nc4cc(OCC)ncn4)(C2)C3)=O)ccc([N+](=O)[O-])c(O)c1 c1(C(N2CC3CC3(CNC(C34CCCC3OCC4)=O)C2)=O)n[nH]c2c1COCC2 C1(CC)CN(C(=O)CC(C)N(C)C)CCN1C(c1ccc(OC(F)F)cc1F)=O N1(C(c2c(C)n(C)cc2)=O)CCOC2(C1)CN(C(c1cccc3c1OCC3)=O)C2 CCCCC(O)CCC(=O)N1CC(NC(=O)C#CC2CCCCO2)C(C)C1 N1(C(CSN(CC)CC)=O)CCC2CN(C(=O)CSc3cccs3)CCC2C1 C(=O)(NNc1cc(CC(N)=O)ccc1Br)C1N(C(=O)OCC(C)(C)C)CCC1 C(C(O)CN(C)N1CCC2(Cc3ccccc3C2)C1)OC(C)C CC[Si]1(CC)CCN(C(=O)NC(c2cccc(C)n2)C)CC1 c1(C(=O)NC2(CC)CN(C(=O)CC(C)(C)O)C2)ccccc1Oc1cccnc1 C1(C(N(CC(=O)Nc2cnn(CCF)c2)C)=O)CCC(=O)CC1 N(C(=NCc1ccnc(OC(C)C)c1)NC1CCC(C(F)(F)F)CC1)C(C=C)C C1(C(=O)NCCC(C)NC(=O)CSc2n[nH]c(=N)s2)CCCCCCC1 C1(NC(CNC(C)=O)=O)CN(C(=O)CC2CC3(COC3)C2)CC1S(C)(=O)=O N1(C(C2=NOC(C)(C)C2)=O)CC(NC(c2cn(C3CC3)nn2)=O)CC12CCCC2 CC(C)(C)C1=NOC(C)(C(=O)NC2CC3CCC2(NC(=O)COC2CCC2)C3)C1 N1(C(c2c(F)ccc(C)c2)=O)CCOCC(C)(CNC(C2C3(CC3)C23CC3)=O)C1 CCC(CC(=O)NCC(CC(=O)NCC1(CC(=O)OC)CC1)OC)C(C)C n1(CC(=O)N(CCNC(CN(CCOC)C)=O)C)ncc(Cl)c1C c1(CC(=O)NC2(CO)CCN(C(=O)CCc3cnn[nH]3)CC2)ccc2c[nH]nc2c1 C1(NC(CCC#C)=O)CCN(C(c2ccc(OC)cc2OC)=O)C12CCC2 CN1CC(C)(C)CC1C(N1CC(CNC(=O)CSc2cccs2)C1)=O N1(C(c2c(OC)ccc(F)c2)=O)CCc2sc(CNC(=O)C(C)(C)OC)nc2C1 C1(NC(c2ccn(CCC)n2)=O)CCC2CN(C(=O)C(C)COC)CCC2C1 CC(C)C(C)N(C)CCN(C)CCN(C)C.C1(=O)C(C)O1 c1(C(=O)NCC2(NC(C3C(OC)C3)=O)CCCC2)[nH]c2ccc(F)cc2c1C n1(C(C)C)ncc(C(N2CCCC2C(C)NC(C2(C(F)(F)F)CCC2)=O)=O)c1N c1(C(=O)NCCCOCCN(C)C(C2CCC3(CCC3)C2)=O)cc(F)cc(Cl)c1 c1(C(N2C(CO)CC(NC(C3(C)COC(=O)C3)=O)C2)=O)cc2ncccn2n1 c1(C(N(C2CCN(C(=O)CCn3ccnn3)C2)CC#C)=O)csc(CCC)n1 C12(NC(CCCOC(C)C)=O)CCN(C(c3cncc(N(C)C)n3)=O)CC1C2 c1(C(=O)NC(C)C(C)NC(c2ccc(F)cn2)=O)cc(N)nc(Br)c1 C1(CCCC)CN(C(C2CC(C3CC3)=NO2)=O)CCN1C(c1sc(C)cc1Cl)=O c1cnc(N2CCNCC2)c(-c2nc(-c3cnc(-c4ccccc4)s3)no2)c1 C(=O)(CCS(N)(=O)=O)N1CCC(C(CNC(C2N(C(=O)OCC)CCC2)=O)F)C1 Cc1[nH]c(=N)[nH]c(=NCCC2CC(C)(C)NC2=O)c1Cl C(CC(=O)N(CCCC(C)C)C)(C(F)(F)F)NC(C(CC)C(C)C)=O C(=O)(C1=CCCOC1)NC1CCN(C(c2c(C(C)C)ncnc2)=O)C1 C1(C(=O)Nc2cccc(CNC(C=C(COC)C)=O)n2)CCC=CCCC1 c1(C(N2CC(NC(=O)C#CC3CC3)CC(C)C2)=O)ncnc2sccc12 CC(C)CC(CNC(c1cn(CC(F)(F)F)nn1)=O)NC(=O)C(F)C(C)C c1(OCC(=O)NC2CCN(C(CC)=O)CC2O)cc(F)c(F)cc1F N1(C(=O)OC(C)(C)C)CCC(CO)(CNC(=O)CC2CC=CCC2)C1 N#CCCCCCC(=O)N1CCC2CN(C(=O)CN3CC4CC4C3)C2C1 c1(C(=O)NC2CCN(C(Cc3scc(CC)n3)=O)C(C)C2)ccc2ccsc2c1 c1(C(N2CC(C(C)NC(C3C(C=C)C3)=O)C2)=O)cc(OC)cc(Br)c1N CC1CCN(C(c2cn(C(C)(C)C)nn2)=O)C1CNC(c1ncoc1C1CC1)=O CC1(C)OCC2CC12C(N1CCOCC(NC(=O)CCCC2CCCC2)C1)=O CC(C)CC(C)C(=O)N1CCCC(CCNC(=O)Cc2ccn(C)n2)C1 c1(C(=O)NC(C2(CNC(C3(C)CCCCC3)=O)CC2)C)ccnc2ccncc12 C(=O)(CC1=CCN(C)CC1)N1C(C)CCN(C(=O)CC2(C)CCOC2)CC1 c1(OC)cc(C(=O)N(CC(C)NC(C2CSCN2C(C)=O)=O)C)ccc1F C1(NC(c2cnc(Cl)[nH]2)=O)CN(C(c2scc3c2CCCC3)=O)C2(CCC2)C1 C(=O)(C(O)CC(N)=O)NCC1(O)CC(CNC(c2cnn(C)c2C(F)(F)F)=O)C1 C(=O)(C1CCc2cccc(F)c21)N1CCN(C(C(CCSC)OC)=O)C2(C1)CC2 c1(CC(C)C)nccc(C(=O)NCC2(C)CCN(C(C3(F)CCOC3C)=O)C2)n1 N1(S(CCOC(=O)CCc2ccc(F)cc2)(=O)=O)CCN(CC)C(C)C1 N1(C(c2n(CC=C)ccc2)=O)CCC2(CCN(C(C3CCCN3C)=O)C2)C1 c1(NC(C2N(C(c3c(C)nc(Cl)s3)=O)CC2)=O)c(Br)cc(Br)c2ccccc12 C(C(C)(C)CC(=O)O)NCCCc1c[nH]c(C)c1CCC(=O)OC.C(C)C c1(C(=O)NCC2(CNC(COCC=C)=O)CC2)ccc(F)c(C(=O)CCC)c1F C1(CNC(c2n(C)ncc2)=O)COC(C)(C)CN1C(=O)Cc1cn(C)nc1Cl C1(C(=O)NC2CC(NC(CC(C=C)(C)O)=O)C2)CCC2C(C1)C2(F)F C1(O)(CNC(=O)CC2CC2)CC(C(=O)NC2CC(N(C)C)C2)C1 c1(C(=O)NC2(CCNC(CC3C(C)C3)=O)CCC2)ncccc1C(F)F N1(C(C2N(C)C(=O)OC2)=O)CCOCC(C(=O)NCC2CCCS2)C1 c1(SC)ccc(NCC(N2CCN(c3ncccn3)CC2)=O)c(Cl)c1 c1(CC(=O)Nc2c(C)nn(CC(=O)OC)c2C)ccc2c(cnn2C)c1 CCC(C)C(C)C(=O)N1CCOCC1CN(C(=O)C(F)CC1CCCC1)C c1(NC(N2C(C(=O)NC3CCN(C(C)=O)C3)CC3CC32)=O)cnccc1C(F)(F)F Cc1cc(C)c(C(N2CC(NC(=O)CC3CCC(F)(F)C3)C(C)C2)=O)c(=O)o1 Cc1nnc2n1C(C(=O)NCCC1CCN(C(C3CCS(=O)(=O)N3)=O)CC1)CC2 c1(C(C(=O)NCCCNC(Cn2c(C(=O)OC)cnc2)=O)CC)cccc(Cl)c1 C(C1CCN(C(=O)COC2CC3CC3C2)CC1)=CC(=O)N(C)C c1(SC(C)C)ccc(C=CC(=O)Nc2cc(C(F)(F)F)ccc2C)cc1 n1(CCOC)nnnc1C(CC1CCOCC1)NC(C1(n2cc(Br)cn2)CC1)C CC1CN(C(c2sccc2Cl)=O)CC1NC(c1ccc(C2CC2)cn1)=O N1(C(c2c(C)cncc2Br)=O)CCC2CN(C(C3CCCCC3O)=O)CC12 c1(CC(CNC(=O)CCSC2CCCC2)NC(=O)CC2C=CCC2)ccccc1 CCC(C)C(C(=O)NCc1cncc(OC)n1)NC(=O)CCC(C)(C)F Cc1cc(F)cnc1C(N1CCCCC1CCC(C)(C)NC(=O)C(C)O)=O C1(n2cc(C3(N4CCCC4)CCOC3)nn2)(C(=O)OC)CN(C(=O)C(C)=O)C1 C1(NC(C2CC(SC)C2)=O)CC(NC(C2(C(C)(F)F)CCC2)=O)CC1O CN1C(=O)C(=O)N(CC(=O)NCC2C=CC(NC(c3ccc(Cl)o3)=O)C2)C1=O C(=O)(CCCCC(N)=O)N1CCC(C)(NC(c2ccc(COC)cc2)=O)C1 c1(CC(=O)NCCCCc2cn(C3C(C)(O)CCC3)nn2)cc(F)c(Cl)cc1F C1(C(N(C)CC2COCCN2C(c2ccnc(S)c2)=O)=O)CCCCC2(CC2)C1 Cc1nc2ccccn2c1CC(=O)NCC1C2CN(C(=O)CN(C)C(N)=O)CC12 C1(C(=O)NCc2occ(C(N(C)CC3NC(=O)NC3=O)=O)c2)CC2C(C1)C2(C)C C1(CC)CC(C(=O)NCc2c[nH]nc2C(=O)Nc2ccc(C(C)C)nc2)CCO1 C(C(O)CNC1C2CCCC12)(OCC)OCC N1(C(c2c(C)ccc(O)c2)=O)CCC2CCN(C(c3cc(C(C)C)no3)=O)C2C1 C1(C(=O)NC(C(N2CCCC(CCF)C2)=O)C2CCOC2)CC2CC1CC2O c1(C(N(CCCNC(=O)C=C2CCSCC2)C(C)C)=O)ccn2nccc2n1 C1(CC(=O)OC)COC(CNC(=O)CC2CSCCO2)C1 c1(CSCC(=O)NCCC(C)NC(c2ccccc2)=O)csc(=N)[nH]1 C(=O)(CC(C)CC(C)C)NC1(CNC(C2CCCN(C(CC)=O)C2)=O)CCCC1 c1(C(=O)NC(CNC(c2ccc[n+]([O-])c2)=O)C2CC2)cccc2c1COCC2 C(CCS(C)(=O)=O)(C(=O)NCC1CCCCN1C(C1(SC)CCC1)=O)OC C=CCCCC(C(=O)NCC12CC(CN1C)C2)NC(=O)Cn1ccc(C)n1 C1(NC(CN(C2CC2)CC)=O)CCC2CN(C(C3CCCS(=O)(=O)C3)=O)CC2C1 CC1CCN(CCC(=O)NC2CC2NC(=O)CC2CC(=O)NC2=O)CC1 C1(C(=O)NCCCCC(N)=O)CCN(C(=O)CC2(O)CCOC2)C12CC2 C(C(=O)NCc1ccc2c(c1)OCO2)(C1=NOCC1)N1C(C)COCC1 N1(Cc2c(C)ncc(Br)c2)CC(NC(C2(CO)CC2)=O)CC2(CCC2)C1 N1(C(C2OCCN(C)C2)=O)CC2(CC2)CC1CNC(=O)CC1CC1 N1(C(C(CC)(F)F)=O)C(CC(=O)NCCS(C)(=O)=O)C2CCCC12 C1(O)(C(=O)NC(C2CN(C(C3CCc4nc[nH]c4C3)=O)C2)C)CCCC(C)(C)C1 O=S(=O)(c1cncc(Br)c1)NCC1C=CC(NC23CC4CC(CC(C4)C2)C3)C1 c1(C(=O)NCC2(C)OCCN(C(C(C(CC)C)C)=O)C2)cccc2sccc12 C1(NC(CSCC(=O)OC)=O)CCC(NC(=O)CC2CCC(C)CC2)CC1 c1(COC)cccnc1C(=O)NCC1(CNC(=O)Cc2scnc2C)CC1(F)F C1(C(=O)NC(CNC(CCOCC#C)=O)COC)CCC2(CC2)C1 N#Cc1cc(C(N2CC(NC(=O)COCC(F)(F)F)C(F)C2)=O)ccc1O N1(C(C(CC#C)C)=O)CCC2(CCCN2C(=O)CC2(COC)CC2)C1 C1(NC(c2ccc(NS(C)(=O)=O)cc2)=O)CCN(C(C2(CO)COC2)=O)CC1O N1(C(c2ccc(C=C)cc2)=O)CCC2(CC(NC(C3CS(=O)(=O)C3)=O)CO2)C1 c1(CN(CC(C)NC(C2(CCOC)CCC2)=O)C)ccc(C(=O)OC)cn1 CC1CCCC(CC(N2CCC(CC(=O)NOCCF)C2)=O)O1 CC(C)CC(C(=O)NCc1cn(C)nn1)NC(c1nnc(O)nc1O)=O C(=O)(C(C)(C)C(C)(F)F)NC1CC(NC(c2nc(C(C)C)sc2)=O)C12CCC2 C1(COC)(NC(=O)CCC2(C)CC2)CCN(C(=O)C#CC2(C)CC2)CC1 N1(S(CC)(=O)=O)CCC(Oc2ccc(NC3CCCC3C3CC3)cc2)CC1 c1(CC(=O)NC(C)CCCNC(c2ccc(F)cc2)=O)ccc(OCF)c(F)c1 N#Cc1ccc(C(=O)NCCC2CCCN(C(=O)Cn3ccc(C4CC4)n3)C2)o1 C(=O)(CCCCCC(C)O)NCC(CN(C(C=CC(CC)C)=O)CC)(C)C C1(NC(C(CC)CC)=O)CC(CNC(=O)CC=CCc2ccccc2)C12CCC2 CC1CC(C(=O)N(CCCn2cc(COCC(N)=O)nn2)C)CO1 c1(C(=O)NCC2(CCNC(C(CSC)C)=O)CC2)ccc2n[nH]cc2n1 c1(C(=O)NC(C)(C)CCNC(C2CCCS2)=O)ccnc(-c2nccs2)n1 C(CC(=O)N1CC2CC1CN2c1nc(C2CC2)nc(=N)[nH]1)(C(F)(F)F)OC N1(C(C2C(C#C)C2)=O)CC(NC(C2(n3cncn3)CC2)=O)CC(F)C1 C1(C(=O)NCC2CC(NC(CCCC#C)=O)C2(C)C)SC2C=CC1CC2 C(CC(C(C)(C)C)NC(=O)CP(C)(C)=O)N(C(=O)CN1CCCCC1)C c1(OC)cc(CCC(N2CCC(C)CC2CNC(=O)C=CS(C)=O)=O)ccc1F c1(CC)c(C(=O)NC2CCOCC2NC(c2[nH]cnc2C)=O)sc2ccccc12 C1(C(N2CC(N(C(CN(C3CC3)CC)=O)C)C2)=O)CCOC1(C)C c1(C(=O)NC(CCCCNC(C(CC)(C)OC)=O)C)ccc(C)c(OC)c1 C1(C(=O)NCC)CCN(c2cc(NCC(F)C3CCC3)ncn2)CC1 n1(CC)ccnc1C(=O)NC12CC(C(=O)Nc3cnsc3)(C1)C2 C1(C(=O)NCC(C)(C)NC(C(CC)=CC)=O)CCC2(CC2)N1C(=O)OC(C)(C)C N(C(=NCc1ccccc1C)N1CCC(F)(C(=O)OC)C1)CC(C)(C)OCC NS(=O)(=O)CCC(=O)N1CCCC1CNC(=O)CC1CC(O)C12CCC2 CCC(C)CC(C(=O)NCCc1ccns1)NC(=O)C(C#N)C(C)C C1(C2(O)CCCOC2)(C(N2C(C)CN(C(c3ccco3)=O)CC2)=O)CC1 c1(CC)cnccc1C(=O)NC(CCF)C(=O)NC1(COC)CC(O)C1 C(=O)(C#CC(C)(C)CNC(c1cccn1C)=O)NCc1cc(OC)nn1C C1(C(C)C)CCC(C)CC1C(=O)NC1CC12CC(NC(C1(F)CCCOC1)=O)C2 c1(C(c2nnnn2C(C)(C)CC)NC(CC)(C)C)nc2ccc(Br)cc2o1 N1(C(c2c(CC)n[nH]c2)=O)CCCC(C(=O)NC2CC(CCC(=O)O)C2)C1 n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N2CCC(SC)C2)c(C)n1 C1(NC(C(CNC(C2(C)CC=CC2)=O)OC)=O)CN(C)C(=O)C12CC2 CCCC#CC(C)(C)NC(C1CCOCC1NC(=O)CC1CC=CC1)=O C1(N(C)C)CCCCC1(c1nnnn1C1CC1)Nc1cncs1 C(=O)(C1=NOCC1)N1CCC(NC(=O)COCCF)C1 C1(C)(CNC(CC2(C=C)CC2)=O)COCCN(C(c2cnc(Cl)n2C)=O)C1 n1(CC)ncc(C(=O)NC2CCCC2NC(c2csc(C(=O)OC)c2)=O)n1 C(=O)(C1Cc2ccccc21)N1C(C)CC(C(N2CC(Cc3ccco3)C2)=O)CC1 CCCC(C(N)=O)NC(=O)CC(CNC(=O)C=CC(C)(C)C)OC Cc1cc(C(=O)NC(CNC(C2CC2(C)C(F)F)=O)C(C)C)cc(C)c1F O=C(C#CC1CCOCC1)N1CCN(C(C2CCCC3(CC3)C2)=O)C(CCO)C1 CC(C)CS(=O)(=O)CC(=O)NC12CCOCC1CN(C(=O)C#CC(C)(C)C)C2 C(=O)(CCCCN(C)C)NCCCOCCN(C(CC(C)C)=O)C C1(NC(c2c(Cl)cnc(C)n2)=O)CN(C(C2CC2CC(C)(C)C)=O)C2(CCOC2)C1 C1(NC(C2CCCC(=O)N2)=O)CCN(C(C23CCC(CC2)CC3)=O)CC1F c1(C(=O)NCC2(F)CCC(NC(C(CCC)(C)C)=O)C2)cnn2ccnc(N)c12 c1(C(N2CC(NC(C(CCC)NC(N)=O)=O)C3(C2)CC3)=O)ccnc2cc[nH]c12 C1(C(=O)NCC(CN(C(C2CCCN2N=O)=O)CC)(C)C)(N(C)C)CCCSC1 C1(C(N(C(CC(C)C)C)C)=O)CCN(C(c2ocnc2C2CC2)=O)C12CCC2 c1(OCC(=O)N(CC=CC#C)CC2CC2)ccc(CO)cc1.C1(C)CC1 C(=O)(NN1CCCOC1=O)NC(=O)COCCc1cn(-c2cccc(F)c2)nn1 C1(CC(=O)NC2CC2)CCC2(CC1)CCN(C(=O)C(F)(F)c1ccncc1)CC2 C(CCCCC(=O)N1CC(NC(=O)CP(C)(C)=O)C1)=CCCC C1(C(=O)NC23CC(C)(C2)C3)CCN(C(=O)CC2OCCC2(C)C)C1(C)C C(=O)(CCS(=O)(=O)N(C)C)N(C)CC1C2CN(C(C(CC#C)C)=O)CC21 c1(NC(N2CC(C(=O)Nc3ccc(N(C)C)cc3)C(O)C2)=O)cc(Cl)ccc1Cl N1(C(c2c(CC)nco2)=O)CCCC(NC(C2CN(C(=O)N(C)C)C2)=O)C1CC N1(C(CCN(C2CCC2)CC#C)=O)CCOC(C(=O)N(CC(=O)NC(C)C)C)C1 CCCC(C)(O)CC(=O)N1CCCC(C)(CNC(C2CN(C)CC(C)O2)=O)C1 C(C(=O)NCC(C)NC(=O)CCc1cn[nH]c1)(C(C)C)NC(C)=O c1(CNC(c2ccccc2)CCc2cn(C)nn2)nc2cnccc2s1 c1(N2CCCC(F)(CO)C2)nc(N2CCC(C)(CO)CC2)c2c(F)cccc2n1 CC(C)C(CO)CCNC(=O)C=CCC1(NC(=O)CCc2nncs2)CCC1 C1(NC(CCc2c(C)cccc2)=O)CCN(C(=O)C(C)(C)n2cccn2)CC1O c1(C(N(C(c2ccccc2)CNC(C(CO)OC)=O)C)=O)cccn2ccnc12 N1(C(C2(C)CC2)=O)CCC2CCN(C(=O)CCC(=O)NC3CC3)CC2C1 C(CC(C)(C)C)(c1ccccc1)NC(c1n(C(C)(C)C)nnn1)c1ccno1 c1(OC)ncc(F)c(=NCc2ccc(C(N3CC4CC4C3)=O)[nH]2)[nH]1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NC1CC1CNC(=O)CC1CCCO1 Cc1ccnc2sc(C(=O)N(C)CC3(CNC(=O)C4=COCC4)CC3)c(C)c12 N1(C(c2c(C)[nH]nc2C(C)C)=O)C2CCCC1CC(NC(c1ccoc1)=O)C2 CCC(C)C(C(=O)NCC1CC(C)(C)CO1)N(C)C(c1n[nH]c2c1COC2)=O c1(SC)c(C(=O)NC2CCOC(c3cccs3)C2)cccc1Cl c1(C(N2CC(O)(CNC(C(CCOC)C)=O)C2)=O)cc(OC)cc(C(F)F)c1 Cc1ccncc1C=CC(N1CCC(F)(CNC(=O)CC2NC(=O)NC2=O)C1)=O C1(CC)(CC)CC(C(N2CCCC2C(C)NC(c2ccn(CC(F)F)n2)=O)=O)C1 C(=O)(C(CN(C)C)C(C)C)N1C(C(=O)NCc2cc(C)sc2C)(CC)CCC1 C(C(C)(O)C(=O)NCCCOCCC(=O)NCCc1ncnn1C)OC N1(C(C(C)C)=O)CC2CC1CC2CNC(C1CC(C(C)C)C1)=O c1(C(N2C(C)C(NC(C3CN(C4CCOC4)C3)=O)CC2)=O)ccc(F)cc1O CC(CC(=O)NC(C1CCCCCC1)CNC(c1nocc1C1CC1)=O)C(F)F C1(CNC(C2(CC#C)CC2)=O)C(C)CCCN1C(c1cc(C)sn1)=O N#Cc1cc(F)c(F)cc1NC(C1CC(F)CN1Cc1sccc1Br)=O CC(C)CC(CNC(C1CC1C)=O)NC(=O)CN1CCS(=O)CC1 Cc1cc(C(=O)NCC(O)CNC(C2CN(C)C(=O)N2)=O)cc2ccoc12 N1(C(C)=O)CC(C)CCC1Nc1cc(OC(F)(F)F)cc(Br)c1 c1(OCC(=O)NCC(CNC(C2(COCC)CC2)=O)F)ccc(OCCF)cc1 C1(C2CC2)(NC(c2csc(C)c2C)=O)CCN(C(=O)C(c2cccc(F)c2)C)C1 C1(COC)(CNC(=O)CCCC2CCC2)CCCN1C(c1ocnc1C1CC1)=O n1(CC(=O)OC)nc(C)c(S(=O)(=O)Nc2csc(Br)c2)c1C c1(OC)cc2ccccc2cc1CN1CCC(O)C(C(N2CCOCC2)=O)C1 c1(Cn2cc(CC(CC)C(=O)O)nn2)ccc2c(c1)CCCS2 c1(CNCC2N(C(CCc3c(C)ncs3)=O)CCOC2)cc2ccccc2[nH]1 c1(NC(Cc2cnn(C)c2Cl)=O)cccc2c1CCCN2C(=O)CSC1CC1 n12nc(cc1C)NC(=O)C2.c1(N2CCC(CC)C2)c(OC)nsc1OC c1(C(N(C2CCC(C(N3CCCC(F)C3)=O)CC2)C)=O)ccc([Si](C)(C)C)cc1 C1(C(N(CC(=O)NCCC2CCC(C)O2)CC)=O)CC2(CSC2)C1 Cn1c(C(N2CCC(C(F)F)(CNC(C3CC(F)C(=O)N3)=O)C2)=O)nnc1S C12(C(N3C(CNC(C4C=CC=CC=C4)=O)COCC3)=O)CC1CCC2(F)F c1(C(N2CC(NC(CC=C)=O)C(O)C2)=O)cc2cn[nH]c2cn1 c1(C(N2CCC(F)(C(=O)Nc3nccc(I)n3)C2)=O)cc(Cl)c2cn[nH]c2c1 c1(C(=O)NC(c2cccnc2O)C)cnc(CNC(=O)C#CC2CC2)nc1 CCCN=C(NCC(C1CCN(C)CC1)(C)C)N1CCN2C(=O)CCC2C1 C1(CNC(CCC=C(C)C)=O)CCN(C(=O)CCc2cn[nH]c2)C1(C)C C1(COC)CC2(CCN2C(=O)C(CN(C)C)NC(c2occ3c2CCC3)=O)C1 c1(NC2C(C)CN(C(c3ccc(Cl)cc3)=O)C2)ncnc2c([N+](=O)[O-])cccc12 n1(CCC(=O)Nc2cc(C(F)F)nc3ncnn23)c(=O)oc2ccccc12 C1(C(N(CCN(C(CSCC(=O)OC)=O)C)C(C)C)=O)CC2C=CC1C2 N1(C(CCCOC(CC)=O)=O)CCN(C(c2cc(OCC)n(C)n2)=O)CC2(CC2)C1 C1(C(N(CC(=O)OCC)C)=O)CN(C(=O)C(O)CCSC)CC(C)(C)C1 c1(OC)cc(CC(=O)NCC2CCCN2C(c2n[nH]c(C)n2)=O)ccc1C Cc1nn(C)c2c(NCc3csc(Br)c3)nc(N3CCc4[nH]c(=N)sc4C3)nc12 N1(C(c2ccc(Cl)o2)=O)CC(CO)C2(C1)CN(C(=O)C1=CC3(CCOC3)C1)C2 c1(C(C)=O)ccc(NNC(=O)NC2CCS(=O)CC2)cc1 C12(C(N(CC(C)C(=O)N3CC(C4CCCOC4)C3)C)=O)CCC(C1)OC2C c1(C(=O)NC2CN(C(C3CCCC3)=O)CC23COC3)cc2ncccc2[nH]1 S(=O)(=O)(c1cc(C)cnc1NC(CO)C1CC1)N(C)Cc1ccc(OC)cc1 N1(C(CC(C)CN(C)C)=O)CCCCC12CN(C(C1CC1C1CCC1)=O)C2 C1(C(C(=O)N(CC(C)CNC(C2(CO)CCC2)=O)C)F)CCCCC1 O=C1Cc2cc(CN3CC(=O)N(Cc4nccn5nccc45)C3=O)ccc2CN1 CC(CC(=O)N1CCC(C)(NC(=O)C(O)C(F)(F)F)CC1)P(C)(C)=O C(c1ccc(Cl)cc1Cl)=CC(=O)NC(C1CN(c2nnnn2C2CC2)C1)C C=C1CC(C(F)(F)F)(C(=O)NCC2CCN2C(=O)CSc2cnn(C)c2)C1 CC1=C(C(=O)NC2(CN(C)C(c3nc(C)nn3C)=O)CC2)CCC(C)(C)C1 C1(CCNC(C(C)NC(CC)=O)=O)CCCCN1C(=O)CCc1ccc(C)s1 Cc1nc2ncc(C(=O)NC3CC3CNC(=O)Cc3nn(C)cc3Cl)c(=O)n2[nH]1 CC(C)(C#N)CCC(=O)NCC1CN(C(C2Cc3cccnc3C2)=O)C1 C1(CC=C)(C(=O)N(CCCOC)C)CN(C(=O)C(CC)=CCCC)C1 CCC(C)(C)CC(=O)N1CCCC1C(=O)NCc1oc(CSC)nc1C N1(C(CCC#C)=O)CCN(C(C2C=CC2C(=O)OC)=O)CC1CC(F)F c1(C(N2C(CCNC(Cc3c(C)nccc3)=O)COCC2)=O)ccc(=O)n(C)n1 C1(CC(=O)NC2CC(C(C)NC(c3cnsn3)=O)C2)CCC2(CC1)CCC2O N1(C(=O)Cc2csc3ccccc23)CCN(C(C2CC=CCC2)=O)C2CCCC12 C1(C(=O)NCCC(CC)CO)C2CCCC2CN1C(=O)C(C(=O)OC)OC Cc1cnc(F)cc1C(=O)NCC1CCCC1NC(c1cn(C)nn1)=O N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CN(C(=O)C(N3CCOCC3)C)CC2C1 C1(CC(=O)NC2(CNC(C3(F)CCC3)=O)CCCC2)CCc2ncc(Br)n2C1 c1(COC)ccnc(C(=O)NCC23CC2CN(C(=O)C=CC2CCC2)C3)c1 C1(OC)CCCC(CC(=O)NC2CCCC2NC(=O)CCCCn2ccnn2)C1 c1(C(=O)NC2CC(CNC(C3CC3CF)=O)C2)nccn2nccc12 c1(C(N2C(CNC(CC(COC)C)=O)CC(C(F)(F)F)C2)=O)ccc(S(N)(=O)=O)s1 c12cc(sc1C)NC2.c1(C(c2nnnn2C)OCC)cn(C)nn1 CCCCS(=O)(=O)CC(=O)NCC1CCN1C(=O)CCCCC#N c1(NCC2CC(NC(c3cc(C)sc3C)=O)C2)ccc(C#N)cc1[N+](=O)[O-] N1(C(C(C2CCCC2)OCC)=O)CCC(NC(c2nc(C)n(C)n2)=O)C1C c1(C(N2CCC(C)(CNC(CC(CC)C3CCC3)=O)C2)=O)cnc(OC)c(C)n1 N1(C(CSC)=O)CCCCC(CNC(c2ccncc2Oc2ccccc2)=O)C1 N1(C(CC2(C)OCCO2)=O)CCCC(C)(NC(=O)C(F)CC2CCOC2)C1 c1(C(N2OCC(n3cc(C(C=C)(C)O)nn3)C2)=O)cc(S(N)(=O)=O)ccc1Br N1(C(c2ccc(CC)cn2)=O)C2CCC1C(NC(=O)Cn1cc(C)cn1)C2 c1(OC)cccc(Br)c1NC(=O)CC1CCN(Cc2cccc(C3CC3)c2)CC1 c1(C(=O)NCCCN(C(=O)C(c2cccnc2)O)C)cc(=O)c(Br)c[nH]1 C(C)(CCC(=O)N(CCCCCNC(c1ccnc(S)c1)=O)C)OC C12(NC(CC3CCCC(OC)C3)=O)CCCC1N(C(C1(C)CC=CCC1)=O)CC2 C1(CC(=O)NCCNS(CC)(=O)=O)CCN(C(C2CN(C(C)C)C2)=O)C1(C)C CC1(CNC(=O)C(C#N)CC2CC2)OCCc2ccccc21 N1(C(CC=C)=O)CC2CCC1CN2Cc1ccc(Br)c(C)n1 C(CC1CCCCC1)(C(=O)NC(C)CCCNC(C1(C)CC=CC1)=O)OC N1(C(CC2(C=C)CC2)=O)CCC(C2CCN(C(=O)C(C)OC)CC2)C1 c1(C(=O)NCCC2CN(C(C(C)NC(C)=O)=O)C2)cccc2cccc(Cl)c12 C1(CC=C)(NC(C2CC(=O)N(C3CC3)C2)=O)CCN(C(c2ccn(C)n2)=O)C1 CC1CCC(NC(c2sc(Cl)cc2Cl)=O)CN1C(c1ccc(F)cn1)=O N1(C(c2nn(CC)c(O)c2)=O)CC2CC(NC(c3cc(C(F)F)on3)=O)C2C1 c1(C2(NC(=O)NCC(C)N(CC)CC)CCC2)cccc(C#N)c1 c1(CNC(=O)CC2OCCCO2)cccc(NC(c2ccc(F)o2)=O)c1 C1(C(=O)NCC2(OC)CC(C)C2)CC12CCN(C(=O)CC1CCSC1)CC2 CC1(C)COCCC1CNC(=O)CC(C(F)F)NC(=O)CC1CCCCCC1 c1(C(N(CCC(C)NC(COC(C)C)=O)C)=O)cnc2c(c1)c(O)nc(=O)n2C Cc1ccc(C(=O)NC2CC(C(=O)Nc3ccc(Cl)c(Cl)c3Cl)C2)c(I)c1C C1(NC(c2cccn2C2CC2)=O)CCCCC1C(=O)NCc1cccnc1O Cc1cc(F)cnc1C(=O)NC1(CCCC(=O)N2CC(CC(N)=O)C2)CCC1 C(=O)(C1CCc2cc(F)ccc21)NCCCN(C(COCCC=C)=O)C1CC1 c1(C(=O)NC2CCCN(C(c3nnc(CC)s3)=O)CC2)c(O)nnc(C)c1C C1(NC(c2cccnn2)=O)CCN(C(C2(CC3CC3)CCCO2)=O)CC1O S(=O)(=O)(c1ccc(Cl)cn1)N1C(CC(=O)NCc2cn(C)nc2)CCC1 Cc1cc2c(C(=O)NCCC3CN(C(=O)CCc4cnn(C)c4)C3)nccn2n1 CCC(CC(=O)NCC1(O)CCN(C(c2cc(N)ccn2)=O)CC1)C(C)(C)C C#Cc1ccc(C(N2CCCC2CN(C(=O)C(O)C=C)C)=O)cc1Cl N1(C(C)C(=O)NC(N)=O)CC2CC1CN2C(C1CC12CCCC2)=O C(=O)(C(CO)NC(=O)C1CC1)N(CC(CC)NC(=O)C(CC)C1CCOCC1)C N(C1c2ccc(OC)cc2CC1(C)C)C(=O)NCCc1ccc(C(=O)OC)s1 c1(C(N2C(C(N3CCC(c4ccccc4)C3)=O)CCC2)=O)ccc(F)cn1 C1(C(N2C(C)(C(=O)NCc3cc(Br)ccn3)CC2)=O)C=CC(=O)N=N1 C1(NC(CSCCC)=O)COC2C(NC(=O)CCc3nc(C)cs3)COC12 N1(C(c2c(C(=O)OC)scc2)=O)CCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C(F)C1 N1(C(c2cnn(C3CC3)c2)=O)CC2(C1)CN(C(C1(CC(F)(F)F)CC1)=O)CC2CO Cc1c(C(=O)NCC(O)CN(C(=O)Cc2cccc(C(N)=O)c2)C)cccc1F c1(C(N(C(C)CCNC(C2(C)CCCOC2)=O)C)=O)c(O)cccc1Cl N1(C(C(C)CN(C(=O)C=CCO)C)=O)CC2C3CCC(C3)C2C1 n1(CC(=O)NC2C(C)N(C(C34COCC3C4(F)F)=O)CC2)ncc(C#N)c1N N1(C(CC=C)=O)CC2(CCC(C(N3CCCCC3CCO)=O)O2)C1 c1(OC)cccc(C(C)=CC(=O)N(CCC(C)NC(=O)CC23CCCC2C3)C)c1 C(=O)(CCCCCC#N)N(CCNC(C1(OC)CC(C)CC(C)C1)=O)C1CC1 CC1CN(C(C2COCCOC2)=O)CC1(C)CNC(=O)CN(C)S(N)(=O)=O c1(CNC(C2CCc3n[nH]cc3C2)=O)cnn2cc(Br)ccc12 c1(OC)ccc(-n2nc(C3CC3)nc2-c2cc(C3CCOCC3)on2)cn1 C=CC1(CC(=O)NC(C)CC(C)(C)O)CN(C(=O)C2CC2)C1 CN1CCC(CCC(=O)NCC(C)(CO)NC(c2ccc(F)s2)=O)C1 c1(CC)cc(CC)[nH]c(=NCCC(C)NC(=O)C(N2CCCCCC2)C)n1 C1(C(=O)NC(C(=O)NC(C)Cn2cccn2)c2cccs2)CCCC1C1CC1 C(=O)(CCCC(F)(F)F)NC1(CF)CCN(C(C(=Cc2ccccc2)OC)=O)C1 CCCCC(CC)CC(=O)NC1CCC1CNC(c1ccc(Cl)c(N)c1Cl)=O C(CC(C(=O)Nc1nccs1)N1CCC(CO)CC1)C1CC(=O)NC1 c1(C(=O)OC)ccc(C=CC(=O)NC(CNC(C23CCCC2C3)=O)C2CC2)cc1 C1(COC)CN(C(C2CC=CC(n3cc(-c4cncnc4O)nn3)C2)=O)CCO1 c1(C(C)NCC(=O)NCC2CCOCC2)n[nH]c(C(C)(C)C)n1 c1(C(=O)Nc2cnc(F)cc2CNCC(O)C(F)(F)F)ccc(O)c([N+](=O)[O-])c1 Cc1coc(C)c1C=CC(=O)NCCC1(C)CCN(C(=O)C(C)C2CC2)C1 c1(C(=O)NCC2N(C(C#CC(C)C)=O)CC(C)CC2)ccc2cnoc2c1 Cc1cc(CC(=O)NCCN(C(C2CCC(C(N)=O)C2)=O)C(C)C)sn1 c1(COC(C2(n3ncc(C)c3)CCCC2)=O)ccc(C(C)C)nc1O O=S(=O)(c1ccnc(C(F)(F)F)c1)NCCOc1ncccc1Br C#CC1(CNC(C2CC2CCNC(C2(CC3CC3)CC2)=O)=O)CC2CCCC12 C#CCC(CC(F)F)C(=O)NCCC(C)(C)NC(=O)CC1CCCCC1 C12(C(N3CCN(C(CCC)=O)CC3CF)=O)CCCCCC1OCC2 c1(C(=O)Nc2scc(-c3c(C)noc3C)n2)cc(F)ccc1O N1(C(c2c(CC)ncs2)=O)CCC2(CCN(C(c3cc(C)c(F)cc3O)=O)C2)C1 c1(C(=O)NCC(C2CCOC2)NC(c2c(C#N)ccs2)=O)ncnc2sccc12 C1(C(=O)NCCCCC(C)NC(=O)C(C)Cc2cnco2)CCc2c[nH]nc2C1 C1(C(N(C)CC2CCN(C(c3c(OC)csc3)=O)C2)=O)Cc2c(C)cccc2O1 C(C(C)(C(=O)NC(c1nc(C)no1)C)NC(=O)CCCc1ccco1)SC Cc1cc(F)ncc1NC(C1(CNC(=O)C(O)Cn2cncn2)CC12CCC2)=O N1(C(CCOCC#C)=O)CCC2CCN(C(c3cnc(OC)c(C)c3)=O)CC12 N1(C(C(N2CCSCC2)C)=O)CCN(C(=O)CCCc2cncs2)C(C2CC2)C1 S(=O)(=O)(c1ccc(I)cc1)NCC1(C(=O)NC2(C#N)CCC2)CC1 c1(C(N2CC3C(NC(C(C)OCC=C)=O)(C3)C2)=O)cnn2c1CC(F)(F)C2 c1(C(=O)NC2C3(NC(C(C)OC)=O)CCC(C2)C3)nc2ccccc2cc1Cl N1(C(C(CC)C)=O)CCC2(CC1)CC2C(=O)Nc1ccnc(C(=O)OC)c1 N1(C(c2cccc(CC)n2)=O)CC=C(CNC(C2CCC=CCCC2)=O)CC1 CCCC(C#N)C(=O)NCC(CC(=O)NC1C2CCC(F)(F)C12)C1CCC1 C1(C(=O)OC(C)(C)C)CCCC(NC=O)C1.C12(C(=O)NC(C(C)O)=O)CC(C1)C2 c1(C(=O)NC(C2(O)CCN(C(=O)C(O)CC3CC3)C2)C)cn(C)c2ncccc12 CC1CCc2nc(S(=O)CCNS(=O)(=O)c3cc(Cl)c(F)cc3F)sc2C1 c1(CNC(c2cc3c[nH]cnc-3n2)=O)cccc2c1CCN(c1ncns1)C2 C(C(C)CC(=O)N=c1cc(C2CC2)n(C)[nH]1)NC(C(CCC(C)C)O)=O C1(CNC(CCCC(=C)C)=O)CN(C(c2cccn2C(C)C)=O)CCC12CCC2 N1(C(CCCN(C(=O)CC2CCCC(=O)C2)C)=O)CCC2(CC1)N=N2 c1(C(N(CCCN(C(C(C)OCCC#C)=O)C)C)=O)cc(C(C)(F)F)ccn1 CC(CC(=O)NCC(C)CNC(C1(C)CC1(C)C)=O)N1CCCC1=O C1(NC(CC(C)NC(N)=O)=O)CC(CNC(c2cncnc2)=O)C(O)C1 C1(C(N2CCC(NC(C(C)(C)OC(C)C)=O)C(O)C2)=O)CCC2(CCC2)CC1 C1(CC)(NC(=O)CC2(N(C(=O)CCc3cccnc3)C)CC2)CCNC1=O CC1(C)CCCCC1CC(=O)NCC(C)(C)NC(=O)CC1CCCNC(=O)C1 CC(C(=O)NCC1CCC(NC(C2COC(=O)N2)=O)CC1)C1=CCCC1 C12(C(=O)NCCOCCCNC(c3n[nH]c4c3CCC4)=O)OCCCC1C2(F)F C1(C)(C(=O)NCCCn2c(C)nnc2)C=CCN1C(=O)CCC1CCCO1 c1(C(=O)NCCCC2(NC(C3C(C=C)C3)=O)CC2)cc(O)nc(C2CC2)n1 C1(C(N2CCC(N(C)CC)C2)=O)CCC2CCC1N2C(=O)CCN1CCCCC1 c1(C(C(N)=O)NC(N(C)CC2CC2c2cn[nH]c2)=O)ccc(Br)cc1 c1(C(C)C)nnc(N2CC(C(C)CN(C)C(=O)OC(C)(C)C)C2)o1 CC1(C)CCCC(C(=O)NCC2CCN2C(=O)CCC2CCOC2)CC1 c1(OC(C(=O)NCC2C3CN(C(=O)CC4CCC4)CC32)F)ccc(Cl)c(F)c1 c1(C(=O)NC(C(C)C)CNC(=O)Cc2cnccn2)ccc(N)c2ccncc12 N1(C(C(C)(C)OC(C)C)=O)CCCC2(C1)CN(C(=O)CCn1ccnc1)CCO2 c1(C(=O)NCCN(C(=O)C(C)NC(c2ccco2)=O)CC)cncnc1.C1CC1 CCC(CC)(CC)C(=O)N1CC2CC1C2NC(C1OCCC1C)=O CCC(CC(=O)C1C(C(=O)NCCC2(CO)CCCCC2)CC1(C)C(C)(C)C)SC.OCC N1(C(CCc2n(C)c(S)nn2)=O)CCC2(NC(c3cscc3Cl)=O)CC2C1 N1(C(C2(CC)CCCO2)=O)CC(CCNC(c2cnc(O)n2C)=O)C(C)C1 c1(C(N2CC(CNC(C(C)(Cl)Cl)=O)OCC2)=O)cc(S(=O)(=O)NC2CC2)c[nH]1 C(CF)(C(=O)NC1CC(CNC2CN(C(C3(Cc4ccncn4)CC3)=O)C2)C1)OC c1(CC(N2C(CNC(CCCSC)=O)C(C)CCC2)=O)c[nH]c2cc(Cl)ccc12 C1(N(c2n(C(C)C3CC3)ncc2)C(=O)C2CC2)CCC2CCC12 N1(C(C2(C#C)CCCC2)=O)CC(C)OC2(CCN(C(=O)COC(F)(F)F)C2)C1 C1(NC(C(=C)Cc2ccccc2)=O)COCCN(C(=O)CSC)C1 C1(C(C)NC(c2cscc2C(F)F)=O)CN(C(=O)CC2(N3CCCC3)CC2)CCO1 c1(C(N2CCC(C(C)NC(Cc3ccc(SC)cc3)=O)C2)=O)cn2ccnc2s1 c1(C(=O)Nc2nc(Br)cs2)cccc2c1CN(Cc1ccn3ccnc3c1)CC2 c1(C(N(CC(C)N(C(C(CCC)C)=O)C)C)=O)ccc2cc(C)ccc2n1 NC1CCOCC1C(=O)NCC(F)(F)CN1CCCC1 c1(CNC(c2cc(C)on2)=O)csc([N+](=O)[O-])c1.C12(CCOCC1)C(=O)N2 C(=O)(C(C)CC(F)F)N1CC(CC(C)NC(C2CCC(CCCCC)CC2)=O)C1 C1(NC(C(N(C)C)C2CC2)=O)CN(C(c2cc(F)c(F)c(F)c2)=O)CC2(CC2)C1 C1(C(=O)NC2(CNC(c3nc(C4CC4)cs3)=O)CC2)CC2C=CC1C2 N1(C(c2nc(NC(C)=O)sc2)=O)CCN(C(=O)C2=CCCS2)CC1C c1(OC)cccc(C2=NOC(C(=O)OCc3cnsc3)C2)c1 O=CN1CCCC1C(=O)NCC12CC(CNC(=O)Cc3ccnnc3O)(CO1)C2 N1(C(C2CCN(C)C2)=O)CC2(CNC(c3cccc4nncn34)=O)CCC1CC2 N1(C(=O)CC2CCCCO2)CCC2CCN(C(c3nccc4occc34)=O)C2C1 N1(C(Cc2n[nH]c(=N)s2)=O)CCOC2(CCN(C(C3CCCC(F)C3)=O)C2)C1 N1(C(CCCCC=C)=O)CC(C(N2CCOC(C(C)(C)C)C2)=O)C2(CCC2)C1 C12(C(N3CCC(NC(C(C)(C)C)=O)C(CO)C3)=O)CC(C)(C1)OC2(C)C C1(C)(CC)CC(NC(c2c(F)cccc2F)=O)CN1C(c1cncnc1C)=O C(=O)(C(O)C(F)(F)F)N1CC(CC)C1.c12n[nH]cc1C(CN(C)CC1CC1)NC2=O c1(CC(=O)NC(c2cnn(C)c2)C(=O)N(C(C=C)C2CC2)C)csnc1C C[Si](C)(C)C1(C(N2CCCC2C2CCCCC2O)=O)COC1 c1(C2(NC(C(c3ccccn3)OCC)C)CC2)ccccc1F c1(C(N2CC3N(C(COCCC)=O)C(CC3)C2)=O)cc(C)nc(O)c1[N+](=O)[O-] N1(C(COCCC#C)=O)CC2CC(C1)N(C(c1sc(C(C)(C)C)nc1C)=O)C2 c1(NC)cnc(F)cc1C(N1CCOC(CNC(c2csc(C3CC3)n2)=O)C1)=O N1(C(c2cccc(COC)n2)=O)CCC(NC(C2CC(OC)C2)=O)C12CCC2 NC1C=CC(NCC2CCCC2OCc2ccccc2)C1 c1(-c2onc(CC(N3CCN(C(CC)(C)C)CC3)=O)n2)coc2cc(O)ccc12 C1(C(=O)NCCC(=C)CO)CC(C)(C)CN1C(=O)CC(C)(C)O CON(CCC(=O)NOCc1nc[nH]n1)C(=O)C(C)CC(F)(F)F c1(CC(=O)NC23C(n4cc(C(C)(C)C)nn4)CC(CC2)C3)ccc(C#N)c(Cl)c1 N1(C(CC2(OC)CCC2)=O)CCC=C(C(=O)NOCC(C)(C)C)C1 N1(C(=O)NCCCCN(CCCCC)C)CCCC1C(=O)NCC.C(C)(C)(C)O N1(C(CC2(C)CCCC2)=O)CCC(O)(CNC(c2coc(C3CCC3)n2)=O)C1 N(C1CC(C)(C)Oc2ccc(F)cc21)C(c1c(OC)cns1)=O CC(O)CCCCCC(=O)NC1CC12CC(NC(=O)CCC=CBr)C2 N1(C(C(c2n(C)ccc2)=O)=O)CC=C(C(=O)NC2CCC(C)(C)C2)CC1 C1(CC(=O)NC2C(C)=C2)CCCC(NC(=O)CCCOC(C)(C)C)C1 N1(C(C2CC(C)(C)C2C(F)(F)F)=O)CCC(CO)(NC(c2ccnnc2)=O)CC1 C(C)(CO)(C(=O)NCC(C(=O)NCC(=O)NOC)N(C)C)OC C(C(CC1CC1)C(=O)Nc1cnccc1CO)NC(C(C)OCOC)=O C(N=c1[nH]c(N(CC(C)(C)CO)C)nc2c1CCC2)C1C(CCC)CCC1 N1(C(c2cc(OC)c(Cl)cc2)=O)CCC(C)C(NC(c2cccnc2)=O)C1C c1(N2CCC(CNC(C)=O)C2)cc(N2CCC(C(F)F)CC2)ncn1 c1(C(N2C(C(=O)NC(CC=C)CO)CC3CC32)=O)c[nH]c2nccc-2c1 N1(C(C(C)=CCC)=O)CCC2(CC1)CC2C(N1CCOCC1c1ccccc1)=O c1(CC)cnc(NC(C2CC(n3cc(CCN(C)C)nn3)C2)=O)s1 C1(NC(c2cc(C)no2)=O)CCN(C(=O)Cn2ccc(=O)n(C)c2=O)CC1(C)C c1(C(N(C(C)CCNC(C2CCC(C)O2)=O)C)=O)cccn(C2CCC2)c1=O CC1C(c2ccccc2)CCN1Cc1cn(C2(C)CCC(C)C2)nn1 N1(C(C2N(CC)CCC2)=O)CCCC(CC)C1C(=O)NCCCSC c1(-c2cn(C)c(=O)cc2)nc(C(=O)Nc2cccc(C#N)c2Cl)n2ccccc12 N1(C(C=Cc2n(C)ncc2)=O)CCN(C(=O)CCc2cncs2)C(CO)C1 N1(C(CC2C(C)=NNC2=O)=O)CC2(C(=O)NCc3cnn[nH]3)CC1CCO2 CCC(CCCO)N=c1[nH]c(=NC2CCOc3c(OC)cccc32)c2ncccc2[nH]1 C1(NC(C2(CC)CCNC2=O)=O)CC=C(C(=O)NC2(CF)CC2)C1 N1(C(c2cccc(-c3cn[nH]c3)c2)C(=O)NCC(=C)C)CCC(O)C(F)(F)CC1 C(=O)(C1=NOC(C)C1C)NC1C(SC)CN(C(C2CCCOC2)=O)C1 c1(NC(c2ccccc2F)CNC(C(C(C)C)NC(C)=O)=O)ncccc1C#N n1(CC(=O)NCC(CNC(CC2C(CC)C2)=O)OC)cc(Cl)c(C)n1 c1(Cc2cc(C(N3CCCC(C(=O)OCC)C3)=O)no2)cc(Cl)ccc1[N+](=O)[O-] c1(CC(=O)NC2CN(C(C(c3ccc(C)cc3)=O)=O)C(C)C2)cc(O)nc(O)n1 C(CC(C(=O)NCC1CCCO1)NC(=O)CCOCC(C)(C)C)=CC C(C(O)CC(=O)NCC12CCC(CC1)O2)NC(CN(CC(C)(C)C)C)=O C1(C(=O)NCC(C)CNC(=O)CCn2cncn2)CC2OC1C1CC21 C#CC1(C(=O)NCC(c2ccccc2)C)CCN(C(=O)C(O)c2ccsc2)C1 N#Cc1ccc(O)c(NC(=O)C(Cn2ccnn2)NC(c2c[nH][nH]c2=N)=O)c1 c1(OC)ccc2[nH]cc(C(=O)NC3CCOCC3NC(C3CSC3)=O)c2c1 C1(C)(CC)CCC(CNC(=O)C(C)(CO)NC(c2csnc2OC)=O)O1 c1(C(N2CCCC(C(C3CC3)NC(CN3CCC(C)C3)=O)C2)=O)ccnc2[nH]cnc12 N=c1nc(Cl)cc(C(N2CCCC(CNC(=O)CCN3CCCCC3)CC2)=O)[nH]1 Cc1nn(C)c2sc(C(=O)NC34CCCC3CN(C(=O)C=C3CCC3)C4)cc12 CCC(CC)C(C)C(=O)NCC1(F)CCCN(C(c2sc(C)cc2C)=O)C1 c1(C(C(=O)O)N(C(CC#C)C)C2CC2)cccc(N2CCCC2=O)c1 C(=O)(C1=CCCO1)N1C(CN(C(CCSCC)=O)C2CC2)CCC1 CC1CCC2(CC1)CCN2CC(=O)NCc1ccc(F)c(Cl)c1F C1(C2CCC2)(C(N(C(C)CN(C(=O)CC(C)n2cccc2)C)C)=O)CC1 N1(C(C=CC(C)(C)SC)=O)CCCCC1C1CCN(C(c2ccc(Cl)s2)=O)C1 C1(OC)CN(C(c2ncc(F)cn2)=O)CC1NC(=O)C(c1ccc(Cl)s1)=O c1(N(C2CCN(C(c3nc(O)n[nH]3)=O)C2=O)C)cccc(N)c1F N1(C(C2C(C=C)C2)=O)CC2CC2(CNC(C2(C3CCCO3)CCCC2)=O)C1 Clc1cscc1CNC(c1ccnn1CCF)c1nnnn1C1CCC1 c1(CC)ccc(O)c(CNC(C2CC2NCc2csc(Br)c2)=O)c1 Cc1cc(C(N2CC(C3(NC(=O)Cc4nccn4C)CC3)C2)=O)c(C)n1C(C)C Cc1cc(=NC(=O)CN(C(C)(C)C)C(c2cccc(F)c2C)=O)[nH]o1 c1(C(CNC(=O)NC2CCC(N(C)C)CC2)(F)F)c(F)cccc1F N1(C(COCCC(C)C)=O)CCC2(NC(=O)CCCn3c(O)nnc3O)CC2C1 C(=O)(C(C)(C)CC(F)F)NCC1C(NC(CCOCC#C)=O)CCCC1 c1(C(=O)NCC2(C)OCCN(C(C=NOC)=O)C2)cccc2c1CCS2(=O)=O C1(CCNC(=O)CCc2ccc(C)o2)(OC)CN(C(c2ccoc2)=O)C1 CCS(=O)(=O)CC(=O)N1CCC(n2cc(-c3ccccc3O)nn2)C1 C1(CC)CCCN(C(c2cc(C3CC3)n(C)n2)C(=O)NCC2CCCO2)C1 C1(NC(C(c2ccoc2)NC(C(C)CO)=O)=O)CCCC(C2CC2)C1 c1(C(N2C(CCNC(c3c(C)cnnc3)=O)COCC2)=O)ccc(Br)c(F)c1 C1(C(N(C2CCN(C)C2C)C2C(CC)C2)=O)COCCN1C(=O)Cc1cocn1 c1(NC(C2C3CN(C(C(CCC)CCC)=O)C2C3)=O)ccc2c(c1)OCCO2 c1(C(=O)OCC)c[nH]ccc1=NCCC1CCN(C(c2conc2C2CC2)=O)C1 N#Cc1cc(C(N2CCCC(CS(c3ccccc3)(=O)=O)C2)=O)sc1Br C1(C(N2C(CNC(CCNC(N)=O)=O)CC2)=O)CCNC(=O)C1 c1(C(C(C)NC(=O)NCc2c(I)ccnc2F)OC)cc(Cl)cc(Cl)c1 C1(C(=O)NC(C2CCN(C(=O)CC(C)(C)O)C2)C)COC2CCCCC12 CCC(CC)CC(F)C(=O)NC(C)CC(=O)N(C)CC1CCCN(C)C1 c1(NC(C(C=C)N(C)C)=O)ccc(C(N2CC(OCC)C2)=O)cn1 c1(C(=O)NCC2(C)CC(NC(C(CCOC)C)=O)C2)cc([N+](=O)[O-])c(C)s1 C1(CC)(NC(=O)CN2CCCOC2=O)CCCN(C(c2cc(Cl)nnc2O)=O)C1 CC(C(=O)N1CC(CN(C(=O)C(c2ccccc2)O)C)C1)C(C)(C)C C1(NC(c2ccc(Cl)s2)=O)CN(C(=O)Cc2ccc(Br)cn2)CC2CC12 c1(N(C)Cc2cc(F)cc(Cl)c2)nc2ccc(Cl)cc2c(=NCC2CC23CC3)[nH]1 C1(C(F)(F)F)(NC(C2CCN(C(COC)=O)C2)=O)CCCCC1 CC(=O)CCCC(=O)NC1CCCC(CC(=O)Nc2ccccc2F)C1 c1(C(N2CC(OC)(CNC(C3CC4CC3C3CC43)=O)C2)=O)scc2c1OCCO2 C1(NC(C(C2(O)CN(C(C3(C)CCNC3=O)=O)C2)F)=O)C2CCC3C(C2)CC13 CC1CN(C(c2cc(C3CC3)cs2)=O)CCC1N(C)C(c1cn(C)ccc1=O)=O CS(=O)(=O)c1cnn(CCNC(=O)C(=O)NC2CC2(F)F)c1 c1(C(N2CC(NC(C3CCN(C(C)=O)C3)=O)C2)=O)cc(Br)nn1C CCC(CC)CCC(=O)N1CCOCCC1C(=O)NC(C)CC(F)(F)F CC1CCCC=C1C(=O)N1CCC2CN(C(c3ncc(C#N)cc3Cl)=O)CC12 N1(C(C23C(NC(c4c(C)cccc4)=O)C4CC2C3C4)=O)CCOC2(CCC2)CC1 N1(C(C)=O)CCCCC1C(=O)N(C)CC1CN(C(C2CN(C)C2)=O)C1 C1(C(N(CCC)CCNC(=O)C=Cc2ccc(Cl)cc2)=O)Cc2ccncc2C1 C(=O)(C1=C(C#N)CCC1)NC1CCCC(CC(N2CCC(C)C2)=O)C1 CC(C)(CCNC(=O)CC1CCSC1)C(=O)NC1CCN2CCC1C2 C(=O)(CC(C)C(C)C)N1CCC(C)(C(NOCCC(=C)C)=O)C1 C1(C(N2CCCC(NC(CC(CC)CN(C)C)=O)C2=O)=O)CNC(=O)CC1(C)C C(=O)(C1CCc2cccnc21)N1C(C)(CC)CC(NC(=O)COC2CCC2)C1 Cc1nn(C)c(C(N2CC3CC3(NC(=O)CC3CCC(C)(C)C3)C2)=O)c1Br c1(C(N2C(C)(CNC(C34CCCN3CCC4)=O)CCC2)=O)ccc(Cl)c(F)c1 c1(C(=O)NC2(CN(C(CCC(CC)OC)=O)C)CC2)cc2nccnc2cc1F CC1(C)C2CCC(C2)C1C(=O)NCC1(NC(=O)CC2CCCSC2)CCC1 C1(C(N2CCCC(CC3CC3)C2)=O)CCCCN1C(c1ccc(Cl)cc1)=O C1(C(N2CCC(NC(C(N3CCCC(C)C3)=O)=O)CC2)=O)CC2C(C1)C2(F)F c1(NC(N2CC(C(CC)C)C2)=O)ccn2nccc2n1 CC(C)C(F)(F)CC(=O)N1CCC1NC(=O)CNS(=O)(=O)C1CC1 N1(C(=O)NC2CN(C(C)=O)CC23CCC3)CCCc2ccccc2C1 C(C(=O)NCC(c1ccc(F)cc1)C(=O)OC)(C(CC)CC)N(CCC)CCC c1(CNC(CC)C(=O)OC(C)=O)ncccc1C(N1CCCCC1C(N)=O)=O C(=O)(C(C)(C)C(C)(C)C)NCC(CC(F)(F)F)NC(Cc1cc(C)c(F)cc1)=O C(=O)(C1COc2ccccc21)NC1CCCC(NC(C(CSC)(C)C)=O)C1 CCC(CC)(CCC(=O)NC1COCC1NC(C12CCC(OC)C1C2)=O)[N+](=O)[O-] C(=O)(C(CNC(=O)C(C1CCC1)OCC)CC1CCCC1)N(CCCF)CC C(c1ccccc1F)=CC(N1CCC(C)(NC(=O)CCC2CC(F)(F)C2)C1)=O C1(OC(C(=O)NCCC(=C)CNC(=O)C(CO)N(C)C)C)CCCCCC1 c1(C(N2CC(CNC(CC(CC)C)=O)N(C)CC2)=O)ccc2c(C)[nH]nc2c1 C1(NC(C)=O)CCCN(C(=O)CCn2cc(-c3ccc(N(C)CCO)nc3)nn2)C1 c1(NC(C2C(O)CCN2C(c2cc(Br)ccc2F)=O)=O)ccnc(Cl)c1I N1(C(Cc2cnc(C)s2)=O)CCOCC1CC(=O)NC1CN(C2CCC2)C1 Cc1occc1C(N1CCCC1C1CCN(C(=O)CNC(=O)C(F)(F)F)C1)=O c1(C(=O)NC2(CF)CCN(C(C(C)OCC=C)=O)C2)cc(=O)c(Br)c[nH]1 c1(C(N2CCC(CNC(c3c(OC)scc3)=O)C2(C)C)=O)nc2ccccc2[nH]1 c1(C(N2CCCC3CC23)C(=O)NCSc2ccc(F)cc2)nc2ccc(F)cc2s1 N1(C(C=C(C)C)=O)CC(CC(=O)NCC2CC(F)C2)C2(CC2)C1 C1(C(=O)NCC(C)N(C(c2c(Cl)c(C)n(C)n2)=O)C)CC(C(C)(C)C)=NO1 N1(C(Cc2ccc(C)o2)=O)CCN(C(=O)CC2=CCCC2)C2CCCCC12 c1(CNCC2CCN(C(COCC)=O)C2c2cccnc2)scc2c1OCCO2 C#CCCC(C(=O)N1CCC(CN=[N+]=[N-])C1)NC(c1cnc(C)nc1C)=O C(=O)(C1=NOC(CNC(c2cnnc(O)c2)=O)C1)NCCC#CCC C1(CNC(C2C=CCC2)=O)CCCC2(CN(C(=O)CCC3CCC3)C2)O1 CC1CN(C(c2ccc(F)c(Cl)c2)=O)CCN1C(=O)CC1CC1C C=CC1(C(=O)NCCCCC(CO)NC(=O)CCn2ccnc2)CCOCC1 S(=O)(=O)(c1cnn2ccc(=NCC(C)(C)C3CC3)[nH]c12)NC(C1CCCC1)CC c1(C(C)C)conc1CC(=O)NCC(C)N(C(=O)C(F)(F)C1(O)CCC1)C N1(C(Cc2cnc(C)s2)=O)CCC2CN(C(c3cccc(Br)c3F)=O)CC12 C1(NC(c2nc(CC)oc2)=O)CN(C(c2c(Br)cncc2Br)=O)CC12CC2 CC(C)C(O)C(=O)N1CCC(C)(CNC(=O)CCc2cccc(O)n2)C1 C(=O)(N=c1cnc(I)c[nH]1)C1C(O)CCN(C(C2CCCC(C)CC2)=O)C1 Cc1cc(Cl)ccc1OCC(=O)N(CC(C)NC(C1CCC(C)(C)C1)=O)C C(C1CN(C(C2(C#N)CCCO2)=O)CC1C(=O)NC1(C)CCCC1C)=CC Cc1c(C(=O)NCCOC2CCN(C(=O)CCS(N)(=O)=O)CC2)cccc1F C1(NC(=O)CC2C3CN(C(c4coc(C5CC5)n4)=O)CC23)CCN2CCC1C2 N1(C(C2(CC#C)CCCO2)=O)CCC2(CCCN(C(=O)Cc3nccn3C)C2)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC2CC(O)C1C2NC(c1c(OC)csc1)=O c1(CNC(CC2(N(C)C)CCC2)=O)ccc(C(=O)NCC2CSCCO2)cc1 c1(C(=O)NCC2CC(C)N(C(=O)CC34CNC(=O)C(C3)C4)C2)ccc(F)c(O)c1 N1(C(c2c(NCC)cccc2)=O)CCCC(C)(CNC(C2CCC(F)C2)=O)C1 N1(C(C2C(=C)CC2)=O)CCC(CN(C)C(c2cn(CC3(C)COC3)nn2)=O)C1 c1(C(=O)NCC(CNC(c2ccc(C(N)=O)o2)=O)O)cccc2ncnc(O)c12 N1(C(C2CCCN(CCC)C2)=O)CCC2(CCCN2C(=O)C=Cc2cscn2)C1 C12(C(=O)OCC)CCC(NC(c3cc(Cl)cnc3F)=O)(CC1)C2 c1(C(N(C2CC(NC(C(Cc3c(C)cccc3)C)=O)C2)C)=O)ccc(F)c(Cl)c1 C1(C(C)NC(CC2(C=C)CCC2)=O)CCN(C(C2CCCCC2)=O)CC1 O=S(=O)(c1cnc(N2CCOCC(O)C2)c(Cl)c1)NCC1(CCCO)CCCC1 C1(NC(Cc2c(C)nc[nH]2)=O)CCN(C(C2CC2CC(C)(C)C)=O)C1(C)C C1(c2cccs2)(N(C(=O)CC(C)(C)C2CCCC2)CC(=O)OC)CCCCC1 CN1CCC(CNCc2cc(C3CC3)ns2)C1c1ccc(F)cc1 C1(c2ccccc2Cl)(C(=O)NC2C(NC(C3(CCC=C)CC3)=O)C2)CCCCC1 C(c1nc2ccccc2s1)=CC(=O)NCCN(C)C(C1CCC=CCC1)=O C1(NC(C(C)N(C(C=CC(C)C)=O)C2CC2)=O)C2CCCCCC12 C#Cc1cnn(C)c1C(=O)NC(CC(C)C)C(=O)NCC12CCC(CO1)C2 c1(C(=O)NC)ccc(NC2CCNC2Cc2ccccc2)c(F)c1 c1(CC(=O)NCC23CC(CNC(C=CCC)=O)(OC2)C3)cn2cccc(C)c2n1 c1(NCC(CC)(CC)NC(=O)CC2CC=CC2)ncc2ccnc-2[nH]1 C1(NC(CCCOCC=C)=O)COCCN(C(=O)C(c2ccccc2)C2CC2)C1 C(=O)(CC(=O)Nc1cnn(CC2(C(C)(C)C)CCCO2)c1)OC c1(OC)ccc(C(=O)NCC2CCCCN2C(=O)C=CCO)cc1C1CC1 C12(C(N3CC(C=C)C(NC(=O)CCCCC)C3)=O)CCC(OC)(CC1)CC2 CCC(C)CC(=O)N1CCCCC1CCNC(=O)Cn1cnc(C(N)=O)n1 CCCCC(CC(=O)N1CCCC(N(C)C)CC1)NC(=O)CCC(C)OC Cc1cc(C(=O)NCCCN(C(=O)CC(C)(C)C)CC2CCCC2)nn1C C1(CN(c2nccc(N3CCC(CC)(CO)C3)n2)C)CCC2(CCOCC2)CO1 c1(C(=O)NC(c2c(CC)cccc2)CNC(C2C(C)C2C)=O)c(N)cccc1Cl CN1CCN(C(C2CC3(C2)CC(O)C3)=O)CC1C(N1CC(F)(F)C1)=O N1(C(c2cnn(C)c2Cl)=O)CCCCCC(NC(c2n[nH]cc2Cl)=O)C1 c1(OC)cnc(Cl)cc1C(=O)NCC1CCCC(CNC(=O)C2=C(C)CCC2)C1 c1(CN2C(C(N3CCC(O)C(F)C3)=O)CC(F)C2)c(Br)cccc1[N+](=O)[O-] C1(CNC(C(C2CCCCC2)C)=O)CN(C(c2cnc(O)n2C)=O)CC1O C1(CCNC(c2cncc(OC)n2)=O)CCN(C(c2nccnc2N)=O)C(C)C1 C1(C(=O)Nc2ccccc2)CCN(CC(O)COCCC2CCCC2)C1 c1(OC)ccc(Cl)cc1C(=O)NCC(C)(C)CN(C)C(C1CCOC1C)=O C(CC(=O)N(C(CO)C(C)C)C)(C(C)C)NC(C(C)NC(CC)=O)=O Cc1scc(C(=O)NCC(O)CN(C(=O)CN2CCN(CC(F)F)CC2)C)c1N C(CC(C)(C)C(=O)NCC(C)O)NC(c1c(C)cccn1)=O N1(C(C(C)OCCC=C)=O)CCC(CNC(c2coc(Br)n2)=O)(OC)C1 c1(C(=O)NC2CCC(N(C(c3cc(C)sn3)=O)C)C2)c(Cl)ccc(C)c1O C(=O)(C(O)C1=CCCCC1)NCCC(C(=O)NCC(CC)(CC)CO)(C)C c1(OC(C(N2CC(O)(CNC(C=CC)=O)C2)=O)C)ccc(C)cc1C CS(=O)(=O)c1ccc(C(c2nnnn2C2CCC2)NCc2ccnc(Cl)c2)o1 CCN=c1cc(C(=O)NC2(CNC(=O)C(F)(F)c3ccncc3)CCC2)cc[nH]1 c1(C(C)OC(C(C)Sc2ccc(NC(C)=O)cc2)=O)cc(=O)n2c(C)cccc2n1 C1(C2CCN(C3C(=O)N3)C2)COCCC1(C)O.c1(CCCSC)sc(Cl)nc1Cl C1(CNC(C2C(C)(C)COCC2)=O)CCN(C(C2(O)CCCC2)=O)CCC1(F)F C(CCN=C(NCCC(C)(C)C)NC1C(C)(C)C1(C)C)SC N1(C(C(C)SC(C)C)=O)CCOC2(CCN(C(=O)CC3CCC(F)(F)CC3)C2)C1 O=C1CCC2(CCC(NC(=O)CNC(=O)NCc3cccc(O)c3)CC2)N1 c1(SC(C2CCCN(C(C(C(C)(C)C)NC(N)=O)=O)C2)C)ccccc1S(N)(=O)=O N1(C(C(C(C)C)N(C)C)=O)CC2OCC(NC(=O)CCc3cccc(F)c3)C2C1 Cc1ncnc(C)c1CC(N1CCC(OCCNC(=O)C=CC2CCCC2)C1)=O C1(NC(C(CC)OC)=O)CCCC12CCN(C(=O)COc1ccccc1F)CC2 c1(-c2nc(C3C(C)C3)n(Cc3cncc(F)c3)n2)cccc(S(C)(=O)=O)c1 N1(CC)CCCC(ONC(=O)C2CC2C(C)NC(C2CCC(=O)O2)=O)C1 c1(C(=O)NCC(C)NC(C2(CCC)CCNC2=O)=O)ccnc(O)c1F Cc1cc(C(=O)NC(C)CNC(=O)CC2NC(=O)NC2=O)n(-c2ccccn2)n1 C(=O)(CC1=CCN(C(=O)C(C)C(F)F)CC1)NC(CC(C)C)C CC(C)C(CCCC(=O)O)NC(c1ccc(-n2cc(C(C)(C)O)nn2)cc1)=O CC1=C(CNC(C2CN(C(=O)C(C)N3CCCC3)CC(C)O2)=O)COCC1 C1(CNC(=O)CCC2CC2)CC2(CCOCC2)CN1C(=O)CCCC1CC1 c1(-n2c(CCOC)nc(CCN3CCCC(C)C3)n2)ccc(S(C)(=O)=O)cc1C Cc1ccc(C(N2CCC(C)C(CC(=O)NCC(C)N(C)C)C2)=O)cc1C#N Nc1c(CC(N2CCNC(=O)C2c2cccc(Br)c2)=O)cccc1Br n1(CC)ccnc1-c1cn(C(C)C(=O)NC2CC(CC(=O)OC)C2)nn1 c1(CCNC(CC2N(C(C3CN(C(=O)NC)C3)=O)CCC2)=O)nnc(C)n1C c1(CNC(CC(CC)N(C(=O)CCC(C)(C)N(C)C)C)=O)ccc(F)c(O)c1 c1(CC(N2C(CNC(C3CC(C(F)F)(OC)C3)=O)CCC2)=O)ccc(O)c(F)c1 c12cccc(c1)C(=O)N2C.C1(OC)CCCC1NC(C)C N1(C(C2C(C(C)C)C2)=O)CCC(NC(c2cn3c(n2)CCCC3)=O)C12CCC2 C1(CC(=O)NC2C(C(N(C(CC(=O)OC)C)C3CC3)=O)C2)CCCCC1O c1(C(N2CCC(CNC(C=COCC)=O)(CO)C2)=O)cnc2nccn2c1 Cc1cc(F)cc(C(=O)NC2CN(C(c3c(O)cccc3F)=O)CC23CC3)c1C Cc1nc2cc(C(=O)NC(C3CN(C(=O)Cc4cnco4)C3)C)ccc2o1 Cn1nc(-c2ccncc2)cc1CN(C(N1CC(c2ccc(F)cc2)(C)C1)=O)CCl C1(C2CC2)(NC(CC(CC)C2CCC2)=O)CCN(C(=O)COC2CCC2)C1 C1(CNC(C(C2CC(NC(c3cnn(C)c3Cl)=O)C2)F)=O)CC2(CCC2)CO1 C1(CN(C(=O)CCc2ccccn2)C)COCCN1C(c1ncc[nH]1)=O N1(C(c2c(CC)n(C)nc2)=O)CCC(NC(C2(C)CC2Br)=O)C(CO)CC1 N1(C(c2cc(CC)[nH]n2)=O)CC2(C1)CN(C(c1cccc3scnc13)=O)CCO2 Cc1cc(C)c(C(N2CC(CN(C)C(c3cnc(C)o3)=O)C3(CC3)C2)=O)c(C)n1 N1(C(C2C(CC)C2)=O)CC(O)(C(C)NC(=O)Cc2cc(C)no2)C1 C1(CC=C)(NC(=O)CSC(C)C)CCN(C(c2c(C)nn(C(C)C)c2C)=O)CC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CO)NC(C(C(C)(F)F)(C)C)=O C1(C(N2CCC(NC(C3(F)C(C)C3)=O)C2c2ccccc2)=O)CCC2(CC1)CC2 C(=O)(C(C)C(=O)OC)NC1CC(C(=O)NC(CCC=C)C)C1 C1(O)(C(=O)NCC2CC(COC)CN2C(=O)CCSC)CC2CCC1C2 CC1(C)CC=C(C(=O)N2CCCC(CO)(NC(C3CCS3(=O)=O)=O)C2)CC1 Cc1ccc(CC(=O)NCCOCCNC(c2occc2C)=O)c(Br)c1 C(=O)(CCN=c1[nH]ccs1)NC1CCCN(C(C2C(C)C2)=O)CC1 C1(OC)CC(C)CN(C(C2(C)CCN(C(=O)Cc3nocc3C)C2)=O)C1 c1(C(=O)NCC2(NC(C(C)n3cncn3)=O)CCOC2)csc2nccn12 CCCCC(C)CCC(=O)NCC1CCC(NC(c2ccc3n[nH]cc3n2)=O)C1 C1(CC(N2CCC(C)C2c2cn(CCF)nn2)=O)CCC2(CC1)OCCO2 N1(C(CCC)=O)CCCN(C(C2(n3cc(Br)cn3)CC2)C2CC2)CC1 C1(NC(CCC(=O)NCCC)=O)CCN(C(=O)C(OC)OC)CCC1CO C=C(Cl)CC(C(=O)NCC(CC1CC1)CO)NC(=O)CNC(=O)CC C1(C)(C(N2CCC(N(C(CN(C(C)C)C)=O)C)C2)=O)Cc2ccccc2C(=O)O1 c1(CC)c(C(=O)NCC(C)NC(=O)C=CC2C(C)C2(Cl)Cl)[nH]c(C)c1C(N)=O CC1(C)COC(C)(C(=O)NC2CCCN(C(=O)CCCc3ccncc3)C2)CO1 c1(C(=O)NC2(CF)CCN(C(=O)CN3CCCCCC3)C2)cc2c(s1)CCCC2 C1(CNC(CC2ON=C(CC)C2)=O)CC2CCC(C1)N2C(=O)C(C)(C)CC(C)C c1(C(N2CC3C(C(=O)NC)(C3)C2)=O)cc2cc(O)ccc2cc1O N1(C(C(CC=CCC)C)=O)CCC2(C1)CN(C(c1ccc(O)c(F)c1F)=O)C2 CCCC(CC)C(=O)NC1CCC(C)N(C(=O)Cn2ncccc2=O)C1 c1(C(c2n(CCSC)nnn2)Nc2cnc(O)c(Br)c2)cccc2sccc12 C1(F)(CNC(c2cnc(CC)[nH]2)=O)CCC(NC(c2cncc(SC)c2)=O)C1 c1(CNCCOCCN(C(C(C(=O)OCC)F)=O)C)c(C(F)(F)F)cc[nH]c1=N N1(C(c2cnn(-c3cccc(F)c3)c2)CC)CCOCC1c1n[nH]c(C)n1 N1(C(Cc2ccc(OC)cc2)=O)CC2(CNC(=O)C=C3CCCC3)CCC1CC2 c1(C(=O)NC2C(NC(CSCCC)=O)CCOC2)ccc2nncn2c1 CCCCCC(O)CC(=O)N1CCCC1CCNC(c1ncsc1CC)=O Cc1nccc(Cl)c1C(N1CC(Cn2cc(-c3ccnn3C(C)(C)C)nn2)C1)=O c12nc(nc3sccc13)CN2CCCN(C)C.C(CC(C)(C)C)Sc1cocn1 N1(C(CC2C(C)(C)C2)=O)CCC(CCNC(c2csc(F)c2)=O)C1 c1(NC(c2scc(C(=O)Nc3c(I)ccc(C)c3)n2)=O)cc(F)cc([N+](=O)[O-])c1 N(C(=NCCC1=CCCCC1)NCc1ccco1)Cc1nc(C(=O)OCC)on1 CCC(CC(=O)N1CC(C(N2CC(C)(C)CC2C)=O)C(C)(C)C1)C(F)F C1(C(=O)NCC2C(C(=O)NCCc3c(C)ncs3)CCO2)CC12CCOCC2 c1(CNC(C23N(C(c4c(C)nc(CC)o4)=O)CCC2C3)=O)ccc(O)cc1C c1(C(N2CCC(C(C)NC(C3CSC3)=O)C2)=O)ccc(Br)nc1O C(=O)(C1=CCC(NC(c2sc(F)cc2C)=O)C1)NC(C#C)(C)C1CC1 c1(C(N2CCC(N(C(CNS(CCCC)(=O)=O)=O)C)C2)=O)c(C)cccc1F c1(CCCNC2(CNCC3CCC(F)C3)CCC2)cc(O)ccc1Cl c1(C(N(C2CN(C(=O)COC(F)F)CC2F)C)=O)cc(F)cc2nn[nH]c12 C1(CNC(C=CC(C)(C)NC(c2ccc(CC)s2)=O)=O)CCC(C)(C)CC1 N1(C(C2CC(C(=O)OC)C2)=O)CC2CCCCC2C1C.N12CCOC(C1)C2=O c1(CCC(N2CCC(C3N(C(C4(C=C)COC4)=O)CCC3)C2)=O)ccnc(Cl)c1 N1(C(CCC=CC)=O)CCCC(NC(=O)Cc2cc(C)no2)CC1 c1(C(=O)NC2CC3(CN(C(C(CC)C(C)O)=O)C3)C2)cc(C)c(C)c2ncsc12 Cc1c(C(N2CCCC(CN(C(=O)CCN3C(=O)C=CC3=O)C)C2)=O)ncn1C N1(C(c2cc(C#N)no2)=O)CC2(CC2)CC1CNC(=O)CCc1nncs1 C1(C)(C(=O)NCCCN(C(C2CC2(C)C(F)(F)F)=O)CC)CC=CC1 N1(C(CCN(C)CCO)=O)CC2CC(N(C(=O)CCc3ccsc3)C)C1C2 N1(C(C(C(C)(C)C)NC(C)=O)=O)CCC(C)N(C(=O)CC2CCCCCC2)CC1 Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)Nc1cc(Cl)cc(F)c1O C1(NC(c2cnc(OC)nc2)=O)C2CC1N(C(c1cc3n(n1)CCC3)=O)C2C C(CCCCC(=O)N1CCCC(NC(=O)CCP(C)(C)=O)C1C)OCC C12(NC(C3CCN(C)C3)=O)COC(CNC(c3cn(C)nc3C(C)(C)C)=O)(C1)C2 c1(CNC(=O)NC(COC)C)ncccc1OCC1CC1(Cl)Cl Cc1oc(C(=O)N(C2C3CN(C(=O)C(C)(C)CO)CC23)C)cc1CO c1(NC(N)=O)ccc(CC(CC(=O)NCC(CNC(c2nnc(C)o2)=O)O)=O)cc1 n1(CC)nnnc1CNC(=O)CCN(C(=O)CC1CC1CC)CCO C1(CNC(c2snnc2C2CC2)=O)CN(C(=O)C2=COCC2)CC1C(F)(F)F O=C(CCCC1CC1)N(CCc1cc(C(=O)NC2CCOC2=O)no1)CCO C(=O)(C(CC(F)F)N(C(=O)C=Cc1cc[nH]c1)C)N(CCC(N)=O)CC N1(C(CC2C(C)C2)=O)CCC(NC(=O)C(N2CCCCCC2)=O)C(CO)C1 C1(CNS(C)(=O)=O)CN(C(=O)CCOCCOCCO)CCC12CCC2 CC#CC1CCN(C(=O)C(C2CCC2)NC(C2COCC2(C)C)=O)CC1 c1(C(N(C2CCN(C(C3CC(C)OC3)=O)CC2)CCO)=O)cnc2[nH]ncc2c1 CCC(CC)(CN=c1[nH]nc(C)o1)NC(c1cn(CCC(C)C)nn1)=O Cc1ccc(C(=O)NC2CCCCN(C(c3ccn(CC#N)n3)=O)C2)cc1F c1(CC(N2CCC(N(C(C=CC=CC)=O)CC)C2)=O)cc(Cl)ccc1Br c1(C(=O)NCC2CN(C(C3CC(=C)C3)=O)C3C2C3)cc(F)c(C)cc1Cl N1(C(CNS(N)(=O)=O)=O)CCC(N(C(=O)C(F)CC2CCCC2)CCO)C1 c1(CCSC)nc(-c2cc(-c3ccccc3)no2)n(C2COC(C)(C)C2)n1 C(CCCCC(=O)NC(c1nn(C)cc1O)C)NC(C1CC(C)SCC1)=O N1(C(C=CC(C)C)=O)CCOCC1C(=O)NCc1cnn(CCO)c1 C1(F)(CNC(C(n2cc(Cl)cn2)C)=O)CCN(C(C2CCC(=O)N2C)=O)CC1 c1(N(C(=O)NC(C2CCCO2)(C)C2CC2)CC)ccccc1[N+](=O)[O-] c1(C(N2CC3(CCN(C(C(C)OCCN(C)C)=O)C3)C2)=O)cc2c([nH]1)CCC(C)C2 c1(C(=O)NCC2(OC)CN(C(CCN(C)CC)=O)C2)cc(OC)c2c(c1)OCO2 C(=O)(C1CCc2nccn21)N1CCC(C(C)(C)NC(=O)Cc2cnoc2)C1 N1(C(C(C)OC)=O)CCN(C(C2(C3CCCO3)CCC2)=O)CCC1C C1(N(C)C(C2(C)CCCCO2)=O)CCCN(C(c2[nH]ncc2C2CCC2)=O)CC1 CCC(C)(C)CCCC(=O)NCCC1(C)CCN(C(C2CCOC(=O)N2)=O)C1 Cc1cc(NC(=O)C(=O)Nc2ccc(-c3ccc(CO)o3)c(F)c2)cc(Br)c1C CC1(C(N2CCCC2CCNC(=O)COc2ccc(Cl)cc2)=O)CCCNC1=O O=C(C(O)CC(F)(F)F)NCC1CCN(C(=O)CCCN2CCOC2=O)CC1 CC(CNC(=O)C(=O)N(C)C)CN(C)C(C1(CNc2cnn[nH]2)CCC1)=O C1(NC(=O)C2CC2)CN(Cc2cnc(-c3ccccn3)s2)CC1CCC(C)(C)C C1(C(=O)NC23CC(NC(c4c(COC)cco4)=O)(C2)C3)CN2CCN1CC2C c1(C(N(C(C(=O)NC(C)Cc2cncs2)=O)C)C)ccc(F)c(F)c1 C1(F)(CNC(C=C(C)C(C)C)=O)CCCN(C(c2cc(C(N)=O)cn2C)=O)C1 N1(C(=O)CC2CC2)CC(NC(C2(C3CC3)CCOCC2)=O)C(c2ccccc2)C1 CC1CN(C(=O)Cn2ncnn2)CC1(C)CNC(c1ccc(=O)n(C)n1)=O N1(C(C(C2CCCC2)OCC)=O)CCOCC1CNC(=O)CC1COC2CC1C2 C1(CNC(CC2C(CC)C2)=O)CC(C(=O)N(CC(C)C#N)C)C1 N1(C(C(C)OCCN(C)C)=O)CCCC(CNC(=O)C(C2CCCCC2)O)C1 Cc1ncnc(C)c1CC(=O)NCC1CC1CNC(c1ncccc1F)=O N1(C(C(C)(Cl)Cl)=O)CC2CS(=O)(=O)CC2(NC(=O)C=CC2CCC2)C1 c1(CNC(C(CC)NC(=O)CSC)=O)n[nH]c2c1CCC2 Cc1nc(CO)sc1C(=O)N(CC(O)CN(C(=O)C(O)Cc1cn(C)cn1)C)C N1(C(COCCC#C)=O)CCCC1(C)CNC(C1(F)CC(C(=O)OCC)C1)=O CC1CCN(C(C23CCCC2C3(F)F)=O)CCN1C(=O)CCC(=O)N(C)C c1(OC)nn(C)cc1C(N1CCCC1CNC(=O)C(F)(F)c1ncccn1)=O C1(OCCNC(C=CC(=O)OC)=O)CCN(C(C2CC23CCC3)=O)CC1 C(Cc1ccccc1)(C(=O)NCCC(N1CCOCC1)C)OC C1(C(=O)NCC(CC(C)C)NC(C(CC)N(CC)CC)=O)CC=C(C(C)C)CC1 C1(NC(COC(C)(C)CNC(=O)CC(Cl)Cl)=O)CCN2CCCCC12 c1(N2CCC(NC(C(CC)C(C)O)=O)C(O)C2)cc2nnc(C)n2cn1 C(=O)(CC(C)C(=O)NCC1CCC(C)CN1C(c1ccc(C)n1C)=O)OC N1(C(C(C=CC)O)=O)CC(F)(F)CC1CCNC(c1cc(C)sn1)=O CCC(C(=O)NCC(F)(F)CNC(=O)OC(C)(C)C)C(C)(F)F N1(C(C2N(CC)CCC2)=O)CC(CNC(c2cncnc2C(C)C)=O)CC1(C)C C(=O)(C(C)(C)C(=O)NCC1(CNC(c2ncn(C)n2)=O)CC1(F)F)NC n1(CC)cnc2[nH]c(=NCC(C)C(F)F)nc(N3CCC(CC)(CO)C3)c12 c1(SC)ccc(C(=O)NC(C)CCCCNC(=O)C=Cc2sccc2C)c(Cl)c1 CC(N=[N+]=[N-])C(=O)NC(c1cn(C)nn1)C(=O)N(C(C)CC(N)=O)C C1(CC)(NC(C2C3CC2N(C(=O)CNC(=O)NC)C3)=O)CC(F)(F)C1 Cc1nnc(O)c(C(N2CC(NC(=O)C(C)(O)C3CCC3)CC3(CC3)C2)=O)c1C c1(NC(C2CN(c3cccc(C)c3)C(=O)C2)=O)ccc2c(c1)CCN(C)C2 c1(C(C(=O)N(CCN(C(C(C2CCOC2)OC)=O)C)C)(C)O)ccc(Cl)cc1 N1(C(C2CCC2)=O)CCC(C2CCN(C=O)C2)C1.c1(C=O)cc2cn[nH]c2cn1 C(=O)(CC(C)(C)C(C)(F)F)N1CCC(C)C1CNC(=O)C(=O)NCC(F)(F)F C1(NC(C2CCN(C(N)=O)CC2)=O)COC2(C1)CN(C(C1CCCC1O)=O)C2 C(=O)(C(O)CC(C)(C)C)NC1C(CNC(c2cn(CCC)nc2C)=O)CCC1 C1(CC)CN(C(=O)C(=O)NCc2cc(Br)ccc2Br)CC(CC)O1 c1(CC)cc(C(=O)NC2CC(CNC(C3CCOC(C)C3)=O)C2)c(C)nn1 c1(C(CC)C(=O)NCC(CO)NC(c2cnc(C)o2)=O)ccc(Br)cc1 C(=O)(C(CCS(C)=O)N(C)C)N1CC(C(C)NC(Cc2c(C)cccc2C)=O)C1 Cc1cccc(NC(C2(F)CCN(Cc3cc(C(=O)O)ccc3O)C2)=O)c1Cl C1(C(=O)NC2CCCN(C(C=CCC)=O)C2C)CCOCC12CCCCC2 c1(C(CNC(CCSC)=O)NC(=O)C(C)OCCc2ccccc2)ccccc1 Fc1ccc2c(c1)CCN(c1nc(Br)cs1)C2 c1(NC(C2CC3CC3N2C(=O)COCC2CCCC2)=O)nccc2nc[nH]c12 Cc1cc(C2(C(=O)N(C)CC3CCCN(C(C4CC4(Cl)Cl)=O)C3)CC2)cc(C)c1 c1(OC)ncc(C(N2CC3CC(N4CCC4N)C2C3)=O)cc1Br.N1CCCC1 c1(OC)ccc(CCC(=O)NCC23CC2CN(C(c2cc(F)n(C)n2)=O)C3)cn1 C(=O)(C(C)CCC)NC(CNC(C1(CC=C)CCCC1)=O)CCOC CCC(C(C)O)NC(C1(CCNC(c2cn(C3CC3)cn2)=O)CCCC1)=O N1(C(c2n[nH]c(C)c2F)=O)CCC(CNC(=O)C(N2CCSCC2)C)C12CCC2 C(CC)(CCCO)NC(N(C(CC(=O)OCC)c1ccccc1)C)=O C1(=O)CCC2(CC2)NC(=O)C=CC(=O)C(=O)NCCN1.C1(C(=O)N)CCC1.CO c1(C(N2CCCC(C)(CNC(c3cn(C)nc3O)=O)C2)=O)nc2ccccc2[nH]1 C1(O)(NC(N2CC(F)(F)C2)=O)CCN(C(=O)COc2ccccc2)CC1 C(C1CN(C(C23CCC(C2)C3)=O)CC1C(=O)NC1CC(N2CCC2)C1)=CC C1(NC(C(C)(C)C2CC2C2CC2)=O)CCC(NC(=O)CC2CCOC2)CC1 CCCC(C(=O)N1CCC(C(=O)NCCc2cc(C)on2)(CC)C1)NC(N)=O C#CCC(C)(CC)C(=O)NCC1(CC(=O)NCc2cnn(C)c2C)CC1 C1(NC(C2(C(C)C)COC2)=O)CCCN(C(C2CC(O)CN2C)=O)C1 C1(NC(C(C)OCCC(C)C)=O)CC(NC(c2c[nH]nc2C2CC2)=O)CC1O C1(C(=O)NC(C2CN(C(c3ccc(N)c(Cl)c3)=O)CCO2)C)CN2CCN1CC2 c1(SCc2nc(-c3c(OC)ccnc3)on2)ncnc2sc(C)nc12 c1(C(=O)NCC(CNC(C(C)C2CCC2)=O)F)nc[nH]c2ncc(Br)c1-2 C(C(N=c1[nH]ccn2nnnc12)C(C)C)NC(c1nc(C(C)C)sc1)=O N1(CCNC(C2CC2CSc2cnn(C(F)(F)F)c2)=O)CCOCC1 c1(CN(CC(=O)NC2CCCOC2)C)coc(Br)n1 c1(SCC(=O)NCCN(C)C(c2cn(C3CCCCC3)nn2)=O)n[nH]c(=N)s1 Cc1cc(=O)n(CCC(=O)N(c2cccc(C#N)n2)C(C)C)cn1 C1(NC(c2c(C(C)C)occ2)=O)CCC2CCN(C(=O)C(C)(C)CF)C1C2 C(=O)(C=C1SCC(=O)N1C)N1C(CNC(C=CC)=O)CCCC1.C(=O)N c1(NC=O)ccc(N(C(=O)C2=CSCS2)CC2CC2)cc1.C12C=CC(C1)NC2=O C1(C(C(N2C(CNC(C3CCN(CCO)CC3)=O)CC2)=O)O)CCCCCCC1 N1(C(C(C)OC2CCCC2)=O)CCC2(CN(Cc3ccncc3Cl)C2)C1 N1(C(c2c(CC)noc2)=O)CCCC(CNC(C2(CO)CCCC2)=O)CC1 N1(C(c2cc(C)oc2C)=O)CC2CCOC2(CNC(C2CCN(C)S2(=O)=O)=O)C1 C1(NC(C=COCC)=O)CC2CN(c3nc(C(F)(F)C(F)(F)F)nc(=N)[nH]3)CC12 C(=O)(C(CC)CC)NCC1(CC=C)CN(C(=O)Cc2ccccc2SCC)C1 CC1CN(C(c2cnc(S)nc2)=O)CC(C)N(C(c2ccc(Cl)c(F)c2N)=O)C1 N1(C(CSC(C)C)=O)CCOCC1CNC(=O)C=Cc1ccc(C(N)=O)o1 c1(NC(C2CCCN(C(c3ccc(Br)nc3)=O)C2)=O)cc(Cl)ncc1Br CC(CC(=O)NC1(CC(N2CCC(CC(F)F)C2)=O)CCCCC1)C(F)F C1(C(=O)NCC2C(C)CN(C(C3CC3(C)C)=O)C2)COC2COCC12 Cc1ccc(CNC(=O)C(C)NC(=O)CN2CC3CC3C2)c(O)c1 N1(CCNC(=O)C=Cc2nccs2)CCCN(C(C2CCC2CF)=O)CC1 c1(C(=O)NCC2CC(NC(c3c(C(C)=O)ccs3)=O)C2)ccnc(F)c1Cl c1(C(N2CC(N(CC=C)C)C2)=O)cn2cccc(Br)c2n1 Cc1cnc2n1CCN(C(=O)Oc1ccccc1F)CC2 C1(C(=O)NC23CC(CNC(c4n(CCC)ccc4)=O)(C2)C3)CCC(C)(F)CC1 CC1(C)CC(CNC(C2CC(O)C2)=O)CN(C(=O)CC(C)(O)c2ccccc2)C1 c1(NCC(c2ccc(OC)cc2)OC)cc(P(C)(C)=O)ncn1 N1(C(C)=O)CCCC(CCN2CCCC2CC(N2CCCCC2)=O)C1 C1(CN(C)C(C2C3CCC2(c2ccco2)C3)=O)COCCN1C(=O)CC1CC(F)C1 C(=O)(C1=NNC(=O)C1)NCCN(C(c1nc(C)c(C)s1)=O)CC C1(NC(c2ccc(C)o2)=O)CN(C(c2cnc(Cl)s2)=O)CCC1CO Fc1ccc(CNCC23CCCCC2NCC3)c(OC(F)F)c1 c1(C(=O)NC2CN(C(c3nccc(C(F)F)n3)=O)CC2O)cc2n(n1)CCCC2 N1(C(CC2CCCC(C)(C)C2)=O)CCC2CCC(NC(c3cc(N)ccc3F)=O)C12 CC(Cc1ccccc1)(C(F)F)NCc1nnc(-c2ccccc2)s1 c1(OC)cc(C(=O)NCC2CCN(C(=O)C(C)(C)c3nccs3)C2)ccc1O c1(CC(=O)N(C(CNC(c2cnc[nH]c2=N)=O)C2CC2)C)ccc2c(c1)OCO2 C1(C(C)(C)NC(CC(C)O)=O)CCN(C(c2cc(C3CCCCC3)on2)=O)CC1 C(=O)(CC(C)C(F)(F)F)NC1CC(CC(=O)NC(COC)(C)C)C1(C)C C=CCC(C)(CC)C(=O)NC1CCCC(N(C)C(c2cnc(OC)c(Cl)c2)=O)C1 N1(CC)CCc2cc(-c3cccc(CC(C(=O)OCC)NC(=O)CSC)c3)ccc21 c1(OC(C)C)ncccc1CC(=O)NCC1(F)CC(NC(=O)CC2CCCO2)C1 C1(CNC(C=CC(CC)C)=O)(CO)CN(C(=O)CCNC(=O)OC(C)(C)C)C1 N1(C(CCSCCCC)=O)CC(C(=O)NC(=O)C(CCC)N(C)C)CC1(C)C N1(C(CC2N(CC)CCC2)=O)CCC2CC1CN2C(=O)CCCN(C)C(C)=O S(=O)(=O)(c1csc(C2CC2(F)F)n1)N(CC(CC)O)Cc1ccccc1 c1(C(=O)NC23CC(C(NOCC4C(OC)CCC4)=O)(C2)C3)c(C)ncnc1C N1(C(c2nnn(CC)c2C)=O)CC(CCNC(=O)CC(=O)N(C)C)OC(C)C1 N1(C(C(CC#CC)NC(C23CSCC2C3)=O)=O)CC2(CCC(=O)N2)C1 c1(C2C(C(=O)Nc3n(CC(=O)OC)ncc3)C2)ccc(OC)c(OC)c1 c1(C(=O)NC2CC3CC2CN3C(C2CCCCC2)=O)csc2c1CCCC2 C1(NC(C2(NC(c3cc(Cl)cn3C)=O)C(C)C2)=O)CCCN2CCCC12 C1(OC)CCCCC1C(=O)NC(C)CNC(C)=O CN1CCCC1(C)C(N1CC(CNC(c2ncnn2C2CCOCC2)=O)C1)=O C1(C(=O)NCC2(C(N)=O)CN(C(=O)CCC3CCCC(=O)N3)C2)CC(F)C(=O)N1 C=CC(C(F)(F)F)NC(C1C(NC(=O)CCNC(=O)COC)C1(C)C)=O c1(NC2CC(C)N(C(c3cnc(Cl)s3)=O)C2)ncc(C#N)cc1Br C1(CNC(C(COCC)(C)C)=O)CC2CC(C1)N(C(c1c[nH]cc(Cl)c1=O)=O)C2 C(=O)(C(C)CC(C)CC(C)C)N1CCC(CC)(NC(c2cc(OC)no2)=O)CC1 n1(CC)nnnc1C(CC)(C1CC1)NCC1CC12CC2 CC(CC1CCOCC1)N=c1cc[nH]cc1S(=O)(=O)NC1(c2cnn(C)n2)CC1 CC12COC(C(=O)NCC(C)(C)NC(c3cc(C4CC4)[nH]n3)=O)(C1)C2 C12(C(=O)NC3CC(n4cc(CCCOC(=N)O)nn4)C3)CCCC(CC1C(=O)O)C2 N1(C(c2cccc(CC)c2)=O)C(C)CC2CN(C(C3OCC4CCCC34)=O)CC12 Cn1c(O)nc2cccc(C(N3CC(CCNC(C4CCCC(O)C4)=O)C3)=O)c12 C(=O)(C1=CCCCC1)N1CC(C=C)(CC(=O)NCC2(F)CCOCC2)C1 N1(C(C2(CNC(c3c[nH]c(=N)o3)=O)CC(=C)C2)=O)CCC(F)(C(N)=O)C1 CC1(C(N2CCCC(CNC(=O)Cc3ccc(F)cc3)CC2)=O)CCNC(=O)C1 Cc1cc(N)ccc1C(=O)NCC12CC1CN(C(=O)OC(C)(C)C)C2 C1(N(C(CCC2(NC(C=NOC)=O)CCC2)=O)C)CC2CCC1CC2 C(=O)(C#CC1CCCCC1)NC(COC)CC(=O)NCC(N1CCCCC1)C C(=O)(C(F)CCC(C)C)NC1CN(C(C2CCC(C(=O)OC)CC2)=O)CC(O)C1 N1(C(CN(C)C)=O)CCCCC1CC(=O)N(CC(C)(C)CO)C CCCCC(O)C(C)C(=O)C(CC(C)N(C(=O)C(O)CCC)C)C(=O)N N1(CC(=O)NC2C(CNC(c3c(COC)nn[nH]3)=O)CCC2)CCNC(=O)C1 c1(CC(C)C)ccc(C(=O)NC2CCC2NC(=O)CCc2ccc(O)nc2)cc1 C1(OC)CC(NC(c2ccc(C(F)F)o2)=O)CN(C(C2CC2(F)F)=O)C1 c1(N2CC(C)(C)C(NC(C3(C(F)F)CCOCC3)=O)C2)c(Cl)cncc1[N+](=O)[O-] n1(CC)cnnc1CNC(=O)C(=O)Nc1cnnn1Cc1ccccc1 n1(CCC)cc(C(=O)N(CC(C)NC(C2CCCC2O)=O)CC)nn1 N1(C(c2n(CC=C)ccc2)=O)CCN(C(c2cscc2C)=O)C(C)C1 Cc1nc(C(N2CCC(C(=O)NC3CCCC3N(C)C)C2)=O)co1 C(CC1=CCC2CC1C2(C)C)OC(c1c(C(C)C)n(-c2cccc(Cl)c2)nn1)=O Cc1nc(Cl)ccc1C(N1CCCC(n2cc(CN3CCOCC3)nn2)CC1)=O C1(C2CN(C(C3CN(C(=O)NC)C3)=O)C2)(NC(C2(C(C)C)CNC(=O)C2)=O)CC1 c1(CC(CNC(C(=C)Cc2ccccc2)=O)C(=O)OC)c[nH]c2cc(F)ccc12 c1(C(N2CCC(O)(CNC(=O)CCn3cccn3)C2)=O)cnc2ncccc2c1 C(=O)(C(CO)C(C)(C)C)NC1CN(C(C(C(C)O)NC(C)=O)=O)C1 N1(C(CC2CCCC(NC(C(C3CCOCC3)C)=O)C2)=O)CC(N(C)C)C2(CC2)C1 C1(NC(c2c(CCC)nns2)=O)(CNC(=O)Cc2ccno2)CCOCC1 c1(C(N(CC(C)(C)NC(C2C(CC)OCC2)=O)C)=O)nc(C)n(C)c1C N1(C(CC)=O)CCC2(C1)CN(C(=O)C(C)NC(S(=O)(=O)Cc1ccccc1)=O)C2 N1(C(C23CCC(NC(CC4C(C)(C)C4)=O)(CC2)C3)=O)CCN2CC(O)CC2C1 c1(C(C(=O)NCC(Cn2cc(CN(C(C)=O)C)nn2)(F)F)C2CC2)ccc(Cl)cc1 c1(NC(c2n(Cc3nnn(C)n3)nnn2)C2CC2)cn(C)nc1Oc1ccccc1 C12(C(=O)NCCc3c(CNC(COCC)=O)cccc3)CCCC1C2(F)F C(c1ccc(C)cn1)=CC(N1CC(C(C)NC(CC2(OC)CC2)=O)OCC1)=O CC(F)CC(=O)N1CCC(CCNC(=O)CCCF)C1 c1(NCCC(C)C)[nH]c(=NC2CSCC2C)nc2scnc12 C(=O)(CC(O)CNC(c1ncncc1Cl)=O)NC(C(=O)NC)(C)C c1(CC)ncc(C(=O)NC(C2CC(NC(C3CC(CC(C)(C)C)C3)=O)C2)C)cn1 Cc1nc([N+](=O)[O-])cn1CC(N1CCOC(CCNC(=O)C(C)CC(F)F)C1)=O C#Cc1ccc(C(N2CCC(CC(N)=O)(NC(C3CC3COC)=O)CC2)=O)cc1 C1(NC(C=CCC)=O)CC2CCC(C1)N2C(C1(CO)CCC1)=O N1(C(C2C(CC)CCO2)=O)CC2CC1C2CNC(=O)Cc1ccn(CC(C)C)n1 C(=O)(C1c2ccccc2Oc2ccccc21)NC1C(NC(=O)CCF)C1 C1(C(=O)NCC(CO)NC(=O)CC(=O)NC2CC2)(C(F)F)CC(F)(F)C1 C12(C(N(CCC)CCNC(C34COC(C3)C4)=O)=O)CCCC1(C(N)=O)C2 CC1(C)CCC(C(=O)NCC2CCC2)(NC(C23C(=O)C4CC2C3C4)=O)C1 c1(C(N(CCN(C(C2CC2F)=O)CC)CC)=O)cc(C)nn1CC(=O)OC C1(SCC)CCC(C)N(Cc2ccc(Nc3cn(C)nc3C#N)cc2)C1 Cc1cccn(CC(=O)NCC2CC(C)CCN2C(C2CCCC23CC3)=O)c1=O CC1CN(C(=O)NCCc2cnco2)CC(C)(C(F)F)O1 C1(CCNC(CC2(OC)CN(C(C3CCS(=O)CC3)=O)C2)=O)CCC(C)(C)C1 C(=O)(CCCC(CC)CC)NCC(CCC)C(=O)N1CCC1C1CCCCC1 c1(OC)ccc(C2CC2)c(C(=O)NCCC(C(C)C)NC(=O)C2=C(Cl)CCC2)c1 c1(C(N(C2CC(NC(C3(OC(C)=O)CC3)=O)C2)C)=O)cc2c(C)c(Cl)ccc2[nH]1 Cc1ccc2oc(N3CCC(C(C4C5Cc6ccccc6C45)=O)CC3)nc2c1 N1(C(c2c(C)cc(C3CC3)cc2)=O)CC2CCC1CC2NC(C1SCCCS1)=O c1(C(=O)NCC(CC)NC(=O)CCC=C(C)C)cnc(C)[nH]c1=N C1(CNC(c2c(OC)c(C)sc2)=O)CCC(C)N(C(C2OCCN(C)C2=O)=O)C1 C1(C(=O)OC)Cc2ccc(S(=O)(=O)NC(c3ccoc3C)=O)cc2C1 CCCC(C(=O)NCC(O)CC(=O)NCC(=O)NOC)OCC C1(NC(CCc2scc(C)c2)=O)CC2(C1)CN(C(C13CCC(CC1)CC3)=O)C2 C1(CNC(c2c[nH]c(=N)o2)=O)CCCC(NC(=O)C(c2ccccc2)O)C1 C1(OC)CC(OC)CN(C(C2CCCCN2C(=O)C(C)C)=O)C1 c1(OC)ccc(OC)c(C(N2CCCC(CCNC(=O)C=CC(C)C)C2)=O)c1 c1(NC(C)=O)ccc(CC(=O)NC(C)CNC(c2c(C)ncn2C)=O)cc1 N1(C(C(CC)n2cncn2)=O)CCC(C(=O)NCc2ccc(Cl)nc2)C(C)(C)C1 N1(C(C(C)Cn2ccnc2)=O)CCN(C(c2cncc(O)c2)=O)CC(C)(F)C1 c1(C(N(C2CCN(c3nnc(O)s3)C2)C)=O)c[nH]nc1C1CCOCC1 C1(NC(=O)NC(CC(C)C)c2ccccn2)CC2CCCC2C1 c1(C(=O)NC(CN(C(=O)C(=O)N(c2ccccc2)C)CC)C)nn(CC)nc1C C1(CC)CN(C(C23CC(CCO2)C3)=O)CCN1C(=O)Cn1nc(C)cc1C C=CCC(CNC(=O)CNC(=O)C(C)(C)C)NC(=O)CSc1ccccn1 CCCCC(F)C(=O)N1CCC(C)(NC(C2CCCN2C=O)=O)CC1 C1(C(C)C)CN(C(=O)CC2CCCC(NC(C3CCC4(CC4)C3)=O)C2)CCN1C N#CC1CCCC(C(N2CCCN(C(c3ccc(C4CC4)s3)=O)CC2)=O)C1 C1(CN(C(c2cc(CO)[nH]n2)=O)CC)CCCCN1C(=O)CN1CCCCCC1 c1(C(N2C(CN(C(=O)C3=C(Cl)CC3)C)CCCC2)=O)ccc2c(O)n[nH]c2c1 N1(C(CC(CC)C)=O)CCCC(NC(C2(C)CCOCC2)=O)C1C c1(C(N2CCCC(NC(C3CCC(OC)CC3)=O)C2)=O)ccc2ncccc2c1 C12(C(=O)NCCOCCOCC)COCC1CN(C(=O)CC1CCC(=O)N1)C2 CC1(CO)CC(NC(=O)CCOCCNC(C2(O)CCC2)=O)C1 c1(-c2onc(CC3Cc4c(nc(C)s4)CC3)n2)cc(C)cc2c1NCCC2C N1(CC(=O)N(C(CCNC(C2ON=C(C)C2)=O)C)C)CC2CCC1C2 c1(CC)nn(C)c(Cl)c1C(=O)NC1(COC)CN(C(C2CC(SC)C2)=O)C1 c1(CC)cccc(CC(N2CCN(C(=O)CN(CC)CC)CC2)=O)c1 C1(CNC(c2cc(C)on2)=O)CC(C)CN(C(C2(CN(C)C)CC2)=O)C1 S1(=O)(=O)c2ccc(cc2)CN1C.C1(OCC(F)F)CC1CC Cc1cc(C(=O)NC(CNC(=O)C(F)(F)c2cncs2)C(C)C)co1 Cc1cc(C(=O)NCCC(C)NC(C2(CN(C)C)CC2)=O)on1 C=C1CCC(C(=O)NCc2nocc2C(=O)NC(C)(CO)CCF)CC1 N1(C(C(c2c(CC)cccc2)(F)F)=O)CCCC(O)(CNC(C2CC2(C)C)=O)C1 N1(C(COCCCC)=O)CCCC(NC(c2cccc(C3(C)CC3)c2)=O)C1C C12(CNC(c3ccncc3)=O)CC1CN(C(=O)CNC(C1CCCCC1)=O)C2 C(CCC(C)C(=O)N1CCCC(NC(c2nonc2N)=O)C1)OC C1(C(=O)NC(CC=C)CC)(CC)CCN(C(C2CCCCC2O)=O)CC1 c1(C(N2CCC(C)(CNC(CC3CC(C)C3)=O)C2)=O)ccc2c(=O)ccoc2c1 c1(OC)noc(-c2nc(C3CCCC3)nn2-c2cccnc2)c1Br C1(CNC(c2c(OCC=C)cccc2)=O)CC2CCC1N2C(=O)CC1(OC)CC1 C1(C(=O)NC2CC(NC(=O)CCCn3cccn3)C2)(OC)CCOC1 c1(C(=O)NCC(C)CNC(=O)CSc2cccc(F)c2)cccc2nonc12 N12CCCC1(C1CC1)C(=O)NOCC2=O.CCCC(C)OCC N1(CCC)CC(CNC(c2ccccc2I)c2nnnn2C)CC1=O C1(C(=O)NC2C(C)CN(C(c3cnn(CC(F)F)n3)=O)C2)CCCCC1(F)F c1(C(N(CC(CC)NC(=O)C(c2cnn(C)c2)OC)C)=O)[nH]c(C)nc1C N1(Cc2c(C)nc(-c3ccc(OC)cc3)s2)C(=O)CCN(CC2C3CCC23)C1=O c1(C(=O)NC(Cn2cccn2)C(=O)O)ccc(C(F)(F)F)c(Cl)c1 C1(NC(C(CC)OCC)=O)C2CC3C1C3C2C(=O)N(CCF)C1CC1 c1(C(N2C(C(CNC(c3cn(C)nc3)=O)(C)C)CCC2)=O)cc(O)cc(C#N)c1 c1(C(N2CC3CC(CNC(=O)COCCF)C3C2)=O)ccc2cncn2c1 C(=O)(CC(C(F)F)C(=O)OC(C)(C)C)NCCCC(C)NC(C1(C)CC(=C)C1)=O C1(C(N2CCC(F)(C(N3CC4C(CO)C4C3)=O)C2)=O)CCCC2(CC2)C1 C1(CNC(Cc2cn(CC)nc2)=O)CCCCN(C(c2nnc(C)s2)=O)C1 C1(C(=O)Nc2cccc(C)c2)CN(Cc2csc(-c3ccco3)n2)CC1(F)F c1(C(=O)NCCC=C)n[nH]c2ccc(-c3cnn(CCCNC(C)=O)c3)cc12 C(=O)(CC(O)CC(C)(C)C)N1CCCCC(N(C(C(=O)NCC)=O)C)C1 N1(C(C(C)N(C(c2ccc(C)[nH]2)=O)C)=O)CCC2CCN(C)CC12 c1(C(N(CCN(C(C2CC(=O)N(O)C2)=O)CC)CC)=O)cc(CC(C)C)nc(O)c1 c1(C(C(N2CCCC(CN(C(c3cc(C)on3)=O)C)C2)=O)O)ccc(C#N)cc1 c1(CNC(c2ccc(C)cn2)=O)nc2c(s1)CN(C(c1csc(S)n1)=O)CC2 C#CCC(C)(C)C(=O)NCC(CC=C)C(=O)N1CC(N2CCC2)C1 CC1Cc2n[nH]cc2CN(CN(c2ccc3c(c2)CC(SC(C)(C)C)CC3)C)C1 c1(C(=O)NC(CCCNC(c2c(CC)occ2)=O)C)ccc2ccccc2n1 N1(C(C2CCN(C)C2)=O)CCCC2CN(C(=O)Cc3ccc(F)c(Cl)c3)CC12 C1(CN(C(C2C(C)C2C)=O)C)CCN(C(=O)CC2(N(C)C)CCCC2)C12CCC2 CC(C)CC(C(=O)NCC1CNC(=O)CO1)NC(c1cccc(=O)o1)=O c1(OCC)ccc(C(=O)Nc2nccc(C#N)c2OC)c2ccccc12 c1(C(=O)NCC(CN(C(C(CC)(F)F)=O)C)O)cccc(F)c1C C(CCCCCNC(C1CCCCO1)=O)N(C(C(c1cccc(Cl)c1)OC)=O)C C(=O)(CCC(=O)NC(CO)C(=O)NC(C1CCCC1O)C)NCCC Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(C)(C)Cl)cnn1 N1(C(C2(C)CCC(F)(F)C2)=O)CC2(CCCN(C(c3nocc3Cl)=O)C2)C1 C1(NC(c2n(CCCSC)nnn2)(C)CCBr)CC12CCCCC2 C1(NC(CCC(=C)Cl)=O)CCN(C(=O)C(C)NC(=O)CC)C2CC12 C1(C(N2CCC(COC)C2)=O)CC(F)CN1C(c1ccc(Cl)o1)=O C(=O)(C1=CCCSC1)NCC1(OC)CCN(C(c2cccc(F)c2F)=O)C1 C(=O)(C1=NOC(CNC(=O)C(F)(F)CC)C1)NCCN(CCO)CC c1(NC(=O)NCCN(CC(c2ccnn2C)O)CC)c(C)noc1C C1(S(C)(=O)=O)(C(=O)NCCN(C(=O)CC2CCCS2(=O)=O)C)CCC1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC(O)CNC(=O)CC1CCCC(=O)N1 CC(C)C(C(=O)NC12CC1CN(C(=O)CCCCn1ccnn1)C2)c1cccs1 C1(C(=O)NCC2(CNC(CC)=O)CCCC2)CCCCC1C1CC1 c1(C(=O)NC2CC(CCNC(C3CN(C(C)=O)C3)=O)C2)ccnc(C2CC2)c1 CC1CN(C(c2cnc(O)o2)=O)CC(CCNC(C23CC(F)(C2)C3)=O)O1 CCC(C)CC(C(=O)NC1CC(CO)C2CC12)NC(c1c(CO)n[nH]c1C)=O Cc1cnc(C(=O)NC2COCC2NC(=O)CSc2ccc(C(C)C)cc2)cn1 N1(C(CCC=C)=O)CC(C(F)(F)F)OCC1CNC(=O)Cc1cccc(O)c1 C1(C(N2CC(CC=C)C(O)C2)=O)CN(C(C2CC3(CCC3=O)C2)=O)CC1(F)F C(=O)(C1CCCc2cccnc21)N1CC(OC)(CNC(=O)C=C2CCC(C)C2)C1 N1(C(C(CC#C)O)=O)CC2(C1)CN(C(c1cc(CC)ccn1)=O)C2 C(=O)(C1CCCc2cncn21)N1CCC(NC(c2ccnc(S)c2)=O)CC1 N1(C(=O)CC2COCCN2C(c2cccnc2Br)=O)CCc2ccsc2C1 N1(C(CC)C(=O)NC2(CO)CC(O)C2)CC(C)OC(C)C1 C1(C(=O)NC(CC=C)C2CC2)CCCC(NC(C2CC(C)=NO2)=O)CC1 N1(C(CCC(C)SC)=O)CCOCC(CNC(c2ccc(C(N)=O)o2)=O)C1 N1(C(c2snc(C)c2Cl)=O)CC(F)(F)CC1Cn1cc(CC(C)O)nn1 c1(C(=O)NCCN(C(c2c(C)snn2)=O)C)ccnnc1NC1CC1 c1(NC(C2CC3CC3N2C(c2sc(Br)cc2Br)=O)=O)cc(Cl)cc(Cl)c1F c1(CC(=O)NCC2N(C(c3cccc(OCC)c3)=O)CC2)ccc(C)c(F)c1 CCC(CCCC(=O)NCC1(C2(O)CCC2)CC1)NC(=O)CSC CC(c1ccsc1)=CC(=O)NCCCN(CCO)C(C1CC1c1cccnc1)=O N1(C(=O)Nc2cnn(-c3cccc(C)c3)n2)CCCc2c(N(C)C)cccc21 C1(NC(c2ccnn2CC(F)F)=O)CCN(C(=O)C2=COCCC2)C12CCCC2 c1(CNC(=O)NC2C(OC(C)(C)C)CCCC2)cccc([N+](=O)[O-])c1 C1(C2CCN(C(c3nncs3)=O)CC2)(NC(=O)COCCF)CCC1 C1(=O)CC(C(F)(F)F)N1.c1(C(=O)NCc2sc(C)c(CO)n2)cc(Cl)cc(F)c1N C1(OC)CCC2CN(C(=O)CCCCN(C(=O)CCCC3CC3C)C)CC12 c1(C(=O)NC(CNC(c2ncn(C(C)C)n2)=O)C)ccccc1F c1(CN(C)C(=O)OC(C)(C)C)ccc(C(=O)Nc2ccccc2C2CC2)cc1 C1(C(=O)NC(CNC(C2(CCN(C)C)CC2)=O)C(C)C)(CC)CCCO1 c1(C(N(C)CC2CCCC(NC(c3c(C)nn[nH]3)=O)C2)=O)cc(Cl)c(Cl)cc1N Cc1c(C(=O)NCC2CN(C(=O)C(C)(O)C3CC3)CCO2)ccn1C(C)C C(=O)(C(O)CC[S+](C)C)NC1C(NC(Cn2ncc(C)c2)=O)CCC1 C(=O)(CC(C)CNC(c1cc(OC)nn1C)=O)N1CC(O)(CCC)C1 C1(OCC)CC(NC(=O)N(C2(C)CCCC2)C)C12CCCO2 C1(CC)(CNC(C2CCN2C2CCCC2)=O)CCN(C(C2CC3CC3C2)=O)CC1 C1(CNC(c2cnc(NC(C)=O)s2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 c1(-c2ccc(CN3C(C)(C(=O)OC)CCC3)s2)cc(C(F)(F)F)ncc1F N#CC1(CC(=O)NCC2CC2CNC(C2(OCc3ccccc3)CC2)=O)CCC1 C1(CC(=O)N(CCC(C2CCCC2)NC(C(C)=C(CC)C)=O)C)CSCCS1 CCC(C)(CC)C(N)NCc1c(C)nn(C(C)(C)C)c1C C=CCC(CC)C(=O)NCCOCCN(C(=O)Cc1cc(C)cc(C)c1)C C1(NCc2nccc(C)n2)CC(=O)N(c2cccc(C(C)C)c2)C1=O c1(SC)cccc(CNC(c2nnnn2C2CC2)c2ccno2)c1 CC(C(=O)NCC(F)CNC(C1(CO)CCCC1)=O)C(=O)N1CCOCC1 C(CNC(C1C=CC=CC=C1)=O)(CC(C)C)NC(C1(OC)CCC1)=O C1(N(CCC)C(C2CSCN2C(C)=O)=O)CCN(C(=O)C(CCO)N(C)C)CC1 N1(C(C(=O)Nc2c(OC)cc(SC)cc2)=O)CCC(O)(C2CCC2)CC1 c1(C(N2CCC(O)(C(C)NC(C(C)N(CC)CC)=O)C2)=O)ccn2nccc2c1 N1(C(c2ccc(C)o2)=O)CCCC2(C1)CN(C(=O)CC1CCC13CCC3)CCO2 c1(OC)ncnc(C(N2CCC(NC(C3(C#N)CCCC3)=O)C(C)C2)=O)c1F C1(NC(COCCOC)=O)CC12CCN(C(c1cnc(Br)o1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NC1(COC)CCN(C(=O)Cc2sc(O)nc2O)C1 C(=O)(C(C)(C)C1=CCN(C(c2ccsn2)=O)C1)NCC(C)Cc1cn[nH]c1 c1(C(F)F)ccc(CNCc2sc(-c3ccccc3)cc2Br)cc1 Cc1n[nH]c(=NCC(C)N(C)C(c2ccc(OCC(N)=O)cc2)=O)o1 N(C(=NCc1cc(C(F)(F)F)cs1)NC(c1nnc(C)s1)C)C(CC)C C1(CNC(c2sc(CC)c(C)c2)=O)CC(C)(C)CN1C(C1CCCC(C)(C)C1)=O Cc1cc(NC(C2CC(F)CN(C(=O)Cc3cnc(C)s3)C2)=O)cc(Br)c1 CC(CC(=O)NCC(c1ccccc1F)NC(=O)C#CC1CCC1)C(C)(C)C C1(C(=O)NCC2(SC)CCC2)CCC(C(F)(F)F)N1C(=O)CN1CCSCC1 c1(C(=O)NCC(C)N(C)C(C2CC(C)(C)CN2C)=O)nc[nH]c2ncnc1-2 C1(NC(=O)Nc2cccc(O)c2)CCCN(C(c2cnccn2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CCOCC(CNC(c2cnsc2C)=O)C1 Cc1cnc(C(=O)NC2C3CC2CN(C(=O)CCc2nc(=N)[nH][nH]2)C3)cc1C c1(C(N2CCN(C(c3ccc(C(C)=O)[nH]3)=O)CC2CO)=O)csc(S(N)(=O)=O)c1 Cc1nc(F)ccc1-c1cn(CC(C)NC(=O)CCCN(C)C)nn1 c1(CC)cc(NC(=O)C(C)(C)CCNC(=O)CN2CCCC2C)cc(O)c1 N1(C(CCC#C)=O)CCC2(CC2C(=O)NC(CN(C)C)C(C)(C)C)C1 C(=O)(C(O)C1=CCCCC1)NC(C(NOCC(=O)OC)=O)C1CCC1 O=S1(=O)C=C(CNS(=O)(=O)c2cnn(-c3ccccc3F)c2)Cc2ccccc21 C1(C(C)(C)C)CCCCN1C(C1(NC(=O)CC2(O)CCCCC2)CCC1)=O C=CCC(C(=O)NCc1cc[nH]c1C(N1CC(O)(CCC)C1)=O)C(C)C C1(NC(C(C)SC(F)(F)F)=O)C2CC3CN(C(=O)C=C4CCN(C)C4)C1C3C2 n1(C(CC)CC)ccc(C(=O)NCC(C)(O)CNC(c2ccc(C(C)C)[nH]2)=O)n1 N1(C(CC=CCC)=O)CC2(CCC(CNC(C3CC(O)CN3C)=O)O2)C1 c1(OC)ccc2oc(C)c(C(=O)NC3CCCCN(C(=O)C(C)(C)OC)C3)c2c1 N1(C(C(C)(C2CC2)OC)=O)CCOCC(C(=O)NC2(CCO)CCCC2)C1 CC1(C)CN(C(=O)C2=COCC2)CC1CNC(=O)C=Cc1cnccn1 S(=O)(=O)(c1cccc2c(N(C)C)cccc12)NC1CCN(C(C(CC)CC)=O)C1 c1(C(N(C(CNC(c2ccnc(C)c2C)=O)C)C)=O)cnc2ccoc2c1 Cc1ccc(C(=O)N(C(CO)C(=O)N(C)C)C)cc1.C1=CCNC1=O C(=O)(C(C)(CCC)CCC)NC(CC#C)CC(=O)NCc1cncn1C N1(C(C2CCC(NC(C)=O)CC2)=O)CC2CN(C(c3ocnc3C)=O)CC12 Cc1cnc(N2CC3CN(C(=O)C(O)C4CCC4)CC3C2)nc1S(C)(=O)=O Cn1ccc(C=CC(N2C(C(=O)NCCOCCN=[N+]=[N-])CCC2C2CC2)=O)c1 c1(C(N(CC(CC)NC(=O)CC2CCCOC2)C)=O)ccc2cnccc2c1 C1(C(=O)NCCCCCN(C(c2cc(OC)no2)=O)C)CNC(=O)C(C)(C)C1 c1(N(C)C)ncc(C(=O)NCCC2CCN(C(C3CCOCC3)=O)C2)cn1 C1(CC(C)(C)C)COCCN1C(=O)Nc1ccncc1F c1(C(c2nnnn2CCC2CC=CC2)NC(=O)OC(C)(C)C)nc(C2CC2)no1 C(CCC(=O)NC1(C(=O)N(CC(N)=O)C)CC1)SC C1(NC(CSCC(C)C)=O)CCC(CNC(c2ccsc2)=O)C1 C1(C2(O)CN(C(=O)C(CO)C(C)C)C2)(CNC(c2c(C)ccc(N)c2)=O)CC1 c12ccc(cc1)COC2=O.c1(CC(=O)NCC)ccc(OCCO)cc1 C1(C(=O)NCC(CNC(COCCC)=O)(C)F)CCc2nc(C)cn2C1 c1(C(=O)NC(CNC(C(C=C)O)=O)C2CCC2)cccc(C(F)(F)F)c1 C(=O)C(O)CCC(C)C.n1(CCNCC)cc(C(c2cccnc2)O)nn1 C1(CNC(CNC(C)=O)=O)CC2(CCN(C(=O)C=C(C)c3cnn(C)c3)C2)CO1 Cc1noc2nc(C(C)C)cc(C(=O)NCCN(C(=O)C(=O)NC3CC3)C)c12 c1(N(CCOC)C)nc(NC2CC(C)(C)C2OC)nc2c1CCC2 c1(C(=O)NC2(C)CC(NC(CCNC(=O)NC)=O)C2)cnc2c(cnn2C)c1 c1(OC)ccc2cc(C(=O)NC3CN(C(c4cc(C)c(C)o4)=O)CC3C)[nH]c2c1 c1(NC)cc(C(=O)N(CCCNC(=O)C(C)C(F)F)CCO)cc(Cl)n1 c1(C(N)=O)nccnc1C(=O)NCCOCCCNC(=O)CC1CSCCS1 C(=O)(C(C)(C)CC#N)N1CCCC(N2CCN(C(Cc3cnn(C)n3)=O)CC2)C1 c1(C(=O)NCCN(C(c2cc(C(N)=O)co2)=O)CC)cc(C(C)(C)C)no1 Cc1ccc(-n2cc(CCNC(c3cc(C(F)(F)F)on3)=O)nn2)nc1 c1(CC)cc(C(=O)NC2CC3CC2N(C(C24COC(COC)(C2)C4)=O)C3)cc(O)n1 C1(C2CCN(C(=O)CN3CC4CC4C3)CC2)(NC(=O)C(O)C2CCCC2)CCC1 C1(NC(=O)COCC2CCOC2)CCCCCC1.C12CN(C1)C2 C1(NC(C2(C)CC=CCC2)=O)CCN(C(c2ccc(O)c(N)n2)=O)CC1F C1(C(=O)NC(CN(C(C2CN(C(=O)OC(C)(C)C)C2)=O)CC)C)CCCC(F)(F)C1 CCCC(C)(CCC)C(=O)NC(CC1CC1)C(=O)NC(c1cccc(O)c1)C N1(C(c2c(OCC=C)cccn2)=O)CCCCC(NC(=O)CCCC(=O)OC)C1 N1(C(c2[nH]cc(C)c2)=O)CCC2CCCN(C(c3nnn(C)c3N)=O)C2C1 C1(C(C)C)CC(C(=O)N(C)Cc2cn(-c3ccccc3Cl)nn2)CCO1 c1(C(=O)NCCN(C(=O)CC2(COC)CC2)CC)ccc(C(C)C)nc1C N1(c2nc(C)cc(OC)n2)CC(NC(=O)CN2CCCCCC2)C2CCCCC12 C(=O)(CCOC1CN(C(=O)CSc2nc[nH]n2)C1)NCCCC1C(C)C1 C1(C)(CC)C=C(C(=O)N2CCC(CC(=O)NCC(O)C(C)(C)O)CC2)C1 c1(N2CCC(c3ccc(C(C)C)cc3)(C)C2)c(F)cc(C#N)cc1F c1(C(N2CC(NC(CC(=O)OCC)=O)C3(C2)CC3)=O)c(F)ccc(I)c1F N1(C(c2cc(OC)ncc2Cl)C(=O)NCCCSC)CCCC2(CCNC2=O)C1 N1(C(C2CCC3(CC3)N2C(C2CC(O)C(F)C2)=O)=O)CC=CC12CCOCC2 C1(C(N2CC(N(CCOC)C)C2)=O)OCCC1CNC(C1CCC1COC)=O C1(NC(C2(C)C(C)C2)=O)CCN(C(C2CC2c2ccnn2C)=O)C1 C1(CC)CCN(C(c2ncn(C)c2C)=O)C1C(=O)NCC(C)(C)n1cccn1 c1(OCC=C)cccc(CN2CC(NC(c3ccc(CO)o3)=O)C(F)C2)c1 c1(C(=O)NCC(CNC(CCCCOCC)=O)C)ncc2[nH]ncc2n1 n1(CCC)nnc(NC(=O)C(C(C)O)NC2CC2C2CNC2)c1C#N c1(C(N2C(C(=O)O)CSCC2)=O)sc2sccc2c1Cl N1(CC)CC(C(=O)NC2CC(CCF)C2)CC1=O.C(=O)(CN)NC(=O)NC1CC1 Cc1nc(CC(C)C)oc1C(=O)N(C(C)CCNC(=O)CNC(N)=O)C N1(C(CC2(OC)CCC2)=O)CC2CC1CN(C(c1c(C)ccc(F)c1O)=O)C2 C(=O)(CN=c1ccc(C#N)c[nH]1)N1C(C)CN(C(=O)Cc2ccnn2C)C(C)C1 C1(NC(c2cc(OC)ncc2)=O)CCCCCN(C(=O)C(C2CCCCC2)=O)C1 C1(C(N(CCCCNC(CCc2cncc(C)c2)=O)C)=O)CN2CCN1CC2C C1(C#N)(C(N(CCCN(C(=O)C(C)(C)c2cnco2)C)C)=O)CC2CCC1CC2 c1(SC)cccc(CC(N2CCCC(CCc3cnc(N(C)C)nc3)C2)=O)c1 c1(CCOCCC(=O)N(CCNC(C2(SCC)CC2)=O)C)ccc(C)cc1 C12(C(=O)NCC3CN(C(CC4CC(C)C4)=O)CC3O)CCC(C)(CC1)OC2(C)C CCCCC(O)CC(=O)NCCN1CCCN(C(c2cc3scnc3[nH]2)=O)CC1 C1(CC(N2C(CN(C(CCOCC)=O)C)CCC2)=O)CCC(=O)CC1 c1(OC)cc(C(N2CCCC(NC(C3CC(C)C3)=O)C2)=O)ccc1C CN1CCC(C#N)(C(=O)N(C2CC(NC(=O)C(C)(F)F)C2)C)CC1 C1(C(N2CC(SC)(CNC(c3cccc(OC)n3)=O)C2)=O)CC2CC1CC2=O c1(CC(C)C)c[nH]c(C(=O)NC2COCC2n2cc(C3(C(=O)O)CC3)nn2)c1 c1(CC)cc(NC2(CCSC)CCC2)ccc1O CCC(C)(C)C(O)C(=O)NCC1(CNC(c2cc(CO)[nH]n2)=O)CC(F)(F)C1 CC(CC(=O)NCC1CCCCCN1C(=O)Cn1cnnc1O)CC(F)(F)F Cc1ccc(SCC(=O)NCC(C2CC2)N(C(=O)CCc2cccs2)C)cc1 C(=O)(C#CC1CCOCC1)N1CCN(C(CN(C2CC2)CC)=O)CC1C(F)F N1(C(CC)=O)Cc2ccccc2C(CNC(c2cnc(O)n2C)=O)C1 N1(C(C=CC(=O)N(C)C)=O)CC(OC)C(C(=O)NC2(C(N)=O)CC2)C1 C1(CCNC(c2cnc(C(C)C)[nH]2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC(C)O1 N1(C(CCSCC)=O)CCC(C2CCN(C(c3cn[nH]c3)=O)C2)C1 C1(C(=O)Nc2ccc(C#C)nc2)CCCCCCN1C(=O)CC1CCCOC1 N1(C(c2c(NC)cccc2)=O)CCOC(C)(CNC(=O)CCn2ccnc2)C1 C=CCCC(F)(F)C(=O)NC(CCC)CCCNC(c1[nH]nnc1C1CC1)=O c1(C(=O)NC(CNC(c2c(OCC)n[nH]c2)=O)C)ccc(C)c(F)c1Br c1(CN(C2CCN(C(C)=O)C2)C(=O)OC(C)(C)C)nccc2c(C)cccc12 N1(c2sc3cccc(C)c3n2)CC(C(=O)N(C)C)Oc2ccccc21 c1(C(=O)NC(C)CN(C)C(C2C3(CC3)C23CC3)=O)cc([N+](=O)[O-])cc(Cl)c1Cl N1(C(CCCOC)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C(C2CC2)C1 c1(OCC(=O)N(CC(C)NC(CSCC#C)=O)CC)ccc(F)nc1 C1(CC(=O)N(C2CCCCC2)C(=O)OCC2CC(F)(F)C2)COC(C(F)(F)F)C1 C1(CNC(C(CC)OC)=O)CC2CCCCC2N1C(=O)CCOC1CCCCC1 C12(CC(=O)NC(C3CCCN(C(=O)CS(N)(=O)=O)C3)C)CC3CC(CC(C3)C1)C2 Cn1nc(C(=O)NCC(C2CC2)NC(c2c(Cl)n[nH]c2C2CC2)=O)cc1CO c1(C(N2C(CN(C)C(C3COC4COCC34)=O)CCCC2)=O)cc2c(s1)CCC2 CCC(N=c1[nH]c(=NCCCc2cnn(CC)c2)[nH]c2c1CCCC2)C1CC1 C(=O)(C1=C(C2CCCCC2)N(CC(F)F)C(=S)NC1c1cnn[nH]1)OCC c1(C(=O)NCCOCCn2cc(C3(C)CCOCC3)nn2)cnn2c1OCC(F)C2 c1(C(N2CCCC(C(C)NC(=O)CCC(=O)N(C)C)C2)=O)cc(N(C)C)ccc1F C1(C(=O)NC(C2(O)CCN(C(c3cnc(N)cn3)=O)C2)C)Cc2ccccc2O1 C1(C(C(=O)N(CCCCN(C(C(c2cnccn2)C)=O)C)C)F)CCCCC1 CCCC(C(=O)OC)C(=O)NCC#CC(N1CCC2C(C(N)=O)C2C1)=O c1(C(=O)NCC2N(C(CC3OCC(C)(C)C3)=O)CC(O)C2)cnc(S(C)(=O)=O)s1 O=C(CC1CCc2ccccc21)NC1(CNC(C2CC2C2CCCC2)=O)CC1 c1(CC(=O)NC2(CN(C)C(C3CC(F)C(=O)N3C)=O)CCC2)c(F)cncc1Cl N1(C(C(C)OC2CCCC2)=O)CCN(C)C(C(N2CC(F)CC(F)C2)=O)C1 N1(C(c2n(C)ncc2C2CC2)=O)CC2CN(C(C34CCCC3(CO)C4)=O)CC2C1 N1(C(CC(CC)C2CCC2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1C(C)C C(=O)(CCC(C)(C)F)CC(C)N(C(=O)C(c1ccccc1)F)CCNC c1(C(N2CC(CNC(c3n(OC)cnc3C)=O)OCC2)=O)cnc2[nH]cnc2c1 Cc1cn(CC(=O)NC2CCN(C(C3CCC3(C)C)=O)C23CCC3)c(=O)nc1O C(=O)(C1=CCSC1)N(CCCOCCNC(=O)C(=O)NCC(N1CCCCC1)=O)C C1(N(C(=O)CCc2cnco2)C)CCCN(C(=O)C(c2cccnc2)N(C)C)C1 Cc1nn(C)c(NC(=O)CC2COCCN2C(c2cc(CO)ccn2)=O)c1C=O CC1CN(C(=O)CCc2nccs2)CC(C)N(C(c2ccc(C3CC3)nc2)=O)C1 C(=O)(C(C)(C)CC(=O)N1CCC(CN(C)C(c2nccc(F)c2Cl)=O)C1)OC c1(C(N(C)CCN(C(=O)C(=Cc2ccccc2)C#N)C)=O)nnc(O)cc1O c1(OC)cccc(CC(N2CCCC2CN(C)C(c2cc(N)ccn2)=O)=O)c1 C(C(=O)N1CCC(C(N2CC3CC3(CO)C2)=O)(CC)C1)(C(C)C)SCC c1(C(=O)NCC(C)N(C(CNC(CCNC(C)=O)=O)=O)C)cnc(N(C)C)cn1 N1(C(C=C(C)C2CC2)=O)CCOC(CCNC(C2CCN(C)C2)=O)C1 N1(C(=O)CC2CC(Cl)(Cl)C2)CCc2ccc3ccccc3c2C1 N1(C(C(=O)NCCC2C=CCOC2)=O)CCOCC1CC1CC1 C(=O)(C(F)C(C)C(F)(F)F)N(CCCNC(c1cncc(Br)c1)=O)CC c1(CC(=O)NC2C(NC(C3(CC=C)COC3)=O)CC2)csc(N2CCCC2=O)n1 C12(C(=O)OC)CCCCC1(C(=O)N(Cc1ccco1)CC1CCCO1)CC2 CCC(C)CCCC(=O)N1CCOCC1CNC(=O)CCCC(N)=O CCCC(CC(C)C)C(=O)NC1(C)CC(C(=O)N(CC(C)C#N)C)C1 C(=O)(C1c2c[nH]nc2CCC1C)NCCC(C)NC(c1cc(Cl)ccc1Cl)=O C#Cc1cncc(C(=O)NC(C)C=CC(=O)NC(c2ccccc2)CC)c1 C1(C(c2ccc(Cl)nc2)N(CCNC(C2(CCC)CC2)=O)C)Cc2nncn2C1 C(=O)(CC(C)(C)C#N)N1C(C(C)(C)NC(C(C)Cc2ccc(F)cc2)=O)CCC1 C(=O)(NNc1cc(Cl)cc(Cl)c1)NC(C#C)Cc1ccc(Cl)cc1 c1(OC)ccc(C(N2CCC(NC(c3cc(Cl)cc(I)c3)=O)C2)=O)c([N+](=O)[O-])c1 CC(C)(O)C(F)C(=O)NCC(O)CC(=O)NCC(O)CNC(N)=O C1(CCC(C)C)CCC(C(N2CC(CNC(c3nncs3)=O)C(C)C2)=O)CC1 CC1CC(C(N2CC(CN=[N+]=[N-])C2)=O)CN1C(=O)CC1CSC1 Cc1ncc(C(=O)NCC2(F)CCN(C(=O)CN3CC(=O)NC3=O)C2)n1C c1(C(=O)NCC2(C(N(C(C=C)C)C)=O)CC23CCC3)cn(C)c(=O)n1C CC1CC(NC(=O)CCSCC2CCCCO2)CN(C(c2ccncc2F)=O)C1 OCC1(c2ccccc2)CCC(NCCCOC2CCOC2)CC1 C(C(CO)(CO)NC(=O)C=Cc1ccccc1)N(C(C1C(C(=O)OC)CC1)=O)C C1(NC(c2c(C)n(C)nc2)=O)CC1C1CCN(C(C2CCOC(C)C2)=O)CC1 c1(NC)ccc(F)cc1C(=O)NC(CNC(=O)C(C)Cc1ccnn1C)C(C)C N1(C(c2occ(C)c2C)=O)CCCC(CNC(c2cccc(C(N)=O)n2)=O)CC1 c1(C(=O)NCC2CN(C(C3(CC(C)=O)CC3)=O)CC2C)cc(F)c(F)cc1F C(CC(C(C)C)NC(C1OCC1(C)C)=O)NC(CC=CCC)=O C(=O)(C(=O)CC(C)C)NCCC(CC)(CC)NC(CCC(C)OCC)=O c1(C(=O)NCCC2(CNC(C3C(CC)C3)=O)CC2)cc2n(n1)CCCC2O CCCCC(O)C(C)C(=O)N1CC(F)(F)CC1CNC(c1cnc(CC)[nH]1)=O N1(C(C(C)OC)=O)CC2CN(C(C3(c4cc(C)no4)CCOCC3)=O)CC2(C)C1 Cc1cc(CN=c2[nH]c(NC(c3nc4ccccc4[nH]3)=O)cs2)c(F)cc1Cl C(CCCC(=O)N(CCC(c1cccs1)NC(c1scnc1C)=O)C)OCCC=C c1(CN2CCC(CNC(C(CCC)OCC)=O)C2)ccc(Cl)nc1C c1(C(=O)NCC2(CNC(C3(F)C(C)OCC3)=O)CC2)ccc2cccc(F)c2n1 CCCCC(C(=O)NCC1(F)CCN(c2cc(OC(C)CC)ncn2)CC1)C(C)C C1(C(=O)NCC2CN3CCC2C3)CCC(O)CN1C(C1CCC1(F)F)=O N1(C(c2nn(CC)c(C)c2)=O)CC(NC(C2CCOC(=O)N2)=O)CC1(C)CC Cc1nc(C)c(C(=O)NCC=CCNC(c2cc([N+](=O)[O-])c[nH]2)=O)c(C)n1 N1(C(C(C(C)C)CO)=O)CC(C)OC2(CCN(C(=O)CC3CC(C)(C)CO3)C2)C1 C1(C(=O)NCC(C(=O)NC)C)CCC2CCC1CN2C(=O)CCc1ccco1 c1(C(N2CCC(N(C(CCC(=C)Br)=O)C)C2)=O)cc(-n2ccnn2)ccc1F C1(NC(N2CCOC(C3CC3)CC2)=O)CC[Si]2(CCCC2)CC1 c1(C(N2CCCC(CCNC(C3COC(=O)O3)=O)C2)=O)ccc(Cl)nc1O N1(C(c2c(=O)ccn(C)c2)=O)CC2CCC(NC(C3CCC(=O)NC3)=O)C2C1 c1(OC)ccc2c(CCNC(=O)C(N3CCCC3c3ccc(Br)s3)=O)c[nH]c2c1 C1(C(=O)NC2(C)CC(F)(F)C2)CC(NC(=O)Cc2ccco2)C12CCC2 N1(C(C2(NC(C)=O)CCC2)=O)CCC(CCC(C)(C)NC(=O)C(O)C(C)C)CC1 C(CN=[N+]=[N-])(C(=O)NC1CCCN(C(C)=O)C1)NC(CN(CCC)C)=O c1(C(N2C(CCCC)CCC2)=O)cc(CNC(C2(F)CCOC2C)=O)ccn1 c1(CNC(C(CN(C)C)NC(COCCC=C)=O)=O)ncc[nH]c1=O C1(CCC=O)CCCN(C(=O)C(O)C2CC2)C1.N(CCF)(CC)CC CN1CC(CNC(=O)C(O)C2(O)CNC2)C(F)(F)C1 C1(C(N(CCCNC(C2C(CCC)C2)=O)C(C)C)=O)CS(=O)(=O)CC(=O)N1 CCC(O)C(C)(C)C(=O)N1CCC1CNC(c1c(-c2ccccc2)c[nH]c1C)=O N1(C(C(=O)N(C)C)=O)CCC(NC(c2ccc(C3CC3)cc2F)=O)C(F)C1 c1(OCCCCC)ccc(C(=O)NC2CC(NC(C3(C)CC3(C)C)=O)C2)cc1 C#CCCCCCC(=O)NC1CCC1CNC(=O)Cc1cnccc1OC C1(NC(C2(NC(C)=O)CCCCC2)=O)CC2CN(C(=O)Cc3cc[nH]n3)CC12 C(N=c1nc(N2C3CCC2CN(C)CC3)c2c([nH]1)CSC2)c1cccc(C)c1Cl S(=O)(=O)(CCCC(CCCCC)OCC(F)F)NCC1(C=C)CCC1 C(c1ccc(F)cc1F)=CC(=O)N(CCCNC(=O)CC1CC1(C)C)C(C)C c1(C(c2nnnn2C2COC2)NCCCCOCCO)ccc(F)cc1 c1(C(=O)NC(CC=C)CNC(=O)Cc2ncc(C)o2)cc(F)cc2cc[nH]c12 c1(C(N2C(C)(CCC)CC2)=O)c(CNC(c2cccnc2CC)=O)cnn1C c1(CC(=O)NC2CC(F)(CNC(C(=C(C)C3CC3)F)=O)C2)ccc(C)c(Cl)c1 c1(NC(C2CCC(C)N(C(=O)CCCCC(N)=O)C2)=O)ccn2nccc2c1 C1(=CC(=O)NC2(CO)CN(C(CCCC)=O)C2)CN2CCC1CC2 c1(OCC(N2CC(C)C(NC(=O)CC3CC4(CC4)CO3)C2)=O)ccc(Cl)cc1Cl N1(C(=O)NC2CCC(CC(N)=O)C2)CC2(CCC2)C12CCC2 C1(NC(COCC=C)=O)CN(C(c2cc3scnc3[nH]2)=O)C(C)(CC)C1 C(=O)(CP(C)(C)=O)NCCN(CCOC)C(c1cnc(COC)nc1)=O C=CCCCCCC(=O)N1CC(OC)CC1CCNC(C1CN(C2CCC2)C1)=O C1(C)(C(N2CC(OC)(CNC(=O)C(C)CCN(C)C)C2)=O)C(C)(C)C1(C)C CC1(C)CCCN(C(=O)NC(c2cccc(O)c2)(C)C(=O)NCCCl)C1CO c1(CCNc2ccccc2)cn2c(n1)CCCC2.CC1(C)CC12CO2 Cc1c(C(N2CCCC2C2CCCN(C(=O)C(C)CO)C2)=O)cccc1[N+](=O)[O-] CC1=NOC2(C1)CC(c1nc(-c3ccccn3)nn1C1CCOC1)C2 C1(C(N(C)C)=O)C2CCC(C2)C1NC(c1ncccc1NC1CCCC(N)C1)=O C(CS(=O)(=O)c1ccc(F)cc1)NC(C(C(=O)OCC)OC)=O C1(NC(COCC)=O)CCCC(NC(c2nn(CC(F)(F)F)cc2Cl)=O)CC1 N1(C(C2(OCC)CCOCC2)=O)CC2(CNC(C3CC(C)CO3)=O)CCC1CC2 c1(C(=O)NCC2CC(C)(C)CN2C(=O)CNC=O)cnc2ncnc(O)c2c1 C(=O)(CCCC(=O)NCCC1CCCN(C(=O)Cc2nc(C)sc2C)C1)OCC C1(C(N(CCC(C)NC(CCC(=C)C)=O)C)=O)C(C2CC2)C1(F)F c1(SCc2c(OC)c(Br)cc(Cl)c2)nc(Cl)nc2c(F)cc(C)cc12 C1(CNC(c2cc(OC)ns2)=O)CCN(C(=O)C(C)=CC(C)(C)C)C(C)C1 C(N=c1ccnc(-c2cccc(C(N)=O)c2)[nH]1)C1CN(C(C2C(=C)C2)=O)C1 C1(C)(C(C)C)CCN(C(=O)CONC(=O)CN2CCC(F)CC2)CC1 CC(CC(=O)N1C2CCC1CC(NC(c1nc(C3CC3)cs1)=O)C2)P(C)(C)=O N1(CC(=O)NCCN(C(=O)C(F)CC2CCOC2)C)CCOCC1 N1(C(c2ccc(CC3CC3)o2)C(=O)NC(CC)C)CC(c2ccccc2)C(C)(C)C1 Cc1c(CC(C(C)C(C)C)=O)cnn1C.N c1(CC)nc(C(=O)NC2CC(NC(c3cnc(OCC(F)F)cn3)=O)C2)c(C)o1 C(=O)(C(CC)CCOC)N(CC(CC)NC(c1ccc(O)c(Cl)n1)=O)C C#CC1(C(=O)NC2CC(=O)N(CC)C2)CCN(C(=O)CCN(C)CCC)CC1 C(=O)(CC(C(C)C)C(C)C)N1C(C(C)NC(c2ccnc(CO)c2)=O)CCC1 CN1CCN(C2CCC(C(N3CCCCC3COc3ccccc3)=O)C2)CC1 c1(C(=O)NCC2C(C)CN(C(=O)C(C)(C)C3CCC3)CC2)ccc(F)c(C#N)c1 C(C)(C)(CCC(=O)N1CCCC(NC(=O)C=CC(=O)NC2CC2)CC1)OC C1(NC(C23CC(c4ccc(F)cc4)(C2)C3)=O)CCCC12CCN(CC#N)C2 c1(CC)nc(C)[nH]c1C(=O)NC(C)CN(C(=O)CC1CCCO1)C c1(C(=O)NCC(C)CNC(=O)CC2COC3CC2C3)ccc(F)cc1C(F)F C1(C(N2CC(NC(c3n(CC)ccn3)=O)C(C)C2)=O)CCc2ncnc(C)c2C1 C1(CC=C)(NC(=O)CCCCCO)CCCN(C(=O)Cc2ncccc2C)C1 n1(CC2CCN(C(=O)NC3CCC(C(=O)O)C3)CC2)cnc2ccccc12 N1(C(CN2C(C)CCC2C)=O)CCN(C(=O)C=Cc2cccc(CO)c2)CC1C CC1(C)OCC2CNCC12NCCCOC1CC1(F)F C(=O)(C(C)C(C)C1CCCC1)N(CCCCN(C(C)=O)C)C.C12CC(F)(C1)C2 N1(C(C2CC(N(C)C)C2)=O)CC2CCC1CN2C(c1csnc1Br)=O N1(C(CCNC(=O)NC)=O)CCC(C)(C)C1CNC(=O)CC1C(=O)N(C)N=C1C C12CC3CCC1CN(C3)C(=O)C1(CC1)C(=O)N2.C1(CN(C)C)CCCC1(C)C c1(OC)ccc2[nH]c(=NC(C)CCSC)[nH]c(=NC3CC(O)CC(C)(C)C3)c2c1 Cn1cc(C#N)cc1C(N1CCC(CCNC(c2c(Cl)nsc2Cl)=O)C1)=O C(N=c1[nH]nc(CC(C)C)s1)C1OCCN(C(C(=Cc2cn[nH]c2)C)=O)C1 N(C1CCCc2ccc(O)cc21)C(=O)SCC=CCc1cn(C)nc1 Cc1cn(C)cc1C(=O)NC1CCC(CNC(=O)Cc2ccccc2CC#N)C1 c1(C(N2C(CNC(C=NOC)=O)CN(C)CC2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(NC(C(CC)CCOC)=O)CN(C(C2(C)CC(C)(C)C2)=O)CC2(CCC2)C1 C(=O)(C(O)CCCNC(C1(O)CC1)=O)NC1CCN(CCC)C1 CC1CC(=O)NCCN1C(c1cc(CNC(=O)CC2CCCN2C)on1)=O CC(C)CS(=O)(=O)CC(=O)NCC(C)CNC(=O)CSc1cccc(O)c1 N1(C(c2nc(C)[nH]n2)=O)CC(NC(C2CCC2(F)F)=O)C(C(F)F)C1 c1(C(=O)NCC(C2CCOC2)NC(c2cnc(C)o2)=O)c(C)nn(C)c1C(F)F C1(CN(C(=O)NCc2n(CC)ccn2)CCO)CCC(C(F)(F)F)CC1 C1(NC(C(C)N2CCC2)=O)CCCC(CNC(=O)CN2CCS(=O)CC2)C1 C(C(C)(C)CCNC(c1ccc(C(C)(C)C)o1)=O)NC(C1(CCC)CCC1)=O c1(C(C(=O)NCC)N(C2CCC(C)C2)C)ccc(OC)c(OC)c1OC.C1CCC1 CC(=O)CCCC(=O)N1CCN(C(c2ccnnc2O)=O)CC1CC(C)(C)C c1(-c2c(F)ccc(NC(c3c(OC)ccc(C)c3)=O)n2)ccc2occc2c1 N(C1COc2c1ccc(Cl)c2Cl)C(C(=O)NC(C)(C)CN1CCC(O)C1)=O C12(NC(c3c(OC)ncc(Cl)c3)=O)CCCCC1N(C(=O)CCC(F)(F)F)CC2 C1(NC(C(C2CC2)OC)=O)CCN(C(=O)CCc2ccn(C)c2)CC1O C(=O)(C(C(=O)NC1(CNC(=O)C(F)C2CCC2)CCCC1)C(C)C)OCC c1(OC)cnc(Br)cc1C(N1CC(CC(N2CCC3CC23C)=O)C1)=O N1(C(C)C)CCOC(C(=O)NCC(O)CNC(c2ccccc2C2CCC2)=O)C1 c1(C(=O)NCC(CNC(c2c(C)snn2)=O)CO)ccc2c(c1)CC(=O)NC2 N1(C(C(C(CC)O)C)=O)CC(NC(=O)CC(C)(C)C(C)(F)F)CC12CCOCC2 C1(CNC(CC(C=C)C)=O)Cc2ccccc2CN1C(c1cc(F)cnc1O)=O c1(C(N2CC(NC(CC(COC)C)=O)C(SC)C2)=O)c(C)nn2cc[nH]c(=O)c12 C(C(=O)N1CC(O)CCO1)(C1CCCO1)NC(Cc1c(C)ncs1)=O N1(C(c2c(C)csc2Cl)=O)CC(C2CCCN(C(c3ccc(Cl)[nH]3)=O)C2)C1 C1(C(=O)NCCOCCN(C(=O)C(CCSC)N(C)C)C)(CC)CCNC1=O C1(S(N)(=O)=O)(C(=O)NCC2N(C(Cc3c(C)n(C)nc3)=O)CCOC2)CCCC1 c1(C(N2C(CNC(=O)Cn3cnnc3)CCC2)=O)ccncc1Cl c1(NC(C2OCC(C)OC2)=O)ccc2ncnc(O)c2c1 Cc1cc(C(=O)NC2CC2NC(c2cccc3c2CCCC3)=O)cc2ccoc12 c1(C(=O)NC(CC)CO)cc(O)nc2c1CN(C(C1(O)CC1)=O)CC2 c1(CC(c2ccccc2)NC(C2(NC(=O)OC(C)(C)C)COC2)=O)ccc(O)nn1 c1(C(N2CCOCC(CNC(CCOCCC)=O)C2)=O)cc2ccncc2[nH]1 c1(C(=O)NC(CNC(Cc2cc(C)no2)=O)(C)CC(C)C)cc2c[nH]cnc-2n1 N1(C(C(COC)C)=O)CCC(NC(=O)C(=Cc2cnn(C)c2)C)C12CCCC2 C1(C(C)C)CCN(S(=O)(=O)NC(C2(C(F)(F)F)CCCCCC2)=O)CC1 c1(CCCCC)cc(C(=O)N(CCC(C)NC(=O)CC2(C)CCOC2)C)n[nH]1 C(=O)(CCCC(=O)NCC(C1CC1)NC(=O)CCc1ccc(Cl)s1)NCC c1(CCC(=O)N(CC(CNC(C(C)C2CCOC2)=O)(C)C)C)ccc(F)c(F)c1 c1(C(=O)NC(CC(C)NC(c2cc(CCOC)on2)=O)C)cnc2n1CCOC2 C1(CCNC(C2CC23CCCC3)=O)CCCN(C(=O)C(=C2CCCCC2)F)C1 C1(C(N2CCN(CCc3cccc(Cl)c3)CC2)=O)C2CC3C(C2=O)C13 C1(C(=O)NCC(C2(O)CCN(C(=O)C=Cc3cnc[nH]3)C2)C)(CC)CCOCC1 C1(NC(C=CCN(C)CC)=O)CCN(C(c2cc(O)nc(Cl)c2)=O)CC(C)(C)C1 C(=O)(CN=S(C)(C)=O)NCC(C)(CO)NC(C1CC1c1ccccc1F)=O C(=O)(C(CC(C)C)C(C)C)N1CC(OC)(CNC(=O)Cc2cccn2C)C1 C(=O)(CCCC(C)C)NC1CCN(C(C(C)OCc2cccc(C)c2)=O)C1 c1(C(=O)NC(CC)CNC(c2csc(Cl)c2Cl)=O)cc2c(s1)COCC2 c1(OC)ccc(OC)c(C2CC2)c1.N12CCCC1CNC2=O c1(OC(C)C(=O)N(C2CCC(NC(C3CCC3(F)F)=O)CC2)C)ccc(F)cc1 c1(C(c2nnnn2CC(F)F)N(c2ccccc2I)C)cc(C(=O)OC)cn1C CC1CC=CCC1NC(=O)C(c1ccco1)NC(=O)C=CC(F)(F)F CCCCCCC(C)C(=O)NC(Cc1ccccc1)CCOC(F)(F)F C1(C(N2CCCC(C(C)NC(Cc3cc(CC)no3)=O)C2)=O)CCC(=O)NC1=O c1(C(=O)NCC2C(NC(c3cnc(C(=O)OC)s3)=O)CCC2)ccc(C)cn1 CCC(CC(=O)NC1CN(C(C2CCC=CCCC2)=O)C2(CCC2)C1)CC(C)C c1(OC)ncc(Cl)cc1C(=O)NCC(C)CNC(C1CC(N2CCOCC2)C1)=O C1(C)(NC(CSCC=C)=O)CCCN(C(c2nc(Br)c(C)s2)=O)C1 C12(NC(c3cnc(SC)n3C)=O)CC3CCC(C1C2)N3C(C1(C)CCC(=O)C1)=O Cc1cn2cccc(C(=O)NC(C)CC(C)NC(=O)C(C)Cc3cnc[nH]3)c2n1 c1(N(C2c3nc(oc3)NC2=O)C)ccccn1.C(=O)(CC1CCO1)OC c1(C(=O)NCCNC(c2c(CC)noc2)=O)ccc2c(ccn2C)c1 c1(C(N2CC(C3(NC(C(C=C=C)C)=O)CC3)C2)=O)cn2c(Br)c(C)nc2s1 N1(C(c2scc(C(N)=O)c2)=O)CCC(CNC(=O)C(F)=CCCF)CC1 Cc1scc(C(N2CCN(C(=O)COCC3CCCO3)CC2)=O)c1C1CC1 Cc1cc(CC(=O)NC(CNC(C2CCOC2c2ccnn2C)=O)C2CC2)n[nH]1 c1(C(=O)NCC2N(C(C(C=C)O)=O)CC(F)(F)C2)c(C)cc(C#N)cc1C C1(N(C(C=CC)=O)C)CCCC(N(C)C(c2cnc(-c3cccs3)o2)=O)C1 C1(CC(C)C)(C(=O)NC(C)Cc2nc(-c3ccccc3)no2)CCCNC1 c1(C(c2n(CC(=C)C)nnn2)NCC2(CCO)CC2)cnn(C)c1C(F)(F)F C=CCC(C)(CC)C(=O)N1CC(CNC(c2csc(C)n2)=O)C(F)(F)C1 N1(C(C2(CCC=C)CN(C(=O)C(=O)CCCC)C2)=O)CCN(C)CC(C)C1 c12ccc(cc1)NC(=O)CO2.C1(C(=O)OC)(CF)COC1 c1(C(=O)NCCOC2CCN(C(C(C)SC)=O)CC2)ccnc(O)c1Br C1(C(=O)Nc2n(C)nc(Br)c2)CC(F)(F)CN1C(c1cc(F)ncc1Br)=O Cc1cccc(F)c1CC(=O)N(CC(C)N(C(=O)COc1ccccc1F)C)C CC(C)(CN(C(=O)CC1CCN(CCc2ccccc2Cl)C1)CCO)C(=O)O c1(C(C)C(=O)NC2CC(CNC(C3CCC(C)O3)=O)C2)ccc(Cl)c(Cl)c1 C(=O)(C1=CCCSC1)NC(c1ccnn1C)C(=O)Nc1c(CC)cccc1 C1(CNC(C2CCC(CC)O2)=O)CN(C)CCN1C(=O)CC12CCC(CC1)OC2 c1(C(=O)NCC2CN(C(c3ccc(C)nc3C)=O)C3C2C3)ccc([N+](=O)[O-])cn1 N1(C(C(=O)N(CC(=O)NCCC(N)=O)C)=O)CCC(NC(=O)CN(C)C)CC1 C(=O)(C1CCc2c[nH]nc21)N1CC(NC(c2c(N)sc(C)c2C)=O)CC1(C)C C(C(N=[N+]=[N-])C(=O)N1CCC(NC(c2ccc(OC(C)C)nn2)=O)C1(C)C)OC c1(-c2nn(C)c(Cc3cccc(O)n3)n2)ccc(Cl)cc1O C1(C(=O)NCC2CC(NC(C3CC(F)(CO)C3)=O)C2)CCCCCC1(F)F c1(C(=O)NC2(C)CN(C(C3CCn4nncc4C3)=O)C2)cc2cccc(Cl)c2s1 C1(c2cn(CC(CC)C)nn2)CN(C(=O)CCCOC(C)=O)CCN1C O(NC(=O)C(CCC=C)CC(C)C)C(C(=O)NCC(CCCC=C)(C)C)CC N1(C(COCCC=C)=O)Cc2n[nH]cc2C1C(=O)NCCCc1cc(C)[nH]n1 c1(C(=O)NCC2CN(C(CSC)=O)C(C)C2)ccc(C)c(O)c1 C(C(C)(C)C(=O)NC1(c2cn(CC3CCCO3)nn2)CC1)N(C)C Cn1cc(C(N2CC(F)(CNC(C3CCC(C)(C)OC3)=O)C2)=O)n(C)c1=O c1(C(N2CC(NC(C(C)C#N)=O)C(CC(C)(C)C)C2)=O)cc2cnccc2o1 c1(C(=O)NC(CNC(c2cnc(C)o2)=O)(C)C(C)C)cccn2ncc(Br)c12 c1(C(N2CCCCC2C(O)CC(F)(F)F)=O)cccc(Br)c1Cl C12(CNC(c3ccns3)=O)CC1CN(C(=O)Cn1ncc(Br)n1)C2 c1(C(=O)OC)cc(C(N2CC(O)CC2C(=O)Nc2sccc2CO)=O)cc(F)c1 Cc1ccc(C(=O)NCCNC(=O)C(c2cccc(Br)c2)(C)C)c(N)c1 C(C1CC(C)Oc2ccccc21)NC(C1(c2c(OC)cccc2)CC1)=O C1(O)(CC(N2C(C(=O)NCc3ccc[nH]3)CC2)=O)CCCOC1 C1(C(N(CCN(C)C)CC)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O C1(CC(=O)NC2CN(C(C(C)(C)OCC)=O)C2)CC(F)(F)C1(F)F C(=O)(C(C)(C)CCC#N)NCC1(CCNC(C(n2c(C)cc(C)n2)C)=O)CC1 Cc1nc(N2CCC(C(C)NC(C3(O)CC3)=O)CC2)c2scc(C)c2n1 N1(C(CC2C=NN(C)C2=O)=O)CCCC(F)(C(=O)NCC(C)(CO)CO)C1 c1(C(N(CCN(C(C(C=CCCC)O)=O)C)C)=O)csc(C)c1Br c1(CN(C(=O)C(C)(C)CCl)C)ccc(CCCCc2cc(C(C)C)[nH]c2)cc1.N C(=O)(CC1=CCCCC1)NC(C1CN(C(C2(C(=O)NC3CC3)CC=CC2)=O)C1)C C1(C)(C(=O)NC(C2(CNC(=O)C(C)N(CC(F)(F)F)C)CC2)C)C=CCC1 C(=O)(C(C#N)C(C)(C)C)N1C(C)CC1C(N1CC(c2ncccn2)C1)=O C=CCC(CNC(=O)CCC(C)(C)OC)C(=O)NCC(C)CC(C)(C)C C(=O)(C(C)(C)CCC(=O)NC1COCC1CNC(C1CN(CC(C)C)C1)=O)OC N1(C(CC2(C)CCOCC2)=O)CC2(C1)SCCC2NC(c1cscc1Cl)=O c1(C(=O)NC23CC(C(=O)NCC4CC4c4ccsc4)(C2)C3)cc2ccccc2[nH]1 CC1CC(C)N(C(=O)CSC2CC2)CCN1C(=O)C#CC1(C(F)(F)F)CC1 N1(C(C2CC(NC(C=CC3(C)COC3)=O)C(O)C2)=O)CCCCC(F)(F)C1 C1(CNC(c2c(C)n(C3CCOC3)nn2)=O)CCC(C)CN1C(=O)CC1CC1 C1(COC)(NC(c2c[nH]c(C)c2)=O)CCCN(C(=O)C(C)C2CC2)C1 C1(CN(C)C(C2COC2)=O)CCN(C(c2sc(Br)cc2F)=O)CC1 C1(CN(C(C(CC=C)c2nn[nH]n2)=O)C)CCC(C)(C)CC1 C1(NC(c2ccn(CC#N)n2)=O)COCCN(C(=O)Cc2ccc(F)cc2Cl)C1 CC1(C)CN(C(C2CCCC(F)C2)=O)CC1NC(C1C2CCC(=O)C12)=O Cc1nccnc1C(C)NC(=O)C(C1CCCN(C(=O)CC2(C)CC2)C1)C C(C(=O)N1CCN(C(c2cc3sccc3[nH]2)=O)C(CC2CC2)C1)(C(C)(C)C)SC Cc1cccc(C(C(c2ccccc2)CC#N)CNC(=O)N(C)C)c1 C1(C2CCN(C(C3CCCS3(=O)=O)=O)CC2)(NC(c2c(C)nn(C)c2)=O)CC1 c1(SCC(=O)NC2C(C(=O)Nc3cc(OC)ns3)C2)ccc2c(c1)OCCO2 N1(C(CS(CC)=O)=O)CCC(C2CC2)(CNC(c2conc2C2CCC2)=O)C1 C1(NC(Cc2c(C)nc(Cl)cc2)=O)CC2CC1CN(C(=O)CCc1ccoc1)C2 C(=O)(C(C)(CCc1ccccc1)N(C)CCOCCOCC1CC1)OCC c1(C(C(=O)NCC2CC2)N(C)CC2CCN(C)C2)csc2c(F)cccc12 c1(OC)cccc(NC2=CCCCC2)c1.C1C(=O)OCCN1C(C)=O C1(C(=O)NCC2(CC3CC3)CCC2)CC2C=CC1N(C(=O)C=Cc1ccncn1)C2 C(c1cocn1)=CC(=O)N(CC(C)NC(C1CC2(CC2)C1)=O)C CCCCC(F)C(=O)N1CC2CC1CN2C(=O)C(CN(C)C)C(C)C c1(C(=O)NC(CC(=O)NC(CC)CCO)COC)nnc(O)nc1O c1(C(N2CCN(CC(=O)Nc3ncc(Br)s3)C(=O)C2)=O)ccc(Br)c(Cl)c1F c1(OC)ccc(CC(=O)NC2CC23CC(NC(C2CCCO2)=O)C3)cc1O c1(C(N(C(CC)CC(=O)NC2CCCC2OC)C)=O)coc2c1COC2 O=C1C2CC3C(C2)C13C(=O)NC(C(=O)NCc1ccc2c(c1)CC2)C1CCCO1 Cc1cnc(OCC(=O)OC2C=CCC2)nc1 N1(C(CC2CC(CC)C2)=O)CCC(C(=O)NCC(C)CC2CC2)(CC)C1 n1(CC)nccc1C(=O)NC1(CNC(=O)CN2CCC(C)C2)CCC1 C(=O)(N=c1nco[nH]1)NC1(COC)CNCCO1 c1(OC)ccc(C2CCCN2C(c2ccccc2SCc2cccs2)=O)cc1F C1(CC(=O)NC2C3CN(C(c4c(CC)nns4)=O)C2C3)CC2(CCCC2)CO1 c1(SC)ncc(N)c(C(=O)NCC2CCCC2NC(c2cc(C)ncn2)=O)n1 C=C(Cl)CC(C(=O)NCC(CO)N(C)C)NC(C1CC1c1cccs1)=O c1(C(N(C)CC2CCCN(C(C3(C)CCCCO3)=O)C2)=O)nccc(N)c1Cl N(C(=NCCC1CC(F)C1)NC1CCC1)C(COC)C C1(C(=O)OC)CC12CN(C(=O)CC(C)CNC(=O)CNC(C)=O)C2 C(=O)(C1CCCc2cccnc21)NC(CNC(CCC(=O)NCCC)=O)C(C)C C(c1ccc(OC(F)F)c(OC)c1)=CC(=O)NC1CCN(CC(=O)NCC)CC1 C1(NC(c2cccc(N=[N+]=[N-])c2)=O)CCC2CN(C(C3C=CCC3)=O)CCC2C1 CC1C(NC(C2CC(N(C)C)C2)=O)CCCN1C(c1cc(N(C)C)ccc1N)=O C1(C(N(CC(=C)C)CCOC)=O)CCCN1NC(=O)CCC1CC1C Cc1ccc(Br)c(F)c1C(=O)NC1(CNC(C2(C#N)CCC2)=O)COC1 c1(C(=O)NCC2CC(NC(c3c(NC)snc3C)=O)C2)nccn2cc(C)nc12 C1(NC(C2(NC(=O)C=CCO)CC(O)C2)=O)CC2(CNC(=O)O2)C1 c1(OC)ccc(F)cc1CC(N1CCCC(NC(C2C3COCC23)=O)C1)=O c1(C(=O)Nc2ccc(CN3C(=O)CSC3=O)cc2)ccc2nccc(Cl)c2c1 N1(C(C(n2ccc(C)n2)C)=O)CC(NC(C2CC2c2oncc2C)=O)C2(CC2)C1 O=C1NCC2(CCCN(C(=O)C3=CCNC3)C2)O1 c1(N2C(CNC(C3(CO)CC3)=O)CC3(CC3)C2)cc(C(F)(F)F)nc2ncnn12 C(=O)(CCCCC(N)=O)NC(C)CN(C)C(c1cc(-c2ccco2)c[nH]1)=O c1(C(=O)NC(CC(=O)NC2CC23CCCCC3)C2CC2)c(F)cncc1F C12(NC(C3(C(F)(F)F)CC3)=O)CC(CNC(c3ccc[nH]3)=O)(C1)OC2C.CCC CC1(C(=O)NC2CN(C(=O)CN3CC(=O)NC3=O)CCC2F)CCC(F)(F)CC1 c1(OC)ccc(NC(C2CC(NC(c3cccc(C)c3)=O)C2(C)C)=O)cc1C c1(C(=O)NCCC(C)N(C(C(C=C)c2ccccc2)=O)C)ccccc1C(C)C N1(C(C(C(C)C)NC(CCOC(C)=O)=O)=O)CC2CC1CN2C(C)C C(=O)(C(C)(C)CC(=O)N1CCCC(NC(=O)CNC(=O)C2CC2)C1)OC CC1OCCCC1C(=O)NCCCN(C(=O)CCOC1CCCC1)C C12(NC(c3n(CC)c(O)nc3)=O)CCC(C1)N(C(=O)COC1CCC1)C2 CC(CC(C)(F)F)C(=O)NC1CCC1NC(=O)CCc1c(F)cccc1Cl c1(CN(C2CCCN(C(=O)Nc3cn(C)nc3CCC(=O)O)C2)C)ccc(F)cc1 c1(C(=O)NC2CC(C)(NC(C(CCCC)C)=O)C2)ccc(OC)c(F)c1N c1(C(=O)NC(CNC(C2C(C)CCC2)=O)(C)C)cc2ncccc2cc1Cl CC(C)CC(CNC(C1(CCF)CCC1)=O)NC(C1CC1(C)C)=O.C1(C)CC1 C(=O)(CCCCCCn1cc(C2CC2)nn1)NCCOC1CCCC(C)C1 NS(=O)(=O)c1ccc(C(=O)NCC(CO)NC(=O)Cn2cnnn2)o1 N1(C(C=CCC)=O)CCCC(O)(CNC(=O)C(c2c(Cl)cccc2Cl)C)CC1 C(=O)(C1CCCNc2ccccc21)NCC1N(C(c2cc(C)sn2)=O)CCC1 c1(C(=O)NOCCO)n[nH]cc1CNC1(C2CCCCO2)CC1 c1(CCC(=O)NCC2(NC(C34CC(C)(C3)C4)=O)CCOCC2)ccc(F)cc1Cl N1(C(CCC=C)=O)CC(CC(=O)NC2(CN3CCCC3)CC2)C2(CC2)C1 c1(C(=O)NC2CCC(NC(C(C)OCC)=O)CC2)c(C)[nH]c2ccc(Cl)cc12 Cc1cc(C(N2CC=C(C(=O)Nc3cnn(C)c3)C2)=O)nnc1C N1(C(c2n(CC#C)ccc2)=O)C(C)CN(C(=O)C=C(Cl)Cl)CC1C N1(C(C2C(C)(C)CO2)=O)CC(CO)C2(C1)CN(C(c1cncc(Cl)c1Cl)=O)C2 c1(CC(C)(C)C)ccc(C(=O)NCCC(O)CNC(=O)C(CO)N(C)C)cc1 c1(CCCC)nc(C(=O)NCC2CCN2C(c2ccsn2)=O)cs1 C(=O)(C1=C2CCCN=C2NN1)N1CCN(C(Cn2ncn(C)c2=O)=O)CC(O)C1 N12CCOC3CC(CCC13)C2=O.C1(NC(C)=O)CCOC(C)(c2ccccc2)C1 c1(C(=O)NC(C(=O)NC(CCC)C(=O)NC)CN(C)C)cc(C)n(C)c1C C=CC1(O)CCN(C(C2CCCN(C(c3cncc(OC)n3)=O)C2C)=O)C1 C1(CCC)CN(C(c2c(Cl)c(CC)nn2C)=O)CCN1C(=O)CCOC C1(OCCCNC(C2C(C)C2C)=O)CCN(C(C2(N(C)C)CCC2)=O)CC1 c1(C(=O)NCCCOCCNC(C(C(CC)CC)C)=O)n[nH]c2nccc(Cl)c12 C=CCC(C)C(=O)NCC1(OC)CN(C(c2ccc(CN3CCCC3)cc2)=O)C1 c1(OC)cncc(CNC(C2CC(C)N2C(c2cccc(CO)c2)=O)=O)c1 C12(CNC(CSCCC#N)=O)CCCC(CN(C(c3ccc([N+](=O)[O-])s3)=O)C1)C2 C1(NC(C(COC)O)=O)CCCCC1CNC(C1CCCC1)=O c1(OC)ccc(C(c2cn(CC(O)CCC3CCCOC3)nn2)OC)cc1 N1(C(c2c(CC)[nH]cc2)=O)CCCC1(C)CNC(C1(C)CNC(=O)C1)=O c1(C(=O)NC(CNC(C(C2CC2)OC)=O)(C)CO)cc(C)ccc1Br c1(OCC)ccc2c(c1)C(C(=O)NCCNC(=O)Cc1nc(=N)[nH][nH]1)CC2 C(=O)(CC1=CCCCC1)NC(CC(C)C)CN(C)C.C12(CC1)C(=O)NCC2 C1(NC(CNC(COCCOCC)=O)=O)CN(C)CCC1O C1(NC(C2CC(CCC)C2)=O)CN(C(=O)COC2CC2)CC1C1CC1 c1(OC)ccc(F)c(C(=O)NC2CC2NC(=O)C(O)C(C)(C)C)c1F Cc1cc(C(=O)NC(CC2CC2)CC(=O)NCCCCN2CCC2)c(C)o1 CC1(NC(=O)C(=O)NCC(F)(F)F)CN(C(C2CCC2(F)F)=O)C1 N1(C(C(N2CCNC2=O)C)=O)CCC(CF)(NC(c2cncc(CO)c2)=O)C1 Cc1cc(C(=O)NC(C(=O)NC(C)CN(C)C(C)C)C2CC2)nn1C C(=O)(CC(C)(C)CC(C)=O)N1CC2(CN(C(C3CCC(CC)O3)=O)C2)C1 c1(C(=O)NC2CCCC(CN(C(c3c(C)nns3)=O)C)C2)cc2n(n1)CCC2 c1(SC(C)C(N2CCC(NC(=O)CC3CCCCCO3)CC2)=O)ccc(Cl)cc1 C1(C(=O)NCC(CNC(COCCOCC)=O)OC)CCOCC1(C)C c1(NC(CC2CCN(Cc3ccc(OC)cc3)C2)=O)c(C)nn(C(F)(F)F)c1C CC1(C)CCc2c(C(N3CCCC(CNC(=O)Cc4cscn4)C3)=O)n[nH]c2C1 C=CCC(C)(C)CC(=O)N1CCC(=CCNC(c2nnc(C(C)(C)C)s2)=O)CC1 c1(C(=O)NC2CC(F)(CNC(C(F)OC)=O)C2)nnn(-c2ccn(C)n2)c1C C12(CCCC1)C(=O)N2.C(=O)(C(=O)N1CC(C(N)=O)C1)N(C)C N1(C(CC(C)C)=O)CCOCCC1C(=O)NCC(C)(O)C1CCC1 C(=O)(C1=CC2CCC=CCCC12)N1CC(Nc2nccc(SC)n2)C(C)C1 N1(C(CCc2ccc(OC)cc2C)=O)CC(NC(=O)C(N)=O)Cc2ccccc21 c1(C(N2CCN(C(c3c(C(C)C)onc3)=O)CC2)=O)cc2c(F)ccc(Cl)c2[nH]1 Cc1ccc(F)c(C(=O)NC23CCCC(NC(=O)C(C)CS(C)=O)(C2)C3)c1 C(=O)(C1=CS(=O)(=O)CCC1)NC1CC(NC(c2c(C)nc(CC)s2)=O)C12CCC2 N1(C(C)C)CCC2(CC1)CC2(C)C(N1CCN(C2CCOCC2)CC1)=O c1(C(=O)Nc2scc(-c3c(F)ncc(OC)c3)n2)nn(C)cc1[N+](=O)[O-] c1(CN2CC(=O)N(CCCN(CCOCC)C)C2=O)c(F)ccc(Br)c1Cl c1(C(=O)NCc2cn(CC(=O)NCC3CNC(=O)C3)nn2)ccncc1F C1(=O)C(F)CC2CN1C2.N1(CC)CCC1CNC(C1(n2cnnn2)CC1)=O Cc1[nH]c(=NCc2cccc(O)n2)sc1C(=O)Nc1cccc(Br)n1 Cc1nsc(C(N2CCC2CNC(C2COCC2(C)C)=O)=O)c1N N1(C(COCCSC)=O)CCC(F)CC1C(N1CCSCC1C)=O C1(CC)CCCN(C(c2cnc(C)nc2C)=O)C1C(=O)NCCC[Si](C)(C)C C1(CC)CC(CC(=O)NC2C=CCN(C(=O)CC#N)C2)CCO1 CCCC(CCCO)C(=O)NCC1CCCC1NC(c1cc(OC)ncn1)=O c1(NC(C(CC)(C)O)=O)ccc(NC(=O)CCC(=O)N2CCOCC2)c(F)c1 N1(C(CC=CC=C)=O)CC2CCC2(NC(c2ccnc(CC)c2)=O)C1 C1(C(N2CC(OC(=N)O)C2)=O)(NC(C(C2CCC(=O)N2)C)=O)CC1(C)C N1(C(C=C2CCC(C)CC2)=O)CC2CCC1C(CNC(C1CCC(O)CC1)=O)C2 c1(C(=O)NCC2N(C(C(C)OC)=O)CC(F)(F)C2)c(C)sc2ccccc12 Fc1ccc(C(c2nnnn2C2CC(F)(F)C2)NCCc2ncccn2)cc1Cl C(c1ccc2occc2c1)=CC(=O)NCC(CNC(C=C(C)C1CC1)=O)(C)O Cc1cccc(C(=O)NCC(CC2CC2)C(=O)NC(Cc2cnc[nH]2)CO)c1N c1(OC)cc(C(=O)NC2CCC(NCc3c(F)cccc3Cl)C2)c(OC)cc1Cl c1(C(N2CCCC(O)(CNC(CCOC(C)C)=O)C2)=O)cn(C)c2ccccc12 c1(C(C(=O)NC(CC)C)N(C)Cc2c(I)cnn2C)c(C)nn(C)c1Cl C1(CC)CN(C(c2cnc(O)cc2C)=O)CCC1NC(=O)CCc1ccco1 C(=O)(CCCN=[N+]=[N-])N(CC(O)Cc1ccccc1F)C(C)(C)C Cc1cc(C#N)nc(N2CC(CNC(=O)Cn3ncnn3)CC2C)n1 CC(Cc1cnc[nH]1)C(=O)NCC(C1CCOC1)NC(c1ccn(C)n1)=O C(=O)(C(CC(C)C)CC(C)C)NCC(CC)NC(C1Cc2cc(F)ccc2O1)=O c1(C(=O)OC)ccc(N2CCN(CCCOC3CCOC3)CC2)nc1C Cc1[nH]c(=N)sc1CC(N1CC=CC(NC(c2ccc(C(N)=O)[nH]2)=O)C1)=O CC1CC(C(N2CC(c3ccccc3)(NC(C3CC4CCC3C4)=O)C2)=O)CCO1 Cc1ccsc1CC(=O)NC(CN(C)C(C1CC1F)=O)Cc1ccccc1 c1(C(CC)NC(C2CCN2Cc2noc(C)n2)=O)cccc(C(F)(F)F)c1 C1(C2CCCCC2)(C(=O)NC(CCNC(C(C(C)C)OC)=O)C(C)C)CC1 N(S(N)(=O)=O)CC(=O)N(CC(C)NC(c1cnc[nH]1)=O)C N1(C(C(C=C)(C)O)=O)CCC2(CCC2)C(NC(c2oc(CC(C)C)nc2C)=O)C1 c1(C(=O)OC)c(C(N2CC(n3cc(CNC(=O)CNC=O)nn3)C2)=O)n[nH]c1C C1(NC(c2c(C)cc[nH]2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC1C C1(CCC(=O)N(CC(CC)NC(c2c(CC)nns2)=O)CC)CCC(=O)NC1 c1(OC)ccnc(OC)c1C(=O)N(C1CC2CC1N(C(=O)C(C#N)C(C)C)C2)C CCC(C#N)(CC)C(=O)N1CC(NC(=O)C(C)Cc2ccnn2C)C(O)C1 CCC(CNC(c1c(Br)c(C)nn1C)c1nnnn1C1CCOC1)(CC)C(N)=O c1(C(=O)NCC(C)(CO)NC(C2CCC(=O)N2)=O)cccc2c(O)nncc12 c1(CCC(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2O)nc2ccccc2[nH]1 c1(C(N(CCC(c2cccs2)NC(C(C2CC2)SC)=O)C)=O)csc(=NC)[nH]1 C(=O)(C(F)n1ccnc1)NCC(=O)NCC(c1ncc[nH]1)O N#Cc1ccc(CC(N2CC3CC3(CNC(=O)CC3NC(=O)NC3=O)C2)=O)cc1 C1(C(c2n(CC)nnn2)NCC2CC(CC(C)(C)C)C2)C(C)(C)C1(C)C c1(C(N2CCC(C(N(C(CC(=O)NC)C)C)=O)C2)=O)cccc(C)c1C N1(CCNC(N(CC(CC)O)C)=O)CCOC(C)C1 CCC(C)C(CC(=O)NC1CCCC(O)CC1)NC(c1ccnc(OC)c1)=O c1(C(=O)NCCCNC(C2CCC(C(N)=O)O2)=O)ccc([N+](=O)[O-])s1 c1(NC(C2(CNC(c3cnc(Cl)nc3)=O)CC2)=O)cnn2ccc(Cl)nc12 N1(C(C(CC2CC2)NC(C(n2c(C)ccn2)C)=O)=O)CC2(C1)NC(=O)NC2=O Cn1nc(C(=O)NC2COCCC2NC(=O)Cn2cnnc2)cc1C(F)(F)F C=CCCC(C)(C)C(=O)NCc1cccc(NC(C2CCN(C)S2(=O)=O)=O)c1 C1(COC)CN(C(c2ccc(Br)cc2)=O)CCN1C(=O)COCC(C)C C1(n2cc(-c3c(C)nsc3)nn2)CC2(CC2)CN1C(C1CC(C)(C)C12CC2)=O Cc1nc(C2CCCC2)sc1C(=O)NCC1CC(NC(C2CN(C(N)=O)C2)=O)C1 CCCCCCC(CNC(c1ncoc1C(F)(F)F)c1nnnn1CCC1CC1)CC c1(C(N(CC(=O)N(CC(F)F)CCOC)C2CC2)=O)nc(C)sc1C N1(C(CCCC(=C)C)=O)CCC2(CC1)CC2NC(=O)CCN(C)CCO c1(C(=O)NC2CC(C)(NC(CCC(C)(C)C#N)=O)C2)cc2ccncc2cc1F c1(C(N(CC(CNC(C(COC)(C)C)=O)C)C)=O)cc(OC)ccc1F c1(C(N2CCCN(C(C(C)NC(=O)NC)=O)CC2)=O)ccc2nn[nH]c2c1 c1(CC=C(C)C)cc(C(=O)NC2CCN(C(C3(C)CC3C)=O)CC2O)ccc1F C1(C)(NC(C(CCC)O)=O)CCN(c2nc(OC)cc(OC)n2)CC1 CC(C)C(CNC(=O)CC1CCC(=O)N1)N=c1[nH]c2cc(F)ccc2o1 C1(C(=O)NCC2CC[Si](C)(C)C2)CC(C)(C)S(=O)(=O)C(C)(C)C1 N1(C(C2C(C)(Br)C2)=O)CCC(c2cn(Cc3cc(C4CC4)no3)nn2)C1 C(C(CC(F)(F)F)NC(c1c[nH]cc1Br)=O)NC(CCCN(C(C)C)C)=O O=C1CN(C(=O)NC2CC2C(=O)Nc2ccc(C(F)(F)F)cc2)c2ccccc2N1 c1(C(N(CC(CN(C(C(CCC)C)=O)C)O)C)=O)cccc(C#N)n1 c1(C(N(CC(N2C(CC)C(O)CC2)=O)C2CC2)=O)c[n+]([O-])c(C)cn1 c1(-c2c(CN(CCN(C)C)C)cc(Cl)cn2)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NC(C(=O)NC(c2n(C)ncc2)CO)C2(C)CC2)cc(Cl)cn1C c1(C(N2C(C(=O)Nc3cnn(CC)c3)CC(=C)C2)=O)cnc(Cl)cc1OC C1(C(=O)NCCN(C)C(C2CC(=O)N(C3CCCC3)C2)=O)CCC2(CCC2)CO1 C1(=O)C(C(C)O)N1.N1(CCC)CCC(C(=O)N(C2CCCN2C(C)C)C)C1 Cc1cn2c(n1)C(C)CC(C(=O)NCC1CN(C(c3cnn[nH]3)=O)CCN1C)C2 c1(C(C(=O)NCCN2CCC(O)CC2)Nc2ccco2)ccc(F)c(Cl)c1 C(=O)(CCC(=O)NN(C)C)N1C(C)CN(C(c2cnc(SC)n2C)=O)C(C)C1 Cc1nc(C)c(C(=O)NC(c2nc(C(F)(F)F)n[nH]2)C)c(C)n1 c1(C(=O)NCC(C2CCCC2)NC(c2c(CC)occ2)=O)ccn2ccnc2c1 C1(N(C)C(c2ccc(C3CCC3)nc2)=O)CCCC(NC(=O)Cc2cscn2)C1 N1(C(COCCNC(c2c(C)nc(C)s2)=O)=O)CCN(C)C2(CC2)C1 C12(NC(=O)COc3cccnc3)COCCC1CN(C(=O)CN1CCCC1)C2 Cc1c(C(=O)NCCC(O)CNC(=O)CC2CCCOC2)sc2[nH]cnc(=O)c12 N1(C(C2CCCOC2)=O)CCN(C(=O)CCc2cnco2)C(CC2CC2)C1 C12(C(=O)NC3CC(C)N(C(=O)COCc4ccncc4)C3)CCCC(C1)OC2 CC(CC(=O)NC1CCN(CCNC(=O)C(c2cncnc2)C)CC1)C(C)(C)C C(C(CO)(CO)NC(=O)C(F)CC1CCCC1)N(C(=O)CNC(C1CCC1)=O)C c1(CCC)cnnc(C(N2CC(CC(C)(C)CNC(C3CC(CC)C3)=O)C2)=O)c1 c1(C(N(C(C)C)CCNC(=O)C(c2ccccc2)F)=O)cncc(C(F)F)c1 O=C(C#CC1CCCC1)N1C(C(=O)Nn2cnnc2)CCC1CF C(CCCC(=O)N(CCCCC(=O)NCCN(C)C)C)OC CC(C)(C)C(=O)NC1CC1C(=O)NCC1COC(=O)N1 c1(C(N2CCC(N(C(=O)C(F)C(C)C)CC)CC2)=O)cncc(Cl)c1C C(C(=O)N1CCC(C)C1CNC(c1cc(C(N)=O)c[nH]1)=O)(C(C)C)NC(=O)OC Cc1noc(C(=O)NC(CNC(=O)CCC2CC2(F)F)C2CC2)c1C C1(NC(=O)OC(C)(C)C)CCN(Cc2cccc(CO)c2)CC1CC#N C(C1=NOC2CN(C(c3nocc3C(C)(C)C)=O)CC12)NC(COCCC=C)=O C(=O)(C(C)(C#N)CC)N1CCC(C(C(=O)N(CCN(CC)CC)C)C)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(C(=O)NCc2cn[nH]c2)C(C)(C)C1 c1(C(N(CC(CNC(CC(C)c2ccncc2)=O)O)C)=O)ccc(=O)n(C)n1 C(=O)(CCCC(C)=O)NCC1(C(=O)NC(C)COC(F)(F)F)CC(=C)C1 N1(C(C(c2cccc(C(F)(F)F)c2)(C)O)=O)CCCNC(=O)C1 C(C(=O)NC1CCN(c2cc(C)ncn2)C1C)(C(C)C)NC(C)=O c1(SCCCCN(C(=O)CCN2CCOC2=O)CCOC)c(C)noc1C c1(C(=O)NCC(C)(C2CC2)NC(C(C)n2cccn2)=O)ccc(C#N)[nH]1 C1(NC(C2C(C)(CC)C2)=O)CC2(CCN(C(=O)CC3=CCCC3)CC2)C1 C1(COCC)(CNC(CNC(=O)CSCC2CCCO2)=O)CCCCC1 N1(C(C(C)NC(=O)NC)=O)CC2CCC(C1)C(NC(=O)CC1CCC(=O)C1C)C2 N1(C(CC2N(C(CCC(CC)OC)=O)CCOC2)=O)CCCNC(=O)C1C N1(C(C(C(C)C)C2CCC2)=O)CCC(C)N(C(C2SC3C=CC2C3)=O)CC1 Cc1cc(C(C(=O)NCC(C)C)N(CCC(=O)N(C)C)C)c2ncccc2c1 N1(C(c2c(C)cco2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2(CC2)C1 N1(C(C2C(C)C2C)=O)CC2CCN(C(c3cc(Cl)c(Br)cn3)=O)CC2C1 c1(CNC(C(C2CCCCC2)C)=O)cc(C(=O)N(C2CC(C)(C)C2)CCO)cs1 CC(C)CC(C(=O)NCC1(F)CCC(NC(c2ncoc2C2CC2)=O)C1)C(C)C C1(OC)(CO)CCN(C(C2(N(C)C(C3CC(C)CCO3)=O)CCC2)=O)C1 N1(C(CC(C)OC)=O)CCC2(CC1)C(NC(=O)CC1(CO)CC1)CS(=O)(=O)N2C N1(C(COCCNC(c2c(CC)cncc2)=O)=O)CCCC2(CC1)CC2 c1(C(=O)NCC(CCCC)NC(=O)CCC(C)(C)C)cnc(N)c([N+](=O)[O-])c1 CCC(CC(=O)NC1CC2CC(NC(c3ccoc3Cl)=O)C2C1)CC(C)C C1(C(C)C)CCCN(C(=O)C(N2CCCCC2C(O)N(C)C)=O)CC1 C(S(=O)(=O)CCCC(=O)NCCc1ccco1)c1ccc(C)o1 C1(C(N(CC=C)Cc2cccc(-n3cncn3)c2)=O)Oc2ccccc2OC1C N1(C(C2N(C)CCCC2)=O)CC2(CCC2NC(=O)CN2CCCCC2=O)C1 C1(CNC(C2CN(C(C)C)C2)=O)CCOC1C(N1CC(N2CC=CC2)C1)=O C(N=c1cccc(S(=O)(=O)N2CCOCC(C)C2)[nH]1)c1c(OC)ccnc1 N1(C(C(CC)n2cccn2)=O)CCOCC(NC(C2CC(C)(F)C2)=O)C1 c1(OCC)n[nH]cc1C(=O)NC1(CCNC(=O)Cc2cnnn2C)CCC1 C(CC(=O)N1CC=CC(NC(C2(OC)CCC2)=O)C1)(C(C)C)OCC c1(C(N2C(C(=O)NC(c3ccc(F)cc3F)CO)CC2)=O)c(Cl)cc(Br)cc1Cl C1(CC(C)NC(c2cncc(F)n2)=O)CCN(C(=O)Cc2cc[nH]n2)CC1 C(=O)(C1=CCN(C(=O)CC2CC2(C)C)CC1)NC(CCOC)C N1(C(C2CCCCO2)=O)CCCN(C(C2CC3CC3C2)=O)CC1 C1(OC)CCN(C(c2cncc(F)c2Br)=O)C(C2CC2)C1 C(=O)(CCCC1OCCO1)NCCC1(NC(C(C)SC(C)C)=O)CCC1 c1(C(=O)NC2CCCN(C(CCCOCCC)=O)C2)ccc(O)c(CO)c1 c1(C(N2CCCC(NC(C3C(C)CC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1Br c1(C(=O)NCCN(C(c2ccc(OC(C)C)o2)=O)CC)ccc2n[nH]cc2c1 N1(C(C23OCC(C)(C2)C3)=O)CCCC(F)(CNC(c2cscc2F)=O)C1 c1(C(N2CCN(C(C(c3scc(C)n3)C)=O)C(C)C2)=O)ccc(N)c(Cl)c1O C(=O)(CCCC(C)(F)F)N1C(CCCNC(c2c(NC)ccc(Cl)c2)=O)CCC1 C(CCCCC(=O)NC(C1CC=CCC1)C(=O)NC1C(O)C2CCOC12)OC C(=O)(C1CCCc2cncn21)N1CC2CCC(NC(Cc3c(C)non3)=O)C2C1 S(=O)(=O)(c1ccc(Br)cn1)N1CC(NC(C2(C(=O)OCC)CC2)=O)C(C#N)C1 Cc1ccc(S(=O)(=O)NC(=O)CCc2ccccc2N)cc1C C1(C#CC(=O)NC2(C)CCN(C(=O)COC(F)F)C2)(CC)CC1 C=CCC(C(=O)N1CCCCC(N(C)C(c2nnn3c2CSCC3)=O)C1)C(C)C C1(C(C)C)CN(C(C2CCC(N(C)C)CC2)=O)CCN1C(=O)C(=O)N(C)C C1(NC(COC2CCC(C)CC2)=O)CC2(CCCN(C(c3cc(Cl)no3)=O)C2)C1 C(=O)(C(CNC(C1CC(F)(CF)C1)=O)C(C)(C)C)NCCc1n(C)cnc1 c1(C(=O)NC(C(C(=O)OC)(C)C)c2ccccc2)ccc2nccc(=O)n2c1 N1(C(CC(C(C)C)(F)F)=O)CC2CCCN(C(c3cn4c(n3)COCC4)=O)C2C1 CC1CCC(NC(c2ccc(C(F)F)o2)=O)CN1C(c1ncc(Cl)nc1Cl)=O c1(C(C)C)c(C(=O)OC(C)(C)C)cnn1-c1ccccc1.C1CNC(=O)O1 Cc1c(CC(N2CCC(CC(=O)N(C3CC4(CC4)C3)C)C2)=O)ncn1C c1(C(=O)NCC2(O)CC(C(=O)NCC(C)C(C)(C)C)C2)ccn2cncc2c1 CCCCCCC(CC)NC(=O)CC1CCN1C(C1(C)CC2CCC1C2)=O CCC(CC(=O)N1CC2CC2(CNC(=O)CC(=O)NCC(F)(F)F)C1)C1CCC1 C1(CNC(c2c(C)ccc(C)c2)=O)CN(C(C2COCCOC2)=O)CCC1(F)F c1(C(=O)NCC2(NC(c3cc(CO)cc(F)c3)=O)CCC2)cc2cccn2cn1 Cc1cc(C(=O)NCCC(C)N(C(=O)C(n2ccc(C3CC3)n2)C)C)ccc1Cl C1(C(=O)NCC(CC)NC(=O)C(C)CC(C)(C)C)Cc2ccccc2N1C(C)=O n1(CC)ncc(Cl)c1C(=O)N(C)CC1COCCN1C(C1CC(F)C(=O)N1)=O C(C)(N(C)N1CCOC(CCO)C1)c1ccc(OC)nc1 CN1CCOCC1C(=O)NCC1(C)N(C(=O)C(C)(C)N2CCCCC2)CCC1 C1(NC(Cc2ccc(C)s2)=O)CC2CCC(C1)N2C(=O)COC1CCOCC1 C1(CNC(C=CC)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1C C1(CCN(C)C(C23CCCC2C3)=O)CCCCN1C(=O)COc1ccn(C)n1 Cc1ccc(C(N2CC(NC(=O)Cc3sc(O)nc3O)C(C)C2)=O)c(O)c1 N1(C(C2C(C=C)C2)=O)CCN(C(c2cccc(SC)n2)=O)C(C(C)C)C1 Cc1ccnc2ccc(C(N3CCCC(NC(=O)CCOCC4CC4)C3)=O)cc12 C(C(C)(F)C(C)(C)F)(c1n(CCSC)nnn1)NC(N1CCCCCC1OC)=O N1(C(C)C(=O)N(C2CCCOC2)C)CCN(C(c2ccoc2Cl)=O)CC1 c1(C(N2CCC(CCNC(c3c(C)cc(SC)o3)=O)C2)=O)ncc(C)cc1C C(=O)(CC(C(F)(F)F)NC(C1(CO)CCC1)=O)N(C)Cc1ncccn1 CC1CCC(CNC(=O)Cc2cccs2)N(C(=O)C(=O)Nc2ncc[nH]2)C1 C1(C(N2CCCC(CCCCNC(c3cc(C)sc3)=O)C2)=O)CC12CCOCC2 c1(OC)cc(C(=O)OCc2ccc(O)c(Cl)c2)nc(C(C)C)n1 CCCC(CCC)C(=O)NCC1(CNC(C2CCN(C3CCSC3)CC2)=O)CC1 C(=O)(C(CC(C)C)N(C)C)N(CCCOCCNC(CC)=O)C c1(C(N(CCC(C)NC(=O)Cc2cnns2)C)=O)ccc([N+](=O)[O-])cc1F Nc1cc2c(cc1C(N1CCC3C(NC(=O)C4=COCCC4)C3CC1)=O)CCC2 C1(C2CCCC2)(C(=O)NC(C(C)(C)O)C(=O)O)CCNC1=O N1(C(c2oc(CC)c(C)c2)=O)CC(NC(=O)C(COC)OC)CC12CCC2 CCCCCC(=O)N1CCC(CCOC)(NC(=O)CCCn2ccccc2=O)C1 c1(OC)c(NC(CNC(=O)CC2CC(C)(C)C2)C2CC2)ccc(Br)c1F c1(C(c2nnnn2Cc2ccccc2)NC(COCC)(C)C)c(C)cncc1C O(NC(=O)C(O)CCCNC(c1cccc2c[nH]nc12)=O)CCC(=C)C c1(C(CC)C(=O)NCC(C)(C2CC2)NC(C2CSCCS2)=O)cccc(Cl)c1 C#CCCC(C(=O)NCC1CC2CCC(C1)C2)NC(c1nocc1Cl)=O N1(C(C(CCCCC)F)=O)C2CCCC1CN(C(=O)CC(C)F)C2 c1(CNC(=NCCC)NCC2(SC)CCOCC2)ccc2ccccc2n1 C(C(C)(C)CC(=O)NC1(CCCCO)CC1)NC(C1N(CC)CCOC1)=O c1(C(N2CCC(N(C(C3CCC(=O)O3)=O)CC)CC2)=O)cnn(C)c(=O)c1 c12ccccc1OCC(=O)NCC(OC)CNC2=O.c1(CC)ccc(Cl)cc1 c1(OC)nc(N)cc(C)n1.N1CCCC(F)(CNC(C2C3C4CCC(C4)C23)=O)C1 Cn1ccc2cc(C(=O)NCC3CCCN3C(C3(C)CC3(C)C)=O)cnc12 C#CCC(C)(CC)C(=O)NC1CCCC1NC(=O)COc1cnn(C)c1 C1(C)(C(=O)NC(C)(C)C)CC12CCN(C(=O)Cc1ccccc1O)CC2 C(=O)(CC(C)(C)C(=O)OC)N(CC(N1CC(C)(C)CC1CO)=O)CC#C c1(C(N2C(CNC(c3c(CCC)nco3)=O)C(C)CC2)=O)cccc2c1CCC2 c1(NC(c2sc3n[nH]c(C)c3c2)=O)ccc([N+](=O)[O-])c(OC(C)C)c1 C(=O)(CC1CC(=O)Nc2ccccc21)NCCN(C(=O)Cc1ccn(C)n1)CC Cc1cc(C(=O)NC2CC(NC(C3(CO)CCOC3)=O)C2)c(F)cc1Cl Cc1ccc(CC(=O)NC2CCCC2NC(C2(C)COC(=O)OC2)=O)cc1Cl N1(C(CC(C)CN(C)C)=O)CC(C)(CNC(=O)CNC(N2CCCC2)=O)CC1(C)C CCC(C)C(O)CC(=O)NCCCCN(C)C(C1(C2(O)CCC2)CC1)=O C(=O)(CC(C)(C(F)(F)F)N(C)C)N(C(CCCC)COC)C.C(=O)(C)NCCSCC CC1CCN(Cc2nc(C(C)(C)C)cs2)CC1NC(=O)CSCCOc1ccccc1 c1(C(N2C3C(NC(C(CC)CC)=O)CC(C3)C2)=O)cc2ccccc2s1 C(=O)(C(C)(O)C(C)C)N(CCOC)CCNC(=O)C(c1cccc(C)c1F)O c1(CNC(C2CCN(C)C2)=O)ccc(CNC(=O)CC2CC3CC3C2)cc1F N12CCOCC(C1)C2=O.c1(NC)n[nH]cc1C(N1CCCC1CN(C)C)=O N1(C(CC(C)(O)c2ccccc2)=O)CCC(NC(=O)C=CI)C(CO)CC1 c1(C(N2CC(OC)C(NC(c3ccc(C(F)(F)F)o3)=O)C2)=O)ccc(N)c(F)n1 C(=O)(CCCn1cc(COc2ccccc2)nn1)N(CC(=O)OCC)CCOC C1(NC(C(C2CCCCC2)NC(C(C2CCOC2)OC)=O)=O)(CO)CCOCC1 CCCC(CNC(=O)C(C1CCOC1)OC)NC(c1c[nH]nc1C(C)(C)C)=O C(=O)(C1=NOC(C)C1C)N1CCC(CCOC)(C(=O)NC2(CF)CC2)C1 N1(C(c2cc(C)sn2)=O)CCCC2(C1)CN(C(c1ccnc(C)c1C)=O)CCO2 c1(OC)cc(NC(=O)CC2CCN(Cc3ccc(Cl)nn3)CC2)c(C)cc1[N+](=O)[O-] C1(C(N2CCC3C2CCCN3C(c2ccccc2)=O)=O)CCc2nccn2CC1 c1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CCC2)cccc(OC)c1O N1(C(C=C(C)C)=O)CCC(F)(C(=O)NC2(C(N)=O)CCOC2)CC1 c1(C(N2CCCC(NC(C3CC(=C)C3)=O)C2C)=O)cccc(SC)c1[N+](=O)[O-] CC(C)(C)CC(C)(C)C(=O)N1CCN(CCCNC(=O)C2=CCCCO2)CC1 Cc1ccc(-c2cc(NCC3(O)CCN(C(=O)OC(C)(C)C)C3)n(C)n2)cc1C C(=O)(C(CC(F)F)NC(C1CC(C)(C)CN1C)=O)NCc1cc(C)on1 C1(CC(=O)NC2(CNC(CC3CC(CC)C3)=O)CCC2)CCC2(CC2)CO1 C=CCCCCCCC(=O)NCc1n[nH]c2cc(Br)ccc12.C12CC(C1)NC2=O N1(C(CCC)=O)CCCN(C(c2nnc(S)n2C)=O)CC1C(C)C C1(C(N(C)Cc2ccc(Cl)s2)=O)C2CCC1(c1ccc(Br)cc1)C2 O=C(CC1CCc2ccccc21)NC1CCN(C(=O)Cn2cc(Cl)cn2)CC1F C1(CC(=O)NCCOCCNC(=O)CC23CCCC2C3(F)F)CN2CCN1CC2 n1(CCCOCC)cc(CC(=O)OC)nn1.n12nnnc1C1(COC1)NCC2 c1(C(N(C2CCN(C(c3cnc[nH]3)=O)C2)CCC)=O)cnc(NC)cn1 C1(CC)CCCN(C(C2CC2CCC=CCNC(=O)CC2CCCN2C)=O)C1 c1(C(N2C3CCC(NC(C(C#N)C4CC4)=O)(C3)C2)=O)cc2ccnc(Cl)c2[nH]1 N1(CCNC(C2CC(C)(C)OCC2)=O)CCN(C(C2CCC2(F)F)=O)CC12CCC2 O=C1CC2CC(C(N3CC(O)(c4ccccc4)C3)=O)C1O2 Cc1cc(C(=O)NC(c2ccccc2)CNC(C2CC3(CCC3)C2)=O)oc1C N1(C(c2cn(CC)nc2)=O)CC(CNC(=O)C(N2CCSCC2)C)C(F)(CO)C1 C1(C(=O)NCc2scc(CNC(C(C)n3cncn3)=O)n2)CC2CCC1O2 c1(CN(C2CCCC(n3ccnc3)C2)CC)ccc(C#N)cc1F C1(NC(c2c(OCC)oc(C)n2)=O)CN(C(=O)C(C)(O)CC)CC1S(C)(=O)=O C1(C)(C(N2CCC(N(C(Cn3c(CCC)ncc3)=O)CC)C2)=O)CC(C)(C)C1 c1(NC(C=CCN(C(C(C=CC)O)=O)C)=O)cnn2c1OCCC2 C1(NC(CCC)CC)CCOCC1C(=O)OC(=O)CC1(CS(C)(=O)=O)CC1 c1(SC)cnc(OC(C)C)nc1.C1(C)(C)CN(C)CC(=O)N1 c1(C(N2CC(CC(C)NC(=O)CC3CCCCC3)C2)=O)ncoc1-c1ccon1 c1(OC(C)CNCC(c2ccccc2)C)ccccc1C(F)(F)F c1(COC)cc(=NCC2CCC(NC(=O)CCCC3CCC3)C2)[nH]cn1 CCCC(C)(C)CC(=O)NCC(CNC(C1C2CCCOC12)=O)C(F)(F)F CCC(CC)C(C(=O)N1CCCOC(CCNC(C2(C)CC=CC2)=O)C1)OC C1(NC(CCc2n(C)ncn2)=O)CC2CCC1N2C(=O)COCC1CCCOC1 CN1CC(C)(C)CC1C(=O)NC1CCCCN(C(C2(C)CCC2)=O)C1 c1(C(N2CCC(C)C2CNC(C2CCC(O)C2)=O)=O)cccc(C#N)c1 C(=O)(C(C(=O)N1CCC(C(C)NC(=O)CCCOC(C)=O)C1)C(C)(C)C)OCC N1(C(COCCC)=O)CC2CCC1C1CN(C(c3csc(C)n3)=O)CC21 c1(OC)ccc(C=CC(=O)NC=CC=C)nc1.C1CC(NC(=O)C=CC2CC2)C1(C)C CCCC(C)C(=O)Nc1ccccc1Br.N12CCSCC1NC2=O CN1CC(NC(=O)C(C2(C)CC2)NC(c2ccc(=N)[nH]n2)=O)C(=O)N1 c1(C(=O)NCCCCNC(C(CCSC)O)=O)cc2ccccc2nc1C(F)F C1(OCCNC(C2C(=C)C2)=O)(CNC(=O)COC2CC2)CCOCC1 C1(OCC)CCCCC(c2nnnn2C(C)COCc2sccc2C(=O)OC)C1 CC1CCN(C(=O)CC2CCC(=O)NC2)C(CNC(=O)CCc2cnco2)C1 c1(NC)ccccc1C(=O)NCCC1CC(C(=O)Nc2ccsc2C(C)C)C1 N1(C(CSCC#C)=O)CCC(NC(=O)CN2CCc3sccc3C2)CC(O)C1 CC(CCCCCO)NC(=O)C(C1CCCO1)NC(=O)CCc1ccccc1 c1(CCC)nc(C)c(C(N2CC(N(C)C(c3ccn(C(C)C)n3)=O)C(F)C2)=O)s1 Cn1cccc(C(=O)NCC2CCCCN2c2nnc(-c3ccccc3)o2)c1=O CC1C2C(CCN2C(c2csnc2Cl)=O)CN1C(=O)C(F)CC1CCOC1 C1(C(N2CC(C3(NC(C4CSC4)=O)CC3)C2)=O)CCOC2(CCCC2)C1 CC1CN(C)CCN1C(=O)C(C(C)(C)O)NC(=O)COCCCN(C)C c1(OC)ccc2ncnc(N3CCCC4C3CCN4c3ncncc3F)c2c1 Cn1cnc2c1CCC(C(N1CC(NC(C3CCCC(=O)N3)=O)C(O)C1)=O)C2 Cc1cc(=NCCCOCCO)[nH]cc1S(=O)(=O)NC1CCCOc2ccccc21 C1(Nc2nc(C(CC)OC)cc(C)n2)CC12CCc1ccccc12 c1(CC(=O)NCC2(O)CCN(Cc3n(C)cnc3)C2)ccccc1[N+](=O)[O-] c1(C2N(C(=O)Nc3c(C4(OC)CCC4)cccc3)CCC2)cc(F)cc(F)c1 c1(C(C(=O)NCC=C)NC(C)(C)C)ccc(C)c(Br)c1C.c1(OCC)ccc(F)cc1 c1(-n2c(C(C)OCC)nc(-c3ccc(Cl)s3)n2)ccc2nccnc2c1 S(=O)(=O)(c1ccc(COC)cc1)C(CSCCC(=O)N(CCC)CCC)=O C(=O)(C1=C(Cl)CCOC1)NC(C1CCCN1C(c1cc(C(N)=O)c[nH]1)=O)(C)C c1(C(=O)NC2C(C)CCN(c3ncnc(CC)c3F)C2)ccc2ccnn2c1 Cc1c(C(N2CC(CNC(c3ccc(N(C)C)nn3)=O)CC2C)=O)n[nH]c1C1CC1 Cc1ccc(CC(N2CCN(CC(=O)NCc3cc(C4CC4)n[nH]3)CC2)=O)cn1 C12(C(N(CC(C)(C)NC(C3(C(=O)NC)CC3)=O)C)=O)CCCCC1CCC2 C(CCC(C(=O)NN1CC(C)(CNC(=O)C2CC2)C1)NC(=O)C1CC1)OC Cc1cc(=O)n(C)cc1C(=O)NCC(O)CNC(c1cn(CCO)nn1)=O c1(CCNC(C(C)SCCCC)=O)ocnc1CNC(C1CCC(CC)O1)=O C1(NC(COC(C)(C)C)=O)C2COCC1CC(NC(C1(CO)CC1)=O)C2 N1(CC(=O)NCCCC)CCC2(CCN(C(c3cccc4ncccc34)=O)C2)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(CO)C1 CC1CCC(CNC(C2CCSCC2)=O)N(C(c2ccc(C(F)F)c(F)c2)=O)C1 c1(C(=O)NC2CC(C(C)NC(Cc3cc(C)[nH]n3)=O)C2)ccccc1Br c1(C(C(=O)NC(C)CC)N(CC(C)C)CCC)cc2c(cc1OC)CCC2 C(CN=c1[nH]nc(C(F)F)o1)(CC(C)C)CN(C1CCN(CC)CC1)CC C1(N(C(c2c(C)snn2)=O)C)CN(C(c2cc(-c3ccccc3)no2)=O)CC1O c1(OC)nc(Cl)ccc1C(=O)NCCC1(O)CN(C(=O)C(O)Cc2cnc[nH]2)C1 c1(C(N2CCCC(NC(=O)CC3CS(=O)(=O)C3)CC2)=O)cc2c(O)cccc2[nH]1 c1(Nc2cnn(CCOC)c2C)nc(=NC2CCC3(CC3)C2)[nH]c2c(C)nn(C)c12 c1(C(N(C)CC2CN(C(CC=CCC)=O)CC23CC3)=O)nn(CC)cc1[N+](=O)[O-] N1(C(C(CC)C2CC2)=O)CCC2C(CCCN2c2cc(SC)nc(SC)n2)C1 c1(NC(C2CC(NC(c3c(CC)n(C)nc3)=O)C(O)C2)=O)cc(C)c(C)c(C)c1 N1(C(C=CC2(C)COC2)=O)CCCC(CNC(=O)CC2CCC23CCC3)CC1 CC(O)(CNC(=O)CCCC1CCCC1)CNC(C1CCCCC1)=O Cc1nnc2n1C(C(=O)NC1CC1CNC(c1cccc3c1CCCC3)=O)CC2 C1(COC)(NC(C2CCOC2)=O)CCCN(C(=O)C=Cc2cnccc2C)C1 C1(NC(=O)CC2(N3CCCC3)CC2)CC2(NC(C3C4COCC34)=O)COC1C2 C#CC(CNC(=O)CCCCCN(C(=O)Cc1ccccn1)C)CC(C)(C)C CC1(C)CC2(CC(C(N3CCC(CCNc4nccnc4F)C3)=O)C2)C1 C1(C2=CCCCCC2)(C(=O)NCC2(O)CCN(C(C(CCC)(C)C)=O)CC2)CC1 c1(C(=O)NCC2C(NC(CC(C)CF)=O)CCCC2)cc(F)c(Cl)cc1Cl C1(C(CNC(c2cncs2)=O)F)CCN(C(=O)C(c2ccc(F)cc2)F)CC1 C(CC)(C(=O)NC1(CNC(c2cc(C(C)=O)on2)=O)CC(OC)C1)OCC.C1CC1 C1(NC(c2c(C)noc2)=O)CC(F)CN(C(c2ccc(OC(C)C)cc2)=O)C1 N1(C(c2c(CC)c(C)sc2)=O)CC2C3CCC(C2C1)N(C(=O)C(F)(F)C1CC1)C3 n1(CC(N2CCC(C)(NC(C(C)C(C)(C)C)=O)CC2)=O)cc2ccccc2n1 N1(c2ccc(S(=O)(=O)NCC(C)F)cc2Cl)CCc2ccc(C#N)cc2C1 c1(CC(N2C(CNC(C3(C)CCC(=O)NC3)=O)C=CC2)=O)c[nH]c2cnccc12 N1(C(Cn2ccc(C)n2)=O)CCC(C)(C)C1C(=O)NCCC1(CN(C)C)CC1 Cc1nc(C)c(CC(N2CCCC(C)(NC(C3CCCC(F)C3)=O)C2)=O)c(O)n1 c1(C(N2CC(n3cc(C4CCN(C)CC4)nn3)C2)=O)cc2c(Br)cccc2s1 C1(C(=O)OC)C=CCCN1C(C1CCN(C(c2cscc2OC)=O)C1)=O c1(C(N(CCCNC(c2nc(Cl)oc2C)=O)CC)=O)ccc(F)c(C#N)c1 C(=O)(C1CCSc2ccccc21)NC1CCC(NC(CCC(C)(C)O)=O)CC1 c1(C(=O)NC2CC(F)(CNC(C(C)NC(CC)=O)=O)C2)ccc(Br)c(N)c1 C1(C(=O)NC(C2CCOCC2)C)CC(NC(=O)C(F)(F)C(F)F)C12CCC2 Cc1nccc(C(=O)NC2CC2CNC(=O)CCCSc2ccccc2)n1 N1(C(CC2CN(C(C(CCC)C#N)=O)C(C)(C)C2)=O)CCCC(C2(C)CC2)C1 c1(C(=O)NCC(C=C)(C)C)coc2c1CN(C(=O)CCN(C)CCC)C2 n1(CC)c(C)cc2c1CCCC2NCCCc1c(C)oc2cc(C)ccc12 C1(CC(=O)NC2CCN(c3nc(C)cc(OC)n3)C2)Cc2ccccc2C1 c1(C(N2CCCC(N(C)C(C3CC(=O)CCO3)=O)C2)=O)[nH]cc2c1CCCC2 c1(C(N2CCOCC(NC(C=CC(C)C)=O)C2)=O)nnc(O)c2ccccc12 C(=O)(C1CCc2c[nH]nc21)NCCCCNC(c1cncc(OC)c1)=O c1(CC=C)cccc(C(=O)N(CCC(=O)NCC2C3COCC23)CC)c1 C12(CNC(C3CCN3C(=O)COC3CC=CC3)=O)CCC(CC1F)C2 CCC(C)CCCCC(=O)NC1CN(C(c2cccc3c2OCCO3)=O)CC1O C1(CC=C)(NC(C(C=C)(C)O)=O)CCN(C(C2CN(C(C)=O)C2)=O)CC1 N1(C(c2c(C)nn(C)c2)=O)CCOC2(CCC(NC(=O)Cn3cnnc3)CC2)C1 C(=O)(CCCC(F)(F)C(F)(F)F)NC1COCCN(C(C(C(C)C)C#N)=O)C1 c1(C(=O)NC2CCN(C(C(C)C(C)O)=O)C2C)coc2c1CCCC2 C1(CC(N2C(C)CC(CCNC(C(CSC)C)=O)C2)=O)CCCCC1(F)F C#CCN(OC)C(=O)C(O)CC1CCCN1C(=O)CC(C)(C)C C12(CCNC(C(F)=C(C)C)=O)CCC1CN(C(C1(c3cccs3)CC1)=O)C2 c12cnc(cn1)C(=O)NC(C1CC1)CNC2=O.c1(C(=O)OC)cc(C(F)F)cs1 C1(CNC(CC(C)(C)N(C)C)=O)CN(C(=O)C(F)(F)C2(O)CCC2)CC12CCC2 CC(CNC(=O)CC1CCC1)C1CC1.C1(C2(C(=O)NCC(F)(F)F)CC2)CCCO1 c1(NC(c2cscn2)C)[nH]c(=NC2CCCC(O)C2)nc2c1cnn2C C1(C)(CC)CCC(c2nnnn2CCCSC)(NCc2ncn(C)n2)CC1 c1(C(=O)NC(CC(C)NC(c2ccc3sncc3c2)=O)C)cc(S(N)(=O)=O)co1 C#CCCC(C(=O)N1CCC(F)(CO)C1)NC(c1cccc(C)c1O)=O c1(OC)cnc(NC(c2ccsc2COC)=O)nc1SC(C)C C(=O)(C(C)(C)C#N)NC1C(NC(C(C)CSCc2ccccc2)=O)C1 C(CCCN=c1[nH]c2cc(Cl)cc(Cl)c2o1)NC(C1CCCC(NC(C)=O)C1)=O C1(CNC(C=NOC)=O)CC(C)(C)CN1C(=O)CS(N)(=O)=O O=C(N=c1cccn[nH]1)C1CC(O)CN(C(c2ccnc(-c3cccs3)c2)=O)C1 C1(CNC(C(CC#C)(C)C)=O)COCC2(CCN(C(=O)CC(C)(C)SC)CC2)O1 CCC1=NOC(CC(=O)NCCN(CC(C)O)C(=O)C=C(C)c2ccco2)C1 C1(C(=O)NC(CCC)CNC(c2cc(C)sc2C)=O)CCc2nc(C)[nH]c2C1 C1(c2nnnn2C2COC2)(NC(CC=C)CC)CSCCSC1 C1(C(=O)OC)(C(=O)NCC=CCC(=O)NCC2CC2)CC1C.c1(C2CCC2)ncc[nH]1 C1(C)(CNCc2n(C)ccn2)CNCCO1 C1(CCNC(c2cnc(C(C)O)s2)=O)CCCCN1C(C1CCC=CCC1)=O CC(C)(F)C(C)(F)C(=O)NC1CC(NC(c2cnc3ccnn3c2)=O)C1 N(C1CCCc2c1cnn2-c1ccccc1)C(=O)NCc1c(C)scc1 CC1COCCCN1C(=O)C(CC(F)F)NC(=O)Cc1ccon1 C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])c1c(CNC(c2c(C)noc2)=O)cccc1 C=CCC(CNC(=O)Cc1nc[nH]n1)NC(=O)CC1CCSCC1 N1(C(C2(COC)CC=CC2)=O)CC(NC(C2CCC(F)CC2)=O)C(C)(C)C1 c1(C(N2C(C)CN(C(C3(C)CC3Br)=O)CC2)=O)ccc2ncsc2c1 c1(C(N(CCN(C(=O)COc2ccc(Cl)nc2)C)C)=O)cccc2nc(O)[nH]c12 N1(C(c2cn(C(C)C)nn2)=O)CCOCC(NC(C2(CCF)CCC2)=O)C1 S(=O)(=O)(c1csc(C(=O)NC(C(C)NC(C23CCC(CC2)C3)=O)C(C)C)c1)NC N1(C(C2C(C)CCC2)=O)CCCC(C)(C)C1CNC(C1CCCSS1)=O C1(NC(C(=O)NCC)=O)COC2C(NC(C3CNC(=O)N3)=O)COC12 c1(C(=O)OCc2ncccc2Oc2ccc(F)cc2)cc2cccnc2cn1 c1(C(=O)NC(C)CN(C(=O)CCc2nccs2)C)sccc1S(N)(=O)=O N1(C(C=NOC)=O)CC2CCCC(CNC(c3cc(O)nc(O)n3)=O)(C2)C1 c12c(cccc1C)NC(=O)NC2.C(CCO)N(CCC)CCOC N1(C(C(COCC)C)=O)CC(OC)CC1C(=O)NCc1c(C)cnn1C C1(C(F)(F)F)(C(N2CCC(N(CCC)C(C3COC(C)C3)=O)C2)=O)CCOCC1 c1(C(N2CC=CC(C(N3CC(OC)C(O)C3)=O)C2)=O)cc(O)ccc1C c1(CC(CC)C)nc(-c2nnn(CC)c2C)n(C2CCOC(C)C2)n1 c1(OC)cc(CC(=O)N(C)CCN(C(=O)C(C)(C)CF)C)cc(F)c1 c1(C(=O)NC(C(=O)N(C)CC2(O)CN(C(CC(C)C)=O)C2)C)ccc(F)cc1F S(=O)(=O)(c1ccc(NC(=O)NNC(=O)c2ccccc2N(C)C)cc1)NC C(=O)(CCC(=O)N1CCC(C)C1CNC(=O)CCCc1sccc1C)NC c1(SC)cc(C(=O)NC2CC(CNC(c3[nH]cnc3C#N)=O)C2(C)C)c(C)o1 C1(C(=O)NC(c2ccco2)C)CC(O)CN1C(C1C=CCC1)=O Cc1nnc(C(N2CC(c3ocnc3Cn3cc(C4CC45CC5)nn3)C2)=O)s1 N1(C(=O)OC(C)(C)C)CC2CC1CN2C1CCCC1.c12ccccc1CS2 c1(CC)cc(C)c(C(=O)NCCCN(C)C(C2C3CC(=O)CC23)=O)o1 c1(C(N2C(C)CC(CNC(C(CC#C)CC#C)=O)C2)=O)cnc2cnccc2c1 c1(C(=O)NCCC2CN(C(CCCC(N)=O)=O)C2)cccc2[nH]ccc12 C1(C)(C(=O)NCC2C(C)CN(c3ncnc(=N)[nH]3)CC2)CCCNS1(=O)=O N1(C(C2CC2C2CCC2)=O)CCC(NC(C2(Sc3ccccc3)CCC2)=O)CC1 c1(C(=O)NC(C(C(C)C)C)CNC(C2(CO)CCCC2)=O)ccc(C#N)cc1F c1(NC(C2(C(N(C3(C#C)CC3)C)=O)CC2)=O)nn(C)cc1C C=CC(C)CC(=O)NC(CCNC(=O)C(CCC)N(C)C(C)=O)C(C)C NS(=O)(=O)C1(C(=O)NCC2(F)CCC(NC(C3CCNC3=O)=O)C2)CCCC1 N1(C(CC)=O)CC2CN(C(c3cc(C4CC45CC5)ccc3Cl)=O)CC2C1 C(=O)(C1=C(Cl)CCOC1)N1CC(CCNC(c2ccc(F)s2)=O)OCC1 C(=O)(C1=CN=C2N=CNN2C1)N1C2CN(C(C3=CC(C)(C)C3)=O)C(C2)C1 C1(NC(C(C(CC)C)OC)=O)CC2CN(C(=O)C(=Cc3ccccn3)C)CC2C1 C(=O)(C(CCCN)NC(c1ccc(NC(=O)C2CC2)nc1)=O)OC Cn1c(C(N2CC3CC2C3CNC(C2C=CC=CC=C2)=O)=O)cccc1=O c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)C(C)C)ccc(O)nc1Cl C=CC(CCC)CC(=O)NC(C(=O)NCC1([Si](C)(C)C)CC1)C1CCCC1 C1(C(N2CCC(CNC(c3cc(F)n[nH]3)=O)C2)=O)CC2CCC(C1)S2 c1(C(N2C(C(C)NC(CC)=O)CCC2)=O)cnc2ccncc2c1 CCCC(O)C(=O)N1CCC(CN(C(=O)CCc2c(C)noc2C)CC)CC1 N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC2CC2(C)C)C(O)C1 C(CCC(C)C(=O)NC1CC(NC(c2ncoc2C)=O)C1)OC C1(C(N2C(C=C)CCC2)=O)C2CCC(C2)N1C(=O)C=C(C)COC N1(CC(=O)N(CCC(=O)NCC2(O)CSC2)C2CC2)C(=O)CNC1=O CN1CCCC(CNCC2NCC23CCCC3)C1c1ccccc1 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)CC2CCCO2)cn(C)nc1C C1(NC(c2c(C)nc[nH]2)=O)CCC(NC(=O)CCNc2ccccn2)CC1 N#Cc1cc(C(N2CCCC2CC(=O)N(CCO)CCO)=O)ccc1O C(CC1=CCN(C(=O)CN2CCC2)CC1)NC(=O)CC(c1ccccc1)C1CC1 c1(OCC(=O)NC(CN(C(C(C)OCC#C)=O)CC)C)cccc(Br)c1 c1(C(=O)NC(c2cncnc2)C)coc(CNC(=O)CCCSC2CC2)n1 c1(C(N2CC3CC(NC(c4cnsc4)=O)C3C2)=O)cncc2c(O)nccc12 S(=O)(=O)(c1ccc(Cl)nc1)N1C(CC)CN(C(C2CN(C)C2)=O)CC1 C1(C(=O)NCCC(C)NC(C2CCN(CCC)CC2)=O)CCc2n[nH]cc2C1C c1(C(C(=O)NCC(C)N(C(=O)CC2CCC(O)C2)C)(C)C)cc(Cl)ccc1F N1(C(C(CC=C)C)=O)CCC2C(NC(=O)Cc3ccsn3)C2C1 C1(COC)(NC(=O)CC=Cc2ccc(C)cc2)CCCN(C(C2CCSC2)=O)C1 C1(C(N(CC(CC)NC(=O)CC2(O)CCCC2)C)=O)C(c2ccccc2)C1(F)F N1(C(c2ccn(CCCF)c2)C(=O)Nc2ccccc2)Cc2ccc(Br)cc2C1 c1(OC)ccc(C(N2CC(CC(C)NC(=O)CCc3cnc(C)o3)C2)=O)c(F)c1 n1(CC(=O)NCCN(C(=O)C(C)CC(F)F)CC)c(C)cc(C)nc1=O CC1CCC(F)(C(=O)NCC2CCN(C(c3ncoc3C3CC3)=O)C23CC3)CC1 N1(C(C)C(=O)N(C)CCN(C(=O)C(C)Oc2cccnc2)C)CCCCC1=O N1(C(C(C)(C(C)C)OC)=O)CCN(C(c2csc(C(C)(C)C)n2)=O)CC(O)C1 N1(C(C2(O)CCC(C)CC2)=O)CC(C)N(C(C23CC(F)(C2)C3)=O)C(C)C1 n1(CCNC(C(CCOCCO)NC(COC)=O)=O)ccc([N+](=O)[O-])n1 C(=O)(C(F)CC(C)(C)NC(=O)CC1CSCCO1)N1C(CC(=O)OC)CC1 Nc1ncc(Br)nc1C(=O)NCC1CCC(NC(=O)CCOCC2CC2)C1 C(=O)(C1=CCCN(C(C2CCCSC2C)=O)C1)N1CCC(C=C)(O)C1 N1(C(c2cnn(CC)n2)C(=O)NCCCF)CCc2oc(C)nc2C1 c1(C(N(C(C)C(C)(C)C)C)=O)cc(CNC(=O)CC(C)C2CCCO2)nn1C C1(C)(N(C)CC)CCN(C(c2coc(CN(C(=O)C(C)(C)CF)C3CC3)n2)=O)C1 C1(OC)CC2CCCCN2C1=O.c12cc(C#N)ccc1[nH]c(=O)[nH]2 c1(OC)nn(C)cc1C(=O)CNC(c1cnn(C)c1F)=O C1(C(=O)Nc2cccc(OCC(=O)OC)c2)C2CCC1N(C(=O)CCN(C)C)C2 N1(C(CN(C(COC)=O)C)=O)CCC(C)N(C(C2CNC(=O)C(C)(C)C2)=O)CC1 N1(C(C(C)NC(C)=O)=O)C2CN(C(C3CCC(=O)N3c3ccccc3)=O)CC12 c1(C(=O)NCC(=C2CN(C(c3cnc[nH]3)=O)C2)F)cnn2ncccc12 C1(NC(CC2CN(C)C2)=O)CC2CCCC(C1)N2C(c1csnn1)=O C1(NC(C(c2ccn(CCF)n2)C)=O)C2CC(NC(C3(C)C=CCC3)=O)CC12 CC(C)CC(C(=O)NCC(O)CCNC(c1ccc(C#N)o1)=O)C(N)=O c1(C(C(F)F)NC(c2ncc(Cc3cccc(Cl)c3)s2)=O)ccccc1Br c1(OC)cc(C)c(C(=O)N(C)CC2CCN(C(c3cnoc3C)=O)C2)cn1 C1(CCC)CN(C(=O)CC2OCCO2)CC1C(N1CC2(CC2)C1)=O C1(CC(=O)NCC2CCCC2NC(c2cncn2C2CC2)=O)CC(=O)NC1=O C(=O)(CC(C(C)C)C(C)C)N1CC(OC)C(NC(=O)CCC2CCN(C)CC2)C1 c1(C(=O)NC2CCCC(NC(=O)COC(F)F)C2)ccc(C(C)(C)C)cn1 Cc1cn(C(C)C)cc1C(=O)NCCCC1(NC(=O)Cc2ccc(F)cn2)CC1 C1(C2CCN(C(C3CSCCS3)=O)C2)(NC(=O)C(CC(F)F)C2CCC2)CC1 c1(C(=O)NCC2CN(C(C)=O)C(C)C2)coc2c(C)cccc12 C1(C(=O)Nc2cc(OC)nc(C(=O)O)c2)CC12CCN(C(=O)CCN(C)C)CC2 CS(=O)(=O)c1ccc(CC(=O)NCC2(F)CCN(C(=O)Cn3cncn3)CC2)cc1 O=C(CCCCCO)NCC1(NC(=O)CC2(N3CCOCC3)CCOCC2)CC1 N1(C(C2(CF)CCN(C(C(C(C)C)O)=O)C2)=O)CC2(COC(C)(C)C2)C1 c1(C(N(CC(C)NC(C2CCC2C(F)F)=O)C)=O)c(C(F)(F)F)ncn1O N1(C(=O)NC(c2ccc(C#N)cc2)CC(C)C)CCN(C2CCOC2)C(=O)C1 CC1=CC(C)CN(C(C2C(C)CN2C(C2CCN(C)C2)=O)=O)C1 Cc1cccnc1CNC(=O)CC1CCC(NC(=O)C=CC2CCOC2)C1 C=CC1(CC(N2CCOC(CNC(=O)CCOCCOC)C2)=O)CCCCC1 N1(CC(=O)N(C(C#C)C)C)CCN(C(c2cnccc2OC)=O)CC1 C1(NC(CSc2cccc(C)c2)=O)CS(=O)(=O)CC1NC(c1cc(C#N)on1)=O c1(OC)ccc(C)c(C(N2CC3CC(NC(=O)C=CC(C)(C)C)C2C3)=O)c1N N1(C(c2ccc(CC)cc2N)=O)CCN(C(c2cn(CCO)nn2)=O)C(C)C1C N1(C(=O)CC2CCCS(=O)(=O)C2)CCC2CCC(NC(C3(Br)CC3)=O)C1C2 C1(CC(=O)NC2CCC(CNC(CN(c3ccccc3)C)=O)C2)COC2CC1C2 Cc1ccccc1C(C)CC(=O)N1CC(N(C)C(c2cc(O)n(C)n2)=O)C1 c1ccc(NC2(CCCC3CCCCO3)CCC2)cc1 c1(C(N(CCNC(C2CC(=C3CC3)C2)=O)CC)=O)ccc(C2CCCO2)[nH]1 c1(COC(C)(C)CNC(=O)NC(C)CCCc2ccccc2)cccc(F)c1O C1(NC2C(C)(CC)CC2OC(c2cnn3c2CCC3)=O)CC(S(C)(=O)=O)C1 C=CC1(CC(=O)NCc2cccnc2F)CN(C(=O)C=C2CCOCC2)C1 c1(NCCC(=O)NC(CC)C)nc(N2CC(O)CC(F)C2)cc(C)n1 C1(C(=O)NCC(CNC(COCCC)=O)F)CCSCC1 N1(C(C23CN(C(C4CCO4)=O)C(C2)CCO3)=O)CC2C3CCC(O3)C2C1 C(=O)(C#CC1CCCCO1)NCC(CNC(C1N(C(C)=O)CCC1)=O)C c1(SCC(=O)NCCC(C)(C)NC(CC=CC)=O)nc2ccc(C)cc2[nH]1 CC1CCN(C(=O)Cc2c(C)noc2Cl)C(C)C1NC(=O)C1=COCC1 N1(C(CN(C(C(C)C)=O)C)=O)CC2(CC2)CC1CNC(C1CC12CCSCC2)=O c1(OC)cccc(C2CCN(C(=O)NCCc3cn(C4CCCCC4)nn3)C2)c1 CCC(CN(C)C)CC(=O)NCC(C)(C)NC(=O)C=Cc1cncs1 c1(C(=O)NC(CC=C)CNC(=O)C=C2CCC(C)CC2)cncc2ccccc12 CN1C(=O)NCC1C(N1CC2C(NC(C3CC(CF)C3)=O)C2C1)=O C(N=c1[nH]cnc(NCC23CCC(CC2)CC3)c1C)c1scc(CC)n1 N1(C(c2c(CC)nc[nH]2)=O)CCC(C)C1CNC(=O)C(=O)NCCOC CC(C(C)C(=O)NCCN(C1CCCC1)Cc1cc(F)ccc1F)S(C)(=O)=O c1(CN(C)C)cc(C(=O)NCC2(CN(C(=O)CCC3CCCOC3)C)CC2)no1 C1(N(C(C2CCCC2)=O)CC)CCCN(C(=O)CC2CCS(=O)(=O)C2)CC1 CCCC(C#N)C(=O)NCCCCc1cn(-c2ccc(C)c(Br)c2)nn1 c1(C(N(CCNC(C(F)(F)C2(OC)CCC2)=O)C2CC2)=O)cnc2cccnn12 C1(NC(c2cncc(C)n2)=O)CC2CN(C(C3CN(C)CC(C)O3)=O)CC12 c1(C(N2C(CNC(C3N(C(C)(C)C)CC3)=O)CC2)=O)cc2c(s1)CCCCCC2 C1(C(=O)NCCCCCCNC(C2CC2F)=O)CS(=O)(=O)c2ccccc2O1 c1(OC)cccc(C2CCN(Cc3cc(Cl)ccc3N(C)C)C2)c1F c1(CNC(=NCC)NC2CC(OC(C)(C)C)C2)nnc(O)c2ccccc12 CN1CCc2[nH]nc(C(=O)NC3CC(NC(=O)C(CC(F)F)C4CCC4)C3)c2C1 c1(C(N2CCC3(CCC3)C2)=O)csc2c1CCN(Cc1cccc(F)c1Br)C2 C1(SCC(=O)N(C2CN(C(c3cc(Cl)ccn3)=O)C2)C)CCS(=O)(=O)C1 c1(-c2cncc(C3CCN(C(CCOCC)=O)CC3)c2)ccc2sc(C)nc2c1 C(C(C)(C)C(=O)N1CCOC(C(=O)NCCSC(F)F)C1)OC(C)C Cc1nc(C(N2CC(O)(C(F)C(=O)Nc3ccccc3F)C2)=O)sc1C N1(C(COCC(=O)NC)=O)CCCC2C(CCCN2C(c2ccc(F)cn2)=O)C1 N1(C(C2N(Cc3c(OCC)ccs3)CC(C)C2)=O)Cc2ccccc2C1 N1(C(c2nc(CC)sc2)=O)CCCC(C2(NC(C3(OC)CC3)=O)CC2)C1 N1(C(C2CC(OCC)C2)=O)CCC(NC(=O)CCN(CC(C)C(C)C)C)C(O)C1 O(NC(=O)C(F)C(C)(F)F)C(C(=O)NCC(NOC)=O)CC(C)C c1(C(CC)C)nc(NC(=O)CCOC)cc(C)n1 CCC(CC)(CC)C(=O)Nc1ccc(CC(C)NC(=O)NN2CCCC2=O)cc1 C1(C(N(CCS(C)(=O)=O)C)=O)CC2CC2N1C(C1(C#N)CCCC1)=O C(N=c1cc(C(F)(F)F)nc[nH]1)C1(NC(C2CCC(C)C2)=O)C(C)CCCC1 Cc1cccc(C(N2CCOC(C(=O)NC(c3ccc(Br)cc3)CO)C2)=O)c1O C1(CCNC(C2C(C)CC(C)O2)=O)CCCN(C(c2nnn(C)c2N)=O)CC1 C(=O)(CCCCC(C)(C)OC)NC(CC)CNC(=O)C(COC)NC(C)=O C1(C(=O)NCC(C)C(=O)O)CCCN(C(C)Cc2ccco2)C1 c1(CC)cc(C(=O)NC2(CNC(c3ccc(-n4cncn4)cn3)=O)CC2)sc1C O=C(CC(F)(F)C(F)(F)F)NC1CCC12CN(C(c1cccc3[nH]ncc13)=O)C2 C1(C)(C(N2CCC(C)(NC(CCCCCOC)=O)C2)=O)CCCC(F)(F)C1 C(=O)(CC(C(=O)OC)OC)NCC1c2ccc(cc2)OC1.C(C)(C)(C)OCC=C N1(C(C(CSC)O)=O)CCC(C(O)CNC(C2CC(F)(F)CS2)=O)CC1 Cc1ccc2sc(NC(CNC(=O)C(=O)N=S(C)(C)=O)C(C)C(C)C)nc2c1C Cc1nn(Cc2ccccc2)cc1CN(C(=O)C(F)C(=O)O)CCN(C)C c1(C(=O)NC(c2cnn(C3CCCC3)c2)C(=O)OC)csc2cncn12 C1(CC(C)(C)C)(C(=O)N(CCCO)C2CCC2)CCNC1 c1(CNC(=O)NC2(CCO)CCCOC2)ccc(Cl)c(F)c1F c1(CNC(=O)NCC2CCC(C(F)(F)F)C2)cccc2ccc(Cl)cc12 C(N=c1[nH]c(N2CCOC(CCF)C2)nc2c1COC2)C1(C)COCCO1 CCCC(O)CCNC(C1(CNC(c2sccc2F)=O)CC(C)(C)C1)=O N1(C(c2c(OC)ncnc2OC)=O)CCC2(CCCN2C(=O)C(C)C(C)C)C1 C(CCC(C)(C)C(=O)NCC1(O)CCCC1(C)C)NC(CCc1ccn(C)c1)=O C1(O)(C(=O)NCCN(C(C(C)CC(F)F)=O)CC2CC2)CN2CCC1CC2 c1(NCC2CCCN(C(C(CC)(CC)CO)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 N1(C(C(C(C)C)OCC)=O)CCC2C1CCCN2C(c1ccc(C#N)cc1F)=O Cc1ccc(F)cc1N(C=O)C(COCc1c(F)cccc1Cl)Cc1ccccc1 c1(C(=O)NC(CN(C(=O)CC(C2CC2)C2CC2)CC)C)sccc1Br c1(Nc2cccc(CNC(=O)Nc3c(C)coc3C)c2)ccc2c(c1)CCCO2 C(=O)(C1=CCCCC1C)NC1CC(C)(CNC(Cc2c(C)cco2)=O)C1 CCC(CC)C(C)C(=O)N1CCC(CNC(C2CCCCS2(=O)=O)=O)C12CC2 CC1N(C(C2(C(C)NC(c3ncccc3O)=O)CC2)=O)CCOC1(C)C c1(COC)ccc(C(=O)N(CC(=O)NC(CC)C(C)O)C2CC2)o1 c1(C(=O)NCC(O)CCNC(c2ccc(O)nc2Cl)=O)ccc2c[nH]nc2n1 C12(C(C(=O)NCCC(O)CNC(=O)C(C)CN(C)C)OC)CCC(CC1)C2 CCCCCC(C(C)(C)C)NCc1cnc(CCC(F)(F)F)s1 c1(C(N(CCN(C(c2ccc(C(=O)OC)[nH]2)=O)C)C(C)C)=O)cc2n(n1)CCCO2 c1(C(N(C)CCNC(C2CCCC(C(N)=O)C2)=O)=O)cc(C(C)(C)C)ccc1N c1(C(N2CCN(C(CS(CCC)(=O)=O)=O)CC2)=O)cc2cccc(C)c2s1 c1(SC)ncc(C(=O)N(C2CN(C(=O)C(C)C3CCC3)C2)C)n1C c12ccc(cc1)[nH]c2=O.C12CCC(CC1)OCC(=O)N2.C1(CO)CCCO1.CC CN1CCc2cc(C(=O)N(C3CCC(NC(=O)Cc4nccn4C)C3)C)sc2C1 C1(C(N2CCC(CC)C2)=O)CN(C(=O)C2=CCCOCC2)CC(C)(C)C1 Cc1ncc(CC(=O)NC2CCCC(NC(c3cc(CCO)on3)=O)C2)c(O)n1 N1(C(C(=CC2CCCC2)C)=O)CC2CCCN(C(c3cnncc3O)=O)C2C1 C1(CCNC(CC2C(C)C2(F)F)=O)CCCCN1C(c1cc(C(F)F)no1)=O N1(C(=O)NC2(c3ccc(OC)c(Br)c3)CCOCC2)CCCCCCCCC1 C1(=O)CCN1.C(=O)(C(C)=CC(C)(C)C)N(CCN(C(=O)NC)C)C(C)C C1(NC(C(COC)O)=O)CN(C(=O)C=Cc2cncc(O)c2)C(C)(C)C1 C1(N(C(=O)C(=O)Nc2nnc(O)s2)CC)CC(N(C)C)C1(C)C c1(C(=O)NCC2CCN(C(C(CC(N)=O)O)=O)CC2)[nH]nc2ncccc12 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CC2CC2(NC(=O)CCC2CCC(=O)NC2)C1 C1(NC(=O)CN2C(=O)CCC2=O)CCC2CN(C(C3CCOC3)=O)CC2C1 C1(CC(N2CCC(C(C(N3CC(N(C)CC)C3)=O)F)C2)=O)CCC(=O)NC1 C(=O)(C1=Cc2ccccc2C1)N1CCC(NC(c2ncc(Cl)cc2Cl)=O)C(O)C1 C1(CN(C(CC2CC(SC)C2)=O)CC(=O)O)CCc2ncnc(C)c2C1 Cc1ccc(C(=O)NCCCNC(=O)CC2(C)CCCO2)c2c1NCCC2 Cc1cc(S(N)(=O)=O)oc1C(=O)NC1CCN(C(=O)Cn2cnnc2O)C(C)C1 C(=O)(C1=NOC2(CCC2)C1)N1C2CC(NC(Cc3ccc(C)cc3)=O)CC1CC2 CC1(C)COC(CCC(=O)NC2CC3(C2)CC3NC(c2coc(CO)c2)=O)C1 c1(C(N(C)CC2CCN(C(CSCC#C)=O)CC2)=O)cc(C(=O)OC)ccc1Cl N1(C(=O)NC2CC(Cc3n(CC)ncn3)C2)CCCC2CC12 C(CCCC)(CC(=O)NCC1(C)CCCC(=O)N1)NC(C(CC=CCC)C)=O C1(CCC)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN1C(=O)CC(C)O C(C(=O)Nn1cnn(CC)c1=O)N(C(=O)COC)CCC.C1CCCOC1 Cc1nc(Cl)sc1C(N1CCC(CC(=O)NCc2nccnc2Cl)C1)=O C12(C(=O)NC3CC(C(N4CC(C(F)(F)F)C4)=O)C3)CCCCC1C2 c1(C(=O)NC2(C(N(CCC(=O)NC3CC3)C)=O)CC2(C)C)cc(N)cc(F)c1 N1(C(C(CCC)N(C)C)=O)CC2CC(CNC(C3(SC)CCC3)=O)C2C1 C1(COCC)CC(F)(NC(=O)C(C)(C)c2cnsc2)C1.C1(C2CCC2)C(=O)N1 CC(CC1CCCCC1)C(=O)NC1(CNC(=O)COc2cccnc2)CCOC1 c1(COC)cccc(NC(=O)NCC(c2cccc(OC(F)F)c2)SC)c1 c1(C(N2CC(CNC(CN(C3CCC3)C)=O)OCC2)=O)cccc(N=[N+]=[N-])c1 N1(C(c2cc(CC)sn2)=O)C(C(=O)N(CC(C)N(C)C(C)=O)C)CCC12CC2 c1(CC(N2C(CCCNC(=O)C=CC(F)F)CCCC2)=O)ccn2cncc2c1 n1(CC)ncnc1C(N1CC(O)(CCNC(C2(C3CCCO3)CC2)=O)C1)=O CC1(C)CC(=O)NCC1C(=O)NCC=CCNC(c1ocnc1C1CC1)=O c1(C(=O)NC2(C3N(C(CCCC#C)=O)CCCC3)CC2)cnn(C)c(=O)c1 c1(CC)noc(CC)c1CC(=O)N(C(C)CN(C(=O)CCCCNC(N)=O)C)C C1(NC(C)=O)CC12CCN(C(=O)COC(c1ncsc1)=O)C2.C1(SC)CCCCO1 CN(C)S(=O)(=O)NC1CC1NC(=O)C(c1ccc(F)cc1)O C(CC(C)(C)C(=O)NCC1CCC(NC(C2CCCC3CC23)=O)CC1)OC N1(C(C(C2CCCCC2)OC)=O)CCCC(CC(N2CCC(C(C)O)CC2)=O)C1 O=C1Cc2cnc(N3CC4CC4(C(=O)Nc4cc(Br)ncc4F)C3)nc2N1 CCCCCC(O)C(=O)NCC12CCC(CC1)N(C(=O)CC(C)(C)O)C2 c1(C(N(CC(C)NC(C(C)C2CCC2)=O)C)=O)sc(Cl)cc1Br C1CCCCN1C(=O)CNC(=O)NC1CC1.C12(CCCC1)C(=O)N2.C(COC)OC c1(C(=O)NCC2(C)OCCN(C(C(C)OCOC)=O)C2)cccc2c1CC(=O)N2 c1(C(N2CCC(NC(c3nc(C)oc3)=O)C(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(CCCC)CCCN(C(c2ncoc2C2CCCNC2)=O)C1 Cc1c(C(=O)NC(CO)C(C)NC(c2cc(C3CC3)no2)=O)nn2ccccc12 c1(C(=O)NC(C(=O)NC)(C)C)ccc2c(n1)CCN(C(=O)C(O)C(C)C)C2 c1(OC)cncnc1C(=O)N(C)CC1(O)CN(C(=O)C(C)(C)c2ccccn2)C1 C1(C(=O)NCCC2(NC(c3c(CC)non3)=O)CCC2)CCCC1S(C)(=O)=O C1(CC(=O)NCC2COCC2O)CCN(c2ncccn2)CC1 Cn1cc2c(n1)CCCC2NC(=O)NCC(C(F)(F)F)n1cncn1 c1(N(C)CC2CCN(C(=O)CC3CCCOCC3)CC2)nc2ncc(Cl)cc2o1 C1(C(=O)NCC(CSC)OC)(CF)CCN(C(=O)CN2CC=CC2)C1 C1(CC(=O)N(CC(CC)NC(=O)C(C)(C)n2cccn2)C)CC(C)(C)CO1 c1(CCC(=O)NCC(CC)NC(C2CC2C(=O)OC)=O)ccccc1Cl c1(OCC)ccccc1C(C(C)CCCC1(CO)CC1)NC(=O)C(=O)N(C)C CC1(CS(=O)(=O)NC2COC(c3ccccc3)C2)CCCCO1 C(=O)(CCC(C)(C)C)N1CCC(CC=C)(NC(C2CC(=O)N(C(C)C)C2)=O)C1 N1(C(c2ncc(OC)nc2)=O)CC=C(C(=O)NCC2(O)CC(O)C2)CC1 c1(NC(=O)NC(C)C(=O)Nc2ccccc2)ccc(Cl)cc1CN(C)C CCC(C)CC(C(=O)NCCC1(OC)CCC1)NC(c1ncccc1CC)=O C=Cc1ccc(C(=O)NC(CN=[N+]=[N-])C(=O)NCCC2CCCC2(C)C)cc1 CC(CC(=O)NCC1CCN(C(C2CCC3(CCC3)CC2)=O)C12CC2)C(C)(C)C C(N=c1[nH]c(=NCc2ccc(F)cc2F)[nH]c2cc[nH]c12)C1N(CC)CCCC1 N1(C(c2c(C)non2)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(F)(F)C(C)(C)O c1(SC)nc(C(=O)NCCCCCN(C(=O)CSC2CC2)C)c2ccccn12 CC(F)(F)C(F)(F)CC(=O)NC1CCCC1NC(=O)CCc1ccccc1 c1(CC(N2CC(C)N(C(=O)Cc3cnn(C)c3)CC2)=O)cc(F)c(Br)cc1F N1(C(C2N(CC)CCC2)=O)CCCC(O)(CCNC(=O)CCc2cccnc2)C1 N1(CC)CCCC1CC(=O)NCCC(C)N(C(=O)CCc1nc(C)cs1)C N1(C(C2(S(C)(=O)=O)CCC2)=O)CCN(C(=O)C(C2CCCCC2)F)CC12CCC2 O=C(CC1OCc2cc(Cl)ccc21)NC1CN(C(C2CCCC2)=O)C1 C1(NC(c2cc(C(C)NC(C3CCC3CN)=O)on2)=O)CCCC1C1CC1 c1(OC)cc(N)c(C(=O)NCCN2CCN(C(=O)C=CC3CCC3)CC2)cc1F c1(OC)cc(C(=O)NCCN(CC(C)O)C(=O)Cc2cn(C)nn2)cc(Cl)c1 c1(C(=O)NC2CCC(NC(c3cn(CC=C)nn3)=O)C2)noc(C)c1C(=O)OC C(=O)(CCCCCC#N)N1C(CN(C(c2cnc(C)c(N)c2)=O)C)CCC1 c1(C(=O)NCC2CC(N3CCCC3)C2)cccc(S(=O)(=O)CC(F)(F)F)c1 c1(CCC(N2CC(C(=O)OC)C(N)C2)=O)c(I)ccnc1O C(CC)(CCCC(=O)NCc1nn[nH]c1C1CC1)NC(CSCCC)=O c1(C2(C(C)NCc3ccnc(Br)c3)CC2)c(F)cccc1F C(=O)(CC(C(F)F)NC(C1(C)CCN1C(=O)C(=O)N(C)C)=O)NC C1(C(=O)NCCc2c(C)nn(C)c2)CCN(C(c2cc[nH]c2)=O)CC1O N1(C(C2CC(C)C2)=O)CC=C(CC(=O)NCCn2cnnc2C)CC1 Cc1cn(C)cc1C(=O)NCCn1cc(-c2cccnc2C)nn1.C12CCCC1C2 CC1CCn2ncc(C(=O)NCCCC3(NC(=O)CCc4cc[nH]n4)CC3)c2C1 C(=O)(C1CCCn2cnnc21)NCC(CO)NC(CCNC(=O)NC)=O C1(NC(C2(SCC)CC2)=O)CN(C(=O)CNC(c2ccnc(O)c2)=O)CCC1C N1(C(CC=C)=O)CCC2(CC1)CCN(C(=O)C=C(C)C1CCCCC1)C2 Cc1nc2c(N3CC4(C3)CN(C(=O)C(O)Cc3ccc(O)cc3)C4)ncnc2[nH]1 C(C)(CO)(C(=O)NC1CC=CCC1)NC(Cc1c(CC)con1)=O C1(CNC(C2(C=C)CCCC2)=O)CCC2(CCC2)C1NC(c1cccnc1C)=O c1(C(N2CCC2CSc2ocnc2CO)=O)csc(-c2ccsc2)n1 c1(OC)cc(OC)nc(CC(N2CCC3C(NC(c4cn(C)cn4)=O)CC23)=O)n1 C(CN=c1ccc([N+](=O)[O-])c[nH]1)N(C(NNC(C)=O)=O)CCO C(=O)(CC(C)(C)C)NC(C)(CSC)CC.C1=CCNC1=O.CC=C C1(C(=O)OC)CCS(=O)(=O)C12CN(C(c1c3c(c[nH]c1=N)CCC3)=O)C2 C1(NC(C(=O)NCC(CC=C)NC(=O)OC(C)(C)C)(C)CO)CCS(=O)(=O)C1 N(C(=NCCCS(=O)(=O)c1ccccc1)NC1CCCn2nc(C)nc21)CC c1(C(=O)NC2(CNC(C3CCC4CCC34)=O)CCC2)nccc2[nH]ccc12 N1(C(C2N(C)CCC2)=O)CC2CC1CN2C(=O)Cc1ccncc1 C=CCCC(C(=O)NC1(c2ncc[nH]2)CC1)NC(C1CC(=O)N(C)C1)=O CN(C)S(=O)(=O)N(C)CC(N1CCCC(O)(CCNC(c2ccns2)=O)C1)=O c1(NC2(CC#C)CCC2)ccc(-c2ccon2)cc1 N1(C(c2ccc(C=C)cc2)=O)CCCC2CN(C(c3cccc(=O)n3C)=O)CC12 C1(CC(N2CCC2(C)CC(N2CCC(OC3CCC3)CC2)=O)=O)CCC(C2CC2)C1 C1(CNC(=O)CC2CC=CC2)CC2COCC2N1C(c1ccc2cc[nH]c2c1)=O C(CN1C(=O)C(=O)c2cc(F)ccc21)N1CCN(C(C(C)(C)C)CN)CC1 N1(C(C(C)n2cccn2)=O)CCC2(C1)CN(S(=O)(=O)c1ccn(C)n1)C2 c1(OC)ccc(C(=O)NC2CC2CNC(C2(F)C(C)(C)C2(C)C)=O)c(N)c1 N1(C(C(C=C)CC)=O)CCC(NC(c2ccc(C)o2)=O)CC1C1CC1 c1(N2CC(CC)SCC2)ncnc(NC(COC)COC)c1C C(=O)(CCC(C)(F)F)NCC1(COC)CN(C(c2cc(C)nc(C)n2)=O)C1 C=CCC(C(=O)N1CC(C(C)NC(C2(F)CCCCC2)=O)C1)c1ccccc1 c1(C(=O)NC2CC3C(NC(=O)CCn4ccnn4)C3C2)ccnc2ccsc12 CCC(CCCC(=O)N1CC(NC(=O)CC(C)C)C(F)C1)NC(=O)OC(C)(C)C c1(NC(C2CCNC(c3ccc(F)cc3Cl)C2)=O)cnc2c(c1)CCC2 C1(C(=O)NCCC2CCN(C(C3(CCC)CCC3)=O)C2)CC2COCC(C1)C2 N#Cc1ccc(C(N2CCN(C3CC3)CC2)C(=O)NCCC2CCC2)c(F)c1 C12(CNC(C(C#C)(C)C)=O)CCCC1N(C(c1nn(C)cc1C#C)=O)CCC2 CCCCCCC(F)C(=O)NC1CN(C(=O)Cn2cc(F)ccc2=O)CC1F N1(c2ccc3c(c2)CCC3)CCN(C(=NCCc2cnccn2)NC2CC2)CC1 c1(C(=O)OCC)ccc(C(N2CC3C(C2)C3(C)C)C(=O)NCCOC)c(Cl)c1 c1(C(=O)NC(CCC)C(=O)NCC(C2CC2)SC)nccc(C)c1F C1(C)(C(=O)NCc2cn(CC)nc2)CCCN1C(=O)CCC(=O)OC C(CC(C(=O)NC1(CCNC(=O)CCc2cn(C)nc2C)CCC1)N(C)C)SC N1(C(C(C)OCC(C)C)=O)C2CCC1C(CNC(=O)Cc1ccsc1Cl)C2 O=C(C1=CSCCO1)NC1CCCCC1CNC(=O)COc1ccccc1 Cc1ccc(C)c(OCC(=O)N(C2CCN(C(=O)C=CC3CCOC3)C2)CCO)c1 c1(C(=O)NC(C)CN(C(=O)CCSc2ccc(Cl)cc2)C)cccn(C)c1=O c1(C(=O)NCc2c(=N)cc[nH]c2)cnn2cnnc2c1 C12(C(=O)OCC(CCC(=O)OC)(C)C)CCCC1CC(F)(F)CC2 CN(C)S(=O)(=NCC(=O)O)NC(C1COC(C)(C)OC1)=O Cc1ccc(C(=O)OCC(=O)N(C(c2ccc(F)cc2)C)C(C)C)cc1 C1(C(=O)NCCC)CCCN1CCC(=O)NCCC(C)(F)F C12(CC)CN(C(c3coc(CO)c3)=O)C(CNC(=O)Cc3ccsc3)(C1)C2 N1(C(C=CCNC(C(C(C)C)C#N)=O)=O)CCCNC(=O)C1C(C)C C(C(C)(O)CNC(=O)COCC1CCCO1)N(C)C(c1cnn(C2CC2)c1)=O c1(OC)cccc(CCC(=O)NCCN(CC(C)O)C(C2CC(F)(F)C2)=O)n1 CN1N=C(CC(=O)N(C)CC2CN(C(c3ccc(F)c(C#N)c3)=O)C2)CC1=O CC(C)CCC(C(=O)NCC1C(CO)C1(C)C)NC(=O)CC(C)O C12CCCN(C1)C(=O)NCC2.C(CS(=O)(=O)Nc1ccn(C2CC2)n1)OC C1(F)(CNC(=O)C=CCn2cncn2)CCCN(C(C2CCS2(=O)=O)=O)C1 C1(C)(C(=O)NCCC2N(C(c3cccc(OC)n3)=O)CCOC2)CCC(=O)NC1 c1(CC)ccc(C(=O)N(CC(CC)NC(=O)C(C)C2(O)CCC2)CC)cc1 Cn1nc(O)cc1C(N1CC(CCCCNC(C2CCC(=O)NC2)=O)C1)=O C1(CC(N2CCCC2)=O)C2CCCC2N1C(=O)C(O)Cn1cncn1.CC(C)N CCCCC(CC(=O)NC1CC=C(C)CC1)NC(=O)CC1(CSC)CC1 C1(CCC(=O)NCC2(NC(C3CNC(=O)N3)=O)CCOCC2)CCC(F)(F)CC1 CCCCC(COC)NC(c1cn(CCNC(c2nnn(C)c2N)=O)cn1)=O C(=O)(CCC(=O)C(C)(C)C)NCCN(CCC)C(c1ccc(CN(C)C)nc1)=O N#Cc1cccc(Cl)c1C(=O)OCc1ccnc(O)c1 c1(C(N(CCNC(=O)CCCc2ccc(F)cc2)C2CC2)=O)cc(Cl)ccc1F CC1CC(NC(C2COC3(CCC3)C2)=O)CCN1C(=O)CC(F)(F)F N1(C(c2c(C)nc(CC)s2)=O)CC2CCC1CN2C(c1cc(F)c(F)cc1O)=O C1(C)(C(C)C)CCCN1N(CC1CCCO1)Cc1ccc2c(c1)CCC2 c1(CC(C)C(=O)NC2CCCC(CNC(=O)CC(C)(C)O)C2)ccc(Cl)cc1 CCC(CC)(CC)C(=O)NCC(C)NC(c1sc(-n2cccc2)nc1C(C)C)=O c1(C(N2C(CCCNC(COCC(=O)NC)=O)CCCC2)=O)cc2scnc2[nH]1 Cc1nn(C)c(=O)c(C(=O)NC2CCCN(C(=O)C(C(C)O)N(C)C)C2)c1C c1(C(=O)NC2CCCC(NC(C3C(=C)CC3)=O)C2)ccc2c(c1)CCCO2 n1(C(C)C)cnc(C(N2CCCC2CNC(C2CC2F)=O)=O)n1 c1(C(=O)NCCC(CNC(c2cnc3c(c2)CCC3)=O)O)cc2c(nn1)CCC2 C(N=c1nc(N2CCC(C)CC2)c2c([nH]1)CSC2)C1N(CCS(CC)(=O)=O)CC1 C1(C(=O)NC2CC(CNC(c3cc(COC)on3)=O)CC2O)CC12CCOCC2 N1(C(CC(CC)O)=O)CCCC(CNC(c2ccc(-c3cnco3)cc2)=O)CC1 C1(C(=O)NCC(CNC(COCC(=C)C)=O)CO)CC2CC(=O)C1C2 c1(NC)snc(C)c1C(=O)NC1CCC(NC(=O)CC2CCCC(C(F)(F)F)C2)C1 C(=O)(CC1CCc2cc(Br)ccc21)NCC(CNC(CCCC=C)=O)CO N1(C(c2cccc(CC=C)c2)=O)CCCN(C(=O)C(C)n2cccn2)CC1C c1(OC)ccc(C(N2CCN(Cc3cc4n(n3)CCC4)C3CC23)=O)cc1C C(C)(CCNC(=O)C=CCOCC(F)(F)F)N(C(C=CCC)=O)C N1(C(c2n(C(C)C)ccn2)=O)CCC2(CCCN2C(c2cc[nH]n2)=O)CC1 CCC(C)(C#N)C(=O)NC1CC(C(=O)NCc2ccc(N3CCNC3=O)cc2)C1 c1(C(=O)NC(CC(=O)NC2C(C)(C)C2C#N)C2CC2)cc2occc2[nH]1 c1(C(=O)NCC(CNC(c2c(C)c(Br)no2)=O)C)c[nH]c2cccnc12 c1(C(=O)NCCC2CCCN2C(=O)Cc2cc[nH]n2)sc(F)cc1Br Cc1ccc(NC(=O)C(C)NCCC2CCCC2(F)F)cc1 N1(C(C(CC)O)=O)CCC2(CCN(C(=O)CCN3CCc4ccccc4C3)C2)C1 C(C)(CN=c1[nH]c(=N)[nH]c(=NC2CCCC(C(C)(C)C)C2)[nH]1)c1ncc(C)s1 c1(C(=O)NC(CC=CC)C(=O)NCc2n[nH]cc2CC)cc(C#N)nn1C S(=O)(=O)(c1cc(C(=O)NCC2(NC(C3CC3CF)=O)CCCC2)ccc1F)NC CC1CCC(C)N1CC(N1CC=CCC1C(=O)NOCC1CCCO1)=O c1(C(=O)NC(CCCNC(CN(S(CC)(=O)=O)C)=O)(C)C)ccc2occc2n1 Cc1ncc(Cl)cc1NC(C1CCCC1NCc1ccc(-c2ccccc2)o1)=O C(CC(C)C)(C(=O)Nc1ccc(N(C)C)nc1)ONC(CCc1ccc(C)o1)=O c1(C(=O)OC)cnc(N2CC3CC2CN3C(=O)Cc2cnn(C)c2)nc1C C1(C)(C(N2CC(OC)(CNC(c3cn[nH]c3)=O)C2)=O)C=CCCC1 C1(CC(=O)NCc2c(C)cco2)CC(C)(C)CN1C(C12CC1CNC2=O)=O N1(C(=O)C=CC2CC2)CCC2(C1)c1[nH]cnc1CCN2C(C1CCCOCC1)=O c1(CCC=C)ccc(C(=O)N(CC(C)N(C(=O)C=Cc2ccncn2)C)C)cc1 c1(C(N2CCC(C)C2CNC(=O)C2=CCSC2)=O)ccc2c(c1)C(=O)NC2 c1(OCC=C)cccc(COC(C)=O)c1.C1CCSCCO1 C1(CNC(c2c(C)nc(C(C)C)o2)=O)CN(C(=O)C(F)CC2CCC2)C(C)(C)C1 O=C(C1=CCC(F)(F)CC1)NC1CCC(O)CN(C(=O)C2CC2)C1 c1(CC(N2CCCC(NC(C(CC)OC)=O)(CC)C2)=O)noc2ccccc12 C1(C(=O)NCC(C)NC(c2c(F)ccc(C)c2)=O)CCN(S(=O)(=O)N(C)C)C1 c1(C(=O)NCC2OCCCN(C(C=NOC)=O)C2)nc2ncc(Br)cn2n1 c1(CC)ccc(C(N2CCC(C(C)NC(C3(C)CCN(C)C3)=O)CC2)=O)c(O)c1 C1(C(=O)OCC)C2CC(CN(C(=O)C(C)(C)O)C2)N1Cc1csnc1C C#CCCN=C(NCC#CC1CC1)NC(C1CCCO1)C c1(C(=O)NC2CC(CNC(CC3C(C)CCC3)=O)C2)cccc(=O)o1 C1(NC(CC=CCC)=O)CCC2(CCN(C(c3n[nH]c(CC)n3)=O)C2)C1 C1(OCC)CCCCC1NC(C1(NC(=O)CCC2CCCCC2)CC1)=O c1(C(=O)OCC)cncc(C(=O)NC2CC(NC(c3nn(C)cc3Cl)=O)C2)c1 c1(CN2CCC(NC(c3ccccc3CO)=O)C2)ccc(Cl)cc1-n1ccnc1 N1(C(CSC)=O)CCCC(CCNC(C2CCN2C2CCCC2)=O)C1 c1(C(=O)NCC(CC)(C)NC(C2(N(C)C)CCC2)=O)cc(OC)cc(OC)c1 C(C(CC(C)C)C(=O)NC1CC2(C1)CC2C(N1CC(N(C)CCO)C1)=O)OC CCC(C)C(C(=O)NC1CNC(=O)C12CC2)NC(c1csc(=N)[nH]1)=O C1(CNC(C(c2ccccc2)C)=O)(CNC(C2CCSC2)=O)CC1(F)F N1(C(=O)OC(C)(C)C)CCC(C(=O)NC2CCCCC2)C(F)C1O C1(OC)(CNC(C2COCCN2C)=O)CCN(C(c2nc(Cl)cs2)=O)CC1 Cc1ccc(F)c(C(N2CCC3CN(C(C4(C)CCC(=O)CC4)=O)CC23)=O)c1F c1(C(N(C(CCNC(C(C(CC)O)(C)C)=O)C)C)=O)cc(C)c2c(O)n[nH]c2n1 CC1(C)CN(CCC(N2CC(O)(CCNC(=O)Cn3cnc(=N)[nH]3)C2)=O)CCS1 N1(C(C2C(C)CCC2)=O)CC2(CCCCN2C(=O)CCn2ccnc2)C1 c1(C(=O)NCCNC(CC2N(C(C)=O)CCC2)=O)cccc2c1CCC2 N1(C(c2c(C)con2)=O)CCCC2(C1)CN(C(=O)Cc1ccns1)C2 N1(c2cc(SCC)ncn2)CC2CN(C(c3ccncc3O)=O)C2C1 CC1(C(=O)NC2(C(F)(F)F)CC2)CC(O)CN1C(c1ccsc1)=O C(=O)(C(CCCC(C)C)N1CCOC(c2cccc(S(N)(=O)=O)c2)C1)OCC C12COCCN1C(=O)CC(C)NC2=O.C(CC(=O)NC(C)(C)C)N(C(C)=O)C CC12CC(C(N3CCC(NC(c4ccccc4F)=O)CC3)=O)(C1)C1(CCC1)O2 C1(C(N(CCC)CCO)=O)CC12CCN(C(c1sc(F)cc1C)=O)C2 N1(C(c2ncc(OC)cn2)=O)CC(NC(c2cc(Br)c(C)o2)=O)C2(CC2)C1 CCCCC(CNC(c1ccccc1OC(C)C)=O)NC(=O)CCCF C(=O)(CCCCCC#N)NCC(C(=O)NCCN1CCC2CC12)N(C)C C1(C2CCCN(C(c3ccc(N)cc3)=O)C2)(NC(CCC=C(C)C)=O)CC1 C(=O)CCCCCC(C)O.C(CC(=O)N1CC(NC)C1)OCC(C)C CC1(CNC(=O)C(CNC(C2CCC=CCC2)=O)CC2CCCC2)CCCC1O C1(CNC(CC(c2ccc(C)cc2)C)=O)CC(F)(F)CN1C(=O)C(C)CF N1(C(c2c(=O)ccn(C)c2)=O)CCC2(NC(=O)Cc3ccsc3)CCCCC12 C1(CNC(C(CCOC)C)=O)(NC(=O)CCC(C)SC)CCC(C)(C)CC1 CC1(NC(=O)Nc2ccc(N3CCC(C(F)(F)F)CC3)cc2)CCC(CO)CC1 N1(C(CC2CCN(C(C(=O)NC3CC3)=O)CC2)=O)CCC(O)C(F)(F)C1 c1(-n2ncc(OC)c2)nc2ccc(C)cc2s1.C12(CO)CCCN(C1)C(=O)C2 N1(C(C2CC(CC)C2)=O)CCCCC(NC(c2cccnc2SC(F)F)=O)C1 n1(CC)nc(C(=O)NC2COCC2C(N2CCSCC2CO)=O)cc1O CCCCC(C)C(=O)NC1CN(C(c2cnc(Cl)cn2)=O)CC1(C)C N1(C(C23CC(CC)(C2)C3)=O)CC2CN(C(C3(C)C=CCC3)=O)CC2C1 C12(C(=O)NC3C(CNC(=O)CCCCC4CC4)CCCC3)CCCC1OCC2 CCC(CC)C(F)C(=O)NC(CNC(=O)CSC)C1CC1 Cc1cc(C(N2CCCC(CO)(Nc3ncnc4sccc34)C2)=O)cc(C)c1F CN1CCCCC(C(N(CCOCCC(=O)NCC2(C)CCC(=O)C2)C)=O)C1 C(=O)(C(CCC(N)=O)N(C)C)N(CC(CC)NC(C1CN(C)CC1C(F)(F)F)=O)C Cc1cc(=NC2CCCN(C(=O)C(F)C3CCOC3)C2)[nH]cc1C#N Cc1nccc(C(=O)NC(C)CCNC(c2ncsc2Br)=O)c1Cl C1(C(=O)NC2CC(CNC(c3ncccn3)=O)C2)CCn2ncnc2C1 C(CC(C)N=c1cc(C)nc(N2CCC(Oc3ccc(CO)cc3)CC2)[nH]1)SC CCC(CC)(CCNC(C1CCCC1C(F)(F)F)=O)NC(c1cnnn1C)=O N1(C(=O)CSC2CC2)CC(NC(C2(C3CCCCO3)CCOCC2)=O)CC(F)C1 n1(CC(=O)NCCN(C(=O)C(F)CC2CC2)C)c(C(F)(F)F)nc2ccccc12 c1(C(=O)NC2C(C(=O)NC(c3cn(CC)nc3)C)OCC2)sc(C)cc1C c1(NCCN2CCN(C(C3(C)CCN(C(C)=O)C3)=O)CC2)ccc(Cl)nc1O N1(C(C(=O)Nc2cc(F)cc(Br)c2)=O)CCc2nc3ccccn3c2C1 Cn1cc(NC(=O)C(c2ccco2)NC(=O)C(N2CCOC2=O)C)cn1 CN1C(=O)COCC1CNC(C1CN(C(C2CCCCC2F)=O)C1)=O Cc1nc(N2CCC(C)C2CNC(c2cc(C(N)=O)[nH]n2)=O)cc(O)n1 c1(CCC(=O)NCC(CNC(Cc2ccc(C)o2)=O)C)ccc(=N)[nH]c1 C=CCCCCCCC(=O)NCC1CCCCN1C(=O)CC1CC2CCC1C2 N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(CCC(NC(C3CC3c3ccco3)=O)C2)C1 C(=O)(C(N)CN(c1ccco1)CCCN(CCCO)Cc1ccccc1)N(C)C C(C(C(=O)N1CCC(C(C)NC(C2CCN(C)C2)=O)C1)C(C)(C)C)OCC(=C)C C=CC1CN(C(c2cccc(N)c2)=O)CC1NC(c1csc(-c2cnc[nH]2)n1)=O c1(C(=O)NC(CN(C(C(C)OCCCC)=O)C)(C)C)ccoc1Br C1(C(=O)NCC(CNC(c2n(C)ncc2)=O)(C)O)CC2(CO1)CC(F)(F)C2 C1(C(C)C)CN(C(=O)C(O)C(F)(F)F)CCCN1C(c1ns[nH]c1=O)=O C(=O)(C(F)(F)CC)N1CCC(OCCNC(C23CC(CC)(C2)C3)=O)C1 c1(CC(N2CC3C(NC(c4csc(Br)c4)=O)(C3)C2)=O)n[nH]c2c1CCCC2 C1(C(C)NC(C=C(C=C)C)=O)CCCN(C(=O)C(c2cccc(OC)n2)(F)F)C1 c1(C(=O)NC(C)CN(C)C(c2cccc(C(N)=O)c2F)=O)cc(Cl)c(N)c(Cl)c1 C(C(C(=O)NC1CC(O)C1OC)NC(c1cnns1)=O)OC CC1CN(C(=O)C2=CCCSC2)CC(C(=O)Nc2ccc(F)cc2Cl)O1 c1(OC)ccc(-c2ccc(CNC(=O)CCc3ncccc3Cl)cn2)cc1OC Cc1nc(C(=O)NC(C(N2CC(S(C)(=O)=O)C2)=O)C2CCC2)ccc1C#N c1(CC)oc2ccccc2c1C=CC(=O)NCCNC(=O)C=C(C)C1CC1 C(C(C)(O)C(=O)N1CCC(CF)(NC(=O)CSc2ccncc2)C1)OC C1(C(C(=O)NCCCC(C)NC(Cc2c(C)scc2)=O)(C)C)CCCN(C)C1 c1(NC(CC2CC(C)N(C(=O)CC3C(C)(C)C3(C)C)C2)=O)cc(Cl)cnc1O Cc1cccc(OCC(N2CCCC(C(=O)Nc3ccc(Br)nc3)C2)=O)c1 c1(C(=O)NC2(CC)CCCN(C(=O)CC(C)CF)C2)nccc2occc12 C(=O)(C(C)(C)CCC#N)NCC1C(C)CN(C(=O)COCC(F)F)CC1 C(=O)(CCCCCCNC(C1CCCS1)=O)NCC(C)Cn1cccn1 Cc1nn(-c2ccc(Cl)cc2)cc1C(=O)NC1CCCN(C(C2CC23CC3)=O)C1 C1(CC)C(NC(c2cc(C3(C)CC3)on2)=O)CCCN1C(=O)Cc1ccc(C)s1 N1(C(C=C(C)Cl)=O)CCC(NC(=O)CCSc2ccc(F)c(F)c2)C(F)(F)CC1 N1(C(C(C)=O)=O)CCn2c(C(N3CCC4(CNC(=O)O4)C3)=O)cnc2C1 N1(C(C2(C)ON=C(C)C2)=O)CCC(C)(NC(C2CCCC(C(F)(F)F)O2)=O)CC1 C(=O)(C1CCc2c[nH]nc21)NCCOC(C)(C)CNC(c1cncc(Cl)c1)=O N1(C(COCCC)=O)CC2(CCCCN(C(C3CC34CC(C)(C)C4)=O)C2)C1 Cc1c[nH]c(C(=O)NCC2(CCNC(c3c[nH]nc3C(F)(F)F)=O)CC2)c1 N1(C(c2ccncc2Cl)C(=O)NC)CCN(C2=NCC(C)S2)CC1 Cc1ccc(C(=O)N(C)CCN(C(=O)C(c2ccc(Cl)c(F)c2)O)C)cc1Cl c1(NC2CCC(NC(C(C)C3CCCC3)=O)CC2)ncc2c(n1)CCCC2 C=C1CCC(C(=O)NCCSCc2ncc(C)s2)C1 N1(C(CCN(CCCO)C(c2c(CC)n[nH]c2)=O)=O)CCC(C)C(C)C1 c1(C(=O)NCC=CCNC(C(CC)N(C)C)=O)cnn2c1CCCC2 N1(C(CC(COC)C)=O)CCC(F)(CNC(=O)CC(C)C(F)F)CC1 c1(CN(C(=O)CC2(C)CCN2C(=O)CSC(F)(F)F)C)ncccn1 c1(NC(=O)NC(CNC(C2CCN(C(CC)=O)C2)=O)CO)scc(C)c1Cl C1(C(=O)NCC2CC3CN(C(c4scc(C)c4C)=O)CC32)CN2CCN1C(C)C2 Cc1cn2c(C(=O)C(=O)NC3(C(=O)N(CC(C)N)C)CC3)c(C)nc2s1.C(C)(C)N C1(NC(c2c(CC)c[nH]c2)=O)CC2C1CCN2C(=O)CCC1C(=O)ON=C1C c1(C(=O)NC2CCCCN(C(C=C(COC)C)=O)C2)c(Cl)ccc2ncccc12 Cn1nnc2cc(C(=O)NC3CCCC3NC(=O)Cc3cccnc3Cl)cnc12 CCCCCC(O)CC(=O)N(C)CC1CCCN(C(=O)CC(C)(C)F)C1 c1(OC(C(=O)NC(CC=C)CNC(c2ccoc2Cl)=O)C)ccccc1OC C1(CC(C)Nc2ccn(C3CCCNC3)n2)CCCCN1 C(=O)(C(C)OC)N(CCNC(=O)CCNC(=O)OC)CC N1(C(C(C)n2ccnn2)=O)CC(C2CC2)(C(=O)NCC2CCOCC2(C)C)C1 Cc1ccc(C=CC(=O)NC2C3CN(C(=O)CCc4nc(=N)[nH][nH]4)CC23)o1 c1(C(=O)NCCC2N(C(c3ncn(C)n3)=O)CCC2)nn(C)c2ccc(F)cc12 C=CC1(CC(=O)NC2CN(C(C)=O)C2)CN(C(=O)NCCN2C(=O)CCC2=O)C1 N1(C(C(c2ccc(Cl)s2)C)=O)CC(F)(CNC(=O)C=CC2CCCO2)C1 C=CC1(CNC(=O)CC2CCN2C(c2cc(COC)on2)=O)CCOCC1 C(C(=O)Nc1cc(C)ccc1O)(C(C)CC)N(C(c1c(CC)[nH]cc1)=O)C N1(C(c2ccc(OC)cn2)=O)CCC(C)(C)C1C(=O)NCCN1C(=O)CNC1=O C1(C(N2CC(OC)C(F)C2)=O)CCCC12CCN(c1ccnc3ccnn13)C2 c1(C2CC(=O)NN2)ccc(F)c(NC(=O)CCc2cnccn2)c1 C1(CNC(C(CC)(C)CO)=O)CCC2(CN(C(C3CSC3)=O)C2)O1 N1(C(C=CCC)=O)CCN(C(c2cncnc2CC)=O)C(CCC)C1 C1(NC(c2cc(OCC)c(C)cc2)=O)CCN(C(=O)CNC2CC2C)CC1(C)C C1(OC)CCC(C(=O)NC2COCC2F)N(C(=O)OC(C)(C)C)C1 CCC(O)C(C)C(=O)NCCN(C)C(c1cc(C)n(C)c1C)=O c1(C(=O)NC2CCCC(NC(=O)Cc3cnc[nH]3)C2)cc2ccc(Cl)cc2[nH]1 c1(C(N(CC(CC)(C)OC)C)C)cccc(F)c1F C1(NC(CS(=O)(=O)NCC)=O)CC2CCC(C1F)N2C(C1CC1C#N)=O C12(C(=O)NC3(C)CC(NC(Cc4c(C)noc4Cl)=O)C3)CCC(F)(CC1)C2 C12(CN3C(C(=O)NCc4cnn(CCO)c4)(CC)CCC3)CCC(F)(CC1)C2 c1(CC(=O)OCCc2ccsn2)c(F)ccc(Cl)c1Br c1(CC)ncc(C(=O)NCc2nc(C(=O)NCc3nc(=O)o[nH]3)co2)cn1 C(C1CCOCC1)=CC(=O)N(C(C(N1CC(C)(C(=O)OC)C1)=O)C)C1CC1 C1(C(N2CC3(CN(C(C)(C)C)C3)C(CO)C2)=O)CCN(C(=O)CCS(C)(=O)=O)O1 CC1(C(=O)NC(CC(=O)NCCC2(C)CC2(F)F)C2CC2)CC(=O)C1 C12C(C1(C)C)C(=O)N2.C(C(C)(O)CSC)NC(CN(CCOC)C)=O c1(CNC(CC)=O)ccc(-c2nnc(CN(C(=O)C(C)O)C)n2C(C)C)cc1 N(C(=NCCN1CCCC1)N1CCC(C2(O)CC2)CC1)C1CCCC(OC)C1 c1(OC(C)C)ccc(F)c(C(N2CCC(NC(=O)C(C)C(F)F)C2)=O)c1F C(C(C)N=c1[nH]c(=NCC2CC2)[nH]c2ncn(C)c12)(c1ccc(C)cc1)C1CC1 CCCC(C(=O)N1CC(OC)C(NC(c2cc(F)n[nH]2)=O)C1)OCC CCCC(C)(C)CC(=O)NCCCOCCN(C)C(C1(CO)CCOC1)=O CN1CCCCC(CNC(C23CC2CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C3)=O)C1 C12(NC(c3c(C)nc(O)[nH]3)=O)CCCN(C(C3(CC(C)C)CC3)=O)CC1C2 c1(OCC)ccc(N2CC2=O)cc1.n1(CC(=O)N(C(CC)C)C)cnnn1 N1(C(C(C)NC(=O)Cn2cnnn2)=O)CC=CC1CNC(=O)Cc1ccon1 C1(C(=O)Nc2c(C(=O)OCC)occ2)CN(C(=O)Cc2cccc(C)c2)CC1C Cc1n[nH]c(C)c1SCC(=O)NC1CCCC(NC(=O)CC2CCC(C)CO2)C1 C1(CCNC(c2c(CC)csc2)=O)CCCCN1C(=O)Cc1nncn1C(C)C Cc1nc2cc(NC(=O)CC3COCCN3C(c3sccc3F)=O)ccc2o1 c1(CC(C(=O)NCC(CN(C(=O)COC2CC2)C)(C)C)(C)C)ccc(C#N)cc1 N1(C(CC)=O)CCC(C)(NC(=O)NC2CC(OC(C)(C)C)C2)C1 N1(C(C2(NC(CCOCCOC)=O)CCCC2)=O)CC2(CC(CO)CO2)C1 CC1CN(C(c2ccc(Cl)cn2)=O)CC(C)C1Nc1nc(Cl)ncc1Cl C1(C(=O)NCC(CN(C(Cn2c(C)ncc2)=O)C)O)CC12CCC1(CC1)CC2 CC(C)CS(=O)(=O)CC(=O)N1CC(CNC(c2csc3cccnc23)=O)CC1C Cc1ccc(C)c2c1N(c1ccc(Br)cc1C(F)(F)F)CCC2 N1(C(CCNC(COC)=O)=O)CC2CC(NC(=O)CCc3ccncc3)C1C2 C1(CNC(CC(COC)(C)O)=O)CC2(CCC2)CN1C(=O)CCc1cc(C)on1 C(=O)(C(F)(F)Cc1ccc(Cl)cc1)N1CC(C(C)(C)C)C1 N1(C(=O)NC(c2ccc(O)cc2)C)CCC(Cc2ccccc2Cl)CC1 CCCC(CCC)CC(=O)NCC=CCNC(=O)CCc1ncc[nH]1 C(CCC(N)=O)(C(=O)NC(C)(CNC(=O)CCCCCF)C1CCC1)NC(C)=O c1(C(=O)NC23CC(NC(=O)C(O)C(F)F)(C2)C3)cc(F)cc(F)c1O C1(NC(C(C)SCCCC)=O)CC(NC(C2CC=CCO2)=O)C(O)C1 Cc1c(C(=O)NC2C3CN(C(c4cc(F)ncc4Br)=O)CC23)cncc1Br N1(C(c2cc(OC(F)F)cc(F)c2)=O)CCCC1C1CCCN1C(=O)C(Cl)=CCl c1(OCC)nc(N2CC(C(C)NC(=O)C(C)(C)c3ccccc3)C2)ncc1Cl N1(C(CC2(C)CCOC2)=O)CCCN(CCNC(C2CCCN2C(N)=O)=O)CC1 N1(C(CCSC)=O)CCC2CCCC(C1)N2C(=O)CCc1cnn(C)c1 C1(CC(=O)NC2CN(C(CC(CC=C)(C)C)=O)CC2F)Cn2ccnc2NC1=O c1(C(N2CCN(C(c3c(CC)[nH]c(=N)s3)=O)CC2)=O)cc(C)ncc1C CS(=O)(=O)c1c[nH]ccc1=NC(=O)N(CCN1CCOCC1)CCO C(=O)(C1CCc2c(Cl)cccc21)NCC1N(C(CC2CC=C(C)CC2)=O)CCC1 N1(C(C(CC)(C)OC)=O)CCN(C(c2ccc(C3CC3)s2)=O)CC12CC2 C1(NC(c2ccc(OC)nc2Cl)=O)C2CCC1CN(Cc1ccnn1C)C2 N1(C(C=C2CCC(C)CC2)=O)CCN(C(C2CCC(=O)CC2(C)C)=O)CC(O)C1 Cc1ccc(S(N)(=O)=O)c(C(=O)NCC2C3CN(C(C45CC(CO4)C5)=O)CC23)c1 N1(C(C2(OC(C)C)CCC2)=O)CCOCC2(COCCN2C(c2ccc[nH]2)=O)C1 c1(C(=O)NCCC(=C)CNC(C2CC2C)=O)cc(Br)cc2scnc12 CC1(C)C(CC(=O)NCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1O N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC1(C)CN(C(=O)CN2OC(C)(C)CC2=O)C1 C1(C(=O)NCCN(C(c2cc3cnccc3[nH]2)=O)CC)OCC2COCCC12 C(CCC(O)C(=O)NOCCN(C)C)NC(c1cnc(OC)s1)=O CC(C)(CO)C(CNC(=O)C(=O)Nc1cccc(F)n1)c1ccco1 C(=O)(C(C)(O)CSc1cccc(F)c1)N(CCCNCC)NC(=O)C(C)OC CCC(CC)C(C)C(=O)NCC1CN(C(=O)Cc2cc(F)ccc2OC)C1 N1(C(c2c(C)nc(C(C)C)cc2)=O)CC2CN(C(c3cnoc3C)=O)CC2(C)C1 N1(C(CCC(N)=O)=O)C(C(=O)NCc2cc(O)cc(F)c2)CCC12CC2 C1(C(N2CC(CC#C)OCC2)=O)N(C(c2cc[nH]n2)=O)CC12CCCC2 C1(CC(=O)NCCC(C)N(C(c2cn(CCC=C)nn2)=O)C)CCCC(=O)C1 Cc1cc(C)n2ncc(C(=O)N(C)Cc3nc4ccccn4n3)c2n1 c1(CC(=O)NCCN(C(CC(C(C)C)OCC)=O)C(C)C)ccccc1[N+](=O)[O-] C(=O)(C1=C2CCN=C2NC=C1)N1CC2OCC(NC(CCSC)=O)C2C1 C1(C(=O)NCC(CCOC)NC(c2ccc(C(N)=O)cc2)=O)CC=C(C)CC1 N1(C(C2(CC)CC2)=O)CCC(C)C(NC(c2cc(C3CCCCC3)[nH]n2)=O)C1 c12ccc(cc1)CN1CCC(C1)CNC(=O)CCO2.CCCCCOC(F)(F)F c1(CC(=O)NCC(N(C(C2C(=C)C2)=O)C)C2CC2)c[nH]c2cccc(OC)c12 CC1(CO)CC(O)CN1C(C1CCC1)=O.O1NC(=O)CNC(=O)C1 CCCC(CC)C(=O)N1CC(CNC(=O)CNC(C)=O)C(C)C1 C1(CNC(c2c(CC)occ2)=O)CN(C(=O)CSc2n[nH]c(C)n2)CCO1 C1(C(N(CCCNC(c2ccc(C(C)C)o2)=O)C2CC2)=O)CC2(C1)CC21CCC1 CCCCC1CC(=O)N1.C12(NC(=O)C=C(C)COC)CC(C1)C2 c1(OC)ccc(Br)cc1NC(=O)NC(c1nc(C2CC2)no1)(C)C N1(CCN(C(=O)C(=O)Nc2scc(C)c2)C)CCc2c(Br)cccc2C1 N1(C(C(C)n2cnnn2)=O)CC2(CCC2CNC(c2cc(Br)no2)=O)C1 c1(C(C)C)ncoc1C(=O)NCC#CCNC(c1cc(Cl)ns1)=O C(=O)(C(O)C(C)(C)CC)N(C1CC2CN(C(CN(C(=O)OC)C)=O)C1C2)C C1(OC)CCCCC1C(N1CC(C(C)NC(c2cc(CC(C)C)nn2C)=O)C1)=O CCCCC(F)C(=O)NCC1CCCCC1C(=O)NOC1CCC(O)C1O CN1CCC2CN(C(=O)CC3(CNC(=O)C=Cc4ccoc4)CC3)CC2C1 Cc1c(C(=O)N(C)CCNC(=O)CCCc2nccs2)cccc1F C1(CC(=O)NCC2(C)CC(NC(c3c(SC)ccs3)=O)C2)C(=O)NN=C1C CC(CC(F)(F)F)C(=O)NC1CCC(CNC(c2ccc3[nH]ccc3n2)=O)CC1 c1(C(=O)NCC(CNC(c2cc(C)nc(O)n2)=O)F)ccnc2cc[nH]c12 Cc1nc(=NC2CC(NC(C34CC5CC(CC(C5)C3)C4)=O)C2)[nH]c2ccccc12 C#Cc1cccc(CC(=O)N(CCCCN(C)C(C2(C)CC2(F)F)=O)C)c1 N1(C(C=Cc2ccn(C)c2)=O)CCCC12CCN(C(C1CCC(C)(C)CO1)=O)C2 N1(C(c2[nH]cc(C#N)c2)=O)CCC(O)CC1C(=O)NC1CCC(F)(F)CC1 C1(C(=O)NCC2(C(N3CC(CN(C)C)C3)=O)CCCO2)COCC1(C)C C1(C)(NC(C(C)SCC)=O)CCN(C(=O)C2=C(C)OCC2)CC1 c1(C(=O)NC2(C)CC(NC(c3cnc4ccnn4c3)=O)C2)cnc2[nH]cnc2c1 N1(C(c2c(C)snc2)=O)CCCC(O)(CNC(c2ccc(CCF)cc2)=O)CC1 C1(CNC(C(C=C)(F)F)=O)(CO)CC12CCN(C(c1coc(OC)n1)=O)CC2 c1(C(=O)NC(CC)(CNC(C2(C)COC2)=O)CC)cc(Cl)c2ccncc2n1 c1(C(=O)NC2C(OC)CN(C(C3C(C=C)C3)=O)C2)cc2c(F)cccc2s1 Cc1cccnc1C=CC(=O)NCC(C)N(C(=O)CC(C(F)F)n1ccnc1)C c1(CC)cscc1C(=O)NC1CCCC1CC(=O)NCC1SCCS1 C1(CNC(C2(CC)CN(C(C3CC(O)CN3C)=O)C2)=O)COCC(C)O1 C1(NC(c2ccc(COC)o2)=O)CN(C(=O)C(F)CC2CCOC2)CC1C c1(C(=O)NCC(CO)NC(c2ccc(C)cc2O)=O)cc([N+](=O)[O-])c(C)cc1C C1(CC2CCN(C(=O)NC3(C)CNC(=O)C3)CC2)CCC(F)(F)CC1 c1(C(=O)NCC(F)CNC(C2CC=CCC2)=O)c[nH]cc1Br C12(NC(=O)C3=COCCO3)CCCC(CN(C(C3CC4(C3)CC3(CC3)C4)=O)C1)C2 c1(C(N2CC(C)C(CNC(=O)C(C)N(C)C)C2)=O)cc2cccc([N+](=O)[O-])c2[nH]1 N1(c2cc(NC(c3ccc(F)c(Cl)c3)(C)C)ncn2)CCOCC(O)C1 N1(C(C2CC2N(C)C(C2CCCCC(=O)N2)=O)=O)CC2(CC(NC(C)(C)C)C2)C1 Cc1[nH]c(Cl)nc(=NC2CN(C(C3C4CC5C(C4)C35)=O)CC3(CCC3)C2)c1C#N N1(C(=O)Cc2cc[nH]n2)CCC2(CC1)CN(C(c1cc(F)cc(Cl)c1O)=O)C2 Cc1cc(C(=O)NC(c2cccc(C(=O)O)c2)Cc2ccccc2)nn1C Cc1cc(NC(=O)C(=O)NC(c2cnn(C)c2)CN(C)C)c(C)s1 CCC(C(=O)NCc1csc(C(=O)NC(c2ncc(C)s2)C)c1)OC N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCC(C(C)C)CC2)=O)C1 N1(N(c2ccccc2)C(CC(CCCC(N)=O)(F)F)=O)CCC(c2cccnn2)C1 C1(OC)(CNC(C2CC2CNC(C2CCC2)=O)=O)CCCC1 N1(C(C2(C#C)CCCC2)=O)CC2CC(NC(C3(C)CCN(C)C3)=O)C1C2 C1(CN(C(=O)CC2CC(F)C2)CC)CCN(C(=O)CC2(N(C)C)CCCC2)CC1 C(=O)(C(C(C)C)n1ncc(N)n1)NCC(=C)CCNC(C1C=CCC1)=O c1(Cn2cc(-c3c(COC)c(Cl)cc(Cl)c3)nn2)n[nH]c2cccc(C(N)=O)c12 C1(C(=O)NCC(CC)(CC)NC(=O)C(C)N2CC(C)C2)CC2C=CC1C21CC1 C1(CNC(C=CCOC)=O)CN(C(c2sc(OC)nc2Cl)=O)C2COCC2O1 Cc1ccc(C(N2CCC2(C)CC(=O)NC23CCC(CC2F)C3)=O)c(C)c1 C(=O)(C1Cc2ccc(Cl)cc21)NCC1N(C(c2ccc(OC)cc2O)=O)CCC1C N1(C(c2c(N)non2)=O)CCOC(CNC(C2CC3CC3C2)=O)C1 C(CC(CNC(=O)C(C)(C)NC=O)NC(=O)C(Cc1ccsc1)NC=O)OC c1(C(=O)NCC2C3CN(C(C4CC(=O)N4)=O)C2CCC3)ccc2cnccc2c1 C12(NC(CC3(C=C)CN(C(=O)CC(C)C4CC4)C3)=O)CCCC1OCC2 CC1=NOC(C(=O)N(C2CC(C(=O)NCCc3cnc(C)[nH]3)C2)C)C1 CC(C)C(Cc1ccccn1)N=c1cc[nH]c(=NCCCCF)[nH]1 N1(C(c2cccc(C)c2O)=O)CCC(C2(NC(=O)C(n3cc(Cl)cn3)C)CC2)C1 Cc1cc(C(N2CCN(CCNC(c3ccc(F)s3)=O)CC2)=O)c2c(c1)CCC2 CC(CS(C)(=O)=O)C(=O)NCC(C1CCC1)NC(=O)CCc1ccc(O)nn1 CC1CN(C(=O)CC2CC2C(F)(F)F)CCCN1C(=O)C=CCO C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC1(O)CC(NC(C(=O)N(C)C)=O)C1 CCC(CC(=O)N1CCCCC(NC(C2CCC2)=O)C1)C(C)(C)C.C(C)=O C12(C(=O)NC3CCC(NC(CC(CN(C)C)O)=O)C3)CC3CC1C2C3(F)F n1(CCC)nccc1C(=O)NC1CCCC1CNC(=O)C(C)Cc1cnc[nH]1 c1(C(=O)NC(CCNC(c2cc(OCC)no2)=O)C)cnn(C)c1CC c1(NS(CCC2CC(OC)(OC)C2)(=O)=O)cc(Cl)c(F)cc1[N+](=O)[O-] O(N(C(=O)C1CCCCN(C(=O)C(C)C(C)C)C1)C(C)C)CC N1(C(C2(OC)CCC2)=O)CC(C(F)(F)F)C(CNC(C2CCN(C(C)C)CC2)=O)C1 C1(CCNC(c2n(CCCC)nnn2)c2cscc2F)CCCS1(=O)=O Cc1ccc(C(CCO)Nc2cc(NCC3CCCS3(=O)=O)ncn2)cc1 CC1(C)CC=C(C(=O)NC2CC2NC(C2CC3(C2)CC(C)(C)C3)=O)CC1 CCC(C)CC(C(=O)N1CCCCC1CCCO)NC(=O)CC(C)(C)C(C)=O c1(C(N2CCCC(N3CCN(C(C4CCC4)=O)CC3)C2)=O)ccc(F)cc1F C12(C(N3CCC(C#N)(F)C3)=O)CCCC1CN(C(=O)CC1(O)CCOC1)C2 c1(OC)ccccc1NC(=O)C(c1cccc(Br)n1)N1CC=CCC1 c1(NC(=O)CC2C3CN(C(c4ccc(CO)o4)=O)CC23)ccc2n[nH]cc2c1 N1(C(C(C(C)C)O)=O)CCC(n2cccn2)(CNC(c2cc(C#N)cs2)=O)CC1 N1(C(c2ccc(C(C)=O)s2)=O)CCOCC1CNC(=O)C(C1CCOCC1)C c1(NC(C)=O)cc(S(=O)(=O)NC(C2CCOCC2)C(=O)OC(C)=O)ccc1N c1(C(N(CCNC(C=CC(=O)OC)=O)C2CC2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 c1(NCC)ncccc1S(=O)(=O)NC1(c2nnnn2C)C(CC)CCOC1 N1(c2nc3ncn(C)c3cn2)CC2C3CCC(C2C1)N(C(=O)C1=CCOCC1)C3 C1(C(N2CCCC(CCNC(C3(C)CC3(F)F)=O)C2)=O)CCCC12CCOCC2 C(CN=C(NCC(c1cccs1)(C)C)N(C)CC1CCC1)N1CC(C)CC(C)C1 c1(N(CC(CN(CC)CC)O)CC)cccc(C#N)c1 c1(C(=O)NC(CCC)CC(=O)N(CC(C2CC2)OC)C)cccc2[nH]ncc12 N1(C(C(=O)NC2CC(C)N(C3CC3)C2)=O)CCc2cc(F)c(F)cc2C1 c1(C(=O)NC2(COC)CN(C(=O)CCc3nc(C)cs3)C2)nnccc1C Cc1cc(C(=O)NC(Cn2cccn2)C(N2CCN(C(C)(C)C)CC2)=O)ncn1 C1(NC(C(C)C(F)F)=O)CN(C(c2cccc(OC3CC3)c2)=O)CC(C)(C)C1 C1(C(=O)NCc2c(C)occ2)COCCC1NC(c1csc(F)c1)=O c1(CC)n[nH]cc1C(=O)NC1CCC(N(C)C(c2cc(-c3ccco3)on2)=O)C1 c1(NC(c2cc[nH]n2)C)[nH]c(=NCCCCO)nc2c1cnn2C C1(C(=O)NCC2(NC(=O)CC3CCCC3)CCOC2)CC2(CCCC2)CO1 C(CCCCCCO)(C(=O)NCCC#N)N(CC(=O)NC1CC1)CCC c1(CC)cccnc1C(N1CCC1CC(=O)NC1CCC(CO)CC1)=O C1(C(=O)NC2C(F)CCN(C(Cc3c(C)scc3)=O)C2)CCc2[nH]nc(O)c2C1 c1(C(=O)NC(CC=CC(=O)NCC2(OC)CC(C)(C)C2)(C)C)cn(C)c(=O)n1C c1(CC)cc(C(=O)NC(C)(CNC(C2CCS(=O)(=O)N2)=O)C2CCC2)ccc1F N1(C(c2cnc(C(C)C)s2)=O)CCC(NC(=O)CCN2CCCC2)C(O)C1 CC1(C)CCC(CC(=O)NC(C)(C)C(=O)ON)N(C(=O)OCc2ccccc2)C1 C1(NC(CCC(=O)NC)=O)CCN(C(=O)Cn2cnc(C(N)=O)n2)C12CC2 C(=O)(CCCCCCCCCO)N1CC2CN(C(C(C(CC)O)C)=O)C2CC1 CC1CN(C(=O)Cc2ccccc2I)CC1C(=O)NCC1C=CC(=O)N=N1 Cc1nn2c(c1C(=O)NCC(C)CNC(=O)CC1CCCCO1)CCCC2 c1(C(N2C(C(C)NC(C3CC(C)(C)C3C(F)(F)F)=O)CC2)=O)ccc(Cl)c(C#N)c1 c1(OCC(=O)NCCN(CCC)C(c2[nH]cnc2C#N)=O)cc(Cl)ccc1Cl c1(CC(N2CCC(C(=O)Nc3ccc(O)nc3)CC2)=O)cccc2ncccc12 N1(C(C2(OC)CCOC2)=O)CC(F)CC1CNC(=O)COCc1ccnn1C CN1CCN(C(=O)NCCC2COCCN2Cc2ccc(O)cc2Cl)C(CO)C1 C12(C(=O)OCC)COC(C(=O)N(C)CC3CCCN3C(=O)C3=COCC3)(C1)C2 C1(C(=O)NCC(=C2CN(C(C3CCCN3C3CCCC3)=O)C2)F)CC2CCC1C2 C1(C(N2CCC(N(C(CCc3c(C)noc3C)=O)C)C2)=O)CCCC(F)(F)CC1 Cn1cnnc1CCCC(=O)NC1COCC1NC(c1cc[nH]c1C1CC1)=O C1(C(=O)NC2CCN(C(=O)CN3CCCC3CO)CC2)CCCC2(CC2)C1 CC(F)(F)C(C)(C)C(=O)NC1CS(=O)(=O)CC1NC(=O)C(O)(C1CC1)C1CC1 c1(-c2ccc(CNC3CON(CC)C3=O)s2)ccc(SC)c(C)c1 C(C)(C)(CC(F)C(=O)NCc1csc(CO)n1)NC(C(C(C)C)SC)=O c1(C(N(C(C)C(N2CCC(CCOC)C2)=O)CC)=O)cc2ccccn2c1 Cn1cc2c(C(N3CCCC(NC(=O)C4=CC5C=CC(C4)C5)C3)=O)cccc2n1 Cc1ncccc1CC(=O)NCCCOCCNC(=O)CN1CCCC1=O C1(NC(C2(OCC)CCC2)=O)CN(C(=O)Cn2ncccc2=O)CCC1CO C1(C)(C(=O)NC(CNC(CCSC)=O)CO)CCN(C)C1=O C1(NC(NCC2CCC(C(N)=O)O2)=S)CCC(=O)NC1 c1(C(N2CCC(CNC(C(C(C)(C)C)OC)=O)CC2C)=O)c(C)cc(O)cc1C C1(NC(C(C=CC)O)=O)CC2(CCN(C(c3cccc4nncn34)=O)C2)C1 c1(N(CC(CCC)C)C)cc(NCc2ncoc2C(=O)NC)nc(C)n1 C(CC(=O)NNC(=O)C(C)N)NCC(C)C(C)C.CCO C1(NC(C2CN(CCC)C(=O)C2)=O)CCN(C(c2c[nH]nc2OC)=O)CC1O C(CCC(=O)NC(c1n[nH]c(CO)n1)C)(C(C)C)NC(C(c1ccc(C)o1)C)=O C1(N(CC(=O)N(CC(C)NC(=O)NC)C)C)(C=O)CC1.CCOCC CC1CCCC(C)C1NC(c1cc(CNC(c2cc(Cl)cn2C)=O)no1)=O C1(C(N2CC3C(CNC(C4C(C)C4C)=O)(C3)C2)=O)CC2CCCC2C1 C1(C)(NC(C2C3N(C(c4c(C)csn4)=O)C(CC3)C2)=O)CN2CCC1CC2 C1(CCNC(c2nc(C)oc2)=O)CCCCN1C(c1cnnn1C)=O Cc1cn2c(n1)CC(C(N1CC(NC(=O)Cc3c[nH]nc3O)CCC1C)=O)C2 N#Cc1ncc(Br)cc1NC(C1C2CCC(C2)N1C(c1ccc(O)c(Br)c1)=O)=O CCCC(CNC(c1c(C)nsc1N)=O)C(=O)NC(c1nc[nH]n1)C1CC1 c1(Oc2cccc(-c3ccc(NC(C4CCCCO4)=O)s3)n2)ccc(Br)cc1F N1(C(C2CN(C(c3ccc(C)cc3)=O)C2)=O)CCc2c(n(C)c3ncccc23)C1 CN1CC(C(=O)NCC2CCN2C(=O)CNC(c2ccccc2)=O)OCCC1=O C(CC(C(C)(C)C)NC(C1CCCC1C1CC1)=O)N(C(=O)Cc1ccsc1)C C1(C)(CNC(CC(C)NC(N)=O)=O)CCCN1C(=O)COc1ccon1 N1(C(Cc2ccc(C)s2)=O)CC2(C1)OC1(C)CC2(NC(C2CCCCN2C)=O)C1 CC1OC(=O)NC1C(N1CCCC(CNC(=O)CC2C=CCC2)C1)=O c1(NC2CC(NC(c3c(C)[nH]nc3Cl)=O)C2)ncnc2cccc(Br)c12 C1(C(=O)NC(CC=C)C2CC2)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C(=O)OCC)cnc2nc(OC)ccn12.C12(C(F)F)CCN(CC1)C2=O N1(C(c2nc(CNC(CCC=C)=O)oc2)=O)CCN2CC(C)CC2C1 N1(C(C(COC)OC)=O)CC2(C1)OC1(C)CC2(NC(c2cn(C)nn2)=O)C1 CP(C)(=O)c1cccc(S(=O)(=O)NC2(C(F)(F)F)CC3C=CC2CC3)c1 Cc1cc(C)c(C(=O)N(C(CNC(c2ccc(C(N)=O)[nH]2)=O)C2CC2)C)c(S)n1 C1(C(N(C)CC2CCCN2C(C2(C)CCC(=O)N2)=O)=O)CSC(c2ccccc2)=N1 C1(NC(CCC)=O)CCCN(C(c2ccnn2C)C(=O)NCCC2CC2)C1 CCC(CC(=O)NCCC1CCOC1(C)C)NC(=O)CC(C)n1ccnc1 c1(-c2cc(C(=O)NCC(CN(C(CC(C)N(C)C)=O)C)O)n[nH]2)cccc(Cl)c1 NS(=O)(=O)c1ccsc1C(=O)NCC1CCC(NC(C2CC(F)(CO)C2)=O)C1 Cc1cccc2c1CC(C(=O)NC1CN(C(C3(C)CCCCCC3)=O)CC1C)N2 C1(C(=O)NCCN(C(C)C)C(C2(CN(C)C)CC2)=O)COC(C)C1 c1(N2CC(NC(C3(C)CC=C(C)CC3)=O)C(C)C2)cc(C#N)ccc1[N+](=O)[O-] c1(C(=O)NCC2CC(OC)CN2C(=O)CC(C)OC)ccc2nc(C)cn2c1 N1(C(C2C3(CC(NC(C4CC(=C)C4)=O)C3)C2)=O)CC2CC=CC1C2 C1(C(N2CC(NC(c3cc(O)ccc3F)=O)C(F)C2)=O)CCCCNC1=O N1(C(CNC(CCC)=O)=O)CC2CN(C(c3ccc(N)cc3F)=O)CC2(C)C1 c1(C(=O)NCCCN(C(=O)C(F)C2CCC2)CCC)coc(C)n1 CCCCCCN(CC(=O)NC1CC(NC(=O)Cn2cc(C(=O)OC)cn2)C1)C C12CCN(C1)C(=O)C(C)(C)CC(C)NC(=O)C2C.C(C)(=O)NC(N)=O C1(OCC(=O)NC(C2CCN(C(Cc3cc(C)ns3)=O)C2)C)CCN(C)CC1 CON=Cc1ccc(C(=O)NCC2CN(C(=O)CC=C(C)C)CC23CC3)cc1 C1(C(F)F)(NC(c2cscn2)=O)CCN(c2ccnc(C(F)F)n2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1C2CN(C(C3N(S(C)(=O)=O)CC3)=O)CC1CC2 C1(C(N2CC(N(C(=O)CC3(C)CCOC3)C)C2)=O)CC(OC(C)(C)C)C1(C)C N1(C(Cc2ccc(C)o2)=O)CCCC2(NC(c3cnn(C)c3F)=O)CC2C1 C1(NC(C(C)Sc2ccc(Cl)cc2)=O)CC2C1CCN2C(=O)Cc1c[nH]nc1O N1(C(C2CC(=C)C2)=O)CCC2C(CCN2C(c2ccc([N+](=O)[O-])cc2I)=O)C1 C1(OC)CC(CC(=O)NC2(CO)CN(C(=O)C(F)(F)CN(C)C)C2)C1(C)C C12(C(N3CCC(CC)C3)=O)CC(CNC(=O)CC3(C)CC3(F)Cl)(C1)OC2C Cc1cc(C(=O)N(C)CCNC(c2c[nH]nc2C2CCC2)=O)c(N)c(F)c1 CC(C)C(CN(C)C)N=c1[nH]c(=NCc2c(Cl)cccc2Cl)[nH]c2cccnc12 C1(C(N2CCC(NC(CCc3ccc(SC)cc3)=O)C2)=O)CN(S(N)(=O)=O)C1 c1(C(N2CC3N(C(C(CC#C)C)=O)CC(C3)C2)=O)[nH]c2ccc(OC)cc2c1C C(=O)(N=c1ccn(CC(N)=O)[nH]1)C1N(C(C2N(C(=O)OC)CC2)=O)CC(O)C1 C(=O)(C(C(C)C)NC(N)=O)N1CC(O)(CCNC(C(C)NC(COC)=O)=O)C1 C1(=CC(=O)NCCOCCNC(C2C(C)OC(C)C2)=O)CCC(C)(C)CC1 N1(C(c2c(CC)ccs2)=O)CCN(C(=O)C2=CCC(C(F)(F)F)OC2)CC(O)C1 C12(CC)CCCN1C(=O)C(C1CCC1)CN(C)C2=O.N1(C(COC)=O)CCCC1 N1(C(C(COC)OC)=O)CC(OC)CC1CNC(=O)CCCN1CCCCC1 CC1(C)CC(CC(=O)NC2CCN(C(c3cnc(C(N)=O)s3)=O)C2)CCO1 O=C(C1=CCN(C(=O)C=C2CCCCC2)CC1)NCC12CCCCC1C2 C1(CNC(C2(C)CC(C)C2)=O)CN(C(c2ccoc2C(C)C)=O)CCO1 O(S(=O)(=O)c1ccccc1)c1ccc(N2C(=O)N(c3ccccc3Cl)CC2)s1 c1(C(=O)NCC2CC(NC(=O)Cc3cncnc3)C2)cc2c(cc1F)NCCC2 C1(CNC(=O)CCc2cnoc2)CN(C(=O)C2CC2)C2CCN1C2 c1(C(N2C(CNC(C(C)SCC)=O)C(CC)CC2)=O)nccc(N)c1Cl Cc1cc(NC(C2CN(C(c3c(C)nn(C)c3C)=O)CC2(F)F)=O)ccc1F C1(NC(C2(C)CCSCC2)=O)CCN(C(C2CC=CCC2)=O)CC1CO N1(CC)CCCCC1c1nc(O)n[nH]1.C(CC)(CF)N C(=O)(C(C)(F)CCCC)N1CCC(CN(C(C(C=C)(C)C)=O)C)C1 c1(CN(C(=O)NCC2C(C)OCC2)C)ccc(-n2cccn2)nc1 N1(C(CC(CC)(C)C)=O)CCN(C(=O)CCn2ccccc2=O)C(C)C1C C1(C(N(CCC(=O)NCC(c2nccs2)C)C)=O)CC1C1CCCC1 C1(CNC(c2cnn(C)n2)=O)CN(C(c2cnn(CCO)c2)=O)C2CC12 N1(CC(=O)NCCCCCNC(=O)CNC(=O)Nc2ccccc2)CCOCC1=O C1(C(=O)NCC(C)(CO)NC(c2coc3c2COC3)=O)CCc2[nH]nc(O)c2C1 c1(C(=O)NCC(CN(C(c2cncc(OC)c2)=O)C)C)ccc2oc(C)nc2c1 N1(C(C(C)C#N)=O)CC(C(=O)Nc2cc(C#N)ccc2F)C2(CCC2)C1 c1(C(=O)NC23CC(NC(=O)CSC(F)(F)F)(C2)C3)ncc(Br)cc1F CC(C(Cc1ccsc1)CO)NC(=O)NCC1(C(F)F)CC1 CC(C)(CO)C(C)(C)NC(C1CCCCN(C(=O)C=Cc2ccncc2)C1)=O C1(OC)CC(F)CN(C(=O)CC2CCCN2C(=O)CC2(C)CC2)C1 N1(C(C(CC)C)=O)CCC(F)C(NC(=O)C(c2ccccc2Cl)O)C1 C1(=CC(=O)NCC2(F)CCN(C(C(=O)NC(C)C)=O)C2)CCC(C)(C)CC1 c1(OC)ccc(NC(C2(NC(=O)CC3CCOC3)CCSC2)=O)cc1 N1(C(C(C)(C2CC2)OC)=O)CCC(CNC(c2c[nH]cc2C(C)(C)C)=O)C(C)C1 C1(C(N2CCOCC(F)(CNC(=O)C(C3CC3)C3CC3)C2)=O)CCOCC12CCC2 C#CC1(C(=O)NC2CCN(C)C2=O)CCN(C(c2cnn(C)c2CC)=O)C1 c1(OC)ccc(O)c(OCC(O)CN(C)CC2C3COCC23)c1 C(=O)(C(N=[N+]=[N-])C(C)C)N1C(CN(C(C2CC(CC(=O)OC)C2)=O)C)CCC1 N(C1CC2(CN(C(c3c(C)cnn3C)=O)C2)n2ccnc21)C(CCCC(=C)C)=O Cc1cc(C(=O)NC2CC(CNC(=O)C(F)=C3CCC3)C2)c2[nH]cnc2c1 CC1(C)CN(C(=O)Cn2cnnn2)CC(CNC(c2cc(Cl)ns2)=O)O1 C12CCCC(C1)N(C)CC(C)CNC2=O.c1(N(C)C)cc(-n2ccnc2)ncn1 c1(C(=O)NCCCN(C(C2(C(C)C)CCCO2)=O)C2CC2)cnnc2ccccc12 C(=O)(C(=O)CC(C)CC)NC1CCCC(C(=O)NC(CC#C)CO)C1 c1(C(=O)NCC(CC)NC(=O)C(O)CCC(C)C)c(C)cc(C)cc1C CCCCCC(O)C(=O)NC(C)(CN(C)C)CNC(=O)C(O)CN(C)C(C)=O CC1CC(=O)NCC1C(=O)N(C)CCN1CCN(C(C2OCCCO2)=O)CC1 C=CCC(C)C(=O)NCC1(C(N)=O)CN(C(C2(CF)CC2(F)F)=O)C1 C1(NC(c2c(C)noc2)=O)C2CC3CN(C(=O)CS(=O)(=O)C(C)C)C1C3C2 c1(C(N(CC(C)NC(=O)C(C)NC(c2cnccn2)=O)C)=O)ns[nH]c1=O Cc1nc2cc(C(=O)NCC(C)(CO)NC(=O)CC3CCC(=O)N3)cnc2[nH]1 Cc1cc(C(=O)Nc2cnc(Cl)cc2C(=O)Nc2c(C)cccc2Br)ccc1O c1(N(C)C)ccc(NC(c2cccc(C(C3CN(CC(F)F)C3)=O)n2)=O)cc1 C(=O)(C(O)CC[S+](C)C)NC12CC(NC(c3nccc(OC)c3N)=O)(C1)C2 C(N=c1nc(N2C3CCC2CC(F)C3)c2c([nH]1)CCC2)c1ccc(Cl)c(Cl)c1 N1(C(c2c(CC)cccc2)=O)CC2CN(C(=O)C(C)OC3CCCC3)CC2(C)C1 C#CC1(C(=O)NC2CN(CC)CCO2)CCN(C(c2cccc(O)n2)=O)C1 c1(SC)ncc(Cl)c(C(N2CCN(C(c3cc4ncsc4[nH]3)=O)CC2C)=O)n1 N1(C(=O)NCC(C)(C)Oc2ccc(Br)cc2)C2CCC1C(N)C2 c1(N(S(C)(=O)=O)CCn2cc(C(C(N3CC(SC)C3)=O)=O)nn2)ccc(C)cc1 CCC(C)C(O)C(C)C(=O)N(C1(C(=O)NCCC(Cl)Cl)CCC1)C1CC1 N1(C(=O)Cc2cccnc2Cl)CCC2CCN(C(=O)C(n3cccn3)O)C2C1 C1(NC(N(CCC)Cc2cccc(Br)c2)=O)CC2CC3C(C2)C13 N1(C(C2(C)CN(C(CCn3ccc(C)n3)=O)C2)=O)CCC(F)(COC(C)C)CC1 C1(C(=O)NCC(CC(=O)NCc2cnns2)C2CCC2)CC2(CCO1)CC2 c1(C(=O)NCC2C(NC(c3ccc(N(C)CC)cc3)=O)C2)ccc2nncn2c1 c1(N(C)CC2CCN(C)C2)nc(N2CC3(C)COCC3(C)C2)nc2c1COCC2 C1(C(c2ccccc2)C)CN(C(=O)Cn2cc(C(=O)OC)nn2)CC1N(C)C.C(=O)O N1(C(C2C(CNC(CC=CCCCCC)=O)OCC2)=O)CCC(COC)C(C)C1 N1(C(C2C(C=C)C2)=O)CCN(C(c2ccn(CC)c(=O)c2)=O)C(CC)C1 C1(NC(c2c(C)n(C)c(C3CCCC3)c2)=O)CC(=O)N2CCCCC12 C1(CC)CN(C(c2sc(C(C)OC)nc2C)=O)CCC1NC(=O)CCF O=C(NNc1ncnc(Cl)c1CO)C1CCOC12CCOCC2 Cc1nc(Cl)ccc1S(=O)(=O)N(CC1CC1c1ccccc1)CC1COCCN1 S(=O)(=O)(c1ccc(N2CCCC(C(F)F)C2)c(F)c1)NCCCOCC(C)C C(=O)(CCCC(CC)NC(=O)CCOC(C)=O)N1CCC(OCC=C)C1 N1(C(C2N(C(c3ccc(C#N)[nH]3)=O)C(C3CC3)CC2)=O)CCC2C(C(N)=O)C2C1 N1(C(COCCN(C)C)=O)CCC(C=CC(=O)N(CC(F)F)CCO)CC1 Cc1ncnc(C(=O)NCCC2(C(=O)N(C)CC3CCCOC3)CCC2)c1C N1(C(C2ON=C(C)C2)=O)CCC(NC(c2cc(Br)no2)=O)C(C)(C)C1 CCCC(C(=O)NC(CCC)CC(=O)NCCN(CC(F)F)C)C(C)C c1(CC(C(=O)NCCCNC(C(C=C)O)=O)NC(=O)OC(C)(C)C)ccccc1Cl C(=O)(C(C)CC(C)C)NCCC1N(C(c2n(CC)ncc2)=O)CCSC1 C1(NC(c2c(CSC)cccn2)=O)CCCN(C(=O)CCC2CCN(C)C2)CC1 N1(C(C(C)=C(C)C)=O)CC(C)CCC1CNC(=O)Cc1cnn(C)c1C C(=O)(C(O)P(C)(C)=O)N(CCC)CCC.C(CC)NC(=O)COC(C)CC c1(N2CC(C)(CC(=O)Nc3c(OC)cc(Cl)nc3)C2)ncc2cn[nH]c2n1 C1(CNC(C2CCC2)=O)C2CC1N(C(=O)CCC1CCCC1)C2.O=C1C(CO)N1 Cn1cc(C(=O)NCCN(C(C2C3COCC23)=O)C2CC2)c(C(C)(F)F)n1 c1(C(=O)NC(CCCC)CNC(=O)CC2(C)CC(F)(F)C2)cc(O)nc(O)n1 Cc1nc2ccc(C(N3CC4CCCN(C(C5CC(C)CO5)=O)C4C3)=O)cc2o1 C1(CC(=O)NCC(CN(C(c2cnc(CCCC)s2)=O)C)(C)C)CCCCC1F c1(C2(C(=O)NCC3(F)CCN(C(=O)C(F)(F)CO)C3)CC2)ccc(F)c(Cl)c1 N1(C(C(=O)NC(C2(O)CN(C(C3N(C(C)=O)CCC3)=O)C2)C)C)CCCC(O)C1 c1(NCc2cccc(C(=O)OCC)c2)cc(-c2n[nH]c(C)n2)ccc1C c1(C(=O)NC(C2CCCN(C(C(C#C)(C)C)=O)C2)C)cccc(C)c1F CC1CCN(CCC(=O)NC(CCN(C(C2(C(F)(F)F)CC2)=O)C)=O)C1 C(CNC(=O)CC1(O)CCCOC1)(C(C)(C)C)NC(CN1CC(C)C1)=O C1(CNC(N(C(c2c(C)cccn2)C)C)=O)COc2ccccc2O1 C1(OC)CC2CC1CN(c1nnc(-c3ccc(F)c(F)c3)s1)C2 C(=O)(C1CCCc2n[nH]cc21)N1C(CNC(c2ccc(C(C)C)cc2F)=O)CC1 CC1c2ccccc2CC1C(=O)NC1(C)CN(C(=O)Cc2cc[nH]c2)C1 C1(CC(N2C(CNC(C=C(COC)C)=O)CCC2)=O)Sc2ccccc2NC1=O N1(C(C(CC(=C)C)C)=O)CC(NC(=O)Cc2ccccc2Cl)CC2(CC2)C1 c1(CCC)cc(C(=O)N(CC(C)NC(=O)C(c2cccnc2C)C)C)ccn1 CCC(C(=O)N1CCCC1CC(=O)NCc1cnc(C)[nH]1)N(C)C c1(OC)ccnc(C(=O)NCC(C)CC(=O)N2CCC2CO)c1 CC#CC1CCN(C(C2CCCN(C(=O)CCC(=O)NC)C2)=O)C1 N1(C(C(CCC(C)C)F)=O)CCCC2C1CCCN2C(=O)CCN1CCCC1 CC1=C(C(=O)N2CC(F)(C(=O)NCC3CCOC3)C2)CCC1 n1(CC(=O)N(C2CCN(C(C3CCC(F)(F)C3)=O)C2)C)ccc2ccc(F)cc12 c1(C(N2CC3CC(CN(C(C(CC)F)=O)C3)C2)=O)nc(C2CC2)n2ccccc12 C1(C(=O)NCC2CCCN(C)C2)CN(C(=O)C(O)CN2CCCC2)CC12CCC2 C12(C(C)C)CCC(NC(=O)NC(C)(Cc3ccccc3)C(F)F)C1C2 CCCCCC(=O)NCC(=O)NC(CNC(C1CC1C(F)F)=O)CC(C)C N1(C(CC(CC)NC(=O)C2=NOC3COCC23)=O)CCC2(CCN(C)C2)C1 CC(O)(CC(=O)N1CC2=C(C1)CN(C(=O)COCCCN=[N+]=[N-])C2)C(F)(F)F N1(C(C(C)S(C)(=O)=O)=O)C2CCC1CC(O)(CNC(=O)CCCNC(N)=O)C2 c1(C(=O)NC2CCN(C(C3C(CC)N(C)CC3)=O)C2)cc(O)nc2cnccc12 Cc1cc(N)cc(C(N2CCCC2CNC(=O)C(C)(C)c2cnco2)=O)c1F C1(CCNC(C(C)(C)C2CCC2)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1 C1(CNC(c2nc(NC(C)=O)sc2)=O)COCCN(C(=O)C#CC(C)C)C1 Fc1ccc(Br)c(-n2nnnc2N2CCN(CC3C4CCCCC4CN3)CC2)c1 c1(CN(C2CCCN(C(c3ccn(CCOCC)n3)=O)C2)C)ccc(F)nc1C C1(C(N2C(COC)C(C)(C)C2)=O)CNC(=O)CN1C(=O)Cc1cncn1C c1(C(N2C(C)CC(NC(=O)CC3CCC(=O)N3)C2)=O)ccn2nncc2c1 N1(C(C(C2CC2)OCC)=O)CC(CC)CC1C(=O)NCC(=O)N(C)OC C1(CCNC(c2cn(C(F)(F)F)cn2)=O)CCCN1C(=O)CNc1ccccn1 C(=O)(C1CCc2sc(NC(=O)NC3CCC(S(=O)(=O)NCC)CC3)nc21)OCC CC(C)C(N=[N+]=[N-])C(=O)NCC1COC(CNC(=O)CCc2cncs2)C1 C1(NC(=O)Cc2ccsc2Cl)CCC12CN(C(c1cccn(C3CC3)c1=O)=O)C2 c1(C(N2CC(CC(C)NC(C(CCOC)(C)C)=O)C2)=O)cc(C)c(F)cc1Cl c1(OCCC(=O)NC(CC)(CNC(C2(O)CCCC2)=O)CC)cc(Cl)ccc1Cl N1(C(c2cc(C)[nH]n2)=O)CCC2CN(Cc3c(Cl)ccnc3Cl)CC12 Cc1cc(C(=O)C(=O)NCC2CCC(F)C2)c(C)o1 N1(C(C2C(C(=O)OC)CC2)=O)CCC2CCCC12C(=O)NC(C)CN=[N+]=[N-] C(=O)(CC(C(F)F)NC(=O)CCC(N)=O)N1CCC(NC(C)=O)CC1 c1(-c2ccc(C(=O)NCCN(CC(F)(F)F)C)o2)ccc(F)c(F)c1 c1(C(N2CCC(N(C(c3csc(CC(C)C)n3)=O)CC)C2)=O)ccc(F)nc1F c1(CC)c(C(=O)NCCCOCCNC(C2CCCO2)=O)oc2ccccc12 C1(C(N2CC(=C(CNC(c3cccc(C4CC4)n3)=O)F)C2)=O)CC(=O)CC2CC12 C1(C(=O)NCC(C)(C)OCCO)CCN(C(C2CC2Cl)=O)C1 C(c1cccc(Cl)c1)=CC(=O)NC1(CO)CN(c2nc(C3CC3)ns2)C1 C12CCC(CC1)n1cc(nn1)C(C)(C)NC2=O.c1(CC)ncoc1C(=O)N(C)C c1(OCC)ccc(CNC23CC2CN(C(c2cc(Cl)nc(Cl)c2)=O)C3)cc1Br C1(NC(c2ccccn2)=O)CN(C(=O)Cn2cncn2)CC1C1CCCC1 Cc1nn2ccccc2c1C(=O)NCC1(F)CC(NC(=O)C(C)(C)C(C)C)C1 c1(C(N(C2CC2)Cc2ccc(OC(C)=O)cc2)=O)cc(C)nc(Cl)c1 C(=O)(C(C)C(=O)N1CCOCC1c1ccc(C(=O)NCCC2(C)CC2)n1C)OC C(=O)(CC(C)CC(=O)NC(CC1CC1)C(=O)Nc1cccc(F)c1)OC C1(CC(=O)N(C2CCN(C(C=CC=CC)=O)C2)CCC)SC2=NCCN2C1=O C(=O)(CCCn1cc(CCCO)nn1)N(C(C)(C)C)NC(=N)N c1(CNC(C2(C)CC=C(C)CC2)=O)nc2c(s1)CN(C(c1ccoc1)=O)CC2 N1(C(C2(C(F)F)CC(=C)C2)=O)CC2C(NC(c3cnc(C)[nH]3)=O)C2C1 C1(NC(C(c2cccc(C)c2)C)=O)CCC(C)N(Cc2cc(C)on2)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CCC(CNC(CCC=C)=O)C(F)(F)C1 c1(C(=O)NCC2(F)CN(C(C34CCC(CC3)CO4)=O)C2)cc2ccc(Cl)cc2o1 N1(C(CCCN(CCC)CCC)=O)CC2(CC(NC(C3CCN(C)C3C)=O)C2)C1 C1(C(=O)NC(CNC(C2(C(C)C)CCC2)=O)(C)CO)CS(=O)(=O)CC(=O)N1 CC(C)(C)C(=O)C(=O)NCC1CCCN1C(C1(Cl)CC12CCC2)=O C1(CCOC)(C(N2CCC(O)(CCNC(=O)C(C)(C)CF)C2)=O)CCN(C)CC1 S(=O)(=O)(c1ccc(Br)cc1)NC1C(C)(C)CN(S(=O)(=O)CC2CCC2)CC1 N1(C(CC(C)C2CC2)=O)CCC2(CCN(C(=O)CC(C)(C)C)CC2)C1 N1(C(CC2(COC)CC2)=O)CC2C3CCC(C2C1)N(C(=O)C(C)(O)C1CC1)C3 CCC(C)(C)CC(C(=O)NCCCF)N1CCOC(CN=[N+]=[N-])C1 C=CC1(CC(=O)OC2(OC)CCC2)CCC1 C1(C(N2CC(NC(C(C)(C)N(C)C)=O)C(F)CC2)=O)Cc2ccccc2S1 S(=O)(=O)(c1nc2c(s1)CCCC2)NC(C1(C2CC2)CC1)=O C(=O)(C(C)N(OC)C(=O)C1COCCC1NC(C12CC(F)(C1)C2)=O)OC C=CCC(C(=O)N(C)CCN(C)Cc1nnc(C)n1CC=C)NC(C)=O c1(C(N2CCN(Cc3ccc(C)o3)CC2CC#N)=O)cccc2ccnn12 C(CNC(=O)C(C(C)OC)NC(c1c(C)csc1C)=O)(CC(C)C)OC c1(C(=O)NCC2CCC(C(=O)NC(CC(CC)C)C)O2)cc2cccn2cn1 CC(C)C(=O)NC(=O)CNC(CC(CO)NC(N1CCCC1)=O)=O N1(C(c2cc(C)cc(Br)c2)C(=O)NC(C(=O)OC)C)CCc2ccc(F)cc21 N1(Cc2n(CC(F)F)ncc2)CCC(F)(F)CC12CCC2 N1(C(C(C)OCC=C)=O)CCC(C)(C)CC1C(=O)Nc1cnc(CO)nc1C C1(C(N2CCN(C(c3cc(O)cs3)=O)CC2)=O)CC12CCC(F)(F)CC2 CC(C)(O)C(O)C(C)(C)C(=O)NC1CC2(CCC2)CN1 c1(C(C)=O)ccc(CC(=O)NCCC(C)(C)NC(=O)C(=Cc2ccco2)C)cn1 CCCCCCC(C)C(=O)NC12CCC(C(=O)NCCCn3cnnc3)(CC1)C2 C12(NC(C(CCCC)F)=O)CCCC1N(C(c1cnn(C3CC3)c1)=O)CC2 C=Cc1ccc(C(N2CCC(CNC(c3cc[nH]c(=N)n3)=O)C(O)C2)=O)cc1 N1(C(C2(C)CCCS2(=O)=O)=O)C2CCC1CC(CN=c1ncc(F)c[nH]1)C2 Cc1ccc(Br)c(CN2CCC(F)(C(=O)NC(C#N)C(N)=O)C2)c1 CC1CCCC(C(=O)NCCC2(C(=O)NC3CCCCC3CCO)CC2)O1 C1(C(N(CC(C)NC(c2nccc(C)n2)=O)C)=O)CC(C2CCC2)C1 C1(NC(CCCOC(C)C)=O)C2CCC1N(C(=O)CC1CCCCN1C)C2 c1(CNC(=O)C(O)Cc2ccccn2)cccc(NC(C2CCC3(CC3)C2)=O)c1 C(CCNC(C1COCC1C(F)(F)F)=O)(CNC(=O)C(=O)N(C)C)OC CCC1=NOC(C(=O)NC2(C)CC(NC(c3cc(C)c(C)[nH]3)=O)C2)C1 c1(CC)ccc(C(C)=CC(=O)NCCN(C(=O)C(=O)NC2CC2)CC2CC2)cc1 C1(CCOC)(NC(=O)C(C)NC(C2CCC2)=O)CCN(C(c2csc(C)c2)=O)C1 C1(Cc2cc(NC(C3(c4oncc4C)CC3)=O)no2)CCCC(NC(=O)NC)C1 c1(CNC(C(c2nc[nH]n2)N(CCC)C)=O)nncn1CC1CC1.OC Cc1cnccc1N1CCN(C(=O)NC(c2ccc(Br)cn2)C(F)(F)F)CC1 CC(CC(=O)N1CC(S(C)(=N)=O)C1)CC(C)(C)C.C12(CCCCC1)C(=O)NC2 c1(C(=O)NC2C(CNC(C(C)CS(C)=O)=O)CCC2)ccc(F)c(O)c1F C(=O)(C(C)(O)CC(C)C)NC1CCN(c2nnc(-c3cnc(C)s3)o2)CC1 c1(C(=O)NCC(CC(=O)OCC)C)cc(I)ccc1O Cn1nnc2c1CC(C(=O)NCC1(O)CCCN(C(C34CC(C3)C4)=O)CC1)CC2 CC1CC(c2ccccc2F)C(C)CN1CC(=O)Nc1ccco1 C(N=c1[nH]c(=NCC(C)OC2CCCCC2)[nH]c2c1COC2)C1C(CCC)C1 C1(F)(C(=O)NC(C2CC(NC(C3CCC(C)CC3)=O)C2)C)CCCN(C)C1 CCS(=O)(=O)N(CC(=O)N(CCNC(=O)COC(F)(F)F)CCOC)C C(=O)(CCCS(C)(=O)=O)N1CC(N(C(C2CC=C(C)CC2)=O)C)C2(C1)CC2 c1(CC)cnccc1C(=O)NCC(C)CN(C)C(c1nc(Br)c[nH]1)=O C(=O)(C(CC(F)F)NC(C1C=CCC1)=O)NCC(C)(O)CO C(=O)(CC(C)n1cccn1)NC(C(=O)NCCC(=O)N(CC)CC)c1cccs1 C1(C(=O)NCC(CCOC)NC(=O)CC2CN(C)C2)CC(C)CC(C)C1 c1(C(N2CCN(C(=O)Cn3ccnn3)C(C(F)F)C2)=O)cnc2ncccc2c1 c1(OC(C)C(=O)N(c2ccc(I)cc2)C(C)(C)C)ccc(Cl)c(F)c1 C#CCC(CC(F)F)NC(C1(F)CN(C(=O)C(C)(O)CCC)C1)=O n1(CC(=O)NC2CCC(NC(CN3C(C)CC3)=O)CC2)cc(C#N)c(O)nc1=O Cc1cc(=NCC2(S(=O)(=O)NC(C)(C)C)CC2)[nH]c(=NCC2OCCC2C)[nH]1 N1(C(Cc2cnc(C)s2)=O)CCC12CN(C(=O)C(C1CCS(=O)(=O)CC1)(C)C)C2 C1(C(=O)NC(C)(CNC(c2ccc(CO)nc2)=O)CO)CCc2nc(O)[nH]c2C1 c1(C(=O)NC(C(C)C)CNC(C2CCOC2=O)=O)cc(F)c2[nH]nnc2c1 C1(CNC(c2ccc(CC(F)F)cc2)=O)COCCN(C(=O)CC2CCCC2)C1 C1(NC(c2ccn(C(F)F)n2)=O)CCOCC1NC(C1CC(CF)C1)=O CC(C)C(=O)C(=O)N1CC2C(NC(=O)C(C)Oc3ccc(Br)cc3)C2C1 C=C1CCN(C(c2ccsc2)=O)C(C(=O)NCC2CC(O)C(O)C2)C1 c1(CN(C2CCN(CC)CC2)CCO)ccc(S(C)=O)cc1.C12CCN(C1)C2=O c1(NCC(=O)NCC2CCC(NC(=O)COC3CC=CC3)C2)ccc(F)c(F)c1 c1(C(=O)NCC2(F)CC(NC(CCOCCOC)=O)C2)nccc2c1CNC2=O C1(CNC(c2n[nH]c(C)c2O)=O)CN(C(=O)C(C)N2CCC2)CCC1(C)C C(CC(F)(F)F)N(C(C)C(=O)NC1CC1CNC(=O)CSc1ccccc1)C CC1CN(C)CCCN1C(C1CC2CC1CN(C(C1SCCS1)=O)C2)=O C1(C(=O)NCCN(C2CC(C#N)C2)C(C2CC(F)(F)C2)=O)CCC(C(F)F)CC1 C1(NC(C2CCSC2)=O)CC(C(=O)NCC2(CO)CCC2)CC1O C1(C(=O)NCc2c(C)ncs2)(NC(=O)CC23CCCC2C3)CCN(C)C1 N1(C(=O)CCCSC2CC2)CCN(C(C2CC=CC2)=O)C2CCCCC2C1 C(=O)(C1CCCc2ncnn21)NC1C(CNC(=O)CCn2cccnc2=O)CC1 N1(C(C2CCN(CC)C2)=O)CC(C)C(C)(CNC(c2[nH]cc(C)c2C)=O)C1 C1(NC(C2C(CC)C2)=O)CCN(C(c2cc(C)c(O)c(Cl)c2)=O)CC(C)(C)C1 C1(NCCC2(C)CCNC2)C=CC2(CCCCCC2)CC1 Cc1ccccc1-c1cnc(CN2CCC(NC(c3cn(C4CC4)nn3)=O)C2)o1 C1(C(=O)NC2C3CCN(C(=O)CCc4cnccn4)C23)COCC2(CCC2)O1 c1(C(=O)NCC#CCNC(C(=Cc2cccs2)C)=O)c(Cl)cccc1[N+](=O)[O-] C1(CC(N2CCC(CCNC(CCCN=[N+]=[N-])=O)CC2)=O)CCn2cncc2C1 c1(C(N(C(C)C(=O)NCCC2CCC(C)O2)C)=O)cccc(CO)c1 Cc1c(Cl)cc(Cn2ccccc2=O)c(Cl)c1C.C1(C(=O)O)(CN)CCC(C)(C)C1 Cc1cc(Cl)c(C(=O)NC2CC(C)CN(C(=O)CSC3CCOC3=O)C2)cc1C N1(C(c2cc(CCC)nn2C)=O)CCN(C(C2(CC)CCCC2)=O)CCC1C CC(=O)CCCC(=O)N1CCC(C)CC1CNC(c1cc(F)n[nH]1)=O Cc1cccc2c1C(C)CC2CNc1c(F)cc(Br)cc1F N1(C(CCN(CC)CC)=O)CC(NC(c2c[nH]c(Br)c2)=O)C2CC12 c1(C(=O)NC(CC)CNC(=O)C(C)OCC2CC2)cccc(CC(C)C)c1 n1(C(C2CCCCC2)C)nc(-c2cccs2)nc1-c1ccon1 CC1CN(C(C2(C)CC3CCC2C3)=O)CCC1NC(C1(C#N)CC1)=O C1(C)(CC(=O)OC2CCC(OC)CC2)Oc2ccccc2O1 N12CC3CC(C3)(C1)CNC2=O.C1(C)(OC)CN(Cc2ccccc2)C1C1CC1 Cc1cc(F)c(C(N2C(C(=O)Nc3cnn4cccnc34)CCC2C)=O)c(F)c1 C1(NC(C(CCC)F)=O)CCCN(C(c2cccc(F)c2N)=O)C1C c1(Sc2nnc(S)s2)ccnc2cc(Cl)ccc12.C12CCN(C1)C(=O)CNC2=O c1(-n2ncc(CN3CC(O)(c4nnc(C)o4)C3)c2)cccc(Cl)c1 c1(C(CNC(C2(CC3CC3)CC2)=O)NC(c2cc(Cl)cs2)=O)ccc(F)cc1 N1(C(CC(N)Cc2csc3ccccc23)=O)CC2(CCC2)CCC1CO C(=O)(C(C)(C)C(O)C(C)C)NC1CC=C(C(=O)NC2C(CC=C)CCC2)C1 C(=O)(C(C)(C)CC(=O)OCC)NC1CC(=C)CN1Cc1cc(C)cc(OC)c1C(N)=O N#Cc1ccc(C2CCN(CC3(C(F)(F)F)CC3)C2)s1.c12ccc(cc1)s2 c1(C(N(C2CCN(C(c3cc(C(N)=O)cs3)=O)C2)C)=O)c[nH]c2ncnc(O)c12 C1(CNC(C(C=C)(C)O)=O)CC(C)(C)CN1C(=O)C(c1ccc(Cl)cc1)C c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CS(=O)(=O)C2)cccc2c1oc(=O)n2C C1(NC(c2c(C)noc2)=O)CCCCN(C(C2CCC2)=O)C1 N1(C(c2nnc(C)s2)=O)CCOC(CNC(c2c(C)nsc2Br)=O)C1 Cc1sc(C(=O)N(C2(Cc3cc(C(F)(F)F)nc(C)n3)CCC2)C2CC2)c(C)c1C c1(CNCCC)ccc(C)c(O)c1.C1C(O)CN(C)CC(=O)N1C n1(CC)cccc1C(=O)NCC1(F)CC(NC(C2CC(=C3CC3)C2)=O)C1 CC(C)CC(C(=O)NCC(CNC(=O)CCCN(C)C(C)C)CO)C(N)=O N1(C(CN(C(C)=O)C)=O)CCC2CCN(C(=O)CCc3nc(C(C)C)no3)CC12 c1(SCC(=O)OCC(CCCC)OC)c(C(C)=O)oc2ccccc12 CC1OC2(C)CC1(C(=O)NC13CCC1CN(C(c1ccc(N)c(Cl)c1)=O)C3)C2 c1(SCC)cccc(CC(=O)NC(C)Cn2cc(Cn3cc(Cl)cn3)nn2)c1 N1(c2nnc(COCC)n2CC2(OC)CCC2)CCC2C(C1)C2(F)F.C1(C)CC1 C(=O)(C1=NOC2COCC12)N1C2C(NC(c3c(CC)[nH]cc3)=O)CC(C2)C1 C1(NC(c2cnc(CC)o2)=O)CC(NC(C23CCC(CC2)C3)=O)C(O)C1 C1(C(=O)OCC)CCC2(CC(C(=O)OC)C2)N(CC)C1.c12cnc(O)c(c1)NC2 C1(C(N2CC(C)CC(CC)C2)=O)CC2(CCN(C(=O)CCCCC(C)C)C2)C1 N1(C(CCSCC(N)=O)=O)CCCN(C(c2cnc3nccn3c2)=O)CCC1 c1(C(N2CC(C(Cn3cc(C(CCCC)CC)nn3)F)C2)=O)ccc(F)cc1N c1(C(=O)NCCOC2CCN(C(c3c(CC)nc[nH]3)=O)C2)ccc(C)nc1O C1(CC)C(C(=O)NCc2c[nH]nc2C2CC2)CCCN1C(c1c[nH]c(=O)cn1)=O CC1=C(C(=O)NCC2CCN2C(C2CC3(C2)OCCO3)=O)COCC1 N1(C(C2C(C)(C)N(C(=O)C(F)CC3CCOC3)CC2)=O)CCc2cccc(O)c21 O=S(=O)(c1cccc(N2CCC(CCO)CC2)n1)NCC1CC12CC2 C1(O)(C(C)NC(C=CCCC)=O)CCN(C(=O)CC2CCC(C)CO2)CC1 Cc1cc(C(=O)NC(C(N2CC3(CCCO3)C2)=O)C2CC2)ncc1N C1(C(F)(F)F)(N(C(=O)OC)C)CCCN(S(=O)(=O)N=S(C)(C)=O)C1 c1(C(=O)NC2CN(C(C3N(C)CC(O)CC3)=O)CC23CC3)ccnc2c1CCO2 C(=O)(C(C)CC(C)C)N(CC(C)NC(C1CC(OC)C1)=O)CC C(C)(C)(C(C)NC(=O)CCc1nc(C2CC2)no1)NC(C(=O)NCCOC)=O C(=O)(C1CC(C)(C)Oc2ccccc21)NC1(C)CN(C(C(COC)OC)=O)C1 c1(C(=O)NC23CCN(C(c4c(C)nc[nH]4)=O)CC2C3)cc2c(o1)CCCNC2=O c1(C(=O)O)ccc(CNC2CCC(N3CCOCC3)C2)cc1 C1(C(=O)NC(C)CSC(F)F)CCCCCC1NC(c1cc(O)nc(O)n1)=O C(=O)(CCCC(F)(F)CO)N(C1CCCN(C(=O)CC2CCC(C)CO2)C1)CC c1(OC)nc(C)c(Br)cc1C(C(=O)NCC(C)C)N(C)CC1CCCC(F)(F)C1 c1(C(N2C(CCC(=O)NC3CC(O)C3)CCC2)=O)cc(F)c([N+](=O)[O-])cc1F c1(OC)ccccc1CCN(C1CC(OC)CC(Nc2ccc(C(F)(F)F)o2)C1)C=O c1(C(N2CCC(NC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)c(Cl)nn(C)c1Cl C1(NC(c2ccn(CC)n2)=O)CC2CC(C1)N(CC(N1CC(C)CC(C)C1)=O)C2 c1(C(N2C(CCNC(=O)COC(F)(F)F)CCCC2)=O)c(F)ccc2n[nH]cc12 N1(C(C2CC(C#N)C2)=O)CC(F)(F)CC1CCNC(=O)CC1C=CCC1 c1(CC)c[nH]c(C(=O)NC(C2CC=CCC2)C(=O)NCC(=O)N(C)C)c1 N1(C(CC(C=C)C)=O)CCC2(CC2NC(c2cnn(C3CCC3)c2)=O)C1 c1(OC)ccccc1C(CNC(C1CC1CF)=O)NC(=O)Cc1nc(C)sc1C c1(OC)cc(CNc2ccc(C(=O)Nc3cncs3)nc2)ccc1C c1(C(C)(F)F)ccc(Cl)c(C(=O)NC(CC2(O)CCC2)C(F)F)c1 C(CC(C)(C)C(=O)N1CCC(N(C)C)C(C)C1)NC(CC1C(C)OCC1)=O N1(C(N(C)C)=O)CCCC(C(N2CC3CC2C3NC(=O)C(C)(C)N(C)C)=O)C1 Cc1cc(S(=O)(=O)N2CC(C)(C)OC(C)(C)C2)ccc1-c1cccnc1 C#Cc1ccc(C(=O)NCC2CCN2C(=O)C(C)N(C)C(C)=O)cc1 N1(C(Cn2ccc(C)n2)=O)CCC2(CCN(C(c3cnc(N)c(Cl)c3)=O)CC2)C1 c1(C(N(C2CC(NC(C3C(=C)CC3)=O)C2)C)=O)cc(Cl)cs1 Cn1ccc(C(N2CCC2CNC(c2cn(CCO)nn2)=O)=O)cc1=O N1(CCNC(C2CC(CNC(CC3CC(=C)C3)=O)OC2)=O)CCCC(O)C1 c1(C(C(=O)N(C(CNC(C2(C(=O)NC)CC2)=O)(C)CO)CC)C)ccccc1C c1(C(=O)NCc2nc(-c3cccc4c3COC4=O)no2)ccc2c(c1)C(=O)NCC2 C1(C2CN(C(C3CC3Cl)=O)C2)(NC(C2CCCCC2)=O)CC1 C1(C(N2C(CN(C(=O)CN3CCCCC3)C)COCC2)=O)CCn2nncc2C1 CCCC(C(=O)OC)C(=O)NC1(CC)CCCN(Cc2ccc(C)nn2)C1 c1(C(C)(C)C)cccc2c1CCN2C(c1cccc(-c2cc(Cl)ccc2Cl)c1)=O c1(N(C(=O)CN2CCCC2)C=O)cccc(F)c1N.C(=O)(OC)OC c1(CCC(=O)NCC2CC2CNC(=O)CSCC(C)C)cc(SC)c(C)o1 c1(C(=O)NC(CC)CNC(=O)CC2CCC(=O)N2C)cc(C)c(O)c(C)c1 C(CCC)(CC(=O)NC(C)CC(C)C(F)F)NC(CCC)=O N1(C(CCCN(C(C)C)C)=O)CCN(C)CC1C(=O)NC1CN(C(N)=O)C1 N1(C(CC(CCN)O)=O)CC(NC(=O)CN2CCCC2)CC12CCC2.C(C=O)SC c1(C(=O)NCCC(=O)NCc2c(C(C)C)ocn2)cnn(C)c1N c1(C(N2CC(O)CC(NC(C3CC4(CSC4)C3)=O)C2)=O)c(Cl)ccc2ccoc12 C=CCCC(C)(C)C(=O)NC(C)CC(C)NC(C1(c2cc[nH]n2)CC1)=O N1(C(Cc2ccc(CC(C)C)cc2)=O)Cc2[nH][nH]c(=NC(=O)c3cnco3)c2C1 c1(NC(=O)COCC2CCC2)cccc(CN(C(COCCOC)=O)C)c1 N1(C(=O)NCCOC2CCS(=O)(=O)C2)CC2CCCN2Cc2ccccc21 Cc1cc(Cl)c(C(=O)NC2CN(C(=O)C(F)CC3CCC3)CC2O)cc1C C1(C=O)CCCN(CC#N)C1.C1(N(C(C=CCC)=O)CCCC(F)(F)F)CCCC1 Cc1cc(C(=O)NCCC(O)C(=O)NCC2(C)CC=CCC2)c(C)cn1 CC1NC(=O)CCC1CNC(=O)C(O)CNC(C1(F)CC=CCC1)=O CC1OCCC1C(N1CCC(C(=O)NC2(CCF)CCC2)C1)=O C(C(C)(CC(=O)O)NC(=O)C(C(C)C)OCc1cccs1)OC c1(C(=O)NCCC2CC(C(=O)NC(CSC)(C)CO)C2)nc(C)ccc1C C#CCCCCS(C)(=O)=NC(=O)C(=O)C1CC(C)(C)CC(C)(C)C1 CC1CCN(C(c2cnc(S)n2C2CC2)=O)CC1NC(=O)C=Cc1cccnc1 C1(C(=O)NC2CON(CC)C2=O)CN(C(=O)CC(C)OC)CCC1(C)C C1(C(=O)NCC2C(NC(C(CCC)OC)=O)C2)CCC(N=[N+]=[N-])CC1 c1(C(c2n(CCOC)nnn2)NC(C(N)=O)C2CC2)ccccc1C(C)(F)F Cc1ccc(-c2cc(C)n(CC(=O)NCc3cc(-c4ccco4)[nH]n3)n2)cc1 c1(-c2cc(C(=O)NC3C(NC(C(CSC)O)=O)C3)on2)ccc(Cl)cc1 N1(C(c2cn(CC)nc2C2CC2)=O)CCC2C(CCN2C(=O)C(F)C2CC2)C1 S(=O)(=O)(c1c(F)ccc(C)c1F)Nc1sc(CCC)c(-c2nn[nH]n2)c1 CC(C)C(C(=O)N(CCCNC(c1ccc(C(F)F)cc1)=O)C)NC(N)=O C1(CN(C=O)Cc2cccc(OC(F)F)n2)CC2OCCC2O1 c1(C(=O)NC(C2CC3CCC2C3)C#N)cc(C(=O)O)c(Br)cn1 c1(C(N(C2CCN(C(c3nc(CCC)oc3)=O)C2)COC)=O)nnn2c1CCC2 N1(C(c2c(F)ccc(OC)c2)=O)CCCCC(NC(=O)CC(C)SC)CC1 c1(CCC2CCCN(NC(C(N3CCCCCC3)C)=O)C2)nnn2c1CCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CC23CCCC2(C1)CN(C(=O)CSC(F)(F)F)C3 C(=O)(CC(C)(C)C(F)F)N1CC(C)C(CNC(=O)CSc2nnc(S)s2)CC1 C1(SCC)CCC(C(=O)N(CCNC(C2(C)CC3CC3C2)=O)CC)CC1 Cc1cccc2nc(CCC(=O)NC3(C)CCN(C(=O)CCCC4CC4)C3)[nH]c12 Cc1nn(C)c2cc(C(=O)NCc3cn(-c4cnc5c(c4)CC(=O)N5)nn3)ccc12 C1(COC)(CNC(c2n[nH]c(C)c2C)=O)CCCN1C(c1[nH]cnc1C)=O Cc1cc2[nH]c(C(=O)NC3C4CC3CN(C(c3ccc(F)cc3Cl)=O)C4)cc2o1 C=CC1OCCCC1C(=O)NCC1CCN(C(=O)C=C(C)Cl)C(C)C1 CCC(CCC(=O)NC(C)CC(C)O)NC(c1cccc(OC)c1)=O c1(SC)nc(N2CCC(NC(C3(C)CCCS3(=O)=O)=O)C(C)C2)cc(Cl)n1 C(CC(=O)NC1CC1c1cncs1)(CC(C)C)NC(c1c(C)nncc1)=O C(c1ccccc1C)=CC(N1CC(CC)C(C(N2CC(C3CC3)C2C2CC2)=O)C1)=O c1(OC)ccc(CCCNC(Cc2ccccc2)C(C)C)cc1O C=CCC(C)C(=O)NCCCC1(NC(=O)CCc2nc(-c3nc[nH]n3)no2)CC1 c1(C(N2CCC(C3N(C(C(N4CCCCCC4)C)=O)CCC3)C2)=O)cncc(N)n1 CC(C)(C(=O)N1CC2(CCN(C(c3coc(CS(C)(=O)=O)n3)=O)C2)C1)S(C)(=O)=O c1(C(=O)NC(CNC(C(C)NS(C)(=O)=O)=O)(C)C)ncc(F)cc1N c1(CC(=O)N(CCCCN(C(=O)C(O)CF)C)C)ccn2cncc2c1 C1(CNC(c2cnc(CC)s2)=O)CCN(C(C2CC2c2cccnc2)=O)CC1C C=C1CC(C)(C(=O)NCC2OCCC2C(=O)NCc2nc(C(C)C)n[nH]2)C1 Cc1csc(CCC2CC2NC(N2CCC(Cc3cccs3)C2)=O)n1 c1(C(C(=O)NC2C(NC(C(CSC)(C)C)=O)C2)C)ccc(F)c(Cl)c1 Cc1nc(C)n(CCCC(=O)NCCC(C)NC(=O)C=CC(=O)N(C)C)n1 c1(SC(C(=O)NCC#C)CCF)cc(C)nc(C)c1.C12(CC1)C(=O)N2 BrC1=CC=CCC2C3(CCOC1CNCCC2)CC3 C1(COC)CC(C)CN(C(C2CS(=O)C2)=O)C1 c1(OC)cc(C(=O)N(C)CC2CCCN2C(C2CC2C(N)=O)=O)c(Cl)cn1 CC(C)(O)C(C)(O)CNC1CC(c2ccccc2)CN1 CC(F)(F)C(C)(C)CC(=O)N1CCC2CC1CN(C(c1ccc(Cl)c(F)c1)=O)C2 N1(C(c2n(C)ccn2)=O)CCOC2(CCN(C(C3CCC(C(N)=O)CC3)=O)C2)C1 Cc1c(C(N2CCC(CNC(=O)CSC(C)C)CC2)=O)ncn1C C1(CC)CN(C(c2ccc(OC)nc2Cl)=O)CCN1c1ncccn1 CC1CCCCC1CC(N1CCC(C)(NC(N)=O)C1)=O.c12cn(nn1)C1CC23CC13 c1(OC)cc(C(=O)NCC2CN(C(c3cnc(C)[nH]c3=N)=O)C2)ccc1[N+](=O)[O-] c1(C(C(=O)NCC(=C)C)N(C(C)C)C2CC2)cncn1C C(=O)(C1CCCc2ccccc21)NC(C(C)NC(CCCOC(C)C)=O)CO CC(C)(CNC(C1CCCO1)=O)CCNC(c1ncoc1C1CC1)=O C#CCC(C(=O)NC(CCF)C(=O)NC(c1ncc(C)cn1)C)C1CC1 c1(C(=O)NC(CC)(C)CNC(C2CC2C(C)(F)F)=O)cncc(C#N)c1 C12(NC(c3c(C)cc(F)cc3)=O)CCCN(C(c3ccsc3C#N)=O)CC1C2 C(=O)(C(CCCCC)C(C)C)NCC1CCC(CN(C(C(CC#C)O)=O)C)CC1 c1(CC)ncc(C(=O)N(C2CCC(NC(c3nc(O)sc3C)=O)CC2)C)c(O)n1 C(N=c1[nH]cnc(Cl)c1OC)C1CCCC(NC(CC(C)SC)=O)C1 c1(C(N2C3CN(C(c4c(C)cn(C)c4)=O)C(C3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(C)(CCNC(C2(NC(=O)OC)CCCC2)=O)CCN(C(c2cnn(C)n2)=O)C1 c1(C(N2CC(C(C)NC(C(C)OCC)=O)C2)=O)cc(C#N)c(F)cc1F C1(NC(C=CSC)=O)(CNC(=O)CCC2CCCC(O)C2)CCCCC1 C1(OC)CCCCC1NC(c1cc(CN=C(NCc2ccco2)NC)c(C)o1)=O C1(C)(C(NOCCC=C)=O)CCCN(C(C2CC(=O)OC2(C)C)=O)CC1 N(C(=NCCc1ccsc1)NCCSC)C.Cn1nc(C(F)(F)F)cc1C1CCCC1 C(=O)(CC(C)C(F)(F)F)N1CCC(OCCNC(C2(COC)C=CCC2)=O)C1 CCCC(O)C(CO)NC(=O)C1=CCN(C(c2n[nH]c(C)c2C)=O)C1 N1(C(Cc2nn(C)c(Cl)c2)=O)CC(NC(=O)CCS(C)=O)C2CCCCC12 N1(C(c2c(CC)n(C)cc2)=O)CC2CCCC1CN(C(=O)Cn1cnnn1)C2 C1(NC(c2ncc[nH]2)=O)CC2(CCN(C(C3C4CCCCCCC34)=O)C2)C1 N1(C(c2ccn(C)c2CC(=O)O)=O)CCn2cc(C(=O)NC3CCOC3)nc2C1 N1(C(C2(CCC)CCCC2)=O)CC2(C)CN(C(C3(NC(N)=O)CC3)=O)CC2(C)C1 N1(C(C2CCC3(CCC3)O2)=O)CCC2(C1)CN(C(C1(c3cc[nH]n3)CCC1)=O)C2 N1(C(CC=CCC)=O)CCC(CNC(c2ccn3ncnc3c2)=O)C12CCC2 N1(C(c2cc(Cl)ns2)=O)CCC2(C1)CN(C(=O)CCc1ccc[nH]1)C2 C1(NC(=O)Cc2cc(Cl)cs2)CC2CCC1(NC(=O)CC1(O)CCCC1)C2 N1(C(C(=O)Nc2cn(CC)nc2)C)CCC(N(C(=O)COCC(=O)OC)C)CC1 C1(CNC(c2nccc(C)n2)=O)COCCN(C(=O)C(C)C2CCC2)C1 c1(CC(=O)NC2CC3CC2N(C(c2ccco2)=O)C3)ccc(Br)cc1F Cc1ccc(CC(=O)N(C)CC2C3CN(C(=O)C(C)(C)CO)CC23)cc1Br CCC(CCC(=O)N1CC(C(F)Cn2cc(CS(=O)(=O)CC)nn2)C1)OC(C)=O c1(CNCc2cc(Br)sc2)cc(N2CCCC2)ccn1 C(CCN=C(NCCCN(C1CCN(C)CC1)C)NCC1CC1)SC N1(C(C(C)CNC(c2ccc(CO)cn2)=O)=O)CCC(=C(F)F)CC1 N1(C(CC=CC)=O)CC(NC(C2(OC)CCSCC2)=O)CC1C N(C1CCCn2cnnc21)C(=O)NCc1ncccc1-c1nn[nH]n1 N1(c2nc(C)nc(Cl)c2)CC(NC(=O)C2=C(Cl)CC2)C2CCCCC12 C1(C#C)(C(N2C(C#C)CC2)=O)CCN(C(=O)C(C)C(C)COC)C1 c1(OC)cc(C(=O)NCc2ncccc2C(=O)NC(C)CC(C)(C)OC)ncn1 N1(C(CCC(C)(C)NC(C(n2ccc(C)n2)C)=O)=O)Cc2cccc(F)c2C1 c1(N(C(C2C(NC(CCSC)=O)CCC2)=O)C)cc(C)cc(F)c1 C#CCCCCCCC(=O)N1CCC(NC(c2cnc(C)[nH]2)=O)C1 c1(NC(=O)NC(C(=O)OC)C)ccc(C(F)(F)F)cc1[N+](=O)[O-].C12CCCN1C2 CC1CN(C(=O)CCOCC2CC2)CCC1NC(C1(C)CCSCC1)=O C1(C(=O)NCC(CC=C)CC=C)CN(C(c2cc(C)cc(C)n2)=O)CCC1(C)C N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)Cc2ccc(Cl)cc2Cl)CC1C(C)(C)C N1(C(c2c(CC)c[nH]c2)=O)CCC2C1CCCN2C(C1CN(CP(C)(C)=O)C1)=O C1(C(=O)NCC(C)N(c2ncc(C)c(O)n2)C)CC2(C1)NC(=O)NC2=O N1(C(CC(C(=O)OC)(C)C)=O)CCC2(CCC(NC(C3CC4(CCC4)C3)=O)C2)C1 N1(C(CN(CC(C)C)C(c2ccn(C3CC3)n2)=O)=O)CCCC2(CC2)C1 N(C)(S(=O)(=O)N(C)C)CC(=O)N(CC(CO)(CO)NC(c1cc(C)oc1C)=O)C C1(N(C(C(C(C)C)SC)=O)C)CCCCN(C(c2ccc(C)nc2O)=O)C1 C1(C(=O)NCC2CCN(C3CC3)C2=O)CCN2CCOCC12 c1(C(=O)NCC(=C)CCNC(=O)CCc2ccccn2)ccc(Cl)c(F)c1 C12(CC(N3CCC(OC)CC3)=O)CCC1CN(C(C1CCC(N(C)C)C1)=O)C2 c1(NC=O)ccc(C(=O)NC2CN(C(c3cc[nH]n3)=O)CC2F)cc1 N(C1c2ccccc2CC1NC(=O)C=CC=C(Cl)Cl)C(c1cncn(C)c1=O)=O N1(C(c2nc(C3CC3)n[nH]2)C)CC(O)CCC1c1ccccc1.C1(C)(C)CN1 c1(C(N(CCNC(C(C2CCC2)OCC)=O)C2CC2)=O)cc(I)c[nH]1 C(N=C(NN(C)CC1(O)CCOC1)NC1CCC1)c1ccc(N(C)C)s1 N1(C(c2n(CCOC)ncc2)=O)CCC(C)(NC(c2cc(Br)ccc2F)=O)CC1 c1(C(=O)NC2(CC=C)CN(C(C3CCCN4CCCC34)=O)C2)cncc(C)c1C N(C1CCCc2c1cnn2C)C(=O)NCCc1c(C)n(C)nc1 C12(NC(CC(C=C)(C)C)=O)CCCCCC1N(CC(=O)NC1CCCC1)CC2 CCCC(CCCNC(C1CC1C)=O)NC(=O)C=Cc1cncs1 c1(NC)cncc(C(N2CCC(C(C)NC(c3cc(C(F)(F)F)no3)=O)C2)=O)c1 N1(C(CSC)=O)CCC2(CCOC2)C(CNC(c2n[nH]c3cc(C)ccc23)=O)C1 c1(CC(=O)NC(C)CCNC(C2(CO)CCOC2)=O)ccc(Cl)cc1Br CC1(CNc2cc(CC#N)ncn2)CCN(C(=O)CCC2CC2)CC1 n1(CC)nc(C(C)C)cc1C(N1CCN(C(=O)NC=O)CC1)=O.C1(=O)CC(C)O1 CC(CC(=O)N1CC(C)(NC(=O)CC2C=CCCC2)C1)C(F)F N1(C(CC(C)N(C(=O)C=Cc2ccoc2)C)=O)CCCC(C)(O)C1 C(C)(C)(C(C)CC(=O)NOC(CO)C(C)C)NC(CC1CC(=C)C1)=O C1(C(N2CC(CNC(C(C)OCC3CCCCO3)=O)C2)=O)CCC(C)(C)CC1 CCCCC(CCCC)NC(C1C(C)OCCN1C(c1ccnn1C(C)C)=O)=O N1(C(CCCOCC=C)=O)CC2(CC2)CC1CNC(=O)C(C)(C)c1cnn(C)c1 C1(CC(N2CCC(CNC(C3(OCC)CCCC3)=O)C2)=O)CCCC(C)(C)CC1 N1(C(C2CC=C(C)CC2)=O)CC(O)C(O)C1CNC(=O)CCCN1CCCC1 c1(C(N(Cc2cn(C(C(OCC)OCC)C)nn2)O)=O)cc2c(Cl)cccc2[nH]1 c1(C(=O)NC2CCN(C(C34OCC(C)(C3)C4)=O)CC2)ccc2c(c1)OCCO2 C1(CC)CN(C(=O)CCC[N+](=O)[O-])CCC1NC(=O)C(c1ccccc1)O N1(Cc2cn(C(C)C)nn2)CC2C(NC(=O)CC3CCCOC3)C2C1 c1(CC(=O)N(CCNC(=O)CNS(=O)(=O)N(C)C)CC)c(C)[nH]c2ccccc12 CCC(C)C(C(=O)N1CCC(NC(=O)CC2(C(=O)OC)CCCCC2)C1)OC CC1CN(C(C2(CO)CCC2)=O)CC1(C)C(=O)N(C)CCOC(F)F C1(NC(c2c(C)cns2)=O)CCC(F)(CNC(=O)Cn2cnc(C#N)n2)C1 CON1CC(NC(CCC2(C)CN(C(C3CC4(CCO3)CC4)=O)C2)=O)CC1=O c1(C(=O)NC2(C)CN(C(c3coc(C(F)F)n3)=O)C2)cccc2c1OCC(=O)N2 c1(C(=O)NCCc2c(CNC(CC=C)=O)nco2)sc(F)cc1Br S(=O)(=O)(CCC(F)(F)F)N1CC2CN(S(CC#N)(=O)=O)CC21 N1(C(C(CCC)c2ccc(Cl)cc2)=O)CC2(CNC(=O)CSC)CC1CCO2 c1(CCCNC(=O)C(=O)NC2CCCC2)ccc(F)cc1Cl N1(C(C(C)OC)=O)CCCCC1C1CCN(C(C2CN(C)C2)=O)CC1 C12(CCCSC1)NC2.S(=O)(=O)(CCN(C)C)N(CC)CC C12CN(C)C3CC(OC)(CC13)OC2.c1(OC)ccc(Oc2ccccc2)c(OC)c1 CC(CS(C)(=O)=O)C(=O)NC1CC2(CCN(C(c3cn(CC(N)=O)nn3)=O)C2)C1 CCCC(C)C(=O)NCCN(C(C)C)CC1CCCCCC1 CCC(CC(=O)NC1(CN(C(=O)C(C(C)C)n2cccc2)C)CC1)C1CC1 C1(O)(CNC(CCCN(C(C)=O)C)=O)CCCN(C(c2cncc(N)c2)=O)CC1 c1(OC)ncc(C(=O)NC(C)CCCNC(c2coc(C(C)=O)c2)=O)c(C)n1 c1(C(=O)NCC2(NC(CC3CCCN(C)C3)=O)CCOC2)cc(F)c(Cl)cc1Cl c1(C(=O)NCc2c(C(N3C(C)(CCO)CC3)=O)[nH]cc2)cc(CO)ccn1 N1(C(C2N(C(c3ccn(C)c3)=O)CC(O)CC2)=O)CC2(CCCCC2)C1 N1(C(CCCN(C(C)=O)C)=O)CC(O)CC1CNC(=O)CC1CCSC1 N1(C(C(CC#C)NC(c2ccc(CC)cc2)=O)=O)CCN(CC)C(C)C1 CCC(C)C(=O)NCC(C(C)C)NC(C1CC(CC(=O)OC(C)(C)C)C1)=O N1(C(CC(C)(C)F)=O)CCC2C(CCN2C(C2CCC(=O)N2)=O)C1 S(=O)(=O)(c1ccc(N(C)Cc2cc(C)ccc2C)cc1Br)NC(CCC)C C1(C(=O)NCCN(C(=O)C(C)(C)C2CCOC2)C)CC(=O)OC1(C)C C1(C(N(CCO)CC)=O)CCc2nc(-c3cccc(C)c3OC)sc2C1 N1(C(C2N(C(C3N(C)C(=O)CC3)=O)CC=C2)=O)CC(F)(F)C(F)(F)C1 C1(C(N(C2CCCN(C(C3(C=C)CCC3)=O)C2)CC)=O)CCc2ccccc2C1 c1(NC2C(SCC)CCC2)cc(N2CCCC(F)(CF)C2)nc(C)n1 CC1CCCn2c(CC(=O)NC3C4CC3N(C(C3CC3C(C)(F)F)=O)C4)cnc21 C12CCN(C(C(=O)NC(CO)C3CC3)C1)C2=O.C1(CC)C=CCC1 C(=O)(CC(CNC(=O)CC(Cl)Cl)OC)NCC1(OC)CCC1 Cc1nn(C)c(C(=O)NC23CC2CN(C(=O)CNC=O)C3)c1[N+](=O)[O-] c1(C(N2C(CNC(=O)C=CC(=O)N(C)C)CC(OC)C2)=O)ccc2ccsc2c1 c1(CCC(=O)NCC2CC3CC3N2C(=O)CC2CC2)ccc([N+](=O)[O-])cc1Cl N1(C(=O)OC)CCS(=O)(=O)CC1.c12cccc(c1)NC(=O)CO2.C12CN(C1)C2=O N#Cc1c[nH]c2c(F)cc(F)cc2c1=NCC(O)CNC(=O)Cc1cscn1 c1(OC)c(C(=O)N(C)CC2CCCN2C(C2CC23CCOCC3)=O)cccc1Cl C1(NC(C2CCC(=O)C2)=O)CC2CCC1CC2NC(c1ccncc1Cl)=O n1(CCCOCCOC)ncc(-c2nc(COc3ccccc3)no2)c1C(F)(F)F N1(C(C2CN(C)C(=O)CC2)=O)C2CCC1CN(C(=O)Cc1cnns1)C2 c1(C(N2CC(n3cc(CCCCC)nn3)C2)=O)cccc2nn[nH]c12 c1(CN2CCC(NC(c3n[nH]cc3[N+](=O)[O-])=O)C(F)C2)cc2ccccc2cn1 C(=O)(C(C)C(O)C(C)C)N1C(CNC(c2ncc(OC)cn2)=O)CCC1 C1(C(C(=O)N(CC(C)NC(C2(CCC)CCC2)=O)C)C)CCOCC1 Cc1cc(N)c(C(N2CCCC(NC(=O)CC3CC3(Cl)Cl)C2C)=O)cc1C C1(NC(C2CC(OCC)C2)=O)CC(C)(NC(=O)C=C(CC)CC)C1 c1(OC)cncc(C(=O)NC2CC(N(C)C(c3ccc(C(N)=O)nc3)=O)C2)c1 Cc1[nH]cc(C(N2CCC(CCNC(=O)CCC3CCCC3)CC2)=O)c(=O)c1Cl C1(SC)CC(C(=O)NCCN(C(=O)NC(C)(C)C)CC2CC2)C1(C)C N1(C(c2cnc(OC)c(Cl)c2)=O)CC(C)CN(C(C2(C#N)CCCC2)=O)CC1C C1(CNC(COCCN(C)C)=O)(CO)CCCN(C(C2CCCO2)=O)C1 C1(NC(C(c2cnn(C)c2)NC(c2ccc(C)[nH]2)=O)=O)CCC=CCCC1 c1(N(C)CCC2CCCCN2C)nc2c(c(=NC3CCN(C)C(=O)C3)[nH]1)SCC2 CC1CCC1CC(=O)N(CCC(=O)N1CC(N2CCCC2)C1)C CCCCCC(C)(C)C(=O)NCC(C)(O)CNC(c1c(C)[nH]c2ccccc12)=O c1(C2C(C)C2)[nH]c(=NCc2cn(C)c3ccc(C4CC4)cc23)nc2sccc12 C1(CN(C(C2CCN(C(C)=O)C2)C(=O)NCCOC)CC)CCS(=O)(=O)C1 C1(N(C(C2CCC(C)(CC)O2)=O)C)CCC2CN(C(c3ccc(F)s3)=O)CC12 C1(CC(=O)NCC2(CN(C)C(c3ccccn3)=O)CC2)CCCCCCC1 N#CC1(C(=O)NCCC2CCN(C(=O)C(F)=C3CCCC3)CC2)CCCO1 Cc1cc(CNC2CCCN(CCF)C2)c2cn[nH]c2c1 CC1=NNC(=O)C1CC(N1CCC(CCC(=O)N(C(CF)CF)C)CC1)=O CCCCCC(CC)C(=O)N1CC(NC(c2cc(CC)on2)=O)CC12CCOC2 c1(-c2onc(-c3c(CSC)cccc3)n2)ccc(S2(=O)=NCCC2)cc1 CC(C)(O)C(F)CNC(=O)Cn1cc(-c2nc(Cl)cs2)nn1 CS(=O)C=CC(=O)NCC(c1cccc(C(F)(F)F)c1)NC(=O)CC1CSCCS1 Cc1cc(C(N2CCC(N(C(=O)COC(F)(F)F)C3CC3)CC2)=O)c(C)n1C N1(C(CN(C)C(N)=O)=O)CC2(CCC2)CC1C(=O)NCc1ncsn1 N1(C(C(=O)NC2CCOC2)c2cccs2)CCC(C2(O)CCOC2)CC1 C1(CCOC)(NC(=O)C(F)C(F)(F)F)CCN(C(c2coc(C(N)=O)c2)=O)CC1 c1(NC2CC(NC(C3N(C)C(=O)OC3)=O)C2)ncc2ccsc2n1 c1(C2(C(=O)NC(c3ccsc3)CO)CC2)cccc2c([N+](=O)[O-])cccc12 c1(OC)ncnc(OC)c1CNc1cnc(F)cc1C(=O)Nc1ccncn1 N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC(NCc2c(C(=O)O)cccc2F)C(F)(F)C1 c1(C(=O)NCC2C(NC(c3cncn(C)c3=O)=O)C2)cn2cccc(F)c2n1 Cc1ccc(C(=O)NC2CS(=O)(=O)CC2NC(=O)CC2CC=CC2)c(C)c1 C(C)(C1=CCN(C)CC1)NC(CN(C(=O)Cc1cn(C)cn1)C(C)C)=O C1(NC(CNC(C2C(C)C2)=O)=O)CC=C(C(=O)N2CC(O)(C(N)=O)C2)C1 N1(C(C2C(C)=C2)=O)CCN(C2CCN(C(c3cnc(Cl)cc3Cl)=O)CC2)C(=O)C1 C1(O)(CNC(C(C)N(CC)CC)=O)CCCN(C(c2cc(CO)on2)=O)CC1 N1(C(Cc2n(C)ncc2)=O)CC(NC(C2CC2[N+](=O)[O-])=O)CC1(C)C C=CC1(CO)CCN(C(=O)C(c2cccs2)NC(c2cn[nH]c2)=O)CC1 c1(NC2(CNC(c3ccc(O)nc3Cl)=O)COCCC2O)ccc([N+](=O)[O-])c(O)n1 N1(C(Cc2cc(C)nn2C)=O)CCC2(CC2C(N2CCS(=O)(=O)CC2)=O)C1 CCCC(C(=O)NCC1CC(NC(=O)CC23CCC(CC2)C3)C1)NC(N)=O C(C(C)(C)C(=O)NCC1CC(NC(=O)C(c2cncc(F)c2)C)C1)OC c1(C(N(C2CN(C(C(C)SC)=O)CC2(C)C)C)=O)c(C)ccc2n[nH]cc12 CS(C)(=O)=NC(=O)C(=O)N1CC2(C1)CN(C(c1c(N)cccc1F)=O)C2 N1(C(c2ccn(C)c2)C(=O)NCCCSC)CCN(CCNC2CCC2)CC1 CN1CCN(C(C2CCCO2)=O)C(CNC(=O)CCn2cc(Cl)cn2)C1 C1(NC(c2scc(C)c2)=O)CN(C(C2C3CCC2(c2ccco2)C3)=O)CCC1F N1(C(c2c(C)ncc(Cl)c2)=O)CCN(C(=O)CNC(c2ccoc2)=O)C(C)C1C N1(C(=O)COCC2CCCC2)CCC2CN(C(c3ccc4[nH]ccc4n3)=O)C2C1 C1(CNC(CCC(C)SC)=O)CC2(CCN(c3cc(=O)n(C)c(=O)n3C)C2)CO1 CN1CC2(CCN2C(c2c(CNC(C3(C)CCOC3)=O)nnn2C)=O)C1 N1(C(c2c(CC)cno2)=O)CCC(C(N2CCOCC2CC)=O)(CO)C1 c1(C(N(C2(CC(=O)N(C3CC(O)C3)C)CC2)C)=O)ccc(C#N)[nH]1 c1(C(=O)NC2CCCC(CCC)C2)cc(C)ccc1N(CC)CC N1(C(C(C)CC2CCC2)=O)CCN(C(c2cc(O)cnc2N)=O)C(C)C1 C1(C(C)N(C(=O)COC2CN(C(=O)CC3(C)CC3)C2)C)CC(F)(F)C1 c1(NC(C2N(Cc3cccc(N(C)C)c3)CCC2O)=O)c(F)ccc(Br)c1F N1(C(c2c(C)oc(CO)c2)=O)CCOC2(CCN(C(=O)C#CC3CCOC3)C2)C1 C1(C(N2CCC(COC)CC2)=O)C2CCC1CN(C(C1(F)CCCC=C1F)=O)C2 N1(C(c2cnc(CC)nc2C)=O)CCC2CC1CN(C(=O)C(C)(C)C(C)O)C2 C1(NC(c2n(CC)ccc2)=O)C2CCN(C(C3SCCCS3)=O)CCC12 C1(C(N2CC(O)C(O)C2)=O)CN(Cc2cc(F)cc(Cl)c2O)CC(F)(F)C1 C1(C(N(C)Cc2cc(CNC(=O)C(O)c3ccsc3)[nH]n2)=O)COCCN1C C(=O)(C(C)(C)CN(C)C(C1CCCN1C=O)=O)NCCC1CC(C)C1 CC(CF)CC(=O)NCC1(C(C)(C)C)CCNC1=O C(=O)(C1c2c[nH]nc2CN1C(=O)CCC1CCC(=O)NC1)N(CCOCC)C c1(C(=O)NCCN(C)C(C2CC23CCOCC3)=O)cccc(Br)c1Cl c1(NC(C(=O)Nc2ccc(NCC(F)F)cc2)=O)nc2c(s1)CC(O)CC2 n1(CCOC)cc(C(=O)NCc2nc(CNC(=O)CC(C)F)cs2)nn1 c1(NCC23CC2CN(CC2(C(C(CC4(C=C)CC4)=O)=O)CC2)C3)ccc2c(c1)OCO2 C(C)(CCCC(=O)N1CCN(C)CC1)NC(C1(CCC)CC(=O)C1)=O N1(C(CCC(C)(F)F)=O)CC2(CNC(=O)C(CO)C(C)(C)C)CC1CCO2 C(=O)(C(F)C(C)(C)O)N1C(C2(O)CN(C(Cn3c(C(C)C)nnn3)=O)C2)CCC1 Cn1ncc(S(C)(=O)=NC(=O)C2CC3CC2(c2cccnc2)C3)c1C(N)=O Cc1cnnc(NC(c2nnnn2C2CC(F)(F)C2)CC2CCC2)c1 c1(OC)c(Cl)cc(C(=O)NC2CCN(C(C3COC(=O)O3)=O)C2)nc1Cl Cc1ncc(C(N2CCC=CC2C(=O)NCCCOC2CC2)=O)cc1C#N C1(c2nn[nH]n2)(N(C(=O)C(C)(C)C)C(C)C(=O)NCc2ccco2)CCCCC1C N1(C(c2ccc(CC)cc2)=O)CCN(C(C2CCCCO2)=O)C(c2ncc[nH]2)C1 c1(OC)ccc(C(=O)NC2CC(C(=O)Nc3ccnc(C)n3)C2)c(F)c1F C(=O)(CC(F)(F)CC(=O)N1CCOCC(F)(CNC(C2(C)CCCO2)=O)C1)OC C1(CNC(=O)C(c2ccccc2)O)CC2(CO1)CN(C(=O)Cc1cc[nH]c1)C2 C(c1ccccc1)=C(OC)C(N1CC2CC1C2NC(=O)CSc1nnc(C)n1C)=O c1(C(N2CC(C(=O)Nc3cc(OC)c(Br)cc3)OCC2)=O)cc(F)cc(C)c1O C(CC(C)(C)C(=O)NC)N(C1CC(C(F)C(=O)C(N)=O)C1)C.c1(N)cc(C2CC2)no1 Cc1c(NC(C2C(C)CCN2c2nccc(C(C)(C)C)n2)=O)ccc2n[nH]cc12 C(=O)(CC(C)(C)CC(F)F)N1CCC(C2(NC(CCS(C)=O)=O)CC2)C1 CC1(C)CCC(CNC(c2cncnc2C2CC2)=O)N(CCC2CCC2)C1 c1(C)ccccc1CC.n1(CCOC)nnnc1C(c1cccs1)NCCSC c1(C(=O)NCC2C(NC(CCCC(N)=O)=O)CCC2)coc2c1C(O)CCC2 CCC(C)CCCCC(=O)N(C(C)CNC(c1cc(C)c(F)cn1)=O)C O=C1OCc2cc(C(=O)NC3CCCCN(C(c4c[nH]c(=O)cn4)=O)C3)ccc21 N1(C(C2(CC)CCC(O)CC2)=O)CCC2(CCC2CNC(=O)C(C)(C)CF)CC1 C(=O)(C(F)C(C)(C)O)N(CC(N1CCCC(OCC)C1)=O)C1CC1 Cc1csc(C(N2CC(CNC(=O)C=C3CCCCC3)C3CC23)=O)c1C C1(CN(C)C(c2ncn(C)n2)=O)CCCCN1C(=O)C(F)=C1CCCC1 N1(C(c2c(C)cnn2C)=O)CC2CCC2(CNC(=O)CSCCC(C)C)C1 N1(C(CCC=C=C)=O)CCC(NC(=O)COc2cncc(Cl)n2)C(CO)CC1 C(=O)(C1=CCc2ccccc21)NC1CC2CN(C(C(=O)NC(C)C)=O)CC(C1)C2 c1(C(=O)NC(C)CC(C)NC(C2(NCCO)CCC2)=O)cccc(=O)n1C c1(CSCC)cn(CCN(C(=O)C(CC)N2CCCC2=O)C)nn1 N1(C(C(C(C)O)C)=O)CCN(C(c2nccc3cc[nH]c23)=O)C2(CCC2)C1 N1(C(C2(OC)CCSC2)=O)CCCN(C(=O)C(C)c2ccsn2)CC1 C1(NC(CC2C(C)C2)=O)CC2CC(C1)N(C(c1cc(O)c(F)cc1N)=O)C2 Cc1cc(C(=O)NC(c2ccc(CNC(C3(Br)CC3)=O)cc2)C)cc(N)c1O C1(NC(C(CC=C)C)=O)CC2CC(C1)N(C(c1ccc(OC)s1)=O)C2 Cc1ncc(C=CC(=O)NC(CNC(=O)Cc2nnc(C)o2)C(C)C)c(O)n1 c1(C(CNC(c2c(CCC)n[nH]c2)=O)NC(=O)C(C)SC(C)C)cccc(C)c1 c1(CNC(C(C)CN(C(=O)CCN2CCCC2=O)C)=O)ccccc1C#N C(=O)(CC(c1ccccc1)C1CC1)NCC(C)NC(=O)CCC1(C)CCCN1 c1(OCCOC)ccc(CNC(=O)C(=O)Nc2cnc(CCN)nc2)cc1 CC1CN(CC(=O)NCC(C)(C)NC(=O)COCC(F)F)C1 N1(C(C=CC=CC)=O)CCCC(C)(C)C1C(N1CC2(CO)CC2(CO)C1)=O N1(C(C=C(CCC)CCC)=O)CCOC2(CCN(c3ccc(C#N)nc3)C2)C1 C1(C(N2C(CNC(CCOC)=O)CC(F)(F)C2)=O)CC2CC1C1C2C1(F)F N1(C(Cc2nc(C)sc2)=O)CCN(C(c2coc3c2COC3)=O)C(CF)C1 c1(C(N(CCNC(C2CCN(CC)C2)=O)CC)=O)cc2n(c1)CCC2 C1(C(N(C2CCN(C(c3nc(CCC)sc3)=O)C2)CC)=O)CCC(=O)NC1 c1(NC(C)=O)ccc(NCC(n2cc(C3(OC(C)C)CCOC3)nn2)C)c(F)c1 N1(C(C(C(C)C)O)=O)CC2CS(=O)(=O)CC2(NC(=O)C(F)=CCCF)C1 Cc1ccc(NC(=O)NCc2ccnc(N3CCCCCC3)c2)nn1 C=CCC(CC=C)C(=O)NC(CC=C)C(=O)NCCC1CC=CC1 c1(C(N(CC(C)(C)NC(C2CC(C)(C)CCO2)=O)C)=O)n[nH]c2ccccc12 c1(-n2ccc(CCNC(=O)NC34CC(CO)(C3)C4)n2)cccc(F)c1 c1(NCC(CC)C(C)C)[nH]c(=NCC(C)(C)N(CC(F)(F)F)C)nc2sccc12 C1(CNC(C(C)CNC(=O)C(C2(O)CCCC2)F)=O)CC12CCOCC2 C#Cc1ccc(C(N2CCN(C(=O)CCCc3cccs3)CC2C)=O)cc1C S(=O)(=O)(c1cccnc1)NC(C(=O)NCC1(NC(COC(C)C)=O)CC1)C(C)C C(=O)(CCC(C)(C)C(=O)OC)N1C(CNC(C(C(CC)O)(F)F)=O)CCCC1 N1(C(C2ON=C(C)C2)=O)CCC(O)CC1C(=O)NCC1CCCCN1C C1(NC(C=CC(C)C)=O)CCCC(CC(=O)NCC2(F)CCOCC2)C1 C=C1CC(CONC(=O)C2CC(NC(=O)CNC(=O)NC3CC3)C2)C1 S(=O)(=O)(c1c(OCOC)ccc(Cl)c1F)CCOc1ccc(C(=O)OC)cc1 C1(C)(C(=O)NCC(C(C)C)NC(c2ccccn2)=O)CC(C2CC2)=NO1 c1(-c2scc(C(=O)NC(c3ncc(F)cc3F)C)n2)c(Cl)cccc1Cl CC(F)(F)CC(=O)NC1CCC(NC(=O)CC2CCC23CCC3)C1 Cc1cc(C2CC2)ccc1C(=O)N(C)CC1CCCN1C(c1ncoc1C)=O Cc1c[nH]ccc1=NC(=O)c1cc(NC(C2CCC(F)(F)CC2)=O)cn1C C(CNC(=O)Cn1nnc(C2CC2)n1)(CC(F)(F)F)NC(Cc1c(C)n[nH]c1C)=O c1(C(=O)NC2C(C)CCN(C(c3cccn3C)=O)C2C)cccc2c1nnn2C c1(C(=O)NCCCOCCNC(C(C)C2CC2)=O)ccc(N(C)C)cc1 C1(C)(C(N2CC(O)(CNC(C3(OC)CCCOC3)=O)C2)=O)CCC(C)C1(C)C C(=O)(C1CCCn2cncc21)NC(CC=C)CNC(c1cn(C)ccc1=O)=O c1(C(=O)NC2(C#N)CCN(Cc3ccc(Cl)cn3)C2)cc2ccoc2cn1 CC(c1cnn(C)c1)=CC(=O)NCC1C2CN(C(=O)CCc3ccoc3)CC12 c1(NC(c2nc(C(=O)Nc3ccc4c(c3)OCO4)cs2)=O)cccc2ccnn12 c1(CC(N2CC(NC(C3(C#C)CCCC3)=O)C(OC)C2)=O)cnc2ncccn12 C1(CNC(c2c(CC)nco2)=O)CN(c2ccnc(Cl)n2)CCN1C C1(NC(Cn2ncc(CC)c2)=O)CCCN(C(C2CCC=CCCC2)=O)CC1 Cc1sc(C(N2CCC(C3CCCN3)C2)=O)cc1[N+](=O)[O-].C12=CC=C(C=C1)C2=O CCC(CC(=O)NC1CC(NC(C2CCCN2C2CC2)=O)CC1O)SC N1(CC)CCC(C(N2CCSCC2CCNC(c2cnn(C(F)F)c2)=O)=O)CC1 c1(C(=O)NCC(C)(C2CCC2)NC(C2Cc3nccn3C2)=O)cc2n(n1)CCC2 c1(C(=O)NC2CC3CN(C(c4cn(CC=C)nn4)=O)CC32)cnn2ccn(C)c12 C1(C(N(CCC(C(C)C)NC(CCCC=C)=O)C)=O)CC12CC(C)(C)C2 N1(C(C2CN(C)C(=O)CC2)=O)CCC2C(CCCN2C(c2cnc(S)nc2)=O)C1 c1(C(=O)NC(C(=O)N2C(CC)CC2)CO)ncncc1OC C1(C(N2CCN(C(C(C(CC)C)=O)=O)CC2C(C)C)=O)Cc2cccnc2C1 O=C1C2Cc3ccc(F)cc3N2C(=O)N1CC1(Br)CCOCC1 N1(C(C=COCC)=O)CCOC2(CCC(NC(=O)C(C)CSC)CC2)C1 CC(=O)CCCC(C)C(=O)NC(Cn1cncn1)C(=O)NCCCCC(C)(F)F C(C)(CCC(=O)NC1(CO)CN(C(=O)Cc2cccnc2Cl)C1)OC c1(C(C(=O)NCCSC)N(C2CCCC2(C)C)C)cc(S(N)(=O)=O)cs1 C1(C(N2CC(C(C(=O)NC3C(C)C3C)OC)C2)=O)(COC)CCCC1 C1(CN(S(=O)(=O)CCN(C)C(C)C)CC)C2CCC1(c1ccnn1C1CCC1)C2 C12(NC(=O)CSCc3ccc(N)cc3)CCC(C1)N(C(C1CCCCS1)=O)C2 C1(NC(CCCCCN(C)C(c2cc(C(F)F)[nH]n2)=O)=O)CCn2cnnc2C1 c1(C(N(C(C)C(=O)NC(CO)CCCO)CC)=O)ccc(=O)n(C)c1 C1(C(=O)NC2(CC(C)C=CCc3ccncc3)CCC2)CCCCCC1 C(=O)(CCCCN(C(=O)CCC1CC(F)(F)C1)C)N(C)Cc1cncn1C Cc1ccc(C(=O)NCC(=O)Nc2cn[nH]c2)cc1Br.C12CCCN1C2=O c1(C(=O)NC(C(C)NC(C(CCC)OCC)=O)CO)cc2ccncc2s1 CC(F)(F)C(=O)NC1CCCC1NC(=O)CNC(c1ccco1)=O Cc1ccc(C(=O)NCC(C)(F)CNC(=O)C(C)C#N)cc1F C12(NC(=O)Cc3cnns3)CCCCC1N(C(=O)CS(=O)(=O)C1CC1)CC2 c1(C(=O)NC2CC(NC(=O)CC(c3ccc(F)cc3)O)C2)ccnc2ncnn12 N1(C(=O)NC2C(c3c(-c4c(C)n[nH]c4C)cncc3)C2)CCc2cccnc2C1 C(=O)(C(O)CCC(C)C)NC1(C(N2CC(CCCCC)C2)=O)CCSC1 c1(NC(CCCC)(COC)c2nnnn2C)ccc2oc(C(F)F)nc2c1 C1(C(N(C)CCc2ccccc2)=O)CC12CCN(c1nnc(C(F)(F)F)o1)CC2 c1(OC)ccc(Cl)cc1C(N1CC2CC1CC2NC(c1ccnnc1O)=O)=O C=CCC(CNC(C1CCCN1CC(C)C)=O)NC(c1cc(CO)[nH]n1)=O c1(CC(=O)NCCN(C)C(c2ccc3nonc3c2)=O)cncc2ccccc12 C1(SC)CN(C(C2CC(n3cccn3)C2)=O)CC1NC(=O)CNC(C1CCC1)=O C(=O)(CCCCC(F)(F)F)NCC1N(C(C=C(C)Cl)=O)CCC1(C)C C1(NC(CC(n2ccc(C)n2)C)=O)CN(C(c2cc(C#N)cs2)=O)CC(C)(C)C1 C1(NC(CCC(C)OCC)=O)CCC(C)N(C(=O)Cn2ccsc2=N)C1 C1(O)(C(C)NC(c2occc2C(C)C)=O)CCN(C(=O)CCSc2ccccn2)C1 C1(CNC(C(C=C)O)=O)CC12CCN(C(=O)CCCCC#N)CC2 C1(CC(=O)NCC2(F)CC(NC(CCC3(C)N=N3)=O)C2)CCC(F)(F)C1 Cc1ncnc(O)c1C(N1CCC(CCCNC(C2(CO)CCCO2)=O)CC1)=O Nc1cc(CC(=O)NCC(CNC(C2(C(F)F)CCC2)=O)CO)ccc1[N+](=O)[O-] n1(CC)cc(Br)c(C(=O)Nc2ccc(NC(=O)CNC3CC3)cc2)n1 C1(C)(C(=O)NC2C=CC(C(=O)NC(c3cn(C)nc3)CO)C2)CCSCC1 c1(CC)cccc(OCC(N2CC(O)(CN(C(=O)CCC(C)OCC)C)C2)=O)c1 Cc1cc(C(=O)NCC(CC(F)(F)F)NC(=O)CC2CCCCN2C)cc(C)n1 N1(C(C(C)(C)CF)=O)CCC(C2(O)CC(NC(C3C=CCCC3)=O)C2)CC1 N1(C(C(CCCC)O)=O)CCN(C(=O)Cc2ccoc2)CC(C)(F)C1 c1(CC2C(C(=O)NC(c3n(C)ccn3)C(F)F)C2)cccc(I)c1 c1(C(=O)NCCC)ccc(-c2cncnc2C(N2CCN(CCC)CC2)=O)cc1F CC(C)CC(O)C(=O)N(C)CC1(O)CCN(C(=O)Cc2ccc(F)cn2)C1 Cc1cc(Cl)n[nH]c1=NC(=O)C1CCN1C(=O)C1=NOC(C)(C)C1 C1(NC(C2N(C(C)C)CCC2)=O)CCN(C(C2CC3(CCC3)CO2)=O)CC1F c1(CN(c2n(CCC=C)c(CC3CC3)nn2)C)ncc2n1CCCC2 N1(CC)C(=O)CCC1CC(=O)N(C1CCN(C(c2cc(C)sn2)=O)CC1)C C1(NC(c2c(C)cnn2C(C)C)=O)CC2CCC1N2C(=O)CCC1CC1 N1(C(C2C(CC)CCO2)=O)CC2(NC(=O)C(=O)Nc3ncc[nH]3)CCC1CC2 C1(CNC(c2c(C)oc(-c3ccccc3)n2)=O)C(C2CC2)CCN1C(=O)CC#N Cc1c(C(N2C3CN(C(=O)CCC(N)=O)CC23)=O)ccc2c1OCCO2 C(=O)(C(C)(C)CCC(C(=O)NCCC#N)N1CCOCCC1C(C)C)OCC c1(C(=O)NC(C(C)NC(C(=O)NCCOC)=O)C)ccc(OCC(F)F)cc1 c1(CC)ccc(F)cc1NC(=O)CCCCNC(=O)C=Cc1ccn(C)c1 C1(NC(C2(S(C)(=O)=O)CC2)=O)CCCN(C(=O)C2=COCCO2)CC1 c1(C(=O)NCC2C(NC(c3c(C)nc(C)s3)=O)C2)cc(N)c(F)c(O)c1F c1(C(c2n(CC=C)nnn2)NC(C2CC2)C2CC2)ccc(-n2cncn2)c(F)c1 N1(Cc2ccc(N(C)C)cc2O)CC2CN(C(c3ccc(F)c(Cl)c3)=O)CC2C1 c1(C(=O)NCC2CCC(NC(c3cnc(COC)s3)=O)C2)c(C)nc(C)o1 C1(CC(=O)NC(CC#C)CCOC)N(C(c2ncc(CC)cn2)=O)CCC1(C)C c1(C(=O)NCC2CCN(C(Cc3cccc(OC)c3)=O)C2)nc(Br)cnc1N N1(C(C2(COC)CC2)=O)CCC(C(C)C(=O)N(C2CC(C)C2)C)CC1 c1(C(=O)NC(CC(C)NC(c2cn(CCF)nn2)=O)C)cccc2sncc12 CCCCCCC(F)C(=O)N(CCNC(=O)CS(=O)(=O)N(C)C)C1CC1 Cc1c[nH]cc(C(N2CCC(OC3CN(C(C4CNC(=O)C4)=O)C3)CC2)=O)c1=O C1(CC(N2C(C)CC2)=O)COCCN1C(C1CCCC(=O)C1)=O c1(N(CC(C)(C)CO)C(c2ccccc2OC(F)F)=O)ncnc2cc[nH]c12 c1(CC)ncc(C(=O)NC(C2CN(C(=O)CCc3cc[nH]n3)CCO2)C)c(O)n1 c1(C(C)C(=O)NC2CCCC(C(F)(F)F)C2)cccc(-c2nn[nH]n2)c1 C1(CC(=O)NCC2(COC)CN(C(=O)CCc3nccn3C)C2)COC(C)(C)C1 c1(C(N(CC(O)CNC(=O)CN(C2CCCC2)C)C)=O)cc(=O)n(C)cn1 N1(C(C(CC)(C)C)=O)C2CCC1CC(CC=C)(NC(c1ccn(C)c(=O)c1)=O)C2 c1(CC(C)C)cc(C(=O)NC2CCC(NC(C3(C(N)=O)CC3)=O)CC2)cc(O)n1 O=C(CCCCC(F)(F)F)NCC1CC2(CCC2)CN1C(=O)Cn1cccc1 C12(NC3CCN(c4cn(C)nc4)C(=O)C3)CCN(C1)C(=O)NC2=O N1(C(C(CCC)n2cccc2)=O)CCOC(C(=O)NCCCOCC)CC1 c1(NC(C(N2CCC(F)(C(=O)OC)C2)=O)=O)ccc(F)cc1C1CC1 C1(CNC(COCCSC)=O)CCN(C(=O)Cn2cccn2)CC1(F)F c1(NC(N2CC(C(C(=O)OCC)F)C2)=O)ccccc1OCC c1(N2CCC(N(C(=O)C(F)=C3CCC3)CC)C2)ncc([N+](=O)[O-])cc1C(F)(F)F N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCN(C)c2ccc(C)cc21 N1(Cc2ccccc2)C(=O)CN(CCC2(C)CC2)C1=O.CCC1(C)CN1C C(CCN(C)C(c1ccc(C(F)F)o1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O N1(C(c2ccc(CC)s2)=O)CCC(C)(C)C1C(=O)NCCF C1(NC(C2CC(C3CCC3)C2)=O)CCCCN(C(c2ccco2)=O)C1 Cc1cc(C(=O)N(CC(C)NC(c2ccnnc2C)=O)C)cc(C)c1F C1(NC(CC2N(C)CCC2)=O)CCC12CCN(C(c1cscn1)=O)CC2 CC1(C)CCN(C(=O)C#CC2CCC2)C1C(=O)NCc1ncc(F)cc1F c1(COC)ccoc1C(=O)N(C)CC1CCCN1C(=O)C(F)Cc1ccccc1 c1(C(=O)NCC2(O)CCN(C(CCCCOC)=O)C2)cc(Cl)c2ccccc2n1 C12(CNC(CC3OCC(C)(C)OC3)=O)CCCC1N(C(c1csc(Cl)c1)=O)CC2 CC(C)C(C)(CNC(=O)CSC1CCCO1)NC(c1cccn(C2CC2)c1=O)=O C(=O)(CC(C)(C)CCOC)N1CC(N(C(c2c(CC)nccn2)=O)C)C(O)C1 C(=O)(CC(=O)N(C)C)N(C(C)C(=O)NCC(CC1CCCCC1)(C)C)C N1(C(C(n2ccc(C)n2)C)=O)CC(O)CC1C(=O)NCC(C)(C)CC1CC1 C(C)(C(C(=O)NCCC1CCOC1)NC(c1cc(C)sc1N)=O)OC c1(C(N2CC(C(C)NC(c3ccc(Cl)s3)=O)C2)=O)cn2c(n1)CCCC2 c1(CC)cc(F)cc(C(=O)NCC#CC2CCCCO2)c1C N1(C(C2CN(C(N)=O)C2)=O)CCCCC1C1CCN(C(=O)CCc2cn[nH]c2)C1 C1(C(N2C(C(C)C)CC2)=O)CN(C(=O)C(C)C2(O)CCC2)CCN1C C(=O)(CCCCCC#N)NC(C1CCN(C(C2CCCC(F)C2)=O)C1)C Cn1cnc(C=CC(=O)NCCCCC2CN(C(c3cc(C(F)F)cs3)=O)C2)c1 C1(CN(C(C2CC2c2cccnc2)=O)CC)CC(F)CN1C(=O)C(Cl)=CCl CN1CCN(C(=O)CCC2(C#N)CCC2)CC1CNC(c1cnn(C)c1N)=O c1(C(=O)OC)ccc(=NC(=O)CCc2ccccc2OC)[nH]c1F N1(C(C2(C)CCSCC2)=O)CC2CCC(C1)C(NC(=O)CC1CSCCO1)C2 C1(NC(=O)Cc2csnn2)CC2(C1)CN(C(c1cnc(-n3cccn3)cn1)=O)C2 C1(C(=O)NC(C(C(=O)OC)C)C)CC2CC1CN(C(=O)C(c1ccn(C)n1)C)C2 C1(NC(C2C(=C)C2)=O)C(C)(C)CN(CC2CN(C(=O)C(C)(C)C)CCO2)CC1(C)C c1(C(=O)NC(CNC(C2(CC)CCCCC2)=O)CO)cccc2c1COCCN2 N1(CCNC(=O)C(O)CF)CCCN(C(c2ccn(-c3ccccc3)n2)=O)CC1 c1(OC)cc(CO)ccc1CCNC(N1CC(CO)OCC1C)=O N1(C(C(C)(CO)OC)=O)CCOC2(CCN(C(c3cc(Cl)cnc3C)=O)C2)C1 C1(C(=O)NCC#CC)(NC(=O)C(=Cc2ccco2)C)CCSC1 Cc1cncc(C)c1C(=O)NCCCC1CCN(C(C2C(C)C2C)=O)CC1 c1(OC)cc(F)c(C(N2CC(=C(F)CNC(C3(O)CCC3)=O)C2)=O)cc1N S(=O)(=O)(c1ccc(=NCc2ccno2)[nH]c1)NCc1cccc(OCC)c1 c1(CC(=O)O)ccc(-c2csc(CN3CCCC3CCOCBr)n2)cc1 C1(C)(C(=O)NC(CN(C(=O)CSS(C)(=O)=O)CC)C)COCCO1 C(=O)(C1=NN(CCO)C(=O)CC1)N1CC2(CC(CNC(C(CC)C(C)O)=O)C2)C1 C12(CC(=O)NC3(COC)CN(C(C4CC5CCCC45)=O)C3)CCCCC1C2(F)F N1(S(CCC=CCOc2c(C(C)(C)C)ccc(Cl)c2)(=O)=O)CC(C(=O)O)C2(CC2)C1 C1(C(=O)NCC2(NC(CCN3CC(=O)NCC3)=O)CC2)CCC(C2CC2)C1 CC1CN(C(c2coc(O)n2)=O)CC1NC(c1ccc(SC(F)F)cc1)=O C(C#Cc1cn(C2CCCC2(C)O)nn1)NC(Cn1ncc(C)c1)=O C(=O)(CC(O)CNC(C1CN(C)CCO1)=O)Nc1c(CC)csc1 CCC(C(=O)NC1(CNC(C2(C)CC2(C)C)=O)CCCCC1)C(C)C c1(C(=O)NC2CN(C(C(C)NC(N)=O)=O)CC2C)cc(O)nc(N(C)C)n1 C(=O)(CC(C)(C)C(F)F)N1CCC(C(N(CC)CC2CC2)=O)OCC1 Cn1c(=O)oc2cc(CN3CC4C(NC(c5ccc(O)cc5)=O)C4C3)ccc12 N1(C(C2(N(C(c3nc(C)c(C)s3)=O)C)CC2)=O)CCCC2(CCC2)C1 N1(C(C(c2ccncc2)OC)=O)CCCC2(CCN(C(C3(F)CCCC3)=O)C2)C1 N1(C(C2(NC(C3CN(C)C3)=O)CC(O)C2)=O)CC(CO)C2(CCC2)C1 Cc1cccc(C)c1OCC(O)CNCc1ccnc(NC(=O)OC(C)(C)C)c1 C1(CNC(=O)C(N2CCC(CO)C(O)C2)c2cncc(F)c2)CCC(F)(F)CC1 CCCCC(C(=O)NC)N(C)CC.C(=O)(C(C)(C)N1CCCC1)N1CC(=O)OCC1 N1(C(C(N)=O)=O)CCN(C(C2CC3CCC3C2)=O)CC1CF C(CCC(C)(C)O)NC(C1C(NC(C(C)N2CCC2)=O)COC1)=O N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(=O)C(Cl)=CCl)C(C)(C)C1 C1(C(N2CC(CC(C)NC(=O)CC(C)(C)C3CC3)C2)=O)CC2(CCOCC2)C1 N1(CCCC)CCC(NC(c2cn(-c3ccc(C)cc3OC)cn2)=O)C(O)C1 c1(-c2cn(CC)nc2)ccc2cc(C(=O)NC(C)(CO)CO)cn2c1 N1(C(C)C)CCOC(C(=O)NCC(C2CC2)NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 CC1CN2CCN1CC2C(=O)N(CCCCCNC(=O)Cc1ccsc1Cl)C CC1(C)COC(CC(=O)NC2(CF)CCN(C(=O)CC3CCCCC3O)C2)C1 N1(C(c2c(C#N)scc2)=O)CCCC2(NC(C3CCCOCC3)=O)CCCC12 c1(C(N2CCC(N(CCC)C(c3cccc(OC)c3)=O)C2)=O)ccc(N)c(N)n1 C12CCN(C13CC3)C(=O)CC1CC(C1)C(=O)N2.Cc1nccn1CCC(=O)N(C)C c1(NC(c2nnnn2C2CCOC2)C2(CO)CCC2)cc(Cl)c(Br)cn1 CC(C(=O)N1CC(CNC(=O)C(=O)N(C)C)C1)n1ccnn1 c1(SCCC(=O)NC2CC(NC(C3CCC(OC)C3)=O)C2)ccc(F)c(F)c1 C1(CCNC(C(=O)NC2(C#N)CCC2)=O)CCC(F)(F)CC1 c1(C(N2CC=CC(NC(C3CCC3(F)F)=O)C2)=O)ccc(F)c(O)c1 c1(C(=O)NCC(C(C)(C)C)NC(CCC#C)=O)cc2n(n1)CC1(CC1)C2 C(=O)(CC1=CCN(C(=O)CC(C)F)CC1)N1CCCC(C)(OC)C1 c1(C(=O)NC2(C)CC(NC(C3C(CC)OCC3)=O)C2)cc[n+]([O-])cc1 Fc1ccc(C(C2CC3CC3C2)Nc2nnnn2CC2CC2)nc1 N1(C(CCCOCC)=O)CCN(C(=O)COc2ccc(OC)cc2)C2CC12 CC(C(C)C(=O)NC1CC2(CCN(C(c3coc(O)n3)=O)CC2)C1)S(C)(=O)=O CCC(CNC(c1c(CNC(c2cc(C3CC3)[nH]n2)=O)nnn1C)=O)CCO C(CCCCC(=O)N1CC(C)OC(C)C1)N(C(CC(C)OC)=O)C c1(NC(CC2N(CC3(C)CC3(Cl)Cl)CCCC2)=O)ncncc1C#N n1(C2CCN(C(C(N3C(=O)CCCCC3)C3CC3)=O)CC2)cnc2cc(Cl)ccc12 c1(C(=O)NC2(CC)CN(C(C34CCC(OC)C3C4)=O)C2)ccc(F)cc1 CCC(C)C(CS(=O)(=O)c1ccccc1)NC(=O)C(C1CCCCC1)C CC1=CCC(NC(=O)C(Cn2cncn2)NC(C23CSCC2C3)=O)CC1 Cc1nnccc1C(=O)NC(C1CCCC1)CNC(C1(C2(C)CC2)CC1)=O N1(C(c2cc(C)c(Cl)cc2)=O)CCC(C)N(C(c2nocc2Br)=O)CC1 C(=O)(C1=Cc2cccc(OC)c2OC1)NCC1CCC(NC(CC)=O)C1 c1(OC)cc(CN(C)C(C2CNCCO2)=O)cc(Br)c1OC C1(NC(CN(C(C)C)C)=O)COCC1CNC(C1CCOC1)=O c1(N(C)CC2CCCN2C(Cc2cccc(OC)c2)=O)ccc([N+](=O)[O-])c(C)c1 CCC(C)(CC)C(=O)N1CCN(C(c2cccc(OC(C)C)c2N)=O)C(CO)C1 c1(NC(N2CC3CCCC(C3)C2)=O)cnc2[nH]cnc2c1 C1(OC)(CNC(=O)CN2CCNC(=O)C2)CCN(C(=O)CCCn2ccnn2)C1 c1(C(CCC(=O)NC2(C)CCN(C(CCOCC#C)=O)C2)=O)ccc(O)c(F)c1 c1(SC)ncc(C(=O)NCC2CCC(NC(=O)CCC3CC3)C2)s1 C1(N(C(=O)CCCF)CCC)CCN(C(=O)CC2(C)CCCO2)CC1 Cc1ccc(C=CC(=O)NC2CCC(CNC(=O)COCc3nc[nH]n3)CC2)s1 c1(-c2cc(CNC(Cc3nc(C(=O)O)sc3)=O)no2)c(Cl)cccc1Cl C(=O)(CCC(CF)CF)NC(CC(=C)Cl)C(=O)N1CC=C(CO)CC1 O=C(CC(F)(F)C(F)F)NCCCNC(c1ccnn1CCF)=O N1(C(CC=CCC)=O)CCC2CCC(NC(=O)CCNC(=O)CO)C1C2 C1(C(=O)NCC(C)(C2CCC2)NC(CC=CCC)=O)Cc2nn(C)cc2C(=O)N1 C(=O)(C(C)CCC(C)(C)C)N1C(CNC(c2cc(OC)n[nH]2)=O)CC2CC21 N1(C(c2cccc(C)c2N)=O)CC2CCCC2(C(=O)NOC(C)C)C1 C1(C(NOCC)=O)C(C)OCCN1C(=O)C(C)OC(C)=O Cc1ccc(N(C)C)c(N2CCNC2=O)c1.c12cc(ccc1O)NC2 N1(C(C(=O)NCCCC=C)=O)C2CCC1CC(F)C2 C1(C(N(CC(C)(C)NC(c2cc(C(F)(F)F)n[nH]2)=O)C)=O)CCn2ncnc2C1 C1(C(N2CCCC(C(=O)NC)C2)=O)COCCN(C(C2CN(C(N)=O)C2)=O)C1 C#Cc1cnc(N2CCC(CNC(c3cnc(F)c(F)c3)=O)C2(C)C)nc1 C1(C2CN(C(=O)CCCC(F)F)C2)(NC(C2CCCC(C)C2)=O)CC1 N1(C(C(CC)COC)=O)CCCN(C(c2cc3sccc3[nH]2)=O)C(C)C1 c1(N2C(C)(CNC(C3(C)CCCS3(=O)=O)=O)CCC2)nccn2nnnc12 N1(C(c2csc(Cl)n2)=O)CCC(CNC(C23CC2Cc2c[nH]nc23)=O)C12CCC2 c1(CN(C)C(=O)NCC2CCOC(C(=O)OC(C)(C)C)C2)c(Cl)cncc1Cl N1(C(c2ncc(C)cc2C)=O)CC(C)(C)OC2(C1)CN(C(c1[nH]cnc1C)=O)C2 C(c1ccc(C)cn1)=CC(=O)N(CC(CC)NC(C1CCC=CCCC1)=O)CC Cc1ccc(F)c(C(N2CC(NC(=O)CCOC3CCCOC3)CC(O)C2)=O)n1 CCCCC(CNC(c1sccc1OC(F)F)=O)NC(C1(CF)CC1(F)F)=O CCC(CC(=O)NC(COC)C(C)C)N(C)C(c1cc(C)c(C)[nH]1)=O C1(C(N2CC(F)(CNC(C(C)OCC)=O)C2)=O)CCC(C(N)=O)CC1 Cc1ccn(CC(=O)NC2(C)CC(NC(=O)CCCN(C)C(C)C)C2)c(=O)c1 Cc1cc(CC(N2CCC(CNC(c3cnn[nH]3)=O)C2)=O)no1 N1(C(COC)=O)CC(CC(=O)NCC(C2CCC2)OC)CC1(C)C Cc1nnn(CC(=O)NC(C(=O)NC(C2CCCO2)CO)C2CCCC2)n1 C1(NC(C2(NC(=O)CN3CC(=O)NC3=O)CCN(C)C2)=O)CC1C1CCOCC1 N1(C(C2(C(=O)OC(C)(C)C)CCC2)=O)CCC(F)(C(N2CC(N3CCCC3)C2)=O)C1 C12(NC(=O)Cc3ccc(CO)cc3)CCCC1CN(C(=O)C1=COCC1)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCC2CN(C(=O)Cc3cc(C)sc3C)C2C1 CCCCCCN(CC(N1CCC(N(C(=O)CC2CCCSC2)CC2CC2)C1)=O)C C12(NC(COCCC#C)=O)CCC(C(=O)NCC3CCCC3CF)(CC1)C2 C(CCN=c1[nH]c(=NCc2cccnc2N(C)C)[nH]c2ccsc12)N(C(C)=O)C N1(C(C(c2cnccn2)C)=O)CC(NC(=O)CN(C)Cc2ccco2)CCC1C c1(CCC)ncc(C(=O)NCC2CC(NC(=O)CCc3ccc(C4CC4)o3)C2)s1 c1(C(N(CCC2N(C(C=CC(CC)C)=O)CCCC2)C)=O)cc(Cl)ccc1C c1(C(N)=O)nccnc1C(=O)NC(c1ccccc1F)CNC(=O)C(O)C1CC1 N1(C(C(=O)NC)=O)CCOCC(C(=O)NCCC(C)N2CCCC2)C1 c1(C(=O)NC2CCCC(N(C(CCOCC#C)=O)C)C2)ccc([N+](=O)[O-])cn1 C1(OC)CN(C)C(C)(C(=O)NC2CCN(C(c3nccnc3C)=O)CC2)C1 C1(C(=O)NC2(CCNC(C=CC(C)(C)C)=O)CC2)CCN(C2CC2)C1=O c1(OC)ccc(COCC(=O)NC23CC(C2)N(C(C2CC24CCOC4)=O)C3)cc1 N1(C(Cc2c(C)noc2C)=O)CCC2(CCCN2C(=O)CC2CCC(C)(C)C2)C1 c1(C(N2CC3N(C(C(CC)=O)=O)C3C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1Cl Cc1cc2[nH]c(C(N3CCCN(C(=O)CC(=O)NCC4CC4)C(C)C3)=O)cc2o1 c1(CC(=O)OCC)cc(Cl)ccc1NC(c1csc(N(c2ccccc2)C)n1)=O C1(c2n(C)ncc2)CC(CNC(=O)C(=O)N(CCCCCCO)C)C(O)C1 c1(OC)cc(C=CC(N2CC3CCN(C(=O)C(C)CBr)C3C2)=O)ccc1O N1(C(c2cc3nc[nH]c3cn2)=O)CCN(C(c2cnns2)=O)C2CCCCC2C1 CC(C)C1=CCC(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])o3)=O)C23CC3)CC1 C1(NC(c2c(OCC)cccn2)=O)COC2(CCCN(C(=O)CC3(C)CC3)C2)C1 C1(NC(=O)COC2CC=CC2)CCC(NC(=O)Cc2ccnc(O)c2)CC1 c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)C)c[nH]c2c(F)c(F)ccc2c1=O c1(NC(c2c(-c3cnn(CC)c3C)csc2)=O)cccc([N+](=O)[O-])c1Cl N1(C(c2n(CC=C)ccn2)=O)CCCC2(C1)CN(C(=O)CC(O)C(C)C)CCO2 N1(CC)CCOCC1CC(=O)NC1CN(C(=O)C=CSC)CC1C(=O)O N#CC1(C(N2CCCN(C(=O)COCC3CCCO3)CC2)=O)CCSCC1 c1(OC)ccccc1C(=O)NC1CCCC1C(=O)Nc1ccccc1N(C)C C(c1c(C)nn(C)c1Cl)=CC(=O)NCCCCNC(CC1CC(CC)OCC1)=O CCC(COCC1CC1)N=c1[nH]c(=NC)[nH]c(=NCC2(C)CC2(C)C)[nH]1 N1(C(CC2N(C(C3(C(=O)NCC(=O)OC)CC3)=O)CCCC2)=O)CCC(O)C(C)C1 C(=O)(CC1=CCN(C(C2CCCN2C(C)C)=O)CC1)NCC1N(C(C)=O)CCC1 c1(C(=O)NC2CN(C(C(CC)C)=O)C2)cc(Br)c(Cl)s1 C1(C(=O)NCC(C2CCCC2)NC(C(C(C)C)(C)C)=O)CCCCN1S(N)(=O)=O N1(C(C2CN(C(CCCCSC)=O)CC23CC3)=O)CCC2(CCCC2)C1 C1(NC(C2CCCC23CCC3)=O)CC2CCC(C1)N2C(=O)Cc1cc(C2CC2)on1 c1(C(=O)NCC2(NC(CS(CC)=O)=O)CCCCC2C)cn2c(n1)COCC2 c1(C(=O)NCCCCC(C)NC(=O)C=C2CCN(C)C2)ccn2ncccc12 C12(C(=O)NCC3CC(C)N(C(C4C(C)(C)C4(F)F)=O)C3)CCC(F)(CC1)CC2 N1(C(C(=Cc2cn[nH]c2)C)=O)CCCC(CNC(C2C(C)C2C)=O)C1 C=C=C(C)CC(=O)NCc1cccc(NC(C2CCC(C(F)(F)F)O2)=O)c1 C(=O)(C1=CCN(C(c2cnn(C3CC3)c2C)=O)C1)NCCC1ON=C(C)C1 c1(OC)cc(NC(c2n[nH]cc2NC(c2ccc(Cl)c(F)c2)=O)=O)cc(Br)n1 Cc1cc(=NCc2cccc3c2CCN3)[nH]c(NC2CCCC(C)(C)C2)n1 Cc1nn(C)c(C)c1C(=O)NCC1(F)CCCN(C(C2C3CCC(=O)C23)=O)C1 c1(N2CCN(C(C)=O)CC2)nc(=N)nc(N(CCC#N)C)[nH]1 CC(C)=C=CC(=O)N1CC(O)CC1CNC(C1CC2(CC2)CO1)=O CCC(CC)CC(=O)NC1(CNC(C2CC23CCCOC3)=O)CCCC1 Cc1cc(F)c([N+](=O)[O-])cc1NC(C1CCN(C(c2cc(F)ncc2Br)=O)C1)=O Cc1cc(C(=O)NC2CN(C(=O)C(C)(C)O)CC2F)c(S(N)(=O)=O)s1 N1(C(C2CCN(C(CC(CC(C)C)O)=O)C23CCC3)=O)CCc2cccnc2C1 Cn1cc(C(F)(F)F)c(NC(C2CC2NC(C2(c3cn[nH]c3)CC2)=O)=O)n1 N1(C(C(C=C)O)=O)CCCC2C1CCN2C(c1cc(Br)cn1CC)=O Cc1nc(F)ccc1NC(C1CC(C)N1C(C1CC(=C2CC2)C1)=O)=O c1(C(=O)NC(C(=O)N(CC(CC)(F)F)C)CC(F)F)cncc2[nH]ccc12 N1(C(C(CCC=C)NC(C23CC(CN2C2CC2)C3)=O)=O)CCOC2COCC12 C#Cc1cc(C(=O)NC2(C)CCN(C(c3ccnn3C(F)F)=O)C2)cc(F)c1 C1(NC(Cn2nc(C)c(Cl)c2)=O)C2CC1N(C(c1cn(C3CC3)cn1)=O)C2C CC(C(=O)N1CCC(CNC(c2ncn3c2CCC3)=O)C(C)C1)P(C)(C)=O CC1CCCCN1CCCC(N1CCC(N(C)C)C1)=O.c12ccc(cc1)c(=O)[nH]2 CCCC(C)(O)C(=O)N(CC(O)CN(C(=O)Cn1nc(O)ccc1=O)C)C c1(CCC)ccc(C(=O)NC2CCC(NC(=O)CCc3ccc(Cl)cc3)C2)cc1 C1(C(N2CC(C=C)C(OC)C2)=O)CC2CCC(C1)N2C(=O)Cn1ncnn1 c1(CC(=O)NCC2(F)CC(NC(CCCN(C)C)=O)C2)c[nH]ccc1=O N1(C(C2(C)C(C)CCCC2)=O)CC=C(CC(=O)NC2CC(CCF)C2)CC1 N1(C(c2cc(C3C(C)C3)no2)=O)CCC(c2cn(-c3ccncc3)nn2)C1(C)C Cc1cccc(C)c1NC(N(C)Cc1ccc(F)cc1Br)=O c1(SCC(N2CC(CCC(F)(F)F)C2)=O)scnc1C1CCCC1 CC(CCNC(=O)CCc1nc[nH]n1)CCNC(=O)C=Cc1nnc(C(C)C)o1 N1(C(c2cnc(Cl)s2)=O)CCC2(CCCN2C(C2CCC23CCCO3)=O)CC1 N1(C(C2(CC=C)CN(C(=O)CNC(=O)OCC)C2)=O)C2CCCC1CN(C)C2 c1(C(N(C)CCOCCN(C)C(C2CC(F)C(=O)N2)=O)=O)cc(N)ccc1Cl c1(C(=O)NC(C)CCCNC(=O)C(F)=C2CCC2)ccc(C(F)F)cc1Cl c1(C(=O)NCC2(CSC)CCC2)cn(C2CCN(C)C2)nn1 N1(C(CNC(=O)Nc2ccco2)=O)CC2CCC(NC(=O)C3=CCOC3)(C2)C1 S(=O)(=O)(c1cccnc1NCc1cn(C)c(=O)n1C)N1CCCC(CC)CC1 N1(C(c2ccn(CC)n2)=O)CCC(C2(O)CN(C(=O)C3=C(C)CC3)C2)CC1 N1(C(C(C(=O)OC)C)=O)CCC2(CCCN(C(=O)Cc3ccnc(F)c3F)C2)C1 CC(O)(CNC(=O)CSC1CCCO1)CNC(C1CCCC1)=O CCCCC(CNC(c1oc(Br)cc1C)=O)NC(=O)C(C)Cn1cccn1 c1(C(N2CC(CNC(C(COCC)(C)C)=O)OCC2)=O)cnc2n1CCOC2 C1(CC(N2CCCC2CNC(c2n(CC)ccc2)=O)=O)CCCC(OC)C1 c1(C(=O)NCC(CNC(c2c(C)n(CCC#N)nc2)=O)(C)C)cc(O)nc(O)n1 C1(NC(C2(CCNC(c3c(C)nc(C)[nH]3)=O)CC2)=O)CC(C)CC(C)(C)C1 N1(C(c2c(C(C)C)ocn2)=O)C(C(=O)NCCNC(=O)C(C)C)C2CC(O)C1C2 Cc1c(C(=O)NCC2CCCCN2C(C2CC(O)C2)=O)[nH]c2c1CCCC2 C(N=c1cccc(NC(=O)C(F)(F)F)[nH]1)c1ncn(C(C)(C)C)n1 N1(C(c2nc(C(CC)NC(c3coc(C)n3)=O)oc2)=O)CCCC(F)(C(N)=O)C1 N1(C(c2nn(CC)nc2Br)=O)CC2(CCCC2NC(C2CC2C(C)C)=O)C1 N1(C(C2(C)CCN(C(c3cccc(C=C)c3)=O)C2)=O)Cc2ccnn2CC1C N1(C(C(C)(C)C2CC2)=O)CC2(C=C(C(=O)NCC3CC3Cl)CO2)C1 C1(CNC(=O)CSCC(N2CC(F)C2)=O)CCCC(F)C1 N1(C(c2nccc(CNC(CCCC3C(C)C3)=O)c2)=O)CC2C(C1)C2(C)C c12ccc3c(c1)C(C(=O)N2)CCC3.c1(-c2cn(C(C)C)nn2)cnc(C)n1C C(CNC(=O)Cc1ccn(C)c1)(CC(=O)Nc1ccc(SC)nc1)OC c1(CCC(=O)NCCN(CCOC)C(C2COCC(C)O2)=O)ccc(C)cc1C CC1CC(C)CN(C(C)(C)COC(c2cnoc2C2CC2)=O)C1 c1(SC)ncc(Br)c(N(C(=O)Cc2ccc(Cl)cc2F)CC2CCCNC2)n1 c1(C(N2CC(CC(=O)NC(C=C)C)OCC2)=O)ccc(OC)cc1O N1(C(Cc2n(C)cnc2)=O)CCC2(CC(C(=O)NOCC3C=NNC3=O)C2)C1 c1(C(=O)NC2CCN(C(c3c(C)c(Cl)ccc3)=O)C(C)C2)cc2cnccc2[nH]1 c1(C(=O)NC(C2CCCC2)CNC(=O)CCOC2CCC2)ncoc1C1CCCO1 N1(C(C2(C)C=CCC2)=O)CCC(CN=c2[nH]nco2)C(F)(F)CC1 CC(C)C(F)(F)CC(=O)NC1CCN(C(c2cn(Cc3ccccn3)nn2)=O)C1 c1(C(N2CC3C(NC(C(CC(C)C)F)=O)C3C2)=O)cccc2nccnc12 C1(CCC)CN(C(c2ccc(CC)cc2)=O)CCN1C(=O)C(CC#N)n1ccnc1 CC1CCN(C(=O)CCC2CC2)C(CNC(c2ccc(C(C)(C)C)o2)=O)C1 N1(C(C(CC)OC)=O)CCC2(CCCN(C(=O)CNC(C3CCC3)=O)C2)CC1 c1(OCCC(=O)NCc2nc(-c3cccc(F)c3)no2)ccc(Br)cc1 c1(C(=O)NCC2(NC(C3CC4CC4C3)=O)CC2)ccc(CO)o1 C1(C(=O)NC(C)C(CO)NC(=O)Cc2ccsc2C)(CC)CC(C)(C)C1 C1(C(=O)NC2(CNC(=O)COC3CCC3)CCC2)CC(F)C(=O)N1 CCC(CCC(=O)NCc1cccc(C)c1C)NC(=O)C(C)(COC)OC Cc1cnc(C(=O)NC2CCCCC2C(N2CCC2C2CCC2)=O)c(F)c1 Cc1ccc(C)c(C(N2CCC(CNC(C3(C)CCC(=O)NC3)=O)C2(C)C)=O)c1 c1(OC)c(C)cc(CN2CCC3(CC3C(=O)Nc3nc(Br)ccc3C)C2)cc1C N1(C(Cc2c(OC)nccc2)=O)CC(NC(=O)C=Cc2cscn2)C(C2CC2)C1 c1(C(N(C=O)CC2CN(C)C2)C2CC2)ccc(F)cc1 C1(N(C(=O)CCn2cccn2)CC)CCCN(C(c2ncccc2C)=O)C1 C=CC(CCC)CC(=O)N1CCC(NC(c2ccccc2N2CCCC2=O)=O)C1 C#Cc1ccc(C(N2CCCC(CC)(NC(=O)CCNC(=O)C=CCl)C2)=O)nc1 N(C1c2ccccc2CC1C)C(N1CCCC(COC)C1)=O C1(CC)CN(C(=O)CC23CCC(CC2)CC3)CCC1NC(c1cscn1)=O CCCC(O)C(C(=O)O)NCC1CC(CC(C)(C)C)C1 N1(C(CNC(c2c(C(C)C)onc2)=O)C)CCN(C(=O)CC2(O)CCOC2)CC1 C1(NC(c2cnc(C)nc2)=O)CCN(C(c2cccc(N(C)C)c2)=O)C(C)C1 N1(C(C=Cc2c(N)cccc2)=O)CCC2(CCN(c3nnnn3C3CCC3)C2)C1 C=CCC(CC(C)C)C(=O)N1CCCC1CN(C)C(c1n[nH]cc1CC)=O C1(C(=O)NC23C(CN(C(C=C(C)C)=O)C2)C3)CCC(F)(F)CC1 N1(C(c2c(C(C)C)[nH]cc2)=O)CCCCC1C1(NC(C2CCN(C)C2=O)=O)CC1 C(=O)(C(C)(CNC(c1n[nH]cc1C#C)=O)CC)N1C(C#C)CCC1 Cn1ncc(C(=O)NC2CN(C(=O)Cc3cccnc3O)C3CC23)c1Cl N1(C(CCS(C)(=O)=O)=O)CC2CCC(C1)N2C(c1ccc(F)cc1Br)=O n1(CCN(C(C(F)=C(C)C)=O)C)cc(CC(C(=O)N(C)C)C2CC2)nn1 c1(C(N(C2CCCC(NC(Cc3c(C)scc3)=O)C2)C)=O)ccc(N)c(F)c1 C1(CNC(c2cccc(OC(F)F)c2)=O)CC2CC2N1C(=O)C=Cc1ccco1 N1(c2nccc(C(=O)OCC)n2)CCS(=O)(=O)C(CCNC(=O)CSCC)C1 c1(C(=O)NC(C2N(C(C(=O)NC(C)C)=O)CCC2)C)ccnc2c1nnn2C CCC(CNC(c1sc(NC2CC2)nc1C)=O)(CC)NC(C1CC=CCO1)=O N1(C(=O)C2=CCOCC2)CC2CCC(NC(C3CC4CCC(C3)S4)=O)CC2C1 c1(CC)c(C(N2CCCC(CCNC(=O)C(O)C(F)F)C2)=O)cccc1C c1(C(=O)NCC(CNC(CC=CC=C)=O)C)cc2cccnc2s1 C(=O)(C(CC=C)C(C)C)N1C(CN(C(c2nccc(C#C)c2)=O)C)CCC1 C1(C=O)C2CCC(F)(F)C12.N1(C(CCC2(OCC)CCC2)=O)CCC(C(C)N)C1 C1(CC(=O)NC(C)CCN(C(=O)CSc2ccccc2O)C)CC2(CCC2)CO1 Cc1n[nH]c(C)c1S(=O)(=O)N(C1(C#N)CCNC1)Cc1ncnc2c(Br)csc12 c1(C(=O)NC2CCC(C(N=c3cc(C)o[nH]3)=O)CC2)c(F)ccc([N+](=O)[O-])c1F N1(CC(=O)NC(C2CCN2C(=O)C=CSc2nc[nH]n2)C)CCCC1C(=O)NC c1(OC)ccc(C(=O)N(C(=O)CC2CCC(C(F)(F)F)N(C)C2)C2CC2)nc1Br c1(CC)cc(F)ccc1C(=O)NCC1CCCC1NC(=O)C1=C(Cl)CCC1 C(C(F)(C(=O)Nc1cc(C)c(F)cc1O)C(C)C)NC(C1(OC)CCOC1)=O c1(C(=O)NCC2CCC(NC(C3(CC)COC3)=O)C2)ccc(-c2ccsc2)cc1 C1(CC(=O)NC(CN(C(c2ncn(C)n2)=O)CC)C)CCc2ccccc2C1 C12CCN(CC1)C2=O.c1(CC(N2CCC(C(CC)=O)C2)=O)cccnc1 O=C(C1=CCOC1)NC1CN(C(c2cccc(-c3ccccc3)n2)=O)C2CC12 Cc1csc(=O)n1CCC(=O)NCC1CCC(NC(=O)CSC2CC2)C1 CC1=C(C(=O)NCC2CN(C(=O)C(C)CC3CCC3)C(C)(C)C2)CCO1 c1(N(C)CCN2CCCCC2)ccc(-c2cc(CN)[nH]n2)cc1 C1(NC(c2ccc(C(F)F)cc2)=O)CN(C(=O)Cc2sc(O)nc2O)C2CC12 CC(C)C(C)(CNC(c1cc[nH]c1)=O)NC(C1CC1F)=O C1(C(=O)NC2CCN(CC)C2)(CC)CCN(C(=O)C=CC2CCC2)CC1.CCF Cn1nc(Br)cc1C(=O)NCC1(C)CCCC1NC(C1CC1(C)C)=O C1(C)(C(NOCCCOC)=O)CC(O)CN1C(c1c[nH]nc1C1CC1)=O c1(C(N(C(C)CNC(=O)CCN2CCCCC2)C)=O)cc(N)cc2ccccc12 C1(NC(C#CC(C)(C)C)=O)CN(C(=O)CN(C2CCSC2)C)C2(CCC2)C1 C=CCCC(=O)NC(CC1CC1)C(=O)NCC(=O)NC(C)C c1(CC(=O)NC2C(C)(CNC(CNS(NC)(=O)=O)=O)CCC2)c[nH]c(=N)nc1O C1(NC(C=C(C)C(F)F)=O)CCN(C(=O)C=Cc2ccoc2)CCC1(F)F N1(C(C(CCC)CCC)=O)CCc2sc(CNC(=O)COCC(=O)OC)nc2C1 N1(C(=O)OC(C)(C)C)CCC(CN(CC(F)(F)C(=O)O)CC(=O)O)C(F)(F)CC1 N(C(=NCC1C(C)(C)C1(C)C)NCC1(C#N)CC1)C(c1cccs1)C c1(C(C(=O)NC(C)C)N(c2ccccc2C)C(C(C)SC)C)nc(Cl)ccc1Cl CCN=c1[nH]c(C)c(C(=O)NC2CN(C(=O)C(C)=CC)CC23CC3)s1 c1(CN=[N+]=[N-])c(N2CCS(=O)(=O)CC2C2CC2)nc2n1CCCC2 C=CC(C)(CCOC)C(=O)N1CC(C(C(N)=O)NC(c2ccc3nccn3c2)=O)C1 c1(C(=O)NCCC(C)NC(c2cc[nH]c2-c2ccccc2)=O)ccc(F)cc1Cl C(=O)(CC1=CSC2=NCCN12)NCC1COCCN(C(C(CC)CO)=O)C1 N1(C(c2[nH]ccc(=N)n2)=O)CCN(C(=O)C2=CCC2)C2CCCCC2C1 C(=O)(CCCCCC(C)(C)C)N1CC(C)CN(C(COc2cc(C)on2)=O)CC1C N1(C(C(CC(N)=O)O)=O)CC2CN(C(c3cc(O)nc(O)n3)=O)CC2C1 N(C1CCCn2cnnc21)C(=O)CC1CCN(C(C2CC3CCCC3C2)=O)CC1 c1(NCC(CC)C)ccc(S(=O)(=O)N2CCOCC2CC2CC2)cc1Cl C=CCCCCCCNC(C1(NC(C2C(C)(C)C2(F)F)=O)CCC(C)(C)C1)=O C(CCCC(=O)NC(C)CCF)NC(C(C)C1CCOC1)=O C(=O)(CC(C(F)(F)F)NC(c1ccc(F)c(C2CC2)c1)=O)OC C1(COC)(NC(=O)CCc2cnn(C)n2)CN(C(=O)Cc2ccc(C)o2)C1 c1(C(=O)NC(CC)CN(C(=O)CNS(=O)(=O)N(C)C)CC)ccc2cnnn2c1 C1(CNC(c2cc(C)ncn2)=O)N(C(=O)CN2CCCC2C)CCC1(C)C N1(C(C(c2ccccc2)OC)=O)CCC(C2CC(NC(c3cc(C)c[nH]3)=O)C2)C1 C12(C(=O)NCC3CCN(C(CC(OCC)OCC)=O)C3)CCCCC1NC(=O)C2 C1(C(=O)NCCCC(C)NC(c2c(C)ccs2)=O)COCCN1CC(F)F c1(OC)cc(C(F)(F)F)c2cc(C(N3CC(P(C)(C)=O)C3)=O)[nH]c2c1 Cc1cccc2cc(C(=O)NCC3CN(c4cncc(Cl)n4)CCO3)[nH]c12 N1(C(C2(CC#C)CC=CCC2)=O)CCN(C(c2ncc(Cl)n2C)=O)C2(CCC2)C1 N1(C(C(N2C(CC)CCC2)=O)=O)CCC(C)(NC(C2CCCS(=O)(=O)C2)=O)CC1 O=C(Cc1csc2ccccc12)NNC(=O)N=c1cc2n([nH]1)CCCC2 CCC(O)C(C)C(=O)NCC1(O)CCN(C(c2cnc(C(C)=O)s2)=O)C1 N1(C(c2c(OC)ccs2)=O)CC(C(=O)NC2(C)CCC(=O)N(C)C2)C2(CCC2)C1 C(N=c1[nH]c(N2CCC3C(C2)C3(F)F)nc(=N)[nH]1)c1cc(C(C)C)no1 N1(C(c2ncccc2Cl)=O)CCC2C(C1)CN2C(=O)CCSCc1ccccn1 C(C(O)CCNC(c1coc(Br)n1)=O)NC(c1cc(CO)[nH]n1)=O c1(OC)cnc(Cl)cc1C(=O)NC1CC(C)CN(C(c2cc(C)nc(C)n2)=O)C1 C(CC(C(=O)NCC1(C(C)(F)F)CC1)NC(C12CC(F)(C1)C2)=O)N(C)C c1(C(N2C3(CN(C(c4cc(OC)c(I)cc4)=O)C3)CC2)=O)ccc2c(c1)OCC2 c1(C(N2CC3(CCN3C(c3ccc(C4CC4)c(F)c3)=O)C2)=O)cnc(O)cc1O C(C)(C)(C(C)CC(=O)N1CCC(C2CC2)CC1)NC(C1CN(CC)C(=O)C1)=O CC(=O)CCCCC(=O)N1CC2(CCCC2NC(c2sc(C)cc2C)=O)C1 N1(C(C(CCOCC)NC(C2C=CCC2)=O)=O)CC2(CC=CC2)C1 C1(CNC(C2C(CC)C2)=O)C(C)CCN1C(=O)CCN1CCNC(=O)C1 Nc1cccnc1C(=O)NC(CC1CCCC1)C(N1CCCC(F)C1)=O c1(N(CCC(C)N)C(=O)NCc2c(Br)nnn2C)ccc(F)cc1 C(=O)(C(F)(F)CO)N1CC(CC(C)NC(c2cnc(-c3ncccn3)s2)=O)C1 CCCS(=O)(=O)C(C)C(=O)N1CCCCC1CNC(=O)C(C)c1ccco1 C(=O)(CCCC(=O)NC(C)C)N(C1(C)CC(NC(=O)CC(O)CC)C1)CCC C(C(CNC1(c2nnnn2CCN2CCOCC2)CCOC1)C(C)C)OC C12(CNC(CCC)=O)COCCN1C(=O)CN(C(c1cccc(CO)c1C)=O)C2 C(=O)(C(Cc1cccnn1)OC(c1ccsn1)=O)OC C(=O)(CC(C)(O)CCC)N(C1CCN(C(=O)C(CC)N(C(N)=O)CC)C1)CC#C c1(NC(N(CC)Cc2c(F)cccc2F)=O)ccc(OC)c2c1OCC2=O C1(NC(C2(C=C)CCC2)=O)CCN(C(=O)C(C)=CC(C)(C)C)O1 N1(C(=O)CCC2CCCO2)CCC2CCC(C1)N2Cc1cccc(F)c1F N1(C(COC(CC(C)c2cccnc2)=O)=O)CC(O)C(O)C1 Cc1n[nH]cc1CCNC(C1(NC(c2csnn2)=O)CC1(C)C)=O c1(N(C)CC2CC2)nc(N2CCS(=O)C3(CCC3)C2)nc2c1CCCCCC2 C1(C(=O)NC(C2CCCN2C)C)CC2CC2N1C(C1CCN(C)CC1)=O C12(C(=O)NC(C)C(CO)NC(=O)C(C)OC3CCCCC3)CCC(CC1)CC2 c1(CC)c(C(=O)NC2CCCC2CNC(=O)C(C)C(C)(C)C)cccc1F Cc1nc(NC2CCN(C(=O)CC3CC4CCC(C3)N4C)C2)c2c(C)csc2n1 N1(C(C(CC=C)NC(C)=O)=O)CCC2(CC1)CC2C(=O)N(CCCF)C N1(C(C2(C)CN(C)C(=O)C2)=O)CCN(C(C2CC(F)(F)C2)=O)CC12CC2 C=CCC(C(=O)NCCNC(=O)CCOCC1CCCO1)c1ccccc1.COC CCC(C)(C)C(O)C(=O)NCC(CC1CC1)C(=O)N1CC(C(F)(F)F)C1 C1(C(=O)NCC(C)NC(=O)C(c2cccnc2)C)CCC2CC2CC1 c1(C(=O)NCCC2(N3CCCC3)CCC2)ccnn1CC1CC1.C12(CC1)C(=O)N2 C(C(COC)C(=O)NCC(c1ccc(C)cc1)NC(c1sc(F)cc1Cl)=O)OC N1(C(C2(COC)CCOC2)=O)CCC2C(C1)CN2C(c1cccc2scnc12)=O C1(NC(C=C(C)C(F)F)=O)CN(C(c2ccc(C3CC3)c(F)c2)=O)CCC1C C1(NC(c2ccc(CNC(=O)C=Cc3ccsc3)s2)=O)CC2C=CC1CC2 Cc1ccc2occ(C(=O)NCC34CC3CN(C(c3ccc(Cl)cc3)=O)C4)c2c1 CN1CC(O)CC1(C)C(N1CCCC(NC(c2cc(O)ccc2F)=O)CC1)=O C1(N(C(C(COC)C)=O)C)CN(C(C2(O)CCC2)=O)CC1F C1(CNC(Cc2c(C)cccc2C)=O)CC2CC(C1)N(C(=O)CC1CC(F)(F)C1)C2 N1(C(c2ccn(CCF)n2)C(=O)NCCCOC)CCN2C(CNS2(=O)=O)C1 c1(NCC2OCC(CNC(c3cc(C)c(CSC)o3)=O)C2)cnc(C#N)cn1 C1(C(C)=O)CC(C(=O)NC2CC(NC(=O)C(C)(C)c3cccs3)C2)C1(C)C C1(O)(CN(C(COC)=O)C)CCCN(C(C2CCC(=O)N(C3CC3)C2)=O)C1 CCC(CCC(=O)Nc1cnn(C)c1C)NC(c1cnn(C)c1CC)=O c1(CC(N2C(CNC(=O)Cc3cnsc3)CC(F)C2)=O)coc2ccc(F)cc12 N1(C(C2C(c3n(C)cnc3)C2)=O)CCC(F)(NC(c2cccc(Br)c2F)=O)CC1 N1(C(C2CC(N(C(=O)CC3(O)CCCC3)C)C2)=O)CCc2ccsc2C1 CC1CC2(CCN(C(=O)C3=COCCC3)CC2)CN1C(C1CCCC(C#N)C1)=O c1(OC)c(NC(C2C3CCC2(c2ccccn2)C3)=O)cccc1C(=O)O c1(CN2C(C(C(=O)OC)(C)C)CCCC2)cn2c(n1)CCCCC2 C1(SC)CCCC1n1cc(C2(C)CN(C(C3CCCN3C(C)C)=O)C2)nn1 C1(CN(C(C(C)n2cccc2)=O)C)CN(C(c2cc(C(N)=O)c[nH]2)=O)CCO1 C1(NC(C(CCCC)=O)=O)CN(C(c2cn(C(F)F)cn2)=O)C2(CCC2)C1 C1(NC(c2coc3c2COC3)=O)CC2CN(C(C3CN4CCN3CC4)=O)CC2C1 O=C(C1=C(c2ccc(F)cc2)CCOC1)NCC(CO)C(F)(F)F C1(C(=O)OC)CCC(C)(C(=O)NCC2CCCN2C(C2(C)C=CCC2)=O)C1(C)C c1(C(=O)NCC(c2ccccc2)NC(CSC(=N)N)=O)[nH]cc2c1CCCC2 CN1N=C(C(=O)NC2CC(NC(c3c[nH]nc3Br)=O)C23CCC3)CCC1=O CC1(CC(=O)O)CCN(CCNC(C2(c3ccccc3)CCC2)=O)C1 C(C)(CCC(=O)N1CCOC(CNC(c2cn(CCC(C)C)nn2)=O)C1)OC N1(C(C(C)n2ccnc2)=O)c2ccccc2CC1CN c1(C(C)C)cc(O)nc(SCC(=O)NCCc2ccc(N3CCOCC3)nc2)n1 c1(OC)ccc(C(=O)NC(C)CC2CCN(C(c3cccs3)=O)CC2)c(C)n1 N1(C(c2nc(C)oc2)=O)CCC(NC(=O)C(c2cnn(C)c2)=O)CC1C c1(OCCC(=O)NCCN(CCC)C(C2CCN(C)C2)=O)ccccc1C(C)C c1(C(=O)NCCC2CCN(C(c3cc(C(=O)OCC)n[nH]3)=O)C2)cncc(C)n1 C1(C(N2C(CNC(CCN(C)CCO)=O)CCCCC2)=O)CCc2nccn2C1 C1(NCCC2(C)N=N2)CN(C(=O)OC(C)(C)C)CC12CCC2 CN1CC=C(CC(=O)N2CCC(C)(C(=O)NCC(c3cccnc3)O)CC2)CC1 C12(C(=O)OC)CCN(C)CC1CN(c1nnc(C(C)(C)O)n1CC(C)C)C2 N1(c2snc(CCC)n2)CCC(C)C(NC(=O)C(C)(c2ccccc2)OC)C1 Cc1csc(C=CC(=O)NC23CC2CN(C(C2(c4ncco4)CC2)=O)C3)n1 N(C1CCOc2ccc(O)cc21)C(C(c1ccccc1-c1ccccc1)OC)=O c1(CC(C)=O)cccc(C(=O)NC(C)CN(C)C(c2nnc(C)o2)=O)c1 C(=O)(C1CCCc2ncnn21)NC1(C)CCCN(C(CCC#C)=O)C1 c1(C2(NC(C(Cc3ccc(OCC)cc3)C)=O)CCC2)cc2ccccc2o1 CCCC(C#N)C(=O)N1CC(NC(c2cc(-c3cnn(C)c3)on2)=O)CC1(C)C N1(C(COCC#C)=O)CC(NC(=O)C(CC#C)C2CC2)C(O)C1 N1(C(C=CCOC)=O)CC2CCC1C(CNC(=O)C(F)CC1CC1)C2 N1(C(CC2(CNC(Cc3nc(C)sc3)=O)CC2)=O)CCc2cc(F)c(F)cc2C1 c1(OC)ccc(C(=O)NCC2CC(OC)CN2C(C2CNC(=O)N2C)=O)cc1F c1(CN(C(=O)NCC(=O)OCc2ncc[nH]2)CC2CCOC2)ccc(Cl)cc1 CC1(C)CCC(C(=O)NC2(C(=O)Nc3cc(F)ccc3O)CCSC2)CO1 N1CCCC12CCN(C(C1N(C)CCC1)=O)C2.c1(C2(CC)CC2)cc(O)cc(Cl)c1 N1(C(CC(C)(C)NC(=O)CCN=[N+]=[N-])=O)CCC12CCC(O)CC2 Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(=O)CC=C(Cl)Cl)C(C)C1 C(C)(c1ccccc1C)=CC(N1CC(CC)C(NC(C2CC(C)=NO2)=O)C1)=O CC1(C)COC(CCNC(C2(NC(=O)C(F)F)CCCC2)=O)C1 C(=O)(C(COC)CC)N1CCC(CN(C(c2c(CCC)nco2)=O)C)C1 Cc1cccnc1C=CC(=O)NCCN1CCN(C(C2(C)C=CCCC2)=O)CC1 N1(C(CNC(c2n(CC)ncc2)=O)C(F)F)CCN(C(=O)CC2CCOC2)CC1 c1(OC)cc(N2CC3CC(NC(c4csnn4)=O)CC2C3)ccc1[N+](=O)[O-] C1(C(=O)NC2CCC23CN(C(c2cc(Cl)c[nH]2)=O)C3)CCc2nccn2C1 C1(COC)CN(C(c2ccnn2-c2ccccc2)=O)CCN1C(C1CC1(F)F)=O CC(O)C(C)(C)C(=O)NC1CN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 NS(=O)(=O)c1n[nH]cc1C(N1CCC12CN(C(c1ccnc(Cl)c1O)=O)C2)=O C1(O)(CNC(=O)NCCN2CC(C)OCC2)CCC(C)(C)C1 N1(C(c2cccc(C(=O)OC)n2)=O)CC2(CCC(CNC(C3CC3CF)=O)O2)C1 C(c1cncc(F)c1)=CC(=O)NC1CC(NC(c2cccc(Br)c2)=O)C1 C(C)(C)(CC(=O)NC12CCN(CC1)C2)NC(C(C)c1cccs1)=O N(C(=NCCN1CCN(C)CC1)NCC1CC1)C(c1ccc(N(C)C)cc1)C c1(C(=O)NCC(C)N(C(C(C)OCC#C)=O)CC)cnc(CCC(F)(F)F)s1 C(=O)(CCC(=O)N1CCC(F)(CNC(C2CCC(C)(C)O2)=O)C1)NC N1(C(C2C3CN(C(C(C)Sc4cccc(C)c4)=O)C2C3)=O)CCCC2(COC2)C1 N1(C(C(CCSC)O)=O)CCN(C(=O)C=Cc2ccc(F)cc2)CC1CC(F)F C1(CNC(C=CCC)=O)CCCC(OC(=O)C=Cc2ccncc2)C1 C(=O)(CCC(C)(C)C)N1C(CN(C(C2CCCN(C(CC)=O)C2)=O)CC)CCC1 N1(C(C2CCC(C(C)(C)C)CC2)=O)CC2CCC(NC(=O)C=C3CCC3)CC2C1 C12(C(N(CCCNC(=O)CC3C=CCCC3)C)=O)CCC(CC1)C2 c1(C(N(C(C(=O)NCC2N(C)CCOC2)CC(F)F)C)=O)cc(C#N)ccc1N c1(OC)nscc1C(=O)NC1CC(O)C1CC(=O)NCC1CCC(C2CC2)O1 C1(NC(c2cn(CC=C)nn2)=O)CCN(C(=O)Cc2c(Cl)cccc2Cl)C(C)C1 CCC(CC)(CCC(=O)OC1CCCC(S(C)(=O)=O)C1)[N+](=O)[O-] C(=O)(C(O)C(F)(F)F)NCC(C)(C)CNC(=O)CC1(n2cccn2)CCC1 c1(C(N2C(CCNC(CC#C)=O)CCCC2)=O)ccc(NS(C)(=O)=O)cc1Cl c1(COC)nc(C)c(C(N2CC(C)(NC(=O)C(C)NC(=O)COC)C2)=O)s1 N1(C(C(C2CC2)OC)=O)CC(C2CN(C(c3ncc(Cl)cc3Cl)=O)C2)C1 CCC(C)(CNC(=O)C(F)(F)C1CCCC1)NC(c1cccnc1)=O C1(C(=O)NCC=C2CCN(C(c3c(C)ccnn3)=O)CC2)CCC2(C1)CC2(F)F Cc1ccnc(CNC(=O)N(C)Cc2nnn(C(C)C)n2)n1 CC1(C)CCOC1C(=O)NCCC1(C)CCN(C(c2cccc[n+]2[O-])=O)C1 CCCCC(CC)C(=O)N1CCN(C(c2cc3n(n2)CCOC3)=O)CC1CCC O=C1COc2cc(F)c(C(N3CCC(NC(C4CNC(=O)N4)=O)C3)=O)cc2N1 C1(C(=O)NCC(C)NC(=O)C(=O)NCC(F)(F)F)CCCN1C1CCCC1 C1(CNC(c2ccc(C)cn2)=O)COCCN(C(=O)CC2(C)CCCO2)C1 c1(OC(C(=O)NCCN(C(=O)C(C)(O)CC)CCC)C)ccc(F)c(F)c1 c1(C(=O)NCC2CCN(C(C(n3c(C)ccn3)C)=O)C2)nnc(Cl)cc1N c1(C(N2C(CNC(=O)C3=CCCC3)CC3(CC3)C2)=O)cnc2[nH]ccnc1-2 O=[N+]([O-])c1cnn(CCN2CCOC(c3cn(CC(O)CO)nn3)C2)c1 c1(-c2nc(C)c(F)cc2)n[nH]c2c1CN(C(c1c(F)cc(O)cc1F)=O)CC2 c1(OC)ccc2ncc(C(=O)NC3CN(C(=O)CN(C)S(N)(=O)=O)CC3F)n2n1 N1(C(CCC2CC(OC)C2)=O)CC(C2CN(C(=O)C(C(C)(C)C)NC(N)=O)C2)C1 c1(C(=O)NN(CC=CC(=O)NC(C23CCC(CC2)C3)C)C)ccnc(C2CC2)c1 Cc1cc(-c2cn(CCCC(=O)NC3CCCOC3(C)C)nn2)c(C)cc1Cl CCC(C)(COC)CNC(=O)C(c1cn(C)nn1)NC(=O)C(C)=CC1CC1 C(=O)(C1CCc2cccnc21)N1CCCCC(N(C)C(c2csc(CO)n2)=O)C1 C1(C(=O)NC(C)(CNC(=O)CC2C=CCC2)C2CC2)CC2(C1)CC(F)(F)C2 N1(C(c2nnn(CC)c2C)=O)CCN(C(c2csc(Cl)n2)=O)CC1CC(C)(C)C C1(C)(C(=O)NCCCNC(c2c(OCC(C)C)nccc2)=O)CCCC1(F)F C(=O)(C(C)Cc1ccncc1)NCC(C1CCCCC1)NC(CC=CCC)=O CC1CCC(C(N)=O)CN1C(C1(C)CCCN1C(=O)CC1(C)CCC1)=O CCCC(C)CC(=O)N(CC(=O)NCC(C)OC)CCn1cc(C)cn1 c1(C(=O)NC2CC(F)(CNC(CC(C)C)=O)C2)cnn2c(=O)cc[nH]c12 C(C(C(C)(C)C)NC(=O)Cn1ccc(C(F)F)n1)NC(C1(C)C(C)C1)=O C(C)(C)(CCCNC(=O)C(C)(C)F)NC(C1C(C(=O)OC)COC1)=O C1(CNC(C(n2ccc(C)n2)C)=O)CC2(CCC2)CN1C(=O)OC(C)(C)C N1(C(C=C(C)C(C)(C)C)=O)CCC(O)(CNC(=O)CCc2ccnc(Cl)c2)C1 C1(NC(=O)C=C2CC2)CC12CCN(C(=O)Cc1ccc(F)cn1)CC2 c1(CC2CCCN(CCCl)C2)cccc2ncnn12.C12(CC1(F)F)C(=O)N2 c1(CC)ccoc1C(=O)NC(CNC(C1CC1(F)F)=O)C(C)C c1(COC(C2C(NCc3cccc(SC)c3)C2)=O)ccc(OC(F)F)cc1Cl C1(C(=O)NCc2cccnc2F)CCC2(CC2)N1C(c1csc(Cl)c1)=O CC1(C)CN(C(=O)COCC2CC2)C(CNC(c2coc(Cl)c2)=O)CO1 N1(C(c2c(C)[nH]cc2)=O)CCC(C)CC1C(=O)NC(C1(CO)CC1)C N1(C(C(C)(C)SC)=O)CCCC(F)(CNC(c2cc(C)c(O)nn2)=O)C1 C#CC1(C(=O)NCCCC(O)CO)CCN(C(=O)C(C)CSC)C1 C1(COC)CC2(CCN2C(=O)CC(CNC(C2CN(C3CCC3)C2)=O)C2CCC2)C1 N1(C(C(C)OCCOC)=O)CC(C2CN(C(c3sc(F)cc3Cl)=O)C2)C1 C1(NC(Cc2cn(C)nc2)=O)CCN(C(=O)CN2C(=O)CNC2=O)CC12CCC2 C1(C#N)(C(=O)NCCN(C(c2c(N(C(C)=O)C)cccc2)=O)C)CCCOC1 N1(C(C(C)=C(C)C)=O)CCCCC1CC(=O)NCc1nn[nH]n1 c1(C(N2CC(C(=O)Nc3ccc(CC#N)cc3)C2)=O)cc(Cl)cc(Cl)n1 C1(NC(c2cc(C(C)=O)sc2)=O)CC(C(=O)N(C2CCOC2)CCF)C(O)C1 c1(CC(=O)NC(C)CCCNC(c2c[nH]cc2Br)=O)noc2ccc(F)cc12 c1(C(N(C2CCN(C(c3cc(C(N)=O)no3)=O)CC2)C)=O)cc2cccnc2s1 N1(C(C(CCC)C)=O)CC2CC(NC(c3cccn(C)c3=O)=O)CC1C2 C1(CC=C)(C(N2CCOCC2C)=O)CCCN1C(=O)C(O)C=CC C1(S(C)=O)(C(=O)OCC)CCN(C(C2CC(=O)N(c3cccc(C)c3)C2)=O)CC1 CC1(C(=O)NCC2(CCNC(c3cc(F)ccc3F)=O)CC2)CCC(=O)CC1 C(=O)(C1=CC2CCC(C1)C2)NCC#CC(N1CC(C)CN(C)CC1)=O c1(CC)ocnc1C(=O)N(C(C)C(=O)NCCCN1CCOCC1)C c1(CCN(C(C(=O)N(C)CC2CCCO2)=O)CC(F)F)cccc(F)c1 C(C(O)CN(C(=O)CCC1CCCO1)C)N(C)CC1CCOC1 C1(C2CC2)(C(=O)NC(c2cn(C)nc2)C(=O)NC2C3CCC(F)C23)CCC1 c1(C(=O)NC2(CF)CCN(C(=O)CCCC3CCCCC3)C2)n[nH]c2c1COC2 C1(CNC(CC2CC(CC)C2)=O)CC12CCN(C(=O)COc1cncc(C)n1)CC2 N1(C(c2c(C)nncc2)=O)CCC2CN(C(c3oc(Br)nc3C)=O)CC12 N1(C(COCC=C)=O)C2CCC1(CNC(=O)Cc1c(C)cccc1C)CC2 c1(C(=O)NCC(CCCC)NC(C2COCC2(C)C)=O)ccc2nccnc2n1 N1(C(C)C)CCCC1C(N1CCC1C(=O)NC1CCCC1F)=O c1(OCC(=O)N(CCCC(=O)NC(c2ccnn2C)CC)C)ccccc1C C1(CN(C)C)CC(O)CN1C(C1CCOCC1NC(c1cnn(CCO)c1)=O)=O C(C)(CCCC(C)C)NC(C=C1CCN(Cc2onc(C)n2)CC1)=O N1(C(c2c(C(=O)O)cn[nH]2)=O)CCC2CC1CN(Cc1ccccc1)C2 Cc1cc(CCC(N2CCCC(CNC(=O)C(C)(C)c3cncs3)C2)=O)n(C)n1 c1(C(=O)NC(C(C)C)C)occc1CNC(=O)CC1(C(=O)O)CCC1 C1(NC(C(C)CO)=O)CCN(C(=O)C(c2ccc(F)cc2F)(C)C)CCC1CO Cc1csc(C(=O)NCCC(O)CNC(c2ccccn2)=O)c1 C1(C(N(CCCCCCCC)C)=O)CN(C(=O)C(CCC)OCC)CC12CCC2 C(=O)(C1=NOC(C)C1C)N1CC(C(=O)Nc2cnn(CC)c2C)(CC)C1 CC1(C)CCN(C(=O)CP(C)(C)=O)CC1C(=O)NC1CCCSCC1 N1(C(C2C(C)CC(=O)NC2)=O)Cc2[nH]nc(C(=O)NCCCC3CC3)c2C1 N1(C(c2c(C(C)(C)C)ocn2)=O)CCOCC1CC(=O)NC1CC(CC2CC2)C1 CC1CC(NC(C2CCC(F)CC2)=O)CN1C(C1CC(=O)N(C)C1)=O C(=O)(C(CC1CCCC1)NC(=O)C(C)OCOC)NCCCC c1(CC(N2CC(C(N(c3csc(Cl)n3)C(C)(C)C)=O)C2)=O)ccccc1C(F)(F)F C1(CCNC(CSCCC)=O)CN(c2cc(C)nc(CO)n2)CCS1(=O)=O C(CCCCCC(=O)NCC1(C2CC2)CC1)NC(c1n(C)c(Cl)nc1)=O N1(C(C2C(C(C)(C)C)C2)=O)CC2(CNC(=O)CCCOC(F)F)CC1CO2 C1(CC(N)=O)CN(CC(=O)NC2CCNC(=O)C2)CCO1 c1(N2CCC(N(C)C(C3CCCN3C3CC3)=O)C2)ncnc2c(Br)nn(C)c12 C=CCC(C)(C)CC(=O)N1CCCC(C)(C)C1CNC(c1cc(=O)n(C)cn1)=O C(CC(C)C)(C(=O)NCC(C)C)N(C(COC)=O)C N1(C(c2scc(C)c2)=O)Cc2c([nH][nH]c2=NC(=O)c2ncccc2Br)C1(C)C N1(C(C2N(CC)CCCC2)=O)C(CC(=O)NCC2OCCC2C)C2CCCC12 N1(C(C(C)OCC)=O)CCC2(CCCC2NC(=O)Cc2csc(Cl)n2)CC1 n1(C(C)(C)C)ccc(C(=O)NCCC2CC2CNC(=O)CC2CCOCC2)c1 C1(NC(C2C3CCCC23)=O)CC2(CCN(C(c3cc(CO)ccc3O)=O)CC2)C1 CC1ON=C(C(=O)N2CCN(C(c3cnc(N)c(Br)c3)=O)CCC2C)C1C Cn1ncc(Cl)c1CC(=O)NC1CCC(F)(CNC(=O)Cn2nnc(=O)[nH]2)C1 C1(NC(C(C#C)(C)C)=O)CCN(C(=O)CCN(CC(F)(F)F)C)CC1(C)C Cc1ncc(Cl)c(C(=O)NC2CCC(NC(C3CC34CC4)=O)C2)n1 N1(CC(=O)N(CC#C)CCN)CCCC(NC(=O)OC(C)(C)C)C1.CO C#Cc1ccc(C)c(NC(C2CC(NC(=O)CCc3cncnc3)C2(C)C)=O)c1 CC(CCNC(=O)CCc1cccc(F)c1)CCNC(C1CC1(C)C(F)F)=O c1(N2CC(C)(C(F)F)OCC2)ccc(S(=O)(=O)NC(C)(CO)CCF)cc1C#N CC(C(C)(C)C)=CC(=O)NC(C1CCCN1C(=O)C(C)n1cccc1)C N1(C(c2ccn(CCC)n2)=O)CC2CCC(C1)N2C(c1cncc(C(F)F)c1)=O CCC(CC)CC(=O)N(C1CCC(NC(c2cnc(C(=O)OC)cn2)=O)CC1)C Cc1ccc(O)c(CC(=O)NCC2(NC(C3CC(C(F)(F)F)C3)=O)CCOC2)c1 CON=CC(=O)N1CCC(CCNC(=O)CCC2CC2(Cl)Cl)C1 c1(NC(C(C)N(C(COC(CC)C)=O)C2CC2)=O)cc(C)cc(Cl)c1 N1(C(COCc2c(C)cccc2)=O)CCC(NC(=O)CN=S(C)(C)=O)C(C)C1 Cc1cc(C)c(C(N2CC3(CCN3C(=O)C(C)C(O)C(C)C)C2)=O)cc1N C12(C(=O)NCCCC(c3ccccc3)NC(C(C)SC)=O)CCCC1C2(F)F C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CC2CCC1CN(C(C1CSCCS1)=O)C2 c1(C(Cc2nc(CC)sc2)=O)cc(C(=O)NCC2CC2)nn1C.C1=CCNC(=O)C1 C(CCC[Si](C)(C)C)N(C(=O)C(C)(C)n1cccn1)C.c1cccc(F)c1 C1(NC(=O)CSc2ccccn2)CC2CN(c3cncc(Cl)n3)CC12 C1(NC(C(C)C2CCC2)=O)CCCCN(C(=O)C(c2ccccc2)O)CC1 N1(C(C2CC(OC)(OC)C2)=O)CCC(CC(=O)NCC(F)(F)Cl)CC1 N1(CC(=O)NC(CNC(c2c(C)ncs2)=O)C(C)C)CCCCCCC1=O c1(C(=O)NCC2N(C(C(C)(C)C)=O)C3C(C2)C3)cnc2c(Cl)cccn12 Cn1nc2c(c1C(=O)NCC1C=CCN1C(=O)CC1CCOC1)CSCC2 c1(NCC(=C)Cl)cc(Br)ccc1S(=O)(=O)NC1CCOC(c2ccncc2)C1 c1(C(N2C(CC(=O)NCCC3=CCCCC3)CC(F)C2)=O)cnc2c(c1)COC2 c1(C(=O)NC2CCC(C)(CNC(C3(COC)CCC3)=O)C2)cccc2[nH]ncc12 C(=O)(CCCCN=[N+]=[N-])N1CC2C(CC(=O)NC(c3nc[nH]n3)CC)(CC2)C1 c1(OC)nccc(NC(=O)COCC2CC2)n1.C12CCCC(C1)NC1CC(C1)N2 C(F)(C(=O)N(CC(=O)N(CC(C)OCCOC)C)C)=C(C)C.CCO Cc1cccc(C(N2CCCC(NC(=O)CC3CN4CCN3CC4)CC2)=O)c1O N1(C(C2CCCCO2)C(=O)NCCCOC)CC(C)CSc2ccccc21 C1(CNC(C(c2c(C)cccc2)C)=O)CN(C(c2cc[n+]([O-])cc2)=O)CC1(C)C C1(C(=O)NC(C2CN(C(=O)CC(C)(C)O)C2)C)CCC2(CC1)CC2 c1(CCN(C(NNC(c2cncc(CC)c2)=O)=O)CC)cn(C)c2cc(F)ccc12 N1(C(CCC=C)=O)CCC(C)C1CNC(c1cnccc1OC)=O N1(C(=O)OC(C)(C)C)CC2(C1)CN(C(C1(Cc3ccc(C#N)cc3)CC1)=O)C2 C1(N(C(C2CCCCC2)C(=O)NC2CC2)C)CCCN(C(=O)CSC2CCC2)C1 c1(CC(=O)NCC2(C(N)=O)CN(C(=O)CCC=CBr)C2)ccccc1[N+](=O)[O-] C1(C(C)C)CC(NC(N2CCOCC2CC(c2ccccc2)O)=O)CCO1 c1(C(N2CCC(NC(C3CC(OC)C3)=O)C2)=O)cccc2c1COCC2 c1(CC(=O)NCC(C)N(C(=O)C(C)SC)CC)csc(C(C)OCC)n1 c1(C(N2CCC(C)(CNC(Cc3c(C)ocn3)=O)C2)=O)ccc(C(F)(F)F)nc1N N1(C(CC(=C)C)=O)CCC(CNC(c2sc(Cl)c(Cl)c2OC)=O)C12CCC2 C(CC(F)CN=[N+]=[N-])NC(C(CC=CC)NC(C1CCCCN1C)=O)=O C1(NC(C2N(C(=O)OC(C)(C)C)CC(C)OC2)=O)CCOCC12CCC2 C1(C)(CNC(CCCC=C)=O)CN(C(=O)C=Cc2cncs2)CCO1 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCCNC(c1sc2cc(C)sc2c1)=O C1(C(N2CCC(N(C(=O)CC3CC(C)(C)C3)CC)C2)=O)CC(=O)OC1(C)C N(C1CS(=O)(=O)c2ccccc21)Cc1nc(-c2ccc(SC)s2)sc1 C1(CNC(CCc2ccc(C)cc2)=O)N(C(=O)C2=CCCC2)CCC1(C)C C=CC1COCC1NC(c1ccoc1CNC(=O)C(CN(C)C)CC)=O C(C(C)(C)CC(=O)N1CCCC1(C)CNC(=O)CCC=C(C)C)OC C=C(C)CC(=O)N(CC(CC)NC(C1CCCC1)=O)C N1(C(C)C(=O)NC2CC2)CCCC(NC(c2ccc(C3CCCO3)[nH]2)=O)C1 N1(C(CC(C)(C)OC)=O)CC(C)N(C(=O)Cn2ccc(C(=O)OC)n2)CC1C C1(N(C(c2ccc(C)n2C)=O)C)CN(C(=O)C(F)(F)C2CCCC2)CC1(C)C CC(C(=O)NN1CCCC1C(=O)N=c1ccn(C)[nH]1)C1CCCC1 c1(COCC2C=CC(Nc3ccc(C(CF)OC(C)=O)cc3)C2)ccc(C)cc1 C1(C2CCN(C(=O)CC3CC=CC3)C2)(NC(c2c(Cl)ccc(OCC)n2)=O)CC1 C1(OCc2cn(CC(COC)O)nn2)CCCN(C(=O)COCC(=O)NC)C1 C1(C(=O)NC(CC)(C)CNC(=O)Cn2ncnn2)CNC(=O)C(C)(C)C1 n1(-c2ccc(C(=O)NC(C)C(c3ccccc3)C)s2)nnc2ccccc12 C(=O)(C1CCc2cccnc21)N(C)CC1(O)CN(C(C2CC(F)C2)=O)C1 CS(=O)c1cc(C(=O)NC2CC(F)(CNC(C3CCC(=O)O3)=O)C2)ccc1F C1(C(=O)NCC2(O)CN(C(C3CC4CCCC34)=O)C2)(COC)CCOCC1 Cc1cc(C(N2CCC(NC(=O)C=CC3CCC3)C2C(C)(C)C)=O)ncc1C#N N1(C(C(C)NC(=O)NC)=O)CCC(NC(C2(C)CC3CCC2C3)=O)C(F)C1 CC(C)(CC(=O)O)NC(=O)CC1CCCC1(C)C CC(C(=O)NCCCCC(C)NC(C1CCC2(CCC2)O1)=O)S(C)(=O)=O CN1CCN(C(C2COCCN(CC(O)CO)C2)=O)CC1c1nccn1C C(=O)(C(C)C(O)C(C)CC)N1CCCC(F)(CNC(CC(=O)NCC#C)=O)C1 C(=O)(C1CCCc2nc[nH]c21)NCC#CCNC(C1=NOC(C)C1)=O C1(NC(=O)C2=COCCO2)CCOC2(CCN(C(C34CCC(C3)C4)=O)CC2)C1 C(C(C)(O)CC(=O)N1CCN(CC(=O)Nc2c(C)cccc2O)CC1)OC c1(OCC(=O)NC2N(C(C(C(=O)OC)C)=O)C3C(C2)C3)ccc2c(c1)CCC2 N1(C(=O)C(N2CCOCC2)Cc2cccs2)CCCC1C=Cc1ccccc1 N1(C(CCC=CC)=O)CC2CC2(NC(=O)CSc2ccccc2Cl)C1 C=CCCC(C(=O)NCCCCC(C)(F)F)NC(=O)CCCN=[N+]=[N-] N1(C(c2csc(C)c2C)=O)CC(C)CCC1CNC(c1ccc(C(N)=O)s1)=O CC1(C)C2CC(C(N3CCCC3(C)Cc3ccccc3Cl)=O)CC12 C1(C(=O)NCCC2CCCCN2C(=O)CSCCC(C)C)(CC)CCC(O)CC1 c1(C(N2CCC(=CCNC(C(C)SCCCC)=O)CC2)=O)coc2c1CCCC2 N1(C(C(CC(CC)C)=O)=O)CCC2(CCCCC2NC(=O)C=C2CCC2)CC1 Clc1ccccc1C1CCN1Cc1c(CNc2nccc(N3CCCC3)n2)n[nH]c1 C1(NC(c2cn(C(C)C)nc2)=O)CCC12CCN(C(=O)CN1CC3CC3C1)CC2 c1(C(N2CCN(Cc3cccc(OC)c3)CC2)C(=O)NCCC)cccnc1C C1(C(=O)OC(C)(C)C)N(C(=O)OCC(N2CCCC2)=O)CCC1(C)C.CC1CO1 c1(C(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)c(Cl)sc2nnsc12 C(C(=O)NCC(F)CNC(=O)CNS(N)(=O)=O)(C(C)C)OCC Cc1noc(C)c1C(C)C(N1CCC(Cn2cc(C(C)CC3CC3)nn2)CC1)=O O=C1OC2CCN(C(=O)Nc3ccc(N4CCCCC4)c(Cl)c3)CC2O1 c1(NC(C(CCCOC)NC(C2OCCC2(C)C)=O)=O)cnc2ccnn2c1 C12(NC(=O)Cc3sc(O)nc3O)CCN(C(c3cc(Cl)sc3Cl)=O)CC1C2 CCCCC(=O)C(=O)NC1CCN(C(=O)C(C)(C)Oc2c(F)cccc2F)C1 CC1CN(C(c2ccoc2)=O)CCC1CNC(C1(CC#N)COC1)=O C(=O)(C(C)(C)N=[N+]=[N-])NCC(CC(=O)N(CC(C)(C)O)C)O c1(CC)cnc(C(=O)NC2(C(=O)NC3CC4(CCC4)C3)CC(F)C2)nc1 c1(NC(N2CCC(CC3CCNCC3)CC2)=O)cc(-c2cccc(F)c2)ccn1 C1(C(N(CC(COCC)O)C)=O)CN(C)CCN1C(c1cnc(O)c(C)c1)=O C1(C(=O)NC2(CC)CN(C(c3cnn(C)c3)=O)C2)CCCC(C(N)=O)CC1 C1(C(N(CCCC)CC(=O)NCC(C2CCCCC2)C)=O)Cc2nccn2C1 N1(C(CC2(C)OCCO2)=O)CC2CCC1C(NC(C1(F)CCOCC1)=O)C2 c1(C(=O)NCCN(C(C)C)C(C2CC3CCC2O3)=O)ccc(N2CCCC2)cc1 C(C(C(C)(C)C)NC(=O)C(C)(C)N(C)C)NC(c1ccc(C(C)=O)o1)=O N1(C(C=Cc2n(C)ncc2)=O)CCC2CN(C(c3nocc3Cl)=O)CCC2C1 c1(C(N2CC(C)C(NC(c3cccc4nonc34)=O)C2)=O)cc2ccncc2s1 c1(C(=O)NC2C(SC)CN(C(=O)C(C#N)C(C)C)C2)cc2cccc(N)c2cn1 N1(C(c2c(C)ccnc2)=O)CCN2CCN(C(c3ccsc3C(F)F)=O)CC2C1 c1(OCC)cccc(NC(C2CCCN(C(C)=O)C2)=O)c1 N1(C(C2(OCC)CCOC2)=O)CC2(C)CC1(C(N1CC3CC3C3CC13)=O)C2 C=C(Cl)CCC(=O)NC1C(C(N2CCCC2C(C)(C)CO)=O)C1(C)C N1(C(Cc2nc(CC)sc2)=O)CCOCC1CN(C)C(C1(C)CCCOC1)=O N1(C(c2ccc(C#C)o2)=O)CCC(NC(=O)C2=CCCCC2C)C(CO)CC1 C(=O)(C1=CCOCC1)N(CCN(C(c1cnc(C(C)C)nc1)=O)CC)CC N1(C(C(C=C)C)=O)CCN(C)C(C(N2CCC(C(C)O)CC2)=O)C1 N1(C(c2c(CC)noc2)=O)CCC(C)C1CNC(C1(NC(C)=O)CCC1)=O C(CC(C(=O)OC(F)(F)F)NC(=O)C=CC(=O)Nc1ccccc1F)SC C1(C(N2CCC(N(C(=O)Cc3cscn3)C)C2)=O)CCS(=O)(=O)N1 N1(OC(C)C)C(C)CN(C(c2cccc(C#N)c2)C(=O)N(C2COC2)C)CC1C c1(C(=O)NC2C(CNC(CCSC)=O)CC2)ccc(C2(F)CC2(F)F)cc1 CC1(C)C2CCC1(CC(=O)NC1CC=CC1)CC2.C1CCOCCNCC(=O)N1 c1(C(N2CC(CC(C)NC(CCOCCOC)=O)C2)=O)noc2cc(Cl)ccc12 CC1(C)CC2(CC(C(=O)NCC(F)CNC(C3CC4CCCC(C3)C4)=O)C2)C1 c1(CC)ccccc1C(=O)NC(C)C(C(C)C)NC(c1cnc(C)s1)=O C1(NC(c2cc(CC)on2)=O)CN(C(=O)OC(C)(C)C)CC(C)(C)C1 C(=O)(CC(O)CC(C)(C)C)NC1CCCN(C(C2(CCCC)CCC2)=O)C1 c1(CC(=O)NCC2CCCCC2NC(c2ccon2)=O)ccc(F)cc1C(F)F CC(CF)N=c1ccn2ncc(S(=O)(=O)N3CCOC(C)CC3)c2[nH]1 CS(=O)(=O)c1cccc(Cl)c1CNCC1CCC2(C1)CC2(F)F C(=O)(C(O)CC(F)(F)F)N1CC(O)(CCNC(C2N(C=O)CCC2)=O)C1 C1(O)(CCNC(C2(CCOC)CCC2)=O)CN(C(=O)C(C)C2CCC2)C1 N1(C(C2(C#N)C(C)C2)=O)CCN(C(=O)CC(=O)N(C)C)CC(C)(C)C1 c1(CNC2N(C)S(=O)(=O)CC2)ccc2c(c1O)CCCC2 c1(C(=O)NC2C(C)N(C(c3ccc(C(C)(C)C)nc3)=O)CC2)ccc(F)cc1F C1(C(C)C)CCCN(C(=NCc2cccc3c2OCCO3)NCC2CCCO2)C1 c1(C(=O)NC(CCN(C(CC(C=C)CC)=O)C)C)ccn2cc(C)nc2c1 Cn1ncc(C(N2CC(n3cc(-c4cccc(N(C)C)c4)nn3)C(O)C2)=O)c1C#N Cc1cccc(Cl)c1C(N1CC(NC(c2cnnc(O)c2)=O)C(F)C1)=O c1(C(N2CC(NC(C=C(CC)C)=O)CC2(C)C)=O)ccc(Br)c2c1OCCC2 c1(C(=O)NCCOCCNC(c2cc(C)on2)=O)nc(Cl)c(Cl)s1 C1(NC(CCOCCN(C)C(C2CCS(=O)CC2)=O)=O)CCCC(O)C1O C(CC(O)C(=O)NC(C1CCOC1)CO)NC(Cc1cnc(C)s1)=O C(N=C(NCc1cncs1)NC1CCOc2ccccc21)c1cc(C)c(Cl)cn1 c1(C(N2CCC(C(N3CCC(COC)C3)=O)(CF)C2)=O)cccn(C)c1=O c1(CC(=O)NC(C2CCN(C(=O)C(N)CC(N)=O)CC2)C)ccc(F)c(Br)c1 C1(C(c2ccc(Cl)cc2)NCCOCCCC)CCCC(C)CC1 N1(CCNC)CCC(N=c2[nH]c(N(C)CCc3c[nH]c(=N)s3)nc3c2COC3)C1.CS C(=O)(C#CC1CCOC1)N1CCC(CC(=O)NC(c2nncn2C)C)CC1 C(CC(=O)NC1(CC(C)C)CC1)OCCN(C(CSCC=C)=O)C C1(F)(C(=O)OCC(=O)Nc2n(C)cnn2)CCS(=O)(=O)C1 N1(C(c2c(C)nc(C)s2)=O)CC(C)CN(C(C2CC3C=CC2C3)=O)C(C)C1 CC1=C(COC(=O)C2=NNC(C(F)(F)F)C2)C(C)(C)CCC1 c1(C(N2CCC(=Cc3cccnc3)CC2)=O)ccc(Cl)c(C(F)(F)F)c1 c1(OC)ccc(NC(=O)C(C)CCOC)cc1OCC(F)(F)F N1(C(C(C(CC)C)O)=O)CCC2CN(C(c3cc(C(N)=O)co3)=O)CC2C1 CC1(C)CCN(C(C2CCOC2(C)C)=O)C1C(=O)NCc1ncc[nH]c1=O CCCN=C(NCc1cc(C)cc(Cl)c1)NC1CC(=O)N(c2ccccc2F)C1 CC(C)CC(C(=O)N(C1CCC1)C(C)C)ONC(C1(C)CCC(=O)C1)=O c1(C(=O)NCc2cccc(CNC(C(C)=CC)=O)c2)ccc2nc(Cl)nn2c1 N1(C(c2ncc(C3CC3)cn2)=O)CC2CC(C(N3CCCC3)=O)(C2)C1 N1(C(Cc2nnc(C)o2)=O)CC2CCC2(CNC(C2CC(C(C)C)=NO2)=O)C1 C1(n2cnnn2)(C(=O)NCC(CO)NC(=O)C(C2CCCCC2)O)CCOCC1 C(=O)(C(O)CC(F)(F)F)NCC1(OC)CCN(C(c2cc3ccncc3[nH]2)=O)C1 C1(NC(COCC#C)=O)CCN(C(c2cccnn2)=O)C1 C(=O)(C(CC(F)F)NC(c1coc(C(F)F)c1)=O)N(CC(COCC)C)C Cc1csc(C(N2CCCC(C(=O)Nc3cn(C)nc3C)C2)=O)c1C c1(C(=O)NC2CCN(c3cccc(C)c3)C2=O)cc(C)c(Br)c(C)c1 N1(C(C(C)NS(C)(=O)=O)=O)CCCC(NC(=O)CCC2(O)CCC2)C1C N1(C(C2(C)ON=C(C)C2)=O)CCCC2(C1)CN(C(=O)CC1OCCC1C)CCO2 N1(C(c2nc(C)[nH]n2)=O)CCC(C2CCN(C(=O)C=C3CCC(C)(C)CC3)C2)C1 N1(C(CCCC#C)=O)CCC2(CC1)CCN(C(=O)CN=c1cc[nH]cc1)C2 C1(CNC(CC=CC=C)=O)CN(C(=O)CC(c2ccc(F)c(F)c2)C)CCN1C c1(C(N2CC(C)C(NC(c3cc(C(C)C)ccc3N)=O)C2)=O)cn2c(n1)SCC2 c1(C(N2CC(C)(NC(=O)CC3(C)CCS(=O)(=O)N3)C2)=O)cc(Cl)c(F)cc1O C1(C(N(C)CC2CC2(C)C)=O)N(C(c2cnn[nH]2)=O)CCC1(C)C CC1CCn2cc(C(N3CCCC(F)(CNC(C4CC(O)C4)=O)CC3)=O)nc2C1 C#CCC(C(=O)NC1CC1C(F)(F)F)NC(=O)C=CC(C)C C1(CC(N2C3CN(C(c4n(C)ncc4)=O)C(C3)C2)=O)Cc2cccc(Cl)c2O1 C(C(=O)NCCCC1CCCN1C(=O)CCn1ccnc1)(C(C)C)OCC(C)C N1(C(C(CCC)C(C)C)=O)CCC2CCN(C(c3nn[nH]c3Cl)=O)CC12 c1(NC(C(C)S)=O)n[nH]c2c1CN(C(=O)CN1CCNC1=N)CC2 Cc1c(F)ccc(C(N2CCC3C(NC(=O)CCCCC(N)=O)C23)=O)c1C#N c1(NCC(CCCC)NC(C2CCN(C)C2=O)=O)nc(Cl)nc2[nH]cnc12 CCCC(C)C(=O)N(C1CC(NC(c2c(C(F)(F)F)noc2C)=O)C1)C Cc1ccc(NC(C2CN(C(=O)C(C)(C)C(C)O)C2)=O)cc1CO Cc1cc(C2CCC2)ccc1C(=O)NCC(C)N(C)C(C1CN2CCC1CC2)=O N1(CCN2C(c3ncc(-c4ccccc4)o3)CCC2)CCCC1(C)C1CCCCC1 C1(C(N2CC(C(C)NC(c3cc(Br)c[nH]3)=O)C2)=O)Cc2cncn2C(=O)N1 CCC(CC)CC(F)C(=O)N1CC(NC(c2cncnc2)=O)CC(F)C1 c1(NC(=O)NCc2cccc(OC)c2OC(F)F)c(Cl)cc([N+](=O)[O-])cc1Br C1(NC(C(CCSC)O)=O)CCN(C(c2cc(N)cc(O)n2)=O)C(C)C1 C(=O)(C(C)CC1CCCCC1)NCC(C)NC(c1coc(-c2ccccc2)n1)=O C1(C(=O)NCC2CC(NC(c3c(C)snn3)=O)C2)SC2C=CC1CC2 C1(N(C(C2CCN(C(C(CC=CCC)C)=O)CC2)=O)C2CC2)CCCN(C)C1=O Cc1cc(F)ccc1C(=O)CNC(=O)C(F)CC1CCOC1 CCC(C(=O)OC)C(=O)N1CSCC1C(=O)NC1(C)CCC(C)(C)C1 C12(CNC(c3c(C)noc3N)=O)CCCCC1N(C(=O)CN(C)CCO)CC2 N1(C(C(C)(CO)NC(C)=O)=O)C2CCC1C1CC1(NC(c1cc[n+]([O-])cc1)=O)C2 C(CCCC(CO)NC(=O)C(COC)CC)NC(CNS(NC)(=O)=O)=O c1(NC(c2n(C(C)C)ncc2)=O)ccc(NC(C2CC(O)CN2)=O)c(F)c1 c1(C(=O)NCC(CN(C)C(C2CCC(F)(F)C2)=O)O)cc2cccnc2nc1O CCC(C(=O)N1CCN(C)C(CNC(C2CNC(=O)O2)=O)C1)C(C)(C)CC C1(NC(c2cnc(C)s2)=O)CC(CNC(=O)C(C#N)C2CC2)C(O)C1 c1(CN2CCN(C(CC)C(=O)NC3CC3)CC2)c(Cl)nc2ccccn12 n1(CC(=O)NCC(=O)Nc2ccc(Br)cc2)cccnc1=O N1(C(CCCSC)=O)CCN(C(c2ncc(C(F)(F)F)s2)=O)C(CCO)C1 c1(C(=O)NC(CCOC)Cc2cccc(Br)c2)cc(C(F)(F)F)ccc1C(=O)O N1(C(C(CNC(=O)OCC)(C)C)=O)CC(C(=O)N(CC(=O)OC)C)CC(C)(C)C1 CCCCCC(C)(C)C(=O)NCCC1CN(C(=O)Cc2cc(F)ccc2Cl)C1 C1(NC(C2CC3(CC(=O)N3)C2)=O)CCCC12CCN(C(c1ccco1)=O)CC2 c1(-c2cn(C(c3ccc(OCC)cc3)CC=C)nn2)cc(F)cc(Cl)c1 C(=O)(CC(C)C(C)(C)NC(c1cccc(C)c1F)=O)NCc1ccc(C)nc1O N1(CC)Cc2ccc(NC(C3CCNC3c3ccccc3)=O)cc2C1 C12(NC(C3CN(C)C3)=O)CCC1CN(C(c1ccc(NCC(N)=O)cc1)=O)C2 C(=O)(C(CNC(=O)CC1OCCCO1)CC1CC1)NC(c1n[nH]c(CO)n1)C C1(C(=O)NC2C(SC)COC2)CCCCCCN1C(=O)CCCc1ncco1 C1(NC(=O)CNC(C2CCCCO2)=O)CN(C(C2OCCCO2)=O)C2(CCC2)C1 c1(CNC(C(N2CCCCCC2)C)=O)cc(O)nc(CNC(=O)CC2CC2C)n1 CCC(O)(C(=O)N1CC(CNC(=O)CC2(C)CC2(F)Cl)C1)c1ccccc1 CCCCC(CCCC)C(=O)NC1CC(CNC(=O)Cc2ccc(OC)cc2)C1 C1(N(C(c2occ(C)c2)=O)C)CCC(NC(C2CC2c2ccsc2)=O)CC1 C(=O)(CC(C)(C)C)NCC(=O)NCC(C)N(C)C(c1cnc(-c2cccs2)o1)=O c1(CC)ccc(C(=O)NC(CNC(c2cnn(C)c2C)=O)CC(C)C)c(Cl)c1 C(=O)(C(O)CCC(C)C)N1C(C(=O)NCCN(CCC)CC)CC(OC)C1 c1(OC)cnc(N(CCc2c[nH]c(=N)s2)CC2CN(C)CCO2)nc1C C1(C)(CC)CC(NC(=O)CCOC2COC2)CN1C(c1c[nH]cc(Cl)c1=O)=O C1(C(=O)NCC2C(C(C)(C)C)C2)(NC(=O)Cn2ccnc2)CCC1 Cc1c(Br)ccc(-c2noc(CSc3cccc(F)c3Br)n2)c1F O=S(=O)(c1ccc2[nH]c(=NCc3ccsc3)sc2c1)NCC1CSCCS1 O=C(CC1OCc2cc(Cl)ccc21)NC1CCN(C(C2CSC2)=O)CC1O Cc1ccc(SCC(=O)N(CC(O)CNC(=O)COC2CCC2)C)c(C)c1 C12(NC(c3n(C)c(S)nc3)=O)CCC(CC1)N(C(C1CCC3C(C1)C3(F)F)=O)C2 N1(Cc2c(C(=O)O)c3c(s2)cccc3)CC2CS(=O)(=O)CC(C1)C2(F)F S(=O)(=O)(c1c[nH]c(C(=O)NC2(C)CCN(C(=O)C(C)S(C)(=O)=O)C2)c1)NCC c1(C(N2CC(O)(CN(C(C(CC#C)CC#C)=O)C)C2)=O)n[nH]c2ccc(F)cc12 c1(-c2cn(C3CCN(C(C4CCS(=O)(=O)C4)=O)C3)nn2)ccc(F)nc1 C1(NC(c2n[nH]cc2F)=O)CN(C(c2cnn3c2CCC3)=O)CC12CCOCC2 N1(C(CCCCOCC)=O)C2CCC1CN(C(=O)CC(n1nc(C)cc1C)C)C2 c1(COC)nc(C(=O)NCCC2(OC)CN(C(c3conc3C)=O)C2)co1 CC1(CNC(C2CCC(OC(F)F)CC2)=O)CCCN(C(c2c[nH]c(=N)s2)=O)C1 c1(C(=O)NC(CNC(CCCC#C)=O)CC(C)C)c(OC)cc(OC)cc1N Cc1ncc(C(=O)NCC2CN(C(c3cc(C(F)F)on3)=O)C2)n1C N=C1NC(=O)C(CC(N2CCN(C3CCCN(C(=O)CC4(O)CC4)C3)CC2)=O)S1 CC1CN(C(c2cscc2C#N)=O)CCC1C(=O)N(C1CC(C(N)=O)C1)C S(=O)(=O)(c1ccc(Cl)c2nonc12)Nc1ccc(NC(c2ccc(Cl)cn2)=O)cn1 C1(NC(CS(CC)(=O)=O)=O)CCC2CN(C(c3ccc(C)nc3OC)=O)CC2C1 c1(C(=O)NC2CC(NC(C(CC)(F)F)=O)C(O)C2)ccc2cc(C#N)ccc2c1 N1(C(C2(C(=O)OCC)CCC2)=O)CC2CCC2(CCNC(c2cscn2)=O)C1 N1(C(CC2C(CC)C2)=O)CCC2(CCCC2NC(c2ccc3c(c2)CCC3)=O)CC1 c1(OC)cc(N2CCC(NC(C3CC3C3CC3C)=O)CC2C)c(Cl)cc1[N+](=O)[O-] CC(C)C(C(=O)N(CC(C)CNC(C1CCCC1C(C)C)=O)C)n1cccc1 C1(CNC(=O)CCc2ncccn2)CCC2(CCC2)CN1C(=O)C=CCF C(=O)(CC(C(F)F)n1cccn1)NCc1ccc(CNC(C(C)=C(C)C)=O)cc1 Cn1ccc(=O)c(C(=O)N(CC(=O)NCCC(=O)NC2CC2)CCO)c1 C1(C(N(C(CNC(=O)CN2CSCC2=O)C2CC2)C)=O)CCCC2(CCC2)C1 C1(C(=O)NC2CCN(C(c3cc(Cl)ns3)=O)CC2O)(OC)CCC(C)(C)CC1 N1(CC(N2CCCCC2c2cc[nH]n2)=O)CCN(Cc2ccc(F)cc2)CC1=O N1(C(C2(C3CCCCO3)CC2)=O)CC2=C(C1)CN(C(C13CC(F)C1C3)=O)C2 C1(CNC(C=CCC)=O)C(C)CCN1C(C1CCCN(C)C1)=O c1(C(=O)NC2CC(CNC(c3cccc(C)n3)=O)C2)cnc(C)c(N)c1 c1(CC)cc(Cl)ccc1C(N1CCCC1CCNC(c1cnnn1C)=O)=O C1(C)(OC)CC2CC1CC2NCC1CC2(C1)N=N2 N1(C(C2(NC(=O)CN3CC(C)(C)C3)C(C)CCC2)=O)CCCNC(=O)CC1 C12(CC(C)(C)C1)C(=O)NC2.C1(C(=O)NC2C=CCC2)(OC)CC(C)C1 Cc1csc2nc(CC(=O)NCC3(O)CC(CNC(C45CC(F)(C4)C5)=O)C3)cn12 c1(NC2C(C)C2)nc2c(c(=NCC3Cc4ccccc43)[nH]1)CCC2 C1(CNC(CNC(C)=O)=O)CN(C(=O)COc2cncc(Cl)n2)C2CCCC2O1 N1(c2nc(C)cc(OC)n2)CC(NC(=O)CC(C)(O)C2CC2)CC2(CCC2)C1 c1(C2C(CNC3(c4n(CCSC)nnn4)CC(C(C)C)C3)C2)ccc(C)cc1 Cc1cc(C)c(CN(C(CC2CCN(CC(=O)NCc3nc(O)n[nH]3)C2)=O)C)s1 C(=O)(CC1=NN(C)C(=O)C1)NC(CCC)CCCNC(=O)CCCN1CCCC1 N1(CC)CCOCC1C(=O)NCCCN(C(=O)C(n1ccnc1C)C)C(C)C C1(CNC(=O)COC2CCCCC2)C(C2CC2)CCN1C(=O)C(F)C1CCC1 c1(CNCC(C)(CC2CCOCC2)NC(C)=O)cn(C)c(=O)n1C c1(C(=O)NCC2(F)CCC(NC(C3(C)ON=C(C)C3)=O)C2)cccc(N)c1O C1(C(N(C)CC2(CNC(CCOC)=O)CC2)=O)(OCC)CCCCCC1 CC(C)CCC(O)C(=O)NCC(C)CNC(=O)C(F)(F)c1cnccn1 c1(CC)cc(C(=O)NC(C(=O)NC2CCCN(C)C2)c2ccco2)c(C)o1 c1(C2(C)CC2CNC(c2cnn(CCc3ccccc3)c2)=O)cn(C(C)C)nn1 c1(C(N2CCC(CNC(C(CN(C)C)N(C)C)=O)C2)=O)c(F)cccc1[N+](=O)[O-] Cc1cc(C(N2CC(C(=O)NC(=O)CNc3cccc(Cl)c3)C2)=O)cnc1O c1(C(=O)NCCOCCN(C(C2C(OC)C2)=O)C)cnn2cc(C)cnc12 C#CCCCC(=O)N1CCC(NC(c2cn(-c3ncccn3)cn2)=O)C1C C1(CC(=O)NCCC2CC(NC(C(C)OCC3CC3)=O)C2)COCCN1C c1(CC)nc(C)c(CNC(C2CCN(C(=O)C(C)NC(C)(C)CC)C2)=O)o1 Cc1nnccc1C(=O)NC(C)C(C(C)C)NC(C1(C)COC1)=O C1(C)(C(=O)NC(C2CCN(C(=O)C(C)=CC3CC3)C2)C)CCCC1 c1(C(N2C(CNC(C(CCC)OC)=O)CC(O)C2)=O)sc2ccc(Cl)cc2c1C c1(C(N2C3CC(NC(C4CCNC4=O)=O)CC2CC3)=O)cc([N+](=O)[O-])ccc1O c1(C(=O)NCC2CN(C(CNC(CC)=O)=O)C(C)C2)cnc(N)c(CO)c1 N#Cc1cccc(C=CC(=O)NC2CC2C(=O)NCc2cc[nH]n2)c1 C=C(Cl)C(C)(C)C(=O)N1CCC(NC(=O)CSc2c(C)noc2C)C(F)C1 C=C(Cl)CCC(=O)NCCOC(C)(C)CNC(=O)C(CC1CCCCC1)CC c1(C(N(CC(C)NC(=O)CC2CC23CC3)C)=O)ccnc(N2CCCC2)c1 c1(C(N2CC(CCNC(=O)CSCC(F)(F)F)OCC2)=O)cc(C(F)F)cnc1O CC(C)C(CC(=O)O)NC(=O)Cn1cc(-c2ccc(C(N)=O)nc2)nn1 c1(C(=O)NCC(CCOC)NC(c2[nH]c(C3CC3)nc2C)=O)ccc(C)nn1 C(CC(=O)N1CCCC1(C)C(=O)OC)(C(F)(F)F)NC(C1(CC#C)CCC1)=O N(C(=NCC(C)c1ncc(C)s1)NCN1CCOC(CC)C1)C(CC)CC c1(N2CCC(N(C(c3cc(SC)sc3Cl)=O)C(C)C)C2)cccc(Cl)c1Cl O=C1CCC(C(=O)NCC2COCCN2C(=O)CC2CCC(=O)NC2)=NN1 CC(c1cccc(C)c1)=CC(N1CCC1CNC(c1cn(C2CC2)nn1)=O)=O N1(C(c2cc(-c3c(OC)cccc3)no2)=O)CC(=O)N(C2CC2)C1=O c1(OC)cc(C(=O)NC2(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)cnc1O C=CCCCC(=O)NC(C)CCCNC(=O)Cc1nncn1C c1(SC)cccc(F)c1C(N1CCC(C)C1CNC(=O)Cc1cnn(C)c1)=O Cc1ccc(N)c(C)c1C(=O)N(CCCCN(C(=O)C(C)C(F)(F)F)C)C CC1=C(C)CC(C(=O)NC2CCCCN(C(=O)CN(C)C(=O)C3CC3)C2)CC1 c1(CNC(=O)C(C(C)C2CCOC2)OC)cc(F)cc(F)c1.c1(O)ccccc1F c1(C(N2CCC(COC(CC)(C)C)CC2)=O)cc(C(F)(F)F)cc(C(C)C)c1 N1(C(C(C(C)C)NC(C)=O)=O)CC2CC(C1)N(C(=O)C(C)(C)OC(C)C)C2 CC(CC(F)F)C(=O)N1CCC(C(=O)Nc2cccc(OCF)c2)C1C N1(C(CCC=CCC=C)=O)CC(NC(c2conc2C(F)(F)F)=O)C(C)(C)C1 C1(NC(C2CCCC(C)(C)C2)=O)CCN(C(c2csc(Cl)c2Cl)=O)CC12CCC2 CCC(CC)(CO)C(=O)NCC1CCCCC1NC(c1nc(=O)n(C)[nH]1)=O N1(C(C)=O)CC2CCN(C(C3CC3Cl)=O)CCC2C1.NC(C=O)=Cc1cccs1 c1(-c2cn(C(C)CNC(=O)C(F)C(F)(F)F)nn2)c(F)cccc1F c1(CC)cnc(C(N2CCC(NC(c3cnn(C(C)C)c3Br)=O)C2)=O)cn1 C1(C(N2CC(C)C(C)C2C)=O)(CC)CCN(C(=O)C=CC(=O)NC2CC2)CC1 c1(C(N2CCC(CC(=O)NC(C)C(F)(F)F)C2)=O)cc(Cl)nc(Cl)c1F c1(CC)[nH]nc(C(N2CCC(CO)(NC(=O)Cc3cncs3)C2)=O)c1Br C(N=c1nc2sccc2c(N2CCCCC(C)(F)C2)[nH]1)c1nn(C)c(Br)n1 C1(C(NOCCC)=O)CN(C(=O)CC23CCCC2C3)CC1CCCC.C(CCO)O C(=O)(C(C(C)(C)C)NC(=O)CCCC)NCC1(CO)C(C=C)C1 N1(C(CC2(C(=O)OC)CCOCC2)=O)CCCC(CNC(c2ccns2)=O)CC1 C1(NC(=O)NCC(C)S(C)=O)CCCC1P(C)(C)=O CC1CN(C(=O)C=C2CCC2)CC2(CCN(C(C3CC(=O)N(C4CC4)C3)=O)C2)O1 C1(CC)CN(C(=O)C(C)CC(=O)OC)CCN1C(c1cccc(C)c1F)=O c1(CN(CCN(C)C)C(c2ccnc(CN)c2)=O)ccc(F)nc1 N1(C(CNC(C(C)(C)C)=O)=O)CCC2(CCC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 C=CCCC(O)CNC(C1CC1C(C)NC(c1c[nH]nc1C(C)C)=O)=O C1(NC(CCN(S(C)(=O)=O)C)=O)COCCN(C(c2cncnc2)=O)C1 CC1(C)CCN(C(=O)CCF)C1CNC(c1ccc(C(F)(F)F)nc1)=O CC(C)C(CNC(=O)C=C1CCCC1)C(=O)NCCCN1CCCC1C c1(NC(C(C)C)C)ccc(S(=O)(=O)NC2CN(C)CC2O)cc1C#N C1(C(=O)OC)CN(C(=O)C(=O)N(C)Cc2c(C)nn(C)c2C)CC1(C)C C12(C(N(C(CC)CCOC)C)=O)CC(CN1C(=O)C(C)(C)COC)C2 CC12CC3CC(CC(C(N4CCCC(O)(CNC(C5CC5F)=O)CC4)=O)(C3)C1)C2 c1(C(N2C3C(NC(C(C)NS(C)(=O)=O)=O)CC(C3)C2)=O)ccc([N+](=O)[O-])cc1N c1(C(=O)NC(CCCNC(C(C)NC(CC)=O)=O)CO)c(C)cccc1Cl N1(C(C2(C(=O)NC)CC2)=O)CCC(NC(C2CSC2)=O)CC1C Cc1nc(NCCc2nc(Br)n[nH]2)cc(=NCC2(c3ccccc3)CC2)[nH]1 CC(CC(C)C(F)F)NC(C1(NC(=O)C(C)SC(C)C)CCC1)=O c1(CS(C)=O)c(C(=O)NC2(CO)CCN(C(=O)CO)CC2)oc2ccccc12 c1(C(=O)OC)c(C)[nH]c(C(N2CC(NC(c3ncc(C)cn3)=O)C2)=O)c1C C1(COC2CCN(C(=O)NCCC)C2)(Cc2ccccc2)CCCC1O N1(C(C=COCC)=O)CCC2CC1CN(C(c1sccc1OC)=O)C2 CP(C)(=O)CCC(=O)N1CCCC1C1(C(=O)Nc2ccc(SC3CC3)nc2)CC1 Cn1nc(C(=O)NCC2CC3CN(C(=O)C=C4CCC4)CC23)c2c1CCCC2O C1(C(=O)NCc2ccc(CNC(C(C)NC(C)=O)=O)cc2)CC(=O)N(OC)C1 c1(NC(=O)CCNCC2NCCC23CC3)ccc2c(c1)CCCO2 C1(CNC(c2cn[nH]c2)=O)(NC(c2scc(Cl)c2Cl)=O)CCC(F)(F)CC1 C1(CC)(CC)CC(NC(=O)C#CC(C)(C)C)CN1C(=O)CN(C)C N1(C(C)C(=O)NC2COCC2CNC(c2cc(Cl)cs2)=O)CCCCC1=O C(CC(CC)C(=O)N1CCC(CNC(=O)Cc2ccsc2Cl)C1(C)C)=CC Nc1ccc(NC(=O)C(F)CC2CC(C(=O)NCCCN)C2)cc1 Cc1noc(C)c1C(=O)NCc1ncoc1C1CN(C(C2C=CCC2)=O)C1 C(CC1CCCC1)(C(=O)N1CC(OCC(N)=O)C1)NC(COCC#C)=O N1(C(C2N(C(C(C)Oc3ccccc3)=O)CCCC2)=O)CCNC(=O)CC1 Cc1cccc(C(C)C(=O)NC(C2CCCN(Cc3ccc(CO)cc3)C2)C)c1 N1(C(c2cc(C(=O)OCC)c(C)[nH]2)=O)CC2(CCC(NC(C3(C)CC3)=O)CC2)C1 N1(C(C(C)OC)=O)CCN(C(=O)C(F)(F)CCn2ccnn2)CCC1C Cc1nc(C(=O)NC(C)CCNC(c2coc(Cl)n2)=O)c(C(F)(F)F)[nH]1 c1(NCC(C)CCO)cc(Br)ccc1S(=O)(=O)NC(C1CCCCO1)(C)C c1(NC(c2c(CNC(C3(C)CCNC3=O)=O)noc2)=O)cc(C#N)ccc1O N1(C(C(CO)NC(N)=O)=O)CCN(C(=O)CCc2ccc(F)cc2)CC12CCC2 c1(CCC(=O)NC(C(C)NC(c2n(CC)ccc2)=O)C)ccc(C)nc1 c1(C(=O)NCC2C(CNC(Cc3cn(CC)nn3)=O)C2)ccc2nn[nH]c2c1 C1(CC(=O)NCC2N(C(CC)=O)CC2)SC(=N)NC1=O CC1(CO)CCN(C(=O)CCOC2CN(C(C3CC(=O)CCO3)=O)C2)C1 c1(OCCCCC)cc(C)ccc1CNc1ccc(NC(=O)C2CC2)cn1 C1(CNC(C(C)Nc2scc(C)n2)=O)CCCN(C(C2(CC(C)C)CCC2)=O)C1 C1(NC(CCc2c(C)ncs2)=O)CCN(C(C2(COC(C)C)CC2)=O)CC1C c1(CC)ccc(C(=O)NC(C)C(CO)NC(C2(C(F)F)CCC2)=O)c(C)n1 c1(CNC(c2n(CCCSC)nnn2)C2CCCSC2)cn2cccc(F)c2n1 C#CCC(C(=O)N1CCC1C(N)=O)NC(c1csc(CO)n1)=O Cc1nc2c(o1)CCN(C(C1CC1NC(=O)Cc1noc(C)c1C)=O)C2 C12(CC3CCCC13)C(=O)NOC2.CCC(C)(C)NC(C)C(=O)NC1CCCO1 c1(C(=O)NC2(CCNC(C(C)n3ccnn3)=O)CCC2)ccc(N)c(F)c1F C1(NC(c2cc(OC)c(F)cc2)=O)CCC2(C1)CN(C(=O)C=C(C)C)C2 Cc1nn(C)c2c(NCC3CSC3)nc(=NCCC3(C(F)(F)F)CC3)[nH]c12 CCC(C)(CNC(c1ncoc1CCC#N)=O)NC(c1cnc(C2CC2)[nH]1)=O C1(NC(c2cc(-c3cn(C)nc3)no2)=O)CCN(C(C2(C)CC=CC2)=O)CC1O C1(NC(C(N2CCOCC2)C)=O)CC2CC(C1)N(C(C1CC1C)=O)C2 C(=O)(C(C)CC(C)(C)C)N1CCCC(NC(C2COCCN(CCCC)C2)=O)C1 c1(COC)nc(CC2CCCCC2)n(-c2ccccc2F)n1 C1(O)(C(CNC(C2(COC)CC=CC2)=O)C)CCN(C(c2csc(C)n2)=O)C1 C1(C)(CNC(C(C)Cc2ccncc2)=O)CCN(C(c2ccncn2)=O)C1 S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1C2C(N3CC(C)C4(C3)CNC4)CC(C2)C1 N1(Cc2cnc(C)o2)CC2CCC(NC(=O)CCC3CCCCO3)CC2C1 N1(C(CC(C)n2ccnc2)=O)CC2CC2(CNC(C2CC(O)CN2C)=O)C1 N1(C(CCCC=C)=O)CC(NC(C2(C)CCC2C(=O)OC)=O)CC12CCOCC2 C1(C(=O)NCCC2CCCCN2C(=O)CN2CCCCC2)CC2CCCCCC12 c1(CC(=O)NCCCC(C)NC(Cn2cc(C(=O)OC)nc2)=O)ccc(C)cc1F Cc1ccc(CSCC(=O)OCC(=O)N(C2CCCC2)C)nc1Br C1(CC(=O)NCCN2C(C)CCC2)CCN(C(c2scnc2Cl)=O)C1(C)C CC(C)CC(CNC(C1(C)CCC(=O)N1)=O)NC(=O)CCSCc1ccccn1 Cc1ccc(C=CC(=O)NC(C)C(C)NC(c2ccc(Br)s2)=O)cc1C C(C1CCOCC1)=CC(=O)N(C)CC1CCCN1C(C1CCC1(F)F)=O c1(CCC(=O)NCC2(O)CN(C(C3C(C)CC3)=O)C2)ccc(Br)c(Cl)c1 C(CCCCn1cc(C2(n3nccn3)CC2)nn1)NC(C1CC2CC2C1)=O c1(C(=O)NC(CCN(C(C(CC)(C)O)=O)C)C)oc(P(C)(C)=O)cc1C N1(C(C(C)SCC)=O)CCOCC(CNC(=O)C(C2CC(F)(F)C2)OC)C1 C1(NC(C2CCCS2)=O)(CO)CN(C(=O)CNc2ncccn2)C1 c1(C(=O)NC(C)C(CO)NC(=O)C(c2ccccc2)O)cc(Cl)ccc1O N1(C(Cc2c(C)ccs2)=O)CCCC(CCCCNC(C2OCC2(C)C)=O)C1 N1(C(C(C)N2CCC2)=O)CC2CCN(C(C3CCOC3c3ccncc3)=O)CC12 c1(C(=O)NC(C(=O)N2C(COC)CC2)CCF)cc2occc2[nH]1 C1(COC)CC(CNC(c2csc(C)c2C)=O)N(C(=O)CCc2cncn2C)C1 c1(C(=O)NCC(C)CNC(=O)CCOCCN(C)C)ccc(C2CC2)nc1 c1(C(N2CCC3C(NC(C(C)C(C)(C)C)=O)C32)=O)cccc2sncc12 c1(CN(C2CCCC2)C(CC2CCN(C(C(CC)C)=O)C2)=O)n[nH]c(C)c1Br C(CCCC(C)NC(C1(F)CCCCC1)=O)NC(c1c(C)scc1)=O O=C(C1=C(Cl)CC1)NC1CCOC(C(=O)NCCC(O)CO)C1 c1(C(N2CC(CNC(C(C3CCOCC3)C)=O)C(C)C2)=O)ccn(O)c(=O)c1 C=C=C(C)CC(=O)NCC1CCCCC1C(=O)Nc1cnc(C)nc1 C#Cc1ccnc(C(=O)NC2CN(C(=O)CNS(=O)(=O)N(C)C)C(C)(C)C2)c1 C1(NC(C2CCC(C)O2)=O)CCC2CCN(C(c3ccc4nc[nH]c4c3)=O)C12 c1(NC)nc(C)cc(=NC(CNC(c2cccc(Cl)c2)=O)C2CCC2)[nH]1 C1(C(N(C2CCN(C(C3CC=CCC3)=O)CC2)CC)=O)CC(C(C)=O)C1(C)C N1(C(C(=O)NC(c2ccncc2Cl)C)=O)CCC(C)C(N)C1 c1(C(N2CCC(F)(CNC(c3n(C)ccn3)=O)CC2)=O)ccc2ncncc2c1 c1(CCNOC)nc(N2CC(C(N3CCOC(C)C3)=O)C2)c(F)c(Cl)n1 C1(C(=O)NCC(CC)NC(C=CC(=O)NC)=O)CCC(CN2CCOCC2)O1 N1(C(C(C)OCOC)=O)CCCN(CCNC(=O)CCc2cscn2)CC1 c1(SC)ccc(N2CC(C(=O)NC3CCN(C(=O)C=C4CCC4)C3)CC2=O)cc1 C1(C(N(C(C)CNC(=O)C(C)(C)n2cc(Br)cn2)C)=O)CC2CCC1C2 c1(OC)ccc2c(c1)CCN(C(C1CCC3(CC3)C1)=O)C2C N1(C(c2n[nH]c(CC)c2Cl)=O)CC(CNC(C2CC(C)C2)=O)C(F)(CO)C1 C(N=c1[nH]nc(OC(F)F)s1)C1OCCN(C(C(N2C(C)CCC2C)C)=O)C1 c1(OC)cc(C(N2CC(C)(CC(=O)Nc3cc(F)cc(F)c3)C2)=O)ccc1I CCC(CC)C(C)C(=O)N1CC(CCNC(=O)CC23CCC(CC2)OC3)C(C)C1 C1(C)(OCC)CCN(C(C2CC(C)CN2C(c2cc[n+]([O-])cc2)=O)=O)CC1 C1(NC(COCC#C)=O)CCCC(NC(c2nnc(S)n2C)=O)C1 C1(CN(C)C)(NC(=O)C(C2CC2)N(C(=O)C=C2CCOCC2)C)CCCC1 C(=O)(C(CC(C)C)C(C)C)NCC1C(NC(C(C)N(C(C)=O)C)=O)C1 C(=O)(CCCCCCCCCO)N(C(C)CN(C(=O)C(Cl)=CCl)C)C c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC2O)ccc2ccc(Cl)cc2n1 N1(C(c2c(OC(C)C)nccc2)=O)CCCN(C(=O)C(C)n2ccnc2)CCC1 c1(C(C)C)ccc(F)cc1C(c1ccccc1)OCN1CCNCC1C(=O)NCCF c1(CCC(=O)NC2C(C)CCN(C(CC(CCC)O)=O)C2)c(C)nc(O)nc1C C12(CCCCC1C)C(=O)N2.C(CC(=O)NC)OC.S(C)(=O)(=O)N(CCN)C CCCC(C(=O)NC(CO)C(C)NC(c1ncn(-c2ccccc2)n1)=O)OC N1(C(c2cn(C(C)C)nc2)=O)CCC(C(=O)NCCn2ccnn2)C1C c1(C(=O)NCC2CCC(NC(C3(C4CCC4)CCC3)=O)C2)cc2c[nH]cnc-2n1 N1(C(c2c(CCC)nns2)=O)CCC2CN(C(C3CCSC3)=O)CC12 N1(C(=O)OC)C2CCC1CN(c1nnc(-c3n[nH]c(C)c3Cl)n1CC1CC1)C2 c1(C(=O)NC2C(NC(COC(C)C)=O)CCCC2)nn(C)c2c1CC(F)(F)CC2 N1(C(c2nnn3c2CCC3)=O)CC2CCN(C(=O)C(C3CCCCC3)F)CC2C1 c1(CCNC(c2n(CCSC)nnn2)c2nc(C)cs2)cncc2ccccc12 C1(C(C)C)CCCC(N=c2[nH]c(=NCC3(C)CCN(C)CC3)[nH]c3c2SCC3)C1 C(=O)(C1=CCCOCC1)N1CC(C)(C)C(NC(=O)Cc2ccc(Br)s2)C1 Cc1nc2sccn2c1C(=O)NC(=O)Cc1c(C)noc1C.C12CC1C2 CCC(CC)CCC(=O)NCc1ccc(C(N2CCc3ccsc3C2)=O)nc1 C1(C(N(CCCCN(C)C(c2ccc(-c3ccco3)o2)=O)C)=O)CC2CCC1C2 c1(C(N2CCC(CCNC(c3nc(C4CC4)cs3)=O)C2)=O)ccc(O)cc1 C1(N(S(=O)(=O)Cc2ccccc2)C(C)=O)CC2(C1)CN(Cc1ccc(O)nc1)C2 Cc1ccc([N+](=O)[O-])c(CC(=O)NCCCN(C)C(c2c(N)sc(C)c2C)=O)c1 N1(C(C(=Cc2ccco2)C)=O)CCCC2CN(c3ncc(C#N)cc3Cl)CCC12 N1(C(c2sc(CC)c(C)c2)=O)CCC2CCC12CNC(c1cnc(O)c(F)c1)=O C(C(F)(F)C(F)(F)F)n1c(-c2csc(CO)n2)nc(C(CC)C)n1 C#Cc1ccc(C(=O)NC2CN(C(c3ccc(SC)s3)=O)CCC2C)nc1 C1(C(=O)NCCCC(C)(C)NC(c2nc(C)oc2C)=O)CCOC(=O)CC1 N1(C(CC2C(=O)NC(=N)S2)=O)CC2CC1CN2C(=O)CCc1cncnc1 C1(CNC(C=C(CCC)C)=O)CCCC(NC(=O)CCSCC(C)C)C1 c1(C(=O)NC2CC(NC(CN(CCOC)C)=O)C2)cccc2[nH]nc(O)c12 C12CCCN(CC1)C(=O)C1(CC1)N(C)C2=O.C1(C(=O)OC)CCNC1=O CC#CCCCC(=O)NC1CCC(N(C(=O)CCCc2sccc2C)C)C1 N1(C(C2CC(C)CN(C(=O)C3=CC(C)(C)C3)C2)=O)C2CCCC1COC2 C1(c2ccc(OC)cc2C)NC(=O)N(CCC2CC2)C2=C1C(=O)NCC2 N1(C(N(C)Cc2ccccc2)=O)CCC2CCNC(=O)C2C1 c1(-c2ccc(C(=O)NCC(CCOC)OC)o2)ccc(F)c(OC)c1 Cc1ccc(C(N2CC3CC(C2)N(C(=O)CCCC(C)(F)F)C3)=O)c(=O)n1C C1(CNC(c2c(C)ccn2C)=O)C(O)C(O)CN1C(c1cnc(CC(C)C)s1)=O c1(CNC(C2(C=C)CCC2)=O)nc2c(s1)CN(C(=O)Cc1ccsc1Cl)CC2 O=C(CCCC1CCCO1)NC(c1ccccc1)C(=O)NC1C=CCC1 C12(C(N(C(CNC(c3cc(C4CC4)on3)=O)C3CC3)C)=O)CCC(F)(CC1)CC2 C1(C2CN(C(C3(C)CC=CCO3)=O)C2)(NC(CC=C(C)C)=O)CC1 N1(C(C(c2cnn(C)c2)C)=O)CC(C)N(C(=O)CC2COCC(C)O2)CC1C N1(C(C(C)(C)SC)=O)CC2(NC(c3cc(N)c(F)cn3)=O)CCC1CC2 CC(CC(=O)NC1CC(O)(CNC(c2cc(C(N)=O)co2)=O)C1)N1CCCC1=O C1(C)(C(=O)NCCN(C)C(c2ccnn2C2CC2(F)F)=O)CCNC1=O CCC(COC)C(=O)NCCCC(=O)Nc1cnn(C(C)(C)C)c1 O=NN1CCCC1C(=O)Nc1cccc(NC(C2CCCCNC2)=O)c1 N1(C(C2N(CC)CC2)=O)CC2CC1C2CNC(=O)CCC(C)N(C)C c1(C(=O)NC(C(C)(C)C)CNC(c2cccc(O)n2)=O)cc2sccc2n1C c1(SCCNC(=NCC)NCCC(c2ccccc2)O)ccccc1S(N)(=O)=O C1(CCC)(NC(c2cn(C)cc2C)=O)CCN(C(c2cnnn2CC)=O)CC1 C1(OC)CCN(C(=O)CSCCNC(=O)Cc2ccnc(O)c2)CC1C C1(C(=O)NCC(C)(C)NC(C2CCN2C2CCCC2)=O)CCC2(CC2)C1 N1(C(CCN(CC(F)(F)F)C)=O)CCC(CF)(NC(c2cnc(Cl)[nH]2)=O)C1 c1(C(N2C(CNC(C3(C)C=CCC3)=O)CC2)=O)cccc(C(OCCN(C)C)CC)c1 CC1CC(C(=O)N2CCCC(NC(=O)CCS(C)(=O)=O)C2C)=NO1 c1(CC(=O)O)coc2c1CN(C(C1CCC(Oc3ccncc3)C1)=O)C2 c1(N2CCC(NC(C34C(C)(C)C(CC3)CC4)=O)C2)nnc2c(c1C#N)CCCC2 C1(C)(C(=O)NCC2C(C)CN(C(C3CCC(O)CC3)=O)CC2)CC2(C1)CC2(F)F n1(CC(=O)N(C)CC2N(C(C3C(C)=C3)=O)CCC2)ccc2c(N)cccc12 Cc1ncc(Br)c(C(=O)NCCN2CCN(C(=O)CC3CCCCCC3)CC2)n1 C1(NC(CCc2c(C)nccc2)=O)CC(C(=O)O)C12CCC2 c1(NC(N(CCC)C(c2ccccc2)C)=O)c(Cl)cc(Cl)nc1C c1(OC)cc(C(=O)NC2CC(C)N(C(c3ccc(SC)o3)=O)C2)nn1C CC1CN(C(C2CCS(=O)CC2)=O)CC(C)N(C(c2cnc3n2CCS3)=O)C1 c1(CN(C)C)cc(NC(=O)NCCCCCN(C)C)cc(Br)c1 c1(SC)cc(C(=O)N(C)Cc2ccccc2CNC(=O)CC(F)(F)F)c(C)o1 NC(=O)CCC(=O)NCCC1(O)CN(C(=O)C=CC(=O)NCc2ccccc2)C1 c1(C(N2CCN(C(c3[nH]cc(C)c3)=O)CC2CCO)=O)ccc2nc(O)sc2c1 C1(C(=O)NC(CC=C)CO)CC(NC(=O)CC2CC(OCC)C2)CCO1 c1(C(N2CC(OC)C(NC(=O)C(C)(C)c3ccsc3)C2)=O)nnn2c1CCCC2 C(=O)(CC(CC=C)NC(=O)C(C(C)OC)N(C)C)N(CCC=C)CC C(=O)(C(F)C(C)C)OCc1nnc(CC)s1 C(C(=O)N(CCCNC(=O)CCSC1CCCO1)C(C)C)(SC)SC C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(=O)C(F)C(C)(C)O)C2(CCCCC2)C1 C1(C)(NC(c2nccc(CC)c2)=O)CCCCC1C(=O)NCC(C1CCCC1)OC N1(C(CC(C)c2cnn(C)c2)=O)CCC2CN(C(=O)CC3CCC3)CC2C1 N1(C(C(C)NC(C)=O)=O)CC2(C)CN(Cn3ccc(C4CC4)n3)CC2(C)C1 c1(C(=O)NCC(CCNC(=O)CC2CCOC2)O)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC2(C)CN(C(c3cc(OC)cc(OC)c3)=O)C2)cc2sc(F)cc2[nH]1 CC(CC(=O)NC(C1CCN(C(c2scnc2C(C)(C)C)=O)CC1)C)P(C)(C)=O CCC(CC(C)C)C(=O)N1CCC(CC(=O)NCC2(CN(C)C)CC2)CC1 C12(C(=O)NCCN(CCO)CC)CCCCC1N(C(=O)C(C)CCOC)CCC2 Cn1cnc(C=C(F)C(N2CCCC2CC2C(C)(C)C2(C)C)=O)c1 c1(C(N(C2CCCN(C(C3CS(=O)C3)=O)CC2)CC)=O)cccc2occc12 C12(C(CNC(Cn3ncc(C)c3)=O)NC(=O)CC3CC3(Cl)Cl)CCC(CC1)C2 Cc1nn(CC(C)C)c(C)c1CN1CCN(C(=O)NC(C)(C)C)CC1C(F)(F)F c1(N2CCN(C(C(C(=O)OC)(C)F)=O)CC2)cc([N+](=O)[O-])ccc1Br CC1CC(C(=O)N2CCC(C)(C)C2CNC(=O)CC(C)(C)C)=NO1 CCCC(C)(O)CC(=O)N1CCOC(C(=O)NCCc2ocnc2CO)C1 c1(C(=O)NCC(c2ccccc2)N(C(C(C)C2CC2)=O)C)cnn(C)c1 C12(C(=O)NCCCN(C(c3ccc(COC)cc3)=O)CC)CCC(O)(CC1)CC2 N1(C(c2cc(C(C)C)no2)=O)CCC2C(CCN2C(=O)CC2(C)CCCCC2)C1 Cc1nocc1C(=O)N(C(C)CC(=O)N1CC(c2cccnc2)C1)C C(=O)(CC(C)CC(C)C)NCCC1(OC)CN(C(c2nnsc2N)=O)C1 c1(C(N2CC(NC(c3cnn(CCC)c3C)=O)C(O)C2)=O)ccc(C#N)cc1C c1(C(=O)NCCC(C)(C)NC(CN(C2CC2)CC)=O)cc2cc(F)cc(F)c2[nH]1 C1(C(=O)NCC2(CC(=O)NCCCN3C(C)CCC3)CC2)CC(=O)OC1(C)C CC1CN(C(=O)CN(C)CCO)CCCN1C(c1ccc(OC(F)(F)F)nc1)=O c1(OC)cc(C(=O)Nc2cccc(F)c2Cl)c(NCc2cc(Cl)cnc2Br)cn1 N1(c2ccnc(NCCCc3c(OC)cccc3)n2)CC2(C1)CN(C)CCO2 CC1CC(C(=O)NC2COCC2CO)CN(C(c2ccnc(O)c2)=O)C1 CC1(C)CCN(C(c2nc(Cl)cs2)=O)C1C(=O)NC1CCCC1N=[N+]=[N-] Cc1cccn2cc(CC(=O)NCC3CCC(NC(=O)C(O)C(F)(F)F)C3)nc12 Cn1cc(C=CC(=O)NC2(C)CC(NC(c3cn(CC(F)(F)F)cn3)=O)C2)cn1 N1(C(C2N(C(C)=O)CSC2)=O)CCCC(N(C)C(C2COCCO2)=O)C1 C(=O)(C(C(C)C)OC(c1cncc(-c2cccnc2)c1)=O)NC C=CC(C)(CC)C(=O)N1CC(CNC(C2CCC3(CC2)CC3)=O)C(F)(F)C1 C=CC(CCC)CC(=O)NCCN(C)C(c1c(F)cc(OC)cc1Cl)=O CC(O)(Cc1ccccc1)C(=O)NCC(CC(F)(F)F)NC(C1(CO)COC1)=O N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2cccc(F)c2C)=O)CC1CC(C)(C)C C1(OC)CN(C(=O)C(C)(CSC)NC(C2CC(SC)C2)=O)CC12CC2 Cc1cc(Cl)c(C)c(C(N2CC(CO)(NC(=O)CCC=CC(C)C)C2)=O)c1N CC1(C)CN(C(C2CCNC(=O)CC2)=O)CC1c1cn(-c2ccc(F)cc2)nn1 c1(NC(C(N2CCC(CNC(C3CC(=C)C3)=O)C2)=O)C)ccc(Br)cc1 c1(NCC2CCN(CC)CC2)nc[nH]c(=NCC2(F)COCCOC2)c1C Cc1cn2c(C(=O)NCC3CCN(C(C4CCCS(=O)(=O)C4)=O)C3)c(C)nc2s1 CC(=O)CCCC(C)C(=O)NCCC(=O)N(C)C(c1nccs1)C NS(=O)(=O)c1ccc(F)c(NC(c2ccccc2CF)=O)c1 C=C(Cl)CCC(=O)NC1C2CC(NC(c3cn(CCC)nn3)=O)CC12 C(=O)(CCC(CF)CF)NC1C(C(N2C(C(=O)NC)CC(O)C2)=O)COCC1 C#Cc1ccccc1CNC(=O)CC(C(C)OC)NC(=O)C(C)OC NC12CCOCC1CN(C(=O)C=CCN1CCOCC1)C2 C1(C)(NC(Cc2nc(C(C)(C)C)sc2)=O)CCN(C(=O)C(=O)NCC(F)F)C1 N1(C(Cc2ccc(C)o2)=O)CC(CCNC(=O)CC2(C#N)CC2)OC(C)C1 C12(CNC(c3ccc(CC)cc3)=O)CC(NC(c3ncccc3Br)=O)(CCO1)C2 C1(NC(C2(N(C)C)CCC2)=O)C2CC1N(C(C1CC1c1cccc(Cl)c1)=O)C2 CCC(C)C(O)CC(=O)N1CCCC(C)(C(=O)NC2CCN(C)C(C)C2)C1 c1(C(N2C(CNC(C3N(C(C)=O)CCCC3)=O)C=CC2)=O)nccc2n[nH]cc12 N1(C(C(C)=C2CC2)=O)CCC(F)CC1C(=O)N(C1CC(C)C1)C N1(CC(C)(C)NC(C(CN(C)C)O)=O)CCN(C(=O)CC2CCC(=O)N2)CC1 S(=O)(=O)(c1cccnc1N1CC(F)C(F)C1)NC(C)C(C1CCCCC1)C C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(Cc2nc(CC)sc2)=O)CC1C1CC1 Cc1cccn2cc(C(=O)NC(C)CCCNC(=O)C(CO)C(C)C)nc12 CCCCCCCC(F)C(=O)NC1CCCCC1CNC(=O)C=C1CCOCC1 C1(NC(c2nc(C)oc2)=O)CN(C(c2cnsc2)=O)CCC1C C(=O)(C(C)(CC)C(N)=O)NCC(C1(O)CCN(C(C=CC=CCC)=O)C1)C C(C)(C)(C(C)CC(=O)N1CC(C)(O)C1)NC(c1nc(C)oc1)=O C1(C(=O)NC2C(C)(C)CN(C(c3cnc(O)n3C)=O)C2)CCCC2(C1)CC2(F)F c1(C(N2CC=C(CCNC(CC(C)(C)SC)=O)CC2)=O)ccc2cn(C)nc2c1 C(CC(C)(C)C)(C(=O)Nc1cnc(F)c(C)c1)NC(C12CCC(OC)C1C2)=O c1(C(=O)NCCC(C)NC(C(C)C#N)=O)cc(Cl)ccc1OCC(F)(F)F c1(CC(N2CCC(CNC(C(F)=CCC)=O)C23CC3)=O)ccc2nc[nH]c2c1 c1(N(CCCCOC)C)cccc(S(=O)(=O)NC2CCS(=O)(=O)C(C)C2)n1 CC(C)CCC(=O)N(C(C)C(N1CCC1(C)CCO)=O)C1CC1 c1(OC)ccc(CCC(=O)NC2CC2NC(=O)CNS(N)(=O)=O)cc1OC C12(NC(C=C(C)C)=O)CC1CN(C(=O)CCc1ccccc1OC(F)(F)F)C2 C1(CC)CN(C(C2CCC(C(=O)NCc3ccc(CC(=O)O)cc3)C2)=O)CCO1 C1(CC(N2C(C)(C(=O)OC)CC2)=O)CC(NC(=O)CNC(=O)CC(C)C)C1(C)C CN1CCC(C(=O)NCCC2(O)CN(C(c3[nH]ccc3-c3ccccc3)=O)C2)C1 c1(OC)ccc(CCC(N2CCCC2c2cccc(Br)c2)=O)cc1 C1(NC(C(C)OCCCCCC)=O)CC(CNC(c2cc(=O)n(C)o2)=O)CC1O c1(CC)c(C(=O)NC2CCN(C(C34CCCC3CC4)=O)CC2)oc2ccccc12 N1(C(c2c(COC)scc2)=O)CCC(N(C(=O)C2=CCSC2)C2CCOCC2)CC1C Cc1nc(N2CC3(CCCC3NC(=O)C3=C(Cl)CCOC3)C2)c2ccsc2n1 C=C(Cl)CCC(=O)NC(C)CCCCNC(=O)C(C)COC(C)=O C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CCC(NC(CCSCCC)=O)CC1 c1(CC(N2CCC(N(C(C=CC)=O)C)C2)=O)ccc(OC)cn1 C12(NC(C(CC=C)(F)F)=O)CCC(CNC(=O)COCCOCC)(CC1)OC2 c1(C(=O)OCC)cc(NCc2cn(C)nc2C(F)F)ccc1C C(=O)(C1CCc2nnc(C)n21)NCCC1N(C(Cc2cc(C)no2)=O)CCSC1 N1(C(CC2CCC(OC)CC2)=O)CC2CC(C1)CN(C(=O)Cn1ccc(C)n1)C2 C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(CNC(CCC(CC)OC)=O)C N1(Cc2cc(C(=O)OC)n[nH]2)CCC2C(C1)NC(=O)CCN2C C(CNC(C1COC(C)(C)C1)=O)(CC)(CC)NC(c1nc(CCC)oc1)=O C1(CNC(CCC#C)=O)COC(C)(C)CN1C(c1ccc(-n2cccn2)c(C)c1)=O c1(C(=O)OC)cc2c(s1)CCN(C(c1cccnc1C)C(=O)NC1CCCC1)C2 C#Cc1cccc(CC(=O)NC2CC3C(NC(C4(OC(C)=O)CC4)=O)C3C2)c1 C(=O)(CC(C)C(C)(C)C)NCC(C)(CC(C)C)NC(c1c(CCC)sc(S)n1)=O C(=O)(C1=CC(C)(C)C1)NC(C1(C(N(CC)Cc2cnn(C)c2)=O)CC1)C N1(C(CCC)=O)CCCC(C(N2CCCC2COC)=O)C1CC C=CC(C)CC(=O)NC(CCOC)C(=O)NC1CCCC1CCOC c1(CNC(=O)Nc2ccc(OC)c(F)n2)c(O)cc(F)cc1F C1(C(N2CC(OCCOC)C2)=O)CC12CCN(C(=O)Cc1ccsc1C)CC2 C1(C(=O)NC(C(C)F)C)CCC(C2CC2)N1C(=O)C=Cc1nccs1 CCCCC(C(=O)NC1CCN(C(N)=O)C1)NC(=O)C(CCC)N(C)C CC1CC(C(=O)NC2CC3CN(c4ccnc(C#N)n4)CC23)=NO1 C12(C(=O)NCC(N(C(C3(OC)CCSC3)=O)C)C3CC3)CC(C)(C1)OC2C N1(C(c2ccc(C3CC3)cc2)C)CC(Cc2c(C)cccc2)CCC1C N1(C(C2(CSC)CC2)=O)CCC(F)(C(=O)NC2(CF)CC2)C1 C1(C(=O)N(C)CC2CCCC2(C)C)(SC)CCN(C(=O)C(C)SC(C)C)C1 c1(CN2CC3N(C(c4c(C)cnn4C(C)C)=O)C3C2)ccc2ncnn2c1 N1(C(C(CC)C2CCOCC2)=O)CCC(C)(CCNC(c2c(C)ncn2C)=O)C1 c1(NC(C(=O)N(CCC2CCOC2)CC)=O)cc(OC)c(OC)cc1OC N1(C(c2ccccc2)C)CCC(C)(NCc2cn(-c3cccc(Br)c3)nn2)C1 CC(C)(C(=O)NC1CCCC(CNC(c2c[nH]nc2Cl)=O)C1)C(F)F C(=O)(C(C)(C)CCCO)NC1(CC=C)CN(C(=O)C=CC(c2ccccc2)=O)C1 c1(OCC)cc(C(=O)NCC(C)N(C(=O)Cc2cnccc2C)CC)ccc1C c1(C(=O)NCC(C)CNC(=O)C(C)C2CCCO2)ccc(C2CCC2)nc1 C1(C(=O)NC2C(C)N(C(c3cnn(C)c3N)=O)CC2)CNC(=O)CC12CCOC2 c1(SC)ncc(N)c(C(=O)NC(C)CCNC(=O)Cc2cc(F)cc(Cl)c2)n1 C(=O)(N=c1cc(C(=O)NC2CCC3(CC2)CNC3)[nH][nH]1)c1c(N(C)C)nccn1 CC(C)CC(=O)C(=O)NCCC1(C(N2CCC(CCCO)C2)=O)CCC1 C1(CC(=O)NC2CCC(CCNC(c3c(C)ccs3)=O)C2)CCCC(C2CC2)O1 C(N=c1ccnc[nH]1)c1nc(CNC(=O)C=Cc2cc[nH]n2)nc(O)c1 C(=O)(CC(CC)C(C)(C)C)N1CCC(N(C(c2ncc(C#C)cc2C)=O)C)C1 c1(CCC(=O)NC(C2(O)CN(C(c3cc[nH]c3)=O)C2)C)ccc(Br)s1 c1(OCCC)ccc(N(C(c2ccnc(F)c2)C(=O)NC)C)cc1 c1(C(=O)OC)ccccc1CNC(=O)CC1(C(N(C)C)C2CC2)CC1 O=C(CCS(=O)(=O)C(F)(F)F)NCC1CC(O)CN1C(=O)CCC(F)(F)F C1(C(=O)NCC2CCC23CCC3)CCC2(CC2)N1C(=O)CN1CCSCC1 N1(C(C(CCC)OC)=O)C2CCC1CC(F)(CNC(C1(CC)CCC1)=O)C2 Cc1cc(C(N2CC3CC2C3CNC(=O)C(C)(C)COC(C)C)=O)c(C)n1C1CC1 C1(OC)(CNC(=O)C=CCCc2ccccc2)CCN(C(C2(C)CC2C)=O)C1 C1(C(N2CC(C(=O)NCC(=O)OC(C)C)(COC)C2)=O)CC2CC(=O)C1O2 C(=O)(C#CC1(C)CCCO1)N1CCC2(CC(C(N(CC(F)F)C)=O)C2)C1 c1(C(=O)NCCC(C)NC(=O)COC2CC2)ccc(Cc2cccs2)cc1 c1(NC(CCCCC)C2CC2)nc2ccccc2nc1NC1CCN(CC)C1 C1(C(=O)NC2CN(C(C(CC)OC3CCCCC3)=O)C2)CC(S(C)(=O)=O)C1 C1(NC(c2ccc(OC)nn2)=O)CCCCN(C(C2OCCC2C)=O)C1 c1(NCC2C(C(=O)OC)C2)cccc(NC(C2CC(F)CN2C(C)=O)=O)c1 c1(C(=O)NCCCC(C)NC(=O)C=CCN(C)C)ncnc2c1cnn2C c1(C(N(C2CN(C(c3c(SC)csc3)=O)CC2(C)C)C)=O)cccn2nncc12 C1(CC(=O)NC2CN(C(C3CCC(=C)CC3)=O)C2)CCCC2CCCCC12 c1(C(=O)NC(CN(C(=O)CC2CC3CC3C2)C)(C)C)ccc(S(N)(=O)=O)s1 C1(NC(CSc2ccc(OC)cc2)=O)CN(C(=O)CC2CCN(C)C2)CCC1F Cc1ccc(CC(=O)NC2CC2CNC(c2cn(C(C)(C)C)nc2C)=O)c(C)c1 c1(N(CC=C=C)C)nc(-c2ccccc2)nc(=NCCCOCCCO)[nH]1 C1(c2nnnn2C2(C)CC2)(NC(c2cccc(NC)c2)=O)CCOCCC1C c1(CC(C2CC2)NC(=O)NC2CCCCC2)ccccc1 CC(C(=O)NC1(C)CC(NC(=O)CCOc2ccc(F)c(F)c2)C1)S(N)(=O)=O CCCC(C)(CC)C(=O)NCC(C)(C)CNC(c1ccc(=O)n(CC(C)O)c1)=O N1(CC)CC(NC(=O)C(c2ccco2)NC(c2cc(C(F)F)[nH]n2)=O)CCC1=O C#Cc1cncc(C(=O)NCC2CN(C(=O)CC(=O)NCC3CC3)CC2(F)F)c1 C1(CNC(CC(C)SC)=O)CCN(C(c2cc(Cl)nn2C)=O)C1(C)C N1(C(C(COC)(C)C)=O)CCC2CN(C(=O)C=CC(=O)N(C)C3CC3)CC2CC1 c1(C(=O)OC(C(=O)NCCC2C(C(=O)OC)CC2)=O)ccc(C(F)(F)F)cc1 C1(C(N2CCC(F)(CNC(C(C)(C)CF)=O)C2)=O)CC2CCC1CC2 C1(NC(C(C)NC(N)=O)=O)CCC(CNC(=O)CCCn2ccnn2)CC1 C(C)(CN=c1nc(C(C)(C)C)nc[nH]1)N(C(CC(CC)CNC(C)=O)=O)C c1(NC(CC)=O)ccc(C)c(C(=O)NC2CCCC2NC(=O)C(Cl)=CCl)c1 c1(C(C)C)n[nH]cc1C(=O)NC1COCC1C(=O)N(C)Cc1ccon1 CCC(CC(F)F)C(=O)N1CCOCC(NC(C2(C)CCC(=O)NC2)=O)C1 C1(NC(c2c(C)nc(CO)s2)=O)COC2(CCN(C(c3ncn(C)c3C)=O)C2)C1 C(CCCCCCCC1CC1)(N(C)Cc1ccc(F)cc1)C1CC1 C(c1cccc(C)c1)=CC(=O)N(CCNC(=O)CC(C)(O)C1CC1)CC N1(CC)CCN(CCC(=O)NCC#CCNC(C2(O)COC2)=O)CC1 C(C)(C)(C(=O)NCCCCCNC(C1CC(O)C1)=O)OCC C1(CNC(C2CN(C(C)=O)C2)=O)CC(C)CCN1C(=O)C(O)C1=CCCC1 c1(NC(c2ccc(NS(=O)(=O)CCCl)cn2)=O)cc(Cl)nc(Cl)c1Cl c1(C(N2CCCCC(CNC(=O)Cn3cncn3)C2)=O)ccn2c(O)nnc2c1 C1(C(N(CCCC)CC)=O)(NC(c2cncn2C)=O)CC(O)C1 CCC(C)C(CC(=O)NC1CCC(=O)NC1(C)C)NC(=O)C(C(C)C)N(C)C C1(C)(C(=O)NC2C(NC(C3(CCOC)CC3)=O)CCC2)CC2(C1)CC(F)(F)C2 c1(C(=O)NC2C3CN(C(c4cocn4)=O)CC23)ccc(Br)cc1I N1(C(CCOC(CC(C)C)C)=O)CCCC(N(C)C(C2(O)CCOCC2)=O)CC1 CCCCC(CNC(=O)CCC(C)OC)NC(C1CCCN1C1CC1)=O C1(NC(c2cnc(CC)o2)=O)CN(C(C2CC(C)CC(=O)N2)=O)C(C)(C)C1 Cc1cc(C(=O)NCC2(NC(=O)CSc3cn[nH]c3)CC2)c(C)n1C(C)C c1(NCC)ncccc1C(N(C1CC(NC(=O)CCCCNC(=O)OC)C1)C)=O N1(Cc2ccc(C(=O)OC)cc2)CCC(CN2CCCC3(CC3)C2)CC1C C1(C(C)CO)CCN(C(C2C3CN(Cc4cc(Cl)ccn4)CC23)=O)CC1 C1(C(CNC(C=C(CCC)C)=O)(C)C)CCN(C(=O)CCC(C)SC)CC1 C1(C(C)(C)C)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CCN1C(C1CCOC1)=O C#CCC(O)C(=O)N(CCCOCCNC(c1n[nH]c(C)c1Br)=O)C N1(C(=O)N(C(C2CC2C(C)(F)F)=O)C2CC2)CCCCC1C(O)C1CC1 C1(CCCC)(C(=O)NCC2CCN2C(C2CC3CC3C2)=O)CCCC1 Cc1cc(C(N2CC(NC(c3c(C)ncn3C)=O)CC(C)C2)=O)ncc1N N1(C(C=Cc2cn(C)nc2)=O)C2CCC(C2)C1C(=O)NCC1CC(=O)N(C)C1=O c1(C(=O)NC2(COC)CN(C(C3CCCS3)=O)C2)ccc2nnc(S)n2c1 C(CO)(C(=O)NCC1(NC(=O)CN2CC3CC3C2)CCCC1)N(C)CC N1(C(CC(C(C)C)O)=O)CCC(C(=O)N(c2cccc(C#N)c2)C)C(C)(C)C1 c1(C(N2CCC2CNC(C2C(=O)NCCC2C)=O)C)cccc2ccccc12 N1(C(c2cnc(C)nc2)=O)CCC2(CC1)CCN2C(c1cc(Br)c(C)cc1O)=O C#CCC(C)(CC)C(=O)NCC(C)(C)C#CC(=O)Nc1ccc(F)nc1 Cn1nc(Br)c2cnc(N3CCCC34CCN(C(=O)CC3C=CCCC3)C4)nc12 CC1SCCCC1C(=O)NCCNC(c1cc(-c2ccn(C)n2)on1)=O c1(C(N2CCC3CN(C(C4C5CCCOC45)=O)C3C2)=O)cccc2nc(Cl)cn12 C(=O)(CC(C)(C)CC(=O)NCc1cn(C2CC2)cn1)c1ccc(C)cc1 c1(C(N2CC3C(N(C(C=CC=CC)=O)C)C3C2)=O)cc(O)ccc1CC C1(NC(=O)Cc2ncc(Cl)s2)CC2CC1CN2C(=O)CN1CCOCC1=O CCCCS(=O)(=O)CC(=O)NC1CCCC(NC(c2nc(C)c(N)cc2C)=O)C1 C1(CNC(CC=CCC)=O)CN(C(=O)COc2cc(C)on2)CC1(F)F C(C1(C)Cc2ccccc21)NC(C)(C)C.c12nc(SCC)cc(n1)N(C)C2C C1(CNC(CCCNC(C)=O)=O)CCN(C(c2cc(C(F)F)nn2C)=O)CC1C C(=O)(C1CCc2nccn21)N1CCN(C(C2(C)CSC2)=O)CC1CO C#CCC(C)(CC)C(=O)NCC(C)(CC)NC(c1ncc(C(N)=O)cc1Cl)=O C(=O)(CC(C)(C)CC=C)NC1CCC(C(=O)NCC2(C#C)CCC2)CC1 c1(C(=O)NC2CC(NC(COc3cccc(C)c3)=O)C2)cn(C)c(=O)nc1O C(=O)(CCC1(NC(c2ccon2)=O)CCC1)NC(C1(C)CC1)CO C1(NC(COC(C)=O)=O)CCCC12CCN(C(c1cccc3nsnc13)=O)CC2 N1(C(c2c(C)ccnc2)=O)CC2CCC(C1)C2NC(=O)C(C)Cc1ccccn1 C(=O)(C1=NNC(C(F)(F)F)C1)NCC1C2CN(C(c3nn(C)c(Cl)c3)=O)CC21 c1(CNC(C2(COC)CN(C(=O)CC3CC4CC4C3)C2)=O)cc(OC)ncn1 Cc1ccccc1C(C)CC(=O)NC1(CN(C(=O)C(C(C)C)N(C)C)C)CC1 N1(C(C23C(NC(C4C(CC(C)C)C4)=O)CC(CC2)C3)=O)CCC(=C(F)F)CC1 CN1C(=O)CSC1=CC(=O)N1CC2C(CNC(C3CCCS3(=O)=O)=O)C2C1 CCCC(CC(C)C)C(=O)N1CCOC(C(=O)NCCCCCC(C)C)CC1 c1(C(N2CCC(C)(CNC(C(C)SC(C)C)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(=O)NC(CNC(CCOCC)=O)(C)C)ccnc(OCCO)c1.CC(F)(F)F c1(N(C(c2cccc(Cl)c2Cl)C(=O)NC(C)C)C(C)C)cccc2ccccc12 N1(C(CCCCCNC(=O)C2=C(Cl)CCC2)=O)CCC2C(C1)C2(F)F c1(OC)ccc(-c2cnccc2C(=O)Nc2sncc2C(N)=O)c(OC)c1 c1(C(=O)NCC(C)CNC(C2CC2c2ccccc2F)=O)cc2cccnn2n1 N1(C(C(C2CCC2)NC(Cn2ncc(C#N)c2)=O)=O)CC(=O)NC(=O)C1 n1(CC)cc(Cl)cc1C(=O)NC(C1CCN(C(C2(C3CCCO3)CCC2)=O)C1)C C1(C(N2CCCC2CC2CC2)=O)(OC)CCN(C(c2cnco2)=O)C1 C1(NC(c2c(C)c[nH]c2)=O)CC(O)CN(C(c2cn(C)nc2-c2ccoc2)=O)C1 c1(C(=O)NCCNC(C2N(CC)CCCC2)=O)c(Br)nc2n1CCC2 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CC(CNC(=O)Cc2cn[nH]c2)C2(CC2)C1 C(CCC(C)CC(=O)NC1C2CN(C(=O)CS(=O)(=O)N(C)C)CC12)=C(C)C C(C1CCCc2ccccc21)NC(C1N(c2nc(OC)c(C#N)cn2)CCOC1)=O c1(C(n2cc(-c3ccc(Br)s3)nn2)COC)ccccn1 c1(C(=O)NCCC2CCCN2C(C2C=CCCC2)=O)ncncc1Br N1(C(C(CC=C)NC(c2cc(CC)no2)=O)=O)CCCN(C)CC1CC c1(C(=O)NC2CCN(C(C=NOC)=O)C2)nc2c(cc1Br)OCCO2 C=CCC(CC(C)C)C(=O)Nc1ccccc1OCc1cccs1 c1(C(=O)NCC(C(C)(C)C)NC(c2ccc([N+](=O)[O-])s2)=O)cnc2[nH]ccc2n1 Cc1cc(C)n(C(C)CC(=O)NC(CCNC(=O)Cc2cnc(C)s2)C(C)C)n1 CC(CC(=O)N1CCCC1CN1CCCCC1)C(=O)c1cccc(F)c1 c1(CC)cc(F)ccc1C(=O)NC(CNC(=O)C(CSC)c1ccccc1)CC Cc1cc(F)c(NC(=O)CC(=O)c2ccccc2)c(Br)c1 Cc1ccc(OC(C)C(=O)NC2C=CCN(C(c3c[nH]nc3C)=O)C2)c(C)c1 N1(C(c2ccn(C)c(=O)c2)=O)CC2=C(C1)CN(C(C1CCc3ncsc3C1)=O)C2 CC1CC(=O)NC(C(N2CCCC(CC(=O)NCC3CNC(=O)C3)C2)=O)C1 C(=O)(C(C)(C)C(F)(F)F)NC(CC1CN(C(CC2CC(OCC)C2)=O)C1)C c1(N)nc2cc3ccccc3cc2s1.C1(CN)CC(=O)N1.C(C(=O)O)OC c1(C(=O)NCCC(C)NC(C23CCC(CC2)C3)=O)cc(N)cc(S(C)(=O)=O)c1 N1(C(=O)OC(C)(C)C)CCCCCCC1C(=O)NCC1(O)CC(CN)C1 c1(OC)ccc(CC2CCCN2C(C2CCN(C)CC2)C(=O)NC)c(Br)c1 C1(C2(NC(CCNC(N)=O)=O)CC2)CCCCN1C(=O)CC1CC2(CC2)CO1 C1(C(C(=O)NCCCN(C(=O)C(C)N=[N+]=[N-])CC)(F)F)(OC)CCCCC1 c12ccnc(c1)NC(=O)C2.CC1(CC2CC2)CN(C(=O)CCC2CCCC2)C1 c1(C(=O)NCC=CCCNC(c2cc(OC)ncn2)=O)cc2sccc2[nH]1 c1(C(=O)NC(C(C)NC(=O)C(C2CCOCC2)O)CO)c[nH]c(=N)c2[nH]ccc12 Cc1sc(NC(c2cnc(NCCc3c(Cl)ccc(Cl)c3Cl)s2)=O)cc1[N+](=O)[O-] O=C(C1=CNC2=NCCCN12)N1CC2CCN(C(C3CC34CC4)=O)C(C2)C1 c12ccc(cc1)s2.N#CC(C(=O)NCC1CCN(S(C)(=O)=O)C1)C1CC1 c1(C(=O)NCC2N(CCC)CC2)sc(Cl)nc1C N1(CC(=O)NC)CCCC2(CCN(C(=O)C3CCCc4c3ncn4C)C2)C1 C(=O)(CCC(C)(C)NC(=O)COCCN(C)C)NCC(C)(C(N)=O)OC N1(C(c2ccc(O)cc2Br)=O)CCCC2(C1)CN(C(c1cc(O)no1)=O)C2 CCCCC(CC)CC(=O)NC1CC(CC(=O)NCCOCC)C1(C)C N1(CC=C)CCC(C(C)(C)CNC(=O)C(c2ccc(F)cc2)C)CC1 C(=O)(CCCC(=O)N(C1CN(C(C2CC(F)(CO)C2)=O)CC12CC2)C)OCC C1(CCC(=O)N(C)Cc2snc(C)n2)CCCCN(C(=O)C(C)c2ccsc2)C1 N1(C(C2N(CC)CC2)=O)CCC2CN(C(c3cc(C)cnc3F)=O)CC2CC1 CN1CCC2(CC1)CC2CNC(c1ccc(C(F)F)nc1)=O Cc1ccnc2c(C(N3CCC4(CCN(C(=O)C(C)(C)C)CC4)C3)=O)cccc12 N1(C(CC2C(SCC)C2)=O)CCN(C(C2CCSC2)=O)C(C2CCC2)C1 c1(OC)noc(C)c1C(=O)NCC1(F)CN(C(C2CN(C)CC2C)=O)C1 C1(N(C)C)CCCN(N(C)C2CN(c3ccccc3)CC23CCC3)C1 N1(C(CC(C=C)C)=O)CCC2(CC1)CN(C(=O)CCc1cc(Cl)no1)C2C(C)C Cc1ccnc(N2CCCC2c2cnc[nH]2)c1-c1ccc(CO)cc1 C(=O)(CC(CC)NC(c1ccn(COC)n1)=O)N(CC#C)Cc1ccco1 c1(C(C(=O)NC(CC)CNC(=O)CCc2cccs2)C)ccc(OC)cc1C c1(C(=O)NC2CC(CNC(C(C)(C)OC(C)=O)=O)C2)n[nH]c(C)c1Cl CC(CC(N)=O)C(=O)N1CCC(CCN(C)C(c2ncncc2N)=O)CC1 C1(C(=O)Nc2c(OCC)nccc2)CCC2(COC2)N(C(=O)OC(C)(C)C)C1 c1(COC)ccnc(C(=O)N(C2CCN(C(=O)C(C)SC3CCCCC3)C2)C)c1 c1(CC(C(=O)O)NC(CC2CCC(C)C2)=O)cc(F)ncc1Br C(=O)(CCCC(C)C)NC(c1c(OC)cccc1)C(C)NC(c1ccoc1)=O N1(C(C(C)(F)F)=O)CCCC(N(CCO)C(C2CCN(S(C)(=O)=O)CC2)=O)C1 N1(C(CCCCCC)=O)CCc2nc(CNC(=O)C(CC(C)C)C(C)C)sc2C1 c1(C(=O)NC2CN(C(COCCC#C)=O)C(C)C2)cc(Cl)c2ccccc2c1O N1(C(c2c(C)cc(C)[nH]2)=O)CC2CC(NC(c3ccc4c(c3)CCC4)=O)C(C2)C1 c1(C(N(C2CCN(C(c3cc(C)[nH]c3C)=O)C2)CC)=O)cc(C)n(C)n1 C1(NC(CCc2n(C)ccn2)=O)CC(C(=O)NCc2ccnnc2O)C12CCC2 C1(=CCNC(Cc2cc(C)on2)=O)CCN(C(C2(CC(C)C)CCNC2=O)=O)CC1 Cc1cccc(C(O)C(=O)NCCOCCOCCNC(C2CC2(F)Cl)=O)c1F CC(CC(=O)NCCC1(CNC(C2CC(=O)NC(=O)N2)=O)CC1)C(F)F C12CCN(CC1)C(=O)C2N1CCC1Cc1cncn1C.N1(CC)CCC1C(=O)OC C(=O)(C1=CCCCC1C)NC1CN(C(C(COC)C)=O)CC(C)C1 N1(C(Cc2cc(C)no2)=O)CC(N(C(=O)Cc2c(C)n[nH]c2C)C)C2(CC2)C1 C1(CC(=O)OC)CCCN(C(c2cn(C)nn2)C(=O)NC2CCOC(C)C2)C1 C1(NC(C2CCC(=C)CC2)=O)CC2CC(NC(=O)CC(O)CN(C)C)C1C2 c1(OC)nc2ccccc2c(=NCC2CC2CN2C3CCC2c2ccccc23)[nH]1 CC(C(=O)N1CCC1CNC(c1ccc(C(N)=O)o1)=O)C(C)(C)C C(CC(C(=O)NCCNCCN=[N+]=[N-])NC(=O)C(C)CC1CCC1)SC C1(N(C(Cc2c(C)occ2)=O)C)CCN(C(=O)C(F)=CCCF)CC1C c1(OC)ccc(C(N2CC3CC(NC(=O)C(C)C4CCC4)C2C3)=O)cc1O CN1CCCC(C)(C)C1CNC(=N)N1CCC1 O=S(=O)(c1[nH]c(=NCC23CCCC(CO2)C3)ccc1Br)NCC12CCCC1C2 C1(C(=O)NCCC(=C)CNC(=O)CCCOC)CN2CCN1CC2C C1(NC(C=C(C)C2CC2)=O)CCCC(CNC(=O)C=CC2CCOCC2)C1 CC1(O)CCCC(CC(N2CCCC2c2ccccc2Br)=O)C1 c1(C(=O)NCC2(C)CCN(C(c3c(CC)[nH]cc3)=O)CC2)cc(F)c(F)cc1N Cc1nc2ccc(C(=O)NC3CCC4CN(Cc5cncs5)CC4C3)cc2n1C Cc1c(C(=O)N(CCCCN(C)C(C2CCCOC2)=O)C)sc2cncn12 Cc1ccncc1C(=O)N(C1CCCN(C(=O)Cc2ccoc2)C1)C c1(OC)ccccc1C1(C(=O)NCC(C)NC(=O)CC2CCC(C)(C)C2)CC1 C(=O)(C(O)CC(C)(C)C)NCC(CC)NC(c1nc(CC)oc1C)=O N1(C(CC=CC=C)=O)CCN(C(c2[nH]cc(C)c2C)=O)C(c2ccc(F)cc2)C1 C(C(C)(CC)CC)(c1n(CCOCC)nnn1)NCC1(C(=O)NC)CC=CCC1 c1(SSC)c(F)cc(C(=O)O)cc1F.C1(C2CC2)(C)CCCN1OC c1(C(N2CC(NC(C(C=C=C)C)=O)C(F)C2)=O)ccc(Cl)c(OC)c1F C1(C(=O)NC(C2CN(C(C(C3CC3)SC)=O)C2)C)CCN(C(N)=O)CC1 C12(NC(CC=C)=O)CN(C(c3cccnc3)=O)C(COC)(C1)C2 Cn1nc([N+](=O)[O-])cc1C(N1CCC2CCCC12CNC(c1ccc(F)o1)=O)=O C1(C(=O)NC2C(CC)CN(C(C3(F)CCOC3)=O)CC2)Cc2ccc(C)cc2S1 N1(C(CC2CC(OC)C2)=O)CCSCC1C(=O)NC1CC1(C)C c1(NC(CCN(C(=O)C2=C(C)CCOC2)CC=C)=O)cc(C#N)ccc1F C(C(CC(F)(F)F)NC(c1cccc(C(F)F)n1)=O)NC(c1ccccn1)=O c1(C(=O)NC2(C3CCCN3C(=O)CC3CCOC3)CC2)nc[nH]c2ncnc1-2 N1(C(C(C2CCC(=O)N2)C)=O)CC2(C1)CN(C(=O)CCc1nc(O)n[nH]1)C2 C(C1=CCCN(C(=O)Cc2ccc(OC)cc2)C1)NC(CC=CC=C)=O C1(C(=O)NC)(NC(C2CN(C(C(CC)(C)C)=O)CC2F)=O)CCC(C)(C)CC1 O(N=C1CCCCCC1)CC(N1C2CC(NC(c3ccc(OC)nn3)=O)(C2)C1)=O C(CC(=O)N1CCC(NC(c2cccc(N)c2O)=O)CC1C)(C(F)(F)F)OC c1(CC)cc(C(=O)NCC2COCC2NC(C2(OC)CCSC2)=O)cc(O)n1 C(=O)(C1CCc2cc(Br)ccc21)NC1C(CNC(c2cn(CC)nn2)=O)CC1 C(C(C)(O)CC(=O)N1CC2C(CNC(C34CC5CC3C4C5)=O)C2C1)OC c1(CNC(C2CSCCN2)=O)cccc(F)c1Br C1(C(=O)NCCCN(C(=O)CN2CCCCCCC2=O)C)OC(C)(C)OC1(C)C C(c1ccc2c(c1)OC(F)(F)O2)=CC(=O)OCC(c1c(Cl)ccc(Br)c1Cl)=O c1(C(=O)NCC(C(C)C)NC(CC(c2ccc(C)cc2)C)=O)cc(Cl)ccc1F C1(CC(=O)NC(c2cscn2)=O)CCN(Cc2ccccc2F)CC1 c1(C(N(C2CCN(C(C=C(CCC)C)=O)C2)C)=O)cc(=O)n(C)cn1 C1(C(N2CC(O)(C(C)NC(C(C3CC3)OCC)=O)C2)=O)CCC(=C(F)F)CC1 c1(C(C(=O)NC)(F)F)ccccc1C.N12CCC(C1)NS(=O)(=O)CC2 C(N=c1ccnc(N(C)Cc2cc(OC)ncc2F)[nH]1)C1CC(CC)(CC)C1 CN1CCC(C(=O)NC2CC3CC3C2)CC1.C12CCC1C(=O)N2CCO C12(C(N(CCCCCNC(C(C)Cc3ccccn3)=O)C)=O)C=CC(CC1)C2 Cc1c(Br)sc(C(N2CCC2CNC(c2cc3sccc3[nH]2)=O)=O)c1C C1(CNC(CN(C2CCSC2)C)=O)COCCN1C(=O)Cc1cncc(F)c1 C12(NC(=O)CC3CC4(CC4)CO3)CCCC1N(C(=O)CCn1cccc1)CCC2 c1(C(N2CC(O)(C(C)NC(C3CCC3(F)F)=O)C2)=O)cccc(C(F)F)c1F C(CC)(CC)(CCNC(C1(CF)CC1)=O)NC(C1CC(O)(CC#C)C1)=O c1(C(N2CC(Cc3cn(CCCO)nn3)C2)=O)cc(Br)ccc1N1CCOCC1 N1(CC)N=C(C(=O)NC2(C3CC3)CCN(C(=O)CCc3cc(Cl)no3)C2)CCC1=O c1(C(=O)NC2CC2NC(=O)CSc2ccccc2)ccnc(O)c1Br C(CCCNC(=O)C(C)N(C)C)(c1ccccc1)NC(C1C(COC)C1)=O N1(C(C=CC(C)(C)C)=O)CCC2CCCC12CNC(c1ncc(C(F)F)s1)=O C1(C#N)(C(N2CC(C(C)(C)O)(CNC(CCNC(COC)=O)=O)C2)=O)CC(C)C1 c1(C(=O)NCCN(CC(=O)NCCCC)C(C)C)cc(C(C)(C)C)nn1C Cc1oc(C#N)cc1C(=O)NCC(C)C(=O)NC1(C)CS(=O)(=O)C1 c1(CNC(=O)NC(CC(=O)OCC)C)ccc(OC)cc1 C1(C)(CNC(c2n(CCC3(C)CC3)nnn2)c2ccns2)C=CCCC1 CC1(CNC(C2CCCN2C(=O)CCc2cc[nH]n2)=O)CCCCCC1 c1(C(=O)NCC(CO)NC(C(C)Cc2ccccc2F)=O)cc2cccnc2o1 C(=O)(C1=CCCOCC1)NC1CCN(C(c2n(CC#N)ncc2)=O)CC1O CCCCCC(=O)N(C1CCN(C(=O)CC2OCCC2C)CC1)C C1(C(N(C)CC2(Br)CC2)=O)CCCCC1CNC(=O)CN1CCSCC1 C1(C(N2CC(O)CCC(NC(=O)CC3(C4CC4)CC3)C2)=O)CC2C=CC1C21CC1 C1(C(=O)NCc2c(C(N(CC(N)=O)CC)=O)nco2)CCC(C2CC2)C1 C1(C(=O)NCC(CCC)NC(=O)C(C)(C)O)CCCC(F)(F)C1 C(c1cccc(N)c1)=CC(N1CCC(C)(NC(C(C2CC2)SC)=O)C1)=O C12(C(N(C3CCN(C(c4cnccn4)=O)C3)CCCOC)=O)CC(C1)C(C)O2 C1(NC(CC2C(C)(C)C2)=O)C2CC3C(C2)C13C(=O)N1CC(O)CO1 CC1(C)CC(C(=O)NCCOCCC(=O)NCC2CC3CCCC3C2)CCO1 c1(C(=O)NCC(CC=C)NC(=O)CCC2CC(C)(C)CO2)ncc(N(C)C)cn1 c1(C(=O)NCC2C(NC(C=C(CCC)C)=O)C2)cc(C)nc2[nH]nc(O)c12 CN1Cc2c(-c3nc(COc4ccc(F)c(F)c4)no3)cccc2NC1=O N1(C(C2N(C(C(CCOC)OC)=O)CCC2O)=O)CC2(CCOCC2)C1 N1(C(CC2COCC(C)O2)=O)CC2CCN(C(=O)C3=NNC(=O)CC3)C2C1 c1(OC)c(Br)cc(CN2CCCC(C(=O)NCc3ccc(O)nc3)C2)cc1Br O=C(CCC(=O)N1CCCC1C1CCCCCC1)c1ccncc1 CC1(C(=O)NCCC2CCC2)C=CCCC1.N12CC3CC1C3C2=O C(=O)(CC(C)CC(F)(F)F)N1CCCC(C)(NC(c2ccc(C(C)C)cn2)=O)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)CC2C(C)(C)C2(C)C)noc2ncccc12 N1(C(C2(c3ccc(OC)cc3)CCC2)=O)CC2CC(CO)CC(C1)C2O c1(C(=O)NC2(C)CN(C(C3CC=C(C)CC3)=O)C2)cc2n(n1)C(C)CCC2 C1(C(=O)NCC2(C(=O)NC)CCC2)CN(C(C2CN(C)C2)=O)CCC1O C1(NC(C(=O)NCC(CCSCC)N)=O)CCC(C)(C)CC1CN N#CC1(F)CN(C(C2N(C(C3C4CCC(F)C34)=O)CC23CC3)=O)C1 c1(C(=O)NC2CCCN(C(C3CC34CCSCC4)=O)CC2)scc2c1CCCC2 C1(NC(C2CCC(C(C)C)CC2)=O)CCCCN(C(C2(F)CCOCC2)=O)C1 C1(C)(CNC(c2c(C)onc2)=O)CCN(C(C2CCC(CC(C)C)CC2)=O)C1 N1(C(C2CCN(SCCCOC)CC2)C(=O)NCC)CCCCC1c1ccon1 c1(NC(C2N(Cc3ccc(C)c(Cl)c3)CC(C)C2)=O)cccc([N+](=O)[O-])c1Br C1(CNC(C(C)NC(CC)=O)=O)(CO)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C1 C=CCC(C)(C)CC(=O)NC1CCN(C(c2cc(C)cc(Br)c2)=O)CC1F N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CC1CN2C(=O)CC(=O)c1ccco1 CC1(C)CCCC(C(C2(C)OCCO2)O)O1.C1(C(=O)O)CCC(CC)CC1 c1(C2C(C(=O)NC3(CC(=O)NC4CN(C)C4)CCC3)C2)ccc(Cl)c(C#N)c1 C1(CNC(=O)CC2CCSCC2)C2CCC1(c1cccs1)C2.C12CCN1C2=O c1(OC)c[nH]c(C(N2CCCC2N(CC(F)(F)F)C)C(=O)NCCCF)cc1=O N1(C(C2CCCN2C(=O)C(F)Cl)=O)CCOC2(CCC2)C1.c12cccc(c1)NC2=O C(=O)(C(O)CCC(C)C)N1CCC(N(C(c2nc(OC)c(F)cn2)=O)CCO)C1 CCCC(CC)CCC(=O)N1CCC(OC2CN(CC3CC3[N+](=O)[O-])C2)CC1 n1(C(C)C)ccc(C(N2CCC(Cc3cn(CC(=O)O)nn3)C2)=O)n1 c1(NC(=O)NC2CCC(NC(Cc3ccc(C)cc3)=O)C2)cc(C)c(O)cn1 C(N(O)C(=O)Cc1cccc(Cl)c1)c1cn(C(C)C(=O)N(C)C)nn1 N1(C(C2N(C(C3N(C)C(=O)CCC3)=O)CC(O)C2)=O)CC2C=CCC(C2)C1 CC1(CC(N2CC(CNC(c3cn(C(F)(F)F)cn3)=O)C(O)C2)=O)CCCCC1 C1(OC)CCCC(NC(c2nc(C(c3ccccc3)(F)F)no2)C)C1 CC12CCC(C(=O)NC(CNC(=O)C=C3CCC3)CO)(CC1)CO2 N1(C(CCN(CCOCCOC)C)=O)CC(NC(=O)C(F)(F)CO)C(C)C1 C1(C2CC2)(NC(CC(C=C)C)=O)CCN(C(c2noc3c2CCCC3)=O)C1 CC1(C)CCC(C(=O)Nc2cnn(CCO)c2)(NC(C2CCC3(CCC3)O2)=O)C1 Cc1ccnn1C(C)C(=O)NC(C1(O)COC1)C c1(C(=O)OC)ccc(NC23CC(C2)N(C(=O)C(C)(C)N(C)C)C3)cc1OC C1(CNC(c2c(OC)c[nH]n2)=O)CCCC2(CN(C(=O)C(F)C(F)(F)F)C2)O1 C=C1CCN(C(c2cc(C(C)C)no2)=O)C(C(=O)NCC2C=CCCC2)C1 c1(Cc2nc(-c3nccc(OC)c3)nn2C)onc2ccccc12 C1(C(C)C)CN(C(N)=O)CCN1C(=O)C(Cc1ccc(O)cc1)NC(N)=O CC1(C)CC(CC(=O)NCCCNC(c2cccc(C(C)(C)C)c2)=O)NC1=O C1(CNC(C(C(C)C)NC(COC)=O)=O)COCCN(C(c2cc(C)c[nH]2)=O)C1 N1(CC=C)CCC(NC(=O)NC(C)CC(C)c2ccco2)CC1 C1(NC(c2ccc(-c3ccco3)o2)=O)CCCN(C(C23CC(O)C2C3)=O)CC1 c1(C(N(C2CN(C(Cc3cc(C)[nH]n3)=O)CC2F)C)=O)cc2nccn2c(O)n1 C(=O)(CCCc1sccc1C)NC1(CN(C(=O)CC2(CO)CC2)CCC)CC1 C12(CNC(CC(CC)CC)=O)CCCC1N(C(=O)C=C1CCCCC1)CCC2 C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NC(C)CCNC(c1ccccn1)=O CC(C)S(=O)(=O)C(C)C(=O)N1CCC2(C1)CN(C(c1cc(Cl)c(F)c(Cl)c1)=O)C2 Cc1cccc(C)c1C(=O)NC1CC1C(=O)OC(=O)C(C)N(C)C CCC(C(=O)NC(c1ccccn1)C)N(C(=O)Cc1cnsc1)C C(CCCC(=O)NCc1ocnc1C(N1CCOC(C(N)=O)C1)=O)OCC C1(NC(c2c(OC)cc(C)cn2)=O)CC2CC1CN(C(C1CCC(C)C1)=O)C2 C1(C(=O)NC2CCN(C(CC3(C=C)CCC3)=O)CC2F)C2CCCCCCC12 c1(CCC)nc(C)c(C(=O)NCC2CC(NC(=O)C(F)(F)CC3CCCO3)C2)s1 c1(NC)ccc(C(N)=O)cc1C(=O)NCC(C)NC(C1CC=CCC1)=O c1(CC)nc(C)oc1C(=O)NC12CC1CN(C(c1csc(O)n1)=O)C2 C(=O)(CCC(F)(F)F)N1C(C(=O)NC(COC)C2(C)CC2)CCC1 C(=O)(CCCC(CC)NC(c1c(C)ncnc1C)=O)NCC(CCC=C)O C1(O)(CCNC(=O)COC2CC=CC2)CCN(C(C2CC3CCC3C2)=O)C1 C1(C(N(C2CCN(C(=O)CCc3cnccn3)CC2)C)=O)CC(=O)N(C2CC2)C1 c1(C(=O)NC2CC(CNC(CSc3n(C)nnc3)=O)C2)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC(C)CCNC(=O)C(c2cccc(F)c2)C)cnc2n(c1=O)CCS2 c1(C(=O)NCCC(=C)CNC(c2n[nH]cc2F)=O)cncc2[nH]ccc12 C=CCCCC(C(=O)NCC(C)C(F)(F)F)NC(C1COCOC1)=O c1(CNCC2(C(=O)Nc3ccc(C#C)cc3)CC2)n[nH]c2ccc(Br)cc12 c1(CC(N2C(CNC(CC=C)=O)C=CC2)=O)ccc(F)c(Br)c1 c1(NC(C)CNC(=O)C(C2(O)CCCCC2)(F)F)nc(O)n(C)c(=O)c1[N+](=O)[O-] c1(C(C(=O)OCC)N(c2ccccc2)C(C)=O)cccc(Cl)c1 C(c1ccc(OC)c(F)c1)=CC(=O)NC(C(=O)OC)Cc1cn(C(C)(C)C)nn1 CC1=C(C(=O)N2CCCOC(CNC(c3nc(C)nn3C)=O)C2)CCO1 N(C1CCc2cc(CNC(c3cc(CO)on3)=O)ccc21)C(c1cn(C)nn1)=O N1(C(CC(=O)N(C)C)=O)Cc2ccccc2C1CNC(=O)CCC(C)(C)F c1(SC)c(C(=O)N(CCCNC(c2cnc(NCC3CC3)s2)=O)C)csc1C C(C)(C(=O)NCCCCO)N(CCC)C(C1CCO1)=O C1(NC(C(CSC)c2ccccc2)=O)CCCCC1NC(=O)C=Cc1cncn1C C1(NC(Cn2ncc(CC)c2)=O)CCC(C)(C)CC1CNC(c1nnsc1C)=O C(=O)(C1CCCCc2ccccc21)NC1CC(CNC(=O)C2=CCOC2)C1 C12(CNC(C(C)(C)CF)=O)CCC(C1)N(C(=O)C(F)CC1CCC1)C2 CC(=O)C(C)CC(C)C(=O)N1CC(NC(c2ccc(O)nc2)=O)CC12CCC2 C1(CNC(C(CCOC)C)=O)CCCCN(C(c2cc(C3CCC3)no2)=O)C1 c1(OC)ccc(-c2n[nH]cc2C(=O)N(C(C)CNC(=O)C(CO)N(C)C)C)cc1 c1(NC(=O)C(C2CCCCC2)F)nc(C(N(c2ccccc2)CC#C)=O)oc1C C(N=c1ccc2ncc[nH]c-2n1)C1(C)CCN(C(C2CC(F)(CO)C2)=O)C1 C1CCCCCNC(=O)CC(=O)N1CC.C1(C(=O)NC)CCOC(C(C)C)C1 Cc1nc(CC(=O)NC(C2CN(C(c3ccc(C4CCCCC4)[nH]3)=O)C2)C)cs1 c12nocc1C(=O)NC2C.C(CC(C1CC1)C1CC1)NC(C1C(CC)C1)=O C1(NC(C(=O)NCC2CC2)=O)CCCC2CN(C(c3nccc(Cl)c3F)=O)CC12 N1(C(c2c(CC)nc[nH]2)=O)CCN(C(=O)CC2=CCN(C)CC2)C(C)CC1C CC1(C)CC(NC(c2cccc(Cl)c2F)=O)CN1C(C1CCC(=O)C1)=O CCS(=O)(=O)CC(=O)NCC(CC#N)C(=O)NC(CF)C(F)(F)F c1(CNC(C2(NC(c3n[nH]c(C)c3Cl)=O)CCOCC2)=O)ccnc(F)c1F C(=O)(C(C)CC(N)=O)N(C(c1ccccc1)CNC(CC1(C(=C)F)CCC1)=O)C CC1CN(C(c2ccnc(N(C)CCOCCO)c2)=O)CCC1CO C(C(F)(F)CCNS(=O)(=O)CC1(C(=O)OC)CCC1)n1cc(C(C=C)(C)O)nn1 N1(C(C(C)N(C(Cn2ccc(C)n2)=O)C2CC2)=O)CCCN(C)CC1 c1(C(=O)NC(CC)CC(=O)NC(c2ncn(C)n2)C)ccnc2cc[nH]c12 Cc1n[nH]c(=NCC(C)(C(C)C)NC(=O)CC2CCNC2=O)s1 c1(C(N2CC=CC(C(N(CCSC)CC)=O)C2)=O)cnn2cccc2c1 CC1CN(Cc2ccccc2)CC(C)N(C(c2ccc3ocnc3c2)=O)C1 C1(NC(C2(c3ccn(C)c3)CC2)=O)COCCN(C(=O)Cc2ccsc2)C1 CC1CC(NC(c2cc(Br)c[nH]2)=O)CCN1C(c1ncccc1Cl)=O CC1=NN(C)C(=O)C1CC(N1CCCN(CCNC(=O)CN(C)CCO)CC1)=O C(=O)(CCCCC(=O)NC1CC(F)(CNC(C2CCc3cnnn3C2)=O)C1)OC C12(C(=O)NC3CC(C)N(C(=O)C(=O)Nc4ccccc4O)C3)CC3CC1C2C3O CC1(C(=O)NCC2(F)CCC(CNC(=O)C3=NOCC3)C2)CCC(O)CC1 c1(C(N2C(=O)C2)=O)cnc2c(Br)n[nH]c2c1.c1(C(C)(C)C)cnc(C2CCC2)o1 C(=O)(C(O)CC(C)(C)C)N1CCN(CC2CN(C(CCC(=C)Cl)=O)C2)CC1 C(=O)(CCCC(=O)N(C)C)NC(C(=O)NCC1(O)C(C)CCC1)Cn1ccnn1 c1(OCCC(=O)NC(C)C=CC(=O)N(C)CCO)ccc(F)cc1Cl Cc1cc(CNc2ccc(-c3ccc(N(C)C)nc3)cn2)cc(C#N)c1 c1(OC)cnc(F)c(C(=O)NCC(n2cc(-c3cnccc3Cl)nn2)C)c1 C1(NC(CNC(C(CC)CC)=O)=O)CCN(C(=O)C(=O)C(C)(C)C)C(C2CC2)C1 C1(C(C(=O)N(CCCN(C(Cc2c(C)n[nH]c2)=O)C)C)(C)C)CCCN(C)C1 C1(CC)C(NC(c2cccnc2C)=O)CCCN1C(=O)CN1CCC(OC)C1 C1(C(N2C(COC)C=CC2)=O)CC2CC2N1C(=O)C(n1ccnc1C)C c1(N2CC(NC(CCN(C)CC)=O)CC3(C2)CC3)nc(CC)nc2c(C)csc12 C1(NC(c2c(CC)cccc2)=O)CC2CCC(C1)N2C(C1(Br)C(C)C1C)=O N1(C(C(C)CCO)=O)CCN(C(=O)Cc2csc(NC=O)n2)CC(O)C1 C1(C(=O)N(CCCCN(C(=O)Cc2c[nH]nc2O)C)C)(OC)CC(C)CC(C)C1 Cc1cn2c(C(=O)NCC3(NC(c4cc(O)nc(C)n4)=O)CC3)c(Cl)nc2s1 C(=O)(C(C)CCO)NCC(CN(C(c1cc(COC)on1)=O)CC)(C)C c1(C(=O)NCC(C)NC(C2COC3(C)CC2C3)=O)cccc(C(F)(F)F)c1O C1(CC(=O)NC(CN(C(c2ccoc2CC(N)=O)=O)CC)C)CCCS(=O)(=O)C1 C1(CCNC(C2CC(OC(F)F)C2)=O)CCN(C(=O)CSC2CCCCO2)C1 C1(C(=O)NCC(C)CNC(C2(C)CC2C(F)(F)F)=O)CS(=O)(=O)CC(=O)N1 C1(NC(c2ccc(C)c(O)c2)=O)CN(C(=O)C(O)C2CCC2)C2(CCOCC2)C1 S(=O)(=O)(c1c[nH]ccc1=NCC1CCOC1C)N(CCCSC)C N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCC(NC(=O)CC(C)N(C)C)C1(C)C C1(NC(C2(Oc3ccccc3F)CC2)=O)C2CN(C(c3ccccc3)=O)CC12 N1(C(CCSC)=O)CCC(NC(C2CN(C)CC(C)O2)=O)CC1C CC(C(=O)NNc1ccc(Br)nn1)c1c(F)cccc1Cl c1(-c2onc(CC(c3ccc(CC4CC4)cn3)=O)n2)ccc(OC(F)F)cc1Cl C1(C(c2cn(Cc3c(C(=O)O)cco3)nn2)O)CCN(C(C2(Br)CC2)=O)CC1 C1(NC(c2ccc(SC)cc2)=O)CN(Cc2cccnc2)CCC1(F)F N1(C(C(C)OCCOC)=O)CCC(C)(Cn2cc(COC(C)C)nn2)CC1 C1(O)(CCC(=O)NCC=CCNC(C2C(C)(C)C2N2CCC2)=O)CCCOC1 CN1CCN(C(=O)C(CNC(C2OC3CCC2C3)=O)N(C)C)CC1CO c1(C(=O)NC2C3CN(C(CC=C(C)C)=O)C2C3)cc(S(N)(=O)=O)c(Cl)cc1Cl c1(CNC(C2C(C)C2)=O)ccc(CNC(=O)C(C)CC2CCCC2)cc1 C#Cc1ccc(C(N2CCCC(NC(=O)C(C)N(C)C)C2C)=O)cc1 CCCCC(CNC(=O)C(C)CCOC)NC(c1onc(CC)c1C)=O C1(C(N(C2CCN(C(C(c3cn(CC)nc3)(F)F)=O)C2)C)=O)CCCS1(=O)=O N1(c2nnc(-c3c[nH]c(Br)c3)n2CCC2CCOC2)CCNCC1.CSC CCC(CC(F)F)C(=O)N1CC(CNC(c2cnoc2CC(C)C)=O)CC1(C)C N1(C(C(C)OCCOCC)=O)CC2(C1)CN(C(=O)C(C)OC1CC1)C2 c1(-c2c(NC(C(C)S)=O)c3c(nc2)cccc3)cccc2c([N+](=O)[O-])cccc12 C1(C(=O)NCC2N(C(C3(F)CC3)=O)CCC2)CC12CCOc1ccccc12 c1(OC)cc2ccc(Cc3ccc(C#N)cc3)cc2cc1OC c1(C(=O)Nc2ccc(-c3cnn[nH]3)cc2)ccc(O)cc1Cl c1(OC)cccc(COCC(=O)NC2CCN(C(=O)CCC(C)SC)C2C)c1 c1(CNC(=NC)NC2CCC(C(F)F)CC2)ccc(F)c(OC)c1F.C1(=O)CO1 c1(C(N2CC(OC)CC(NC(C(C=C)(C)C)=O)C2)=O)ccc2nn[nH]c2c1 N1(c2c(Br)cn(C(C)C)n2)C(=O)C2c3ccccc3OCCN2C1=O CC(C)(C)CS(=O)(=O)NCCc1c(Cl)cccc1Cl C1(C(=O)NC(C)CNC(=O)Cc2nnco2)CCCC12OCCO2 N1(CCNC(Cc2cc(C)no2)=O)CCN(C(C2CCCC23CC3)=O)CC1 c1(C(=O)NCC(CN(C(C)=O)C)O)n[nH]c2ccc(Cl)cc12 c1(CC)ccc(C(N2CCC(NC(c3cc(COC)no3)=O)C2(C)C)=O)cc1F N1(C(C2CC3(ON=C(C)C3)C2)=O)CCCCC2(C1)CN(C(=O)CSCCC#N)C2 NS(=O)(=O)c1cc(C(=O)NCCOC2CCN(C(C3CNC(=O)N3)=O)C2)c(Cl)o1 C1(C(=O)NC(C2(C(=O)OC3CC3)CC2)C)C(C(C23CCC(C2)C3)=O)C1(C)C CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(C2COCCO2)=O)C2CC12 c1(C(N2CC(C(C)NC(c3c(C(C)C)nns3)=O)C2)=O)cc2ccsc2[nH]1 Cc1ccc(C=CC(=O)NCC(C)CNC(=O)CC2CCCS(=O)(=O)C2)cn1 N1(C(c2cnc(C)nc2C)=O)CCCC2(NC(c3cnc(C)[nH]3)=O)CCCC12 Cc1ccc(N)cc1OCC(N1CCC1CNC(=O)C(c1ccc(Cl)s1)C)=O N1(C(C2(OC)CCC2)=O)C(C(=O)NC2CCC3CCC23)CCC12CC2 N(C1CCc2c(Cl)cccc21)C(c1c2ncc(C(N)=O)c(N)n2nc1)=O C1(C(=O)NCCC2CCN(C(C3CC(C(=O)OC)C3)=O)C2)CCC(C)(C)OC1 c1(N(CC(C)C(F)(F)F)C)ccc(S(=O)(=O)NC2CC2C2CCOCC2)c(Br)c1 C=CC1(C(=O)NCC2(OC)CN(C(=O)CC(C)(O)COC)C2)CCCCC1 c1(NC(C)=O)ccc(C(=O)NC(C)CNC(C2(C#N)CC(C)C2)=O)c(Cl)c1 C1(C2(NC(Cc3ncc(C)s3)=O)CC2)CCCCN1C(C1C2CCCC12)=O N1(S(CC(=O)OCC)(=O)=O)CCCC2(CCN(C(c3ccc(S)cc3)=O)C2)C1 c1(NCCCC(N)=O)nc(N2CCSCC2)nc2scnc12 C1(NC(CCC2(C)CC2)=O)CC2CCC1N2C(=O)Cc1ccc(OCC#N)cc1 C(=O)(CCCS(C)(=O)=O)NCC(c1ccccc1)CNC(CC(CC)SC)=O CC(C)C(C(=O)NC1CN(C(=O)C(C)C2CCC2)CC1C)NC(c1cccs1)=O N1(CC(C)(C)NC(CCCOCC)=O)CCN(C(c2ccc(F)cn2)=O)CC1 CCC(C)(C(=O)NC(C)CCCCNC(=O)CCc1ccc(O)nn1)OC N1(C(c2c(C)n(C)cn2)=O)CC2CN(C(C3CC3c3ccncc3)=O)CC2(C)C1 c1(C(=O)NCCSc2ccc(C)cc2)c[nH]c2ccccc2c1=N c1(OC)cc(Cl)c(C)cc1C(=O)COC(=O)C(F)(F)CC(C)C c1(CCNC(C2(OC)CCCCCC2)=O)c[nH]c2cc(C(C)C)ccc12 CC1CN(C(=O)CC(F)(F)F)CCN1C(C1CC(O)C(F)C1)=O N1(C(c2cc(C#N)sc2)=O)CCCC2(CCCN2C(c2ccc(Cl)nc2O)=O)C1 N1(C(Cc2cc(C)nn2C)=O)CC(C2CN(C(c3cc(F)c(F)cc3Cl)=O)C2)C1 Cc1cncc(OCC(N2CC(CN(C)C(c3ccn(C(C)(C)C)n3)=O)C2)=O)n1 CCCC(C)(C)C(=O)N1CCC(C)(NC(C2CCC23CCOCC3)=O)C1 CCCC(CCC)CCCC(=O)N1CC(CCNC(=O)CN(C2CCSC2)C)C1 C1(C(=O)OC)CC(=O)CN1C(c1c(O)n[nH]c1-c1ccccc1)=O c1(CCC(=O)NCC(CNC(C2=C(C)OCC2)=O)C)cccc(S(N)(=O)=O)c1 O=C(C1CCCc2nc[nH]c21)NCC1C2CC1N(C(=O)CCC1CCCCO1)C2 CCC(C(=O)OC)C(=O)NC(C)CNC(c1ncc(Br)cc1C(F)F)=O CN1CCc2c(NC(=O)NC3(c4ccncc4)CCC3)cccc2C1=O Cc1ncc(CCNC(=O)C(C2(O)CN(C(C3CC3[N+](=O)[O-])=O)C2)F)[nH]1 C1(CCC(=O)NCC(C2CCCC2)NC(C2(CC)CC2)=O)CCC(=O)N1 C(=O)(C1=CCCOC1)NC(C(C)C)CCN(C)C(c1cnc(C(F)(F)F)cn1)=O c1(N2CCCC(CNC(=O)CC3CCCS3(=O)=O)CC2)c(Br)cccc1[N+](=O)[O-] c1(NCc2cc(C)ns2)cc(NCC(Cl)=CCl)ncn1 c1(-c2cn(C3C(C)CN(C(C4(CCF)CC4)=O)C3)nn2)ccc(F)cc1Cl CC(C)CCN=C(NCc1ccc(Br)o1)NC(C1CCCO1)C C(=O)(C(C)(C)CC(=O)NC(C)CNC(c1ccccc1C(C)(C)C)=O)OCC CCC(C)CCCCC(=O)N1CCC(N(C(=O)CCSC)CCO)C1 CC1(C)C2CCC1(C)C2C(=O)NC1CN(C(c2cc(F)ccc2F)=O)CC1F c1(CC)cc(C(=O)NCC2CCC(C(=O)NCCC(C)(C)F)O2)n[nH]1 O(C=C(C#N)C(=O)N1CC(NC(c2cc(C3CC3)cnc2Cl)=O)C(C)(C)C1)CC C1(C(N2CCCC(c3ccccn3)C2)=O)COc2ccccc2C1 c1(SCC(=O)NCCN(C(=O)C(C)(C)C)CC)nc(C)nc2sc(C)c(C)c12 C1(C(=O)NC2(CN(C(=O)Cn3cccn3)C)CC2)CCC1C(C)(C)C C(C(COC)C(=O)NC1CC2(C1)CC2C(=O)NCC(C)(C)OCCO)OC C1(NC(=O)Nc2c(C)cccc2)CC(F)CN(C(C2CCCS2)=O)C1 c1(C(=O)NC2C(NC(C(C)NS(C)(=O)=O)=O)CCOC2)cn2c(n1)CCC2 C(C)(C(=O)NCCCN(C(=O)CNC(=O)Cn1cncn1)C)=CC Cc1ccc(C(=O)NCC2CN(C(c3cnnn3C(C)C)=O)CCO2)c(C)n1 C#Cc1ccc(C(N2CCC3CC23C(=O)NC(CC2CC2)C(=O)NC)=O)cc1 N1(C(CC(CCC)C)=O)CC2C3CCC(C(NC(c4sccc4C)=O)C3)C2C1 C#CCCCC(=O)N1CCCC1C(N1CC(NC(=O)C2CC2)C1)=O CC1CC(C(=O)NCC2CCN(C(=O)CCc3cn[nH]c3)CC2)Cc2nn[nH]c21 C1(C)(C(=O)NCCC(CC)(C)NC(C2COCCO2)=O)CCCN(C)C1 C1(OC)CCN(C(C2CSCCN2C(C2CCCC(=O)C2)=O)=O)CC1(C)C C1(NC(c2cc(C(F)F)cs2)=O)CCC12CCN(C(=O)C(F)CC1CCC1)CC2 c1(N(CCOCCNC(C)=O)C)nc(N2CCCC(F)C2)c2c(n1)CCC2 c1(OC)cccc(CN2CC3CC(C2)N3C(=O)C2=CCC2)c1Oc1ccccn1 CCC(CC(F)F)C(=O)NCC1(NC(c2ccn(C(C)(C)C)n2)=O)CCOC1 C1(C(N(CCCNC(=O)Cc2cncc(C)c2)CC)=O)CC(C)CC(C)C1 C1(C(N2C(CNC(COCCCCC)=O)CC2)=O)CCCC(F)(F)C1 C1(NC(CC)=O)CC(C2CCN(C(=O)CN(C3CCSC3)C)C2)C1 CC1C(C)N(C(c2cccc(C#N)c2Br)=O)CCN1Cc1ccccc1 c1(CNC(CNC(=O)OC)=O)nc(OC(=O)C(F)C(F)(F)F)cc(O)n1 n1(C(c2nc(CC(C)C)on2)C)cc(Br)cn1 C1(CNC(c2[nH]cc3c2CCC3)=O)CN(C(=O)C(F)(F)CO)CCC1(F)F C1(CNC(N(C)CC2CC2C)=O)C=CCC1 O=C1CCC(CC(=O)NC2CN(C(C3CCS(=O)(=O)N3)=O)C2)CN1 C(=O)(C(O)CCC(C)C)NCC(CC(N1CC(CC)C(F)C1)=O)C1CCC1 C1(OCCC)CCCCC1Cc1nc(-c2cc(C)oc2C)nn1CCC(C)(C)C Cn1cc(-c2nnc(C3CC3F)o2)c(Oc2ccccc2)n1 c1(C(=O)NC2C(NC(Cc3ccc(C)c(Cl)c3)=O)C2)cccc(S(N)(=O)=O)c1C CCCCC(C)(N=c1ccn(C2CC2)[nH]1)c1nnnn1C1CCC1 C1(C(N(C2CCN(C(C3(SC)CCC3)=O)CC2)CC#C)=O)CCC(=O)NC1 Cc1n[nH]c(=NC2=CCCC2)o1.N1(C(C(=O)N2CCC2)C)CCCC(O)C1 C1(NC(=O)NC(C)C(=O)NCc2ccco2)CCNC(=O)C1 c1(C(N(C(CN(C(C(CC=C)N(C)C)=O)C)C)C)=O)cccc2[nH]ccc12 c1(C(N2C(C)CC(NC(c3c(C)c(N)n(C)n3)=O)C2)=O)ccc2cncn2c1C c1(C(=O)NCC2CC(F)CN2C(c2cc(Br)n[nH]2)=O)csc2ccncc12 C1(C(=O)NCCC(C)(C)NC(c2cc(C(C)(C)C)ccn2)=O)CCC2C1C2(F)F C1(CN(CC(=O)NCCC)C)CCN(C(=O)C(CC)SC)CC1 C1(OC)C(NC(C2(CNC(=O)Cn3cncn3)CC=CC2)=O)CC12CCC2 N1(C(CCCOCC)=O)CC2(CCCCN(C(C3(Cl)CC3(F)F)=O)C2)C1 CC(C)(C(=O)N1CCC(NC(c2cnn(C(C)(C)C)c2)=O)C(CO)C1)S(C)(=O)=O C1(NC(C(CC)NC(N)=O)=O)CCC2CCN(C(C3(CO)CCC3)=O)C1C2 C1(C(N(CC)Cc2cnc(Br)cn2)=O)CN(C(=O)OC(C)(C)C)CCS1(=O)=O CC1(C)CC(=O)NC1CNC(C1CCC(CNC(=O)C(Cl)Cl)O1)=O CC1CCCC(CNC(=O)C(=O)NCc2ccsc2)CC1 C1(CN(C(=O)Cc2ccccc2C(F)(F)F)C)CCCCN1C(=O)CC1(C)CC1 C1(NC(CC2N(C(c3c(C)n(C)cn3)=O)CCCC2)=O)CC1C1CCCC1 C1(CC)(CO)CCN(CCC(=O)Nc2cnn(C3CCCCC3)c2C)C1 N1(C(COCCC=C)=O)CCCC(CCC)(NC(c2cccn2C)=O)C1 n1(CC)c(N2CCC(c3ccon3)CC2)nnc1C1CCC1c1ccsc1 C1(NC(C(=O)NCC(c2ccncc2)C)=O)CCCN(Cc2cccc(F)c2)C1 Cc1sc(C)c(C(=O)NCC2(NC(C34CC(F)C3C4)=O)CCOC2)c1C#N C(=O)(C(F)(F)c1cscc1Br)N(C1CN(C(C2(C)CC2(C)C)=O)C1)C C=CC(F)(F)C(=O)NCCCC(C)NC(C1CSCN1C(C)=O)=O Cn1cncc1C(=O)NC1CC(NC(=O)CC2C(C(F)(F)F)C2(F)F)C1 N1(C(C(C)=C(CC)C)=O)CC(OCC)C(NC(=O)CNC(=O)C(C)(C)C)C1 Cc1ccc(C(N2CC3CC3(NC(C3(C4CCCO4)CC3)=O)C2)=O)cc1Cl c1(C(C)=O)ccc(Cl)cc1S(=O)(=O)Nc1cc(C)nc(N2CCOCC2)n1 C(CN=c1cc(C)c(S(=O)(=O)N2CCN(c3ccncn3)CC2)c[nH]1)SC C1(C)(NC(C(CCN(C)C)NC(COCCOCC)=O)=O)CN2CCC1CC2 c1(OCC(C)(C)NC(C(CC)N(C)C)=O)cccc(C)c1.C1(=O)COC(C)N1C c12ccc3c(c1)n(CC(F)(F)F)c(=O)n3C2.CCCCC(C(=O)O)OC c1(C(=O)OCC)ccc(CNC(=O)CC2(C)CCN2C(c2ccsc2C)=O)cc1 N1(C(c2c(C)nc(COC)s2)=O)CCN(C(=O)CC(C)SC)CC1CO N1(C(CSC)=O)CCN(C(C2CCCN(C(C)(C)C)C2=O)=O)CC1C(C)C C1(C)(C(N(C)CC2CC(O)C2)=O)COCCO1.c12cn(nn1)C1CN(C1)C2=O N1(C(C2(C=C)CCN(C(=O)Cn3cccc3)C2)=O)CCCC(C)(C)CC1 C(C(=O)C(=O)NC(COCC)C1CC1)(c1ccco1)NC(=O)OC.C1(=O)C(C)N1 c1(C(=O)NCC(CCCC)NC(=O)C(C(C)C)NC=O)nc(C)c(C)nc1C C1(CCC)CN(C(=O)CCC(=O)NC)CC1NC(=O)COCc1nc(C)no1 CC1CCC(NC(c2cccc(C3CC3)n2)=O)CN1C(C1COC2(CCC2)C1)=O Cc1c(C(N2CCCCCC2c2ccc(Cl)cc2)=O)oc2ccc(F)cc12 C#CCCCCC(=O)NC1(CNC(c2c[nH]nc2CC)=O)CC2CCC1C2 c1(SC(C(=O)NC(CNC(CCCc2onc(C)n2)=O)C)C)ccc(F)cc1 c1(C(N2C(C)CC(CNC(c3cccc(OC)n3)=O)C2)=O)ncc(Cl)cc1Cl C#CC1CCC(C(=O)N(C2CN(C(C3OCCC3C)=O)CC2(C)C)C)CC1 N1(C(c2c(C)[nH]nc2Cl)=O)CC(NC(=O)C(C)NC(c2cccs2)=O)C(C)(C)C1 c1(OC)nccc(Sc2noc(C34CC3CN(C(=O)C(C)CC(N)=O)C4)n2)c1F c1(C(C)C)ccc(C(=O)NCC2CN(C(=O)C(C)OCCN(C)C)CCO2)cc1 C1(CC)(CC)CN(Cc2ccccc2)CCS1(=O)=O.c1(C)nccn1C(F)F C1(CNC(c2c(OC)nsc2)=O)N(C(C2CC2C(C)(C)C)=O)CCCC1(C)C C=CCC(CC(C)C)C(=O)N1CCN(C(=O)COCC=C)CC1C1CCC1 c1(CNC(c2n(C)ccc2)=O)nc(CNC(C2C(C3CC3)C2(F)F)=O)cc(O)n1 Cc1cc(C)c(COC(C2Cc3ccccc3C2)=O)c(C)c1O N1(C(=O)CCC2CCOC2)CC2(CCCCN2C(=O)COC2CCCOC2)C1 Cc1cc(CN(C=O)Cc2ccc(O)c(Br)c2)ccc1N(C)C Cc1ccc(C)c(CC(=O)NC(C2CCCCN2C(=O)C(C)OCC2CC2)C)c1 N1(C(c2ncc(OC)cn2)=O)CCc2sc(CNC(C3CC3C(C)C)=O)nc2C1 c1(C(=O)OC(CC(=O)N(CCN(CC(=O)OC)C)C2CC2)=O)cccn2nncc12 c1(CCC(N2CC(O)(C(C)NC(C3CCCOC3)=O)C2)=O)cccc(N(C)C)n1 c1(C(=O)NCC2(OC)CCN(C(c3cncs3)=O)C2)cc2c(F)cc(F)cc2[nH]1 C=CC(C)(CC)C(=O)NCc1cn(C2CN(C(=O)CSCC(N)=O)C2)nn1 N1(C(CNC(=O)OCC=C)=O)CCC(NC(C2CCCCN2N=O)=O)C(C)C1 c1(C(N(CCOCCNC(C2(COC)CC2(F)F)=O)C)=O)cc(Cl)ccc1OC c1(C(=O)OC)ccc(C)nc1NC1CCN(C(c2cc(C)cs2)=O)C1C CC1CCCCN1S(=O)(=O)N1CCN(C(c2cc3c(Br)c(Cl)ccc3[nH]2)=O)CC1 N1(C(CN(CCC#C)C)=O)CC(NC(C2CCC2C(=O)OCC)=O)CC(C)C1 C#Cc1cccc(C(=O)NCC2CCN2C(=O)Cc2cc(F)ccc2C)c1Cl c1(CNC(C(C)(C2CC2)OC)=O)ccccc1CN(C)C(c1c(C)cnn1C)=O Cc1cnncc1C(=O)NOCC(N1CCOCC1c1ccccc1OC1CC1)=O c1(C(N2C(C)CCN(C(=O)C(F)OC(F)(F)F)CC2)=O)c[nH]c2cc(F)ccc12 Cc1nc2ccccn2c1CC(=O)NCCN(C(=O)C(C)C(C)(F)F)C N1(C(C(C(=O)OC)C)=O)CCC2CCN(C(=O)C(=O)NC(C)C)CC12 c1(C(=O)NC2C(NC(CC(C=C)(C)O)=O)C2)cccc2c1COCC2 c1(CC)cc(C(=O)NC2CC2CNC(c2cc(Br)n[nH]2)=O)c(C)o1 Cc1ccc(-c2nc(C)sc2CC(=O)N(C(C)(C)C)CCOCCO)cc1 c1(C(=O)NCCCC2N(C(C3CC(OC)C3)=O)CCCC2)cc(Cl)c(F)c(Cl)c1 CC1CN(S(=O)(=O)N2CCC(NC(N)=O)CC2)CCO1 C12(C(N(C)CCC3CCN(C(C4(N=[N+]=[N-])CC4)=O)CC3)=O)CCCC(CO1)C2 C1(C2CCC2)(CNC(=O)C=CC2CCOC2)CCN(C(=O)COCCCF)CC1 C12(CN(C(C(c3ccc(N(C)C)cc3)C)=O)CCO)CCCC1OCC2 Cc1nn(CC(N2CC(C)CCC2CNC(=O)CC(C)C)=O)c(C)c1Cl C1(CC(=O)NCC(=O)N(C)C)CCN(S(=O)(=O)CCc2ccno2)CC1 N1(C(Cc2ncc(C)nc2)=O)CCC2CCCC12CNC(=O)C(C)(C)CC#N C1(C(=O)NCCCCCNC(c2cn(CC)nc2C)=O)CCc2[nH]nc(O)c2C1 c1(OC)ccc(CC(=O)NCCn2cc(CCC#N)nn2)cc1O c1(C(=O)NC2CC3(C(C(=O)NC(C(=O)OCC)C)C3)C2)cnc(C)nc1C C1(CN(C(=O)CC2COCC2(C)C)C)C2CN(C(C3CC(F)(F)CS3)=O)CC12 N1(CC)CCC(CCNC(=O)CC2CC(C)=NO2)CC1.C12C=CC(C1)CNC2=O c1(C(=O)NCC2C(C(=O)OC)CCC2)ccc(-c2ncco2)cc1F c1(C(=O)NC(CC)CNC(=O)CCC2CCC(=O)N2)cncc2[nH]ccc12 C(=O)(CCS(C)(=O)=O)NC(C)C(C)NC(=O)C(F)(F)c1ccsc1Cl C(=O)(C(CC(=O)O)n1cc(-c2cn(CC(=O)O)nc2)nn1)NN1CCOC(CO)C1 C1(C(N2CCC(NC(c3cc(C)on3)=O)C(O)C2)=O)CC(O)c2ccccc2O1 c1(NC(C23CC(C(N(CC(C)C)CCC)=O)(C2)C3)=O)c(Cl)c(F)nc(F)c1Cl c1(NC(c2nc(-c3c(C)ccc(OC)c3)sc2C)=O)ccc2scnc2c1 n1(CC(=O)NC2(C)CC(NC(C(C)(C)OC)=O)C2)c(O)nc2ccccc12 C1(C(=O)NCC2CCCN(C)C2)CCN(C(=O)Cc2ccccn2)C12CC2 Cc1nc(Cl)ccc1CC(N1CCN(C(=O)CC2CCCOCC2)C(CO)C1)=O O(NC(=O)C(CC(N)=O)NC(=O)CCCOC)CCOCC#C Cc1cc(C(N2CC(O)(C(F)C(=O)NCC(CC3CC3)CO)C2)=O)ccc1F C1(CC(C)CNC(=O)C#CC2CC2)CCN(C(=O)Cc2ccon2)CC1 c1(NC(=O)CC2CCCN(C(=O)CC3CCOC3=O)C2)cccc(F)c1F CCC(C(=O)NC1CC(CCNC(=O)CCc2cncn2C)C1)OC C12(NC(c3c(Cl)cncc3Cl)=O)CCCC1N(C(=O)CC1CC1)CCC2 c1(C(N2CC(COC)N(C(=O)C=Cc3cccs3)CC2)=O)cc(C)c(Cl)c(C)c1 C1(C(=O)NC2CC(=C)CN2c2cc(O)nc(C)n2)CCc2nc[nH]c2C1 c1(N2CC3(C(NC(C4CC45CC5)=O)CCS3)C2)c(Cl)cncc1[N+](=O)[O-] CC1CN(C(c2cc(Cl)no2)=O)CCCN1C(=O)CCCCC1CC1 N1(C(C2C(C(C)C)N(C(c3cnc(S)nc3)=O)CC2)=O)CC(O)CC1(C)C C(=O)(C(=O)C(F)(F)F)NCCC1CCN(C(C(C)CC2CCC2)=O)CC1 c1(C(=O)NCC2(O)CCN(C(c3c(C)nn[nH]3)=O)CC2)cc(S(N)(=O)=O)oc1C c1(C(=O)NCCN(C(=O)Cn2cnnc2O)CC)cnn(CCC(F)(F)F)c1 C1(C(=O)NC(COC)CNC(C2CC(OC)C(OC)C2)=O)CCn2c(O)nnc2C1 C1(NC(C2C(C)CCC2)=O)CCCC2CN(C(c3cccc(C4CC4)c3)=O)CC12 C12(C(=O)NC3CCN(C(C(c4ccc(F)cc4)CC)=O)C3)CCC(C1)OC2 c1(NC(C(C)(C2CCC2)NC(N)=O)=O)ccc2cccnc2c1 N1(C(c2ccc(OC)c(F)c2)=O)CC(NC(=O)CCC(C)N(C)C)C(C2CC2)C1 C1(C(N2CCC(CNC(c3csc4ccccc34)=O)C2)=O)COCC2(CCC2)O1 C#CC1(O)CCN(C(=O)CC2CC2CNC(=O)C(COC)CC)C1 c1(C(=O)OC)ccc(NCCCNC(=O)CC2CC3(CCC3)CO2)c([N+](=O)[O-])c1 c1(C(N2CC(OC)C(CNC(C3(C#N)CC(C)C3)=O)C2)=O)ccc(F)c(C)c1C N1(C(c2n(C)c(Cl)nc2)=O)CC(F)(F)CC1C(=O)NC1(C)C(C)(C)C1(C)C c1(C(=O)NCC(C)(C2CCC2)NC(=O)CCS(C)(=O)=O)cccc2[nH]nc(O)c12 c1(C(N2CC(NC(CC(n3c(C)ncc3)C)=O)C(C)C2)=O)cc(Cl)ccc1F CC(C)CCCC(C)NC(c1cc(CCNC(c2cnncc2O)=O)on1)=O c1(N(C2CNCC(F)C2)C(c2scnc2C(F)(F)F)=O)ncc(Cl)cn1 O=C1NCC2(CCN(C(=O)CC3(NC(C4CC(O)C4)=O)CCCCC3)C2)O1 N1(CCOCC)CCC(N=c2[nH]c(=N)[nH]c(=NCCCn3cccn3)[nH]2)CC1 N1(C(C(C)OCC)=O)CCCC(N(C)CC2CCOC(C)C2)C1 C1(CNC(C2=CCC(C)CC2)=O)CN(C(=O)C=Cc2cc[nH]n2)C2COCC2O1 N#Cc1cn(CC(N2CCCC23CCN(C(=O)C2=CCCC2)C3)=O)c(=O)nc1O c1(C(N2CCC(C(=O)NC)C2)C(=O)NC2(C)CC2)cc(Cl)ccc1C C(=O)(C(C)C(F)(F)C(F)F)N1CCC(CCNC(C2(CC#C)CCOCC2)=O)C1 C1(NC(c2c(CC)nns2)=O)CCN(C(C2(N=[N+]=[N-])CC2)=O)CC1CC N1(C(CCOC)=O)CC(C)CCC1C(=O)N(C)CCc1cnn(C)c1 c1(CNC(COCC(=C)C)=O)cn(C2CN(C(=O)CCc3ccncc3)C2)nn1 c1(COC)nc(C(=O)NC2(C)CC(NC(c3snnc3CC3CC3)=O)C2)cs1 C(c1ccc(NC(=O)C(=O)NC2C3CCC(O3)C2N)cc1)=CC(=O)OC(C)(C)C c1(C(=O)N(C)C)ncc(F)cc1N.CC1C(N(C)C)C(=O)N2CCC2C(=O)N1 C(=O)(CS(=O)(=O)CC)N1CCC(N(CC#C)C(C2C3CN(C)CC23)=O)C1 N1(C(Cc2cnc(C)[nH]2)=O)CCCC(C)C1CNC(=O)CCc1ccn(C)n1 C1(NC(c2n(CC)ccn2)=O)C(CNC(=O)C(C)=CC2CC2)CCC12CCC2 c1(OC)sc(C(=O)NCC2CC2CNC(c2ccnc(C)c2)=O)cc1Br N1(C(CS(CC)=O)=O)CCCCC(NC(c2cncc(C(N)=O)c2)=O)C1 c1(C(=O)NCc2c(C)cccc2)csc2c1CCN(C(=O)C(C)(C)F)C2 C1(NC(c2nc[nH]c3nccc2-3)=O)CCCCCN(C(=O)CC(F)(F)Cl)C1 c1(C(=O)NCC(C)CNC(=O)COCc2nc[nH]n2)ccc(F)c(N)c1 c1(CNC(CC2(OC)CCC2)=O)ncccc1CNC(c1cnccc1C)=O N1(c2nc(=NC)[nH]c(=NCc3ncc(C)cn3)[nH]2)CCOc2ccc(Br)cc2C1 N1(C(=O)COCCO)CCOC2(CCCN(C(C3CCC=CO3)=O)C2)C1 Cc1cc(=NC(=O)C2CCN(C(c3cc(Br)cc(I)c3)=O)CC2O)[nH]c(Cl)n1 Cc1ncc(CC(=O)NCC2(C(=O)NCC3CCCN3C)CC2)s1 C(=O)(CCC1=CCCCC1)NC1CC2(CC(C(=O)NCC(COC)(O)CO)C2)C1 C(CCCCC(=O)NCC1CC(NC(c2ncc(Cl)cc2F)=O)CC1O)SC S(=O)(=O)(c1ccc(C#N)cc1Cl)N1CC2N(S(CC(=O)OC)(=O)=O)C(COC2)C1 c1(-c2n(C(COCC)C)nc(C(C)O)n2)cc(C)c(Br)cn1 CC1C(C)N(CC(F)F)CCN1C(c1cc(Cl)nc(Cl)c1)C(=O)NC1CCOC1 C1(N(C)C(c2cc(=O)cc(Cl)[nH]2)=O)CN(C(=O)COC2CCCCC2)CC12CC2 C1(CNC(CCOC)=O)COCCN1C(c1nccc(SC)n1)=O N1(C(CC2CC(C)C(C)CC2)=O)CCCC2(CCN(C(=O)CSC(F)F)CC2)C1 c1(OC)ccc(O)cc1C(N1CC(O)(C(C)NC(c2csc(Cl)c2Cl)=O)C1)=O c1(CN(C(C2CCOCC2)C)C)ccc([N+](=O)[O-])c2cccnc12 CCC(CN(C)C)CC(=O)NCC1C2CN(C(c3ccnc(Cl)c3OC)=O)CC12 C(C(C(=O)NCCCc1ncco1)NC(=O)Cn1ccnn1)SCC C1(C(=O)NC2(CC=C)CCN(c3nnc(C(N)=O)s3)C2)CCC(C)(C)CC1 N1(C(c2cc(C)n(C)n2)=O)CC2CN(C(C3CCN(CC(C)C)CC3)=O)CCC12 CC(C(=O)NCC1CC2CCC1N2C(c1cc(Cl)ccc1F)=O)C(C)(F)F C(=O)(C(C(C)O)NC1CCN(C(C)Cc2ccccc2)C1)OC C1(N=[N+]=[N-])(C(=O)NCc2nccc(C)c2F)CCN(C(=O)CC2CCC(=O)C2)C1 c1(C(N2CCC(C)(CCNC(c3ccc(C)cc3)=O)C2)=O)ccc(F)cc1C c1(C(N(CCC(C)NC(c2c(C)cccn2)=O)C)=O)ccc(C#N)cc1O C1(OC)COCC1n1cc(C(N2CCCC2CNC(c2cscc2Cl)=O)=O)nn1 c1(C(N2C(C)CC(NC(c3cc(F)c(F)c(F)c3)=O)C2)=O)cc(Cl)cc(F)c1N Cc1cc2c(C(N3CCCC(CO)(NC(c4cnns4)=O)C3)=O)ccc(C)c2[nH]1 C1(C(N2CC(c3ccccc3)(NC(CC3(C=C)CC3)=O)C2)=O)COC2(CCC2)C1 c1(C(c2nnnn2C2CC2)NCC2(CCF)CCC2)ccc2ncsc2c1 c1(SC)nocc1CCNC1CC1.C1C(=O)N1CCO C1(C(=O)NCCCCNC(c2ncc(Br)cn2)=O)CCCC(F)(F)C1 N1(C(=O)OC(C)(C)C)CCC(O)C(C)(C(=O)Nc2cc(Br)ccc2C(C)(C)C)C1 C1(CC(=O)NC2(CNC(c3cnn(C)c3N)=O)CCC2)CCC(C)(C)CO1 c1(C(CC)C)ccc(C#N)c(N2CCCN(C(c3c(Cl)csc3Cl)=O)CC2)n1 c1(CNC2(CO)CC2)ccccc1C(C)(C)N(C(C1C(C(=O)OC)C1)=O)C1CC1 N1(C(C2(OC)CC2)=O)CCC(C(F)(F)F)C(NC(=O)C=CC2CCC2)C1 CS(=O)CCC(O)C(=O)NC1CCN(C(=O)Cn2nnc3ccccc23)CC1 N1(C(c2c(C)ccs2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C2(CCC2)C1 CS(=O)(=O)c1cccc(Cl)c1NCC1=CCN(C(=O)NC2CC2)CC1.c1(SC)ccccc1 CC1(CCNCc2ccc(-c3cccc(Cl)c3)cc2)CCNC1=O C1(C)(C(N2CC(CC)C(CNC(c3cc(C)ns3)=O)CC2)=O)CC(C)OC(C)C1 C1(NC(C(N2CC(C)C2)C)=O)CC=CCC1C(=O)NCC1(CO)CCCO1 N1(C(C(C(C)O)N(C)C)=O)CCN(C(=O)C=Cc2cccc(F)c2)CC(CO)C1 c1(C(C(=O)NCCC(CNC(c2c[nH]nc2C(C)C)=O)OC)C)c(C)n[nH]c1C c1(C(=O)NC2CCSCC2)cccc(CN(C)C)c1.CC1C=CC(=O)N1 Cc1nc(CC(=O)N(CC(O)CN(C(=O)CN(c2ccccc2)C)C)C)cs1 c1(CC(=O)OCC)cc(Br)c2c(c1)CCO2.c12ccsc1COC(=O)C2 C(=O)(C(F)(F)C(C)O)NC1CN(C(C(CC=C)OC)=O)CC1F O=C(C(O)C(F)(F)F)NCc1cccc(-c2cn[nH]c2)c1 N1(C(C(C2CCOC2)NC(CC=CCC)=O)=O)CCCC(CCC)CC1 Cc1noc2ccc(NC(C3CC(Nc4ncnc5cc(I)sc45)C3)=O)cc12 C1(OC)CCCC1C(=O)NCC(C)N(C)C(C1CC(C)(C)C1)=O c1(CN(C(C(=O)NC(C2(C)OCCO2)C)=O)C)nc(Br)cs1 C1(C(=O)NCC2CCC(NC(C(C)OCCN(C)C)=O)C2)COC2COCC12 CC1CCN(C(C(=O)NCc2ccccc2)C2CC2(Br)Br)Cc2ccc(O)cc21 C(=O)(CCS(=O)(=O)NC)N(CCCCN(C(CCCN(CCC)CCC)=O)C)C CCC(C)C(O)C(=O)N1CC(C)(NC(c2cccc(C(F)(F)F)c2O)=O)C1 c1(NC(C2(CNC(c3cccnc3CO)=O)CC2)=O)cc(F)c(Cl)cc1F Cc1nc(N2CCCC(C(=O)N(C(C)C)Cc3cccc(Cl)c3)C2)nc(O)c1C Cc1nc2c([nH]1)CC(NCc1c[nH]nc1-c1ccccc1Br)CC2 Cc1c[nH]c(C(=O)NCC2(C(=O)NC3CC(CC(N)=O)C3)CCCO2)c1C c1(CNC(C2CC3(C2)CN(Cc2cccnc2)C3)=O)cc(Br)cc(Cl)c1F C(C)(C(CC(=O)NCC1CCOC1C)NC(C1CCC1C(C)(C)C)=O)OC N1(C(COC(CC)(C)C)=O)CC(N(C(=O)CN2CCC(O)CC2)C)C(O)C1 C(=O)(CCC(N)=O)NCC1(NC(c2n(C(CC)C)ncc2)=O)CCOC1 N1(C(C)C)CCC(C(N2CC(N3CCN(c4ccc(F)cn4)CC3)C2)=O)C(C)C1 c1(C(=O)OC)ccc2c(c1)C(NC(=O)NC(C)C(=O)N(C)C1CC1)CC2 N1(C(CCC(C)(C)C)=O)CC2(CNC(=O)CC3CC=CCC3)CC(F)(C1)C2 C1(CN(C(=O)C(N2CCCC(F)CC2)=O)C2CC2)CCC2(CCCCCC2)O1 N1(C(CC2(NC(CCC)=O)CC2)=O)CCC(CCCO)C1.C1C(=O)N1 CS(=O)c1ccc(CC(=O)NCC(=O)NC2CC2)cc1.c1ccc(N)c(Cl)c1O C=C(F)C1(CC(N2CCN(CC(=O)NCc3n[nH]cc3C)CC2)=O)CCC1 C(=O)(C(F)(F)C(C)(C)O)NCC12OCC(NC(C(CC)NC(N)=O)=O)(C1)C2 c1(OCCC(=O)NCCCCNC(c2ccc(C)cn2)=O)ccccc1[N+](=O)[O-] N1(C(c2c(CNC(C(C(C)C)C3CCC3)=O)cc[nH]2)=O)CC(CO)CC1(C)C c1(CC(=O)N(CC(CNC(C(CC)C)=O)(C)C)C)c[nH]c2cc(F)ccc12 c1(COC(CN(C(C)=O)C)=O)ccc(O)cc1.C12CC(CO1)NC2=O C1(C)(C(=O)NCC(n2cc(C3(C)CCCC3)nn2)C)CCCS1 N1(C(=O)C=CC2CCCCCC2)CC2CCN(C(C3C=CCCC3)=O)C2C1 Cc1cc(C(=O)NC2(C(=O)N(C3CCN(C4CC4)C3)C)CC(F)C2)sc1C c1(CCc2c(C)c(N3CCC(C4CCCC4)C3)ncn2)ccc2oc(=O)n(C)c2c1 c1(C(=O)NCCCOCCCNC(C(C(C)(C)O)F)=O)cn2cccnc2n1 Cc1cc(C(=O)NCC(C)CC(=O)NC2CC(n3cccn3)C2)nc(O)c1 n1(CCC(=O)NCCN(C(=O)CC2CCC3CC23)C)cc([N+](=O)[O-])cn1 N(C(=NCCC(C)C)NCc1cn(C2CCOC2)nn1)CC1CCC(=C)CC1 c1(C(=O)NCCC2CC(OC)CN2C(c2ccc(C)s2)=O)cc(C)c(C)c(F)c1 C=CCCCCCC(=O)N1CCN(C(=O)C(C)(CC)OC)CC(CO)C1 N1(Cc2cn(CC(=O)NC3(C(N(CCC)CC)=O)CC3)nn2)CC2CCC1C2 N1(C(C(c2cccc(C)c2)O)=O)C2CCC1CC(O)(CNC(=O)CCF)C2 c1(OCC(=O)N(C)C)ccccc1NC(CNC(c1snnc1C1CC1)=O)CO C1(C)(NC(C(C)Oc2ccc(O)cc2)=O)CCCN(C(=O)CCP(C)(C)=O)C1 C1(NC(C=Cc2scc(C)n2)=O)CCCC(NC(c2cn3c(n2)CCC3)=O)CC1 CC1=C(C)CC(C)(NC(=O)CNC(c2ccc(C#N)n2C)=O)CC1 C(=O)(CC(C)C(C)(C)C)N1CCC(C=C)(C(=O)NCC(c2cnc[nH]2)C)C1 C1(C2CCN(C(=O)Cc3cc[nH]c3)C2)(NC(c2cc(CCC)c(C)s2)=O)CC1 N(C(=NC)N1CCC(n2cc(C)cn2)C1)Cc1nc(C(=O)OCC)nn1C C1(COCC)CN(c2ncncc2OC2(C(=O)NC)CCCC2)CC(C)(C)O1 CC(CC(=O)NC(C1CCN(C(=O)CC2CC2C)C1)C)CC(C)(C)C Cc1cc(F)sc1C(=O)NC(C)CNC(C1CC12CCC2)=O CC(C)C(O)C(=O)N(CC(C)CNC(=O)Cc1ccc(SC2CC2)cc1)C c12cccc(c1)NC2=O.C1(SCCC(=O)OCC)CCCCC1 N1(C(C2C(C)C2C)=O)CCCC1CN(C(=O)CO)C1CC1 C1(c2ccc(C)cc2)NC(=O)N(CCCNC(c2nnnn2C)=O)C1=O c1(C(N2CCN(C(C=CC=CC)=O)CC(O)C2)=O)ccnc2c1ccn2C c1(C(N2CC(=C(CNC(C3C(OC)CCC3)=O)F)C2)=O)ccc(C(C)C)cc1 C12(C(=O)NCC(CO)NC(c3cccc(OC)c3)=O)CC=CCN1CCC2 CC1CCN(C(c2ccc3n[nH]cc3c2)=O)C(C)C1NC(C1CCC(C)O1)=O C1(C(=O)NC(CSC)(C)C)C2CN(C(c3cc(Cl)n[nH]3)=O)CC12 c1(C(N2CCC(OC)(CNC(=O)C(O)C(C)C)C2)=O)cc(C)nc(CC(C)C)n1 C1(OC)(COC)CCCC(C)C1.c12cncc(n1)C(=O)N1CCC1c1cn-2nn1 C=C(C)C(CC(=O)NCCOC1CCN(C(=O)CS(N)(=O)=O)C1)OCC CN(CCCC(=O)NCC1CC1NC(=O)Cc1cc2ccccc2o1)N=O C1(CC=C)(C(=O)Nc2ccc(SC)nc2)CCCN(C(=O)C(O)C=CCC)C1 CC(F)(F)C(F)C(=O)N1CC=CCC1C(=O)NCC1Cc2nccn2C1 N1(C(C2CC(F)CN2C(c2cc(F)c(F)c(Cl)c2)=O)=O)Cc2ccc(F)cc2C1 C1(CC(=O)NCC(CC)NC(c2ccc(OC)c(C)c2)=O)CCCC2(CCC2)O1 c1(C(=O)NC23C(CN(C(CC(C)F)=O)C2)C3)cc(N)c(Cl)cn1 N1(C(C2(CC)CCC2)=O)CC(NC(c2cc(N)ccc2Cl)=O)C2(CC2)C1 N1(C(CN(C(C(C)C)=O)C)=O)CCC(C)(CCCC2(C(=O)O)CCCO2)C1 C1(NC(C2(C(C)C)CCCC2)=O)CCN(C(c2cnoc2C2CC2)=O)CC(O)C1 CC(CCN=c1ccc(Br)c(S(=O)(=O)NCCC2=CCN(C)CC2)[nH]1)N(C)C O=C(C1=C2CCN=C2NC=C1)NCC(C1CCCCC1)NC(=O)CSc1cccs1 C1(C)(C(=O)NC2(C(C)NC(C3CCC3C(F)F)=O)CC2)CCCC1O N(C(=NCC(C)(C)CC1(C)OCCO1)NCC1CC1)C(c1ccc(Cl)c(F)c1)C N1(C(c2cc(C)[nH]c2)=O)CCCC(C(=O)NCCc2cc(C)[nH]n2)CC1 C(=O)(C1=CCCN(C(=O)CC2C=NN(C)C2=O)C1)NCC(C#C)C(C)C C1(C(=O)NC(C)CNC(c2cccc3c2OCCO3)=O)Cc2c(F)cccc2O1 C1(c2cn(CC(F)(F)CO)nn2)(NC(C2CCC(F)C2)=O)CCCCC1 N1(C(C(CC)Sc2nc(C)cs2)=O)CCC(C2CN(C(=O)CCSCC)C2)CC1 Cc1c(C(F)(F)F)cc(NC(N2CCN(CCC(=O)O)CC2)=O)cc1O C1(NC(c2c(C)cc[nH]2)=O)CCCN(C(c2cc(C3CC3)on2)=O)CC1F Cc1cc(CNC(C)(CCCl)c2nnnn2-c2ccc(F)cc2)cnc1C c1(C(=O)NC2C(CNC(CCC(C)OC)=O)CC2)sc(C#N)cc1Cl N1(C(CC(C=C)C)=O)CCCC(CO)(CNC(c2ccc(OCCO)cc2)=O)C1 c1(N2CC3N(C)C(CCC3)CC2)nc(=NCC23CCC(CO2)C3)[nH]c2ccsc12 c1(C(N(CC(C)NC(C2COC(=O)N2)=O)C)=O)cnn(C2CC2)c1Cl C1(C(CNC(COCC(=C)C)=O)(C)C)CCN(C(C2CCCC2OCC)=O)CC1 c1(C(=O)OCC)c(NC2CC(C)N(C(=O)CC(C)(C)OC)C2)cc(C)nc1O CCCCC(=O)C(=O)N(CCCN(C(=O)C(C)c1cc[nH]n1)C)C N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)C(C)(O)C3CC3)C(C2)C1 c1(SCC(N2CCCC(CNC(C3(CC=C)CC3)=O)C2)=O)ccsc1[N+](=O)[O-] N1(C(c2cc(C)oc2C)=O)CC2CCC1C(CNC(C1CC1F)=O)C2 C12(C(N(c3cccn3C)CCNC(C)=O)=O)CC3CC(C1)CC(O)(C3)C2 c1(CNC2(CC(=O)NC(c3ccccc3F)C)CCC2)ccc2[nH]ccc2c1 Cc1cc(C)c(CC(=O)N(C2CCN(C(=O)COc3ccc(F)cc3)C2)CC)s1 C1(c2cn(CCC3CN(C(C4OCC(C)C4)=O)C3)nn2)CCCC(F)(F)C1 CCC(CCC(=O)NCC1CCCC(NC(=O)CCc2cc(C)nn2C)C1)OC N1(C(c2c(OC)cnnc2)=O)CCCC(CC(N2CCC2C)=O)CC1 NS(=O)(=O)CCCC(=O)NC1COCC1NC(c1cc2c(s1)CCOC2)=O CCC(CC(=O)NCCNC(C1(C)CCC(=O)N1)=O)C1CC1 Cc1cn(C)cc1C(=O)NC1(C(=O)NC(C(N)=O)C2CCCC2)CC1C Cn1[nH]c(C2CCN(CCN3CCOCC3)CC2)nc1=N N1(C(CC2(C)OCCO2)=O)CCC(CF)(NC(=O)Cc2cc(C3CC3)no2)C1 Cc1ccc(CNC(N2CCN(C(c3cn(CC4CC4)nn3)=O)CC2)=O)cc1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)Cn2ccsc2=N)c2c(c1)CCO2 CCC(C)C(O)C(C)C(=O)N1CCOC(CN(CC(=O)NC)C2CC2)C1 c1(CC)cccc2c(F)c(C(N3CC4C(NC(=O)C=C(Cl)Cl)C4C3)=O)[nH]c12 Cc1ccc(Cl)cc1C(=O)NC1(CNC(C2CCN(CC(C)C)C2)=O)CCCC1 N1(C(c2c(F)ccc(N)c2)=O)CCCC(C2CCCNC2)C1 c1(OC(C)C)n[nH]c(C(=O)NC2CN(C(=O)Cn3cccc3)CC2F)c1Br C=CCCC(C(=O)NC(c1cnns1)C)NC(=O)CCC(C)OC c1(C(=O)NCC(C)NC(C(C)NC(CC)=O)=O)ccc(C(F)(F)F)cc1[N+](=O)[O-] N1(C(CCCc2ncc(C)o2)=O)CCC(CNC(=O)CSCC(C)C)C(C)C1 C1(C(N(CC(C)NC(c2ccc(SCC)cc2)=O)CC)=O)CCCCC(F)(F)C1 c1(C(N2CCC(F)(CNC(C3(CF)CCC3)=O)C2)=O)cccnc1F C=CCCCC(C)(C)C(=O)N1CCC(C)N(C(=O)CC2CCS(=O)(=O)CC2)CC1 C1(C)(CNC(C2C(CC=C)CCC2)=O)COCCN(Cc2cn(C3CC3)nn2)C1 c1(C(C(=O)NCC2N(C(CCOCC)=O)CCCC2)C)ccc2ccccc2c1 C(=O)(CC(F)(F)C(C)C)N1CC(CC)N(C(c2nnn(C)c2C(F)(F)F)=O)CC1 C1(C(C)NC(c2ccc(C3CC3)o2)=O)CN(C(C2CCCC2)=O)CCO1 CC(CS(C)(=O)=O)C(=O)Nc1ccc(Cl)c(C#N)c1.C12CN(CC1O)c1cn2nn1 c1(C(N(C2CN(C(C3CC4(CSC4)C3)=O)C2)C)=O)nnc2ccccc2c1N C1(CNC(C(COCC)C)=O)CN(C(c2ccccc2OC(C)CC)=O)CCN1C c1(C(N2CC(NC(CC3(C)CC3(F)F)=O)C2)=O)ccc(C(=O)CF)cc1 c1(C(N2CCC(OCCNC(C(C)n3cncn3)=O)C2)=O)cc(C2CC2)nn1C c1(C(N(CC(C)N(C(=O)CC2CCN(C)C2=O)C)C)=O)cc2n(n1)CCC2 Cc1nc(N2CC3CCCC(NC(C4CC(C(C)C)C4)=O)C3C2)ccc1[N+](=O)[O-] N1(C(CN(C(C(C)C)=O)C)=O)CCC2CN(C(=O)CN3CCN(C)C(=O)C3)C2C1 C1(C(N(OCC(=O)OC)C)=O)CC(NC(c2cc(OC)n[nH]2)=O)CCO1 CC1(C)COCC1C(=O)NC1CN(C(C2CC3CCC(C2)C3)=O)C1 CCC(C)(CNC(C1CCC(=O)O1)=O)C(=O)NC(c1nnc(C)o1)C C1(CNC(C2CN(C(C3C4CCC(F)C34)=O)CCO2)=O)CC2(CCC2)C1 c1(OC)cc(C(N2CCC(F)(CNC(=O)C=Cc3nc(C)co3)C2)=O)c(F)cn1 c1(OC)ccc(C2CCN(C(c3csc(-c4cccc(F)c4)n3)=O)CC2)nc1 CCC(CC(F)F)C(=O)NCC1CN(C(=O)CC(C)C(=O)OC)CC(C)(C)O1 C(CC(C)(C)CC(=O)NC(c1nc2ccccc2o1)C(C)C)OC C1(C(=O)NC2CC(CC(=O)NC(CC(C)O)C)C2)CCC(C)(C)OC1 c1(CCC)nc(=NCC2(O)CCCN(C(=O)CC(=O)N(CC)CC)C2)s[nH]1 Cc1cc(C)c(NC(C23CC(CN(C(c4cnc(N)c(N)c4)=O)C2)C3)=O)cc1O C1(C(=O)NCC2CCC(C(N(c3ccc(OC)cc3)C)=O)C2)CCOC(=O)CC1 c1(CC(=O)N(C(C)CNC(=O)C(c2cncnc2)C)C)cccc2ncccc12 Cc1ncc2n1CCC(C(=O)NC(C)CNC(C1CC1C(C)O)=O)C2 N1(C(C(CCN(C)C)N)=O)CCC(OC(F)F)C(O)C1 c1(C(=O)NC23CCN(C(=O)C=Cc4nccs4)CC2C3)cccc2[nH]nc(O)c12 N1(C(C(=Cc2cn[nH]c2)C)=O)CCOC(CCNC(=O)CC2CCC(=O)N2)C1 c1(CNC(C(C)SCC)=O)ccc2c(c1)CCN(C(=O)Cc1cc(C)nn1C)C2 C(CC(C(C)(C)C)NC(C1CC1c1ccco1)=O)N(C(C(C=C)(C)C)=O)C C1(=CC(=O)N(C(C)CNC(=O)C=CCN(C)C2CC2)C)CC2CCC(C1)N2C C(CCC)(C(=O)NCC1CCC1N(C)C)NC(COCC(=C)C)=O C(=O)(C1CCCc2n[nH]cc21)N(CC(C)CNC(=O)Cc1cccnc1Cl)C c1(C(N2CC3(CCN(Cc4cc(F)cc(Br)c4Cl)C3)C2)=O)nc2ccccn2n1 Cc1nc(C)c(C(=O)NCC(O)CN(C(=O)COCCCN(C)C)C)o1 c1(C(=O)NCC)ccc(OC(C2CCC(C#N)CC2)=O)c([N+](=O)[O-])c1 C=CCC(CC)C(=O)NC1(C)CN(C(c2cc(OC(F)F)cc(F)c2)=O)C1 c1(OCC)ncccc1N(C)C(c1cccc[n+]1[O-])=O c1(C(C(=O)N(CCCCN(C(C2CC(=C)C2)=O)C)C)=O)cc(Br)cs1 CCC(C)C(O)CC(=O)NCCC1CC(NC(=O)CNS(=O)(=O)C2CC2)C1 c1(C(N(C2(C#N)CCN(S(=O)(=O)c3cn[nH]c3)C2)C)=O)cccc2c(O)nccc12 C(C(CC(C)C)C(=O)NCc1ccc(C(=O)NC(C2CCCO2)C)nc1)OC c1(C(=O)NC(CNC(Cc2c(C)n[nH]c2C)=O)CO)onc2ccccc12 N1(C(CCCCC)=O)CCC2(CC1)CC(NC(=O)CCn1cncn1)CO2 c1(CC(=O)NC2C=CCN(C(c3cc(O)ncn3)=O)C2)cc(F)cc(Br)c1 C(C(=O)N1CC(O)(C2CCCN2C(=O)COCC2CC2)C1)(C(C)(C)C)NC(C)=O CC(CCC(=O)N1CCC(CNC(=O)Cc2cncnc2)C12CC2)S(C)(=O)=O C1(C)(CC)CN(C(c2[nH]cnc2C)C(=O)Nc2ccc(F)cc2C)CCO1 CCCC(C(=O)N1CCN(CC(C)NC(c2cn(CC)nn2)=O)CC1)NC(N)=O C1(CNC(CCCC(C)=O)=O)COC(C)(C)CN1C(=O)CC1CCOC1(C)C C(C(O)C(=O)NC(C)CC(=O)NCCc1ccon1)=CC N1(C(CCC2(NC(=O)CCc3ccsc3)CCC2)=O)CC(O)(C2CCC2)C1 C(=O)(C(CC1CCCC1)NC(=O)CC(C)N(C)C)NCCCNC(C)=O c1(N2C(CNC3CN(c4ccc(C(N)=O)cc4)C(=O)C3)CC2)ccnc2ncnn12 N1(C(C2(CC)CCOC2)=O)CC(CCNC(C2C(CN=[N+]=[N-])C2(C)C)=O)C(C)C1 N1(C(=O)C=C2CCCC2)CCC(O)(C2(NC(C34CCC(CC3=O)C4)=O)CC2)CC1 CC1(C)CCCCCC1S(=O)(=O)Oc1cnnn1-c1ccccc1 Cc1cnc(C(N2CCOCC2CNC(=O)CCS(C)(=O)=O)=O)c(C)c1 N1(C(CCCOC)=O)CCCC(CO)(CNC(=O)CC2CCSC2)C1 C1(NC(c2cscc2F)=O)CC2CCC1CN(C(=O)C1CCc3c[nH]nc31)C2 N1(C(C(C2CCCCC2)C)=O)CC2CC(NC(c3ccc(Cl)s3)=O)CC1C2 c1(OC)cnc[nH]c1=NCC1(O)CCCN(C(=O)CSc2cccc(F)c2)C1 C(=O)(C(C)(C)C(C)O)NCC(=O)NC(C)C(C)C(=O)O n1(CC)nnc2c1C(C(=O)NCc1ccc(F)cc1F)CN(C(C1CC1C)=O)C2 Cc1cc2nc(NC(=O)N(c3ccc(=N)[nH]c3)C)sc2cc1F O=C(C#CC1CCCO1)NCC1CCCN1C(c1scnc1C1CC1)=O c1(C(N2CC(C)(O)C2)=O)nc(-c2cccc(F)c2C#N)c2ccccn12 n1(CC(=O)NCC2CC(NC(C(CCCC)O)=O)C2)ncc2ncccc12 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2SCCS2)=O)CCC1C C(C(F)(F)CO)N(C(=O)C(c1cccs1)NC(c1cccn1C1CC1)=O)C N1(C(c2c(C)cn(C)n2)=O)CC2CC1CCC2NC(=O)Cc1c[nH]nc1C Cc1cnc(C(N2CC(NC(=O)Cc3cc(C4CC4)on3)CC2C)=O)cc1C#N N1(C(C(C)Cc2ccc(Br)cc2)=O)CCOC2C(C(=O)OC(C)(C)C)CC12 c1(C(N2CCC(C)(NC(C(C(=O)OCC)F)=O)C2)=O)nc2ncc(C)cn2n1 N1(C(=O)Nc2cc(CC(C)C)ncc2)CCC2C(CC(=O)N2C)C1 NS(=O)(=O)c1coc(C(N2CCC(NC(=O)CC3CCC(=O)N3)C2)=O)c1 C1(NC(C(C2CC2)OC)=O)COC2(C1)CN(C(c1c(N)cccc1F)=O)C2 N1(C(C)C)CCOC(C(=O)NCCCC2CN(C(c3cc(F)n[nH]3)=O)CCO2)C1 C1(NC(c2c(NC)cncc2)=O)CCN(C(=O)C(F)(F)CN(C)C)CC1F c1(CCC(=O)NCCC2CCN(C(C3(F)CCOC3)=O)C2)ccc(F)cc1 c1(OC)ccc(C2C(C(=O)Nc3nccs3)C2)cc1OCC(N)=O C1(NC(c2c(C)occ2)=O)CC2CC(NC(c3cnc(Cl)c(N)c3)=O)C1C2 C(=O)(C(C)C(C)COC)NC1CC(NC(c2n[nH]c(CC)c2Br)=O)C1 Cn1cnc(=N)[nH]c1=NCc1cc[nH]c1-c1ccncc1 Cc1cccc2c(N(C(=O)C=Cc3ccc(F)cc3)CC3CCNC3)ncnc12 C(=O)(CC1=CCCC1)N(C(C)CNC(=O)C(c1cc(Cl)ccc1F)(C)C)CC Cc1ccc(CNC(C2CC2C(=O)Nc2oncc2C#N)=O)c(F)c1 Cc1cc(C)nc(N2CC(NC(c3cn(CC4CCCOC4)nn3)=O)CC2C)n1 N1(C(CCC2CC(NC(C3(C)N(C)CCC3)=O)C2)=O)CC2CC3CC2C1C3 C1(CCC(=O)NCCN(C(=O)Cc2nc(C3CC3)nn2C)CC)CCN(C)CC1 C1(CNC(c2c(C)n(C3CC3)nc2)=O)CN(C(c2cnc(N)cn2)=O)C(C)(C)C1 c1(C(=O)NC2C(C)N(C(=O)CC3CC3(C)C)CC2)c(Cl)c([N+](=O)[O-])nn1C C1(NC(c2cc(Cl)no2)=O)CC2CC1CN2C(C1(C(c2ccccc2)=O)CC1)=O CCCCN=C(NCC1(C)CCC(=O)N1)NC(C)CC.C12CCN1C2 C(=O)(C(CC(C)(C)C)NC(=O)CC1CC(C)C1)N1CC(CC(C#C)C)C1 C(C(=C)C1CCOCC1)NC1(c2n(CC=C)nnn2)CC(C2CCNC(=O)C2)C1 C1(N(C(=O)COCc2ccccn2)C)CN(C(=O)CN2CCSCC2)CC1(C)C C1(N=[N+]=[N-])(C(=O)NCC(C#C)C(C)C)CCN(C(=O)C(N)=O)C1 C(CC1=CCCCC1)N(C1CCCN(CCC)CC1)CCCS(=O)(=O)CC c1(C(C(=O)NC(CNC(C2(C(N)=O)CC2)=O)(C)CO)=O)cc(F)ccc1C C1(C(=O)NCC2(NC(CCC=C)=O)CC3CCC2CC3)Cc2c(C)cccc2O1 c1(C(=O)NC2CCN(C(c3cc(CC)on3)=O)CC2)cc(C)c(O)c(C)c1 CN1C(=O)CCC1C(=O)NOCCCC(F)(F)F.c12ncccc1C(=O)NC2 c1(C(=O)NCCOCCNC(CCC2CCN(C)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(CC(=O)N(C)CC2CCCN(c3nnn(C)n3)C2)CCOC(C)(C)C1 C1(C(=O)NC(Cn2cc(C(C=C)(C)O)nn2)C)CC2(CCNCC2)CO1 Cc1cc(C(=O)NCC2CC2NC(=O)CC2(n3ccnn3)CC2)cnc1C(F)F C(=O)(C1=NN(C)C(=O)CC1)N(C)CC1(CNC(c2nc(CC)oc2C)=O)CC1 C(C(C)N=c1[nH]c(CC#N)nc(Cl)c1C)(C1CC1)NC(C(C)C)=O C1(NC(C2(CO)CCN(C(C(C)OCCN(C)C)=O)C2)=O)C(C)(C)C(O)C1(C)C C1(C2(O)CCN(C(=O)C=CCN(C)C)CC2)(NC(C(C)NS(C)(=O)=O)=O)CC1 C(=O)(CCCC(C)=O)N1C(C(=O)NCC2(F)CCCCC2)(COC)C=CC1 c1(OCC)cccc(C(=O)NC2CCC(CNC(=O)CNC=O)C2)c1N C1(COC)CN(C(c2ncc(C(C)(C)C)cn2)C(=O)NCCCSC)C(C)(C)C1 C(C1(O)CCc2ccccc21)NC(CC(C=C)(C)C)c1nnnn1C1COC1 c1(SCC(N2C(c3cc(C)[nH]n3)CSCC2)=O)cccc(F)c1[N+](=O)[O-] C1(C(C)N(C)C(C2CC(CCNC(=O)CC(C3CC3)C3CC3)C2)=O)CCOCC1 CC1CN(C(=O)CCC2(C)CN(C(C3CCN(C)CC3)=O)C2)CC1(F)F CC1COc2c(C(=O)NC3CCCC3NC(=O)CCCC(N)=O)cccc21 CC1(C)C=C(C(=O)N2CC(NC(c3cc(-c4cccs4)[nH]n3)=O)CC(F)C2)C1 N1(C(c2c(CC)onc2C)=O)CCCC(C2(NC(=O)C(F)=C(C)C)CC2)C1 C12(CC(=O)NCC3C(CNC(c4nn(C)c(F)c4)=O)C3)CCC(CC1)CC2 c1(C(N2CC(C)C(CNC(=O)CCCC(F)F)C2)=O)coc2c1C(=O)NCCC2 C1(C(=O)NC2(CSC)CCC2)CCN(C(c2cnnc(O)c2)=O)CCO1 C1(OC)CC(CCNC(C)=O)N(C(C2CCN(CCC3CC(F)C3)CC2)=O)C1 C1(C(=O)NCC(CCC=C)O)CN(C(=O)Cc2c(C)noc2C)CCN1C c1(OC)cccc(C(=O)NC(C)CC(C)NC(=O)CCNC(C)=O)c1F N1(C(c2cnc(C)c(N)c2)=O)CCC2CN(C(=O)Cc3cccn3C)CC2C1 c1(SC(C(=O)OC(CCC)C)C)ccc(Cl)cc1 C1(C)(NC(C(CNC(C2N(CC)CCC2)=O)N(C)C)=O)CC(C)(C)C1 C1(NC(CC2(C)N(C(c3cc(C)cc(O)n3)=O)CCC2)=O)CCn2ncnc2C1 c1(C(=O)NCC(CC(C)C)NC(C(C(CC)O)C)=O)nc(N)cc2ccccc12 CC1(CNC(N)=O)CN(C(=O)C(C2CCCC2)NC(=O)CCCCO)CCO1 C1(NC(C2CCN(C)C2)=O)CN(C(c2cc(C(C)(C)C)on2)=O)CC2(CC2)C1 C1(C(=O)NCC(CSC)(C)C)C2CCC(C2)N1C(=O)C(C1CCCCC1)C c1(NC(C2CC(NCc3cccc4cc[nH]c34)C2)=O)c(Cl)cc(Cl)cc1[N+](=O)[O-] C#CCCCCCC(=O)N1CC=CC1C(=O)NCc1cc(F)ccc1Cl N1(C(c2c(C)c(Cl)ccn2)=O)CCC2(CCCCC2NC(c2cc(Cl)no2)=O)C1 N1(C(C2C=C(C)CS2)=O)CC(C(=O)Nc2cc(C)cc(O)c2)CCC1(C)C c1(N2CCCC(CC)C2)nc(N(CCS(=O)(=O)NC)C)nc2ccc(Cl)cc12 c1(CC(CC(F)(F)F)NCC2C(C)(C)COCC2)ccc([N+](=O)[O-])cc1F N1(C(C(n2c(C)cc(C)n2)C)=O)CC(NC(=O)CC2OCCO2)CC12CCC2 C1(NC(c2c(SC)ccs2)=O)CCN(C(C2(C)COCCO2)=O)CC1CO Cc1cc(-c2csc(C(N3CCn4cccc4C3)=O)n2)c(F)c(F)c1 C1(CC)CN(C(C2CN(C(C)C)C2)=O)CC1C(=O)NCCSC c1(C(C(=O)NCC(C)(C)NC(C2(CC)COC2)=O)O)cccc(OC)c1 O=C(CCCC(=O)c1ccc(F)cc1)NCC(F)CNC(C1CCCC12CC2)=O C1(C(=O)NC2CN(C(=O)CC3CNC(=O)O3)CC2O)(CC)CCCC1O C#CCC(C)(C)C(=O)N1CC(CNC(c2ccccc2C(C)C)=O)C(O)C1 Cc1ccc(F)c(C(N2CCC(C)(NC(C3CC34CC4(F)F)=O)CC2)=O)c1 c1(C(=O)NCCOC2CCN(C(CC3(C)CCCO3)=O)C2)cc(Cl)ccc1CO Cc1cc(C(=O)N(C2CC(NC(=O)Cc3cc(C)on3)C2)C)c(C)cn1 CC#CCCCC(=O)NC(CC#CC)C(=O)NCCC(=O)NC(C)CC N1(C(c2cnc(C(C)C)s2)=O)CCOC(CNC(=O)C=Cc2cnc[nH]2)C1 Nc1cc(F)cnc1C(N1CC2CCC2(CC(=O)NCc2cnsc2)C1)=O C1(C(=O)NC2CC(OC3CCCC3NC(CC)=O)C2)CN(C(C)=O)CCO1 CC1(C)CCCC(C(=O)NCC2CN(C(c3ccnc(F)c3N)=O)C2)CC1 C1(CCC)(NC(=O)COc2cn[nH]c2)CCCN(C(C2CCC(CC)O2)=O)C1 c1(CCC(=O)N(C(=O)CSc2ccccc2)CC)cc(C)nc(C)c1 C(=O)(CCCC1CC1)N(CC(C)O)CCNC(C(C)OC1CCCC1)=O C12CC(CN1C)OC2=O.c1(C(C)CN(C)C)ccc(CN2CCCCC2C)cc1 C(C)(C(=O)N1CC(NC(=O)C(C)=CCO)CC(F)C1)(C(C)C)OC N1(C(C(C)OCCC#C)=O)CCC(CCCCNC(C2C3CC4C(C3)C24)=O)CC1 c1(N(C(=O)C(C)=CC2CC2)CCOCC)nc(CC(=O)OC)cs1 CCC(C)C(C(=O)NCC(C1CCCC1)C)N(C)C(c1cnccc1C#N)=O N1(C(c2c(CC)nco2)=O)CC(CNC(C2CCC(C)(C)CC2)=O)C2(CCC2)C1 Cc1cc(=O)oc(C)c1C(N1CC2CC1C2NC(C1(Br)CC1)=O)=O C1(O)(CCNC(=O)CCF)CCN(C(c2ccccc2C(F)F)=O)C1 C1(OC)CC2(C1)CN(C(=O)CNC(=O)C(F)CC1CCC1)C2 C(C(C)(O)CC(=O)NCC1CC(NC(c2cnc(C3CC3)s2)=O)C1)OC N1(C(C(C(C)C)(C)C)=O)CC(NC(C2(C)CC2(F)F)=O)CCC(O)C1 c1(C(=O)NCCSCC)cc(-n2cc(C)cn2)cc(F)c1.O(C=CC(=O)NCCO)CC c1(C(=O)NC(CC)CNC(c2c(C)nn(C)c2C(F)F)=O)nn(C)c2c1CCC2 c1(C(=O)NC(c2ccccc2)CNC(C(C(C)C)O)=O)csc2ncnc(O)c12 N1(CCOC)CCN(c2nnc(-c3cc[nH]n3)n2CCc2cccs2)CC1 N1(C(c2n(COC)ncc2)=O)CC=C(C(C)(C)C(=O)N2CCC(F)(C#N)C2)C1 c1(OC)cc(C)c(C(=O)NC2CCCCN(C(=O)C(F)C(F)(F)F)C2)c(F)c1 N1(CC)CCC(NC(c2sccc2CNC(C2COC(C)C2)=O)=O)CC1 c1(C(=O)NC(CNC(C2CC(C)=C(C)CC2)=O)CO)n[nH]c2c1CCSC2 C1(C(=O)NC2CCN(C(CCOCCCOC)=O)CC2C)CCC(C2CC2)CC1 c1(C(C(=O)NC2(CN(C(=O)CN3CCOCC3)C)CC2)F)ccccc1 N1(C(CNC(C(CC)C)=O)=O)CCOC(C)(CNC(=O)CCS(C)(=O)=O)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(C(C)C)NC(C1CC1C#N)=O Cc1cccc2cc(C(=O)NCC3CCCN3C(c3cc(Cl)ncc3O)=O)sc12 CCC(O)C(=O)N1CCC(C(=O)NC2CSC2)C1 c1(SCC(=O)OC(C)=O)ccc([N+](=O)[O-])c(OC)c1.C1(=O)C=CCN1 c1(CC)ccc(C)cc1NC(=O)C(O)C(C)(C)NC(=O)OC(C)(C)C N1(C(c2nccc(-c3ccccc3)n2)C)CCN(CC(O)CNC(C)(C)C)CC1 c1(CC(=O)NC2C=CCN(C(c3ncc(F)cn3)=O)C2)c[nH]c2cccc(F)c12 C1(C(N2C(CN(C(Cn3c(C)nnn3)=O)C)COCC2)=O)CC2(C1)CC21CC1 N1(C(CCCC)=O)CCC2(CCOCC2)C(CNC(=O)CCCCC(F)F)C1 C1(CNC(c2ccc(Cl)nn2)=O)CCN(c2ncc(C(F)F)cn2)CC1(F)F C(=O)(C1=Cc2ccccc2C1)N1CC(C(=O)NCC(COC)(F)F)CC12CCC2 CC1C(CC(=O)NCCC2CC2)CCCN1C(c1cc(F)cc(Cl)c1)C(=O)N(C)C C1(C(N(CC(N2CCC3(CC3)C2)=O)CC)=O)CCn2ccnc2C1 Cn1cc2c(n1)CC(C(=O)NC1CCC(CCNC(=O)CNC=O)C1)NC2=O CC(F)CC(=O)N(C(c1ccccc1)CNC(=O)Cn1ncnn1)C c1(C(N(C)CCNC(c2cc(C(N)=O)ccn2)=O)=O)ccn2ccnc2c1 CC1CCC2(CC2)N(C(C2CC3CC2CN(C(c2cnccn2)=O)C3)=O)C1 c1(C(=O)NC2C(CNC(c3c(C)n[nH]c3)=O)CCC2)cc2cccnc2nc1O C#CCC(C)C(=O)NCCCNC(c1ccoc1I)=O c1(N2C(CCCNC(C(C)NC(COC)=O)=O)CCC2)nc(Cl)nc2[nH]cnc12 c1(CC)nocc1C(=O)NCC(CCNC(=O)Cc1ncoc1C)OC N1(C(Cn2cc(CNC(=O)Nc3cccc(N)c3)nn2)=O)CC2COCC2C1 CC1(C)COCC1C(=O)NC1CC2(C1)CC2NC(C1CC1c1ccccc1)=O C1(C(N)=O)CCCN(N2CCC(SCC(F)(F)F)CC2)C1 CN1CCOc2ccc(-n3cc(CC4(C(=O)O)CCC(CO)CC4)nn3)cc21 c1(C(C)=O)cc(CNC(CC2N(C(C34CC(CSC)(C3)C4)=O)CCC2)=O)oc1C CON(C)CCCNC(=O)C(CNC(c1ncoc1C(C)C)=O)N(C)C C(=O)(C(CCOC)NC(C12CCCC1C2)=O)NCC1CC(CN(C)C)C1 Nc1cc(C(=O)NC2CCC2NC(c2n[nH]cc2Cl)=O)c2ccccc2c1 N1(C(Cc2ccc(C)cc2)=O)CCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1 C1(C(=O)NCC2(C(N3C(CCC=C)CCC3)=O)CC23CCC3)CC(=O)CC(=O)N1 c1(OCCC)cccnc1CC(=O)NCCC1(O)CN(C(=O)CCC=C(C)C)C1 N1(C(C(CC)CCOC)=O)CC(NC(C2CCc3ccnn3C2)=O)CC12CCC2 c1(C(=O)NC2C3CN(C(c4c(C)cc[nH]4)=O)CC2C3)ccc2[nH]c(C)c(C)c2c1 c1(C(N2CCOCC(NC(C3C(=C)CC3)=O)C2)=O)cc(C)nc(Cl)c1N c1(CCC(=O)OC(CN(C)Cc2c(OC)cccc2)C)ccc(Cl)c(Cl)c1 CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(C2CCCCS2)=O)C(C2CCCC2)C1 N1(C(c2cnc(CC)s2)=O)C2CCC1CC(CNC(=O)C(O)C(F)(F)F)C2 C1(O)(C(=O)NCCNC(=O)Cc2cncs2)CCC(C(F)F)CC1 c1(C(=O)NC2CN(Cc3cncs3)CC2(F)F)ccc2ccccc2n1 C1(NC(C2CC(C)(CC)C2)=O)CCN(C(c2ccc(C(N)=O)cc2)=O)CC1 C1CC(=O)N=C2C=CN(N2)C12CC2.C(CC)(C(=O)NC)=CC CCC(C)(C(=O)N1CC2CCC1CN2C(=O)C=C1CCCCC1(C)C)C(N)=O C12(NC(C(CC)=CCCC)=O)CCCC(CN(C(c3cnc(C4CC4)s3)=O)C1)C2 N1(C(C(C(C)C)NC(C)C)=O)CC2CCC1C(NC(C1(O)CC1)=O)C2 C=CC(C)CC(=O)NC(C)(CNC(c1cscc1Cl)=O)C1CC1 c1(OC(C)C(=O)NCC(F)CNC(=O)CC2CC(=O)C2)ccc(Cl)cc1Cl C1(C(=O)NCC2CC(C)(NC(CSCCC)=O)C2)CNC(=O)CC1C C1(NC(c2c(CC)nco2)=O)CCN(C(=O)Cc2ccoc2)CC1CO N1(C(c2c(OC)scc2)=O)CCN(C(=O)C=CC=C(C)C)C(c2cn[nH]c2)C1 C1(NC(C(c2ccnn2C)C)=O)CCC(NC(c2cn(C(C)(C)C)nn2)=O)CC1 n1(CC)cc(C(=O)NC2CC(CNC(C3CCC(OC(F)(F)F)C3)=O)C2)c(C)n1 CCC(Cc1nc(CCN2CCCCCC2)no1)C(C)(C)C c1(C(N2CCC(O)(CN(C(c3c(OC)noc3C)=O)C)C2)=O)cc(C)cc(C)c1 C(=O)(CS(=O)(=O)c1ccccc1C)NC1CC(NC(CC2CC(CC)OCC2)=O)C1 c1(CNC(C2N(C(CCc3ccc(OC)nc3)=O)CCC2)=O)ccnc2[nH]ccc12 C1(C(=O)NCC(C)NC(=O)C(F)=CC2CC2)CCc2nnnn2CC1 Cc1nc2[nH][nH]cc-2c(=NC2CCC3CN(C(=O)C(F)(F)C(C)(C)O)CC23)n1 CC(C)(O)C#CC(=O)NC1CC1CNC(c1ccccc1N1CCCC1)=O C1(NC(C(Cc2ccc(C)cc2)C)=O)CCN(C(=O)CCC2CC2(C)C)C(C)C1 C1(O)(C(=O)NCCN(C(c2cccnc2)=O)C2CC2)CC2(CCOCC2)C1 c1(N2CCC(=C)CC2)ncnc2n[nH]cc12.C12CCCCC1N2 c1(OC)cc(C(=O)N(C)CC2(O)CN(C(=O)C(O)CN3CCCC3)C2)ccc1C N1(C(=O)NC)CCC(N=c2cc[nH]cc2S(=O)(=O)N2CCC(F)C(O)C2)C1 c1(-c2cccc(CC(=O)NC(c3cccc(F)c3Br)=O)n2)c(O)cccc1F N1(C(c2c(C)c[nH]n2)=O)CC2(CCCN(C(c3ccc(C(C)(C)C)cc3)=O)C2)C1 N1(C(c2ccc(COC(C)C)cc2)=O)CCC(O)(CNC(=O)C(C)O)CC1 C1(CNC(C(C)N(C)C)=O)CCN(C(=O)C(CO)N(C)C)C(C)C1 N1(C(c2ncc(OC)nc2)=O)CCCCC(C(=O)N(C(C)C(C)SC)C)C1 c1(C(=O)NC2(C)CC(NC(C3CC4COCCN4C3)=O)C2)cnn2c1NCCC2 C1(NC(C(C(C)C)CO)=O)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CC2(CCC2)C1 NC(=O)CCCCC(=O)N1CCC2(CC1)CC2NC(c1ccc(=O)oc1)=O C(=O)(C(O)CCC(C)C)NCC1C(CC(=O)NCc2ncc(C)[nH]2)C1 c1(C(N2CCN(C(C=CSC)=O)C(C)CC2)=O)ccc(C#N)c(F)c1Br Cn1cc(S(=O)(=O)NC(C2(C)C=CCC2)=O)ccc1=O N1(C(c2cc(CC)c(CC)o2)=O)Cc2nccn2CC(NC(C2CC2(Cl)Cl)=O)C1 CC(C)CCCCC(=O)NC1CN(C(=O)C(C)(C)Oc2ccc(Cl)cc2)C1 N1(Cc2cn(CC(CNC(C#CCOCC)=O)(C)C)nn2)C(=O)CNC1=O c1(C(N2CC(N(C(C(C(C)C)n3cnnc3)=O)C)C2)=O)cc(F)cc2nn[nH]c12 C(=O)(C(C)(C)C(C)C)N1CCC(CC=C)(NC(=O)C=Cc2ccc(C)s2)C1 S(=O)(=O)(c1ccccc1F)N1C(C(=O)OCc2nc(Br)c[nH]2)CCC1 N1(Cc2nccc(OC)c2)CCC2(CC1)CN(C(c1ccoc1C1CC1)=O)C2 Nc1ccc(F)c(F)c1C(N1CC(NC(=O)Cc2cnns2)CCC(O)C1)=O Cc1sc(Br)cc1C(=O)NCC(C)(CO)NC(C1CCS(=O)CC1)=O C1(CNC(C(COC)NC(c2ccoc2)=O)=O)(CO)CCN(C)C1 c1(C(=O)NCCCC(=O)NC)ccc2nnc(C(F)F)n2c1 C1(CC(N2C(CNC(c3c(C)cc(C)s3)=O)CC2)=O)OCCCC1(C)C CC(CC(C)(C)O)C(=O)NC1CC(N2CCN(C)CC2)C1 C#CCC(C)(C(=O)NCC(c1ccnn1C)O)NC(C1CC(F)(CF)C1)=O N1(C(C2(C(C)C)CC2)=O)CC(F)(CNC(=O)C(F)(F)Sc2cnn(C)c2)C1 N1(C(CSCCCC)=O)CC2CC2(CNC(C2CC2F)=O)C1 CC(C)(Cc1nn[nH]n1)C(=O)NC1(c2cccc(Br)c2)COC1 Cc1cccc(C(=O)NC2CC2CNC(c2cncc(N(C)C)c2)=O)c1C S(=O)(=O)(c1cccc(F)c1)N1CC(NC(c2c(C)ccc(C(=O)O)c2)=O)C(O)C1 C1(C(=O)NCC2(CCC)CC2)CC(NC(C2CCC(F)CC2)=O)CCO1 N1(C(c2ccncc2Cl)=O)CC2CCC1CN2c1nc(Cl)ncc1F CCC(CC)C(C(=O)NCC1COCCN1C(C1OCCCO1)=O)OC c1(SCC(=O)NCC2CN(C(C=CC)=O)CC2O)ccc(NS(=O)(=O)CC)cc1 C1(O)(C(=O)NC2CC3CC2N(C(=O)CC2CCCC2)C3)CC2(CCOCC2)C1 c1(CC)ncc2c(n1)CCC(C(N1CCCC(CNC(=O)C(C)(C)F)C1)=O)C2 C(C(C)(O)CC(=O)NCCCCCCn1cc(C2CC(F)(F)C2)nn1)OC CC1CC(NC(c2cc(OCC(F)F)ccn2)=O)CN1C(c1csnn1)=O C1(CC)CCC(C(N2CCOC(CNC(=O)C(O)CSC)C2)=O)CC1 C1(NC(=O)CCCn2ccnc2)COC2(C1)CN(C(C13CCCC1C3(F)F)=O)C2 N1(C(c2c(C)ccc(F)c2)=O)CC(C2CN(C(c3cc(C(C)(C)C)c[nH]3)=O)C2)C1 C=C=C(C)CC(=O)N=S(C)(=O)c1cnn2c1CN(C(C13CCC(C1)OC3)=O)CC2 C(=O)(CC1=NNC(=O)C1)N1CCC(NC(CCCN(C(C)=O)C)=O)C12CC2 CC1CN(C(=O)C(C2(C)CC2)NC(C2CCC2C)=O)C(C)C(C)(C)O1 C(=O)(C(F)(F)C(F)F)NC1CN(C(C2C(C(=O)OCC)C2)=O)CC1C(F)F CCC(CC(C)C)C(=O)NCC#CC(=O)N(CCCF)C c1(C(C)NCCCF)cccc(N2CCOCC2=O)c1 c1(CNC2CC3CC(CC(=O)OC)C2C3)c(C)cc(CN)cc1C C1(CC(=O)NCC2CC(O)CN2C(c2cccnc2S)=O)(COC)CCOCC1 C1(C(C)(C)C)CN(C(=O)CC(F)(F)F)CCN1C(=O)C(F)CC1CCCC1 C=CC(C)(C)NC(C1(NC(=O)CCOCCN(C)C)CC1)=O c1(C(=O)NCCCCNC(C2C(C)(C(C)C)C2)=O)cnnc(C2CC2)c1 CCC(CC(=O)NCCCc1cccs1)N(C(=O)C(CSC)OC)C c1(-c2cncc(C)c2)ccc(C(=O)Nc2ccnc(CC3CC3)c2)c(C)n1 c1(C(N2C(CNC(=O)CCC3CCOC3)C3CCC2C3)=O)cccc2c1OCO2 C(=O)(C1=CCS(=O)(=O)C1)N1CC2(CC(NC(=O)C(F)CC3CCCCC3)C2)C1 c1(CN2C(C)(C(=O)NCc3nc(Cl)ccc3F)CCC2)ccncc1[N+](=O)[O-] CN1CC(=O)NC12CCN(C(C1CCC(=O)CC1(C)C)=O)CC2 c1(NC2C3(CN(C(C4C(C)(C)CC4)=O)C3)CCC2)ncc2cccnc2n1 Cc1cc(C)n(-c2ccc(CC(=O)NC(C3CN(C(=O)C(C)(C)O)C3)C)cc2)n1 CC(C)(CCCNC(C1CCCO1)=O)C(=O)NC1C2CCCCC12 Cn1c([N+](=O)[O-])cnc1C(=O)OCC1CCCC(C)(C)C1 Cc1ccncc1C=CC(=O)NC(C1(O)CN(C(C2CC3CC3CC2C)=O)C1)C N1(C(C(COC)C)=O)CCN(C(c2ccccc2-n2ccnn2)=O)CC(O)C1 c1(SCC(=O)NCCC(O)CNC(C2CCCCO2)=O)ccc(F)cc1 C#CC1CCCN(C(=NCCF)NCc2cccc(C(F)(F)F)c2O)C1 C(C)(N=c1[nH]nc(C(N)=O)s1)C1(O)CN(C(Cc2c(C)nc(C)s2)=O)C1 c1(C(N(CC(CNC(CC(C(=O)OC)C)=O)O)C)=O)cnc2cc[nH]c2c1 c1(C(=O)NCCC2N(C(CC(CC)C)=O)CCSC2)ccc(F)cc1C#N c1(C(N2C(C)CCC(NC(c3cc(OC)ns3)=O)C2)=O)cccn2nccc12 c1(C(=O)NC2CN(C(C3CNC(=O)O3)=O)C(CO)C2)cc2ncsc2[nH]1 C1(CC#C)CCCN(C(C2C(C)CCN2C(=O)COCC(=C)C)=O)C1 N1(C(C(C)OCCOC)=O)CC2CCC2(NC(=O)C=CBr)C1 C1(CNC(c2nnc(CC)s2)=O)CCN(C(=O)CSC(F)(F)F)CC1C C1(NC(CCC(C)(C)N(C)C)=O)CN(C(=O)OC(C)(C)C)C(C)(CO)C1 C(C)(CC(=O)NC1CC(=CC(=O)NOC(C)C(=O)OC)C1)OC CCCCC(O)CC(=O)N1CCC(F)(CNC(=O)CCc2cc[nH]n2)C1 c1(C(=O)NCCC(CNC(c2cn(C3CC3)nn2)=O)OC)ccccc1C c1(C(=O)NCC(CNC(c2cc(Cl)cc(C)c2N)=O)O)ccc2c(c1)CCC=C2 CCC(C)CC(C)C(=O)N1CCC(CCNC(C2CC(C)(C)C2)=O)CC1 c1(C(N2C(C(=O)Nc3cc(OC)ncc3)CCC2)=O)ccn2cncc2c1 Cc1cc(N)c(C(N2CCC(OC3CN(C(C4CC(F)C4)=O)C3)CC2)=O)cc1C CCCC(C(F)(F)F)NC(C1CCCN(C(c2cc(C)nn2C2CC2)=O)CC1)=O C1(C#N)(C(=O)NC(CN(C(c2ccsc2C)=O)CC)C)CCC1 C1(CNC(C2C(OCC)C2)=O)CC2(CC2)CN1C(C1CC12CCSCC2)=O N1(C(C(CC)OCC)=O)CCC(N(CCO)C(c2cnoc2CC)=O)CC1 c1(C(N2CC(NC(C(CC)(C)OC)=O)C(C)C2)=O)c(N)cccc1Cl Cc1cc(CC(=O)NC(C)CCCNC(=O)C(C)Cc2cnc[nH]2)c(C)s1 S(=O)(=O)(c1ccc(Cl)c2cccnc12)NC(C(c1ccc(CC)cc1)N)=O CC1CCc2[nH]nc(C(N3CC4CC(NC(=O)CCCC(N)=O)C3C4)=O)c2C1 C1(COC(C)C(=O)OCc2ccccc2)CCCN1Cc1nc(C(C)(C)C)no1 C(=O)(C1=Cc2ccccc2C1O)N(CCNC(c1cc(C2CC2)nn1C)=O)CC C1(C(=O)NC(C)CCNC(=O)C(C)CCO)CC(=O)CC1(C)C c1(CC(=O)NCCc2cn(-c3cc(C)cc(N)c3)nn2)cccc2cccnc12 S(=O)(=O)(c1nccs1)NC1CCCN(C(c2cccc(Br)c2F)=O)C1 N1(C(CCCCN(C)C)=O)CC2CC(C1)N2C(C1CC2(CC2)CN1C)=O C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(CNC(C(C(CC)C)O)=O)C12CCC2 N1(C(C2CCC(NC(C(CCC)C)=O)C2)=O)CC(C2CC2)(CC)C1 C12(C(=O)NCC3(NC(Cc4c(C)n[nH]c4C)=O)CCOC3)COCC1C2(F)F c1(C(c2nnnn2CC)NC(c2ccccc2)(CSCC)C)ccc(F)c(Br)c1 N1(CCNC(CCC2(NC(C(C)c3cccs3)=O)CCC2)=O)CCCCC1 c1(C(N2CC(NC(C(C)C3CCCO3)=O)(CO)C2)=O)cc2c(Cl)cc(F)cc2[nH]1 C(=O)(C(F)C(C)(F)F)N1C(C(N2C(C)(C(=O)NC)CCC2)=O)CC(O)C1 C=C(C)CN=C(NCC1CCOC1)N(C)CC(=O)NC(C)(C)C C1(CC)CN(C(c2nn(CC)cc2Cl)=O)CCC1NC(C1(O)CCSCC1)=O N1(CC)CC(C(=O)NC2CN(C(=O)CCc3nc(C)no3)C2)CCC1=O c1(C(=O)NCCC(C(C)C)NC(c2cscn2)=O)c(F)cccc1[N+](=O)[O-] N1(C(c2cc(C)nnc2)=O)CCN(C(=O)CCCCCF)CC1CF C(=O)(CC1=CSC2=NCCN12)NCC(C)NC(=O)C(C)CS(C)(=O)=O CC(=O)CC(C)(C)CC(=O)N(C)CCN(C)C(C1CCC(=O)N(C)C1)=O C12(CC(N3C(C(=O)OC)CC3)=O)CCC1CN(C(=O)CCC1CCCCC1)C2 c1(NC(CCSC)C)ccc(S(=O)(=O)N(C)CCc2c(F)cccc2Cl)c(Cl)c1 C(N=c1[nH]c(=NCc2ccoc2)[nH]c2c1CC(C)CC2)c1cc(OC)c(C)cc1 CCC(C(=O)NCC1COCCN1C(=O)C(C)C1(O)CCC1)C(C)(F)F c1(CC(=O)NCCC(C)NC(C(C(CC)C)NC(C)=O)=O)ccc([N+](=O)[O-])c(N)c1 N#CCCCCC(=O)N1CCC(NC(C2CC3CCC2O3)=O)CC1 c1(NCC#C)nc(C)sc1C(=O)N(CCO)CCc1cccc(Br)c1 CCCCC(O)CC(=O)NC1CCN(C(=O)CCc2c(C)noc2C)C12CCC2 Cc1cc(NC(=O)C(C2(O)CCC2)NC(=O)C#CC2CCC2)cnc1Cl c1(C(=O)NC(CNC(CSCC=C)=O)C(C)C)cccc(C)c1N N1(C(C2CCN(CC(C)C)CC2)=O)CCN(C(=O)CC2CC2(C)C)CC(CO)C1 CCCCC(O)CC(=O)N(CCCNC(c1ccc(C)nc1)=O)CCC c1(C(=O)NC(CN(C(=O)CCn2cccn2)CC)C)cnn(C(C)C)c1Br C(CC(C)C)(C(=O)NCC(O)C(=O)NC)N(C(C1CC(=C)C1)=O)C N1(C(CC(=O)NCC)=O)CC2(CNC(=O)CC(C)(C)CC)CC2(C(F)(F)F)C1 O=C1C2COCC1CC(C(=O)NC1CCN(C(C3CCC3)=O)CC1CO)C2 c1(C(N(CCC(C)NC(c2cc(N3CCCC3)ccn2)=O)C)=O)ccncc1O C1(C(=O)Nc2ccc(F)cc2CO)CC2(C1)CN(C(=O)CC1CC1)C2 C1(OC)CN(C(=O)C(CCC(C)C)NC(C2COC(=O)N2)=O)C2(CCC2)C1 CN1CCC(C(=O)NCC2CCC(NC(c3cc(C(F)(F)F)cs3)=O)C2)CC1=O C(N=c1ncc(F)c[nH]1)C1N(C(CCCC(=C)C)=O)CCCC1 c1(NCC(CNC(CC(C)C(F)F)=O)O)ccc([N+](=O)[O-])cc1F C(COC)(CC(=O)N1CCC(O)(CO)C1)NC(C1CCC(CC)O1)=O N1(C(C2(C#N)CC2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C2(CCC2)C1 CC(CCC(C)(C)C)C(=O)NCC(c1ccccc1)N(C(=O)CP(C)(C)=O)C c1(N2CC3CN(C(=O)Cc4cc(F)ccc4Cl)CC32)ncc2cc(Br)cnc2n1 N1(C(c2cccc(C)c2)=O)CC2CC(CNC(=O)CN3CCOCC3)CC1C2 c1(OC(C(=O)NCC2CC(NC(C(C)C)=O)C2)(C)C)ccc(F)cc1 C(CC1=CCCCCC1)NC(CC1CC(NC(C2(CC(C)C)CC2)=O)C1)=O c1(CC(=O)N(C2CCCN(C(c3c(CC)nns3)=O)C2)C)ccc(C#N)cc1 C=Cn1nncc1C(=O)NC(c1ccccc1)CNC(=O)C=CCOCC c1(C(=O)NC2C(NC(C(C=C)(C)C)=O)CC2)c(F)ccc(C)c1Cl C1(C(N(C2CCN(Cc3cnsc3)CC2)CC#C)=O)CCCC(F)C1 CC1(C(=O)NCC2(NC(c3cccc(CC(F)(F)F)c3)=O)CCC2)COCCO1 Cn1nc(CNC(=O)NCC2(NC(=O)OC(C)(C)C)CCC2)cc1Br c1(CNC(=O)NCC2(C(=O)OCC)CC2C(F)(F)F)c(C)ccc(C)c1O Cc1cc(C(N2CCCC2(C)C(=O)Nc2cncnc2O)=O)ccc1Br c1(C(N(CCNC(=O)COc2ccsn2)C2CC2)=O)ccn2ccnc2c1 c1(C(N(CCC(=O)NC(C2CCCC2)CC)C)=O)ccc(O)nc1 c1(NC(C(=O)NC2(CCCNC(C=CC=CCC)=O)CC2)C)ccc(F)cc1 C1(NC(=O)OC(C)(C)C)CC2CC(NC3CCN(C4CC4)C3=O)CC12 c1(SC)ccc(C(N2CC3C(NC(c4cn5c(n4)SCC5)=O)C3C2)=O)c(Cl)c1 CC1(NC(c2ccncn2)=O)CN(C(=O)C(C)(C)c2ccc(Cl)s2)C1 C(C(O)CC(F)(F)F)NC(C(C(C)NC(c1cccc(CO)n1)=O)C)=O Cc1nc(CC(=O)NC2CC(O)(CNC(c3ccsc3CN(C)C)=O)C2)sc1C CCCCC(CNC(c1ccc(C(F)(F)F)nn1)=O)NC(=O)C=CCF c1(C(=O)NCC2(COC)N(C(C(CCCC)O)=O)CC2)ccc2c(C)noc2c1 CCCC(CNC(=O)C(C)(C)C(C)(C)O)C(=O)NCC1CC(O)C12CCC2 C1(NC(c2ccc(OC)s2)=O)CCCCC1CNC(c1c(C)[nH][nH]c1=N)=O c1(NC(C2(C)N(c3cc(OCC)ncn3)CCC2)=O)ccnc(Cl)c1OC c1(C(N2C(CNC(c3c(C)snc3)=O)CCCC2)=O)cc2c([nH]1)CCC(C)C2 c1(C(=O)NCC2CC(CC(=O)OC)C2)c(Br)ccc(F)c1I C12(NC(=O)NCC3CCC(N4CCOCC4)CC3)CCCC1C2(F)F C1(C(N2CC3(CCNC3=O)C2)=O)N(C(C2CC23CC3)=O)CC12CCCC2 C(C)(CNC(c1ccsc1CC)=O)(CC(C)C)NC(c1cccc(CCC)c1)=O N1(Cc2nc(-c3ccn(C)n3)nn2CCN(C)C)CCC2(CC1)N=N2 c1(C(N)=O)cc(C(=O)NCC(O)Cn2cc(CC(C)(C)O)nn2)c[nH]1 C1(NC(CSCCCCC)=O)C=CC(CC(=O)NC(C)CC(C)O)C1 CCC(C)CC(=O)N(CCNC(=O)C(N1CCC(O)CC1)C)C(C)C c1(C(=O)NCC(F)(F)F)c(-c2ccccc2C(=O)NC2CCCC2)cncc1F N1(C(C2(CC)CCOCC2)=O)CCC(C)C(NC(c2ccncc2)=O)C1 CCC(CC(=O)NCC(O)CN(C)C)N(C(=O)C(F)n1ccnc1)C C1(NC(C2(CNC(C(CC=C)NC(C)=O)=O)CC3(CC3)C2)=O)CCOC(C)(C)C1 C1(NC(c2nc(C)sc2)=O)CN(C(=O)CCc2ccc(F)nc2)CC2CCCC12 c1(C(=O)NC(C(C)C)CNC(=O)CC2CC=CCC2)ccc2c(=O)cc[nH]c2c1 c1(C(=O)NCCC2CCCN(C(COCCC)=O)C2)ccc(C(C)CC)nc1O C1(=CC(N2CC3C(NC(=O)C=CCn4cncn4)C3C2)=O)CN2CCC1CC2 c1(C(N2CCC(CC=C)(NC(=O)C(O)CCSC)C2)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(CC2N(C)CCC2)=O)CCCCN(C(c2cncnc2)=O)CC1 CC(CN(C(=O)C(F)C(C)C)C)N=c1ccn2c(Br)cnc2[nH]1 c1(OC)cc(Cn2nc(C(C)O)nc2CC(C)P(C)(C)=O)cc(OC)c1OC CCN(C(C)c1cccc(C(F)(F)F)c1)N1CCN(C)CC2(CCCCCC2)C1 N1(C(c2[nH]cc(CN(C)C)c2)=O)Cc2ccccc2C(NC(=O)C=CCF)C1 c1(Nc2ccccc2)ccccc1O.n1(C(CN)=O)nncc1C(CCC(F)(F)F)=O C#CC1(C(=O)NC(CNC(=O)C(F)(F)c2nc(CC)cs2)CC)CCCC1 Cc1noc(Cl)c1CC(=O)NCCN(C(c1conc1C(C)C)=O)CC1CC1 c1(C(=O)NCC(CNC(c2cc(CCC)ncc2)=O)(C)OC)cc(C)cc(C)n1 C1(N(C(C(=O)NC2COC2)c2cscn2)C)CCC(C)(C)C1 CN1CCC(CNC(=O)N=c2ccn(CCS(C)(=O)=O)[nH]2)c2ccccc21 c1(C(=O)NC(C)CN(C)CCOC2CCOC2)ccc2ccc(Cl)cc2n1 C=CC1CCCCN1C(=O)C(C(C)(C)C)NC(C1CC(C)N(C)C1)=O Cc1oc(CNC(=O)CCCC#N)nc1C(N1CCC(C(C)C#N)CC1)=O Cc1cn(C(C)(C)C(=O)NCC(C)NC(=O)CCc2nncn2C)cn1 C(CC(O)CCO)NC(C(C1CCCC1)NC(=O)CCc1ccccc1)=O c1(C(=O)NCC2CCN2C(=O)C=C(Cl)Cl)ccc(=O)n(CC(F)(F)F)c1 CC(C)(CCCF)C(=O)NC1CC(CNC(C23CCCC2C3(F)F)=O)C(O)C1 [N-]=[N+]=NCCC(=O)N(CCC(=O)NC1CCCC(C(N)=O)C1)CCCO CC(O)(CC(F)F)C(=O)N1CCCC(NC(C2(C(F)(F)F)CCOCC2)=O)C1 C(CC(C)C(=O)N1CCCC1C=CC(=O)NCC1C=CCOC1)=CC c1(C(C(=O)NC(C)COCC(F)(F)F)F)ccc(Cl)nc1 c1(C(N2CCCC(CNC(c3c(OC)csc3)=O)C2)=O)ccc(O)nc1Cl N1(C(CC#N)=O)CCC2(C1)CN(C(=O)Cc1csc3cccc(F)c13)CCO2 C1(N(C(C2CN(C)C(=O)N2)=O)C)CCC2CN(C(c3csc(O)n3)=O)CC12 c1(COC)ncc(C(N2CCCC(NC(c3n[nH]c(SC)c3Cl)=O)C2)=O)c(O)n1 Cc1cc(C(=O)NCC23CC2CN(C(c2ccc(C(F)F)cn2)=O)C3)cc(F)c1 CC(F)(F)C(=O)NCC1CC(NC(C2CC2[N+](=O)[O-])=O)C1 CC(C)C1=CCC(NC(=O)COC(C)(C)C)CC1.c12ccccc1SC2 C1(Nc2ncn(C)c(=O)c2)(CNC(=O)C(=O)NC2CC2)CCC(F)(F)CC1 n1(CC(=O)NCC2(NC(=O)CSC3CCCC3)CCCC2)ncn(O)c1=O N12CCC(CC13CC3)CC(=O)COC2=O.c1(C2C(C(C)(C)C)C2)ncco1 CC1CN(C(=O)C(F)F)CC1CCc1cn(Cc2nc(C(N)=O)cs2)nn1 C(C(=O)O)(C(O)c1cccnc1)NC(C(n1cc(Cl)cn1)C)=O c1(C(=O)NC(C2(O)CN(C(C=CCC)=O)C2)C)cc(C)c(Cl)cc1C N1(Cc2cccc(OCC)n2)CC2(CCC(NCc3cc(C)cc(Cl)c3)C2)C1 c1(CC(=O)NCCC2CC(NC(C(C)c3ccco3)=O)C2)ccc(Cl)cn1 C(CCCCC(=O)NCC1(O)CC(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1)SC C1(NC(c2cn(CCOC)nn2)=O)C=CCN(C(=O)C(F)C2CCC2)C1 Cc1c(C(N2CC(O)CC2CNC(C2CC3(CC3)CO2)=O)=O)nn(C)c1Br C1(c2ccc(CC)cc2)CN(C(C2(CCF)CC2)=O)CCN1C(C1SCCS1)=O C(C)(C)(CC(F)C(=O)NC(C)C(=O)N(C)C1CC1)NC(c1c(CC)cco1)=O c1(C(=O)OCC)c(C)nc2scc(C(=O)NC)c2c1C.N12CC(C(C)C1)NC2=O C(=O)(CC(CC#N)c1ccccc1)NCC(C)NC(C1(c2ccccc2F)CC1)=O Cc1ccc(C(F)(F)F)cc1C(=O)NCC1CC1NC(c1ccc(F)cn1)=O C1(C(=O)NC(C)C(C)(C)NC(=O)CS(=O)(=O)C2CC2)Cc2cc(Cl)ccc2O1 c1(CC)noc(C(N2CCC(N(C(=O)Cc3ccoc3C)C)CC2)=O)c1C Cc1cccc(C(=O)NCC(C)C(=O)NC(C2CCC2)C2CC2)c1F N1(C(c2c(C)cccc2N)=O)CC(C2CCCN(C(c3cn(C)nc3O)=O)C2)C1 C1(CCNC(Cc2nnc(C)s2)=O)CSCCN1C(=O)CSC(F)F c1(C(=O)NC(C)Cc2cccc(C(F)(F)F)c2)cc2nccc(C(F)F)n2n1 n1(CC)nc(C(=O)NCC(O)CNC(=O)CCc2csc(=N)[nH]2)c(Br)n1 c1(OC)cnc(C(C)C)c(C(=O)NCCNC(=O)CNC(c2ccoc2)=O)c1 c1(C(=O)NCC(CC(=O)NCC(C)CN(C)C)C2CCC2)ccc([N+](=O)[O-])o1 c1(CC(N2CC3CN(C(c4c(C)c[nH]n4)=O)CC3C2)=O)ccc([N+](=O)[O-])cc1F N1(C(c2cn(CCC(F)(F)C(F)F)nn2)C(=O)NC)CCCC1C1OCCO1 c1(C(=O)NC2C(CNC(C=CC(=O)OCC)=O)C2)c(C(F)(F)F)cccc1F c1(C(N2CC(C(C)NC(=O)C(C)(Cl)Cl)OCC2)=O)ccc(=O)n2c1CCC2 c1(NC(C2(CNC(c3ccc(OC)cc3)=O)CC2)=O)scc(O)c1C#N C#CCCCC(C)C(=O)NC1C2CCN(C(=O)CCc3ccncc3)CC12 c1(C(C(=O)NC(CNC(Cc2nc(C)[nH]n2)=O)CO)(C)O)ccc(F)cc1 CCC(Cc1cccc(F)c1)C(=O)NCC(c1cn(C2CC(O)C2)nn1)(C)O c1(C(=O)NCC(CC(C)C)NC(=O)CSC(F)F)ccc2nc(O)[nH]c2c1 C#CC1(C(=O)NCc2nonc2C)CCN(C(=O)C(O)C2CC2)CC1 N1(C(C2(F)CCN(C)CC2)=O)CCC2(CNC(=O)Cc3ccsc3)CCCC12 CC(C)(CNC(=O)C(C1CCOCC1)N1CCCC1)Cn1cc(C2CC2)nn1 CC1(C)CC(NC(=O)C=CCO)CCN(C(C2CC3(CCCC3)CO2)=O)C1 C(=O)(C(C)C(F)(F)C(F)F)N(CCNC(C(C(CC)(C)C)O)=O)C(C)C c1(CC(N2CCN(C(COCCCC)=O)C3C2C3)=O)c[nH]c2c(CC)cccc12 N1(C(C(CCCC)C)=O)CC2(C1)CN(C(=O)CCCOCCOCC)CCO2 C1(NC(c2c(C)nc[nH]2)=O)CN(C(c2cncc(Cl)c2)=O)CCC1F Cc1ccc(O)cc1CN1CC2(CC2)CC1C(=O)NCCC(C)CO Nc1c(C(=O)NC(c2ccccc2Cl)CCO)cc(F)cc1Br C#CCCCC(C)C(=O)N1CC=C(C(=O)NC(C)(C)CCO)CC1 O=C(C1=CCCCO1)NC1CCN(c2ncnc(O)c2Br)C1 C(=O)(C1=COCCO1)NCC1(CNC(=O)CCc2cn[nH]c2)CC12CCC2 c1(N2CCC(C(C)NC(c3cnc(Cl)cn3)=O)CC2)nc(C(C)(C)C)nc(=N)[nH]1 N1(C(C(CCSC)NC(C)=O)=O)C2CCC1C(F)C(NC(c1coc(Cl)c1)=O)C2 C=CC1(C(=O)N(C)CC)CCN(C(c2ccc(N)c(F)n2)=O)C1 c1(C(=O)NC(CNC(CN2CC(C)C2)=O)C)ccc(-c2ncno2)cc1 N1(C(C2C(OC)(OC)CC2)=O)CC(CNC(c2ncoc2C)=O)CC1(C)C CC1CCN(C(=O)CCCc2cnn[nH]2)C(C(=O)NCCCC2CCCCO2)C1 C1(C(=O)NC2C(NC(=O)CCc3ccsc3)C2)CCCC2(CCC2)O1 c1(C(N2CC(C(N(C)CC3C(C)C3)=O)OCC2)=O)cc(F)ccc1F c1(C(=O)NCC)ccc(C(CC)NC(C2CCCN2N=O)=O)cc1 c1(CN(C)CC2(C)CC2(F)F)cc2cc(Cl)ccc2s1 CC(C)CCCN=c1[nH]c(N2CCC3(CCCN3C)C2)nc2ccc(Cl)cc12 c1(OC)cc(-c2nc(CCCOC)nn2C(C)C(F)(F)F)c(C)cc1C1CC1 C1(C)(CC)C=C(C(=O)NCC2CN(C)CCN2C(c2csc(C(C)=O)n2)=O)C1 C(C(=O)N(C1CCCN(C(c2c[nH]c(Br)c2)=O)C1)CCO)(C(C)C)OC C=C(C)CC(C(=O)N(CCCNC(c1ccc(C(=O)OC)s1)=O)C)NC(C)=O c1(C(=O)NCC2CC(NC(c3c(N)ccc(O)c3)=O)C2)ccnc2c1CCC2 N1(C(c2ccc(SC)o2)=O)CCCC(O)(CNC(=O)Cc2cc(C)cc(C)c2)C1 N1(CC(=O)N(C(=O)Cc2ccc(F)c(Cl)c2)C(C)C)CCCCC(C(C)(C)C)C1 C1(CNC(CNC(=O)OC)=O)CC(OC)CN1C(=O)C(C)(C)NC(=O)C=COC C1(OC)CC(NC(c2cncc(C(C)C)c2)=O)CN(C(=O)C(F)OC(F)(F)F)C1 N1(C(c2c(C)nc(=N)[nH]c2)=O)CC2(NC(=O)CC3CCN(C)C3=O)CCC1CC2 C1(NC(CNC(c2ccc(C)s2)=O)=O)CC2CN(C(C34CC(C3)C4)=O)CC12 C1(NC(C2N(C)CCC2)=O)CN(C(c2cc(O)ccc2F)=O)C2(CCOCC2)C1 N1(C(c2scc(OC)c2OC)C(=O)NCCC)CCCC(C)(C)C1C(=O)OC C1(NC(CSCC)=O)CN(C(=O)C=Cc2cncc(O)c2)C(C)(C)C1 N1(C(C(C)OCCC=C)=O)CCC2(CCOCC2)C(NC(=O)CC(C)CCC)C1 C(=O)(C(C#N)CC)NC(CCC)CNC(c1ccncc1OC(C)C)=O CCC(C(=O)NC1(CO)CCN(C(=O)C(=O)NC)C1)C(=O)NCCOC c1(C=C(COC(c2c(CCC)n[nH]c2)=O)C)ccc(OC)c(OC)c1OC N1(C(=O)Nc2cnc(C)s2)CC2(CCN2C(=O)Cc2ccc(Cl)cc2)C1 c1(C(=O)NCC(C(C(C)C)C)NC(c2ccc(Cl)cn2)=O)cnc2[nH]ncc2c1 C(C(O)(C(=O)NC1CC2C1CCN2C(C1CCCC(=O)N1)=O)C(F)(F)F)N(C)C C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(C)C2CC2)CC1F c1(C(=O)NCCOC2CN(C(C(C)SCC)=O)C2)csc2cc(OC)ccc12 C1(NC(Cc2c(C)cccn2)=O)CC(F)CN(C(C2CCC(=O)N2)=O)C1 CC1C(=O)N(C)CCN1C(=O)CCC1(NC(c2ccncc2O)=O)CCC1 C(=O)(C(C)(C)C(=O)NCC(C1CCN(C(c2cnc(O)c(C)c2)=O)CC1)O)NC N1(C(c2c(CC)ncs2)=O)CCCC2CN(C(=O)C(c3ccccc3C)C)CC12 c1(C(=O)NC2(CN(C(C3C(OC)C3)=O)C)CC2)cc(=O)c2ccccc2[nH]1 C1(NC(C(CC)OC2CCCCC2)=O)CN(C(=O)C=CC=C(Cl)Cl)CC1SC c1(C(=O)NC2C(NC(C3(C(F)(F)F)CC(=C)C3)=O)COC2)cc(F)cnc1OC N1(C(CNC(C2CCCCCC2)=O)=O)CCOC2CCCCC12 c1(C(=O)NC(C2CCCCC2)CNC(C2N(CC)CC2)=O)cscc1Cl C=CCC(CC=C)C(=O)NCC(CCCC)NC(c1ccnc(CN(C)C)c1)=O CC1=C(C)CC(C(=O)NCC(C(=O)NC2CN(C(N)=O)C2)N(C)C)CC1 CC1Cc2cc(C(=O)NC34CCC(C3)N(C(=O)CN(C)C3CC3)C4)ccc2O1 C1(CN(C(=O)COCCCF)C)CCCC(NC(c2ncccc2F)=O)C1 c1(C(=O)NC(C2CCN(C(c3c(C)c[nH]n3)=O)C2)(C)C)nn(C(F)F)cc1Cl C(=O)(C(CCC(C)C)CC(=O)OC)NCC1CC(F)(C(=O)NC)C1 C1(CN(CC)CC)CCCCN1C(=O)CCc1ccc(N(C)C)nc1 N1(C(C(C)(C)OC(C)C)=O)CCN(C(C2(C)CCCS2)=O)CC12CCC2 n1(CC)cc(Cl)c(C(=O)NC(C(C)NC(c2conc2COC)=O)C(C)C)n1 c1(C(=O)NCc2cc(C(N(CC(C)O)CCF)=O)on2)cc2occc2[nH]1 c1(CC(=O)NCCN(C(=O)C2=C(C)CCC2)CC)ccc2ocnc2c1 c1(COC)ccccc1CC(=O)N(CCNC(c1cc(=O)cc[nH]1)=O)CC1CC1 C12(NC(COCCSC)=O)CCC(CC1)N(C(=O)CC1CCCS1(=O)=O)C2 n1(C(C)C)nccc1-c1cn(C2CC(NC(C3CCC(C(N)=O)C3)=O)C2)nn1 c1(CC(N2CC(CC(C)NC(c3c(CC)cno3)=O)C2)=O)ccc(F)cc1 c1(C(=O)NC2CN(C(C(CC)C(C)O)=O)CC2(C)C)ccnc2[nH]ncc12 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CN(C(=O)C(F)C1=CCCCC1)CC2CO N1(C(c2c(C)cccn2)=O)CCn2c(CNC(c3cccnc3N)=O)nnc2C1 C1(NC(C(c2ccccc2)OC)=O)COCCC1NC(c1nc(C)oc1C)=O C(CCCC(=O)N1CCC(F)(CNC(C2C3CN(C)CC23)=O)C1)SC C1(CNC(c2ccc(SCC)nc2)=O)CCC(C)CN1C(=O)CNC(N)=O c1(SC)cc(C(=O)NCCC2(O)CCCNC2)cc(SC)c1 N1(C(c2cc(C)ns2)=O)CCN(C(=O)C(n2nccc2C)C)C2CCCC12 C1(CCNC(c2cc(OCC)no2)=O)CC(F)(F)CN1C(=O)C(N)=O C1(NC(C2(CC)CC2)=O)CC2CC1CN2C(C1(c2ccccc2)CC1)=O C1(C(=O)NCC2CCCN(C(c3ccccn3)=O)C2)CC12CCC(F)(F)CC2 C1(OC)(CNC(=O)C(O)CNC(c2cc(C)ns2)=O)CCOC1 C1(CCOC)(NC(C(=O)NC(c2ccccc2)CSCC)=O)CCCC1 C(=O)(C(C)C(O)C(C)C)NCCN(CC(C)O)C(c1nc(C(C)C)oc1)=O CC1(C)CCC(CC(c2nnnn2C2(C)CC2)NCc2cc(C(C)(C)C)no2)C1 CCC(CC)C(C)C(=O)NCC1(C(N2CCCC3C(=O)NCC23)=O)CC=CC1 c1(C(N(C2CC(NC(CC3(CC)CCC3)=O)C2)C)=O)nc(C)oc1C N1(C(C(CC(C)C)C)=O)CCCN(C(C2(n3cc(Cl)cn3)CC2)=O)CC(CO)C1 c1(C(=O)NCC2(C(C)(C)O)CN(C(C3C(CC)CCC3)=O)C2)cccc(CO)n1 N(C1CCCc2sccc21)C(CCCCCO)c1n(CC(=C)C)nnn1 C1(C)(CC)CC1C(=O)NCC1CC(C(=O)NCC(C)(C)n2ccnc2)C1 CCC(CC(=O)NCC1CN(C(C2OCCC2(C)C)=O)CCO1)OC C1(OC)(CNC(C2CC(F)(CO)C2)=O)CCN(C(=O)CC2OCCC2(C)C)C1 C(=O)(C(C#N)C(C)C)NCC(c1ccccc1)N(C(c1[nH]cc(C)c1)=O)C c1(OCC)cnc(C(=O)NC(CNC(=O)CCOC2COC2)CC(C)C)cn1 c1(OC)nccnc1C(=O)NC1CC(C)(NC(C2CCCN2C(C)=O)=O)C1 C1(C(=O)OCc2coc(Cc3ccccc3)n2)CNC2(CC2)CO1 CC(C)CC(C(=O)Nc1cc(Cl)cnc1O)NC(=O)C(C)CC#N Cc1c(F)cc(C(=O)NC2CCCCN(C(=O)C=Cc3cscn3)C2)c(F)c1N Cc1ncsc1C=CC(=O)Nc1cccc(NC(=O)C(F)(F)c2cncs2)c1 C1(COC)CCC(C(=O)NCC(C(=O)NCC2(C)CCOC2)N(C)C)O1 N1(C(C(CC)C)=O)CC2(C(=O)NC3CC(n4cncn4)C3)CCC1CC2 N1(C(C(C)=NOCC#N)=O)CCCC(CC(=O)N(C(C)CO)C2CC2)CC1 C(=O)(C(C)(C)CC(=O)N1CC2CCCC2(NC(c2ccoc2C)=O)C1)OCC C#CC(C)(C)C(=O)N1CC2CC2(CNC(=O)COCC2CCCCO2)C1 c1(C2(C(=O)NC3C(NC(c4[nH]cc(C)c4)=O)C3)CC2)cc(F)cc(C#N)c1 c1(C(=O)NCC2(CNC(C(C(C)O)N(C)C)=O)CC2)cc2cc(O)ccc2[nH]1 c1(C(N2CC(CNC(C(C)(C)OCC)=O)C3C2C3)=O)nc(C)ccc1C C1(CC(=O)NCCC(CNC(CC=CCC)=O)O)CCC(C(=O)OCC)CC1 N1(C(COCCCC#C)=O)C(CNC(=O)C2=C(Cl)CCOC2)CC2CCCC12 c1(OC)ccc(C(=O)N(CCC(C)NC(C2CC23CCCC3)=O)C)c(O)c1F C1(C(N(CC(C)(C)CNC(=O)Cc2ccoc2)C)=O)CCCCS1(=O)=O CCN=c1ccc(C(=O)NCC(C)(C(C)C)NC(=O)CC2CC23CC3)c[nH]1 C1(NC(C2C(CC)OCC2)=O)CC12CCC(NC(=O)C=C1CCN(C)CC1)CC2 Cc1cc(C)c(C(=O)CCCC(=O)OCCc2cc(C)n(C)n2)c(C)c1 O=S(=O)(c1c[nH]ccc1=NC1CCC(F)C1)NC1CCN(c2cccc(Cl)c2)C1 N1(C(CC(C)C(=O)c2cccc(F)c2)=O)CC2CCC1CN2C(=O)C=CC1CC1 c1(C(=O)NCC2CCN(C(C3(CC#C)CCCO3)=O)C2)cc(C)c(C)c(C)c1 Cn1nc(CN2CCC(O)(c3ccccc3Br)C2)cc1C1CC1 [N-]=[N+]=NCC(C(=O)N1CCSC2(CC2)C1)NC(=O)C(O)C1CCCC1 CC1CC(CNC(c2ccn(-c3ccccc3)n2)=O)CN1C(=O)CSCCC#N c1(OC)ccccc1C(CNC(c1ncc(F)cn1)=O)NC(=O)Cc1ccon1 N1(Cc2ccc(OC)c(Br)c2)CCn2c(nc3c2CCCC3)C1 CCC1CC(=O)N1.C1(CCNC(=O)COC)(OCCOC2CC2)CCOCC1 C1(C(N2CC(O)(CCNC(COC3(C)CCC3)=O)C2)=O)CC(C2CCCC2)C1 c1(C(=O)OC)cnc(C(=O)NC(C)CCCNC(=O)C(C)n2ccnc2)cn1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(COC)(CNC(=O)C(C)CC(C)C)C1 c1(C(=O)NCCN(C(C(c2ccccc2)SC)=O)C)cc2cc(Cl)ccc2s1 C(=O)(C#CC1(C)CCCO1)N1C(C(=O)Nc2c(OC)n(C)nc2C)CC=CC1 C1(NC(c2cnc(C3CC3)s2)=O)COCCN(C(c2ccccc2Br)=O)C1 c1(C(=O)NCC2C(CNC(c3nncn3C3CC3)=O)C2)cn(CCO)nn1 C1(CC(=O)NCCCC2N(C(CCC(=O)OC)=O)CCCC2)CCCCC1(F)F c1(C(=O)NC(C(C)NC(c2csc(S)n2)=O)CO)ccc(Cl)c(Cl)c1 c1(C(=O)NC(c2nocc2C(=O)NCc2ccncn2)C)cccc2cncn12 C#Cc1ccc(NC(C2CN(C(C3(C#N)CCCCC3)=O)CCO2)=O)cc1 c1(SC)ccc(CN(C)C(N2CCOCC2C2CCC2)=O)cc1 C=C(C)CCCC(=O)NCc1nc(C2CCN(C(C3CC3(F)F)=O)CC2)n[nH]1 N1(C(c2c(C)nc(Cl)cc2)=O)CCC2(CCCN2C(=O)C(C)n2cccn2)CC1 CC(C)C(C)(CNC(C12CC(C)(C1)C2)=O)NC(=O)CCc1ccsc1Cl CC1CC(=O)NCCN1c1nnnn1C1CCC2CC2CC1 CN1CC(C(=O)NCCNC(=O)CN2CCOCC2=O)CC1=O c1(N(C)CCC2CC2)ccc(S(=O)(=O)NCC(O)CCC2CC2)c(Br)c1 C=C(CNC(=O)C(c1ccccc1)OC(C)C)CCNC(=O)CC1CSCCS1 c1(NC(=O)CCF)ccc(Cl)c(CNC(c2cnccc2N2CCOCC2)=O)c1 C=CC(C)(CCOC)C(=O)NC(C)CCCNC(C1(F)CCCN(C)C1)=O C1(CNC(c2c(CC)n[nH]c2)=O)CN(C(=O)C(=Cc2cccnc2)C)C(C)(C)C1 N1(C(C2C(=C)C2)=O)CC(F)CC1CN(C(=O)C(CC)=CCCC)C C=Cn1nccc1C(=O)N(C1CCC(O)C1O)Cc1c(OC)nsc1OC c1(-c2nccc(C(C3CCN(C)CC3)(C(C)C)C)c2)ccc(Cl)c(Cl)c1 C(=O)(CCCN=[N+]=[N-])NC(C=CC(=O)Nc1c(C)n(C)nc1)C C1(C(N2CCC(N(C(c3ccc(F)s3)=O)CC)C2)=O)CCCC(OC)C1 N1(S(CC)(=O)=O)CCC(C(N2CC(CNC(c3cn[nH]c3)=O)(OC)C2)=O)CC1 CCC(CC)CC(=O)NCC1CCC1C(=O)NC1(C(C)(F)F)CCC1 CCC(C(=O)NC(C1CCN(C(c2cnc3n2CCC3)=O)C1)(C)C)C(C)C C1(NC2(CNC(CCN(C)C3CC3)=O)CC2)C2CCCCC12.C12(CC1)N(C)C2=O C(CCNC(C1(C#N)CC1(C)C)=O)(C(=O)NCc1nn[nH]n1)OC CC(C)C(C)(CN=c1[nH]c(=NCCC(C)CO)[nH]c2cc(CO)ccc12)NC C(=O)(C(C)(C)CC(F)F)NC1C(C(=O)NCC(CSC)(C)C)CCC1 c1(OC)cccc(C(CNC(C)=O)NC(C2C3CCC2(c2ccncc2)C3)=O)c1 c1(C(N2CCC(CN(C(C(C(CC)CC)C)=O)C)C2)=O)cc2c(cc1Cl)OCO2 c1(C(N2CCCC2)=O)ccc2c(c1)CN(N1CCC([N+](=O)[O-])CC1)C2 O(NC(=O)CCCC(C)NC(C1CCOC1C(C)C)=O)CC(=C)C C1(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)CCCCC(C)(C)C1 N1(C(c2nc(CCC)sc2)=O)CC(C2CN(C(c3cccc(F)c3C)=O)C2)C1 CC(CC(=O)N(CCCCN(C(=O)CN1CC2C=CC1C2)C)C)CC(C)(C)C c1(C(N2CC(OCCNC(CC(C)CF)=O)C2)=O)cc(F)c(O)c(F)c1 c1(OC)n[nH]c(-c2nc(CC(C)OC)nn2-c2ccnn2C)c1Cl c1(C(N(CCCNC(CCN(CC)CC)=O)CC)=O)ccc(C)c(P(C)(C)=O)c1 c1(-c2occ(C)n2)cc(CN2CCCC(C(F)(F)F)(CO)C2)ccc1C C1(OC(=O)CN(C)C(c2ccc(C)cc2)=O)CC(O)CN(C(=O)OC(C)(C)C)C1 CC(C)CC(C)(C)C(=O)NCC1CCC(C(N2CCCCCC2C)=O)O1 O(NC(=O)CC(C1CC1)NC(=O)CNc1ncccn1)CCCC#C C12(CNC(CC(C)SC)=O)CC1CN(C(c1cnn(CC(C)C)c1)=O)C2 Cc1cc2c(C(=O)N=c3ccn(-c4ccc(F)cc4C#N)[nH]3)cccc2[nH]1 C1(NC(c2nc(C(=O)OC)sc2)=O)CC2CC(NC(=O)C(C)N(C)C)CC2C1 N1(C(C)=O)CC2CCN(C(C3CCN4CCC3C4)=O)CC12.C(=O)CCS(C)(=O)=O C1(=CC(=O)N(C(C2CCCCC2)CNC(=O)C(N)=O)C)CCCCC1 C1(O)(CCOC)CCN(C(=O)Cn2nc(C)nc2C)CC1 N1(C(CCC(C)N(C)C)=O)CCC2(CC(NC(c3ccsc3)=O)C2)C1 c1(C(N2CC3CC2CN3C(c2cccc3cncn23)=O)=O)ccc2ncsc2c1 N1(C(C#CCNC(C2(C)CC(=C)C2)=O)=O)CCC2(CCOC2=O)C1 C(CC(C(=O)NCC(O)CCO)NC(=O)C=CC1CCCC1)OCC c1(C(N(C2CCCCN(C(C(C=C)C)=O)C2)C)=O)cc(C)cc([N+](=O)[O-])c1 c1(NC(COC)=O)cccc(C(=O)NCc2ccc(CC(F)(F)F)cc2)c1O c1(OC)ccc2c(=NCCC3CC=CC3)[nH]c(=NCc3cccc(O)n3)[nH]c2c1 C1(CNC(c2ncccc2CO)=O)CC(O)CN1C(c1cnc(C2CC2)s1)=O N(C1CCc2c(C(F)(F)F)cccc21)C(C1C(CC)OCC1)=O c1(C(N2CCN(C(CS(CC)(=O)=O)=O)CC2CCO)=O)nccn2nccc12 C1(C(=O)NCCn2cc(C3(OC)CCOC3)nn2)CCS(=O)(=O)CC1 C1(CNC(c2cnc(C)nc2)=O)COC(C)(C)CN1C(C1CCCN(C)C1)=O C(=O)(C1=C(Cl)CC1)NC(CC)(C)CNC(=O)CCc1ncc[nH]1 N1(C(C2C=CCC2)=O)CCC2CCC(C1)N2C(c1ccc(O)cc1Cl)=O N1(C(C)=O)CCCC(C(N2CC(O)(CNC(C34CC(CCO3)C4)=O)C2)=O)C1.OC CC1CN(C(=O)Cc2cn[nH]c2)CC(C)CN1C(=O)C(C(F)(F)F)C(F)(F)F N1(C(Cc2cnc(C)s2)=O)C2CCC(C(N3CCCCC(CO)C3)=O)C1CC2 Cc1nc(=N)[nH]c(=NCC2CC(CNC(c3ccncn3)=O)CO2)[nH]1 N1(C(C2C(C)C2)=O)CCOC2(C1)CN(C(=O)CN1CCCC(C(F)(F)F)C1=O)C2 C1(NC(c2sccc2C2CC2)=O)CC2CC(C1)CN(C(C1(CO)CCCO1)=O)C2 C1(OC)CC(C)CN(C(C2CCCN(C(=O)CC3CCC(=O)C3)C2)=O)C1 N1(C(C(c2cn(C)nn2)OC(c2c(C(=O)NC)ccs2)=O)=O)CCC(C)C(CO)C1 CC1(C(=O)NCc2ccc(C(=O)N(CC3CC3)CC3CC3)cn2)CCC(O)CC1 C1(C(N2C(CC(N3CC=C(C)CC3)=O)CC(F)C2)=O)CC12CCCCC2 Cc1nn(-c2cccc(F)c2)cc1C(=O)NCC1(NC(C2CC23CC(O)C3)=O)CC1 c1(C(C(=O)NCCC2(CO)CCC2)NC(=O)Cn2ccnn2)cccnc1 C(N=c1[nH]c(=NCC(CC)(CC)CCO)[nH]c2c1COCC2)c1c(CC)c[nH]n1 Cc1ncsc1C=CC(N1CCCCC1CCCNC(C12CC(F)C1C2)=O)=O O(N(C)C(=O)CCN(C(c1cc(Cl)cn1C)=O)C1CC1)CC(=O)OC N12CCC(CC1C(=O)O)C2.c1(C(=O)OC)ccc(-c2ccc(C(F)(F)F)s2)cc1 CN1CC=C(CC(=O)NC2CCC(C(N3CCC4NCCC4C3)=O)CC2)CC1 c1(C(N(C2CCCN(C(CN(C)CC)=O)CC2)C)=O)cnn2c(=N)[nH]cnc12 N1(C(CCOCC)=O)CCN(C(=O)CNC(C2CCC2)=O)CC1c1ccccc1 C1(CNC(C(CC)OC)=O)CC2(CCC2)CN1C(=O)Cc1cn2c(C)csc2n1 N1(C(CNC(C)=O)=O)CC2(C1)CN(C(C1CN(C3COC3)C1)=O)CCO2 C1(NC(Cc2ncn(C)c2)=O)CN(C(=O)CC2=CCCC2)CC2(CC2)C1 C=CC(C)(C)CC(=O)NC1CCN(C(c2ccc(CN(C)C)nc2)=O)C1(C)C N1(C(C=C(CC)CC)=O)CCc2[nH]nc(CNC(c3ccncc3Br)=O)c2C1 c1(-c2cc(C(=O)NC(CCC)CCC)c(F)nc2)cc([N+](=O)[O-])ccc1F Cc1cc(C(N2CC3(C2)CN(C(C2Cc4nccn4C2)=O)C3)=O)ccc1C#N n1(CC)cc(CC(=O)N(C(=O)CCc2cocc2Br)CC2(O)CC2)cn1 c1(C(=O)NCC(C)NC(c2cc3cc(F)ccc3[nH]2)=O)n[nH]c2c1CN(C)CC2 CCCC(C)C(=O)N1CCC(C(=O)Nc2ccccc2C(C)(C)C)C1 c1(C(=O)NC2CCCN(C(C3CCN(C)CC3)=O)CC2)ccc2nccnc2c1 C1(c2ccccc2)(C(N2CC(N(C(=O)CC3(C(F)(F)F)CC3)C)C2)=O)CCCC1 C1(C(=O)NC2CCC(C(=O)NC3C(C)(C(F)F)C3)CC2)CC12CCOCC2 N1(C(CC(=O)OC)=O)CC(CNC(=O)C(C)CN2CCCCC2)OC(C)(C)C1 Cn1nnc(C(=O)NC2CCN(C(C3CC(O)(c4ccccc4)C3)=O)C2)n1 c1(NC(C2CCC(NC(c3c(Br)cnc(C)n3)=O)C2)=O)ccc2nn[nH]c2c1 C1(O)(C(=O)NCC2C(NC(c3cnc(CC)s3)=O)CCC2)CCCC(C)(C)C1 CC1(CNC(=O)CC2(NC(c3ccncc3F)=O)CCC2)CCC(=O)N1 c1(C(=O)NC2(C)CC(NC(COC(CC)C)=O)C2)cccc(C)n1 N1(C(=O)NCCCOC(C)(C)C)CC(F)(F)C1C1CC1 c1(OC)ncc(Cl)c(=NCC2CC(NC(c3cccc4cnccc34)=O)C2)[nH]1 C(=O)(CCCC(F)(F)C(F)(F)F)N(CCCNC(c1c(C)con1)=O)C CCC(CC(=O)N1CCC(C(C)(C)C(=O)NCC(Cl)=CCl)C1)C(C)(C)C CC1(NC(=O)C(C)(C)NC(C23CC2CNC3=O)=O)CCC(=O)NC1=O C(CCC(C)C)(C(=O)NC1CCN(C(c2cnc(N)c(N)c2)=O)C1C)NC(C)=O C(N=c1nc2c(cnn2C)c(NCc2cnc[nH]2)[nH]1)c1c(CC)con1 N1(C(c2nccc(CC)c2)=O)CCC2CN(C(=O)CSCCC(C)C)CC12 n1(C(C)C(=O)NCCC2CC2(Cl)Cl)cc(C2(C)CCCO2)nn1 N1(C(COCC(=C)C)=O)CCCCC(NC(c2ccnn2C(C)CC)=O)C1 CCCC(C(=O)N1CCCC(CCNC(C2(CO)CCOCC2)=O)C1)S(N)(=O)=O N1(C(C(CC(=C)C)C)=O)CCCCC(C2CN(C(c3cncc(Cl)c3Cl)=O)C2)C1 c1(C(=O)NC2C3CN(C(C(C)(F)F)=O)C2C3)cnc2c(n1)CCCC2 N1(C(CC2CCC(C)CO2)=O)CCC2(CC2)CC1C(=O)NCc1cc(CO)on1 C1(NC(c2c(CSC)cccc2)=O)CC2(CCN(C(=O)CC(=O)NC3CC3)C2)C1 N1(C(C(CC)F)=O)CCN(C)CC1CNC(c1sc(-c2ccc(C)o2)nc1C)=O c1(C(=O)NC(C)CCCNC(=O)CC#N)ccc(-c2ccccc2)cc1F C1(NC(CCC(C)NC(Cc2c(C)ocn2)=O)=O)CC12CCCCCC2 CC1CCN(C(c2cccnc2O)=O)CC1CC(N1CCC(C(N)=O)CC1)=O c1(CC)ccc(NC)cc1.O1NC(=O)CN(C)C(=O)C1 C12(NC(=O)C3=COCC3)CC(C(C)NC(=O)C(O)Cn3cncn3)(CO1)C2 n1(CC)ncc(C(=O)NC2CCC(CNC(=O)CCC(C)SC)CC2)c1C C=CCN(OC)C(=O)c1cn(CCN(C(=O)C(CCC)OCC)CC)nn1 C(CC(C)C)(C(N)=O)NC(CC(CC)NC(c1sccc1C#N)=O)=O c1(C(=O)NCC(CN(C(c2c(C)cccc2O)=O)C)C)cc2c(C)sc(C)c2s1 C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CC(NC(c3cc(C)c(C#N)cn3)=O)C2)C1 C1(NC(C2C(C)OCC2)=O)CN(C(c2cnn3cccnc23)=O)C2CCCC12 N1(C(CC2CCN(C(C3CC(O)(CC#C)C3)=O)C2)=O)CCC=CC1COC C1(C(C)(C)O)CC(NC(=O)C(c2ccc(-c3ccccc3)cc2)(C)C)CCN1 N1(CCNS(CC2(C)CCNC2=O)(=O)=O)CCCOC(c2ccc(C)cc2)C1 Cc1cc(C(=O)NC2CC(C)CN(C(=O)C(C)NC=O)C2)cc(O)n1 C1(C(=O)NC(C(=O)OC)C(C)O)CCCN(C(c2cc(C3CC3)on2)=O)CC1 C=CCN=c1[nH]cc(C(=O)NC(CN(C(=O)Cn2ccc(C)cc2=O)C)CC)s1 CC1=C(C(=O)NC2CCC(NC(c3cncc(C(F)F)c3)=O)C2)CCO1 C(=O)(C1=CCC2(COC2)OC1)NC(C(C)NC(=O)Cn1ccc(C(F)(F)F)n1)C N1(C(C(CSC)O)=O)CC2CC3CC2C1C3NC(C1Cc2cc(C)ccc2S1)=O N1(C(C(C)n2ccnc2)=O)CCC(CNC(=O)COCCOCCO)C(O)C1 CC1CN(C(=O)CC2(N(C)C(c3ncc(F)cc3N)=O)CC2)CC(CO)O1 c1(OC)c(F)ccc(C(N2CC3CN(c4ncc(C)c(C)n4)CC3C2)=O)c1F N1(c2n(C)c(=O)n(C)c(=O)c2)CCC2CCC(C1)N2C(C1CC1(C)Br)=O c1(C(=O)OC)cc(NC(c2ccc(C#N)c(O)c2)=O)cc(OC)c1OC C1(CC)C(=O)NCCCN1C(C1CC(C)CN(C(c2cccc(Cl)c2)=O)C1)=O Cc1ccc2ncc(C(=O)NC3CCC(NC(=O)CC45CCCC4C5)C3)n2c1 C(=O)(CC(C(=O)NCCC(C)CCNC(c1cncc(C)c1)=O)NC(C)=O)OC c1(SC)ccc(C(=O)NC(C)CCNC(=O)C(C)(C)c2ccsc2)s1 C(c1ccc(F)cc1)=CC(=O)NC1CCC(NC(=O)CC23CCCC2C3)C1 N1(C(CCN(C)CCO)=O)CCC(C2CC2)C1C(=O)NC1CC2(CCOC2)C1 C1(CNC(c2ccc(COC)o2)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1(F)F C(N=c1cc[nH]cc1[N+](=O)[O-])C1CN(C(Cc2c(C)non2)=O)CC12CCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CCCN(C(C2CCN(C3CC3)C2=O)=O)CC1 c1(OCC)ccncc1C(=O)N(c1ccccc1)CC(F)F CC(O)C(C)(C)C(=O)N1CC(n2cc(-c3ccc(Cl)cn3)nn2)C1 CCCC(CC(=O)NCC(C)NC(c1cccc(F)c1C)=O)NC(=O)OC(C)(C)C c1(C(N(C2CC(C#N)C2)CC(=O)NC(c2ncc[nH]2)CC)=O)ccc(Cl)o1 C1(C(=O)NC(C)CCCNC(=O)C(C)(C)O)CCC2CCCCC2C1 c1(Cc2nn(-c3cccc(OC)c3)c(CCCF)n2)coc2c(C)c(Cl)ccc12 C1(CNC(C(C)(C)SC)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 N1(Cc2cccc(C#N)n2)CCC2(CC(C(=O)N=c3cncc(Br)[nH]3)=NO2)C1 N1(C(C=COCC)=O)CCC(c2ccccc2)(NC(=O)C(C)SCC)C1 C(=O)(C1CCNc2ccccc21)c1onc(-c2c(C)cc(F)cc2Cl)n1 O=C1CN(CC(N2CCC3CC23CC(=O)NOCCOCCO)=O)C(=O)N1 C1(c2cn(CCC=C)nn2)CN(C(C2CC=CCO2)=O)CCO1 C(=O)(C(C)(C)N(C)C)N(CCC(=O)NCCC1CCNC1=O)C C(=O)(CCC(C)NC(c1ncn(C)n1)=O)NCc1ncc(C)o1 C=CCC(C)(C)C(=O)NCc1occc1C(=O)NCc1nocc1C(C)C C1(N(C)C(c2csc(C3CC3)n2)=O)CN(C(C23CC(F)(C2)C3)=O)CC12CC2 N1(C(C(CC)C)=O)CCCC2(CCCN2C(c2n[nH]c3c2CCC3)=O)C1 C1(C(=O)NC(C#C)C2CC2)(CNC(=O)Cn2nnc(C)n2)CCCO1 CC1(C)CC(=O)N(CC(=O)NC2CN(C(C3CC4CCC4C3)=O)CC2C(F)F)O1 C1(NC(CC2(C)CC2(F)Cl)=O)CCC(NC(=O)C=CCOC2CCOCC2)CC1 C1(C)(NC(C(CCC)NC(=O)C(C(C)C)SCC)=O)CC(F)(F)C1(C)C c1(C(=O)NCC2(C)CCCN(C(C3(CC)COC3)=O)C2)cc2c(=O)[nH]ccn2n1 N1(C(C2CC=C(C)CC2)=O)C2CCC1C(NC(c1cc(C)[nH]n1)=O)C2 c1(CC(N2CC3(CN(C(=O)CCc4cnn[nH]4)C3)C2)=O)cncc2ccccc12 C1(CC(=O)N(CC(N2CC(CCC)C2)=O)C2CC2)CC2CCC1C2 c1(C(N(C)CC2CCN(C(=O)C=CCF)CC2)=O)cccn2ncnc12 C1(CC)CN(C(c2cc(C)c[nH]2)=O)CCC1NC(C12CC3CC1C2C3)=O N1(C(c2c(COC)nn(C)c2)=O)CCOCC(C(=O)NC(CO)C(C)(C)C)C1 N1(C(c2ccc(N)cn2)=O)CCC(NC(=O)CC2CC(O)C23CCC3)C(O)C1 c1(C(N(C)CC2CCN(C(c3c(C)nc(CC)o3)=O)C2)=O)cc(F)cc(Cl)c1N O=C(C#CC1CCCCO1)N1CCC(F)CC1c1ccco1 CCCC(C(=O)NCC(CC)N(C(c1ccn(CCC)n1)=O)CC)C(C)C N1(C(COCCOC)=O)CC(C(=O)NC(C2CCCO2)(C)C)C(C(C)C)C1 C1(NC(C(C)=C(CC)C)=O)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1C C(CCO)(C(F)F)N(C(CNC(CN1C(C)CCC1)=O)=O)C C1(C(C)NC2CCOC2)CCCN(C(=O)CN2CCOCC2)C1 N1(C(C2(OCC)CC2)=O)CC2C(CN(C(=O)CC3COCCN3C)C)C2C1 N1(C(CCSCC)=O)CC(NC(C2CCCCCN2C)=O)CC1(C)C C12(C(=O)NC3CC(OCC(=O)N(CCC(O)CO)C)C3)CC(CO)(C1)C2 C(CN=c1[nH]c(=NCCc2nc(-c3cccs3)n[nH]2)[nH]c2ccsc12)SC(C)C N1(C(=O)C(=O)NCCOC2CCOC2)CCC(c2cccnc2)C1 c1(C(=O)NC2CCC(NC(COCC#C)=O)C2)c[nH]ccc1=NC(=O)C(C)(C)C C1(N(C(=O)Cn2cccn2)C)CCCC(NC(c2cscc2F)=O)C1 c1(OCc2cn(C(C)CNC(=O)Cc3cc(Cl)cs3)nn2)ncc(C#N)cc1Cl Cc1ccc(C=CC(N2CCC(F)(CNC(=O)CCc3ccc(CO)cc3)C2)=O)s1 C1(C)(CC)CCC(C(=O)NC2CC2CNC(=O)CCc2cn[nH]c2)O1 c1(OC)ccc(Br)c2c1C(NCC1CCNC3(CCC3)C1)CC2 C(=O)(C(C)CS(C)=O)N(CCCNC=O)C.c1(C(=O)OC)ccc(N2CCC2)nc1 Cc1cc(C(=O)NC(CNC(=O)Cn2nccc2C)C(C)C(C)C)cc(C)c1Cl CC(C)CCC(=O)O.C1(CC(=O)NC)CCOC1=O.C1C(=O)N1.C1C(=O)N1 c1(C(N(CCNC(C(C(C)C)SCC)=O)C)=O)cc(F)cc2cnccc12 O(NC(=O)C(CCC(C)C)NC(=O)C(C)NC(N)=O)C(CC)CC c1(OC)ccc(C(CNC(=O)NC(C(F)(F)F)C2CC2(C)C)N(C)C)cc1 C=CCC(C(=O)OC)NC(=O)Cn1cc(-c2cccc(SC(F)(F)F)c2)nn1 C=CC1(C(=O)NCc2cnns2)CCN(C(=O)CC(C)C(F)F)C1 N1(C(C(COC)N(C)C)=O)CCN(C(=O)Cc2ccsc2C)C(CCOC)C1 N1(C(C(CCC)CNC(C2CC2Cl)=O)=O)CCC2(CC(CO)C2)C1 Cc1cc(=NC(=O)C(C(C)NC(=O)C(c2cnn(C)c2)C)C(C)C)[nH]n1C1CC1 C(CCO)(C(C)(C)C)NC(CCN(C)C(c1cnc[nH]c1=N)=O)=O N1(C(C(C)(C)CO)=O)CC2CN(C(C3(S(C)(=O)=O)CCCC3)=O)CC2(C)C1 CC1CN(C(c2ccccc2CO)C(=O)NCCCC2CC2)CC1(C)C(N)=O c1(C(=O)NC(CNC(CC2CC(C)OC2C)=O)C)c2c(nn1C)CCOC2 N1(C(C(COCC)N=[N+]=[N-])=O)CCCC(C2CN(C(c3cc(=O)cc[nH]3)=O)C2)C1 Cc1nc2c(s1)CCCC2C(=O)NCC1CC(F)(NC(=O)CCCS(C)(=O)=O)C1 c1(CC(=O)N(C(CCNC(C(C)OCCC#C)=O)C)C)cc(C)n(C)n1 n1(C2(C(CCCC)=O)CC2)cc(CN2CCOCC2)nn1.C1COO1.C1(CC)CC1.O.C C1(NC(c2c(F)cc(OC)c(F)c2)=O)CC12CCN(C(C1CCCC1)=O)CC2 CCCC(CCC)C(=O)N(CCNC(C1CCCC1C1CC1)=O)CCOC c1(C(=O)NCCCN(C(C(C)OCC#C)=O)Cc2ccccc2)cc(O)ncn1 C#Cc1ccc(F)c(C(=O)NCCC(CC)(CC)NC(=O)CC2CCOCC2)c1 c1(CC(N2CCC(C(C)NC(=O)C(C)C3CC3)C2)=O)c(F)cccc1F C1(C(=O)NCC(CCCC)NC(C=COCC)=O)CCOC(=O)CC1 C(CC(F)CN=[N+]=[N-])NC(C(C1(O)CN(C(c2cn(C)nc2)=O)C1)F)=O C12(C(=O)NC(CC=C)C3CC3)CC1CN(C(=O)CC1CCCCN1C)C2 c1(C(N2CCC(C)(CNC(C(C)N(C)C)=O)C2)=O)c(C(F)(F)F)cccc1Cl C1(NC(CN(CCC#C)C)=O)CCCN(C(c2cccc(N)n2)=O)C1C C(C)(C(=O)NC1CCOC(C(=O)NC2CC(O)C2O)C1)(C(C)C)OC C#CCCCCCCC(=O)N1CC2CC1(c1cn(-c3ccccc3SC)nn1)CO2 Cc1ccc(C(N2CC(NCc3cc(C)n(C)c3)CC(C)C2)=O)cc1C(F)(F)F c1(SC)ccc(Cl)c(C(=O)NC2CCN(C(=O)Cc3ccc[nH]3)CC2C(C)C)c1 c1(C(C(=O)NC2CN(C(c3cc(C)cc(F)c3)=O)C2)C)cn(C)c2ccccc12 N1(C(c2c(CC)ccc(F)c2)=O)CCC2(NC(=O)Cc3cccnc3)CCCC12 C1(NC(=O)NCc2nc(COC)sc2)(COc2ccccc2)CCCC1C1CC1 C1(C(=O)NC(CCNC(C2CCC(CCC(C)C)CC2)=O)C)CC(C)CC(=O)N1 c1(C(N2CCCCC(NC(CN(C)C)=O)C2)=O)cc([N+](=O)[O-])c(Br)cc1F C1(N(C(=O)Cn2cccn2)C)CN(Cc2sccc2OC(F)F)CCC1O C1(C(N(C)CC2CN(C(c3ccc(C)o3)=O)C2)=O)CCC(=O)NC1 Cc1nc(C(=O)NCC2CN(C(=O)Cc3sccc3C)CC2C)ccc1[N+](=O)[O-] CN1CC(C(=O)NC2(CCNC(c3nc[nH]c3C(F)(F)F)=O)CCCC2)NC1=O c1(C(=O)NCC2C(NC(C(n3ccc(C)n3)C)=O)C2)cc(Br)c(C)cn1 C(CCCC(=O)NCC(C(=O)N1CCC(CO)C1)N(C)C)SC c1(C(=O)NC2C3CN(C(c4c(N(C)C)ccnc4)=O)CC32)ccc(F)c(F)c1F C12(C(=O)NC(C(C)F)C)CCCC1CCN2C(=O)C(c1cnn(C)c1)C C1(NC(C2COCCOC2)=O)COC2(C1)CN(C(c1cnc3nccn3c1)=O)C2 C=CC(CC)C(=O)NC(C(=O)NCC1(OC)CCC1)c1ccco1 N1(C(c2noc(CSC)n2)=O)CCC2(NC(=O)Cc3cnn(C)n3)CCCC12 N1(CC)CC(NC(=O)C(CC2CCC2)NC(=O)C=CC2CCCC2)CC1=O c1(C(C(=O)NC(C2(O)CN(C(C3(O)CC(C)(C)C3)=O)C2)C)CO)ccc(F)cc1 C1(C(=O)O)CCC(C(=O)NC(c2cccc(Cl)c2)CF)CC1 c1(C(=O)NC2C(NC(COC)=O)CCCC2)ccc(C)c(OCC(C)C)c1 C1(C(N(CC(C)NC(c2c(C(=O)OC)n(C)nc2)=O)C)=O)CN2CCC1(C)CC2 N1(C(C(C(C)C)SC)=O)CCC2C(C1)CN2C(=O)CC(C)(C)CN1CCOCC1 c1(CC(C(=O)NCC(C)NC(CC(=C)C)=O)C)ccccc1Cl Cn1cc2c(n1)CCCN(C(C1C3CN(C(=O)C(C)(C)n4cccc4)CC13)=O)C2 Cc1coc(C(=O)NC2CCC(CNC(=O)C(F)(F)c3nccs3)C2)c1 N1(C(C(=O)N(C)C)=O)CCC(NC(c2nc(Cl)sc2Cl)=O)C(CO)CC1 C=C(C)CCCC(=O)NCCC1CN(C(=O)C(C(=O)OCC)OC)CCO1 C1(C(=O)CC2(c3ccccc3Br)CC2)CNC(C2CC2)CO1 Cc1cc2cc(C(=O)NCC3CN(C(=O)C(C)(F)C(F)(F)F)C3)[nH]c2cc1Cl C1(CC(=O)NC2C(N(C)C)COC2)CCOC1(C)C S(=O)(=O)(c1ccsc1C(N1CCC(NC(=O)C=Cc2cncs2)C(O)C1)=O)NC Cc1ccccc1C(=O)NCC(=O)NCC(F)CNC(c1sccc1Cl)=O c1(C(N2CC(OC)C(NC(c3cnnc(C)c3)=O)C2)=O)cccn(C)c1=O c1(NC(C(CNC(C2CC(COC)C2)=O)C)=O)c(C)[nH]c(C)cc1=O N1(C(C=C(C)Cl)=O)CCC2CC(NC(c3cnc4nccn4c3)=O)CCC2C1 c1(C(=O)NC(CNC(c2ccc(C)o2)=O)C)cnc2c(c1)c(C)nn2C S(=O)(=O)(c1ccc(F)c(Br)c1)N1CCN(C2CCN(C(=O)C(F)F)C2)CC1 C1(NC(CCC2N(C(C=CC(CC)C)=O)CCC2)=O)COC2(CCCC2)C1 N1(C(COCC=C)=O)C(C(=O)N(C(C)C(C)(C)O)C)C2CC(O)C1C2 C1(CC)C(C(=O)NCCCC(C)(C)OC)CCN1C(c1ccccc1NC)=O c1(NC2C(C)C(c3ccccc3)C2)ccc(Cl)c(C2=CCNCC2)c1 c1(C(N2C(C(C)NC(c3cnc(O)o3)=O)CCCC2)=O)cccc2oc(O)nc12 N1(C(c2c(C)nco2)=O)CCCC(N(C)C(c2cc(F)c(N)cc2F)=O)CC1 N1(C(c2c(C)cccn2)=O)CC2CCC(CNC(C3CC3Cl)=O)C2C1 C1(n2cc(C(C(C)(C)C)O)nn2)(CNC(C2CCC(F)(F)C2)=O)CCCCC1 c1(C(=O)NC2CC(N(C)C(c3nccnc3C(N)=O)=O)C2)ccnc2c1CCO2 Cc1[nH]nc2cc(C(N3CCN(C(=O)CC(C)CF)CCC3C)=O)ccc12 c1(C(=O)NC2CCCN(C(C3CC34CC4)=O)CC2)c[nH]c2cc(O)ccc12 C1(NC(=O)CC2COCCOC2)CC(NC(=O)Cc2ccsn2)C12CCC2 CCC(CC(C)C)C(=O)NC(CNC(c1sc2ccsc2c1C)=O)CO C1(NC(C2CCN(C(C)C)CC2)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)C1(C)C C1(S(C)(=O)=O)(C(=O)NCC2(NC(CCC(C)(F)F)=O)CCOC2)COC(=O)C1 c1(C(=O)NNC(=O)C23COC(C2)C3)cccc(S(=O)(=O)C(F)(F)F)c1 c1(CC(=O)NCCCCCCNC(CCS(=O)(=O)NC)=O)ccc(C)c(F)c1F Cc1nn(CC(=O)NC(C(C)NC(C2(O)CCC2)=O)C(C)C)c(C)c1[N+](=O)[O-] CC(C)(C)C(CNC(=O)CCC(F)(F)F)C(=O)NC1CCC2CCC12 c1(OC)cccc2c1CCCC2NC(=O)C(C)(C)c1ccns1 C1(NC(C(Br)=C(C)C)=O)CN(C(=O)CCC(C)C#N)CCC12CCC2 CCCCCS(=O)(=O)CC(=O)NCC(C)CN(C(=O)CC12CC(C1)C2)C C(C(F)(C(=O)NCCCC(=O)NC1CC1)C(C)C)NC(c1c(CC)cccc1)=O CC(C)C(C(=O)NC(C)CN(C(=O)Cc1n[nH]c(=N)s1)C)c1ccncc1 c1(OC)ccc(NCC2(C)CCC(C(=O)OC(C)(C)C)C2)cc1N1CCOCC1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(C2CN(C(c3c[nH]c(=N)o3)=O)C2)C1 CN1C2CCC1CN(C(=O)C(CO)NC(c1ccncc1N)=O)CC2 Cc1cc(C(C)(C)C)ccc1C(=O)NCCN(C(C1CC1(F)Cl)=O)C(C)C c1(OC)cnncc1C(=O)NC(C1CCN(C(C2CCC(=O)N2)=O)C1)(C)C CC1CCC(NC(c2cnc(-c3ccccc3)[nH]2)=O)CN1C(=O)CNS(N)(=O)=O c1(CNC(C=C2C(C)(C)CCCC2)=O)c(F)ccc(N)c1F CCCC(C)CCCC(=O)NCCCNC(=O)C(c1cccnc1)O C(=O)(CCCCCF)N1CCC(C(C)NC(CCc2cccc(OCC)n2)=O)C1 C(CCC(C(=O)N(C1COCC1OC)C)NC(c1scnc1Cl)=O)OC C(Cn1cncn1)(C(=O)NCCC1COCCO1)NC(CCOC(C)=O)=O CCCC(CC(C)C)C(=O)N(CC(C)NC(=O)CN(CC)CC)CC N1(C(c2c(C(C)C)ccs2)=O)CCC2CCN(C(C3CC(=O)N3)=O)CC2C1 C(CCCCCCO)NC(C(C1CCCN(C(=O)C=CC(=O)N(C)C)C1)C)=O Cc1cc(NC(=O)CSCCC(C)C)ccc1NC(C1CCCC(C)O1)=O N1(C(c2cnn(C)c2N)=O)CC2CCN(C(=O)CC3CC4(CCC4)C3)C2C1 c1(OC)c(NC(C2CC(C)CN2C(c2nc(C(C)C)cs2)=O)=O)c(C)nn1C Cc1cccc(C(=O)NC2(CCNC(=O)C(F)C(C)(C)O)CCCC2)c1C C(C(C)(C)C#CC(=O)NCCC1COC(C)(C)C1)NC(C(C)S(C)(=O)=O)=O c1(CC(=O)N(C(CNC(C2(C(=O)OCC)CCC2)=O)C)C)cscc1Br C(=O)(C(C)(C)n1cc(Cl)cn1)NCC(C)(C)OCC(=O)N(C)CC1CCCO1 N1(C(c2n(CC#C)cnn2)=O)CCN(C(c2scnc2Cl)=O)C(CC)C1 C1(C(=O)OC)CC(C(=O)OC)CC(C(N2CCC(CCF)CC2)=O)C1 Cc1cc(C(=O)NCC2CCCC(NC(=O)COCc3scnc3C)C2)n(C)n1 C1(C(N2CCC(C)(CC)CC2)=O)CCC(C)(C)N(C(=O)Cc2nc(=N)[nH][nH]2)C1 C(CC(C)C)(C(=O)N(C1CN(C(C)C)C1)C)ONC(c1cc(CC)[nH]n1)=O c1(NC(C2(C(C)C)CCNC2=O)=O)cc(Cl)cc2c1OCC(=O)N2 CN1CCOC(C(=O)NC23CC(NC(C4CCCC(C(=O)N(C)C)C4)=O)(C2)C3)C1 CCC(O)C(C)C(=O)N1CCC(C(C)(C)NC(c2cnn(C(C)(C)C)c2)=O)C1 C1(C(=O)NCCOCCOC)CCCC(NC(c2nccn2C2CC2)=O)CC1 C(C1CCCCCC1)=CC(N1C(CO)CC(NC(Cc2c(C)noc2)=O)C1)=O C1(NC(c2cncc(CNC(=O)Cc3cnccn3)c2)=O)CCCCC1(F)F C1(CNC(C2N(CC)CC2)=O)CC2(CO1)CN(C(=O)CCC1CCC(=O)C1)C2 c1(OC)ccc(C=CC(=O)NC2(CN(C(=O)CC3CCC(C)CC3)C)CC2)cc1 c1(C(=O)NCC(CC=C)NC(=O)CC2COCCN2C)cc2c(C)nn(C)c2s1 C1(CNC(COCCCCC)=O)COC(C)(C)CN1C(c1cccc(C)c1)=O C12CN(CCC1C)C(=O)C2.C1(CCC)(CC)CCCN1C(=O)CCC1CC1 Cc1ccc(C(=O)NCC2CN(C(=O)CC(c3cccc(F)c3)O)CCO2)nc1 C1(NC(Cc2c(C)n[nH]c2C)=O)CC2CC(C1)N(C(=O)Cc1cncnc1O)C2 c1(CC(=O)NC(c2nn[nH]n2)C2CC2)ccccc1OCCCC#N CC(C)C(O)CC(=O)NCC(F)CNC(c1cc(-c2ccncc2)no1)=O C=CC(CC)CC(=O)N1CCCC(CNC(c2coc(-c3cn[nH]c3)c2)=O)C1 C1(C)(C(=O)NCC2N(c3ncc(OC(C)C)cn3)CCC2C)CCCCCC1 c1(C(N(CC(N2CCN(CC(C)C)CC2)=O)C)=O)cc2cccnc2o1 c1(C(N2C(C)CC(NC(=O)Cn3nccn3)C2)=O)cc(=O)c2ccc(O)cc2o1 N1(C(=O)NC(C)CN2CCCN(C)CC2)CCNc2cc(Br)ccc2C1 C1(NCCNC(Cn2cnc(C(=O)OC)n2)=O)CCCSC1 C1(C(N(CCCCCNC(C(CSC)OC)=O)C)=O)CC2(C)CC1CO2 C1(CNC(C2CC(CC)C2)=O)C2CN(C(=O)CN(C3CCC3)C)CC12 N1(C(C(C)Oc2ccc(C)cc2Br)=O)CCCC2CCCCC12 N1(C(C(CSC)O)=O)CCC2(CC1)CCN(C(C1CCC3(CCOCC3)C1)=O)C2 c1(C(N2CC(F)(CNC(CC(C)C(C)(C)C)=O)C2)=O)cc2c(F)c(F)ccc2[nH]1 c1(C2(COC)CC2)ccc(C(N)=O)nc1.C1(CCN)(NC(=O)C=CC)CCC1 CC(O)(C(=O)N1CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C(F)C1)C(F)(F)F C(=O)(C1=CCc2ccccc21)NCCC(CCNC(CC(=O)OCC)=O)C c1(CC(=O)NC2CC(C(C)NC(=O)CCC3CCCOC3)C2)cc(C)nn1C c1(C(=O)NCC2(F)CCN(C(c3ncc(OC)nc3)=O)C2)ccc2c(c1)CCC2 c1(C(=O)NC2C3(CC(NC(CCNC(=O)NC)=O)C3)C2)cccc(C)c1C C1(CNC(c2ccc(C(F)(F)F)[nH]2)=O)CC(O)CN1C(C1CCC(F)(F)C1)=O C(=O)(C(C)(C)C(=O)NCC(CC(F)(F)F)NC(=O)C=Cc1ccc(F)cc1)NC C1(c2n(C)ccc2)CN(C)CCN1C(c1ccc(C2CC(C)(C)OC2=O)cc1)=O C#CCCCC(C)C(=O)NC1(CC=C)CN(C(c2cc[nH]c2)=O)C1 c12cccc(c1)CNC2=O.C1(C(=O)NCC(C)(C)OCCO)OC2CCC1C2 c1(C(=O)NC(C)C)nnc(N2CCOC3CC23)n1Cc1cccc(Cl)c1 c1(C(=O)Nc2ccc(-n3c(C)ccn3)cc2)cc2cccc(C)c2s1 C1(CCNC(CCCOC)=O)C(C)CCCN1C(C1CCCCC1)=O N1(C(C(CO)OC)=O)CCCN(CCNC(=O)C(F)CC2CCCC2)CC1 N1(C(=O)CC(F)(F)C(=O)O)CC2CCN(C(c3cscn3)=O)CC2C1 C1(CNC(CSCCC)=O)CC2(CCC2)CN1C(c1sccc1C)=O C(C)(C(C)(C)C(=O)NC1(c2cccs2)CC1)NC(C(CO)OC)=O CN1CC(C(=O)NC2CN(C(=O)C=Cc3ccc(=N)[nH]c3)CC23CC3)CCC1=O N1(C(c2c(C)cc(F)s2)=O)CCC2CC(NC(c3csnn3)=O)CCC2C1 c1(CN2C(CC(C)C)CCCC2=O)cc(=O)[nH]c2ccccc12 C1(CNC(C(C)OC(C)C)=O)CCC2(C1)OCCO2 N1(C(c2c(CC)n[nH]c2)C(=O)NC2(C)CC2)CC2CC3CC2C1C3C(=O)OC c1(Cc2occc2)ccc(F)c(-c2ccc(C)cc2)c1.n12nnnc1C2.C1CCC1 CCCC(C)(CCC)C(=O)NCC1C=CC(NC(=O)Cn2ccnc2C(C)C)C1 N12CCCC(C)(C1)C2.N1(C(=O)OC(C)(C)C)CCC2CC12C(F)(F)F c1(NC)c(C(=O)NCCN(C)C(c2c[nH]cc2C(C)C)=O)cccc1F C1(C(=O)NC(C)CCN(C(=O)CCc2ncco2)C)OCCN(C)C1=O c1(C(=O)NCC2(C(=O)Nc3c(C)cc(Br)cc3Cl)CC2)ccc2nc(O)oc2c1 c1(NC(C2C(NC(c3c(O)ccc(C)c3)=O)C2)=O)cc(Cl)c(Cl)cc1[N+](=O)[O-] C12(NC(=O)COC(F)F)CCCC1N(C(=O)C(c1cc(F)c(F)cc1F)O)CC2 Cc1cc(CC(=O)NCC2CCN(C(c3ccccc3)C)CC2)n(C)n1 CC(N=c1nc2scnc2c(NCCOc2ccncc2)[nH]1)C1CCOC1 c1(C(=O)NCCC2OCCN(C(CC3(C)CC3(F)F)=O)C2)cccc2c1CCC2 C1(OC)CC2CC1CN(C(c1conc1CNC(c1cnccn1)=O)=O)C2 N1(C(C(CSC)OC)=O)CCCC(C)(C)C1CNC(=O)C(=O)N=S(C)(C)=O C1(O)(CN(C)C(C2(F)CCOC2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1 c1(C(=O)NCCC(C)NC(c2cnc(NC(C)=O)o2)=O)nn(C)c(N)c1C c1(C2(C)CC2)ccc(C(=O)NCC2(NC(c3cc(C)c[nH]3)=O)CCOC2)cc1Cl C(=O)(CCC(=O)N1CC(NC(=O)Cc2c[nH]nc2O)CC1C)N(CCC)CCC N1(C(C(CC(C)C)O)=O)CCN(C(=O)C(=CC2CCCCC2)F)C2CCCC12.CC=CC C1(C(C)NC(C2(C(N)=O)CC2)=O)CCN(C(c2ccc(CCF)cc2)=O)CC1 CC1(C)CC1(c1ccccc1)C(=O)NCC1CN(C(C2(CF)CCC2)=O)C1 c1(CCOC)ccc(OC(C)CCF)c(C)c1 N1(C(Cn2ncc(CC)c2)=O)CCCN(C(=O)CCCC(=O)N(C)C)CC1C Cc1cc(F)c(C(N2CCC(C)C(NC(=O)Cc3csc(S)n3)C2)=O)cc1F c1(C(N2C(CO)CC(NC(CN(CCOC)C)=O)C2)=O)ccc2nnc(O)n2c1 C1(O)(CCC2(C)CN(Cc3cccc(N4CCOCC4)c3)C2)CCCCC1 C(=O)(CCC(C)C#N)N(CCC(=O)OCC)C1CC1 N1(CCNC(C(n2cc(-c3cc[nH]n3)nn2)C)=O)CCCC1CO C1(C)(NC(C2C(OC(C)=O)C2)=O)CCN(C(c2cc(CC(C)C)on2)=O)C1 N1(C(Cc2cn(C(C)(C)C)nc2)=O)CC(CO)C(CCO)C1 N1(C(C(C)(C)N(S(C)(=O)=O)C)=O)CC2CC1CN2C(c1cncn(C)c1=O)=O c1(CC)ccc(C(F)(F)F)c(C(=O)OCC23CC(OC)(C2)C3)c1 C1(S(N)(=O)=O)(C(N(C)CC2CN(C(C3CCCCN3C)=O)C2)=O)CCC1 C1(CNC(Cn2ncc(CC)c2)=O)CCC2CN(C(=O)C(F)=CC3CC3)CC12 N1(C(CC(C)SC)=O)CCC(CCC(=O)NC2CN(C)CC2C)CC1 C1(CCCNC(c2ccc(CCC)s2)=O)CN(C(c2cc(C)co2)=O)CCO1 N1(C(Cc2c(SC)cccc2)=O)CCC2(CC1)CN(C(=O)CC1CCOC1=O)C2 C#Cc1cccc(C(=O)NC2CC(CCNC(c3ncccc3F)=O)C2)c1F c1(C(N2CC(CCC)N(C(=O)C(C)=C(C)C)CC2)=O)oc2cc(Cl)ccc2c1C C1(CNC(CCCC#C)=O)C(C)CCCN1C(=O)C(C)SCCCC N12CCCN(CC1)C(=O)C2.c1(CCC(=O)OCC(=O)NC)nnc(C)n1C C1(NC(c2cc(CO)[nH]n2)=O)CCC2CCN(C(C3(CO)CCC3)=O)C1C2 N1(C(C2C(C)(COC)C2)=O)CC2CC(C1)C2NC(c1cc(O)cc(F)c1)=O Cc1[nH]cc(C(N2CC(NC(C3CC4CSCC(C3)C4)=O)C2)=O)c(=O)c1Cl C1(N(C)C(C2(C)CC(C(F)(F)F)C2)=O)CCC(NC(=O)Cc2ccco2)C1 C1(C(=O)N(c2ccncc2)Cc2ccccc2)CSc2ccccc2O1 c1(CCCC(=O)NCC(C)(C2CC2)NC(CC(C)O)=O)ccc(F)c(F)c1 C(=O)(CCCC(=O)NC1(C)CCN(C(=O)CC2CCCN2C(C)C)CC1)OCC N1(C(=O)CCC2CCCC2)CC2CC(NC(C3(COC)CC(=C)C3)=O)C(C2)C1 c1(C(c2nnnn2CCCC)NC(CCCC)CCC)sc2ccccc2c1Cl N1(c2ncc(C)cn2)CC(NC(=O)C(CO)c2ccccc2)CC(C)C1 CC(C(=O)NCC(O)CC(=O)N1CCCC1CCCO)C(C)(C)C c1(C(=O)NCC2N(C(CN(C(C)C)C)=O)CCCC2C)c(F)cccc1[N+](=O)[O-] c1(CC(=O)N(C)CC2N(C(CC3(C=C)CCC3)=O)CCC2)cn2c(n1)CCCC2 C1(C(=O)NC(CNC(c2ccnc(CO)c2)=O)C2CCC2)CC2(C1)CC(F)C2 C1(C(=O)NC2C3CC2N(C(C2CCO2)=O)C3)CC(c2ccccc2[N+](=O)[O-])=NO1 C(C(C)(COC)C(=O)NCc1cccc(NC(C2CCC(C)(C)OC2)=O)c1)OC N1(C(c2ccc(OC)nn2)=O)CCCC(NC(=O)CC2(C)CCCCC2)C1C c1(CCC(N2C(CCCNC(C3CCSC3)=O)CCC2)=O)nc2ccccc2[nH]1 N1(C(C2(OCCOC)CC2)=O)CCN(C(c2conc2C(C)(C)C(F)F)=O)CC1 N1(C(C(C)OCC=C)=O)CC2CCC1CN2C(c1c(C)[nH]c(C(=O)O)c1CC)=O Cc1cc(C(N2CCCC(CNC(=O)C(F)C(F)(F)F)CC2)=O)c2occc2c1 N1(C(C(C)O)=O)CC2(CCN(C(c3ccc(F)cc3Br)=O)CC2)C1 C1(C)(C(N(C)CCNC(=O)CC2CCC(=O)N2C)=O)CCCCNC1=O C1(N(C)C)CCCC(C(N2CC(O)(CN(C(=O)CC3CCOC3)C3CC3)C2)=O)C1 C(=O)(C(C)(O)C(F)(F)F)N1CC2C(N(C(=O)CCCCCc3cccs3)C)(C2)C1 C(=O)(C(F)CC(C)(C)C)NCCn1ncc(C(=O)NC(C)CC(N)=O)c1 N1(C(CC(CC)N(C(c2c(CC)c[nH]n2)=O)CC)=O)CCN(C2CC2)CC1 Cc1sc(C)c(C(=O)NC(CNC(C2CCCN2C)=O)C2CCC2)c1C#N c1(OCC)ccc(-c2cc(C(=O)Nc3cnccc3Br)n[nH]2)c(C#N)c1 C(=O)(C1=NOC(C)C1C)NC(C(N1CCC(O)(CC)CC1)=O)CCN(C)C CCC(C)(C(=O)O)N(c1ccccc1F)C(=O)CCCC1(c2cccc(Cl)c2)CC1 c1(NC(=O)NCC2CC(NCc3ccc(OC)cc3)C2)cc(F)c(C)cc1Cl C(C)(CCC(=O)NC1(CCNC(=O)C(=O)NC2CC2)CCC1)OC c1(OC)ccccc1CCC(N1CCOCC1CNC(=O)C=CC1CCOC1)=O C(=O)(C1COc2ccc([N+](=O)[O-])cc21)NCC(CC)(C)NC(=O)C(N)=O N1(Cc2nccc(OC)c2)CCOCC(C2CCC2)C1 C(C(C(=O)NC(c1ccon1)(C)C)C(C)C)NC(c1c(C)coc1)=O N1(C(CCP(C)(C)=O)=O)CCN2C(=O)C(NC(c3cnc(=N)[nH]c3)=O)CC2C1 C(=O)(C1=NNC(=O)C1)NCC1CN(C(c2c(COC)cco2)=O)C1 CC1(C)CC(C(N2CC=CCC2)=O)CCN1C(=O)CCn1cccc1 N1(c2nc(C)nc(C#N)c2)CCC2CCC(NC(=O)C=CC=C(Cl)Cl)C1C2 c1(C(=O)OC)ncccc1NC(=O)C(=O)NCC1CCCSCC1 C1(COC)CN(C(c2ccnc(CNC(C3CCCS3)=O)c2)=O)CCO1 c1(CNC(c2c(CNC(C3(COC)CCOC3)=O)cco2)=O)nn(C)cc1SC c1(C(N(C2CCC(NC(C3CC34CCC4)=O)CC2)C)=O)cc(Cl)cc(F)c1N C(=O)(CN=c1[nH]c(=NCCC2CC2(Cl)Cl)c2ccc(OC)cc2[nH]1)OCC=C C=C(C)C1OCCCC1C(=O)NC1CCC1NC(c1cc(Cl)cs1)=O CC1OCCC1C(=O)NCC(=O)OC1CC(C(=O)N(C)C)C1 Cc1c(F)ccc(C(=O)NCC2CCCN2C(=O)Cc2ccc(Cl)cc2F)c1Cl c1(C(N(CC(CN(C(C2C(CC)C2)=O)C)O)C)C)nc(C(C)C)no1 n1(C(C)C)ncc2cc(NC(=O)C3=CC(C)CC3)ccc12 CS(=O)(=O)c1ccnc(N(C2CC2)CC2CN(C(C3CCCC3)=O)C2)n1 C1(CNC(C2N(C(Cc3n(C)ccc3)=O)CC=C2)=O)CC12CCOCC2 C(C1=CCN(C(=O)CCN2CCCC2)CC1)NC(c1cncc(CC)c1)=O C1(NC(c2ncn(C)c2)=O)CCC(CNC(=O)CCC2NC(=O)NC2=O)CC1 C1(C)(C(=O)NC2CCC(N(C(CCC=C)=O)C)CC2)CCCN(C)C1 C1(CC(=O)NC2(CNC(c3n(CC#C)cnn3)=O)CCC2)CC(C)(C)C(=O)N1 N1(C(CCC=C(C)C)=O)CCC(C(=O)NCc2ccnc(C#N)c2)CC1(C)C N1(C(C2(F)CCN(Cc3cc(OCC)c(Br)cc3)C2)=O)CCCC(F)C(F)(F)C1 C1(N(CCCSC)C)CC2CC1CN(C(=O)CCOc1cccnc1)C2 C1(CNC(c2ccn(CCC)n2)=O)CC(C)CN(C(c2ccc[nH]2)=O)C1 c1(C(=O)NC2CCC(CNC(Cc3nn(C)c(Cl)c3)=O)C2)cnn2c1CCCC2 c1(C(N2CCC(C(CC)NC(=O)C(c3cnn(C)c3)C)C2)=O)ccc(C)nc1N c1(CS(=O)(=O)NCCCNC2CCCN2CCN2CCOCC2)cccc(Br)c1 CCC(C(=O)N1CCC(n2cccn2)(CNC(=O)C2=COCC2)CC1)C(C)C c1(NC(C2CC(CC(C)(C)C)C2)=O)c(CO)cnn1C.C12CC(C)(C1)CNC2=O C1(C(=O)NCCC2(O)CCN(C(=O)C(O)CCSC)C2)(CC)CC(C)(C)C1 N1(C(C(C)CO)=O)CCC(O)(C2(NC(=O)CC3COCC(C)(C)O3)CC2)CC1 Cc1cccc(CCCN(C(=O)CC2CCCC(O)C2)C)c1.C(=O)(CO)N c1(C(C23CCCC2NCC3)N2CCC(c3nnc(C)o3)CC2)cccc(Cl)c1F N1(C(C(C(C)C)C)=O)CCn2ncc(CNC(C3(c4cccs4)CC3)=O)c2C1 C1(OC)(NC(C2CC2c2ccc(Cl)cc2F)=O)CCC(C)CC1 N1(C(c2cc(CC)no2)=O)CC2CCCC2(Nc2cc3nncn3cn2)C1 C1(NC(c2[nH]cc3c2CCCC3)=O)C2CC3CN(C(C4CC=CCC4)=O)C1C3C2 CC(Cc1cnc[nH]1)C(=O)NCC1CN(C(c2ncoc2C2CCC2)=O)C1 C(=O)(CCCC(=O)N(CCCN(C(=O)CC1CCCCN1C)C)C)OC C1(Cl)(C(N2CCCC(N(C(CCCCOCC)=O)C)C2)=O)CC2CCC1O2 CCC(CC(F)F)C(=O)NCC1CCCN1C(=O)Cc1cccc(C(=O)OC)c1 N1(C(CCc2n(C)cnc2)=O)C2CCCC1CN(C(C1CCCCS1(=O)=O)=O)C2 Cc1nc2sc1NC(=O)C(C)CN1CCC2CC1.C1(C2(C(=O)O)CC2)CCCO1 N1(C(c2nc(C)co2)C(=O)NCC)CC(Cc2ccccc2)OCC1C C1(C(=O)NCC2N(C(CCCNC(N)=O)=O)CCC2)Cc2ccc(F)cc2O1 Cc1[nH]nc(C(F)F)c1C(N1CCCC(NC(=O)Cc2ccc(Cl)s2)C1)=O c1(C(=O)NCCNC(=O)CC2(O)CCCOC2)cc2cscc2s1 c1(C(=O)NCC2C(C)CN(C(=O)CC(O)CN(C)C)CC2)c(N)cc(Cl)cc1F CCCCCCC(=O)N(C)CC1C2CN(C(c3nc(C)c(C)[nH]3)=O)CC12 C(=O)(C(C)CC(C)(C)C)NC1CCCN(C(c2nc(CCC)sc2)=O)C1 Cc1cnc2n1CCC(C(=O)NCCCN(C(=O)C(C)Oc1ccccn1)C)C2 N1(C(c2cc(NC(C)=O)ncc2)=O)CCC2(CCCC2NC(c2cscn2)=O)C1 Cc1ccc2nc(C(=O)N(C)CCN(C)C(C3CCCO3)=O)ccc2c1 c1(SC)cc(C)ccc1C(=O)NC(C1CCCN1C(C1COCOC1)=O)C c1(C(=O)NC2(C(=O)N(C)Cc3c(C)noc3C)CC(F)C2)cncc(CC)c1 C1(C(N2CCC(C)(CNC(c3cncnc3C)=O)C2)=O)(CC)CNC(=O)C1 Cn1ccc2[nH]c(C(=O)NC3CC(NC(c4c[nH]c(=O)cn4)=O)C34CCC4)cc12 N1(C(C2CCN(C(C(CCC)O)=O)CC2)=O)CC2CC1CS2=O c1(CC)ccc(C(=O)N(CCNC(=O)C(C)OCCOC)C(C)C)c(N)c1 C1(Nc2cc(N(C3CCC(O)CC3)CCCC)ncn2)CC2(CCC2OC)C1 C12CCN(CC1)C2=O.C1(C(C)(C)C)(CN(C(=O)Cc2cn(C)nn2)C)CCCC1 c1(SC)ccc(C)c(C(=O)NC(c2ccccc2)CNC(c2cc(Cl)no2)=O)c1 C1(C2CC2)(NC(COCC(=C)C)=O)CCN(C(=O)C(C)SC(C)C)C1 c1(CC)conc1C(=O)NC1COCC1C(=O)NCC(C)O n1(CC)ccc(CC(=O)NC2CCC2CNC(=O)CC2(SC)CCC2)n1 C#CCC(C)(C(=O)N=c1ccn(C2CC2)[nH]1)NC(C1C2CCC(=O)C12)=O C12(C)CCN(C1)C2=O.CC1(N2CCCC2)CN(C(C2CCCOC2)=O)C1 c1(C(=O)OCC)ccccc1COC(=O)C(F)(F)c1nc(C)cs1 C1(CN(CCCN(c2ccncc2)C)CC)CCCCN1C(=O)CCCF CCCCCCCC(O)C(=O)NCc1c[nH]nc1C(=O)O C1(CC(=O)NC(C)Cn2ccnc2)CCN(C(=O)C(C2(O)CCCCC2)O)CC1 C1(COC)(CNC(=O)CCn2ccc(C)n2)CCCN1C(c1ccccc1)=O c1(C(=O)NC(C(=O)NCCCNC(C)=O)C(C)O)ccc(=O)n(C)n1 c1(C(=O)NC(CNC(c2cc(C)ncn2)=O)C(C)C(C)C)ccc(C)c(Cl)c1Cl C1(O)(CNC(c2c(CC)nn(C)c2Cl)=O)CCCN(C(=O)CSS(C)(=O)=O)CC1 C1(CC)(CC)CCN(C(=O)C(CC(C)C)NC(=O)C(C)N=[N+]=[N-])CC1 N1(C(C(COCC)NC(CCC=CCC=C)=O)=O)CC2CC1CN2C(=O)NC C1(C(=O)NCCNC(CC(C)C(F)F)=O)CC2CCC(C1)C2F c1(C(=O)NC(C2CCCCN2C(=O)C2=CSCS2)C)cccc[n+]1[O-] C#CCCC(C(=O)NC(c1ccc(C)cn1)C)NC(=O)CCn1ccnc1C C1(C(=O)NC(C2CCCC2)CNC(CNC(COCC#C)=O)=O)CCSC(C)C1 C1(C(=O)NCC2CCN2C(C2CCC(=O)O2)=O)(OC)CCC12CCC2 C1(O)(C(C)NC(C=CSC)=O)CCN(C(C2CC(C)CO2)=O)CC1 C(=O)(C(CC(C)C)n1ccnc1)N(CCCCN(C(C(F)=CCC)=O)C)C c1(C(=O)NCC(CNC(C(COC)C)=O)O)cn(CCO)c(=O)nc1O C(=O)(C1=C(c2ccccc2)CCCC1)N1C(CNC(CC(CC)(C)C)=O)CC1 CC(CNC(N1CCOCC(C(=O)O)C1)=O)CC(F)(F)F c1(CC)cc(C(=O)NC2CC2NC(=O)CN(C)C(C)=O)ccc1F N1(C(C2CCC(CC)O2)=O)CCC2CCCC(C1)N2c1nnc(CC(=O)NC)s1 CC1=C(C(=O)NC(C(=O)NCC2=CCCC2)C(C)(C)C)CCC1 C1(NC(C(C(=O)OC)C)=O)CC2CCC1CN2C(c1cnc(OC)nc1C)=O C1(NC(C2CCN2C(=O)CC2C=CCC2)=O)C(O)CC1O CC1(C)CCC(C)(C)c2cc(S(=O)(=O)N3CCC(OCC(F)F)C3)ccc21 c1(C(=O)NC(C2CC=CCC2)CNC(C)=O)cccc(C(N)=O)c1F C(CCC(=O)N(CCC(=O)NC(C)(CO)C1CC1)CCO)C1C(C)C1 CCC(O)C(C)(C)C(=O)N1CCN(C(c2ccnc(S)c2)=O)C(CO)C1 N1(C(CCC=C)=O)CCN(C(=O)C=Cc2ccoc2)CC1CC1CCCC1 CC(C)C(O)C(C)(C)C(=O)NCCC(C)(C)CNC(=O)CCCCC1CCCC1 N1(C(C(C(COC)C)C)=O)CCCN(C(=O)Cc2cc(OC)ccc2Cl)CCC1 C1(c2n(C)nnn2)(NCCc2ccc3c(c2)CC3)CCCC(OC(C)(C)C)C1 C1(C(=O)NC2CCCN(C(C3(CC(=O)OC)CC3)=O)CC2)CCN2CCOCC12 CC1(C)NC(=O)CC1C(N1CCCC(C)(CNC(C2CC2c2ccoc2)=O)C1)=O N1(C(C2(CC)CCOCC2)=O)CC2CCC(CNC(=O)C3=C(Cl)CCOC3)C2C1 CCC(CC(=O)NCCCC(O)C(=O)N1CC2CCC(C1)O2)C(C)C N1(C(C(=O)NC(C)(C)C)CCc2ccco2)CCCC(C(F)F)(C(=O)OC)C1 c1(C(=O)NC(CCC)C(=O)NCC2CCC(C)C2)ncc(F)cc1C C(C(C)(COC)C(=O)N1CCC(CO)C(NC(=O)CCc2cnccn2)C1)OC N1(C(C(C)NC(c2ccco2)=O)=O)CCC2CCN(C(=O)CSC3CC3)CC12 CCC(CC(=O)N(CC(C)(C)CNC(C1CC(=C2CCC2)C1)=O)CC)SC C1(NC(C=CCC)=O)COC2C(NC(c3c(F)ccc(F)c3OCC)=O)COC12 S(=O)(=O)(c1ccc(Br)cc1)N(C(CN(C1CCSCC1)C)=O)CC1CC1 C(CCC1CCC1)(C(=O)NC(c1cccs1)C)NC(c1ccc(SC)o1)=O Cc1nn(C)c(Cl)c1C(=O)NCCN(C(=O)CCOc1cccc(C#N)c1)C1CC1 N(C(=NCCOC1CCSCC1)NCc1ccccc1)C1CC(CN)C1 CCC(C(C)C)S(=O)(=O)NCC1CCCC2(CCC2)C1 c1(C(=O)NC(C2(C)CN(C(=O)CCc3cn[nH]c3)C2)C)cc(O)cc(F)c1 c1(NCC2(CNC(C3(C)CC4CCC(C3)S4)=O)CC2)nccc(S(C)(=O)=O)n1 N1(C(c2ccn(C(C)C)n2)=O)CCC(CO)(NC(=O)C(c2cnn(C)c2)C)CC1 C1(N(CC(=O)NC2(C)CC=CCC2)C)C2CC(O)C1N(C(c1ccncc1)=O)C2 C(=O)(CCCC(=O)NC1CC1NC(c1ccc(C2CCC2)cc1)=O)OCC C1(C(=O)NC(COC(C)=O)CO)CC(F)(F)CN1C(C1OC2CCC1C2)=O c1(-c2c(CC)ncs2)nc(CC(C)OC)nn1C.n1(CC)ccnc1 C1(C2(O)CCOC2)(NC(C(C(C)NC(CSCC)=O)C)=O)CC1 Cc1ccc(CC(C)C(=O)N(CCC(C(C)C)NC(c2csc(F)c2)=O)C)cc1 C(=O)(C#CC1CCOCC1)NC(C1(C2C(C(C)(C)C)C2)CCC1)=O.C1(C)CCCC1 N#CC1CCCC(CC(N2CCCC(CCC3CCC(OC(F)(F)F)C3)C2)=O)C1 c1(C(C(N2CCCC(CNC(CC(C)OC)=O)C2)=O)(F)F)ccc(=O)n(C)c1 Cc1cc(CC(=O)NCCC2(O)CCCN(C(=O)C(C)N(C)C)C2)ccc1Cl N1(C(CCCOCC)=O)CCC(O)(C(C)CNC(c2cccc[n+]2[O-])=O)C1 N1(C(c2c(C)n(C)cn2)=O)CCN(C(c2ccsc2C#N)=O)CC1C c1(C(N2CCCC(N(C(C34CC(OC)C3C4)=O)C)C2)=O)cc2n(n1)CCNC2=O c1(OC)cc(Cl)c(Cl)cc1CNC1C=CC(C(=O)Nc2cc(CO)cc(C)c2)C1 c1(CCCC(=O)N2CC(=C(CNC(C3CC(C)(F)C3)=O)F)C2)ccc(F)c(F)c1 Cc1ccc(C(=O)CN2CCN(C(=O)Cc3ccsc3)CC2C2CC2)cc1Cl CON1CCC(C(=O)NC2CN(C(=O)CSC(C)(C)C)CCC2C)CC1 N1(C(CC(C)OC)=O)CCC(C)(C(=O)NCCC(F)(F)F)C1 CC1CCN(C(=O)C=Cc2cnc[nH]2)CC1NC(=O)C=CCN1CCCC1 c1(NCC2OCCN(C(C3(COC)CCOC3)=O)C2)ncc([N+](=O)[O-])cc1F c1(SCC(c2ccccc2)OCC)cccnc1-c1ncccc1Cl C(C(F)C(=O)NCCNC(=O)NC1(c2cccnc2)CCCC1)N(CC)CC C1(C)(C(=O)NCc2onc(C)n2)CCCN(C(C2CCC=CCCC2)=O)C1 C1(NC(CCC(=O)NC)=O)CCC2CN(C(c3ccn(C)c3)=O)CC2C1 N1(C(C(C)OC)=O)CCC2C1CCN2C(=O)C(c1ccccn1)Nc1ccccn1 c1(C(N2CC(COC)N(C(=O)CCS(C)=O)CC2)=O)cc2c(C)ccc(F)c2o1 Cc1cc(CC(=O)NCCC2CN(C(C3(C#N)CC3C)=O)C2)nn1C C=C(Br)CCC(=O)N(C1CN(C(C2(O)CCC2)=O)C1)C CC(C)(CNC(=O)NC1(Cl)CC1(F)F)CSc1ccccc1 C1(NC(CC(CC)(C)C)=O)CC2CN(c3cc(C)c([N+](=O)[O-])cn3)CC2C1 n1(CCC)cc(C(N2CCC(N(C(=O)C(C)CC(C)C)C)C2)=O)c2ccccc12 c1(C(=O)NCC2C(NC(C(C)c3cccs3)=O)COC2)cnn(C)c1Cl c1(C(=O)NCC(CNC(c2c(CCC)nsc2N)=O)C)cccc2cncn12 N1(C(C(CCCC)N(C)C)=O)CCC2(CCN(C(c3ccnnc3)=O)C2)C1 c1(C(=O)NC2CCCN(C(c3cnc(CC)[nH]3)=O)C2)cnc2ccnn2c1N N1(C(CCC=C)=O)CCOC2(CCN(C(c3cnc4cc(C)nn4c3C)=O)C2)C1 c1(C(=O)NC(C(=O)OC)C)n[nH]cc1CNC(=O)CCOC1CCCC1 C(C)(C)(CC(F)C(=O)NCC(C)(O)COC)NC(C=C(CCC)CCC)=O C1(CNC(=O)CSc2cccnc2)CC(F)(F)CN1C(=O)C(C1CC(F)(F)C1)O c1(OC)cc(N2CC(C)(C)OC2=O)cc(OC)n1 C1(C(=O)NCC(CC=C)NC(c2oc(C)cc2C)=O)(N(C)C)CCCOC1 CCCC(O)CC(=O)NC1CCN(C(=O)Cn2ccc(C)n2)C1 CC1CCC(=CC(=O)NCC2CN(C(=O)Cc3ccc(C(F)(F)F)cc3)C2)CC1 N1(C(C2CCN(C)CC2)=O)CCCCC12CN(C(c1cc(C(N)=O)c[nH]1)=O)C2 c1(-c2cc(C(N=c3[nH]nc(SC)s3)=O)n[nH]2)ccc(S(=O)(=O)NCC(C)C)cc1 n1(CC)ncc(C(=O)NC2(CF)CCN(C(=O)Cc3cc(C(C)C)no3)C2)c1Cl N1(C(CC)CC)C(=S)NC(c2cc(OC)c(O)cc2F)C2=C1C1(CCC1)NC2=O C1(CSC)(CO)CCCN(C(C2(NC(C(CCC)NC(N)=O)=O)CC2)=O)C1 C(C(=O)NC1(CNC(=O)C2=CSCCO2)CCC1)(C(C)(C)C)OC O=S(=O)(c1nc(N2CCC3(CCCCC3)C2)ccc1Br)N.N1CC2CC2C1 N1(C(c2c(C)c(Br)no2)=O)CCOCC(NC(C2(C)CCCS2)=O)C1 N1(C(CN(C2CCSC2)C)=O)CCC(CO)(CNC(=O)Cc2cncs2)CC1 N1(C(CCC2OCCN(C(CCC(=O)NCCC)=O)C2)=O)CCCC(C)(O)CC1 c1(C(C)=O)c(C)[nH]c(C(N2CCCC(N(C)C)C2C)=O)c1C(C)C N1(C(c2nccc(NC(c3cccc(N(C)C)c3)=O)c2)=O)CCN2CCCC2C1 CCC(CC(=O)OC)NC(c1oc(CNC(=O)Cn2nnnc2C)nc1C)=O c1(C(N2CC(CNC(CNC(CCC)=O)=O)N(C)CC2)=O)cc2nnn(C)c2s1 C#Cc1cn(C)nc1C(N1CCOC(C)(CNC(C2CCCCS2(=O)=O)=O)C1)=O C1(NC(CCC=C)=O)CCN(C(=O)C(c2ccc(F)cc2)F)C(C)C1 c1(C(=O)NCCC2(CNC(c3n(CC)nnc3)=O)CC2)cc2c(s1)CCCC2 CC1CN(C2CC2)Cc2cccc(Br)c21.N12C(=O)OC(C(F)(F)F)C1C2 C(=O)(C1=CC(O)C(NC(C2CC3CC3C2)=O)C1)NCC(=O)NCC1CC1 C1(NC(C=CC=CCCCCC)=O)CCN(C(c2ccc(C)cc2Cl)=O)CC1C C(CCC(C)C)(C(=O)N(C)CC1CCOCC1)NC(CC(CC)C1CC1)=O C1(C(N(CC(O)C(F)(F)F)C)=O)CC2CCC(C1)N2C(C1(F)CCCC1)=O c1(CN2CC(NC(CC(CC)O)=O)C(F)(F)CC2)ccc(C)cc1[N+](=O)[O-] C=CCCCCCCC(=O)NCCOCCC(=O)NCCc1cnc(C)[nH]1 FC(F)(F)C(CC(F)F)c1nc(-c2cccc(Br)c2)nn1CC(F)F C(=O)(C1CCc2cc(F)ccc21)N1CCC(NC(c2n(CC)nnc2)=O)CC1C CCCCCCNC(C1(NC(=O)CC2C=CCCC2)CC(F)C1)=O c1(C(=O)NCCCN(CCC)C(c2cc(C)nn2CC)=O)ncc(C)cc1C N1(C(C(CC)F)=O)CCCC(CC)(NC(c2cc(C)c(C(=O)OC)o2)=O)C1 c1(CNC(C(CC)SC)=O)cncc(CNC(=O)C(C)Cc2ccccc2F)c1 Cc1ccc2sc(C(N3CC4CC(C3)C4NC(=O)CC3CCCO3)=O)c(C)c2c1 C(=O)(C1=C(Cl)CC1)NC(C)CCCNC(c1cc(Cn2cccn2)on1)=O N1(C(C(CNC(=O)NCC#C)O)=O)CCC(CNC(C)=O)(NC)CC1 C#Cc1cccc(NC(C)C(N2CCN(C(=O)C(F)n3cccn3)CC2)=O)c1 C1(NC(COc2cc(C)on2)=O)CCC12CN(C(=O)Cc1cc(Cl)cnc1C)C2 N1(Cc2cn(CCCCOCC(=O)OC(C)(C)C)nn2)CCCCC1C(=O)O O=C1CC(=O)NC(C(=O)NC2C=CC(C(=O)NCc3ccncc3Cl)C2)C1 Cc1cc[nH]c1C(=O)N(C1CN(C(=O)C(F)n2cccn2)C1)C c1(N(C(=O)CN2C3COCC2C3)C(c2cn[nH]c2)=O)ccccc1F C1(CNC(c2cocn2)=O)C(C2CC2)CCN1C(c1csnc1Cl)=O C12(CNC(c3ccc(C)cn3)=O)CCC1CCN2C(=O)CSc1nncn1C C=CC1CN(C(=O)CNS(=O)(=O)CCCC)CC1NC(=O)Cc1ncccc1C c1(CC)cccc(CC(=O)NCCN(C(c2cc(C)c(Br)o2)=O)C2CC2)c1 c1(C(N2CCC(C(C)NC(=O)Cn3nccn3)C2)=O)cnc2[nH]nnc2c1 C(=O)(C1CCCc2nc[nH]c21)NCC1(F)CC(CNC(=O)CCOC2CC2)C1 CC1C(=O)OC2C1CCC1(C)CCC3(C=CCCN(C)C3)CN2C(=O)C2CC1CCN2 C1(CNC(Cc2ccn(C)n2)=O)CC2COCC2N1C(c1ccncc1)=O Cc1ccc(CN2CC3(CC3)CC2C(N2CCOC(C#N)C2)=O)cc1O C(CCC(=O)N1CCCC1CC(=O)NCC(C1CC1)SC)OC C1(C(=O)NCCC#C)CC(O)CN1C(=O)C(c1ccccc1Br)OCC.C(C)(=O)O N1(C(c2c(OC)c(C)sc2)=O)CC2CN(C(c3cc(C)c(O)nn3)=O)CC2(C)C1 c1(OC)c(C(=O)NC(CNC(c2ccoc2)=O)C(C)C)cccc1C(F)F c1(C(=O)NC2C3CN(C(C4C(C)C4)=O)C2C3)ccn2c(C(F)(F)F)nnc2c1 N1(C(C(CC)CC)=O)C2CCC(C2)C1C(=O)NC1C=CC(C(=O)NC)C1 Cc1nnn(CC(=O)NCC(C2CCCC2)NC(C2(O)CCOC2)=O)n1 C1(C(=O)NCC2CC(NC(C(CC(C)C)C)=O)C2)CN2CCN1CC2C C1(NC(c2ccc[n+]([O-])c2)=O)CCN(C(=O)Cc2ccnnc2O)CC1 c1(OC)ccc(CC(=O)NCC2CC(C)N(c3nnc(O)s3)C2)c(C)c1 c1(C(N2C(CO)CC(NC(C3CCCS3)=O)C2)=O)c(Cl)ccc2c[nH]nc12 C(=O)(C(O)CCCc1ccccc1)NC(CC)CNC(C1(N(C)C)CCC1)=O FC(F)(F)C(F)(F)N(CC(O)Cn1cnnc1O)Cn1ccnc1 C1(CC(C)NC(=O)CC2(C)CC2(Cl)Cl)CCN(C(c2nnn(C)n2)=O)CC1 CC1(C)CCCC(C(=O)NC(Cc2ccccc2Br)Cc2c(Cl)cccc2Cl)C1 C1(C(=O)O)CCN(N(C(CC)C)C)CC1.c1(C=O)ccncc1F C(=O)(C1=CCCCO1)NC1CN(C(=O)C2=CCCC2)CC1c1cccc(F)c1 C(=O)(C1=C(C#N)CCC1)NC1CCC(N(C(=O)CC2CC(F)(F)C2)C)C1 c1(C(=O)NCC2COCCN(C(CC3C(C)C3)=O)C2)cccc(C#CC2CC2)c1 C1(CN(C(=O)C2=CCOC2)C)COCCN1C(=O)CCCc1ccsc1 N1(C(CCC)=O)CCC(NC(=O)COc2ccc(Br)cc2CC)C(C)C1 S(=O)(=O)(c1ccc(NC2CC3CC3C2)c(Br)c1)N(CCCO)CC CC(=O)CCCC(C)C(=O)NCC1(C(N2CCC3(CCC(O)C3)C2)=O)CCCC1 c1(SCC)cnc(O)c(C(=O)NC2CCN(C(c3cc(C)n(C)c3)=O)C(C)C2)c1 C1(C#N)(C(=O)NCCNC(C2C(=C)CC2)=O)CC12CCC2 C1(C(N2C(C(=O)NC)CCC2)=O)CC(C2CNC2)C1 c1(CNC(C2(F)CCN(C(C)=O)C2)=O)ccc(F)c(C#N)c1 C1(C)(C(=O)NCCC2CCCN(C(C3C(C)OCC3)=O)C2)CCN(C)C1=O N1(C(C(Br)=C(C)C)=O)CCC(C(C)CNC(=O)C(C)Cn2cccn2)CC1 c1(C(N2CCC(C(C)N=c3nc(C(C)(C)C)[nH]s3)C2)=O)ccc2ccncc2n1 C1(NC(c2ccc(C)nn2)=O)CCC12CN(C(=O)CC1CCCC1)C2 N(C1CCCc2c1cnn2-c1ccccc1)C(C1CC(CS(C)(=O)=O)C1)=O CC1=C(C(=O)N2CCSCC2c2ccc(C(F)(F)F)o2)S(=O)(=O)CCO1 CCC(CC)CCC(=O)N1CCCC1C1CCN(C(=O)CCCC(N)=O)C1 C(C(C)(F)C(C)(C)F)n1cc(C2CN(C(C3(C)CCN(CCO)C3)=O)C2)nn1 c1(C(C(=O)NCCCC2CC2)N(CCCO)C(C)C)ccc(C2CC2)cn1 c1(CC)ccc(C(=O)N(C2CCN(C(C3C=C(C)CS3)=O)C2)CCOC)s1 CC(C)CCCC(C)C(=O)NCC(C)(C)C(=O)NC(C1CCOCC1)C C1(CNC(C)=O)C2CCC1CN(C(=O)Cc1cncnc1)C2.C1CCCC(=O)N1 N1(C(CC2CC(=C)C2)=O)CC2(CO)CC1(C(=O)NC(CO)CCC1CC1)C2 CCC(CCC(=O)N(CC(O)C(F)(F)F)C)NC(=O)CCNC(C)=O n1(CC)nc(C)c(NC(C2CC23CCN(C(=O)CN2CCCCC2=O)C3)=O)c1C C1(NC(Cc2c(C)nc(S)s2)=O)CC(O)CN(C(=O)COCC2CC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC(CNC(=O)Cc2cncs2)OCCC1 Cc1ccc(F)cc1-c1nnc(CN2CCCC2c2ccco2)o1 C(C1CC1)(C1CC1)=CC(=O)N(CC(C)C(=O)NC1CCN(CC2CC2)C1)C Cc1cccc2c(C(N3CCC(CNC(=O)CC(C)(C)C)C3)=O)coc12 CC1CN(C(=O)C(F)(F)c2cccnc2)CCN1C(=O)CC1CCCC1 N(C1CCCc2ccoc21)C(C1CN(C(C=CC=CC)=O)CC12CC2)=O c1(C(=O)NC2CCC2NC(c2cccc(C3CC3)c2)=O)ccc2oc(S)nc2c1 CC(CC(C)(C)C)C(=O)N1CC(C)(C)CC1C(N1CCOC(C)(CO)C1)=O C(=O)(C(C)(C)CS(=O)(=O)N1CC(N=[N+]=[N-])CC1C(=O)OC)OC C1(NC(CCNC(C)=O)=O)CCN(C(C2CSC2)=O)CCC1CO n1(CC)nc(C(N2CCCC(CC(=O)N(CC(C)O)C(C)C)C2)=O)cc1C C12(Nc3ncc(C)c(C)n3)CCCC1CN(C(c1cc(C)c(C)nc1O)=O)C2 CC1CC(NC(c2cc(C(F)F)nn2C)=O)CN(C(c2nn(C)cc2N)=O)C1 C1(OC)CSCC1.C1(C(F)(F)F)(C(=O)OC(C)(C)C)CC1 C1(C(N2CC(C(=O)NCC3CCCC3C)(COC)C2)=O)CCCC(=O)C1 N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)CCC1CCC(=O)N1)C2C(C)C Cc1cc(NC(=O)C(O)CCNC(C2(C)CCC(=O)NC2)=O)cnc1O C(=O)(C(O)CC(C)(C)C)NCC1N(C(c2nc(C)c(C)s2)=O)CC1 C1(C#N)(C(N2CC(C(C)NC(=O)Cn3cc(Cl)cn3)C2)=O)CC1(C)C CCCCC(CC)C(=O)N1CC2CCC(C(=O)NC3CCC(N(C)C)C3)(C2)C1 N1(CC(=O)NC(C2CCCCC2)CNC(COCC(=C)C)=O)CCOCC1 N1(C(C(CC=CC)C)=O)CC2(CC(NC(C3(CSC4CC4)CCCO3)=O)C2)C1 CCCCC(CNC(=O)CC(C)n1cc(Br)cn1)NC(=O)CCSC Cc1[nH]c(C#N)cc1C(N1CCC(CF)(NC(=O)Cn2cccn2)C1)=O C1(O)(CNC(C#C)=O)CCN(C(=O)C(c2ccc(F)cc2)F)CC1 c1(OCCC)ccccc1C(N1CC(NC(=O)Cc2ccsc2)C(O)C1)=O N1(C(C2(N(C(c3ncc(C)[n+]([O-])c3)=O)C)CC2)=O)CC2(CNC(=O)C2)C1 C1(CNC(c2cc(C)ns2)=O)CCC2CN(C(c3ncoc3C(C)C)=O)CC12 Cc1ccn(C)c1C(N1CCCC(CNC(c2cc(Cl)ccn2)=O)C1)=O O=C(C1=CC2CCC(C1)C2)N(CCC(=O)NCC1CCC(F)C1)C1CC1 Cc1cnc(C(N2CCOCC2c2cn(Cc3nccs3)nn2)=O)c(Cl)c1 C1(C(=O)NCC2(O)CC(NC(=O)CSC(F)F)C2)CN2CCC1(C)C2 c1(C(N)=O)ccccc1C(N1CCC(C(=O)NCC(CO)CO)C1)=O C12(CC(=O)N(C3CCCN(C(c4snc(C)c4N)=O)C3)C)CCCN1CCC2 N1(C(C(C(C)C)n2cccc2)=O)C2CCC1CC(NC(=O)C(F)(F)C(C)O)C2 Cc1cc(C(=O)N(CCCC(=O)NC2CCN(C(C)(C)C)C2)C)c(C)n1C CC(N=c1[nH]c2c(c(=NCc3cn[nH]c3)[nH]1)SCC2)c1ncnn1C c1(C(=O)NC2(C)CCCN(C(C3(CO)CC(F)(F)C3)=O)C2)cnn2cnnc2c1 c1(C(N2CCC(CCNC(C(CC)OC)=O)C2)=O)ccc(OC2CC2(F)F)cc1 N1(C(C(F)=CC)=O)CCC2(CC1)CC2CNC(c1ccc(CS(C)(=O)=O)cc1)=O C1(NC(C(CC)=CC)=O)CC2CCC1CC2NC(=O)CCOC(C)CC(C)C N1(C(CCCOC)=O)CC(CNC(=O)C(C)Cc2ccccc2)CC(C)(C)C1 C(C1=CCCN(C(=O)CC(C)c2ccco2)C1)NC(C(CO)OC)=O CCC(CC)C(=O)NCC1CCCN1CC.c12ccccc1CNC2=O C1(CC#C)(C(N2CC(OC3C=CC(CCC(=O)NCC(N)=O)C3)C2)=O)CCOC1 c1(C(N)=O)cocc1C(=O)NCC1CCCN1C(=O)CC1CC2(CC2)C1 C1(O)(CCNC(C2C(C=C)C2)=O)CCN(C(C2(C)CS(=O)(=O)C2)=O)C1 C#CCCCC(=O)NC(C1CCCCN1C(=O)C=C(CCC)CCC)C C1(NC(c2c(OC)ccs2)=O)CCCC(C(=O)NCC2(CCO)CN(C)C2)CC1 C(N=c1nc2sccc2c(N2CCc3c[nH]nc3C2)[nH]1)C1N(C(CC)=O)CCC1 CCCCCC(O)CC(=O)NC1CN(C(c2cocc2C)=O)C(C)(C)C1 Cn1cc(CC(N2CCCC2C(C)(C)NC(C2(F)CC=CC2)=O)=O)cn1 N1(C(C(CCC)NC(C)=O)=O)C2CCC1CN(C(C1CC(OC)C1)=O)C2 c1(C(=O)NCC(C(=O)NC2CCC(F)(F)C2)N(C)C)ccc(O)cc1 C1(NC(c2cc3nc(C)sc3[nH]2)=O)CCN(C(=O)COCCF)CC(C)(C)C1 c1(CC)nc(=N)[nH]cc1C(=O)N(CC(O)CN(C)C(C1CC(=O)NC1(C)C)=O)C C(=O)(C1CCCn2cnnc21)N(C1CCC(C)(C)C1)CCOC c1(OC)cc(C(N2CCCC2CCCNC(=O)CSCC2CCCCO2)=O)sn1 C1(C(=O)NCc2c(SC)c(F)ccc2)CC2COCC(C1)C2 O=[N+]([O-])c1ccn(-c2ccc(F)c(CNC3CCOC3c3ccccc3)c2)n1 c1(C(N2CCC(C(C)C(=O)N(C)Cc3cncs3)C2)=O)ccc(O)c(F)c1 C1(c2nnnn2C)(NC2(CCOC)CCOC2)CC2CC(O)C(C1)N2C c1(N(CCC)C(=O)Oc2ccc(-c3cccs3)cn2)ccc(-c2cscn2)cc1 C1(COC)CCN(C(=O)Cc2c[nH]c(C(N3CCC3C(=O)OC)=O)c2)CC1 N1(C(CCS(=O)(=O)NC)=O)CCC(C)(C)C(C(N2CCCC2CO)=O)C1 C(=O)(C(C)(C)C(C)(C)O)NCC(C(C)(C)C)NC(c1ccc(Br)o1)=O C(=O)(C1CCc2c[nH]nc21)N1CC(CC(CNC(c2c(C)sc(O)n2)=O)(C)C)C1 C1(NC(c2n(CC)ncn2)=O)CC2CC(C1)N(C(c1ccnc3c1CCC3)=O)C2 c1(C(=O)NCC(CC)NC(C2C3CCC(F)(F)C23)=O)cc([N+](=O)[O-])cnc1N C(CC(O)CNC(=O)CCN(CCC(C)(C)C)C)NC(C1(CC(C)=O)CC1)=O C1(OCCCN(C)C(c2cnc(Cl)[nH]2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1 CC(=Cn1ccnn1)C(=O)NCCC1CN(C(=O)CC2CCCCN2C)CC1C C#Cc1cccc(C(=O)NC2(C)N(Cc3cccc(CC)c3)CCOC2)c1 C1(CC)CN(C(C2CCCCN2C)=O)CC1NC(c1ccc(C(N)=O)cn1)=O C(CCCC(=O)NC(C1CCCN1C(=O)C(C)C)C)(OC)OC C1(C(N2CC(O)CC2C2CC2)=O)CCN(C(=O)CC2(O)CCCCC2)C12CCC2 CC1CC(=O)NC1C(=O)NC1(CNC(c2[nH]c(O)nc2C)=O)CCC1 C1(OC)CCCN(C(C2CCCC2CNC(=O)C(C)(C)n2cccn2)=O)C1 C(=O)(C(O)C1=CCCCC1)NCC(CCCC)NC(c1cccc(Cl)c1F)=O N(C1CCC(NC(=O)C(CC)(CC)OC)c2ccccc21)C(CSCCC)=O C1(NC(COC(C)=O)=O)CCC(C#N)CC1.C12CCC1NC2=O N1(C(C(C)OCCC(C)C)=O)CCC(C2(NC(C3CC4(CC4)CO3)=O)CC2)CC1 N1(C(C2CCCC(C)C2)=O)CC2CC(NC(c3cccc(N(C)C)n3)=O)C(C2)C1 C1(C(=O)NCC(CO)NC(C2OCCO2)=O)(OC)CCCOC1 C1(NC(C2(CC)CCCC2)=O)CCCCC1NC(C1CCC(C)CC1)=O C1(SC)CN(C(c2ccc(C#N)[nH]2)=O)CC1NC(C1CS(=O)C1)=O c1(C(N2CC(NC(CC(CC)C)=O)CC2(C)C)=O)cc(=O)n(C)cc1Br C1(N(C(C(C)C#N)=O)CCF)CCCN(C(=O)C(=O)NCCC(N)=O)C1 c1(NC(N2C(C)(CNC(c3c(OC)cccc3)=O)CCC2)=O)oc(C)nc1C#N C(CCCCC(=O)NC1CCCC1(C)CN(C(=O)CC(C)(C)SC)C)SC C1(C(=O)NC(C2CCC2)C)CN(C(C2CC(F)(CF)C2)=O)CC1C1CC1 c1(CNC(=O)NC(c2ccccc2F)C)ccc(C(C)(C)C)cn1 c1(NCc2cc(C)[nH]n2)nc(N2CCC(N(C)C)C(C)C2)nc2c1cnn2C NC(=O)C1=NOC(CNC(=O)CCNC(c2csc(Cl)n2)=O)C1 N1(CC2(NC(C(C3CCSC3)N(c3cc[nH]n3)C)=O)CC2)CCCCC1 c1(NC(C(C)N(C(c2n(CCC)ncc2)=O)CC)=O)ccc(F)cc1CO c1(C(C(=O)Nc2ccc(OC(F)F)cc2)(F)F)c(F)cccc1Cl.N1CCCC1 Cc1ccc(C)c(C(=O)NCCCCCCNC(c2occ3c2CCC3)=O)c1C c1(CC(=O)NCC(C2CC2)NC(C=CC2N(C)CCC2)=O)ccc([N+](=O)[O-])c(N)c1 CN1CC(C(N2CCOCC2C(=O)Nc2cccc(CCF)c2)=O)CCC1=O C(N=c1cc(C)nc(NC2CCCCN2CC)[nH]1)C1(OCC)CCCSC1 C1(O)(CN(C(c2c(C)nns2)=O)C)CCN(C(c2ccncn2)=O)C1 C1(OC)CN(C(c2cn(CCO)nn2)=O)CC1C(NC[Si](C)(C)C)=O C1(CNC(=O)C=C(C)CNC(C2(COC)CC(=O)C2)=O)(OC)CCCCC1 C1(NC(C=CSC)=O)CCOC2(CCN(C(C3CC3CC(C)C)=O)CC2)C1 c1(N2C3CN(C(C(CC)CCOC)=O)C(CC3)C2)nc2ccc(Br)cc2s1 c1(C(=O)NCC2C(C)CN(C(C3CNC(=O)N3)=O)CC2)cnn2ccccc12 C(C(C(=O)N(C)Cc1cnc(C)s1)NC(=O)Cc1cnnn1C)OC c1(CC)cnccc1C(=O)N(C)CC1C2CN(C(=O)CSCC(N)=O)CC12 c1(C(N(CCCN(C(c2c(C#N)cnn2C)=O)CC)C)=O)ccc(=O)n(C)c1 N1(C(CN(CCCCCC)C)=O)C(CNC(=O)CCN(C)CC)CC2COCC12 N1(c2n(C)c(C(c3cccnc3)O)nn2)CCC(C2CC2)C1c1nnc(O)o1 C(CCCCCC(=O)N1CC(SC(F)F)C1)NC(=O)CN1CCCCCC1 C1(CNC(C(CC)C(C)(F)F)=O)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)CC2)O1 CCC(C)(CO)C(=O)N1CC(NC(=O)COc2ccc(F)cn2)C2(CC2)C1 C12(C(=O)NC(CC)C)CC(CO1)N(C(c1c(C)coc1CN)=O)C2 CC1C(C(=O)NCc2nc(N(C)C)n[nH]2)CCCN1C(c1cccnn1)=O CC(C#N)C(=O)N1CC(N(C)C(c2cc(C3CC3)no2)=O)C1 C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(=O)CC(F)(F)F)C2(CCC2)C1 C1(C(N2C(CNC(c3cc[nH]n3)=O)CCC2)=O)CCCCC12CC2 C(CNC(C1CC(OCC)C1)=O)(CC)(CC)NC(c1ccccc1-c1ncc[nH]1)=O c1(NC2CCC(C(=O)NC(C(=O)N(C)C)(C)C)OC2)ncnc(C(F)(F)F)c1Br C1(C(N(CC(CC)NC(COC2(C#C)COC2)=O)CC)=O)C(F)(F)C12CC2 C1(C(C)C)CN(C(c2cnc(OC(C)C)cn2)=O)CCN1C(=O)CCS(C)=O c1(C(=O)OCC)cncc(CN(C2CCCC2)CC2CCNC2=O)c1 CC1CCC(NC(c2cc(C(F)F)n(C)n2)=O)CN1C(c1cnsc1)=O N1(C(CCCCOCC)=O)CC(C)(C)OC2(C1)CN(C(C1CCC(F)CC1)=O)C2 C(=O)(C(C)(F)C(=O)NCCC(C)(C)NC(=O)COC1CCCC1)OC c1(-c2n(CC)cnn2)cccc(NC(C2CCC(NS(=O)(=O)C3CC3)C2)=O)c1 c1(NC(C2CCCO2)COCCCOC)nccc(=NCCC#N)[nH]1 c1(C(N2C(CC=C)CCCC2)C(=O)NCCCC)csc2ccccc2c1=O C1(NC(C2CCC(NC(C3(C=C)CCCC3)=O)C2)=O)CCCCNC1=O n1(CCC)ccc2cc(NCCC3COC4(CCC4)CO3)ccc12 c1(C(N2CC(NC(=O)Cc3cnc[nH]3)C2)=O)cnc(COc2ccccc2)s1 N1(C(c2cc(C(=O)OC)ncc2F)=O)CCC2CN(C(c3ccoc3)=O)CCC12 C1(C(=O)NCCCSCC)(NC(c2conc2C2CC2)=O)CC(O)C1 CC1(C)CCC(C(=O)NC2CCN(C(C3CCCS(=O)(=O)C3)=O)C2(C)C)CC1 CCCC(C(=O)N(C(C)CNC(c1nsnc1O)=O)C)S(N)(=O)=O CS(=O)(=O)c1cc(C(N2CCC(NC(C3CC=CCC3)=O)C23CC3)=O)cc(N)c1 C(=O)(CCCCCNC(c1coc2c1COC2)=O)N(CC(C)(C)C)C1CC1 O=C(CCC#Cc1ccccc1)NCC1COCC1NC(C1(CO)CC1)=O C(C)(CCC(=O)NC(C)C(CO)NC(=O)C(c1ccnn1C)C)SC C(C(CC(C)O)c1ccccc1)NC(N(CCCCC)CCO)=O c1(OC)cc(N)c(C(=O)NCC2CCN(C(C3(C)CCCC3(F)F)=O)C2)cc1F N1(C(C2CC3CC3C2)C(=O)NCCCSC)C2CCC1CN(CC(F)F)C2 c1(CN(C(C)C(O)Cc2ccccc2)C=O)ccc(CC#N)c(F)c1 C(=O)(C1CCCn2cc(C)nc21)NC(C(C)(C)NC(CSCCC)=O)C C1(CC(=O)NC(CC(=O)NC2C(OC)CC2O)C2CC2)CCC(C)(C)O1 CCN(OC)C(=O)C(C)N(C)C(c1nscc1C)=O c1(OC)ccc(C(N2CCCC(O)(CN(C(=O)Cn3cnnn3)C)C2)=O)c(O)c1 c1(-c2cn(C(C)(C)CO)nc2)cccc2[nH]c(C(=O)Nc3coc(Cl)n3)cc12 N1(C(C(=Cc2ccccn2)C)=O)CC2CCC1C2NC(=O)C1=COCC1 CCCCC(CNC(=O)C=C(CC)CC)NC(=O)CC1(O)CCOC1 c1(NCC(N2CCN(CC)CC2)(C)C)ccc(Cl)c(C)c1Cl c1(C(=O)NC(CCNC(c2cc(C)nc(O)c2)=O)(C)C)cc(F)c(C#N)c(F)c1 c1(NC(CNC(C(C)OCC=C)=O)=O)sc2c(c1C(N)=O)CCC2.c1(N)cnsc1 C12(CNC(CCCCCSC)=O)CCC(CN(C(=O)C3=CCC(C)CC3)C1)C2 N1(C(COC)=O)CC(C(=O)NCCCCc2cnn(C)c2O)C(C)(C)C1 C1(CC)(CC)CC(C(=O)NC(COC(C)C)C(=O)NC2CCN(CC)C2)C1 C1(C(N2C(CN(C)C(c3ncc(Cl)nc3Cl)=O)CCCC2)=O)CC2C(C1)C2(C)C Cc1cccc(Cl)c1C(=O)N(C1CCC(NC(c2cc(Cl)cn2C)=O)CC1)C Cc1cnn(C(C)C)c1C(=O)N(C)CC1CCN(C(=O)CC(C)(C)C2CC2)C1 c1(OC)cc(NC(c2ccc3c(cnn3C(F)F)c2)=O)cc([N+](=O)[O-])c1 C1(C(N2CC(C)C(NC(=O)C(C)NC=O)C2)=O)CCCCCN1C N1(C(CCCOCC)=O)CCCC(NC(c2cn3ccsc3n2)=O)C1C N1(C(CCC(=C)Cl)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1C1CCCC1 N1(C(c2cccn3nccc23)=O)CCn2c(n[nH]c(=O)c2=O)C1 Cc1nc(C(C)NC(=O)CC(C2CC2)NC(c2cc(Cl)cs2)=O)n[nH]1 c1(OC)ccc2cc(C(=O)NC3CN(C(c4cnn(C)n4)=O)CC34CC4)[nH]c2n1 C1(O)(C(N(C)CC2CCCN(C(C3(CSC)CC3)=O)C2)=O)CCC(C)(C)CC1 C=C(Cl)CCC(=O)NC(CN(C)C(c1coc(-c2ccccn2)n1)=O)CC CC1C2CCN1C(=O)C1(CC1)CN2.C1(C(=O)ON)CCCCC1c1cccnc1 C(=O)(CCCC(C)NC(=O)CCC1CCC(=O)C1)N(CC(=O)OC)C1CC1 Cc1cccc(C(O)C(N2CCC(NC(c3nccn3C)=O)C2)=O)c1 C(c1nc2ccccc2s1)=CC(=O)NC1CCC1NC(C1CCCCC(=O)N1)=O N1(CC(CC)CC)CCCC(C(=O)NC2CONC2=O)C1 Cc1cc(F)c(C(=O)NC(CO)CCCNC(c2ccn(CCF)n2)=O)cc1F c1(C(n2cc(C3CC4CC4N3C(=O)C(O)C(C)(C)C)nn2)C)c(F)cc(Cl)cc1F CCC(C)(C)C(O)C(=O)NCC(C)NC(c1coc2c1CCCC2)=O c1(C(=O)NC2CCC(NC(CC(CC)C3CC3)=O)CC2)cc2c(Cl)cccc2s1 C1(C)(CNC(c2c(C)n[nH]c2)=O)CN(C(C2CCOC2=O)=O)C(C)(C)C1 C1(CNC(COCCCCC)=O)CN(C(c2cc(CC)[nH]n2)=O)CCC1(F)F NS(=O)(=O)c1n[nH]cc1C(N1CC=CC(NC(=O)C(F)OC(F)(F)F)C1)=O N1(C(CC(C(C)OC)NC(C(CC(CC)(C)C)=O)=O)=O)CCCC(N=[N+]=[N-])CC1 N1(C(C2(C)CCCO2)=O)CCN(C(=O)CNC(C2CC2C(F)(F)F)=O)CC1 N1(C(c2cnn(C)c2Cl)=O)CCC2C(C1)CN2C(=O)Cc1csnn1 c1(NC(COCc2ncc(C)o2)=O)cccc(NCc2c(C)coc2C)c1 C1(CC(=O)NC(C2(C(=O)N(C)CC3CCCC3)CC2)C)CCCCC1 C=C(Cl)C(C)(C)C(=O)N1CC2(C1)CN(C(C1CCCCC1(C)C)=O)C2 N1(C(c2c(C)ccc([N+](=O)[O-])c2)=O)CCC2C(CCCN2C(c2ccsc2)=O)C1 c1(C(N(C2CCN(Cc3nc(CC)sc3)C2)C)=O)cnn2cccnc12 c1(CC(=O)NC2C(CNC(CC(=C)C)=O)CC2)c(F)cccc1Br c1(C(N(CC(=O)NC(CC=C)C)CCOC)=O)cnc(COCC)s1 c1(C(N2CC3(CC(NC(C4CCCCS4)=O)C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1O C(C(C)(C)C(C)(F)F)NC(C1(NC(CCSC)=O)CC1)=O.C(C)(=O)O Cc1nn(C)c(C(N2CCC(N(C)C(c3cncc(N)c3C)=O)C2)=O)c1Br C=CCC(C)(C)CNC(=O)C(C1CCN(C(=O)CN(C2CC2)CC)C1)F C1(N(C(=O)C(C)(C)C2CCOCC2)C)CCN(C(c2ccc(Cl)o2)=O)CC1 c1(C(C(=O)NC2CC(C)(NC(C(C)SC)=O)C2)C)ccc(CC(C)C)cc1 N1(C(CSc2n(C)cnn2)=O)CCCC12CCN(C(c1c[nH]c(C(N)=O)c1)=O)C2 c1(C(N2C3CC(NC(C)=O)CC2CC3)=O)cc2nccc(Cl)c2s1 c1(CO)nc2n(n1)Cc1cc-2nn1C.C1(C)(C2CC2)CC1 N1(C(C(CC)C)=O)CC2(C)CC1(C(=O)N(C)CC)C2 N1(C(Cc2c(C)non2)=O)CC(NC(=O)C(C)OCC2CC2)CC12CCCC2 C1(NC(c2cc(C)c(C)[nH]2)=O)COCCN(C(C2CC23CC(O)C3)=O)C1 c1(CC)nc(=N)[nH]c(=NCCC2CCN(C(c3ccccc3COC)=O)C2)[nH]1 C1(CC(=O)OC)CC2(CCC2)CN1C(=O)NC1CC1C1CCC(N)CC1 C1(NC(CC2C=CC(NC(CC=CCC)=O)C2)=O)CCCCNC1=O C#CCCCC(=O)NC1C2CN(Cc3sccc3Br)CC12 Cc1c(C(=O)NCC=C2CCN(C(=O)CC3(C)CC3(F)F)CC2)cnn1C1CC1 c1(C(N2CC=CC(NC(CCc3c(C)n[nH]c3C)=O)C2)=O)ccc2nccn2n1 c1(C(=O)NCCC2CC(NC(CNS(CC)(=O)=O)=O)C2)ccc(SC)nc1 N1(C(C)C)CCC(C(=O)NC2CN(C(C3CC4CC4C3)=O)CC2O)CC1 c1(CC(N2C(C)CCC(NC(=O)CC(C)(C)C)C2)=O)ccc2nc(O)[nH]c2c1 CN1C2CCC1CC(C(=O)NCC1CN(C(c3ccncc3F)=O)CC1O)C2 N1(C(CCN(c2ccccc2)C)=O)CC(CO)(NC(=O)Cc2n[nH]c(=N)s2)C1 CC(C)C(O)CCN=c1[nH]c(=NCc2ccnc(OCCO)c2)c2[nH]ccc2[nH]1 c1(OCC(N2C(CNC(c3c(C)ocn3)=O)CCC2)=O)ccc(Br)cc1 c1(C(N2CC(O)(CNC(c3c(C)n(C)nc3Cl)=O)C2)=O)n[nH]c2c1CC(C)CC2 Cc1ccc(C(=O)NCC2C=CCN2C(=O)Cc2nncn2C)cc1C C1(C(=O)NCC2(CO)C(C=C)C2)CCN(C(c2c[nH]c(=NC)s2)=O)C12CC2 C(=O)(C1=CCCN(C(=O)CCc2cnc(C(C)NC(=O)OC(C)(C)C)o2)C1)NC c1(C(C(=O)NCC2C(NC(CCC3CC(OC)C3)=O)C2)OC)ccccc1Cl C1(NC(C2C(NC(c3cc(OCC)no3)=O)CC2)=O)CC(C)OC1=O N1(C=O)CC(F)(F)OC(F)(F)C1.N1(N(c2ccccc2)COCC)CCOCC1 C1(CNC(C=C(CCC)C)=O)CC(CNC(c2cnc(CC(C)C)[nH]2)=O)CO1 c1(CCC)nc(C(=O)NCC(C2CCCCC2)NC(=O)COCC(F)F)cs1 C(=O)(C(C(=O)N(C1CCCCC1NC(C12CC(C)(C1)C2)=O)C)C(C)(C)C)OCC C1(C(=O)NCC(C2CCCCC2)NC(c2ccc(C(C)C)s2)=O)CC=CCC1C CCCCCC(F)C(=O)NCC1CC(C)CCN1C(=O)C(C)SC N(C1c2ccccc2CC1O)C(N1CC(C)N(CC(N2CCOCC2)C)CC1)=O N1(C(CNC(c2ccccn2)=O)=O)CC=C(CNC(C2CNC(=O)N2)=O)CC1 Cc1oc(C(C)C)nc1C(=O)NCC1CCCCN1C(C1CCCC(=O)N1)=O c1(C(N2CC3C(CCNC(CC=C)=O)(CC3)C2)=O)nc2ccccc2cc1Cl C(C1(C)CCOCC1)=CC(=O)NCCNC(CN1CCC(C)C1)=O Cc1nccc(C(=O)NC2C=CC(CC(N3CCC(C)(C(N)=O)C3)=O)C2)n1 C1(N(C(c2cncnc2)=O)CC)CCCN(C(=O)C(C2CC2)C2CC2)C1 C1(O)(C(N2CCC(NC(C(=O)NCC)=O)C2)=O)CCSCC1 c1(C(=O)NC(CN(C(C2C(C)OCC2)=O)C)(C)C)ccc(C#N)[nH]1 c1(C(C)C(=O)NCC2CC(NC(=O)C(F)(F)c3ccnn3C)C2)ccc(F)cc1 C1(C(=O)NCCC(C)NC(=O)C(C)(C)c2cc[nH]n2)CCC2(CC1)COCCO2 Cc1cc(CNC(C2CCCC(NC(=O)Cc3cnoc3)CC2)=O)cc(C)n1 CC1(C)CCC1C(=O)NCC1(CNC(C2CS(=O)(=O)C2)=O)CCC1 c1(NC(C23CC(NCc4ccc(OC)c(C)c4)(C2)C3)=O)ccc(C#N)c(Cl)c1 C1(NC(Cc2ncc(C)s2)=O)CCCN(C(c2c(Cl)c(C)nn2C)=O)CC1 c1(C(C)(C)C(=O)NC2CCC(NC(C3CCOC3C)=O)C2)cccc(O)c1 c1(C(=O)NCC2(O)CN(C(C3CC(=O)N3)=O)C2)ncc(Br)cc1F C#CC1CCC(C(=O)NCC2CN(C(=O)Cc3ccc(F)c(CC)c3)C2)CC1 N1(CC(C)C)CC(C(=O)NCC(F)CNC(C2(n3cccn3)CC2)=O)CC1=O c1(C(=O)NC2CCC(C)N(C(c3nccnc3N)=O)C2)c[nH]c2cc(Cl)ccc12 N1(C(C(C(C)c2ccccc2)O)=O)C2CCC1CC(c1cn[nH]c1)C2 c1(NC(C23CC(C(N4CC5CC4CO5)=O)(C2)C3)=O)ccc(Br)c(C(F)(F)F)n1 C(=O)(C1=C(C)OCCS1)N1CC(NC(CCOCC#C)=O)C(OC)C1 Cc1cccc(CC(=O)NCC2CC(F)(CNC(=O)CC3CCCSC3)C2)c1C CC(C)C(O)C(C)C(=O)NCCCCCN(C)C(C1(O)CCCC1)=O C1(NC(c2c(C)cno2)=O)Cc2ccccc2C1NC(=O)C(C)CS(C)(=O)=O CCC(C)CC(=O)C(=O)NC1CCCC(C(=O)NCCSC(F)F)CC1 C1(NC(C2(NC(CC3CCN(C)C3)=O)CCCCC2)=O)CCC(=O)N(C)C1=O C(=O)(C(O)CCNC(=O)C=CCN(C)C)NC1(CC=C)CC1 C1(NC(C2C(C)=CCS2)=O)CCC(C)(CNC(=O)CN2CCNC(=O)C2)CC1 c1(OCC(=O)NC(CCN(C(C)=O)C)C(C)C)ccc2c(c1)CCCC2=O C12(CNC(CC3(C=C)CC3)=O)CC3CC(CC(C3)C1NC(=O)C(F)CC1CC1)C2 Cc1cn2c(n1)CCC(C(=O)NC1CC3CC(O)C1C3)C2 C1(C(N2CCN(CCN(C(c3c(C)occ3)=O)C)CC2)=O)CCC2(C1)CC2(F)F c1(CC(=O)NC2CCC(C(N(CCCC)CCCO)=O)CC2)cccc(C#N)c1 N1(S(C)(=O)=O)CCN(CC(=O)NC2CC(NC(C3(N=[N+]=[N-])CC3)=O)C2)CC1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)NC1CN(Cc2cn(C)nc2)CC1C#N c1(N2CCC(NC(CC(CC=C)(C)C)=O)CC2C)cc(S(C)(=O)=O)ncn1 c1(C(C)=O)ccc(C(N2CCC(N(C(=O)CSCC3CCCO3)C)C2)=O)[nH]1 Cc1ccc(F)c(C(=O)NC(CCN(C(=O)CCCCCF)C)C(C)C)c1O CCCC(C)(CCC)C(=O)NC(c1ccc(C)cc1)CNC(c1cocn1)=O NC1CCc2cccnc2N(C(c2cc(C(F)(F)F)c(Br)s2)=O)C1 C1(CNC(=O)CCF)CC=CCN1C(=O)C(O)CC1CC1 c1(C(C(=O)NC2(C#C)COC2)O)ccc(OC)c(OC)c1 C=CCCCCCC(=O)NC(C)CC(C)NC(c1cc2sccc2[nH]1)=O N1(C(c2cnc(OCC)s2)=O)CC(NC(=O)CC2CNC(=O)O2)C(SC)C1 C=CCCCC(C(=O)NCC(=O)NC(C)(C)C)NC(C1CC12CCCC2)=O c1(C(N2CC3CCN(C(c4[nH]n(C)c(=O)n4)=O)C3C2)=O)cc2ccc(Cl)cc2o1 c1(C(N2CCCC(C)(NC(COCCCOC)=O)C2)=O)cc2c(s1)CCOC2 C1(NC(C=CSC)=O)CC(NC(C2CC2c2cncn2C)=O)C(O)C1 C(=O)(C(Cn1cccn1)NC(=O)NCCC1CC1)OC(C)(C)C N1(C(c2c(OC)cccc2)=O)CCC(C)C(CC(F)(F)F)C1.C1CC(=O)O1 C1(CNC(c2nnn(C)n2)=O)CCC(CNC(C2C3CCC(F)C23)=O)CC1 N1(C(c2cc(C)c(N)cn2)=O)Cc2nccn2CC(NC(=O)CC2CC2(C)C)C1 Cn1cc(C(=O)NCCN(C(C2CCO2)=O)CS(C)(=O)=O)c(C2CC2)n1 Cc1ocnc1C(N1CC(NC(=O)CCN(C)C(=O)OC(C)(C)C)C1)=O C1(NC(C(=O)NC2C(OC)COC2)=O)CCN(C(=O)NCc2ccccc2)CC1 CC1(C)CC(NC(C2CN(C(=O)CC3CC3(C)C)CC2F)=O)CO1 N1(C(c2occ(C)c2)=O)CC2(CCN(C(=O)C=Cc3ccccc3Cl)C2)C1 N1(C(C(c2ccccc2)N(C)C)=O)CCC(N(C(=O)CC2CC=CC2)CCO)C1 CN1CCOC(CONC(c2cccc(C(=O)NS(C)(=O)=O)n2)=O)C1 C(=O)(CN=c1[nH]c2ccccc2s1)N(CCN(C(C(COC)C)=O)C)C CC1CC(NC(=O)CSc2ccccc2)CN(C(=O)Cc2n[nH]c(=N)s2)C1 C(CCCCC(=O)N1CCN(C(c2n[nH]cc2C(C)C)=O)CC1)SC C(CCC(=O)NCC(O)CCC)N(C(CCSCCCC)=O)CCC O=C1NCC2(CN(C(c3nccc4[nH]ccc34)=O)C2)N1.C1(=O)C2=CCN(C2)N1 N1(C(C(CC)Nc2ccccc2)=O)CCCC(NC(=O)CC2CCNC2=O)CC1 N1(C(COCCCC(C)C)=O)CCC(NC(C2CC(C(C)(C)C)C2)=O)CC1C CC(N=[N+]=[N-])C(=O)N(C(C)(C)CC(=O)N1CCN(C(=O)CCO)CC1)C c1(SC)cc(N2CCN(C(c3sc(C)nc3C)=O)CC2)nc(SC)n1 C(=O)(C(CC(F)F)N(C(=O)C=Cc1cnccn1)C)NCC(n1cccn1)C O=C(CCS(=O)(=O)c1ccc(F)cc1)OCc1cscc1C(F)(F)F C1(CNC(C(C)c2ncco2)=O)CC12CCN(C(c1ccoc1Cl)=O)CC2 C(C(CC(=O)N(C)CCS(C)(=O)=O)C(F)F)NC(C(C)(C)NC(C)=O)=O C(=O)(C1Cc2c(Cl)cccc21)NC1CCN(C(c2c(OC)cnc(F)c2)=O)C1C C(Cc1ccccc1)(CC(F)(F)F)NCc1nc(N(C)C)sc1 N1(C(c2cc(C)sc2)=O)CCC(Nc2ncc(C#N)c3ccsc23)C2(CCC2)C1 N1(C(C(COC)O)=O)CC2CCC1C2NC(c1ccc(N2CCCC2)cc1)=O Cc1nc(N2CCC(CCNC(=O)NC3CC(C)OC3C)C2)c(C)c(Cl)n1 C(C)(c1ccccc1OC)=CC(N1C2C(CNC(C(CC)(C)CO)=O)C(C2)C1)=O C=CCCC(C(=O)NCC1CN(C(=O)OC)C1)NC(c1cn(CC)nc1C)=O c1(NC(N2CCCC(CCCC)C2)=O)sc(OC(=O)C2CC2)cc1C N1(C(C=COCC)=O)CCC(C2CCN(C(c3cn(C4COC4)nn3)=O)C2)C1 CCC(C)(CN=c1[nH]c(NCCCc2cnccn2)nc(=N)[nH]1)C(C)O c1(C(N(CC(C)O)CCNC(C2(C)CCCCC2)=O)=O)ccc2c(c1)nnn2C C(=O)(C1=Cc2ccccc2OC1)NC1C2CCN(C(C(C)CC(N)=O)=O)C2C1 C1(NC(C(n2c(C)ccn2)C)=O)CCCC(NC(=O)C(C)OCOC)C1 O=C(CS(=O)(=O)CCO)NCCC1CCCN(C(C2CC3C=CC2O3)=O)C1 c1(NC(COC)CC2CCOCC2)cc(C(=O)NC(C)C)ccc1[N+](=O)[O-] CC1(C)CC(C(=O)NCC2(CNC(C3CC(=C4CC4)C3)=O)CC2)CNC1=O N1(C(CSc2c(C)n[nH]c2C)=O)CCN(C(=O)C(N2CCCCC2=O)C)C(C)C1 C(CC(=O)NC1CCOC1=O)(C(F)(F)F)NC(CCCC=C)=O S(=O)(=O)(c1cnn2ccc(NNCC3CCOCC3C)nc12)N(CC#CC)C C1(CC(=O)N(CCOC)CCNC(c2ccn(C(F)F)n2)=O)CC2CCC1O2 C1(CCCNC(CCN(C(C)=O)C)=O)CCN(C(c2ncsc2N(C)C)=O)CC1 CN=c1[nH]cc(C(N2CC(OC)CC2CNC(=O)C2=CCOC2)=O)o1 c1(-c2nc(C)c(NS(=O)(=O)c3ccc(Cl)s3)s2)c(C)ccc2ncccc12 c1(C(=O)NC2CCCN(C(CC=CCC)=O)C2)ccc2c(c1)oc1ccccc21 c1(C(N2CCC(C(CNC(C(CC)O)=O)(C)O)CC2)=O)ccn2cncc2c1 N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2ncncc2Cl)=O)C2COCC12 CCC(C)(O)C(=O)NCc1c[nH]nc1C1CCN(C(c2cc(C(F)F)n[nH]2)=O)C1 C(=O)(C(F)C(C)(F)F)NC(COC(C)C)C(=O)N1CC=CC1CF N1(C(CC(CCC)O)=O)CCC2CC1CN(C(=O)Cc1cccc(C3CC3)c1)C2 C(=O)(C(CCS(C)=O)N(C)C)N(CC(C)CNC(C1CCC(CC#N)CC1)=O)C c1(CNC2CCC(C(=O)Nc3cc(C)c(Cl)cn3)OC2)c(O)cc(F)cc1F C1(C)(C(=O)OC)CCN(C(=O)CC2CCCN(C(c3cccn3C)=O)C2)C1 O=C1Cc2c(C(=O)NCC(F)CNC(=O)Cn3cnnn3)ccnc2N1 N12CC(O)CC1C2=O.C1(NC(=O)OC)(CNC(=O)C(=O)NCC(F)F)CCC1 c1(CN2C(C(=O)NCCC(=O)OC)CSCC2)ccc(Cl)cc1OC N1(C(C2=C(C)CCC2)=O)CC2=C(C1)CN(C(=O)C(C)(C)C(C)C)C2 C(=O)(C1CCCc2sccc21)N(C1CN(C(CC=CC=C)=O)C(C)(C)C1)C1CC1 C(CC(N)=O)(C(=O)NCC1(F)CCCN(C(=O)C(=O)NC2CC2)C1)NC(CC(C)C)=O c1(C(=O)NCC(CC)NC(c2cccc(=O)o2)=O)c(OC)c(Cl)cc(O)c1Cl C1(C(=O)OCC)CN(C(=O)CC2COCC(C)O2)CCC1=O S(=O)(=O)(c1ccc(Br)cc1N)N(C)Cc1ccc(SC)o1.N12CCCCC1C2 c1(OC)ccc(OCC(=O)NCC2CC(O)CN2C(C2CCCNC2=O)=O)cc1 C#CCCCCCC(=O)NC1CCN(C(c2cnc(C)[nH]c2=N)=O)C1(C)C c1(C(N2CCC(NC(Cc3ncc(C)s3)=O)C(F)C2)=O)ccc2oc(S)nc2c1 N1(C(CCC(C)=O)=O)CC(NC(C2CC2C2CCCC2)=O)Cc2ccccc21 C1(NC(C2CCN(C(C)=O)C2)=O)(CF)CCN(C(c2cncnc2)=O)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(C)(CNC(c2n[nH]c(C)c2F)=O)OCC1 C1(CNC(C2(C#C)CCCC2)=O)CC2COCC2N1C(c1ccco1)=O C1(CNC(C(C2CC2)SC)=O)CCC(NC(c2ccc(C3CC3)o2)=O)C1 c1(C(N2CCOC(C3CC3)C2)C(=O)NCCCF)cnn(C(C)C)c1F C1(C(N2CC(n3cc(CN(CC(C)(C)C)CC)nn3)C(C)C2)=O)CC(=O)NC(=O)N1 C(=O)(C(O)C(C)(C)CC)N1CC(NC(CC(CC)CNC(=O)OC(C)(C)C)=O)C1 N1(C(COCC)=O)CCC(N2CCN(C(c3csnc3Br)=O)CC2)CC1 N1(C(c2cc(OC)ns2)=O)CCC(C2CCN(C(c3ccnn3C)=O)C2)CC1 N1(C(=O)NCc2csc(N3CCCCC3)n2)CC(CC)OC1=O N1(C(CCOCC#C)=O)CC(CC(=O)NCC2(C)CC(C)(C)C2)CC1C c1(C(c2nnnn2-c2ccccc2)NCC(C)OC)cc(F)c(F)c(F)c1 c1(OCC)ccc(NC(=S)Nc2cnc(C(C)O)cn2)cc1OC(C)C c1(C(=O)NCC2CCN2C(=O)CC2(CSC)CCCC2)ccc(F)cc1Cl c1(C(c2nnnn2C2CCOC2)NCCCOC(=N)O)occc1Br c1(NC(C(CC)(C)O)=O)ccc(CNC(=O)C(C)(C)N2CCCC2)c(C)c1 N1(C(C2(SCC)CC2)=O)CCC(C(C)NC(=O)Cc2cc(-c3cccs3)on2)C1 c12ccc3c(c1)C(=O)N(C3=O)COC21CCCC1.COCC C1(NC(C(C=C)OC)=O)CN(C(=O)Cc2cccc(OC(F)F)n2)CC12CC2 N1(C(CN(C)C)=O)CCCCC(NC(=O)COc2ccccc2C(N)=O)CC1 Cc1cc2c(CC(=O)NC3CCNCC3c3ccccc3)csc2s1 c1(C(=O)NC2CC(CCCN(C(=O)C(F)C3CCCC3)C)C2)ccc(C#N)cc1 Nc1c(C(=O)NCC2(NC(C3CC4(CCC4)CO3)=O)CCCCC2)cccc1F N1(C(c2n(C(C)C)ncn2)=O)CCCC1(C)CNC(c1sccc1CC#N)=O c1(-n2cc(CCC3N(C(CCS(C)=O)=O)CCC3)nn2)ccc(Cl)cc1Cl C12(CNC(C(CC)C(C)C)=O)CCC(CNC(=O)CC34CCCC3C4)(CC1)CO2 c1(C2N(C(=O)Cc3n[nH]cc3Br)CCC2)nnc2n1CCC2 Cc1cc(C(N2CC(CNC(=O)CN3C(=O)CNC3=O)C3CC23)=O)cn(C)c1=O CC(C)CC(C)(CO)NC(=O)COC1CN(C(C2CCCCCCC2)=O)C1 Cc1oc(-c2ccco2)nc1C(N1CCOC(CS(N)(=O)=O)C1)C(=O)NC1CC1 c1(C(=O)NCCN(C(c2cn(CCC)nc2C)=O)C)cnc(O)c2cccnc12 N1(C(c2cn(C)[nH]c2=N)=O)CCC(CO)(CNC(C2(Cl)CC23CCC3)=O)CC1 c1(OC)ccc(C(N2CCOC(C(C)Nc3cc(C(N)=O)ncn3)C2)=O)c(C)c1 C1(COC)(NC(=O)Cc2cccn2C)CN(C(=O)CCC2CCOC2)C1 C#CCCC(=O)NC(C1CC1C(=O)NC(c1nn[nH]n1)C1CC1)C N1(C(C2C(C(C)(C)C)CC2)=O)CCCC(C(=O)NCC2CCCC23CC3)CC1 C1(NC(C2C(C=C)OCC2)=O)CCN(C(=O)CC2CCC(OC)CC2)CC1CC C(=O)(C(O)CC1CCOCC1)NCCN(C(=O)C(O)CC1CCOCC1)C(C)C c1(C(N2C(CCOC)CN(C(=O)C=C(C)Cl)CC2)=O)cnn2cc(C)cnc12 O=C(N=c1ncnc2[nH][nH]cc1-2)C1CC12CCN(Cc1cccc(F)c1O)C2 C1(NC(c2c(OC)ncc(Cl)c2)=O)CN(C(=O)CSCCC#N)C2(CCC2)C1 N1(CC#N)CCC2(CCCCN(C(C3(C4CCCO4)CCCO3)=O)C2)C1 c1(C(=O)NCC(n2cc(Cc3nn[nH]n3)nn2)C)cccc(C2(F)CC2(F)F)c1 C(CC(O)C(=O)NCC(CC(C)C)NC(C1CC1C(=O)OC(C)(C)C)=O)SC c1(CCC(=O)OCC(c2c(OC)ccc(F)c2)=O)ccc2ncccc2c1 N1(C(=O)Cc2nc[nH]n2)CCN(C(c2ccc(OC(F)F)c(F)c2)=O)C(C2CC2)C1 N1(C(CCN(C)CC)=O)CC2CCC2(CC(N2Cc3ncsc3C2)=O)C1 N#Cc1cccc(S(=O)(=O)Nc2cc(C(N3CCC(O)(CF)CC3)=O)n(C)c2)c1 CC1CN(C(=O)C(C2CC2)N(C(=O)Cc2ccccn2)C)CCS1=O C1(C(=O)NCC(CNC(c2cnn(CCN(C)C)c2)=O)OC)CCCCO1 c1(N2CCC(NC(C3CN(C)C3)=O)C(F)C2)nc2ccc(O)cc2s1 Cc1cc(C(N2CC(F)(CNC(=O)C(N3C(=O)CCC3=O)C)C2)=O)cc(N)c1 N1(C(c2nc(C(C)C)oc2)=O)CC2CC1C2NC(=O)COc1ccsc1Cl c1(C(C(N2C(CNC(C(C)(C)OC)=O)C=CC2)=O)C)ccc(C(C)(C)C)cc1 CCC(C)(C(=O)NCCCNC(c1ccc(Oc2ccccn2)cc1)=O)OC c1(C(=O)NCC2(NC(C3C(C(C)(C)C)C3)=O)CCC2)ccc2nccn2c1 C(c1ccncn1)=CCc1csc(CNC(CCC(CC(C)(C)CO)(C)O)=O)n1 C1(CC(=O)NCC2C3CC2N(C(c2nocc2Br)=O)C3)CCS(=O)(=O)C1 C1(OCC)CN(C(=NCCN)NCC2CCCCN2C)CC1N(S(C)(=O)=O)C c1(OC)cc(O)ncc1C(=O)NCC(C)CNC(c1cccc(C2CCC2)c1)=O C12(C(=O)NCC3N(C(CCC(CC)CC)=O)CC(O)C3)CCCC(=O)N1CCC2 c1(SCC(=O)NC2(CCCNC(C3(CC)CC3)=O)CC2)ccc(O)cc1 N1(C(C(N2CCOCC2)C)=O)CCC(CNC(=O)Cc2cncn2C)(OC)C1 c1(OC)ncc(Br)c(C(N2CC3CC(C2)N3C(=O)CC2CCCC2O)=O)n1 C1(C(=O)NCC2(CC(=O)NCCCCC#C)CC2)CCCCC1O C(CC(=O)NCc1cccc(C)n1)(C(C)CC)NC(c1c(C#C)c[nH]n1)=O c1(SC)ccc(C(=O)NC2CC2NC(c2n[nH]cc2C(F)(F)F)=O)s1 N1(C(C(CCN(C)C)NC(=O)C#CC(C)(C)C)=O)Cc2cccc(O)c2C1 CCCC(CC(C)C)C(=O)N1CCC(C(=O)N(C2CCCC2)C)C(C)C1 C1(NC(c2sc(CC)c(C)c2)=O)CCN(C(=O)COCC2CCCCO2)C1(C)C c1(C(N2CCN(C(CC=C(C)C)=O)CC2CF)=O)[nH]c2ccc(C)cc2c1Cl c1(CN2CC(NC(c3ccc(O)c(O)c3O)=O)C(F)(F)C2)cc(F)c(Cl)c(Cl)c1 N1(C(C=CC(C)C)=O)CC(NC(c2ccc3nn(C)cc3c2)=O)CC12CCCC2 c1(NCCOCCN(C)C(C2CCC3CC3C2)=O)ncnc2c1nnn2C1CC1 C1(C(C)C)CCc2[nH]nc(C(=O)NC(=O)C3CC3)c2C1.C12CN(CCN1C)C2=O CN1C(=O)CCC1CNC(c1cc(C2CCCC2)nn1C)=O c1(NCC(=O)NCC2CCC(N(C(C(CCC)O)=O)C)CC2)c(C)cccc1Cl C1(C(N(CC(CC)C)C)=O)CCN(C(C2CCCOCC2)=O)CC1 c1(OC)ccnc(C(=O)NC2CCCCN(C(C3CC4(C3)CC4F)=O)C2)c1OC C1(OC)CN(C(C2NC(=O)OC2C)=O)CCC1NC(c1sccc1C1CC1)=O C1(CNC(C2CC(N(C)C)C2)=O)CCC(NC(=O)C(O)CC2CC2)CC1 O=C(C1=CCCOCC1)NC12CCCC1N(C(c1cnns1)=O)CC2 O=C1CCN(C(c2cccc3ncnn23)=O)C2CCCCC12 C1(OC)CC(CC(=O)NC(C(=O)NCCC(=O)NC(C)(C)C)C2CC2)C1 c1(C(N2C(CNC(CC3(C)CC3)=O)COC(C)(C)C2)=O)cc([N+](=O)[O-])ccc1N N1(C(c2ccc(C(C)C)o2)=O)CCCC(O)(CNC(c2nnn3c2CCC3)=O)C1 c1(C(=O)NC2C(NC(C(c3ccccc3O)OC)=O)CCC2)ccc([N+](=O)[O-])[nH]1 C1(NC(=O)Nc2ccnc3c2CNCC3)CCc2nnc(-c3ccccc3)n2C1 C(=O)(C1=NOC2COCC12)NC(CCNC(C=CC)=O)C(C)C C(=O)(C#CC1CCOC1)N1CCC(C(=O)Nc2cccc(F)c2)OCC1 C1(NC(c2n(CC)ccn2)=O)(CO)CCN(C(=O)C(c2ccccc2Cl)O)C1 CC(CC(=O)NCC12CCC(CC1)O2)C(C)(C)NC(=O)C1=NOCC1 CC1CCC(CC(=O)NC2CCCC2CC(=O)Nc2ccc(N(C)C)cc2)OC1 c1(C(=O)NC2CC(C)(CNC(C3(C(=O)NC)CC3)=O)C2)c[nH]c2c(Cl)cccc12 CCC(CCC(=O)NCCOc1ccncc1)NC(=O)C(C)CC(F)F C1(CC)CNC(=O)CN1C(=O)C(CC(C)C)NC(=O)CC1CCCSC1 CC1=C(C)CN(C(=O)CC2CC3(C2)CN(C(c2ccoc2Cl)=O)C3)CC1 c1(C(=O)Nc2c(C(C)(C)C)cccc2)ccc2c(=O)c(C(C)(C)C)c[nH]c2c1 CS(=O)(=O)c1ccc(Br)cc1CC(=O)OCC(=O)N(c1ccccc1)C1CCC1 C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC=CCNC(C(C)C(F)(F)F)=O Cc1nc(C2CC2)ncc1C(=O)NC1CCN(C(C2(C3CC3)CC2)=O)CC1O C1(CC(=O)NCCN(CCC)C(C2CCCCCC2)=O)CCC(F)(F)CC1 C(=O)(CCCCC(=O)NC1CC(CO)N(C(=O)CCNS(C)(=O)=O)C1)NC c1(OC)cccc(Cl)c1C(N1CCN(CCN(C(=O)C(C)CC(C)C)C)CC1)=O c1(C(=O)NCC(CC=C)NC(c2c[nH]cc(C)c2=O)=O)c(F)ccc(C#N)c1F C1(NC(CCCN(C)C)=O)CC(NC(C2OCCC2C(F)(F)F)=O)C(O)C1 c1(C(=O)NCC2(CNC(C(c3c(C)noc3C)C)=O)CC2)nn(C)cc1[N+](=O)[O-] C1(C(C)C)CN(C(=O)C(=O)C(C)(C)C)CCCN1C(c1ccnc(N(C)C)c1)=O N#Cc1cc(C(=O)NCC=CCC(=O)Nc2cccc(CCO)c2)co1 C1(C(=O)NC2CC(OCC(=O)NCc3ccc(F)c(O)c3)C2)CCCC12CCC2 C1(NC(C2(C=C)CCOCC2)=O)CCN(C(=O)CC2CCCN(C)C2)CC(O)C1 CCCC(C(=O)NC1CCOCC1NC(C1(C(C)C)CC1)=O)C(C)C C1(OC)CC(NC(=O)C=C(Cl)Cl)CN(C(c2nn(C)cc2Cl)=O)C1 c1(CSC)ccc(C(=O)NCCCCNC(C2(n3cncn3)CC2)=O)cc1 N1(C(C(COCC)N=[N+]=[N-])=O)Cc2n[nH]cc2C1C(=O)NCC=CCOC C1(CNC(c2c(COC)cc[nH]2)=O)CCCN(C(c2c(Cl)cnn2C)=O)C1 CN1CCn2nc(C(=O)N(CCc3nn[nH]n3)CC3CNC3)cc2C1 N1(C(C2C(NC(c3cnn[nH]3)=O)C3CCC2C3)=O)CCC(C2CCC2)C1 c1(C(N2CC3CC(NC(C4(CCF)CCC4)=O)CC3C2)=O)ccn2cncc2c1 CC1=NC=COCCN2N=NN=C3C=CC(OC(F)F)=CC=C1CCC2NC3 Cc1cc(CC(N2CCN(C(=O)CC3(O)CCCN(C)C3)C(C)C2)=O)ccc1Br c1(C(=O)NCC2C(CNC(c3ncn(CC)c3)=O)C2)cccc(N2CC=CC2)c1 C(=O)(C(C)(C)C(=O)N1CC(NC(=O)CC(C)NC(C2CCCC2)=O)CC(F)C1)NC N1(C(C(C)CSc2ccccc2)=O)CCCC(CO)(NC(=O)C2=CSCCO2)C1 C1(C)(CC)CC(NC(C2CC=CC(NC(=O)CCC3CC3(C)C)C2)=O)CCO1 C1(N(C(C(CCC)N(C)C)=O)CC)CCCN(C(c2nn(C)cc2C)=O)CC1 c1(OC)ccc(C=CC(=O)NCC(O)CNC(=O)C(C(C)C)NC(C)=O)c(C)c1 c1(N2C(C)CC(F)C2)ccc(S(=O)(=O)NCCN2CCOCC2)cc1Cl Cn1ncc(C(N2CC(NC(=O)C3=CCCC3)CC(C)(C)C2)=O)c1S(C)(=O)=O C(=O)(C(F)(F)C(F)(F)F)N(CC(C)(C)NC(c1cc(C)[nH]c1C)=O)C CC(C(=O)N1CC2(CC(NC(C3(OCCNC)CCOCC3)=O)C2)C1)C(C)(C)C c1(C(C(=O)NC(C2CCCN2C(=O)Cc2cocn2)C)(C)C)ccc(Cl)cc1 N1(C(CNS(C)(=O)=O)=O)CCC(C)(C)C(NC(C2(O)CCSCC2)=O)C1 c1(C(=O)NC2CCCC(NC(c3cc(C)c(C)[nH]3)=O)C2)cnc2nccn2c1 Cc1nn2c(c1C(N1CC(NC(c3nccn3C)=O)CC1C)=O)NCCC2 C(=O)(CC1=CCCC1)NCC1C(C)CCN1C(=O)CCOC1CC1 c1(CN2CC(CC(=O)Nc3cccnc3F)OCC2)ccc2c(Cl)ccnc2c1 C1(NC(Cc2cc(C)n(C)n2)=O)CCN(C(c2nnn(C)c2C(F)F)=O)C12CC2 C1(C(=O)NC(C2CCCC2)CNC(c2ncnc(O)c2F)=O)CC12CCSCC2 C1(C(=O)NCCCN(C(CC2C(C)(C)COC2)=O)CCO)CC12CCOCC2 C1(NC(=O)CC2CCOC2)CCN(C(=O)CNC(C2CCC2)=O)CC1CO c1(C(=O)NC(CC2CCN(CC(CC)OC)CC2)C)cnc(C2CC2)nc1C N1(CCC(CC)(C)C)CCC(=O)N(Cc2ccc(CC(N)=O)cc2)C1=O CCCC(C(=O)NCC(C)(C)C1CC1)N1CCNC(=O)C1 N1(C(C2C(NC(C(C)OCOC)=O)COCC2)=O)CCn2ccnc2C1 C#CC1CCN(C(=O)C(CC)NC(c2c[nH]c(C(N)=O)c2)=O)C1 c1(NC(C2CCCC(NC(c3scc(C)c3C)=O)C2)=O)c(F)c(F)cc(F)c1F S(=O)(=O)(c1ccccc1[N+](=O)[O-])NCCCNC(=O)C(=O)NC1CCCC12CC2 c1(N2CCN(c3ccnc(C(C)C)n3)CC2)ccc2c3c(cccc13)CC2 C#Cc1ccc(C(=O)NCC2CC2CNC(=O)Cn2cc(Br)c(C)n2)c(C)c1 CCC(C)C(=O)C(=O)NCC1CC2(CC(NC(=O)CC3CC=CCC3)C2)C1 N1(C(C2(CCC)CCC2)=O)C(C(=O)NCCNC(C2CCCS2)=O)CCC12CC2 C1(NC(C23CC(NC(C(CC)OC)=O)(C2)C3)=O)CCCC(C(C)(C)C)C1 N(C(=NCCCCl)N1CCC(C(=O)NC(c2c(CSC)ccs2)=O)C1)C(C)C N1(C(CCC)=O)CCCCC1C(N1CCC(N(C(c2ccncc2)=O)CC)C1)=O C(=O)(CC1OCc2ccccc21)N1CCC(CCNC(CC(C)O)=O)C1 N1(CC(=O)NC(C)CCN(C(=O)C(F)=CC2CC2)C)CC(=O)Nc2ccccc21 N1(C(C2CCCC23CCC3)=O)CC(C2CC2)(C(N2CCOC3CC23)=O)C1 C1(NC(CC(C2CC2)SC(C)C)=O)CCCCC1NC(C1C(C(N)=O)C1)=O c1(C(=O)NCC2(NC(C(C(C)C)NC(COC)=O)=O)CC2)c(O)nnc(C)c1C C(=O)(C1=CCCCC1)N1C(CC=C)(C(=O)OC)CCC1.C(=O)CCCn1ccnc1 C1(c2cn(CCc3cn(C)nn3)nn2)CCC(N)CC1 CC1CCC(CO)(NC(=O)CCN(C)C(c2cccc(CC#N)c2)=O)C1 N1(C(COCCC)=O)CC2CCN(C(=O)Cc3csc(S)n3)CC2C1 C1(C(N(C2CCCC2)CCC=C)=O)Cc2c(F)ccc(F)c2CN1 Cc1oc(C(N2CCC(CNC(=O)C(O)Cn3cncn3)C2)=O)cc1Br Cc1cc(C#N)nc(N(C2CCNCC2F)C(c2ccc3c(c2)CCO3)=O)n1 N1(c2cc(N(CC)Cc3ccccc3Cl)ncn2)CC2CC(C1)C2C(=O)O c1(-c2cn(CC(=O)NCC(CC)(C)CO)nn2)ccc(C)c(F)c1 CC1=C(C(=O)N2CCC(CC(=O)N(C(C)C)Cc3cnccn3)C2(C)C)CCO1 N1(C(c2cc(C)nc(O)c2)=O)CCC2CN(C(c3cc4sccc4cn3)=O)C2C1 c1(C(=O)NC2CC(C)(CNC(C3CC4CC4C3)=O)C2)cccc2[nH]ncc12 N1(C(C2(CC)CCCC2)=O)CC(N(C(=O)Cc2n[nH]cc2Br)C)C(O)C1 C1(CC=C)(C(=O)NCC(=O)OC)CCN(C(=O)CCCOCCC)C1 c1(CC)nn(C)c(C(N2CCC2CNC(=O)CC2CCC3(CCC3)O2)=O)c1Cl N1(C(C(=O)NCCOC)C(C2CCC2)OCC)CCC2OCCCC2C1 N1(C(C(C)n2ccnc2)=O)CCC2(NC(=O)Cc3ccc(O)nc3)CCCC12 Cc1ccc(Cl)cc1NC(=O)C(C1CCN(C(C2C(C)(C)C2(F)F)=O)C1)F C1(NC(CC=C)=O)CCC2(CC1)CC2NC(=O)CC(CN(C)C)CC c1(C(N(C(CNC(c2nnc(C)s2)=O)C)C)=O)ccc(=O)n2c1CCCCC2 N1(C(c2sccc2I)C(=O)NC(CC)(C)C)CC(=O)NC(C(C)C)C1 c1(N2CCC(NC(c3cc(SC)c(F)cc3)=O)C(O)C2)ncc2c(n1)COC2 c1(N(C)CC2N(C(C(C)OCCN(C)C)=O)CCC2)nccc(S(C)(=O)=O)n1 c1(C(N(CCCCNC(C(C)NC(C)=O)=O)C)=O)c(Cl)cc(C#N)cc1Cl Cc1oc(C(=O)NC(CCN(C)C)C(=O)NC2CCN(C(C)(C)C)C2)cc1CO CCS(=O)(=O)CC(=O)NC1CCCC1CN(C)C(c1ncnc(C)c1C)=O C(=O)(C(C)CS(C)(=O)=O)N1CC2(N(C(COCCCCCCOC)=O)CC2)C1 C1(CC(N2CC(C)(NC(=O)CC3CCCC(C#N)C3)C2)=O)CC2CCC1C21CC1 Cc1c(C(=O)NCCC2(O)CN(C(C3(C)CC=CCC3)=O)C2)[nH]c2ccccc12 N1(CC(=O)NCCSCCCl)C2CCCC1CC(=O)NC2.CC(C)(C)S C1(C(=O)Nc2cnc(-c3ccccc3)s2)CCS(=O)(=O)CC1.C12CCN(CC1)C2 C12(C(=O)Nc3cc(SC)n[nH]3)CC1CN(C(c1ncoc1C)=O)C2 Cc1c(Cl)ccnc1C(=O)NCCC1CCCN(C(=O)COCP(C)(C)=O)CC1 C1(CNC(CC2CCC2)=O)CC(O)C(O)C1.C12CCOC1CNC2=O.CCOC C(CCC(=O)NC(C)CNC(=O)C(C)(C)C1CC1)NC(=O)OC CC1CN2CCN1CC2C(=O)NC1CCCCC1CNC(C12CCCC1C2)=O C1(OC)CC2(C1)CC(C(C(=O)NC1COC1)N(C)Cc1nccn1C)C2 N1(C(C2(CC#C)CCC2)=O)CCC(C(O)CNC(=O)CSC(C)(C)C)CC1 c1(C(=O)NCC2(OC)CN(C(C3CCC(F)C3)=O)C2)cnn2c1CCC2 C1(C(N2C(CCC)COCC2)=O)CC(C)(C)CCN1C(C1CC(=O)CCO1)=O c1(C(=O)NC(C)CF)ccnc(CNC(C2CCCC(F)C2)=O)c1 c1(C(=O)NCCC2CCCN2C(=O)CCc2ncc[nH]2)cc2n(n1)CC(F)C2 N1(C(C(C2CCC2)OC)=O)CCN(C(=O)CCc2conc2C)CCC1C c1(CNC(=NCCOCC=C)NCCC(O)C(C)(C)C)c(C)cc(C)cc1C Cc1cccc2ccc(C(=O)NC3CCC(NC(=O)C(C)O)C3)nc12 Cc1cccc(N)c1C(=O)NC1CCCC(NC(=O)C=C(Cl)Cl)CC1 CCCCC(CCC)NC(=O)C(=O)Nc1cccc(COC)c1 C1(CNC(C(CSC)(C)C)=O)CN(C(=O)CC(F)(F)F)CCC1C c1(N(CCCF)C)nc2c(c(=NCC3(CO)CCCO3)[nH]1)CCC2 Cc1cnc(C(=O)NCC2CN(C(C3CC34CCSCC4)=O)CC2(C)C)cc1Cl c1(OC)ccc(C=CC(=O)NC2CN(C(c3nocc3C)=O)CC2C)c(C)c1 c1(C(=O)OC)ccc(C(CO)N(c2cncc(C(F)(F)F)n2)CCO)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C2C(CNC(C(C(C)C)O)=O)CC(CC2)C1 c1(NC(C2(CC)CN(C(c3cc(O)ccc3C)=O)C2)=O)cnc2ncnn2c1 N1(C(Cc2c(C)cccc2C)=O)CCC2CN(C(c3ccnnc3S)=O)C2C1 N1(C(C(CC=C)C)=O)CCN(C(c2cc(C)c(C)o2)=O)C(C2CC2)C1 C1(CNC(C2(OC)CCC2)=O)CCC(C)(C)CN1C(c1ccncc1)=O c1(NCC2(C)CCCN(C(CC(CN(C)C)O)=O)C2)ncc2c(n1)CCCCC2 C1(NC(C2CC23CCC3)=O)CCCCCN(C(=O)C(F)(F)c2nccs2)C1 Cc1cc(C(F)(F)CNCC2(N)CCOC2)cnc1Cl C=CCC(CC)C(=O)NCCOC(C)(C)CNC(=O)C(C1CCC(C)(C)CC1)C C12(C(C=Cc3cc(C(=O)OC)c(OC)cc3)=O)CCC(C#N)(CC1)CC2 CC(C)C(C(C)NC(=O)COC1CCCCCC1)NC(=O)CCc1cnc[nH]1 c1(C(=O)NC(C)CNC(=O)CC2CCC(=O)N2)cc(=O)n(C)o1 c1(C(=O)NCC(CCNC(c2ccc(C(C)=O)[nH]2)=O)O)ccc(C(C)C)nc1O C(=O)(CC(O)C(C)(C)C)N1CCN(C(C(C(C)C)NC(=O)OC(C)(C)C)=O)CC1C C=CC(CCC)CC(=O)NCC1CCC1NC(c1cc(C#N)c[nH]1)=O C(=O)(C(F)(F)C1=CCOCC1)N1CCC(CCN(C)C(c2ccsn2)=O)CC1 N1(C(CC(CCC)O)=O)CCN(C(=O)CSc2cccs2)C2COCC12 C12(NC(C=CCCC)=O)CC(CNC(=O)C(N3CCN(C)CC3)C)(C1)OC2(C)C c1(C(N(C(c2ccccc2)C(=O)OC)C)=O)ccc(OC(C)C)cc1OC N1(C(C(F)=CCC)=O)CC(OC)CC1(C)CNC(=O)CSc1n[nH]c(C)n1 C1(C(=O)NCCN(C(C)C)C(c2cnn(-c3ccncc3)c2)=O)CCCN(C)C1 c1(C(C(=O)NC(C)CC)N(CCCOC)C)sc(C(=O)OC)cc1C Cc1cccc(OCC(=O)NCC2C3CN(CC4CCCCO4)CC23)c1C c1(SCC(N2CC(C(C)NC(=O)CCn3cccc3)C2)=O)ccncc1 C=CC(CC)CC(=O)NC1CN(C(c2cc(C(F)(F)F)cnc2N)=O)C(C)(C)C1 Cc1cc(CC(=O)NC(C)CC(C)NC(c2cnsn2)=O)ccc1CO CCCCC(C)C(=O)NCc1cccc(CN(C(=O)C=C(C)C(F)F)C)c1 N1(C(C(C)N2CCC2)=O)CC(C(C)(C)O)(CNC(C2CC2(C)Br)=O)C1 CCC(C)(C)C(C)NC(=O)C(C)(C1CCC1)NC(=O)Cn1ccnc1 c1(C(=O)NCC2(CNC(C(CSC)O)=O)CC2(F)F)cc2c(F)ccc(F)c2[nH]1 C(=O)(CC1=CCCCC1)NCCC(=C)CNC(=O)C(F)(F)c1ccnn1C C12(NC(CC(=O)OC)=O)CCN(C(=O)CSc3ccc(C)cc3)CC1C2 N1(C(c2c(Cl)cc(C)s2)=O)CCC(C)C(NC(C2CC3CCC2CC3)=O)C1 C1(CNC(c2cnc(CCCC)s2)=O)CCCC2(CN(c3ncc(O)cn3)C2)O1 S(=O)(=O)(c1ccc(NCc2csc(CO)n2)c(F)c1)NCC1C(C)OCC1 N1(c2n(C(C)C)nnn2)C(C)CCCC1C.C(=O)CCN=[N+]=[N-] C#CCCCCCCCNC(=O)C1=CCC(NC(=O)C(C)=CC=C)C1 C=CC1(C(=O)N(CC(C)(C)COC)C)CCN(C(=O)C(C)CC(=O)OCC)CC1 N1(C(c2c(OC)nsc2)=O)CC2CC(C(=O)NC(C)(C)CNC(N)=O)C(C2)C1 C1(NC(=O)Nc2ccc(OC)cc2)CC2(C1)CC(Nc1nccnc1C#N)C2 CC(C)CCCCCC(=O)N1CCC(C)C1C(=O)NCCN1CCOCC1 C1(C)(CNC(CC2CC(OCC)C2)=O)CN(C(c2cnc(C)c(N)c2)=O)CCO1 C1(C(N(C2CCN(C)CC2)C)=O)CCC(O)CN1C(c1nnc(S)n1C)=O C=CC(C)(C)CC(=O)NC(C)CCN(C(=O)C(O)C1CCCC1)C O=C(CC1=CCCCC1)NCC1CCCC(NC(=O)CCCc2cnccn2)C1 C1(CNC(c2cnn(-c3nccs3)c2)=O)CC(F)CN1C(=O)CO CN1CCC(C(N2CCCC(CCCO)C2)=O)(NC(c2scnc2C(F)F)=O)C1 C1(NC(c2ccc(C)c(C)c2)c2nnnn2C(C)C)CC2(CCCOC2)C1 N1(C(C(COC)OC)=O)CC=CC(NC(C2(CC3CC3)CCC2)=O)C1 N1(CCCc2ccccc2Sc2ccc(Cl)cc2)CCOC2(CCCC2)C1 C1(CSC)CCCCN1C(C1CC1C(C)NC(c1cn(C(C)C)nc1C)=O)=O c1(CCN(C2CCN(C(=O)CC3COCCO3)C2)C)c[nH]c2ccccc12 Cc1cncc2nc(CC(=O)NCC3(C4=CCOCC4)CC3)cn12 CC1(C)CCC1C(=O)NCC1(NC(C2(c3ccccc3)CC2)=O)CCC1 CN=c1ccc(Br)c(C(=O)NC(C)CN(C(=O)CCC=CC(C)C)CC)[nH]1 c1(C(N2CC(CC(N3CCC(CO)C3)=O)C2)=O)c(OC)cccc1CC C(=O)(CC(C(=O)N1CCC(C2CCCN2C(c2ccns2)=O)CC1)N(C)C)OC N1(C(CCC2(NC(CCCC)=O)CCC2)=O)CCN2CCCC2C1 C1(OC)CC(NC(C2(C3CCC3)CC2)=O)CN(C(=O)COC2CCCC2)C1 C=CCC(CC)C(=O)N1C(CC(N2CC(C)CCC2CC)=O)C2CCCC12 Cc1ccc2c(C)c(C(=O)NCC34CC3CN(C(=O)CCC3CC3)C4)[nH]c2c1 c1(CN=C(NCC2(CC)CCC(=O)N2)NCCSCC)ccc2c(c1)oc(=O)n2C C1(C(N2CC(CNC(=O)Cc3ccno3)C2)=O)CC12C(=O)Nc1ccccc12 C(=O)(C(CO)C(F)(F)F)NCC(=O)NCc1nccc(OC)c1 C(=O)(CC(c1ccccc1)Nc1ccc(SC(=O)OC)o1)OCC C(=O)(C(C(=O)OCC)C(C)C)NCC1(F)CN(C(CSCC(=O)NCCOC)=O)C1 C1(NC(C2(C)CC(N(C)C(c3cc(C(N)=O)co3)=O)C2)=O)CCN(C)C1=O C(CC(C)(C)C(=O)N1CCCOC(CNC(c2cc(C)sn2)=O)C1)OC c1(CC(=O)NC(CN(C(C2C(OC)CCC2)=O)C)C)ccc(Cl)cc1 C(C1=CCN(C(C2(C)CCCC2)=O)CC1)NC(C(CC)Oc1ccccc1)=O C(CCCC(=O)N1CCC1C(C)C)N(C(C(C)(C)OC(C)=O)=O)C C1(C(N(C(C)C)CCN(C)C(C2CCC(F)C2)=O)=O)CCn2ncnc2C1 C1(CC#C)(C(=O)NCCCCCNC(c2cnc(COC)[nH]2)=O)CC=CCC1 N1(C(C(=O)NCCOC)=O)CCC12CN(C(c1ccc(C(C)=O)nn1)=O)C2 C1(NC(c2c(C)cno2)=O)CCCC(NC(c2c(Br)n[nH]c2C)=O)C1 C1(C#CC(=O)NC2COCCN(C(=O)CC(C)C3CC3)C2)(CC)COC1 c1(C(N2C(CC)C(NC(c3csc(C)c3)=O)CC2)=O)csc2ccccc12 C1(C2CCOCC2)(C(N(C)CCN(C(=O)C(C)(C)C(N)=O)C)=O)CCOCC1 N1(N(C(=O)Cn2cccn2)CCC2(C(F)(F)F)CC2)CC(C=O)CC1=O.C C1(CC)CCCN2C1C(=O)NC(C(C)OC)C2=O.C1(C)CCCN1C(C)=O Cc1cccc(C(=O)NC(C2CN(C(c3cc(Cl)ccn3)=O)C2)C)c1[N+](=O)[O-] C1(NC(C(COC)(C)C)=O)CC12CCN(C(C1CC(CF)C1)=O)CC2 N1(S(c2c(CC(=O)OC)cccc2)(=O)=O)CCS(=O)(=O)N2CCOCC12 CC1(C(N2CC=CC(NC(=O)Cc3ccsn3)C2)=O)CCC2(CC1)OCCO2 C12(C(=O)NCC#CCNC(c3nc(C)n(C)c3)=O)CC(CO)(C1)OC21CCC1 c1(CNC2C(C(=O)Nc3nc(C)c(Cl)s3)C2)ccc2cc[nH]c2c1 CCCCCCCCCCOc1c(Cl)cc(C(=O)OC)cc1Br C1(CN(C(=O)CCC2CCCCO2)C)COCCN1C(=O)Cn1cnnn1 C1(O)(CCC)CCN(C(c2c(CNC(=O)C(C)NC(C)=O)nnn2C)=O)CC1 N1(CC)N=C(C(=O)NCC(O)CCNC(=O)CC2CSCCS2)CCC1=O Cc1nc(NC(c2sc(Br)nc2C)=O)sc1C(N1CC2C(CO)C2C1)=O C1(NC(N)=O)CCN(C(=NCC2CCCN(CC(F)F)C2)NC2CCC2)C1 c1(C(N2CCC(NC(C(C)SCCCC)=O)C2)=O)cccc(C)c1[N+](=O)[O-] N1(C(C2(COC)CC2)=O)CC2CCC1C(CNC(=O)C(O)CC(C)C)C2 CC1CCN(C(c2nncn2C2CC2)=O)CC1NC(=O)CSCCC(F)(F)F c1(SC)cc(C(=O)NCC2CN(C(=O)CCC3CC3(C)C)CCO2)c(C)o1 N=c1nnn(CC(=O)NC2CC(CNC(c3ccsc3Br)=O)C2)[nH]1 CC12CN(C(c3ccc(OC(F)F)cn3)=O)CC1CN(C(C1CCCCS1)=O)C2 C1(CNC(C(C=C)O)=O)CN(C(C2CSC2)=O)CCN1C c1(N(CCCCCNC(C2C(C(=O)OC(C)(C)C)CCO2)=O)C)c[nH]ccc1=N CCC(CC(=O)NC1CC=C(C(=O)NCCCCS(C)=O)C1)C(C)C c1(C(=O)NC2CCCN(c3nnc(C)o3)C2)ccc(O)nc1C N1(C(C23N(C(C#CC)=O)CC(CO)(C2)C3)=O)C2CCC1CC(OCC)C2 C(c1ccc(F)cc1)=CC(=O)NC1CC(CNC(C(COC)C)=O)C(O)C1 N#Cc1cc(N(CCNC(c2csc(Cl)c2Cl)=O)C2CC2)nc(C2CC2)n1 Cc1cc(C)c(S(=O)(=O)N2CCC(N(C)Cn3nc(C)cc3C)C2)c(C)c1 Nc1ccc([N+](=O)[O-])c(C(N2CCN(C(=O)Cc3cocn3)C3(CC3)C2)=O)c1 C1(C(=O)NCCN(C(=O)C=C2CCCC2)CCC)CCCN(c2nccn2C)C1 CC(C)CC(CC(=O)NCC1(NC(=O)CC2(C)CCC2)CCCC1)CC(N)=O Cc1ccnc(-n2cc(C3(F)CN(C(C4CC5(C4)CC5F)=O)C3)nn2)n1 C1(NC(C2CC(=C)C2)=O)CCCCC12CCN(C(C1CCCN1C(C)=O)=O)CC2 c1(C(N2C(C)CC3CNCC23)C(=O)NC(C(=O)OC)C)ccc2ncccc2c1 c1(C(N2C(C)CCC(NC(c3c(C)cncc3)=O)C2)=O)cc(C)cc2c1CCC2 Cn1ncc(C(=O)NC2CC(F)(CNC(c3ccc(C(F)F)cn3)=O)C2)c1F C(=O)(CS(=O)(=O)C1CC1)N1C(C(C)C)C(NC(c2cc(F)cnc2O)=O)CC1 c1(C2C(C(N(C(C(=O)N3CC(COCC)C3)C3CCC3)C)=O)C2)ccccc1F N1(C(C)=O)CC(F)(F)CC1C(=O)N(CCc1ccccc1)Cc1ccccc1C C(=O)(C1CCCc2nn(C)cc21)NCC1(O)CC(NC(c2n(CC)ccc2)=O)C1 CC(C(=O)NN1CCCCC1=O)NCC.c1(O)ccc(Cl)cc1 C(CCC(O)CO)NC(C=CCN(C(c1ccc(COC)s1)=O)C)=O n1(CC(=O)NCC(CCNC(CC(C)CN(C)C)=O)O)sc(=O)c2ccccc12 c1(C(N(CCCNC(c2c[nH]cc2-c2cnn(C)c2)=O)C)=O)ccc(N)cn1 Cc1ncc2n1CC(C(=O)NC(C)CC1(O)CCC1)CC2 N1(C(C2(C(C)(F)F)CC2)=O)CCCCC(NC(c2ccc(CO)cn2)=O)C1 c1(C(N(CCNC(c2cccc(OC)n2)=O)CC)=O)ccc2c(c1N)CCCC2 N1(C(CCC=C(C)C)=O)CCN(C(=O)C#CC(C)(C)C)C(C)C1 C1(C(=O)NC(C2(O)CN(C(=O)CCCn3cncn3)C2)CC)CCCCC1OC N1(Cc2c(C)scn2)CC2C(C(=O)Nc3n[nH]c(C)c3Cl)C2C1 c1(CC(=O)NCCCNC(=O)Cc2cn[nH]c2)c(F)cccc1F c1(C(N2CC(CC(=O)NCCOc3ccccn3)C2)=O)ccc(C(F)F)cc1F c1(C(N(C)CCC2CCN(C(c3cnc(Cl)cn3)=O)CC2)=O)cnc(O)nc1O Cc1cc(Br)c2nc(CNCc3cc(F)c(C#N)c(F)c3)ccc2c1 C(CNC(=O)Cc1cncc(C)c1)(CC(C)C)NC(C1CCC(OC)C1)=O C1(NC(c2ncccc2CO)=O)COC2(CCN(C(=O)C3=CCOCC3)CC2)C1 c1(OC)cc(C(=O)NCC(F)CNC(=O)C(C(C)O)N(C)C)cc(Cl)c1O N1(C(c2nc(CC)oc2C)=O)CC(OC)CC1(C)CNC(c1cc(C)cc(C)c1)=O C1(CNC(c2cnn(C(C)C)c2Cl)=O)(NC(C2CCC2)=O)CCCCC1C N1(CC(N2CC(O)(CN(C)C(c3n[nH]c4c3COC4)=O)C2)=O)CCS(=O)(=O)CC1 C(=O)CC(C)(O)CCC.N1(CCCC)CCC(NC(=O)CC)CC1 CCC(C)CCC(=O)NC1CCN(C(c2cc(Br)cn2CC)=O)C1C C1(OCC)CC2CN(C(=O)C(C(C)CC)NC(c3nscc3C)=O)CC12 Cc1cc(C(=O)NC2C3CN(C(c4nocc4Cl)=O)CC23)cn1C(C)C Cc1cc(Br)cnc1C(=O)N(C)CCN(C(=O)CC1OCCC1(C)C)C C1(CC(=O)NC(C2(NC(=O)CN3CCCC3)CCC2)C)COC(C)(C)C1 CCCCC(C)C(=O)NC1(COC)CCN(C(=O)C(C2CCCCC2)O)CC1 C=C(C)C(C)(O)C(=O)NC1CCCC1NC(c1ccn(C(C)C)n1)=O C(=O)(C1Cc2ccc(F)cc21)N1CCC(CNC(CCC(C)C)=O)C(C)C1 c1(OC)ccccc1C(=O)NCC(C(C)(C)C)NC(=O)CCc1cc(C)[nH]n1 c1(N(C(CC)(C)C)C(CCOC(C)C(C)CC)c2nn[nH]n2)nc(C)c(C)o1 N1(C(CCCCCCCSC)=O)CCN(C(=O)CSC)C2CCCCC12 C(=O)(CCN(C)CCNC(=O)CSC)NC(C#C)C1CC1 N1(C(c2cnc(OCC)nc2)=O)CCOCC(NC(=O)CC2CC(C)C2)C1 N1(C(C2CC(NC(c3c(C)cn(C)c3)=O)C2(C)C)=O)CCS(=O)CC1C c12ccc(cc1)C(c1ccccc1)Nc1cc-2cs1.c1(S(C)(=O)=O)ccccc1 c1(C(=O)NCc2cn(C3N(C(C=CC)=O)CCC3)nn2)ccc2cnc(C)n2c1 C12(OC)CCCC1N(C(=O)CC1CCOCC1NC(=O)OC(C)(C)C)CC2 C(=O)(C1=CNS(=O)(=O)N=C1C)N1C(C)CCC(CNC(CCCOCCC)=O)C1 c1(C(=O)NC(CN(C(=O)Cc2ccc(Cl)c(F)c2)CC)C)cc(N)ccc1C C(=O)(C(O)CC(F)(F)F)NC(C)CC1CN(C(C2CCCCN2C)=O)C1 N1(C(C(C)(C)c2ccno2)=O)CCCC(CNC(=O)CSc2ccccc2O)C1 c1(CC)ccc(C(=O)N(CCCCCNC(=O)Cc2cnccn2)C)c(F)c1 c1(C(=O)NCC(CNC(CCC(C)OC)=O)OC)ccnc(C)c1C C1(C(=O)NC2CCN(CCCNC(C(C)(C)C(F)F)=O)C2)CCOC2(CCC2)C1 N1(C(C2(C)CC2(F)F)=O)CCOC2(CCCN(C(=O)Cc3cnns3)C2)C1 CCC(C(=O)NCC1CCCN1C(C1CCC=CCCC1)=O)C(C)C N1(C(CCCCC(N)=O)=O)CCC(C2(NC(C3(F)CCCCC3)=O)CC2)CC1 Cc1ccc(O)c(C(=O)N(CC(C)C(=O)NCC2CC(C)(C)CO2)C)c1 c1(C(=O)NC2CC(NC(c3c(OC)c(Cl)ccc3)=O)C2)cc2ncn(C)c2cn1 c1(C(=O)NCC2C(C)CCN2C(c2cccc(N)n2)=O)cnc(O)n(C)c1=O CCCC(O)CC(=O)NC1CC(C)CN(C(=O)CCC(=O)c2cnn(C)c2)C1 c1(CC(=O)N(C(C(=O)N(C(C(C)SC)C)C)(C)C2CC2)C)ncccc1F C=C(C)CN=C(NCC(c1ccncc1)C)N1CCC(NC(=O)NC)C1 c1(C(C(=O)NC2CCN(C(c3nn[nH]c3Cl)=O)CC2)(F)F)cc(Cl)ccc1F c1(C(=O)NC(CCC)C2CC2)sccc1CNC(=O)CCc1ncnn1C c1(N(CCC(CC)O)C(=O)C(N2CCC(O)CC2)=O)ccc(C(=O)OC)cc1 CCC(C)CCC(=O)NC(C)(C(=O)N(CC(C1CC1)OC)C)C1CCC1 c1(CC(=O)N(C)CC2N(C(CN3C(C)CC3)=O)CCOC2)noc2ccccc12 C(=O)(C1CCCc2ncccc21)NCC(CNC(c1scc(C)c1C)=O)C C1(C#CC(=O)NCC2C3CCC(C3)N2C(=O)COCCOC)(CC)CC1 C1(C(C2(O)CCOCC2)C)NC(=O)N(CCc2nccs2)C1=O c1(CC(N2CCC(Sc3cc(C(=O)OC)c(O)cc3)C2)=O)cc(C)cc(C)c1C C(=O)(C(O)CC[S+](C)C)N1CCC(N(C(=O)COCC2CCC2)C)C1 C1(C(=O)NCC2=CCN(C(c3c(C)nco3)=O)CC2)CCC2C(CC1)C2(F)F Cc1cc(NCCC#CCN=[N+]=[N-])cc(C)c1S(N)(=O)=O c1(NC(C(C)NC2(C(=O)NC34CC(C)C3C4)CCCC2)=O)ccccc1Cl c1(C(c2n(CCCC)nnn2)NCc2cnn(CCF)c2)cnc(OC)c(F)c1 C1(n2c(COC)ncc2)CCN(C2CNC(C)C2)CC1 C1(COC)(CNC(=O)CCF)CN(C(C2(C)CCCO2)=O)C1 N1(C(=O)C2CC2)CCN(C2CCN(C(=O)C(=O)Nc3n(C)ccn3)CC2)CC1 S(=O)(=O)(c1cccc(N2CCCC(CC(F)(F)F)C2)n1)NCCC(=O)N(C)CC C1(CNc2n(C(CCC)C)ncc2)COCCN1Cc1ccccc1 C1(C)(CC(=O)N(CC#C)CC2CCCC2)CCN(C(=O)C(C)CN(C)C)C1 c1(C(=O)NCC23N(C(CCC)=O)CCC2CCCC3)cc2ccccc2c(O)n1 C(N=c1[nH]c(=NCCCCS(N)(=O)=O)[nH]c2c1SCC2)C1CCCC(CC)C1 C(=O)(N=c1ccn(CC2CC2)[nH]1)C1N(C(C=CC2C(C)C2(Cl)Cl)=O)CC(C)(C)C1 C1(CCCNC(C(C2CCC2)OC)=O)CN(C(=O)CC2CCCC(C)O2)CCO1 CCCC(O)C(=O)N1CC(CNC(C2CCCN(C(C)=O)C2)=O)C(C(F)(F)F)C1 Cc1cc(C(N2CCC(C)(NC(=O)Cn3ccnn3)C2)=O)ncc1Br C1(C(=O)NC(CC)CNC(c2ccnn2CC2CCC2)=O)CC2C=CC1C21CC1 C(CCC(=O)N(C)CC1(CSC)CN(C(=O)C=CC(=O)N(C)C)C1)OCC c1(C(C)C)cc(-c2nc(CN3CCC(CC(=O)N(C)C)CC3)cs2)ccc1F N1(C(c2c(CC)occ2)=O)CC2(C1)CN(C(c1cnn(C)c1Cl)=O)CCO2 c1(OC)cccc(C(=O)NC2(C3CN(C(C4NC(=O)CC4C)=O)C3)CC2)c1O C(Cc1cc[nH]n1)(C(=O)NCC(C)CC1CCC1)NC(C=CCC)=O CCCCCC(C)CC(=O)NC1CC(F)(CNC(c2cnc(C(C)(C)C)o2)=O)C1 N#Cc1cc(S(=O)(=O)N2CCC(F)(C(=O)O)C2)ccc1NC1CC1 N1(C(C2N(C(c3ncc(OC)nc3)=O)CC(O)C2)=O)CC2(CNC(=O)N2C)C1 Cc1cc(C)c(C(=O)NC2CCN(C(C3COC4(CCC4)C3)=O)CC2O)c(S)n1 c1(OC)cc(C(F)(F)C(=O)NC2CC(CNC(C3CCCO3)=O)C2)ccc1C C1(CNC(c2ccc(CC=C)s2)=O)CCCCN1C(=O)C(C)CC1CCCC1 C(C(C)(CC(C)C)NC(c1cnc2n1CCC2)=O)NC(c1c(C)sc(Cl)n1)=O Cc1c(C(=O)NC(CC2CC2)C(=O)NCC(c2ccsc2)C)nnn1C C(=O)(CCC(=O)N1CCCC(N(C(=O)CCCc2cc[nH]n2)C)C1)NCC c1(C(N2CC(NC(C(C)NC(=O)NC)=O)C(C)C2)=O)n[nH]c2cccc(OC)c12 C(C)(CC(=O)NCC1C2CC1N(C(=O)C=Cc1cc[nH]c1)C2)(C(F)F)N(C)C C(N=c1[nH]c(C(=O)Nc2ccnc(Br)c2F)cs1)c1cc(OC)ncc1 c1(C(=O)NCCC(C)NC(=O)Cc2nnc(O)s2)cc(Cl)cc(Cl)c1 C1(C(=O)OC)CCC(C(N2CCCC2CCNC(=O)C(C)SC(F)(F)F)=O)CC1 N1(C(C(N2CCOC2=O)C)=O)CC2CCC(C1)C2CNC(=O)C(C)C1CCCC1 N1(C(C2(C#N)CC3(CC3)C2)=O)CC2COCCC2(NC(=O)CC2CCCC2)C1 C1(C(=O)NCC(C)(C)CNC(=O)CCC(=O)N2CCC2)CCC(C(F)(F)F)N(C)C1 N#CC(C(=O)N1CCCC1C(=O)NCCCc1ccccc1)c1ccccc1 N1(CC(C2CCOCC2)OCC)C(=O)CN(CC(n2cc(Br)cn2)C2CC2)C1=O C1(c2n(CC=C)nnn2)(NCc2n[nH]c(C3CC3)n2)CC2CCCCC12 N1(N(c2n[nH]cc2I)C2CCN(C(C)=O)C2)CCC2(CCOC2=O)C1 N1(S(=O)(=O)c2cc(Br)c(Br)s2)CCc2cc(F)ccc2C1 C(=O)(CCC(C)NC(c1cnn(C)c1N)=O)NC(C)C(=O)NCC(F)F c1(CNC2(C(C)O)CCOCC2)[nH]nc2c1CNC2(C)C C(c1ccccc1)=CC(=O)NC(C)C(=O)N(C1CCN(C)C1=O)C C1(C(N2C(C(N3CC(F)C(F)C3)=O)C=CC2)=O)C2Sc3ccccc3C12 c1(C(N(CCNC(c2cnn(CCOC)c2)=O)CC)=O)cc(Cl)sc1Cl C(=O)(C1CC(=O)c2c(F)cccc21)NCC(CO)NC(C(CC)=CC)=O c1(C(=O)NCC2(NC(C3CC(=O)NC3)=O)CCOC2)ccc2nc[nH]c2c1F c1(CCC(=O)NCCN(C)C(C2CC2Cl)=O)ccc2ncsc2c1 C(=O)(C1=CCCOC1)NCC(c1ccccc1)NC(C12C(CN(C(C)=O)C1)C2)=O C1(C(N2CCN(C(CC(C)C)=O)C(C3CCC3)C2)=O)CN(S(=O)(=O)N(C)C)C1 Cc1c(C(=O)NCC2CCC(NC(c3occc3C(C)C)=O)C2)c(Cl)nn1C C(=O)(CCCC(=O)N(C)C)NCC=CCNC(CCC=CC(C)C)=O S(=O)(=O)(c1cc(Br)c(F)cc1F)N1C(C)(C(=O)Nc2c(Cl)ccc(OC)n2)CC1 c1(CC(N2CC(NC(C(CC=C)C)=O)C(CC)C2)=O)cc(Br)ccc1C N1(C(CCc2cn(C)nc2)=O)Cc2[nH]nc(NC(C3CCSCC3)=O)c2C1 c1(OCC(=O)NCC(C)(C)CNC(c2csc(O)n2)=O)ccc(F)nc1 c1(CC(=O)NCC2CCCC(NC(=O)CSC(F)(F)F)C2)cccnc1Cl CC(C)CC(C(=O)N(C(C)C(=O)NCC1CNC(=O)CO1)C1CC1)C(N)=O CC(C)(C(=O)NCC1(F)CC(NC(=O)CCc2cnco2)C1)n1cnnn1 C1(OC)CCCC(C(N2CC(CO)(NC(=O)Cc3conc3C)C2)=O)C1 c1(C(N2C(CNC(C(C)Cc3cnc[nH]3)=O)CC(F)C2)=O)c[nH]c2ncccc12 c1(NCC2CC(F)C23CCC3)ncnc2[nH]c(I)cc12 CCN=c1[nH]cc(C(=O)NCC(C2CC2)NC(c2cccc(C3CC3)c2Cl)=O)s1 c1(CN2C(C)CCC2C(=O)NC2CN(C)C2)ncn2ccccc12 c1(CCC(=O)NCCCCN(C(=O)CC2CC(O)C2(C)C)C)cccc(F)c1F C(=O)(C(O)CC(N)=O)NC(C1CN(C(=O)CCc2cncs2)CCO1)C c1(SCC)ccnc(NS(=O)(=O)CCCn2cnnn2)c1.C=O c1(CCC(N2CC(NC(C3C4CNC(=O)C34)=O)C2)=O)cc(Br)ccc1F C=CC1(CNC(=O)C(C2(O)CCC2)NC(C2CCC(=O)N2C)=O)CCOCC1 c1(NC(C(COCC)C)=O)ccc(O)c(C)c1C C(=O)(CCP(C)(C)=O)N(C1CCCCC1NC(=O)CCc1csc(=N)[nH]1)C c1(CC)ccc2c(c1)C(NC(C13CCCCC1NC(=O)C3)=O)C(=O)N2 C1(CNC(C2(NC(CCCOC(C)=O)=O)CCOCC2)=O)CC1C1CCCC1 c1(C(=O)NC2(CCNC(C(C)=Cc3ccsc3)=O)CC2)cc(C2CCCC2)on1 c1(C(N(CC(C)NC(c2cc(C(C)=O)cn2C)=O)C)=O)c[nH]cc(F)c1=O c1(C(N2CC3CC2CN3C(c2cnc(Cl)s2)=O)=O)cc2ncccn2n1 CC(C(=O)NCc1ccc(CNC(c2cnc(S)[nH]2)=O)c(F)c1)C(C)(C)C c1(CC)nn(C)c(OC)c1C(c1nnnn1C1COC1)NCC1CCSC1 Cc1cn2cc(C(N3CCCC(NC(C4CC(C)C4)=O)CCC3)=O)cc(C)c2n1 c1(C(N2CCC(NC(CCC=C)=O)CC2C2CC2)=O)ccnc2c1cnn2C Cc1cc(C(N2CCC(O)(CCNC(c3ccco3)=O)CC2)=O)c(Cl)cc1F C(N=c1cc[nH]cc1S(=O)(=O)NCC1CC12CCOC2)c1c(OC)cccc1F c1(COCCSCC(=O)NCC(CNC(C2(C)CCC2)=O)O)ccccc1 Cc1cc(NC(=O)CCC2CCCN2C(=O)Cc2ccccn2)cc(C)c1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC2CN(C(=O)Cn3cc(OC4CC4)cn3)CC12 N1(C(C2(CC)CCCN2C(c2ccc(C)o2)=O)=O)CCC(OC)C(C)(C)C1 c1(OC)nc(C(N2CCC(NC(c3ccc(C)c(C)c3)=O)CC2C)=O)cc(O)n1 c1(C(N(CC(C)O)CCF)=O)cc(Br)c2occc2c1 C(=O)(C(C)CC(C)C)N(CCCNC(C(=Cc1cnc[nH]1)C)=O)C1CC1 CCCCC(C)(F)C(=O)NCC1CCCCN(C(c2cn(C)nc2C)=O)C1 N1(C(CCC(=O)N(C)C)=O)CCCCC(C(=O)NCc2ccc(CO)cc2)C1 N1(C(C(COCC)C)=O)CC(C)(C)CCC1CNC(c1cscc1C(F)(F)F)=O C1(C)(CNC(C(C)(C)N(C)C)=O)COCCN(C(=O)C2=CCCCC2)C1 N1(C(c2cc(F)c[nH]2)=O)CC2(CCN(C(c3ccccc3C3CC3)=O)CC2)C1 C=C1CCC(C(=O)NC2CC3(C2)CC3NC(=O)CNC(=O)OC)CC1 CC1CC(CNCCCN2CCCN(C(=O)OC(C)(C)C)CC2)CC(C)C1 c1(CC(=O)NCCCCCCNC(CSS(C)(=O)=O)=O)ccc2cccnc2c1 c1(N2CC3CN(C(C4CCN(C(C)=O)C4)=O)CC3C2)ccc2nccnc2n1 CC1=C(F)CN(C(=O)CNC(c2cc(C)n(C)n2)=O)CC1 c1(C(N(CCCNC(C(C(C)C)SCC)=O)CCO)=O)cn(C)c(=O)cc1OC CCCCC(O)C(C)C(=O)NCC(CNC(c1cnc2cc[nH]c2c1)=O)CO N1(C(C2C(C)(C)C2C#N)=O)CCOC(C)(CNC(c2coc(C(F)F)c2)=O)C1 c1(CNC(C2CC(F)CN2C(C2CCCS2)=O)=O)c[nH]c2ccc(Br)cc12 N1(C(c2ccc(C)nc2)=O)CC(O)CCC1C(N1CCC(C(C)C)CC1)=O N1(C(C2CC(C(=O)OC)C2)=O)CC(CNC(=O)CC2CCCN2C)CC1(C)C N1(C(C(c2ccc(C)s2)C)=O)CC(NC(C2CC2C)=O)CC(C)(C)C1 c1(C(=O)NC2CC(CNC(C3(C)CCCCO3)=O)C2)cc(N)ccc1Br c1(OC)nc2ccc(CC(=O)NC(C(F)F)c3ccco3)cc2s1 C1(NC(CC(=O)NC2CC2)=O)CC(NC(=O)CCN2CCCCC2=O)CC1O N1(C(C2CNC(=O)N2)=O)CC(CNC(c2cccc3[nH]ccc23)=O)C2(CCC2)C1 C1(NC(c2ccsc2C(F)F)=O)CC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 N1(C(C2(CC#C)CCC2)=O)CCC2(CC1)CC2C(=O)NC1CCC(O)(CC)CC1 CCC(CN(C)C)C(=O)N(C(C)CCNC(=O)CSc1ccc(OC)cc1)C c1(CNC(C(c2ccsc2Br)N(C2CCC2)C)=O)cccc(Br)c1 c1(SC)nc(N2CCOC(C(C)NC(C3(C4CCC4)CC3)=O)C2)cc(C(F)F)n1 N1(C(C2(CCN(C)C)CCCC2)=O)CC2CC(NC(=O)C3=CCCC3)CC2C1 CCCCC(O)C(=O)Nc1cccc(-c2c(OC)cccc2O)n1 N1(C(CC(C(=O)OC)(C)C)=O)C2CCCC1CC(CNC(=O)Cc1cn[nH]c1)C2 c1(C(=O)NCCC(=O)NC2CC2CF)c(F)cccc1F C1(NC(CCOCCN(C)C)=O)CCC12CN(C(=O)CCn1ccc(O)nc1=O)C2 C1(C)(C(C)(C)C)CC(C(=O)NC2CC2CNC(C2CC3CC3C2)=O)C1 N1(C(=O)NC(CC(C)C(F)F)C)CCCCC(C)(F)C1 C1(N(CCC(=O)NC2CCOC2)C)CCN(C(C2CN(S(C)(=O)=O)C2)=O)CC1 C1(C(=O)Nc2c(CNC(CC=CC)=O)c[nH]n2)CC(SCC(F)(F)F)C12CCC2 c1(C(N2CCC(NC(C(CC)=CC)=O)(CF)C2)=O)cc(OC)cc(C)n1 c1(C(N(C2CCN(C(C(COC)C)=O)C2)C)=O)cncc2[nH]ccc12 CC(C)(CC(F)(F)F)C(=O)NCCC1CCCN1C(=O)CN1CCOCC1 C(=O)(CC(C)C(C)(C)C)N1CCC(O)(CCNC(C=COCC)=O)C1 C1(C(=O)NCCc2ncccn2)(NC(C(C)C2CC2)=O)CC1(C)C C(=O)(C1=NOC2COCC12)N(C1CN(C(=O)CCn2cccn2)CC1(C)C)C N1(C(C(=CC2CCCC2)C)=O)CCCCCC1CNC(c1snnc1C1CC1)=O C1(NC(CCNC(CC(C)C)=O)=O)CC(CNC(=O)CC=C(Cl)Cl)C12CCC2 c1(C(N2C(CNC(c3cnn4cc[nH]c34)=O)CCC2)=O)cccn(O)c1=O c1(OC)ccc2c(c1)NCCN(C(c1ccn3ncccc13)=O)C2 N1(c2nc(C)cc(CC)n2)CC2CCC1C1CN(C(=O)CCS(C)=O)CC21 c1(N2C(=O)CC(C(=O)NCC(CNC)(C)C)C2)ccc2nc(CN)oc2c1 C1(O)(CNC(C2(C)CC2(Cl)Cl)=O)CCCN(C(=O)C(F)(F)C(F)F)C1 CCC(CC(C)C)C(=O)NCCN(C(C1C(F)(F)C12CC2)=O)CC1CC1 N1(C(C(C)(C)OCC)=O)CCCC(C(C)C(=O)NC(c2cn(C)nn2)C)C1 C1(C(N2CCC(CNC(C34CCC(F)(CC3)C4)=O)C2)=O)CCCCC(F)(F)C1 c1(NC(=O)NC(C(=O)OC)OC)ccc(CS(C)(=O)=O)cc1 C(=O)(CC1COc2ccccc21)NC(CNC(C(C(=O)OCC)(C)C)=O)C c1(N2CC3C(C(F)(F)F)(C3)C2)nccc(-c2ccncc2)n1 c1(C(N2CCC(NC3C(OC)COC3)CC2)=O)ccnc2c1CCC2 c1(CCNC(c2cnc(C)o2)c2nnnn2C(C)(C)C)c(C)noc1C CC1=C(C(=O)N2CC(NC(=O)C3=NOCC3)CC2(C)CO)SCCO1 C1(CC(=O)NCC(CNC(Cc2n[nH]c(=NC)s2)=O)(C)O)CCCC12CC2 c1(CC)nc(C(=O)NC(CNC(=O)C(CC)CC)C2CC2)c(N)s1 c1(NC(=O)NCc2cc(N(C)C)ncc2)sc2ccccc2c1C#N CCCCC(CNC(=O)C(c1ccc(Cl)cc1)=O)NC(c1cnn(C)c1)=O CC(C)C(C(=O)Nc1cncc(C(=O)NC(C2CCOC2)C)c1)c1ccccc1 CCCC(CC)CC(=O)NCC(CNC(c1ccc(CO)c(Cl)c1)=O)CO c1(CN2CCC(NC(c3ccc(Cl)cc3)=O)CC2)c(F)ccc(F)c1Cl N1(C(CCCC(C)=O)=O)CCC(O)(C2(NC(c3cc(Br)no3)=O)CC2)CC1 C1(N(C(C(C)OCC#C)=O)C)CC2CCC(C1)N2c1ncns1 C1(OC)CC(CNC(=O)C(C2CC2)N(C)C)N(C(C2CC3(CC3)CO2)=O)C1 CNS(=O)(=O)N1CCN(C(=O)C2CCc3ccc(Br)cc32)CC1 N1(C(C2N(C(C)(C)C)CC2)=O)CCCC(C2CC2NC(c2ccsc2)=O)C1 N1(C(C2C3(CC(NC(C(C)SC)=O)C3)C2)=O)CCCC(C)(C)C1 C1(C(=O)NC2C(OC)COCC2)COCCN(C(C2(Cl)CC2(F)F)=O)C1 c1(C(N(CC(CNC(CCOCC(C)C)=O)C)C)=O)sc(=N)[nH]c1C1CC1 c1(CCC(=O)NC2C(NC(C(C)NC(CC)(C)C)=O)C2)ccc(OC)c(O)c1 C1(NC(c2cc(SCC)ncc2)=O)CCCCN(C(C2(CO)CCCO2)=O)C1 C(=O)(C1CCc2nccn21)NC(C(=O)N(CC(CC)C)C)C(C)(C)O NS(=O)(=O)c1cccc(CCC(N2CC3(CCCCC3)C2)=O)c1 Cc1ccc(C(=O)NC23CC(NC(=O)Nc4ccc(COCO)cc4)(C2)C3)cc1 C1(C(N(C)CC2(CNC(c3cnco3)=O)CC2)=O)CCCCS1(=O)=O C12(C(C)NC(N3CCC(NCCC(C=C)(C)C)CC3)=O)CC3CC(CC(C3)C1)C2 C1(CNC(c2c(SC)snn2)=O)CCC(N(C(=O)CCc2nncn2C)C)CC1 C1(CNC(C2N(C(C)C)CCC2)=O)CCCCN(C(=O)C(C)c2cccs2)C1 C1(NC(CCNC(COC)=O)=O)CCC12CN(C(=O)C(F)C(F)(F)F)C2 N1(C(CCOc2ccc(OC)cc2)=O)CC2CC1CC2NC(=O)C(C)=C1CCC1 C(=O)(CCCCC#N)NCCOCCCN(C(=O)CCC1(C)CC1)C c1(C(N2CC(NC(c3ccc(OC)c(O)c3)=O)C(F)C2)=O)cc2ccccc2o1 Cc1ccc(-c2cn(-c3ccccc3C(=O)N(C)C(C)C)nn2)c(C)n1 N1(C(c2cc[n+]([O-])cc2)=O)CC2(CCCN2C(c2ncn(-c3ccccc3)n2)=O)C1 N1(C(C(CSC)(C)C)=O)CC=C(CC(=O)NCC2(O)CC3C=CC2C3)CC1 c1(N2CCC(C)(C(=O)NC3CC3)C2)ccn2nccc2n1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2(CC1)CC2C(=O)NC1CCCC(O)C1 c1(C(CO)NC(C2CCCCC2O)=O)ccc(C(F)(F)F)cc1 c1(CC(=O)NCc2nc(C(C)(C)C)sc2)c[nH]c2ncc(Br)cc12 C1(C(N2CC3CC3(CNC(C3(CF)CCC3)=O)C2)=O)Cc2nccn2C1 CC(C)(C)C(=O)C(=O)NCCCCCCNC(=O)COc1cccc(C#N)c1 S(=O)(=O)(c1ccc2ccccc2c1)NC(C)C(=O)NC1CCCNCC1 C1(NC(C2C(CC)C2)=O)C2CCCN(C(=O)CCOCC(C)(C)C)C2C1(C)C Cn1nc(-c2cccnc2)cc1C(=O)NC1CC1NC(c1ccon1)=O CC#CCC(CO)NC(=O)CC(C)CNC(c1ocnc1CCC)=O C1(C(=O)OC)CCCCN1C(c1nc(C(C)NC(c2ccc(F)nc2)=O)cs1)=O c1(CNC(C2C(CC)N(C(=O)Cc3ccn(C)c3)CC2)=O)ccc(C)cc1O N1(C(C2(CC)CC2)=O)CCN(C(=O)Cn2cc(C3CCOC3)cn2)C(CCO)C1 C1(C)(C(N(CCOCC)C)=O)CN(C(=O)CSc2ccc(F)cc2)C(C)(C)C1 Cc1ccc2c(c1)CN(C(C1C(O)CCN1C(C1C3C4CCC(C4)C13)=O)=O)C2 C1(C(=O)NC(C)C(=O)O)CC2CCN(C(=O)CSCC3CCCC3)CC12 c1(CCNC2(c3n(-c4c(C)cccc4)nnn3)CCC2)cc2[nH]nc(C)c2cn1 c1(C(=O)NC2(CNC(c3ccoc3Cl)=O)CCC2)cc2c(Cl)cccn2n1 N1(C(C2C(OC)CCC2)=O)CCOC(CNC(=O)C(c2nc(C)cs2)C)C1 C12(C(=O)OCC3CCCCN(C(=O)OC(C)(C)C)C3)CCCCN1CCC2 c1(CNCCP(OCC)(C)=O)c(F)ccc(Cl)c1Br CC(C)(C(=O)NCc1cc(C(=O)NC2CCN(C(N)=O)C2)n[nH]1)C(F)F Cc1nc(NCc2nc(C3CC3)cs2)cc(=NCC2(C)C=CCCC2)[nH]1 N1(C(=O)NCCc2cccc(CC)c2)CC(=O)OCC1c1ccccc1 c1(CC2C(C(N(CC(C)(C)NC(=O)C(C)(C)c3ncco3)C)=O)C2)sccc1C#N C1(NC(=O)CCF)CC2CC(C1)CN(C(=O)C(c1ccc(F)cc1Br)O)C2 C1(NC(C(CC=CCC)C)=O)CCCN(C(C2CCC(=O)CC2)=O)CC1 CC1=C(C(=O)N2C(C(=O)Nc3cc(CO)ccc3C)CC2C)CCO1 c1(C(C(=O)N(CCCNC(=O)C(CSC)OC)CC)(F)F)cccc(C)c1 C1(NC(COC2C(C)CCCC2)=O)CCSC12CN(C(=O)C(C)(C)C1CCC1)C2 c1(CNC(NC(CC)C)=NCC2CCCC(=O)N2)c(C)ccc(Br)c1F C12CN(CC1(C)C)C2=O.c1(NC(C)=O)ccc(NC(c2cccn2C)=O)cn1 C1(NC(c2nc(-c3ccccc3F)cs2)=O)NCCCC1C(F)(F)F c1(C(CNC(C(CC)SC)=O)NC(=O)Cc2nn(C)cc2Cl)ccc(F)cc1F C#CC1(C(=O)NCC2(O)CC(CNC(=O)CSCC)C2)CCC1 C1(C(=O)NCCCc2cc(C(=O)OC)c(C)o2)CC12CCC(C)(C)CC2 c1(NC(C(=O)NCc2c(C)cccc2)=O)ccnc2c1CCO2 C(CC(C)(C)C)(C(=O)NCCc1ccncc1)NC(C(C(C)C)C1CCC1)=O C1(C(=O)NC(c2cccc(OC)c2)c2ccccn2)CC(C)(C)OC1=O C1(NC(c2cnn[nH]2)=O)CCCC12CCN(C(c1cc3n(n1)CCCN3)=O)C2 C1(C(N(CCC(C(C)C)NC(C(C=C=C)C)=O)C)=O)CC2CC(C1)CC(F)(F)C2 Cc1n[nH]cc1CC(=O)NC(C)(C)CNC(=O)CCOCC1CC1 C(=O)(C1=CCCC1)N1CCC(N(C(=O)COCC(=O)NC)CCOC)C1.CC CC(c1ccccc1F)=CC(=O)NC(Cc1ccccc1)CCC(=O)O CCC(C)(CCNC(=O)C(C)COC)NC(=O)C=Cc1ccnn1C C(CC(C(=O)N(C)CP(C)(C)=O)NC(=O)Cc1cnccc1C)=CC N1(C(C(=O)NC(C)C)=O)C(C)CC2CN(C(c3ccc4ncncc4c3)=O)CC12 C1(C(N2CCC(CC(N3CCOC(CN=[N+]=[N-])C3)=O)C2)=O)CC2(CC2)CO1 C1(CC(=O)NCC2C=CCN2C(c2ccnnc2O)=O)(OC)CCCCC1 c1(C(=O)NCC(C2CCCC2)NC(c2c(CC)ocn2)=O)c(O)cccc1O N1(C(C(CC#C)O)=O)CCCC(NC(c2cccn2Cc2ccncc2)=O)C1C C1(CNC(C2CCS(=O)(=O)C2)=O)CC2(C1)CN(C(=O)Cc1cccnc1)C2 C1(CC=C)(C(N2CCC(CN(C)C(C3CC(O)C3)=O)C2)=O)CCOCC1 O(NC(=O)C(CC(C)(C)C)NC(=O)CC1CC2CC2C1)C(CC)CC CCCC(C)(O)C(=O)NC1CC(N(C(=O)CCCc2ccc(C)cc2)C)C1 Cc1cccn2ncc(C(=O)NCC(C3CC3)NC(=O)C(C)(O)CC(C)C)c12 c1(C(N2C(=S)NC(c3c(C)cccc3)C2=O)=O)c[nH]c2c(F)c(Cl)ccc2c1=O Cc1ncnc(N2CCN(C3CCN(C(c4cc(F)ccc4Cl)=O)C3)CC2)c1Br c1(NC(C)C(C2CCCCC2)NC(=O)CCC2CCCCCC2)ncc(I)cn1 c1(C(=O)NC2(CNC(=O)CC3(O)CCOC3)CCC2)sc(Cl)cc1Cl CCC(CC)CCC(=O)OCC(C1CCN(C(=O)C(COC)N(C)C)CC1)C c1(C(=O)OC)ccc(N2CCN(C)CC2)nc1C.c12nccnc1C(=O)N2 C(c1ncco1)=CC(N1CCC(C2CCCN2C(=O)Cc2cscn2)C1)=O Cc1c(N)ccc(C(=O)NC2CS(=O)(=O)CC2NC(c2coc(O)n2)=O)c1Cl C=CCC(C(=O)N1CC(CC(=O)NC2(CO)CCOCC2)C1)c1ccccc1 C1(C(N2C(C)C(NC(=O)C(F)=C3CCCC3)CC2)=O)CCCS(=O)(=O)C1 CCCCCCCCC(=O)N1CC2(C1)CN(C(C1CC(OC)C1)=O)C2 CC1CCC(NC(c2cn[nH]c2)=O)CN1C(c1cc(Cl)cc(Cl)c1)=O Cn1nc(Br)c2ncnc(N3CCC(NC(=O)CC4CC(O)C45CCC5)CC3)c12 N1(C(C=C(CCC)CCC)=O)CC(N(C)C(c2[nH]c(=N)ccc2C)=O)C2(CC2)C1 c1(OC)cccc2cc(C(=O)NC(C)CC(C)NC(=O)C(C)(C)N3CCC3)[nH]c12 C1(C(N2CCC(CC(C)NC(c3occ(C)c3)=O)CC2)=O)CCC(N=[N+]=[N-])CC1 c1(CC(C)C(N(C(c2ccc(F)nc2)C)C)=O)ccc(F)cc1F C1(NC(CCN(C)CC)=O)C(CNC(=O)Cc2ccccc2Cl)CCC12CCC2 c1(CC)cc(C(=O)Nc2cccc(NC(=O)CN3CCCCC3C)c2)oc1CC N1(C(C2(COC)N(C(C3C(=C)C3)=O)CC=C2)=O)CCC2(CCOCC2)C1 N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCN(C(=O)C#CC2CC2)CC(C)(F)C1 c1(C(=O)NCC(C2CCCCC2)OCC)nc(Cl)ccc1Cl S(=O)(=O)(C1CN(C(C2(O)CC2)=O)C1)N1CCN(C(C2CCCC(C)C2)=O)CC1 c1(CNC(CC2(C)CN(C(C3COC3)=O)C2)=O)ccc(Br)c2ccccc12 C1(C(=O)NC2(CNC(c3c(C)n[nH]c3)=O)CC2)CC2CCCC12 C12(C(=O)NC(C3(O)CCN(C(CC(C)CF)=O)C3)C)CC3CC(C1)CC(O)(C3)C2 Cc1cc(C)c(C(=O)NCC2CC(O)CN2C(c2cnn3c2OCC3)=O)cc1N C=CC(F)(F)C(=O)N(CC(C)N(C(=O)OC(C)(C)C)C)C.C1(OCC(=O)N)CCCC1 C1(F)(CNC(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)CCCN2CCCC2)C1 C1(O)(CNC(c2cn(C3COCC3F)nn2)=O)CCN(C(=O)Cc2cnsc2)C1 c1(C(=O)NC2C3CN(c4nc(C#N)c(F)cn4)C2C3)ccc2[nH]nc(Br)c2c1 c1(NCC(O)CC(C(C(C)C)n2cncn2)=O)ccc(Cl)c(Cl)c1 C1(CC)(NC(=O)CN(c2ccccc2)C)CCCN(C(=O)Cc2ccc(C)o2)C1 CON=C(C(=O)N1CCCC(N(C(=O)CSC(F)(F)F)C)C1)c1ccco1 CCC(C)(O)C(=O)N1CC(CCNC(=O)C(C)CC#N)C(C)C1 N1(C(C(CC)(C)CNC(=O)CCc2ccoc2)=O)CCCC2C(=O)NCC12 c1(CC(=O)NC23CC2CN(C(C2(C(F)F)CC2)=O)C3)nsc2ccccc12 C(=O)(C#CC1CCOC1)N1C(CC)C(C(=O)NCc2cc(C)cnc2O)CC1 CCC(C)C(C(=O)NC1CCC(O)CC1)N(C(=O)C1=CCCCC1)C c1(C(N(C2CCC(F)(F)C2)CC)=O)cccnc1O N1(C(C(CC)(C)C)=O)CCC2(NC(c3cn(CCCC#N)nn3)=O)CCCC12 C1(NC(C(CC=CC)C)=O)CCC2CN(C(=O)CNc3ccccc3Cl)CC2C1 N1(C(C2C(=C)C2)=O)CCC2(CC1)CC2c1cn(CCc2ccc(O)c(O)c2)nn1 C(=O)(CCC(C)(C)F)N(C1CCCC(NC(CCCc2scc(C)n2)=O)C1)C c1(C(N2CCN(C(c3ccc[nH]3)=O)CC2c2cn[nH]c2)=O)cc2c(s1)CCOC2 C1(C(=O)NC2C(C(=O)NCc3n(C(C)C)ncc3)C2)C2CCCOC12 N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(=O)C(C)CCC(C)(C)C)C2(CCC2)C1 C1(CNC(c2n(CC)cc(Cl)c2)=O)N(C(=O)C(F)=C2CCCC2)CCCC1(C)C N1(C(C(=O)Cc2ccc(F)cc2)=O)CC2(CC2)CC1CNC(=O)Cn1nccn1 C1(NC(C(C)SC)=O)COC2(CNC(=O)C(c3ccc(C)cc3)(F)F)CC1C2 c1(C(=O)NC(C)CNC(C2CC2CF)=O)cn(-c2ncccn2)cn1 c1(C(N2C3C(C(=O)NCCC4C(C)CCCC4)C(C3)C2)=O)cc(F)c(F)cc1Cl N1(C(CCC=C=C)=O)CC2CCC(N(C(=O)COCC(C)(C)C)C)C2C1 c1(COC)cccc(NC(C2CC=CC(NC(=O)C(C)(CO)OC)C2)=O)c1C N1(C(CC(=O)OC)=O)CCC(C)C1CNC(=O)CC1CCC(C)CO1 C1(NC(c2cc(CCO)on2)=O)CN(C(=O)C2=C(Cl)CCC2)CCC1O C1(CC(N2CCC(CCN(C(=O)C(C)CC)C)CC2)=O)(COC)CCOCC1 S(=O)(=O)(c1ccc(CCC(=O)O)cc1)N(c1ccccc1)CCC(=O)O C=CCCC(O)CN(C)C(C1(C)C=CCN1C(=O)Cc1c(C)noc1C)=O CCN=c1[nH]c(C)c(C(=O)NC2CCCCCC2NC(=O)C(C)=CC(C)(C)C)s1 Cc1cccc(OCCC(N2CC3CC3(NC(=O)Cc3ccc(F)cn3)C2)=O)c1 c1(C(=O)NCCC2(O)CCN(C(C3C=CCCC3)=O)C2)noc2ccc(Cl)cc12 O=C1CCC2C(C(=O)NCc3ocnc3C(=O)NCC=CCl)C12 c1(C(C(=O)NCC(C)N(C(=O)CC2CCC2)CC)(F)F)ccc(C(C)C)cc1 C(=O)(C1CCCc2n[nH]cc21)NCCC(C)Nc1nccc(CC(=O)OC)n1 CC(CC(C)(C)C)C(=O)NC1CCC1C(N1CCC(O)(C(N)=O)CC1)=O C(=O)(C1=C(C)OCCS1)N(CCC(=O)NCCOC(CC)CC)CCO CC1CCC(NC(c2cn3c(n2)SCC3)=O)CN1C(c1nnn(C)c1N)=O C(=O)(CCCCCOC)N1CCC(CN(C(C2C(C(=O)OC)CCC2)=O)C)CC1 C1(NC(CC2(C)CCC2)=O)CCCC(CNC(c2cc(Cl)ns2)=O)C1 c1(C(=O)NC2C(NC(c3nc(C)oc3C)=O)CCC2)ccc2c(c1O)CCCC2 c1(NC(=O)NCC2CC3C(C2)C3(F)F)nc2c(s1)CC1(CCCCC1)CC2 n1(C(C)C)ncc(-c2noc(C3CCCO3)n2)c1F C1(C(=O)NC2C(NC(C(C)(C)Cc3cccc(Cl)c3)=O)CC2)NC(=O)OC1(C)C C#Cc1ccc(C(=O)NCCN(C)C(c2cnc(CC)[nH]2)=O)nc1 O=C(CC1=CCCC1)NCC1C2CN(C(=O)CCN(CC(F)(F)F)C)CC12 c1(-c2cn(C)nn2)nc(CCn2cc(Br)cn2)nn1CC(N)=O C1(NC(CCSCC#C)=O)CC(C(=O)NCc2cccc(C=C)c2)C12CCC2 c1(CC(C)C(=O)NCC2CN(C(C3(C#N)CCC3)=O)C2)ccc(Br)cc1 Cc1ccn2nc(C(N3CC(CNC(=O)CC4CC4C)C3)=O)nc2n1 c1(C(N2CCCC(N(C(C(CC)NC(N)=O)=O)C)C2)=O)cc2occc2[nH]1 C12(C(=O)NCC3CCN(C(c4ccoc4)=O)C3)CC3CC1C2C3 CCC(C)(C)C(C(=O)N1CCOCCC1c1cccc(C(F)(F)F)c1)NC(C)=O CCCCC(CNC(c1ccc(-c2cccs2)s1)=O)NC(c1nc(O)sc1C)=O C1(F)(CNC(c2cnc(O)s2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1 c1(CNC(=NC)NCc2c(F)cc(F)c(F)c2F)cccc(S(N)(=O)=O)c1 c12ccc(cc1Cl)[nH]c2=O.c1(CC(=O)Nc2ncc(CC)s2)ccc(Br)cc1C Cc1cnc(C)c(C(=O)NCCC2CCN(C(=O)CC3CCCC(C)O3)C2)c1 C1(CNC(C(C)(C)C)=O)CC2(CCC2)CN1C(C1CC=CCC1C(F)(F)F)=O N1(C(c2n(CC(C)C)ncc2)=O)CC2CCC(NC(=O)Cc3cn[nH]c3)CC2C1 C=CC(CC)CC(=O)NCCCCC1CCCN(C(=O)Cc2cn[nH]c2)C1 c1(C(=O)NCC2N(C(c3ncc(NC)nc3)=O)CC(OC)C2)c(C)[nH]c(C)c1C c1(OC)c[nH]c(C(=O)NCCN(C(C2CCOC(C)C2)=O)CC2CC2)cc1=O c1(C(=O)NC)ccc(C(=O)N(C)CC2(O)CN(C(=O)C=CCCC(C)C)C2)cn1 N1(CC2CN(C(C3CN(C(C(C)SCCCC)=O)C3)=O)C2)CCN(C)CC1 C1(C(=O)Nc2cccnc2C)(CC)CCN(C(c2cn(C3CC3)cn2)=O)C1 C(c1ccc(I)o1)=CC(=O)NC(C(=O)NC(C)C)C C(=O)(CC(C)(C)CC(=O)OC)NC1CC(F)(CNC(c2c(COC)noc2)=O)C1 C1(NC(C(CC#C)O)=O)CN(C(=O)C(CSC)c2ccccc2)CCC1O c1(CCC)cc(C(=O)NC2CCN(C(=O)CCCC3CCC3)C2C)cc(O)n1 Cc1cc(C(=O)NCC2CC(C(=O)NN3CCC3C)C2)ccc1N1CCOCC1 N1(C(=O)CC(F)(F)F)CCC2CCN(C(C3(F)CC4(CCC4)C3)=O)CC2C1 N1(C(C=COCC)=O)CCC2(CCC(CNC(C3CN(C)C3)=O)O2)CC1 C(=O)(C1=CCSC1)NCCNC(C1CN(C(C(N2CCCCC2=O)C)=O)C1)=O C1(CNC2C=CC(C)(C)CC2)CCCC(C2CC2)C1 c1(CCC(=O)OCc2n(CCC)ccn2)cccc(F)c1Br c1(OC)c(NC(C2CCCN2C(=O)CC2CCCN2C(C)=O)=O)cnn1C C1(C(C)C(=O)NCC(O)CO)CCCN(C(C2(CF)CC(=O)C2)=O)C1 N1(C(C(C(C)C)(C)O)=O)Cc2ccccc2CC1CNC(=O)CC1CCN(C)C1 Cc1oc(C)c(C(N2CC(NC(=O)CCc3cnoc3)C(C)C2)=O)c1C c1(C(N2C(CN(C(CCOCCOCC)=O)C)COCC2)=O)cccc(C)c1F C1(NC(Cc2nnc(C)o2)=O)CC(O)CN(C(=O)CC2(n3ccnc3)CC2)C1 C1(C#N)(C(N2CCC(OC)(CNC(C3CCC3(F)F)=O)C2)=O)CCCCCC1 C1(C(N2CCC(NC(Cn3nnc(=N)[nH]3)=O)(CO)C2)=O)CCc2nc[nH]c2C1 C1(NC(COC(CNC(C2(C(C)(F)F)CC2)=O)(C)C)=O)CC(F)(F)C1(C)C CS(=O)(=O)C(C(=O)Nc1ccc(NS(C)(=O)=O)cc1Cl)C1CC1 N1(C(c2c(C)n(C)nn2)=O)CCN(C(C2COCCN2C(=O)N(C)C)=O)CC1C c1(C(N2C(CN=c3nnn(C)[nH]3)(C)CCC2)=O)csc2c1CCCC2 C(=O)(CC(C(C)C)OCC)N1CCC(N(C(C2(CC)CC(OC)C2)=O)C)CC1 C1(CNC(COCCOCC)=O)CNCCN1C(C1CN(C2CCOC2)C1)=O c1(C(=O)NC(C)CCC2CCCC2)cc(CNC(=O)CC(C)C2CC2)on1 CCCCC(CC)CC(=O)NC1CCC(N(c2nc(C)nc(Cl)c2C)C)CC1 c1(C(=O)NC(C)CNC(C2CCOC(=O)N2)=O)ccc2c(c1)NC(C)CC(=O)N2 C(c1ccc(F)cc1)=CC(=O)NC1CCC(N(C)C(c2ccco2)=O)CC1 N1(CC(=O)NCC)CCCC1C1CCCCN1C(=O)C=C1CCCCC1 c1(C(=O)NCCN(C(=O)CCN2CCCC(C(C)(C)C)C2)CC)cccc(NC)c1 C1(C)(CCC)CCN(C(=O)C(C)(C)CNC(C2CC=CCO2)=O)C1 c12ccnc(c1)NC2=O.C1(=O)C(C2CCOC2)N1.N(CCC1CC1)(CC)CC c1(C(=O)NC2(C(=O)O)C(C)C2)cccc(Cn2cc(-c3ccccn3)nn2)c1 CC1(C)CCCCC1C(N1CCCC1CN(C(C12CCC(CC1)CO2)=O)C1CC1)=O N1(C(CCCC#C)=O)C2CCC1C(F)C(NC(C1CCC(N(C)C)CC1)=O)C2 C1(C(=O)NCC(CO)NC(C)=O)CCN(C(c2cc(CO)on2)=O)CC1 C1(NC(C2(C)CC(C)C2)=O)CCC(CNC(=O)Cc2ccsn2)CC1 CCCCC(C)C(=O)NC12CC1CN(C(c1coc(C(F)F)n1)=O)C2 c1(C(N2C(C(=O)Nc3cc(C)cc(O)c3)CC2C)=O)cc(C#N)ccc1C c1(C(C=CC(=O)NCCN(CC(C)C)CCOCC)C)ccccn1 N1CCC(CCn2nccn2)CC1.n1(CC)ccnc1 CC(C)S(=O)(=O)C(C)C(=O)N1CC(NC(=O)Cc2nc[nH]n2)C(CC(C)(C)C)C1 N1(C(C2N(C)CCCC2)=O)CCN(C(c2cnc(-c3ccsc3)s2)=O)CC1CF C1(CN(C(CC(C)n2cccn2)=O)C)C2CN(C(c3ncccc3F)=O)CC12 C(=O)(C1CCCc2sccc21)NC(C)CNC(C1(C2CCC(=O)NC2)CCC1)=O C(=O)(C(=O)N=S(C)(C)=O)NC(CCCNC(CN1C(C)CCC1C)=O)(C)C C(=O)(C(F)C(C)(F)F)N1C(C2(C(=O)NCc3n(C)cnc3)CC2)CCC1 C(=O)(CCCC(=O)NC1CC1)NCC1CC(C)N(C(=O)Cc2ccnc(O)c2)C1 CS(=O)(=O)c1ccnc(NCCCC(CC)Nc2cc(C#N)ccn2)n1 N1(S(CC)(=O)=O)C2CCC1CC(C(=O)NCC1(O)CCCN(CCO)C1)C2 Cc1cnc2ccc(C(=O)NC3(CNC(C4(Cl)CC4(C)C)=O)CC3)cn12 Cc1nn(C)cc1C(=O)NC1CCN(C(C2CCN(Cc3ccsc3)CC2)=O)C1 c1(CC)cccc(C(=O)NCC2C=CC(NC(c3ccc(C4CC4C)o3)=O)C2)c1 N1(C(CCC)=O)CCCCC1C(=O)NCC(c1scnc1C)N1CCOCC1 Cc1nc(-c2c[nH]cc2C(=O)NCCC2CCCN2C(C2CC2C)=O)cs1 C12(C(=O)NCC3(NC(CCN4CC(=O)NCC4)=O)CC3)CCCC1C2(F)F N1(C(c2cn(CCC)nc2C)=O)CCCN(C(C2CCCCO2)=O)C(CO)C1 c1(CNCC2N(C(C3CCO3)=O)CCC2)ccc(Oc2ccccc2)cn1 Cc1cncc(C)c1C(=O)NCC(C)(C(C)C)NC(C1CC2CCC1CC2)=O C1(F)(NC(C2CCOCC2)C)CCN(Cc2cccc(C(F)(F)F)c2)C1 N1(C(Cc2ccn(C)c2)=O)CCC(C(=O)NC(CO)CC(F)(F)F)C1(C)C c1(OCC(=O)NCC(CO)NC(c2nc(C)sc2)=O)ccccc1O.C(C)C CCCC(CCC)NC(C1CCC(C2CC2)N1C(=O)CCCOC(C)=O)=O C=C1CCC(C(=O)NCCC2CCN(C(C3CC(OC(C)(C)C)C3)=O)C2)CC1 C1(NC(C(C)OCCC#C)=O)COC2(CCN(C(c3ccnnc3O)=O)CC2)C1 CCC(C)CCCCC(=O)NC1C(C)(C)C(NC(c2ocnc2C)=O)C1(C)C c1(C(=O)NCCCC(C)NC(C2(CC#C)CCCCO2)=O)nccc(C)c1F N1(C(C(C)c2ncco2)=O)CC2(NC(C3CC(=O)N(CC(F)(F)F)C3)=O)CC2C1 Cc1ccc2sc(C(=O)NCCNC(=O)Cc3ccc([N+](=O)[O-])cc3Cl)cc2c1 N1(C(CN(C(=O)OC)C)=O)C(C(=O)N(CC(O)C2CCC2)C)CCC12CC2 C1(NC(c2c(SC)scc2)=O)CCCCC1NC(c1[nH]c(C)nc1C)=O O=C(CCCCCc1ccc(O)cc1)NCC1(CNC(c2nsnc2O)=O)CC1 Cc1csc2ncnc(N3CCC(C)(C)C(CNC(=O)CCCS(N)(=O)=O)C3)c12 N1(C(C(C)OCC)=O)CCCC(N(C(=O)Cc2ccccc2Cl)C)C1 CC(C)CC(CNC(=O)CCC(C)(C)N(C)C)C(=O)NC(c1ccc(F)cn1)C C12(C(=O)NCC3N(C(C4CCCC(O)C4)=O)CCC3)CCCN(CCC1)C2 CC(CCN1CCC(CS(C)(=O)=O)C1)C(=O)NC1CCCCC1 C12(CCNC(C3N(CCC)CCC3)=O)CCC1CN(C(=O)Cc1c[nH]nc1O)C2 c1(N(C(C2CCCCC2)C(=O)NC2CCCCC2)C)cncc(C(N)=O)c1 C1(NC(C(Cn2ccnn2)NC(Cn2nnc(C)n2)=O)=O)CCN(C)CC1 c1(C(=O)NC(C(=O)NCC2N(C(C)=O)CCCC2)CO)cc2ccsc2s1.C(N)=O c1(OC)cc(OC)nc(C(N2CCC23CC(c2ncc[nH]2)C3)=O)c1 c1(C(C)OCC)noc(CC(=O)N(C)CCCCCNC(=O)Cn2ncnn2)n1 c1(SCCCC(N2CCCC(NC(C(CSC)O)=O)C2)=O)ncnc2[nH]cnc12 C#CC(CC(C)(C)C)NC(C1C=CCN(C(c2cc(O)cc(F)c2)=O)C1)=O C(CN=c1nc(N2CCC3(CCCC3)C2)c2[nH]ccc2[nH]1)OCCC(C)C C(=O)(CCCCCC(C)O)NC1C(CNC(c2ccc(CC)cn2)=O)COC1 N1(C(C)C)CCC(CC(=O)NC(C)(CNC(=O)CC2CC2C2CC2)CO)CC1 CC(C)C(C)C(=O)N1CCC(CNC(C2CCCC(CF)C2)=O)CC1 CCC(C)(CC(=O)NCCN(CC(C)O)C(c1cccc(COC)c1)=O)C(=O)OC N1(C(C2C(C)C2)=O)CCCC12CCN(C(c1cc3c(s1)CC(C)(C)C3)=O)C2 C(c1ccc(S(C)(=O)=O)o1)=CC(N1C(C#C)CN(C(C2CCC2(F)F)=O)CC1)=O C(C(C(C)(C)C)Nc1cc(CN2CCC(O)CC2)ncn1)NCc1ccc(C)o1 c1(OC)cccc(NC(=O)CCN(CC2CC2)CC2CCCO2)c1 N1(C(C=C(C)C)=O)CC(C)CN(C(c2ccnc(O)c2Br)=O)C(C)C1 CC(CNC(=O)C(F)(F)c1ccccn1)(Cn1cccn1)N=c1cc(Cl)c(O)n[nH]1 O=C1CC2(CCN(C(=O)C(c3cccc(Oc4nccs4)c3)(F)F)C2)CN1 c12cc(Br)ccc1S(=O)(=O)N2.c1(CCN(CCOCCC=C)CC)ccncc1 Cc1noc(C(F)(F)F)c1C(N1CC(CC(=O)NC2COCCC2C)C1)=O c1(C(N2CCC(N(CCC)C(C3CC3CC)=O)C2)=O)ccc2cn(CC)nc2c1 CCC(O)C(F)(F)C(=O)NC(C1CN(C(c2cc(=O)n(C)cn2)=O)C1)C CCC(CCC(=O)NCCc1ccncc1F)NC(C1CNC(=O)O1)=O CC#CCCC(=O)NC1CC(CNC(=O)CCCCC2CCCCC2)C1 C(=O)(C(C)(C)C(=O)NC1CCN(C(=O)CN2CCC(F)(F)C2)CC1C)NC CCC(C)(CNC(=O)CCC1CCCN1C(=O)C(C)N1CCCC1)CO C1(C(N(C2CCN(c3ccc(C#N)nc3)C2)CC)=O)CCc2cncn2C1 CC12CC(C(=O)NC3CC(NC(c4cccnc4O)=O)C3)(C1)C1(CCC1)O2 c1(-c2cn(Cc3ccc(N4C(=O)NCC4)cc3)nn2)ccc2nccnc2c1 C1(C(=O)NC2C(NC(c3cc(C(N)=O)[nH]c3)=O)CCC2)Cc2ccccc2C1 c1(C(=O)NCC(CCNC(C(C)(C)OC)=O)O)[nH]cc2c(=O)n(C)ccc12 C1(C(N2CC(C#C)(F)C2)=O)CC(F)CCN1C(c1ncoc1C)=O c1(NC(C)=O)ncc(S(=O)(=O)NC2CN(Cc3nccs3)CC2F)s1 N1(Cc2cccc(CC)c2)Cc2[nH]nc(NC(c3cccc4[nH]ccc34)=O)c2C1 c1(C(=O)NCCCCCN(C(c2c(CC)ccs2)=O)C)cc(OC)cc(C)n1 C=CCC(CC)C(=O)N1CCC(CCN(C(=O)Cc2sc(C)nc2C)C)CC1 c1(N(Cc2c(C)cccn2)CC2(C)CCCC(=O)N2)ccccc1[N+](=O)[O-] CC1CCCN(C(=O)CCn2ccnn2)C1CNC(=O)CN1CCN(C)CC1 C1(C(=O)NC(C)C(C)(C)O)CCN(C(=O)C(F)C2CCC2)O1 CCC(C)C(O)C(C)C(=O)N1CCC(CCNC(=O)CCc2ccsc2)C1 Cc1cc(C(=O)NCCC2(O)CN(C(c3cn(C)nc3Cl)=O)C2)cc(C)c1F C1(C(=O)NCC(C)(C)CNC(=O)C(F)F)CC12C1CC3CC(C1)CC2C3 c1(C(CNC(c2ccnn2CC(C)C)=O)NC(C(=O)NCC)=O)cccc(C)c1 C1(OC)CN(C(=O)C(C)(C)OCC(F)(F)F)CC1NC(C1CCCCCS1)=O C1(N(c2c(SCC)cccn2)C(c2ccnc(C(N)=O)c2)=O)CCCN(CC)C1 c1(C(=O)NCC(C)CNC(=O)C(C(C)(C)C)n2ccnn2)ccc([N+](=O)[O-])cc1 C1(NC(CCCC#N)c2n(C)nnn2)CC2CC3C(C2)C13 N1(C(CNS(CC)(=O)=O)=O)CC(NC(=O)Cn2cc(C3CCC3)nn2)C(C)(C)C1 c1(OCC)nc(Cl)ccc1C(=O)NCCC(C)NC(C1CCCC1O)=O CC1CCN(C(c2c[nH]c(=N)nc2O)=O)CCN1C(c1noc2c1CCCC2)=O Cc1ncn(C)c(=O)c1C(=O)NCCNC(C1(C#N)CC2(CC2)C1)=O C1(OC)CC2(C1)CC(C(=O)NCC(CO)NC(=O)CC1CCC(F)(F)CC1)C2 C=C(C)C(C)(C)C(=O)NCCC1(NC(c2cc(C#N)n(C)n2)=O)CCC1 N1(C(CC(CC)(C)C)=O)CCCN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1C N1(C(C(CCC2CCC2)NC(c2ccn(CC)n2)=O)=O)CCc2ncncc2C1 C(c1c(Cl)cccc1Cl)=CC(=O)N(CC(C)(C)NC(c1c(C)snc1)=O)C Cc1nsc(N2CCC(N(C(=O)C=C3CCCCC3)C)CC2)c1C#N CCCCC(O)C(=O)NCC1CN(C(c2ccccc2O)=O)CC1O c1(OC)ccc2[nH]cc(CC(=O)OCc3noc(COCC(C)C)n3)c2c1 N1(C(CC(CCC)C)=O)CC(NC(=O)Cn2ncc(Br)n2)CC(C)(C)C1 c1(C(=O)NC(c2ccc(C)cc2)CNC(=O)CN2CCCC2)cc(N)c(F)cc1C C1(CC(=O)NCC(C)NC(C=C)=O)CC(=O)NC(=O)C1 C(=O)(CC1(O)CCOc2ccccc21)NC1CCN(C(C(CCC)CCC)=O)C1 N1(C(CC2(OC)CCC2)=O)CC2(CC(NC(c3ccccn3)=O)c3nccn32)C1 C1(C(=O)NCC2(O)CN(C(c3cc(OC)c(F)cc3)=O)C2)CC2C=CCC(C1)C2 c1(C(N2CC(C(C)(C)O)(CNC(CCCCCC)=O)C2)=O)cc2n(n1)CCCO2 c1(CNC(COCC#C)=O)cc(C(=O)NC2(C(N)=O)CC(CO)C2)n[nH]1 c1(N2C(CCC=C)CCC2)nc(=NCC23CCC(C2)C(C)(C)O3)[nH]c2ccsc12 Nc1cc(Cl)nnc1C(=O)NC1CS(=O)(=O)CC1NC(c1c[nH]cc1C1CC1)=O C(CC(=O)N(CC(O)CN(C(=O)Cc1c(C)cccc1F)C)C)(C(C)C)OCC CCC(N=c1cc(NCC(=O)N(C)C)nc(C(C)C)[nH]1)C1CCOC1 c1(C(N2CC(CCNC(C(C(C)C)O)=O)C2)=O)cc2ccnc(Cl)c2s1 C1(CCNC(c2ccc(C)nc2)=O)CN(C(c2ncsc2C2CC2)=O)CC(C)O1 c1(OC)cc(C(N2CC(CNC(c3ccsn3)=O)CC2C)=O)cnc1O CCCC(C(=O)OC)C(=O)NC(CO)C(=O)NCCc1cnn(C)c1C C(=O)(CC1=CSC2=NCCN12)NC1C(C2CCN(C(c3cc(C)on3)=O)CC2)C1 S(=O)(=O)(c1c(C)cccc1Cl)N(C(C=CCCC=C(C)C)=O)CC(F)F N1(C(c2nnn(C)n2)C(=O)NC(=O)OC(C)(C)C)CCn2cncc2C1 Cc1c(C(=O)NC(C2CCCN2C(=O)CC2CCCC(C)(C)C2)C)cccc1F C1(CC=C)(C(=O)NCC(=O)N2CCCO2)CCN(C(=O)C(F)C(C)C)C1 c1(C(=O)NC2CCCC(CNC(CCC#CC)=O)C2)cc(OC)c(S(N)(=O)=O)s1 C1(C(N(C)CCC2CCCCN2C(=O)CS(C)(=O)=O)=O)OC2CCC1CC2 c1(OC)ccc(NC(=O)C(=O)NC(C)C(=O)NO)cc1S(C)(=O)=O CC(C)(C)C(C(=O)NCC1CNC(=O)CO1)NC(=O)CCn1cnnn1 c1(C(N2CCCC(N(C(C(C)NC(N)=O)=O)C)C2)=O)cc2ccccc2s1 CC1CC2(CCO1)CC2C(=O)NC1CCCCN(C(c2ncn(C)n2)=O)C1 C1(C(=O)NCC2C=CC(NC(c3cc(OC)no3)=O)C2)CCCOC1C c1(C(N2C(CNC(CC3C(C)C3)=O)CC2)=O)cccc(-c2cnn(C)c2)n1 C1(O)(CNC(CC(C)C(F)(F)F)=O)CC2CCC(C1)N2C(=O)C(O)C(C)(C)C N1(C(c2ccc(CSc3scc(C)n3)cc2)=O)CCN(C)C(=O)C1C C12(C(N3CC(O)(C(C)C)C3)=O)CCCC1CCN2C(=O)CC1=CCCCC1 C1(NC(C(C)Cc2ccc(F)cc2)=O)CN(C(=O)C(F)=C2CCC2)CC2(CC2)C1 c1(CC2(C(=O)NN3CCC(C(=O)OCC)(CO)C3)CC2)ccc2c(c1)OCO2 C1(NC(C(=O)NCCC(N)=O)=O)CC2CCC1N(C(=O)Cc1ccc(O)cn1)C2 N1(C(C)=O)CCC2(CCCN2c2nc(N3CCOCC3)c3sccc3n2)CC1 CC1CCN(C(=O)COCc2ccccc2Cl)C(CNC(c2cc[nH]n2)=O)C1 N1(C(c2cnc(O)c(F)c2)=O)CCC(C2CN(C(C3CC3(F)Cl)=O)C2)CC1 N1(C(C(C)N(C(CCCOCC)=O)CC)=O)CCC(F)(F)C(C)C1 c1(C(N(CCC(C(C)C)NC(=O)CC(C)(C)C)C)=O)ccc2c(c1)CN(C)CC2 Cc1sc2ncnc(N3CCCC(C)(CNC(=O)C=Cc4cnc[nH]4)C3)c2c1C N1(C(c2nc(Br)sc2C)C(=O)NCC(=C)C)CCOC(C)(CC)C1 C(=O)(C1CCCc2c[nH]nc21)NC1(CC)CCN(C(C2CCC(C)C2)=O)CC1 Cc1ccc(C)c(C(=O)NC2CC(C)(CNC(=O)CC3CCCOC3)C2)c1 N1(C(c2c(C)ocn2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)C(CC(C)(C)C)C1 c1(C2C(NC(c3c(Br)n[nH]c3Br)c3n(CC=C)nnn3)C2)ccc(F)cc1 CCCC(C)(CCC)C(=O)NCC(C)CNC(c1cnn2c1OCC2)=O Cc1cc(C(=O)N(C2CN(C(=O)C(c3cccnc3F)(C)C)C2)C)c(C)s1 C1(NC(C(C)OCC#C)=O)C2CC1CN(C(=O)C(N1CCC(C)C1)=O)C2 C1(N(C(c2ccc(SC)s2)=O)C)CN(C(c2ccc(F)cc2O)=O)CC12CC2 C1(C(=O)NCC2CC(C(=O)NCC3CC(OC)C3)CO2)(CC)CCCCO1 Cc1cnc(C(=O)NC2CC(NC(c3cn(CCO)nc3C)=O)C2)cn1 C=CCCCCCN=c1[nH]c(N2CCC3CCCC3C2)nc2cccnc12 C1(CC=C)(NC(c2nc(Cl)ccc2Cl)=O)CCCN(C(C2(Br)CC2)=O)C1 C(CO)(C(C)NC(c1cc(CNC(=O)CSCCC(C)C)[nH]n1)=O)SC c1(C(=O)NCc2c(C(=O)NC(CCSC)CO)n[nH]c2)cnn(C)c1Cl CC1(C)CCOC1CC(=O)NC1COCC1CNC(c1cccnc1C(F)F)=O C1(CNC(C2(CC)CCNC2=O)=O)CN(C(C2(C)CCC(=O)N2)=O)CCC1(F)F C(=O)(C1CSc2ccccc21)NC1C(NC(C=Cc2c(C)n(C)nc2)=O)COC1 C1(CC)(CNC(=O)C(=O)Nc2cc(I)ccc2N(C)C)CCCC(=O)N1 N1(C(CC(C=C)C)=O)CC(CNC(c2cncc(NC)c2)=O)CC1(C)C C1(C(=O)NC(C#C)CC2CC2)CCc2nc(C#N)sc2C1 c1(CC)ccc(Cl)nc1NC(=O)C(C)NC(C(=O)OC(C)(C)C)C(C)C CCCCC(CNC(C1CN(C(c2ncncc2Cl)=O)CC(C)O1)=O)CCC N1(S(C)(=O)=O)CCN(C(=O)COC(C2(C)C=CCC2)=O)CC1 c1(OC)ccc(CCCNS(C)(=O)=O)cc1Cl.c1(C(=O)O)cnn(C)c1 C1(NC(c2cccc(=O)o2)=O)CCC2(CC1)CC(NC(=O)C(O)CC1CC1)C2 c1(C(N(CC(C)N(C(=O)C(C)OCCN(C)C)C)C)=O)cnc(C(C)(C)C)o1 c1(CC)cc(C)c(C(=O)NCCC(C)(C)CNC(=O)CC2(O)CCCCC2)o1 c1(C(=O)NCC(CC)(CC)NC(=O)C(O)C(C)OC)c(Cl)nc2ccccn12 c1(C(N(C2CC(C(F)C(=O)NCC(C)(O)C3(C)CC3)C2)C)=O)ccn(C)n1 N1(C(c2c(C)nc(COC)nc2C)=O)CCC2(CC(C(=O)NC(CF)CF)C2)C1 N=c1c(C(=O)NC2CCCCN(C(C3CCC=CCC3)=O)C2)c[nH]c2ccc(Br)cc12 NC(=O)CC(O)C(=O)NC1CC2(C1)CC2C(=O)NCCOc1ncccn1 C1(C(N(C2CCN(C(CCc3n[nH]c(=N)s3)=O)C2)CCO)=O)CC12CCCCC2 N1(C(c2ccc(C)cc2F)C(=O)NCCC#N)CCCSc2cc(C)ccc21 C1(O)(C(=O)NCCNC(C2CCC3(CCOCC3)C2)=O)CCc2ccccc2C1 N1(C(Cn2cc(COC)nn2)=O)CC(NC(C2(C(C)(F)F)CC2)=O)CCC1C c1(N2CCC(N(C(=O)C(C)CSSC)CC)C2)cc(SC2CC2)nc(C)n1 Cc1ccc(C(=O)Nc2cc(Cl)ccn2)cc1Cl c1(C(C2CCCCC2)C(=O)N(C)CCN(C)C(C2CCO2)=O)ccccc1F c1(C(=O)NC(c2ccc(F)cc2)CNC(C2(C=C)CCC2)=O)csc(=NC)[nH]1 CCC(C(=O)NCC(C)CN(C(=O)CCc1ccc(C)s1)C)OC Cc1ccc(OCCC(=O)NCC(C(C)(C)C)NC(c2nn(C)cc2N)=O)cc1 CC(C(=O)N1CCC(CNC(=O)COCC2CCCC2)C1)S(N)(=O)=O N1(C(Cn2c(C)ncc2)=O)CC(NC(c2cc(C(F)(F)F)cc(F)c2)=O)C(C#N)C1 C1(CCOC)(NC(=O)C(C)CS(C)=O)CCN(C(c2ccnc(CO)c2)=O)CC1 C(CCCCCNC(c1ccc(Cl)cn1)=O)NC(c1c(COC)ncs1)=O C(c1ccc(F)cc1)=C(C)C(N1CC2CC1(CNC(=O)CC(C)C1CC1)C2)=O C1(CC(=O)NC(CC)C(=O)NC23CC(F)(C2)C3)CCOC1(C)C N1(C(C)C)CCNC(=O)C1.C1(CO)C(=O)N1 N1(C(c2c(CC)c[nH]c2)=O)CC(N(C(=O)CC2CC(C)(C)C2)C)C(F)C1 CC(C(=O)NCC1CC(C(=O)NC2(CN(C)C)CC2)C1)N1CCCC1 Cc1c(NCC(F)(F)CC2CC2)ncnc1N1CCC(CO)CC1 N1(C(CC(c2ccc(OC)cc2)C)=O)CCN(C(=O)CCCOC)C2CSCC12 CC(CC(=O)N(C)CC1(O)CCN(C(=O)CN2CCOC2=O)CC1)P(C)(C)=O C1(O)(CNC(=O)CN2CCCS2(=O)=O)CCCN(C(=O)C(c2ccccc2)O)C1 N1(C(C(N)CC2CCOC2)=O)CCC2(CC1)NC(=O)N(Cc1ccccc1)C2=O C=C(C)CC(C(=O)NCC#CC(F)(F)F)NC(=O)CCn1ccnn1 c1(C(N2CC3(CC(NC(C(C)n4cccn4)=O)C3)C2)=O)cc2cccnc2[nH]1 c1(C(=O)NC2CN(Cc3cc[nH]n3)CC2O)ccc2c(c1)OCCO2 C(=O)(C(C)CCC(C)(C)C)NC(CNC(C1CCN(CC(C)C)C1)=O)C C1(NC(C(CC)N(C)C)=O)CC1C1CCCN(C(c2cc(C)n(C(C)C)n2)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCCC(O)(CCNC(C2CC(OC)C2)=O)C1 O=C(CC1=Cc2ccccc2C1)N1CCCC(NC(C23CCC2C3)=O)CC1 CCCC(CC)C(=O)N(C)CC1CCN(C(=O)C2=CSCS2)CC1 c1(CC)ncncc1C(=O)NC1CC1CNC(c1ccc(CO)s1)=O CN1CCCC2C1CCN2C(=O)CC1CC2CCC1O2 N#Cc1ccc(CN2CCC(F)(C(N3CCC(O)(C(F)(F)F)C3)=O)C2)c(O)c1 CC(CCC(=O)N1CCC(C)(O)C1)NC(=O)CSC1CC1 C1(NC(c2c(CC)nns2)=O)CN(C(C2CC(F)C2)=O)C2(CCOC2)C1 c1(C(=O)NCCC2CCN(C(C)=O)C(C)C2)c(F)ccc2[nH]ccc12 CC1(C)OCCC1C(N1CCSCC1C(=O)NC1C=CC(CO)C1)=O c1(C(=O)NC2CC3(CC(NC(C(COC)C)=O)C3)C2)nc(Cl)c(Cl)c(N)c1Cl C1(CCCNC(CC2CC(=C)C2)=O)CCN(C(=O)CC2(N(C)C)CC2)CC1 C1(CC(=O)NCC2CC(NC(C3(CC=C)CCCC3)=O)C2)CC(CC)=NO1 c1(C(C(=O)N(CCC)CCNC(C2(COC)CC2(F)F)=O)C)cc(F)cc(F)c1 C12(C(=O)NCCCCCNC(C(CC=C)CC)=O)CC(CO)(C1)OC2(C)C c1(NC(COC)=O)ccc(NC(=O)C(C)(C)OC2(OCC(F)(F)F)CC2)cc1 c1(NC2CCCN(CC)C2)ccc(S(=O)(=O)NCCC#CC(C)C)cc1Cl.C1CS1 c1(C(=O)NC(c2ccccc2)CNC(=O)CCc2nccs2)cc(Cl)nnc1O CC1CCCC(CCNC(=O)CCC(=O)C2CCCCC2)C1 c1(C(=O)NCC23CC2CN(C(c2cnc(S)[nH]2)=O)C3)ccc2oc(O)nc2c1 C1(NC(C(c2cncn2C)C)=O)CCC(C(=O)NCCCn2ccnc2)C1 n1(CC)ccc(CNC(=O)CC2CCN(C(C3(CCN=[N+]=[N-])CC3)=O)C2)n1 C1(NC(C2(C)CC=CCO2)=O)CCN(C(c2scnc2Cl)=O)CC1O c1(C(=O)NC2C(N(C)C)CC2)cccc2cncn12 N1(C(c2noc(CC)c2C)=O)CC2CCCC2(C(N2CC(SC)C2)=O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC2OCCN(C(=O)C(C)C(F)(F)F)C2C1 C1(C(C)(F)F)(C(=O)NCC(C)CNC(=O)C(F)=C2CCCC2)CCOCC1 c1(OCC)cncc(C(=O)NCC2C3CN(C(=O)C(O)C(C)C)CC23)c1 C1(C(=O)NCC2C(NC(c3ccc(-c4ccccn4)s3)=O)C2)CCC(F)CC1 CC(C)CCCCC(=O)NCC12CN(C(=O)C(C)OC(C)(C)C)CC1CCO2 c1(NC)ncccc1C(=O)NCC1CC(C)N(C(=O)CCN2CCC2)C1 N1(C(c2cncc(C)c2)=O)CCC2CCC(NC(C3CC(C)CCO3)=O)C12 C1(C(C)C(=O)NC(c2scc(CC)n2)(C(C)C)OC)CCN(CC)CC1 C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CC2CN(C(CCSCCC)=O)C1C2 CCCCC(CNC(c1cc(C)n(CCO)n1)=O)NC(C1CCCO1)=O CCC(CC)C(=O)N1CCCC1CC(=O)N(c1cncc(C(=O)OCC)c1)CC c1(C2C(C(=O)O)C2)ccccc1C(=O)Nc1ncc(CCN2CCOC3CC23)s1 C(=O)(C1CCCc2c(O)cccc21)NC1(COC)CN(C(=O)C(O)C(F)(F)F)C1 c1(N(CCNC(c2ncoc2-c2ccon2)=O)C2CC2)ncc2scc(Br)c2n1 C(CCN=c1ncc(C2CC2)c[nH]1)NC(c1ccc(C)nc1)=O Cc1nn(C)cc1CC(=O)N(C1CN(C(c2nn[nH]c2C(F)(F)F)=O)C1)C CCC(CC1CC1)C(=O)N1CCC(C)(NC(c2cc(COC)on2)=O)C1 C(=O)(CCC(F)F)NC(C)CCCNC(C1(C)CC1C(F)(F)F)=O Cn1nc([N+](=O)[O-])cc1CNC(=O)NCC(=O)NCC1(C)CCC1 N1(C(C(C)OCC)=O)CCOC2(C1)CN(C(c1cccc(Cl)c1F)=O)C2 N1(C(CCC(N)=O)=O)Cc2ccc(CNC(=O)CCn3ccnn3)cc2C1 c1(C(N(C(CNC(CSCC=C)=O)C)C)=O)ccc(NS(=O)(=O)CCCC)cc1 Cc1cc(C(=O)NCCCN(C)C(c2cn(C)nc2C2CC2)=O)nnc1O N1(C(c2ncn(C)c2)C(=O)NC2CC2)CCSC2CCCCC12 c1(OCC(=O)NC2(CN(C)C(c3cnn[nH]3)=O)CC2)ccc(F)cn1 c1(C(=O)NC2C(NC(C3(OC)CCOC3)=O)C2)sc(C#N)cc1C N1(C(C(c2cccnc2)OC)=O)CC(NC(=O)C(O)CC(N)=O)C2(CC2)C1 C1(CC#C)(C(=O)N(C2CCC3CC23)C)CCN(C(C2CC2(F)F)=O)C1 N1(C(C2C(C)CCCC2)=O)CCCC2(CCN(C(C3CCC(C)(C)OC3)=O)C2)C1 C1(NC(=O)CC(O)CNC(C2CCN(CCC)C2)=O)CCC(=O)N(C)C1 CC1C(NC(c2cccc(S(C)=O)c2)=O)C(C)CCN1C(c1cnn[nH]1)=O N1(C(c2c(O)ccc(C)c2)=O)CCC(N2CCCC(Cn3cc(Br)cn3)C2)C2(CC2)C1 CC1CN(C(=O)Cc2nccn2C)C1C(=O)NC(C1CCCCC1)C C1(CNC(C2ON=C(C)C2)=O)(CO)CC12CCN(C(c1sccc1F)=O)CC2 N1(C(C2(O)C(C)(C)C2)=O)CC(C2CCCCN(C(c3ccc(C4CC4)s3)=O)C2)C1 N1(C(c2c(O)cncc2F)=O)CC=C(c2ccnc(Cl)c2F)CC1 N1(S(C(C)C)(=O)=O)CCOC2(CCCN(C(c3cc(Br)cc(F)c3C)=O)C2)C1 CCC(CC(=O)NC(C)C(=O)NCC(C)(F)F)OC C1(C(N2C(C)CN(C(C3(O)CCOCC3)=O)CC2)=O)CC2CSCC(C1)C2 C1(C(N2CCC(N(C(=O)C=CCO)CCO)C2)=O)CCc2nnc(C(F)(F)F)n2C1 c1(C2C(C(=O)NC3C(NC(C=C(C)Cl)=O)CC3)C2)cnn(C(C)C)c1 c12cn(nn1)C(C)C(=O)N2.C(C)(C(C)(C)C)N(CC(=O)OC)C1CC1 C1(CNC(CCS(C)=O)=O)CN(C(=O)CC(F)(F)Cl)C2(CCC2)C1 Cc1ncc(CNC(=O)C(CC2CCOCC2)NC(=O)Cc2nonc2C)[nH]1 N1(C(C(N2C(C(=O)O)(Cc3c(C)cccc3)SCC2)C)=O)CCS(=N)(=O)C(C)C1 N1(C(C=CCC)=O)CCC2(CC1)CN(c1ccnc(C(=O)OC)n1)CCO2 N1(C(c2c(SC)cn(C)n2)=O)CCCC(NC(=O)CC2CCOC(C)(C)C2)CC1 N1(C(Cc2cnc(C)s2)=O)CCC2CCC12CNC(=O)C#CC(C)(C)C c1(C(N2CC3CCN(C(=O)CCC(F)F)C3C2)=O)cc(Cl)c(F)cc1F CCC(C)C(C(=O)N1CCCOC(CNC(c2cc(C)c(C)[nH]2)=O)C1)OC N1(C(c2c(CCC)n(C)nn2)=O)CC(NC(=O)CN2CCSCC2)C(C2CC2)C1 c1(OC)cnc(Cl)cc1C(N1CCC(N(C(=O)CCC(F)(F)F)C)C1)=O CC#CCCC(=O)NC(C)CC1CCN(C(C2(c3cc(C)no3)CC2)=O)CC1 CC(C)C(CCC(=O)NOCC(O)CO)NC(C1CCCCC1O)=O CCC(C(=O)N1CCCC1CNC(=O)C(C)=C1CCC1)SC N1(C(CC(C)(C)SC)=O)CC2CC(C1)N2C(C1CC1C(F)F)=O c1(C(N2CCC(C)C(N(C(=O)Cc3cncnc3)C)C2)=O)cc(F)c(O)c(F)c1 c1(C(N(CC(O)CF)CC)=O)ccc(CNC(C2CC(=O)N(C)C2)=O)cn1 Cn1ncc([N+](=O)[O-])c1N1CCC(NC(=O)C=Cc2ccsc2)C(CO)CC1 C1(NC(C2C(OCC)C2)=O)COC2(CCN(C(=O)C=Cc3cnc[nH]3)CC2)C1 n1(CC)[nH]cnc1=NC(=O)C(=O)NCC1=NOCC1 N1(C(c2nc(C)n(C)n2)=O)CC2(CCN(C(C3CCCNC3=O)=O)CC2)CC1C C(=O)(C1=CS(=O)(=O)CCC1)N1C(C)CCC(NC(=O)C=Cc2ccc[nH]2)C1 C1(CC)CC(CC(=O)N(CC(C)(C)CNC(=O)CC(=O)N(C)C)C)CCO1 N1(C(C2CC(n3cc(CNC(=O)NC)nn3)C2)=O)CCOC(C(C)(C)C)C1 CCC(C)(CO)C(=O)N1CC2CC2(CNC(=O)CNC(c2ncccc2O)=O)C1 N1(C(C(C=C)c2ccccc2)=O)CCCCCC(NC(=O)CCc2cscn2)C1 c1(SC)cccc(N(C(C)C(=O)NC2CN(C(C3CC(NC(C)=O)C3)=O)C2)C)c1 N1(C(CSc2ccc(C)cc2)=O)CC2=C(C1)CN(C(=O)CCc1cncnc1)C2 c1(CCC(=O)OC)ccc(F)c(CN2CCN(C(C)CN)CC2)c1 C1(NC(C2(CCNC(C3CCC(=O)C3)=O)CCC2)=O)CCC2(CCC2)C1 CC1=C(C(=O)NCC2(CNC(=O)C(O)C3CC3)CCC2)Cn2nnnc2N1C c1(C(N2CCC(NC(c3c(C)cc(F)cc3)=O)C2)=O)cnn2c(C)cccc12 C(=O)(C1CCCc2nc(C)[nH]c21)NCC(C)(CO)NC(c1cncc(C)c1)=O c1(CN2CCC(C)(C(N3CCS(=O)CC3)=O)C2)cc([N+](=O)[O-])ccc1Br c1(SCC)ccc(C(N2CCCC2C2(c3ccc(C(=O)NC)cc3)CC2)=O)cn1 CN1Cc2ccc(C(N3CCC(CNC(c4ncc[nH]4)=O)C3(C)C)=O)cc2C1 c1(C(=O)NCCC2(O)CCN(C(CN=S(C)(C)=O)=O)C2)scc2c1OCCO2 N1(C(C(CCC)OC)=O)C2CCC1CC(F)(CNC(C1(C(=O)NC)CCC1)=O)C2 N1(C(c2c(C)cccc2Cl)=O)CCC2(CCC(NC(=O)CC34CCCC3C4)C2)C1 Cc1ccn(C(C)C(=O)N(C(C)CN(C(=O)CN(C)C(N)=O)C)C)n1 c1(C2N(CC(=O)NC(C3CC(F)(F)C3)C)CCC2)ccc(C(F)(F)F)cc1 c1(NC(Cc2cn(CC(CC(C)C)OC)nn2)=O)ncc2nccnc2n1 Cc1cc(C(N2CCOCC2CN(C(=O)Cn2cncn2)C)=O)c2n[nH]cc2c1 C1(NC(CCSC)=O)Cc2ccccc2C1NC(c1ccc([N+](=O)[O-])cc1F)=O CC(=O)CCCC(C)C(=O)NC1CN(C(c2cc(CO)oc2C)=O)CC12CC2 c1(C(N2CCC(C(=O)Nc3ncccc3F)C2)=O)cc2c3c(ccc2[nH]1)NCC3 C1(C(=O)NC(C(O)CO)C2CC2)CC(O)CN1C(=O)CCc1cncnc1 N1(c2ccnc(NC(c3csnn3)C)n2)CCC(C)(C2CC2)C1 C1(NC(=O)Cn2cnnc2O)CCCC2CN(C(c3ccc(F)nc3F)=O)CC12 c1(C(=O)NCC2CCN(C(C(N3C(CC)CCC3)=O)=O)CC2)cc2scnc2[nH]1 c1(C(N2C(CC(=O)NC(C#C)C(C)OC)CCC2)=O)cccc(CC)c1 C1(CN(C(=O)CN(S(C)(=O)=O)C)C)CC(F)CN1C(C12CCC1C2)=O C(CCCC(=O)N1CC(N(C(=O)C(C)CCOC)C)C1)OCCC=C c1(C(=O)NCC(CNC(c2c(CCC)nco2)=O)O)cncc(OC(C)C)c1 N1(C(c2c(OC)cccc2I)=O)C2CCCC1CC(NC(C1CCCOC1)=O)C2 c1(OCC)ccc(C(N2CCC(F)(CNC(=O)CNC(=O)OC)C2)=O)cn1 C(=O)(CC(=O)NCC(C)N(C)C(c1cnn(C2CC2)c1)=O)OC c12ccc(cc1)S(=O)(=O)N2.C1(N(C)CCO)CCN(CC2CNC2)CC1.C1C(=O)N1 C(=O)(C1=CCCCN1C(=O)OC(C)(C)C)N1CC(N(CC(F)(F)F)C(C)=O)C(C)C1 c1(NCC(C)(C2CC2)OC)ccc2c(C)[nH]nc2c1 C(C1=CCN(C(=O)C(c2ccccn2)O)CC1)NC(C=C(C)Cl)=O C(=O)(C(O)P(C)(C)=O)NC1CC(NC(c2cc(NC(C)=O)ncn2)=O)C1 c1(CC(=O)NCC2CC(F)(CNC(CN(C)CC)=O)C2)ccc(C)cc1 N1(C(C(C)(C)c2cc[nH]n2)=O)CC2CC2(NC(c2cncc(C(F)(F)F)c2)=O)C1 C1(NC(C2CCCN(C(C(CO)OC)=O)C2)=O)CC12CCOCC2 C1(NC(C2CCN(C(C)C)CC2)CC)CCCC(C)(C)C1 C#CC1CCCN(C(C2CCN2C(=O)CN(C)CCOC(C)=O)=O)C1 CC(CNC(=O)Cc1ccc[nH]1)C(F)C(=O)NC1CN2CCCC1C2 N1(C(COCP(C)(C)=O)=O)CCOCC(NC(=O)C(c2cccnc2)O)C1 C1(C(N2CCCC(C)C2CCO)=O)(OC)CCN(C(=O)CCc2ccoc2)CC1 Cc1cc(CC(=O)NC2CN(C(=O)Cc3nocc3C(C)C)C2)sn1 C1(CC)CC(C(=O)N(CC(=O)N(CC(C2CC2)OC)C)CC2CC2)CCO1 c1(C(C(=O)NCCC(=O)OCC)N(C(C)CCC(C)C)C)nn(C)nc1Br c1(CC(N2CCCC(C(=O)NC3CCN(CC=C)CC3)C2)=O)c(Cl)cccc1Cl C1(CNC(C2CCN(CC)C2)=O)CC2(C1)CN(C(=O)COc1ccon1)C2 C12(C(N(CCN(C(C(CC)COC)=O)C)C)=O)CCC(C(F)F)(CC1)CC2 CCCC(CCC)C(=O)N1CCCC1C(C)NC(=O)COCc1nc(C)no1 C1(C(N2CCC(C(CNC(CCSC)=O)O)CC2)=O)C2Cc3ccccc3C12 c1(OC)cccc(CCCn2nnnc2C2(NCCF)CCC3CC23)c1 c1(CC)ccc(F)c(C(=O)NCC2(C)CCN(C(C3CC4CCC3O4)=O)C2)c1 Cn1ncc(C#N)c1NC(C1CC(O)CCN1C(c1ccc(Cl)cc1F)=O)=O N1(C(c2cncc(OCC)c2)=O)CCC2(CC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 c1(CN2CC(C)(CC(=O)Nc3c(C(=O)OC)ccs3)C2)nc(Cl)ccc1F c1(NCCN(CC)CC)cc(=NC(C)c2ccc[nH]2)[nH]c(C(C)C)n1 c1(Cc2nnc(-c3ccc(OC)cc3OC)o2)cn2cc(Cl)cc(Cl)c2n1 N1(C(C2C(CNC(c3ccc(O)nc3)=O)CC2)=O)CCC2CCCC2CC1 N1(CC(N2CC(CC(F)C(=O)NCc3ccc(O)cc3)C2)=O)C(=O)CCCC1=O CC1(C)CC(=O)N(CC(=O)NCCNC(C2(C3CCCO3)CCCO2)=O)C1=O c1(C(N(C2C(C)(C(=O)O)CCC2)C(=O)CCN2CCC2)=O)cc(Br)cnc1O c1(Oc2c(CNC(CC(C)C3CC3)=O)cccc2)ccc(Cl)cc1Br C12(CNC(C3(C)COC3)=O)CCC(CNC(=O)C#CC(C)(C)C)(CC1)CO2 C=CC(C)(O)CC(=O)N1CCC(C(C)(C)NC(=O)CCc2ccc(C)c(C)c2)C1 C1(CN(C)C(C2(C(F)F)CC2)=O)COCCN1C(=O)C(O)C1CC1 C(CC(=O)NCC1(F)CCOCC1)(C(F)(F)F)NC(C(COC)C)=O C#Cc1ccccc1CC(=O)NC(C)(C)CCN(C(=O)CCCC#CC)C CC(C(=O)NCC1(NC(C2CSC2)=O)CCOC1)C(=O)N1CCOCC1 C1(NC(c2cc(CNC(C3CCCC3)=O)oc2)=O)CC2CC1OC(=O)N2 CC(O)C(C)(C)C(=O)NCCC(C)NC(C1CCN(C)C1)=O Cc1ccc(Cl)c(N)c1C(=O)NC1CC1CNC(C12CC(C(F)(F)F)(CO1)C2)=O C1(NC(c2csc(Cl)c2)=O)CCOCC1NC(C1CC(F)(F)C1)=O c1(CNC(C2C(C)CCCC2)=O)ccc(C#N)cc1F.C12CC(C)(C)CN1C2=O N1(C(CNS(C)(=O)=O)=O)CC2ON=C(CNC(c3ccc(C(N)=O)cn3)=O)C2C1 CCC(C(=O)NN(C(=O)NC(=O)OC(C)(C)C)S(C)(=O)=O)C1CCOC1 C(=O)(C1c2ccccc2C2CC1C2)NC1CC(NC(C(CC=C)CC)=O)C1 C(=O)(C1(C)CCCc2ccccc21)N(C)C.C12CC3CCCC(C1)N3C2=O c1(C(=O)NCCN(C(C)C)C(c2cccc(N)c2F)=O)ccc(F)cc1F C1(NC(CSC(=N)N)=O)COC2(C1)CN(C(c1cc(C(F)(F)F)on1)=O)C2 C1(NC(=O)NC2(c3cccc(Cl)c3)CCC2)CC2C(C1)C2(F)F c1(C(=O)NC2C(C)CCN(C(c3c(C(C)C)ncs3)=O)C2)n[nH]c2ccccc12 CC1CCN(C(C2CCSC2)=O)CCN1C(c1ccc(CO)c(F)c1)=O C1(NC(C=C(COC)C)=O)CC2C1CCN2C(c1nnn(-c2ccccc2)n1)=O Cc1cc(C(=O)NCC2CCN(C(=O)CCc3ccoc3)C(C)C2)cc(N)c1O N1(C(c2c(N)nccn2)=O)CCC2CN(C(=O)CC3CS(=O)(=O)C3)CC12 CC1C2C(CCN2C(=O)C2=CCCC2)CN1C(=O)CC1(O)CCCCC1 C1(CCC)(NC(=O)COC)CCCN(C(c2cc(C)ccc2-n2cncn2)=O)C1 c1(C(=O)NCC(CNC(Cc2nc(C)sc2)=O)CO)nnc2n1CCCCC2 C(CC1=CCCCCC1)NC(C1N(C(CCCOC)=O)CCC(C)C1)=O C1(C(C)NC(C2(O)CCC2)=O)CCN(C(=O)Cc2ccccc2)C1 c1(C(=O)NC2CN(C(C(=CC3CCCC3)C)=O)C2)ccc(Br)cc1O C12CCCC3CN(CC13)C(=O)N2.CC(CCC1CC1)NC(=O)OC(C)(C)C c1(C(N2CCC(C(=O)NCC3CN(CC)C(=O)O3)(CF)C2)=O)cncc(F)c1C c1(NCC2CC(C)(COC)C2)ncnc2onc(C)c12 CCC(C(=O)NC1CC(NC(c2c(Br)ccc(F)c2F)=O)C1)C(C)(F)F C(=O)(C(CC(C)=O)NC(=O)C(C)CN1CCCC(C=O)C1)OC.c1(C)ccccc1 N1(C(CCC(=C)Cl)=O)CCCC(NC(=O)C(O)Cn2cncn2)CC1 c1(C(C)=O)cc(=NCc2ccccc2CNC(C2CCc3nncn3C2)=O)[nH]cn1 c1(CCN2CC(=O)N(CCc3nnn(C)n3)C2=O)nc2cc(F)c(F)cc2[nH]1 Cc1ccccc1C(C)C(=O)NCC1COCCN1C(C1CC1(C)C)=O Cc1nncc(CNC(C2CN(C(C3(C)CCCOC3)=O)CC2(F)F)=O)c1C C1(C(N(C2CN(C(=O)C(F)=C3CCC3)C2)C)=O)CCC(=O)N2CCCC12 C1(C(=O)NC2CC(O)C2)CN(C(c2ccc(Br)cn2)=O)Cc2cccn2C1 Cc1cc(-c2cn(CC3CCCN3C(=O)CCOC(C)C)nn2)sc1C N1(C(=O)OC(C)(C)C)CCC2(CCC(C(N3CCC(C)(NC(=O)C4CC4)C3)=O)C2)C1 Cc1nnn(NC(=O)CC2CN(C(=O)CCN3CCOC3=O)CC23CC3)c1C CC1(C)CCC(=CC(=O)NCCC2CN(C(C3(Cl)CC34CCC4)=O)CCO2)CC1 c1(OCCC)ccccc1NCC(O)CNC(=O)C1CC1.C1(=O)C(C)(C)CN1 c1(-n2c(-c3nc(OC)ccc3Cl)nc(CCCCC)n2)cc(Cl)ccc1OC c1(C(=O)NCC2(C)OCCN(C(Cc3cn(C)nc3)=O)C2)cnc2[nH]nnc2c1 CC1=C(C(=O)NCC2CCCN(C(=O)CCc3ccoc3)C2)CCCC1 c1(C(=O)NCCCC(C)NC(c2c(OC)n[nH]c2)=O)nn(C)nc1C C1(C(=O)OCC)(CO)CN(N2CC(CO)C(C)(COC)C2)C1 C1(C(=O)NCC(=C)C)CCC2(CN(C(c3cc(F)c(Cl)cc3C)=O)C2)O1 c1(C(=O)NC2C(CNC(Cc3cc(C)ns3)=O)C2)c(C)cc[nH]c1=N CC(CC(N)=O)C(=O)N1CC2(CCN2C(=O)C(O)CC(=O)c2ccccc2)C1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(CC(C)NC(C(C(CC)C)OC)=O)C1 Cc1ccc(C(c2nnnn2C2COC2)NC2CC(=O)N(O)C2)c(C)c1C N1(C(=O)OC(C)(C)C)CCCC12CCCN(c1ccc([N+](=O)[O-])cc1C#N)C2 Cc1cc(C#N)ccc1NC(c1cnn(-c2ccccn2)c1C)=O N#Cc1cc(C(=O)NCC2CCN(C(c3cc(F)c[nH]3)=O)CC2)ccc1[N+](=O)[O-] c1(C(=O)NCC2CN(C(CC=CCC)=O)C(C)C2)cn(C)c2ncccc12 c1(C(N2CC(NC(C(CN(CC)CC)F)=O)(CO)C2)=O)cc2ncccc2o1 CC1(CCNC(C2(F)CC2)=O)CCN(C(c2cccc(O)c2F)=O)CC1 C1(C(C)(C)C)C(NC(C2CCC(C)(C)C2)=O)CCN1C(=O)CNc1ncccn1 Cc1nc(C(=O)NCCn2cc(CCc3ncccc3F)nn2)c(C)o1 c1(C(=O)NCC2CC(NC(C(C)N(CC(F)(F)F)C)=O)C2)c[nH]nc1C(C)(F)F c1(C(N2CCN(CCCNC(C)=O)CC2)=O)c(C)nc2ccc(N(C)C)nn12 c1(NC(N2CC(CC)(CO)C2)=O)ccccc1OC(c1ccc(Cl)cc1)C(C)C N1(C(c2oc(C)c(Br)c2)=O)C2CCC1CC(CNC(C1CC1(C)C)=O)C2 C1(NC(CCOCCOCC)=O)CCC(CNC(=O)C=CC2CCCO2)CC1 Cc1nc(Cl)[nH]c(=NC(C)C2CN(C(c3cccc(OC(F)F)c3)=O)C2)c1F C1(C(N2CCC(CNC(=O)CC3OCCCO3)C2)=O)(OC)CC(CF)C1 c1(OC)nc(N(CC(O)CN(C2(C)CC2)C)C)nc2[nH]cnc12 c1(C(C)(C)C)cc(C(=O)NCCC2(NC(C3(C)CCCO3)=O)CC2)no1 N1(C(C(F)=CC)=O)CCC(CNC(c2nc(-c3cccs3)oc2C)=O)CC1 C=CCC(C(=O)N1CC=CC1C(=O)NC1CCOC(C2CC2)C1)NC(C)=O C1(NC(c2cnnc(O)c2)=O)COC2(C1)CN(C(=O)Cc1cscn1)C2 C12(CNC(C(CC=C)(F)F)=O)CCCCC1CN(C(c1cc(OC)n[nH]1)=O)C2 C1(C(=O)Nc2c(CC)nn(C)c2)C(C)OCCN1C(=O)C(N1CCOC1=O)C c1(C2CCN(C(c3ccc(-c4ccc(F)cc4)nn3)=O)C2)ccnc(Br)c1 c1(C(=O)NC(C)CN(c2nc(-c3ccccc3)ns2)C)coc(C2CCC2)n1 C(=O)(C(F)C(C)(C)O)N1C(CCNC(c2c(C)oc(C(F)(F)F)n2)=O)CCCC1 c1(C(N2C(C3(NC(CCCOC)=O)CC3)CCC2)=O)cccc2c1NCC(C)C2 Cc1nc(O)sc1C(=O)NCC(C)NC(=O)C(C)CN(C)C C(=O)(C1Cc2ccccc21)NCC(C(=O)NCC1CCN(C(CC)=O)C1)O C1(C(N(CCOC)CC)=O)CCCCCN1C(c1cnncc1OC)=O C1(CC(=O)NC2CC(C(C)C)OC2)CCN(C(=O)CN2CC3CC3C2)C1(C)C N1(C(C(C2CCOC2)NC(=O)CC2CCCC2)=O)CCCC2(CC2)C1 c1(C(=O)NC(CSC)(C)C(=O)N(C)CCOCCCO)ccc(C)c(O)c1 C1(CNC(C(C=C=C)C)=O)CN(C(c2ccnc(CC(C)C)n2)=O)CCC1(F)F C1(NC(=O)C=Cc2ncc[nH]2)CC2CCC(C1)N2C(c1ccc(F)c(Cl)c1)=O N1(C(c2ccc3nc(C)sc3c2)=O)CCC(N=c2[nH]c(C(C)C)ncc2Br)C(C)C1 C(=O)(Nn1ccccc1=O)C1(NC(C2CC(C)OC2C)=O)CCCC1 CC(O)CCC(=O)N1CC(C)CC1C(=O)Nc1ccnnc1O c1(CN2CCC(CC(=O)Nc3c(C)c(Br)ncc3)C2)ccc2c(c1)OC(F)(F)O2 N1(C(C)=O)CCCC1CC(=O)N(C(C)CNC(C1OCCCO1)=O)C N=c1[nH]cnc2c1CN(c1nc(N3CCC(CCO)C3)c3c(n1)COC3)CC2 c1(CC(=O)Nc2cccc(NC(C(CCCC)O)=O)c2)ccc2c(c1)CCCS2 N1(C(CC(C)F)=O)C2CCC1CC(CNC(c1ccc(Cl)cc1C(F)(F)F)=O)C2 C1(NC(C2N(C(Cc3c(C)n[nH]c3)=O)CC=CC2)=O)COC2(CCCC2)C1 C(CCC(O)C(=O)NC1(CSC)CCCC1C)NC(CCSCCCC)=O C(=O)(C(CO)C(C)(C)C)N1CCC(NC(COCCCCCC)=O)C1 C(C(CC1CC1)C(=O)N1CCC(N(C)C)C1)NC(c1cnc(CC)o1)=O C1(CC)(NC(c2cnc(OC(C)C)cn2)=O)CCCN(C(c2occc2C)=O)C1 CC1(C)CN(C(c2cccc(Br)c2F)=O)CC1NC(c1ccncc1N)=O C(=O)(C(C)(C)C(=O)NC1(CNC(C2(OC)CCSC2)=O)CCCCC1)OC CC1(C)CN(C(C2CC3CCC3C2)=O)CC1CNC(c1ccnc(C(N)=O)c1)=O c1(C(N(CCCCNC(=O)COC2CC=CC2)C)=O)ncccc1N(C)C C1(OC)CCC(C(N2CCC(F)(CO)C2)=O)CC1.C12(CC1)C(=O)N2 c1(CCC(=O)N(C)CCNC(C2(F)CC(C(=O)OC(C)(C)C)C2)=O)ncccc1F c1(OC)ccc(Br)nc1CNC1C=CC(C(=O)NCCOC(F)(F)F)C1 c1(C(N2C3CC(NC(C(C)=C4CCC4)=O)(C3)C2)=O)ccc(Br)cc1Cl CC(CC#C)(C(=O)N1CCCc2ccnn21)NC(=O)Cc1ccc[nH]1 N1(C(c2ccc3n[nH]cc3n2)=O)CCC2CN(C(C3(CF)COC3)=O)CC2CC1 N(C1CCCc2ccc(F)cc21)C(c1cc(CC)on1)c1nnnn1CCSC CC1(C)C(NC(=O)CCc2cc(F)c(F)c(F)c2)C(C)(C)C1O Cc1cc(C(=O)N(C2CCC3CC23)C)c(O)c(C)n1 C1(O)(CCNC(=O)Cc2nc[nH]n2)CCN(C(=O)CC2CC(=O)NC2=O)CC1 N1(C(c2ccn(CCCC)n2)=O)CC(C)N(C(=O)CCN2CCOCC2)CC1C C1(C(N(CC=CC(=O)N(C)Cc2ccn(CC)n2)C)=O)CC(=O)CC(=O)C1 c1(CNC(C2(CC)COC2)=O)ccnc(C(=O)NOC2CCC(O)C2O)c1 N1(C(CC(=O)OCC)=O)CCN(C(c2cc3sc(CC)cc3s2)=O)CCC1C C1(CC(=O)OC(C2CC(OCC)C2)=O)CCC2CN(C(=O)OC(C)(C)C)CC12 C#CCC(C)C(=O)NCC1C(C)CCN1C(=O)CN(S(C)(=O)=O)C c1(C(=O)NC(C2N(C(CC(CCC)C)=O)CCC2)(C)C)cc2ccccn2c1 c1(OC)ccc2c(c1)N1CCN2Cc2ncc(s2)C1=O.C(CN)SC c1(C(=O)NCC(C)N(C(=O)C(O)C(F)F)C)ccc2c(c1)CCCC(=O)N2 c1(OC)ccc2ccccc2c1CN1CCC1C(=O)NCc1cn[nH]c1 C(C1=Cc2ccccc2OC1)NC1C(SCc2c(F)cccc2)CC1 C(=O)(C(CCNC(c1cc(CO)oc1C)=O)OC)NC(C1CCCOC1)CC N1(CCS(N)(=O)=O)CCC(NC(=O)NC(CC(=O)O)c2ccccc2)CC1 CCCCC(C)C(=O)NCC1(CCNC(C2CCC(N(C)C)C2)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)NC1CCC(CNC(=O)CC2CCNC2=O)C1 Cc1[nH]nc2c(C(N3CCCC(C(N4CCOC(C(=O)O)C4)=O)C3)=O)cccc12 C1(NC(CN(C(c2ccc(Cl)cc2)C(=O)NC(CC)C)C)=O)CC(N=[N+]=[N-])C1 C1(C(=O)NC(CC(C)C)C(=O)NC)(NC(C(C=C)CC)=O)CCC(C)(C)C1 N1(C(C23N(C(=O)OC(C)(C)C)C(CC2)CC3)=O)CC(C2CCCCC2)C1 c1(N2C(C(C)O)CC2)nc(=N)c2ncc(Br)n2[nH]1 C=CCC(C)(CNC(=O)C(c1ccoc1)NC(=O)C(F)n1ccnc1)CO N1(C(c2c(C)scc2)=O)CCC(OCCNC(=O)CC23CCCC2C3)CC1 N1(CCC)CCCC(C(=O)NCC2CC(F)CN2C(c2cn(C3CC3)nn2)=O)C1 C(=O)(CC(C)CNC(C1(C)CC1(C)C)=O)NCCN1CC(OC)C1 N1(C(COCCOCC)=O)CC(N(C)C(C2CC3CCC2CC3)=O)C(C)(C)C1 C1(C(N2CC(CNC(CN(CCCCCC)C)=O)C2)=O)CC(C(C)=NO)C1(C)C C1(C)(CNC(c2c[nH]c(=NC)s2)=O)CN(C(C2(C)C=CCCC2)=O)CC1C Cc1nc(NC2C(C)CCC(C)(C)C2)c2cc(C)sc2n1 C1(NC(c2ccc(SC)s2)=O)(CO)CCN(C(c2nc(C)ccc2C)=O)CC1 c1(C(N2C(=O)NC(CC(C)C)C2=O)C)ccccc1[N+](=O)[O-] c1(C(=O)NCCCN(C(=O)Cc2ccc(C)cc2)CC)nn(C(C)(C)C)cc1Cl c1(C(N2CC(NC(c3sccc3Cl)=O)C(O)C2)=O)cc(F)c(F)cc1Cl C1(NC(c2ccccc2Cl)c2n(CCC)nnn2)CCCCC12CC2 N1(C(CN(c2ccccc2CO)C)=O)CCCC2(C1)CN(C(c1cc[nH]c1)=O)C2 c1(C(N(CC(C)(C)NC(C(=O)NCCOC)=O)C)=O)cc(Cl)c(OC)c(Cl)n1 c1(C(N2CCC(N(C(=O)CCn3cnnn3)C)CC2)=O)cc(F)c(CO)c(F)c1 N1(C(c2sc(C)c(O)n2)=O)CC(NC(=O)C(O)C2CCCC2)C2CCCC12 N1(C(c2cccc(CC=C)c2)=O)CC2CCN(C(c3cc(C)c(Cl)s3)=O)C2C1 Cn1cc2c(n1)CCCC2C(=O)NCC1(C)CCN(C(c2ncc(F)cn2)=O)C1 C(C(F)(C(=O)NC(C)(C)CCCO)C(C)C)NC(CCNC(=O)OCC)=O c1(C(N(CC(CO)(CO)NC(Cc2c(C)non2)=O)C)=O)cccc2ncsc12 N1(C(C2N(C(=O)NC)CCC2)=O)CCCCCCC1C(=O)NC1CCNC(=O)C1 N1(C(c2c(OC)scc2)=O)CCCC(C2(NC(C3COC4COCC34)=O)CC2)C1 C1(CC)CCCCCCN1C(=O)CNC(C1CC(=O)C12CCC2)=O N1(C(CC(C)c2ccco2)=O)CCCOC(CCNC(=O)CC2CCN(C)C2)C1 N1(C(CCCOCCC)=O)CC(C(F)(F)F)CC1CNC(=O)C(CC)SC C1(CC(=O)N(C2CCN(C(c3cnco3)=O)CC2)CC#C)CCCS1(=O)=O C(=O)(C(CC)CC=C)NC(CCC=C)C(=O)NCCCCC(C)(F)F CCC(C(C)C)NC(=O)C#CCNC(c1cnc(C)o1)=O C1(N(CCNC)C(C2(C)CC2C(C)C)=O)CCNCC1 C1(C(=O)NC)CCCCN1C(=O)CSC1CCN(c2cccc(F)c2)C1=O C(=O)(C1=C(C)CCOC1)N(CCCN(C(CCC(=C)C)=O)C)CC CCCCCC(C)(C)C(=O)NC(C1CC=CCC1)C(=O)NCCc1cnn(C)c1 CCC(CC(=O)N(CC(O)CN(C(=O)CCn1ccnc1)C)C)C(C)(C)C c1(N(C(C(CC(=O)OC)CC2CC2)=O)C(C)C(=O)N2CCCC2)ccnnc1O Cc1ccc(C(=O)NCC(C)(C)CN(C)C(C2CS(=O)(=O)C2)=O)cc1Cl C(CCCCNC(C1CC(C)C1)=O)N(C(CCSCC)=O)C c1(C(=O)NC(CCNC(c2nn(C)c(Cl)c2)=O)(C)C)ccc(O)c(Cl)n1 N1(C(C2(COC)COC2)=O)CCC(C)C(NC(c2ccncc2C(F)F)=O)C1 C1(CC(=O)NCC(F)(F)F)(OC)CN(C(C2(c3ccccn3)CCC2)=O)C1 C12(C(C(F)(F)F)NC(C3CC3OCC3CC3)=O)CC3CC(CC(C3)C1)C2 c1(C(N2C(C(=O)Nc3cnc(C(N)=O)nc3)C(O)CC2)=O)cccc(F)c1F Cc1cc(NC(C2CC2)=O)ncc1-c1nc(C2CCC3CC3CC2)no1 N1(C(COCCCCC)=O)CC2CC2C1C(=O)N(C)CC1(COC)CCC1 C1(NC(c2cc(C(N)=O)oc2)=O)CC(=O)N(C2CN(C(C3CC3C(N)=O)=O)C2)C1 c1(CNC(=O)NC(CCOC)C)c(C)cccc1O N1(C(=O)NC(c2ncc(C)[nH]2)C(C)(C)C)CCOc2ncccc2C1 c1(C2C(C(=O)NC(CNC(CS(C(C)C)(=O)=O)=O)C)C2)ccnc2ccccc12 Cc1ccc(C)c(C(N2CC(CC(=O)NOCC(O)C(C)C)CC2C)=O)c1 C1(C(=O)NCCc2c(C)cnn2C)CCC(=O)N(C2CC2)C1 C1(C(=O)OC(C)(C)C)(CF)CCN(N2CCC3CCN(C)C3C2)C1 c1(OC)ccccc1C1CNCCN1Cc1noc(-c2ccccc2)n1 c1(CNC(c2ccncc2-c2ccc(CO)cc2F)=O)cccc(Cl)c1Cl c1(C(N2CCOCC(CNC(C3CC34CCCC4)=O)C2)=O)cc(Cl)cc(F)c1F c1(CCC)c(C(=O)NC(C)C(CO)NC(c2csc(C(C)(C)C)n2)=O)nnn1C C(CCCCC(=O)NCc1c[nH]nc1C(=O)NC1COCCC1(F)F)OCC CC1OCCC1CC(=O)NCc1cc(C(=O)NCCc2c[nH]nc2O)co1 c1(NCc2c(CC)nns2)ccc2ccccc2c1 C1(C(N2CC(OC)CC(CO)C2CO)=O)CCC2(CC1)CC(CN)C2 N1(C(C)C)CC2CC1CN2C(=O)CCC1CCN(C(C2CCOC(C)(C)C2)=O)C1 c1(CCOC)cc(Cl)cc(Cl)c1NC(c1cccc(F)c1-c1c(OC)cccc1)C N1(C(CCCNC(C)=O)=O)C2CCC1CN(C(C1COCC1C(F)F)=O)C2 C1(CNC(CCCN(C(C(C)CC2CC2)=O)C)=O)CCCOC1(C)C n1(CC(=O)NC(C)CC2CN(C(=O)CC3CCC3)C2)cnc(Br)c1 C1(NC(CC2C=CC(NC(c3cnn(C)c3C#N)=O)C2)=O)CC12CCCCCC2 n1(CC(N2CC(CCCCNC(CCOCCOC)=O)C2)=O)ccnc1C CCCC(C(=O)NCCC1(O)CN(C(c2ncsc2C2CC2)=O)C1)NC(N)=O C=C1CCN2C(C1)C2=O.N1(CCC(=O)NC)CCC(C)CC1 C1(NC(C(CC)Oc2ccccc2Cl)=O)CCN(C(=O)CC(C)C)CC1(F)F CC1(F)CCN(c2nnc(-c3cccc(Br)c3)n2CCN2CCCCC2)C1 c1(NC(c2n(C(CC)(C)C)nnn2)C2CN(CC(F)F)C2)ccc2nccn2c1 n12cc(nn1)C2.n1(NC(C2CC(N(C(C)=O)CC)C2)=O)cc(C)cn1.C1(=O)CCO1 C1(CNC(c2cncc(Cl)c2)=O)CC2CN(C(=O)C(F)n3cccn3)CC12 O=C(C1=CCSC1)NCC1(CNC(=O)CCc2ccoc2)CC1(F)F c1(CC)nnc(N2CC3C(CNC(=O)CN4C(C)CCC4C)C3C2)c(C#N)c1CC c1(CN(C)Cc2c(F)cc(Cl)cc2F)cccc2c[nH]nc12 N1(C(C2C(CCC)C2)=O)CCCC(C(=O)N(C)CCC)C1CC CCCCC(O)C(=O)NC1C2CC1N(C(C1CCN(C3CC3)CC1)=O)C2 c1(C(=O)NC(C2CCN(C(CSC)=O)C2)(C)C)cc(C(=O)OC)oc1C CCCC(O)C(=O)N1CCC(CN(C)C(c2ccc(-c3ncnn3C)cc2)=O)C1 CC1OC2(C(=O)NC3CN(C(=O)Cc4cnccn4)CC3C)CCC1CC2 C(CC(C)(C)CC(=O)NCc1cnc(OC)cn1)OC c12ccc(OC)c(c1)ON(C(C1C(C)(C(=O)OC)C1)=O)CCNC2=O.C1(C)CC1 CCCCCCC(CC)C(=O)NCC1CCN1C(C12CCC(CC1)C(C)O2)=O C1(NC(C(N2CCC(O)CC2)C)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1F C1(OC)CC(C(=O)NCC2CCC2NC(=O)COc2ccccn2)N(C(C)=O)C1 C1(NC(C(C(C)C)OC)=O)CCN(C(=O)C=Cc2cnn(C)c2)C12CCC2 c1(C(=O)NC2C(NC(C3N(C)C(=O)OC3)=O)CCC2)ccc([N+](=O)[O-])cc1F C=CCCCC(C)(C)C(=O)N1CC2CC2(CNC(c2oc(C(F)F)cc2C)=O)C1 CC1=C(C(=O)NCC2CC(C)CN(C(=O)CCC3CCCO3)C2)CCC1 C1(CC=C)(C(=O)NCC(=O)NOC)CCCN1C(=O)CCC1CCCCO1 c1(OC)c(Cl)nc[nH]c1=NCC1(NC(=O)COC(=O)C2CC2)CCCC1 c1(C(=O)NCC(CC)NC(=O)CCF)cc(OC)c(Cl)cc1Cl CCC(C)(COC)C(=O)NC1CC(O)CN(C(=O)C(C)(C)COC)C1 c1(OC)cccc2c1OCCC2OC(=O)CS.c1(CC#N)ccc(F)cc1 C1(NC(C(CC)O)=O)CN(C(=O)C(c2csc(C)n2)=O)CCC12CCC2 c1(C(C(=O)NCCC(C)N(C(=O)C(C)=C(C)C)C)OC)ccccc1SC c1(OC)nc(C(N2CCC(OCC(=O)N(CC(C3CCCC3)O)C)C2)=O)co1 CC1CC(C(=O)NCC2CCN(C(c3cnn(CCF)c3)=O)CC2O)CC(=O)N1 C1(CC(N2C(COC)CC2)=O)N(C(c2csnc2OC)=O)CC1(C)C N1(C(CCC=C)=O)CCC(C(=O)NCc2ccnc(F)c2)C(C)(C)C1 c1(C(=O)OC)cc(S(=O)(=O)NC2CCS(=O)(=O)C2)ccc1C c1(C(=O)NC2(C(=O)NCC#CCN(C)C)CCCO2)cccc(OC2CC2)n1 C(CC(C)(C)C)(C(=O)N1CC(C(=O)NCc2ncc(CO)o2)C2(CCC2)C1)OC N1(C(CC=C=C)=O)CC2CCN(C(c3scnc3C(C)C)=O)CCC2C1 C1(NC(c2cnc(OC)nc2)=O)CCN(C(=O)C(C)CSC)CC(C)(C)C1 CC(C(=O)O)C(C)(C)CC(=O)NC(C)CCNC(c1ccccn1)=O c1(C(N2CC(C(=O)Nc3cc(C)c(F)cc3)CC2(C)C)=O)cc2cccnn2c1 N1(c2ccn(C)n2)CCCCNC(=O)C(F)(F)C1.C1CCCCCC(=O)N1 C(=O)(C1=CCCCC1)N1CCC(C)(C(=O)NC(CCO)C(F)F)C1 CCC(C)CC(=O)C(=O)N1CCC1CC(N1CCCC(C)(C)C1)=O C#CC1CCN(C(C2COC(CNC(=O)C(O)C3CCCC3)C2)=O)C1 N1(C(C=CC(CC)C)=O)CC(C(F)(F)F)CC1CNC(=O)C(c1ccccc1)O C(=O)(CCC(C)=O)NCC1C(C(=O)NCC(COC)(F)F)OCC1 C#Cc1cnn(CC(N2CCC(C(=O)NC(C)Cc3cccs3)(CF)C2)=O)c1 C(=O)(C(C)(C)C(C)(C)O)NCC1N(C(Cc2c(C)cccc2Cl)=O)CCCCC1 c1(C(=O)NCC(C(C)C(C)C)NC(CCCSC)=O)c(C)ccc([N+](=O)[O-])c1C c1(OC)ccc(-c2cn(C3CCN(C(C4CC(O)C(F)C4)=O)C3)nn2)cc1Br c1(C(=O)NC(C2CCN(C(=O)Cc3sc(O)nc3O)C2)C)cncc(C2CC2)c1 c1(C(=O)NCC(CC=C)NC(c2cn(C)c(C)n2)=O)cccc2c1CCC2 c1(C(N2CC(NC(=O)OCC)C2)=O)cc(CNC(c2csc(Cl)c2)=O)ccn1 N1(C(CCCOC)=O)CCCOC(CCNC(=O)CC=Cc2ccccc2F)C1 C1(C(C)C)CCCN(C(=O)CCN(CCO)C(C2(Cl)CCC2)=O)CC1 c1(C(N2C(C(=O)NC(C#C)C)CC3CC32)=O)cc(Br)c(C)c(Br)c1 NS(=O)(=O)c1ccc(-c2csc(CNC(=O)COCC3CCCO3)c2)cc1 N1(C(=O)Nc2nn(CC)c(O)c2)CCC2(CC1)CC(NC(=O)OC(C)(C)C)C2 C(CCN(C)C(c1ccc(C)nc1O)=O)(C(C)(C)C)NC(CC(=C)C)=O c1(CC(=O)NC2C(C)CN(CCc3ccc(F)cc3)CC2)cccc2nsnc12 c1(C(=O)NCc2ccc(C(=O)OCC)cc2)n[nH]c2cc(OC)c(OC)cc12 Cc1nc(C)c(F)c(=NCC2C(C)CCCN2C(c2scnc2C)=O)[nH]1 C1(CC)CCOCCN1C(C1CC2C(C1)C2(F)F)C(=O)NC C1(CNC(CCCCCC)=O)(NC(=O)CC(C)CN(C)C)CCC(F)(F)CC1 C(CO)(CCCCNC(C1CCCC1)=O)NC(CCNC(C)=O)=O CN1CC=C(CC(=O)NCC2CCN(C(=O)CC3CCCC34CC4)CC2)CC1 CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC(C(=O)NC1CC(=O)NC(=O)C1)C2 C1(C(=O)N(CCCCNC(=O)CCC2CCCCO2)C)(COC)CC(=O)C1 Cc1cncc(C(=O)NCC2C(C)CCN2C(c2cnn(C(C)C)c2)=O)n1 C#CC1(C(=O)NCCCNC(C)=O)CCN(C(=O)COC(=N)O)C1 C12(C(N3CCCC3CCSc3ccccc3)=O)CCC(CC1)CC2.C12CCCN1C2 N1(C(CSCCC(C)C)=O)CCCC1CNC(C1(CCN(C)C)CCC1)=O C1(NC(C2(CC(C)C)CC2)=O)(CO)CCCN(C(=O)Cc2ccno2)C1 N1(C(CCC(=C)Cl)=O)CCCC2(NC(c3ccc(C4CC4)c(F)c3)=O)CC2C1 c1(C(NOCc2cn(CC3CC(C(C)C)OCC3)nn2)=O)c(Cl)nnc(Cl)c1O C(=O)(C1=NNC(=O)CC1)NCC1C2N(C(C3C4CC(C)(C4)OC3)=O)C(CC2)C1 Cc1ccc(-c2noc(C3CN(C(=O)OC(C)(C)C)C(C(F)(F)F)C3)n2)cc1F C1(NC(C(CC#C)C)=O)CC2CC(C1)N(C(C1(c3cccc(OC)c3)CC1)=O)C2 C#CCCCCCCNC(=O)C(C)CNC(=O)CC1(O)CCOCC1 CC1CCN(C(c2ccno2)=O)C1CNC(c1cc(Br)n[nH]1)=O C1(C(=O)OC)CC(CNCc2cccn2CF)N(S(C)(=O)=O)C1 N1(C(CC#C)=O)CCCCC1CCNC(c1cncc(Br)c1)=O c1(NC(c2n[nH]c(=N)s2)C)ncc(S(=O)(=O)NCCc2cccnc2)cc1Cl N1(C(C(C)CN(C)C)=O)CC2(CNC(c3ccc(CC4CC4)o3)=O)CCC1C2 c1(C(=O)NC2CCN(C(c3ccn(C(C)C)n3)=O)C2)n[nH]c2c1CCOC2 C=CCC(CNC(c1cnc(=N)[nH]c1)=O)C(=O)NC(C)(C)CCF c1(C(C)C(=O)NC2CC2NC(=O)CC2=NNC(=O)C2)ccc2ccccc2c1 N1(C(Cc2n(C)ccn2)=O)CC(O)CC1C(=O)NC1CN(C(N)=O)C1 C1(NC(C2(CC=C)CCCCC2)=O)CC(NC(C2(OC)CCCC2)=O)C12CCC2 C1(CNC(C=CCC)=O)CC(NC(c2ccn(CC)n2)=O)C(O)C1 c1(OC)c(C(=O)NCC(C2CC2)NC(c2ccc([N+](=O)[O-])o2)=O)cc(Cl)cc1C N1(C(CC2(OC)CC2)=O)CCCC2(C1)CN(C(=O)C(C)N=[N+]=[N-])C2 C=CCC(C)(C(=O)NC1(CNC(c2cc(OC)nc(Cl)c2)=O)CCC1)N(C)C N1(C(c2occ(C)c2C)=O)CCC2CC1CN(C(=O)CC(C)c1ccncc1)C2 C12(C(=O)NC(CCNC(c3cc(C(C)C)nn3C)=O)(C)C)CSCC1C2(F)F c1(C(=O)NC(CN(C(C(C=C)(F)F)=O)C)C)cncc2ccccc12 c1(C(=O)Nc2ccc(NC(c3cccc(C)n3)=O)cc2C)c(C)cc(O)cc1C Cn1cc(C(=O)NC2CCN(C(C3(C#N)CC3)=O)CC2)c(C(C)(C)C)n1 CCC(CCOC)C(=O)NC(C)(C)C(C)NC(c1csc(C(F)F)n1)=O C1(C=O)CC1C1CN(N(CCC(=O)OC)C2CC2)C1.C1(C=O)CC2CC(=O)C1C2 Cc1cccc(C2(CC3(C4CC4)CCCC3)CCC2)c1 c1(C(N(C(CNC(c2cc(C(C)C)n(C)n2)=O)C)C)=O)nn(C)c2c1CSCC2 C1(NC(C=Cc2c(C)ncs2)=O)COCCN(C(=O)C=CSCc2ccco2)C1 N1(C(C)=O)CCN(C(=O)Cc2cc(=O)n(-c3ccc(C)cc3)[nH]2)C2CCC12 CCC(CC)C(C)C(=O)N1CC2CC2(CNC(C2CC(n3ccnn3)C2)=O)C1 C12(CNC(C(CC)F)=O)CCCC1N(C(c1ccc(Br)c(F)c1)=O)CC2 C(=O)(C(CC(F)F)NC(c1nccnc1N)=O)NC(C#C)CC(C)C C(=O)(C(CC(=O)OC)NC(C)=O)N(C1CC(NC(COCCCC)=O)C1)C c1(OC)ccc(C(N2CC(C(C)NC(C3CC(OC)C3)=O)C2)=O)cn1 CC(F)(F)C(F)C(=O)N1CCCC1(C)CNC(=O)CCc1cn[nH]c1 C1(C(N(C(C)C(=O)N(C)CCn2cncn2)CCC)=O)CCN(C)C1 C(=O)(CCC1=CCCCC1)NCC(CCNC(C1(C)CCC(C)CC1)=O)O C1(CN(C(c2cnc(CC(C)C)[nH]2)=O)C)CCCN(C(=O)CC2CCNC2=O)C1 CCS(=O)CC(=O)NC1CCN(C(c2cccc(C(C)(F)F)c2)=O)C1C(C)(C)C N1(C(C2(F)CN(Cc3ccncc3Cl)C2)=O)CCc2nc[nH]c2C1 c1(C(=O)NCC(CC=C)NC(c2cc3ccccn3n2)=O)ccc2c[nH]nc2c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC2CCCN(C(=O)CN(C)C(C)=O)C2C1 c1(C(N2C(CCC)CN(C(C3(CO)CCCC3)=O)CC2)=O)ccc2occc2c1 c1(CC)nc(C(=O)N(C)CC2CCCCN2C(=O)CC(C)C2CC2)c(N)s1 c1(C(=O)NCC23N(C(C4(c5n(C)ccn5)CC4)=O)CC(C2)C3)cnc2n1CCC2 C1(CNC(C(CC)OCC)=O)(NC(=O)CCCSC(C)(C)C)CCCCC1C N1(C(c2c(C)ncn2C)=O)CCC(NC(=O)C=C2CCN(C)C2)C(CO)CC1 C1(C(N(C2CCN(C(CCc3c(C)nn(C)c3)=O)C2)C)=O)OCCN(C)C1=O c1(C(=O)NC(C2CCCN2C(C2CCC(=O)N2)=O)(C)C)cccn2ccnc12 C1(C(N(C2CCN(C(=O)C(C3(O)CCCC3)F)C2)CC)=O)CCCCN1C C(C(C)(C)C1=CCCC1)NC(C(Cc1ccoc1)NC(C(SC)SC)=O)=O C(C)(CO)(C(=O)N(CC(O)CN(C)C(C1CCC(F)(F)C1)=O)C)OC c1(C(C(=O)NCc2ccc(F)cc2)N(CC(CC)O)C)nc(Br)ccc1OC CC1OCCC1(C)C(N1CC(OCCNC(=O)Cc2ccnc(O)c2)C1)=O c1(N2C(CCCNC(c3cccc(F)c3F)=O)CCC2)ncnc2c1SCCC2 N#Cc1cn(CCC(=O)NCCCC2NC(=O)NC2=O)c(=O)nc1O N1(CCNC(CC(CC)C2CCC2)=O)CCCN(C(c2snc(O)c2Cl)=O)CC1 C(=O)(CCC(C)S(C)(=O)=O)NCC(C)(C)NC(CC(COC)C)=O Cc1cccc(C)c1N1CCN(C(=O)CC(O)C(C)C)CC1 N#Cc1cc([N+](=O)[O-])ccc1N1CCC(CN(C(=O)COC2CCOC2)CCO)C1 C12(NC(=O)CCSC(F)(F)F)CCCN(C(=O)Cc3cnoc3)CC1C2 CC1SCCC1(c1nnnn1CC1CC1)NCCCc1cccs1 CC1CC(O)CCN(C(C2CCCN(C(C3C4CN(C)CC34)=O)C2)=O)C1 C1(C(=O)NCCN(C(CCSCC(C)C)=O)CC(C)O)CCCC(O)C1 N1(C(C(CC)N(C)CC)=O)CCC(C2CCCCN2C(=O)CC2OCCO2)CC1 CC(=O)CCCC(=O)N(C1CCCN(C(c2cnc(C)nc2C(C)C)=O)CC1)C C1(C)(C(=O)NC2CCC(NC(c3c(C)c(=O)cc[nH]3)=O)CC2)CCC(F)(F)CC1 Cc1cc(C(N2CC(O)CC2(C)C(C)(C)C)=O)ccc1S(=O)(=O)C(C)C C1(NC(CCCCC)=O)CCCCCN(C(=O)CCc2ccncn2)C1 C1(NC(CCN(C)CC)=O)CCN(C(c2ccccc2C)=O)C12CCC2 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCc2ccc(C)cc2)=O)CC1C c1(OC)ccccc1C(C1CC1)NC(C1CC2(CCC2)C1)=O c1(NCC2(NC(C(CC(CC)C)C)=O)CCCCC2)nc2c(cc1C#N)CCC2 c1(C(=O)NCC(CNC(Cc2ccc(C)o2)=O)F)ccc2ncccn12 N1(C(C(C=C)C)=O)Cc2occ(C(=O)N(C(C)COC)C)c2C1 CCC(CC(=O)NCCCCCCNC(=O)CCCC(OC)OC)C(F)F N1(C(c2n(CC)ncc2)=O)CCC2(C=C(C(=O)NCc3cccc(OC)n3)C2)C1 CCC(CCOC)C(=O)NCC1CCN(C(=O)COc2cc(C)cc(C)c2)C1 CC1(C)CCC(NC(C2COCCC2NC(=O)Cc2cncs2)=O)C1 c1(NC(C2CCN(C(c3ccccc3F)=O)C2)=O)ccc2cc[nH]c2c1 C1(C(N2CCC(C)(NC(C(C)c3ccco3)=O)C2)=O)CCc2ncnn2C1 C1(CCC)CN(C(=O)C(C)CSC)CCN1C(c1[nH]nc(OC)c1Cl)=O c12cc(C#N)ccc1NC2.Cc1ccc(N2CCCCC2c2nncn2C)cc1 N1(C(c2ccc(=N)[nH]c2Cl)=O)CCC2(CC1)CN(C(C1CCCCC1F)=O)C2 c1(OC)nccc(C(=O)N(CC(C)CNC(=O)CNC(N)=O)C)c1Br c1(C(=O)NC(C)CCN(C)C(C2(C#N)CC23CCC3)=O)c(F)cccc1Cl C(=O)(C(C)(C)S(C)(=O)=O)NCC(CCOC)NC(C12CCC(CC1)O2)=O Cc1ccc(-c2cc(C(=O)NC3CC3CNC(=O)C3CC3)n[nH]2)c(C)c1 c1(C(C)C)cc(C(N2CCC(F)(CNC(=O)C(C)(C)N3CCCC3)C2)=O)nn1C c1(CC(=O)NCC2CC(NC(=O)C3=C(Cl)CC3)C(O)C2)ccc(C(F)F)c(F)c1 c1(CC(C(=O)NCC2C(CNC(C3CN(C)C3)=O)C2)O)ccccc1Cl C1(NC(CNS(N(C)C)(=O)=O)=O)CC2CC1N(C(=O)CC1CN3CCC1CC3)C2 c1(OC)c(C(N2C3COCC2C3NC(=O)CC2CCCCC2)=O)nc(O)nc1O C1(C(=O)NCC=C2CCN(C(=O)CC=C(Cl)Cl)CC2)(OC)CCC(C)C1 c1(C(C)NC(C2CCCN(CC(C)C(C)(F)F)CC2)=O)ccc(F)cc1Cl C1(NC2(c3n(C(C)C)nnn3)CC3CCC(C3)C2)CCCC2(CC1)CC2 CC1(C(=O)NCc2ncoc2C2CN(C(C34CCC3C4)=O)C2)C=CCC1 C#CCCCC(C)C(=O)N1CCN(C(c2occc2COC)=O)C(C)C1 N1(C(C(C)OCCC(C)C)=O)CCCN(C(C2CC3CCC2O3)=O)CC1 N1(C(CCN(C2CCCCC2)C)=O)CC2CCN(C(c3ccc(Cl)cn3)=O)C2C1 C(=O)(C(C#N)C(C)(C)C)N1C2CC(NC(c3cc(CC)no3)=O)C1CC2 c1(C(N2CCC(CN(C(C(c3ccccc3)C)=O)C)C2)=O)cccc(O)c1F C1(N(C)C)CCC(C(=O)NC2CCCC2(C)CNC(C2CCN2C2CC2)=O)CC1 c1(CC)ccc(C(=O)NC2CCC(CCNC(c3sccc3OC)=O)C2)c(F)c1 N1(C(C2N(C)C(=O)CC2)=O)Cc2ccccc2CC1CNC(=O)C=CI C1(CC(=O)NCCN(C(=O)OC)C)CCN(C(C2CC(=O)N(C)C2)=O)CC1 Cc1nn(C(C)(C)C)cc1C(N1CCC(NC(=O)C=Cc2cc[nH]n2)C1C)=O C(=O)(CCC(=O)NCC1CC(C)N(C(c2cc(COC)oc2C)=O)C1)NCC C(=O)(C1=C2CCCN=C2NN1)N(C)CC1CCN(C(C2CCCC(C)C2)=O)CC1 C(C)(C(C(=O)Nc1cnn(CCF)c1)C(C)C)NC(CCC)=O c1(C(C)C)ccccc1C(NC(=S)NC(c1ccccc1)C1CCOCC1)=O C1(N(C(=O)C(CC)N(C)C(c2cnc(Cl)s2)C)CC#C)CCN(C(C)=O)CC1 C12(NC(CCCC)=O)CCN(C(c3ncc(Br)cn3)=O)CC1C2 CCCCC(CC(=O)N1CCC(C)CC1)NC(c1[nH]nnc1CC)=O C(CC(=O)NC(C1CCN(C(=O)CCC2CCC(=O)N2)CC1)C)(C(F)(F)F)OC c1(-c2nc(C(C)O)nn2C2CCCOC2)ccc2ncn(C)c(=O)c2c1 C1(O)(CN(C(CN(C(COCCCC)=O)CCOC)=O)C)CCCCC1 C1(CCC#C)CCCCN1C(=O)CN(C(=O)CN1CCCC(O)C1)C c1(CC)nc(C)c(C(N2CCCC2(C)C(=O)N(CC)CC2(O)CCC2)=O)o1 O=C(C1=CS(=O)CCC1)N1CCC2CN(C(=O)CCC3CCCCC3)C2C1 C(CC(=O)N=c1ccn(C)[nH]1)C12CN1C2.C12(OC)CCCC1C2(F)F C(C(CC(=O)NCC1CC(NC(c2ccc3nn[nH]c3n2)=O)C1)C(F)F)N(C)C C1(C(N2C(C(=O)NC3(COC)CCOCC3)CCC2)=O)CC2C(C1)C2(F)F C1(CC)CCCCC1C(=O)NCCOCCOCCNC(c1n[nH]c(C)n1)=O C1(C#N)(C(=O)NC(CNC(c2cccc(OC)n2)=O)CCOC)CC2(CCC2)C1 CC1C(NC(C2(C)CCCCC2)=O)CCN1C(C1CCC1CF)=O C1(C(=O)NC(c2cccnc2)C(=O)NCCOCC(F)(F)F)CC2(CCC2O)C1 N#CC1CCN(C(=O)COC2CCN(C(=O)CC3CCC(=O)N3)C2)C1 N1(C(C2CCC(=O)NC2)=O)CC2CC(CNC(=O)Cc3ccc(O)cn3)C2C1 NC(=O)C(F)(F)CNC(=O)CNC(c1cn(CCO)nn1)=O C(=O)(C(F)CCC(C)(C)C)NC(c1nc(-c2noc3ccccc23)no1)C c1(C(=O)N)cc2c(C3CC3)cccc2[nH]1.C1(CC)CCN(C(c2coc(CO)c2)=O)C1 C1(CNC(C(CC)NC(N)=O)=O)CC2CCC(C1)N2C(=O)CC(C)(C)OC C1(C(N2C(CCC#C)CCC2)=O)C(C)CCN1C(=O)Cn1nnnc1CC N1(C(CC2C(CC)C2)=O)CCCN(C(C2(CF)CC2)=O)CC1 c1(C(C)(C)C)cnc(CCC(=O)NCC2(NC(C3CSCCS3)=O)CCOC2)o1 c1(OC)ccc(C(=O)NC(C)(C)CNC(C2CCC(NC(N)=O)C2)=O)nc1N c1(C(=O)NC2CC(CNC(C3C(CC)C3)=O)C2)cn(C)c(C)cc1=O N1(C(c2c(CC)cccc2)=O)CCC(C(=O)N(C2CCC(CC)CC2)C)C(C)C1 C1(CC)(NC(c2c(C(=O)OC)cnn2C)=O)CCN(C(c2cn(C)cn2)=O)CC1 C#CCCCC(C)C(=O)NCCCCCCN(C(=O)C=CC(C)(C)C)C C1(CC)CC2(CCN2C(=O)C(C)(CSC)NC(=O)C(F)C(C)(F)F)C1 Cc1cnc(Cl)c(S(=O)(=O)NC2CN(C(c3cc(Br)c(C)s3)=O)CC2F)c1 c1(CCC(=O)NC(CC)CNC(=O)C(CO)N(C)C)n[nH]c2c1CCCC2 CCCCCS(=O)(=O)CC(=O)N1CCCN(C(c2ccc(Cl)c(C)c2)=O)CCC1 CCC(C)(C)CCCC(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C Cn1ncc(C(N2CCOCC2CC(=O)NCC2=CCCCC2)=O)c1Cl c1(CNC(C2N(C(CCCC)=O)CSC2)=O)c(C)cnn1COC c1(C(=O)NC2CC(C(=O)Nc3ncc(F)cc3Cl)C2)c(Cl)cnc(Cl)c1Cl C(=O)(CCC(C)(C)C(=O)NC1CC1CNC(c1ccc2c(C)noc2n1)=O)OC CC1(C)CN(S(=O)(=O)COc2ccc(Br)cc2)CCC1CNc1ccccc1 CCC(C(=O)N1CCN(C(=O)CSCC(N)=O)CC12CC2)C(C)(F)F C(=O)(CC(C)(C)C(F)F)NCC(C1CCN(C(=O)Cc2ccsc2Cl)CC1)(C)O CC(C)C(C)(CNC(=O)OC(C)(C)C)NC(c1ncc(Br)cn1)C S(=O)(=O)(c1cccnc1NC1CCCCC1C(F)(F)F)NCC(CN(C)C)(C)C C1(c2n(CC)ccn2)CCCCN1C(c1conc1CC)C(=O)NC1(C)CC1 C(=O)(C(C(C)(C)O)NC(c1cnn2c1CCC2)=O)NC(c1nccs1)C N1(C(c2cccnc2C2CC2)=O)CCN(C(c2cc(F)n[nH]2)=O)C(C2CC2)C1 C(CC(C(=O)N(C1C2CN(C(C34COCC3C4)=O)CC12)C)NC=O)SC S(=O)(=O)(c1ccc(=NCC(O)c2ccnn2C)[nH]c1)N(CCN(C)C)CCO c1(C(=O)NCCNC(C2CC=CCC2)=O)ccnc2cc(F)cnc12 c1(OC)c(CC(=O)NCC(O)CCOC)cccc1F c1(C(C)C(=O)NC(C(=O)NCc2ccon2)C2CCC2)ccnn1C Cc1cn(C)nc1CN1CC(C)(O)C1.N12CCC(CC1)C(=O)N1CC2C1 Cc1cc(NC(=O)CCc2cnn(C)c2)ccc1NC(=O)CC1CCC1C C1(C(C)C)CC(C(=O)NOCC(O)C(F)(F)F)CCO1.C1C(=O)N1C(C)C C1(NC(=O)NCc2nccc(C(C)C)c2)CCc2nnc(C(F)F)n2C1 CC(CC(=O)NC1CCCC1CNC(c1cccnc1OCC(F)F)=O)C(F)F C(=O)(CCCCCCN=[N+]=[N-])NC1(C2N(C(C(CCC)OC)=O)CCCC2)CC1 N1(C(CNC(C(C)N(C(C)=O)C(C)C)=O)=O)CCN(C(=O)CSC(F)F)CC1 C1(C)(CNC(c2c(CC)oc(C)c2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CCO1 c1(C(C(=O)NC(CNC(C2CC=CCO2)=O)CO)(F)F)cccc(Cl)c1 N1(C(C2(CCNC(c3cccc(C)c3F)=O)CC2)=O)CCCCC(F)(F)C1 N1(C(CC(C)c2cccnc2)=O)CCCC(CNC(C2(CO)CCCO2)=O)CC1 c1(C(C(C)O)NC(=O)CCC2CCOC2)cccc(OCCN(C)C)c1 C1(CNC(C(CC)SC)=O)(NC(=O)C=Cc2cnn(C)c2)CCCCC1 C(=O)(N=c1cc(C2CC2)n(C)[nH]1)C1N(C(C(C)OCCC(C)C)=O)CC1 c1(C(=O)OC)c(Cl)nc[nH]c1=NCCC1CCCCN1C(=O)CC1CCOCC1 c12cnccc1NC1CCN(C1)C(=O)c1cc(n[nH]1)C(=O)N2.C(C)(C)(C)OC Cc1cccc(N)c1C(N1C2CCC1C(CNC(=O)CCF)C2)=O C1(NC(c2c(C)cns2)=O)CCOC(C(=O)NCCS(N)(=O)=O)C1 c1(CC)cc(NC(C2(CNC(=O)CN3CSCC3=O)CC23CCC3)=O)ccc1F C1(OC)CC(CNC(c2c[nH]nc2C(C)C)=O)N(C(=O)C(F)CC2CCCC2)C1 c1(C2CCN(c3ccnc(NCC4(C(C(C)C)O)CC4)n3)C2)cc(F)cc(Cl)c1 C(=O)(CS(=O)(=O)c1cccc2nsnc12)N1CC=CC(NC(C2CC2(F)F)=O)C1 C1(C)(C(=O)NC2C(NC(c3cc(COC)on3)=O)CCC2)CCNC(=O)C1 CCCC(CC)N=c1cc(C)[nH]c(=NCc2cc(C)cs2)[nH]1 C1(O)(CN(C(c2c(NC)cccc2)=O)C)CCCN(C(C2C=C(C)CS2)=O)C1 CCCCC(C)NC(C1CCN1C(c1cncnc1)=O)=O c1(C(=O)NC23CC(CNC(C(C(C)C)(C)O)=O)(OC2)C3)sccc1S(N)(=O)=O C1(C(N2CC(C(=O)NCC)C2)=O)CC2CCCC2N1C(=O)CON(CCO)CC Cc1ccc(C(C)C(=O)NC2CC(CNC(c3c(Br)noc3C)=O)C2)cc1 c1(CN(C(=O)CC2CCC3CC23)C(N)=O)nnnn1C1CC1.C12CCCN1C2=O c1(C(=O)NCC(CC(C)C)NC(C(CC=CC)C)=O)cc(C(C)C)n(C)c1C c1(CNC2C(C)CN(C(=O)C(c3cnn(C)c3)=O)C2)ccc(F)c(O)c1F CCC(C)CC(C)C(=O)N1CC(CC)(NC(=O)CN(c2ccc(Cl)cn2)C)C1 c1(CNc2cc(C)nnc2)cnn2cccc2c1 C1(OC)CCN(CC(=O)N(C)CCNC(c2csc(Br)n2)=O)C1 CC1CN(C(=O)C(F)(F)C(O)C2CC2)CCC1CNC(=O)CSC(C)(C)C C#CCCCC(C)C(=O)NC(CC(C)(C)C)C(=O)Nc1ccc[n+]([O-])c1 c1(OC)ccc(CN2CCC2(C)C(N2CCOC(C)C2)=O)cc1-c1ccccc1 c1(C(=O)NCC2CCC2NC(C2CCC(=O)N2C2CC2)=O)cccc2occc12 CC1CN(C(c2cnsc2)=O)CC(C)CN1C(=O)C(N1CCCCC1=O)C N1(C(C2COCCN(C(C(C(C)C)C)=O)C2)=O)CC2CCCCC12C N1(C(c2csc3ccccc23)=O)CC(CO)C2(C1)CN(C(C13COCC1C3)=O)C2 C1(CNC(CSCC(=O)OC)=O)CCN(C(=O)Cc2cc[nH]n2)C1 C1(O)(CNC(C(CCNC(C(C)(C)CO)=O)O)=O)CC2CCC1O2 C=Cn1nccc1C(=O)NC1CCCN(C(=O)C(c2cnn(C)c2)=O)C1 S(=O)(=O)(c1cccc(S(=O)(=O)N(n2cccn2)C)c1)N(C(CN(C(C)C)C)C)C C1(NC(C(F)=CC)=O)CCCC(NC(=O)C(c2cccc(OC)c2)(F)F)CC1 C12(C(=O)NCC(C)OCC)CC(CN)(C1)OC2(C)C.c12cccc(c1)N2 C(=O)(CCN=C(NCc1cc2cc(Cl)ccc2[nH]1)NCC1(SC)CCC1)NC C(=O)(C1=NOC2COCC12)N1C(C)CC(NC(=O)CC2CCN(C)CC2)CC1 Cc1cc2ncnc(N(C)CC3CCCN3C(=O)COCC(C)(C)C)c2[nH]1 N(C1c2ccccc2CC1NC(c1ccc(CO)o1)=O)C(C1C(C)CCO1)=O N1(C(C(C)OC)=O)CCC2(CCN(C(c3cc(N)ccc3C(F)(F)F)=O)C2)C1 C1(CC(=O)NCC(C)(C2CC2)NC(CCSC)=O)C(=O)ON=C1C CCCCCCCCCCC(C)NC(=O)C(=O)Nc1cc(Cl)cc(Br)c1F C1(NC(c2c(C)ccs2)=O)CC12CCN(C(c1c(F)ccc(O)c1F)=O)CC2 n1(CC(=O)OC)c(C)cc(C(=O)NC(CNC(=O)CC23CCC(CC2)C3)CO)c1C C(c1ccncc1)=C(C)C(N1CCOC(CN(C)C(C2CC2C(F)(F)F)=O)C1)=O C1(NC(C(C)CC2CC2)=O)(CO)CCN(C(c2coc(CO)c2)=O)CC1 c1(C(CC)C(=O)N2CC(NC(c3ccc(CN(C)C)o3)=O)C2)ccc(F)cc1 C1(C(=O)NCCn2c(C)cc(C)n2)CC12CCN(C(=O)C(C)(C)C1CC1)C2 N1(C(c2cc(Cl)ccc2C(F)(F)F)=O)CCn2ncc(C3=CCCC3)c2C1 c1(C(N2CCCC(NC(c3cc(O)ccc3Br)=O)CC2)=O)ccc2sccc2c1 N1(C(c2cc(C(=O)OC)n(C)c2)=O)CCN(C)C(CNC(=O)C(F)OC)C1 N1(C(C(C)Cc2ccncc2)=O)CCN(C(=O)CSc2cn[nH]c2)CC(C)(F)C1 N1(C(=O)NC(c2cccc(Cl)c2)C(C)C)CC(O)C2(CCCC2)C1 c1(C(N2CCN(C(c3ccc(C)c(O)c3)=O)C(CF)C2)=O)[nH]nc2ncccc12 c1(C(=O)NCC2N(C(CC)=O)CC2)cc(C2(C)COC2)no1 c1(CCCC)cc(=NC(=O)CC(=O)N(C)Cc2ccc(OC)cc2C(=O)O)[nH]o1 CC1CN(C(C2C(C)(C)C2(C)C)=O)CC(C)C1NC(c1cc(Cl)c(Cl)s1)=O C1(C(CC)C)CCCN1C(=O)C(C)N(C(=O)CCNC(=O)C1CC1)C N1(C(C2CC(O)(CC#C)C2)=O)CC(C)(C)OCC1CNC(C1(CC)CCCO1)=O c1(C(N2CCC(CCNC(C(C)CC(N)=O)=O)C2)=O)cnn2c1CCCC2 C1(CC=C)(NC(=O)CC(C)N(C)C)CCN(C(=O)Cc2cc(C)ccc2F)CC1 C1(C(=O)NCC(C(C)(C)C)NC(c2c(CC)nco2)=O)CC(C2CC2)=NO1 N1(C(c2c(C)n(CCO)nc2)=O)CC(C2(NC(=O)C=Cc3ccncc3)CC2)C1 c1(C(N2CCC(CNC(CCCCCSC)=O)C2)=O)cc2n(n1)CC(C)NC2=O N1(C(CCCC=C)=O)CC2CN(Cc3ccc(O)c(C)c3)C2C1 c1(C(=O)Nc2c(C)nc(F)cc2)n[nH]c2c1CN(Cc1sc(Br)nc1Br)C2 N1(C(Cc2c(C)nc[nH]2)=O)CC2CC(C1)CN(C(C1CCCNS1(=O)=O)=O)C2 CCCCCC(C)(CC)C(=O)NCCCCCCn1cc(CC2CCCC2)nn1 N1(C(CC(CC)CC)=O)CC2(CCC2)CC1CNC(c1c(C)ccc(C)c1C)=O C(C(C(F)(F)F)n1cccn1)NC(=O)NC(c1ccncc1)C C1(CC(=O)NC(C(=O)OCC)C)CC2(C1)CN(C(=O)CN(C)C(N)=O)C2 CCCCC(C)(CO)NC(=O)CC(C(F)F)NC(=O)CC(CC)CC C(=O)(N=c1cnn(C2CCC2)[nH]1)c1cccc(NC(=O)OCc2ccccc2)c1 C=C=CCCC(=O)NCCC(=C)CNC(c1occc1Br)=O c1(CN(C)C(c2ccc(O)cn2)=O)ccccc1CNC(c1cn(CCO)nn1)=O C1(NC(c2cnc(C(C)C)nc2)=O)CC(C)CN(C(c2cc(Cl)ccc2N)=O)C1 C=CCCCCC(=O)N1CCC1CNC(C1(CF)CC1(F)F)=O C=C(C)CC(C(=O)NC(C)CCC(=O)NCCc1ncoc1C)OC Cc1ccc2c(c1)CC(C(=O)OCC1CCCN1)S2(=O)=O CC1=C(C)CC(C(=O)NC2CN(C(C34CSC(C3)C4)=O)CC2C)CC1 CC1(NC2c3nnnn3CCOCCC23CCC3)CC(F)(F)C1.C1(CF)CC1 c1(COC(CSC)=O)nc(C)c(NC(c2ccccc2C)=O)s1 c1(C(N2CC(NC(C(C)OCCOCC)=O)C2)=O)cc2c(nc1O)CCOC2 N1(C(C2CN(C(N)=O)C2)=O)CC(C2CC2)(C(N2CC(O)(CO)C2)=O)C1 N1(C(C=C(C)C(F)F)=O)CCOC2CN(C(c3cc4[nH]ccc4s3)=O)CC12 c1(-c2cnc(CNC(c3cccc(CO)c3O)=O)nc2)cccc2c1OCC2 C(=O)(C(O)C(F)(F)F)NC(C(=O)NC1CCC(C(N)=O)C1)CC1CCC1 c1(C(N2CC(CC)C(NC(C3CCSC3)=O)CC2)=O)cncc2sccc12 N1(C(CCC(=O)NC)=O)CCCC(OCCNC(CCOCC)=O)C1C N1(C(C=CSC)=O)CCN(C(c2nnccc2C)=O)C(C)C1C C1(NC(c2c(C)nsc2C)=O)CC2CC(C1)N(C(C1CN(C3CCCCC3)C1)=O)C2 S(=O)(=O)(c1cc(C(=O)O)cs1)NCC(=O)Nc1c(C)noc1-c1ccccc1 c1(CC(=O)N(CCC(C)NC(CSCC)=O)C)nc(Br)n(C)c1C C1(CC(=O)NCC2(NC(CCc3cc(C)[nH]n3)=O)CCCC2)CCCCC1(C)C c1(OC)cccc(CC(N2CCCC2C(c2cn(CCC(C)C)nn2)(C)C)=O)n1 C1(C(N2CC(Nc3ncncc3F)CC(F)C2)=O)CN2CCC1CC2 C(N=c1[nH]c(N2CCCC3(C=CCO3)C2)nc2cccnc12)c1nnc(C)o1 Cc1c(C(N2CC(NC(c3ccsn3)=O)C(C)C2)=O)cnc2ccnn12 c1(C(=O)NC(c2ccccc2)C(C)NC(CCCOCC)=O)cc(C)n(C)n1 CC1(C)CC(NC(=O)CC(CNC(=O)CC2OCCO2)C2CCC2)C12CC2 Cc1cc(CC(=O)NCC2(CO)CCN(C(C3OCCC3(C)C)=O)C2)cc(F)c1 c1(C(N2CC(NC(C(C)(CO)OC)=O)C(F)C2)=O)cccn2nccc12 C(=O)(CCC(C)(C)C)NC(C)CCNC(=O)CNC(c1ccccc1)=O N1(C(C(CC)C2CCC2)=O)CCN(C(C2(C#N)CC2)=O)CC(C)C1 N1(c2nc(Cl)nc(C)c2F)CCC(C2CCCN(C(C3(Cl)CC3)=O)C2)C1 C(=O)(C1=C(C2CC2)N(C)C(=O)N(C)C1c1cncc(C(=O)OC(C)(C)C)c1)OC Cn1cnc2c1C(C(=O)NNC(=O)c1ccc(Br)cc1OC(F)(F)F)CCC2 C1(C)(CC)CC(NC(=O)CNC=O)CN1C(c1oc(C)nc1C)=O c1(C(=O)NC2C(NC(CC=C=C)=O)CC2)ccc(C#N)c(Cl)c1 c1(C(=O)NC(C(C)NC(=O)CC2CCCC2)C)ccc2c(c1)NC(=O)CCN2C C1(c2n(C(C(=O)OC)C)nnn2)(NC2CC(C)CC(C)C2)CCC=CCC1 c1(-c2ccc(SC)cn2)nc2ccc(C(=O)Nc3ccc(C#N)cc3Cl)cc2s1 CCCC(CCC)CC(=O)NC(C)C(=O)Nc1ccc(CCO)cc1 CCCCCCCC(=O)NC1CC(C(=O)N(CC(=O)OC)C)=CC1O c1(C(=O)NC2CCC(C(=O)NCC3CCN(CC)CC3)C2)cc(F)cc(Br)c1F C1(C(=O)NC(CC)COC)CC2CCCC2N1C(C1CC(=O)N(C)C1)=O C1(NC(c2cc(C)sc2C)=O)C2CCCN(Cc3snnc3C)C2C1(C)C c1(CNC(C2CCCN2Cc2cc(O)ncc2Br)=O)cc(Cl)cc2nc[nH]c12 C12(CNC(C3C(C=C)C3)=O)CCC(NC(=O)CC3(NC(C)=O)CC3)(CC1)CO2 c1(CCOC(C)C(=O)NC2CN(C(=O)C(c3ccccc3)F)C2)ccccc1 c1(CN(CC(=C)F)C(C2(n3nccn3)CC2)=O)cn(CC(=N)O)cn1.c12cn-1nn2 c1(OC)ccc(C(N2CC(CNC(=O)CCc3cnc(C)s3)C2)=O)cc1C1CC1 N1(CC(=O)NC2CCCN(C(=O)Cc3cc[nH]c3)C2)CCCCC(O)C1=O c1(C(N(CCOC)CCNC(=O)Cn2cccn2)=O)c(F)cc(C)cc1F C12(C(=O)NC(C=C)(C)C3CC3)COC(C1)C(NC(c1cnc(C3CC3)o1)=O)C2 c1(OC)oc(C)nc1C(=O)NC(C1CN(C(=O)C2=C(C)CC2)CCO1)C CC1(C)CCN(C(=O)C(C2CC2)C2CC2)C1CC(=O)NCC(F)CO C1(CNC(C(F)=CC)=O)CC2(C1)CN(C(c1cnc(OCC)s1)=O)C2 C(=O)(C(CO)C(F)(F)F)N1CC2C(CC(=O)N(C(C(=O)NC)C)C)C2C1 C(=O)(C(O)COC)NCC1(CC(=O)NCC(C)OC)CC1 c1(C(=O)NC2(CNC(c3cccc(Cl)c3F)=O)CCOC2)ccc2c(c1)NCC2 C(=O)(CC(C(=O)NCC(O)CNC(=O)CCN1C(=O)CCC1=O)NC(C)=O)OC c1(C(N(C(C)CCNC(c2cc(Cl)cnn2)=O)C)=O)ccnn(C)c1=O c1(C(=O)NC2C(CNC(Cc3cn(C)nc3)=O)CCC2)cc2n(n1)CCCC2=O C1(C(=O)NCC(C)Cn2ccnc2)CN(C(C2(C(N)=O)CCC2)=O)CCO1 C1(C(=O)OCC)CCCN(S(=O)(=O)N2CC(CNC(=O)NCC3CC3)C2)C1.OCC CCS(=O)CC(=O)N1CCC(C)(CCNC(c2ccnn2C2CCCC2)=O)C1 c1(C(=O)NCC(C)CN(C(=O)CSc2cnn(C)c2)C)ccoc1Br N1(C(c2cn(CC)nc2)=O)CCC2CCN(C(=O)CC3=CCCC3)C2C1 C1(NC(C2C(C)CCO2)=O)CCCC(CNC(c2cccn2C2CCCC2)=O)C1 c1(-c2nc(O)cc(C)n2)nc(C2COc3ccccc32)nn1CC1CCCO1 Cc1nc(O)ccc1C(=O)NC1COCCN(C(C2CC2C)=O)C1 n1(CC(C)C)[nH]c(CC(=O)NCCCC(C)NC(C2CCCOC2)=O)cc1=O C1(C(N2CCC(CNC(C3(O)CCOC3)=O)C2)=O)CN2CCN1CC2 C#CCCCCC(=O)NCCN(C(=O)Cc1ccc(F)cc1C)CCOCCO S(=O)(=O)(CC(=O)NCC(C1CC1)NC(=O)C(=O)C(C)C)NCC N1(C(C2C(CC)CCC2)=O)CC2CC(C1)CN(C(c1cnc(S)nc1)=O)C2 C(=O)(C1CCCc2ccnn21)N(C1CCCN(C(c2c[nH]c(=N)s2)=O)C1)CCF CCC(C)(CNC(c1n[nH]cc1Cl)=O)NC(C1CC(=O)C1C(C)(C)C)=O c1(N(C)C)cnc(C(N2CCCC(CNC(c3cocc3C(N)=O)=O)C2)=O)cn1 c1(OC)cc(Cl)c(Br)cc1NC(CCC(C)C)C(=O)OCCCF C1(C(C)(CNC(C2CCSC2)=O)NC(=O)OC(C)(C)C)CCOCC=C1 N1(C(CC(C)(C)C)=O)CC2(CCCC2NC(c2noc3ccccc23)=O)C1 Cc1c(C(N2CC(CNC(C3(C)CC(C)OC(C)C3)=O)C2)=O)cccc1[N+](=O)[O-] N1(C(c2c(C)nn(C)c2)=O)CC2(C)CC1C2NC(c1c[nH]ccc1=O)=O N1(C(C2CCN(CC)C2)=O)CCC(NC(c2snnc2C2CC2)=O)C12CC2 C(=O)(C(C)S(N)(=O)=O)N1CC(C(=O)NC(c2ccncc2)C)C(C)C1 c1(C(=O)NC)ncc[nH]c1=NCc1ccc(-c2cccc(C(=O)N(C)C)c2)cn1 c1(C(C)C)ccc(C(=O)NC(C)CC(C)NC(c2ccc(C3CC3)cc2)=O)cc1 N#CC1(C(=O)CCCc2nc(-c3sccc3CO)no2)CCC1 n1(CCC(=O)NCCC2(OC)CN(C(=O)CCC3CC3(F)F)C2)cnccc1=O C1(CN(C(c2sc(C(C)(C)C)nc2C)=O)CC)CCCCN1C(=O)C1=COCC1 c1(C(=O)NCCCCN(C(=O)CCc2cnc(O)[nH]2)C)cccc2nsnc12 c1(C(N2CCC(CNC(C3(C)CC(=C)C3)=O)C2)=O)cc2c([nH]1)CCC2 c1(CNc2c(CC(N3CCC(F)CC3)=O)cccc2)cccc2nccnc12 C1(C)(C(N2CC3C(NC(c4ccc(CC)s4)=O)(C3)C2)=O)CC(C(F)(F)F)=NO1 C(=O)(C(C(C)(C)C)OC)N1C(C(N2C(C=C)CC2)=O)CSCC1 c1(C(N2CC(NC(C3CC(=C)C3)=O)C(OC)C2)=O)ccc(C(F)(F)F)cc1SC CCC(CNC(=O)C(CN(C)C)N(C)C)(CC)NC(C1OC2CCC1C2)=O C1(CNC(CC2(CSC)CC2)=O)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 C1(N(C(Cc2scc(C)n2)=O)C)CCCN(C(C2CNC(=O)N2C)=O)CC1 N1(CCS(CC(C)OC)(=O)=O)CCC(C(=O)NC(C)C)c2ccccc21 N(C(=NCC1CCC1c1cncnc1)N1CCc2c(F)ccc(F)c2C1)CC(F)F C(=O)(CC(F)(F)CS(C)(=O)=O)N1C2(CCN(C(C(CC)C)=O)CC2)CC1 N1(C(C2N(C(C)=O)CC(O)C2)=O)C2CCC1CC(NC(c1ncccc1Cl)=O)C2 C1(CNC(C(C)SC(C)C)=O)CCC2(CN(C(C3CCC4(CCC4)CC3)=O)C2)O1 C1(C(=O)NCC2(CN(C(C(F)=C(C)C)=O)C)CC2)OCCC1(C)C Cc1sc(C(=O)NCCOCCNC(=O)Cn2[nH]cnc2=N)c(C)c1C Cc1cc(C(=O)NCC(C)(F)CNC(=O)CC2=CCOCC2)c(C)c(C)c1 N1(C(CC(CCCCC)O)=O)CCC(C2CCCN(C(c3cnn(C)c3)=O)C2)C1 C1(C#CC(=O)N2CCC(C(C)NC(c3nc(C)ccc3C)=O)CC2)(CC)COC1 c1(C(=O)NC(C2CN(C(C3(O)CC(C)(C)C3)=O)C2)C)cccc(-c2ccc[nH]2)c1 C(CC(C)C)(C(=O)N1CCCC(N(CCF)C(c2ccc(Cl)s2)=O)C1)OC C12(NC(c3nc(C(C)(C)C)oc3)=O)CC(C1)N(C(C1CCCOC1)=O)C2 c1(C(N(C2CN(C(C(C)=C(CC)C)=O)CC2F)C)=O)cc(F)c(F)cc1OC c1(C(=O)NC(C)(CO)C(=O)N2CCC(n3ccnc3)C2)cccc2cc[nH]c12 C1(CCC)CN(C(c2cn(C)nc2OC)=O)CCN1C(=O)CC1CCC(=O)N1C c1(OCC)cccc(CNC(c2c[nH]nc2CNC(=O)C(C)C#N)=O)n1 c1(CC(=O)NCCC2CC(NC(=O)C(O)CC3CC3)C2)cccc(OC(F)F)c1 c1(C(N2CC(CCNC(c3n[nH]c(C)c3Cl)=O)OCC2)=O)cc(Cl)c(F)cc1F c1(C(N2CCC(C(=O)NC(COC)C(C)C)C2)=O)c(OC)cccc1C N1(NC(=O)NC(C2CCN(C(C)C(=O)N3CCCC3)C2)(C)C)C(=O)CCC1=O S(=O)(=O)(c1cccc(F)c1C#N)NC1C(C)(C)CN(C(=O)C2CC2)C1 CCC(CC)CCCNC(c1c(O)cccc1F)c1nnnn1CC N1(C(C2(C)CC=C(C)CC2)=O)C2CCC1CN(C(c1nnn(C(C)(C)C)n1)=O)C2 c1(C(=O)NCCC2OCCCN(C(C(C=C)O)=O)C2)cc2ccccc2c(=O)o1 CCS(=O)c1ccccc1NC(=O)NCCC(C)(O)C1CCCCC1 C1(NC(c2ccc(CCC)s2)=O)CC2CCC1C(NC(=O)C#CC(C)(C)C)C2 C1(CCC)CCN(C(=O)C(F)C2CC(NC(C3CC3Cl)=O)C2)CC1 N1(C(CC2C(CC)C2)=O)CC(NC(C2(C)CCCN(C)C2)=O)C(N=[N+]=[N-])C1 c1(NCC2C(C)C2C)[nH]c(=NCc2ccccc2C(C)(F)F)nc2ncn(C)c12 C1(C(N(CCNC(C2CN(CCC)C(=O)C2)=O)C)=O)COc2ccccc2C1 C1(NC(c2cccc(CC)c2)=O)C(CO)C2CCCCC12 c1(C(=O)NC23CC(NC(c4n(C)ncc4)=O)(C2)C3)nccc(F)c1Cl N1(CCC)CCN(C(=O)C(C(C)O)NC(C2CC(C)(F)C2)=O)CC1 c1(C(N2C(C(=O)NCC(CC)C(C)C)CC(OC)C2)=O)cc(C)nc(C)n1 N1(CC(=O)CC2CCOC2)CCN(C(C2CCCC2(F)F)=O)CC1 CC1=C(c2ccco2)CN(N(C)CC(O)C2CC2)CC1 c1(N2CC(OCCNC(c3c(C(C)C)noc3)=O)C2)ncccc1C#N C1(CNC(=NCC=C)NCC(C2CCOCC2)(F)F)CCc2ccccc2O1 N1(C(CCCCCC)=O)C2CCCC1CC(CNC(=O)Cc1cncc(F)c1)C2 C1(C)(CNC2(c3n(CC=C)nnn3)CCSC2)CCCCC1 Cc1cc(C(=O)N(C2(CC(=O)NOCC3CCOC3)CC2)C)ns1 c1(C(=O)NCCCCNC(c2ccccc2OC2CCC2)=O)ccc(Cl)cn1 c1(C(N2CCC(O)(C(C)NC(CNC(C)=O)=O)C2)=O)c(C)ncc2ccccc12 c1(N2CCC(c3nc[nH]n3)CC2)nc(N2CCN3CCCC3C2)nc2ccsc12 CC1=NN(C)C(=O)C1CC(=O)NC1CC(NC(c2cn(C)cc2C(F)(F)F)=O)C1 c1(C(=O)NCC2(C)CCC(NC(c3cc(CC)[nH]n3)=O)C2)cnn2cnnc2c1 C(c1ccncc1)=CC(=O)NCC(CC)N(C(=O)C(CC1CCCC1)OC)C N1(C(CCC2N(C(C(c3ccn(C)c3)C)=O)CCCC2)=O)CCOCC(O)C1 C1(C(=O)NC2(CNC(COC3(C)CCC3)=O)CCCC2)CC12CCOCC2 Cc1cc(Cl)c(Cl)cc1C(N1CCOC(C(C)NC(=O)C=CCN(C)C)C1)=O N1(C(C(=O)NC(C2COC2)C)C)CCN(C(=O)C2CC2)CC1 C1(C(=O)NC(C2CN(C(=O)C(c3ccccc3)F)C2)C)CCCOCC1 c1(C(C)C(=O)NC2C(NC(=O)C3=C(C)OCC3)CCOC2)c[nH]c2ccccc12 C=CCC(CC(C)C)C(=O)NC1(C(=O)NC2CC2O)CCC1 c1(CCNC(C2CCC(C)C2)=O)ccc(CNC(c2n[nH]c(C3CC3)n2)=O)cc1 C1(CN(C(CN(C)C)=O)C)COCCN1C(=O)CC1CCC(O)C1 c1(C(N2C(C)(CNC(Cc3ncc(C)o3)=O)CCC2)=O)ncnc2c1CCCC2 CN1CC2(CCN2C(C2(F)CCN(CC)C2)=O)C1.C(=O)C=CC(F)F C1(NC(c2c(C)n(C)nc2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 N1(C(C(c2ccncc2)C)=O)CCC(C)C(CNC(c2cccc(Cl)c2)=O)C1 c1(C(N)=O)cnc(Cl)[nH]c1=NC1CCC2CN(C(c3c[nH]c(=O)cn3)=O)CC2C1 C1(C(=O)NC(CNC(C(c2nc(C)sc2)=O)=O)C(C)C)CC2CCC1O2 Cn1nc(C(=O)NCC2CN(C(c3ccc(C(N)=O)cc3)=O)CC2O)ccc1=O CC(CCC(=O)N1CCC(O)(CCC(=O)O)C1)NC(c1cnns1)=O C1(C2CCN(C(C34CC=CC(C3)OC4)=O)CC2)(NC(C(C)C2CCCC2)=O)CC1 C#CCCCC(C)C(=O)N1CCC(C)(NC(=O)Cc2sc(C)nc2C)C1 N1(C(C(=O)NCC)=O)CCn2c(CNC(C3CC(=O)C3)=O)nnc2C1 N1(C(c2nn(C)cc2I)C(=O)NCCOC)CCCCCC1c1cccc(C)c1 N1(C(c2nc(C)n(C)n2)=O)CC2CC(NC(c3ccc(N=[N+]=[N-])cc3)=O)CC1C2 CN1CCN(C(N2CCOCC2CCCc2ccccc2)=O)CC1C1=CCN=C1 C(=O)(C1=CCCSC1)NCCC(C(=O)N1CC(COC)C1)O C1(NC(c2cncc(NC)c2)=O)CC2CC(NC(c3cc(C)n(C)c3)=O)CC2C1 c1(CC(=O)NC2N(C(CC3C(=O)NC(=N)S3)=O)CC2)coc2cc(F)ccc12 CCCCCCC(C)NC(C1(F)CCCN(C(c2cnc3n2CCC3)=O)C1)=O C1(CC=C)CCCCN1C(=O)C(Cc1ccccc1Br)NC(=O)Cc1ccsn1 C1(C2CCCCC2)(C(N(C)CC2CN(C(C3(CCN(C)C)CC3)=O)CCO2)=O)CC1 c1(NC(C2C(NC(c3ccc(C)cc3F)=O)CCC2)=O)ncc2ccccc2n1 C(=O)(C1CCc2nccn21)NCCN(C)C(C1CN2CCN1CC2)=O C=C(Cl)C(C)(C)C(=O)NC1CCN(C(=O)CCCN(C)C)C1 CN=c1[nH]c(=NCC2(C)CCCCO2)[nH]c(=NCc2ccnc(SCC)c2)[nH]1 CCC(CN=c1nc2c(ncn2CC)c(NCC(C)(CC)OC)[nH]1)OC c1(C(N(C2CCCN(C(=O)CCOC3CCC3)C2)C)=O)cc(C2CC2)ccn1 Cc1ncccc1C(=O)NC(c1ccccc1)C(=O)NCCn1cccnc1=O c1(CN2CCN(C(c3c(CC)c(Br)ccc3)=O)C(CC)C2)cc(F)cc(C)c1O CC1(C(N2CCCC2c2cn(Cc3cccc(Cl)n3)nn2)=O)Cc2ccccc2C1 Nc1ccc(C(=O)NCCN(C(c2ncc(Br)cn2)=O)CC2CC2)c(Cl)c1 O(NC(=O)C(C)(C)C(C)NC(c1cnn2c1CCC2)=O)C(CC)C C12(NC(c3ccc(CC)cc3O)=O)CCC(CNC(=O)C=CCOC)(CC1)OC2 N1(C(C)=O)CCC2(CC1)CN(C(=O)C(c1ccccc1)=O)C2 N1(C(=O)CC2CNC(=O)O2)CC2CC(C1)N2C(C1(F)CCCC1)=O c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCCOCC)=O)ccc(N)c(Cl)c1 CC1N(C(=O)CN(C)C(C2COC2)=O)CCCC1(C)C N1(C(c2ncc(OC(C)(C)C)nc2)=O)CC2CCC1CN2C(c1cnccn1)=O C1(SC)CCCC1C(N1CC(C(N)=O)(CNC(=O)CC2(NC(C)=O)CC2)C1)=O C1(C(C)OCC)CCN(CCC(=O)NC(=O)NCc2ccccc2Br)CC1C C=C1CCC(CNC(C2CCCN(C(=O)Cc3nc[nH]n3)C2)=O)CC1 C12(C(=O)NCC(CCOC)NC(c3nnc(C)s3)=O)CCC(CC1)CC2 C1(NC(C2(NC(C)=O)CCC2)=O)CC2(CCCCN2C(C2SCCC2C)=O)C1 N1(C(C2(CC(=O)OC)CC2)=O)CCC2CCCN(C(=O)CCc3nc(=N)[nH][nH]3)C2C1 C1(C(=O)N(C2CC2)C(C2CC2C(=O)N(CCO)CCO)=O)CCC(O)CC1 c1(C(C)C)cc(C(=O)NCC2CC(C(=O)NCc3cn(C)nn3)C2)on1 c1(CCC(=O)NC2C(NC(CCC#CC)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] N1(C(c2c(C#C)c[nH]n2)=O)CCC2(CC1)CN(C(=O)C(C)CCCCCC)C2 N1(C(CCCNC(C)=O)=O)CCC(C(=O)N2CC(C)C2(C)C)=C(F)C1 N1(C(C(=O)Nc2ccc(OC)cc2)=O)CCC(C)C(NC(C2CSCCS2)=O)C1 C(C(=O)NCC1(NC(=O)C2=CCCS2)CCCCC1)(C(C)C)SC C1(NC(c2cnc(C)[nH]2)=O)CN(C(C2Cc3nccn3C2)=O)C2CCCC12 c1(C(CC(=O)NC(C)CCNC(C2CC(=C3CC3)C2)=O)C)cccc(F)c1 N1(C(C2CCN(C(=O)C3(C4OCCO4)CC3)O2)=O)CC23CCC2(COC3)C1 C=CCC(C)C(=O)NCc1ccc(CN(C(=O)CC(C)COC)C)cc1 C(N=c1[nH]c(N2CCCC(CF)C2)nc2ccccc12)C1(CO)CCC(C)(C)C1 Cc1nc(C)c(CN2CCC(NC(c3cc(I)c(F)cc3Cl)=O)C(F)C2)nc1C N1(C(C(CCC)NC(c2ncn(C)n2)=O)=O)CCC(C)=C(F)C1 c1(C(=O)NCC(C2CCOC2)NC(c2cc(C(=O)OC)on2)=O)ncncc1Cl N1(C(C(CC#C)NC(C)=O)=O)CCC(NC(C2CC3CCC2CC3)=O)C(C)(C)C1 c1(C(=O)NC2CCCC(Nc3ncc(I)cn3)C2)cc2ccccc2oc1=O c1(C(=O)NC(CCOC)C(=O)N(C)CC2CCCO2)cnn2ccccc12 N1(C(C(C=C)CC)=O)CCC(CCOC)(NC(c2ccc(=N)[nH]n2)=O)CC1 c1(CC(=O)NC(CCNC(CC)=O)(C)C)ccc(F)cc1Br Cc1ccc(C(N2CC(O)(CN(C)C(c3c(C)coc3C3CC3)=O)C2)=O)c(C)c1 CC1CCCCN(C(=O)C(C(C)(C)O)NC(=O)COC(C)(C)C)C1 C1(C(=O)OCC)CN(C(=O)OCc2c(C)nn(COC)c2C)CCC1O C#CCCC(O)C(=O)NC(C)C(C)(C)NC(c1ccn(CC(C)C)n1)=O C(=O)(C(C)(C)CC(F)F)NC(CCN(C(=O)C=Cc1cnc[nH]1)C)C(C)(C)C CCCC(CCCNC(C1CC12CCC2)=O)NC(c1ccc(OC)cc1Cl)=O N1(C(CCOC)=O)CCC(C(C)(C)C)(CNC(=O)C(C(C)C)c2cccnc2)C1 C1(C(=O)NCc2n(CCC)ccn2)CN(C)CCN1C(=O)CC1(N(C)C)CCC1 c1(C(=O)NCc2c(C(N3CCC(C(N)=O)C3)=O)scc2)ccccc1Cl C1(c2cc(C)sc2)CCN(C(=NCC2CCC2)NCc2cccc(Br)c2O)C1 N1(C(CC(C)C2CCCC2)=O)CC2CCCCC2(NC(=O)Cn2ncnn2)C1 c1(-c2cn(CCC(=O)NC(C)CCN(C)C)nn2)ccc(C(F)(F)F)cn1 CC(C)(C)CC(C)(C)C(=O)NC1CCCN(C(=O)CCCc2cnccn2)CC1 CCCC(O)C(CO)NC(=O)CN(C(c1cc(C)nnc1C)=O)CC1CC1 N1(CC(C)(C)NC(=O)C=Cc2cccnc2)CCN(C(C2CCNC2=O)=O)CC1 C1(NC(C2(CC=C)CCOCC2)=O)CCN(C(C2(C#N)CC2)=O)CC1F S(=O)(=O)(c1cccc(NCC(C)Oc2ccc(F)c(Br)c2)c1)N(CCC(C)C)C c1(OC)cc(C(=O)N(CC(c2c[nH]c3ccccc23)=O)C)cc2c1OCO2 C1(NC(c2c(C)cc(F)nc2)=O)CCN(C(=O)CC2CCC3CC23)CC(O)C1 n1(CC)c(-c2nc(CCCO)nn2CCN2CCC(O)CC2)cnc1O CC1(C)CCCCCC1NC(C1CCC(C(=O)NCc2cc[n+]([O-])cc2)O1)=O Cc1cnccc1C(N1CC(c2ccccc2)(NC(C2COC(=O)C2)=O)C1)=O C=CCC(CC)C(=O)C(C)=O.C(=O)(C(C)C)N(CCCOCCN)C N1(C(CN2CC(C)C2)=O)CC2CC(C(=O)NC3CC3)CC(C2)C1.C1(=O)C=CCN1 C1(CC(=O)NCCN(C(=O)CCc2cnn(C)c2)CC)Cc2ccccc2C1=O CC1CCN(C(=O)CC2(CO)CC2)C1CNC(c1c[nH]ccc1=N)=O c1(C(CC)N(CCNC(=O)C(C)(C)C)Cc2occc2Br)ccccc1F c1(CC(=O)NC(CNC(C(C)OC)=O)C2CCC2)ccsc1Cl O(NC(=O)CN(C(=O)CC)CCN(C)C)CCC.C1(C)CCCO1 CN(CCCC(=O)N1CC(NC(c2cnn(CCC#N)c2)=O)C2(CC2)C1)N=O CC1CN(C(=O)CS(C)(=O)=O)CCC1N(C(=O)C(F)(F)C1CCOCC1)C c1(C(C(C)NC(c2c[nH]c(C(C)(C)C)c2)=O)C)ccc(C(F)(F)F)cc1 c1(NC(N(C(C(C)SC)C)C)=O)ccc(OCCCF)cc1 C1(NC(C2C(CC)OCC2)=O)CCS(=O)(=O)C12CN(C(=O)C=C(Cl)Cl)C2 C(=O)(CCCC(F)F)N(C(CNC(C1CCN(C)C1)=O)C1CC1)C CCCCCC(C)(C)C(=O)NC1CCCCN(C(=O)C(CCSC)OC)C1 CC1CN(C(C2CCC(F)CC2)=O)C(C)CN1C(=O)CCc1ccccc1C#N CCC(CC(=O)N1CCC(C)(C)C(C(=O)N(C)Cc2cnc[nH]2)C1)C(C)(C)C N1(C(=O)C2=CCOC2)CCN(C(c2ccc(-c3cccs3)o2)=O)C(C2CCC2)C1 C1(CC(=O)NCC(CNC(C2(C(C)C)CCCO2)=O)(C)C)CCCCCC1 N1(C(C2(O)C(C)(C)C2)=O)CCC2(CCOCC2)C(NC(=O)Cc2cn[nH]c2)C1 N1(C(CCCOC(C)C)=O)CCC(C(C)(C)NC(C2CC(N(C)C)C2)=O)CC1 n1(CC(=O)OC)c(C)cc(C(=O)C(Cl)(Cl)Cl)c1C.C1(C2C(=O)O2)CCCCO1 c1(-c2ccc(CN3C(CC(=O)NC4CCCCC4)CCC3)o2)ccc(F)cc1 Cc1cnc(O)c(NC(=O)C(C2CC=CCC2)NC(=O)C=CC2CC2)c1 C1(NC(c2cnn(C)c2Cl)=O)CN(C(C2CC(=O)N(CC3CC3)C2)=O)CC1(C)C C1(N(C)C(=O)OC(C)(C)C)CC2CC(NC(=O)C(c3ccc(O)cc3)=O)C1C2 C1(CNC(CCN(C(=O)C=Cc2cocn2)CC#C)=O)(CF)CC(=O)C1 C1(C)(CSC)CCN1C(=O)C(F)CC1CN(C(=O)COc2cc(C)on2)C1 C1(N(C(=O)Cn2nnc(C)n2)CC)CCCN(C(C2CC3CCC2O3)=O)C1 C1(CNC(CC(=O)OC)=O)CCN(C(c2nn(C(C)(C)C)cc2Cl)=O)C1(C)C c1(NC(C2CC2NCc2ccc(F)s2)=O)ccc2sc(Cl)nc2c1 C(=O)(C(C)(C)C(=O)OC)NC12CC(NC(COCCCC#C)=O)(C1)C2 C1(CC)CN(C(=O)C(CC2CCC2)NC(=O)C(=O)NC(C)C)CC1O N1(C(C2N(C(c3c(C)cccc3O)=O)CCC2)=O)CC(=O)NC2(CC2)C1 N1(C(c2cncc(O)c2Cl)=O)CCCC(C2CN(C(=O)C(O)C(F)F)C2)C1 CCCC(C)(C)C(=O)NC1CC(F)CN(C(C2(C)CCC(=O)NC2)=O)C1 CCC1=NOC(C(=O)NC2(C)CCN(C(c3nnn(CC)c3C(C)C)=O)C2)C1 CCCC(C#N)C(=O)N1CCC(C)C1c1cn(CCOCc2ccccc2)nn1 c1(COC)nc(Cl)cc(=NC2CC(NC(C3Cc4ccccc4CO3)=O)C2)[nH]1 C1(NC(c2onc(C)c2C)=O)CCCCC12CCN(C(C1(CF)COC1)=O)CC2 c1(C(=O)NCCCN(C(C(C=CCCC)O)=O)C)cc2c(Cl)nccc2s1 N1(C(C(CC)OC)=O)CCC(C2CC2)(NC(c2csc3ccccc23)=O)C1 N1(C(Cc2cc(C)sc2)=O)CC2CC(NC(=O)CC3CCOC3(C)C)CC1C2 n1(CC)cc(C(=O)NC(C)(C)C=CC(=O)NCC(F)(F)CC2CC2)nn1 Cc1cccc(F)c1C(=O)NC1C=CC(C(=O)NCc2nocc2C(C)C)C1 C#Cc1ccc(C)c(NC(=O)C(=O)NC(CSC)C(=O)N2CCCCC2)c1 c1(OCC(=O)NCC(C)NC(C(C(C)C)O)=O)c(Cl)cccc1F Cc1cccc(CC(=O)NCc2cc(C(N3CCCC3CN(C)C)=O)co2)c1 C1(CCC2N(C(c3nc(C)[nH]n3)=O)CCC2)CCN(C(=O)CC2CC2C)CC1 c1(C(=O)NCC2C(C(=O)NC(C=C)CO)C2)cccc(CN2CCSCC2)c1 C1(CNC(C2N(N=O)CCC2)=O)CC2CCC1N2c1cc(C(F)(F)F)nc(Cl)n1 C(C(C)(CNC(=O)CCN(C(c1ccc(C#N)s1)=O)CC1CC1)CO)OC N1(C(C(C(C)C)F)=O)CCC(O)(C(C)NC(=O)CCCCCn2cnnn2)CC1 CC1CCN(C(=O)N(C)Cc2ncnn2C)c2ccccc21 C1(C(=O)NC(C2CCN(C(C3(C)CCCC3)=O)C2)C)CCC1(C)C C1(NC(CCC(=O)NC)=O)CCCC12CN(C(C1CC3(C1)CC3F)=O)C2 N1(C(C2(CC)COC2)=O)CC(CO)(NC(=O)CSc2cccs2)C1 C12(NC(c3c(C)cc(SC)o3)=O)CCCC1N(C(c1ccc(Cl)cc1C)=O)CC2 C12(C(N(C)CC3CN(C(C4OCC4(C)C)=O)CCO3)=O)CCC(CC1)CC2 CC1(C)CCCC(CC(N2CCC(C(C)(C)NC(=O)Cn3cnnc3O)C2)=O)C1 c1(CC)cc2c(NC3(CNC(c4coc(CC)n4)=O)CCC3)ncnc2s1 n1(CCC)cc(C(=O)NCC2(CN(C(=O)CC(C)OC)C)CC2)c(C)n1 c1(CN2C(C(=O)NCC3(O)CCOCC3)CC(=C)C2)c(Cl)cccc1B(O)O Nc1cc(F)c(-c2cccc(C(=O)NC3(CO)COC3)c2)c(F)c1 N1(C(C(CC=CC)C)=O)CC(CC(=O)NCC(C)(O)CSC)CC1(C)C CCCCCC(O)CC(=O)N1CCC(C(C)NC(C2CC3(C2)OCCO3)=O)CC1 C1(CNC(C(CC)CCOC)=O)CN(C(=O)COC(C)=O)C2COCC2O1 CC(CC(=O)N1CC2CN(C(c3nc(Cl)ccc3N)=O)CCC12)C(F)(F)F CC1(O)CCN(CC(=O)NC2(CNC(=O)CN3C(=O)CNC3=O)CCCCC2)C1 C(CC(N=c1cc[nH]cc1C#N)C(C)C)N(C(c1ccc(C)nc1)=O)C C(CCC(C)C)(C(=O)NCc1ccnc(Cl)c1)NC(Cc1cc(C)n(C)n1)=O C1(C(=O)OC)CCCCC1(C)C.c1(CCC23CN(C2)C3=O)ccc([N+](=O)[O-])s1 c1(C(N2C(C)CN(C(=O)CC3CCCNC(=O)C3)CC2)=O)nc2cccnc2s1 O=C(N=c1nn[nH]n1-c1ccccc1Cl)NC1CC1C(=O)Nc1ncccn1 N1(C(C2CC2c2c(Cl)cccc2Cl)=O)CC2(CCOCC2)C1c1ccco1 c1(OCCOC)ccc(-c2cncc(C(=O)NCCc3ccccn3)n2)cc1 C1(C(=O)NCc2c(C(C)C)con2)CCN(C)CC1.C12(CCCO1)C(=O)NC2 Cc1nn(CC(=O)NC(C2CCCN2C(=O)CC2CCSC2)C)c(=O)o1 c1(CNC(=O)NC2C(CC(C)C)CCCC2)ccc(F)cc1O C1(C2CCOCC2)(NC(C2CC(CNC(=O)C=Cc3nccs3)OC2)=O)CC1 C1(NC(=O)CCCC(=O)N2CCC2)CN(C(=O)C=CC2CCC2)CC12CCOCC2 C1(C(=O)NCC2(F)CC(CNC(c3nnsc3C)=O)C2)(OC)CCCOC1 c1(CN(CC(O)CNC(C2CC2C(C)(C)O)=O)C)ccccc1 c1(C(C(F)(F)F)OC)ccccc1NC(c1nc(C)cn1C)c1ccccc1Cl c1(C(=O)NC2C(C)(CNC(c3coc(CO)c3)=O)CCC2)ccnc2[nH]cnc12 c1(C(N(CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC)CC)=O)ccc(Cl)c(C)c1 N1(C(CCOC2CN(C(CC(C)N(C)C)=O)C2)=O)CCC(C2=NOCC2)C1 C=CCCN=C(NCc1cc(C)ccc1Br)NC1CCC(=O)NC1 N1(C(c2cc(C)c(C)o2)=O)CC(C2CCN(C(C3CCOC3(C)C)=O)CC2)C1 C1(OCCNC(C(C)c2cncs2)=O)CCN(C(c2coc(Cl)n2)=O)C1 c1(C(=O)NC(C)C(=O)N(CCCNC(C2C(Cl)(Cl)C23CC3)=O)C)ccccc1Cl N1(C(CCOCC)=O)CC(NC(c2nscc2C)=O)C(n2ccnn2)C1 CCCC(C(=O)N1CCCCC1CNC(=O)C(C(C)CC)OC)S(N)(=O)=O CC1CN(C(=O)COc2cccc(F)c2)CC1NC(=O)C=Cc1cnc[nH]1 Cn1ccc(-c2noc(C3(C4CCNCC4)CCC3)n2)n1 N(C)(S(=O)(=O)N(C)C)CC(=O)NC1CCC(CCNC(COCCC#C)=O)C1 c1(C(=O)NC(C)CCNC(=O)C(c2ccccc2F)O)cccc(P(C)(C)=O)c1 CC(=Cn1ccnn1)C(=O)NCCCCN(C)C(C1CCC(F)(F)CC1)=O C1(C(N2CC(OCCNC(C(C)S(C)(=O)=O)=O)C2)=O)CCc2nn(C)cc2C1 N1(C(C2C(=C)C2)=O)CCC2CC12C(=O)NCCN(C)C(C)C CC(C)C(CCN(C(=O)CCc1cc[nH]n1)C)NC(C1(O)CCCC1)=O C1(CNC(CCSC)=O)CN(c2nccc(C(C)(C)C)n2)CCCO1 C(CCN(C(=O)C(c1ccc(F)cc1)CO)C)(C(C)C)NC(c1c(C)cc[nH]1)=O N1(C(C2C(CC)N(C(c3ccc(F)cc3)=O)CC2)=O)CC(OC)CC(C)C1 C1(C(N(CCCN(C(C2C(C(=O)OC)C=C2)=O)C)C)=O)CCCCN1C Cc1ccc(C(C)(C)C(=O)NCC2CN(C(=O)C3=CCC3)C3CC23)cc1 c1(C(N(C2CCC(NC(C3CC34CCOC4)=O)CC2)C)=O)c[nH]c2cnccc12 Cc1ccc(S(=O)(=O)NC(c2ccccc2)C(=O)O)cc1.N12CCC(C1)CC2=O c1(CCNC(C2CC2F)=O)ccc(CNC(C2CC(F)C2)=O)cc1 C(CCF)(C(=O)NCCCc1nccs1)NC(C1C(C)OCC1)=O c1(C(N(CC(CC)NC(c2cc(C(CC)CC)no2)=O)C)=O)nnc(O)cc1O C(=O)(C(=O)NCC(C)CNC(C1CCN1C(=O)OC(C)(C)C)=O)NC c1(C(N2CC(O)(CC=C)C2)=O)ccc(CNC(=O)CN2CCSCC2)cc1 C1(C(N2CCC(COC)(CNC(=O)C(O)C(C)C)CC2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NC(c2ncc(C)o2)C)CC(C)CN(C(C2C=CC=CC=C2)=O)C1 C=CCN(OC)C(=O)C12C(NC(=O)CCc3csnn3)C3CC1C2C3 C1(NCCCC(C)OC)CC12CCN(C(=O)OC(C)(C)C)CCCO2 c1(OC)ccnc(OC)c1C(=O)NC1CCN(C(C2COC(=O)O2)=O)C1 C1(CC(N2CCN(CCNC(CS(CC)(=O)=O)=O)CC2)=O)COC2(CCC2)CO1 N1(C(c2c(COC)cco2)=O)Cc2ccccc2C(NC(=O)C(F)C(C)(C)O)C1 c1(SCCC)cccc(C(=O)NC2CN(C(=O)C=NOC)CC2C(F)(F)F)c1 S(=O)(=O)(c1cscc1F)Nc1c(CC(=O)OC)cccc1 c1(OC)c(C(=O)NC2CCC2CNC(C2CCC(O)CC2)=O)cnn1C C1(CC(=O)NC(C=C)(C)CC)CC2(CC2)CN1C(=O)CSC(C)(C)C c1(OC)cc(NC2CN(C3CN(C(C4C=C4C)=O)C3)C(=O)C2)nc(OC)n1 C(c1cnc2ccccc2c1)=CC(=O)NCc1cnn(C)c1Br C1(NC(CSC(C)C)=O)CN(C(c2cnc(N)c(Cl)c2)=O)CC1S(C)(=O)=O C(=O)(CCC(F)F)NCC(CNC(=O)Cn1ccc(C(F)(F)F)n1)O [N-]=[N+]=NC1CC(C(=O)NC2CC3CCC2O3)N(C(c2ccc(C#N)cc2)=O)C1 Cc1ccc(-c2ccc(C(=O)NC3CC(F)(CNC(c4ccsn4)=O)C3)s2)s1 C1(OC)C(NC(=O)CC(C)(C)n2cc(CC(C)(C)O)nn2)CC12CCC2 c1(C(N2CCC(CNC(c3cn[nH]c3)=O)C(F)(F)C2)=O)ccc2nc(O)[nH]c2c1 C(=O)(C1=Cc2ccccc2C1O)NC1C(C)(C(C)C)C1 C1(C(N(C)Cc2n(CC)cnn2)=O)CCN(C(C2CC(=O)N(C)C2)=O)C1(C)C c1(OC)c(C(c2nnnn2CCC2(C)CC2)NC(C)(C)CF)ccc(Br)c1F C1(NC(CN(c2ncccn2)C)=O)CC2CC(C1)N(C(=O)Cc1ccc(Cl)s1)C2 C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)CSc2nnnn2C)CC1C C#CCC(O)C(=O)N(C)CC1CC(F)CN1C(=O)CSc1nnnn1C1CC1 N1(C(C(c2ccc(F)cc2)C)=O)CC2CC2(CNC(c2ccsc2C#N)=O)C1 C1(CC)CN(C(=O)C(c2ccccc2F)O)CCC1NC(C1(Br)CC1)=O C1(C(N2CCC(C(=O)OCC)C2C)=O)CC(n2cc(CC3CCC3)nn2)C(O)C1 Cc1ccc(C(=O)NC2CCCC2NC(C2(C(C)(F)F)CC2)=O)c(Cl)c1.C1(C)CC1 N1(C(C(CCOC)C)=O)CCN(C(c2ccc(C)cn2)=O)C(C)C1 Cc1cc(C(c2nnnn2C2COC2)Nc2cn(CCO)nc2C)sc1C C1(C(=O)NCC2(CN(C(=O)C=C3CCC(C)C3)C)CC2)(OC)CCC(C)(C)CC1 c1(OC)ccc(Cl)c(C(=O)NCCC2CCCCN2C(c2cccnc2C)=O)c1 N1(C(C(CC(C)C)O)=O)CCCCCC(NC(c2ccc3ncnn3c2)=O)C1 c1(NCCCCOC)cc(=NCC2CNC(=O)CO2)[nH]c(C(F)(F)F)n1 c1(C(N2CC(F)CC(NC(C(C=C=C)C)=O)C2)=O)ccc2cc(O)ccc2n1 CCCCCC(O)C(=O)NCC(C)(CC(C)C)NC(=O)CCNc1ccccn1 CCC(CCC(=O)N1CCC(SC)C1)NC(c1cc(Cl)cs1)=O N1(C(C(C)=C(C)C)=O)CCC(C(C)C(=O)NCC2CN3CCC2C3)CC1 C=C=CC(C)C(=O)NCC(C(C)C)NC(c1c(C(F)(F)F)coc1CC)=O c1(C(=O)NC2CN(C(C(C)(C)NC(C)=O)=O)CC(C)C2)c[nH]c2ccc(Br)cc12 C1(NC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)COC2(C)CCCC2)CC1F C1(CCC)CC(C(=O)N(C)CCNC(c2nc(C)n(C)n2)=O)CCO1 N1(C(C(CC2CCCC2)NC(C(CC=C)(F)F)=O)=O)CCC2(CC1)CN(C)C2 C1(CNC(CN(C(C)C)C)=O)CCC(CNC(C2CC3C=CC2C3)=O)CC1 C1(NC(C(C)OC2CCCC2)=O)CC2(C1)CC(NC(C1CNC(=O)N1)=O)C2 C(=O)(C(CC(C)C)C(C)C)N1CC(CC)C(CNC(c2cnnc(C)c2)=O)CC1 c1(C(=O)NCCC(CNC(CCOCC#C)=O)=C)nc(C)c(C)[nH]c1=O N1(C(C(C)=C(CC)C)=O)CCCC1(CNC(C1(CC)CCOCC1)=O)COC c1(C(N2CC(NC(c3cc(CCOC)on3)=O)(CO)C2)=O)cc(O)ccc1C S(=O)(=O)(c1cccc(Cl)c1)N1CC(CC(N2CCC(F)C2)=O)OCC1 C12(CCNC(C3C=CCN(C(C4(Cl)CC4)=O)C3)=O)CC(CCO1)C2 C#CC1(C(=O)NCC2(N(C)C)CCC2)CCN(C(=O)CC(C)(O)C=C)C1 N1(C(C2(CC(N)=O)CC2)=O)CC(CNC(=O)CC2CC(N(C)C)C2)C(O)C1 c1(C(N(CC(CC)NC(C2CC2c2ccsc2)=O)C)=O)ccc(F)cc1[N+](=O)[O-] C1(NC(c2cc(CC)no2)=O)CCC2(CCN(C(C3(CF)CC(=O)C3)=O)C2)C1 c1(C(C)C)conc1CC(N1CCC(CNC(c2cc(C3CC3)[nH]n2)=O)C1)=O N1(C(c2cccc(NC(C)=O)c2)=O)CC(C)N(C(c2cccc(=O)o2)=O)CC1C C1(CNC(c2nccc(C)n2)=O)CN(C(C2CC(=C3CC3)C2)=O)CCC1(C)C C(C(C)N=c1[nH]c(Cl)nc(C)c1F)NC(Cc1ccc(C)cc1Cl)=O c1(C(N(C(C)C(=O)NOCC(O)CO)CC)=O)n[nH]nc1OC N1(C(c2cc(CC)c(C)s2)=O)CCCC1C1CCCCN1C(=O)COC(C)(C)C C(CC(=O)NCCCCCC(C)C)(C(F)F)NC(c1ccc(C(C)=O)[nH]1)=O c1(CCC)ccc(C(=O)NC2COCC2CNC(=O)C(C)(O)CC)cc1[N+](=O)[O-] S(=O)(=O)(c1ccc(Cl)cc1Cl)N1C2CN(C(c3cc(Br)cnc3F)=O)CC21 CCC(O)CC(=O)NC1CCN(C(c2nc(Cl)sc2C)=O)C1 C1(C(C)(C)O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C.C12CCN1C2=O N1(C(CC2CN(C(Cc3ccc(C)s3)=O)C(C)C2)=O)CC2CCC(C1)C2O N1(C(CC(C=C)CCC)=O)CCCCC2(C1)CN(C(=O)CC(F)(F)F)C2 C1(C(N(CC(C)OC)C)=O)CN(C(=O)Cn2cc(CO)nn2)C(C)(C)C1 c1(CCCCC)cc(CN2CC(CNC(=O)Cc3ccnn3C)(COC)C2)n[nH]1 Cc1cccc(OCC(=O)OCc2cn(Cc3cccnc3)nn2)c1C c1(C(N2CC3CN(C(C4(n5ccnn5)CC4)=O)CC3C2)=O)cc(Cl)c(F)cc1Cl N1(C(C2CC(C)(C)C2)=O)CCC2(CCCN(C(c3ccc(F)c(F)c3)=O)C2)C1 c1(C(=O)NCC(CN(C(=O)C2=C(C)CCC2)CC)(C)C)c(F)ccc(F)c1O CCC(C)CCCCC(=O)NC(CCCOC)C(=O)N(C)CC1CCCCCC1 c1(C(=O)NCCC(C)NC(=O)CC2COC(=O)C2)ccnc2[nH]cnc12 c1(CCC(=O)NCCN(CCOC)C(C2CC23CCCC3)=O)ccccc1Br C(=O)(C(CO)c1ccccc1)N(CC(C)(C)NC(=O)C(N)=O)C n1(CCNC(=O)OC(C)(C)C)cc(C(N)=O)cn1.C1(=O)C(=O)NCCCN1 c1(OC)cccc(N(CC(C)C)C)c1.c1(C2N3CCCC3NC2=O)nocc1C Cc1ccc(OCC(=O)NCC(O)CN(C(=O)CSc2cnnn2C)C)cc1 CC1(C(N2CC3C(CNC(=O)CC4CCCCCC4)C3C2)=O)COC(=O)N1 c1(CCC)cc(C(=O)N(C)CC2CN(C(c3cnn(CC)n3)=O)CCO2)nn1C C(=O)(C1=CCCSC1)N1CCC(CCCCCNC(Cc2c(C)ocn2)=O)CC1 N1(C(CN(C)C(N)=O)=O)CC2CCCC(C1)N2C(C1CC12CCOCC2)=O c1ncc2c(n1)CC1CCC2N1C(=O)C.C1(C(C)(C)C)CCC(C(F)(F)F)CC1 C12(C(=O)NC3C(NC(=O)CCc4cnco4)CC3)CCCC1C2(F)F C1(NC(c2c(C(C)C)occ2)=O)CCC2(CCCN(C(=O)Cc3cncs3)C2)C1 c1(C(=O)NC(CNC(C=C(C)C(C)C)=O)C(C)C)nc2n(c1Br)CCC2 c1(OCC(C)C)ccc(C(N2CC(O)(CCNC(C3(C)CSC3)=O)C2)=O)cc1 C1(NC(=O)CCc2ccccn2)(CNC(=O)C(F)F)CCc2ccccc2C1 C1(CC(N2CC(n3cc(NC(=O)CN4CCCCC4)cn3)C2)=O)CCS(=O)(=O)C1 C(C=CC(=O)NC1(CNC(=O)CNS(N)(=O)=O)CC1)(CC)=CC C1(C(=O)OCC)CCNCCC1Nc1c(N(C(COCC)=O)CC)cc(Cl)cc1 N1(C(CC=C)=O)CCC2CN(C(=O)C(=Cc3cnn(C)c3)C)CC2CC1 C(CC(F)(F)CC(F)(F)F)ONC=O.C=CCCCn1cc(C(O)C2CC2)nn1 C1(CNC(C(C)NC(CC)=O)=O)CC2CN(C(=O)C=C(C)C(F)F)CC12 CC1CCN(C(=O)OC(C)(C)C)C1C(=O)NCCC(O)C(F)F Cc1n[nH]c2cnc(C(=O)NC3CN(C(C4CC5CCCCC45)=O)CC3C)cc12 n1(CC)ccnc1C(N1CC(O)(CNC(=O)CC2CCOC2C)C1)=O S(=O)(=O)(c1ccc(Cl)cc1Cl)N1CCC2CN(C(C=CC)=O)CC21 C1(c2cn(CC3C(C)C3C)nn2)(NC(CC2CC(CC)C2)=O)CCOCC1 C(C)(C(O)C(=O)NC1CC(CNC(c2cccc(N)n2)=O)C1)OC N1(C(C(CC)=CC)=O)CCC(CNC(c2csc(C(F)F)c2)=O)C1(C)C c1(NC)ccccc1C(=O)OCC(C)C(=O)Nc1ccccc1OC n1(CC=C)c(N(CCO)Cc2cccc(Br)c2)nnc1C(C1CCOCC1)C C1(N(C)C)CCCC(C(=O)NCC2CCN2C(C2CCCO2)=O)C1 c1(C(C)(C)NC(=O)NC(C)C(C)(C)C#N)ccc2c(c1)OCCO2 C1(CNC(CC(CCC)O)=O)CCN(C(=O)Cn2ccnc2C)C12CCC2 c1(CNC(CC(=C=C)C)=O)c(C)nn2c1CN(C(=O)CN1CCCC1CO)CC2 C(=O)(C1=C(Cl)CCCC1)N1C(CCCC(=O)NC2(C(=O)OC)CCCCC2)CCC1 c1(C(N2CC(NC(c3[nH][nH]c(=N)c3Br)=O)C2)=O)ccc2sncc2c1 c1(C(=O)NC2(CC)CCN(C(c3cc(C)n(C)c3)=O)CC2)cc(F)c(C)cc1F c1(NC(C(F)F)Oc2cccnc2)nccc(=NCC2=CCCOC2)[nH]1 Cc1nc(-c2ccccc2)[nH]c1C(=O)Nc1ccccc1OC(C)C N1(C(COC2(C)CCC2)=O)CCCC(NC(=O)C(C)(F)c2ccon2)C1 C1(CNC(Cc2ccc(C)cc2C)=O)CC2CCCC2N1C(=O)CCC1(C)CC1 C(CCC(C)(C)C(=O)N1CC2CCC(CNC(=O)C3=C(Cl)CCC3)C2C1)OC C(=O)(C1=CC2CCCCC12)N1CCN(C(c2cnn(C)c2Cl)=O)C2(C1)CC2 Cc1ccn(CC(=O)NCC2(CNC(c3cncc(Cl)c3Cl)=O)CC2)c(=O)c1 c1(C(=O)NCC2C(CNC(CC(COC)COC)=O)C2)cn2c(n1)CCC(C)C2 N1(C(CCC2CC(NC(c3cncc(C)c3)=O)C2)=O)CC2COCC2C1 N1(C(C(c2ccc(C)o2)C)=O)CC=CC(NC(c2ccc(Br)s2)=O)C1 c1(OC)ccc2[nH]c(=NCCCCCCCO)nc(N3CCC(F)C3)c2c1 N1(C(C2CC3CCN(CC(C4CCCCC4)O)CC23)=O)CCCC2C1CCN2CCO C=C(C)C1OCCC1C(N1CCC(CCC(N2CCCC2C(O)CO)=O)C1)=O c1(C(=O)NC2C(C)CCN(C(c3c(C)c(O)ccc3)=O)C2)cc2ncccc2o1 Cc1cccc2cc(C(=O)NC3C4CCN(C(=O)CC(C)(C)O)C34)oc12 N1(C(c2cc(SC)oc2)=O)CCCC(CNC(=O)C(c2ccccc2)F)C1 c1(C(N(CC(CNC(Cn2ncc(C)c2)=O)O)C)=O)cc(F)c(Cl)cc1F Cc1ccc(Cl)c(OCC(N2CC3CC3(CNC(C3(CF)COC3)=O)C2)=O)c1 C(=O)(CCC1=CCc2ccccc21)N1CCC(NC(C=CC=CCC)=O)C(F)C1 c1(C(=O)NCCC2(NC(c3csc(CN4CCCC4)n3)=O)CC2)ccc(Cl)cn1 c1(C(=O)NC2CN(C(C)(C)C)C(=O)C2)cc(Cl)c(Cl)c(C(N)=O)c1Cl c1(C(N2C(CNC(=O)CC3C=CCC3)CC2)=O)ccc(-c2ccccc2)nc1 C1(CC(=O)NC(CSC)CO)CN(C(C2(OC(C)=O)CCOC2)=O)CC12CC2 Cc1cc(Br)cc(C(N2CCOCC2C2CCC2)C(=O)NC2CC2)n1 Cc1cc(C(=O)N(C2CN(C(=O)Cn3nccn3)CC2F)C)nn1C(C)C N1(C(CC(C(C)C)OCC)=O)CC2(CCC(NC(c3cnc(Cl)s3)=O)CC2)C1 c1(C(C)OC)ncc(C(=O)NC2CC(N(C)C(c3cccn3C(C)C)=O)C2)s1 c1(C(N2CCC(F)(CNC(=O)C=CCF)CC2)=O)ccn2cnnc2c1 c1(CC(=O)N(C2CCC(NC(CCCC)=O)C2)C)ncn2c1CCC2 C1(N(C(C(C2CCC2)OC)=O)C)CCCCN(C(c2ccc(C(N)=O)cn2)=O)C1 C1(CC(=O)NCC2C=CCN2C(c2cc(C3CCC3)[nH]n2)=O)CCCC2CC12 C(CN=C(NCC(OC)OCC)NC1CC(O)C12CCC2)C1(CNCC)CC1 c1(NC(C2CCN2Cc2cc(F)c(F)cc2Br)=O)cc(Cl)c(O)cc1Cl CC1CC(NC(=O)CCOC2CCCCC2)CN1C(=O)CCc1cncc(F)c1 c1(C(=O)NC2C(SC)CN(C(c3cc(Cl)no3)=O)C2)cc(C)c(C)cc1C c1(C(=O)NCCCCNC(C(C)NC(CC)=O)=O)ccc(S(=O)(=O)NOC)cc1 C=CC(CC)CC(=O)N(CCCNC(=O)Cc1ccc(CC)c(F)c1)C c1(CNC(C2(C=C)CCC2)=O)cc(C(=O)NCC(C2CCCC2)O)ccn1 C12(C(=O)NC3CN(C(CNC(=O)CC(F)(F)F)=O)CC3O)CCCC(C1)OC2 CC#CCCCC(=O)NCC=CC(=O)NCC(CC)C(C)(F)F c1(C(N2CC(C3N(C(CC=C)=O)CCC3)(O)C2)=O)cc([N+](=O)[O-])nn1C C(=O)(CCCC(=O)N1CCC(C(=O)NC(c2ccccc2C)C)C1C)OC N1(C(C2CCC(=O)N2)=O)CC(NC(c2cc3cccnn3n2)=O)CC12CCOC2 C1(CNC(CC)=O)CN(C(c2cccnc2OC(C)C)=O)CC1C CC1=C(C(=O)NC(CC2CC2)CC(=O)NC(CN(C)C)CCO)CCCO1 C(C1(O)CCc2cc(F)ccc21)NC(c1cc(C2CCC2)[nH]n1)=O N1(C(CCC)=O)CC(NC(=O)CCc2ccoc2)CC2(CCC2)C1 N1(C(CC2C(C)(C)COC2)=O)CC2CC1CN2C(=O)CCOCC(F)(F)C(F)F C12(C(N3CC(O)(CN(C(=O)CC4C=CCC4)C)C3)=O)CC3CC(CC(C3)C1)C2 N1(C(c2nc(C)oc2)=O)CCC(C)(C)C(NC(c2ccc(OC(F)F)nc2)=O)C1 CCCCCC(=O)OC(C)(C)C.C(CCCCCn1cc(C(C)N(C)CCO)nn1)N c1(C(N2CCC(CN(C(c3c(C)scc3)=O)C)C2)=O)ccc2c(c1)CC2 CC1(C)CC(CO)N(C(c2ccc(CNC(C3CC3[N+](=O)[O-])=O)nc2)=O)C1 C(=O)(CCC(C)O)NC(CNC(CCN(CC)CC)=O)C(C)C c1(OCC)ccc(C2(C(=O)NC)N(C(C3CC4CC4C3)=O)CC2)c(C)c1 C1(C(=O)NC(C(=O)OC)CC#N)C=C(c2ccc(Cl)cc2)CC1 C1(C(N2C3CC(C(N4CCCC5(CC5)C4)=O)C2CC3)=O)C2Sc3ccccc3C12 N1(C(C(CC)C)=O)CCC2(CCCN2C(=O)CCNC(c2cccs2)=O)C1 N1(C(C2C(C)=CCC=C2)=O)CCCCC(N=c2nc[nH]cc2C#N)C1 c1(N(C)C)nc(Cl)c(C(=O)NCCCCCNC(C2(CO)CCOC2)=O)s1 C1(NC(c2n(CC)ccc2)=O)CC(O)CN(C(=O)CC2CCC=CCC2)C1 N1(C(C(CC)(F)F)=O)CCCC(F)(C(=O)NCCNC(=O)NCC)C1 N1(C(=O)CC2CCCCO2)CC2(CCCN2C(c2cccc3ncsc23)=O)C1 c1(C(C)C)cc(C(=O)NCC(CO)NC(c2sccc2OC(F)F)=O)n[nH]1 C1(NC(c2nc(C(C)C)oc2)=O)CC2CC(C1)N(C(C1(C)CC(O)CN1C)=O)C2 C1(NC(=O)C(F)C2CCOC2)CC1C1CCCN(C(c2c[nH]cc2C2CC2)=O)C1 N1(C(C2C(C)C2(F)F)=O)CC(NC(=O)C=C2CCN(C)CC2)C(O)C1 C1(CC)(Nc2nccc(CO)n2)CCN(C(C2(CF)CC2)=O)CC1 CCC(C)(COC)C(=O)NN1CCCC1C(=O)NCCC1CC(C)C1 C1(NC(=O)CCN2CCCCC2)CCCC12CN(CC(=O)N(CCO)CC1CC1)C2 N1(C(C2C(CC)CCC2)=O)CCC(C)C(NC(=O)CC(C)(C)CC)C1C Cc1cnc(CCC(=O)NCC2CCN2C(C2CSCCS2)=O)[nH]1 N1(C(N2CC(C)C(C(=O)OC(C)(C)C)C2)=O)CC(C)C(F)(F)C1 C=CCC(CC(F)F)NC(C1C(CC)CCCN1C(=O)COC1CCOCC1)=O CC(C)CCC(C(=O)NC1(C(=O)N(C)C)CC1)NC(=O)CCC(C)(C)N(C)C N1(C(Cc2c(C)ocn2)=O)CCOC(CN(C)C(C2CCC(=O)N2C)=O)C1 N1(C(Cc2cc(C)n(C)n2)=O)CCN(C(c2ccn(C(C)C)n2)=O)CC(C)(F)C1 C1(NC(C2(CC#C)CCCC2)=O)CCC(C)N(C(=O)Cn2cc[n+](C)c2)C1 CC1CN(C(=O)Cn2cc(C#N)cn2)CC1NC(=O)C(C1(O)CCCC1)F Cc1ccc2c(=NC(=O)NCC3CC3C3CC3)[nH][nH]c2n1 N1(C(c2c(C)n(C)c(-c3ccccc3)c2)=O)CC23CCCC2(COC3)C1 C(=O)(C1CCc2cccc(OC)c21)NC(CC=C)CNC(=O)Cn1cc(Cl)cn1 CC1(C)CC(C(=O)NC2CNC(=O)C2)CCN1C(=O)C(F)=CC1CC1 Cc1[nH]cc(C(=O)NC2CN(C(=O)C(C)C3(O)CCC3)CC2(C)C)c(=O)c1Cl C1(C(=O)NC(CN(C(c2occ(C)c2)=O)C)(C)C)CC12CC(O)C2 C#CC1(C(=O)Nc2ccc(OC)nc2)CCN(C(=O)C#CC2CC2)CC1 C(=O)(CCCCNC(C1CCCCN1C(c1ccc(F)s1)=O)=O)OCC N1(CC)CCC2(CC1)CC(Cn1nc(-c3ccsc3)nc1C(=O)OC(C)C)=NO2 C1(C(=O)NCCN(C(C2(O)COC2)=O)C2CC2)CCCC1n1cccc1 C1(CNC(C2COC3COCC23)=O)CCC2(CN(C(=O)CC3CCOCC3)C2)O1 C1(SC)CN(C(=O)CC2CCCCC2O)CC1NC(=O)CCc1ccncn1 c1(C(=O)NC2CN(C(C(C(CC)O)(F)F)=O)CC2O)sc2cccc(F)c2c1Cl C1(NC(c2cnc(S)[nH]2)=O)CC2CC(C1)N(C(c1ncsc1Br)=O)C2 Cc1nccc(CNC(=O)C=CCC(C)(C)NC(=O)Cc2cc[nH]n2)n1 C(=O)(CCCC(CC)NC(=O)C1=C(C)OCC1)N(C1CC(SC)C1)C c1(C(N2C(CNC(C(C=CC)O)=O)CCC2)=O)cnc2cnn(C)c2c1 C1(C(=O)Nc2scc(C)n2)CC12CCN(c1ncnc(C)c1Br)C2 N1(C(c2cn(C)cc(Br)c2=O)=O)CCCC(N=[N+]=[N-])CC1 C(=O)(C=C1SCC(=O)N1C)N1CC(NC(C(CC=CCC)C)=O)C(OC)C1 C12(C(=O)NC3C(C=C)OCC3)COCC1CN(C(=O)Cc1cccc(F)c1)C2 c1(N2C(C)(CNC(C(C)NC(C)=O)=O)CCC2)ncc([N+](=O)[O-])cc1F CCCC(C)(C)C(=O)NCC1(O)CCCN(C(c2nccc(Cl)c2O)=O)C1 C1(C(=O)NCC2CCC(NC(COCC(C)C)=O)C2)CC2CCC(C1)C2(F)F C1(OC)CC(CCNC(=O)CN2CCC2C)N(C(C2CCC=CCC2)=O)C1 n1(-c2c(C)ccc(C)c2)nc(-c2cccc(Br)n2)nc1C1CCc2c[nH]nc21 c1(CC(=O)N(CC(C)N(C)C(C2CCC23CCC3)=O)C)c(F)cccc1F c1(NC(C2(C)N(C(c3cc(C)on3)=O)CC2)=O)ncc(Br)nn1 C1(C(N2CC(C(=O)NCC(C3CCCCC3)C)(SC)C2)=O)CC2C(C1)C2(C)C C1(N(C(c2c(OC)csc2)=O)C)C2CN(C(C3CC(F)(CF)C3)=O)CC12 C(=O)(CCCCC(C)(C)C)N1CC(NC(C(CCCC)CC)=O)C2(C1)CCC2 C1(CCC=C)(C(=O)NCC(O)CO)CN(C(=O)Cc2ccc(Cl)s2)C1 C(C1CCCC1)=C(C)C(=O)NC(C)C(=O)NC(C)Cc1nn[nH]n1 c1(CN(C(CN2CCC(CCCC)C2)=O)C)ccccc1Cl C1(NC(c2cc(C)nn2C)=O)CCN(C(c2sc(Cl)cc2Cl)=O)C(C)C1 N1(C(C)C(N2CCCC2CNC(=O)CC2CCN(C3CC3)CC2)=O)CC2CCC1C2 N(C(=NCCC(=O)OC(C)C)NC1CC(=O)N(C(C)C)C1)CC(CC)(C)OC N1(C(Cc2c(C)nsc2)=O)CC2CC1CN2C(=O)Cc1sc(=N)[nH]c1-c1cccs1 Cc1nn(C2CCCCC2)cc1C(=O)NCC12CC(CN1C(=O)C=C(Cl)Cl)C2 C1(NC(CC2C(C)OC(C)C2)=O)CCN(C(=O)Cc2nncs2)CC1(C)C c1(N2C(C3CCN(C(CC=C)=O)C3)CCC2)cc(OC)nc(OC)n1 C1(CCC(=O)NC2CC(N(C(=O)C(N3CCOCC3)C3CC3)C)C2)CCCN1C CCC(C(=O)NC(C1CCN(C(c2[nH]nnc2C2CC2)=O)C1)C)c1ccccc1 C1(CNC(c2c(C)nn[nH]2)=O)CN(C(=O)CCc2nncs2)CC1O C(=O)(CCC(F)F)N(CCNC(C(C)SC(C)C)=O)C(C)C c1(C(N2CC(NC(c3cnc(CC)[nH]3)=O)C(C)CC2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(C(N2C(C3(NC(C=CC=CC)=O)CC3)CCC2)=O)CN2CCC1(C)CC2 CC1(C)CCCC(C(=O)NCCC2(NC(c3cnc(O)s3)=O)CCC2)CC1 C1(NC(C(c2ccc(C)cc2)(F)F)=O)COCCN(C(c2cn(C)cc2C)=O)C1 C(CC(=O)OCc1ccco1)(C(F)(F)F)N1C(C)CCC1 c1(NC(C)CCN2CCOCC2)nc(N(CCC#CCO)C)nc2c1CCC2 c1(NCCN(C(C2CC(C#C)(O)C2)=O)CCC(C)=O)ccc(Cl)c(Cl)c1 C1(NC(c2ccc(CN(CC(N)=O)C)cc2)=O)CCOC12CCOCC2 c1(C(=O)NC(C)C(C)NC(C2CN(C)C2)=O)cnn(-c2ccccc2)c1 C1(NC(CCc2c(C)n(C)nc2)=O)CCN(C(c2nonc2N)=O)CC(C)(C)C1 Cc1c(C(N2CCOCC(CNC(C3(C)CCCN3C)=O)C2)=O)sc2cncn12 CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CC1(C)CNC(=O)C(c1ccccc1)F C1(CC(=O)NC(C(C)n2cccn2)C)CCCCN1C(C1OC2CCC1C2)=O c1(C(=O)NC(c2ccccc2)CNC(C2(C(C)C)CC2)=O)ccc(N)cc1Cl N1(C(CSC(C)(C)C)=O)CC2CCC1C(CNC(=O)C1CC1)C2 CCCC(C(=O)N(C)Cc1ccc(C)cn1)NC(c1ccccc1)=O C1(C(=O)NC2(C)CCN(C(c3nn(C)c(Cl)c3Cl)=O)C2)Cc2cc(F)ccc2O1 C(=O)(C(CC(C)C)C(N)=O)N1CC(C(C(=O)N(CC=C)CCOC)OC)C1 Cn1nc2c(c1C(=O)Oc1c(F)cc(OC)cc1F)CN(Cc1ccc[nH]1)CC2 CC1CCCN(C(=O)C2=CCOC2)C1CNC(c1ccoc1C(F)(F)F)=O c1(C(=O)NC2CN(C(C(CCC)OC)=O)CC2C)cc(S(N)(=O)=O)cs1 CCCC(CC)CCC(=O)NC1CN(C(c2ccc(C#N)o2)=O)CC1O N1(C(C(CO)NC(C2N(C)CC(O)C2)=O)=O)CCC(C2CCC2)CC1 C1(C(C)NC(c2coc(CO)c2)=O)CN(C(C2CSCC(=O)N2)=O)CCO1 C(=O)(CC1=NNC(=O)C1)N1CC(C)C(CNC(c2cc(Cl)cc(F)c2N)=O)C1 Cc1cc(F)c(C(=O)NCCCNC(N)=O)cc1Br.C(C)(CCSC)NC C1(CCC(=O)NCCOCC#C)CCN(C(c2c[nH]nc2OC)=O)C1 C1(CNC(CN(C(C)=O)C)=O)(NC(c2ccnc(C(F)F)c2)=O)CCCCC1 c1(CO)ccc2ccccc2c1C.C12CC1C(=O)N(CCC)CCN(CC)C2=O CC(=O)CCCC(=O)NCC1CCN(C(c2coc(C(N)=O)c2)=O)C1 c1(C(=O)NCC(C)C(=O)O)ccc(F)c(-c2cn(CC3(O)CCSC3)nn2)c1F c1(C(=O)NCCC(C)NC(c2cc(C)oc2)=O)oc2c(C)ccc(C)c2c1C C#CCC(C(=O)N(C1(C)CC1)C)NC(C1CCCN1C)=O C1(F)(C(=O)NCC(c2ccccc2)N(C(C=C(CCC)C)=O)C)CC1(F)F CC(O)CCCCCC(=O)Nc1ccccc1CN1CN(C)C(=O)N(C)C1 C1(NC(C2(CCCC)CCC2)=O)CN(C(=O)Cc2cccc(C(F)F)c2)CC1O c1(C(=O)NCCC(CNC(c2c(C)ccnn2)=O)O)c[nH]c(=N)nc1C N1(C(CNC(=O)NC)=O)CCN(C(c2cc(O)nc(C)n2)=O)C(C(C)C)C1 CC(C)CCCC(C)C(=O)N(C)CC1CCN(C(C2COC(=O)N2)=O)CC1 C1(NC(=O)CCC2CCC2)CCCC2CN(C(=O)CNS(N)(=O)=O)CC12 CCCC(C)C(=O)N1CCC(F)(C(=O)Nc2nccnc2C)C1 c1(NC(C2CCCN(c3cc(C)nc(C)n3)C2)=O)ccc(C(F)(F)F)c(F)c1C C1(NC(C(CCN(C)C)O)=O)(CO)CCCN(C(=O)C(c2cccc(N)c2)O)C1 N1(C(C(C(CC)CC)C)=O)CC(CNC(=O)C=Cc2ncc[nH]2)OC2COCC12 C1(C(=O)NCCN(C(c2cc(COC)on2)=O)CC)CCOC(C)C1 CC1CCN(C(C2CC(NC(c3cc(Br)c(F)cc3F)=O)C2)=O)CC1(F)F C1(NC(=O)CCC2CCCC2)CN(C(C2(CC3CC3)CCCO2)=O)CC1F c1(OC)ccc(CC(=O)NC2CC(F)CN(S(=O)(=O)C(C)COC)C2)cc1F C1(NC(Cc2c(C(=O)OC)csc2)=O)C(C)CCN(C(=O)CNC=O)C1C C(C1=CCN(C(C2(F)CCCCCC2)=O)CC1)NC(c1ncc(Cl)cc1F)=O C(CC(=O)NC1CCC(CO)CC1)(C(C)C)NC(c1c(CC#N)cccc1)=O C1(C)(C(=O)NC(C23CCC(CC2)C3)CNC(CCNC(C)=O)=O)CCCS1(=O)=O C1(NC(C2CC(CCC)OCC2)=O)CCCC2CN(C(=O)C(C)=CC3CC3)CC12 C1(NC(COCC)=O)CS(=O)(=O)CC1N=c1ccnc(-c2cccc(Cl)c2)[nH]1 N1(C(c2c(NC)snc2C)=O)CC(NC(=O)CCc2ccccc2)CC(O)C1 C1(CNC(Cn2cc(C(C)=O)nn2)=O)CC(NC(C2C3COCC23)=O)CCO1 c1(C(=O)NC(C(C)C)C(=O)NC(C)CS(C)(=O)=O)cccc2ccoc12 N1(C(CC2(C=C)CC2)=O)CC(CNC(c2nnc(S)n2C)=O)OC2(CCC2)C1 C(c1ccc(C#N)cc1)=CC(=O)NC1CCC(C)N(C(c2cccc(=O)o2)=O)C1 N1(C(C=C(C)CCc2ccccc2)=O)CC2OCC(NC(=O)C3=CCCS3)C2C1 CCC(O)C(F)(F)C(=O)NC(C1CC(NC(c2coc(C3CCC3)n2)=O)C1)C c1(NC(C(c2cc(O)cc(Cl)c2)N2CCC(C(=O)NC)C2)=O)ccc(Cl)cc1F C1(C(N(CC(C)N(C(C(C2CC2)SC)=O)C)C)=O)CC2(C1)OCCO2 c1(C(N2C(CNC(c3c(CC)non3)=O)C(C)CC2)=O)cncc(S(N)(=O)=O)c1 N1(C(c2c(C)n(C)nc2)=O)CC(F)(F)CC1(C)CNC(=O)Cc1ccnnc1O C1(NC(C=CCC)=O)CCC(N(C(=O)C(C(C)C)Oc2ccc(Cl)cc2)C)CC1 C12(C(N3CC(C)(NC(CC(C=C)C)=O)C3)=O)CCCN(CC1)S2(=O)=O c1(C(=O)NC(C2(O)CCN(C(=O)CSCC(N)=O)CC2)C)ccccc1[N+](=O)[O-] C12(CNC(=O)Nc3c(C)c(Cl)ncn3)CCC(CC1)C(C)(C)O2 N1(C(C)C)CCOC(CN2CC(CNC(c3cccc(C(N)=O)n3)=O)C2)C1 Cc1[nH]nc2c1CC(C(N1CC(CNC(=O)CCCCNC(N)=O)C1)=O)CC2 CCCC(C)(CCC)C(=O)NCC12CC(CN1C(=O)C(C)CCC(C)(C)C)C2 Cc1ccnc(C(N2CCOC(C(C)NC(C3CC(C)(C)C3)=O)C2)=O)n1 CC1CN(C(c2c(Cl)nsc2Cl)=O)CCCN1C(c1ccc(C(N)=O)cc1)=O C1(CC)CCCCN1C(=O)CC1C=CC(NC(=O)Cc2ccc(C)o2)C1 Cc1cc(C(=O)NC2COCC2NC(C2(C)CCC(C)C2(C)C)=O)cc(C)c1N CCC(CS(C)(=O)=O)NCc1cccc(-c2nncn2CC)c1 c1(C(N(C2CN(C(C(CC=CC)CC)=O)CC2(C)C)C)=O)[nH]cc2c1CCCC2 c1(C(N2CC(C)(NC(C(CC)C(C)C)=O)C2)=O)cc2c(o1)CCCNC2=O C12(C(=O)NC(c3cn(C)nn3)C)CCC(CC1)N(C(C1CCOC1(C)C)=O)C2 CCCCCCNC(=S)NC(C)C c1(C(=O)NCC(CC=C)NC(c2ccc(COC)o2)=O)ccc(Cl)nc1 Cc1ccc(C(=O)NC2CCOCC2NC(=O)CCNC(C2CCC2)=O)c(F)c1 c1(OC)cc(C(=O)NC(C)CN(C(=O)CCc2ccc(N(C)C)cc2)C)ccn1 C(CC(C)C(F)(F)F)NC(=O)NCC1CC(C)SCC1 C1(NC(c2ccc(C)cn2)=O)CCC2CN(C(c3cc(Cl)cnn3)=O)CC2C1 c1(C(=O)NCCCCC(C)NC(c2c(C)sc(O)n2)=O)cnn2c1CCCN2 N1(C(C(COC)O)=O)CC2(CC(NC(c3cnc(OC)cc3C)=O)CO2)C1 c1(C(=O)NC(C2(O)CN(C(C3CC(F)CN3C)=O)C2)C)c[nH]c2ccc(F)cc12 C(=O)(C1=Cc2ccccc2OC1)N1CCN(C(CC(C)N(C)C)=O)C2(C1)CC2 Cc1ccn2ncc(C(=O)NC3CC(NC(c4cc(CO)[nH]n4)=O)C3)c2c1 C1(NC(CN2C(C)CC2)=O)CCN(C(C2CCN(CCC3CC3)CC2)=O)C12CC2 C1(C(=O)NC23C(NC(C(C)=C4CC4)=O)CC(CC2)C3)CCn2nnnc2C1 C#CC(CC(C)(C)C)NC(=O)C(C)N(C(C1(C)CC(C)(C)C1)=O)C1CC1 N1(C(c2cc(C3CCCC3)no2)=O)CCCC(N(C(=O)CCC(F)F)CCO)C1 c1(N2CCC(COC)CC2)ccncc1S(=O)(=O)NCC1COC(C)(C)O1 N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(c3c(C)[nH]c4ccccc34)=O)CC12 c1(NCC2C(NC(C(CC)OC)=O)CCCC2)cc2nncn2c(C)n1 Cc1nc(-c2ccccc2)oc1C(=O)NC(C)CNC(=O)CC(C)CN(C)C Cc1ccnc2c1N(C(c1cc(Cl)ccc1CN1CCCC(O)C1)=O)CCO2 CCCC(O)CC(=O)N1CC(NC(c2ccc(OCC)cc2)=O)CC1(CC)CC C1(CNC(CCSCCN(CC)CC)=O)C(O)C(O)CN1C(=O)CCS(C)(=O)=O N1(C(C2N(C)CCC2)=O)CC2CC2(CNC(=O)C(C)(C)c2ccns2)C1 C=C(C)C1OCCC1C(=O)NC1C2CC1N(C(c1cnncc1C)=O)C2 C1(NC(c2cc(C(F)F)[nH]n2)=O)CCC2CC1CN2C(c1cnn(CCF)c1)=O C(=O)(CC(C(=C)C)OCC)NC1(CO)CCN(C(CCC(=C)Br)=O)C1 C1(C(N2CCC(CN(C(=O)Cc3cnsc3)C)C2)=O)CC(c2ccncc2)=NO1 C1(CNC(c2c(C)n(C)nn2)=O)CN(C(=O)CC2CCCOC2)CCN1C N1(C(C=C(C)CCc2ccccc2)=O)CC(NC(=O)CC(C)C)CC(C)(C)C1 C1(C2CCCC2)(NC(C2C=CC(NC(=O)CC3CCC=CCC3)C2)=O)CC1 c1(NC2CCCN(C(C(CC)NC(N)=O)=O)C2)ncnc2c1ncn2CC C=CC1CCCN1C(=O)C(C)(CO)NC(C1COCC1C(N)=O)=O C(=O)(C(O)C(F)(F)F)N(C)CCN(C(=O)CCc1cc[nH]n1)C c1(C(c2n(CCC)nnn2)NCc2nnc(C(F)F)s2)ccc(S(C)(=O)=O)s1 CC1CN(C(C2OCCC2NC(=O)CC2CC(F)C2)=O)CCC1(F)F C1(C(C)NC(C=CCC)=O)CCN(C(=O)CC(=O)NCC)CC1 N1(C(C(C)OCC=C)=O)CC(C)(CNC(C2CC2c2ccnn2C)=O)CC1(C)C c1(C(=O)NC(CNC(C2(CC=C)CCOC2)=O)C)sc(C2CCCC2)nc1C C(=O)(C1=NOC(CNC(c2ccc(C(N)=O)[nH]2)=O)C1)NC(CN(C(C)C)C)C N1(C(C(=O)NCC)=O)CC(C)C(NC(=O)Cc2c[nH]c3ccccc23)C(C)C1 C1(CSC)CCCN(C(c2ccc(Br)cn2)C(=O)NCCCSC)C1 CCC(CNS(C)(=O)=O)N=c1[nH]c(=NCC(CC)n2cccn2)[nH]c2cc[nH]c12 N1(C(C(C)OCC2CC2)=O)CC(O)C(O)C1CNC(=O)C(C)(F)F N1(C(=O)OC(C)(C)C)CCCCC12CCCN(C(C1CC1(C)C)=O)C2 N1(C(C(C=C)(C)CC)=O)CC2CCN(C(=O)CC3(OC)CC3)CCC2C1 C1(NC(c2ccc(CC)nc2)=O)COC2(C1)CN(C(c1cc(N)ccc1C)=O)C2 c1(CC(=O)NCCCCCNC(c2ccc(C(C)=O)o2)=O)ccc2[nH]ccc2c1 O=C(CCCc1ccncc1)NCCCNC(c1cc(CO)on1)=O c1(OC)cc(C(=O)NCC#CCNC(=O)COC(C)C)c(Cl)cn1 C(=O)(C1=CCC2CCC1N2C(C1(C)CC2CC2C1)=O)NCc1cc(OC)no1 c1(OCC(=O)NCCN(C(C2CC(N3CCCC3)C2)=O)CC)cccnc1 CCCCCCCCCC(O)C(=O)N1CCCC(NC(c2cnc(C)[nH]2)=O)C1C C1(CNC(c2cc(SC)ncc2)=O)C(C)CCCN1C(c1occc1C)=O C(=O)(C(C)CCC(C)(C)C)N1CCC(O)(CN(C(c2c(C)nc[nH]2)=O)C)C1 c1(OC)cncc(CCC(=O)NCC(O)CCNC(C2CCCC2C(C)C)=O)c1 N1(C(Cn2ccc(C)n2)=O)CCC2(CCCN(C(c3cc(C#N)[nH]c3C)=O)C2)C1 N1(C(c2cncc(OC)n2)=O)CCC(NC(=O)CC2CCC(=O)N2C)CC1C c1(C(=O)NCC(CC)NC(c2ccccc2COC)=O)c(C)nn(CC(C)C)c1Cl Nc1c(C(=O)NCCNC(c2[nH]nnc2-c2ccccc2)=O)cccc1F C1(C(C(C)NC(=O)CN(C)C(C)=O)OC)CCCCC1 c1(-c2cccc(CN(C(C)C)C)c2F)ccc([N+](=O)[O-])cc1O C1(C(=O)NC(CC)CNC(=O)Cc2cnn(CC)c2)C(C(F)(F)F)C1[N+](=O)[O-] c1(NC2(C(=O)NCCNC(C)=O)CC2)cc(C(C)C)cc(N)c1 C(=O)(C(F)C1=CCCCC1)N1CC2CN(C(c3c(C)nsc3N)=O)CC2C1 C1(C(=O)NCC2CC(C)(C)C2)CCN(C(=O)CCCCN(C)C)CC1O N1(C(c2c(CC)nco2)=O)CCN(C(C2CCC(=O)N(CC)C2)=O)CCC1C c1(C(N2CCC(COC)(NC(=O)CCc3nnc(C)o3)C2)=O)cc2n(n1)CCC2 c1(NCc2c(-n3cccn3)c(C)n(N)n2)nn(C)c2ccccc12 N1(C(C(COC)(C)C)=O)CCCC2(C1)C(NC(=O)C1=CSCCO1)CCN2C C#CCC(C)(C(=O)N1CCCCC1C)NC(c1cc(C)ccc1C)=O N1(C(c2n(C)ccn2)=O)CC2CCC1C1CN(C(=O)CCc3ccnn3C)CC21 c1(C(N2CC(CNC(c3c(C)csc3)=O)OCC2)=O)cc(Br)c(F)cc1F C1(C(=O)NCCC2(NC(c3cnc(O)s3)=O)CCC2)(CC)CCCCC1 c1(NC(c2c(C(=O)OCC)c[nH]n2)=O)ccc(NC(=O)C(C)C2CCOC2)cn1 C(CCCCC(=O)N(C(C)(C(=O)NCc1ccc(F)cc1C)C1CC1)C)OC NS(=O)(=O)c1cc(C(N2CC(OCCNC(=O)C(F)(F)CO)C2)=O)co1 n1(C(C)C(=O)N(C2CCCS2)C)cc(C(C)(C)CC2CC2)nn1 N1(C(C2C(C)CCO2)=O)CCOC(C(=O)NC(C2CCOC2)CO)C1 N1(C(C(=O)NC2(C)CC(C)(C)OC2=O)=O)CCC2C(CCCC2(F)F)C1 N1(C(C(=C)F)=O)CCC12CN(C(=O)CCc1ccccc1OC(F)(F)F)C2 c1(OC)nscc1C(N1CC(O)(C2CCCN2C(c2ccsc2Cl)=O)C1)=O c1(C(=O)NCC(C(=O)Nc2ccc(OC)cc2)OC)ncnc(O)c1F C(CC(C(=O)N(C1CCCC1C#N)C)NC(=O)C1=CCCC1)OCC c1(C(=O)NC(CN(C(=O)CCN2CCOCC2)C)(C)C)snc(Cl)c1Cl c1(C(=O)NC2(CF)CCN(C(CCNS(C)(=O)=O)=O)C2)ccc2c(c1)B(O)OC2 c1(SC)c(NC2(c3nnnn3C3CCCC3)C(OC)CCC2)cnnc1COC N1(C(=O)Nc2csc(Br)c2)CC(CO)CC12CCOCC2 CC1(C)CCN(CCNC(c2ccc(CNC(C3CC3(F)Cl)=O)o2)=O)C1 c1(C(N2CCC(F)C2)C(=O)NC2CCOC2)ncc(C2OCCO2)s1 C1(c2nc(C(c3ccoc3)OC)on2)(c2cccs2)CCCCC1 c1(OC)ccc(C(=O)NC2CC3CC2N(C(=O)C(C)(C)C#N)C3)cc1C(F)F CCCCCCCCC(=O)N1CCOCC1CN(C(=O)C(C)(CC)CO)C CC1(C)CCCC1CNC(c1[nH]ccc1-c1cccs1)=O C=CCCCC(C(=O)NC(CC)C(C)(C)C)NC(=O)COCCF c1(NC(=O)NNC(=O)c2ccccc2)cc(F)c(F)c(F)c1 C(=O)(CCCNc1cccnc1)N1CC(OCCNC(c2cnns2)=O)C1 c1(C(N2C(COC)CN(C(=O)C=CBr)CC2)=O)ccnc2ccccc12 C#CC12CCC(C(=O)NC3CN(C(C4COC4)=O)CC(C)(C)C3)(CC1)CC2 C(CNC(C1CN(C2CCC2)C1)=O)(CCOC)NC(C1(OC(C)C)CCC1)=O C1(C(N2CC3CC(CN(C(CNS(N)(=O)=O)=O)C3)C2)=O)CCCC2(C1)CC2(F)F CC(C)S(=O)(=O)c1ccccc1NC(=O)CC1(C)CCN1Cc1cccnc1Cl N1(C(c2cccc(N)n2)=O)CCC2(NC(c3ccn4ccnc4n3)=O)CCCC12 c1(CC(=O)NC2CCN(C(C3CC(C)N(C)C3)=O)CC2)c[nH]c2ccncc12 c1(C(C(=O)NCCNC(C2CCC2)=O)C)cccc(C(=O)OC)c1 N1(C(c2cc(C)ncc2C)=O)CCCC2(CCC2NC(c2cnccc2C)=O)C1 C12(NC(=O)CN3CC=CC3)CCOCC1CN(C(c1cccc(C(F)F)c1)=O)C2 c1(OC)ccc(-c2cc(CN(C3C4CN(C(=O)C(O)CCl)CC34)C)n[nH]2)cc1 CC(C(=O)NCCC1CN(C(c2cc(Cl)c(Br)cn2)=O)C1)C(C)(C)C CCC(C)C(C(=O)NC1CC(NC(c2coc(-c3ccccc3)c2)=O)C1)OC c1(C(=O)NC2C(NC(c3cn(CCC=C)nn3)=O)COC2)cncn(C)c1=O N1(C(CCCOCCC)=O)CCCC(CO)(NC(c2oc(CC3CC3)nc2C)=O)C1 C1(COC)CN(C(c2c(C3CC3)noc2C)=O)CCN1C(c1cscc1C)=O C(=O)(C1CCc2nccn21)NC1(CC=C)CCN(C(c2coc(C(F)F)c2)=O)C1 C1(NC(C2CC(NC(c3ccccn3)=O)C23CCC3)=O)CCc2nncn2C1 C1(NC(C(C(C)C)OC)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1F Cn1cnc(CC(=O)NCC(C2CCOC2)NC(=O)COC2CCC2)c1 c1(C(N2CC(CCNC(C(C(CC)C)O)=O)C2)=O)ccc(F)c(S(N)(=O)=O)c1 c1(CC)ccccc1CCNC(C1CC1CCCC(=O)OC)=O.C(F)(F)F CC(C)CCC(=O)NCC(=O)NC1C=CCN(C(=O)COCC2CCOC2=O)C1 n1(CC)c(CNC(=O)CN(C(=O)CC2CCOCC2)C2CC2)nnc1O C(=O)(C(CC(C)C)OC)N1C(C2(NC(c3c(CC)nc(C)o3)=O)CC2)CCCC1 c1(OC)ccc(C(F)(F)F)cc1CNC12CC(C(N3CCC3(C)C)=O)(C1)C2 c1(C(=O)NC2(CC=C)CCN(C(C3CC(N(C)C)C3)=O)C2)ccc(S(C)(=O)=O)s1 C1(C(c2cn(CCNC(C(C=CCCC)O)=O)nn2)C)CCN(C)CC1 Cn1ncc(C(=O)NCC(c2ccccc2)NC(=O)Cc2sc(O)nc2O)c1Cl c1(C(C)C)ccc(CC(=O)NCC(C)(CO)NC(=O)C(C)C2CCCC2)cc1 C1(CCNC(c2cc(C(F)(F)F)no2)=O)CCCN(C(=O)CC2CCOC2=O)C1 CC1CCCCC1(CO)NC(c1cncc(CNC(=O)CCCN=[N+]=[N-])c1)=O c1(C(=O)NC2CCC(CNC(c3occ(C)c3C)=O)CC2)ccc2nccn2c1 c1(C(N(C2(CNC(=O)CC3(C(F)(F)F)CC3)CC2)C)=O)cnco1 C1(C(=O)NCCC2CC(NC(c3ccc(=O)oc3)=O)C2)CC2CCC1O2 C(C)(C(=O)NCCCn1cc(-c2ccc(C)cc2Cl)nn1)(C(C)C)OC C#CCC(C)(C)C(=O)NCCOCCNC(=O)CCC(N)=O C1(C(=O)NCC2CN(C(C3CCN(C(CC)=O)C3)=O)CC2C)CN2CCC1CC2 CC1(C)CCC(C(=O)NC2(CNC(=O)CCC3CC(F)(F)C3)CCC2)O1 c1(C(c2nnnn2C)NC(CCC)Cn2cncn2)ccncc1COC CC(CN(C)C)C(=O)N1CC(C(O)C(=O)N(C)CCF)C1 c1(C(=O)NCC(CC)(C)NC(c2ccn(C)c2)=O)cc(COC)c(C)s1 C1(C(=O)NC2C(CNC(COC3(C)CCC3)=O)CCCC2)CC(C)(C)C12CC2 C(CC(=O)NCCC(C)OC)(C(F)F)NC(C1(CC)CC(C)(C)C1)=O C1(C(=O)NCC2(C)N(C(c3cc(C)sn3)=O)CCC2)CCc2ccnn2C1 c1(N(CCOC)CCNC(=O)CCN2C(=O)CCC2=O)nccc(C)c1[N+](=O)[O-] c1(NC(C2C3CC2N(C(c2ccc(Br)c(F)c2)=O)C3)=O)ncc(Cl)cc1O c1(C(=O)NCC2CCN(C(=O)Cc3ccc(Cl)cc3F)C2)ccc(Cl)c(Br)c1 c1(C(=O)NC2C(NC(C3CCN(C)C3=O)=O)COC2)cc(F)c2ccccc2c1 N1(C(C(C=C)(C)C)=O)CC(CC(=O)NC2CN(C)CC2C)C2(CC2)C1 C1(NC(COC)=O)CCN(C(c2cc(Br)sc2Cl)=O)C(C)C1 O=C(C1=CC2CCCC12)Nc1ccc(C(=O)OCc2cc(F)cc(F)c2)c(Cl)c1 C(=O)(CCCCCS(N)(=O)=O)NCC1CN(C(c2ccc(OC(C)C)nc2)=O)C1 C(=O)(CC(O)CC(C)(C)C)N1CC2N(C(c3n(CC)ncn3)=O)C(CC2)C1 C(C(C)(C)CC(C)O)NC(C1CN(C(C2(CC=C)CCCC2)=O)CC1F)=O N1(C(C(=O)NC(c2c(Cl)nn(C)c2Cl)C)C)Cc2ccccc2C1CCO CCCCC(CC)CC(=O)NC(CCC)C(O)C(=O)Nc1ccc(OC)cc1F N1(C(C2C(C)OC(C)C2C)=O)CCC(NC(=O)CCCCCO)C2(CCC2)C1 C1(NC(=O)CC(=O)OC(C)(C)C)COCCN(C(CC2CCCC(OC)C2)=O)C1 N1(C(C(CC)SC)=O)CCCC1(CNC(=O)C(C)(C)c1cccnc1)COC C12(CNC(=O)CC3=CCCC3)CCCCC1N(C(=O)COc1ccccc1)CC2 N1(C(C2CC(=C)C2)=O)CCC(O)C(NC(c2c[nH]nc2-c2ccoc2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CC(CNC(c2cnc(SC)s2)=O)CC1(C)C N1(C(C2CCC3(CC3)C2)=O)CCCCC2(C1)CN(C(C1CCCCO1)=O)C2 C1(NC(=O)C(F)CC2CCCC2)CS(=O)(=O)C2CN(C(=O)Cc3ccco3)CC12 Cc1cc(C(N2CCC(CN(C(=O)COCCCF)C)CC2)=O)c(C)nc1C c1(CNCC(C)C2CNC2)ccccc1CNS(C)(=O)=O CCC(C)C(O)CC(=O)NC1(C(=O)NC2CN(C(C)C)CC2C)CCCC1 c1(C(N2CCC(N(C(C=CC(CC)C)=O)C)CC2)=O)ccc(Cl)c(F)c1 C(=O)(CCCCC(F)F)N1CC(F)(CNC(C2(C)N(C)CC(OC)C2)=O)C1 c1(C(N2CC3C(N(C)C(C4CCS(=O)(=O)N4C)=O)C3C2)=O)cc(O)cc(C#N)c1 C1(CC(N2C(C)CN(C(=O)CCc3nncn3C)CC2)=O)CC2(CCCC2)CO1 C(=O)(CCCS(N)(=O)=O)NC1CCC(NC(C(C)Cc2ccncc2)=O)CC1 C1(NC(c2c(OC)csc2)=O)COC2(C1)CN(C(=O)C(C)(O)c1ccccc1)C2 C12(C(=O)NCC(C)CN(C)C(c3cc(F)cnc3O)=O)CCCC1CC(=O)CC2 c1(CC(N2C(COC)CN(C(=O)CCC(=O)NC)CC2)=O)nnc2n1CCCC2 C1(C(=O)Nc2cc(OC)n[nH]2)CCCCN1Cc1cnc(C)cn1 C(C(N)=O)(C(C)CC)N.n1(CC#C)ccc(-c2nccn2C(C)C)c1 Cc1n[nH]c(C)c1C(C)C(=O)N(CC(C)NC(c1ncccc1C(F)F)=O)C C1(C(=O)NC2CCC(CNC(c3scnc3C3CC3)=O)C2)C(F)(F)C12CCC2 N1(C(c2cccc(N(C)C)c2)=O)CC2CC1CC2NC(c1cc(O)cc(Cl)c1)=O C1(C(=O)NCC2C(OC)CC2)CC(c2ccccc2)(NC(C2CC23CCC3)=O)C1 C=C1CCC(C(N2CC3CC3(CNC(=O)C(C)Nc3nc(C)cs3)C2)=O)CC1 C1(C(=O)NC2CC2(F)F)COC2(CCN(C(c3ccncc3Br)=O)CC2)C1 c1(C(=O)NC2(CNC(C)=O)CCCC2)c(F)c(F)cc(F)c1F C1(C(=O)NCC2CCN2C(=O)CN(C(=O)C(C)C)C)(SC)CCC1 C(=O)(C(=O)NOC)NC(c1ccccc1)C(=O)NC1(C=C)CCC1 c1(C(=O)NCC(C2CCN(C(=O)CN3CSCC3=O)CC2)(C)C)ccncc1Cl N1(C(C=CCNC(c2cscn2)=O)=O)CCC(n2cncn2)C1 C1(C(=O)OCC(=O)N(CC#N)Cc2cccc(Br)c2)COC2(CCC2)C1 CCCC(C(=O)NC(C)(CNC(C1(F)CCCCC1)=O)CO)c1ccc(Cl)cc1 c1(-c2n(C(COC)C)nc(-c3ccc(N)cn3)n2)cnn2c(N(C)C)ccnc12 c1(C(C)C)cc(C(=O)NCC(C)(C(C)C)NC(=O)CCc2cocn2)cc(O)n1 CC1(C)CC(C)(C(=O)NC2CC=CCC2)CN1C(c1ccc2[nH]ccc2c1)=O Cc1cccc(C(=O)NC(C)(C)CCNC(=O)C(C)CSc2ccccc2)c1F C(C(C(=O)Nc1cnn(C)c1)NC(C1CC(N(C)CC)C1)=O)SCC C(=O)(C(C)CC(C)(C)C)NC1(C2N(C(CCc3cc(C)no3)=O)CCCC2)CC1 O(NC(=O)CCC(C(C)C)NC(=O)C(CC(C)C)C(C)C)CCOC(C)C c1(CC)nc(C(C)NC(c2nnnn2Cc2ccco2)C2(CC)COC2)cs1 Cc1c(C(=O)NC2CC2NC(=O)C(F)(F)C2(O)CCCC2)cncc1Cl c1(SC)cc(C)c(C(=O)NC(C2CN(C(=O)Cc3cnccc3C)CCO2)C)o1 c1(C(N2C(CC(=O)Nc3c(OCC)cccc3)CC2)=O)ncc(F)cc1N Cc1nnc2n1CCC2(C)C(=O)N(C)C.n1(CC(=O)N2CC2)ncnn1 c1(C(=O)NCC2(NC(CCCC3C(C)C3)=O)CC2)cccnc1F O=C(NNc1ccc(Br)cc1O)c1ccc(CC(=O)N2CCC2)cc1 N1(C(CS(C)(=O)=O)=O)CCCC2(C1)CN(C(C1CC3CC1C3)=O)CCO2 N12CSCC1C2=O.CC(O)(CC(c1ccco1)=O)C1CCNC1 c1(C(N2C(OC)C=CCC2)=O)cc(O)nc2c1CN(C(=O)C(C)CC1CC1)CC2 N1(CC)CC(C(=O)NCCCNC(C2CCCN(C(=O)OC(C)C)C2)=O)NC1=O CC(CC(=O)NC(C)CN(C)C(c1ccnc(Cl)c1)=O)C(F)F CC(C)CCCC(=O)NC(CCN(C(=O)CC1CC1(C)C)C)C(C)C N1(C(=O)COC(F)F)CCN(C(c2ccc(CO)nc2)=O)C(C2CC2)C1 N1(C(C2CCCC(=O)O2)=O)CC(NC(=O)C=Cc2cncnc2O)CC2(CC2)C1 c1(C(=O)NCC(CC(C)C)NC(C2CNC(=O)N2C)=O)c(O)cccc1Cl C(C(=O)N=c1cc(C)o[nH]1)N1CCCC(CN(C(CC(C=C)CC)=O)C2CC2)C1 c1(C(N(C)CC2N(C(C(N3CCCC(O)C3)C)=O)CCC2)=O)nc(Cl)c(Cl)s1 c1(OC)cc(C(=O)NC2CCN(C(=O)C(C)(C)CF)CC2CO)c(Cl)cc1Cl c1(CNC(=O)NC2N(C(CN(CCCN(C)C)C)=O)CCC2)sc(Br)cc1Br c1(CC(=O)Nc2cc(=O)oc3cc(O)ccc23)cc(S(=O)(=O)N2CCCC2)ccc1Cl N1(C(CC(CC)C(F)F)=O)CC(NC(c2ccc(=O)oc2)=O)CC12CCOCC2 C1(c2n(-c3c(C)cccc3)nnn2)(N(c2ccc(Br)nc2)C2CC2)CCCCCC1 C1(COC(C)C(=O)NCCNS(=O)(=O)C2CC2)(CO)CCN(C(C2CC2)=O)CC1 c1(C(N2CCC(NC(c3c(C)nn(C)c3)=O)C2)=O)ccc(=O)n(C(C)C)c1 c1(C(N2C(C)C(O)CC2)=O)cc(O)nc2c1CN(C(C1CCN(C)C1C)=O)CC2 Cc1ncnc(C)c1CC(=O)NC(C)CCCCNC(C1CC1c1cnc[nH]1)=O N1(CCC)CCCC1C(N1CCC(C(=O)NCc2cccs2)C1)=O C1(NC(C(C)OCCC=C)=O)CC2(C1)CC(C(=O)NC1CCN(C)C1C)C2 C1(C(=O)Nc2cccc(COC)c2)N(C(=O)CCc2cccs2)CCC1(C)C C(=O)(C(CC)C(C)(C)CC)N1CCN(C(c2cn(CCOC)nc2)=O)CC(O)C1 C1(CC(=O)NC)CN(C(c2conc2C)=O)CCN1C(=O)C(=O)NC(C)C CC1(C)CN(C(=O)CNC2CCCC2)C1C1CCCO1 CCCCCC(O)CC(=O)NC1CCN(C(=O)C#CC(=O)N(C)C)C12CC2 C1(CC)CN(C(C2CC(=O)N(C)C2)=O)CC1NC(c1cccc(OC2CC2)c1)=O CC1(NC(c2cccc(OCC3CCCO3)c2)=O)CCCN(C(=O)CCC#N)C1 N1(C(C(C2CCOCC2)OC)=O)CCOCC(NC(c2cccc(CO)c2C)=O)C1 Cc1nnc2cc(NCC3CCC(NC(c4cccc5nncn45)=O)C3)ncn12 CCCCCC(C)CC(=O)NCC#CC(=O)Nc1cccc(CO)c1 CC1CCC(CNC(=O)CCCCC2CC2)CN1C(=O)CCc1cocn1 C1(C(N(C)Cc2c[nH]ccc2=O)=O)CN(C(=O)CC2CC(=O)NC2=O)CCO1 N1(C(c2cnn(C)c2Cl)=O)CCC2(CCN(C(C3CC(=O)CCO3)=O)C2)C1 CC(F)(F)CCC(=O)N1CCC(N2CCN(C(=O)Cc3ccsn3)CC2)CC1 c1(C(N2CCC(NC(C(C)C3CC3)=O)C2)=O)ccc2c(c1)OCCO2 C1(O)(CN(C)C(C2CC(=O)CN2C(C2(C)CCCO2)=O)=O)CCCCC1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(CNC(c2cncc(OC(C)C)c2)=O)C1 O=C1CCN(CC(=O)OCC2CC3(CCC3)C2)C(=O)C(CC(F)(F)F)N1 C1(C(=O)NCC2CN(C(Cc3c(C)ncs3)=O)C(C)C2)CCc2n[nH]cc2C1 C(CN=c1cccn[nH]1)NC(N1CCC(n2ccnn2)C1)=O N1(C(CCS(C)=O)=O)C2CCCC1CN(C(=O)CCC1CCC(=O)NC1)C2 c1(N2C(C)CN(C(c3cccc(=O)n3O)=O)CC(C)C2)ncnc2c1SCCC2 Cc1ocnc1C(N1CCC1CNC(c1cn(-c2ccn(C)n2)cn1)=O)=O N1(C(CCCC)=O)C2CCC1C(F)C(NC(C1CCSC1)=O)C2 C1(C(N(CC(O)CNC(=O)CCc2ccon2)C)=O)CC(C)(C)SC(C)(C)C1 c1(N(C)CC2CCN(C(=O)COc3ccsn3)C2)ncc(S(C)(=O)=O)cc1Cl C=CC(CCC)CC(=O)N1CC2(CC2)CC1CNC(c1cc(F)ccc1CC)=O n1(CC(C)NC(C2(C(F)F)CCCO2)=O)cc(CCC2CCCCO2)nn1 c1(CNC(C(=O)NC2C(C)CCC2)=O)ccc(NC2CC=CCC2)cc1 c1(C(C)NC(=O)NC(CCN(C)C)C(F)(F)F)ccc2c(c1)CCC2 N1(C(C2(C#C)CCC2)=O)CC(NC(=O)CCc2cc(C)cc(C)c2)C2(CC2)C1 c1(C(CC(=O)OCCCCC(=O)N(C2CCC2)C)N)ccc(C(F)(F)F)cc1 C1(C(=O)NC(C2CCN(C(c3ccoc3)=O)C2)C)C2CCC3(COC(=O)C13)O2 N1(C(C2CC(OCC)C2)=O)CCCC1c1cn(C2CC(O)C2)nn1 N1(C(CNS(CC)(=O)=O)=O)CC2CC1CN(C(C1CCC(C(N)=O)CC1)=O)C2 N1(C(C2CCC(C(=O)OC)CC2)=O)CCCC(F)(F)C1O C(=O)(C(CCC)OC)N1CCC(C(C(=O)NC(C=C)(C)CC)(C)C)C1 Cn1nc(Br)cc1C(=O)NCC1CCCC1NC(=O)CCC1CCC1 N1(C(CCOCCNC(C(COCC)N=[N+]=[N-])=O)=O)CC=CC12CCOCC2 c1(C(=O)NC(CCNC(CC(CC)OC)=O)C(C)C)cc(F)c2[nH]nnc2c1 C(CCC(=O)NC1(CNC(c2ccc(CN(C)C)s2)=O)CCOC1)=C(C)C C(=O)(C#CC1CCCOC1)NCC(C)(CNC(=O)CC(Cl)Cl)OC C1(CC(=O)NCc2c(C(=O)NCc3onc(C)n3)cco2)CCCC(=O)N1 N1(C(C2(F)C(C)C2)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C(F)(F)CC1 C12(C(=O)NC(C34CCC(CO3)C4)C)COC(C1)C(NC(=O)C#CC1CCC1)C2 C1(OC)CN(C(c2cc(Br)c3[nH]c(C)nc3c2)=O)CC12CCOCC2 c1(C(N2CCC(F)(CNC(C3(C)C(C)C3)=O)C2)=O)ccc2c(c1)CC(C)(C)C2 c1(C(N2C(CNC(C(C)NC(C)(C)C)=O)CC2)=O)c2n(c(=O)n1C)CCCC2 Cc1ccc(C)c(C(=O)NC(C)C(C)NC(c2nn(C)c(C)c2Cl)=O)c1N N1(C(c2cn(C)nc2O)=O)CC(NC(C2C=CCS2)=O)CC2(CCC2)C1 c1(CC)cc(C(=O)NCCCN(CCO)C(c2cnsc2)=O)ccc1C C1(NC(c2sccc2-n2cccc2)=O)COC2CN(C(c3ccnnc3)=O)CC12 C(=O)(CCC(C)N(C)C)NC(C1N(C(C(=O)NCC)=O)CCC1)C c1(CC)noc(CC)c1CC(=O)NCC1CCCC(NC(=O)C(C)(CO)OC)C1 C1(O)(CNC(C2C(C)(COC)C2)=O)CCN(C(c2cnc(C3CC3)s2)=O)CC1 c1(C(N2C(C)(CNC(c3cc(CF)on3)=O)CCC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nn(-c2ccccc2)cc1NC(C1(N2CCOCC2)CCCC1)=O C1(C(=O)NC2C=CC(C(N3CC(CSC)C3)=O)C2)CC12CCOCC2 C(=O)(CCCCC(C)(C)C)N1CC2C(C(=O)NC(C)C(=O)NO)(CCC2)C1 N1(C(c2c(CSC)cccn2)=O)CC2CCN(C(C3CC(SC)C3)=O)CC2C1 c1(OC)ccc(-c2cn(CCNC(=O)Cc3cccc(Cl)c3Cl)nn2)cc1F C(=O)(C(C)(C)c1cncnc1)N(CCC(=O)O)CCCC(c1ccccn1)O CC1COC(C)(C)CN1C(c1cc(O)nc2c1CCC2)=O N1(C(C(CC)(CNC(c2ccc(N)cn2)=O)CC)=O)Cc2ccc(C)nc2C1 N1(C(C(C)OCCCCCC)=O)CCCCC1CNC(=O)C(C)CC C(c1cncc(C(F)(F)F)c1)=CC(N1C(C)CCC1C(=O)Nc1ccccn1)=O C1(NCCc2cccc(C(F)(F)F)c2)CCC2CNCC2C1 c1(C(N(C)CC2CCN(C(=O)Cn3cccn3)CC2)=O)cc([N+](=O)[O-])cnc1O CCC(F)C(=O)N1CCC(N(C(=O)CCC=CCC=C)CC)C1 C1(C(=O)NCC(CC)NC(=O)COCC2(F)CC2)CCC(C(C)(C)C)CC1 c1(NC(C(=O)N(C2CCOCC2)C(C)C(C)n2cccn2)=O)ccc2nccn2c1 Cc1oc(C(=O)NC2CCC2CNC(=O)C(N2CCCC(O)C2)C)cc1CO C(=O)(C(C(=O)N1CCCC(NC(c2cc(C(C)(F)F)on2)=O)C1)C(C)C)OCC N1(C(C2(C)COC2)=O)CCC2(CCCN(C(c3cc4ccnc(Cl)c4s3)=O)C2)C1 c1(C(N2CC3(CC(NC(=O)CC4CS(=O)(=O)C4)C3)C2)=O)noc2cc(Cl)ccc12 c1(OC)c(C(=O)N(CCCCN(C)C(C2CCCC(C)O2)=O)C)nc(O)nc1O N1(C(c2c(COC)ccs2)=O)CC2CCN(C(=O)Cc3cscn3)CC12 c1(CCNC(=O)NC2CCCC2n2cccn2)cccc(F)c1 c1(SCNC(C)CCN=[N+]=[N-])ccc(S(N)(=O)=O)c(C)c1 CC1(C)CCCC(C(=O)NC2CCCCC2CNC(=O)C=CCN2CCC2)C1 c1(OC)ccc(F)c(C(N2CCCC2CNC(c2cncn2C2CC2)=O)=O)c1 C(CC(=O)NOC1CCC1)C1CN(C(CN(C(=O)OCC)C)=O)C1 Cc1cc(F)c(C(=O)NC(C2CCOC2)CNC(=O)CC(C)(C)C)cc1F C1(OC)CC(CNC(=O)Cc2ccc(C(=O)O)cc2)C1(C)C C#CC1(C(=O)NC2C3CC2N(C(=O)CC2OCCCO2)C3)CC(F)(F)C1 C1(O)(CN(C(=O)COC(F)(F)F)C)CCCN(C(=O)C(=O)N(C)C)C1 c1(C(C(=O)NCC2CCN(C(C(CC)F)=O)C23CC3)=O)c[nH]c2ccccc12 CC(C)CC(O)C(=O)N1CCN(CCCNC(c2cc(Cl)no2)=O)CC1 n1(CC)c(C(N2CCNCC2C(=O)O)=O)cc2ccccc12 c1(C(=O)NC2CCN(C(c3c(C)cns3)=O)CC2F)cc(S(C)(=O)=O)c(C)o1 C(=O)(C(O)CCCNC(C1(C#N)CC1)=O)NC(C)(C)C(N)=O c1(OC)ccc(C(=O)NCCN(C(=O)C(CCSC)NC(C)=O)C(C)C)cc1C N#Cc1ccncc1C(=O)NCC1OCCC1C(=O)N(CCCO)CCCO c1(OC)cncc(C=CC(=O)N(CCNC(c2ccc(F)c(Cl)c2)=O)C(C)C)c1 N1(C(C(C)n2ccnc2)=O)CCOC(C(=O)Nc2ccc(F)cc2)CC1 C(=O)(CCN=C(NCc1cccc(SC)c1)NC1CCOC(C)(C)C1)NC N1(C(C(=O)NCCOC)=O)CCN(C(=O)CCc2cnco2)CC1C1CC1 C(=O)(C1=CCC(NC(c2cc[nH]c2)=O)C1)NCCC1C(C)CCO1 CC(C(=O)NNc1ccc(Br)c(F)c1F)OCC1CCCO1 c1(CN(C)CCc2nccs2)nc(-c2ccc(Cl)cc2)sc1-c1ccc(=N)[nH]c1 CCCCCC(=O)N1CC(NC(c2csc(-c3cccc(C)n3)n2)=O)C(C)C1 c1(C(=O)NCCC(C(N2CCCC(C)(O)CC2)=O)OC)ncc2ccccn12 c1(SC)ccc(CCCC(=O)NC2C3CC2N(C(C2CCC(=O)O2)=O)C3)cc1 C1(C(=O)NC(C)(C)CNC(=O)C=C2CCCCC2)(CC)CCC(F)(F)CC1 CC1(O)CCCC(C(N2CCC(CCNC(=O)CC3CN4CCN3CC4)C2)=O)C1 c1(CNC(C2(CCNC(COC)=O)CC2)=O)cccc(CO)c1.c1nc[nH]n1 C(CC(C(C)(C)C)NC(c1cccc(C(F)F)n1)=O)N(C)C(c1cnn(C)n1)=O CC(C)CC(C(=O)N1CC2CC2C2CC12)ONC(=O)CC1C=NN(C)C1=O c1(C(=O)NC(CC(C)NC(C=CC(C)(C)SC)=O)C)c(C)cncc1C c1(C(N2CCC(N(C(=O)C3=CC(C)(C)C3)CC)C2)=O)ccc(CO)c(F)c1 C1(C)(C(=O)NC(C2CCCN2C(=O)Cc2cn[nH]c2)C)CC1(C)C c1(NC(CNC(c2c(C)nc(CC3CC3)o2)=O)C)cc(C#N)c(F)cc1[N+](=O)[O-] Cc1c(NC(c2nc(-c3ccccc3)oc2C(C)C)=O)cnn1CCO C1(C(N2CCC(O)(C(C)NC(CSC)=O)C2)=O)CCC(O)CN1C C(=O)(CC(C)(C)C#N)NC1CCCC(N(C)C(c2ccc(Br)s2)=O)C1 c12ncc(cn1)-c1csc(n1)NC(=O)N2.CC(=O)NCCN(C)C N1(C(C2C(NC(c3scc(OC)c3)=O)CCO2)=O)CCOC(CC(N)=O)C1 c1(OC)cc(OC)cc(CN2CCC(C)(C(=O)Nc3cc(F)cc(Br)c3)C2)c1 N1(C(C(CCSC)NC(C)=O)=O)CCC2CCN(C(=O)C3=CCCC3C)CC12 CC(C)C(=O)CCCN1CCN(C2CCCCC2)CC1 c1(C(=O)NCC2(C)CCN(C(c3c(C)cccn3)=O)CC2)cc2n(n1)CCCO2 C(=O)(C#CC1CCC1)N1CCC(C(C)NC(c2ccn(CC)n2)=O)C1 C(=O)(N=c1[nH]nc(C(C)(C)CN(C)C)s1)N1C(C)CC(O)C1 c1(CN(c2ccccc2)C(=O)NC2CCCC(COC)C2)ccnc(C)c1Cl c1(C(=O)OC)cc2c(c(S(=O)(=O)Nc3cccc(N4CCCC4=O)c3)c1)CCC2 CCC(C)C(C(=O)N(C(C)(C(=O)NC1CC1CC(C)C)C1CC1)C)N(C)C c1(N2C(C(N3CC4CCC(C3)O4)=O)CCC2)ncc(Br)cc1Br Cc1cc(Cl)c(C(=O)NC(C2CCCCN2C(c2cc(F)cs2)=O)C)cc1N C1(C(N(C2(C(=O)OC)CC2)C)=O)CC12CCN(C(=O)C(C)CC(N)=O)CC2 C(=O)(CC1CCCc2ccccc21)NC(C(CCCCC)(O)CC)C c1(C(=O)NC2C(NC(=O)C3=CCCOC3)CCCC2)ccc2c(c1)COCCN2 N1(C(CC2C(OCC)COCC2)=O)CC2CC(N(c3ccc(F)cc3)C)C1C2 C1(C)(C(C)C)CC1C(=O)N(CCNC(=O)Cc1cc[nH]c1)CCOCCO C1(CCC)CN(C(c2cc(C(=O)OC)cs2)=O)CCN1C(c1cccnc1Cl)=O N1(C(C(COCC)C)=O)CCCC(O)(CNC(C2(C)CCC(F)(F)CC2)=O)CC1 c1(C(CNC(=O)NC2CC3(C2)CC3F)(F)F)ccccc1F C(=O)(CCC(C)(C)NC(c1cn(C)c(=O)n1C)=O)NCc1c(C)nn(C)c1 CCC(CC(=O)NC1CN(C(C2CNC(=O)N2)=O)C1)C1CC1 C(=O)(C#CC1CCCOC1)NC1CCCCN(C(C(c2cccs2)SC)=O)C1 Nc1cc([N+](=O)[O-])ccc1C(=O)NC1CC(CNC(c2nsnc2O)=O)C1 N1(C(=O)CC2CC3CCC2C3)CC2CN(C(C3(Br)CC3)=O)CC(C1)O2 C#Cc1ccc(C(N2CCC(C=CC(N3CCC(C(N)=O)C3)=O)CC2)=O)cn1 C(=O)(C1CCCc2ncccc21)NC12C(CN(C(c3c(C)nn(C)c3Cl)=O)C1)C2 c1(C(N2CC(NC(C=CC(CC)=CC)=O)C3C2C3)=O)ccc2nncn2c1 Cc1c(NC(c2cc3c(F)c(Br)ccc3s2)=O)ccc(Cl)c1[N+](=O)[O-] CCCCC(CCCC)C(=O)N1CC(NC(=O)CCSc2nccn2C)C(C)C1 C1(N(C(c2c(CC)c[nH]n2)=O)C)CCC(NC(=O)CC2CCC3CC23)CC1 S(=O)(=O)(c1ccc2c(c1)CN(CC1CC(C)(C)C13CCC3)C2)N(C)C Cc1nc(N(CCCS(N)(=O)=O)CCO)cc(C(F)F)n1 C12(CNC(c3c(N(C)C)cccc3)=O)CCCOC1CCN(C(=O)C(F)Br)C2 C(=O)(N=c1ncnc2[nH][nH]c(C)c1-2)C1C(NC(c2cc(C)cc(C)n2)=O)C1 N1(C(CCSCCC)=O)CC2CCC2(CCNC(c2nccnc2C(N)=O)=O)C1 C1(C(=O)NC2(COC)CN(C(C)=O)C2)CCN(C(=O)C(C)N(C)C)CC1C c1(C(N(CC(=O)NCc2c(C)nc(C)s2)C)=O)ccc(C)c(O)c1 n1(CCC(=O)N(CCC(=O)O)CC(C)C)ccc(O)nc1=O c1(C(N2CCCC2CF)C(=O)NCCN2CCC(O)C2)cc(Cl)cc(Cl)c1Cl C1(C)(NC(C2CN(C(C)C)C2)=O)CCN(C(=O)C(C(C)C)c2ccccc2)CC1 c1(C(=O)NCC(CCCC)NC(=O)C(C)=C2CCC2)ccc(OCCF)cc1F c1(C(=O)NCCCNC(=O)C(F)Cc2ccccc2)cnc2[nH]nnc2c1 C1(C(=O)NC2C(CCOC)CCC2)CC(O)CN1C(=O)C=C1CCOCC1 C=CCCCCCC(=O)NC1CCN(C(=O)COC2(C)CCC2)CC1F c1(C(N2C(C)CC(c3ccccc3)C2)=O)cc2cccc(Br)c2cn1 c1(C(=O)NC2CCCC(C(=O)Nc3cnoc3)C2)cc(F)cc([N+](=O)[O-])c1 c1(C(CC2CC3CN2C3=O)=O)cc(C)nc2ncnn12.c1(C(=O)OC)cscc1F N1(C(COC(C)=O)=O)CCC2(NC(=O)Cc3ccc(F)cc3Cl)CCCCCC12 CCC(CC(=O)N1CC2C(CNC(c3cncc4c[nH]nc34)=O)C2C1)C(C)C N1(C(C=C(C)C2CC2)=O)CCC(C)(C)C1CC(N1CCCC1)=O N1(C(C)=O)CCC2(CCC(C(F)(F)F)N2C(=O)C(C)NC(=S)SCC(F)(F)F)CC1 n1(CC(=O)OC)cc(NC(=O)CC2CC(C(F)(F)F)C2)c(C)n1 C1(C(N2CC(CCNC(c3cc(C)oc3)=O)OCC2)=O)CN(S(N)(=O)=O)C1 c1(CCNC(C(CN(C)C)NC(=O)Cc2ccn(C)n2)=O)cccnc1O N1(C(C(Cc2ccccc2)OC)=O)C2CCC1CC(NC(=O)CC1(C)CCC1)C2 c1(SCC)cc(F)c(S(=O)(=O)Nc2cccc(C(=O)OC)c2)c(F)c1 Cc1cc2c(cc1NCCSCCSCCO)CCO2 N1(C(c2c(C)ccnn2)=O)CCCC(CO)(NC(c2cccs2)=O)C1 Cc1noc2ncc(C(=O)NC3CC(O)(CNC(=O)C=C4CCC4)C3)cc12 C1(NC(=O)CSc2nc[nH]n2)CC(CO)N(C(=O)CCc2ncc[nH]2)C1 C1(C(=O)NC(c2n(CC)ncc2)C)CN(C(=O)CCP(C)(C)=O)CCC1O Cc1nnc(CNC(c2ccncc2)C2CCOC2)n1C O=S(=O)(c1ccc(N2Cc3cnn(CCO)c3C2)cc1Br)NCc1cc(Br)no1 c1(NC(C)CCC(F)(F)F)ccc(S(=O)(=O)NCC2(C)CCCOC2)cc1C#N N#CC1(C(=O)NCC(O)CNC(C2CC23CCCCC3)=O)CCSCC1 c1(OC)ccc(C(=O)NCC2C3CN(C(C4(F)CC4)=O)CC23)c(OC(F)F)c1Cl C(=O)(C(C#N)C(C)C)N1CCC(CC#C)(C(=O)NCc2cnn(C)c2O)C1 C1(NC(C(C)(C)SC)=O)CCC2(CC1)CCN(C(=O)CCc1cc(F)ccn1)C2 N1(C(=O)CCc2ccc(Cl)s2)CC(C2CN(C(C3CC3F)=O)C2)C1 CCC(COC)C(=O)N1CCC(CC(=O)NC(C)CC(C)CC)CC1 Cc1cc(C(=O)NCC=CCNC(C2CC2c2cccc(Cl)c2)=O)ncn1 CC(C)C(CC(=O)N1CC2C(N(C)C)C2C1)NC(C1CCOC1(C)C)=O C1(CNC(CC2CC(NC)C2(C)C)=O)CC(C)CN(C(c2scc(C)c2C)=O)C1 C1(C(=O)NC2CCCC2C(N)=O)(CNC(CN(C(C)C)C)=O)CCCO1 Cc1cc(O)nnc1C(=O)NCCC1CN(C(C2CCC(C)CC2)=O)CC1C c1(CNC(C(Cn2ccnn2)NC(C(CC)O)=O)=O)cccc(O)n1 N1(CC(=O)N(C(C)C)CC2CCCO2)CCC12CCOC(C)(C)C2 C1(C2CC2)(CNC(CN(CCOC)C)=O)CCN(C(C2(C3CCCO3)CC2)=O)C1 c1(OC)ccc(C(=O)NC(C)CCCNC(C2(C)CCOC(C)C2)=O)cc1C N(C1CC2(CCN(c3ccc(C#N)cn3)C2)Oc2ccccc21)C(C=CSC)=O C(=O)(C(C)CC(N)=O)NC1CC(F)(CNC(c2c(C(C)C)scn2)=O)C1 C1(NC(C(C(C)(C)C)NC(=O)OC)=O)CN(C(c2n[nH]cc2F)=O)CCC1(C)C C1(NC(CONC(c2n(C)ccn2)=O)=O)(CC2(F)CCC2)CCOCC1 c1(C(N(C(CN(C(C2(O)CCC(C)CC2)=O)C)C)C)=O)ncc2ccccn12 C1(C(N(CCC#N)Cc2cccnc2)=O)C2C=CC(C2)C1C(=O)O N1(Cc2cccc(C)c2)CCCC(NC(=O)CNC(=O)CC(C)(C)C)CC1 C1(NC(c2nnn(CC)c2C)=O)CC(NC(c2occc2F)=O)C12CCC2 N1(C(CC=CCNC(C2C(C)CCC2)=O)=O)CCCC2(C=CCO2)C1 c1(CC(N2CCCC2)C)nnc(CCN(C)C)n1CC(c1cccs1)N(C)C C1(C(=O)NCC2N(C(CSc3n(C)ccn3)=O)C3C(C2)C3)CN2CCN1CC2 N1(CC(C)NC(c2cncc3c[nH]nc23)=O)CCc2ccccc2C1=O c1(-n2c(C(=O)NC3CC(CNC(CCOCC#C)=O)C3)cnc2)ccccc1Cl C(=O)(C1CCCc2nncn21)N1CCC(O)(CN(C)C(c2ccc(F)cn2)=O)C1 N1(C(C(CC=CC)CC)=O)CCC2CN(C(=O)C=Cc3sccc3C)CC12 c1(C(N2C(CNC(c3n(CC)ncc3)=O)CCC2)=O)c(Br)cc(F)c(F)c1F CC(CC(=O)N1CCCC1CC(=O)N(C)CC1(C)CC1)C(C)(C)C c1(C(N2CCC(CF)CC2)=O)ccc(CNN(C2CC2(F)F)C2CC2)cc1 C(=O)(CCCCC#N)NCC1(F)CCC(CNC(C(C)Sc2ccccc2)=O)C1 C(=O)(CC(F)(F)C(C)(F)F)N1CC(N(C(=O)C=Cc2cccn2C)C)C2(C1)CC2 C1(CNC(C2(COC)CCCN2C(=O)C(=O)NC2CC2)=O)Cc2ccccc2O1 Cc1cc(C)c(C(N2CC(C(F)(F)F)C(CNC(C3CCCC3)=O)C2)=O)c(=O)o1 Cc1cc(C)c(NC(=O)C(C2CC23CCCCC3)N2CCC(C(N)=O)C2)c(C)c1 N1(C(=O)NCC(=O)Nc2c(C)ccnc2C2CCNCC2)CCC2(CC(C#N)C2)C1 C1(CNC(C(C)=C(C)C)=O)C2CCCC1N(C(c1cnn3c1OCC3)=O)C2 C1(NC(CCC=C(C)C)=O)CC12CCN(C(c1nn(C)cc1N)=O)CC2 CC1Oc2c(F)cccc2C1NC(c1ccc(C#N)cc1Br)=O C1(C(=O)N(C)CCC2CCC2)(SC)CN(C(C2CCCC2O)=O)C1 C1(NC(c2cccc(CC3CC3)c2)=O)CCN(C(=O)CN2CCOC2=O)CC1O C1(C(N2CC(CNC(CN3CC(C)(OC)C3)=O)C2)=O)CC2(CCCC2)C1 CCC1=C(C(=O)NCCOCCCN(C)C(C23CC4CC2C3C4)=O)SCCO1 N1(C(C(CC)OC)=O)CC2C(CN(C(=O)CCC3CCCCC3)C)C2C1 C1(C(N2CC(O)(CNC(c3ccc(N)cn3)=O)C2)=O)Cc2nnsc2S1 c1cc2[nH]c(=NC3CC4CC4C3)nc(N3CC4CCC3CC4)c2s1 c1(CN2CCC(C(C(=O)Nc3nc(C)sc3)C)CC2)cc(F)ccc1[N+](=O)[O-] N1(C(COC(CC)C)=O)CCCC12CCN(C(c1cncc(OC)c1)=O)C2 C1(CC)CN(C(c2c(C)cnn2C)=O)CCN1Cc1ncnn1CC C1(C(=O)NC2CN(C(c3ncn(C)n3)=O)CC2O)CCCCNC1=O C#CCC(C)(C)C(=O)N1CCC1CNC(c1nc(C)ncc1Cl)=O C(=O)(CCCC(C)(C)NC(=O)C1=CCCCC1C)N1C(C(=O)NC)CC(O)C1 C1(NC(=O)Cn2cccn2)CCN(C(=O)CC2CC=CC2)CCC1(F)F C(=O)(C(C)CC(C)(C)C)N1CCCC(O)(CCNC(c2ncc(C)c(Cl)c2)=O)C1 c1(C(=O)NCC2(C)CCOC2)cccnc1CNC(C1CCC(F)C1)=O c1(SC)nc(C)cc(=NCC2(CCNC3CC4CCC3O4)CC2)[nH]1 N1(C(COCCCOC)=O)CCCC(OCC(=O)N(C2CCSCC2)C)C1 C1(CNC(Cc2cc(C)ncc2)=O)C(C2CC2)CCN1C(=O)CC1CCC(C)C1 C1(CN(C)C(c2coc(CO)c2)=O)CCCN(C(C2(C)CNC(=O)N2)=O)C1 c1(CC(=O)N(C2CC3CNC2C3)Cc2ccccc2)ccccc1OCCCF Cc1[nH]nc(C(=O)NCCC2CCN(C(=O)Cc3cc(C4CC4)no3)C2)c1F C(=O)(C(C)(C)C(N)=O)N1C(C2(NC(C3CCN(CCC)C3)=O)CC2)CCC1 C(N=c1[nH]c2c(c(=NC3CCc4cccc(CO)c43)[nH]1)COC2)c1c(C)occ1 C(CCCCC(=O)NC1CCCCC1CNC(c1cc(C#N)oc1C)=O)SC C1(CC(=O)N(CCC(=O)NCC(N)=O)CC=C)CC2CC2C1 c1(C(N2C(CNC(CC3(C)CCOCC3)=O)CCC2)=O)cnn2cccc(Cl)c12 C(CNC(c1n[nH]c(O)n1)=O)(C(=O)NCC(CC1CC1)CO)OC c1(CN=C(NC(COC)C)NCCn2ccnc2)ccc(F)c(O)c1 N1(C(C(CCC)OCC)=O)CC2(CCN2C(=O)CCC2CCC2)C1 N1(CC2C3CC(C)(C3)O2)CCCC2(C1)OCC(O)C2O N1(CC(=O)NCCCC)CC(NC(c2cnsn2)=O)CCC1C CC1CC(C(=O)NCc2cn(CCN3CCSCC3)nn2)CCS1 CC1(C)CNC(=O)c2c(C(=O)NCCNC(C3Cc4cscc4C3)=O)coc2C1 N#Cc1cc(C(=O)NCC2CCN2C(c2nccc(Cl)c2F)=O)n2c1CCCC2 C=CC1OCCCC1N(C(=O)C(=O)NCC1CCN(C(=O)OC(C)(C)C)C1)C CCCCC(CC)CC(=O)N1CCC(C)(C)C(C(=O)NC2CC(O)(CO)C2)C1 CCCCCC=CCC(=O)NCCN(C(=O)C(C)OCC1CCCCO1)C(C)C O=C(CCC(F)(F)Cn1cc(-c2cccnc2)nn1)NC1(C(F)F)CCOCC1 c1(NC(C2(C)CCN2Cc2c(OC(F)F)cccc2Br)=O)cc(Br)c([N+](=O)[O-])cn1 c1(C(N2CCC(C(N)=O)C(C)(C)C2)C(=O)NC)ccc2c(c1)CC(C)O2 Cc1cc(C#N)cc(C)c1C(N1CCCC1CCNC(=O)C(O)c1ccco1)=O c1(C(=O)NCC(CC)NC(=O)C(C)S(C)(=O)=O)coc2c(F)c(Cl)ccc12 c1(C(=O)NC(CCCNC(Cc2ccc(C)cc2F)=O)C)cccc2c1NCC2 CCC(CCCC(=O)NC1CC2CC1C(O)C2O)NC(c1cc(C)nnc1O)=O C(CCCCC(=O)N1CCC(F)CC1C(=O)NCC1CCCCN1C)SC C#Cc1ccc(Cl)c(C(N2CCCC(CN(C(=O)C(C#N)CC)C)C2)=O)c1 n1(CCC(=O)Nc2cnn(C(C)C)c2C2CC2)c(=O)oc2ccccc12 N1(C(c2c(OCC)scc2)=O)CCC(C)(CNC(=O)C(C)NC(C)(C)CC)CC1 N1(COC)CCC(COCC)(NC(C2(NC(=O)CC3CC3(C)C)CC2)=O)C1 N1(C(=O)NC(c2ccc(F)cc2)CCC)CCCC1C1OCCO1 CCCCC(O)C(=O)NC1C2CN(C(=O)Cc3ccc(Br)cc3C)CC12 C1(CNC(C=C(C)C(F)F)=O)CCC(CN(C(=O)C=C2CCCCC2)C)CC1 c1(OC)nc(Cl)ccc1CCC(N1CCCC1(C)Cc1cc(Cl)cc(Cl)c1)=O N1(C(c2ccc(CCCC)cc2)C(=O)NCCCC2CC2)CCOC2CCCC12 Cn1nc(C(=O)NC2CC(C)(C(=O)NCCC(N)=O)C2)cc1CO n1(CC(=O)NCC(C)NC(C2CN(C)CC2C(F)(F)F)=O)nnc2ccccc12 N1(C(c2cc(C)cc(Br)c2)C(=O)NC(C)C(=O)OC)CCC(C2CCOC2)CC1 Cc1cc(NC(c2coc(CNC(c3ccnn3C(C)C)=O)n2)=O)cc(CO)c1 C(=O)(CC(O)C(C)(C)C)NCCC(=O)NC(C)C(c1ccccc1)C C1(CC)C(C(=O)NCCOC2CCN(C(=O)Cc3cn(CC)nn3)C2)CCN1C CC1C(NC(=O)C(F)(F)CO)CC2CCC1N2C(c1cccc(Br)c1)=O CC1C(NC(=O)C(C)(C)C2CCCCO2)CCN1C(=O)CC1CCOC1 CCC(CC)CC(=O)N1CCC(CC(N2CCC(C)C(CC3CC3)C2)=O)C1 N1(C(=O)Cc2ccno2)CCC2CCCN(C(=O)CCC3CCCCCC3)C2C1 C1(C)(NC(COCC=C)=O)CC(NC(c2csc(C(C)(C)C)n2)=O)C1 N1(C(Cc2ccc(C)c(Cl)c2)=O)CCC2CN(C(=O)Cn3cnnc3O)CC2C1 C1(CCO)(NC(CCN(C)CC)=O)CN(C(=O)C(CO)c2ccccc2)C1 C(=O)(C(O)C(C)(C)C)NC1(CC(=O)NCc2ccc(OC)cn2)CCC1 C1(C#N)(C(=O)Nc2cccc(CNC(C(CCC)OC)=O)c2)CC12CCCC2 C1(CC(=O)Nc2cccc(C3CCOCC3)c2)CCCS(=O)(=O)C1 Cc1ccnc(C)c1NC(C1CCC(NC(c2nccnc2Br)=O)CO1)=O CC(C)(C)CCCC(=O)N1CCCC(C(C)(C)C(=O)NCc2ccncc2)C1 C1(C(N2CC3C(n4cc(C=CCC=C)nn4)C3C2)=O)CCCCCS1(=O)=O Cc1ccc(C)c(N(C)C(C(=O)CO)=O)c1.c1(N)ccc(F)c(Cl)c1 N(C(=NCCSC(F)(F)F)NCCn1ncccc1=O)CC1(C)CCCS1 C12CC3(CCN(C3)C1=O)C2.N1(C2CN(C(CC3CC(=C)C3)=O)C2)CCOCC1 CCC(C)C(C)C(=O)NCC1(NC(c2occ(C)c2C)=O)CCCCC1C C(=O)(C1NCCc2cc(Br)ccc21)Nc1c(C)n(-c2ccc(Cl)cc2)nc1 C1(CNC(=O)CCn2cccc2)CC2CCC1N2C(=O)CCOCC(F)(F)F N1(C(C2(C)CC2)=O)CCCC(C2CC2NC(=O)CCCCCn2cnnn2)C1 C12(C(=O)NC3COC3)CCCC1CS(=O)(=O)C2.N12CCC(CC1)OC2=O.CC(C)(C)O C(=O)(CCCCCCBr)N1C(C(=O)NC2CS(=O)(=O)C2)COCC1 C1(CC)CN(C(c2c(CNC(=O)C=Cc3cnccn3)nnn2C)=O)CCO1 C1(C(=O)NC(C2CCOC2)(C)C)COCCC1NC(c1cccc(CC#N)c1)=O c1(C(N2CCC(O)(C(C)NC(CCSCC(C)C)=O)C2)=O)occ2c1CCOC2 c1(CC(N2CC(C(C)NC(c3c(C#C)c[nH]n3)=O)C2)=O)c[nH]c2cnccc12 N1(C(C2(C#C)CCCC2)=O)CCC2(CCC(CNC(C3CC3(Cl)Cl)=O)O2)CC1 N1(C(C(=O)NCCCSCC)C(C)CC(C)C)CCC2(O)CCOCC2C1 CCC(CC(=O)NC1(COC)CCCN(C(c2csnc2OC)=O)C1)C(F)F C(CCCCC(=O)NC1CC1C(F)(F)F)NC(C1C(C)CC1)=O O=C(N=c1cc[nH]cc1)Nc1ccccc1F.c12cc(Cl)ccc1NC2=O CCCCC(CC)C(=O)NCC1(F)CC(CNC(c2cn(C3CC3)nn2)=O)C1 Cc1c(NCCCc2ccsc2)ncnc1N1CCC(CC2CC2)C1 C1(NC(C(C)CC2CCC2)=O)CCC2(CCCN2C(=O)CC(C)(C)C(F)F)CC1 N1(C(c2c(C)ocn2)=O)CCC(C2CCN(C(c3ccnn3CC(F)F)=O)C2)C1 CCCCCCC(C)C(=O)NC1CC(C)(NC(c2cncc(Cl)c2)=O)C1 N1(C(C2CC=CCC2C)C(=O)NC)CCCC(C2CCOCC2)C1 Cc1nnc(C(=O)NC2CCCC2CNC(c2ccc(CO)o2)=O)s1 C1(NS(CC)(=O)=O)CN(C(=O)OC(C)(C)C)C2(CCC2)C1.C1C(=O)N1 CCCC(C#N)C(=O)NC1CCCCN(C(c2cc(C)nn2C2CCC2)=O)C1 N1(C(=O)CCCc2cc(C)sc2C)CCN(C(c2c(OC)cc(C)s2)=O)C2CC12 N1(C(=O)Oc2c(C)cccc2)C2CC1CN(Cc1ccnc(F)c1)C2 c1(SCC(=O)NCCC2(C(=O)NC3CCC(CO)C3)CC2)ccccc1 C1(NC(CC=C(C)C)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 C1(C(N2CC(CCC)N(C(c3csnc3C)=O)CC2)=O)CCCN2CCCCC12 c1(C(=O)NCCC2CCCN(C(=O)C(F)C3CC3)CC2)ccc2nn[nH]c2c1 N1(C(=O)CCOC2CC2)CCCC2(CCN(C(=O)CC3CC4CC4C3)CC2)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)N1CC(NC(=O)NC(C(=O)OCC)C)OCC1 Cc1nc(O)[nH]c1C(=O)N(CC(C)(C)CNC(C1CC(C(C)C)C1)=O)C c1(C(=O)NC(C(C)C)CNC(C2(C3CC3)CC2)=O)ccc2c(c1)OCC2 Cc1cnc(N2CCOC(C(C)NC(c3cc(C4CCC4)on3)=O)C2)nc1O c1(CC(=O)NCC(C)NC(CC2C(C)=NOC2=O)=O)ccc(F)cc1F C(=O)(CCCC(F)F)NCCC(C)(C)NC(C12CC(C(F)F)(C1)C2)=O c1(CC)ccc(F)c(C(=O)N(C)CC2CCN(C(c3conc3CC)=O)CC2)c1 c1(C(=O)NCC(C)NC(C23CC(CC4CC4)(C2)C3)=O)c[nH]nc1C1CCOCC1 N1(C(C2(COCC)CC2)=O)CCC(C(=O)Nc2ccccc2C(C)O)CC1 CC1CN(C(=O)CC2C=CC(NC(c3ccc4[nH]ccc4n3)=O)C2)CC(C)(C)C1 N1(S(C(C)(C)C)(=O)=O)CC2CC1CC2NS(=O)(=O)CC#N C#CCCC(O)C(=O)N1CC(C2CN(C(c3ccc([N+](=O)[O-])n3C)=O)C2)C1 c1(C(=O)NCC(CCC)NC(C2COCCO2)=O)cc(F)cc(F)c1 N1(C(c2c(CC)cccn2)=O)CCN(C(=O)Cc2ccn(C(C)C)n2)CC(O)C1 C#CC1COCCN1C(=O)CCC(CC)NC(=O)CC(C)N(C)C N1(C(c2c(C)cc(F)cn2)=O)CCC(N(C(=O)C=C2CCOCC2)C)C2(CC2)C1 C1(NC(C(Cn2ccnn2)NC(CCC(C)N(C)C)=O)=O)CCCN(C)C1=O C12(C(N3CCC(C(C#C)C)CC3)=O)CCCC1CCN2C(c1sncc1CC)=O N1(C(c2c(C)nccc2)=O)CCC(C)(C)C1C(N1CC(c2cc(O)n[nH]2)C1)=O C1(C)(C(=O)NCC2(NC(CCC(C)(F)F)=O)CCOC2)Cc2ccccc2C1 c1(NCCNC(=O)OCC)ccccc1S(C)=O C1(C(N2CCC(O)(CNC(=O)CCc3cc(Cl)cs3)C2)=O)CC2C(C1)C2(F)F c1(OC)ccc(NC(C2CC(C)CN(C(=O)C(C)N(C)C)C2)=O)c(C(N)=O)c1 c1(OC)ncccc1C(N1CCOCC1C1CCOC1)C(=O)NCCCF C1(C(N2CC3CC(CNC(c4cccnc4S)=O)C3C2)=O)CCc2ncsc2C1 N1(C(C2CCN(CC)CC2)=O)C2CCC1C(C(=O)NC(C)CCCO)C2 C(C)(CC(C(=O)NCCSC)N1CCC(c2cnccn2)C1)CCC(=O)N(C)C c1cn(C)c2ccccc2c1=O.C(=O)(C(C(=O)OC(C)(C)C)OC)OCC C(CCO)(C(C)(C)O)NC(C1C(CNC(c2c(CC)nn[nH]2)=O)CCCC1)=O c1(CC(=O)NC(C2CCN(C(COC(CC)C)=O)C2)(C)C)ccc(F)cc1F Cc1ncncc1NC(C1CCC(NC(=O)Cc2cnn(C)c2)CO1)=O c1(OC)c(F)ccc(F)c1C(=O)NCC1CC1NC(C1(P(C)(C)=O)CC1)=O CC(C(C)(C)C)=CC(=O)NC1CC(NC(=O)C(C)(Cl)Cl)C1 Cc1cc(C)n(C(C)C(=O)N(C(C)C(=O)N(C2CC(C)(C)C2)C)C)n1 CN=c1[nH]cc(C(=O)NC2CCC2NC(=O)CCc2ccccc2OC)s1 C1(N(C(C2CCCC2C(=O)OC)=O)CC)CCN(C(=O)Cc2nnc(C)s2)CC1 CCC(F)(F)CCN=c1nc2scnc2c(NCCCOC2CCCCO2)[nH]1 OC1CN(Cc2cn(-c3c(F)cc(F)cc3F)nn2)CCC12CCC2 C(=O)(CCS(C)(=O)=O)N1CCC(N(CC#C)C(c2ccc(O)nc2)=O)CC1 c1(OCC)ncc(CNCCC(=O)C(C)Nc2cccnc2NC2CC(=O)N2)cn1.N c1(C(CNC(CC2CC(OC)C2)=O)CNC(=O)CN2CC=CC2)ccccc1 n1(CC)ccc(CC(=O)NCCN(C(=O)C(C)OCC(C)C)C(C)C)n1 C1(CCNC(c2cccc(C)c2C)=O)CN(CCON)CCS1(=O)=O N1(C(Cc2cn(CC)nc2)=O)CCCCC(NC(c2nn[nH]c2Cl)=O)C1 C1(C(=O)NC(C2CCCC2)CNC(C2(CC(C)C)CC2)=O)CC=CC1 c1(C(=O)NC2C(C)CCN(C(=O)CCC3CC3)C2)cc(F)c2c(c1)nnn2C C1(OC)CN(C(=O)OC)CCC1O.C12CCN(C1)C2=O C1(C(=O)NC2CN(C(c3ccc(C(N)=O)o3)=O)CC2CO)CCCCC1C1CC1 N1(S(CC(=O)OCC)(=O)=O)CCC(F)(F)C(NC(c2cnn(C(C)C)c2)=O)C1 N1(C(C2=NN(C)C(=O)CC2)=O)CCC(C2CCCN(C(C34CC(F)(C3)C4)=O)C2)C1 C1(C(N(C(CC(=O)N(CC#C)CC2CC2)(C)C)C)=O)CCC(C)=C(C)C1 CC1CN(C)CCCN1C(C1CN(C(c2ccc3c(c2)CC3)=O)CCO1)=O C(C(F)C(=O)NC1(CO)CN(C(C2CCC(CC)O2)=O)C1)N(CC)CC N1(C(=O)NCCC2(C)CCOC2)CCC2(O)CC2C1 c1(CN2CCCC(CNC(c3ccc(OC)cc3)=O)C2)ccc(O)c(C)c1 n1(CCC)cc(Cl)c(C(N2CC(NC(=O)C(C)(C)OC)C2)=O)n1 n1(CCCCSc2nc(O)cc(COC(CSCC)=O)n2)c(C)cccc1=O N1(C(c2cc(Br)cs2)C(=O)NC(C(=O)OC)CC(C)C)CCC(C#N)CC12CC2 C1(CC(=O)NC(C(=O)NCC(F)(F)C(F)F)c2ccco2)CC2(CC2)CO1 C(c1ccc2[nH]ccc2c1)=CC(=O)N(CC(C)NC(CCC(C)OC)=O)C Cc1ccc(C(=O)N(C(C)(C(=O)N(C)CC2CCCCO2)C2CC2)C)c(C)n1 Cn1cc(C=CC(=O)N(C(C2(CC)CCC2)C)C2CC2)cn1.C(C1CC1)=C.OC(F)F Cc1cc(F)ccc1CC(N1CCCC(CNC(C2CC(C(C)C)=NO2)=O)C1)=O C1(CNC(C(C(C)C)(C)C)=O)CN(C(c2ccnc(F)c2N)=O)CCC1(C)C Cc1cccc(OCNC(=O)NCC(C)(C)CSCCl)c1C.C(C)(C)(C)O C(=O)(C(C)S(C)(=O)=O)NC1CCCC(CNC(C2C(CC)C2)=O)C1 O=S1(=O)CC2CN(Cc3ccc(Br)c(Cl)c3F)CC2(C(F)(F)F)C1 CC1CN(C(=O)CC2(O)CCCC2)CC1CC(=O)NC1CC(=C2CC2)C1 CC1CN(C(c2ccc(C(N)=O)o2)=O)CC1NC(=O)C(C)(C)OCC1CC1 CCCCC(CC)CC(=O)NCC1(F)CC(CNC(=O)CC2CCCC23CC3)C1 c1(C(N2CC(COC)(CNC(=O)CN(C)CCO)C2)=O)cnn2c1CCC2 N1(C(C(C=C)C)=O)CCCC(C)(C(=O)Nc2cccc(O)c2)C1 C(CCCCCC(=O)NCCCOC1CCC1)NC(C(C)N(CC)CC)=O c1(N2CCC(C)(OCC)CC2)nc(C)cc(=NCCc2ccncc2C)[nH]1 c1(CC)ncncc1C(C(C(C(=O)N(CC(CNC)O)C)OC)=O)=O.OC C1(NC(C2(CSC)CCOCC2)=O)CCN(C(C2(C)CC2(F)F)=O)CC(C)(C)C1 Cc1nc(O)ccc1C(=O)NCCC(C)N(C)C(c1cccc(CC2CC2)c1)=O N1(C(Cc2n[nH]c(=NC)s2)=O)CCC2C(C1)CN2C(=O)COC1CCOCC1 CCC(C)CC(C(=O)NCC(C)(O)C1CCC1)NC(=O)C(O)C1CCCC1 C1(CCNC(=O)C=Cc2cocn2)CN(C(C2CC(n3ccnc3)C2)=O)CCO1 c1(NC(C2CSC2)C)ccc(S(=O)(=O)NC2CCCN(CCO)C2)c(Br)c1 c1(OC)ccc(-c2cscc2C(=O)NCC(=O)NCC2CCC(C)N2)cc1 Cc1cccc(C(N2CCCC2CNC(=O)CC2OCCCO2)=O)c1F c1(OC)ncc(C(N2CCC(O)C2C(=O)Nc2ccc(I)cc2F)=O)cc1F N1(C(c2cc(N)cc(F)n2)=O)CCCC2CN(C(=O)CC3COCCO3)CC12 N1(CC)CCN(C(c2cc(OC)ccc2O)C(=O)NC)NC1=O.c1(C)ccccc1 C(CS(=O)(=O)c1ccc(CC(=O)OC)cc1)NC1(CCC)CC2NCCC12 C1(C)(COC)COCCN1C(c1cccnc1-c1ccc(F)s1)=O CN1CC(NC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)CC12CCCC2 Cc1cc(O)n2ncnc2c1NC(C1CC(C)(C)SC(C)(C)C1)=O C#Cc1ccc(F)cc1C(=O)NC(CC)(CC)CCNC(C1(COC)CC1)=O N1(C(CCNC(=O)NCC)=O)CCN(CCC(=O)OC)C(=O)C1 c1(C(N2CCN(C(CCC(=C)Br)=O)C(C)C2C)=O)ccc2nc(O)oc2c1 c1(C(C)C)ccc(C(c2nnnn2C2CC2)NCC2(CO)CCC2)cc1 c1(C(N2CCC(N(C(c3c(OC)cccn3)=O)C)C2)=O)ccnc2cc[nH]c12 c1(C(N(C(C)C(N2CCCC2CN(C)C)=O)CCC)=O)ccnc(OC)n1 CCC(C)C(O)C(=O)NC(C)(C)CN(C)C(c1ccc(CSCC#N)cc1)=O c1(NCC(C2CCCC2)NC(=O)CCC2CCCCO2)ncc([N+](=O)[O-])cc1Cl c1(OC(=O)CCNC(C)CCn2cccn2)ccc([N+](=O)[O-])cc1 C1(C)(C(=O)NCCN(C)C(c2cc(OC(F)(F)F)cc(Cl)c2)=O)CCC(=O)NC1 C1(C(=O)NC(C(=O)N(CCCC)C(C)CC)(C)C)COCCC1C c1(C(=O)NCCSC)cc(CNC(c2cc(CSC)cs2)=O)nn1C c1(NC(C2CC(NC(c3ccc(Br)c(Cl)c3)=O)C2)=O)nc(Cl)ccc1O n1(CCCCC(=O)N(CCC(F)F)C2CC2)c(=O)oc2ccccc12 C12(C(C)NC(C3CC(O)CN3C(=O)C(F)Cl)=O)CC3CC(CC(C3)C1)C2 C(=O)(C(C)CCCC(C)C)NC1CN(C(C2N(CC)CCOC2)=O)C(C)(C)C1 C(=O)(C(C)CC(C)C(C)=O)N1C(C(=O)NC2(C#C)CC(F)(F)C2)CC=CC1 c1(C(=O)NC2CC(C)N(C(=O)CCSC(F)(F)F)C2)ccc2oncc2c1 N(C1CCCc2cccnc21)(S(=O)(=O)Cc1ccc(-n2cccn2)cc1)CC N1(C(C(CCSC)OC)=O)CCN(C(c2cncc(N)n2)=O)CC1CO CC(C)C(O)C(=O)NC1CC1CNC(=O)CCc1nnc(C2CCCC2)o1 c1(OC)ccccc1NC(=O)C(c1ccc(C2CC2C)o1)N(C)CC1CC1(C)C N1(C(C2C(C(C)C)C2)=O)CCC(C)C(N(C(=O)C(=Cc2cccc(F)c2)F)C)C1 N1(C(C=C(C)C(C)C)=O)CCOCC(CNC(=O)CC(C)(C)C)C1 c1(C2(C(N3C(C(N)=O)CC(F)C3)=O)CC2)c(Cl)cccc1Cl C=C1CC2CCC(C1)N2C(=O)C(c1cccs1)NC(=O)CC(CC)C(C)C N1(C(c2cc(Br)c(C)s2)C(=O)NC(c2ccccc2)C)CCC(O)C(F)C1 CCCCCC(O)CNC(C12CC(NC(C3C4(CC4)C34CC4)=O)(C1)C2)=O N1(C(C(CC=C)CC)=O)CCCC2(C1)CN(C(C1COCCOC1)=O)C2 C1(N(C(c2cnc(CCC)s2)=O)C)CCN(C(=O)CCCCN(C)C)CC1C c1(C(=O)NC2C(NC(=O)Cc3ccc(Br)cc3F)C2)csc2ccccc12 c1(COC(CCC(C)NC(c2ccccc2)=O)=O)ccc2c(c1)CCCS2 CC(C)(C(=O)NC1(CNC(C2CCNC2=O)=O)CC1)C(O)c1cc(Cl)cc(Cl)c1 C(F)(F)(CN=c1ccc(Br)c(S(=O)(=O)N2CCC(C(N)=O)C2)[nH]1)C1(OC)CCC1 Cc1cc(C(=O)NCC2CCN2C(=O)CCSCC(C)C)nn1C(C)C c1(-c2c(OC)c(F)ncc2)cc2c(s1)CCN(Cc1ncc[nH]1)C2 c1(C(N2C(CN(C)C(C3CC34CCC4)=O)CC(F)C2)=O)ccnc2c1CCC2 C1(C(=O)NC2CCN(C(c3onc(C)n3)C)CC2O)CC2(C1)CC(C)(C)C2 N1(C(c2c(COC)cc[nH]2)=O)CC(NC(=O)C(CCSC)N(C)C)CC12CCC2 C(=O)(C1CC(=O)c2c(F)cccc21)NCC1CCN(C(c2cc(OC)ns2)=O)C1 C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2C3CNC(=O)C23)=O)C1 c1(C(N2C3CN(C(C(COC)C)=O)C(C3)C2)=O)cc(S(C)(=O)=O)cs1 N1(C(C(=O)NC(C)C)=O)CC2CC3CC2C1C3NC(c1cn2sccc2n1)=O C(=O)(C1CCc2ccccc21)NC1CC(C)N(C(=O)C(C)Cc2ccccc2)C1 N1(C(CC(C)(C)C2CC2)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)C2 c1(OC)ccc2c(c1)OCCC2NC(c1ccc(Br)c2c1OCO2)=O N1(C(CN(C(C(C(CC)C)=O)=O)C2CCC2)=O)CCC2(CCOC2)C1 c1(C(=O)NCC2(CCNC(C3CC(CC(F)F)C3)=O)CC2)cc(O)cc(Cl)c1Cl N1(C(C2N(C(C(C)OC3CCCC3)=O)CC(C)C2)=O)CCC2(CCOC2)CC1 c1(C(N(CC#C)C)=O)ccc2c(n1)CN(C(C1CCCCC1O)=O)CC2 Cc1cnc2c(C(=O)N(C3CN(C(c4cc(C#N)cs4)=O)CC3O)C)cnn2c1 N1(C(c2c(CC)nccc2)=O)CC2CCN(C(=O)Cc3ncoc3C)C(C2)C1 C1(CNC(c2ccc(Br)cn2)=O)COCCN1C(=O)CC1C=CCC1 N1(C(=O)NC(C2CC2C2CC2)CC)CC(C)CC1CO N1(C(CCC(C)O)=O)CCCC2(C1)C(NC(=O)CC1(C)CCCC1)CCN2C c1(CC(=O)NCCOC2CCN(C(C(CC)n3cncn3)=O)C2)c(C)noc1Cl C1(F)(C(=O)NC2C(NC(CC3CCCN(C)C3)=O)CC2)CCC(F)(F)CC1 C1(NC(c2c(C)cccc2N)=O)CC2(CCCCN2C(C2CCCC(O)C2)=O)C1 c1(CC)noc(CC)c1CC(=O)OCc1cncc(C(C)C)c1 O=C(C1CCCn2cnnc21)NC1CN(C(c2nc(Cl)ccc2F)=O)C1 Cc1cnc(CC(=O)N(C2CC(C(=O)NCc3[nH]cnc3C)C2)CC2CCCO2)o1 N1(C(C)=O)CCCC2(NC(c3ccc(Br)s3)=O)CCCC12 C1(CNC(CC(CC)(C)C)=O)CC2(CCOCC2)CN1C(C1CC(C#N)C1)=O c1(C(=O)NCC(C)N(C)C(c2ccoc2Cl)=O)ccc(F)c(C#N)c1 C=Cc1ccc(C(N2CC(NC(=O)C3=C(Cl)CCC3)C3CC23)=O)cc1 C1(CCNC(C=Cc2ncc(C)[nH]2)=O)CN(C(c2cscn2)=O)CCCO1 C(=O)(CS(=O)(=O)C1CCCC1)NCC(CO)NC(=O)CCCC1CCC1 CC1=C(C)CN(C(c2sccc2CNC(c2ccn(C(C)C)n2)=O)=O)C1 c1(C(=O)NC2CC(C)(NC(=O)CC3(O)CCCN(C)C3)C2)c[nH]c2cccnc12 C1(C(=O)NC(C(C)SC)C)CCN(C(C2CCCCCC2)=O)C(C)(C)C1 c1(C(N2CC3(CC(NC(C(C#C)(C)C)=O)C3)C2)=O)cc(Br)c2[nH]c(C)nc2c1 c1(CN=C(NCC(COC)F)NC(C)C2CC2)nnc2cccnn12 C(=O)(C1=CC2CCC(C1)C2)N1C(C(N(C)CCc2nccs2)=O)CCCC1 CCCCS(=O)(=O)NC(C)C(=O)NCCNC(c1cc(C(C)(C)C)n(C)n1)=O N1(C(C(=O)NCC2CC(C)OCC2)=O)CCC(C(F)(F)F)C1(C)C c1(N(C)C)ccc(NC(=O)CNC2CCCC2Oc2cccnc2)cc1 C1(N(C(c2cc(COC)no2)=O)C)CN(C(=O)CS(N)(=O)=O)CCC1O N1(C(c2c(C)ccnc2)=O)CCC2CCN(C(=O)C3=CCCCC3)CC2C1 C12(CNC(C(n3c(C)ncc3)C)=O)CCCC1N(C(c1cscn1)=O)CC2 CCCC(O)C(=O)N1CCCC1n1cc(NC(c2cccc(SCC)c2)=O)nn1 C(CN=c1[nH]c(=NCCC(O)c2ccccc2)[nH]c2ccccc12)N(C(C)C)C Cn1ncc2c(NC3C4CCCCCCC34)ncnc12 N1(C(CCC2(C)CC2)=O)CC(NC(=O)Cc2ccc(O)nc2)C2CC2C1 c1(C(N2CCC(NC(C(C=C)O)=O)C2)=O)ccc(-c2ccc(F)cc2)n1C C1(CNC(C2N(C(CCSCCC)=O)CCC2C)=O)CCCC(C)CC1 c1(N2CCN(C(=O)NC)CC2)nc(=NC2CC(F)(CO)C2)[nH]c2c1COC2.C1CC1 c1(CNC(COC)C2CC2)cc(Br)cc2nn(C)cc12 N1(C(CCc2ccn(C)n2)=O)CCCN(C(=O)CCC2CCC(=O)N2)CCC1 C(c1cc2ccccc2o1)=CC(N1CC(C(C)NC(c2c(C)ncn2C)=O)C1)=O c1(C(=O)NCC2CC(C)N(C(C3CCC3)=O)C2)nc2n(c1Br)CCC2 n1(C(CC)C)nnnc1C(c1nccs1)Nc1cnn(CCOC)c1 c1(OC)[nH]c(=NCc2n[nH]c(=N)s2)cc(N)c1F CCCCCC(C)(CC)C(=O)N1CC=CC(NC(=O)CSCCCC)C1 C(=O)(CC(P(C)(C)=O)c1ccccc1)NC(C1N(C(CCC)=O)CCC1)C Cc1ccc2c(CC(=O)NCC(CO)NC(C3(n4cccn4)CC3)=O)coc2c1 C(=O)(C1=CCCOCC1)N(CC(CN(C(=O)CSc1nncn1C)C)O)C Cn1cc2c(CN3CCC(O)C(C(=O)Nc4cccc(Br)c4F)C3)cccc2n1 Cc1cc(CNC(C2CC(n3cc(-c4ncoc4C(=O)O)nn3)C2)=O)sn1 O=C(CN=c1cc[nH]cc1)NC1CCCC(NC(=O)C(F)(F)C2CC2)CC1 Cc1c(C(=O)NC(C2CCCN2C(=O)C(C)NC=O)C)cnn1C(C)C C=C(C)C(C)(O)C(=O)NCC1CCCCN(C(=O)CCC2CCN(C)CC2)C1 c1(NC(c2cc(-c3ccccn3)c[nH]2)=O)cccc(C(F)(F)F)c1 Cc1cc(C(=O)N(C)CC2(O)CN(C(=O)CC3CCCC(C)C3)C2)oc1C(=O)O N1(c2snc(SC)n2)CCC2(CC1)CC(NC(c1cnc3c(cnn3C)c1)=O)C2 c1(C(=O)NC2C(OC)CN(C(=O)C(C)c3cncs3)C2)nn2c(c1C)OCCC2 c1(OC)cc(C(N2CC3CC2C3NC(=O)C(C)=C2CCCC2)=O)ccc1C#N C1(C(=O)NCCNC(=O)NC)CCCN(C(c2ns[nH]c2=O)=O)C1 c1(C(C(=O)NCCN(C(c2nnn(C)c2N)=O)CC)(F)F)cc(F)ccc1OC CCCC(CCCO)C(=O)N1CCC(C)C1CNC(=O)CCCn1ccnc1 C1(C(NOCC(C)C)=O)CC2(CC2)CN1C(c1ccc(=N)[nH]n1)=O N1(C(C(COC)Cl)=O)CCC12CCN(C(c1ccc(Cl)c(Br)c1)=O)CC2 C1(C(=O)NC(c2ccnn2C)CC)CC(=O)CN1C(c1csnc1Cl)=O c1(NC(CC=C)C)[nH]c(=NCC2(OC)CCCOC2)nc2scnc12 C1(CCNC(c2ncn(CC)c2)=O)CC(F)(F)CN1C(C1CC(C(=O)OC)C1)=O c1(CC(=O)NCC2(NC(=O)C(O)CN3CCCC3)CCCC2)cccc(O)c1 C(=O)(CCN(OC)C(=O)C(C)CSC)NC(Cc1cn(CC)nn1)=O N12CCC(CC1)C(=O)Nc1cccc(c1)C2.c1(COCC)cc(CSC)no1 C(=O)(C(C)C1=CCCC1)NC1CCCN(C(Cc2nnc(C)s2)=O)CC1 C(=O)(C1=C(C#N)CCC1)NCC1(OC)CN(C(c2ccc3cncn3c2)=O)C1 C(C)(C)(CC(=O)NCC1CN(C(C2CC2c2nc[nH]n2)=O)CCO1)N(C)C c1(C(N(CCCNC(=O)CC2CC2(Cl)Cl)C(C)C)=O)ccc2c(c1)C(C)CO2 C(=O)(C1=CCCC(C)(C)C1)NCC1COCCN(C(c2c(C)ncnc2)=O)C1 C(CCCC(=O)NC1CCCC(NC(c2n[nH]c(C)c2O)=O)C1)OCC C1(CC(=O)NCC(c2ccccc2)N(C(c2cc(C)[nH]n2)=O)C)SC(=N)NC1=O Cc1ncnc(C)c1C(=O)NC1CCC(C(=O)NC2CCCC3(C2)N=N3)CC1 CC1CCC(CO)N1N1CCN(c2cc(Cl)ccn2)CC1 N1(C(C(CC)CC)=O)CC2CCCC(CNC(=O)C#CC3CCCCC3)C2C1 Cc1nc[nH]c1CC(O)C(=O)NC1COCC1CNC(=O)C=CC(F)(F)F C(=O)(CCCCCCCCCO)N1CCC(NC(C=CC(C)(C)C)=O)C1 C1(NC(CC2N(CC)CCC2)=O)CC2(C1)CC2NC(=O)C(COC)COC C1(C(N2CCN(CC(C)F)CC2)=O)CN(C(=O)CC2=CCCC2)CCN1C c1(C(=O)NC(CN(C)C(C23CC(C2)C3)=O)(C)C)cn(C)nc1Cl C1(OC)CN(C(c2ccccc2F)=O)C(C)(CNC(c2ccc(C)c(C)n2)=O)C1 CC(C)C(C(=O)N1C(CO)CCC1CO)C(C)NC(c1cncc2[nH]ccc12)=O C1(OC)CN(C(c2ccco2)=O)CC1NC(C1CCC(C(F)F)CC1)=O C#Cc1cccc(C(=O)NC(CNC(=O)Cc2ccc(Cl)cc2)C2CCC2)c1C N(C1CCOc2ccc(Br)cc21)S(=O)(=O)c1ccc(Br)cc1F C12(C(N(CC(=O)NCCc3cnn[nH]3)C3CCC3)=O)CCC(CC1)CC2 C1(CC)(CC)CCCN(C(=O)C(=O)NN2CCN(c3ccccc3)C2=O)CC1 Cc1nc(O)ccc1C(=O)N(CC(C)CNC(c1cccc(O)n1)=O)C C(CCC(C)(C)C(=O)NC(C1CCCOC1)CO)NC(C1N(C)CCCCC1)=O C(C(C)NC(c1ccc(OC2CCOCC2)cc1)=O)(C(C)C)NC(C=CSC)=O c1(C(N2C(CNC(=O)CC3C4CCCCC34)CCC2)=O)cc2c(s1)CCOC2 Cc1c(C(=O)NCCCNC(c2cccc(Cl)c2)=O)cc(Br)cc1N Cn1[nH]c(=NC(=O)C(Cn2cncn2)Sc2ccccc2Cl)cc1Cl CC1CCCCC1(C)C(=O)NCC1CC(CNC(=O)Cc2c[nH]nc2O)C1 C1(NC(CC2(C=C)CN(C(C3CCC3(F)F)=O)C2)=O)CCN(C)CC1C#N N1(C(N(c2ccc(COC)cc2)C2CC2)=O)CC2CC1CCC2OCCO c1(CC2(NS(c3ccn(C)n3)(=O)=O)CN3CCC2C3)[nH]nc2c(Cl)cccc12 C=C(C(=O)N1CC2CC1C2CNC(c1c[nH]nc1-c1ccccc1)=O)C(F)(F)F C1(CCNC(C(F)=CC)=O)CCCN(C(c2ccc(Cl)c(C(F)(F)F)n2)=O)CC1 CC(C)(CC(=O)NCC1COC(C)(C)CN1C(c1ccc(N)cn1)=O)C(F)F CC1C(O)CCN1C(C1CN(C(C2C(C#N)C2(C)C)=O)CCO1)=O C1(NC(C2(C)CN(C(C(C)NC(C)=O)=O)C2)=O)CN(C(C)C)CC1C c1(C(=O)NCC(C)N(C)C(c2nn[nH]c2C(F)(F)F)=O)cc2c([nH]1)CCCC2=O Cc1ccc(CCC(=O)NC(C2CCOC2)CNC(=O)CCC#N)c(C)c1 C(=O)(C(CC1CC1)NC(=O)C=CC1CC1)N(CCN=[N+]=[N-])CC Cc1nn(C)cc1CCC(=O)NC(CNC(=O)CN1CC2CC2C1)C(C)C C(=O)(CCCC(C)C)N1CC(CCC)C(C(=O)NCCc2cc[nH]n2)C1 c1(C(N2CCN(C(c3c(CC)sc(=N)[nH]3)=O)C(C)C2)=O)cncc2nc(C)[nH]c12 Cc1cc(N)cc(C(N2CC(C(C)NC(=O)Cc3cccnc3Br)C2)=O)c1F C(C)(CC(F)(F)F)N(C(CCN(C(CCn1c(C)ncc1)=O)C)=O)C N1(C(c2cc(CC)cc(C)n2)=O)CCC2CN(C(C34CC5CC3C4C5O)=O)CC12 C1(C(=O)NC(CCC)CCO)CN(C(=O)C(C)(CO)OC)CC(C)(C)C1 c1(CN(C(CCNC(CC(C)C)=O)=O)CCNC(=O)C(C)SC)cccc(Cl)c1 c1(CN2C(C(N3CCNC(=O)C3)=O)CC(=C)C2)nccc2ccccc12 Cc1nn(C)c(C(=O)NC(C)CNC(=O)C(c2ccc(F)cn2)(F)F)c1[N+](=O)[O-] Cc1cc(C(C)C(=O)NC23CC(NC(=O)Cc4cc(C)on4)(C2)C3)cc(F)c1 C1(C(N(CC(=C)C)CC)=O)CC2CC1CC2NC(=O)CNC(=O)OC C1(C(=O)NCC2(OC)CCCC2)CC(C)(C)CCN1C(=O)C(O)CCSC C1(C(N2CC(C)C(CO)CC2)=O)CC2CN(C(=O)C(C)OC(C)(C)C)CC2C1 N1(C(c2ccc(N(CC)CC)cc2)=O)CC2CCC2(NC(C2CC(O)C2)=O)C1 C1(C(=O)NC2OCCN(C)C2)COCCN(C(c2cc(Br)oc2Br)=O)C1 C1(C(N2CC(SCC)C2)=O)CCCC(NC(c2cc(CO)c(C)o2)=O)C1 C(c1cc[nH]n1)=CC(=O)NC(C(N1CCC(n2ccnc2)C1)=O)c1ccoc1 O=C(C1=C(Cl)CC1)NCC1CCN1C(=O)Cc1cc(Cl)sc1Cl C=CC1(C2(C(=O)NC3CCC(CNC(c4ncncc4Cl)=O)C3)CCC2)CCC1 c1(C(=O)NCCNC(CNS(N(C)C)(=O)=O)=O)cc2c(Cl)cncc2s1 C1(NC(c2c(SC)cnn2C)=O)CCCC(NC(c2cc(C(F)F)no2)=O)CC1 c1(C(N2CCC(C(c3ccccc3)CO)CC2)=O)cc(Br)ccc1Cl CC(C(O)C(F)F)NC(=O)CC1CCCC1NC(c1cc[nH]n1)=O CC1CC(C(=O)N(C)CC2CCCN2C(C2CCOCC2(C)C)=O)CC(C)O1 C(=O)(CC1=NN(C)C(=O)C1)NC(CCC(=O)NC(CC(C)(C)OC)C)C(C)C c1(OC)cccc(COCCNC(N2CCC(OC(=O)C(C)C(C)O)C2)=O)c1 CCC(C)CC(C(=O)NCC(C)(C)CC(F)F)NC(=O)CN1CC(C)(C)C1 C(CCN(C)C(c1ccnc(C(C)(C)O)c1)=O)(C(C)(C)C)NC(CC(C)F)=O c1(C(N2CC(C(C(N3CCC(CC(C)C)C3)=O)OC)C2)=O)cc(O)n(CC)n1 C12(CNC(c3nn(CC)c(C4CC4)c3)=O)CCC1CCN2C(c1ccn(C)n1)=O C1(C(=O)NC2(CC=C)CCN(C(=O)C=CC(=O)N(C)C)C2)CCC2CC2CC1 C1(C)(C(N2CC(OCCNC(c3c(F)ccc(C)c3)=O)C2)=O)CCS(=O)(=O)CC1 c1(C(N2CC3C(CN(C(C4CC(C)C4)=O)C)C3C2)=O)ncc(OCC2CC2)cc1F C(=O)(CC(C)(C)C#N)NC(C)C(C)C(=O)N(CCF)C(C)C C#CCCCC(=O)NCC1(C(C)NC(=O)C(c2ccccc2OC)=O)CC1 CCCCC(C)CCC(=O)N(C(C)C(=O)NCc1nncn1CC)C1CC1 c1(C(=O)OC)c(NCC2CC3CCC2C3)cccc1Cl.C(C)=O c1(C(=O)NC(C(C)NC(C2C(COC)C2)=O)(C)C)oc2ccc(Cl)cc2c1C N=c1[nH]c(Cl)c(Cl)cc1C(=O)NCC(C1CCCC1)NC(=O)C=C1CCC1 C1(OC)CN(C(=O)CC(C)(C)OC)C(C)(CNC(=O)CCn2cnccc2=O)C1 CON(CCC(=O)N1CCCC12CCOC2)C(=O)C1CCOCC1(C)C N1(C(C=CSC)=O)CC(C2CN(C(=O)CC3CCC34CCC4)C2)C1 c1(SCCC(=O)N(C)CCNC(C2CCC2(F)F)=O)ccc(F)cc1 C1(CC(N2CCN(c3nc(C)cc(C)n3)C(C)C2)=O)CCCCCC1(F)F c1(C(N2CCC(N(CCC)C(c3cc(CO)on3)=O)C2)=O)ccnc2c1CCC2 N1(C(CCCSC(=N)N)=O)CCN(C(C2(C3CCCO3)CC2)=O)CC1 c1(C(N2C(CNC(C3C4CCCC(F)(F)C34)=O)CCC2)=O)cc(Cl)c(F)cc1O N1(C(C2(NC(c3c(OC)ccs3)=O)CCCC2)=O)CCCC2(CC2)C1 CC(CCCCNC(C1(O)CCOCC1)=O)NC(=O)C(F)(F)CN(C)C Cc1cc([N+](=O)[O-])ccc1NC(C)CCNC(=O)CCCCO C1(C(C)(C)C)CCCN(C(=O)NCCCNC=O)C1.c1(N)ccc(F)nc1 N1(C(c2cnc(C(C)C)s2)=O)CCN(C(c2cc3n(n2)CCC3)=O)C2CCCC12 C1(NC(c2cc(CC)ncn2)=O)CC2CC(NC(=O)Cc3ccsc3)C2C1 c1(C(=O)NC2CN(C(C(C=C)(C)O)=O)CC2O)cnn2ccncc12 N1(C(C(CCC)O)=O)CCCN(C(=O)Cc2cccc(Cl)c2OCC)CC1C c1(C(=O)NCC(C)(C2CC2)NC(C2CC=C(C)CC2)=O)cc(Cl)cc(Cl)n1 c1(C(N2CCC(NC(C3CC(F)C3)=O)C2)=O)cncc(-c2ccco2)c1 N1(C(C=C(C)C(F)F)=O)CC2(C1)CN(C(c1coc(O)n1)=O)C2 N1(C(C(C2CCN(C(c3c(CC)cco3)=O)C2)F)=O)CCC(F)(CO)C1 C(=O)(CCCC(F)(F)F)N(C)CC1(NC(c2ncncc2F)=O)CC1 O=C(N=c1ccnc2[nH][nH]cc1-2)C1CC2CC2N1C(c1csc(C(F)(F)F)n1)=O CC(C)CCC(C)N(C(=O)C(=O)NCC1CCN(S(C)(=O)=O)C1)C C(=O)(C(F)(F)CCc1ccccc1)NC(C(C)C)(C)CNC(c1c[nH]c(=N)s1)=O c1(CC(N2CCC3(C(NC(CCSCC)=O)C3)C2)=O)c(C)nc(O)nc1O c1(C(N2CCC(CC3CC3)C2)C(=O)NCCSC)cn2c(F)cccc2n1 N1(C(C(C(=C)Cl)(C)C)=O)CCC2CCN(C(c3ccn4c(C)cnc4c3)=O)C2C1 c1(C(=O)OC)cc(C(=O)NCCCCCNC(C2(C3CC3)CCCO2)=O)c(C)[nH]1 c1(OCc2ccc(C#N)s2)c(-c2cccc(Cl)c2)cccc1F c1(OC)ccc(SC(C)C(=O)NCCC2CCCN2C(=O)Cn2ncnn2)cc1 CC(C1=CCN(C)CC1)NC(C1CC2CN(C(=O)C(C)(Cl)Cl)CC2C1)=O CCCCC(C(=O)NC1CCCC1NC(=O)CC1CCCCCC1)C(C)C C(=O)(C1CCCn2ccnc21)N1CCC(OC)(CNC(C2CC3CCC2O3)=O)C1 N1(C(C)=O)CCOC(C(=O)N(C2CCCCC2O)C)CC1 C1(C(=O)OC)CN(C(C2CCOC(C)(C)C2)C(=O)NC2CC(CO)C2)C(C)CO1 S(=O)(=O)(c1ccc2[nH]c(=NCC(F)F)sc2c1)N(CCC(C)O)C Cc1cccc(C2=CCN(C(=O)C(=O)N(C)C(C3CCCC3)C)CC2)c1 C1(CNC(c2c(CC)noc2C)=O)CCCCCN1C(C1CCCOC1)=O C(C(=O)NC(CC(C)C)C(=O)NCC1CCCCCC1)(C(C)(C)C)OC CC(C)CC(C)(C)C(=O)NCC(F)CNC(=O)Cc1ccc2nn[nH]c2c1 C1(F)(CNC(C(=Cc2ccco2)C)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC1 N1(C(C=C(C)C)=O)CCC2(C=CCO2)CC1.n1(C2CC2)ccc(C)n1 C1(O)(CCNC(=O)Cc2ccsc2)CCN(C(=O)CC2CCC(F)(F)C2)C1 c1(NC(C(N2CC(OC)C(c3ccncc3)C2)=O)=O)cc(F)ccc1C C1(OC(C(N2CC=C(C)C2)=O)C)CCN(C(=O)CCN=[N+]=[N-])CC1 c1(CCC(=O)N(C)CC2CCCN(C(C3C(C=C)CC3)=O)C2)c(C)ncnc1O c1(C(N(CCCN(C)C(C2CC2C#N)=O)C)=O)cccc(C2CC(F)(F)C2)c1 CC1CCC(C(N2CCC(N(C(c3ccco3)=O)CC3CC3)CC2)=O)C(=O)N1 C1(C(C)C)CCCN(C(=O)Nc2cn(CC(N)=O)nn2)CC1 Cn1nc(C(=O)NCCC2(C(=O)NC(C3CCOC3)CO)CCC2)cc1Cl C12(C(=O)NCCOCCN(C(=O)C(C)(C)c3ccnn3C)C)CCC(C)(CO1)C2 c1(C(N2C(C)C(NC(=O)C(O)Cn3cncn3)CCC2)=O)ncnc2c1CCC2 C1(C(N2CC(C=C)(CC(=O)NCCC(O)C(F)F)C2)=O)CCCCCN1C C#CC1(C(N2CCCC(CC)CC2)=O)CCN(C(c2ccsc2)=O)C1 C(CCCC(=O)N1CC(NC(=O)CC(F)(F)F)CC1C)SC c1(C(=O)NCC(C)N(CC(N)=O)C)ccc(C(F)(F)F)o1 N1(C(c2c(C)n(C)nc2)=O)CCCC(C)C1CCNC(=O)C=C1CCCC1 N1(C(c2ccn(C(F)(F)F)n2)=O)CCC(n2ccnc2)C1 C1(C)(C(=O)NCC(C(=O)NCCn2c(CC)nnc2)O)CCN(C)CC1 C12(C=O)CC1CCN2C(=O)CC1CC(C)(C)CO1.N1(N(C)CCO)CC(NC)C1 c1(C(N2CC(O)(C(C)NC(=O)CN(C)C)C2)=O)cc(F)ccc1OC(=O)C1CC1 CCC(C)(C)C(=O)C(=O)NCCN(C)C(C1CCCC(C(N)=O)CC1)=O c1(C(N2CC(CNC(CC3(C)CC3)=O)C2)=O)c(Cl)n(C)c2cc(Cl)c(Cl)cc12 c12cc3[nH]nnc3cc1C(C=C)C(=O)N1CCC(O)(C1)CNC2=O.C1(C(C)C)(CC)CC1 N1(C(C(C=C)O)=O)C2COCC1CC(NC(=O)CC1CC(SC)C1)C2 N1(CC(N2CCN(C(c3c(C)nncc3)=O)CC2)=O)CC(=O)N(C)C1=O Cc1noc(C)c1C(N1CCCC1CN(C)Cc1ccnc(Cl)c1)=O c1(OC)ccc(C(=O)NC2CC2CNC(c2ncnc(O)c2Br)=O)cc1C CC1(C)CCOC1C(=O)NCCC1(NC(C2CCCC2(F)F)=O)CCC1 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2)ccc(F)c(Cl)c1N N1(C(c2ccc(-c3cc(C#N)on3)cc2)=O)CC2OCCOC2C1 C(C(C)(C)CCl)(c1n(CCCCCC)nnn1)NCCC(=O)N(C)C C1(C(=O)NC2CCCC2)CC2CC2N1C(C1CC1c1ccc(Cl)cc1)=O CC1C(C)N(C(c2nn(C)cc2N)=O)CCN1C(C1CC2(CSC2)C1)=O CC(C)CCC(C(=O)NCCc1ncccn1)NC(c1cc(F)cc(F)c1)=O C12(NC(c3cncc(C)n3)=O)CCOC(CNC(c3csc(C)c3N)=O)(C1)C2 C(=O)(C(CO)C(F)(F)F)N1CC(C(N2CC(=O)NC(C(C)C)C2)=O)(SC)C1 CC(C)C(CC(=O)NC(C)(C(=O)OC(C)(C)C)C1CC1)OC(F)(F)F N1(C(c2ccc(SCC)cc2)=O)CC(C)N(C(c2cnc(N)c(N)c2)=O)CC1C Cc1ccc(C(N2CCCCC(C)C2)C(=O)NCC2CCCO2)nc1Br c1(C(N(CC(CC)NC(=O)C(C)(C)C2CCCCC2)C)=O)scnc1C c1(C(=O)NCC2(NC(C3C(OCC)CC3)=O)CCCC2)ccnc(S)c1 N1(C(C2CC(N(C)C)C2)=O)CCC2(CCCC2CNC(C2CCCC(=O)O2)=O)CC1 C12(NC(c3c(Cl)nc(OC)s3)=O)CCN(C(=O)CCn3cccnc3=O)CC1C2 S(=O)(=O)(c1ccc(-c2nnc(C(F)F)o2)cc1)NC1CCC(C)CC1 c1(N2C3(CNC(C(CC)CC4CC4)=O)CCC2CC3)ccc2c(n1)CCCC2=O c1(C(C)C)n[nH]cc1C(=O)NCc1n[nH]cc1C(N1CCC(CN(C)C)C1)=O N1(C(C2CCCCN(C(CC(=O)OC)=O)C2)=O)CCCC2CCCCC12 CC(C)C(C(=O)N(C)CC1CCCN1C(=O)C1CC1)NC(=O)OC(C)(C)C N1(C(CN(CCC=C)C(C)=O)=O)CCC2CC12CCCN1CC=CC1 N1(C(c2c(C(C)C)ncnc2)=O)CC2CCC(CNC(=O)C(CO)N(C)C)(C2)C1 c1(C(=O)NC2CN(C(c3ccc(CO)nc3)=O)C2)ccc2ccncc2c1 C1(C(=O)NC2CC=C(C)CC2)CC2CCC(C1)C2 C1(C(N(C(C)CNC(c2cc(C3CCC3)no2)=O)C)=O)COCCN1CC(F)F N(C)(C(=NCC1=C(C)OCCS1)NC1CCC1)Cc1ccc(C(=O)NC)cc1 C(C#CC(=O)NCCC(C)NC(=O)Cn1nnc(C)n1)(OCC)OCC CC1CCCC(CC(=O)NC2CC3(C2)CC3C(=O)NC2CN(C(N)=O)C2)O1 C1(NC(CCNC(COC)=O)=O)CC(C(=O)NC2CC3(CCOC3)C2)=CC1O N1(C(C2(C=C)CCN(C(c3ccnc(CO)c3)=O)C2)=O)CC2(CO)CCC1CC2 c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)ccc2cc(Cl)ccc2c1 C1(NC(CC2CC(SC)C2)=O)CC(CC(=O)NC2(CN(C)C)CC2)C1(C)C N1(C(c2coc(Br)n2)C(=O)NC)CC(C(=O)OC)C2(CCCCC2)C1 C1(NC(=O)CN2CCCS2(=O)=O)CS(=O)(=O)C2CN(C(c3cscn3)=O)CC12 C1(N(CCC(=O)NCCN(C(C2CC2c2cccnc2)=O)CC)C)CCCCCC1 C1(CNC(C2(SC)CC2)=O)CN(C2CCN(c3ncccc3Cl)C2)CC(C)(C)O1 CC1CC(CC(=O)NCCC(O)CNC(c2ccc3c(c2)CC3)=O)CC(C)(C)C1 c1(CC)ncc(C(=O)NC(CCN(C(=O)Cc2coc(C)n2)C)C(C)C)cn1 N1(C(c2c(C)nns2)=O)CCCCC1CNC(=O)Cc1ccn(C)n1 C#CCCC(O)C(=O)N1CC(CNC(c2c(Cl)cccc2Cl)=O)CC1(C)C N1(C(C)C)C(=O)COCC1C(=O)NCC1C2CC1N(C(=O)Cn1cncn1)C2 C1(C(=O)NC(C(C)C)CNC(c2cncc(Cl)c2)=O)CN(CP(C)(C)=O)C1 N1(C(C2CN(C(N)=O)C2)=O)CCCC(NC(=O)C#CC2CC2)C1 Cc1cnnc(O)c1C(=O)NC1CCCC1CN=c1[nH]nc(C(C)(C)C)o1 C#Cc1cccc(CC(=O)N(C(CNC(c2ccc(F)cc2C)=O)CC)C)c1 C(CC(=O)NCC(C1CCCN1C(c1cc(C)cs1)=O)(C)C)(C(F)(F)F)OC N1(C(CC(CCC)C)=O)CC(c2cn(-c3cnn(C)c3Br)nn2)C(O)C1 C(=O)(C1=CNC2=NCCCN12)N1CCN(C(c2ccc(C)n2C)=O)CC1C1CC1 c1(C(C(=O)NC(C)CC)N(CCOCC)C)ccc(CO)c(C)c1 C1(C(=O)NCCN(CCOC)C(C2SCCCS2)=O)CCC2(CC1)CC2 c1(CN(CC(c2ccccc2)NC(C2CC(OCC)C2)=O)C)ncncc1OC CC(CNC(c1nocc1Cl)=O)CC(=O)N(C)CCc1nccs1 C(=O)(C1CCC(=O)c2ccccc21)N1CCN(C(c2ncn(C)n2)=O)C(CF)C1 CN1CC(C(=O)NCC23CC(CCO2)C3)N(C(=O)COCC2CCOC2)C1 C(=O)(C(Cc1ccc[nH]1)N(C(C)C(=O)OCC)C1CC1)NCCC c1(NC(C2CC(F)CN2C(c2ccc(Cl)nn2)=O)=O)ncc(Br)nc1Br c1(C(C(=O)NC(CC)(C)C)N(C)Cc2cnn[nH]2)cn(C(C)C)cn1 C12(NC(c3c(CC)c[nH]c3)=O)CC3CCC(C1C2)N3C(=O)CCOC1CCC1 C1(CC)CCN(C(C2CCCC(CF)C2)=O)C1C(=O)NC C#CC1CC1C(=O)NCC1CCC1NC(=O)CCSC CCC(C)CC(C)C(=O)N1CCC(CNC(c2cccc(OC(C)C)c2)=O)C1 C(=O)(CC(C)(C)C=C)NCC1(CNC(CCCOCC=C)=O)CCCCC1 CC1(C)COC(C(=O)NCCCCCNC(C2COCC2(C)C)=O)CO1 C1(C(=O)NCC2(C)CC(NC(CN3CC(CC)C3)=O)C2)CN(C)CC(C)O1 N1(C(CCN(C)CCO)=O)CC2=C(C1)CN(C(=O)CN1CCCC1CSC)C2 C(CCC(=O)N(C(CNC(=O)CCCC1OCCO1)C1CC1)C)=CCC=C C1(C(=O)NC(C2(C(=O)NCC=Cc3cccnc3)CC2)C)CCC2(C1)N=N2 CC(F)(F)CCCC=O.C1(N2CCOCC2=O)CN(c2nnnn2CCF)CCC1O N1(C(=O)Cc2cnccc2Cl)CC(C2CCCN(C(C3CCC4(C3)N=N4)=O)C2)C1 C=CCCCCCC(=O)NC1C=CCN(C(=O)CCOc2ccc(Cl)c(Cl)c2)C1 C1(C(N2C(C(=O)NCC(=O)NC3(CC=C)CC3)CSC2)=O)CCOCC1 C=CCC(CC(C)C)C(=O)NCC1(NC(c2ncccc2C)=O)CCC1 c1(C(N2CC3CC3(C(=O)Nc3cncc(F)c3)C2)=O)c(C(F)(F)F)cccc1Cl Cc1c(CC(N2CC(NC(C3OCCO3)=O)C3(CC3)C2)=O)ccc(Cl)c1Cl c1(CNCC23C(CN(C(c4cc(C)[nH]n4)=O)C2)C3)c(Br)cc(Br)c(O)c1Br C12(C(N3C(CNC(C4N(C(C)=O)CCCC4)=O)CC3)=O)CCC(C)(C(=O)O1)C2(C)C c1(C(N2CCCC(C(=O)NC(C=C)C)C2)=O)cccc(Br)c1O c1(CC(=O)NCC2CC(OC)CN2C(C2CCN(C)C2)=O)c[nH]c2cnccc12 C12(CNC(c3cc(C)on3)=O)CN(C(c3cnc4ccnn4c3)=O)CC1CCO2 N1(C(=O)OCC)CCC(C(N2CC(N3CC4C(C(=O)O)C4C3)C3CC23)=O)CC1 N(C1CCCc2c1cnn2C1CCCC1)C(CNS(C)(=O)=O)=O C(=O)(CC(C(F)F)NC(C1CN(C2CCC2)C1)=O)Nc1c(C)nccn1 C1(NC(C(COC)OC)=O)CCC(O)CN(C(=O)CCN2CCN(C)CC2)C1 c1(C(N2CC(CNC(C(C(CC)C)O)=O)(COC)C2)=O)cn(C)c2ncccc12 c1(C(=O)NC2(C(=O)NCC(c3ncc[nH]3)C)CCC2)cc(C(F)F)cs1 C1(C(N(CCCNC(=O)CC2CCCC2C)CCC)=O)CC(F)(F)C1(C)C C1(CNC(=O)NCCC(C=C)C)(CF)CC(F)(F)C1 CCCCCC(C)(CC)C(=O)NC1CCN(CCOCC(F)F)CC1C C1(O)(CN(C)C)CCN(C(c2ccnc(CNC(C3(C)CCCS3)=O)c2)=O)C1 CCC(O)CC(=O)NCC(C)NC(=O)CCc1cnn[nH]1 c1(N(C)C)nc2cccc(C(N3CCCCCC3CNC(C3(O)CC3)=O)=O)c2o1 c1(CC(N2C3CN(Cc4cccc(F)n4)CC23)=O)ccccc1[N+](=O)[O-] C(F)(C(=O)NCCC1CC(NC(=O)C(C)n2cnnn2)C1)OC C1(NC(CSCC(=O)OC)=O)CC2(CCN(C(c3ccns3)=O)C2)C1 C1(C(N(C)Cc2cn[nH]c2)=O)CC12CCN(C(c1cnc(S)nc1)=O)C2 c1(C(=O)NCC(C(C)(C)C)NC(=O)C(O)C2CCC2)cccc(F)c1C#N CCCCC(C)C(=O)NC(C)CC(C)NC(c1cn(CCO)nc1C)=O C12(C(=O)NC3(CO)CN(C(C=C(C)Cl)=O)C3)CCCC1(C(N)=O)C2 N1(C(C(c2cccs2)NC(c2c(C)n(C)cc2)=O)=O)CC2CC3CC2C1C3 S(=O)(=O)(c1ccccc1COCC1CCCN1C)N(CCC)CCC C(=O)(CC1=NNC(=O)C1)N1CCOCC(CNC(=O)COCC2CCC2)C1 C1(C)(C(N2CC(CC(=O)NCC(C(C)C)O)OCC2)=O)C(C)(C)C1(C)C C(N=c1ccn(CC(=O)NCc2cccc(Br)c2)c(O)n1)c1ccc(C)cc1F C=Cn1nccc1C(=O)NC1(CCNC(C2ON=C(C)C2C)=O)CC1 C(CC(F)F)(C(=O)NCCN1CC2CC2C1)NC(c1nnn(C)c1N)=O CC1CC(=O)NC(C(N2CCC(C)C(CC(=O)NCCC(O)C(F)F)C2)=O)C1 C1(C(=O)NCC(C)(C2CCC2)NC(C=CC(CC)=CC)=O)CC(C)=NO1 c1(OC)ccc(F)c2[nH]c(C(=O)NCC3(NC(=O)CN4CCOC4=O)CC3)cc12 C1(C2CCN(C(C3(CC)CC3)=O)C2)CCCCN1C(=O)CCC(N)=O C1(C(=O)NCC=CCNC(c2nccc(C)c2)=O)CC2CCCC(C1)C2(F)F N1(C(c2ccn(CC)n2)=O)CCCCC(CNC(=O)Cc2conc2C)C1 CCCCCC(C)CC(=O)NCCn1cnnc1C(N1CCCCCC1CO)=O N1(C(c2c[nH]c(=NC)o2)=O)CCC(C)(C)C1C(=O)NC(c1ncc[nH]1)CO C1(CC(=O)NC2(C=C)CCC2)CCN(C(=O)C(F)=C(C)C)C1(C)C C1(CNC(c2c(C)ncs2)=O)C2CCCC1N(C(=O)CSc1cn[nH]c1)C2 C1(C(=O)NC2CC(C)(CNC(C3CC(O)C3)=O)C2)CCCC(C)(C)CC1 C(c1cncc(F)c1)=CC(=O)NC(C1(O)CCN(C(c2cnc(CC)s2)=O)C1)C C1(NC(c2cnc(Cl)s2)=O)CC12CCN(C(=O)CN1CC=CC1)CC2 S(=O)(=O)(c1ccc(Br)cc1)N1CCC(N2CCCN(CCOC)CC2)C12CCC2 c1(C(=O)OC)ccc(F)c2c1CN(S(=O)(=O)Cc1cccc3cc[nH]c13)CC2 N1(C(C(CC#C)C)=O)CCCC2CN(C(C3CC(SC)C3)=O)CCC12 C1(CC)CN(C(C2CCC(=O)N2)=O)CC1NC(c1nn(C(C)C)nc1Br)=O N1(C(C(N2CCCCC2=O)C)=O)CC(NC(C2CC3CC3C2)=O)CC12CCCC2 N1(C(CCn2c(C)csc2=O)=O)CC(NC(C23CC(CCO2)C3)=O)CC(F)C1 C1(CNC(C(CC=C)(C)C)=O)CN(C(c2ccc(SC)[nH]2)=O)CCC1(F)F CCC(CC(F)(F)F)C(=O)NC(CNC(=O)COc1ccn(C)n1)CO N(C1CN(C(=O)CN=S(C)(C)=O)Cc2ccccc21)C(C(C)OC)=O CC1(C)CC(C(=O)NC2COCC2C(=O)NCCOc2ccncc2)CCO1 C(=O)(C(C)C(C)NC(c1nn(C)cc1C)=O)NC1(C)CN(C(=O)OC)C1 C=CCC(C)(C)C(=O)NC1CCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 c1(C(C)=O)ccc(C(=O)NCC2CN(C)CCN2C(=O)C(F)CC(C)C)cc1C C(C1c2ccsc2CCN1C(c1sccc1F)=O)NC(CSCC=C)=O N1(C(=O)NC2CCCCN2)CCc2nc[nH]c2C1c1ccc(F)cc1 C1(C(=O)NCC(CN(C)C(C23CCC(CC2)CC3)=O)O)CS(=O)(=O)CC12CC2 N1(C(C(C(C)C)NC(C)=O)=O)CCC12CN(C(C1CC(=O)NC(=O)N1)=O)C2 CCCCC(C(=O)N(CCOCC)CC1CC1)NC(=O)C(C)(C)Cl C(C(=O)N=S(C)(C)=O)NC(c1ccncc1C)c1n(CCCSC)nnn1 C=CC1CCCN(N2CCN(c3nc(C(C)(C)C)ns3)CC2)C1 CC(C)(C)C(O)C(=O)NC1C2CC(NC(=O)C(C)(F)CC3CCCC3)CC12 C1(C(N2CC3C(CNC(C(C4CCOCC4)C)=O)(C3)C2)=O)(CF)CC2(CCC2)C1 c1(OCCC)cccc(CCC(=O)NCC23CC2CN(C(=O)CC(C)OC)C3)c1 CC1(C)COCCC1C(N1CCC(CNC(=O)Cc2csc(C(N)=O)n2)CC1)=O CC(C)(C)C1CCNc2c(C(=O)NCCNC(=O)CCc3cnccn3)cnn21 N1(C(C=C(COC)C)=O)CCC(NC(=O)CSC2CCCCO2)C1C1CC1 C12(NC(C(CC=C)N(C)C)=O)CCC(CNC(C3(COC)CC(=C)C3)=O)(C1)OC2 C1(NC(c2ccc(=O)n(-c3ccc(I)cc3)c2)=O)CNC2(CCC2)C1 C1(C)(CNC(CCC2(C)CC2)=O)CC(F)(F)CN1C(c1cccc(Cl)c1O)=O C1(CC)CN(C(C2COCC2NC(C2CCC3CC2CO3)=O)=O)CCCO1 C1(CC)CCCN(C(C2CC(=C3CC3)C2)=O)C1C(N1CCN(CC(N)=O)CC1)=O c1(C(N2CC(C)(NC(=O)Cn3nnc(C(C)(C)C)n3)C2)=O)cn2cccnc2n1 C(=O)(CC(CC)NC(C1(CC)CCCN1C)=O)NC(C=C)C N1(C(CCNC(C)=O)=O)CCCCC1C(C)NC(C1CC(CC2CC2)C1)=O C1(Nc2cc(OC)nc(OC)n2)CC(C)(C)C12CCC2 C1(NC(C(CC)CC)=O)C2CCN(C(=O)CC3CCCO3)CC12 c1(C(=O)NCC(N(C)C(C2CCC2C(C)(C)C)=O)C2CC2)cc(Cl)c(Cl)n1C C1(NC(C(C)(C)CC#N)=O)CCC2(CC1)CCN(C(c1conc1C1CC1)=O)C2 c1(CNC(COCC)=O)ccc2c(c1)CCC2NC(=O)C#CC1CCCCO1 CCCC(C(=O)N1CCC(N(C)C)C1)NC(C)=O.C12CC(C1)NC2=O C(=O)(CC(C)C(=O)OC)NCCC1CCN(C(C(CC)CC)=O)C1 C=C=CCCC(=O)NC(C)(C)C=CC(=O)NCC(N1CCOCC1)=O c1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)CO)C2)[nH]c2ccc(Cl)cc2c1Cl c1(OC)c(F)cc(C(=O)NCC(C)(CO)NC(C2CCC(C)(C)CO2)=O)cc1Cl c1(C2C(C(=O)NCCOC)C2)noc(C)n1 Cc1csc(=Nc2cccc(C3CCCCC3)c2)n1C1CCCSC1 c1(CNC(c2ccc(C)n2C)=O)cc(O)cc(=O)o1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCC1(CNC(=O)CCCS(N)(=O)=O)CC2 N1(C(C(C=C)(C)C)=O)C2CCCC1CC(NC(c1ccccc1S(C)(=O)=O)=O)C2 c1(C(N2CCC(c3ccccn3)C2)C(=O)OCC)ccccc1C CCC(C)C(O)CC(=O)NCC1(NC(=O)C2=C(C#N)CCC2)CCCCCC1 CC(C(C)C(=O)NCC1(Nc2ncccc2[N+](=O)[O-])CCOCC1)S(C)(=O)=O N1(C(C2C(C(C)O)C2)=O)CC(CNC(C2CC2(C)C)=O)C1 c1(C(C(=O)NCC(CO)NC(=O)CC2CSC2)O)cccc(Cl)c1 N1(C(C(N2CCC(C)C2)=O)=O)CCCC(O)(CNC(C2(C(N)=O)CC2)=O)CC1 C1(CNC(C2CC(CCC)C2)=O)CCC(NC(=O)CCN2CCC2)CC1 c1(C(=O)OC)ccncc1S(=O)(=O)NC(=O)NC1CC(CCN(C)C)C1 N1(C(C(C2CCCC2)NC(c2ncccc2F)=O)=O)CC2CCC(O)C2C1 c1(N2CC(CN(C(=O)CC3CCCCC3(C)C)C)OCC2)ncc(C#N)cc1Br N1(C(CCCC)=O)CCC(NC(c2cc(C(N)=O)co2)=O)C(CC)C1 C(=O)(C(CNC(=O)CCCn1cncn1)OCC(=O)NC1CC(SC)C1)NC.C1CCC1 C1(F)(C(=O)NCC2C(C(NOCC3(C)CC3)=O)CCO2)CCOCC1 Cc1c(NC(=O)C(CCC2CC2)NC(c2csnc2Cl)=O)cnn1C N1(C(C(F)=CC)=O)CCC(CNC(c2n[nH]cc2-c2ccccc2)=O)C(C)C1 c1(CC(=O)N(CC(O)CNC(C2(C)C=CCC2)=O)C)c(F)cccc1F N1(CC)CC(C(=O)NCc2cccc(C(N3CCCC3C(N)=O)=O)c2)CC1=O Cc1nn(C)cc1C(=O)NC1CN(C(c2nocc2C)=O)CC1C C1(CNC(CN(C(C)C)C)=O)CN(C(C2CC(N3CC(O)C3)C2)=O)C1 C1(C(=O)Nc2c(C)nsc2)(NC(c2cc[n+]([O-])cc2)=O)CCCC1C NC1COC2(C(N3CCOC(c4ccc(F)c(Cl)c4)C3)=O)CC1C2 C(=O)(C1=CC2CCC(C1)C2)N1CC(C)CC(CNC(C(CC#C)(C)C)=O)C1 c1(NC)cc(NCCC(C)(C)NC(=O)C2=C(C)OCC2)ccc1[N+](=O)[O-] C=C(C)CC(C(=O)N(C(C)CCSC)C)NC(c1ncoc1CC)=O C1(CCCC)CN(C(C2CC23CCC3)=O)CCN1C(=O)C#CC1CC1 C1(C(=O)NCCC2CCCC2(F)F)(CNC(=O)OC(C)(C)C)CCOCC1 c1(N2C3CC(N(C)C)CC2CC3)nc(=NCc2cnns2)[nH]c2c1CCCCC2 C(=O)(C1=CCCCCC1)NC(CC#C)C(=O)NCC(C)(O)CCC C(N=c1[nH]c(=NCCC(C)OC)[nH]c2cccnc12)c1n(CCC)ccn1 c1(CNC2C(C(=O)Nc3c(C)ncnc3)C2)c(F)cc(C#N)cc1F N1(C(C(C)C2CCCC2)=O)CC2CC(C1)N(C(c1noc3ncccc13)=O)C2 C1(CNC(CN(C(=O)CSCC(F)(F)F)CCOC)=O)CC1(C)C C(=O)(CC(C)(C)CN(C)C)NC(C)C(C)C(=O)NCCS(N)(=O)=O c1(-n2ncc(C(N(CC(CNC(C(CC)(C)C)=O)O)C)=O)c2)ccc(F)cc1F N#Cc1ccc(CNC2(c3nnnn3CC(F)F)CCNCC23CC3)cc1F C1(N(C)C(c2nnn(-n3cccn3)n2)=O)CCC(CNC(=O)CCC(N)=O)CC1 C1(CC(=O)NCCCOCCNC(C2(C(N)=O)CC2)=O)CC=CCC1 c1(OC)cc2c(cc1CN1CCC(CC(C)C)(CO)CC1)OCO2 c1(NC)ccc(C(=O)NCC2(CNC(C3CC3F)=O)CC2)cc1[N+](=O)[O-] C(C(CC(F)(F)F)NC(C1CC(=O)NC1(C)C)=O)NC(C(CC)=CC)=O N1(C(CCCC)=O)CC(C(=O)NC23CC(F)(C2)C3)C(F)(F)C1 O=S(=O)(c1cccc(N2CCOC(C(F)F)CC2)n1)NCCCOC1CCCC1 N1(C(C2N(C(CCCOC(C)=O)=O)CC2C)=O)CC2(CCN(C)CC2)C1 C1(C(=O)NC2C(SC)CCC2)CC(O)CCN1C(c1cc(F)cnc1O)=O C=C1CC(C(=O)N(CC(C)C#N)CC2CC2)(CNC(C)=O)C1 c1(C(N2CCC(C(C)C#N)CC2)C(=O)NC)ccc(OCC(C)C)nc1C C1(CC)CN(C(=O)CSCC(=O)OC)CCC1NC(c1ccnc(NC)c1)=O C1(NC(Cc2c(C)n(C)cn2)=O)COC2(C1)CN(C(C1CCO1)=O)C2 c1(CNC(C(C(C)OC)NC(=O)CC2CNC(=O)O2)=O)nn(C)c(=O)n1C C1(NC(C(=O)NC(C)C)=O)CCN(C(c2cc(Br)ccc2F)=O)CC1C C(=O)(CC(C(F)(F)F)n1cccn1)NCC1(CCNC(C(C)N(C)C)=O)CC1 N1(C(c2c(C)cccn2)=O)CCC(NC(C2CCC(=O)N2)=O)C(CO)CC1 c1(C2N(C(C=CC(=O)OCC)=O)CCC2)ccc(Br)cn1 c1(NC(c2cnn(-c3ccc(O)nn3)c2C(F)F)=O)nc2ccccc2o1 Cc1ccc(C(=O)N(CC(C)N(C(=O)CCn2cncn2)C)C)c2cccnc12 c1(OC(C)C(=O)N2CCC2CNC(=O)CCC2CCCO2)ccc(F)cc1 C(=O)(C1CCC(=O)c2cccn21)NCCN(C(C=CCCC)=O)CC c12onc(C)c1OC(=O)C2.N1(C2CN(C(C(=O)NCC)=O)C2)CCOC1=O C(=O)(C1=CCC(F)(F)CC1)NCCCOCCNC(C1CCCC(=O)N1)=O C(C(C(=O)N(CCCOCCNC(C1CC1C)=O)C)C(F)(F)F)OC c1(C(=O)NCC2C(CNC(c3c(CC)nns3)=O)C2)cc2c(F)cc(Cl)cc2[nH]1 CC(N=c1nc2c(cnn2C)c(NCc2ccc(C(F)(F)F)o2)[nH]1)C1CC1 Cc1nccc(C(=O)NCC2CCCN(C(C34CC5CC3C4C5)=O)C2)c1Cl CC(C)CS(=O)(=O)CC(=O)N1CCOCC(CNC(=O)C(F)C2CCOC2)C1 C1(NC(C(CC)O)=O)CCN(C(c2cccc(N)c2F)=O)CC12CCC2 CC12CCC(C(=O)NCc3cccc(NC(=O)C(=O)c4cccs4)c3)(CO1)C2 C1(NC(C2OCC(C)C2)=O)CC2CC(C1)N(C(=O)C=Cc1ccccn1)C2 C1(C(C(=O)NCC(CCNC(CCSCC)=O)OC)O)CCCCCC1 C(C(CNC(=O)NC1(c2noc(C)n2)CCC1)C(C)C)OC Cc1ccccc1CC(=O)NC(C)(C)CC(=O)N(C)CCN(C)C1CC1 C1(CNC(C(C2CC2)OC)=O)CN(C(=O)CCc2nc[nH]n2)C2(CCC2)C1 c1(C(=O)NC2CC(CO)NC2=O)cccc2ccc(Br)nc12 Cc1c(C(N2CCCC(CNC(C3(C)CCC(C)C3)=O)C2)=O)cnc2ncnn12 C1(c2cn(CC(N3CCN(C)CC3)=O)nn2)CC2(CCCN2)C1.C(C)(C)C Cc1ccc(F)c(CS(=O)C(C)C(=O)N(Cc2ccccn2)Cc2ccco2)c1 N1(C(c2c(C)nn(CCO)c2)=O)CCCC(NC(c2cn3c(n2)CCC3)=O)C1C CC(=O)C(C)(C)CC(=O)NC1CCC(NC(=O)C2=CCCSC2)C1 N1(C(Cc2c(C)occ2)=O)CCC2OCCN(C(=O)CNC(=O)C(C)(C)C)C2C1 N1(C(CSCC)=O)C2CCCC1CN(C(C1Cc3ccccc3C1)=O)CC2 c1(OC(c2ccc(N(C)C)cc2)CC)cccc(F)c1 N(C(=NCCCOCCN(C)C)NC1CCN(c2ccccc2)C1)CC(=C)C C1(CNC(c2c(OC)cc(C)cc2)=O)CC2CCC1N(C(=O)CC(=O)N(C)C)C2 c1(CC(=O)NCC=CC(=O)NCCC=CC=C)c(C)noc1C C12(C(=O)NCC(=O)OC)CCCCN1CCC2.c12cc(F)ccc1NC2 C1(C(=O)NCC2(C)CCC(NC(CC(CCC)O)=O)CC2)CCc2nccn2C1 C(c1c[nH]nc1C)=CC(=O)NCCNC(C1N(CCC)CCC1)=O C#CC1CCCN1C(=O)C(CC1CC1)NC(=O)C(C)(CO)OC c1(N(C)C)ncccc1C(=O)NC1CCN(C(=O)CN2CCNC2=O)C1 N1(C(CC(CCCC)NC(=O)C(C)(C)OCC)=O)CCC2CCN(C)CC12 c1(C(N2CCC(NC(C(C)OCCC=C)=O)CC2)=O)ccc2cnoc2c1 Cc1[nH]nc2ccc(C(=O)N(C(C)CN(C)C(C3CCCCCC3)=O)C)cc12 C1(C(F)(F)C(=O)N2CCC(N(C)C(c3ccncc3Cl)=O)C2)(OC)CCCCC1 N1(C(C(=O)NCC2CCC(c3nc(O)cc(C)n3)CC2)=O)CCc2n[nH]cc2C1 C(=O)(C#CC1CCCO1)N1CCC(N(C(c2c(CC)nccc2)=O)C)C1 C1(CCC)(NC(c2ccc(=O)n(C)c2)=O)CCN(C(=O)CN(C)C(C)C)CC1 C1(CCC)CCC(NC(=O)C(=O)Nc2ccc(-c3nncn3C)nc2)CC1 C(=O)(C1=CCN(C(C2CC=C(C)CC2)=O)CC1)NCC1(SC)CCC1 CCCC(C(=O)N(CC(F)(F)COC)C)NC(C1(OC)CCOCC1)=O C12(N(C(C=CCCC)=O)CC)CCC(CNC(=O)C(C#N)C(C)(C)C)(CC1)OC2 N1(C(C2C(CCC)C2)=O)CCN(C(c2ccc(F)c(C(C)C)c2)=O)CC(C)C1 Cc1cc(Cl)cc(N)c1C(=O)NC1CCN(C(=O)C(C)CC(F)F)C1 CC1(C)CC(CO)CN(C(c2ccc(CNC(=O)C3=COCCC3)nc2)=O)C1 C=CCC(CN(C)C)C(=O)Nc1c(C)ccnc1OC C1(NC(CCc2ccc(C)nc2)=O)CC12CCN(C(=O)Cc1cnc[nH]1)C2 c1(CN(C(=O)CCn2nc(-c3cccs3)oc2=O)CC(=C)C)cccc(Cl)c1 C1(CNC(c2c(C)c[nH]n2)=O)CC(C(=O)NC(CO)C(F)(F)F)=NO1 C1(C(N(C2CN(C(c3cnc(CC)o3)=O)CC2O)C)=O)CCc2nnc(C)n2C1 c1(C(=O)NC2C(CNC(c3cc(CC)on3)=O)CC2)ccc(=O)n(CCOC)c1 C1(C2CN(C(=O)C=CC3CCCO3)C2)(NC(Cc2cn(C)nn2)=O)CC1 n1(CC)ncc(Cl)c1C(=O)NCC(C)N(C(=O)CC(C)C1CC1)C C(c1cccc(Cl)c1)=C(C(=O)NC1CCN(C(c2c(C)nc(OC)s2)=O)CC1)C c1(NC(CN(CCC=C)CC(=O)C2CC2)=O)cc[nH]c(=NC)c1 N1(C(c2cc(C)nc(C)c2)=O)CCC2(CCCN2C(C2CCOC2(C)C)=O)C1 c1(C(=O)NCCOC2CN(C(C3C(C)(CC)C3)=O)C2)nccn2nccc12 C12(C(N3CCC(C(C)NC(C4CCN(C)C4)=O)CC3)=O)CCC(CC1)CO2 C(C(O)C(F)(F)F)NC(=O)C(=O)NC(c1cccc(Cl)c1)Cc1ccccn1 C1(CC#C)(C(=O)N(CC)Cc2ncc[nH]2)CCN(C(c2nc(C)sc2C)=O)C1 Cc1nc(=NCCC2CCCCN2C(=O)Cc2cccc(C(F)F)c2)[nH]cc1Br c1(C(=O)NC2(C(C)NC(=O)C(N3CCC(C)C3)=O)CC2)ccn2nccc2n1 CN1CCCC(C)(C(=O)NC(CC(=O)NCC2CCCNC2=O)C2CC2)C1 O=S(=O)(c1cccnc1N1CCC2(CCC2)CC1)NCc1ccncc1 C(c1cccnc1)=CC(=O)NCCOCCNC(c1cn(CCC#N)nn1)=O C1(CCC(=O)N(CC(C)O)CCNC(=O)C(C)(C)C2CC2)CCCN(C)C1 C(C#Cc1cn(CC2CC3CC3C2)nn1)NC(Cc1c(OC)nccc1)=O c1(C2CCOCC2)cccc(Cl)c1.Cn1nncc1C(=O)NC(=O)Cn1nccn1 C(=O)(C1COc2cc(C)c(C)cc21)N(C1CCN(C(=O)CC(C)OC)CC1)CC C1(NC(C(C)(C)C2CCN(C(=O)CCn3cccn3)C2)=O)COCC(C)(C)C1 c1(CC(=O)NCC(CNC(=O)C(C)NC(=O)C2CC2)OC)n[nH]c2c1CCCC2 c1(C(C)C)cc(F)c(Cl)cc1Cl.C1C(C(=O)O)NC1=O C1(NC(C(C)OCC(F)(F)F)=O)CCC12CN(C(c1cn(C)[nH]c1=N)=O)C2 O=C(CC(C(F)F)NC(=O)C1CC1)NC(c1cnn[nH]1)N1CCC1 CCCCCC(O)CC(=O)NC(C)CC1CN(C(=O)CC)C1.c1(C(=O)OC)sc(C)cc1Cl C#CCCCC(C)C(=O)N(CC(C)(C)CNC(C1CCc2n[nH]cc2C1)=O)C N1(C(C(C)N(C(c2c(CC)cco2)=O)C2CC2)=O)CCCN(CC2CC2)CC1 c1(CC)onc(C(=O)NC(C)C(C)NC(C2CC(n3ccnn3)C2)=O)c1C N1(C(CSCC)=O)CCC(CNC(c2csnn2)=O)CC1C C1(OC)CC(NC(C2CC=CC2)=O)CN(C(C2(N3CCOCC3)CCC2)=O)C1 N1(C(c2cnc(OC)s2)=O)CCCCC(N(C)C(C2(C)CCN(C)C2)=O)C1 CC(C)CCCC(=O)N1CCC(C(C)CNC(=O)CC(O)CN(C)C)CC1 N1(C(C(=O)Nc2ccc(OC)cc2CNS(C)(=O)=O)=O)CC2CCC1CNC2 N1(C(C(C)C(C)O)=O)CCOCC(CNC(c2scnc2Cl)=O)C1 N1(C(=O)CCC2CCCCCC2)CCC2CN(C(C3(O)CCOCC3)=O)CC12 c1(CNC(C2CC(C)(F)C2)=O)nc(CNC(=O)CS(C)(=O)=O)cc(O)n1 CCC(C)(CNC(=O)CC1CN(C(=O)CC2CSCCO2)CCO1)CO C(CC(=O)N1CCC(C)CC1)(C(C)(C)C)NC(c1nccc(OC)c1)=O c1(OC)cc2[nH]cnc2cc1C(N1CC2CC(C1)N(C1CC1)C2)=O C1(CCC(=O)NCCn2ncc(C)c2)CCCCN1C(=O)CC(C1CC1)C1CC1 c1(C(C)(C)C)ccc(C(N2CCC(NC(C3CC(C)(CO)C3)=O)CC2)=O)c(N)c1 C1(CC(C)O)CCCN1C(C1(CCNC(=O)CN2CCOC2=O)CCCC1)=O Cn1[nH]c(C(=O)NCCC2(NC(=O)Cn3nnc(-c4ccco4)n3)CC2)nc1=O Cc1ccc(C(N2CC(C3CCN(C(C4CC5CC(=O)C4O5)=O)CC3)C2)=O)c(O)n1 c1(C(N(c2nc(C(=O)NC3CC3(F)F)cs2)C)=O)ccc(CCC(=O)N)[nH]1.C(F)(F)F Cc1cccc(C)c1C(=O)NCCC1(C)CCN(C(=O)C2=CCCCO2)C1 N1(C(C(C(CC)O)C)=O)CCC=C(C(=O)NCC2CC(F)(F)C2)C1 CCCCC(O)C(=O)N1CC(CC(C)NC(=O)C(C)C(O)Cc2ccccc2)C1 C1(C(=O)Nc2cn(C)nc2)CCC(NC(=O)CN2CCOC2=O)CC1 c1(C(=O)NCCOCCN(C)C(C2(C)CC2(F)F)=O)cccc2c1COCCN2 c1(C(N2CC(C)(NC(CC3CC(CC)C3)=O)C2)=O)ccc(O)c(Cl)n1 Cc1cc(CC(=O)NCC(C)N(C)C(C2CC3CC3C2)=O)cc(C)c1Br N1(C(CC(CCC)C)=O)CC2CCC(C1)N2c1nc(C2CC3(CCC3)CO2)ns1 c1(OC)ccc(S(=O)(=O)N2CC3CN(Cc4nc5ccccn5c4C)C3C2)cn1 c1(N2CC(N(CCCC)C(c3cncc(C)c3C)=O)C2)ncnc2c1ccn2CC N#Cc1cc(C(=O)NC2CCC2NC(C2CCCCC23CCC3)=O)c(F)cc1F Cc1cc(CC(N2CC(CO)(NC(=O)COc3ccsc3)C2)=O)no1 C12=CC=C(C=C1)C2.c1(NCCNC(C2C(C)C2)=O)ncc(Br)cn1 Cc1onc(C(=O)NC(C)C(C)NC(=O)CCc2ncc(F)cn2)c1[N+](=O)[O-] N1(C(CCC)=O)CC(NC(=O)CC(C)(C)CC)CC2(CC2)C1 c1(C(=O)NCC2C(CNC(CN(CCOC)C)=O)C2)csc(C#N)c1 c1(C(=O)NC(CC)CNC(=O)CC(c2cccs2)NC(C)=O)cc(C)cc(F)c1 CC1=NNC(=O)C1CC(=O)NCC1(F)CCC(NC(c2csnc2C)=O)C1 c1(NC(C)=O)ccc(F)c(C(=O)NC(C)C(C)NC(C23CC(C2)C(C)O3)=O)c1 C1(CN(C(=O)CCC2CCC(NC(c3cncn3C)=O)C2)C)COC(=O)N1 c1(CCC)cc(C(=O)NCCCOCCNC(C2CC2(C)Br)=O)sc1C C(=O)(C1=COCCC1)N(C1CN(C(C2(n3nccn3)CC2)=O)CC1(C)C)C C(C(CC(C)(C)C)NCc1nccn1CCc1ccccc1)OC CCC(C)C(C(=O)NCC1C2CN(C(=O)C3=NOC(C)C3)CC12)N(C)C C(C(=O)N(CC)CC1CCCN(C(=O)C=CCCC(C)C)C1)(C(C)C)OCC C1(C(=O)O)(OC)CCN(C(C2CC(=O)N(CCc3ccccc3)C2)=O)CC1 N#Cc1c(NC2CCN(C(C3CCN3C3CCCC3)=O)CC23CCC3)cccc1F N1(C(=O)OC(C)(C)C)CCC(NC(CCc2cn(C(C)(C)C)nn2)=O)CC1 c1(CNC2CCN(C(c3ccn(C)n3)=O)CC2F)cc(F)c(C#N)c(F)c1 c1(CC(N2CC(NC(C3C(C(C)C)C3)=O)C(C)C2)=O)cccc(Cl)c1F CCC(C)C(O)C(=O)NCC1(C(N2CCCC2C)=O)CCCCC1 C(=O)(C1SCCc2ccccc21)NCCC1CC(NC(c2c(N)nccn2)=O)C1 CC(N=[N+]=[N-])C(=O)N(CC(C)NC(C1(c2cc[nH]n2)CC1)=O)C Cc1nc(C(=O)NCC(C2CC2)NC(=O)CCc2ccc(O)nn2)ccc1C#N c1(C(N2CCC(N(C(c3cccc(C)c3Cl)=O)C)C2)=O)ccc2c(c1)COCC2 c1(C(N2CCCN(C(C(C)C)=O)CC2C(C)C)=O)cc2cc(F)cc(F)c2o1 N1(C(c2ccc(C(C)(F)F)cc2)=O)CC(F)(F)CC1CNC(C1C=CCCC1)=O c1(C(N(CC(C)NC(c2ccccc2)=O)C)=O)cncc2cnccc12 N1(C(c2ncc(C)o2)C(=O)NC2CCC2)CCC(C2CCCC2(C)C)C1 N1(C(C(Cc2ccsc2)NC=O)=O)CCC2(CC1)CN(C(=O)C(C)CO)C2 N1(C(C(C=CC)O)=O)CCN(C(=O)CCCc2nc3ccccc3o2)CC(O)C1 C1(COC)(NC(c2cnc(O)o2)=O)CCCN(C(c2cccc(OC)n2)=O)C1 C1(F)(C(=O)NC2CCC(NC(C(c3cccc(OC)c3)C)=O)C2)CCS(=O)(=O)C1 O=C1C(NCc2cccc(Cl)c2O)CCCN1Cc1ccccc1 C12(NC(c3cscc3C(F)F)=O)CCCC1CN(C(=O)C1=C(Cl)CCC1)C2 Cc1cc(C)c(CC(=O)NC(C)CN(C)C(c2ccn3nccc3n2)=O)c(O)n1 N1(C(C2(SC)CCC2)=O)CCC(C)C(CC(=O)NCc2cc(C)on2)C1 O=C(C1=CCN(C(C2(C3(O)CCC3)CC2)=O)C1)NC1CCOCC1 C1(N(C(c2ccnc(F)c2)C(=O)NCC2CCCOC2)C)(CSC)CCOCC1 C(CCC(C)C)=CC(=O)N1CCN(CCOC)C(=O)CSC1.c1(C(C)=O)nccs1 [N-]=[N+]=NC1CC(C(=O)NC2CC(CNC(c3ccnn3CC(F)(F)F)=O)C2)C1 C(=O)(CCS(N)(=O)=O)NCC(N(C)C(C1CN(S(C)(=O)=O)C1)=O)C1CC1 CCC(C)(C)CCCC(=O)NC(C)C(C)C(=O)NC1CNC(=O)OC1 C1(NC(C#CCNC(C2(C)C(C)OCC2)=O)=O)CC2(C1)CC(C#N)C2 N1(C(C(C)NC(=O)NC)=O)CCCC(COC)(NC(c2c[nH]c(C)c2)=O)C1 C(=O)(C#CC1CCOCC1)NCCOC1CCN(C(C(CC)SC)=O)CC1 c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC(C)C(NC(=O)CCCCOC)C1)=O c1(OC)ccc(-c2nc(C3CCN(C)C3C)n(CCCO)n2)nc1 C1(C(N2C(CN(C(C3CC=C(C)CC3)=O)C)CCC2)=O)CCCCCN1C C1(C(=O)NCC2CCN(C(=O)C(F)n3cccn3)C23CC3)(OC)CCCCCC1 N1(C(CC(CC)(F)F)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)CC2)CC1C c1(OCC)ncc(NC(C2(C)CC(O)CN2C)=O)cc1F C1(NC(CCC(=O)NC)=O)C2CC3CC(C2)CC1(CNC(=O)Cc1cnsc1)C3 C1(C(=O)OC)(CC)CCCCN1C(c1ccc(NC)cc1)=O N1(C(C(CO)NC(N)=O)=O)CC2(C1)CN(C(=O)CC=Cc1ccccc1F)C2 C#CCCCCC(=O)NC1CC(CNC(=O)COc2ccc(C(F)(F)F)nc2)C1 c1(NC)ccc(Cl)c(NC(=O)C(=O)NCCCn2nc(C)cc2C)c1 S(=O)(=O)(c1c(C)nn(C)c1Cl)N1CC(c2nc(C)[nH]n2)OCC1 C=CC(CCC)CC(=O)NC(CCSC)C(=O)NC1CC(=O)N(O)C1 N12CCCCC1CNC(=O)C2.C1(C(N)=O)CC(CSn2ccnn2)C1 N1(C(c2c(C)cc(Br)cc2)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1F c1(NC(C2(CC)CCOC2)=O)ccc(NC(=O)C(C)C(C)(C)C)cc1C S(=O)(=O)(c1cccc2cccnc12)NCCNCC1(F)C(C)OCC1 C(=O)(CC(C(F)(F)F)n1cccn1)N(C1CCCN(C(c2c[nH]c(C#N)c2)=O)C1)C N1(C(C(CC)OC2CCCC2)=O)CCC(C)(C(=O)N(C2CC3(CCC3)C2)C)C1 c1(C(=O)NC2C(NC(c3cnnc(O)c3)=O)COC2)n[nH]c2c1COCC2 c1(C(=O)NCC2(C(C)NC(=O)C(c3ccc(F)cc3)O)CC2)[nH]nc([N+](=O)[O-])c1Cl N(C(=NCc1ccoc1)N1CCN(c2ccc(C)cc2)C(=O)C1)C(C#C)C(C)C N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)Cc2ccccc2[N+](=O)[O-])CC(C)(C)C1 C1(NC(C2CCC(CNC(c3cc(C#N)sc3)=O)CC2)=O)CCc2nn[nH]c2C1 N1(C(C(C=C)CC)=O)C2CC1CN(C(=O)CCC(=O)N(CC)CC)C2 C12(C(N3CC(N(C)C)C4(C3)CC4)=O)CCC(CC1)N(C(c1cnc(S)nc1)=O)C2 C=C1CCN(C(=O)C(C)C(F)(F)F)C(C(N2CC(c3nncs3)C2)=O)C1 O=[N+]([O-])c1cnc2c(F)ccc(Br)c2c1NCc1nc(C2CCCC(F)(F)C2)cs1 c1(C(N2C(Cn3cc(CC=C)nn3)C=CC2)=O)ccc(C(F)F)c(C(C)C)c1 N#Cc1cc(F)c(C(=O)NCCCNC(C2CCc3nncn3CC2)=O)c(F)c1 C(CC(=O)NC1CC(NC(=O)COc2cccc(N)c2)C1)(C(F)(F)F)OC CCS(=O)(=O)NNC(=O)c1c(F)cncc1Br C(CN=c1[nH]c(N2CCN3CCCCC3C2)nc2c1COCC2)N(CCO)CC CC1CN(CCCc2csc(=N)[nH]2)CC(C)N(C(=O)C(N2CCC(O)CC2)=O)C1 C=CCC(C)(CC)C(=O)NC(C1CN(C(c2nnn(C)c2N)=O)C1)C C1(NC(c2ncc(OC(C)C)nc2)=O)CCN(CCCC(F)F)CC1 c1(C(=O)NC(C(C(C)C)NC(=O)C2=CCCCO2)C)ccc2nsnc2c1 C1(CNC(c2n(CC)ncc2)=O)CCN(C(C2CCCN(S(C)(=O)=O)C2)=O)CC1 C(C(O)C(=O)NC(C)(C)C(=O)NCCc1ncn(C)n1)NC C(C(C)(C)CNC(C)=O)N(C)C.C1(N(C(=O)C2CC2)C)CC(n2cnnc2)C1 O=S(=O)(c1ccc(O)nc1)N1Cc2cc(-c3nn[nH]n3)ccc2C1 C1(NC(COCC(c2ccccc2)C)=O)CCCC1(C)CNC(C1CC2(CC2)C1)=O C(=O)(CCCCCC(C)C)NC1C(CNC(C(C(C)(C)C)OC)=O)COC1 CCCCC(C(=O)NCC1(NC(=O)CNC(c2ccco2)=O)CCC1)C(C)C C=CCCC(C)(C)C(=O)N1CCCC(C)(NC(c2cnn(CCF)c2)=O)C1 CN1CC=CCC1CC(=O)NCCC1CN(C(C2(C)CCCOC2)=O)C1 c1(OC)ccc2c(N(CC3=CCSC3)C)nc(=NCC(Cl)(Cl)Cl)[nH]c2c1 N1(C(C2(NC(CC3(C)CCOC3)=O)CC(O)C2)=O)CC2CCC(C1)O2 CC1CC2CN(C(C3(NC(=O)CC(C)C4CC4)CC(CO)C3)=O)CCN2C1 C1(C(=O)Nc2cn(CC)nn2)CC(O)CN1C(c1ccc(SC)cc1)=O c1(CC(=O)OCC(COC)=O)ccc2ncccc2c1 C1(C)(C(=O)NC(CCOC)C(C)C)CC(O)CN1C(c1ccc(F)c(C)c1)=O N1(C(C(C)NC=O)=O)CCC2(CC1)CC(C(=O)Nc1ncc(C#N)cn1)CO2 N1(C(CSc2n(C)cnn2)=O)CCCC(C)(C)C1CNC(C1(C)CCNC1=O)=O CC1=C(C(=O)NC2C3CC4C(C3)C24C(=O)NCCCn2cnnc2)CCCO1 C1(CN(C(C2(C)CC2(C)C)=O)CC)CCCN(C(=O)CC2CN(C)C2)C1 C(=O)(CC(C)(O)COC)NCC(CC)NC(c1sccc1C(C)=O)=O C1(N(C(=O)COc2ccc(F)cc2)C(C2CCCOC2)C)CCCC12CCNCC2 C1(C(N(C)CC2(NC(=O)CSC(F)(F)F)CC2)=O)CCOC1=O CCCCC(C(=O)N1CCC(C(C)CNC(=O)C=Cc2ccoc2)CC1)C(C)C N1(C(c2c(CC)sc(=N)[nH]2)=O)CC2(C1)SCCC2NC(=O)CC1C=CCC1 N1(C(C(n2cc(Cc3cnn(C)c3C#N)nn2)C)=O)CCc2ccc(Br)cc2C1 c1(CC)cccc(CC)c1CC(=O)N(CC(C)N(C)C(c1ccncc1F)=O)C c1(OC(CCN(c2ccc(F)nc2Br)CC)=O)ccc(C)c(F)c1 c1(C(=O)NC(CC=C)CNC(=O)C(C)NS(=O)(=O)CC)ncc(CC)cn1 N1(C(CN(CCOC)C)=O)CCC(NC(c2cccc(CO)n2)=O)C2(CCC2)C1 C1(C(=O)NC(C#C)(C)CC)CC2CC2N1C(=O)C(N1CCCCC1)C N1(C(C2(CC)CCNC2=O)=O)CCC2CN(C(=O)C=CBr)CC2C1 c1(C(N2CCC3(CCC3)C2)=O)coc2c1COC2 N1(C(c2c(SC)nn(C)c2)=O)CCN(C)C(CNC(C2(O)CCSC2)=O)C1 C(C(C)(C)CNC(c1cnc[nH]1)=O)N(C(=O)C(F)(F)c1ccnn1C)C c1(C(=O)NC2(C)CCN(C(c3c(Br)cc(C)s3)=O)C2)cccn2nncc12 c1(CC(=O)NCC(C)CN(C(=O)CC2CCCCC2O)C)ccc2c(c1)CCO2 Cc1ccc(OC(C)C)cc1-c1ccc(NCc2ccc(I)cc2)nc1 N1(C(C2C(C)(CC)C2)=O)CC=C(C(=O)NCCn2cnc(C)c2C)CC1 N1(C(C(C2(O)CN(C(CCC#C)=O)C2)F)=O)C2CCCC1CC2 N1(C(C)=O)CCCN(C(c2c[nH]cc2C2CC2)=O)CC1C C1(N(C)C(c2coc(Br)c2)=O)CCN(C(=O)CCCc2cnn[nH]2)CC1 C1(C)(C(=O)NCC(CCNC(C2(OC(C)C)CCC2)=O)O)CCN(C)C1=O c1(C(=O)OC)ccc(CC(=O)N(C)Cc2ccc(Br)cc2)cc1.C1(C)C(=O)N1 N1(C(C2(CF)CC2)=O)C2CCC1CC(NC(C1(CO)CC(F)(F)C1)=O)C2 Cc1[nH]nc(C(=O)N(CC(=O)NC2C(=O)OCC2CO)C)c1C CC1CCn2ncc(CNCc3c(Cl)nc4ccccn34)c2C1 N1(C(Cc2cnc(C)o2)=O)CCCC(C2CC2NC(C2(C)CCC2)=O)C1 C1(C(=O)NCc2ccccc2)COCCN(C(=O)Nc2ccc(C(F)(F)F)o2)C1 c1(CC)cccc(C(=O)NCCn2cc(COC3CCOC3)nn2)c1F Cc1cnc(F)c(CNC(C2CC23CC(NC(C2CC2C#N)=O)C3)=O)c1 c1(C2C(C(=O)NCC3(SC)CCOC3)CNC2)ccccc1 c1(C(=O)NCCCCCCNC(C2C(C=C)(C(F)(F)F)C2)=O)c(C)nc(C)n1O CC1(C)CCC(CNC(=O)CS(=O)(=O)CCO)N(C(C2CCC(C(N)=O)C2)=O)C1 c1(C(=O)OC)ccc(Cl)c(C)c1NCC1CC(C)C1 C1(C(=O)NCC(F)CO)COCCN(C(c2ccccc2O)=O)C1 C=CCC(CC=C)C(=O)NCC=CCC(=O)NCC1CC1(Cl)Cl c1(C(c2n(CC=C)nnn2)NCc2ccc(OC)cn2)cccc(C(N)=O)c1 C(=O)(C1=CCC(F)(F)CC1)NC1(COC)CN(C(C2(CC)CC(C)(C)C2)=O)C1 c1(C(N2C3CCN(C(=O)Cn4cc(Cl)cn4)C(C3)C2)=O)nncc2c1CCCC2 c1(NC(C)=O)ccc(-c2ccc(-n3nc(C)cc3C)s2)c(C)n1 C1(NC(C)=O)CC(O)CN(C(=O)CNC(c2nnc(S)n2C)=O)C1 CCC(C)(C)C(=O)C(=O)NOCC(=O)NCc1ccccc1F C(C(=O)NCC1CCCN1C(=O)C(O)CN1CCOCC1)(C(C)C)SC n1(CC(N2CCC(CN(C(CC3CC(C)C3)=O)C)C2)=O)cc([N+](=O)[O-])ccc1=O N1(C(C2(C#N)CCSCC2)=O)CC(NC(C2CC(C(F)(F)F)C2)=O)CC2(CC2)C1 C(=O)(CCP(C)(C)=O)NC1(C)CCN(C(C2COCCC2(F)F)=O)C1 Cc1cc2c(cc(C(=O)NC3C(O)CC3O)n2CC(F)(F)F)s1 Cc1cc(C)c(C(=O)NCC(F)CNC(c2[nH]c(=N)ccc2C)=O)c(C)n1 C1(CC)CN(C(c2cn(CCNC(=O)CSC3CC3)cn2)=O)C(C)CO1 CC(C(=O)NCC1CC(F)CN1C(c1cc(Cl)cnc1O)=O)C(F)(F)F Cc1nc2ccc(NC(=O)C3=CCCN(C(=O)C(C)O)C3)cc2o1 C1(C(N2CCCC2CNC(C2CCOC2)=O)=O)CCCC2CCCCC12 c1(C(N(C2CC(NC(c3ccc(CC)[nH]3)=O)C2)C)=O)ccc(OC(F)F)cc1F C1(CNC(c2scc(OC)c2)=O)CC2CCCCC2N1C(c1cc(CO)[nH]n1)=O O=C(C1=CCCOCC1)NCCNC(C1CCCC(O)C1)=O C(=O)(C(F)C(F)(F)F)N(C1CCN(C(=O)CNS(C)(=O)=O)CC1)C c1(OC)ccc(-c2n[nH]cc2C(=O)NCC2CCCCC2c2ccncc2)cc1 c1(C(=O)NC2CN(C(C3(CC)CCCC3O)=O)C2)cc(F)cc2nn[nH]c12 c1(CCNc2nccc(=NCc3cc(SC)ncc3)[nH]2)nn(C)c2ccccc12 C1(CC)CN(C(c2ncccc2F)=O)CCC1NC(=O)C(C1CCOCC1)F c1(C(=O)NC2CC(C)N(C(c3cc(Cl)ccc3N)=O)C2)nc2ncccn2n1 C1(C)(Cn2cc(C(C=C)(C)O)nn2)CCN(C(C2(CC)CCCOC2)=O)CC1 Cc1cc(C(N2CCCC(c3nc(C)cs3)C2)C(=O)NCCC#N)cc(F)c1 CC1CN(CCCCNC(=O)C(=O)NCc2ccc(F)cc2F)CC(C)O1 C1(NC(c2ccccc2O)=O)CC(O)CN(C(=O)C=C2CCCC2)C1 c1(N2CCN(C(=O)NC(C3CC(C)CC(=O)N3)C)CC2)ncc(Br)c(C(F)(F)F)n1 c1(C(=O)NCC2CCC(NC(C(CC)NC(N)=O)=O)C2)cncc(OC(C)C)c1 C=CC(C)(O)C(=O)NC1CC(NC(=O)C=CC=CC=CC=CCC)C1 C(CC(C)(C)CC(=O)N1CCC2C(NC(=O)CNC(=O)CC3CCCC3)C12)OC CCCC(CNC(C12CCC(c3nn[nH]n3)(CC1)C2)=O)CCO C1(NC(C23CCC(N(C)C)C2C3)=O)C2CCC(C2)N1C(=O)CO.C12CN(C1)C2=O C(=O)(CCCCCCNC(c1cc(C)[nH]n1)=O)N1C(CSC)CCC1 C1(C(=O)NCC2CCCC2NC(c2cc(-c3ccco3)c[nH]2)=O)(CC)CC1(F)F CC1CN(C(C)Cc2ccccc2)CC1NC(=O)NCC1CC1(F)F Cc1ccc(F)c(C(N2CSCC2C(=O)NCCCOC(C)C)=O)c1 S(=O)(=O)(c1c(Br)cccc1[N+](=O)[O-])NCCC1C(C(=O)OC)C1 c1(C(N2CC(C3(NC(C4(C(N)=O)CC4)=O)CC3)C2)=O)ccc2c(c1)C(=O)CCC2 C(=O)(C(C)(F)C(C)(C)F)N1CC(O)(C(C)NC(c2cnn(CCC)c2C)=O)C1 N1(C(C2OCCC(C)C2)=O)CCCC(C2CN(C(C3(F)CCN(C)CC3)=O)C2)C1 N1(C(C(CC)n2ccnc2)=O)CCC(CN(C(=O)CC2(N(C)C)COC2)C)CC1 N1(C(c2occ(C)c2)=O)CC2(CCC2)CCC1CNC(=O)Cc1ccc(Cl)cn1 C#Cc1ccc(C(=O)NCC(C(C)(C)C)NC(=O)C=CS(C)=O)cn1 N1(C(c2ccc(OC)nc2)=O)CC2(CC2)CC1CNC(C1CCOCC1CO)=O C(=O)(C(CC(F)F)NC(C1CCCC(C#N)C1)=O)NCCN1CC(C)(O)C1 N1(C(C2CCN(C(c3cc(CC)oc3C)=O)CC2C)=O)CCCC2(CC1)CC2 N1(C(CCCn2c(C)ncc2)=O)CC2(CC(NC(C3CC3(C)C(F)F)=O)C2)C1 c1(C(=O)NC2CC(CNC(C=C(C)Cl)=O)C2(C)C)ccc2ccncc2c1 N1(C(=O)NC(CC(=O)NC2CC2)CSCC2CC2)CCOCC12CCS(=O)(=O)C2 C1(C(N2CCC(CCNC(C3N(S(C)(=O)=O)CCC3)=O)C2)=O)CSCC(=O)N1 N1(C(C2CCCCC(N)C2)=O)CCC2(CC1)CC2N c1(C(N2CC3(CN(C(CC(C=C)C)=O)C3)OCC2)=O)cc(Cl)c(N)c([N+](=O)[O-])c1 c1(CC)cccc(F)c1C(=O)NCC1CCCN1C(=O)CC(C)C(=O)OC N1(C(C(C)SC)=O)CC2CCC(C1)N2C(C1COCCO1)=O C=CCCC(C(=O)N1CCCC(C)(O)C1)NC(c1c[nH]nc1C)=O Cn1nc(C(=O)NCCCC2CCCN2C(=O)C=CCF)c2c1CCOC2 c1(SCC(=O)NC(c2ccccc2)CC#C)ncccc1C c1(N2CCN(N(C(C)=O)C)CC2)nc(Cn2nc(C)n(C)c2=O)c2c(n1)CSC2 c1(C(N2CCC(N(C(C3C(OCC)C3)=O)CCO)C2)=O)cc(CO)ccn1 Cc1ccc(C(N2CCCC(C)(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)c(C)n1 c1(C(N2CC(C)CC(NC(C3C(OCC)C3)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] CC1CN(C(=O)Cn2ccccc2=O)CC1CNC(c1cnccc1Cl)=O N#CC(C(=O)NCCC1CCCN1C(c1cnc(Cl)s1)=O)C1CC1 n1(CC(C)C)ncc(C(=O)NCCC2CC(NC(c3cnsc3)=O)C2)c1C1CC1 n1(CC(=O)NC(CCN(C(=O)CCc2ncc[nH]2)CCCN(C)C)CCl)cnnc1O CCCC(CC)CCC(=O)NCC(O)CC(=O)N1CCC(C#N)C1 C1(CCCNC(=O)Cn2nnc(=O)[nH]2)CCCCN1C(=O)Cn1cnnc1 CCCCCCC(O)CCC(=O)N1CCCC1C1(NC(=O)C(CC)CCOC)CC1 c1(CC)nc(C(=O)N(C)CC2CCN(C(c3cnc(O)n3CC)=O)CC2)c(C)o1 c1(OC)ccc(C)cc1C(N1CCC(C)(C)C1CNC(=O)CC12CCCC1C2)=O C1(CN(C(C2C3CCC(=O)C23)=O)CC)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 c1(C(=O)NCC(C(=O)NC2CCOC(C3CC3)C2)OC)cccc[n+]1[O-] N1(C(c2[nH]c(=N)sc2)=O)CCN(C(=O)CC2CCCC2(F)F)CC1C1CC1 C=CC1(C(=O)NCc2coc(CC)n2)CCN(C(C2CC2(F)Cl)=O)C1 C(=O)(CC(O)CN(C)C)NC(c1cccnc1)C(=O)NCCN(OC)C c1(C(=O)NC2CC(CNC(C(C)OCCOCCOC)=O)C2)cc(C(C)C)no1 C#CCCC(O)C(=O)N1CC(OC)CC1CCNC(=O)CC1COC(=O)C1 C1(C(N2CCC(CCNC(Cc3nc(C)sc3C)=O)C2)=O)CCC2CCC1O2 C(=O)(C(CC(C)(C)C)NCC(CSC)OC)NCc1ccc(OC)cc1 C(CN=c1[nH]c(=NCC2CCC2)c2cc(Cl)ccc2[nH]1)OCCOC N#CC1(C(=O)NCCCCCC(=O)N2CCN(C3CC3)CC2)CCCOC1 C1(O)(C(=O)NC(C2CCCO2)(C)C)CC(F)(F)C1 c1(CC)cccc(C(N2CCCC(C(C)NC(C3(CCOC)CC3)=O)C2)=O)c1F C#CCCCCN(C(C1CCOCC1)C(=O)Nc1ccccc1)C N1(C(C2CCC(=C)CC2)=O)CC2CCN(C(=O)CC3CC3C3CC3)CC(C2)C1 N1(C(CC2CC(SC)C2)=O)CCCC(NC(c2cc(O)ccc2F)=O)C1C c1(N2CCC(C3CCN(C(C(C(C)(F)F)Cl)=O)C3)C2=O)ccc2ccccc2c1 C(=O)(C(C)(C)COC(C)(C)C)N(CCN(C(=O)CCC1CCN(C)C1)C)C C12(NC(c3ccc(O)nc3Cl)=O)CCCC1N(C(=O)C(O)(C1CC1)C1CC1)CC2 C1(C(N(CC)Cc2ccsc2)=O)CCCN(C(=O)CCc2ccoc2)C1 C1(NC(C2C(COC)C2)=O)C=C(C)CCC1 c1(C(=O)OC)ccc(C#N)cc1C.N12CC3C(C1)N3C(=O)c1csc(c1)C2 N1(C(C2(CC)CC2(F)F)=O)CCC2(CCCC2NC(=O)CC2CC=CC2)CC1 C1(C(CO)NC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)Cc2ccccc2)CC1 C1(CC(=O)NC2CC2)CCCN(C(C2CCCCCCC2)=O)CC1 c1(SCC2C(C(=O)NCCNC(C3CCS3(=O)=O)=O)C2)nc2ccccc2s1 C#CCC(O)C(=O)NCC1CCN1C(c1ccc(C(F)(F)F)[nH]1)=O C1(Cl)(C(=O)NCC(C)N(C(CC2(NC(C)=O)CC2)=O)C)CC1C(C)=O c1(C(N(C2CCN(C(=O)CC3COCCO3)C2)CC)=O)ccc(C)c(F)n1 c1(C(N2CC3C(CNC4CCC4)C3C2)=O)ccccc1Br.C12(C=O)CC(F)(C1)C2 c1(CC)ccccc1C(=O)NC(C1CCCN1C(=O)CCC(=O)OC)C c1(C(C)=O)cnc(C2CN(C(C3CCCC3c3cnn(C)c3)=O)C2)cn1 c1(NC(C(C)N(C(C2CCCC(OC)C2)=O)C)=O)cc(C)ccc1F c1(OC)ccc(CC(N2CC(OC)C(NC(C3(N=[N+]=[N-])CC3)=O)C2)=O)c(Cl)c1 C(=O)(CC(C)CNC(c1c[nH]nc1CNC(=O)CC1C(=O)NN=C1C)=O)NC CC(C)(C)C(C)(C)C(=O)NCCN1CCN(C(=O)C#CC2CCCC2)CC1 C12(NC(=O)CC3CCC4CC34)CCCC1N(C(c1cnc3n1CCC3)=O)CCC2 CC1OCCC1NC(=O)CONC(=O)CN1CC2CC2C1 c1(CN2C(C(=O)Nc3ccnn3CCO)CCCC2)c(O)ccc(F)c1Br N1(C(CC=C=C)=O)CC2CC2(NC(c2cnc(S)nc2)=O)C1 Cc1cccc(C(N2CCC(N(C)C(C3(C)CCN(C)C3=O)=O)CC2)=O)c1C C1(C(N(CCCNC(=O)CC(=O)N(C)C)CC)=O)CCCC(C(=O)OC)C1 C=CCC(C)(C)C(=O)N1CCC(NC(=O)Cn2ncn(C)c2=O)C(C(N)=O)C1 c1(OC)c(C(N2CCC(Cc3ccccc3)CC2C2CC2)=O)cc(Cl)cc1Cl C(=O)(C(F)(F)Cc1ccc(F)cc1)NC1CC(CNC(C=CC=CCC)=O)C1 n1(CC)ccnc1C=CC(=O)NC1CN(C(=O)CCC2CC2(F)F)CC1F Cc1nc(C(C)C2CC2)sc1C(=O)NCCCNC(=O)CCNC(N)=O CC#CCC(C(=O)NCC=CC)NC(C1CC=CCO1)=O C1(NC(C(COC)OC)=O)CC2CCC(C1)N2C(C1CCCC1(C)C)=O C1(C(=O)N(CC(=O)NC2CC(C(N)=O)C2)C)(COC)CCC1 C1(C(N2CC(CC(N)=O)C2)=O)CCN(C(=O)C2CCC3(CCC3)O2)O1 c1(CC(=O)NC2CC3CC(NC(C(CC)SC)=O)C2C3)c(C)cc(OC)cc1C C=CC1CCCN1C(=O)NC1CC1c1ccccc1OC(F)F C1(C(=O)NCCN(C2CCCCC2)C(=O)C(C2CCCCC2)O)CC2CCC2C1 c1(OC)cc(-c2nc(-c3cncnc3)nn2CC2CCSC2)n(C)n1 O=C(C#CC1CCCOC1)NCC1CCCCN1C(=O)CCc1ccc(Cl)cc1 c1(C(=O)NC(C(C)NC(=O)C(C)(C)CN2CCOCC2)C)cnn2c1N(C)CC2 c1(CN2CCC(N(C(CCCC(C)=O)=O)C)C2)ccccc1S(C)(=O)=O O=C(C1=CCCCO1)NCC1(O)CCN(C(=O)CCC=Cc2ccccc2)C1 CCC(C)(C)C(=O)N1CC(CNC(c2cncnc2-c2ccccc2)=O)C(O)C1 CC(C)C(C(=O)N1CCCC(CN(C(=O)C(F)(F)C2CC2)C)C1)c1cccnc1 c1(CC)ccc(O)c(NC(=O)CC(CC)NC(c2cc(C(N)=O)[nH]n2)=O)c1 C1(CC(=O)NCC(=O)N(C2CN(C)C2)C)CCCN1C(C1CC1F)=O CCC(O)C(F)(F)C(=O)NCC1CN(C(=O)CC2CCC3CC23)C1 C1(C(=O)NC2CCC(NC(c3ocnc3C(F)(F)F)=O)CC2)CC2COCC2C1 CCCC(C)(C)C(=O)N1CCCC(NC(=O)C(O)CC2CC2)CC1 c1(-c2nc(C)on2)cccc(NC(C2(F)CCN(C(C3(F)CC3)=O)C2)=O)c1 C(CCCCCCn1cc(CCCCCO)nn1)NC(C1CC(=O)N1)=O C(=O)(C#CC1CC(F)(F)C1)N1C(C(C)NC(c2ccc(N)cc2Cl)=O)CCCC1 n1(CC(N2CC(N(C(=O)C3=CCOCC3)C)C(F)C2)=O)ncn2nccc2c1=O C(c1cccc(F)c1Cl)=CC(=O)N(CC(C)(C)NC(C1C(OC)CCC1)=O)C CC1(NC(C23CC(F)(C2)C3)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 n1(CC)nc(C(=O)NCC(CNC(=O)C(F)n2ccnc2)CO)cc1C C(=O)(C1CCc2c[nH]nc21)N(C(N1C(Cc2ccc(OC)cc2)CCC1)=O)CC C1(C(=O)NC2(CO)CC(C)C2)CC(NC(=O)CS(C)(=O)=O)C12CCC2 c1(C(N(C2CCN(C(=O)CCCc3ccc(F)cc3)CC2)C)=O)ccccc1Cl c1(C(=O)NCC(C)(C)CNC(=O)CCc2cncnc2)cc(Cl)c([N+](=O)[O-])[nH]1 c1(CC(=O)NC2(CN(C)C(C3CN4CCN3CC4)=O)CC2)c(F)cccc1C#N n1(CCC)cc(Cl)c(C(=O)NC2CCN(C(=O)CC3OCCC3C)C2)n1 Cc1cc(=O)n(C)nc1C(=O)NCCNC(c1cccc(Br)c1F)=O c1(N(C)Cc2ccsc2Br)nc(NCCC2CCOC(C)C2)c2cnn(C)c2n1 C(=O)(CCC(C)(C)C(=O)c1cccc(OC(c2ccc(Cl)c(F)c2)C)c1)OC C1(NC(C(CC)OCC)=O)CC2CC(NC(c3cccnn3)=O)CC12 C=C1CCN(C(c2cnn(CCNC(c3ncoc3C)=O)c2)=O)C1 C(=O)(N1OC2CCC1C2)C1(NC(Cc2c(C)ccnc2)=O)CCC1 Cc1ncc(C(N2CC(CNC(=O)CCOCC3CCC3)CC2C)=O)cc1Cl c1(C(N2CC(OCCNC(c3cc(C(C)C)[nH]n3)=O)C2)=O)ncccc1C1CC1 N1(C(c2c(C)cc(CC)o2)=O)CCCC(C)(C(=O)NCC2(C(C)(C)OC)CC2)C1 c1(C(=O)N(CC(O)C(F)(F)F)CCO)nc2ccccn2c1-c1cnc2[nH]cnc2c1 c1(CC(C)C)cc(C(N2CCCC2CN(C(C)C)C)=O)cc(O)n1.C1CC1 c1(N2CCCC(C(CC)NC(C3CCCC3OC)=O)C2)nccc(S(C)(=O)=O)n1 C1(C)(C(=O)NCC=CCSC)CCN(C(C2CN(C)CCO2)=O)CC1 c1(N(C)C=O)ccc2n[nH]c(C(C)C)c2c1.c1(SC)cccc(-n2cc(CN)nn2)c1 c1(C(C(=O)N(CCC)CC=CCC(C)C)OC)ccccc1.C(=O)(COCCOC)N C1(NC(CCOCC#C)=O)CCCN(C(c2ccc(OC)c(Br)c2)=O)CC1 C1(C(N2CCC(C)C2CNC(c2cccc(CCO)c2)=O)=O)CC2(C1)OCCO2 c1(C(=O)OCC)nc(=NCC2CC(NC(C3(C(F)F)CCC3)=O)C2)[nH]cc1Cl C1(CNC(C(C)(C)OCC)=O)C(C)CCN1C(=O)CCC1OCCO1 C(=O)(C(CNC(C1OCCC1(C)C)=O)C(C)(C)C)N1C(C)(CC(=O)NC)CC1 C1(CNC(c2ccc(C=C)cc2)=O)CN(C(=O)C(COC)N(C)C)C2(CCC2)C1 CC1CC(NC(C2CC(O)C2)=O)CCN1C(c1cccc(C(F)F)c1Cl)=O c1(OCC)ncc(C(c2nnnn2C2CCOCC2)NCCc2ccc(C)s2)s1 C(=O)(CCCCC(C)C)NC(CC=C)CC(=O)NC(c1cnco1)C C1(C(N2C(C)(CNC(c3ccc(C#N)o3)=O)CCC2)=O)Cc2cccnc2C1 C=CCCC(=O)NC(C1CC=CCC1)C(=O)NC(c1nc[nH]n1)C1CC1 C1(C(C(=O)NCCCCC2CN(C(C3CC(F)(CO)C3)=O)C2)F)CCCCCC1 N1(C(C(C(C)C)F)=O)CCC(C2CCCN(C(c3ccc(F)o3)=O)C2)CC1 c1(C(=O)OC)ccc(NC(=O)CCc2cc(C)ccc2C)cc1OC(C)C c1(CC(=O)NCC2C(NC(C(C)c3ccco3)=O)CC2)sc(O)nc1O C1(CC=C)(NC(C2COCCC2(F)F)=O)CCCN(C(=O)CC(C)(C)CC)C1 N#Cc1ccccc1C(=O)NCC(CC(=O)N1CCCC1C(N)=O)C1CCC1 CCC(C)CCCCC(=O)NCC1(NC(=O)CCOC(C)C)CC1 C1(O)(CNC(C(F)=CC)=O)CC(NC(=O)C(O)c2ccco2)C1 c1(C(N2CCC(C(C)(C)C)(CNC(C(CSC)C)=O)C2)=O)cc(C)c(CO)cn1 c1(C(C(N2CC(N(C(c3c(C)n[nH]c3)=O)C)C2)=O)C)cc(Br)ccc1F C1(C)(N(C)CC)CN(C(=O)C(C)(C)C2CCN(C(=O)CCN(C)CCO)C2)C1 C1(C(=O)NCc2c(C(N3CCC(SC)C3)=O)scc2)CCCC(=O)C1 c1(OCCC(=O)N(C(C)CNC(C2CC3CC2C3)=O)C)ccc(S(C)(=O)=O)cc1 C(=O)(C(C)C(C)COC)N(CCCNC(CCC)=O)C(C)C.c12ccc(cc1)s2 N1(C(C2(OC)CCCC2)=O)CCC(NC(=O)Cn2cncn2)CC(C)(C)C1 C1(C(=O)NC2CC(C)(NC(c3cnc(OCC)s3)=O)C2)CCCCC1(F)F c1(C(N2CC3C(NC(c4c(Cl)ccc(NC)c4)=O)(C3)C2)=O)cc2ccccc2[nH]1 n1(CC)cc2ccc(C(=O)NC(C)C(C(C)C)NC(c3c[nH]cc3C)=O)cc2n1 c1(Nc2cccc(SC)c2)ncnc(NC(C)C(C)Oc2ccccc2F)c1C c1(CC)nc(C)c(C(=O)NCC2(F)CCC(CNC(c3n[nH]cc3CC)=O)C2)s1 C(CCCC(=O)NCC1C=CCN1C(=O)CC1CC1c1ccccc1)OCC C(=O)(C1=C(Cl)CCCC1)NCc1ccc(C(=O)NC2CCN(C(=O)C3CC3)CC2)s1 Cc1ccccc1SCC(=O)NCC1CC2CC2N1C(=O)Cc1sc(O)nc1O c1(COCC)nc(C)c(C(N2CCC(CNC(c3csc(CC)n3)=O)CC2)=O)s1 CCCC(CCCNC(c1sccc1C(C)C)=O)NC(=O)C(C)C(F)F N1(C(CCCSC)=O)CCC(C(C)NC(=O)CC2CCC=CCC2)CC1 c1(C(=O)NCC(C(C)(C)C)NC(C2C(C(C)C)CCC2)=O)cccc2c1OCO2 Cc1nnc2n1CCCC2C(=O)NC1CCN(C(=O)CCCC#N)CC1 N1(C(c2ccoc2Cl)=O)CCC2CCCN(C(=O)COCC(F)(F)F)C2C1 N1(C(=O)CC2CC2)CC2C3CCC(C2C1)N(C(=O)CC(=O)NC1CCOC1)C3 c1(CC)ccc(NC(=O)C(F)CC2CN(C(=O)CCC3CC3C)C2)cc1O C=CC1(C(=O)NCC[Si](C)(C)C)CCN(C(c2ccn(CCC)n2)=O)C1 N1(C(CCC=C)=O)CC(NC(=O)C(C)(O)C(C)c2ccccc2)CC2(CC2)C1 c1(CCCC(=O)N(C(CNC(CC(CC)C)=O)C2CC2)C)nc2ccccc2o1 C1(C(=O)NCc2ncnn2C(C)C)(COC)CN(C(c2cccn2C)=O)C1 C#Cc1ccc(OC)c(C(N2CCC(NC(=O)C(C)(C)C3CCCO3)C2C)=O)c1 C(C(C)C)(C(O)C(=O)NC1CC2(C(=O)N(C)Cc3ccn(C)n3)COC1C2)OC C1(C(=O)NCC2(O)CCN(C(Cc3cc(C)no3)=O)CC2)Cc2cccnc2C1 CC(C)C1C(=O)N1.c1(NC(=O)OC(C)(C)C)cn(CC(F)F)cn1 C(=O)CCC(C)(C)F.N1(C(C(CC2CCC2)N(C)C)=O)CCCCC1C1(O)CC1 c1(NC(C2N(C(CCC3C(C)(C)C3)=O)CCCC2)=O)cccc(C#N)c1 N(C1CCCn2nncc21)CC(C)NC(C1CCN(C(=O)N(C)C)CC1)=O C12(NC(C3CC34CCOCC4)=O)CCCC1(F)CN(C(=O)C(F)(F)C(F)F)C2 c1(C(=O)OC(C)(C)C)cncc(C(=O)OC(CC)C(=O)N(CC(C)C)C)c1 Cn1cnc(CNC2(CNC(C)(C)CC3CCC3)CC2)cc1=O C1(c2ccccc2)(NC(C=CC=CCC)=O)CC(NC(=O)Cc2ccoc2)C1 C1(NC(c2c(CC)scn2)=O)CS(=O)(=O)CC1NC(=O)CCCn1cc(C)cn1 C1(N(c2nc(C)c(CN)s2)C(C)=O)CC(=O)N(C(c2ccccc2)C)C1 C1(C(N2CC(C(C(=O)NC(C)(C)C(F)F)OC)C2)=O)CC(N=[N+]=[N-])C1 N1(C(CC2N(C(CC3CCC(C)CO3)=O)CC2)=O)CC2CN(C)CC2(C)C1 C(=O)(C1CCc2ccccc21)NCC(CNC(=O)COC1CCCOC1)OCC Cc1cc(C(N2CC3CC3(CNC(C34CC(C3)C4)=O)C2)=O)cc(C)c1Cl c1(C(N(CCC(=O)N(CC(C)C)C)C)=O)ccc2occc2c1 C(=O)(C1CCCc2nncn21)N1CCCC(NC(C=Cc2c(C)coc2C)=O)C1 c1(C(=O)NCC2N(C(COc3c(F)ccc(C)c3)=O)CC2)cnc2[nH]nnc2c1 C1(C(N2CC(C(N)=O)C2)=O)COCCN1C(=O)CCc1cncnc1 c1(C(N2C(CC)CN(C(=O)CN(C)C)CC2)=O)cc(Br)cc(F)c1O C(=O)(CCCC(C)(C)C)N1C(CN(C(c2nc(O)nc(O)c2F)=O)CC)CCC1 c1(C(N2CCC(N(C)CCc3c(F)cccc3F)C2)=O)ccc2cc[nH]c2c1 C1(NCCc2ncn(CC)c2)CCNC2CC12 c1(N2CCC(C(F)(F)F)(OC)C2)nc(C)cc(=NCC2(S(C)=O)CCC2)[nH]1 C1(NC(c2c(C)cc(F)cc2)=O)C2COCC1CN(C(c1ccc(C#N)[nH]1)=O)C2 CC1(C)CCN(C(=O)C(N)=O)C(C(=O)NC2(C)CCC(=O)NC2=O)C1 c1(C(C)C)nc(NCC(C)C(F)F)cc(=NCc2cncc(C(F)(F)F)c2)[nH]1 c1(N2CCC(C)C(NC(=O)CCC(N)=O)C2)nccc(S(C)(=O)=O)n1 N1(C(C2CC(OCC)C2)=O)CCC(CN(C(=O)C=CC2CCCN2C)C)CC1 N1(C(CC(c2ccco2)C)=O)CC(C(=O)OCC2CC3C(C2)C3(C)C)CC(O)C1 c1(CC(=O)NC2CC(F)(CNC(=O)CCC3CCCO3)C2)ccc(O)cc1 c1(CC)ccc(C(N2CCOCC2CC(=O)NCC2COCCN2C)=O)cc1N CCC(F)(F)C(C)(C)C(=O)NC1CCCC1CNC(C1(C2CC2)CC=CC1)=O C1(CNC(c2cc(C)cc(Cl)n2)=O)CC2COCC2N1C(C1CCCS1(=O)=O)=O C(CC1CCC1)(CC(=O)N=c1ccn(C2CC2)[nH]1)NC(C1C(C)CCOC1)=O C=C(C)C(C)(O)C(=O)NCC(O)CNC(c1cc(OC)ccc1Br)=O c1(C(=O)NCC=CC(=O)NCC(C)Cn2cccn2)csc2cc(Cl)cnc12 c1(CN(CC(=O)OCC)C(=O)NCC2CC2)ccc(Br)o1 N1(C(c2c(C)snc2)=O)CCC(C)N(C(c2cc3ccncc3o2)=O)CC1 N1(C(c2c(OCC)cccc2)=O)CCN(C(c2[nH]cnc2CC)=O)CC2(CC2)C1 Cc1nn(C(C(CO)NC(=O)COCC(C)C)C)c(C)c1C c1(CC)cc(C(F)(F)F)ccc1C(=O)NC1CCCN(C(=O)C(C)(C)N(C)C)C1 CC(C)(CC(=O)NCC1CCCN(C(c2occc2Cl)=O)CC1)CC(F)F c1(N2CC(C)(NC(CCNC(=O)NC)=O)C2)c(C(N)=O)cccc1[N+](=O)[O-] c1(C(N(C)CC2CCN(C(C(C(C)(C)C)OC)=O)C2)=O)cnc2ccncc2c1 Cc1c(C(N2CC(O)C(F)C2)C(=O)NCC2CCOC2)ccnc1F C(=O)(CC1=CCCCC1)N1CCCC(NC(C2CC(=O)N(c3nccs3)C2)=O)C1 C12(C(N3CC4C(CNC(c5c(C)ncs5)=O)C4C3)=O)CC3CC(C(=O)N1)C2C3 C(=O)(CC1COc2cc(O)ccc21)N1CC(O)(CNC(c2c(CC)[nH]cc2)=O)C1 C#CCC(C)(C)C(=O)NCC(C)(CC)NC(c1cc(C(N)=O)no1)=O Cc1nc2ccc(C(N3C4CC3CN(Cc3cccc5[nH]ncc35)C4)=O)cc2[nH]1 c1(OC)cnc(C(N2CCC3C(NC(c4ncccc4OC)=O)CC23)=O)c(F)c1 Cc1ncc(Cl)cc1C(N1CC2CC(NC(=O)Cc3cc(O)nnc3O)C1C2)=O c1(C(N2CC(CC)N(C(=O)CC(C)F)CC2)=O)ccc(C#N)c(O)c1 C(N=c1cc(C(N)=O)nc[nH]1)c1occ(C(N)=O)c1 C1(CNC(CC)=O)CN(C(=O)CCCC2CCCC2)CCC1CO c1(C(N2CCC(O)(CC(=O)OC)C2)C(=O)NCC)nn(CC(F)(F)F)cc1C C(=O)(C(O)CN1CCCC1)NC1(C)CSC1.N12CC(C1)C2=O C(c1c(Cl)nc2sccn12)=CC(N1CC(NC(c2cc[nH]n2)=O)C(CO)CC1)=O N12CC3=C(C1)CN(C3)C(=O)C1(CCOCC1)N(S(C)(=O)=O)CCC2=O.C1(CO)CC1 Cc1cnc(F)cc1C(=O)NC1CCC(NC(=O)C(C(C)C)OCC(C)C)CC1 C(=O)(CCCCC(F)F)N1CCCC(NC(C=Cc2nnn(C)n2)=O)C1 C1(C)(C(=O)NC(CC(C)NC(c2c(C)ncs2)=O)C)CCc2ccccc2N1 C1(NC(C(CC)c2ccccc2)=O)CCN(c2ncc(C3CC3)cn2)CC1 C1(NC(C23CC(NC(=O)CC4CCSC4)(C2)C3)=O)CCc2nn[nH]c2C1 C1(CNC(C(N2C(CC(=O)N(C)C)CCCC2)=O)=O)CC2CCCC(C1)C2 C1(C(=O)NC(CNC(c2cc(C(=O)OC)ncc2)=O)C2CC2)CC2CCC(C1)C2 c1(OC)ncc(C(=O)NC2COCC2CNC(=O)Cn2ncn(C)c2=O)c(C)n1 CCC(CC(F)F)C(=O)NCC1CCN(C(c2cc(C(N)=O)cc(C)c2)=O)CC1 C1(NC(c2oc(C3CC3)nc2C(F)F)=O)CN(C(C2CCCN2C2CC2)=O)CC1O c1(C(C(=O)N)OC)ccc(SCC)cc1.c12ccoc1CC1(CC1)C(=O)N2 c1(OC)ccc(CC(N2CCCC2(C)C(=O)Nc2c(Br)ccnc2Cl)=O)c(Br)c1 C1(C(NOC(CC)CC)=O)CCOCC1NC(c1oc(CO)cc1C)=O C1(C)(C(=O)Nc2cn(C(C)(C)C)nc2)CCN(C(c2ccncc2)=O)C1 c1(OC)ccc2cc(C(=O)NCC3CC3CNC(c3ccc(C)cn3)=O)sc2c1 C12(C(N3CCC(N(C(Cc4cc(CC)no4)=O)C)CC3)=O)CCCC(C1)OC2 C1(C(N(C(CCNC(C(C2CC2)OCC)=O)C)C)=O)CCCC2(CCC2)O1 C1(C)(OC)CN(CC(=O)NCCOC2CN(C(=O)C(=Cc3cn[nH]c3)C)C2)C1 C(CC(C)C(=O)N(CCC)CCNC(C1CC(=O)N(C2CCCC2)C1)=O)=CCC c1(SCCC)nc(Cl)c(CNC(=O)CC2COCCN2)c(Cl)n1 N1(CCC(N2C(CN(C(=O)C=Cc3ccco3)CC)CCC2)=O)CCC(C)CC1 C1(C(=O)NCCCN(C(C(Br)=C(C)C)=O)C2CC2)CCN(C2CC2)C1=O C12(NC(C(C)N(C)CC3CC3)=O)CC1CN(C(c1sccc1-n1ccnn1)=O)C2 C12(CNC(C(=O)NC(C)C(C)(C)CO)=O)CCC(CC1)C(C)O2 CC1CCN(C(=O)CNC(=O)C=CCN(C)C(C2(CCF)CCC2)=O)C1 C(N=c1[nH]c2c(c(=NCC3CC34CCOCC4)[nH]1)CCC2)c1cc(C(C)C)n[nH]1 C(=O)(C(C)(C)COCC(F)F)NC(C)C(C)NC(c1ccncc1F)=O N1(C(C(c2ccc(C)cc2)C)=O)CCC(C2CN(C(C3(C(C)C)CCC3)=O)C2)C1 N1(C(CC(CC)C2CCC2)=O)CCN(C(c2ccc(C)nc2C)=O)C(CO)C1 c1(C(N(C2CN(C(c3ccc[n+]([O-])c3)=O)C2)C)=O)ccc2c(C#N)c[nH]c2c1 C1(C(=O)NC2CCN(C(C3CN(C(C)=O)C3)=O)C(C)C2)CCc2c(cnn2C)C1 N1(C(C2OCCC(NC(c3c(Cl)cn(C)n3)=O)C2)=O)CC2CCC(O)CC2C1 C1(CNC(N2CCN(c3snc(C)n3)CC2)=O)CCOC2(CCC2)C1 C1(NC(C2CCC(C)O2)=O)CCC(NC(=O)COCC(N2CCCC2)C)CC1 C(=O)(C(O)C(F)(F)F)NC(CNC(=O)CCCCN1CCOCC1)(C)CC1CC1 N1(C(CC2C(C)OCC2)=O)CC2CCN(C(=O)CCCC3CCC3)C2C1 Cc1cc(C(F)(F)F)cc(C(=O)NC(C)CC(C)NC(=O)C=CC2CCCC2)n1 C1(CC(=O)NCC2CCCN(C(=O)COc3cnn(C)c3)C2)(OC)CCCCC1 C(=O)(C(CC(N)=O)NC(=O)CC1CC(=O)C1)NC1CCN(C(C)=O)CC1 c1(C(=O)NCC(C)C(F)C(=O)NCc2conc2C2CC2)cncc2[nH]ccc12 c1(C(=O)NC(C)CCNC(c2ccc3c(c2)COC3)=O)ccc2c(c1)C(C)CO2 N1(C(c2cnc(N(C)C)c(Cl)c2)=O)CC2CC1CCC2NC(c1cc(Cl)no1)=O N1(C(CCCOCC)=O)CCCC(C2CN(C(=O)C(CC)CC(F)F)C2)C1 CC1CCN(C)C(=O)C1NC(=O)C(=O)NCC1(F)CCCCC1 c12ccccc1CC(=O)NC(C)CN(C)C2=O.C1(CC#C)(C(=O)OC)CCCC1 C=C(C)c1cn(C2CC3CC2CC3N(CC(OC)OCC)CC)nn1 c1(CC(=O)OCC)nc(C)c(C(N2CCC2CNC(c2ccon2)=O)=O)s1 c1(C(=O)NC2C(C)CN(C(=O)CC3CCCCO3)C2)c[nH]c2ncccc12 C1(C)(CNC(CC(C2CC2)OC)=O)CCC(NC(=O)CCOCCOC)CC1 CCCC(O)(CNC(=O)Nc1c(Cl)cccc1Cl)CCC C(=O)(C(CC(C)(C)C)NC(=O)Cc1ccnn1C)NC(CC(C)C)CO c1(CCC(=O)N(CC(CC)NC(C2CCC(=O)O2)=O)C)cncc(F)c1 CCCCCC(O)CC(=O)NC1(C)CC(NC(c2coc(CCC)n2)=O)C1 c1(-c2nc(C(c3cn(CCCCC)nc3C)O)on2)cccc2cccnc12 C(=O)(C1=C(C)N(C)c2ncnn2C1)N(C1CCN(C(c2c(CC)c[nH]c2)=O)C1)C N1(C(CCSC)=O)CCC(C2CCN(C(c3cncc([N+](=O)[O-])c3)=O)C2)C1 C(C(CCCC)NC(=O)Cn1cccn1)NC(C(F)=CCC)=O C(CCO)(C(=O)N1CCOC(CCNC(C2(C(F)(F)F)CC2)=O)C1)N(C)C C1(C(=O)NCC(C)(C)OCC(=O)NCC2(C)CCCO2)COCCC1(F)F Cc1nc2ccccc2cc1C(=O)NC1COCCN(CC2(C(=O)NC)CC2)C1 N1(C(=O)CC2CCC=CCC2)CCCC(C2CN(C(C3C=CCC3)=O)C2)C1 C(=O)(C1CCCn2nccc21)NC(CNC(C1N(CC)C(=O)CC1)=O)CC(F)(F)F N1(C(CSCC=C)=O)CCC2(C1)OCc1ccccc12 C1(CNC(Cc2c(C)ccs2)=O)CC(C)(C)CN1C(C1CC12CCOC2)=O CCCC(CNC(=O)Cn1nc(C)nc1C)C(=O)N1CCC(C(=O)OC)C1C C1(C(N(C)CC2CCCN2C(=O)CC2CCC(=O)C2)=O)CC12CCOC2 N1(C(C=CCC)=O)CCC(C(N2CCC(C(C)C)(CN(C)C)C2)=O)C12CC2 C(C)(CCOC)NC(CN(C(=O)CNC(=O)CCOC(C)=O)CC)=O c1(CNC(C(c2cn(C)nc2)O)=O)nc(C)c(C(=O)NCCCC(F)F)o1 c1(NC(C(c2ccco2)NC(C2CC=CCO2)=O)=O)ccc2nccn2c1 CC(C)C(F)(CNC(C1CCC2(CCC2)C1)=O)C(=O)NCCCN(CCO)C c1(-c2cc(C(=O)NC3CC(N(C(CCC=C=C)=O)C)C3)on2)cccc(C#N)c1 C1(CNC(C(C)SC)=O)CCN(C(=O)CNS(=O)(=O)CC)CC1(F)F C1(NC(C(c2c(Cl)cccc2Cl)C)=O)CCN(C(=O)CCF)C12CCC2 Cc1cc(N)n(CC(N2CC(CNC(c3sccc3C3CC3)=O)C(C)C2)=O)n1 C1(CC)CCN(C(c2cc(C(C)C)oc2C)=O)C1CNC(C1CC2CC2C1)=O C1(C(=O)NCC(C)NC(c2[nH]c(=N)sc2C(F)(F)F)=O)(COC)CC=CCC1 N1(C(CC=CCC)=O)CCC(C)CC1CNC(=O)Cn1ccc(C)cc1=O C(c1ccccc1F)=CC(=O)NCC(CC)(C)NC(c1ccoc1C)=O c1(OCC(=O)NC)cccc(CC(=O)N(C2CN(C(C3SCCC3C)=O)C2)C)c1 N1(C(C(c2ccc(C)s2)C)=O)CCC2(CCC(NC(=O)CCC3CCC3)C2)CC1 C1(CC(=O)NCc2cc(O)cc(F)c2)CCC(F)(F)C(=O)N1 C(=O)(C(F)=CCOC(=O)N)N=CCCC.C=C C1(N(C)C(c2ccc(C3CCOC3)s2)=O)CN(C(=O)C(F)F)CC1F CP(C)(=O)c1cnc(C(N2CCN(C(c3sc(C#N)cc3Cl)=O)CC2)=O)nc1 CC12CN(C(c3cnc(C4CC4)[nH]3)=O)CC1(C)CN(C(C1CC(=O)N1)=O)C2 C#CCCCCCCC(=O)NCCOCCC(=O)N1CC(SCC)C1 C12(CNC(c3ccc(OCCC)cc3)=O)CCCC1CC(=O)N2 C(c1ccc(C)cn1)=CC(=O)NC1C(NC(C(CCC)C)=O)C1 C1(C2(O)CN(C(=O)CC3(CO)CC3)C2)(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 C1(C(N2C(C(=O)NCC(C)C#N)CSCC2)=O)CC2C(C1)C2(F)F c1(NC)cccc(C(=O)N(C(C)CCNC(=O)CC2CC(N(C)C)C2)C)n1 C1(NC(c2c(CC)csc2)=O)CCCN(C(c2cnc(OC(C)C)cn2)=O)C1C C1(CNC(C(C=C)O)=O)CN(C(=O)C(O)CCSC)CCC1C N1(C(C(C)SC(C)C)=O)CC2C(NC(=O)C=CC(=O)N(C)C)C2C1 c1(C(C(=O)NCCCOC)N(C(CC)CC)C)c(C)noc1C c1(C(N2C3C(N(C(C(COC)C)=O)C)CC(C3)C2)=O)ccsc1S(C)(=O)=O c1(NC(c2cc(-c3nc[nH]n3)ccc2F)=O)c(F)cc(F)cc1Br C1(CC)CCN(C(C2CC2CCOC)=O)C1C(=O)NCC1(F)CC1 c1(C(=O)NC2(CCOC)CCN(C(=O)C=C(C)C(F)F)C2)cn(C)c(=O)nc1O c1(NCC(C(C)C)O)ccc(S(=O)(=O)N2CCC3C(O)CC23)c2ccncc12 C1(N)C2CN(CC3(c4ccc(O)nc4)CC3)CC12.Cn1cc(C(=O)C(=O)C(C)=O)cn1 c1(C(N2CC(c3cn(C(C)CO)nn3)N(C)CC2)=O)cccc2c[nH]nc12 c1(C(N2C(C(CNC(C(CC(C)C)C)=O)(C)C)CCC2)=O)cccc2c1NCC2 C(=O)(C=CS(C)(=O)=O)NC(C)CCNC(=O)CCC1NC(=O)NC1=O Cc1ccc2c(CC(N3CC(CNC(C4C=CCCC4)=O)C(C)C3)=O)c[nH]c2c1 C(c1ccccc1F)=CCC(N1C(C(C)NC(C2CCCS2(=O)=O)=O)CCC1)=O N1(C(c2c(OC)c(Cl)sc2)=O)CC(NC(c2ccnn2C)=O)CC(O)C1 N1(C(=O)CCc2ccc(F)c(F)c2)CCC2(CC(NC(=O)C(F)(F)CF)CO2)C1 N1(C(C2(C)CN(C(CC3C(C)(C)C(O)C3)=O)C2)=O)CCC12CC(C)(CO)C2 C1(NCCNC(=O)NCc2cnn(Cc3ccccc3)c2)C2CCCCCCC12 C12(C(N(CCNC(C3(C(N)=O)CC3)=O)C3CC3)=O)CCCCC1CS(=O)(=O)C2 c1(C(=O)Nc2nc(CNC(C)CC3CCCCO3)[nH]n2)ccc(Cl)cn1 C(=O)(C(C)(O)C(F)(F)F)NCCN(C(C(n1ncc(C)c1)C)=O)C c1(C(=O)NC2C(NC(=O)CN3CCOC3=O)CC2)ccn2nnnc2c1 Cc1ncc(C(N2CCC(CCC(=O)NC(C)CC(N)=O)C2)=O)c(=N)[nH]1 CC(C)C(F)(CNC(=O)CCN(C)CCO)C(=O)NCc1cocn1 CCC(C)C(C(=O)NC(CN=[N+]=[N-])C(=O)NCC1CC(C2CC2)=NO1)N(C)C CC(=O)CCCC(=O)N1CCN(C(c2csc(C)c2N)=O)C(CC(F)F)C1 CC1C(C)N(C)CCN1C(=O)C(CCF)NC(C12CC(CO)(C1)C2)=O c1(CN(C(=O)C(=O)NCC2CC3CCC2C3)CC=C)ccc(F)cc1 c1(C(N(CC(C)CNC(C2CC23CC(F)(F)C3)=O)C)=O)cccc2[nH]ncc12 C1(C(=O)NCCC(=O)NCC)CCCC(C(=O)NCCOc2ccncc2)C1 N1(C(COc2c(CC)cccc2)=O)CC2(C1)CN(C(=O)C(C)(C)CC1CC1)C2 N1(C(CC2(C)CCCO2)=O)CCCC12CCN(C(c1csc(F)c1)=O)CC2 CC1C(NC(=O)CCc2cc(F)cc(F)c2)CCCN1C(C1CN(C(N)=O)C1)=O Cc1nn2ncccc2c1C(=O)NCC(C)N(C(=O)CC(=O)NCC(F)(F)F)C Cc1ncc(CCC(=O)NCC23CC(NC(=O)C(F)CC4CC4)(C2)C3)o1 c1(C(N2CC(O)CC2CNC(C2(CC(F)F)CCC2)=O)=O)cn2ncccc2n1 c1(C(=O)NCC(C)CN(C)C(c2nn(C)cc2[N+](=O)[O-])=O)nc2ccccc2[nH]1 c1(CC(=O)NC23CCCC2CN(C(=O)C2=CCCS2)C3)ccc2c(c1)CCCC2 N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(=O)CC2CNC(=O)C2)CC12CCC2 C(C(C(=O)NC1CCCCC1NC(C1CC2CC1C2)=O)C(C)(C)C)OCC=C N1(C(COc2c(C)cccc2)=O)C2CC1CN(C(=O)CCC(C)(C)F)C2 c1(C(N(C2CN(C(C(CC)OC)=O)CC2O)C)=O)cc2cccc(C)c2nn1 c1(C(N2CCC3(CCCN3C(=O)C3CC3)C2)=O)c[nH]c2cc(Cl)c(Cl)cc12 Cc1cc(Cl)c(C(N2CCC(O)(CNC(C3COC(=O)N3)=O)C2)=O)cc1F CC(C(=O)N1CC(NC(C2(CCF)CCOCC2)=O)C(F)C1)C(C)(F)F N1(C(c2c(OC)csc2)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC1CC(F)F C(C(F)(F)F)(C(F)(F)F)c1n(C(c2ncc(-n3ncc(C)c3)cn2)C)ccn1 C1(C(N2CCCC(CCO)C2)=O)CC(F)(F)CN1C(c1nccs1)=O c1(N2CCCC(Nc3c(-c4ccc(Cl)cc4)cccc3)C2)cc2ncnn2cn1 CCC(CC(=O)NC(C(=O)NOC(CSC)CSC)C1CC(CO)C1)C1CCC1 CCCCCCC(F)C(=O)NC(C)CN(C)C(c1cn(C)[nH]c1=N)=O N1(C(C2(N(C(=O)Cc3cccc(Cl)n3)C3CC3)CCC2)=O)CCOC2CC12 N1(C(C2CC(OC)C2)=O)CCC(C(C)(C)C)(CNC(=O)CN2CCC(C)(O)C2)C1 c1(NCC2(C=C)CCC2)cc(=NCc2cc(Br)cc(C)c2F)[nH]cn1 c1(C(N(CC(CC)NC(C(CCC#C)O)=O)C)=O)c(C)c(C)cc(C)c1C N1(C(c2c(C)nc(C(F)(F)F)s2)=O)CC(C)N(C(c2ccc(C#N)o2)=O)CC1C C1(C2CCN(C(C3(c4ccccc4)CC3(F)F)=O)C2)(NC(C(=O)NCC)=O)CC1 c1(NC(C(C)OC)=O)ccc(O)c(Br)c1.C12(CO)CC(F)(C1)C2 C12(C(=O)NCCCn3cc(C4CC(C)(C)OC4)nn3)CCCC1C2(F)F C1(C(=O)NC(C(C)C)CCNC(c2ccc(=O)n(C)c2)=O)CCCC1S(C)(=O)=O Cc1ccc(CNC(=O)C(C2CCCC2)NC(c2sccc2CO)=O)c(O)c1 C1(S(C)(=O)=O)(C(=O)NC(C2CCN(C(C3=C(C)CCC3)=O)CC2)C)CCOCC1 c1(C(=O)NC(CC)CN(C(=O)C(C)CF)C)ncc([N+](=O)[O-])cc1Br C1(C(=O)OCC)COC(CNc2c[nH]c(CN(C)C)c2)C1 C12(C(=O)NCCC3CN(C(C(C4CC4)OC)=O)C3)C=CC(CC1)C2 c1(C(=O)NC(C)(C)C=CC(=O)Nc2cnc(F)nc2)cccc(F)c1F CC(C)C(O)C(=O)NCC1CC(F)CN1C(=O)COCC1CCOC1 Nc1cc(Br)cnc1C(=O)NC1CCCN(C(C2CCOCC2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC1COCCN(C(C2CCOC(C)(C)C2)=O)C1 N1(CC(=O)OC)CCN(C(=NCC=CC2CC2)NC2CSC(C)C2)CC1 C(=O)(C(Cc1ccccc1)NC(C1CCCN1C(c1csnn1)=O)=O)NC c1(C(N2CCC(NC(c3c(C)ncn3C)=O)C(O)C2)=O)cc(Cl)cc(Cl)c1O Cc1cc2nc[nH]c(=NCC3CC(CNC(c4ccoc4Cl)=O)CO3)c2[nH]1 Cc1oc(C(F)(F)F)c(C(N2CCN(C(C3CCC(=O)N3)=O)CC2)=O)c1C CCC(F)(C(=O)OC)C(=O)N1CC2CC1C2CNC(C1(O)CCC1)=O C=CC(C)(C)CC(=O)NCC1C2CN(C(=O)C=Cc3ccc(C(N)=O)o3)CC12 N1(C(C(C)=CCC)=O)CCCC(C(=O)NCC(C)(C)CN(C)C)(CC)C1 Cc1cc(NC(C2CCCCC(=O)N2)=O)ccc1NC(=O)CS(N)(=O)=O C1(C(=O)NCC2CCN(C(C(N3CCC(O)CC3)C)=O)C2)CCC2C(C1)C2(F)F N1(C(C(CC=C)c2n(C(=O)CC3CCC(=O)CC3)ccn2)=O)CCCC(C)(C)C1C c1(CCC(=O)N(CCCNC(c2csc(O)n2)=O)C)cc(F)cc(F)c1 N1(C(COCCOC)=O)CC(NC(C2CCC(c3ccccc3)O2)=O)C(O)C1 c1(C(c2nc(-c3ccc(OC)nc3)nn2C2CCC2)C)cn(C)c2ccccc12 c1(Nc2c(NC(CC(=O)OC)C)cccc2)ncc2[nH]ncc2n1 C(C(C)(C(N)=O)NC(C1(CNC(c2cncc(N)n2)=O)CCCCC1)=O)OC C(=O)(CC(C)CC(C)(C)C)N(C)CC1N(C(Cc2cn(CC)nc2)=O)CCCC1 C1(CC(=O)NC(C(=O)OC(C)C)C)CCCN(C(=O)CC2C=CCCC2)C1 C1(N(C(=O)CSCCC#N)CC)CCN(C(=O)CCSC2CCCC2)C1 Cc1ccc(C(C)NC2(c3ccc(F)cn3)CCOC2)cc1 C1(C(N2CCC(O)(CNC(C3(OC)CCOC3)=O)C2)=O)CC2(CCCC2)C1 C1(CO)CCC(C)(C)N(CC)C1.c1(CCN)cc(C2CC2)nn1C(C)C C1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)(COC)CCCCO1 C(=O)(C1=NOC(C)C1C)NC1C(NC(c2c(C)n(C(C)C)nn2)=O)COCC1 CC1CN(C(c2coc(C(F)F)n2)=O)CCCN1C(c1cnn2ncccc12)=O c1(CC)ncc(C(=O)N(C)CCN(C(=O)CCc2cnc(C)s2)C)c(O)n1 c1(C(=O)NCC(CO)NC(c2cccc(OC(C)C)c2)=O)n[nH]c2c1COC2 C1(CNC(C=CCN(C)CC)=O)CN(C)CCN1C(=O)CCNC(=O)CC c1(C(=O)OC)ccncc1-n1cc(SCC(=O)O)nn1 C12(NC(C#CC(C)C)=O)CCCC1N(C(=O)CSCc1csc(=N)[nH]1)CC2 N1(CC(=O)NCCN(C(=O)Cc2cncn2C)CC)CCCNS1(=O)=O CC1CC(CC(N2CCC2CC2CC2)=O)CN1C(=O)Cn1cccc1 c1(CC(=O)NC(C2CCCCC2)CO)ccc(Br)s1 c1(C(N2CCC(C(C)NC(c3c(C)coc3)=O)C2)=O)cc(C(N)=O)ccn1 C#Cc1cnc(C(=O)NC23CCN(C(c4cn(C)cc4C)=O)CCC2C3)c(C)c1 N1(C(Cc2c(C)non2)=O)CC2(CC2)CC1CNC(=O)C(C)(F)F C1(NC(c2c(C#C)cnn2C)=O)CC2CC(C1)N(C(=O)CSc1cnn(C)c1)C2 C1(C(N(CCC(C)NC(=O)CCC=CBr)C)=O)C(C)(C)C1(C)C N1(C(c2cn(CC)nc2C)C(=O)NC(C)C)CCS(=O)C(C)C1C C(=O)(CC(C)C(F)(F)F)NCC(=C)CCNC(=O)Cc1cccc(C2CC2)c1 CC(CC(=O)NC1CCOC1C(N1CC(CC2CC2)C1)=O)N(C)C n1(CC)ncc(CNC(C(C)(C)CC2CCCO2)c2nnnn2CC2CC2)c1C c1(CCC(=O)NCCN(C(c2c(NC)c(F)ccc2)=O)C)cccc([N+](=O)[O-])c1 c1(C(=O)N(C)C)ccc(C=CC(=O)NC2CCCC2NC(c2cnc(C)o2)=O)cc1 n1(CC)cnc2c(NC(C)CC(N)=O)[nH]c(=NC(C)c3ccccc3)nc12 N1(C(c2nn(CC)c(O)c2)=O)CC(O)(C2(CNC(c3cnn(C)c3)=O)CC2)C1 C#Cc1cccc(CC(=O)NC(C)(CO)C(=O)NCC=CBr)c1 c1(NC(N(CCn2cc(CNC(C)=O)nn2)CC)=O)cc(Br)c([N+](=O)[O-])[nH]1 c1(C(C)C)ncc(C(=O)NCC(C)N(C(=O)C=CCF)C)n1C c1(N(C(=O)CN2CCSCC2)C)cc(O)cc(Cl)c1.C12CCN1C2 c1(C(CC)C)nc(NC2CCCCC2NC(C2CCC3CC3CC2)=O)cc(C)n1 C(=O)(CCCCCn1cc(CN2CCCCC2)nn1)N(C)CC1CCCO1 Cc1nc(C(N2CCCC2CNC(c2ncc3ccccn23)=O)=O)c(=O)[nH]c1C c1(-c2nc(CCC(=O)NC(C)(CNC(=O)C=CBr)CO)on2)cccc(Cl)c1 CC(CCNC(=O)CCn1ncn(C)c1=O)CCNC(=O)C=C1CCC(C)C1 c1(-c2c(C)onc2)cccc(NC(=O)NS(=O)(=O)CC(C)C2CC2)c1 C1(NC(c2cc(C)oc2)=O)C(C)CCN(C(=O)Cc2ccc(Cl)nc2)C1C N1(C(c2cc(C)c(O)nc2)=O)CC2CN(C(c3cc(O)nc(O)n3)=O)CC2(C)C1 c1(C(=O)NCC(CC(=O)OC)NC(C(C(=O)OCC)OC)=O)ncc(Cl)cc1Cl N1(C(C(C)(C)NC(=O)OC)=O)CCC2(CC2C(=O)NCC2CC(O)C(O)C2)C1 C1(C(=O)OC)CCCN(C(c2cccn(CC(=O)OC)c2=O)=O)CC1.C1CC1 c1(OC)ccc(N(C)Cc2csc(Br)c2)c(OCc2ccco2)c1 CC1(C)CC(C(N2CCC(C3(NC(=O)C(F)F)CC3)CC2)=O)CC(C)(C)C1 N1(C(Cc2nc(C)oc2)=O)CC2(CCCC2)C1C(=O)NCC1CCCOC1 N1(CC(=O)NCCC2CC(CF)C2)CCCCC1.C1COC1 C1(c2cn(CCCC(=O)N(CCCN(C)C3CC3)C3CC3)nn2)CC2(CCC2)C1 C=CC1(C(N2CCCC3(C2)N=N3)=O)CCN(C(=O)C#CC2CCC2)C1 CN1CCN(C2(CC(N3CCC(NC(C45CCC(CC4)C5)=O)C3)=O)CCC2)CC1 c1(CN2CCC(C(=O)OCC)CC2C)ccccc1S(=O)(=O)NC c1(C(N2CCN(C(c3c(C)cc(C)o3)=O)CC2)=O)cccc2ncnc(O)c12 C(=O)(C(O)C(CCC)NC(c1cc(CO)on1)=O)NC(CC#C)C(=O)NC O=C1CC(C(=O)NC2CN(C(c3cnsc3)=O)CCC2C(F)(F)F)CC(=O)N1 CCCC(F)C(=O)N1CCCC1C(C)NC(=O)CCC1CC(F)(F)C1 C(C1=CCN(C(c2ccn(C(F)F)n2)=O)CC1)NC(C(C)(C)c1ccncc1)=O C(C)(C)(CC(F)C(=O)N1CC(n2cnnc2)C1)NC(C(Br)=C(C)C)=O C(=O)(C1=C(C)CN1)N1CCC(N(C(=O)C(O)C2CC2)CCC)C1 CCCCCC(C)(C)CNC(=O)C(C(C)C)NC(=O)CN(C)C(C)C C1(NC(C2C(C)C2C)=O)CC(C)(CNC(C2CCCCO2)=O)C1 C1(NC(CCn2c(C)cc(C)n2)=O)CCN(C(=O)C(F)(F)CC2CC2)CC1C C(=O)(C(C)(O)C(C)(C)C)N1CCC(CN(C(Cc2c(OC)ccnc2)=O)C)C1 c1(OC)ccc(C(N2CCCC(c3cnc[nH]3)C2)C(=O)NC(C)C)cc1C1CC1 c1(N2CCC(NC(c3ccc(CC)cc3)=O)C(O)C2)ncnc2sc(CC)cc12 N1(CCNC(C(CC)SC)=O)CCN(C(=O)C(C2CCC2)SCC)CC1 N1(C(CCC(=O)NCCC)=O)CCCC(C)(CNC(=O)CCc2cnoc2)C1 C1(NC(C=CC=CCCCCC)=O)CCC(C)N(C(c2cccc(CO)n2)=O)C1 c1(C(=O)NCCCCN(C(C(CC(C)C)OC)=O)C)cc2cn[nH]c2cn1 CCCC(C(O)C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CN=[N+]=[N-] CCCCCC(C(=O)NC)NC(=O)CC1CN(CCc2c(OC)cccc2F)C1 N1(C(c2cc(C)ncc2C)=O)CC2(CCCC2)C1C(=O)NCCC(C)N1CCC1 c1(-n2cc(CCOC)nn2)cccc(C(=O)NC2(C)CCSCC2)c1 c1(CC)cc(C(N2CCC(O)(C(C)CNC(c3cc(CO)[nH]n3)=O)C2)=O)nn1C n1(CC)nnnc1C(c1nc(C)cs1)NC1(c2ccccn2)CCC1 C=CCCCC(=O)NC(C)(CNC(c1sc(=N)[nH]c1C)=O)CO c1(C(=O)OC)cc(NC(=O)NCC(c2cccc(Br)c2)O)cc(Cl)c1 C(=O)(CC1=CCOCC1)N(C)CC1CCCC1NC(c1ccc([N+](=O)[O-])cn1)=O N1(C(C2(C=C)CCN(C(c3n[nH]c(C)c3C)=O)C2)=O)CCCCCCC1CC c1(C(CCOCC)NCC(C2CCCC2)NS(C)(=O)=O)cn2ccsc2n1 C#CC1(C(=O)NCC2COCC2N(C)C)CCN(C(=O)C2=CCSC2)C1 C1(CC)(NC(c2cc(C#N)cs2)=O)CCCN(C(C2CCC(C(N)=O)O2)=O)C1 N1(CCNC(CCCSC(C)(C)C)=O)CCCCN(C(C2CCNC2=O)=O)CC1 c1(C(=O)NC(C2CCCN(C(=O)CCc3cnn(C)c3)C2)C)ccnnc1O n1(CC(C)CO)nc(CCCN2CCCC2)nc1-c1cn(-c2ccccc2)nn1 C1(NC(c2cnc(CC)nc2C)=O)CCN(C(=O)C(C)(O)COC)C12CCCC2 Cc1oc(C(C)(C)C)cc1C(=O)NC1CC1CNC(=O)C(c1ccccc1Cl)O C1(C)(CNC(=O)Nc2c(N(C(C)=O)C)cccc2)CCC(=O)NC1 c1(C(=O)N(C(c2nc(C)no2)CC)NC(C)(C)C)cc(-c2cccs2)[nH]n1 c1(OC)cc(C(=O)NC2CC(O)CN(C(c3cnn(CCO)c3)=O)C2)ccc1O C1(C)(CNC(CCN(C(C=C(C)C2CC2)=O)CC2CC2)=O)CCCCC1O C(C)(CCC#N)(c1nnnn1C1(C)CC1)NCc1scc(C)n1.c1ccncc1Br CN1CC(O)CCC1C(=O)NC1(C(=O)NC(CO)C(=O)NC(N)=O)CC(F)C1 c1(C(N2CC(CC)(NC(c3ccn(C)c3C)=O)C2)=O)cnc(O)cc1C c1(CC)ccc(NC(=O)CC2CN(C(C3CC(=O)CS3)=O)CCO2)cc1 CN1C(=O)C(=O)N(CC(=O)NCC2(C)CCCN2C(c2ccno2)=O)C1=O C1(C(C(=O)NCCC(=O)NC2CC2)NC(C(C2CCCCC2)C)=O)CCCOC1 Cc1nnc(CCC(=O)NC2(C)CC(NC(C3CNC(=O)N3)=O)C2)n1C c1(C(CCCOC)NCCCCOC)ccc(OC)c(F)c1 N12CCC(CC1)C(=O)N2.C1C(CO)CC(=O)N1.C1(COCC)CC1.C1CC1 c1(-c2c(CN3CCC(NC(=O)NCC4CSCCS4)C3)cno2)ccc(F)cc1 Cc1c(C(=O)NC2CN(C(C3CC3C)=O)C2)oc2ccccc12 Cc1nc(C(N2CCN(C(c3cnc[nH]3)=O)C(CC3CC3)C2)=O)c(C)n1C1CC1 N1(C(CC)=O)CCN(C(c2ccc(SC(F)(F)F)o2)=O)CC(C)(F)C1 N1(C(CC=C)=O)CCCC2CN(C(c3nscc3N)=O)CCC12 c1(CC)nnc2n1CC(C(N1CCCC(Nc3cc(NC)ncn3)C1)=O)CC2 C(=O)(C(CO)C(C)(C)C)NCCCN(CCCNC(C(CSC)C)=O)C c1(CC)cc(CNN2CCC(Cc3ccccc3F)CC2)n(C)n1 N1(C(Cc2cc(C)on2)=O)CCC2(CCN(C(=O)C(F)(F)C3CC3)CC2)C1 c1(NC2CCCC(C)CC2)ccc2ccncc2c1[N+](=O)[O-] c1(C(N2C3C(C(=O)NC4CCC(C)CC4)C(C3)C2)=O)cccc2cccnc12 c1(NC(C(=O)N(C(C)CCN2CCCC2)C2CC2)=O)ncc(-c2ccncc2)s1 C(C(C(=O)NC1(CNC(C2CC2c2nc[nH]n2)=O)CC1)c1ccccc1)SC C1(C(NCP(C)(C)=O)=O)CCCC(NC(C2(C(C)(C)OC)CC2)=O)C1 C1(NC(C(CC)OC)=O)CCSC12CN(C(c1cc(C(C)(C)C)oc1C)=O)C2 c1(C(N2CC(N(C)C(c3cc(C(F)F)ccc3F)=O)C2)=O)ccc2cnoc2c1 C1(C(C)(C)C)CCN(c2nc(=N)nc(N3CCC(N4CCCC4=O)C3)[nH]2)CCO1 c1(C(=O)NCCCOCCNC(=O)CC2CCC(O)C2)ccc(F)c(F)c1 CC(Cc1cnc[nH]1)C(=O)NCC(C)CNC(=O)COC1CC1 C1(NC(C=CCC)=O)CCN(C(c2cc(OC)c(Br)s2)=O)CC1(C)C CCCC(=O)N(CC(=O)NCCc1ncc[nH]1)CC(C)C O(NC(=O)C(CC)NC(c1ncoc1CC)=O)CCC#C c1(NC(=O)NC(c2cc(C)ns2)(C)C)nc2cc(Cl)c(C)cc2s1 C1(N=[N+]=[N-])(C(N2CCC(CSC)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)C1 C(CCO)(C(=O)NC1CCCCC1NC(=O)Cc1csc(C2CC2)n1)N(C)C C(C(N=c1ccc2nnnn2[nH]1)C(C)C(C)C)NC(Cc1n(C)nc(CC)c1Cl)=O C1(CC(=O)O)(NC(=O)C(=O)N)CCCCC1.n1(CC)ccc(CC)n1 N1(C2CCN(C(C3C(=C)CC3)=O)C2)CCC(N(C(=O)C(CCC)OCC)CC)CC1 c1(C(=O)NC(C)C(C)(C)NC(=O)CC(C)n2cccn2)cnc(O)c2cncn12 c1(C(=O)NCC(C)CNC(=O)CNC(C2CCOC2)=O)cccc(Cl)c1 C1(C(=O)NC2CCCN(C(CSCC#C)=O)CC2)CC12CCC(C)(C)CC2 c1(C(N(C2CN(C(=O)CCc3nccn3C)C2)C)=O)cc(C(F)(F)F)cnc1N c1(C(=O)NCCC(CNC(=O)C(F)=CC2CC2)O)ccc(C2CCOC2)cc1 C1(C)(COC)CC(NC(=O)C=Cc2nc(C)co2)CN1C(=O)CNC(=O)C1CC1 c1(C(N2CC(C(C)NC(C3CC34CCSCC4)=O)C2)=O)csc2c1CCCC2 c1(C(N2C(C)CCC(CCc3ccc(OC)cc3)C2)=O)cc(F)c(Br)cc1C C(=O)(CCS(=O)(=O)C(F)(F)F)N(C1CCCCN(C(C(CC)(C)C#N)=O)C1)C C1(NC(CCC(C)=O)=O)CN(C(c2cccc(F)c2Cl)=O)CCC12CCOCC2 c1(CN2CC(n3ncc(C(=O)OCC)c3)C2)ccc2oc(C)c(C)c2c1.C1CO1 C1(O)(C(=O)O)CCCN(C(=O)COC(C2(CC(CC)OC)CCCC2)=O)C1 c1(N2C(CCNC(CN(C(C)=O)C)=O)CCC2)ncnc(C)c1OC N1(C(c2ccc(C)s2)=O)CC(C)OC2(CCN(C(C3CCCSC3)=O)C2)C1 N#Cc1ccc(=NCC(=O)NCC2CC2CNC(c2cc(C(F)F)no2)=O)[nH]c1 N12CC3(CC3)CC1CNC(=O)c1nsc2n1.C(=O)(CCC(F)F)OC n1(CC)cnc2c(NCC(CCC)CCO)nc(N3CCSCC3CCO)nc12 C12(NC(CCCCSC)=O)CC(CNC(=O)C(O)CN(C)C)(C1)OC21CCC1 c1(CNC(C(C)=CCC)=O)cc(C(=O)N(CC(O)CC)C)cs1 CCCCC(CC)CCC(=O)N1CCC(S(=O)(=O)NC(=O)OC(C)(C)C)C1 c1(C(=O)NCC=CCNC(C=CC=CC)=O)c(C)cc(C)c([N+](=O)[O-])c1C CC1=C(C)CC(C(=O)N(C(CNC(=O)CS(N)(=O)=O)C2CC2)C)CC1 N1(C(COC)=O)CCN(C(=O)CCS(=O)(=O)N(C)C)CC(C)(F)C1.C1CO1 N1(C(CN2CCN(C(C(c3cccnc3)C)=O)CC2)=O)CCC2(CC1)CC2 c1(C(=O)NCC(CC)N)ccc(Oc2ccc(Br)cc2)c(C(C)SC)c1 C(=O)(C=CS(C)=O)NCCC1CCN(C(C2(CCOC)CCC2)=O)C1 C1(C(=O)NCC2CC2C2CCCO2)CN(C(=O)CC2(O)CCC2)CCO1 CC1=C(C(=O)Nc2cccc(OCCC(=O)O)c2)Cn2ncnc2N1C c1(C(N(CCCN(C(CCC(=C)C)=O)C)C)=O)nccc2ccccc12 N1(C(C2(C)CCCN2C(c2ccc(B(O)O)cc2)=O)=O)CCCC2(CCOC2)C1 c1(C(=O)NCC2CC(NC(c3ccc(F)c(O)c3)=O)C2)cc2c(nn1)CCCO2 CC1(C)CC(=O)NC1NC(=O)C(CC1CCOCC1)NC(=O)CCNC(N)=O C(=O)(C(C(C)C)NC(N)=O)NCC=CCC(=O)N(C1CCCC1)CCOC N1(C(C2=C(C)OCC2)=O)CCCC2(CCN(C(C34CCCC(C)(C3)OC4)=O)C2)C1 C1(C(=O)Nc2cnn(C(F)F)c2)CN(c2ncc(F)cn2)CCC1(F)F N1(C(C(C=C=C)C)=O)CC(C(=O)NCCN(C)C)C2(CC2)C1 C(=O)(C(CC(C)C)NC(C)=O)NCC(CNC(CC1(C=C)CC1)=O)OC N1(C(CC(C)C)=O)CC2CCN(Cc3cc[nH]c3)CC2C1 c1(N2CC(CNC(=O)OC(C)(C)C)C3(C2)CC3)nc2ccccc2s1 C1(c2nn[nH]n2)(C(N(CC(C)OC)C)=O)CC2(CC2)C1 C1(OC)CC(CNC(=O)CCC2CCOC2)N(C(c2n[nH]c(C)c2O)=O)C1 CC1C(NC(=O)CC2(C)CCC2)CCCN1C(c1csc(C(C)(C)C)n1)=O C1(C)(CNC(c2c(OC)csc2)=O)CCN(C(C2(C)CC(O)C2)=O)C1 c1(OC)cc(C(N2CCCC(NC(=O)C(=O)O)C2)=O)cc([N+](=O)[O-])c1 C1(C)(C(=O)NC(C2CCN(C(N)=O)CC2)C)COC(=O)C1.C12CCN(C1)C2=O C1(CC(=O)NCC2(F)CC(NC(CC(C=C)C)=O)C2)CC(C)CC(C)(C)C1 C(=O)(CCCCCO)N1CCC(N(CC#C)C(C2CC2(Cl)Cl)=O)CC1 C1(N(C(C(C)(F)F)=O)CC2CCCO2)CCN(C(c2cc(C(N)=O)no2)=O)CC1 Cc1cccc(COCC(=O)NCCC2CCN(C(C3CCCC(=O)O3)=O)C2)c1 Cc1ccn(CCC(=O)NC2CCCC2NC(c2cnn(CCF)c2)=O)n1 N1(C(c2nnn(CC)c2C)=O)CC2CC1CN2C(=O)C(c1c(Cl)cccc1Cl)C CCC(C)(CCNC(c1cnc(C2CC2)o1)=O)NC(c1cc(Cl)ns1)=O C1(C(N2CC(OC(C)=O)C2)=O)CCN(C(=O)c2cc(C)cc(O)n2)O1 CCCC(C)(C)CC(=O)N1CCN(C(c2cc(C#N)ccc2F)=O)C(C2CC2)C1 C1(NC(CCOCCOC)=O)CCC2(CC1)CC2NC(=O)C(C)C(C)(C)C C(C)(C(=O)N1CC(CNC(=O)C(c2ccns2)NC(=O)OC(C)(C)C)C1)SC N#Cc1cccc(CCC(=O)NCCC2CN(C(C3CCSC3)=O)CCCO2)c1 c1(C(N2CCCCC2C(C)CO)C(=O)NCCOC)cc(C)ccn1 c1(C(=O)NCCOC2CCN(C(C(CC)C(C)C)=O)C2)ccc2nnnn2c1 n1(CC(=O)NCC(CN(C(=O)CC2(O)CCCCC2)C)O)ccc2ccccc12 CC1=NOC(=O)C1CCC(=O)NC(CNC(=O)CC1COCCO1)C(C)C C1(CCC)CN(C(c2[nH]ccc(=O)c2C)=O)CCN1C(c1cnc(O)s1)=O CCC(O)C(C)C(=O)NCC(C)=CC(=O)NC(c1cncnc1NC)=O N1(C(C2C(C(=O)OC)C2)=O)CCCC(C2(NC(C3CN(S(N)(=O)=O)C3)=O)CC2)C1 N1(C(C(CCC)OC)=O)CC(NC(=O)CCc2ccc(Cl)cc2)CC(F)C1 c1(NC(c2nc(N)c(-c3cnc(C(N)=O)nc3)cc2)=O)c(F)c(F)nc(F)c1F C(=O)(C1CCCc2ncnn21)N1C(C)CCC(NC(=O)C(C)(C)n2ccnn2)C1 c1(C(N2C(C(=O)NCCn3cc(C)nc3)C(O)CC2)=O)cc(C)cc(C#N)c1 C(CCCCCC(=O)NC1CC(O)CN(C(=O)CCC2(C)N=N2)C1)SC c1(C(N2C(C(N3C4CCCC3COC4)=O)CC3CC32)=O)ccc2c(c1)CCC2 N1(C(C2(CCC)CC2)=O)CCN(CC2CCN(C(C3CCC(C)C3)=O)CC2)CC1 C1(CC(=O)NC(CC(=O)N(c2ccsc2)C)C2CC2)CC2(CC2)CO1 C1(F)(CNC(c2nn(C)c(C(F)F)c2)=O)CCN(C(=O)COCP(C)(C)=O)CC1 CC1(C(N2CCOC(CC(=O)NCC(O)C3(Cl)CC3)C2)=O)CC(C#N)C1 N1(C(C2CC(CCC)OCC2)=O)CC(C2(NC(=O)CC(=O)N(C)C)CC2)C1 c1(C(N2CCC(C(O)CO)CC2)C(=O)NC(C(=O)OC)C)sc(Br)c(C)c1C N1(C(=O)OC(C)(C)C)CC(NC(=O)OCc2cc(Br)cnc2F)CC12COC2 Cc1ccc(C(=O)NC2CCN(C(c3cc(N)ccc3O)=O)CC2C)c(O)n1 N1(c2c(S(=O)(=O)N3CC(COC)OCC3)cccn2)CCN(C)C2(CCOC2)C1 C1(C(=O)N(CC(C)N(C)C)C)(CC)CCCN(C(=O)C(C(C)(C)C)SC)C1 N1(C(C=CCCC)=O)CCCC(CCNC(=O)Cn2cc(C)cn2)CC1 CC1(C)C=CC(NC(=O)NC2CC(OCC(F)(F)F)C2)CC1 C(=O)(CC(C(C)C)NC(C1CC(C)CCO1)=O)NCc1c(C)scn1 Cc1[nH]nc2cc(C(=O)NC3CC3NC(c3c4c(nn3C)CCSC4)=O)ccc12 C1(OC)CN(C(=O)C(F)CC2CCOC2)CC1C(=O)N(CC1=CCSC1)C C12CC13CCN(C3)C(=O)CCN2.Cc1cc(CNC(C2(F)CC2)=O)no1 CCC(O)CC(=O)NCC1(O)CC(CNC(=O)CN(C)C(C)=O)C1 c1(C(N2CCC(C)(CCNC(CCCOCC=C)=O)C2)=O)cc(C)ccc1N c1(C(=O)NCC(C)CNC(=O)CN(C)C(c2ccccc2)=O)ccn2ccsc12 O=C1CCc2cc(C(=O)NC3C=CC(C(N4CCC5(C=CC5)CC4)=O)C3)ccc21 c1(CN(CC(C)(C)C)CC2CC3C=CC2C3)ccc(C2CC2)cc1 C1(C(N2CCC(c3cccc(Cl)c3)C2)=O)CC(O)CN1C(c1ccccc1F)=O C1(NC(c2c(C)ncnc2C)=O)CCC2CCN(C(=O)C(C)n3ccnc3)C12 C1(C(=O)NCC(CC=C)(C)C)CC(F)CCN1C(c1ccccc1O)=O C1(NC(C(CSC)OC)=O)CN(C(=O)C=Cc2ccc(Br)cc2)C(C)(C)C1 C(=O)(CCCCC(F)F)NC1(C2N(C(c3ccc(OC)cc3)=O)CCCC2)CC1 C1(NC(C(C)OCCCC)=O)CN(C(c2cc(C(F)F)cs2)=O)CC1CC c1(C(C(=O)NCC(COC)NC(=O)Cn2[nH]cnc2=N)C)cnn(C)c1 C(CN=C(NC1CC1)N1CCC(F)(c2cc(C)cc(C)c2)C1)NC(=O)NC C1(CO)(CF)CCOCC1.C1C(CO)CNC(=O)c2ccc(o2)C(=O)N1.C1CO1 N1(C(COC)C)CCN(C(=O)C=Cc2ccccn2)C(=O)C1 C1(CNC(CS(CC)=O)=O)(OC)CCN(C(c2c(OC)ccnc2F)=O)CC1 C1(NC(c2nc(C(C)NC(CN(C(=O)OC)C)=O)oc2)=O)CC(=O)N(O)C1 C1(C(C(=O)NC2CC2)N(C2CCCO2)Cc2ccsc2)CC2CC2C1 Cc1ccc(C)c(SCC(=O)N(CCCNC(C2CNC(=O)N2)=O)C)c1 N1(C(=O)Cc2cn[nH]c2)CCC(C2CCO2)CC1 C1(NC(c2cnc(OC)[nH]2)=O)CCC(C(N2CCC2CC(C)(O)CC)=O)CC1 C1(NC(c2ccc3nccn3c2)=O)CS(=O)(=O)C2CN(C(c3ccsc3)=O)CC12 c1(CNc2ncc(-c3cc(CO)c(F)cc3)cc2O)cc(Cl)cc(Cl)c1Cl N1(OC)CCN(c2cccc(Br)c2)C(=O)C1.c12cc(ncn1)CN1CCCC1C2 c1(C(=O)NC2CN(C(C3(F)CC3)=O)CC2O)cccc(C(F)(F)F)c1Cl Nc1c(C(N2CC3(C2)CN(C(=O)C(O)CF)C3)=O)cc(F)cc1Br c1(C(=O)NCC2CC(NC(c3cc(C)sc3C)=O)CC2O)ccsc1S(C)(=O)=O N1(C(C2N(C(C(C3CCC3)OCC)=O)CCC2O)=O)CCOCC(C2CC2)C1 C1(C(=O)NC(CC)CCCO)C(C)OCCN1C(C1CCCC1O)=O C1(N(C)C(c2ncoc2CNC(=O)CC2COC(=O)C2)=O)CCC(C)(C)CC1 c1(NC(C2CC(F)CN2Cc2ccc(Cl)cc2)=O)cccc(OC(F)(F)F)c1Cl CC1CN(C(=O)C(c2ccccc2F)(C)O)CC1NC(C1COCCO1)=O c1(C(=O)NC(CCN(C(C2CC(SC)C2)=O)C)(C)C)cnc(C)nc1 C12(C(N(C(C)CNC(C3(F)C(C)(C)C3(C)C)=O)C)=O)CCC(N(C)C)(CC1)CC2 c1(OCC)cncc(C(N2CCC(OCCNC(c3ccnnc3C)=O)C2)=O)c1 N1(C(C=Cc2occ(C)n2)=O)CCC2C(NC(c3ncccc3Br)=O)CC12 CC12CC(C(=O)NCC3C4CN(C(c5coc(C(F)F)n5)=O)CC34)(C1)C(C)(C)O2 c1(C(=O)NCC(CO)NC(c2ncc(C#N)cc2Cl)=O)cnc2[nH]c(O)nc2c1 Cc1csc(C(=O)NCC2CCCC2NC(c2cc(CCCO)on2)=O)c1C C1(O)(C(N2CC(CNC(c3cccc(C)c3O)=O)C(C)C2)=O)CCCC(C)(C)C1 c1(NC(C2CN(C(c3cc(C)cc(C)c3)=O)C2)=O)ncc([N+](=O)[O-])cc1Cl Cc1c(C(N2CCC(NC(=O)C(C(C)C)NC3COC3)CC2)=O)ccn1C(C)C C1(c2n(CC(=C)C)nnn2)(NCC(C)(C)C)CCCC1CCc1ccccc1 CCC(CC)C(C)C(=O)NCCC1CCN(C(c2nocc2C(C)C)=O)C1 N1(C(C(C)=C(CC)C)=O)CCCOC(CNC(=O)C(C)C2(O)CCC2)C1 N1(C(C(C)c2ccsn2)=O)CCCN(C(c2ncccc2Cl)=O)CCC1 C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(c2sc(CC)nc2C)=O)CC1O Cc1snnc1C(=O)NC(C1CC1NC(C1(N2CCCC2)CCC1)=O)C c1(C(N(C2C(C)CCN(C(CCC=CC)=O)C2)C)=O)cccc2c(C)ccnc12 Cc1ccc(F)c2[nH]c(C(=O)NC3CN(C(c4nnsc4Cl)=O)CCC3C)cc12 C=CC1(C(=O)NCC2(C)CCC(=O)N2C)CCN(C(=O)C2CC2)C1 CN1CCCC(CNC(C2C=CCN(C(=O)C=Cc3ccncc3)C2)=O)C1 Nc1cccc(CC(=O)NCC2CCCN2C(=O)C(C2CCC(=O)N2)O)c1N c1(CC)noc(CC)c1CC(=O)NCC(C1CC1)N(C)C(C1(C)CC(F)C1)=O N1(C(CCCC(C)C)=O)C2CCC1CC(NC(c1coc(Br)c1)=O)C2 C(=O)(C(CC(C)C)CC(C)C)N1CC(C)(CNC(CCOCCC)=O)OCC1 C12(C(=O)NC3CC(N(C(c4c(C)nc(C5CC5)[nH]4)=O)C)C3)CCCN1CCC2 CC1COCC(CC(=O)NCc2cc(C(=O)N(C)CCN3CCCC3=O)on2)O1 C1(CN(c2nnc(-c3cccc(O)n3)n2CCC#N)C)CCc2c[nH]nc2C1 c1(Cn2cc(CC3CN(CC4CC(C(C(CC)C)=O)C4)C3)nn2)cccc(Cl)c1 C12(C(=O)NC3(C(=O)NC4CCCC(C(=O)OC)C4)CC3)CCCC(C)(C1)OC2 N1(C(C(=Cc2cccnc2)C)=O)CC(NC(C2(C)C(C)(C)C2(C)C)=O)CC(C)C1 N1(C(c2c(NC)c(N)ccc2)=O)CC(NC(C2CCCN2C)=O)C2CCCCC12 c1(C(=O)NC(CNC(c2c(OCCC)cccn2)=O)C)ccc2ocnc2n1 c1(C(N(C)CC2(CNC(=O)Cn3cnnc3O)CCC2)=O)ccc(CSC)nc1 C(=O)(C1=NOC(C)(C)C1)NC(C)C(=O)NC(C)Cc1ccnn1C N1(C(CC2CC(CC)OCC2)=O)CCCC2(NC(=O)C(C3CC3)C3CC3)CC2C1 C1(C(N2CC(C(C(C)C)O)C2)=O)CCN(C(C2CC3CCC3C2)=O)CC1C c1(OC)cc(CC(=O)NC2CCCN(C(=O)C=C(Cl)Cl)CC2)cc(F)c1 c1(C(N2C(CNC(CC=C(C)C)=O)CCCC2)=O)cnc2ccnn2c1C c1(CN(C(=O)NC2CSC(C(F)(F)F)C2)CC)ccc(C)c(C#N)c1 N1(C(CCSCCNC(c2c(CC)nn[nH]2)=O)=O)CCC(C)C(CO)C1 N1(C(CCNC(COC)=O)=O)CC2(COC(CNC(=O)Cc3cnsc3)C2)C1 Cc1ccc(C(=O)NC(C2CN(C(=O)Cn3cnc(Br)c3)C2)C)s1 C1(CC#C)(C(=O)OCC(C2CCCCO2)=O)CCCN(C(=O)OC(C)(C)C)C1 n1(CC(C)C)[nH]c(CC(=O)N(C2CN(C(=O)C(F)C3CCOC3)C2)C)cc1=O C1(NC(c2ncccc2O)=O)CN(C(c2cnn(C3CC3(F)F)c2)=O)CC12CC2 CC1(NC(=O)CCC2CCCCC2)CCN(c2nnc(CC(F)(F)F)s2)CC1 CC1(C)C(NC(=O)CCc2cnn[nH]2)CC1CNC(c1ccc(Br)cn1)=O C1(NC(C(CC)C(C)C)=O)CC2(CCN(C(=O)C#CC3CCCO3)CC2)C1 c1(C(C)NCC(=O)N(CCc2ccc(OCC)cc2)CC)ccc(C#N)cc1 c1(C(N2CC(C)(CNC(CC=C)=O)CC2(C)C)=O)ccc2cncn2c1C C=CC(C)(CC)C(=O)NC1CCC1NC(=O)Cc1cccc(N2CCOCC2)c1 N1(C(c2[nH]cc(C)c2)=O)CCN(Cc2cnn(-c3cccc(C#N)c3)c2)C2CC12 N1(CCC)CCCC1C(N1CC(CNC(C2COCC2C(N)=O)=O)(OC)C1)=O C(=O)(C1=CCC(C)(C)CC1)NCC(C)C(F)C(=O)NCCS(C)(=N)=O CC1COc2c(C(N3CC4(CNCCO4)C3)=O)cccc21 c1(C(N2CC3C(NC(c4cn(C)nn4)=O)C(C3)C2)=O)cccc2nnn(C)c12 c1(C(=O)NC(C)CN2CCN(C(=O)C=C(Cl)Cl)CC2)cnc2[nH]cncc1-2 c1(C(N2CCC(C(=O)NCc3ccno3)C2)=O)ccc(C(F)(F)F)cc1Br CCCCS(=O)(=O)Nc1cccnc1C(N1CCNC(C(=O)OCC)C1)=O c1(C(N2CCN(C(C(C(C)C)OC)=O)C(C)C2)=O)sc(S(N)(=O)=O)cc1C C1(C(N(CCN(C(C2C(=C)CC2)=O)C)C)=O)COCCC1C c1(NC(C2(CNC(CCCCCCC)=O)CC2)=O)ccc2cccnc2c1 C(C(=O)NN1CCCC1C(=O)NC(C)CN1CCCC1=O)SCCC C(=O)(CCCCCCCCC1CC1)NC1C(NC(C(C)(C)OCC)=O)CCC1 c1(-n2c(SCC(=C)C)nnn2)ccc(OCSc2nnn(C)c2C)cc1 N1(C(C2(C)CC(=C)C2)=O)CCC(NC(=O)CC2(C#N)CCC2)C(C)C1 C#CC1(C(=O)NCC2CC3CCC3C2)CCN(C(=O)C=C2CCCCC2)CC1 c1(OCC)cccc(CC(=O)N(CC(C)N(C(=O)C(C)CSC)C)C)c1 C1(CC(=O)OCC)CN(N2CC(c3ccccc3C)CC2C)CC2(CCC2)O1 O=C1CCCCC(C(N2CCCN(C(C3CCC(F)(F)C3)=O)CC2)=O)N1 C1(C(N2CCC(C(=O)NC3C(CN(C)C)C3)CC2)=O)CCC2(CC1)CC2 CC1(C)CC(CO)CCN1C(=O)CC(O)CNC(=O)CCc1cccnc1 CS(=O)C=CC(=O)N1CC(NC(C2(CF)CC(F)(F)C2)=O)C(CC2CC2)C1 c1(C(CNC(COCC(=O)NC)=O)NC(C2CC3CCC2C3)=O)cccc(Cl)c1 C(=O)(CC1CCOc2ccccc21)N1CC(O)CC(NC(CN(C)C(N)=O)=O)C1 C(=O)(CC(O)CC)N(CCC(=O)N(C1CCN(C)C1)C)CC=C N1(C(=O)OC)CCC(N(C(=O)C=CC(C)=O)C2CC2)CC1C c1(NCc2nnc(C)n2C)[nH]c(=NC2CCCN3CCCCC23)nc2sccc12 N1(C(c2c(C)con2)=O)CCC2(CC1)COC(CNC(c1cc(Br)n[nH]1)=O)C2 CCCC(C#N)C(=O)NCC(C)(CC)NC(=O)C=CCN1CCOCC1 N1(C(c2n(CC)nc(C)c2)=O)CC2CCC2(NC(c2ccoc2Cl)=O)C1 C(=O)(C(CCOCCO)NC(=O)C(C)C(=O)OC)NC(C(=O)OC)C1CCC1 c1(C(C)NC(c2cc(CC)nn2C)=O)cc(F)cc(F)c1F c1(C(=O)NCC2(F)CCN(C(COCCOC)=O)C2)ccc2nn[nH]c2c1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1C C(=O)(CC(C)(C)C)NC(C(C)C)C.C12CCN(CC1)C(=O)C1CC1C(=O)N2 CC(C)C(CNC(c1csc(CO)n1)=O)C(=O)N1CC(C(N)=O)C(C)C1 c1(C(CNS(CC2(C)CCNC2)(=O)=O)CC2CCCC2)ccc(Cl)c(Cl)c1 C1(C(C)NC(c2ccno2)=O)CCN(C(c2ccc(OCCO)cc2)=O)CC1 C(=O)(C(CCCC=C)NC(=O)C(C1CCC1)OCC)NCC(CC#C)(C)CO c1(C(N(c2ccnc(-c3cn(CCCC)nn3)c2C)CC)=O)c(F)cc(Cl)cc1Cl C1(SC)CN(C(c2ccc(C(F)F)cc2)=O)CC1NC(c1cc(C#N)c[nH]1)=O N1(C(CN2C(C)CCCC2)=O)CC2(CC(NC(=O)C(C)C(F)F)C2)C1 C1(CNC(C(CCC)F)=O)CCCCN(C(=O)CCOC(C)C)C1 C=CCC(CC(=O)N(C1CCOCCC1O)C)NC(c1[nH]ccc1C)=O c1(CC(=O)NC2C(CNC(C(COC)C)=O)CCC2)ccc2c(c1)CCN2C c1(N(CC=Cc2cc[nH]c2)CC2CN(C(C)C)C2)n[nH]cc1-c1nn[nH]n1 C(=O)(C1=CC2(CN(C(=O)C(C)C3CCOC3)C2)OC1)Nc1cncc(COC)c1 N1(C(CCOCCN(C)C)=O)CC2C(CNC(C3(O)CCC3)=O)C2C1 C1(OCC)COCC1N=c1[nH]c(=NC(C)CC2CCCCC2)[nH]c2c1CSC2 CCN=c1cc(-c2nc(CC(C)OC)n(-c3ccc(C(F)(F)F)cc3)n2)cc[nH]1 CC(C)C(C(=O)NCC(CNC(C12CCCC1(C(N)=O)C2)=O)C(F)(F)F)C(C)C C1(CNC(C(COC)O)=O)CCCC2(CN(C(=O)Cc3ccc(C)c(C)c3)C2)O1 C=CCCC1C(=O)N2CCOCC2N(CC)CC(F)C(=O)N1.C(C)SC C1(NC(=NCCCSCC)NCCSS(C)(=O)=O)C(=O)N(C)CCC1C CC1CC(N=c2c([N+](=O)[O-])c[nH]c3ccc(Cl)cc23)CCN1C(C1CCC1)=O c1(-n2cc(C(CCC)NC(c3ccccc3C(F)F)=O)nn2)cc(F)ccc1C C1(C(N(C2CCCN(C(c3nn(C)cc3CC)=O)C2)CC#C)=O)CC2CC(=O)C1O2 Cc1cc(C(=O)NCCOCC(=O)NCc2cc(C#N)c[nH]2)n(C)n1 N1(C(C(COCC)C)=O)CC2CCC2(C(=O)NCC2(CCOC)CC2)C1 N1(C(c2nc(CC)sc2)=O)CCN(C(c2ncccc2C(C)=O)=O)CC1C N1(C(C(CC=CC)C)=O)CCC(NC(=O)C2=CCOC2)C1(C)C C1(CC)CC(C)N(c2nnc(-c3cncs3)n2CC2(CO)CC2)C1 CC(F)(C(=O)NCCC1CN(C(=O)CCCc2ccccn2)C1)C(F)(F)F c1(C(N2CC(C)C(NC(c3cncc4sccc34)=O)C2)=O)n[nH]c2c1CC1CC21 C1(NC(Cn2c(C)cnc2)=O)CCC(NC(=O)COCCN(C)C)CC1 C1(C(=O)NCCC2N(C(c3c(C)nc(C)[nH]3)=O)CCSC2)OCC2CCCCC12 N1(C(CCCNC(CC)=O)=O)CC(OC)CC(NC(c2cc(C)sc2C)=O)C1 Cc1csc(C(=O)NC2CCC2NC(C23C=CC(CC2)C3)=O)c1Cl CC1CN(C(C2CCCC(F)(F)C2)=O)CCN1C(=O)CN1C(=O)CN(C)C1=O CC1(C)OC(=O)C(CC(=O)NC2CC(NC(=O)CSc3nncs3)C2(C)C)O1 C12(OC)CCCCC(C(=O)NCCNC(=O)C3=CCC(C)CC3)(C1)C2 c1(CC(N2CC(CCNC(CC3CN(C)C3)=O)C2)=O)cc(Br)cs1 c1(C(C)OC)nc(C)c(C(=O)NCCNC(C2CCSCC2)=O)s1 c1(C(=O)NC(CC)CNC(c2cccnn2)=O)ccc2nc[nH]c2c1F N1(C(C(C)(C)OCCC)=O)CC2CC2(NC(=O)CC)C1.C12CC(C1)S2 N1(CC(CN(C)C(=O)OC(C)(C)C)O)CCN(c2ccccc2)CC1.C1CO1 N1(CC)CCCC(C(=O)NC(C)(CO)C(=O)N(CC(C2CCCC2)O)C)C1 C(=O)(C1=COCCO1)N1CC(C(C)NC(=O)C2=COCC2)C1 c1(NCCC(O)C2CC2)cccc(-n2ncc(-c3nn[nH]n3)c2Br)c1 N1(C(C2C(NC(c3csc(Cl)n3)=O)CC2)=O)CCOC(CCF)C1 C1(C(=O)NCC2=CCN(C(C3C(C)(CC)C3)=O)CC2)CC(c2cccnc2)=NO1 C=CCCCCC(=O)N1CCCC(NC(C2CCCC2F)=O)CC1 C1(NC(c2ccc(C3CC3)o2)=O)CN(C(C2CC3CCC2O3)=O)CC2(CC2)C1 C(=O)(CC(C)C(F)F)NCC(CNC(CCc1c(OCC)cccc1)=O)CO C(C(COC)C(=O)N1CC(F)CC1Cn1cc(C2OCCO2)nn1)OC C(=O)(N=c1cccn[nH]1)C12C(CN(C(c3ccc(COC)cc3)=O)C1)CC2 Cc1cccc(CC(N2CCC(NC(=O)CC3CCCCC3F)CC2)=O)c1F C12(C(=O)NCC3C(NC(C(C)(C)C)=O)C3)CCC(C(F)F)(CC1)C2 C1(O)(CNC(C2C3(CC3)C23CC3)=O)CCN(C(C2CCOC2=O)=O)CC1 C1(C#N)(N(C(CSCCNC(c2cn(CC)nc2)=O)=O)C)CCOCC1 C(CC1CC1)(C(=O)NCC1CC(NC(=O)C=CC2CCCC2)C1)OC C(=O)(C(CNC(C1(n2cnnn2)CC1)=O)C(C)C)NCC1(OC)CC1 CC(C(CO)NC(C1(C2CCCCO2)CC1)=O)NC(=O)CC(C)c1ccncc1 C12(NC(c3cc(F)c[nH]3)=O)CCCCC1CN(C(C1CC3C=CC1C31CC1)=O)C2 c1(C(=O)OCC)sc(C(=O)NCCC(O)CNC(C2CC2F)=O)c2c1CCCC2 C1(N(C(c2scc(C)c2C)=O)C)CN(C(C23COCC(C2)C3)=O)CC1(C)C c1(C(=O)NCC2C(NC(c3c(C)snc3)=O)C2)cccnc1Oc1ccccc1 n1(C(C)C)ncc(C(=O)NCC2C3CN(C(=O)Cc4conc4C)CC23)c1N c1(NC(c2ccnc(-c3cccc([N+](=O)[O-])c3)c2)=O)c(F)cc(F)cc1[N+](=O)[O-] C(N=c1cc(CCC2CCCC2)nc[nH]1)C1CS(=O)(=O)CC1O C1(NC(CCCOCCOC)=O)CN(C(c2csc(Cl)c2)=O)CC1n1ccnn1 C12(CNC(c3coc(C4CC4)n3)=O)CCC1CN(C(c1cc(Br)co1)=O)C2 c1(-c2c(C(=O)Nc3ccc(C(=O)OC)s3)ccnc2)ccnc(OC)c1F C1(CNC(C2(CCC)CCC2)=O)CCN(C(=O)CCC=CBr)CC1C CS(=O)(=O)C1(C(N2CCCOC(CNC(c3c(O)cccc3O)=O)C2)=O)CCC1 c1(C(N(CCN(C(C(C)(CO)OC)=O)C)C)=O)cc(C)c2sccc2c1 c1(CC(=O)NCC2(CNC(C3CC(=C)C3)=O)CC2)nnc(O)s1 N1(C(C(n2ccc(C(F)(F)F)n2)C)=O)CCC(N(CC(=O)NC2CCC2)C)CC1 C=CC(CC)CC(=O)NC1CCN(C(=O)CNC(c2c(F)cccc2Cl)=O)C1 C(=O)(CCCN=[N+]=[N-])NC1(C(N(CC(C)C(F)(F)F)C)=O)CSC1 N12CCC(C(O)C1)C2=O.c1(OCC)ccc(CNCC23CC(CO)(C2)C3)cn1 c1(C(=O)NC2CN(C(c3n(C)cnc3)=O)CC3C2C3)cc(S(C)(=O)=O)ccc1O CCCCC(CC)CC(=O)NC(C)(C)CN1CCC1.C1=CCNC1=O c1(-c2nc(CCN(C)C)nn2C2CCS(=O)(=O)C2)ccn2cnnc2c1 N1(C(=O)Nc2ncc(OC)s2)CC(C)SC(C)C1 N1(C(CC(CNC(C2CC=CC2)=O)OC)=O)CC2(CCC(=O)NC2)C1 c1(C(N2CC(C(C(=O)N(C3(OC)CCCC3)C)OC(C)C)C2)=O)cccc(F)c1 Cc1cccc(Cl)c1CC(=O)NCCC1CN(C(C2CCN(C)C2=O)=O)CCO1 C=C=CCC(=O)NC(C)CCNC(C1CCC(C(F)(F)F)C1)=O C#CC1(C(=O)NCC2CCCN2C(=O)C=CC(=O)OC(C)(C)C)CCC1 O=C(CC(O)COCc1ccccc1)NCCNC(C1CCNC1=O)=O C=CCCCCCCC(=O)N1CCCC(CN(C(=O)C(C)(Cl)Cl)CC)C1 c1(C(N2CC(F)(CNC(c3c(COC)ccs3)=O)C2)=O)cccc(Cl)c1Cl N1(C(c2cc(=N)[nH]cc2)=O)CC2CCN(C(=O)CCc3cnoc3)CCC2C1 C(C(CC(C)C)NC(c1csnc1Br)=O)NC(C1(OC(C)=O)CC1)=O C(=O)(CCCC(=O)NCC(CO)NC(=O)C(CCC)c1ccccc1)OCC C1(CC=C)(NC(=O)Cn2cccn2)CCN(C(C2CC2(F)F)=O)CC1 CC(C)CCC(O)C(=O)N1CC=CCC1C(N1CCN2CCCC2C1)=O c1(NC(CC2CCN(C(C=CCC)=O)C2)=O)c(C)nn(CC)c1C C(Cc1ccccc1)(CCNC(C1(Cl)CC1)=O)NC(c1cncnc1)=O Cc1nc(N2CCC(NC(=O)CC3COCCO3)C(C)C2)cc(Cl)n1 C1(COC)(CNC(C2CS(=O)(=O)C2)=O)CCCN1c1cncc(Cl)n1 Cc1ccccc1-c1cn(C(C)CN(C(=O)CCN2CCCC2)C2CCC2)nn1 CC(CCC(C)(C)C)C(=O)NC1(C(=O)NC2CCn3cncc3C2)CC(F)C1 N1(C(CCN(C)CCO)=O)CCCC(C2CCN(C(=O)C(C)(C)CN(C)C)C2)C1 Cn1nc(Br)c2ccc(C(N3CC(F)CC3C(=O)NC(C3CC3)C3CC3)=O)cc12 N1(C(c2c(C)c(Cl)cnc2)=O)CC2CN(C(=O)CC(O)CCN(C)C)CC2(C)C1 Cn1ccc2ccc(C(N3CCCC3CNCc3cncc(O)c3)=O)cc12 C1(C(N2CC(NC(Cc3cc(C)no3)=O)C(C#N)C2)=O)CCc2nc[nH]c2C1 CCC(CNC(C1(F)CCN(C(=O)CC2CCC(C)(C)C2)C1)=O)C(C)(F)F C(=O)(CCCCCO)NCCCCC(C)NC(C=CC)=O c1(CNC(C2CCC(N(C)C)C2)=O)ccc(CNC2N(C(C)=O)CCC2)c(F)c1 C#CC1CN(C(=O)CCN(C(=O)C(CN(C)C)N(C)C)C)CCN1C C1(NC(C(CC)C)=O)CCCN(C(=O)C=Cc2ccc(SC(F)F)cc2)CCC1 C(CCCC(C)(C)C(=O)NNC(=O)C1CCCCCC1)NC(C(C)C(C)(C)C)=O c1(C(=O)NCC2OCCCN(C(c3ncc(C)cn3)=O)C2)cnc(O)n(C)c1=O C1(C(N(CCCn2cc(-c3cn[nH]c3)nn2)C)=O)CC(F)(F)CCC1(C)C C1(NC23CC(C2)CCCCn2c3nnn2)CC(O)C(O)C1.C(C)(C)(C)S.CO N1(C(CC(CCC)O)=O)CC2CC(C1)N(Cc1nn(C)c(=O)n1C)C2 N1(C(C(C=CC)O)=O)CCN(C(=O)CC(C)(C)C2CC2)CC1CF c1(CC)cc(C(N2CCCC(CC(N3CCC3C(=O)NC)=O)C2)=O)ncn1 O=S(=O)(CCc1ccncc1)NCCC1(c2ccccc2)CCCO1 c1(OC)cccc(O)c1C(N1CCN(C(c2cc(C)c(C)o2)=O)C(C(C)C)C1)=O Cc1cc(O)cc(Cl)c1C(=O)NCC(O)COc1ccc(C2CCC(=O)N2)cc1 N1(C(CCOCC)=O)CC(NC(c2cnc(N(C)C)s2)=O)CC(C)C1 c1(OCC)cc(F)ccc1C(N1CCCC(O)(c2cn(C(C)C(C)O)nn2)C1)=O C(=O)(C(F)CC(C)(C)C)NC1CC(CCNC(c2c(C)n(C)nn2)=O)C1 Cc1nnc2ccc(C(N3C4CCC3C3CC3(NC(C3CC3(F)Cl)=O)C4)=O)cn12 CC1CNCC(CC(=O)NC(=O)CC(c2ccc(Cl)cc2)C2CC2)O1 c1(C(N(CCC)Cc2cccc(Cl)c2)=O)cnc2ccccc2c1C C1(C(N2CCCC(SC)C2)=O)C2CC3C(C2NC(=O)C(C)CC2CCCC2)C13 C1(NC(c2nccc(OC)c2OC)=O)C(C)CN(C(c2cnc(O)o2)=O)CC1C C1(NC(c2c(C)ccc(-c3ccncc3)c2)=O)CC(C)(C)OC(C)(C)C1 N1(C(CC2(C)CC2(F)F)=O)CC(NC(c2ccc(Cl)c(O)c2)=O)CC12CCC2 c1(C(=O)NC(CC=C)CNC(c2coc(COC)n2)=O)ccc(C)c([N+](=O)[O-])c1 c1(C(N2CCC(NC(CNC(=O)NC)=O)C2)=O)ccc(C(C)(C)C)cn1 c1(COC)nc(=NC(=O)c2ccc(C(C)(C)S(C)(=O)=O)cc2)o[nH]1 C(=O)(C1c2ccccc2C1)NCCCN(C(C1CCC(C)(C)C1)=O)CC c1(OC)ccc(Cl)c(C(=O)NCC(C)CNC(c2nc(C)ccc2C)=O)c1F n1(C(C)C)ncc2c(NC(c3cnn(C)c3)C)[nH]c(=NC3CC=CC3)nc12 N1(C(CC(C)F)=O)CCc2c(c(CNC(C3CC3F)=O)nn2C)C1 C1(C(=O)NC(CNC(CC2C(SC)C2C)=O)CC(C)C)CCc2nnc(O)n2C1 c1(CC(=O)NCCCCC(C)NC(=O)C(F)=CC2CC2)ccc2oc(O)nc2c1 c1(C(=O)NC2CC(CNC(=O)C(F)n3cccn3)C2)cccn2nncc12 C(=O)(CC1CC(C(C)C)c2ccccc21)N1CCC(NC(CCC#C)=O)C(O)C1 c1(C(=O)OC)ccc2nc(NC(c3ccc(Cl)cc3Cl)=O)[nH]c2c1 Nc1ccc2nc(N3CCCC(CO)(NC(=O)C=Cc4ccccn4)C3)sc2c1 c1(C(=O)NCC2(CNC(CSCC(C)C)=O)CC(F)(F)C2)cc(S(N)(=O)=O)c[nH]1 N1(C(CCCN(C(C)=O)C)=O)CCC(NC(=O)CN2CC(C)C2)C2(CCC2)C1 C(=O)(C(C)CC(F)F)NC(C(=O)NCc1ccc(C)cc1)C1CCC1 N(C1c2cc(F)ccc2CCC1C)Cc1c(C)nc[nH]1 c1(CCC)c(C(=O)OCCCC2CCOC2)cnn1C N1(C(C(CC)(C)O)=O)CCC(O)(CCCNC(C2CN(C(C)=O)CCO2)=O)CC1 N1(C(c2c(C)cns2)=O)C2CCC1C(CNC(c1cnncc1C(F)(F)F)=O)C2 CC(=O)CCN=C(NCc1nnc(-c2ccccc2)s1)NC1CCN(C(C)=O)C1 c1(C(=O)NCC2C(NC(CC3(OC)CCCCC3)=O)C2)c(F)ccc2[nH]ccc12 c1(C(=O)NCC2C(NC(CC(C)(C)c3cccs3)=O)CCC2)cnc2n1CCS2 N1(C(CC(C)C)=O)CCC2(CC2C(N2CCN(c3ccc(Cl)nn3)CC2)=O)C1 C1(NC(CNC(C(COC)(F)F)=O)=O)COCC1C1CC1 CC(C)(CC(=O)N1CC(C2(NC(=O)CCc3ccc(F)nc3)CC2)C1)C(F)F c1(C(N(CC(CNC(C2C(C(C)C)OCC2)=O)O)C)=O)cnc2c[nH]nc2c1 c1(C(N2CC(NC(c3cnn(CCF)c3)=O)C3(C2)CC3)=O)cnn2ccccc12 CC(C)CC(CNC(=O)Cn1nccn1)C(=O)NC(CN(C)C)CCO Cc1cc(C(N2CCC(C)C2CNC(c2cc[nH]c3nccc2-3)=O)=O)c(O)cc1F S(=O)(=O)(c1cnc(NC2CC=CCC2)c(Cl)c1)N(CCCCOC(C)(C)C)C c1(CNC(C(CCOCCO)NC(CC(CC)C)=O)=O)cc(C)nc(C)c1 CN1CC(CCNC(C2(C)CCN(C(C3CCN3C)=O)C2)=O)CC1=O C1(NC(c2c(SC)ccs2)=O)CN(C(=O)C(O)CC(F)F)Cc2ccnn2C1 N1(C(C)=O)CC(C)(C)OCC1CNS(CC(=O)NC1CC(CSC2CC2)C1)(=O)=O c1(NC(c2c(F)cccc2F)C)ccc(S(=O)(=O)NC2CC2C2CCC2)cc1F CC(CCC(=O)N1CC2C(N(C)C)C2C1)NC(=O)C(c1cccn1C)=O c1(C(Cc2c(C)non2)C)nc(CCN(C)C)nn1-c1ccn(C)n1 Cc1c(Br)c(C(=O)N(C)CC2(O)CN(C(=O)C3=CC(C)(C)C3)C2)nn1C C(=O)(C1CCCc2ncc(C)n21)NC(C1CCCC1)CNC(CNC(C)=O)=O c1(C(=O)NCCCN(C(c2ccsc2Br)=O)CC)c[nH]c(=O)cn1 c1(CCCCOC(C)=O)cn(CC(O)CNC(=O)Cc2ccccc2)nn1 c1(C(N2CCC(N(C(c3ncn(CC)c3)=O)C)C2)=O)ccc(=O)n2c1CCCC2 N1(C(C(C)OCC)=O)CCC(C(C)NC(C2(C(=O)NC)CCC2)=O)C1 C1(C(=O)NC(COC(C)=O)CO)CC2(CCN(C(c3c(C)ncn3OC)=O)C2)C1 C1(C(N2CC(C#N)C(NC(C3(Br)CCC3)=O)C2)=O)Cc2ccccc2O1 Cc1ccc(F)c(C(N2CCSCC2C(=O)NC2CC(n3ccnc3)C2)=O)n1 N1(C(C2(CC=C)CCC2)=O)C2CCC1CC(CNC(C1C=CCC1)=O)C2 c1(OC)c(C(=O)N(C)CC2CCCN(C(C3(Cl)CC3(C)C)=O)C2)nc(O)nc1O C(=O)(C(C)(C)C1=CCSCC1)NC(C(C)NC(C1CCOC(C)(C)C1)=O)CO c1(C(=O)NCC2(NC(c3cnsn3)=O)CCC2)ncc(C(F)(F)F)s1 C1(OC)CN(C(=O)C=CC(=O)OC(C)(C)C)CC1C(N1CC(O)CC1C1CC1)=O C(=O)(C(C)C(=O)N1CCCC1CN(C)C(c1csc(-c2cnccn2)n1)=O)OC c1(N(C)Cc2ccc(OC(C)C)cc2)cccc(S(=O)(=O)N2CCS(=O)CC2)n1 C(C)(CCCN=c1[nH]cc(C#N)cc1C)NC(C(C)OCC)=O Cc1cc(O)cc(C)c1C(=O)NCC1CCN(C(=O)Cc2nc[nH]n2)C1(C)C N1(C(C(C)S(C)(=O)=O)=O)CCC2C(CCCN2C(=O)CCCC(N)=O)C1 C1(C2N(C(c3ccc(CC)s3)=O)CCC2)CCN(C(c2ccc(O)nn2)=O)CC1 C1(C(=O)NCCN(C(c2ccc(C3CC3)nc2O)=O)CC)CN2CCN1CC2C N1(C(C=CCC(C)(C)NC(C(C(C)C)C2CCC2)=O)=O)CC(O)CCC1C C12CCC(CC1)CNC2=O.C(CCCCNC(C1CC1Cl)=O)=CC(C)C C(=O)(C(C)(C)C(F)F)NC(C(C(=O)N1C(C(C(=O)OC)(C)C)CCC1)C)C C1(C#N)(C(=O)NC2(C(N(C)CCC3CCCO3)=O)CCC2)CCC1 C(=O)(C1=Cc2ccccc2OC1)N1C2CCC(NC(C(N)=O)=O)(CC2)C1 C(CC(=O)NCCn1ccnc1)(C(F)F)N(C)C(c1cc[n+]([O-])cc1)=O C1(CC)CCCCC1NC(c1c(CNC(=O)C=Cc2ncc[nH]2)cnn1C)=O C(=O)(C1=CCC(C)(C)CC1)NC1CCCN(C(Cc2cnc(C)s2)=O)C1 n1(C(CC)(C)C)nnnc1C(c1conc1C1CC1)NCC1CC1c1ccccc1 c1(C(=O)NCC2C(NC(c3cnn(C)c3Cl)=O)CCC2)cccc(F)c1Cl C(C(CCO)NC(c1cnn(CCNC(C2CC2C#N)=O)c1)=O)OC C1(N(C(CC(C)c2ccco2)=O)C)CCN(C(=O)CN2CCCS2(=O)=O)CC12CC2 N1(C(C2C(C(=O)OC)C2)=O)CCC2CCCC(C1)N2c1nc(C)cc(C#N)n1 C1(C)(C(N2CCC(CCNC(c3cc(COC)no3)=O)CC2)=O)CCC(O)CC1 C1(C(=O)NCCc2nc(C)sc2)C2CCN(C(c3cc4n(n3)CCO4)=O)CC12 C1(C(N(CC(=C)C)C)=O)C(O)CCN1C(=O)COCCF C1(CCNC(C2CC(NC(c3ccc(C4CC4)o3)=O)C2)=O)CCCCCC1 c1(C(=O)NC2(C)CC(NC(c3cnco3)=O)C2)cncc2cccnc12 C1(CC#C)(C(=O)NCC2CCOC2)CCN(C(=O)C(F)n2ccnc2)C1 C1(CN(c2ccncn2)C(C2CCCNC2)C)CCC(F)CC1 Cc1nc(C)c(C(=O)N(C)CC2(O)CCN(C(c3csc(C(F)F)n3)=O)C2)o1 C(C)(CC(C(=O)Nc1nnn(C)n1)N(Cc1cc(C)ccc1F)CC1CC1)SC N1(C(c2n(C)nnc2CNC(=O)CN(C)C)=O)CCCC[Si](C)(C)C1 N1(C(C2OCCCO2)=O)CCn2nccc21 CC1CN(C(C2CCN3CCC2C3)=O)CCCN1C(c1ccc(F)c(F)c1)=O CC(C)(CNC(=O)CO)CNC(=O)CCNC(C1CCCC1)=O C1(C(N2CCCC(CC)(NC(c3csc(=N)[nH]3)=O)C2)=O)CC2(C1)CC(C)(C)C2 O=C(CS(=O)(=O)c1ccc(Cl)cc1)NC1CN(C(C2CSC2)=O)CC1O N1(C(c2ccc(COC)o2)=O)CCCC(CN(C(=O)CCC(=O)OC)C)C1 C(CC1CC1)(C(=O)NCCCN(C)C(C1CC2CC2C1)=O)OC N1(C(Cc2cc(C)sc2)=O)CC2CC1CN2C(C1(n2cccc2)CCCC1)=O C(C#Cc1ccccc1F)N(C(=O)CCc1ccc(F)cc1Br)CCOC C(=O)(C=C1SCC(=O)N1C)NCC1CCCN(C(C2CC(C(=O)OC)C2)=O)C1 N1(C(C(C)CO)=O)CCC2(C=C(C(=O)NCC3CCC3(F)F)C2)C1 C1(NC(c2ccc(CC)cn2)=O)CN(C(c2[nH]nnc2C2CC2)=O)CC1C1CC1 C1(C(=O)NC2CC(=C)C2)CCN(C(=O)Cc2occc2C)C1 c1(NCC)ncc(C(=O)NC(CCN(C(=O)CCNC(N)=O)C)C(C)C)cc1Cl c1(C(=O)OC)cnc2nc(NC(c3cccc(O)c3OC)=O)ccc2c1 C(=O)(C1CCNc2ccccc21)NC(CC(C)C)CNC(c1nccnc1N)=O C1(C(N2C(CNC(C3CC(C)C3)=O)CC(O)C2)=O)CN(CP(C)(C)=O)C1 C=CCCCC(=O)N1CCCC(N(C(=O)Cc2csc(C(=O)OC)c2)C)C1 c1(C(=O)NCCCC2N(C(c3cnn(CC)n3)=O)CCCC2)cccc(C)c1C c1(C(N2CCC(CNC(Cc3cc(C)no3)=O)C(O)C2)=O)ccc2nccn2n1 c1(C(C(N2CCC(NC(C=CCCC=C(C)C)=O)C2)=O)=O)ccc(F)cc1 CC1OC2(C(=O)NCCCC(C)NC(=O)COCC(C)(C)C)CC1C2 C1(C(NNC(c2c(OC)c(Br)ccc2)=O)=O)CCc2nccn2CC1 N1(C(CNS(C)(=O)=O)=O)Cc2ccccc2OC2(C1)CN(C(=O)CSCCF)C2 N1(C(c2c(C)nc(C(C)C)nc2)=O)CC(N=c2[nH]c(Cl)ncc2C(N)=O)CC1C c1(CC(=O)NCC(CCCC)NC(=O)CCS(C)(=O)=O)cc2ccccc2s1 C(=O)(CC1=CCCCC1)NC1C(C)CCN(C(c2c(C)oc(C)c2Br)=O)C1 N1(C(c2c(OC)cc(C)cc2)=O)CC2CCC(NC(=O)C(C)(C)C(=O)NC)C2C1 C(=O)(C1=NN(CCO)C(=O)CC1)N(C1C2CN(C(C(C)C)=O)CC21)C C1(CCC(C)C)(CC)CCCN1C(=O)OCC1(C#N)COC1 C12(C(N3CC4C(NC(C5CCN(C)C5=O)=O)(C4)C3)=O)C3CCC(CC13)C2(F)F c1(C(N2CC(SC)C(n3cc(CC4(O)CCC4)nn3)C2)=O)cc(C)c(F)cc1Br C(=O)(CCCCO)N1CCCC(N(C(c2ccc(Cn3ccnn3)o2)=O)CC)C1 C1(C(=O)NC(CC(C)NC(C#CC(C)C)=O)C)CCCCC1(F)F N1(CC(=O)NC2C3CCN(C(C(C)C4CCC4)=O)C32)CCCCCCC1=O C(C(C)(C)OCC(=O)OC)OC(C1(CC)CC1)=O C1(C(N2CC(CCNC(c3ccc(C(N)=O)nc3)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C(CCSC)O)=O)C2CCC(C2)C1CNC(=O)CSc1cccc(Cl)c1 c1(NC(C=C(C)CNC(=O)CCc2nc(O)n[nH]2)=O)ccsc1C c1(C(=O)NCc2c(CNC(=O)CCF)cccc2)cccc(=S)n1O C1(CNC(C2OCCN(C)C2)=O)CCC12CCN(C(=O)CCC#N)CC2 C1(C)(C(=O)NC2CN(C(CN(C(=O)C3CC3)C3CC3)=O)C2)CC(C#N)C1 N1(C(c2n(C)cc(I)c2)=O)CCC(NC(=O)CC(F)F)C1(C)C N1(CC(=O)O)CCCN(C(c2c(O)cccc2Br)=O)CC1 c1(NC(=O)Nc2ncc(NC(c3ccc(Cl)cc3)=O)s2)ccc(Cl)cc1Cl C1(CC)CN(C(C2(CC)CCC2)=O)CC1C(=O)NCC12CSCC1C2 N1(C(CCC2CCCN(C(c3cnn(C)c3N)=O)C2)=O)Cc2ccncc2C1 C(=O)(C(C(C)C)C(C)C)Oc1ccc(C)cc1.c12cccc(Cl)c1Cn1cc-2nn1 N12CC(C(O)C1)CNC(=O)C2=O.CC1(C)CC1(C)COC(=O)OC(C)(C)C c1(C(N2CCC(n3cc(Cn4ncccc4=O)nn3)C2)=O)cc2cnccc2[nH]1 C1(OC)CN(C(=O)C=CC2CCOC2)CCC1NC(c1cccc(OC)c1C)=O CN1CCC(N(C(=O)C(C2CC2)N(C(=O)Cc2ccc(F)cc2)C)C2CC2)C1=O c1(CNC(C(C)=C2CCCC2)=O)ccc(C(=O)NCc2ccco2)cc1 c1(C(N2CC(CNC(c3csnn3)=O)C(O)C2)=O)cc(F)cc2cnccc12 C1(N(C(=O)NC(C)C(C)n2cccn2)C)CCC(C)(C)C1 N1(C(C(CC=C)CC)=O)CCCC(C)(C)C1CNC(c1ccc(F)o1)=O c1(CN(C)C)ccccc1CNC(c1ccc(CCN2CCCC2=O)cc1)=O c1(C(N(CC(CC)NC(c2c[nH]c(C(N)=O)c2)=O)C)=O)ncc(C)cc1C c1(C(=O)NCC(C)(C)NC(C(C(C)C)c2cnc(C)s2)=O)nccn2nccc12 C1(C(=O)NCC(CC)(C)NC(=O)C(C)Cc2ccncc2)CC=CC(O)C1 CCCC(C(=O)OC)C(=O)NCC1CC(F)CN1C(=O)CC1CCC(=O)NC1=O Cc1conc1CCNC(c1nc(CC(F)(F)F)cs1)c1nnnn1CCC1CC1 C(C1CCOCC1)=CC(=O)NC(C=CC(=O)NC1CCN(CC)C1)C CCC(COC)C(=O)N1CC(NC(c2sc(Cl)cc2Br)=O)C(O)C1 CCC(C(=O)NCc1ccc(C(F)(F)C(F)(F)F)s1)C(C)O C(=O)(C1Cc2ccc(F)cc21)N1CC(CCNC(C2CCCC(O)C2)=O)C1 CC1CCN(c2ccc(CNC(C3CC(O)C3)=O)cn2)CC1 C1(C(=O)NC(CC)CNC(C2CCC(C)(C)CO2)=O)CCC2(CCCC2)CC1 C(C(C(=O)N(C1CC(NC(c2cc(C(C)=O)[nH]n2)=O)C1)C)N(C)C)OC C(=O)(C(C)(C)CCC)N1CCC(CCOC)(NC(C2(CC#C)CCCCC2)=O)C1 N1(C(C(CC=C)(C)C)=O)Cc2occ(C(N3CC(=O)NC(CC)C3)=O)c2C1 c1(CCNC(C(c2ccc(OCC3CC3)cc2)N(C)C)=O)ccccc1Cl c1(CC(N2C(C3CCCN(C(C)=O)C3)CCC2)=O)sc(N(C)C2CC2)nc1C N1(C(C(c2c(C)noc2C)C)=O)CCC2(CCCN(C(=O)C3=CSCS3)C2)CC1 C1(C(N2CCC(C)(C(=O)OC)C2)C(=O)NCC(=C)C)CCCOCC1 c1(OC)c(C(=O)N(CCNC(=O)CN(C)CCO)C(C)C)cc(F)cc1F c1(NC(=O)NC2C(C)(C)CC2)nc2ccc(F)cc2s1 c1(OC)ccnc(O)c1C(=O)NC1CCC(N(C(=O)Cc2ncc(Cl)s2)C)C1 C1(NC(COCCOCC)=O)CCCCN(C(c2ccc(OC)cc2F)=O)C1 c1(C2CC(c3ccc(C)cc3)(O)C2)nn2cc(C)nc2s1 c1(CC)cc([N+](=O)[O-])ccc1Oc1ccc(C)c(NC2CN(C(=O)COC)C2)c1 C1(NC(c2c(C)n(C)cc2)=O)CCN(C(c2cnc(C3CC3)nc2O)=O)CC1C C1(C(=O)NCCn2ncc(C(N)=O)c2)CC(O)CN1C(c1scnc1Cl)=O N1(C(C(C=C)OC)=O)CCCC(O)(CCNC(c2cc(SC)n(C)n2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(c3ccccn3)=O)C2)cc2cc(F)ccc2o1 C1(C2CCOCC2)(C(N2CCC(CNC(CCCC=C)=O)CC2)=O)CC1(F)F CC1CCC(CC(=O)NCCNC(C2(C#N)CC=CC2)=O)CC1C c1(-c2ncc(C(N3CC(NC(CCCC)=O)C3)=O)s2)ccc(C)c(C)c1 N1(C(C2C(C)C2)=O)CCCC2(CCCN2C(=O)C(c2ccc(Cl)cc2)O)C1 N1(C(C)C(N)=O)CCC(C)(NC(=O)CC2C=CCC2)C1 N1(c2nc(N(CC(=C)Br)C)c3c(n2)n(C)cn3)CCc2sc(S(N)(=O)=O)cc2C1 C(=O)(C1=CC2(CCN(C(=O)C(CO)C(F)(F)F)C2)C1)N(CC(C1CCCC1)O)C N1(Cc2cccc(CCF)c2)CCC(C2(C3CCCN3)CC2)CC1 N1(C(C(C)OCC)=O)CCN(C(=O)CC2(OC)CCC2)C2CCCC12 CC(CNC(c1cn(CCNC(=O)C(C)(Cl)Cl)nn1)=O)S(N)(=O)=O c1(C(N2CC(NC(c3nccc(C)c3)=O)C(C#N)C2)=O)ccccc1S(C)(=O)=O c1(C(N2CC(CC=C)(NC(=O)Cc3cnns3)C2)=O)cc(N)cnc1C c1(CCC(=O)NC(CNC(C2CCC(COC)C2)=O)(C)C2CC2)cnn(C)c1C C1(COC)(NC(N2CCCC(CCNC(=O)OC(C)(C)C)C2)=O)CC(F)(F)C1 c1(N2CCC(N(C)C(c3ccc([N+](=O)[O-])s3)=O)C2)nc(Cl)nc2nc(Cl)n(C)c12 C(=O)(CC(O)CCCC)NC(C(N1CC2(CC(=C)C2)C1)=O)C1(C)CC1 N1(C(c2cc(C)ncc2C)=O)CC(F)(F)CC1(C)CNC(=O)CC(C)C1CC1 C1(F)(C(N2CCC(N(C(=O)CCOC3CC3)CC)C2)=O)CCS(=O)(=O)C1 C1(C(=O)NC(c2c(C)nccc2)C)CC1C1CN(C(=O)C(C2CC2)N(C)C)C1 c1(CC2(C(=O)NCC3CC3Cl)CN(Cc3cn(C)nc3)C2)ccc(F)cc1F N1(C(C(C(C)C)SC)=O)CCCN(C(c2ccc(C(F)(F)F)c(F)c2)=O)CCC1 c1(C(=O)NCC2N(C(C3(C=C)CCOCC3)=O)CC2)cccc2ccsc12 c1(C(=O)OC)c[nH][nH]c1=NC(=O)C(CNC(C1CNC(=O)C1)=O)Cc1ccccc1 C1(CC)(NC(c2nc(C)c(C)o2)c2nnnn2CC2CCOC2)CCCCCC1 C1(c2ccc(C)o2)C(C2CC2)CCN1C(=O)C(=O)NC1CC(C)S(=O)(=O)C1 C1(C(=O)NCCC2OCCN(C(c3c(COC)cco3)=O)C2)CCCCC1(F)F C1(OCC)(OCC)CC(C)(C(=O)NC23CC2CN(C(=O)C=Cc2cnc[nH]2)C3)C1 c1(C(=O)NC2C(C(=O)Nc3n(C)nc(Br)c3)C2)nc2ccccc2n(C)c1=O c1(C(N2C(C3(O)CN(C(CC(C)C4CC4)=O)C3)CCC2)=O)cc(Br)n(C)c1 C1(CNC(c2ccc(-c3ncon3)cc2)=O)CCCN(C(C2CCCOC2)=O)C1 c1(C(N2CC(NC(c3c(C)ccnc3)=O)C(CO)CC2)=O)cc(C)c(Cl)c(C)c1 c1(C(=O)NC2C(CNC(C(C)=C3CCCC3)=O)CCC2)c(C)nc2sc(C)cn12 C1(NC(C2CC2F)=O)CCN(C(c2cccnc2C2CC2)=O)CC1F c1(CC)cc(N)ccc1C(=O)NC1CC(NC(=O)Cc2cn(C)nn2)C1 N1(C(CCCCCN(C(=O)CCC2CC2)C)=O)CCC2(CNC(=O)N2)C1 C1(CN(CCNC2CC2)CC)Cc2ccccc2O1 C(=O)(C1=CCC(C)(C)CC1)N(CC(=O)OC)C.c1(=O)[nH][nH]c(=O)c2occc12 Cc1nc2ccccc2n(CCNC(=O)CN(C)C)c1=O C(CC(C)(C)C)(C(=O)N(CCC(C)NC(=O)C(c1cn(C)nc1C)O)C)OC C12(NC(C(C3CCC3)OC)=O)CC3CC(C1)CC(NC(=O)CCC(C)(C)F)(C3)C2 C1(CC)CN(C(=O)COCc2cc(C)no2)CCC1NC(=O)CCCn1cccc1 Cc1[nH]c(C(=O)NCCC2CCCCC2C)c(C)c1C(=O)Nc1sccc1Cl N1(C(C2N(C(CSC(C)(C)C)=O)CCCCC2)=O)CC(CO)C(C2CC2)C1 C1(NC(C(CN(C)C)N(C)C)=O)CC2C(NC(=O)CCc3ccsc3)C2C1 Cc1cccc2c(C(=O)N(CCOC)Cc3ccccc3)cccc12 N1(C(C2CCC(CC)C2)=O)CCC(CN(C)C(C2(CO)CC2)=O)CC1 c1(C(=O)N(CCCSC2CCCN2C(=O)Cc2cscn2)C2CC2)ncc[nH]c1=O N1(C(Cc2cn(C(C)C)nc2)=O)CCC(C)(NC(C2CCC(C)CC2)=O)C1 CC(C(=O)NCCCN(CCO)C(c1cc(Br)ccn1)=O)C(C)(F)F Cc1cc(C)n2nc(CC(N3CCC(NC(c4ccncc4)=O)C3)=O)nc2n1 N1(C(C)=O)CCCN(C(C2CCCC2CNC(=O)CCCSC)=O)CC1 c1(N(C)Cc2c(C)cco2)nc2c(c(=NC(C)c3nnnn3C)[nH]1)SCC2 C(=O)(C(CCS(C)=O)N(C)C)NC(CNC(c1c(C)nc(C)[nH]1)=O)C(C)C C(=O)(CC(C)CC(C)C)NCC(C1CCC1)NC(c1c(C)cno1)=O C1(N)CC12CCC(N)CC2.N1(CC(=O)C(C2(O)CC2)=O)CCN(C2CC2)C1=O c1(CC(N2CCC(N(C(=O)C(F)(F)c3nccn3C)C)C2)=O)ccc(O)c(F)c1 C1(OCC)C(N=c2[nH]c(=N)[nH]c(=NCc3cn4c(n3)CCCC4)[nH]2)CC1(C)C CCCCC(CC(=O)NCCCCCF)NC(c1ncccc1F)=O c1(NC(CSCC(C)C)=O)ncccc1N1CCCC1 c1(C(=O)Nc2scc(-c3cccc(CNC(C)=O)c3)n2)cc(I)ccc1Cl N1(C(C2CCN(C)C2=O)=O)CC(NC(c2cc(CO)ccc2Cl)=O)CC(C)(C)C1 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)CCC2CCCCO2)CC1C C(=O)(CCCC(=O)OC)NCCCCC(C)NC(c1cn(C)nc1C(F)F)=O c1(C(=O)NCC(C)CNC(c2ccncc2N=[N+]=[N-])=O)nc2n(c1Cl)CCCC2 c1(NC(C2CC(=C)CN2C(C2CCN(C)CC2)=O)=O)cc2[nH]ncc2cc1OC C1(C(=O)NC2C(CNC(CC(C)C3CC3)=O)CCCC2)CCC2(C(C)C)CC12 C1(C(N(CCNC(c2ccsc2Cl)=O)C2CC2)=O)COCCC1c1ccccc1 c1(C(=O)NCCCCN(C(C(CCC)O)=O)C)ccc(Cl)c2ccccc12 c1(C(N2CC(C(=O)NCCNC(C=C(C)C(C)C)=O)C2)=O)cn(CCO)nn1 c1(C(=O)NC(CC2CCCO2)C(=O)O)ccc(Br)cc1C(F)F C1(NC(c2ccc(SC)s2)=O)CN(C(c2cnc(C(C)(C)C)s2)=O)CCC1C C=CCC(C)(C)CC(=O)NCC1CN(C(c2cccc(=S)n2O)=O)C2(CCC2)C1 C1(CC#C)(C(=O)N(CC(C)N(C)C(c2ccn(CCC)n2)=O)C)CCOC1 c1(CC(=O)N(C2CCN(C(C3CCCC(F)C3)=O)C2)CC#C)ccccc1F c1(C(N2C(CC(N3CC(CCC)OCC3)=O)CC2)=O)cc(C)cc(O)c1 C1(C)(C(N2CC(C(=O)NOCC(N)=O)(COC)C2)=O)CC(O)CN1C C1(CNc2ccc(Nc3ccccc3)cc2)C2Cc3ccccc3C12 C1(CC(=O)N(CCCCNC(C2CCC2)=O)C)COCC(C)(C)O1 N1(C(c2cc(=N)[nH]cc2)=O)CC(NC(=O)Cc2cnns2)CC2(CCC2)C1 c1(CC(=O)NCC#CCNC(c2ccc(C)cc2)=O)cccc(Br)c1Cl CCCC(C)(C)CC(=O)NC1(CC(=O)NCC(c2ccccn2)C)CCC1 N1(C(C(=O)NCC2CC2)=O)CCCC(CNC(C2COC(=O)N2)=O)C1 C1(CN(C(=O)COCC2CCCO2)C)CCCN(C(=O)C(c2cnn(C)c2)O)C1 c1(C(=O)NC2CCCC2NC(C2CCC2(F)F)=O)cnc2c(F)cccc2c1 C(C(C(=O)NC(C)C(=O)NC(C)(C)C)NC(c1cc(C)c[nH]1)=O)OCC C1(NC(c2onc(C(C)(C)C)n2)=O)CN(C(=O)CC#N)C2CC12 CC1CN2CC1CC2=O.C1(C)(CCC(=O)NCCC23CCCC2C3)CC1(F)F c1(C(=O)NC2(CO)CCN(C(Cc3n(C)cnn3)=O)C2)ncnc2c1CCC2 c1(C(=O)NC(CNC(c2c(CC=C)cccc2)=O)C2CC2)cn2c(n1)CCCC2 Nc1cc(C(=O)NCC2CCC(NC(c3ccc(Cl)cc3Cl)=O)CC2)ncc1F C12(NC(c3cc4c(s3)COCC4)=O)CCCC1CN(C(c1cnn[nH]1)=O)C2 C(C1=NOC2CCCC12)NC(C(CCSC)NC(=O)CCc1cncnc1)=O C(=O)(CCCC(=O)N(C)C)NC(C(C)NC(c1cccc(N)c1)=O)C CN1CC(=O)NC(CC(=O)NC2COCCC2NC(=O)C(C)(C)O)C1=O C1(C(=O)NCCOC2CC2)(CC)CCCN1C(C1CCCC(C(=O)OC)C1)=O c1(C(=O)NC(C(C)NC(C(CC(C)C)OC)=O)CO)ccnc2[nH]nnc12 C1(C(N(C(c2ccc(C)cc2)C)C)=O)CN(C(=O)Cc2ncoc2C)CCC1O C1(C(N(C(C)CCNC(=O)CCCSc2ccccc2)C)=O)CC2CC1CO2 N1(Cc2ccc(-c3n(C)cnn3)s2)CC2(CCCC2)c2cccc(F)c21 N1(C(C(CC)OC)=O)CCC2(C1)CN(C(C13CCCCC1C3(F)F)=O)CC(C)O2 C1(C(N(C(C(=O)Nc2cn(CC=C)nc2)C)CC)=O)CC2(CSC2)C1 N1(C(C2CCC(=O)C2)=O)CCCCC1CCNC(c1cc(Cl)n[nH]1)=O N#Cc1nc(Br)cnc1NC(C1CCCN1Cc1ccc(F)cc1C(F)(F)F)=O Cc1nc(Cl)sc1C(N1CCN(c2noc(C(C)C)n2)CC1)C(=O)NCC1CC1 C(C(O)C(C)(C)C)NC(CCCn1cc(-c2cn(C(C)C3CC3)nc2)nn1)=O CC(C)CC(N)CC(=O)N1CC2CCCC1C2CO C1(NC(C(C)C2CCC2)=O)CCCC12CN(C(C1COC(=O)N1)=O)C2 c1(C(=O)NCC2CCC(NC(CC(C)C3CC3)=O)C2)cn2cc[nH]c(=O)c2n1 N1(C(C(CC=C)C)=O)CCC2CCC(NC(c3cc4n(n3)CCCN4)=O)C12 Cc1cc(F)c(CN(C2CCN(S(=O)(=O)CC3CCCCN3C)C2)C)c(F)c1 c1(CC)nnc(C)n1C.C1(C(N2CCC(N3C(=O)CN3C)C2)=O)C2COCC12 C1(C(CCC=CCCCNC(CCC)=O)=O)CCCCC1C C1(F)(C(N2CC(SC)C(NC(C3CC(C4CCC4)C3)=O)C2)=O)C(C)(C)C1(C)C C1(C(N2C(c3ccc(CC)s3)CCC2)=O)CC(CN)C12CCC2 C1(C(=O)NCC(=O)NCC(=O)Nc2cccc(OC)c2)CCOC(=O)CC1 C1(CNC(C2C(CC)C2)=O)CCCC2(CN(C(c3cccc(C)c3O)=O)C2)O1 c1(C(=O)OCC)cc(NC(C2CC(NC(C3CCC(C)S3)=O)C2)=O)on1 C1(CC(=O)NC2C(N(C)C)CC2O)CCN(C(=O)CC2CC3(CC3)C2)C1(C)C N1(C(CCC)=O)CC2(C1)OC1(C)CC2(NC(=O)C=C2CC3CCC(C2)N3C)C1 c1(CCC(N2CC(C(N(CCOC)C)=O)C(O)CC2)=O)ccc(F)c(F)c1F c1(C(=O)NCCC(CC)(CC)NC(=O)C(O)CN(C)C)n[nH]c2c1CSCC2 C1(C2CCOCC2)(C(=O)NCc2cn(C3CCCC3)cn2)CCNC1 CC1CCCC1(C(N1CCC(CCO)C1)=O)NC(=O)CC1C(C)(C)C1(C)C c1(C(N2C(C)CC(NC(=O)CC(c3ccc(Cl)cc3)O)C2)=O)cccc(F)c1N C1(O)(C(C(=O)NCCCC2CC2)NC(C2C(C(C)C)OCC2)=O)CCCCC1 N1(C(C2C(C(C)O)C2)=O)CCC2(NC(c3cc(Br)co3)=O)CCCC12 C12(NC(C(CCCC)N(C)C)=O)CCC(F)(F)CC1CN(C(=O)C(F)=C(C)C)C2 C1(NC(c2cn(-c3cccc(C)c3)nn2)=O)CCN(C(c2ncc[nH]2)=O)C(C)C1 C=CC1(C(=O)NC(c2noc(C)n2)C)CCN(C(c2ccco2)=O)CC1 N1(C(C(CCC)(C)C)=O)CCOC2(CCCN(C(=O)CNC(C)=O)C2)C1 C1(C(=O)NC(C(C)C)CCN(C(=O)CCN2CCCC2)C)CN(C)CC(C)O1 Cc1cc(C(N2CC(O)CC2C(=O)Nc2cccc(O)c2Br)=O)ncc1[N+](=O)[O-] C12(CNC(C(CC)N(C)C)=O)CCC(CC1)CN2C(=O)CCNC(=O)CO CC1CCCC1(C(=O)N(CCCN(C)C)C)NC(C1CCCC1O)=O CCC(C)C(C)(c1nnnn1C1CC1)Nc1cnn(CCO)c1C c1(OC)cc(F)c(C(=O)NC(C)C(C)NCc2ccc3c(c2)OCC3)c(Cl)c1 Cc1cc(C(N2CC3CCN(C(=O)CS(C)(=O)=O)CC3C2)=O)ccc1[N+](=O)[O-] CC1(C)CCOC1CC(=O)NC(C(N1CC(O)(c2nn[nH]n2)C1)=O)C1CCC1 C12(C(=O)NC3(CNC(=O)CC4CCCCC4)CCOC3)CC3CC1C2C3O c1(OC)ccccc1S(=O)(=O)CCCN1CC2C3CCC(O3)C2C1 CC1CN(C(C2CCCN2C(c2ccc(O)c(F)c2)=O)=O)C(C)CO1 N1(C(C2CC(=C)C3N2CC3)=O)CCC2CCOCC2C1 c1cc(N2CC3CCC3C2)nc(N2CCC(C3CCCO3)C2)n1 C(=O)(C(O)CCCNC(C1CCC(OC)C1)=O)NCc1c(OC)cccc1 Cc1ccc(C)c(OCC(=O)NC2C3CC2N(C(=O)C=Cc2ccco2)C3C)c1 c1(C(=O)NC2CN(C(CCC(C)OCC)=O)CC(F)C2)cc(Cl)cc(C)c1OC C1(CN(C(=O)COCP(C)(C)=O)C)CCCN1C(=O)Cc1cc(C2CC2)on1.OC C#Cc1ncccc1CNCCc1ccc(N2CCOCC2)nc1 C1(CCC(C)C)CCN(Cc2cnc(C(F)(F)F)nc2)CC1 c1(N2CCCC(NC(c3c(C(C)(C)C)noc3)=O)C2)cccc(F)c1[N+](=O)[O-] N1(CC2CC3(C(F)F)C(C2)C3)CC23CCCC2(COC3)C1 c1(CN2C(C(=O)NCCCOC(C)C)CC3CC32)c[nH]c2cc(C#N)ccc12 C(=O)(C1=CC2C=CC(C1)C2)NC1CCC(CC(=O)NC(COC)C)C1 N1(C(C2C(C)(C)C2NC(=O)CC2CCOC2(C)C)=O)CCCC(F)CC1 C(=O)(CCCC(C)NC(c1c[nH]c(C#N)c1)=O)NC(C(=O)OC)CO C1(C(=O)NC(C2CCN(C(c3cn(C)nn3)=O)C2)C)Cc2cc(Cl)ccc2C(=O)O1 Cn1nc2c(c1C(=O)NCCN1CCN(C(C3CCNC3=O)=O)CC1)CCCC2 C1(NC(C=Cc2c(C)ncs2)=O)CCCN(C(=O)CP(C)(C)=O)CC1 C1(OC)(OC)C(C(=O)NC(C2(O)CCCCC2)C)CC1(F)F c1(CC)ccnc(C(N2CCC(F)(C(=O)NCc3nonc3N)C2)=O)c1 N1(C(C=COCC)=O)CCC(NC(c2ccco2)=O)C(F)C1 c1(C(N2CC3(CCN3C(c3ccc[n+]([O-])c3)=O)C2)=O)cccc2c(Br)n[nH]c12 N1(C(c2cn(CCN(C)C)nn2)=O)CCCC(CNC(c2nnn(C)c2N)=O)C1 C12(OC)CCC(C(=O)NC3CC(N(C(=O)C(O)C(C)C)C(OC)OC)C3)(CC1)C2 N1(N(C2CN(C(C3(C(C)(F)F)CC3)=O)CC23CC3)C)CC2(CCCCCC2)C1.C=O C1(NC(C2(CC)CCN(C(C3CCC4CC34)=O)CC2)=O)CCC2(CCC2)CC1 C1(NC(C(CC)OCC)=O)CC12CC(NC(c1cc(-n3nccn3)ccn1)=O)C2 c1(C(N(CC(C)N(C(C2C(CCOC)C2)=O)C)C)=O)ccc(O)nn1 C12(C(=O)NC3CC(F)(CNC(C4(CC#C)CCCC4)=O)C3)CC3CC1C2C3 C1(F)(C(=O)NC2CCN(CC)C2)CCCN(C(=O)C(C(=O)OC)OC)C1 C1(C(=O)NC2CCCCCC2)(COC)CCCCN1CCC(=O)N(C)C C1(OC)(CNC(=O)C(C)SC)CN(C(c2occc2Cl)=O)C1 Cc1cccc(O)c1C(=O)NC1CCCC(NC(C2(CO)CC(F)(F)C2)=O)C1 C(C(C)(CO)OC)NC(CN(C(=O)CC(C)n1ccnc1)CC#C)=O c1(C(=O)NC(CCC)C(=O)N(C)Cc2ccn(CC)n2)ccc2c(c1)COC2 c1(C(=O)NC2CC3CC(NC(C4CC4F)=O)C3C2)cc2ncccc2[nH]1 C1(NC(=O)CC2CCOC2=O)C2CC1CN(C(=O)Cc1c(F)cccc1Br)C2 c1(C(=O)NCC2C(NC(C3(C#C)CCC3)=O)COC2)cnc(C)nc1COC CCC(CN(C)C)CC(=O)NCCCCC(C)NC(c1csc(COC)c1)=O CC1CCN(C(=O)COC2CCCOC2)CCN1C(c1csnc1Br)=O C(C(C)(CC)C(=O)NC(CC)C(C)(C)C)NC(C(C1CC1)OCC)=O NC1(C(=O)NNC(=O)Nc2ccc(F)cc2)CC12CCOCC2 Cc1ncccc1C=CC(N1CC=C(CNC(C2CC(C)CO2)=O)CC1)=O c1(C(N2C(CN(C(=O)C(=O)C(C)(C)C)CC)CCC2)=O)ccc(OC)c(Cl)c1 N1(C(CC2(OC)CN(C(C(C)OCCC=C)=O)C2)=O)CC(CO)C(C2CC2)C1 C1(C)(CCNC(C2C(OC)CC2)=O)CCCN1C(=O)C1CC1 n1(CC)c(CCN2CCCC(C(=O)O)(CO)C2)nc2ccccc12 c1(OC)noc(C)c1C(=O)NCCC1(O)CN(C(c2cncc(O)c2)=O)C1 N1(C(COc2c(C)cc(Cl)cc2)=O)CCC2CCCC12CNC(=O)C(C)(C)C1CC1 CC(=O)CCCC(=O)N1CCC(N(C)C(c2ccc(-c3cscn3)nc2)=O)C1 c1(NC(c2c(CCC)n(CCO)nc2)=O)ccc(C)c(C)c1N C(CCCC(=O)NCC1CCOC1C(=O)NCC(C)C1CC1)NC(C)=O CC1CCN(CC(=O)N(C(C)CN(C)C(c2ccn(CCF)n2)=O)C)CC1 c1(C(=O)OCC)ccncc1NC(=O)NC1CC(C)CCS1 c1(CNC(C2C(C)(C)COCC2)=O)cccc2c1CCC2 C1(C(=O)NCc2scc(CNC(C(F)OC)=O)n2)CCC(=O)N1C(C)C C(CCN(C(=O)C=CBr)C)(C(C)C)NC(C(CC)OC1CCCC1)=O c1(CCC)ccc(CC(=O)NCC(O)CN(C(=O)C(C)=CC2CC2)C)cc1 C1(NC(C(C)=C(CC)C)=O)CN(C(C2COCCC2(F)F)=O)CC12CC2 CCC(C)CCC(=O)N1CCC(Cn2cc(-c3cccc(C(N)=O)c3)nn2)C1 N1(C(CCOCCOCC)=O)CCC2(CCC2)C(NC(=O)C(=O)NC2CC2)C1 c1(OCC)cc(CNC(=O)C(N2CCC(C)(c3cccc(Cl)c3)C2)=O)cc(F)c1 c1(OC)cc(OC)c(C(=O)NC(CNC(=O)C(C)C(C)(C)C)C2CC2)cc1OC c1(C(=O)NC(C(CSC)(C)C)c2nnnn2C)ccc(OC)c(C(F)(F)F)c1 C1(CC)CN(C(C2(C(=O)OCC)CC2)=O)CCC1NC(=O)Cn1nccn1 c1(C(C)NC(=O)NC2C(OCC)(OCC)C2)ncc(Cl)nc1Cl C1(CCC(=O)NCC(COC)NC(c2cn(C(C)C)nc2C)=O)CC(C)(C)CO1 N1(C(C2C(C)CC=CC2)=O)CCCC(O)(CCNC(c2ccnc(CO)c2)=O)C1 c1(C(N2CCOCC2C2CC2)C(=O)NCCCF)cc2nc(F)ccc2o1 N1(C(C2CC(OCC)C2)=O)CCN(C(=O)C2=NOCC2)C(CCSC)C1 C1(CC)CCN(C(=O)CS(C)(=O)=O)C1C(=O)NC(C)C(C)n1cccn1 CCC(C)C(O)C(=O)N1CC(CCNC(c2csc(-c3cnn(C)c3)n2)=O)C1 C1(C(N2C(CNC(C(CC#C)C)=O)CC(F)(F)C2)=O)CC2(C1)CC(C#N)C2 Cc1ccc(-c2ocnc2C(=O)NCC2CC2NC(C2(C)CC2(F)F)=O)s1 C=C(CNC(C1CC1(F)F)=O)CCNC(=O)C(O)Cn1cncn1 C1(C(N2C(C=CC(N3C(CN(C)C)C=CC3)=O)CCC2)=O)CC(=O)CC(=O)N1 c1(-c2c3cc(C(=O)NCC(=C)F)sc3ccc2)cnn2ccc(C)cc12 c1(C2C(c3cc(-c4ccoc4)[nH]n3)C2)ccc(Br)cc1.C12CC1C(=O)NC2=O Cc1cc(-c2nc(-c3cccc(C(F)(F)F)c3)nn2CCC2CC2)c(C)o1 N1(C(C(CC2CCCC2)NC(c2cc(C(C)C)no2)=O)=O)CCC2(CSC2)C1 CP(C)(=O)C1CCCCC1C(=O)NC1C2CC1N(C(C1CC1c1ccsc1)=O)C2 N1(C(CN2C(C)CCC2)=O)CC2(C1)CN(C(c1nnn(C)n1)=O)CC2CO N1(C(C(C2CN(C(C3CC3C(C)C)=O)C2)OC)=O)CCCC2(CCC2)C1 N1(C(c2c(C)nco2)=O)CCC(C)C(CNC(=O)CSc2ccc(F)cc2)C1 c1(C(N(C)CC2(NC(C3C(C=C)C3)=O)CC2)=O)cc(C)c(F)cc1Br c1(CC(=O)NC(CNC(C(COCC)C)=O)CO)coc2cc(CC)ccc12 N1(C(COCC#C)=O)CCCC1C1CCCN1C(=O)CCCOC1CC1 S(=O)(=O)(c1c(Cl)nc2ccc(Br)cn12)NC(Cn1ccc(C(=O)O)c1)=O c1(SC)ccc([N+](=O)[O-])c(NC(C2CC(NC(=O)CC3CC4CCC3C4)C2)=O)c1 S(=O)(=O)(c1ccccc1Br)N1CCC(N2CCN(C(c3cocn3)=O)CC2)CC1 C(CCCCCC(=O)NC12CCC(CC1NC(C1CCCNS1(=O)=O)=O)C2)SC S(=O)(=O)(c1cnc(N2CCC(CCC)C2)cc1C)NC(CCC=C)(C)C CN1CCC(NC(=O)C(CC(F)F)NC(c2coc(C(F)F)c2)=O)C(C#N)C1 CC1(C)Cc2cc(CS(=O)CCc3cccc(O)c3)ccc2CO1 C1(COC(C)C(=O)NC2CC3CCC2C3)COCCC1(F)F N1(C(c2n(C)c(=O)ccc2)=O)CCC2(CCCC2C(NCP(=O)(O)O)=O)C1 C(=O)(C(C(C)(C)C)C1CCC1)NC(CC1CN(c2cc(COC)ncn2)C1)C C1(C(N(C)CCC2CCOC2)=O)CCCCN1C(=O)CCC(=O)N1CCCC1 c1(CN2CC(O)(CCC)C2)c(OC)ccc(F)c1Br C1(OC)CN(C(c2sc(-c3ccn(C)n3)nc2C)=O)CC1NC(c1ccoc1)=O N1(C(c2ccc(C3CC3)nc2O)=O)CCC2(CCC2)C(O)C1 c1(N2CCN(CC(=O)OC)CC2)ccc(CNc2cccc(F)n2)cc1C C1(C(N2C(CNC(C3CC(F)(CO)C3)=O)CC(C)(C)C2)=O)CCc2nc[nH]c2C1 C(CCCCC(=O)N1CC(N(C)C)C1)NC(C1(C(C)=O)CC1)=O c1(-c2ccc(OC)nc2OC)cccc2nc(C(=O)Nc3cc(C)ns3)ccc12 CCC(C)C(O)C(=O)NCCN1CCC(NC(=O)CCCn2cccn2)CC1 Cc1cc(C(N2CCC(CNC(=O)C(F)(F)c3cncs3)C(C)C2)=O)cnc1O c1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCCC2C)cncc2ccsc12 c1(C(=O)NCC2C(CNC(C(F)=CC)=O)C2)c(C)ncn(C)c1=O CC1CCN(C)CCN1C(=O)C(N1CCC(CCP(C)(C)=O)CC1)=O CCC(C)C(C(=O)NCC(C)(C)CNC(=O)CC1(O)CCC1)NC(N)=O Cc1cn2cc(C(=O)NC34CCC(C3)N(C(=O)CC3COCCN3C)C4)nc2s1 N1(C(c2c(CCC)nns2)=O)CC2CC(C1)C(CO)C2NC(c1nonc1N)=O N1(C(=O)COC2CN(C(c3cc(Cl)ccn3)=O)C2)Cc2cncnc2C1 c1(C(N(CCNC(c2occ(C)c2C)=O)CC)=O)cccc2cccnc12 c1(NC(C)=O)ccc(NC(c2cnnc(O)c2S)=O)c(Cl)c1 N1(C(C(F)=CCC)=O)CCC(NC(=O)COCc2ccccn2)C(CC)C1 c1(C(N2CC(COC)N(c3nccc(C)n3)CC2)=O)c(C)ccc(Br)c1F n1(CC)c(SC(C)C(=O)NCCCn2cc(C(=O)OC)nn2)nc2ccccc12 CC(C(=O)NCC1(O)CN(C(c2ccc(O)c(Br)c2)=O)C1)S(N)(=O)=O c1(C(N2CCN(C(c3ccnc(Cl)c3)=O)C3CC23)=O)cccc([N+](=O)[O-])c1Cl C=CCCCC(C(=O)NC(C)(C)CCCC)NC(=O)COCCCN=[N+]=[N-] C1(CCC(=O)NCC(N(C)C(C2(C)CC2(F)Cl)=O)C2CC2)CCCCN1C C(CN=c1ccnc(C(C)C)[nH]1)(CC(C)C)NC(C1Cn2c(C)nnc2CC1)=O C1(CNC(C2(CCOC)CCCC2)=O)CN(C(=O)CS(N)(=O)=O)CCCO1 c1(NCC(C(C)C)C)cc(=NCC(F)CO)[nH]cn1 C1(CNC(C2(COC)CCC2)=O)C=CC(NC(=O)C(C)(C)C2CCCCO2)C1 C(CCC(N)=O)(C(=O)N(C)CC1(O)CN(C(C2(C)CCN(C)C2)=O)C1)NC(C)=O C1(c2n(-c3ccccc3)nc(-c3nc[nH]n3)n2)CCCC2(CCC2)O1 C=CCC(CNC(=O)Cn1cc(C2CC2)cn1)C(=O)NCc1nnnn1CC C12(OC)CCC(C(N3CC4CC3CN4C(=O)C(CCSC)OC)=O)(CC1)C2 Cn1ccc2[nH]c(C(=O)NC3(C)CCN(C(=O)C(F)=C4CCC4)C3)cc12 C(=O)(C(C)(C)CC(C)=O)N1C2(C(NCP(OCC)(C)=O)=O)CC(C)(C1)C2.C(C)(=O)OC C1(NC(C2(C3CC3)CC2)=O)CS(=O)(=O)CC1N=c1[nH]ncs1 c1(OCC(=O)NCC(CNC(C(C(C)C)OC)=O)F)cccc(S(C)(=O)=O)c1 C(=O)(C1=CC2CCC(C1)C2)N1CC(O)(CCNC(c2cnc(OC)c(C)c2)=O)C1 CC1OCCCC1C(=O)NC12CC(C1)N(C(=O)Cn1ncnn1)C2 c1(C(N2CC(F)(C(=O)Nc3cn(CCC)nc3)C2)=O)cccc(Br)c1 C1(CC=C)(NC(C2(C(C)C)COC2)=O)CCN(C(c2ccc(SCC)cc2)=O)C1 c1(CC)cc(C(=O)NCC=CCNC(C2(C)CCCC2(F)F)=O)cc(O)n1 C=CCC(CC=C)C(=O)N1CC(C)N(C(c2nnc(O)cc2C)=O)CC1C C1(c2ccc(C)o2)CS(=O)CCN1C(C1CC1c1ccc(F)cn1)=O C(=O)(CS(=O)(=O)CC(=O)NCC(CO)NC(=O)CC1C=CS(=O)(=O)C1)OC c1(C(=O)NCC2C(C)CN(C(C3(CCF)CCOCC3)=O)C2)cc(N)cc(O)c1 c1(C(=O)NCC(C)N(C(CC2(C=C)CCC2)=O)C)cccn2cncc12 C1(C(=O)NC(CC=CC)CO)CN(C(=O)C(C)CSC)CC1(F)F N1(C(C(C)(C)N2CCOCC2)=O)CC2CC(C1)CN(C(C1CCCCO1)=O)C2 C(=O)(C(O)CCCN1CCCC1c1ccc(Cl)c(Cl)c1)OC C=C=C(C)CC(=O)NCCCC(=O)NCc1cnc(OC)cn1 C1(CNC(C(C)C2CC2)=O)CCC12CCN(C(=O)C=CCN(C)C)CC2 C=C(C)C(C)(O)C(=O)NCC(C(C)C)NC(c1cncc(N2CCCC2)n1)=O O(NC(=O)C(c1cccnc1)NC(c1ccn(CCF)n1)=O)CC(C)C N(C)(C1CN(C(=O)C(=O)NC2CC2)CCc2ccccc21)C(CC(CC)OC)=O c1(C(=O)OCCCN(C(=O)Cc2ccccc2F)CC)ccc(NC)cc1 N1(C(C2(SC)CC(=O)C2)=O)CC(C(=O)NC2CC3(C2)CC(O)C3)CC(C)(C)C1 C=CCC(C(=O)N1CCCC1(C)CCC(=O)NCCOC(CC)CC)NC(C)=O CCC(C#N)C(=O)NC(c1ccccc1)CNC(=O)C(CC)NC1CC1 CCN(C(C)c1ccc2c(c1)OCCCC2)N(C)C1CCOC1 CC1(C)C(NC(=O)CCC2CCCOC2)CCN1C(=O)CCSCCC(F)(F)F Cc1cc(C2CC2)ccc1C(=O)NCC(O)CNC(c1cncc(N)c1)=O c1(C(=O)NCC2(CO)CCN(C(C3CC=CCO3)=O)C2)ccn2c1CCCC2 S(=O)(=O)(C1CCC2(CC1)OCCO2)N(CC(C(=O)OC)Nc1ccccn1)C C(=O)(C(C)CC)NCCNC(=O)COC(C(=O)N(C)CC)C CS(=O)(=O)c1cc(C(N2CC(O)CC2c2ccc(Br)cc2)=O)c(Cl)c(Br)c1 CCC(C(=O)OC)C(=O)N1CC=CCC1C(N1CC(CO)C1(C)C)=O c1(CC(=O)OC)c(C)nn2c1CN(C(=O)COCCCN(C)C)CC2 C1(C(=O)NC2(CO)CN(C(C3(c4ccno4)CC3)=O)C2)C2CCC(=O)C12 C1(C(=O)NC(CCN(C)C)C(=O)N2CCCC(CN=[N+]=[N-])C2)CCC2(CC1)CC2 C1(CC=C)(NC(=O)CO)CN(C(=O)CCc2cncn2C)C1 N(C1CCCc2occc21)C(C1C(C)CCN1C(C1CC(C)(C)CO1)=O)=O CC1CCn2ncc(C(=O)N(C3CCCCN(C(=O)CCF)C3)C)c2C1 c1(OC)ccc(N)c(C(=O)NC(C)CCNC(=O)COC2CCOC2)c1 C(=O)(C(CO)NC(=O)CN1CC2CC2C1)N(C(CO)CO)C C(C1OCc2ccccc21)c1n(-c2ccc(CC)cc2)nc(CO)n1 c1(C(=O)NCC2(F)CCC(NC(C(C)(C)O)=O)C2)cn(CCO)c(=O)nc1O CCCCC(CC)NC(C)(CCC1CC1)c1nnnn1C1CCCC1 CCC(C)(C)C(C(=O)NC1CCCCN(C(c2coc(Cl)n2)=O)C1)OC c1(CC)cc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCc2cc(C)[nH]n2)n[nH]1 c1(C(=O)NC2CC(CCNC(C3CC=CCO3)=O)C2)ccc2nsnc2c1 c1(NC(=O)NCCCC(=O)NCCC2CN(C(C)=O)C2)cc(C#N)ccc1N c1(C(C(=O)NC(CCCNC(c2cnc(SC)s2)=O)C)C)c(C)n[nH]c1C c1(CC(=O)NCC23N(C(C4CCC(C)C4)=O)CC(C2)C3)nn(C)c2ccccc12 C1(C(=O)NCCC(C)C)CCC2(CN(C(=O)CCc3ccoc3)C2)O1 c1(CC(=O)NC(C2CN(C(=O)C=CCF)CCCO2)C)csc2ccc(Cl)cc12 C1(C(=O)NCCCC2C=CCC2)CCOCCN1C(c1scnc1Cl)=O N1(C(C(=Cc2ccncc2)C)=O)CCC2(C1)CN(C(C1CCCC(CF)C1)=O)C2 c1(C(=O)NC2CC(C(C)C)SCC2)cc(C#N)ccc1Cl c1(OC)ccc(CCC(=O)N(CC(F)F)CC2CCCO2)cc1CC(=O)O C1(C(N2C(C#C)CC2)=O)(OC)CCN(C(c2ccc(CC)o2)=O)C1 c1(NC(C2(CF)CCN(C(C(CC)COC)=O)C2)=O)cccc2c1CCC2 C(=O)(C(F)(F)c1csc(=N)[nH]1)NCC(CN(C)C(C1(C(N)=O)CCC1)=O)O O=C(O)CCCCCNC1CCN(C(C2CC2)C2CC2)CC1.c1(O)ncc(Cl)cn1 c1(C(=O)NC2CN(C(CC3(OC)CCC3)=O)CC2C2CC2)cncc2c1CCC2 C1(CC(=O)NCC2(C(N)=O)CN(C(C(C(C)C)F)=O)C2)CCCCC1(F)F N1(C(CC(C)c2cccnc2)=O)CC=C(CNC(c2cc(O)nc(O)n2)=O)CC1 Cc1[nH]nc2ccc(C(N3CC4(CC4)CC3CNC(=O)CC3(C)CC3)=O)cc12 c1(C(=O)NCCCC(c2ccccc2)NC(CCC#C)=O)cc(Cl)c(Cl)s1 C1(C(=O)NCC(C)CN(C)C(C2CCN2C)=O)CCCC1O Cc1ccnc(N(CCCNC(c2cc(O)nn2C)=O)C(C)C)c1[N+](=O)[O-] c1(C(=O)NCC2C(NC(c3n(CC)ncc3)=O)C2)nc(O)nc(O)c1N C1(O)(CNC(Cc2ccc(CC)cc2)=O)CCCN(C(CCCC(C)C)=O)C1 c1(NC(=O)NCCC#C)ccccc1-n1nc(C)cc1C CC1C2CC(C2NC(C2CCN(C)CC2)=O)N1C(=O)C1=CCCOC1 C1(CC)(CO)CCN(C(=O)C(CO)NC(c2ncncc2Cl)=O)C1 C(CNC(N1CCSC1)=O)(CNC(=O)CCSC)OC c1(CC)nc(C#N)cc(=NC(C)CNC(=O)Cc2ccco2)[nH]1 c1(CC(N2C(CNC(C3CCOC3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])cc1 N1(C(CCCOCC)=O)CCCCC12CC(NC(=O)Cc1ccc(CC)cc1)C2 CC1CC2CCC(C1)N2C(=O)CC1COCC1NC(c1ccc2ccoc2c1)=O C(=O)(C(C)(O)C(F)(F)F)NCc1oc(C)c(C(=O)NC2CCOC(C)C2)n1 C1(C(=O)NCC(CNC(c2ccc(C#C)o2)=O)C)CC2(C1)CC2(F)F CC(C)(C(=O)NCCC1CC2CC1CC2O)C1=CC2CCC(C1)N2 C(=O)(C1=C2CCN=C2NC=C1)N1CCN(C(C(N2C(CC)CCC2)=O)=O)CC1 C1(C(N(CC(=O)NCc2scc(C)n2)C(C)C)=O)CCCC1C1CC1 C1(NC(CCCC(=O)NC)=O)C(CNC(=O)C(C)(C)CCC#N)CCC12CCC2 C12(NC(Cc3[nH]nc(C(C)N)n3)=O)CC(N=[N+]=[N-])(C1)C2 c1(OC)cc(I)cc(NCC(C)C(=O)c2ccccc2)c1[N+](=O)[O-] C=CCC(C(=O)N1C(C(N2CC(C#N)C2)=O)CC2CC12)OC c1(C(N2C(CNC(C(C)(C)O)=O)CC2)=O)ccccc1-n1ccnc1O C(=O)(C(O)P(C)(C)=O)C(Cn1cc(CCC2N(C)CCC2)nn1)=O.N1CCC(CO)CC1 c1(C(=O)NCCC2CC(NC(C3(Cl)CC34CCC4)=O)C2)ncccc1F C1(C(=O)Nc2c(C(=O)OC)csc2)CC(C)CN1Cc1cccc(CO)n1 N1(C(CC(C)n2cccc2)=O)CCC(O)C(N(C)C(C2CCCN2N=O)=O)C1 c1(NCC(N2CCN(C(C(C(C)C)SC)=O)CC2)=O)cc(CO)ccc1[N+](=O)[O-] C1(CNC(C=C(CC)C)=O)CN(C(c2ccnn2C)=O)CCC1C(F)(F)F C(c1nc2ccccc2[nH]1)=CC(=O)NC(C)CNC(c1cc(C#N)cn1C)=O C(=O)(CC(C)(CNCC12CCC(O)(CC1)CC2)C(F)(F)F)OCC c1(OCCC)ccc(C(=O)N(C)CCN)cc1OCC1CC1C(=O)C(C)(C)F C1(O)(CN(C(C(CCC)NC(C)=O)=O)C)CCCN(C(C2CC(=O)N2)=O)C1 C=CCC(C)(C)C(=O)N1CCCC(C(N2CCC(OCC3CC3)C2)=O)C1 N1(C(C2CCC(CNC(c3cnn(C)c3Cl)=O)CC2)=O)CC2OCCOC2C1 C(CC(C)=O)(C(=O)NC(C)(C)CCN(C)C)NC(CC1(N)CC1)=O.C1(COC)CC1 C(=O)(CC1=NNC(=O)C1)NCC1(C(C)NC(c2cc[nH]c(=N)c2)=O)CC1 c1(OC)ccc(N(C(=O)C(c2cn(C)nc2C(F)(F)F)C)C)c(F)c1 c1(C(N2CN(C)C(=O)C2C)C)ccc([N+](=O)[O-])cn1 N1(C(c2cc(C(=O)OCC)no2)=O)CC2CC(C1)C2NC(=O)C(O)C(C)CC N1(C(C2CC3CCC3C2)=O)CC2CCC2(C(=O)NC2CCOC2)C1 C(=O)(C(C)C(C)C)NCCN(C(=O)COc1ccsc1)CC=C Cc1nc(C)c(C(N2CCC(NC(c3ccnc(N4CCCC4C)c3)=O)C2)=O)[nH]1 C1(NC(Cn2c(C)nc(C)n2)=O)CC(NC(=O)CC2CC3(CC3)C2)C12CCOCC2 Cc1[nH]nc(C(=O)NC2CCOCC2C(N2CC(O)(C(F)(F)F)C2)=O)c1C C1(CC)CN(C(=O)CCSC2CC2)CCC1NC(=O)CCOCC(F)(F)C(F)F Cn1cc(C(=O)NC2(CNC(c3ccc[n+]([O-])c3)=O)CC2)c(-c2ccccc2)n1 c1(C(N2CCSCC2(C)C)C(=O)Nc2c(CC)cccc2)ccc2c(n1)CCC2 CCC(CC(C)C)C(=O)NC(C(N1CC(=O)NC(=O)C1)=O)C1CCCC1 N1(C(C(C(COC)C)C)=O)CCC2(C1)CN(C(=O)COCP(C)(C)=O)C2 N1(C(c2c(C)nc(O)[nH]2)=O)CCCC2(C1)CN(C(=O)C(O)CCC(F)(F)F)C2 N1(N(CC=C)C)CCC(C)N(C(=O)CC2CCCOC2)CC1.c1(C=O)nccs1 C1(CNC(c2n(CCC)nnn2)c2nnnn2C(C)C)CCC(=O)NC1 c1(C(N2CCN(C(c3c(CC)con3)=O)CC2C(C)C)=O)cc2nnn(C)c2s1 C1(F)(CNC(c2c(C)cccc2)=O)CCCN(C(=O)CCc2nncn2C)CC1 C1(N(C)C)CCCN(CCC(=O)NCC2(O)CN(C(=O)CC3CCCOC3)C2)C1 c1(CNC(C(Cc2ccoc2)NC(C2C3CC(=O)CC32)=O)=O)ccc(F)c(F)c1 N1(C(C2(C)CCCN(C)C2)=O)CCC2(CC(C(=O)NC(CCO)C(C)(C)C)C2)C1 CC(C)C(CCC(=O)NCCCC(C)(C)O)NC(C1CCCC(=O)C1)=O N#Cc1ccc(C(=O)NN2CCC(NC(=O)C(=O)NCCNC3CC3)C2)cc1 c1(C(N2CCCC(c3nc[nH]n3)C2)C(=O)NCCCC)ccc(OC)cc1 c1(OC)c(C)nc(C2CC2)[nH]c1=NCC1(F)CCN(C(c2ccncn2)=O)CC1 c1(C(C(=O)NCCN(C(=O)CC(C)CN(C)C)CC)(C)O)ccc(F)cc1 C=CCCC(F)(F)C(=O)N1CC(CC(F)C(=O)NCC(C2CC(C)(C)C2)O)C1 C=CCC(C)(C)CC(=O)N1CCN(C(c2c[nH]nc2F)=O)CC(CO)C1 N1(C(c2c(C)cco2)=O)CCCOC(CNC(c2ncccc2C(F)(F)F)=O)C1 C(=O)(CC1=NNC(=O)C1)NC(c1c(OC)cccc1)CNC(=O)Cc1cocn1 C1(C2CCCCC2)(C(=O)NC2C(F)CCN(C(C(n3c(C)ncc3)C)=O)C2)CC1 c1(C(N2C3CC(NC(c4cn(C)nc4C(F)F)=O)(C3)C2)=O)ccc2ccnn2c1 C12(NC(c3[nH]cc(COC)n3)=O)CCCC1CN(C(=O)COCC1CCCC1)C2 C1(CN(C(=O)Cn2cnnc2O)C)CN(C(c2ccc(C3CC3)nn2)=O)CCO1 CC#CCCCC(=O)NCC(=O)NCC(=O)NCCCCO c1(OC)cc(N)c(Cl)cc1C(N1CC(NC(=O)C(C)(C)CF)CC1C)=O Cn1cc(C(=O)NC2CCC(NC(c3occc3Br)=O)C2)c(-c2ccco2)n1 C1(CCC)CN(C(c2c(C)nn(C)c2F)=O)CCN1C(=O)COCC(C)C Cc1cccc2c(C(N3CC4(CC4)CC3CNC(C3CC3Br)=O)=O)coc12 C(=O)(C(C)C(F)(F)F)NCC1(COC)CCCN1C(=O)CCC=CBr N1(C(C(CC2CCC2)OC)=O)CCC2CN(C(C3CCCSC3)=O)CC12 c1(OC)nccc(CNC(C2(NC(=O)CCC3CC3(F)F)CCC2)=O)n1 N1(C(c2cnc(CCOCC)s2)=O)CCN(C(C2CCOC2C)=O)CC2(CC2)C1 C1(NC(C(C)NC(=O)Cc2cccnc2F)=O)CC2(CCC2)C1O Cc1nc(NC2CN3CCC2C3)cc(NC2CC(F)C2)n1 c1(CC(C)C)ncc(C(=O)N(CCN(C(=O)COCCCF)C)C(C)C)[nH]1 C1(C)(COC)CC(NC(c2[nH]cnc2C#N)=O)CN1C(=O)CCOCC(C)C N1(CCNC(C2(CC)CCC2)=O)C2CCC1CN(C(=O)C(C)(C)CC(C)C)C2 C(=O)(CC(C)(C)C(F)(F)F)N1CC(C)C(NC(C2CCCS(=O)(=O)C2)=O)CC1 N1(C(c2ccc(C(C)C)nc2)=O)CC2CCC1C(NC(=O)C(C)C(C)C)C2 C(CCN=c1nc(O)c2ccccc2[nH]1)N1CCc2c(CO)ccc(F)c2C1 C#Cc1ccc(C(N2CC(NC(c3coc(CO)c3)=O)CC3(CC3)C2)=O)cc1F c1(C(=O)NC2CC(CCNC(C(C3CCC(=O)N3)C)=O)C2)c[nH]nc1F C1(C(=O)NC(C2CCN(C(=O)COCC(F)(F)F)C2)C)CCC(=O)N1C1CC1 C1(C2CC2)(C(N2CC(N3CCCC3=O)C2)=O)CN(C(C2C3CCCOC23)=O)C1 c1(C(N(C(C)CNC(C2CC2(F)F)=O)CC)=O)cc2cccc(OC)c2[nH]1 CCCCCC(O)C(=O)NC(CC(N)=O)C(=O)NC(C)CC(C)(C)CO CC1CC(NC(=O)C(F)(F)c2ccccn2)CCO1 C=C1CC(C(=O)NC(c2ccccc2)COC)N(CS(=O)(=O)CC2CC2)C1 S(=O)(=O)(C1CCCCC1)N1CCC(NC(c2cccs2)=O)CC1 c1(CC(=O)N(CC(C)NC(c2cc(C)oc2C)=O)C)ccc(O)c(C)c1 C12(C(N3CCC(COC)C3)=O)CC(CO)(CN1C(=O)C(C)c1cc[nH]n1)C2 c1(OCC)cncc(=NC(=O)C(=O)N2CC3CC(OC)C(C3)C2)[nH]1 CCC(CC)C(C(=O)NC1CCC(NC(c2cnoc2CC(C)C)=O)C1)OC c1(CC)cncc(C(=O)NC2CC(C)N(C(=O)C3=CCCC3)C2)c1 N1(C(=O)C2=CSCS2)CCC2C(CCCN2C(c2cccc(C3CC3)c2)=O)C1 N1(C(CC)=O)CCN(C(C2CCC23CCC3)=O)CC1c1cccc(Cl)c1 C1(C(N2CC3C(NC(c4c(CC)ncnc4)=O)C3C2)=O)CCC2CC(C)CN2C1 C(C(O)C(=O)NCC1CN(C(c2ccc(C)o2)=O)C1)SC Cc1c(C(=O)Nc2cnn(C(F)F)c2)cccc1C1CC1 c1(C(=O)NCC2CC(C(=O)NC(c3ncc(C)o3)C)C2)ncccc1F c1(CCC(=O)NCC(c2ccccc2)NC(COC(C)=O)=O)ccc(F)cc1Cl CCS(=O)(=O)CC(=O)N1C2CCC1C(CNC(=O)Cc1ccnn1C)C2 C1(C(N2CC(CNC(C3C(CC)C3)=O)(COC)C2)=O)CC(O)CN1C(C)=O N1(C(CC(C)O)=O)CC2CC1CN2C(c1ccc(Br)cc1O)=O c1(C(=O)NC2C3N(C(C4(C)COC4)=O)C(CC3)C2)cc2c(nn1)CCCC2 N1(C(c2c(C)nsc2N)=O)C2CCC1CN(C(=O)CC(C)c1ccncc1)CC2 c1(C(=O)Nc2c(C)ccc(-c3ncco3)c2)cc(C)nc2[nH]cnc12 Cc1ccc(F)c(N)c1C(N1CC2C(NC(=O)Cc3cnc(C4CC4)[nH]3)C2C1)=O N1(C(C)=O)CCC(C(=O)NC(C2C(NC34CC(CO)(C3)C4)C2)C)C1 c1(C(=O)NC2(CNC(CC3CC(OCC)C3)=O)CCOCC2)ccc(C#N)cc1 N1(C(Cc2c(C#C)cccc2)=O)CCC2CCN(C(=O)CC(CC)OC)CC2C1 C1(CNC(Cc2nnc(C)o2)=O)CN(C(C2CCCC(=O)N2)=O)C2(CCC2)C1 c1(CNC(COCC#C)=O)nc(CNC(c2c[nH]c(=O)cn2)=O)cc(O)n1 CC(CC(N)=O)C(=O)NC1CC(OCC(N2CCS(=O)(=O)CC2)=O)C1 CC(C)(C)C#CC(=O)N(CC(CC1CC1)C(=O)N1CCC1)CC(N)=O Cc1nc(C(N2CCN(C(=O)Cc3ccsc3C)C(CF)C2)=O)ccc1[N+](=O)[O-] C1(NC(C(=O)N(C)C)=O)CS(=O)(=O)C2CN(C(C3Cc4ccccc4CO3)=O)CC12 C1(N(C(C2(CC)CC2)=O)C(c2cn(C)cc2C)=O)CN(CC2CCC2)CC12CC2 N1(C(c2cnnc(Cl)c2)=O)CCC2(CCCN(C(C3CCCC3)=O)C2)C1 N1(C(C2CCCN(C(CS(CC)=O)=O)C2)=O)CCC2CCN(C)CC12 C1(C)(C(N(CC(C)C)CC#C)=O)CN(C(C2C3CCC(F)C23)=O)C(C)(C)C1 C1(C(CNC(C2(CC)CC2)=O)Nc2ccccc2)C(C)(C)C1(C)C.C(=O)CCSC C12(C(N3C(C(=O)OC)C4CC4C3)=O)CC(CN(C(c3cc(F)ccc3F)=O)C1)C2 N1(C(c2cn(CC)nn2)=O)CCC(C)(C)C(NC(=O)CC(C)C2CCCCC2)C1 Nc1ccc(CCCNC(=O)NCc2cc(Cl)ccn2)nc1 N1(C(c2c(OC)nc(C)s2)=O)CC2CCCC(C1)N2C(=O)C(C)CN(C)C c1(CNC(=O)NC(c2cccs2)CC)cc2occc2s1 c1(C(=O)NCC(CC(=O)NCC(CC)(C)CO)C)coc2ccccc12 CC(C(=O)N1CC2CC(NC(C34CC(C)(C3)OC4C)=O)CC1C2)C(C)C(C)(C)C Cc1noc(C)c1CCC(=O)NC(C)(CNC(=O)C(O)Cc1cccs1)CO C(=O)(C(CC(C)C)NC(c1ccc(O)nc1)=O)N1CCC(COC(C)=O)C1 N1(CC)C(=O)CCC1CC(N1CC(F)(CNC(C2(CCOC)CC2)=O)C1)=O N1(C(C(C)(C)SC)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1CC(C)(C)C1 S(=O)(=O)(c1cccc(=NCc2ccc3c(c2)COC3)[nH]1)NC(C)CCC1CC1 c1(C(NC(=NC)NCc2cc(C(F)(F)F)co2)C)cccc(C)n1 C1(CC(=O)N(C2CCN(C)C2=O)C)CC2CCC1(NC(=O)CSC(F)F)C2 N1(C(Cc2cnc(C)o2)=O)CCC(NC(c2cnn(C(F)(F)F)c2)=O)C(O)C1 CC1CC(=O)NCCN1C(C(=O)NC(C)(C)C)c1ccoc1 CC1CCC(N2CCCC2)CN1C(=O)NC(=O)NCC(c1ccc(O)cc1)O c1(C(C(=O)NCc2ccc(-n3cc(C(C)O)nn3)cc2)O)ccc(C#N)cc1 c1(C(N2CC(NC(C3CC3F)=O)(CO)C2)=O)c(F)ccc(F)c1Br N1(C(c2c(CC)nccn2)=O)CC(NC(=O)C(SC)SC)C(C2CC2)C1 c1(N(C)Cc2ccc(SC)cc2)ccc(S(=O)(=O)N2CCOCC3CC23)cc1Cl c1(-n2cc(C3CN(C(C(C(C)(C)OC(F)F)=O)=O)CC3O)nn2)ccc(Cl)cc1F.OC C=CC1(C(=O)NC(C2CN(C(=O)C(C)C(C)O)C2)C)CCOCC1 CC1CCN(C(=O)CC(C)C(C)(C)C)CCN1C(=O)Cc1cccs1 CC(C)C(C)(CNC(=O)C(=O)N(C)C)NC(=O)C(c1cccc(Br)n1)C C1(CC(=O)NC(CC)(CNC(C2(C)CC3CC3C2)=O)CC)COC(C)(C)CO1 C1(C)(CNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)C(CO)c2ccccc2)CC1 N1(C(C)=O)CCc2c(C(=O)Nc3cn[nH]c3)n[nH]c2C1 c1(C(C(N2CCC(N(C(=O)CC3CCOC3=O)C)C2)=O)(F)F)ncc(Cl)n1C CN1C(=O)CSC1=CC(=O)NCC1CCN(C(=O)COC2CC2(F)F)CC1 CCC1=NOC(CC(=O)NCC(c2ccccc2)CNC(c2cnns2)=O)C1 c1(OC)ccc(CCCCC(=O)N(CCCCN(C)C(c2csnn2)=O)C)cc1 C12(NC(C(F)=C(C)C)=O)CCCN(C(c3cc(F)c(F)cc3F)=O)CC1C2 c1(C(=O)NCC(c2cccc(C)c2)NC(CCCOC)=O)scc(C)c1C C1(C(=O)NC(C)CNC(c2c(Br)cnn2C)=O)CC12CCC(C)(C)CC2 C(=O)(C1CCCc2sccc21)NCC1CC(C(=O)OC(C)(C)C)C1 Cc1ccn(C)c1C(N1C(C(=O)NCCc2ncnn2C)CC1C)=O C1(OC)CC(NC(=O)C=Cc2cccc(F)c2)CN(C(=O)C(C)(F)C(=O)OC)C1 Cc1nc2cc(C(=O)NCC3CCCCN(C(C4CC4C#N)=O)C3)ccc2s1 c1(CC)ccc(OCCC(=O)NC(C)(C)CNC(=O)Cc2csc(C)n2)cc1 c1(C(=O)NCC(CC=C)NC(C2(F)CCCOC2)=O)c[nH]c2c(C#N)cccc12 C1(OCCC)CCC(CC(=O)NC(CNC(=O)C(C)(CO)OC)CO)CC1 CC1(C)NC(=O)OC12CCN(C(c1nnc(C3CCCC3)s1)=O)C2 CN1CCN(C(=O)C(c2ccccc2F)O)CC1CNC(c1cccnc1Cl)=O N1(C(C2(NC(=O)CCc3cncs3)C(C)(C)C2)=O)CC2(C1)CC2(F)F C1(C(N(CC(C)(C)CNC(=O)CC(=O)NCC(F)(F)F)CC)=O)CCC2(CC2)C1 CS(=O)(=O)C(C(=O)N1CCN(C(c2cc3n(n2)CCO3)=O)C(C2CC2)C1)C1CC1 c1(OC)ccc(CC(=O)NCC(C)N(C(=O)C(c2cccnc2)C)C)cc1F C1(CNC(CCN(C(C(CSC)OC)=O)C(C)C)=O)CCN(C)CC1 N1(C(=O)COc2cccnc2)CC2CN(C(c3coc(Cl)n3)=O)CC(C1)O2 c1(OCC)noc(C)c1C(=O)NCC1(CNC(c2cc(COC)on2)=O)CC1 c1(OCC)ncccc1-c1cccc(CC(=O)NCc2ccnn2C)n1 c12ccncc1S2.C(=O)(C(Cc1ccccc1)NC(=O)C1CC1)NCC(C)OC c1(NCC(CC)CC)ccc(S(=O)(=O)NC2CC(O)C2(C)C)c(Cl)c1 N1(C(CCNC(N)=O)=O)CC(NC(c2ccc(Br)o2)=O)CC2(CC2)C1 C1(N(CCCC)C(C2CC=CC2)=O)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 C(=O)(C(C)C(C)(F)F)N(C)CC1N(C(C(CC=C)NC(C)=O)=O)CCCC1 C#CC1(C(=O)NCc2n[nH]c(C)c2C)CN(C(=O)CC2OCCC2C)C1 C(C(C)CC(=O)N(C)CCc1cccs1)NC(c1cc(C)oc1)=O C1(O)(c2cn(CC)nn2)CCS(=O)(=O)CC1.C1(C)C(C(=O)OC)C(=O)C12CC2 C1(C(=O)NCCC2CCN(C)C2=O)CC(O)CCN1C(C1CC(N=[N+]=[N-])C1)=O c1(CCC)sc(C(=O)NCCCN(C(=O)C=CS(C)=O)C)cc1Br Cc1ccc(C(N2CCCC2)=O)c(CSCc2cn(C)nc2C)n1 c1(NC(C(N2C(CC(=O)OC)CC2C)=O)=O)ccc(O)cc1Br C(=O)(CCCC(N)=O)N1CCC(C(C)NC(c2c(C)nc(Br)o2)=O)C1 c1(OC(CC)C)ccccc1C(=O)NC1CN(C(c2cccn2CC)=O)CC1C C=CC(C)(O)C(=O)NC1CC(C(=O)NCCc2cncc(C)n2)C1 C(=O)(C(C#N)(CC)OCCCOCCOC)c1cn(SC)nn1.CCCC.C1CS1 C12(C(=O)NC(CCOCC)C(=O)N3CCOC(C(C)C)C3)CCCC1C2(F)F C(C)(CCCCNC(=O)C(C(C)C)C1CCC1)NC(Cc1c(C)con1)=O C1(C(N2CC(OC)(CNC(=O)CC(C)(C)OC)C2)=O)CC2CCC1O2 C1(C(=O)NCC(C2CC2)NC(COC(CC)C)=O)CCc2cncn2C1 c1(C(=O)NCCCCNC(c2n(CC)c(O)nc2)=O)cnc2c(c1)nnn2C C1(CCOC)CN(C(=O)COc2ccc(C)s2)CCN1C(=O)C(CCOC)OC N1(C(C2OCCN(CC)C2)=O)CCOCC(C(=O)NC(C)(CC)CC)C1 c1(CCCC(=O)NC(CN(C(CCN(C(C)=O)C)=O)C)C)csc2ccccc12 N1(C(C2C(C)C2)=O)CCCC(CNC(c2ccc(F)c(Cl)c2)=O)C1c1ccccc1 Cc1cc(Cl)ncc1CNC(C1CCC(OC2CCC2)CC1)=O CC(C)CC(=O)C(=O)NC(c1nocc1C(=O)NCCc1cnco1)C C1(C(=O)NC(C2CCCC2)CO)COC2(C1)CN(C(=O)Cc1cnns1)C2 N1(C(C2CCC(CC)O2)=O)CC=CC(NC(=O)Cc2nnc(O)s2)C1 c1(OC)cc(C=CC(=O)N(C2CCCCN(C(=O)C(F)C(C)C)C2)C)ccc1F C(=O)(CCS(C)(=O)=O)NCC#CC(=O)NCC(c1ccsc1)C CC1CN(C(C2CN(C)CCN2C(=O)CCc2ccn(C)c2)=O)Cc2nncn21 CC(C)CC(O)C(=O)NCC1CCCN1C(c1nncs1)=O N1(C(CCSCCCC)=O)CCN(C(=O)C2=CCOCC2)CC12CC2 Cc1ccc(O)c(C(N2CC(C3CN(C(C4OCCC4(C)C)=O)CCO3)C2)=O)c1 c1(C(N2C(C(C)C)C(NC(C3(C)CC(C)(C)C3)=O)CC2)=O)cccc(C#N)c1 C1(NC(C2(C(=O)NC)CC2)=O)CCC2CCN(C(c3[nH]ccc3C(F)(F)F)=O)C12 N1(C(C=C(CC)CC)=O)CCCC1C(C)(C)NC(c1ccc(COC)s1)=O C(CS(=O)(=O)CC(=O)NC1CCN(C(c2cc(OC(F)F)n(C)n2)=O)CC1)OC Cc1nnc2n[nH]c(NC(c3cc(N)ccc3[N+](=O)[O-])=O)c2c1C c1(C(=O)NC2CCN(C(c3ncc(C)cc3C)=O)C2)c(F)ccc2ccoc12 C1(C(=O)NCCNC(C2CCCC2)=O)CC2(CCN(C(=O)C=CC(F)F)C2)C1 C1(CC=C)COCC1NC(=O)C(C)(C)C1CCN(C(c2cc(C3CC3)on2)=O)C1 Cc1cc(-n2cncn2)ccc1C(=O)NC(C)CCCNC(C1CCCOC1)=O CC(C)C(C(=O)NCCC(F)(F)Cl)C(C)NC(=O)C(C)N=[N+]=[N-] C1(CNC(CC#N)=O)CN(C(c2cc(C(F)F)ccn2)=O)CC12CCOCC2 C1(CC(=O)NC2C(NC(C3(COCC)CC3)=O)C2)OC(C)(C)OC1=O C#CC1(O)CCCN(C(C2CC(C)N2C(=O)COc2ccn(C)n2)=O)C1 C1(NC(C2COCCN(C(C(C(C)C)(C)O)=O)C2)=O)CCOC2(CCC2)C1 c1(CO)nc(Nc2cccc(F)c2C)cc(=NCC2CC23CCOC3)[nH]1.C1CO1 C1(CNC(CCn2ncc(C)c2)=O)CN(C(=O)CCC2CCCO2)CCCO1 Cc1c(C(=O)NC2(CO)CCN(C(C3CS(=O)(=O)C3)=O)C2)cnn1CC(F)F CS(=O)(=O)c1ccc(C(N)=O)cc1F.C1(=O)CC(c2cccs2)C(=O)N1C Cc1nc(C(=O)N(C2CCN(C(C3CCC34CCC4)=O)CC2)CC2CC2)c(C)s1 N1(C(CCNS(C)(=O)=O)=O)CC(CO)C2(C1)CN(C(=O)CC1CCCCCC1)C2 c1(OC)cc(N)c(F)cc1C(N1CCCC1CNC(C1CCC2CC2CC1)=O)=O O=C(NNc1cccc(Br)c1F)C1CCCS(=O)(=O)C1 C(c1ccc(Cl)c(C(F)(F)F)c1)=CC(=O)NCCN(C)C(C1C(F)(F)C12CC2)=O C1(C(=O)NCCC(C)N(C(=O)CCNC(N)=O)C)CCC(=O)C1 C=CCC(C)(CC=C)NC(=O)C(C(C)O)NC(=O)CCN1CCCC1=O C1(C(=O)NC2C3CN(C(C(C)NC(N)=O)=O)CC2C3)CC2CC(O)CC(C1)C2 c1(C(=O)NCC23CC(c4ccccc4)(C2)C3)c[nH]c2ccc(Br)cc12 C1(C(=O)NCCCN(C(c2c(NC)snc2C)=O)C)CCOC2(CCCCC2)C1 C1(NC(C(C)N(CC)CC)=O)CC2CC(C1)CN(C(=O)CCC1CCCCO1)C2 N1(C(C(C2CC2)OCC)=O)CC(NC(=O)CC=C(C)C)C(c2cnn(C)c2)C1 N1(C(CC(C)n2ccnc2)=O)CCOCC1C=NO.c1(C(CO)N)ccccc1 CC(C)CS(=O)(=O)CC(=O)NCCCN(CCO)C(C1CN2CCN1C(C)C2)=O c1(OC)cc(C(=O)Nc2cccc(F)c2)c(-c2cccc(F)c2)cn1.C(C#N)SC C1(C(=O)NCC(C(C)O)C)CCOCCN1C(=O)CC(C)(C)O N1(C(c2cc3ncccc3s2)C(=O)NC(C)(C)C)Cc2ccc(Cl)cc2C1 CCCCCCCCCC(O)C(=O)NC(C)C(C1CCOCC1)O CC1OCCOC1C(=O)NCC1(CO)CCN(C(C2C=CCC2)=O)C1 c1(CNC(C2CC(F)(F)CN2C(=O)Cc2ccsc2)=O)c(Br)cncc1Br CCC(C)CCC(=O)NCCNC(=O)C(C)Sc1ccccc1Cl C(=O)(CCCCN(C)C(C1CCCC1)=O)N(C(C=C)C1CC1)C C12(C(N3CCC(O)(CC)C3)=O)CC(CN(C(c3cn(CCO)nn3)=O)C1)C2 N1(C(c2ccn(CC)n2)=O)CCOCC1CC(=O)NCC(C)(O)C1CCCC1 C1(C(N2CC(COC)C2)=O)CCC(NC(=O)CSc2nc[nH]n2)CC1 CC(CCN=c1ccnc(NCc2nnc(-c3ccccc3Cl)s2)[nH]1)C(F)(F)F C1(CNC(C2N(C(=O)NC)CCC2)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC1(F)F C(=O)(CCCCCF)NCC1(CN(C(c2ccc(OCC)nc2)=O)C)CC1 c1(CC)ccc(C(N2CCOC(CN(C)C(C3(C)CC3(C)C)=O)C2)=O)c(C)n1 N1(C(C(CSC)C)=O)Cc2nccn2CC(NC(C23CC(CC(F)F)(C2)C3)=O)C1 N1(C(C(SC)SC)=O)C2CCCC1CN(C(c1cc(C#N)c[nH]1)=O)C2 C(C(CC(C)C)NC(C1CCCN1CC)=O)NC(C=CCC)=O N1(C(CC(C)(C)C)=O)CC2(CNC(c3ccc(Cl)cc3)=O)CC1CO2 C(C(C)(C)C(=O)NCC(C(C)C)NC(=O)C(C)CN1CCOCC1)NC(C)=O c1(CC(=O)NCCC(C)NC(c2c(SC)cnn2C)=O)ccc2sccc2c1 C1(C)(CNC(C(C)(C)OCCC)=O)CCN(C(C2CC2C2CC2)=O)C1 c1(C(=O)NC2C(NC(c3cccnc3O)=O)CCCC2)cc2c(nn1)OCCS2 c1(C(N2C(C)C(NC(=O)C(C)(C)O)CCC2)=O)cc2cc(O)ccc2cc1O N1(C(c2n(CC)nnc2C)=O)CC2CCC1CN2C(=O)CC1CCCCN1C C(=O)(CC1=CCN(C)CC1)NCC1CCN(C(C(Br)=C(C)C)=O)C1 N1(C(c2cnc(C)s2)=O)CCC(NC(C2(F)CCS(=O)(=O)C2)=O)CC1C c1(C(=O)NC2(CNC(C(COC)(C)OC)=O)CC2)cccc2[nH]c(C)cc12 c1(C(=O)OC)cccn(CC(=O)NCC(F)CNC(=O)CC2CCC2)c1=O c1(CN(c2ccn(S(=O)(=O)F)n2)CC(=O)OCC)cc2nn[nH]c2cc1F N(C1CCCc2c1cnn2CC1CCC(N)C1)C(C(=O)N(C)C)=O Cn1[nH]c(=NC(=O)C2CC(F)CN(Cc3cc(Cl)cnc3Cl)C2)cc1Cl CCCC(C)C(C)(c1nnnn1CC)Nc1ncc(OCC)cc1Br c1(NC(C(C)(C)Br)=O)cnc(F)cc1CNC(c1cc2sccc2[nH]1)=O C(=O)(C1CCc2ccccc21)N1CC(NC(CCc2c(C)noc2Cl)=O)(CO)C1 c1(C(N2CC(NC(CCC(C)SC)=O)C(SC)C2)=O)cc2ccc(F)cc2o1 N1(C(C(C(C)C)n2ccnc2)=O)CC(C(N2CC(O)CC2(C)C)=O)CC(F)(F)C1 c1(C(N2CC(CN(C(C=CC(CC)C)=O)C)OCC2)=O)cn2cccc(F)c2n1 N1(C(C(CC)CC)=O)CCN(N2CCC(Cc3ccc(C=O)cc3)C2)C2CC12 c1(C(=O)NC2C(CNC(C3C(=C)CC3)=O)CCCC2)[nH]c2ccccc2c1C#N Cc1ccc(N)c(C(=O)NCC23CC(NC(=O)CCC4CCC4)(C2)C(C)O3)c1F c1(C(N2CCC(OC)(CNC(=O)C=C3CCOCC3)C2)=O)cnc2ncccn12 CN1CCN(C(=O)CN2CCCC2=O)CC1C(=O)Nc1ccc(C2CC2)cc1 C(C(CC(=O)NC1(CO)CC=CC1)NC(c1nonc1N)=O)OC C1(NC(CC2CN(C)CC2O)=O)CCCCCN(C(=O)Cc2cncc(F)c2)C1 C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1CCC(NC(c2c(CC)nc(C)[nH]2)=O)C1 c1(NC(N2C(CCC(C)C)CCCC2)=O)ccc(F)c(S(N)(=O)=O)c1 N1(C(c2scc(OC)c2)=O)CCOC(C(C)NC(=O)CC2CC3CCC2C3)C1 CC(CC(C)(C)C)C(=O)N(CCCNC(=O)Cc1ncn2c1CCCC2)C C1(S(N)(=O)=O)(C(=O)NC(CNC(c2cc(C)n(C)c2)=O)C)CCCC1 c1(C(=O)NCC(CNC(COCC#C)=O)F)cc(CCOCCOC)no1 c1(OC)cccc(CC(=O)NCC2(F)CC(NC(=O)C=C(C)C)C2)c1Cl C1(NC(=O)Cn2cnc(Br)n2)CCN(C(=O)CCn2cncn2)CC1O c1(C(=O)NC2C(C)CCN(C(=O)C(C)(Cl)Cl)C2)cc2n(n1)CCNC2=O c1(CC(N2CC(C)C(NC(C3CC3C(F)F)=O)C2)=O)cccc(C#N)c1 c1(NCCCSCCCN(CC(C)O)C)cc(Br)no1 N1(C(C(C)O)=O)CC(C2CCCCN(C(c3cc(C4CC4)sn3)=O)C2)C1 N1(Cc2c(C)cccc2Cl)CCC(NC(c2ccc3nc[nH]c3c2)=O)C(C)(C)C1 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)N(CC(C1CCCC1)O)C N1(CCNC(C(c2cnn(C)c2)NC(c2c(C)non2)=O)=O)CCOCC1=O C=CCCC(c1nnnn1C(C)C(=O)OC)(C1CC1)NCc1ccccc1Cl Cc1nc(N2CCC(NC(C3CCCC(C)C3)=O)C2)ncc1Br CC1(CNC(c2ccc(C3CC3)cc2)c2nnnn2CC2CC2)CC2CCC1O2 C1(NC(C2C(OCC)C2)=O)CCCCC1CNC(c1cc(C(C)(C)C)nn1C)=O c1(NCCC2N(C(c3cnccn3)=O)CCCC2)nc(Cl)nc2[nH]c(O)nc12 c1(C(N(C(C)C)CCNC(c2sccc2C(F)F)=O)=O)cccc2c1COCC2 CC(CC(=O)N1CCOC2(CCC2)C1)C(C)(C)NC(=O)CC1CNC(=O)O1 C1(NC(c2cncnc2)=O)CN(C(=O)CC2CCC23CCC3)C2CCCCC12 Cc1cc(C)n2nc(C(=O)NCc3cn(Cc4nc(C(=O)O)cs4)nn3)cc2n1 N(C1CN(C(=O)CC(C)(C)O)Cc2ccccc21)C(CCCCCOC)=O C1(C(=O)OC)CN(C(=O)NCCCC2CC2(C)C)c2ccccc2O1 c1(C(N2CCC(NC(c3cncc(Cl)c3)=O)(CF)C2)=O)cnc2ccccc2n1 C1(CC(=O)NOC2CCOC2)CCCC12CC2.c12cn(nn1)C2 CC(Cn1cccn1)CN=c1nc(N(C)Cc2nc(=N)[nH][nH]2)c2cc[nH]c2[nH]1 N1(C(C(CC=C)(C)C)=O)CCC2CN(C(=O)Cc3nn(C)cc3[N+](=O)[O-])CC2C1 N1(C(C2CC(=O)NC(=O)N2)=O)CC2CN(C(C3CC4OC3C3CC43)=O)CC2C1 Cn1cc([N+](=O)[O-])cc1C(N1CCCC1C1(O)CN(C(C2C=CCCC2)=O)C1)=O N1(C(C(CC(C)C)OC)=O)CCC(C(=O)N(C)OCC(F)(F)F)C(C)(C)C1 Cc1ccc(C(=O)NC23CC2CN(C(=O)CN2CCC(C)CC2)C3)c(I)c1 CCCCC(CNC(c1coc(C(N)=O)c1)=O)NC(=O)Cc1cnc(C)s1 c1(C(=O)NCC(C)N(C(CCCN(C(C)=O)C)=O)C)cc(C)cc(O)c1 C1(CNC(C(C2CC2)OC)=O)CCN(C(=O)CCOCC2CCC2)C1 Cc1cncc(C(N2CCOC(CCNC(=O)Cc3ccc(C)s3)C2)=O)n1 c1(C(=O)NCC2(CF)CCC2)cncc(-n2cccn2)n1 c1(N2CCCN(C(c3cccc(F)c3I)C=O)CC2)nccn2cnnc12 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(C2(CO)CCC2)=O)CCC(C)(C)C1 c1(C(N2C3C(NC(c4nc(C)oc4)=O)CC(C3)C2)=O)c(F)ccc(Br)c1F CC(C)(O)CC(=O)NCC1CN(Cc2ccnc(N(C)C)c2)C1 N1(C(c2cc(C)sn2)=O)C2CCC1CC(C(N1CCC3(CCCO3)C1)=O)C2 C1(C(=O)NC2CC(CCNC(C3(c4cncs4)CC3)=O)C2)CCCOCC1 N1(C(C=C2CCN(C)C2)=O)CC(O)CC1CNC(=O)C(C)(C)c1ccnn1C C#CCC(C)(C(=O)N1CCC(O)C(CO)C1)NC(C1C=CCC1)=O C=CC1CN(C(=O)Cc2ccccc2COC)CC1NC(c1csc(C)c1)=O c1(-n2cc(CCCC(=O)NC(CC(CC)C)C(=O)O)nn2)c(F)c(F)cc(F)c1F c1(C(N2CCCCC2CO)=O)cc(Br)c(F)cc1Cl.N12CCC1C2=O c1(C(N2CC(F)CC(C(=O)NCC3(O)CCC3)C2)=O)ccc2c(Cl)ccnc2c1 N1(C(Cc2nc(C)sc2Cl)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 c1(NC2CCN(C(c3c(C)coc3C)=O)C2)ncc2c(Cl)cccc2n1 C(CC(C(=O)NCCc1nc(C)cs1)NC(=O)C(C)OCCOC)=CC c1(CCC(=O)NC(C)C(C)NC(=O)CC#N)cnn(-c2ccccc2)c1 c1(CN2CC3(C(C(N4CC(=O)NC4)=O)C3)C2)cc(Cl)cnc1Cl n1(CC(=O)NC(CC)CN(C)C(C2CC(F)(CO)C2)=O)nc(C)c([N+](=O)[O-])c1C C1(C(=O)NCc2ccc(C(=O)OC)[nH]2)CC12CCN(C(c1ccc(Cl)cc1Br)=O)C2 C(c1cnc(C)nc1O)=CC(=O)NC1CC(CNC(c2oc(CC)c(C)c2)=O)C1 c1(C(N2CC(CC(=O)OCC)C3(C2)CC3)=O)ccnc2ccccc12 c1(NC(=O)NCC(C)COc2ccc(Cl)cc2)nnc2ccc(C(F)(F)F)cn12 CCC(C#N)C(=O)NC1(C(=O)NC2C=C(C)CCC2)CCOCC1 N1(C(CC(=O)NCC#C)=O)CCN(C(=O)CCn2cc(C)cn2)CC1C#C c1(C(N2CCC(NC(c3cc(OC)ncc3)=O)(CF)C2)=O)ccc(C#N)nc1O c1(C(=O)NC2CCOCC2NC(C2CSCCS2)=O)ccc2nn[nH]c2c1 CC1CN(C(C2(CCF)CCC2)=O)CCC1NC(C1CN(S(=O)(=O)C(F)F)C1)=O Cn1c(-c2nc(C(C)C3CC3)nn2CCCC(F)F)cc2ccsc12 Cc1ncc(C(=O)NCCc2cn(CC3CCC4CC4C3)nn2)c(O)n1 Cc1cc(C(=O)NCC2CCCN2C(C2C=CCCC2)=O)n2ncnc2n1 C1(C(=O)OC(C)(C)C)CC2(C1)C(NC(=O)C1=CC3C=CC(C1)C3)C21CCC1 CCCC(O)C(=O)NCC(CC)NC(=O)CC1(C(F)F)CC1 N1(C(C(C)=C2CC2)=O)CC(CNC(c2ocnc2-c2ccccc2)=O)CCC1C c1(CN(CC(=O)NCC(=O)NC2CC2)CC)ccc(Cl)cc1 N1(C(c2c(C)[nH]c(=NCC)s2)=O)CCC2(CC1)CC(NC(C1CC3(CC3)C1)=O)C2 CC1(C)CCC(C(=O)NC2CCCC2C(=O)NCc2ccc(O)c(F)c2)CC1 N1(C(C2C(=C)C2)=O)CC(O)(C2(CNC(c3ncc(Br)cc3OC)=O)CC2)C1 C1(C)(C(N2CC(C)(NC(C3C(CC)CCC3)=O)C2)=O)CCC(=O)NC1 N1(C(c2c(C)ccnc2)=O)CCC(C)N(C(c2cnc(C3CCC3)o2)=O)CC1 c1(C(=O)NCC(CC)NC(=O)CN2CCCCCC2)cnc2n1CCCCC2 CC(C)C(C#N)C(=O)NC1(C(N2CCCC(CN=[N+]=[N-])C2)=O)CC(F)C1 Cc1cc(Br)c2ncnc(NCc3sccc3C(F)(F)F)c2c1 c1(C(=O)NC2(C)CN(C(C(CC)Sc3ccccc3)=O)C2)nc(C(F)(F)F)sc1C C1(COC)CC(CNC(=O)C(c2ccc(Cl)cc2)=O)N(C(=O)Cc2cn[nH]c2)C1 c1(OC)ccc(C(=O)NC2CCCN(C(C3CC3C(C)C)=O)CC2)cc1O CC1CCN(C(=O)COC2CCC2)C(CNC(C2CCC3(CCC3)C2)=O)C1 Cc1nc(Cl)c(NC(C2CC(F)CN(C(=O)C3CC3)C2)=O)c(Cl)n1 N1(C(C2CC(N(C)C)C2)=O)CCC(C(N2CCC3(CCCO3)C2)=O)CC1(C)C c1(C(N(C2CC(NC(C(C)CC3CC3)=O)C2)C)=O)cc2n(c1)CCOC2 c1(N2C(C(=O)NC(c3ccc4c(c3)OCCO4)C)CC2)ncnc2cccnc12 c1(OC)nscc1NC(=O)CC1(C)CCN1C(=O)C=CCN1CCC1 N1(C(CCOCC)=O)CCC2CCN(C(=O)C(c3ccccc3F)(C)C)CC2C1 C1(CN2CCN(C(c3cc(C)on3)=O)CC2)Cc2ccccc2C1C C1(CC)CN(c2nnc(C(c3ccccn3)(F)F)n2CCC(=O)NC)CC(C)O1 c1(OC(C)C(=O)N(C2CCN(C)C2=O)C)c(Cl)cc(I)cc1Cl C(=O)(C(=O)C(F)(F)F)NC1C(NC(C(C2CCC(=O)N2)C)=O)CCCC1 C1(NC(c2cccc(OC)c2)=O)CCN(C(=O)Cc2ccc(O)cn2)C(C)C1 c1(CC(=O)NC2CC(CN(C(C3C(COC)C3)=O)C3CC3)C2)c(Cl)cnn1C CC1CN(C(=O)CC2CCCN2Cc2ncccc2Br)CC(=O)N1 CC1CN(C(=O)CC(C(F)(F)F)c2ccccc2C(F)(F)F)CCC12CCOC2 C(=O)(CC1CCc2ccccc21)N1C(C)(C)CC(NC(=O)CCCC2CCC2)C1 C#Cc1cnn(CC(=O)NC(CNC(=O)COCCc2cccs2)(CC)CC)c1 C1(C(=O)NCC(CCNC(C2C(=C)C2)=O)O)(OC)CCC(C)(C)CC1 N12CCC(C)(C)C1C(=O)NON1CCC(C1)C(C)C2=O.C(=O)C(C)C1(O)CCC1 C1(C)(C(=O)NC(C)C2CC2)CCCN(Cc2ccnc(-c3ccccn3)c2)C1 c1(N(CC2=CCSC2)C)nc(=N)[nH]c(=NCCc2csc3c(Cl)cccc23)[nH]1 C1(N(C(c2c(-c3cncc(C)c3)nccc2)=O)C)CCCCN(CCO)C1 C(CC)(CCCC(=O)NCC[Si](C)(C)C)NC(C1(CC=C)CCC1)=O CCCCCCC(=O)N1CCC(C(C)C(=O)NCC2(C)CCCO2)CC1 C12(C(=O)NC3CC4C(NC(CCC(=O)N(C)C)=O)C4C3)CCCN(CC1)C2 N1(C(c2nc(CCC)sc2)=O)CCn2c(CNC(C3C=CCC3)=O)nnc2C1 N1(C(CCOCCOC)=O)CCC(O)(CCNC(c2cc(C(N)=O)cn2C)=O)C1 c1(C(=O)NCC23OCC(NC(C(C=C)O)=O)(C2)C3)cc(F)cnc1O C1(C(=O)NCCC(CNC(CSc2cccc(C)c2)=O)O)CN2CCN1C(C)C2 N1(C(CC(C(C)C)NC(c2ccc(CC)s2)=O)=O)CCC2(CCC2)C(O)C1 c1(SCC(N2CC3C(NC(C=CC(=O)OCC)=O)(C3)C2)=O)ccc(C)cc1C Cn1cc2c(C(=O)NC3CCCC3NC(=O)Cc3cnsc3)cc(F)cc2n1 CC1CC(NC(c2ncoc2C(C)(C)C)=O)CN(C(=O)C=C2CCN(C)C2)C1 N1(C(C(C(C)O)N(C)C)=O)CC2(C1)SCCC2NC(c1cc2cnccc2o1)=O N1(C(C(CC)C#N)=O)CC(C2CCCN(C(=O)CNC(c3ccco3)=O)C2)C1 N1(C(C2C(CC)C2)=O)CCC(CF)(NC(=O)C(C)Cc2ccccc2F)C1 CCCCC(C(=O)N(C)CC1CCCN1C(c1ccc(O)c(Cl)n1)=O)NC(N)=O C1(C)(CC(=O)OCc2c(O)nc(C)c(Br)c2)Oc2ccccc2O1 C1(NC(CCOCC(C)C)=O)C=CCCC1C(=O)NC1CC1(C)C(F)F c1(C(N2CCC(C(=O)Nc3ncc(C)nc3Cl)C(O)C2)=O)ccc(I)c(F)c1F c1(CNC(C2(OC)CC(C)C2)=O)ncccc1C(=O)N(C1CCSCC1)C Cc1sc(C)c2sc(C(=O)NC3CN(C(=O)CCCC(N)=O)CC4(CC4)C3)cc12 N1(c2ccnc(NC3C(CCCC)CCC3)n2)CCC2(CC1)CCN(C)C2 C1(C)(CC(=O)N(C(C2CCCCC2)C)C)CCN(C(=O)Cc2ccc(O)cc2)C1 C1(C(N(CC(CC)NC(c2cn(C)c(O)n2)=O)C)=O)CCNC(=O)C1 C(=O)(C1=COCC1)NCC1N(C(C)C)CCC1.C12(CCC1)C(=O)N2C1CC1 N1(C(C2C(OCC)C2)=O)CC2C(N(C(=O)CCc3ccsc3Cl)C)C2C1 N1(C(c2nc(CC)oc2C)=O)CCCC1C1CCCN1C(c1cccnc1C)=O N1(C(CC2CCN(C(C3(C)CNC(=O)N3)=O)C2)=O)CC2CC(O)CC1C2 c1(OC)cc(C(N2CC(O)(c3ccccc3)C2)=O)sn1 C#CC(CC(C)(C)C)NC(=O)C(CCOCCO)NC(=O)Cc1ccccc1C Cc1cc(C(=O)N(CCC(C)NC(C2CCC(=O)N2C(C)C)=O)C)oc1C N1(CC)CCN(N2CCC(S(=O)(=O)CC=O)CC2)CC1.N(C)(CC)CC Cc1nc(O)sc1C(=O)NC1CCCCC1CNC(c1cc(C(N)=O)c[nH]1)=O C(=O)(C(=O)N=S(C)(C)=O)NCCN(C(c1ccc(CN(CC)CC)o1)=O)C1CC1 CCC(C)(CCC(C)C)C(=O)N1CCCCC(NC(C2CN3CCN2CC3)=O)C1 C(=O)(C(O)C1=CCCCC1)NCC(C)(CO)NC(C1CC(CC(F)(F)F)C1)=O S(=O)(=O)(c1cccc(C#N)c1F)Nc1sc2ccc(C)cc2n1 c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC(F)C2)=O)cc2cccnc2[nH]1 Cc1nn(C)c2nc(C(=O)NC3CCC(CNC(c4ccccn4)=O)C3)ccc12 S(=O)(=O)(c1cc(F)c(F)c(F)c1F)C(NNC(c1c[nH]c2ccccc12)=O)=O CC12CCC(C(=O)NCC3CN(C(c4csc(-c5ccncc5)n4)=O)C3)(C1)OC2 CC(C)(CCCNC(C1COCOC1)=O)C(=O)N1CC(CO)C(O)C1 C1(NC(CCOCC)=O)CCCN(C(=O)Cn2cnc(C(F)(F)F)n2)CCC1 C(C)(C(=O)NC1CC(OCC(=O)N(C)CCc2cccs2)C1)OCOC C1(CC(=O)N(C)Cc2nc(C)[nH]n2)CCCCN1C(c1n[nH]cc1Cl)=O c1(OCC)ccc(CNN2CCC(O)(C(C)C)C2)cc1-c1cc(F)ccc1C C1(NC(C2CC23CCC3)=O)CCN(C(=O)CCC2CCOCC2)C(C2CC2)C1 c1(-c2n(C3C(C)OCC3)nc(CCN3CCCCC3)n2)noc2c1CCCC2 c1(OCC)ncccc1C(=O)N(CC(C)CNC(c1cnn(CC(F)F)n1)=O)C c1(-c2cc(C)c(O)cc2)ccc2ccnc(NCc3cn[nH]c3)c2c1 C1(N(C(c2n(CC)cnn2)=O)C)CN(C(=O)C=Cc2cn(C)nn2)CC1(C)C CC1C(NC(=O)CC2OCCOC2(C)C)CCCN1C(c1nn(C)cc1Cl)=O Cn1cncc(C(N2CCC(CO)C(NC(=O)CC3CS(=O)(=O)C3)C2)=O)c1=O C(C(C)(C)C(=O)NC(C)CC(C)NC(C1CN(C2CCC2)C1)=O)NC(C)=O N1(C(=O)NCC2CCCNS2(=O)=O)CCOC2CCN(C(C)(C)C)CC12 c1(OC)cc(O)ncc1C(=O)NC1CCCN(C(C2CCCCC23CC3)=O)C1C C(=O)(C1=CCCCC1)NC(CNC(c1c(C)cnn1C)=O)(C)C1CC1 C1(NC(=O)CCC(F)F)CN(C(=O)C=C2CCCCCC2(F)F)C2CCCCC12 N(C(=NCCCF)N1CC=C(F)C1)CC(C(C)C)CCc1ccccc1 c1(C(=O)NCC2N(C)CCN(C(C3CC4(CC4)C3)=O)C2)[nH]cc2c1CCCC2 N1(C(C2C(C(C)O)C2)=O)CCC(NC(c2cncc(Cl)c2Cl)=O)C2(CCC2)C1 c1(C(C(=O)NC2CCOC2)N(C(CC=C)C)CC)cnc(C)[nH]1 CCCC(C)(O)C(=O)N1CCC(C2CCCN2C(=O)Cn2ccnn2)CC1 c1(C(=O)NC2C=CC(CNC(=O)COCCCF)C2)ccc(O)c(F)c1 N1(C(CCC2(C)CC2)=O)CCC(c2nnc(CNC(=O)CC(C)(F)F)s2)CC1 N1(CC(CC)C)CCC2CCC(C1)N2C(=O)Cc1c(F)cccc1Cl c1(C(=O)NC2CCN(C(c3cccnn3)=O)C2)ccc(C(F)(F)F)nc1O c1(C(N2C(CN(C)C(C3(F)CCOC3)=O)CCC2)=O)ccc2c(c1O)CCCC2 C(C)(C(=O)N1CCC(CC(C)NC(c2ccnc(F)c2O)=O)CC1)(C(C)C)OC c1(C(=O)NCC2CCN(C(C=CCCC)=O)C2)ccc2ccc(Br)cc2n1 C1(NC(CCc2ccc(C(=O)NC(CCC)CCO)[nH]2)=O)CCC(F)(F)CC1 CC(CC(=O)NC1CC(C)N(C(=O)COc2ccn(C)n2)C1)CC(F)(F)F CCCCCCC(C(=O)NCCN(C(c1c[nH]c(=N)s1)=O)CC)NC(C)=O c1(CC)cc(CNC(C2CC(CNC(COC(=O)N)=O)C2)=O)no1.C(C)(C)C Cc1cc(C(=O)NCCOC2CN(C(=O)CCNC3CC3)C2)c(C(F)(F)F)o1 C#CC1(C)CCCN(C(C2C3CN(C(C4(O)CCOCC4)=O)CC23)=O)C1 CCCC(C(=O)NC1CN(C(c2cc(C(F)(F)F)cs2)=O)CCC1C)C(C)C c1(C(N(CC(CCC=C)O)C)=O)cc(C#N)cc(C#N)c1 c1(CC)cccc(NC(c2c(CNC(C34CC(CO)(C3)C4)=O)cncc2)=O)c1F C(CCN=c1nc2scnc2c(N(CC(C)(C)CO)C)[nH]1)N1CC(C)OC(C)C1 Cc1cncc(CNC(C2CC(O)CN2C(=O)C=C2CCOCC2)=O)c1 N1(C(=O)Nc2ccc(SC)s2)CCCC2C1CCN2C(=O)CC1CCN(C)CC1 c1(CC2N(C(C(C)N(CCC)C3CC3)=O)CCC2)cccc2ccccc12 C12(CNC(C(C(C)O)C)=O)CN(C(=O)Cc3ccc4c(c3)OCC4)CC(F)(C1)C2 C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)cccc2)=O)CC2C(C1)C2(F)F C1(NC(C(C)n2cccc2)=O)CCOCC1NC(=O)COCc1cnn(C)c1 C1(C(=O)NCCN(C(CCCOCC)=O)C2CCCC2)Cc2cccnc2C1 N1(C(CNC(=O)OC)=O)CCC(C(C)NC(c2ccnn2C2CCC2)=O)C1 c1(NC(C2(C)CCN(C(c3c(Cl)cccc3Cl)=O)C2)=O)c(O)ncnc1O O=C1CC(C(=O)NCC2(O)CC(NC(=O)CN3CCSCC3)C2)C2(CCC2)C1 CCC(CC)C(C(=O)N1CCCC(NC(c2cnoc2C(C)C)=O)C1)OC c1(C(N2CCC(C(C)NC(C(CC)NC(C)=O)=O)C2)=O)c(Cl)nn(C)c1Cl Cc1ccc(C(=O)NC(c2ccccc2)C(=O)NC2C3COCC23)nn1 c1(N2CCCC(C)(CC)CC2)cc(Br)ccc1S(=O)(=O)NC(CO)C1CCC1 c1(C(N2C(CNC(C(CSC)OC)=O)CC(OC)C2)=O)cn2ccc(F)cc2n1 C1(C(=O)OCC2CCC3C(C2)C3(F)F)C(F)(F)C12CC(C(=O)OC)C2 N1(C(C2CC(O)C(F)C2)=O)CC2CCC(C1)N2C(C1CC(n2ccnn2)C1)=O C1(C(=O)NC2CC(C#C)C2)CCN(C(=O)OC(C)(C)C)C12CCSCC2 c1(CC(N2CCCC(NC(CC3C(C)=NOC3=O)=O)C2)=O)c(O)nc(=N)[nH]c1C N1(C(C2N(CCC)CCC2)=O)CCOC(C(N2CCC(F)CC2)=O)C1 c1(OC)cc(C(F)F)c(C(N2CCCC2CNC(C2CCC(C)CC2)=O)=O)cn1 C1(C(=O)NC2CCN(c3snc(CCOC)n3)CC2O)Cc2ccccc2CO1 CCC(CNC(c1cncc(O)c1)=O)(CC)C(=O)NCC(C)(C)C(C)(C)O C1(CC(N2CCC(CN(C(=O)CC3C=CCC3)C)CC2)=O)CCCCC1(F)F c1(C(N2CCC(c3ccc(OC)cc3)C2)=O)cc(SC)c(Cl)cc1Cl C1(CC)CN(C(=O)CN(c2ccncc2)C)CCN1C(=O)C(C(C)C)OC C1(C(=O)NCC(CN(C(C(CC)F)=O)C)C)CCc2ccccc2O1 c1(NCCNC(=O)NC)nc2ccccc2nc1NC(C1COC(=O)N1)C C1(NC(C23CC(C)C2C3)=O)(CNC(c2cccc(CC#N)c2)=O)CCOCC1 c1(C(N(C2CCC(NC(=O)C(F)=CCCF)C2)C)=O)ccc(P(C)(C)=O)s1 C1(N(C(CCN(C(C(F)=CCC)=O)C)=O)C)CC(C)OC(C)C1 Cc1ccc(Cl)c(OCC(=O)NC2CC(NC(=O)CC3CCC3C3CC3)C2)c1 c1(C(N(C)CC2COCCN2C(=O)CCCC#N)=O)cn2c(n1)CCCC2 N1(C(C(C)CO)=O)CC23CCCCC2(C1)CN(C(=O)C(C1CCCCC1)O)C3 c1(OC)cc(OC)c(C(=O)NCC2CC(F)CN2Cc2ncc[nH]2)cc1Cl c1(C(=O)NCCN(C)C(C23CCC(CC2)CO3)=O)cc([N+](=O)[O-])ccn1 N#Cc1ccc(-c2cnn3cc(C(=O)NCc4ccc(O)nc4)cnc23)cc1F c1(CCC(=O)N(CC(C)NC(C2C3CCC23)=O)CC)ccccc1F N1(C(C2(Cl)C(C)(C)C2)=O)CCC2(C1)CN(C(C1CNC(=O)N1)=O)C2 N1(C(c2cc(OC)cc(F)c2)C(=O)Nc2ccccc2)CCOCC1P(C)(C)=O C1(C(N(c2ccccn2)CCC(N)=O)=O)CCN(C(c2sccc2Cl)=O)CC1 Cn1c(C(=O)NCC2CCOC2C(=O)NC2CC(C(C)(C)C)C2)cnc1Cl c1(C(=O)NC2CC(F)(CNC(c3cnsc3)=O)C2)cncc2[nH]ccc12 c1(C(=O)NC23C(CN(C(c4cccc(CC)c4)=O)C2)C3)cc2ccsc2c(O)n1 C(CC(C(=O)NC1CC(C)C1)NC(=O)CCc1nc(O)n[nH]1)OC N1(C(C2(C)CC(OC)(OC)C2)=O)CC2CCCC2(CNC(=O)CC2CC=CC2)C1 CC1C(=O)NC(=O)CN1C(=O)C(CO)NC(c1ccoc1Br)=O C1(C(N2CC(NC(C(C)N3CCCC3)=O)C(F)C2)=O)CC(C)(C)CN1C c1(C(N2CCN(C(C3CCC(F)(F)C3)=O)CC2)=O)ccc(I)cc1[N+](=O)[O-] C(CC(C)C)(C(=O)NCCCCC1CC1)N(C(C(C(C)C)NC(C)=O)=O)C Cc1cnc2ccccc2c1C(=O)NCC1(O)CC(NC(=O)CNC=O)C1 C1(C(N(CCCOC(C)C)C)=O)CC(C)(C)CN1C(=O)CC1COCCO1 CC1CN(C(c2ccccc2C(N)=O)=O)CCN1C(c1cccnc1N)=O c1(OC(C)C)cccc(SC(c2nnc(C(N)=O)n2C)C)c1 C1(NC(C(=O)Nc2c(C)occ2)=O)(CO)CCCN(C(=O)C(C)CSC(F)(F)F)C1 c1(C(=O)NC(CN(C)C(c2sc(N(C)C)nc2Cl)=O)(C)C)ncccc1C1CC1 c1(CN2CCC(Nc3nc(OC)c(F)cn3)CC2)cccc([N+](=O)[O-])c1 n1(CC(N2CCCC(C)(CNC(C(CCC)O)=O)C2)=O)c(C)nc2ccccc12 c1(CC)cnccc1C(=O)N(CC(C)(C)CNC(=O)C(C)C1CCOC1)C N1(C(CC(=O)OC)=O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)C(C2CCC2)C1 C1(F)(C(N2CC(CC(=O)OC)C2)=O)CN(C(=O)C(C)NC(=O)C2CC2)C1 c1(-c2nc(CN(C(=O)C(=O)NC3(C)CCCC3(F)F)C)sc2)cccc(C#N)c1 Cc1nc(C)n(O)c1C(=O)NCC1(C)CCCC1NC(=O)C=Cc1cnc[nH]1 CC(C)C(C(=O)NCCc1cncs1)C(C)NC(c1ccsn1)=O c1(N(C(C)=O)C(C)C)ncnc2c1nc(NC(c1ccccc1Cl)C(=O)O)n2C N1(C(CCCOCC=C)=O)CCC2(CCC2)C(NC(=O)CC2CCC(=O)C2)C1 C1(CNC(C(C)=C(CC)C)=O)CCCC2CN(C(c3ccsn3)=O)CC12 C=C(Cl)CCC(=O)NCc1cccc(C(=O)NCC2CCC(C)(C)O2)n1 c1(NCC#N)cc[nH]c(=NCCCNC(c2cnn(C3CC3(F)F)c2)=O)n1 C1(CNC(CCC)=O)CCCN(c2ncc(O)cn2)C1 C1(O)(C(=O)NCCC2N(C(C(C)=CC)=O)CCC2)CCCCCC1 C(C(=O)NC(COC)CC(=O)N(C)Cc1ccccn1)(C(C)C)OCC N1(C(C2C(C)(C)C2)=O)CCCC1(C)CNC(c1cc(Br)ccn1)=O C1(NC(COC)=O)CC2(CCN(C(c3ccnc(N(C)C)c3)=O)CC2)C1 C(=O)(C1=CC2(CCOC2)C1)N1CCCC(CCNC(CCCC#N)=O)C1 c1(OC)ccc(Br)c(CS(=O)(=O)NC(C)(CN)C2CC2)c1 C(=O)(CC(C)(C)CNC(C1CC(C)(C)C1)=O)NCC(C)O C1(NC(CN2CCN(C)CC2)=O)CN(C(=O)C(C)(C)n2cnnn2)CC1N=[N+]=[N-] BrC1=Cn2c(-c3noc(COC4CCCCCC4)n3)nc(n2)C=C1 C1(O)(C(=O)NCC2(C)CCCN(C(CC(=O)NCC)=O)C2)CCCC(C)(C)CC1 C1(C(=O)NCC2(F)CN(C(c3n(CC#C)ccc3)=O)C2)CCCCC1(F)F N1(CC(N2CC(F)(CNC(C3C(=O)NCC3)=O)C2)=O)CCCC(N(C)C)C1 C12(C(=O)NC3CC(NC(c4c(NC)nccc4)=O)CC3O)CCCN(CCC1)C2 Cc1cccc(C2(C(CNC(c3ccc(C)n3C)=O)NC(=O)C(C)(Cl)Cl)CCC2)c1 C1(NC(C=C2CCC(C)C2)=O)COC2(CCN(C(c3cc(O)nc(O)n3)=O)CC2)C1 c1(NC(C23C(CN(Cc4ccc(C(=O)OC)cn4)C2)C3)=O)ncc(Cl)cc1F C1(OC)(CNC(=O)Cn2cc(CNC(c3sc(C)cc3Cl)=O)nn2)CCCSC1 C(=O)(CC1CCCc2oc(C)nc21)N(CCN(C(C1CCC1CF)=O)CC)CC CC1=C(C(=O)NC2(CC(=O)NCc3cncc(C#N)c3)CCC2)CCC1 CC(C)C(C)CC(=O)NCC(CC1CC1)C(=O)NC(c1cc[nH]n1)(C)C n1(CC(=O)NC2CC(NC(C=C(CCC)C)=O)C2)c(C2CC2)nc2ccccc12 C(=O)(N1CCCc2nncn21)C1C(NC(c2c(C(N)=O)coc2)=O)CCCC1 c1(C(N2CC3(OCC(NC(CC4(C)CC4)=O)C3)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(Cc2cccc(C)c2F)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 C12(CNC(=O)CCCCCF)CCC(CNC(=O)CC3CC4CC4C3)(CC1)OC2 c1(CC)ccccc1C(N1CCC(N(C(C2CCCS2(=O)=O)=O)CC)CC1)=O C1(NC(C(c2c(C)noc2C)C)=O)CC2CCC1N(C(c1n[nH]c(=N)[nH]1)=O)C2 N1(C(COC)=O)CCOCC1C(=O)NCc1ncsc1-c1ccccn1 c1(C(=O)NCC(CC=C)NC(=O)CC=C(Cl)Cl)cc2cccc([N+](=O)[O-])c2[nH]1 N1(CC2N(C(=O)Cn3cc(CNC4CCCCC4)nn3)CCC2)CCCS1(=O)=O CN1CCCC12CCN(C(C1(CNC(c3cnc(=N)[nH]c3)=O)CCCO1)=O)C2 c1(C(=O)NC(CCOC)CNC(=O)CCn2ccnn2)cc(Br)cnc1O C(=O)(CC(C(F)(F)F)OC)N1CCC(NC(C(CSC)OC)=O)C(C)(C)C1 N1(C(c2cc(OC)n[nH]2)=O)CC2CC(NC(=O)CC(F)(F)C(F)F)C(C2)C1 N1(C(c2cccc(N)n2)=O)CCC2C(C1)CN2C(=O)CCOC1CCOC1 Cc1cc(Br)cc(C(=O)NC2CCN(C(=O)C3=CCS(=O)(=O)C3)C2)c1C c1(C(=O)NCCC2CN(C(C(C(C)C)F)=O)CC2C)nc2c(s1)COCC2 c1(C(N2C3C(NC(C4C(COC)C4)=O)CC(C3)C2)=O)cc(OC(C)=O)cc(F)c1 C1(CNC(C(COC)COC)=O)CN(C(c2cc(C(F)F)cs2)=O)C(C)(C)C1 CCC(C)C(C(=O)N1CC=C(C(=O)N(CC2=CCSC2)C)C1)N(C)C S(=O)(=O)(c1ccc(=NCC2CC2(Cl)Cl)[nH]c1)NCCc1ccc(N(C)C)c(F)c1 N1(C(C2CC(O)(CNC(c3cc(C)sn3)=O)C2)=O)CCC(C2CCC2)CC1 CCCC(C)(O)CC(=O)N1CCN(CC(C)NC(c2cc(CC)ccn2)=O)CC1 C(=O)(CCP(C)(C)=O)NCCCCC1CN(C(C2CC(C)C2)=O)C1 C1(C(=O)NC(c2ccccc2)c2cnco2)CC12CCN(Cc1cnsn1)CC2 c1(C(=O)NC(CC)CNC(c2nn(C)nc2Br)=O)ccc(C#N)nc1O C1(N(C)C(C2COC(=O)N2C)=O)CN(C(C2(CC(F)F)CCC2)=O)CC1(C)C CC1CN2CCN1C(C(=O)NCC(C)CNc1ccc([N+](=O)[O-])cc1)C2 C1(C(=O)NC2C(NC(CCOCC)=O)CCCC2)Cc2cncn2C(=O)N1 C(=O)(CCC(C)(C)C(=O)OC)NC1CCCC(NC(c2c(OC)cncc2)=O)C1 N1(C(CNC(=O)OCC)=O)CCN(CCCN2CCCC2C)CC1 C(CCC(O)C(=O)NCC1(C(=O)NCCCc2nncs2)CC1)OCC C1(CNC(c2nc(C3CC3)cs2)=O)COCCN(C(c2cc(O)cc(Cl)c2)=O)C1 C#Cc1ccc(C(=O)NC(CNC(=O)CC2CCCS2(=O)=O)CC(C)C)cc1F c1(C(=O)NC(C(CO)NC(CC2N(CC)CCC2)=O)C)cc(Cl)cc(Cl)c1 N1(C(C(=O)NC(=O)NCC)C)CCC(NC(c2cnn(CC)c2)=O)C(C)(C)C1 N1(C(CN(S(C)(=O)=O)C)=O)CCOC2(C1)CN(C(C1(C)CC1(F)Cl)=O)C2 c1(CC(=O)NCC(C)N(C(c2cc(C)sc2C)=O)C)cccc(S(C)(=O)=O)c1 N1(C(C(CC)NC(C)=O)=O)C2CCC1C(CNC(=O)C=C1CCSCC1)C2 C1(NC(CSCCOC)=O)CCN(C(=O)CCc2cccc(OC)c2F)C1(C)C c1(C(=O)NC2C(C(C)Nc3cnn(C)c3)C2)ccc(S(C)(=O)=O)c(Br)c1 C(C(C(=O)NC1CCC(NC(=O)C(C)(C)O)C1)NC(C)=O)OC c1(C(N2C3C(NC(C(C)n4cnnn4)=O)C(C3)C2)=O)ccc(O)nc1Cl CCC(C(=O)N1CCSCC1C(N1CCC(C(N)=O)CC1)=O)C(C)C C#CCCCC(=O)N(CCNC(c1ocnc1Br)=O)C1CC1 N1(CC(=O)N(C2CCS(=O)(=O)C2)CC)CCC(C2CC2(F)F)CC1 C(=O)(C(O)P(C)(C)=O)N(CCN(C(C(CC#C)O)=O)C)C c1(CC(=O)NCCN(C(C)C)C(C2CCN(C)C2C)=O)ccc(O)cn1 C1(NC(C(C)C)=O)C2CC1N(C(=O)CC1CC1)C2 C1(CN(C(C(C)CO)=O)C)CC(F)CN1C(c1ccnc(OCC2CC2)c1)=O c1(N(CC)Cc2cc(C)on2)nnc(CC(C)(C)O)n1CCOc1ccccc1 c1(CN2C(C(=O)NCCC3(C)OCCO3)CCCC2)cccc2nonc12 CCCCC(C)CCC(=O)N(C(C)CNC(c1cnc2n1CCCC2)=O)C C(=O)(C(CC(C)C)C(C)C)NC(CC(=O)NCC(CSC)(C)C)C(F)F C1(C(N(C2CCCCN(C(c3ccc(Cl)cc3O)=O)C2)C)=O)Cc2nccn2C1 C1(NC(CC(CC)(F)F)=O)COC2CN(C(=O)C(C(C)C)NC(N)=O)CC12 C(=O)(CC1=CCCCC1)N1CCC(C=C)(C(=O)NCC(F)(F)COC)C1 c1(OC)ccc(CN2CCC(F)(C(=O)Nc3cncc(C(F)(F)F)c3)C2)cc1I C1(CNC(=O)C2CC2)CC2CCC(C1)N2c1ccnc(C(F)F)n1 c1(C(=O)NCCN(CCC)C(C2(C)CC(C3CC3)=NO2)=O)ccnn2ccnc12 O=C1CC(C(=O)NC2CCCCC2C(=O)NC2(c3nccs3)CC2)=NN1 c1(C(=O)NC2C(NC(C3(CC)CC3)=O)CCC2)ccc2c(c1)CCS2(=O)=O N1(C(c2c(OC)cc(OC)c(Cl)c2)=O)C2CCCC1CN(C(C1CC1C)=O)CC2 C=CC1(C(N2CC(N(C)C)C(C)C2)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC1 C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1ccnn1C)NC1CN(CC)C(=O)C1 Cc1csc(C(C)C(=O)NCC2CCCC2NC(c2cnc(C(C)O)s2)=O)n1 c1(-c2nc(-c3c(C)ccnc3)n(C3CCOC3)n2)c2ccccc2nn1C Cc1nc(CNC(c2ncoc2CNC(C2(CO)CCCO2)=O)=O)oc1C N1(CC(N2C(CNC(C(c3cccc(Cl)c3)OC)=O)CC2)=O)CCCCCC1 C1(C(=O)NCCC2N(C(c3c(C)ocn3)=O)CCCC2)CCn2c(C)cnc2C1 C1(NC(=O)Cn2cncn2)CCC12CCN(C(=O)CN1CC=CC1)CC2 Cc1cc(C(N2CCC(NC(=O)N(C)C)CC2)C(=O)NCC2CCOC2)cc(Cl)n1 C1(C2CCOCC2)(C(=O)NCC(CC)NC(=O)C=Cc2ccoc2)CC1(F)F c1(C(=O)NCC(C)(C)CNC(=O)CCNC(=O)CO)ccc([N+](=O)[O-])o1 C=CCC(C(=O)N1CC(C)(C)C1C1CC1)NC(C1CCC(N(C)C)C1)=O C(C1OCCc2sc(I)cc21)SCCNC(c1ccc(C)cc1)=O CCCC(C)(C)CC(=O)NCCC1(O)CCN(C(=O)CC(C)CC(C)C)C1 C1(CNCCC(c2ccnn2C)C)CC2CC1(CO)C2 C(=O)(C1Cc2ccc(Cl)cc21)NC(CNC(c1c(C)c(F)ccc1)=O)C(C)(C)C c12cc(N)ccc1S2.C(CCCOC(=N)O)NC(CC1(C(=O)OC)CC1)=O c1(-n2c(C(n3ccnc3)CC)nc(C(C)C3CC3)n2)cc(F)ccc1F C=CCC(C)(C)C(=O)NC(C)C(C)NC(c1ncoc1C1CC1)=O C(=O)(CS(=O)(=O)N1CCC(CC(=O)NCc2cc(CC)n[nH]2)C1)OCC C12(NC(CCCC3C(C)C3)=O)CCC(CC1n1cc(-c3ccnn3C)nn1)C2 c1(C(=O)NCCCC(C)NC(c2ccc(CCCC)cc2)=O)c(F)cccc1Cl c1(C(N2C(C)CC(CNC(=O)C(F)(F)C3CC3)C2)=O)ccc2[nH]ccc2c1 N1(C(C(C=C)O)=O)CC(OC)CC1Cc1ccc(CNC(=O)OC(C)(C)C)cc1 CN1CC(NC(c2ccnc(CNC(=O)CCc3ccncc3)c2)=O)C(O)C1 Cc1cc(S(N)(=O)=O)oc1C(N1CC2CC1CN2C(c1cnc(O)o1)=O)=O CC(C)(F)CC(=O)NCCCCCc1cn(CCC(=O)N(C(C)(C)C)CC#N)nn1 N1(C(CC2CC(OCC)C2)=O)CC(NC(=O)CN2CCCCC2)CC1(C)CC c1(CC)nc(C(=O)NC2C=CC(CNC(c3cnncc3O)=O)C2)c(N)s1 N1(C(Cc2cc(C)[nH]n2)=O)CC2(CCN(C(c3cnn(C(C)C)c3F)=O)C2)C1 C1(CSC)CCc2nc(C)nn2C1.N12CC(C1)NC(=O)C1(CC1)C(=O)CC2=O C(CC(C)C)(C(C(=O)NC1CC(F)(F)C1)N(c1ccc2[nH]ccc2c1)C)SC CC1(C)OCCN(C(C2C3CCCCC23)C(=O)NC2CCOCC2)C1(C)C CC(CN1CCOCC1)C(=O)N1CC(OCCNC(C2(CCC#N)COC2)=O)C1 c1(C(C)C)nn(-c2ccccc2)cc1NC(c1csc(C2CCOC2)n1)=O c1(C(=O)NCC2C(NC(c3ncc(OCC)nc3)=O)C2)cc2cccc(F)c2o1 CCC(C)C(CC(=O)N1CC(CNC(=O)C(CO)NC(N)=O)CC(C)C1)OC c1(OC)cccc(F)c1CN1CC2C(C(=O)Nc3cccc(C)c3F)C2C1 Cc1c(C(N2CCC(C)(CCNC(=O)CN3CC=CC3)C2)=O)noc1C1CC1 C1(C(=O)NCCOC(C)(C)CNC(=O)Cc2ncc(Cl)s2)CCCN1C=O C1(N(C(CCCCC)=O)C)CN(C(c2c[nH]cc(F)c2=O)=O)CCC1C Cc1ccc2c(C(N3CCC(NC(=O)C4=C(Cl)CC4)C(C)C3)=O)coc2c1 N1(C(CC2CCCC(C)C2)=O)CC2CC(NC(c3cnc(F)c(F)c3)=O)CC1C2 Cn1c(I)cc2c(N(C3CCNC3)Cc3c(F)cc(Cl)cc3Br)ncnc12 c1(NC(c2ccc(-c3ccc(O)cc3O)nn2)=O)ncc(F)cc1Br C12(C(=O)NC3(CO)CCN(C(=O)Cc4ccc(Cl)c(F)c4)C3)CCCC1CCC2 N1(c2cc(CC)nc(C)n2)CC(NC(=O)C2=CCCCCC2)CC2(CC2)C1 CCCCC(CCCC)C(=O)NC1CC2CC(NC(c3cccc(C)c3)=O)C1C2 c1(CCNC(C(=O)NC2C(C)C2(F)F)=O)csc2ccccc12 C(=O)(C(O)CN1CCCC1)N(CC(C)C)CC(=O)NC1(C)CSC1 N1(C(CC2CN(C(C)=O)C2)=O)CC=C(CC(=O)N2CCCNC(=O)C2C)CC1 N1(C(C(c2ccc(O)cn2)C)=O)CC2CN(C(=O)C=Cc3ccc(Cl)s3)C2C1 Cc1c(NC2CCN(C3CCC(C)CC3)CC2)ncnc1N1CCSC(C)C1.OC C(=O)(C1=CCC2CCC1N2C(C12C(=O)C3CC1C2C3)=O)N1CC(OC)C2(C1)CC2 C1(C)(CNC(C(C)=C(CC)C)=O)CCC(NC(c2occc2C2CC2)=O)C1 CCC(C(=O)NCc1cc(C(=O)NCC(CC2CC2)CO)no1)SC C1(NC(C2C(NC(CC3CC(CC)C3)=O)CCO2)=O)CCOCCC1C c1(C(=O)NC2(CNC(CN(CCOC)C)=O)CCOC2)cnn(C(C)C)c1C c1(C(C)C)ccc(C(C)C)c(S(=O)(=O)N2CCCC(c3ncco3)C2)c1 N1(C(CC(C(=C)C)OCC)=O)CC2(CCC2)CC1C(=O)NC12CCC(CC1)C2 C1(C(=O)NCC(=O)NCC2C(NC(CCNC(=O)OC)=O)C2)CCCCC1 c1(C(=O)NC2CC3(C2)CN(C(=O)C(Cl)=CCl)C3)cc(O)c2cc(F)cc(F)c2n1 C(CC(C)(C)C)(C(=O)N1CCCC[Si](C)(C)C1)OC N1(C(C(C2CCCOC2)OC)=O)CCC(N(C(=O)C2=CCOC2)CCO)CC1 CC(C(C)(C)O)NC(=O)C(=O)NCC1CCC1CO C#CC1CCCC(NC(=O)CCCCCN(C)C(C2CCC2C)=O)C1 c1(-c2c(C(N3CC(SC)OCC3)=O)ccnc2)ccccc1-c1ncccc1F Cc1ncnc(C(=O)NC(C)C(C)(C)C(=O)NC2CC(CCF)C2)c1C C(=O)(N=c1[nH]n(C)c(=O)n1-c1ccc(C)cc1)N1CC(OC)OCC1 c1(C(CC)C)ccc(C(=O)NCC2(F)CC(NC(=O)C3=COCCO3)C2)c(C)c1 C#Cc1cc(C(N2CC3(C2)CN(C(C2(C)C(C)(C)C2(C)C)=O)C3)=O)cc(N)c1 c1(OC)cc(CCC(=O)NC(c2csc(Br)c2)C(=O)O)ccc1C Cc1cc(C(N2CCC(NC(=O)Cc3cn[nH]c3)CC2C)=O)ccc1Cl CC(C)CC(C)CC(=O)NC1(C)CCCN(C(C2CCCOCC2)=O)C1 N1(C(C(C(C)(C)F)(C)F)=O)CCC2(CCCCC2NC(=O)CS(=O)(=O)C2CC2)C1 C1(C(C)NC(CCc2cc(C)no2)=O)CN(C(C2(N=[N+]=[N-])CC2)=O)CCO1 C(=O)(CC(C)CN(C)C)N(CC(CC)NC(=O)CCc1ccncc1)C N1(C(=O)Cc2cc(Cl)sc2Cl)CC2CC(C1)N(C(=O)NC1(c3cc[nH]n3)CC1)C2 CCC(F)(F)CC(=O)N1CCOCC(C(=O)NCC2CCC(F)(F)C2)C1 N1(C(C(c2ccc(O)cc2)C)=O)CCC2CN(c3ncc4[nH]ccc4n3)CCC12 c1(CC(=O)NC2C=CCN(C(=O)Cc3cnccc3Cl)C2)ccc(F)cc1F c1(CNC(C2CC(F)CN2C(C2CC(O)CN2)=O)=O)c(Cl)cccc1[N+](=O)[O-] CC(C)CC(C)C(=O)NCC1(NC(=O)Cc2csc(C(F)(F)F)n2)CCCCC1 C(c1csc2ccccc12)=CC(=O)NC1CCC(C)N(C(c2ccncc2)=O)C1 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(C)(F)F)CC1c1ccccc1 C1(C2CN(C(=O)C(C)(C)c3ccno3)C2)(NC(C2CCC(OC)C2)=O)CC1 CCC(C)(C)CC(=O)N1CCC1CNC(=O)CN(C)CCO c1(CC(=O)NC2CCCC(NC(C3(O)CCOC3)=O)C2)nc2ncccn2n1 c1(CNC(C(=O)NC(C)C)=O)nnn(C)c1C(N1CCC2CC12)=O C1(CNC(C=CC(C)(C)NC(C2CC(=C)C2)=O)=O)CC(O)C12CCC2 C1(C)(CNC(C(=O)NCCOC)=O)CN(C(C2(Cl)CC2(F)F)=O)CCO1 C1(C(C)C)CCC(C)(C)CC1c1nc(-c2cc(O)nc(C3CCOCC3)n2)no1 N1(Cc2ncn(C)n2)CC(NC(=O)C=CC2CC2)C(O)C1 C1(C(=O)NCCN2CCC(NC(C(CC)OC)=O)CC2)CC2C(C1)C2(C)C CCC(C#N)C(=O)N1CCC(N2C(=O)c3cccc(c3)C2)C1.S(C)CC C1(CNC(C(C)c2cccs2)=O)CN(C(=O)C2=NOC(C)(C)C2)CCC1(C)C C1(C(=O)NCCCN(C(=O)CCCc2cc[nH]c(=N)c2)C)C2CCCCCCC12 c1(C(=O)NC(C)(CNC(=O)C2=CCC2)C2CC2)cc2ccc(Br)c(F)c2[nH]1 C1(C)(NC(C(C)OCC#C)=O)CCCN(C(C2CCOC2)=O)C1 CCCC(C)(O)CC(=O)N1CCCC1CCNC(=O)C(C)=C1CC1 c1(C(N(CCC)CCNC(=O)Cc2cnn(CC(C)C)c2)=O)cc(OC)ccn1 N1(C(C(C(CC)O)C)=O)CCCN(C(c2cc(Br)sc2C)=O)CC1CO N1(C(CC(C)CNC(c2cc[nH]c2)=O)=O)CCC(C)C(O)C1 CCS(=O)(=O)CC(=O)N1CCC(C(=O)NC(C)CC(F)(F)F)C12CC2 C(c1cccs1)=C(C)C(N1CC(CO)(NC(=O)CC2CCCC2)C1)=O N1(C(CC)=O)CCN(C(c2cscc2Br)=O)CC1c1cccnc1 c1(OCCCN(C(=O)C(=O)N2CC(NC(C)(C)C)C2)Cc2ccsc2)ccccc1 c1(-c2n(CN(C(CC)C)CCc3ccncc3)ccn2)cccc(-c2cscn2)c1 C1(C(C)=O)C(C(=O)NCC(C)(F)CNC(=O)CN2CCCC2=O)C1(C)C C1(CC=C)(NC(=O)C(C)N(C(=O)CC(=O)OCC)CCC)CCOC1 c1(C(N2C(CNC(c3n(CC)ncc3)=O)CCCC2)=O)cc(C2CC2)cc(F)c1 Cc1c(C(=O)N(CCC(=O)NC(C2CCCC2)C)CCCO)cccc1O Cc1cc(-c2ocnc2C(=O)NC(CNC(c2cc(Cl)no2)=O)C2CCC2)on1 n1(CCCC)nccc1C(=O)NCCC(C)N(C(=O)C=CC(C)CC)C CCCCCC(=O)N1CC(CC)(NC(=O)CCc2cnn(C)c2C)C1 c1(C(N2CCN(C(c3c(CC)csc3)=O)C(COC)C2)=O)ccc2cc[nH]c2c1 c1(C(C)CCCCCCC(=O)NC(=O)CC(C)c2ccco2)cnccn1 C12(C(N3CCC(OC)CC3)=O)CCC(C1)N(C(c1ccc(N(C)C)cc1)=O)C2 c1(C(=O)N(C2CC(C(=O)O)N(C(c3ccc(Cl)cc3Cl)=O)C2)C)scc2c1CCCC2 N1(C(C2C(CC)CN(C(c3ccccc3NC)=O)C2)=O)CCCC2(C=CCO2)C1 c1(C(=O)NC(C2(C(=O)NC(C)C(=O)NCCF)CC2)C)cnc[nH]1 c1(NC(Cc2cccc(OCc3ccc(C)cc3)c2)=O)cnc(Cl)c(C)c1 c1(OCC)ccc2cc(C(=O)N(C(C)CNC(C3CCCN3C=O)=O)C)[nH]c2c1 N1(C(C(COC)OC)=O)CCC(NC(C2(CC(C)=O)CC2)=O)C(C)(C)C1 N1(C(c2ccc(CNC(C(C)CC3CCC3)=O)s2)=O)CC2C(C)C2C1 c1(C(C)=O)cc(C(N2CCN(C(c3coc(C)c3)=O)CC2CCO)=O)ccc1C C1(NC(CC2OCC(C)(C)OC2)=O)CC2(CCN(C(=O)C(N)CN)CC2)C1 C1(NC(CNS(CCOC(C)C)(=O)=O)=O)CC(O)CN(C(=O)CN2CC=CC2)C1 C(=O)(C(O)C(C)C)N1CCC(N(C(=O)CCC2CCCC2)CC)C1 C1(NC(C(c2cccs2)NC(=O)Cn2ccccc2=O)=O)CCCC(O)C1O c1(C(N(C2CCN(C(=O)CC3CCC(=O)N3)CC2)C)=O)cc2ccoc2cc1F CCS(=O)(=O)CC(=O)NCC(C)NC(=O)CC(O)C1CCCC1 c1(NCc2c(N)nccc2)cc(=NCCCc2cccc(OC(F)F)c2)[nH]cn1 CC(CN1CCCC1=O)N=c1[nH]c2c(c(=NCc3nncn3C)[nH]1)CSC2 c1(C(N2CCOC(C(F)F)CC2)C(=O)NC(CC)(C)C)cc(C2CC2)cc(C)c1 N1(C(c2c[nH]c(=NCC=C)s2)=O)CCN(C(=O)CCOCC(F)F)C2COCC12 c1(C(N2CC(NC(CCOC(C)C)=O)CC(C)(C)C2)=O)c[nH]c(=N)c2[nH]ccc12 N1(C(C(C2CN(C(C3COC(=O)C3)=O)C2)OC)=O)CC2C(C1)C2(F)F CCC1=C(C(=O)NCC(C2CCC2)NC(C2(F)CCCN(C)C2)=O)CCCO1 N1(C(C)=O)CC2(NC(=O)Cc3cc(OC)cc(Cl)c3)CCC1CC2 C(=O)(C1CCc2nccn21)NCC1(CCNC(=O)CC2CCC2)CC1 c1(C2(C(N3CCC(c4scc(C)n4)CC3)=O)CCC2)ccc(F)cc1Br CCCC(C(=O)N(C)CC1COCCN1C(c1csc(=NC)[nH]1)=O)OCC c1(NC(C2CC23CCN(Cc2cccc(F)c2Br)CC3)=O)cc(F)cc(F)c1Br c1(C(N2C(C)(CNC(C3C(=C)C3)=O)CCC2)=O)nc(C(F)(F)F)n2ccccc12 CC1(C)NC(=O)N(CCCC(N2CC3CC2(CNC(=O)C=C(Cl)Cl)C3)=O)C1=O C1(C2CCCCC2)(C(N2CCN(C(C3C(C(C)C)C3)=O)C(C3CC3)C2)=O)CC1 c1(C(c2nnnn2C)NCC(F)(F)Cl)ccn(C2CC2)n1.C1(C2CCC2)CCOCC1 c1(C(N2CCC(CN(C)C(C3(C)CC=CCO3)=O)CC2)=O)nccc(C#N)c1F C1(O)(CCNC(Cc2cc(C)ns2)=O)CCCN(C(C2CS(=O)(=O)C2)=O)C1 N1(C(c2ccn(C)n2)=O)CCSCC1C(=O)NC1CC(c2ccccc2Cl)C1 C1(C(=O)NC(C2(O)CCN(C(=O)Cc3cnsc3)CC2)C)C2CCC3C(C2)CC13 C=CCC(C(=O)NCC(C(C)(C)C)NC(C1CCC(=C(F)F)CC1)=O)C(C)C c1(C(N(C2CN(C(C3(Br)CC3)=O)CC2O)C)=O)c(Cl)cccc1Cl N1(C(c2ccn(C)c(=O)c2)=O)CCC2CC2(NC(c2csc3nnsc23)=O)CC1 c1(C(=O)NCCCN(C(CN(CC)CC)=O)Cc2ccccc2)csc(C)c1 C=CC1(C(F)(F)F)CCN(C(N2CCC3C(CC(=O)OC)C23)=O)C1 c1(C(N2CCC(c3n[nH]c(=N)o3)CC2)=O)nc2ncc(CCO)cn2n1 N1(C(c2ccc(C)c([N+](=O)[O-])c2)=O)CC(NC(C2(C)CC2)=O)CC12CCOCC2 c1(C(=O)NC2CC(C)(NC(c3coc(Br)c3)=O)C2)cc2nc[nH]c2cn1 C(=O)(C1CCc2ccccc21)NC(C)(C)CCC(=O)NC1CCN(C(N)=O)C1 CC(CCCC(=O)NCc1cnco1)NC(c1cn(CCO)nn1)=O C(c1ccccc1)=CC(=O)NC1CCN(C(C2CC2c2ccc(Cl)o2)=O)C1 CC1(C(N2CCOCC(NC(C3CCCS3(=O)=O)=O)C2)=O)CC2CCC1C2 CC(C)S(=O)(=O)CC(=O)NCCN(C(=O)CN1CCSCC1)CC1CC1 N1(C(C2CCN(C(c3ccc(CC)s3)=O)C2)=O)CC2C(CN(C)C)C2C1 C1(OC)CCC(F)(Cc2cn(CC(=O)Nn3nc(C)cc3C)nn2)C1 CC(CF)CC(=O)NC1(CNC(c2cccs2)=O)CCOC1 Cc1c(O)nc2ccccc2c1C(=O)N(C)CC1CN(C(=O)CC(C)(F)F)C1 c1(C(=O)NC(C(C)NC(CCCCN(C(C)=O)C)=O)C(C)C)ccn(C)c(=O)c1 C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(=O)Nc2ccc(Cl)cc2)CC1O N1(C(C=C(C)C)=O)CCCN(C(=O)Cc2ccccc2C(F)(F)F)CC1C(C)C N1(C(c2n(C)ccc2)=O)CCN(C(=O)CC2CCN(S(C)(=O)=O)CC2)CC1CF c1(C(N(C)CC2(O)CN(C(C3(CCOC)CCCC3)=O)C2)=O)cc(O)ccc1F C(CC(O)C(F)(F)F)NC(CN(C(Cn1ncc(CC)c1)=O)C(C)C)=O c1(NC(C(CCC)C)=O)cc(C)c([N+](=O)[O-])cc1[N+](=O)[O-] Cc1ccc(F)c(NC(C2CC(C)CN2Cc2ccc(O)c(F)c2)=O)c1 c1(-n2c(CCCC(C)(F)F)nc(C(C)OC)n2)ccc(S(=O)(=O)N(C)C)cc1 N1(C(C(C(C)C)F)=O)CCCC(C)(C)C1C(=O)NCCc1ccns1 N1(C(CCCCCOC)=O)CCC(C(=O)NCC(C)CC(C)C)=C(F)C1 C1(C)(C(=O)NC(C(C)CO)C)CCN(C(C2CCCC2)=O)CC1 Cc1c(Br)ccc(CNC2CC2C(N2CCOC3CC23)=O)c1F C1(NC(=O)CCF)CC(NC(=O)C=C2CCOCC2)C(O)C1 c1(CNC)cnn2c1CN(C(=O)COCC1CCC1)CC2.C1(C=O)(CF)CCC1 O=C1NCC2(CC(N=c3[nH]c(N4CCC(F)CC4)nc4ccc(Cl)cc34)C2)O1 N1(C(c2c(Br)cnc(C)n2)=O)CC2CCC(NC(=O)Cc3ccco3)(C2)C1 N1(C(c2nccc(CC)c2)=O)CC2CC(NC(c3ccc(F)nc3)=O)CC2C1 N1(C(c2c(OC)ccc(OC)n2)=O)CC2(C1)CN(C(=O)CC1(C)CC1)CCO2 C(=O)(CC(C)(C)CN(C)C)N(C1CCN(C(=O)C(c2ccccc2OC)C)C1)C.CO N1(C(c2c(CC)onc2C)=O)CCN(C(c2cc(Cl)no2)=O)C(CCOC)C1 C(=O)(C1=CNC2=NCCC2=C1)NCC(CN(C(c1ccc(CC)c(C)c1)=O)C)O N1(C(CC(c2ccc(OC)cc2)C)=O)CC(NC(c2csc(O)n2)=O)CC1(C)C C1(c2n(CC)nnn2)(Nc2cccc(C(F)F)c2C)CCOCCC1C N1(C(c2cc(CNC(C(CCC)C)=O)sc2)=O)CCCC2(C1)N=N2 N1(C(CCC(CC)OC)=O)CC2CCCC(C1)N2C(C1CC1CC)=O C(=O)(C(C)(F)C(=O)NCC1(CN(C(c2cnoc2-c2cccs2)=O)C2CC2)CC1)OC c1(C(=O)NC2CCC(CCNC(C3(CC)CCCC3)=O)C2)ncc(N)nc1C O=C1CC(=O)CC(C(N2CCC2CC(=O)NCCOCC(F)(F)F)=O)C1 C1(C(N2CCC(O)(C(C)NC(c3ccns3)=O)CC2)=O)CC2CC1CC2(F)F O=C(N=c1c(Br)c[nH]cc1I)C1(F)CCN(Cc2ccc([N+](=O)[O-])o2)C1 c1(N(C(C)CNC(c2ccnn2-c2ccccc2)=O)C)cc(Cl)nc(S(C)(=O)=O)n1 c1(CCC)cc(C(=O)NCC(C)(O)CNC(=O)C(C)C(F)F)c(C)o1 c1(C(=O)NC(C2CCCC2)CNC(C(C)SCC)=O)cccn2c(C)cnc12 C12(NC(CCC#C)=O)CCCN(C(c3ccnc(C)n3)=O)CC1C2 C1(CC(=O)NCC(CCOC)NC(C2(C(=O)OCC)CC2)=O)CC(F)C(=O)N1 C(CCNC(C1CCC12CCC2)=O)(C(C)C)NC(Cc1c(C)ncs1)=O N1(C(Cn2ncc(C#C)c2)=O)CCCC2(C1)CN(C(=O)CN1CCC(O)CC1)C2 CCCCC(C)(F)C(=O)NC1CCN(C(C2COC(C)(C)C2)=O)C1 CC1(C)c2[nH][nH]c(=NC(=O)c3ccnc4ncccc34)c2CN1C(=O)C(F)Br c1(C(=O)NCC2(F)CN(C(COCC#C)=O)C2)cncc2ncccc12 c1(CNC)cnn2c1CN(Cc1cnc(-c3ccc(OC(C)C)cc3)s1)CC2 Cc1nc(O)sc1C(=O)NCC1CC(C)N(C(=O)C=CC(=O)N(C)C)C1.C(CO)N N1(C(CCCCCCC)=O)CCCC2C(NC(c3ocnc3CC)=O)C(C)(C)C12 c1(C(N2CCN(C(C3CC4CCCC34)=O)CC2)=O)c(F)ccc2nc[nH]c12 O=C(NNc1ncc(F)cc1F)NCc1ccc2c(c1)CCCC2 N1(c2cc(NC(c3n(CC)ncn3)C)nc(C(C)C)n2)CCn2ncc(C)c2C1 N1(C(CC2N(C)CCC2)=O)CCC2OCCN(C(=O)CCc3cnoc3)C2C1 c1(OCC(=O)NCC(C(C(C)C)C)NC(c2nncs2)=O)ccc2c(c1)CCC2 c1(C(=O)NC(C)CNC(=O)CC(C)(F)F)cc(S(N)(=O)=O)cc(Cl)c1F N1(C(c2c(C)coc2C(C)(C)C)=O)C(C)CC2CN(C(=O)CNS(C)(=O)=O)CC12 C1(NC(=O)NC(CCSC)C(=O)O)C2Cc3ccc(Br)cc3C12 C(=O)(C(C(C)O)NC(=O)Cc1ccsc1C)NCc1c(CC)con1 CN1CC(C(N2CC(CO)(NC(=O)C(c3cccn3C)=O)C2)=O)CC1=O CCC(CC)CCC(=O)NC(CNC(=O)CC(C)(C)C(F)F)C1CC1 N1(C(C(C(C)C)SCC)=O)CCOCC(CNC(C2CCCN2C2CC2)=O)C1 C=C(Cl)CC(C(=O)N(C1CC2CC2C1)C)NC(c1ncc(C)cc1F)=O N1(C(c2ccn(C(C)C)n2)=O)CCCCC(C(N2CC3CCC3(C)C2)=O)C1 Cc1ccc(C(=O)NCCCCCNC(c2cc3occc3s2)=O)c2c1CCC2 C(F)(c1ccccc1)=CC(=O)N(C1CN(C(=O)C(C#N)C2CC2)CC12CC2)C C#Cc1cncc(NC(=O)C(O)CCCNC(=O)C(F)OC(F)(F)F)c1 CC1CCN(C(=O)Cc2csc(N3CCC(O)CC3)n2)CCN1C(=O)CCC#N c1(C(N2C3CN(Cc4cc(Cl)c(Cl)cc4O)CC23)=O)cc(F)c(F)cc1Cl C12(C(=O)NC(C3CN(C(C4CC4c4ccc(F)cc4)=O)CCO3)C)CC(CCO1)C2 c1(C(C)C)cccc(CC(=O)NCCOCCCNC(c2ccon2)=O)c1 C1(N(C)C)CCC(CNc2cc(NC(c3ncc[nH]3)CO)ncn2)CC1 c1(OCCC(=O)NC2CC(N(C)C(c3nccnc3N)=O)C2)cc(F)ccc1F C1(C(N2CC(O)(CC=C)C2)=O)CN(C(C2COCCN2C(C)C)=O)CC1C(C)C Cc1n[nH]c(C)c1CC(=O)NC1(CNC(=O)CCOCC(F)(F)F)CCOC1 C1(S(N)(=O)=O)(CNC(C2N(C(c3n(C)nc(O)c3)=O)CCC2)=O)CCCC1 c1(NC(C(=O)NC2CCCC(C(C)(C)C)C2)=O)cc(C(N)=O)ccc1C CC1CC(CO)N1C(C1(CCNC(c2ccc(Cl)s2)=O)CCC1)=O c1(N2CC(CC=C)(NC(=O)CCc3ccccc3F)C2)cc(C(N)=O)nc(Cl)n1 c1(C(=O)NC2C(C=C)CN(C(=O)C=NOC)C2)nn2c(c1C)OCCC2 N1(C(CC(C)OC(C)(C)C)=O)CCN(C(=O)C(C2CC2)NC(N)=O)CC1C S1(=O)(=O)c2c[nH]c(c2)C(=O)N(C)CCN1C1CC1.C1(C)(NC)CCC(C)C1 C#CC(CNC(=O)CC(C)NC(=O)C=CC(C)CC)C(C)C Cc1cc(Cl)ccc1C(=O)N(C1CCCN(C(=O)Cn2cnc(C#N)n2)C1)C c1(N(C(=O)Nc2cccs2)CC2CCSC2)ccccc1 c1(NC(=O)C(N2CCC3(CCSC3)C2)=O)cccc(P2(=O)CCCC2)c1 N1(CC(F)F)CCCC(N=c2ccnc(N3CCCC(c4nc(O)n[nH]4)C3)[nH]2)C1 CC1CN(C(=O)C(O)(C2CC2)C2CC2)CCN1C(c1coc(Cl)n1)=O c1(CC)cc(C)ccc1C(N1CCCC(N(C)C(c2ccn(C)c2CC)=O)C1)=O C1(NC(c2ncc(OCC)nc2)=O)C(C)CN(C(c2sc(C)cc2C)=O)CC1C Cc1cc2sc(C(=O)NC3CCN(C(=O)Cn4ccnn4)C3(C)C)cc2s1 C1(CC(N2CC(NC(=O)CCc3ccco3)CC2C)=O)(CC)CCOCC1 C1(C(N(CCOCCNC(CCSC)=O)C)=O)CCC(=O)N1C(C)C S(=O)(=O)(c1ccc(N(C)Cc2ccoc2)cc1Cl)NC(CCOC)C(C)(C)C N1(C(C2(CC)CCCO2)=O)CCC(C(=O)N2C3CCC2CC(F)C3)=C(F)C1 N1(C(C(=O)NCC)=O)CC(C)C(NC(c2ccc(-c3cccs3)cn2)=O)C(C)C1 C1(C(N(C(C(=O)OC)C)C2CC2)=O)CCC(c2ccc(C)cc2)CC1 c1(CNC(c2cc[nH]n2)=O)c[nH]nc1C(=O)N(CC(F)F)CC1CCC1 N1(C(C(C(C)C)CN(C)C)=O)CC(NC(=O)CC=C(Cl)Cl)C2CCCC12 c1(C(=O)OCC)cnc(O)c(OC2CN(C(=O)CC3CCC3(C)C(=O)OC)C2)c1 C1(C(=O)NCCCC(C)NC(C(C)OCC)=O)CCOC(C)(C)C1 N1(CC(=O)N(c2nc(C)sc2C)CCC)CC(O)C(O)C12CCC2 N1(Cc2nc(C)c(C)s2)CCN(N2CCCC(c3nncn3C3CC3)C2)CC1 CC1CN(C(=O)CC2CSCCO2)CCC1NC(c1ccc(Cl)c(O)c1)=O N(C1CC2(CCN(C(C3(Br)CC3)=O)C2)Oc2ccccc21)C(=O)Cn1cnnn1 c1(CC(C(=O)NCCCCC=C)NC(=O)C(C2CCOCC2)F)cnn(C)c1O C1(C(=O)NC2(C(N)=O)CC2)C=CCN(C(=O)Cc2ccccc2F)C1 C1(NC(C=C2CCC(C)C2)=O)CC2CCC1CN(C(C13CC1COC3(C)C)=O)C2 C1(F)(CNC(C2CC(=O)OC2)=O)CC2CCC(C1)N2C(=O)C(O)(C1CC1)C1CC1 c1(C(=O)NCC2CN(C(C(COC)C)=O)CC2O)cc(F)cc2cccnc12 C(=O)(C(O)CCC(C)C)NC1CC(NC(C=CSC)=O)C1 Cc1ccc(C(N2CCC(NC(c3oc(Br)cc3C)=O)C(F)C2)=O)cc1Br C1(CC(=O)NC2CN(C(C(C)(C)N(C)C)=O)CC2F)CC(c2ccccc2)=NO1 C=CCC(C(=O)NC1(C(C)(C)NC(c2cnc(CSC)s2)=O)CC1)C(C)C C1(NC(=O)CCc2cnoc2)COCCN(C(=O)C(O)Cc2ccc(F)cc2)C1 CC1(C)CCC(O)(CNC(C2C=CC(NC(C3C=CCC3)=O)C2)=O)C1 CC1CN(C(C2CC23CCOC3)=O)CC(C)N(C(=O)CN2CC(=O)N(C)C2=O)C1 c1(C(=O)NC2CCCN(C(c3ccc(OC)c(N)n3)=O)C2)ccc(S(C)(=O)=O)o1 C(=O)(CC(O)C(C)(C)C)N(CC(C)NC(c1ccc(OCC)cc1)=O)C CC1CN(C(C2CC(=O)NC2(C)C)=O)CCN1C(c1cc(Br)cs1)=O C1(C2CCCOC2)(NC(C(C2(C)CC2)NC(CC(C)(F)F)=O)=O)CC1 N1(C(C2=CCCN(C(C(C(CC)O)C)=O)C2)=O)CC(C)NC(=O)C12CC2 c1(C(=O)OC)ccc(OC)cc1C(=O)NC1CCCCN(C(=O)C(O)C2CC2)C1 c1(OC)cc(C(=O)NCCOc2ccccc2Cl)c2c(c1)CCO2.C1(=O)CO1 C(=O)(CCCCC(F)F)N1CC(CNC(C2(C#C)CCCC2)=O)N(C)CC1 CCCCC(F)C(=O)N(C(CNC(=O)C(C)NC(=O)CC)C1CC1)C C(CCC(C)C(=O)N(C1CCCCN(C(=O)CCc2csc(=N)[nH]2)C1)C)OC CC1CC=CCC1C(=O)N(C1CCN(C(=O)Nc2cc(Cl)cs2)CC1)CC1CC1 c1(C(N2CC(NC(c3cc(CC)oc3)=O)C(OC)C2)=O)cnc2n1CCC(C)C2 c1(-c2n(-c3ccc(COC)cc3)nc(CCC(C)C)n2)ccc(C)cc1C C1(C(N(C2CCN(C(CCC=CCC=C)=O)C2)C)=O)CC2(CCC2OC)C1 C1(NC(C(CSC)(C)O)=O)(CO)CCCN(c2ccnc(Cl)n2)C1 C(C(O)C(=O)NC(c1cnn(C)c1)C(=O)N(C1CCC1O)C)=CC C(=O)(C(C)C(F)(F)C(F)F)NC(CC)(CNC(C1(C)CCNC(=O)C1)=O)CC c1(C(N(CCC(C)NC(C(CC)C(C)C)=O)C)=O)ccc2c(c1)NC(=O)CS2 CC1OCCCC1C(=O)NC1CC(CNC(=O)C=CCOc2ccccc2)C1 c1(C(C)C)ncc(Cl)c(C(=O)NC2CC23CC(NC(c2ncncc2Cl)=O)C3)n1 C1(CNC(C(C(C)C)O)=O)CN(C(C2CC(F)C2)=O)CC1(C)C c1(-c2cn(CCC(=O)N(C3C(OC)CCCC3)C)nn2)ncc(Cl)cc1F c1(C(=O)NCC2C(NC(C(C(CC)C)O)=O)CCCC2)cc(F)c(F)cc1OC Cc1[nH]c(C(N2CCCC(C)CC2)=O)c(C)c1C(=O)NCc1csc(C#N)c1 C#Cc1cnc(N2CC(=C(F)CNC(=O)CCc3ccccc3C(N)=O)C2)nc1 C1(O)(C(=O)NC2CC(N(C(C=CCN(C)CC)=O)C)C2)CCc2ccccc2C1 N1(C(CN(C(C2C(CCC)C2)=O)C)=O)CCC1C=O.C(C)(C)C C1(C(=O)NCC(C2CCCCC2)NC(C(CC)F)=O)CCN(CCO)C(=O)C1 C1(c2ccc(C3(NCCNC(=O)Cc4nn[nH]n4)CC3)cc2)CCCCC(=O)N1 C(=O)(C(C)C(C)S(C)(=O)=O)N(CCCN(C(C(C(CC)(C)C)O)=O)C)C C(=O)(CN1C(=O)COc2ccc(Cl)cc21)NC1C(NC(c2cncc(C)n2)=O)C1 c1(OC)ccc(CC(N2CCC(=O)CC2C(=O)O)=O)c(Cl)n1 c1(C(N(C(C)C)CCNC(c2ccnn2C2CC2)=O)=O)ccc2nccn2n1 N1(c2nc(N(CCC)C)c3c(n2)c(C)nn3C)CCc2c([nH]c3ccccc23)C1 N1(C(CC=C)=O)CCC(NC(c2cc(O)n(CC)n2)=O)CC1 c1(CC(=O)NCCC2CCCN(C(C3CC(C)(F)C3)=O)C2)noc2ccccc12 N1(C(c2c(C)nc(C)s2)=O)CC2OCC(NC(=O)CCOCC(F)F)C2C1 c1(C(N(C)CC2N(C(c3c(CC)onc3)=O)CCC2)=O)nsc2ccccc12 Cc1cc2cc(C(=O)NCC3CC(C)(C)CN3C(=O)CCC(F)F)oc2cc1C c1(C(=O)NC(CCC)CNC(C2CC2C(C)C)=O)c(N)ccc(F)c1F C1(C(=O)NC(CC)COC)(C(c2ccccc2)O)CN(C(C2CCCC2C)=O)C1 c1(NS(CC)(=O)=O)cnc(Cl)cc1C(=O)Nc1nccnc1Sc1ccccc1 c1(CC)onc(C(N2CCCC2C(C)(C)C(=C(C)C)NC(=O)C#CC2CC2)=O)c1C O(C1CCCc2ccccc21)CC(=O)NOc1cccc(F)c1Br N1(C(COc2cccc(C)c2)=O)CCC(C)C(NC(=O)C=CCCC(C)C)C1C CC1CCCN1C(=O)CCSC1CCCC1.C(=O)(CCCn1ccnc1)OC C1(CCCNC(Cn2c(C)nnn2)=O)CN(C(c2cc(O)nn2C)=O)CCO1 c1(C(N2C(c3cn(C(C)CO)nn3)CC(C)(C)C2)=O)cc2n(n1)CCC2 Nc1ncc(C(=O)Nc2nc3c(s2)CC(C(F)(F)F)CC3)cc1[N+](=O)[O-] C1(C(N2C(C)(C)CC(NC(c3cnn4c3CCC4)=O)C2)=O)CNC(=O)CC1(C)C CC(C(=O)NCCC1(O)CCN(C(C2(c3ccno3)CC2)=O)C1)C(F)(F)F C1(OC)(CNC(c2ccc(C)c(Cl)c2)=O)CCN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1 c1(NC(c2cc(C)sc2N)=O)ccc(C)c(Br)c1 C12(C(=O)NC3CCN(C(C=CCC)=O)CC3(C)C)CC3CC(C(=O)N1)C2C3 C=CC(C)(O)CC(=O)N(C1CCN(C(=O)COCCCC)C1)CC1CC1 c1(C(=O)NC(CCCNC(CCN(CCC)C)=O)C)ncnc(C)c1OC C(N=c1[nH]c(Cl)ncc1F)C1N(C(C2(CC#C)CCCO2)=O)CCCC1 CC(CSC1CC(OC(F)F)C1)C(=O)OC(C)(C)C CC1(C)CC(C(=O)NCC2CCCOCC2)N(C(=O)Cc2c(Cl)cccc2Cl)C1 c1(C(=O)NCC23CC2CN(C(C2CCCC(F)C2)=O)C3)cc(O)nc(C2CC2)n1 C1(OC)CC2(C1)CC2C(N1CCCC1CCNC(C1(C)CCCO1)=O)=O N1(C(CCC2(C)N(C(CC(CC)CC)=O)CCC2)=O)CCCN2CCCC2C1 C1(N(C(C2C(C=C)C2)=O)C)CCC(NC(=O)C(c2ccc(OC)cc2)C)CC1 C1(N(C(C2C3(CC3)C23CC3)=O)CC)CCCN(C(=O)CCC2CCC2)CC1 Cc1cc(Br)cc2[nH]c(C(=O)NC3CC(CCNC(=O)C(C)(C)O)C3)cc12 C(c1cccnc1C)=CC(=O)NC1CCN(C(CN(C)CC)=O)C1C1CC1 Cc1ncc(CCOC(=O)Oc2ccccc2)n1C.C12(C)CC(O1)COC2=O CC1(C)CCC1C(=O)NC1COCC1NC(c1nscc1Br)=O N1(C(c2cnc(C(C)O)s2)=O)CCC2(CC1)CCN(C(c1cnnc(Cl)c1)=O)C2 C=CCC(CO)NC(C1(C)CN(Cc2c[nH]nc2-c2ccccc2)C1)=O c1(C(N(C(CCNC(Cc2nc(C)sc2C)=O)C)C)=O)ccc(Cl)cc1O CN=c1[nH]cc(C(N2CC(OC)C(NC(=O)C(n3ccc(C)n3)C)C2)=O)s1 C(=O)(C1=NOC(c2ccccc2)C1)N1C(C(=O)N(CC)Cc2cc[nH]n2)CCC1 CC(C)CC(C)CC(=O)N1CCC(CNC(c2ccc(C(C)C)cn2)=O)C(C)C1 Cc1oc(C#N)cc1C(=O)NCC1(CNC(=O)CC(C)c2ccco2)CC1 C1(C)(C(N2CC(CNC(c3cn(CCCOC)nc3)=O)C2)=O)CCCC1O C1(C(=O)NCC2C(CNC(Cc3c(C)scc3)=O)C2)COC2COCC2O1 c1(C(C)=O)nc(C(=O)N(C(C)CCNC(=O)Cn2ccc(C(F)(F)F)n2)C)cs1 CC1CCCCC1OCC(=O)NCCC1CN(C(c2cnc(C3CC3)[nH]2)=O)C1 c1(CC)cnc(N2CCC(C)(NC(c3cnn(C)c3CC)=O)C2)nc1 c1(OC)ccccc1C=CC(=O)N(CCCNC(C1CCCC1(C)C)=O)CCO N1(C(CCN(C)CC)=O)CCC(C(N2CCCC2C(C)O)=O)C1 C1(CNCCCNC(CCSC)=O)CC(C)N(C(c2ncc(F)cn2)=O)C1 C(CC(CO)NC(=O)CCN(C(=O)C(C)n1cccn1)C(C)C)SC c1(CC(=O)NCC2(F)CC(CNC(CC)=O)C2)cnc2n1CCCC2C C1(CNC(C2C(CNC(CCOCC#C)=O)C2)=O)CCOC(C)(C)C1 C1(C)(NC(c2nc(C(C)NC(c3nc(C)oc3C)=O)oc2)=O)CCC(=O)N(C)C1 c1(C(=O)NCC(CNC(c2ccncc2N)=O)OC)cc2nc(C)[nH]c2cc1F N1(C(C2CCN(C(c3c[nH]c(=NC)o3)=O)C23CC3)=O)CC(C)(C)OCC1C C1(CNC(C2(O)CC(C)(C)C2)=O)CN(C(=O)CCC(CF)CF)CC12CCC2 c1(C(=O)NCC(CNC(=O)CC2CCSCC2)F)cc(Cl)c(F)cc1[N+](=O)[O-] N1(C(C(C(CC)O)C)=O)CC2CCOC2(CNC(=O)CCn2ccccc2=O)C1 CN1C(=O)CC(CNC(C2CC(N(C)C)C2)=O)C1c1cccnc1 C1(CC)(NC(C2CCCC2CNC(C2COCC(C)O2)=O)=O)CCCCCC1 c1(SCC(=O)NCC(CC)(C)NC(=O)C(C)(F)C(=O)OC)cc(C)cc(C)c1 N1(C(=O)C(Cl)=CCl)CCOCC(NC(c2cnc(-n3cccn3)cn2)=O)C1 C1(C(=O)NCc2occ(C(=O)NCC3(CO)CCN(C)C3)n2)CCC(O)CN1C C(=O)(C1=CCC(C)(C)CC1)NC(CC#C)C(=O)N1CC(O)(CO)C1 CCC(C)(C)C(C(=O)N1CC2CCN(C(c3sc(SC)cc3C)=O)C2C1)OC c1(CN(C(COC(C)C)=O)C(C)C)noc(-c2ccco2)n1 n1(CC(=O)N(C)CC2CN(C(=O)COCC(F)F)C2)cnccc1=O CC(C)(CC(=O)NCC1(C)CCCC1NC(=O)C=Cc1cocn1)C(F)F c1(C(=O)N(CCO)C2CC2)cc[nH]c2nccc1-2.C(=O)(N1CCCCO1)C1CC1 C1(NC(c2sc(C)c(O)n2)=O)C(C)CCN(C(c2ccc(C)n2C)=O)C1C C1(C(C)NC(CCCN(C(C)=O)C)=O)CCN(C(=O)CC2(CO)CCC2)CC1 C(CC(C)(C)C)(C(=O)N(CC(C)O)C)NC(c1c(C)ccc(C)n1)=O c1(C(N2C3CC(NC(C4CCC(=C)CC4)=O)(C3)C2)=O)ccc(F)cc1O C1(C(N2CCC(O)C(CO)C2)=O)(CC)CCN(C(c2cc(OC)ncn2)=O)CC1 c1(OC)cnc(C(=O)NCC23CC2CN(C(=O)C2=CCCCC2)C3)c(OC)n1 Cc1ccc2c(CN3CCC(NC(c4ccc(Cl)c(C)c4)=O)C(F)C3)c[nH]c2c1 C12(NC(c3coc4c3CCCC4)=O)CCC(CN(C(=O)C(F)C3CCC3)C1)C2 C1(C(N(CC(CC)OC)C)=O)CC(NC(c2ccc(C)cc2)=O)C(O)C1 n1(CCC(C)(C)NCC)c(N2CCCC2)nnc1-c1ccc(C(N)=O)cc1 C1(C(N2C(CC(=O)OC)CCC2)=O)CN(C)CCN1C(C1CC(=O)C1)=O C1(CCNC(c2n(CC)ccn2)=O)CSCCN1C(c1cn(C2CCC2)nn1)=O CC(CC1=CCCCC1)NC(N1CCCCC1c1nc(-c2cccnc2)no1)=O C#CCC(C)(C(=O)NC(CC)C(C)CN(C)C)NC(c1cc(N)cc(F)c1)=O c1(C(=O)NC2C(CC)CN(C(c3oc(SC)cc3C)=O)C2)c(C)ccc(C)c1C C1(NC(C)=O)CCN(C(C2CN(CC(C)(F)F)C2)=O)C(C)C1 N1(C(COc2ccc(C#C)cc2)=O)CCC2C(C1)CN2C(c1ccoc1Cl)=O c1(C(c2nnnn2C)Nc2c3cn(C)nc3ccc2)cc(Br)cc([N+](=O)[O-])c1 N(C1CCOc2ccc(Br)cc21)C(C1CCCCN1Cc1c(Br)cncc1Br)=O Cc1nc(C2C(C(=O)NC34CC(NC(c5cn[nH]c5)=O)(C3)C4)C2(C)C)n[nH]1 N1(C(c2nn(CC)c(O)c2)=O)CC2(CC(NC(c3nc(O)c(C)s3)=O)CO2)C1 CC(C)C(F)(CNC(=O)C1=NOC(C)C1)C(=O)Nc1ccc(F)cc1 c1(C(=O)NC2CN(C(C(CSC)(C)C)=O)CC(O)C2)ccc2nc(O)sc2c1 C1(F)(CNC(C2(C)C(C)CCC2)=O)CCN(C(=O)C=Cc2ncco2)CC1 C1(NC(C(CC)NC(=O)CC2CCCOCC2)=O)COC2COCC12 Cc1cc(C(=O)NCC(=O)NCCOCCNC(=O)C(C)(C)C)ccc1C(F)(F)F Cc1[nH]nc(C(N2CCC(C(C)C(=O)N(CC(C)O)C3CC3)CC2)=O)c1O c1(C(N(CC(=O)N(C2CC2C)C)CCOC)=O)cn(C2CC2)cn1 C(=O)(CC1=NNC(=O)C1)NCC1N(C(C2(C)CCC(=O)NC2)=O)CC1 c1(C(C)N(C(c2cnn(CCNC(=O)CCCF)c2)=O)C2CC2)ccccc1F c1(NC(CC2N(C(CCN(CC)CC)=O)CC2)=O)cccc(Cl)c1C Cc1nn(CC(N2CC3CC3(CNC(=O)C(C)CN(C)C)C2)=O)c(C)c1Br C1(C(C)C)COCCN(C(C2CCN2C(=O)C(F)=CC2CC2)=O)C1 C1(CCNC(c2c(C)nn[nH]2)=O)CN(C(=O)Cc2cncc(O)c2)CCS1(=O)=O c1(C(N2CCC(NC(C3C(CCOC)C3)=O)CC2C)=O)cc(Cl)cc(Cl)c1OC c1(C(N2CCC(N(C(c3nccc(NC(C)=O)c3)=O)C)C2)=O)c(F)cncc1F C1(C(N(CC(C)NC(c2ccc(F)cc2NC)=O)CC)=O)CCc2nc[nH]c2C1 c1(NC(C(N2CCC(C)(CNC(CSCCOC)=O)C2)=O)=O)c(F)cccc1F C1(C(N(C(CC)COC)C)=O)CCOC1CNC(c1c[nH]nc1Cl)=O c1(C(N2CCN(C(C=NOC)=O)C(CS(C)(=O)=O)C2)=O)cnc2[nH]cnc2c1 c1(C(=O)NCCCN(C(=O)CC(=O)NC2CC2)CC)coc2cc(F)ccc12 C1(C2CCN(C(=O)CCc3cnc[nH]3)C2)(NC(C(CC)c2cnccn2)=O)CC1 c1(CSC)cc(F)ccc1NC1(c2nnnn2CCC2CC2)CC2COCC12 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)COC)ccc(C)c(S(N)(=O)=O)c1 c1(SC)ccc2cc(C(=O)NC3CC3NC(C3OCC4CCCC34)=O)[nH]c2c1 c1(C(N2CC(N(C(CC3C(C)C3)=O)CCO)C2)=O)nc(N)cc2ccccc12 C12(C(=O)NC(CCC(=C)C)C)C(NC(=O)CC3CCC(=O)N3)C3CC1C2C3 c1(C(=O)NCC(CC(C)C)NC(=O)COCC2CC2)ccc([N+](=O)[O-])n1C C1(C)(C(=O)NCCCCCCN(C(c2n(CC)ncc2)=O)C)CCOC(C)C1 c1(CN(C2N(C(C(C3CCCC3)OCC)=O)CCC2)C)ccnc(F)c1 c1(CNC(C2CC(NC(C3(F)CC3)=O)C2)=O)ccc2c(c1)CC2 N1(C(CCCCc2ccc(OC)cc2)=O)CCC(C2(NC(=O)CC3CC3)CC2)C1 C1(COC)(CNC(c2cc(C(N)=O)no2)=O)CCCN1C(=O)C(C)CC1CCC1 C1(CNC(c2csc(F)c2)=O)CC2(CC2)CN1C(c1cc(Cl)ccn1)=O C(C)(CC(=O)N(CCNC(C1(F)CCOC1)=O)C(C)C)SC C(N=c1[nH]c(=NCCOCC(F)F)c2c(F)cccc2[nH]1)c1c(C)cc(Br)cc1 Cc1cc(C(N2C3CN(Cc4ccc(-c5ccccn5)cc4)CC23)=O)c(C)[nH]1 N1(C(c2c(CC)ncs2)=O)CCC(NC(c2cc(C)c(F)cn2)=O)C(CO)C1 Cn1cc(C(N2CCC(CO)C(NC(=O)C3=COCCC3)C2)=O)c(O)nc1=O c1(C(N2CCC(NC(C3(COC)CC=CC3)=O)C2C)=O)noc2c1CCCCC2 c1(OCC(=O)NC(C)CCCNC(=O)C(C)CC2CCCC2)ccc(CO)cc1 Cc1sc(=O)n(CC(N2CC(N(C)C(c3cc(C)n(C)n3)=O)C3(CC3)C2)=O)c1C c1(C(=O)NC(CCN(C(c2cccc(C(C)=O)c2)=O)C)C)ccc(N=[N+]=[N-])cc1 N1(C(c2ccc(OC)nn2)=O)Cc2ccccc2C(NC(C2(F)CCOC2)=O)C1 C1(CC(N2C(C(C)NC(C3CC(F)(CO)C3)=O)CCC2)=O)CCC(F)(F)CC1 N1(C(CCc2onc(C)n2)=O)CCC(O)(CNC(c2ccc(N)c(F)n2)=O)CC1 C(=O)(C1=C(C)C(C)(C)OC1=O)NCC1CCCN(C(CS(=O)(=O)NC)=O)C1 c1(NC(=O)NC2C(c3onc(COC)n3)C2)cc(OC)c(Cl)cc1OC N1(Cc2cc(CC)no2)CCc2[nH]cc(I)c(=O)c2C1 c1(C(=O)NC(C2CN(C(c3cnc(S)nc3)=O)CCO2)C)ccc(F)c(F)c1O CCCC(C)(C)C(=O)N1CCCC(CCC(=O)NC(C)CN(C)C(C)C)C1 c1(C(N2CCC(N(C)C(c3snc(Cl)c3Cl)=O)C2)=O)nnn2c1C(=O)NCC2 C(=O)(C1CCC(=O)c2cccn21)NCC1N(C(c2cn(C)nc2)=O)CCCC1 c1(CN(CC(O)CO)C(=O)OC(C)(C)C)ccc(OCC(F)(F)F)cc1F C1(NC(CC2(CNC(c3ccc(C#N)cc3)=O)CC2)=O)CC2CC1C(O)C2O C1(F)(C(N2CCC(OCC=C)C2)=O)CCCN(C(=O)CN(C2CCCC2)C)C1 N1(C(Cc2cc(C)sc2)=O)CCOCC(NC(c2c(C)nn(CCO)c2C)=O)C1 C1(NC(=O)CN2CCCC2=O)CN(C(C2CCSCC2)=O)C2CC12 N1(C(C2(C)C(C)(C)C2)=O)CCOC(CC(N2CCC(OC(F)F)C2)=O)C1 N1(C(C2C3CN(C(CC(C)n4cccc4)=O)C2C3)=O)CCCN(C)CC1C N1(C(CC2(OC)CCC2)=O)Cc2ccc(NC(=O)C(C)n3cncn3)cc2C1 Cc1ccsc1CC(=O)NCCN(C(=O)C(CO)N1CCCCC1)CCOCCO c1(CC(=O)NCC2CCN2C(c2nc(Br)c[nH]2)=O)ccc(F)cn1 CCCCCC(C)CC(=O)N1CC2(CC(CC(=O)NCCC(C)SC)C2)C1 c1(NC(=O)NCc2cccc(C3CC3)c2)cc2ccccc2c(=O)o1 C1(C)(C(=O)NCC(C)Cc2cn[nH]c2)CC(O)CN1C(c1ccn(C(F)F)n1)=O c1(C(=O)NC2C(N(CCC(=O)NCc3ccccc3)C)C2)cc2ccccc2o1 c1(OC)ccccc1C(C)C(=O)NCC1CCN(C(=O)C(c2ccnn2C)C)C1 c1(C(N2C(C)(CC)CC(NC(c3scc(C)c3C)=O)C2)=O)cnn2ccccc12 C1(NC(CCCC=C)=O)CC2(C1)CN(C(=O)C(C)S(N)(=O)=O)C2 c1(NC(C2CN(C(C(C)c3ccco3)=O)C(C)(C)C2)=O)cnc2ccccc2c1 C1(CNC(c2cc(C)ns2)=O)CN(C(c2cc3ccsc3s2)=O)C2(CCC2)C1 N(C(=NCc1cc(C(F)(F)F)cs1)N1CCC(COC)C1)C(CC)C CCCC(C)(O)C(=O)N1CC(N(C(=O)CCc2ccccn2)CC)C(C)(C)C1 c1(CNC2CC2(Cl)Cl)c(CSC)oc2ccccc12 N(C(=NCCCCC(F)(F)F)NC1CC12CCCC2)CC1(SC)CCC1 C1(C)(C(N2C(CN(C(=O)CC3(COC)CC3)CC)CCC2)=O)CCC(F)(F)C1 Cc1ccc2c(C(=O)NCC3CCCN3C(=O)C(C)CC(F)F)ccnc2c1Cl N1(C(C(C=C=C)C)=O)CCC(C=C)(C(=O)NCC=Cc2ccccc2)CC1 c1(CN(C)C(C2(NC(=O)CCn3cnc(=N)[nH]3)CC2(C)C)=O)cn(C)cn1 N1(C(Cc2cnc(C)s2)=O)CCC(CNC(=O)C(C)C(F)(F)F)C12CC2 C1(C)(NC(C(C)C2CCCO2)=O)CN(C(C2CC3CC2C3)=O)C1 C=CC(C)(CCOC)C(=O)N1CCN(CCCNC(=O)CCC#CC)CC1 N1(C(c2ccc(CC)[nH]2)=O)CC(NC(=O)C(C)CC(C)CC)CC12CCOCC2 O=C(C1=CN2CCS(=O)(=O)N=C2C=C1)NC1CCN(C(=O)C2=CCCOCC2)C1 C=CC1OCCC1C(N1CCCCC1C1(NC(C2CCC2OC)=O)CC1)=O C1(NC(CN(C(C(C)OCOC)=O)C2CCC2)=O)CCn2nnnc2C1 N1(C(c2cc(C)oc2C)C(=O)NC(C(=O)OC)C)CC(C)(C)C1C1CCCO1 N1(c2[nH]c(=N)c3c(n2)CCC3)CCC(N=c2nc3scnc3c(N3CCC3)[nH]2)C1 N1(C(c2cccc(CC)n2)=O)CC2CC(NC(c3ncc(Cl)s3)=O)CC1C2 c1(C(=O)NCC=CCNC(=O)Cc2cccnc2)cnc(Cl)c(Cl)c1 C1(C(N(C)Cc2c(OC)cccc2)=O)CC2OCCC2N(C(=O)C=CCBr)C1 c1(C(N(C(CNC(COCCC#C)=O)C2CC2)C)=O)cn2c(n1)COCC2 C=Cc1cnn(C)c1C(=O)NCC1CCCCC1NC(=O)CCCC(=O)N(C)C CCC(CC)CCCC(=O)N1CC2OCC(NC(=O)CCc3cncn3C)C2C1 c1(C(N2CCC(CC)(NC(=O)C(C)CC(F)F)CC2)=O)cc2c(s1)CCSC2 C#Cc1cc(C(N2CC(NC(c3ccnn3C=C)=O)CC2C)=O)cc(Br)c1 C(=O)(CCC(=O)NN(C)C)N(CC(=O)NCCCC(C)C1CC1)CC#C C(=O)(CCCCC(C)=O)N1C(C(N2CC(CC)OCC2C)=O)CC(=O)C1 Cc1ncc2n1CCN(C(=O)C(CNC(=O)CC1CC(=O)NC1=O)CC(C)C)C2 C(CCC(C)(C)C(=O)N(CCCSC)C)NC(c1c(CC)cccc1)=O c1(C(=O)NC(CN(C(C2C3CCCC23)=O)CC)C)cc(OC)cc(Cl)c1O N1(C(c2c(OC)cccn2)=O)CCN(C(=O)Cc2ccccc2Cl)C(CO)C1 N1(C(=O)NC(C)C)CCOC(C(=O)NCCN(c2ccsc2)C)C1 C1(CS(N2CC3CC(O)CC2C3)(=O)=O)Oc2cc(F)ccc2NC1=O c1(N(C)C)cccc2sc(C(N3CCN(C)C4CC34)=O)cc12 Cc1ccn2cnc(C(=O)NCC3CN(C(=O)C(C)C(C)C4CCC4)C3)c2c1 c1(CC)ccccc1COC(=O)CC(C1CC1)NC(=O)C(C)(C)OCOC C1(NC(C2CC(C#N)C2)C)CC12CCN(Cc1ccc(F)c(O)c1F)CC2 C1(C(=O)NC(CCOC)CNC(C2CN(C(N)=O)C2)=O)(CC)CCC(O)CC1 CCCC(CCCNC(=O)CCC(CC)OC(C)=O)NC(=O)CCC1CCCC1 Cc1ccc(C(=O)NC(C2CC2C(=O)N(C)CC2CC2(F)F)C)cc1O C(=O)(C(F)CCC(C)(C)C)N1C2CC(C(N3C(CCC)COCC3)=O)CC1CC2 N1(C(C2CCN(C)C2)=O)CCC2(CCC(CNC(=O)CC(C)(C)C)CC2)CC1 N1(C(C(C)=C2CCC2)=O)CCCC(CC(=O)NCCC2(C)N=N2)CC1 C12CCCC(C1)C2=O.c12ccc([nH]1)CCC(=O)N2.C1(NC(C)=O)(CO)CCSC1 O(NC(=O)C(c1cn(C)nn1)NC(c1ccn(CC)n1)=O)C(C=C)C C(=O)(C#CC1CCOC1)N(CC(C(=O)NC1(CC=C)CC1)C)C N1(C(C(CC)N(C)C)=O)CCOC(C(=O)N(C(C)CCO)C)CC1 Cc1ccc(F)cc1C(=O)N(CCC(=O)NCc1ccccc1F)C1CC1 c1(C(N2CC(OC)(CNC(c3cc4ccsc4s3)=O)C2)=O)cccn2ncnc12 Cc1nn2ccccc2c1C(N1CC2(CCN(Cc3cnn(C)c3)C2)C1)=O c1(C(=O)NC2CC3(CN(C(C4C(C)(Br)C4)=O)C3)OC2)ccc(F)c2ccccc12 c1(C(=O)NC(C=C)CO)ccc(CNC(=O)C=CC2(C)COC2)cn1 C(=O)(C(CN=[N+]=[N-])NC(c1ccn(C)c1C)=O)NCCn1c(C)nc(C)n1 C1(CCC)CCC(C(=O)NC2CC(NC(=O)C(N3CCC(C)C3)=O)C(O)C2)CC1 N1(C(C(C)SC)=O)CCC(F)(C(=O)N(CC(O)C(C)(C)C)C)CC1 CCCCCC(C)(C)C(=O)NCC1CCCN1S(C)(=O)=O N1(C(C(NOC)=O)=O)CC2CN(C(c3cc4cccnc4[nH]3)=O)CCC12 c1(C(N(CCC(=O)NCc2nncs2)C)=O)cccc[n+]1[O-] CC1CN(C(=O)C=Cc2cscn2)CCC1CNC(=O)COc1ccc(F)cc1 Cc1cc(Br)cc(C)c1CNC(=O)NCC(C)(C)C(C)O C(=O)(C(C)(F)C(C)(C)F)N1C(C(N2CC(OCC)C2)=O)CC(=O)C1 c1(C(=O)NCC(COC)OC(C)C)ccc(CC(C)N)cc1 c1(OC)cc(C(=O)NCC(C)CNC(=O)CC2CCOC2(C)C)sc1Cl CC#CCC(C(=O)N(CC(O)CO)C)NC(C1CCCS1)=O C(=O)(CCCC(=O)NCC1(C)CCN(C(c2ncncc2Cl)=O)C1)N(C)C C1(NC(C2(C)COC2)=O)CC2CCC1N(C(=O)C#CC1CCOC1)C2 c1(C(=O)NC2CN(C(c3ncc(C)c(Cl)c3)=O)CC(F)C2)cn2cc(C)sc2n1 c1(C(N2C(CC)CN(C(C3CCC(=O)N3)=O)CC2)=O)cc2cc(C)ccc2o1 c1(CC)cc(C(=O)NC2C3CN(C(C4CC(F)C4)=O)CC23)cc(N)c1 c1(C(N(CC(CNC(C(COCC)C)=O)C)C)=O)c(C(F)(F)Cl)n[nH]c1C C(C(=O)N1CC(N(C(=O)COc2cc(C)on2)C)C(C)(C)C1)(C(C)(C)C)SC N1(C(C(CCC)C)=O)CC2(CCN2C(c2cnc(C)c(C)c2)=O)C1 c1(C(=O)NC2C(CNC(c3ccc(CS(C)(=O)=O)o3)=O)C2)cc(F)n(C)n1 c1(CC)cc(C(N2CCCC2CN(C(=O)C=C2CCSCC2)C)=O)no1 CCC1c2ccccc2CN1N1CC2CCCC2(CNC(=O)OC)C1=O.C(C)(C)(C)O CC1(CNC(c2ccnc(CNC(=O)C(O)C3CC3)c2)=O)CCCCCC1 c1(C(N(CC(C)CNC(=O)C(=O)C(C)(C)C)C)=O)ccc(N=[N+]=[N-])cc1 C1(CNC(c2c(CC)onc2)=O)CN(C(C2(Cl)CC23CCC3)=O)CCO1 C(=O)(C1=CC2C=CC1C2)NC1(C(NOCC=CC)=O)CCSC1 CCC(C(=O)OC)C(=O)N(CC(N1CCCC(COC)C1)=O)C1CC1 N1(C(C(=O)NC(c2cc(C(C)(C)C)on2)C)=O)CCCC(CN(C)C)C1 C1(NC(c2cc(CC)on2)=O)CCCC(NC(C2(C#N)CCC2)=O)CC1 N1(C(CN(C(C)C)C)=O)CC2C(C(=O)NC3CC(N(C)C(C)C)C3)C2C1 c1(C(=O)NC2(CC=C)CCCN(C(=O)C(F)C(C)C)C2)cc2c(C)sc(C)c2s1 C1(C(N(C(c2ncccn2)C)C2CC2)=O)CC1C1CN(C(=O)C=CC(=O)N(C)C)C1 c1(OC)ccc(Cl)c(CN=c2[nH]cc(-c3ccc(I)c(F)c3F)s2)c1Cl N1(C(c2c(CC)onc2C)=O)CC2CCC2(CC(=O)NC2CCC(O)C2O)C1 c1(NC(=O)CC2CC23CC3)ccc(S(=O)(=O)Nc2ccccc2)cc1 Cc1nn2c(c1CNC(c1cnnn1C)=O)CN(C(=O)Cc1cncn1C)CC2 c1(CCC(=O)NCCN(CCC)C(c2cc(C)sn2)=O)c[nH]c2cc(C)ccc12 Cc1ccc(C2CN(C(C3CCCN(Cc4cnc(O)o4)C3)=O)C2)c(F)c1F CC1=NOC(CCNC(=O)CCOCCN(C)C(C2CCS2(=O)=O)=O)C1 N1(C(C2(OC)CC(C(C)(C)C)C2)=O)CCCC(C2(NC(C)=O)CC2)C1 Cc1ccc2[nH]nc(C(N3C4CCC3CC(CCNC(=O)CNC=O)C4)=O)c2c1 C1(CN(C(=O)C=CC(F)(F)F)C2CC2)CCCN1C(=O)Cc1cc[nH]c1 c1(OCC(NNC(Cn2cc(OC)c(=O)cc2C)=O)=O)ccc2ccccc2c1 n1(CC)cc(Br)cc1C(N1CCC1CNC(C1C(C)CC1C)=O)=O C1(CN(C)C(C2CCOC2)=O)CCCN(C(c2occc2F)=O)C1 CC(C)CC(CNC=O)CC(=O)NC1CC(CNC(C2CCC(=O)C2)=O)C1 N1(C(C(C)C(C)NC(=O)CCc2cccnc2)=O)CC(=O)NC(=O)C1 c1(OC)cc(C(N2CCC(=CC(=O)Nc3ncco3)CC2)=O)ccc1F C1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)N3)=O)C2)CCC2CCCCN12 CCCCC(C)(F)C(=O)N(CCC(C(C)(C)C)NC(c1c[nH]nc1Br)=O)C c1(N2CC(C)(C)NC(=O)C2)nc(NC2CCC3(C2)CC3(F)F)c2ccsc2n1 C1(C)(CC)C=C(C(=O)NC2CC(NC(=O)COC3CCC3)CC2O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CC(NC(CCN(c2ccccc2)C)=O)C1 Cc1cc(C(=O)NC(C2CCCN(C(=O)C(C)(C)F)C2)C)c2cnccc2c1 c1(CNCC(N2C(C)(Cc3ccccn3)C=CC2)=O)cc(O)n2nccc2n1 c1(C(N2CC(CNCc3ccc(C)cc3Br)OCC2)=O)cccc2cn(C)nc12 N1(C(C(C(CC)O)(F)F)=O)CCN2CCN(C(c3cncc(F)c3)=O)CC2C1 c1(CC(=O)NCC2C(C)CN(C(C3CC4CC4C3)=O)CC2)ccc2nn[nH]c2c1 CC(C)(O)C(C(=O)N)NC(=O)C(=O)NC1CCNCCC1CO c1(CNC(C(C(C)(C)C)NC(=O)OC(C)(C)C)=O)nc(=NCC(C)C(C)C)cc[nH]1 N1(C(CSCC)=O)CCOC(CN(C)C(c2c(Cl)n[nH]c2C2CC2)=O)C1 CCC(C)(CNC(=O)COc1ccccc1)C(=O)N(CC(C)SC)C c1(C(N(C2CCCC(NC(c3c(C)snn3)=O)C2)C)=O)cnc2c(c1)CCCO2 c1(C(=O)NCC2C(C)CN(C(=O)CN(C)C)C2)cc(Cl)c(Cl)cc1O N#CCC(C(=O)N1CCOCC1CCNC(C1(C2CC2)CC1)=O)c1ccccc1 CCC(O)C(C)C(=O)NC(C)CC(C)NC(c1ccc(-n2cnnn2)c(C)c1)=O C1(CC(=O)NC2C(C)(C(=O)OCC)C2)CCC(NC(=O)OC(C)(C)C)CC1 c1(OC)ccc(Br)c(NC(=O)CC2CN(C(c3cnco3)=O)C2)c1 C12(C(=O)NCC(C)(CC(C)C)NC(C(C)=CC3CC3)=O)CCOC1CC(=O)NC2 c1(C(N2C(CNC(C(CC)C#N)=O)CC(OC)C2)=O)cnc(C(F)(F)F)c(F)c1 N1(C(c2c(C)c(C3CC3)on2)=O)CCCC2C(NC(c3csnn3)=O)C(C)(C)C12 c1(CC(=O)NC(CCCNC(C2CCC(=C)CC2)=O)C)ccc(O)c([N+](=O)[O-])c1 N1(C(C(C(C)O)(F)F)=O)CC2(COC(CNC(c3cc[nH]c3C3CCC3)=O)C2)C1 C(=O)(C1CCCn2ccnc21)N(C)CC1(NC(=O)CCS(C)=O)CC1 Cc1nc2c(C(N3CCC(O)(CCNC(=O)C=CC(F)(F)F)C3)=O)cccc2o1 CC(C)CC(O)C(C)C(=O)N(C(C)C(N1CCC(N=[N+]=[N-])CC1)=O)C1CC1 N1(C(c2ccn(CC)c(=O)c2)=O)CC2CCCC(C1)N2C(=O)CN1CCCCC1 c12ccccc1COCCOC2=O.N1(CCCOCCC)CC=CC1.C1(=O)CS1 CCC(O)C(C)C(=O)N1CCCCC(N(C(=O)CC2(OC3CCC3)CCC2)C)C1 c1(C(N(C(C(=O)N(CCOC)C)C2CC2)C)=O)csc(C)n1 c1(C(=O)NCc2cccc(NC(c3c(C)n(C)nc3)=O)c2)ncnc2c1CCC2 c1(CC(=O)NC2C(CNC(CCS(C)=O)=O)CC2)ccc(Cl)cc1F CC(C(=O)NC1CC(CNC(C2CCN(C(N3CCCC3)=O)CC2)=O)C1)S(C)(=O)=O c1(CC)ccccc1C(=O)NC1CC(CNC(c2ccn(C3CC3(F)F)n2)=O)C1 c1(C(CF)NC(=O)NC2C(=O)OCC2CO)cccc(F)c1F N1(C(C2(F)CN(C(CC(CC)CN(C)C)=O)C2)=O)CC(C)(C)CCC1C c1(C(=O)OC)ccc(C(=O)NCC2CC2CNC(c2cc(C)n(C)n2)=O)cc1F c1(C(=O)NCC2(CN(C)C(C3CS(=O)(=O)C3)=O)CC2)cnc(O)c2ncccc12 CC(C)CCC(=O)NCCC1(CNC(=O)CC2CCC(C3CC3)O2)CC1 C(=O)(C1CCc2ccc(Br)cc21)NC1C(C)CN(C(=O)Cc2ccon2)C1 c1(OC)cncc(C(N2CCC=CC2C(=O)Nc2conc2C(C)C)=O)c1 Cc1cc(C(F)F)ncc1C(=O)NC1CCN(C(C2CCO2)=O)CC1F CCC(F)(F)CCN=c1[nH]c(=NC(C)c2snnc2C)[nH]c2c1CCC2 C#CC1(O)CC(CNC2CCCNC2CC)C1 CC1COc2c(C(N3CCN(C(c4ccc(O)cc4)=O)CC3C)=O)cccc21 C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(C2CC(CN(C)C)C2)=O)CC1C n1(CC(=O)NCC2C(CNC(c3nnc(C)s3)=O)C2)ccccc1=O Cc1cc(C)c(C(=O)NCCC2CN(C(c3[nH]cnc3C#N)=O)CCO2)s1 c1(C(=O)NCC(C)NC(c2c(C)cco2)=O)ccc2c(=O)ccoc2c1 Cc1oc(C(N2CC3CC2C3NC(=O)CC(C)CC(F)(F)F)=O)cc1S(N)(=O)=O N1(C(CC2CC(NC(COCCC)=O)C2(C)C)=O)CCOC2CCC12 C=CCC(C)(CC)C(=O)NCCC1(CNC(=O)CC2(C)CCCO2)CC1 CCC(C)C(O)C(=O)N(C)CCOCCNC(C1CCN(C(C)=O)CC1)=O C(=O)(CC(CC(N)=O)CC(C)C)NC1C(NC(C2(C#C)CC2)=O)CCCC1 N1(CC2(O)CCN(Cc3ccncc3)C2)CCC(F)(F)CC1 N(C(=NCCc1cc(Br)ccc1OC)NCC1(CO)CCCC1)C(CC)C N1(C(C(CC#C)(C)NC(c2cnc(Cl)n2C)=O)=O)CCCC2(CCC2)C1 C1(CC(=O)NC(Cc2cn[nH]c2)C(=O)NCC(N2CC=CC2)=O)CCCCO1 N1(C(c2cnc(C(C)C)o2)=O)CC2C(C(=O)NC3CCN(C(C)C)C3)C2C1 C1(CC)CC(C(=O)NC2CC23CC(OC)C3)CCN1C(c1ccc(C(N)=O)[nH]1)=O c1(C(C=C)C)nc(-c2ccc(N(CC)CC)cc2)nn1-c1ccnn1C N1(C(C)=O)CCCC1CNC(C1CCC(CNC(=O)COCCC(C)C)C1)=O C(=O)(C1=CCC(C)(C)CC1)C(C(C)CNC(=O)N(C1CCCCC1N(C)C)C)=O c1(SC)nc(O)nc(C)c1C(=O)NCC1CN(C(=O)CCC2OCCO2)CC1C C1(N(C(CN(CC)CC)=O)C)CN(C(c2ccc(OC)cc2Cl)=O)CCC1C C1(C(=O)NC(C)CNC(c2cnccn2)=O)CC2C=CC1O2 N1(C(c2nc(C(C)C)sc2)=O)CCC(OCCNC(=O)C(C)C2CCC2)CC1 CC1CC=C(C(=O)NCC23CC(CN2C(c2ccc(N(C)C)cn2)=O)C3)CC1 N1(C(C(c2ccccc2)NC(c2n(C)ccn2)=O)=O)CC(O)CC(O)C1 N1(C(C2(OC)CCOCC2)=O)CC2CN(C(=O)C=Cc3ccc(OC)o3)CCC12 N1(C(c2ccc(C)nn2)=O)CC2CN(C(C34CCC(C)(CC3)CO4)=O)CC2C1 c1(CC(=O)NC23CCCC2N(C(c2ccsn2)=O)CC3)ccc2c(c1)OCCO2 N1(C(c2c(CCC)nco2)=O)CC2CCC1CN2C(C1(OC)CCC(C)C1)=O C1(NC(CC(=C)Br)=O)CC2CC1CN2C(=O)Cc1c(OC)cccc1F CCCCC(CCCC)NC(C1(C)CC(O)CN1C(c1ccc(O)nc1)=O)=O N1(C(C(Cc2ccc(Cl)cc2Cl)NC(=O)OC(C)(C)C)=O)CCCC(F)(F)CC1 n1(CC#N)ccc(=NC(=O)C2C3CCCC3CN2C(=O)CN2CCCCCC2)[nH]1 N1(C(CCNC(c2c(C(=O)OC)coc2)=O)=O)CC2CC2C(OC)C1 N1(C(CC(=C)C)=O)CCCC(n2cc(CNC(C3CCOC3CC)=O)nn2)C1 C1(C(NOCC)=O)CCN(C(c2cc(C(C)=O)[nH]n2)=O)C1C.c12cn(nn1)C2 CC1C(NC(=O)CCCC(N)=O)CC2CCC1N2C(=O)CC1(CO)CCOCC1 N1(CCN(C(c2c(CC)nc[nH]2)=O)C)CCN(C(=O)CC2(OC)CC2)CC1 Cc1cn2ccc(C(=O)NC3C=CCN(C(C4(C)CC(O)CN4C)=O)C3)cc2n1 c1(C(N2CCC(C)(CCNC(C3ON=C(CC)C3)=O)C2)=O)cccc2nncn12 C1(C(=O)NC2CCC(C(C)C)CC2)(NC(CNC(=O)OC)=O)CCCSC1 C1(NC(C2N(CCC)CCC2)=O)CN(C(=O)C=Cc2cnn(C)c2)CC2(CC2)C1 c1(NC(=O)NC)ccc(Cl)c(C(=O)NC2CC2CNC(c2ncccc2Cl)=O)c1 C1(C(=O)NCC(=O)Nc2c(F)cccc2F)CCc2ccccc2C1 c1(C(=O)NCC(O)CNC(c2cc(F)c[nH]2)=O)ccc2c(c1)OCCCO2 Cc1cc(C(=O)N(C(c2ccc(Br)cc2)C(N)=O)C)nc(-c2ccccc2)n1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(=O)C(O)C(C)(C)C)C12CC2 c1(C(N2CCC3CN(C(C=CC)=O)CC3C2)=O)cc(Cl)cc2ccncc12 c1(CC)cnc2ccccc2c1C(=O)NC1CC(NC(c2cc(C)ncn2)=O)C1 c1(C(=O)NC2CC(CNC(c3nccc(OC)c3)=O)C2(C)C)cc(C)n(C)c1C c1(OC)cc(C)nc(N2CCC(C)C(NC(=O)C=Cc3cncnc3O)C2)n1 CC1CCCC(CC(N2CC(CNC(=O)CCCCNC(N)=O)CC2C)=O)C1 c1(NC2CCN(c3snc(C)n3)CC2)cc(NC2CCS(=O)(=O)CC2)nc(C)n1 CC(CCC(C)(C)C)C(=O)N1CCC1C(=O)NC1CC12CCCC2 c1(N2CC(NC(C3CC(=O)N3)=O)C(O)C2)ncnc2n[nH]c(Br)c12 C1(NC(C(CC)(C)C)=O)CN(C(C2CCC=CCC2)=O)CCC1C C1(NC(CNC(CCC(C)C)=O)=O)CCN(C(C2(C)CCCO2)=O)CCC1(F)F Cn1ncc2c1CN(C(c1c(C3CN(CC4C5CC6C(C5)C46)C3)cnn1C)=O)C2 N1(CC(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)CCC(=O)NC1=O N1(CCCCC)CCC2(CN(C(C3CCCOC3)=O)CC(C)O2)C1 c1(C(c2n(CC)nnn2)NCCC(C)COC)ccc(F)cc1 N1(C(CCCN(C)C)=O)CCCC1(C)CCC(=O)N(C)CC1(CO)CC1 Cc1cc(=O)c(C(=O)NC(C)(CNC(c2sccc2C)=O)CC(C)C)cn1C C1(CCNC(C(=O)NC2C(C)(C)C2)=O)CC12CCCCC2 c1(C(=O)NCC(F)F)ncn2ccccc12.c12ccc(cc1)[nH]2 C1(NC(=O)CNC(=O)C2CC2)CC2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC12 c1(NC(c2cc(C)nn2C(F)F)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(CNC(C)=O)=O)CCCC(N(CCO)Cc2ncnn2C2CCOCC2)C1 C(=O)(C(C)(C)C(F)F)NC1C(CNC(c2c(C)n(CC3CCCC3)nn2)=O)CCC1 Cc1ccc(C(=O)NCCC2CCC(NC(=O)C3=COCCC3)C2)c(C)c1 C1(N(C(=O)CCN2CCC(F)C2)CC#C)CCN(C(C2COCCOC2)=O)CC1 N1(C(c2cc(CC)nn2C)=O)CCOCC(F)(CNC(C2CC2CC)=O)C1 c1(-c2n(CCN(C)C)nc(-c3cc(F)cc(F)c3)n2)n[nH]c2c1COCC2 c1(CNC2(c3n(CCOC)nnn3)CN(C3CC3)CC2C)ccc2sccc2c1 c1(OC)ccc(Cl)c(C(=O)NC2CN(C(C3(C)CC(O)CN3C)=O)C2)c1F O=S(=O)(c1ccc(Br)cc1F)NC1CCC(Nc2ncnc3sccc23)C1 c1(C(=O)OC)cc(F)cc(F)c1NC(C1CSCCN1Cc1cccs1)=O CC1(C)CCCCC(C(=O)NCCCC2CC2(F)F)C1 C1(NC(c2c(C)oc(CO)c2)=O)CC(C(=O)N2CCCC(F)(F)C2)=CC1O CC(C)(O)CC(C)(C)NC(=O)CCCCCNC(=O)CC1CCC(C)(C)C1 C1(NC(c2noc(CC)c2C)=O)CC2CN(C(=O)C3=NOC(C)(C)C3)CC2C1 N1(C(Cc2nc(CC)sc2)=O)CC2(NC(=O)C(CC)N(C)C)CCCC2(F)C1 C1(COC)CN2CCN1C(=O)CCCC2=O.c1(C(=O)NC)sc(Br)cc1F N1(C(C(C)OCCCCCC)=O)CCC(NC(C2(COC)CCCC2)=O)C(F)C1 c1(NC(C(c2cccc(Br)c2)(C)N)=O)ccc(S(F)(F)(F)(F)F)cc1 C=CCC(CNC(=O)C(C)=CCN(C)C)NC(C1CCCN1CCC)=O C1(C(N2CC(CNC(Cc3c(OCC)ccc(Cl)c3)=O)C2)=O)CCC2(CCC2)OC1 c1(CC(=O)NC2C(C)N(C(=O)C(C)O)CCC2)cc(F)c(F)cc1F c1(C(=O)NCCCN(C(=O)Cc2cnc(C)s2)CC)c(F)ccc2[nH]ccc12 CCC(C)C(C)C(=O)NCc1ccc(C(=O)NCC(C)(C)C2CCC2)o1 N1(C(C2(C)COC2)=O)CC2CCC1CN2C(c1cccs1)=O N1(C(C(C)N2CCCC2)=O)CCCCC1CN1CCCC2(CC2)C1 c1(C(=O)NC(C2CCN(C(C(CC)OC)=O)CC2)C)cc(N)cc(O)c1C c1(OC)cc(O)c(C(=O)NC2CN(C(=O)CCNC(C)=O)CC2C#N)cc1OC C1(NC(CCC2CCCN(C(C(C)(C)CC3CC3)=O)C2)=O)CC(C)(C)OC1(C)C n1(CC)cccc1C(=O)NCCC(C)NC(c1ccncn1)=O N12CC(CC(NC(=O)CCCSC)C1)OCC2=O.CCS(=O)(=O)N(C)C(C)C N1(C(C(Cc2ccco2)OC)=O)CC2CCCC2(NC(C2CC2(F)Cl)=O)C1 CC(C)(CC(=O)N1CCCCC(CNC(=O)Cc2ccc(O)nc2)CC1)C(C)C C(CN(C)C)(CN=c1nc(N(C2CCCCN2C)C)c2c([nH]1)CCOC2)OCC C1(NC(Cc2c(C)cccc2)=O)CCCCC12CCCN(C(C1C=C1C)=O)C2 C=CCC(CNC(c1cnoc1-c1ccccc1)=O)NC(C1(C)CC1)=O Cc1cc(C)c(CNC(=O)C(=O)N(C2CCN(c3cccnc3)CC2)C)s1 C1(CC=C)CCCC1N=c1[nH]c(N2Cc3ccccc3C2)nc2ncn(CC)c12 c1(SC)cc(C(N2CC(C(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)c(C)o1 C12(C(=O)NC(C)CNC(=O)Cc3nc(=N)[nH][nH]3)CC(CC(C)O1)C2 CC1CC(C(=O)N(C2CCN(C(=O)CSC(=N)N)CC2)CC2CC2)CCO1 N1(C(C(CCSC)O)=O)CCC(CC(F)F)(CO)CC1 N1(C(C(C)(F)F)=O)CCC2(CC1)CC2NC(=O)CN1C(=O)CNC1=O C(=O)(C(F)(F)C(O)CCCCCCCCC)N(C(C#C)(C)C)C CC1(C)CN(C(=O)CCc2ccoc2)CC1CNC(=O)CSC1CC1 N1(C(CCCC#CC)=O)CCCC2CN(C(=O)C(C(C)(C)C)n3ccnn3)CC12 c1(NC(C2CCCN(Cc3cccc(OCC)c3O)C2)=O)c(C)cc(O)cc1O N1(C(C=CCOC)=O)CC(CNC(=O)CCSCC(C)C)OC2(CCC2)C1 CN1C2CCCC1CN(C(C1CC1C1CN(C(c3coc(C4CC4)n3)=O)C1)=O)C2 c1(NC(=O)NCCN(C)Cc2ccc(C#N)cn2)cn2ccc(Cl)cc2n1 C(=O)(CC(C(F)(F)F)NC(=O)C(C)NC=O)NC1(CNC(COC)=O)CCC1 C(CCNC(C1CC1(C)Br)=O)(C(C)C)NC(C(CC)n1nccc1C)=O C1(C(N2CC(C)OCCC2)=O)CC2CCCC2N1C(=O)CCc1nncs1 c1(NC(C(=O)NC(CC(=O)OC)Cc2cccc(F)c2)=O)cccc([N+](=O)[O-])c1 c1(CC(=O)NC2(CNC(C3(CCC)CCC3)=O)CC2)ccc(OC)c(Br)c1 c1(-n2cc(CNC(C3C(C(=O)OC)C3)=O)nn2)cc(F)cc(F)c1 c1(OC)c(Cl)nc[nH]c1=NCC(C)(C)NC(=O)C1Cc2ccccc21 C(CN=c1ccc(-c2cccc(OC)n2)c[nH]1)Nc1cc(OC)ncc1 N1(C(CC2(OCC)CC2)=O)CCCC2(CCCN2C(C2(C3CCCO3)CC2)=O)C1 Cc1ccc(-c2cccc(-c3nc(COc4ccc(C)cc4C)no3)c2)c(C)c1 C1(CC)C(C(=O)NCC2CCC2(F)F)CCCN1C(=O)CCC1CC1(F)F c1(C(N2CC(CNC(CC(C)OC)=O)C3(C2)CC3)=O)cc2ccccc2o1 Cc1nc(CCC(=O)NC(C2CN(C(C3(C)CC3(F)F)=O)C2)C)oc1C c1(CC)ncoc1C(=O)N(CCCNC(C1CCCO1)=O)CC1CCCC1 Nc1cc(F)cc(Cl)c1C(=O)NCC1CN(C(=O)C2=CCS(=O)(=O)C2)CCCO1 N1(Cc2cc(C)[nH]n2)C(C(N2CCC(Nc3ncccn3)C2)=O)CC2CC12 C(=O)(C(C)CC(C)(C)C)N(CCNC(c1c(C)n(CCO)cc1)=O)CCOCCO C1(CNC(C2(CC#C)CCCC2)=O)CN(c2nc(Cl)ncc2F)CCN1C C1(CN(C(C(C)OC)=O)C)CCN(C(C2CC2C(F)(F)F)=O)CC1 n1(CC)cc(NC(=O)CC2CCCN(C(C3CC3C(N)=O)=O)C2)c(C)n1 C1(C)(C(N2CCC(O)(CNC(c3cncc(CC)c3)=O)C2)=O)COCC1(F)F C(=O)(C(C)Cc1cnc[nH]1)NC(C(n1cc(CCN2CCOCC2)nn1)C)=O C1(NC(C(CC)NC(C)=O)=O)CC(F)CN(C(=O)C(CC)(CC)c2ccccc2)C1 CC(C(=O)N1CCCC(CCC(=O)NC2(C3CC3)CC2)C1)C(C)(C)C CCC(C)CC(C)C(=O)N(C1CCN(C(C2CC23CCCC3)=O)CC1)CC1CC1 Cc1cn2c(n1)C(C)CC(C(=O)NCC(C(C)(C)C)NC(c1ncn(C)n1)=O)C2 Cc1cc2[nH]c(C(=O)NCC3(F)CCN(C(c4cc(Cl)ccc4O)=O)C3)cc2s1 C=CC(C)(CC)C(=O)N1CCCC(CCNC(=O)CC2CC(C(F)F)C2)CC1 c1(CONC(c2cccc(C3CC3)c2)=O)c(Cl)cccc1[N+](=O)[O-] c1(C(N2CCC(O)(CNC(C34CCC(C3)C4)=O)C2)=O)ccc(Cl)cc1Cl C#CC12CC(CN1C(=O)NCc1ncc(-c3cccc(F)c3)s1)C2 c1(C(N(CC(=O)N(CCOCC)C)CC(C)C)=O)cc[nH]c2nccc1-2 c1(C(N2CC(C(C)NC(c3cc(C(C)C)[nH]n3)=O)C2)=O)ccnc2c1CC(=O)N2 Cn1cc(C(N2CC(CNC(=O)C(=O)NCC3CC3)C(F)(F)C2)=O)c(O)nc1=O C1(CNC(C(CC)O)=O)(NC(c2ccc(C(N)=O)nc2)=O)CCOCC1 C1(OC)CC(CNC(C2CC2(C)C(F)F)=O)N(C(=O)CC2CC=CC2)C1 N1(C(CCC#CC)=O)CC2(CCCC(CNC(=O)Cc3ccc(F)cc3C)O2)C1 N1(C(C(C(C)C)C(C)NC(=O)CC23CCC(CC2)C3)=O)CCC2CCC(C1)N2C c1(C(c2n(CCCOC)nnn2)NC(C)CCCCSC)c(F)cncc1F C1(C(=O)N(CCNC(C2(CC(F)F)CC2)=O)C2CC2)CC2CCCC2C1 N1(C(c2c(C)ccc(F)c2)=O)CCC2CC2(C(N2CC(N3CCCCC3)C2)=O)CC1 N1(C(C2(NC(C(c3cncnc3O)C)=O)CCSC2)=O)CCCCCCC1C N1(CCNC(COCCCCC)=O)CCC(N(C)CC(C2CC2COC)=O)CC1 CCCCCC(C1CC1)NC(=O)C(CC1CC1)NC(c1nocc1Cl)=O C(=O)(CCCCCNC(=O)C(C)(C)O)NC1(CCC)CCNC1=O C(=O)(C1(C)Cc2cccc(Cl)c21)NC(CNC(C1CCN(C)C1)=O)(C)C CCC(C)C(O)CC(=O)NCCN(C)C(c1cnc2c[nH]nc2c1)=O Cn1nnc2c1C(C(=O)NC1CCCC1NC(=O)C1=CSCS1)CCC2 C1(C(N(C2CCN(C(=O)CCn3cccc3)CC2)C)=O)CCCC2(CC2)C1 c1(C(N(CC(CC)NC(=O)CCc2ccccc2O)CC)=O)cnc(O)cc1C C12(NC(c3cccnn3)=O)CCCC1N(C(c1cncc(O)c1)=O)CC2 N1(C(CCC)=O)CCN(CC(C)NC(=O)C(C)(C)n2ccnn2)CC1 c1(OCC)ccc(-n2nc(-c3ccccc3Cl)nc2C(c2cnn(C)c2)C)cc1 C(C)(CCNC(=O)C(=O)NCC(F)(F)F)NC(COC)=O C1(NC(C(c2ccc(C(F)(F)F)s2)N(C(C)COC)CCOC)=O)CC(F)(F)C1 N1(C(CC(CC)C2CC2)=O)CC2CN(C(C3(NC(C)=O)CCC3)=O)CC(C1)O2 C1(C(N2CC(C)C(CC(=O)N(CC(N3CC=CC3)=O)CC)C2)=O)CCC(C2CC2)C1 C(=O)(C(O)CCC(C)C)NCC1CN(C(CCCC=C)=O)CC12CC2 N1(C(c2cnn(C=C)c2N)=O)CC2C=CC1C(C(=O)NCC(F)F)C2 N1(C(c2sc(C)c(C)c2C#N)=O)CC(N)CCc2ccccc21 c1(N(CC(=O)OC)C(=O)NC(COC)Cc2ccc(Br)cc2)ccc(Cl)cc1Cl O=C1CCC2(CC1)CC2C(N1CC2CCC(C1)N2C(=O)C=Cc1ccco1)=O c1(C2N(c3ccnc(C(C)(C)C)n3)CCC2)cccc(P(C)(C)=O)c1 c1(C(=O)NC23CC(NC(c4nc(CC)sc4)=O)(C2)C3)ccc2c(c1)COC2(C)C c1(C(=O)NCC2N(C(c3cc(CC(C)C)on3)=O)CC2)ccccc1F N1(C(CCNC(COC)=O)=O)CC(C(C)NC(=O)C(C)OC)C1 C1(C)(CC)CC(NC(c2cn(CCNC(C3(N(C)C)CCC3)=O)cn2)=O)CCO1 CCC(CCC(=O)N1CC(c2ccccc2)(NC(C2C=CCC2)=O)C1)OC c1(OC)ncc(C(N2CCC(C)(NC(c3cn(C)ccc3=O)=O)C2)=O)cc1Cl N1(C(C(C2CCC2)OC)=O)CCCCC1C1CCCN(C(C2(C(N)=O)CC2)=O)C1 CCC(C)CC(=O)N(Cc1cccs1)CC1COCCC1C(=O)Nc1ccccc1 CCC(CC)C(C)C(=O)N(C1CCCN(C(C2(O)CCC2)=O)C1)CC C(CC(C(=O)NC1(C)CCCC1C)NC(c1ccc(N)cn1)=O)SC CC1(C)C(=O)NC2CCC(C(=O)NCC(O)CN=c3cc(F)nc[nH]3)CC12 C1(CC=C)(C(=O)NCCN(CCC(C)C)C)CCN(C(C2CCSCC2)=O)C1 C1(NC(C2(C)CCCC2)=O)CC=C(C(=O)N2CC(OC(=N)O)C2)C1 c1(COC)ccc(C(=O)NC2(CCCNC(=O)C(n3ccc(C)n3)C)CC2)s1 N1(C(CCOCCC)=O)CCN(C(=O)CNC(=O)OC)CC1C1CCCC1 C1(C(=O)NC2(C3N(C(COC(C)(C)C)=O)CCC3)CC2)CCc2nncn2C1 c1(C(N2CCC(C)C2CNC(=O)Cc2cccc(F)c2O)=O)cc(O)ncc1F C1(C(=O)NCC2C(N(C)C)COC2)CN(C(C2CCCC2C2CC2)=O)CC1(F)F CC1(C)OC2(C(=O)NC3COC4(CCN(C(c5cnco5)=O)C4)C3)CCC1CC2 CCC(C)CCCCC(=O)NCCC1CCCN(C(c2cnc(COC)[nH]2)=O)C1 c1(C(=O)NC(C)CC2CN(C(C3(C(N)=O)CC3)=O)C2)nccc2cccnc12 C(CC(C)C)(C(=O)NC(CCO)C(C)C)N(C)Cc1ccc(CC)s1 c1(C(=O)NCC(C)CN(C)C(C2CC2C(F)F)=O)cncn1C C1(NC(=O)CCc2ncc[nH]2)CCCC12CN(C(C13CCCC1CCC3)=O)C2 C1(C(N(CCOCCCNC(CC=CCCCCC)=O)C)=O)CCNC(=O)C1 O=C(N=c1[nH][nH]c2ccc(F)cc12)c1cc(F)c(F)cc1Br N1(C(=O)NC2C(C)(C)COCC2)CCc2c(c[nH]c(=N)c2C#N)C1 N1(C(c2n(CC)cnn2)=O)CCCN(C(=O)CCCc2cc(C)no2)C(CO)C1 Cc1ncnc(C)c1OCC(=O)NCC(C)(C)NC(c1ccsc1C#N)=O C(CC(C)C(=O)NC1CCCC1CNC(=O)CSCC(C)C)=CC c1(C(N(C2CCN(C(c3cc(COC)on3)=O)CC2)CCC)=O)cc(=O)cc[nH]1 c1(C(=O)NC(c2ccccc2)C(C)NC(C=C=C(C)C)=O)cnc(C)c(C)c1 C12(C(=O)NC3CCN(CCNC(=O)CCC4CCCCC4)CC3)CCCC1CCC2 CC1CN(C(C2(c3ccccc3)CCCN2)=O)CC1CC(=O)O C(=O)(CCC(C)(C)C)NC1C2CN(C(c3c(CC)nccc3)=O)CC21 N1(C(C2(C#C)CC2)=O)CCN(CCNC(=O)CC(c2ccccc2)OCC)CC1 c1(NCC2(Cl)CC2)nc2c(c(=NC3CCN(c4ccccn4)C3)[nH]1)SCC2 N1(C(CC)=O)CCC2(CC1)CC2C(=O)Nc1cc(O)ccc1CC N1(C(CCc2nc(C)c(C)o2)=O)CCC2(CC2NC(C2CC2C(N)=O)=O)C1 C1(c2noc(C3(C45CC6CC4C5C6O)CC3)n2)(CO)CCC(F)(F)CC1 CC(C)(O)C(F)(F)C(=O)N1CC2(CCNC(=O)COC3CCC3)CCC1CC2 C1(NC(=O)C(N2CCC(F)(CF)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC2CCCC(CN(C(=O)C3=COCC3)C)C2)cc(F)cc(F)c1 c1(C(=O)NCC(CCCC)NC(C2OCCN(C)C2=O)=O)ccc(C)cc1Cl Cc1ccc(C)c(C(=O)NC2CCN(C(c3ccc(Br)cc3)=O)CC2O)n1 Cc1ccccc1CC1CCCN1C(=O)C(=O)NCC(c1cncn1C)O c1(CC)ccc(C)cc1C(N1CC(CC(C)NC(=O)CCN2CCCCC2)C1)=O C(=O)(C(C)(CC)CCC)N(CCC)CCNC(C1CC(=O)N(O)C1)=O N1(C(COCC#C)=O)CCC2CN(C(=O)C(CC)n3ccnc3)CC2C1 N1(C(=O)Nc2cccc(SCC#C)c2)CCC(C)OC(C)C1 N1(C(C)=O)CCCCC1C(=O)NCCN(C(c1c(O)noc1C)=O)C1CC1 C1(CN(C)C)CCCC1NC(C1CCC1NC(=O)CN1CCCC1)=O CC1(C)C(NC(c2nsnc2O)=O)CC1CC(=O)NC1CCOCC1F CC1(C)CC2(CC(N=c3[nH]c(=NCNC4CCC4)[nH]c4ccc(C(N)=O)cc34)C2)C1 C#CCC(CC(=O)NCC12CCC(CC1)O2)NC(c1c[nH]nc1[N+](=O)[O-])=O C12(CC3(CC3)C1)C(=O)NC2.c1(C(=O)CC2CN(C(=O)OC)C2)cc(C)n(C)n1 O=S(=O)(c1ccc(NC2CCCC3(C2)OCCO3)c(F)c1)NCC1CCCCS1 c1(C(c2n(C(CC)C)nnn2)NCc2cccnc2)cc(C)oc1C N1(C(CC=CC)=O)CC2CN(C(=O)C=Cc3ccoc3)CCC2(CO)C1 C1(C(=O)NCC2N(C(CC(CC)CC)=O)CC(F)(F)C2)CCc2nnn(C)c2C1 N1(C(C(COCC)NC(=O)CC(C)(O)COC)=O)CCC12CCCSC2 N1(C(CCn2cc(CCCS(N)(=O)=O)nn2)=O)CCC(F)(CC#N)CC1 C1(N(C(C=C(CC)CC)=O)C)CCN(C(C2(C(F)F)CC(O)C2)=O)CC1 n1(CCC(=O)NCC2N(C(C(C(C)(F)F)F)=O)CC2)nc2ccccn2c1=O C12CCCC1NC2=O.C(CC(OC)OC)NC(C1(C(=O)OCC)CC1)=O c1(C(N(CCN(C(c2ccc(Cl)s2)=O)CC)CC)=O)cnc(O)c(OC)c1 C1(CC(=O)NC2(C)CN(C(C(C)CSCc3ccccc3)=O)C2)CCN(C)C1=O c1(C(=O)NCCCCN(C)C(c2ccc(CO)o2)=O)ccc(F)c2occc12 Cc1cnc(C)cn1.n1(C(=O)N)cc(C(n2cncn2)C2CC2)nn1 Cc1nc(C(=O)NC2C3CN(C(=O)Cc4ccsc4Br)CC23)c(C)n1C CC1CC(NC(=O)CCC(N)=O)CN1C(=O)CCCc1ccsc1 c1(C(N2C(C)(CC(N3CCC(c4cnco4)C3)=O)CC2)=O)cnn2ccccc12 CC(C)C(O)C(=O)N(C1CC1)CC1CCCN1C(=O)C(c1cccc(F)c1)O N1(C(c2c(C)n(CCC(C)C)nc2)=O)CCC2(CC2NC(=O)CSC2CC2)C1 C1(NC(C=C(CCC)C)=O)CCS(=O)(=O)C12CN(C(c1c[nH]nc1F)=O)C2 c1(C(C)C)ccc(C(N2CC(CC(C)NC(=O)CC3OCCC3C)C2)=O)c(F)c1 CC1CCC=C1C(=O)N1CCCCC1CC(=O)NCCCS(N)(=O)=O C1(CCNC(c2n(CC#C)ccc2)=O)CC(OC)CN1C(c1cncc(N)c1)=O CC(C(=O)NC1CN(C(=O)CN2C(=O)CCC2=O)CC1c1nccn1C)C(C)O C(=O)(C1CCc2cccc(OC)c21)NC1(CCNC(C(CC=CC)C)=O)CC1 N1(C(C(C=C)(C)C)=O)CCC2CN(C(c3n[nH]cc3C(C)C)=O)CC2C1 N1(C(C=CC(C)=O)=O)CC(CCNC(C2(O)CCC2)=O)C(C)C1 c1(C(N2CCC(C(C)NC(=O)CNC(C3CCC3)=O)C2)=O)cccc(C(F)F)c1 c1(C(=O)NC2(C)CCN(C(C3(F)CCCN(C)C3)=O)C2)cc(F)cc(F)c1O C(C(C)(C)C(=O)OC)(c1n(CCCC)nnn1)NCc1csnc1C S(=O)(=O)(c1cc(C)cnc1NCc1cc(Cl)n(C)n1)NC(CC(CC)C)CO C1(NC(c2ccc(C3CC3)s2)=O)CC(F)(CNC(=O)C(F)(F)C2(O)CCCC2)C1 CC1CN(C(C2(C)CCC2)=O)CC1NC(C1(F)CCCOC1)=O N1(C(c2ccnc([N+](=O)[O-])c2)C(=O)Nc2ccccc2)CCC2OCCC2C1 C(=O)(CCCC(=O)NC1CC(F)(CNC(c2csnc2OC)=O)C1)NCCC CC1(C)OC2CN(C(=O)CN3CC(=O)N(Cc4ccc(Cl)s4)C3=O)CC2O1 C(=O)(C(C)(C)CCF)NCC1CCC(CN(C(c2c(C)n(C)nn2)=O)C)CC1 C1(C(=O)NC(CNC(CC=C)=O)CC)CC(F)CN1C C1(NC(CCC(C)O)=O)CN(C(=O)CN2CCC2)CC1(C)C c1(C(=O)NC(CCOCC)C)c(CNC(=O)CC)nnn1C c1(CC)onc(C)c1C(N1CCC(OCCNC(=O)CC2CSCCS2)CC1)=O CC1(F)CN(C(=O)C=CC2CCCCC2)CCN(C(C2(Br)CC2(C)C)=O)C1 C1(C)(CC)C=C(C(=O)N(C2CN(C(c3cnn4cc[nH]c34)=O)C2)C)C1 CCC(CC(C)C)C(=O)NC1CCN(CCCNC(c2csc(C)c2C)=O)C1 c1(OC)ccc2c(=NCc3nc(=N)n(C)[nH]3)[nH]c(=NCCCOC(=N)O)[nH]c2c1 c1(CC)ccc(C(CNC(=O)Cc2cccnc2F)N(C)CCNC(C)=O)cc1 c1(SCC)cc(C(F)(F)F)ccc1C(=O)NC1CC(C)OC1C(F)(F)F c1(CC(=O)NC2C(OC)CN(C(C3CC34CC(O)C4)=O)C2)ccc([N+](=O)[O-])cc1 C1(C)(C(=O)NCC(COC)NC(=O)Cc2nnc(S)s2)CCC2(CC1)CC2 Cc1cc(CNC(=O)C=Cc2cn(C)nn2)oc1C(=O)NCC1(N(C)C)CC1 C1(NC(CCC(C)=O)=O)COC2(CCN(C(=O)Cc3cccc(O)c3)CC2)C1 c1(C(N2CC(C3N(C(C4(CC)CC4)=O)CCC3)(O)C2)=O)n[nH]c2c1CC(C)CC2 C1(NC(C2(SC)CCC2)=O)CN(C(C2CC(C)C2)=O)CCC1C C1(CCN(C(CC)COC)C)CCN(C(c2sncc2C)=O)CC1 C(=O)(C(C)(O)CC(F)(F)F)N1CCCCC(NC(CSC)=O)C1 C12(C(N3C(C(N4CC=C(C)CC4)=O)CC(F)C3)=O)CCCN(CC1)C2 C12(NC(CCc3ccn(C)n3)=O)CCC1CN(C(C1CCOC(=O)N1)=O)C2 C1(CC(=O)NC)CN(C(C2C(F)(F)C23CC3)=O)CCN1C(c1cnc(S)n1C)=O C12(CC(=O)N(C3(C(N(C4CCCCC4)C)=O)CCC3)C3CC3)CCCC1C2.C C1(CNC(CC2(OC)CCC2)=O)CN(C(=O)CCN2CCOCC2)CCC1(F)F C12(CNC(c3ccc(CCC)[nH]3)=O)CC(NC(c3cc(O)n(C)n3)=O)(CCO1)C2 c1(CC(=O)NC(CC)CNC(C2CC(N(C)C)C2)=O)ccnc(Cl)c1F C12(C(=O)NCc3cn(CC)nn3)C(NC(=O)CC3CCSCC3)C3CC1C2C3 c1(C(N2CCC(CC)C2CNC(=O)C2=CCCC2)=O)cc(C)nc(C)n1 C1(F)(CNC(CC(CC)O)=O)CCCN(C(c2cccc(F)c2F)=O)C1 C1(NC(CCCCC)=O)CC(F)(F)CC1NC(c1ccc(SC)s1)=O c1(C(N2CC3C(NC(=O)Cc4ccco4)C3C2)=O)c(O)ccc(Cl)c1F CCCCCCCC(=O)N1CCC(O)CC1C(N1CCC(N2CC(O)C2)C1)=O C#CCCC(C(=O)NC1CC(O)C1(C)C)NC(c1cc(F)cnc1O)=O N#CC1CCC(CC(=O)NCCNC(c2cncc(Br)c2)=O)C1 C(CCCCC(=O)NC1(C(=O)NCC2CC2)CCCCC1)NC(C)=O CCCC(C(=O)N1CCCC1=O)C(C)C.N1C(=S)S1 N1(C(C(C2CCCN(C(=O)Cc3cncnc3)C2)C)=O)CCC(O)C12CCC2 N1(C(c2cn(-c3c(Cl)ccc(OCC)c3)nn2)=O)CC2CCC(COC)C2C1 N1(C(CC(C)(C)O)=O)CCCC2CCN(C(=O)CCCc3ccc(Cl)cc3)CC12 C(=O)(CC(C(F)F)NC(=O)CN(c1nn(C)cc1OC)c1ccccc1)OC c1(C(=O)NCCC2CC(NC(C(=O)NCC)=O)C2)ccc(Br)c(C)n1 c1(OC(C(CC)C2CCOCC2)=O)cn(C)nc1I c1(C(N2C(CCCNC(CCC#C)=O)CCCC2)=O)n[nH]c2ccc(OC)cc12 CC(C)(CNC(c1cc(CNC(c2csnc2Cl)=O)on1)=O)CO c1(CCNC(c2ccc(OC3CCCCC3)c(F)c2)=O)cccc(F)c1Br CC1CCc2ccccc2N1C(N1CC(O)C(O)C1)=O c1(SCC(=O)NC2CCC(N(C(C3(CC(C)C)COC3)=O)C)C2)ccc(F)cc1 N1(C(C2(C)CCCC2)=O)CCCC2(CCC(NC(=O)C=CC3CCCCC3)C2)C1 N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CCCCCC1CNC(C12CC=CC(C1)OC2)=O C1(OC)CCC(S(=O)(=O)Oc2ccc(N3CCOCC3=O)cc2)C1 c1(C(=O)NCCCN(CCCNC(C2CC2Cl)=O)C)ccnc(OC(F)(F)F)c1 C1(C(N(CCNC(c2c(COC)cco2)=O)C)=O)CCCCC(=O)N1 N1(C(c2c(C)nc[nH]2)=O)CC2(C1)CN(C(=O)C(C)N(C)Cc1ccccc1)C2 c1(CNC(C2CC23CCN(Cc2cc[nH]n2)CC3)=O)ccc2cncnc2c1 c1(C(C(N2C(CNC(c3c(C)n(C)nc3)=O)CC2)=O)C)ccc(F)c(Cl)c1 C12(CNC(=O)NC3CCCN(C(c4cc[n+]([O-])cc4)=O)C3)CC3CC(CC(C3)C1)C2 c1(C(=O)Nc2nc(OC)nc(SC)n2)ccc2cc(NC3CNC3)ncc2c1 c1(NC(CCC(C)NC(=O)CSc2nc[nH]n2)=O)ccc(F)cc1O N1(C(C(C(C)C)O)=O)CCOCC(NC(c2cc(C(F)(F)F)ccc2F)=O)C1 Cc1ncc(C(=O)NC2CN(C(=O)CCCc3cnccn3)CC2C)cn1 N1(C(CSC(=N)N)=O)CCN(C2CN(C(=O)CCC3CC3)C2)CC1 C=CCCCCCC(=O)NC1CCN(C(c2nc(C)c(C)s2)=O)CC1(C)C c1(C(=O)N(CCC(N2CCCCCCC2)=O)C2CC2)c[nH]c2ccccc12 c1(C(=O)NC(CNC(C2(NC(C)=O)CCCC2)=O)C)[nH]nc2ncccc12 CC(C)C(C(=O)NCCC(C)(O)C1CC1)C(C)NC(=O)CCC1CC1 c1(C(N2CCC(C(C)NC(=O)C(F)(F)c3nccs3)CC2)=O)cc(=N)[nH]c(=N)[nH]1 O=C1NC(=O)C(C(c2ccccc2)OC)N1.N1(C(=O)O)CC(O)CC1C(=O)O Cc1noc(Cl)c1CC(=O)NCC1CC(CNC(=O)CNS(=O)(=O)N(C)C)C1 c1(CCN2CCCC(C(=O)NC(CC(C)=O)C)CC2)nc2ccc(C)cc2[nH]1 C1(NC(c2c(CCC)occ2)=O)CCN(C(=O)C(F)OC(F)(F)F)C12CCC2 C=CC(C)C(=O)NC1CCN(C(C2CCC2C#N)=O)C1 C1(C(N2CC(CC(C)C)OCC2)=O)C2CCN(C(C3CNC(=O)O3)=O)CC12 c1(CNc2cccc(C(N3CCCC(OC)C3)=O)c2)ccc(Br)cc1I C1(C(N2CCC(C3(C)COC(=O)N3)CC2)=O)CN2CCC1(F)CC2 C12(NC(CNC(=O)OCC)=O)CCCC1CN(C(=O)Cc1ccc(C)c(F)c1)C2 CC1CC(=O)NCC1C(=O)N(CCCCN(C)C(C1(C2CC2)CCC1)=O)C N1(C(CCCC(C)NC(c2cc(=N)[nH][nH]2)=O)=O)CCC2(CCOC2=O)C1 N#CC1(C(=O)CN2C(=O)C=CC2=O)CCNC1.c1(N)ncc(C2CC2)cn1 c1(CNC(c2c(C)oc(Cl)n2)=O)cnc2c(c1)CNC2=O N1(C(c2cccc(C#C)c2C)=O)CCC2(CCN(C(c3cnnnc3C)=O)C2)C1 N1(C(c2c(C)snc2)=O)CCC(C)(C)C1CNC(=O)C(C)C(C)(C)C C1(F)(CNC(c2nc(C)[nH]n2)=O)CCCN(C(C2CCN(C3COC3)C2)=O)C1 N1(c2nnc(COC)s2)CC2CC1CN(C(C1(C)CCC(C)C1)=O)C2 N1(C(c2cc(Br)cc(C)c2C)=O)CCC2CCN(C(=O)C=C3CCCC3)CC12 C(C)(CCS(C)(=O)=O)(c1n(CCCC)nnn1)NCC(C(F)F)c1ccccc1 CCC(CCC(=O)NCCNC(=O)CC1OCCC1C)NC(=O)CO c1(OC)c(C)cc(C)cc1C.c1(C2c3ccc(o3)CN2)ccccc1C C(C)(CCC(=O)N(C1CCN(C(C2OCCCO2)=O)C1)CC1CC1)OC N1(C(c2cc(C)no2)=O)CC2CC1C2NC(C12CCCC1(C(N)=O)C2)=O C1(C2(O)CCOC2)(C(=O)NCCC(C)(C)NC(C(c2cnn(C)c2)C)=O)CC1 C(=O)(CC1=CCN(C)CC1)NC1(C)CC(C(N2CCC(O)(CC(C)C)C2)=O)C1 c1(NC(=O)NCC)cc2[nH]nc(C(N3CCNCC34CC4)=O)c2cc1C(=O)OC.OC C1(CNC(C(CC)C(C)C)=O)CCN(C(=O)CSc2cccc[n+]2[O-])CC1(F)F C12(C(N(CCCNC(C(CO)NC(C)=O)=O)CC3CCCC3)=O)CCC(C1)OC2C C1(NC(Cn2cc(CC)nn2)=O)CN(C(=O)C=C(C)C2CC2)C(C)(COC)C1 C1(C(=O)NC2C(C)CCN(c3cc(CC)nc(CC)n3)C2)COC2(CCC2)C1 C1(OC)C2CCN(C(N3CCOC(CNC(=O)OC(C)(C)C)C3)=O)CC12 Cc1oc([N+](=O)[O-])cc1C(N1CCN(C(C2(C)CC(C#N)C2)=O)CC1C)=O c1(C(C(=O)NC2CC2)N(C)CCOCC2CC2)ccc2c(c1)CCCC2 Cc1cc(C(N2CCN(C(=O)C(C)O)C(CO)C2)=O)n2nc(C(F)(F)F)cc2n1 c1(C(=O)NC2C(NC(=O)CCc3nc(O)n[nH]3)CCC2)cccc2c1CCO2 c1(C(=O)NCCC2CC(NC(CCN(CC(F)(F)F)C)=O)C2)cccnn1 C(=O)(C(C)(O)C(F)(F)F)NC1C(NC(CCN(CCCCC)CC)=O)CCOC1 c1(N(CCCNC(c2ccc(C)s2)=O)C)nc(-c2cccs2)nc2ccccc12 CC(C(=O)N1CC(CN(C)C(c2ccc(CN(C)C)[nH]2)=O)C2(CC2)C1)C(C)(C)C c1(C(c2nnnn2C(C2(C)CC2)C2CC2)Nc2c(C)csc2)ccc(Cl)cc1F C1(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)C)C)COC2(CO)CC1C2 N1(C(c2c(C)n(C)nn2)=O)CCC(F)(C(=O)NC(C)C(C)n2cncn2)CC1 N(C(=NCCN1CCCC1)N1CCC2(CC(C(F)F)=NO2)C1)C(CC)C c1(C(N2CC(N(S(C3(CC)CC3)(=O)=O)C)C2)=O)ccc(O)c(C)c1O c1(OCC)cc(Br)c(ON2CCC(N(C)C)C2)cc1Br c1(C(=O)NCCCCCCNC(C(C)(C)SC)=O)ccc(O)c2ccccc12 C1(O)(CNC(c2c(CC)cncc2)=O)CCCN(C(=O)CN2CC3CC3C2)CC1 CC1CN(C(c2ccc(N(C)C)cc2)C(=O)Nc2ccccc2Cl)CC1C(N)=O N1(C(c2cc(C(N)=O)no2)=O)CC2(CCCCN(C(=O)C(=O)NCC(F)F)C2)C1 C1(NC(CC(C)SC)=O)C(CNC(C2CN3CCN2C(C)C3)=O)CCC12CCC2 C(CCC(C)(C)NC(=O)Cc1cn[nH]c1)NC(CC1(C=C)CCC1)=O C1(C)(OC)C=CCN1C(=O)CCCn1cc(C(c2cccc(N)c2)O)nn1 C1(C(N)=O)CCCCC1C(=O)NC1CCCC(NC(C23CC(CO)(C2)C3)=O)C1 c1(NC(c2n(C(COC)C)ncc2)=O)cccc(F)c1C(=O)OC(C)C N1(C(C2(CC)CCCN2C(c2csc(CO)n2)=O)=O)CCCC(F)CC1 C12(C(=O)NC3CN(C(=O)CC4CC5(CCC5)C4)CC(F)C3)CC1Cc1c[nH]nc12 CCC(CC(=O)NCC(C)(C1CC1)NC(C1CCOC1)=O)CC(C)C n1(CCCC)ncc(-c2nccn2C2C=CCCC2)c1C c1(C(N(CCCNC(=O)CSCC2CCCO2)C)=O)ccc(F)c(O)c1 C(=O)(C(Cn1cncn1)NC(=O)CCc1cc(C)[nH]n1)NC1(CC)CC1 c1(C(N2CC(CNC(C(CSC)OC)=O)OCCC2)=O)ccc2nc(C)cn2c1 C1(C(=O)NCCC2CCCN(C(CC=C=C)=O)C2)CN(CP(C)(C)=O)C1 CC1CC(CNC(c2cn(C3CCC3O)nn2)=O)CCN1C(=O)Cc1cscn1 S(=O)(=O)(c1ccc(C)cc1F)NCC(=O)NC1CN(C(C(CC=CCC)C)=O)C1 CCC(C)C(CC(=O)NC(c1cccc(Cl)c1)C)NC(c1ccnn1COC)=O c1(C(=O)NCC(C)NC(=O)C2=COCCC2)cc2c(s1)C(C)(C)CCC2 C(=O)(C1CCc2c(Cl)cccc21)NCCNC(C=Cc1cnc(OCC)nc1)=O CCCC(C)(CCC)C(=O)NCC(O)CN(C)C(C1CCCOCC1)=O c1(CC(C(=O)NCCN(C(C(C)(C2CC2)NC(C)=O)=O)C)C)ccc(F)cc1F N=c1cc(C(N2CCC(CCCNC(c3cc(Cl)no3)=O)CC2)=O)cc[nH]1 N1(C(=O)CCCCO)CCC2(CCCN2C(C2CCCCS2(=O)=O)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CN(C(C(=O)NCCCC)C)C)C1 c1(C(N2CCOC(CC(F)(F)F)C2)C(=O)NCCC)c(C)nn(C)c1C C1(CC#C)(C(=O)NCC(C)(O)CNC(c2cccn2CC=C)=O)CCCC1 C1(NC(C2(C)CCCC2)=O)CC2CC(NC(=O)CCN3CCOCC3=O)C2C1 Cc1ccc(O)c(C(N2CCCC2C(C)NC(=O)COCc2nnc(C)s2)=O)n1 O=C(C#CC1CCCOC1)NCC12CCC(CC1)N2c1cnc(C(F)(F)F)cn1 Cc1nnc(CCC(=O)NCC2CC2CNC(C2CC=CCC2C)=O)n1C C1(C(=O)OC)Cc2cc(Br)ccc2N1C(c1cccc(C(=O)N(C)C)c1)=O N1(C(c2c(OC)ccnc2)=O)CCOCC(NC(=O)C(C)c2ccsc2)C1 c1(C(=O)NC(CC(C)NC(c2cc(C(C)(C)C)c[nH]2)=O)C)cccnc1O c1(C(N2C(C)CC(CC(=O)NCCc3ncon3)C2)=O)nnc(O)nc1O c1(C(=O)NC2C(NC(C3CCC(COC)C3)=O)COC2)ccc(Br)cc1 c1(NC(C2CC3CC3N2C(=O)C=Cc2cnccn2)=O)ccc(Cl)nc1Cl C1(C(=O)NCCCN(C(c2ccc(SC)s2)=O)C(C)C)CC2CCCCCC12 CCC(C)C(O)C(=O)NCCN(C(c1ccnc(OCCOC)c1)=O)CC C1(NC(C(CC)(C)O)=O)CCN(C(C23CCCN2CCC3)=O)CC(C)(C)C1 Cc1ccc(C(=O)NCC2(F)CC(NC(c3nncs3)=O)C2)cc1 N1(C(C(CCC=C)c2nn[nH]n2)=O)CCC(C)N(C(=O)C=CCOC)CC1 C=CCC(C)C(=O)N(C1CC(NC(c2cn(C)c(O)n2)=O)C1)C N1(C(c2ccc(COC)s2)=O)CCN(C)CC1CNC(C1(O)CCOC1)=O C1(OC)CC(NC(=O)C(C)OCC(C)C)CN(C(c2csnn2)=O)C1 c1(OCC)nc(Cl)ccc1S(=O)(=O)Nc1cccc(C2CCCCC2N=[N+]=[N-])c1 N1(C(CC(COC)C)=O)CCC(C(F)(F)F)n2nccc21 CC1(C)CCC1NC(=O)CCC1CCN(C(C2COCCO2)=O)C1 C1(NC(C2CC(=C)C2)=O)CCN(C(=O)CCC2C(=O)NN=C2C)CC(C)(C)C1 c1(N2CC(SC)C2)ccc(S(=O)(=O)NCc2nn(C)cc2C)cc1C#N c1(CCN(C(=O)CN(C(=O)CC2CCSC2)C2CCC2)C)cccs1 C(CCC(C)C)(C(=O)NC1C2CCCC1COC2)NC(CCCCC#C)=O C(=O)(CC1=NN(C)C(=O)C1)NC1CN(C(CC2(OC)CCOCC2)=O)C(C)C1 C#CC1CN(C(=O)CC2CN(C(c3sncc3CC)=O)CCO2)CC1O O(Nc1cc(OC)cc(OC)c1)Cc1c(C)cc(CC)c(C)c1 c1(NC(=O)NC2CN(C(c3ncccc3F)=O)CCO2)ccc(Br)cc1 Cc1c(C(=O)NCCC2(NC(=O)CCCC(N)=O)CCC2)sc2cccc(F)c12 Cc1cc(CC(N2CCN(C3CN(C(=O)C(C)O)C3)C(=O)C2)=O)cc(C)c1Br C1(C(=O)NCC23OCC(NC(CCCC)=O)(C2)C3)CC(C(=O)OC)=NO1 C(CCc1ccccc1)(C(C)(C)C)NC(COC1(C#C)COC1)=O C1(NC(C(C)Oc2ccccc2)=O)CC2CN(C(=O)CC(C)(C)O)CCN2C1=O C1(CNC(c2c[nH]cc2Br)=O)CCCN(C2CCN(c3cccc(Cl)c3)C2=O)C1 Cc1nc(CC(C)C)oc1C(=O)N(CC(C)(C)CNC(=O)CC(C)(O)C1CC1)C c1(C(=O)OCC(C)CC2CCOCC2)ccc([N+](=O)[O-])c(O)c1 C1(CCNC(=O)CCc2cnco2)CCC(NC(c2ccoc2Br)=O)C1 Cc1cnc(NCC2CN(C(c3csc(Cl)c3C(F)F)=O)CC2C)nc1O C#Cc1cncc(C(=O)NC(C)C(C)NC(c2c(C)ccn2C)=O)c1 c1(C(C)NC(C23C(CN(S(C(C)C)(=O)=O)C2)C3)=O)cc2ccccc2cn1 C1C(=O)N=C2C=CN(N2)C2CN1C2.N1(CCOCCC(C)C)CCc2sccc2C1.NOC N1(C(C(C)(C)C)=O)CCC12CN(C(=O)CC1CCNCC1)C2.c12ccc(cc1)o2 C12COCCN1C2=O.Cc1cc(OCC(N2CCCC2)=O)no1.C1CC(=O)N1 C(C(CC)(CC)NC(=O)C(CC)n1ccc(C2CC2)n1)NC(C(CC)NC(C)=O)=O N1(C(C2CCN(C(C)C)CC2)=O)CC(NC(=O)CN(S(C)(=O)=O)C)C(C2CC2)C1 Cc1ccc2c(=NCc3cccnc3Cl)[nH]c(N3CCCCC(C)C3)nc2c1 CC(C(=O)NCC1(CN(C(=O)C(c2cnn(C)c2)O)C)CC1)C1=CCCC1 Cc1c(Br)c(C(=O)NCCC2CN(C(=O)CCOC(C)C)CCO2)nn1C c1(CC)ccc(C(=O)NC2CN(C(c3ccn(COC)n3)=O)CC23CC3)c(C)n1 c1(CC)onc(C(=O)NC2CC(CCNC(=O)Cc3cncc(O)c3)C2)c1C c1(C(=O)NCC(C)NC(=O)CSc2nc[nH]n2)ccccc1CC(C)(C)C C1(NC(C2CCOCC2)=O)CCN(C(c2cnn3cnnc3c2)=O)CC12CCC2 C1(C(=O)NC(CCCNC(c2c(CC)noc2)=O)CO)CCC(C)(O)CC1 c1(C(N(CC(=O)NCC(C)NC(=O)CC2CC2)C)=O)csc(=N)[nH]1 C(=O)(C1=NNC(=O)CC1)N1CCCC(CCNC(=O)CN2CCCC2=O)C1 C1(O)(C(C(=O)N(C2(C(=O)OC)CC2)C)F)CN(C(C2CS(=O)(=O)C2)=O)C1 CC1CC(NC(=O)C=C2CCCCC2)CCN1C(=O)CCF c1(C(N2C(CN(C)C(C3CCNC3=O)=O)CCC2)=O)cc2c(O)ncnc2cn1 C1(C(N2CC(CCNC(c3cnc(C(C)=O)s3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1oc(C)c(C(=O)NCC2(NC(c3c[nH]c(C#N)c3)=O)CC2)c1Br c1(NCC(N2CCN(c3cccc(C)c3)CC2)=O)c(C)nc2ccccn12 C1(CNC(CNC(CCC)=O)=O)CN(C(c2cccnc2CC)=O)C2CC12 c1(C(N2CC(NC(c3c(COC)cco3)=O)C(C)C2)=O)ncn2c1CCCCC2 N1(CC2N(C(=O)OC(C)(C)C)CCOC2)C(=O)CN(CCOc2ccncn2)C1=O N1(C(C2C(CNC(CC)=O)C2(C)C)=O)CCC(F)(F)CC1 C1(NC(c2cnc(COC)s2)=O)(CF)CCN(C(c2n[nH]c(O)n2)=O)C1 c1(OC)cc(OC)nc(N2CCCC2CNC(c2cc(F)cnc2Cl)=O)n1 CC(C)CC(F)C(=O)NCCOCCNC(=O)CC1CCCCC12CC2 C(=O)(CCC(C)(C)C#N)NCC(C(=O)NCc1c(C)nc(CC)o1)N(C)C N1(C(C(CSC)O)=O)CCCC2(CCN(C(C3(CC(C)C)CC3)=O)C2)C1 N1(C(CCc2onc(C(C)C)n2)=O)CC2(CCN(C(C3COC(=O)N3)=O)CC2)C1 c1(OC)c(C(=O)NC2CCN(C(=O)CN3CCCOC3=O)CC2C)ncnc1C C(CC(=O)NC1CCSC1)(C(F)(F)F)NC(c1nn(C)c(=O)cc1)=O CC(CCC(=O)N1CC=CC1Cn1cc(-c2nccn2C)nn1)N(C)C C1(C(N2CC(N3CCN(C(=O)Cc4cnoc4)CC3)C2)=O)CCCCC2(CC2)C1 c1(C(N2CC3CN(C(c4nn(C)c(F)c4)=O)CC3C2)=O)cccc2cnccc12 C1(NC(COCCCOC)=O)C=CCCC1C(=O)NCCCCSC CC(C)CC(C(=O)NOCCOCCO)NC(C1CCC(=O)C1)=O N1(C(C2(CC(=O)OC)CCCC2)=O)CC(NC(=O)C=C(C)C(F)F)CC(F)C1 CC(C)(C)C(CNC(=O)Cn1cnc(C(N)=O)n1)NC(c1ccc(F)nc1)=O C1(NC(c2ccc(C(C)C)s2)=O)CCN(C(=O)CSCCC#N)C1(C)C C1(NC(C(C)N(C(=O)COCC(C)C)CCC)=O)CCCN1 Cc1ncnc(O)c1C(N1CCC(C2CCCCN2C(=O)C=CCO)CC1)=O CC(C)(C)CC(C(=O)NCCOC(=O)C1CC1)NC(=O)CC1CC=CCC1 C(=O)(C(F)C(C)CC(C)(C)C)NC(C(C)C)CCNC(c1cc(F)cc(F)c1)=O C(=O)(CC1OCCc2sccc21)NCCCNC(c1c(C)c(C(F)(F)F)n[nH]1)=O N1(C(CCOCC(C)C)=O)CCN(C(C2(CF)CCC2)=O)CC1 C1(C(=O)NC(C=C)CO)CN(C)CCN1C(c1cnncc1OC)=O CC1(C)C(=O)Nc2ccc(C(N3CC(NC(C4C=CCC4)=O)CC(F)C3)=O)cc21 C(c1ccco1)=C(C)C(=O)N1CC(=C(F)CNC(=O)Cn2cc[n+](C)c2)C1 C(=O)(CC(C)CC(F)(F)F)NCC1CCN(C(CC(C)C)=O)CC1C Cn1cccc1C1CC1C(=O)NCCNC(c1csc(-c2cnccn2)n1)=O N1(C(C2C(CCC)C2)=O)CC2CN(C(c3cc(CC)ccc3F)=O)CC2C1 N1(C(C(COC)OC)=O)CCC(NC(=O)CNS(N)(=O)=O)C(O)C1 c1(OC)ccc(C=CC(N2CC(C(C)NC(c3ccc(F)cn3)=O)C2)=O)cc1 N1(C(c2cc(C)n(-c3ccccc3)n2)=O)CCC2(C1)CN(C(=O)C=CCO)C2 CC1(C)CN(C(=O)CCc2cnoc2)CC1CC(=O)NCc1[nH]ccc(=O)c1O O=C(CC1CN(C(C2CCCCC2)=O)c2ccccc21)N=c1cns[nH]1 N1(C(c2nccc(C)c2)=O)CCCC(C2CCCN(c3nc(C)ns3)C2)C1 C1(C(=O)NC(C)CNC(=O)CCc2nccs2)CCC2(CC1)CC2 CCC(CC)C(F)C(=O)NC1CC(C)(CNC(=O)CCSCc2ccccn2)C1 CCCC(C)CC(=O)N1CCC(NC(c2cnn(-c3ccccn3)c2)=O)C1 C(=O)(C1=CNS(=O)(=O)N=C1C)NC(CSC)C(N1CCc2nc[nH]c2C1)=O C1(NC(C(CC)(CO)OC)=O)CC12CCN(C(=O)CC1CCCOC1)CC2 C1(NC(=O)Cn2ccnn2)CN(C(C2CCCOCC2)=O)CC1n1cccn1 CC1(C)CCCC(CS(=O)(=O)N(CC(C)(C)NC=O)C)O1 CC(C(=O)NC1CCN(C(c2sncc2Br)=O)C1)S(C)(=O)=O C1(C(=O)NC2C(C(=O)NC3CC(C(C)O)C3)CC2)CC(C)(C)CO1 c1(CC(=O)NCC2(C)CC(NC(C3CC3F)=O)C2)cn2ccccc2n1 C(c1ccc(O)c(O)c1)=CC(N1CC(C(C)NC(c2n(C)cnc2)=O)OCC1)=O C1(CNC(C(CC)OC)=O)CN(C(C2CC3(C2)CC(O)C3)=O)CC1(C)C c1(OC)cncc(C(=O)NC(C2CCCN2C(=O)COC2CC2(F)F)C)c1C O=[N+]([O-])c1cccnc1N1CC(NC2CC2)C1 c1(-c2cc(NCc3nc(C)oc3)ncc2)cc(O)c2ccoc2c1 N1(C(c2ccc(Br)cc2)C2CN(C(c3c(C)cnnc3)=O)C2)CC2CC2C1C#N C1(C(C)C)(C(=O)NCC2C=CCOC2)CCN(C(=O)C(O)Cn2cncn2)C1 CCCC(C)C(=O)Nc1ccc(-c2cnccc2C(=O)OC(C)(C)C)cc1 C1(C(C)O)CCN(C(=O)C(N2CCCC(Cc3nccn3C)C2)=O)CC1 c1(CCOCC(N2CC(CCCCNC(C=CC)=O)C2)=O)cccc(F)c1 c1(CCC(c2n(CCC)nnn2)(C)NC2CCC2C(=O)OC)cccc(Br)c1 C(=O)(C(F)CCC(C)C)NCC1N(C(c2csc(C)c2N)=O)CCC(C)C1 C1(NC(=O)C2=CCSC2)CCN(C(c2csc(F)c2)=O)C(C2CC2)C1 N1(CC2(CS(=O)(=O)Cc3ccccc3)CCCC2)CCCC(S(=O)(=O)N2CCOCC2)C1 c12ccc(C#N)cc1NC2=O.O(N(C)C(=O)C1(OC)CCSC1)CC(=O)OC N1(C(CC(CNC(C(C)CC(F)(F)F)=O)C2CCC2)=O)CCC2(COC(=O)N2)C1 C1(CC(=O)NC(CC#C)CC)C2CCCC2N1C(=O)CC1(C#N)CCOCC1 C(N=c1nc(N2CC(COC(C)(C)C)C2)cc(C)[nH]1)c1cn(CCC)nc1C C1(NC(c2c(OC)csc2)=O)CN(C(=O)C(C)(C(C)C)OC)CCC1CO Cc1ccc2[nH]c3c(c2c1)CC(NCc1ccc(Cl)c(Cl)c1O)CC3 CC(C#N)CCC(=O)N(C1CCCC1)Cc1csc(-c2ccco2)n1 CC1(C)CCC=C1C(=O)N1CCN(C(c2ccc(C(F)(F)F)nc2)=O)CC1C1CC1 N1(C(c2cc(C)nn2C)=O)CCC(NC(C2CC2C(N)=O)=O)C(F)C1 CC1OC2(C(=O)NC(c3cccc(Br)c3)CC3CC3)CCC1CC2 c1(NC(=O)NCc2ccc(C)c(OC(F)F)c2)nnc2c(Cl)cnn2c1O CCC(CN1CCCC(c2n[nH]cc2OC)C1)CC(F)F N1(C(CCC2N(C)CCC2)=O)CCCCC1C(=O)NC1CCN(CC2CC2)C1 C1(NC(C2(CO)CCN(C(C(CC)OC)=O)C2)=O)CC(C)CCC1O n1(C(C)C)cc2c(n1)CC(C(=O)OCC1CCOCC1(C)C)CC2 CC1(C)CN(C(C23CCC(CC2)C3)=O)CC(C)(C)C1NC(=O)CCC1CCOC1 C(c1ccc2ncccc2c1)=CC(=O)NC12CC1CN(C(C1(O)CCOC1)=O)C2 CC1(C)CCc2cnc(CNc3cncc4c3CCC4)nc21 N1(C(CNC(CCC)=O)=O)CCC2(CCN(Cc3ccc4ccccc4c3)C2)C1 c1(N2C3CC(NC(C4(CC)CCC(O)CC4)=O)C2CC3)ncnc2[nH]ccc12 N1(CC(=O)NCC(O)CCNC(c2cncc(Br)c2)=O)CC2CCC1C2 C1(C(=O)NC2CC(NC(c3cc(C(N)=O)[nH]n3)=O)C2)CCn2ncnc2C1 C1(CC)(CC)CCN(C(=O)C(C)N(C(=O)C(CC2CC2)OC)C)C1 C(=O)(C1=COCCO1)N1CCC(N(CCC)C(C2CCC2C)=O)CC1 Cc1nc(N(C)C)sc1C(=O)NCC1CN(C(=O)C=Cc2ccn(C)c2)C1 N(C(=NCCNS(C)(=O)=O)NCC1CCOC1)C(C#C)CCC C1(CC)CC(C)CN(C(C2(CC)CN(C(C3CCN3C)=O)C2)=O)C1 CC1CCCC(C(N2CCC(NC(=O)COc3ccccc3)CC2)=O)C1 N1(C(Cc2c(C)nccc2)=O)CC(NC(c2cncc(CO)c2)=O)CC2(CC2)C1 CCC(C(=O)N(CC(C)N(C)C(c1cc(C(C)(F)F)ccc1C)=O)C)C(C)(C)C C1(NC(C(CCCC)(C)F)=O)CCC2(CC1)CC(NC(=O)CNC(=O)OCC)C2 Cc1ccc(OCC(=O)N(C)C)c(C(=O)NCCCc2ccccc2Cl)c1 CC(C)(O)C(F)(F)CNC(c1csc(CNC(c2cc(Cl)cs2)=O)c1)=O C(CC(C)(C)C)(C(=O)NCC1CCN1C(C1(C#N)CC2(CC2)C1)=O)OC c1(C(=O)NC2C(NC(c3cc(C)sc3)=O)COC2)c(C)noc1C(C)C CC1(CNC(=O)C(O)C(F)(F)F)CCCN(C(=O)CNC(N2CCCC2)=O)C1 Cc1ccc2nc(C)cc(C(=O)NC3CCC(N(C)C(c4cn[nH]c4)=O)C3)c2c1 C(=O)(C(C(C)C)n1cnnc1)N1C(C(C)NC(Cc2c(C)con2)=O)CCC1 c1(CCC)nc(C(O)Cc2ccccc2F)n(-c2cnn(C)c2)n1 C12(CNC(C(CC=C)(C)C)=O)CN(C(c3n[nH]c(C)c3Br)=O)CC(F)(C1)C2 c1(OC)ccc(C(=O)NC(C)CCNC(=O)Cn2c(C)ccc2C)c(F)n1 c1(C(N(C)CC2(NC(C(C)=CC3CC3)=O)CC2)=O)ccc(OC(F)F)c(C)c1 C1(C(=O)NC2(CO)CCCN(C(=O)C3=CCC3)C2)CN2CCCN1CC2 N1(C(C2C(=C)C2)=O)CCCC(CO)(NC(c2cc(CC)ccc2Cl)=O)C1 Cc1nccc(C(N2CCCC(CN(C(=O)CSc3n[nH]c(O)n3)C)C2)=O)n1 Cc1cc(C(=O)NC2CCC(CNC(C3(C)COCCO3)=O)C2)cc(N)c1Cl C1(C)(NC(C(C2CCCC2)OC)=O)CN(C(=O)C=C(C)C(C)C)C(C)(C)C1 C1(C(N2C(CNC(c3cc(OCC)nc(C)c3)=O)CC2)=O)CCn2nncc2C1 N1(C(C(C)CCCc2nn[nH]n2)=O)CC2(C1)CN(C(=O)Cc1ccsc1Cl)CCO2 c1(C(N2CC(N3C(=O)CC(NC(C=CC=CC)=O)C3)C2)C)ccc2[nH]ccc2c1 Cc1nc(C(F)(F)F)oc1C(=O)NC(C1CCCN(C(=O)Cn2cnnn2)C1)C C1(OC)CC(CNC(c2ccc(O)cn2)=O)N(C(c2ccc(F)cc2)=O)C1 c1(SC)nccc(CNC2CC(NC(c3cc(C(F)(F)F)ccn3)=O)C2)n1 CC1CCc2n[nH]cc2C1C(=O)NCCN(C(c1cc(CO)on1)=O)C1CC1 c1(C(N2C(C)(C(=O)Nc3nccc(OC)c3I)CC2)=O)cnn2cccnc12 C(=O)(CCS(C)=O)NC(C1CCN(C(=O)CCCC2CCC2)CC1)C Cc1cncc(C(N2CCCC2C(C)(C)C(=O)NC(C)CS(C)=O)=O)c1 c1(C(=O)NCC(CC(C)C)NC(CCCC(C)=O)=O)c(F)ccc(C)c1Cl C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CN(C(=O)C(C)(C)C(F)F)CCC1CO Cc1nc(N2CCCC(CO)C2)sc1NC(=O)NC(Cc1cccc(F)c1)CO C(CCCC(=O)NOC(CO)C(C)C)N(C(CC(CCOC)C)=O)C N1(C(CC)=O)CCC2CCC(C1)N2C(=O)Cc1c(F)cc(C#N)cc1Br C=CCC(C)(CC)C(=O)NCCC1(CNC(C23C4C5C2C2C3C4C52OC)=O)CC1 c1(C(N(CC(C)NC(c2ccn(C)c2)=O)C)=O)c(Cl)ccc(Cl)c1N c1(N2CCCN(C(CCSC)=O)C(C)C2)ncnc2ccc(O)cc12 C(=O)(C(F)C(C)CNC(=O)C(COC)COC)N(C1CC(=C)C1)C C1(CC(=O)NCC2CCC(N(C)C)C2)(NC(C23CSCC2C3)=O)CCCCC1 C1(NC(C(C)N(C)C)C)CC(=O)N(Cc2ccccc2O)C1 CC1CCn2ncc(C(=O)NC3CCN(C(C4CC(F)C4)=O)C34CCC4)c2C1 Cc1c(C(=O)NC2CC2CNC(=O)C(F)=CC2CC2)cnc2ncnn12 C(=O)(N(CC)OC)C1(CNC(c2cn(CC=C)nc2)=O)CCCC1 N1(C(c2sccc2CO)=O)CCC2CN(C(=O)CCc3ncc[nH]3)CC2C1 c1(NC(C(=O)NC(c2cncc(F)c2)C)=O)ccc2ncn(C)c(=O)c2c1 c1(C(=O)OC)c[nH]c(=NC2CCCC(NC(=O)C(C)n3ccnc3)C2)cn1 CCS(=O)CC(=O)N1CC(C)(CCC(=O)NCC(C)(COC)OC)C1 n1(CC)nc(C)c(C(=O)NC2C=CCN(C(C3CC3C(=O)NC)=O)C2)c1Cl c1(C(=O)NCC(C)(C)N(C(C(C)NC(=O)OC)=O)C)sccc1CO S(=O)(=O)(c1cccc(C(C)C)c1)Nc1c(=O)cc(C(=O)OC)n(C)c1 C12(C(N(CC(=O)OCC)C)=O)CC(C)(CN1C(=O)CSc1cn[nH]c1)C2 C1(CNC(CCCCC)=O)C(C)CCCN1C(c1ccnc(OC(C)C)c1F)=O C#CC(CC(C)(C)C)NC(=O)C(C)(C)CCNC(=O)C(CC)C(=O)OC c1(C(=O)NC(C)C(CO)NC(c2csc3c2CCCC3)=O)cccn2ccnc12 C12(C(N3CCC(NC(C4OCC5CCCC45)=O)(CF)C3)=O)CC3CC1C2C3O N1(C(c2cc(OC)n(C)n2)=O)CCC2CCN(C(c3cncs3)=O)C2C1 N1(C(c2c(C)con2)=O)CC(NC(=O)CC2CCN(C)CC2)CC12CCCOC2 C1(C(N2CCC(OC)(CNC(C3CC=CCC3)=O)C2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NC(COCC)C)CCC(CNC(c2cscc2Cl)=O)CC1 c1(NC(C2=NOC(c3ccc(C)cc3)C2)=O)nc2cc(C)cc(C)c2s1 C(=O)(C1=C2CCN=C2NC=C1)N1C2CC(CN(C(C3(C)CC3(F)F)=O)C2)C1 CC1C(NC(=O)C(Cl)=CCl)CCCN1C(C1CC1c1ccsc1)=O C1(c2cn(CC(=O)NC3CC(C(C(=O)OCC)C)C3)nn2)CC(F)(F)C1(F)F c1(C(N(C2CCN(C(COCC=C)=O)CC2C)C)=O)ccc(Cl)c2ncccc12 C1(CCOCCNC(N)=O)C=CC(CC(CCN2CC(Oc3ccccc3)C2)=O)C1 c1(C(=O)NC2CC(NC(C3N(C)C(=O)CCC3)=O)C2)cc(Br)c(F)cc1F C(=O)(C1CCCc2cccnc21)N1CC(CC(=O)NCC2CC(=O)CO2)(OC)C1 C(=O)(C1=NOC(C)C1)N1CC(C)(NC(c2cnn(CC)c2C)=O)C1 CCC(O)CC(=O)NCCC(C(=O)NCCC1CCN(C)C1)OC C1(NC(COCC)=O)C=CCN(C(=O)C(c2cccnc2)C)C1 c1(C(N2CCCC(N(C(c3c(CC)cno3)=O)C)C2)=O)ccc(F)c(OC)c1F N1(C(CCn2ncc(C)c2)=O)CCC(C2CC2)C1CNC(=O)C1=COCC1 O=C(CCCC1CCCO1)NCC(O)C(=O)NCCc1ccncn1 C1(NC(CC(C)OC)=O)C=CCCC1C(N1CCCC1C(C)C)=O C(=O)(CCCCCCCCCO)NCC1N(C(c2c[nH]c(=N)o2)=O)CCCCC1 C1(C(=O)OC)CC(F)(F)CC1C(N1CCC(O)(CNC(=O)CN(C)C(C)C)C1)=O CC1CC2CN(C(C3CCC4(CC4)N3C(c3cc(CO)on3)=O)=O)CC12 C(c1ccc(F)cc1)=CC(=O)NCCC(C)N(C(=O)Cn1ncccc1=O)C C(=O)(CC(C)C1CCCCC1)NCC(CC)NC(C1CCCCO1)=O C1(CNC(C2CCC(C)CC2)=O)CCN(C(=O)C(F)n2ccnc2)CC1O C1(NCC(C2CCOCC2)OC)CC(NC(c2csc(Cl)c2Cl)=O)C12CCC2 CCC(CC)(CCNC(C1(C)CCCO1)=O)NC(C1CCN(C2CC2)S1(=O)=O)=O C(=O)(C(C)(C)C1=CCSCC1)NCC1CN(C(C=C(C)C(C)(C)C)=O)C(C)CC1 c1(C2(C(=O)NCC3CCC(NC(C)=O)C3)CC2)cccc(Cl)c1F C1(C(=O)NCC2N(C(c3c(C)[nH]nc3Cl)=O)CC(O)C2)COC2(CO)CC1C2 Cc1nc(CC(C)C)sc1C(=O)NCC1C2CN(C3CCSC3)CC12 CCCS(=O)(=O)CC(=O)NC1COCCN(C(=O)COCC(=O)OC)C1 C12(CNC(C(F)=CC)=O)CCCC1N(C(=O)COCP(C)(C)=O)CCC2 C(=O)(CC(C)(C)CCC)N1CC(CCC)N(C(c2cc(Br)ccc2O)=O)CC1 c1(NC(C(N2CCOCC(F)(CC)C2)=O)=O)sc(S(N)(=O)=O)c(OC)c1OC N1(C(CCCNC(C)=O)=O)CC(NC(=O)C2=CCC(C)CC2)CC(F)(F)C1 CC1=C(C(=O)N2CC(NC(c3csc(C4CC4)n3)=O)CC2(C)C)COCC1 c1(C(=O)NC(C2CCN(Cc3nccs3)CC2)C)cc(Br)c2ccccc2n1 c1(C(=O)NC2C(C)(CN(C(CCOC)=O)C)CCC2)ccc(Cl)c(N)c1 Cc1nn(CC(=O)NCC2CC(F)(F)CN2C(=O)Cc2nncn2C)c(C)c1C c1(SC)cccnc1CNC(=O)CN1CCCCC1=O.C123CC(C1)(C2)C(=O)N3 c1(C(N2CC(C)(C(=O)Nc3nc(C)c(C)s3)C2)=O)cc(Br)c(F)cc1C CC1(C)CC(CNC(=O)C=Cc2ccco2)N(C(C2CC=CCC2)=O)C1 N1(C(c2c(Cl)csc2Cl)=O)CC2(C1)CN(C(C1(CF)CCC1)=O)CCO2 c1(C(=O)NCC2N(C(C(CC=C)C)=O)CCCC2)c(-n2cccc2)sc(C)c1C Cc1ccc(C(=O)NC(C2CCN(C(=O)CCOCC(=O)N(C)C)C2)(C)C)cc1 c1(C(N2CCC(Cc3c(C)nn[nH]3)C2)=O)ccnc(NC2CCCC2)c1 Cc1cocc1CN(Cc1ccccc1)CC1CCC1 Cc1cc(F)sc1C(=O)NC1CCCC1CNC(c1csc(Cl)c1Cl)=O C1(=CC=CC(=O)NC(=O)C(O)C2CN(C(=O)CCCN3CCC3)C2)CCCCC1 N1(C(C2(OC)CCSCC2)=O)CCCC2(CCCN2C(=O)C(C)CSC)C1 C1(NC2(OC)CCC(C)C2)CC2(CCNC2=O)C1 C(CC)(CC(F)F)NC(=O)Nc1ccccc1F.c1(CC(CC)OC)ccc(SC)cc1 C(C(C)(C)CNC(=O)COCCN(C)C)N(C(=O)CC1CCC2CC12)C N1(C(C(C)CO)=O)CCCC2C1CCN2C(=O)CC12COC(C)(C1)C2 c1(CCC(N2C(CNC(C3C(CC)CCO3)=O)CCC2)=O)ccc([N+](=O)[O-])cc1 C(CCC(C)(C)C(=O)NCC1CCC1(C)C)NC(C1CN(OC)C(=O)C1)=O C1(N(C(c2cnc(CC)s2)=O)C)CCCN(C(=O)CC(c2cccc(F)c2)C)C1 c1(CN2C(C(=O)Nc3cccc(O)c3)CC3CC32)c(Cl)cccc1[N+](=O)[O-] c1(C2C(C(=O)NC3CC(C)(NC(=O)C=Cc4nccs4)C3)C2)ccncc1F C1(C(=O)NC2(C)CN(C(c3cnc(COC)s3)=O)C2)C(C(=O)OC)CC(=O)N1C c1(C(N(C)CC2CCCN2C(c2ccc(Cl)o2)=O)=O)cnn2c1CC(F)(F)C2 Cc1cc(C(F)F)oc1C(=O)NCC1(O)CC(NC(C2(n3cncn3)CC2)=O)C1 c1(C(=O)NC(C)(C)CCCNC(c2cn(CC3CC3)nn2)=O)ccc(Cl)cc1Cl Cc1ccc(CC(=O)NCCCCC(C)NC(c2cn(C(F)F)cn2)=O)c(C)c1 C(=O)(CC(C(F)F)n1cccn1)NC(CC)(CC)CCN C(C)(C)(CN=c1nc(SC2CC2)[nH]s1)C1CCN(C(C(C)CN(C)C)=O)CC1 CC1CN(C(c2cn(C3COC3)nn2)=O)C(C)CN1C(=O)COCC1CC1 c1(C(N(CCC(C)NC(C2(CC(C)C)CCC2)=O)C)=O)nnn2c1C(=O)NCC2 C(CC(C)(C)C)(C(=O)N1C(CC(=O)NCC(N2CCCC2)C)C2CCCC12)OC c1(CC(=O)NC(COC)C(=O)NCc2cocn2)cncnc1O C1(C(N2C(C(CC)C)CCC2)=O)CCCC(NC(C2CCN(C)C2)=O)CC1 c1(C(=O)NC(CCSC)C(=O)NC(C)C(=O)NO)cncc(F)c1C C1(CCNC(c2cc(CC)n(C)n2)=O)CN(C(=O)Cc2ccno2)CCC1CO N1(C(c2cc(C)[nH]n2)=O)CC2CC(C)N(C(=O)C(C3CCCO3)C3CC3)C2C1 C1(C(=O)NCCCc2cn(-c3ccc(Br)cn3)nn2)CCNCCC1CO CCN=C(NCc1noc(COC)n1)N1CCCC(C2(C)OCCO2)C1 c1(CC(=O)NC(C(C)(C)NC(c2cc(CC)ncn2)=O)C)nc2c([nH]1)CCCC2 c1(C(N(CCCNC(c2coc(Br)n2)=O)C2CC2)=O)cc2ccccc2cn1 c1(SCC(=O)NCC(N(C(=O)C(F)n2ccnc2)C)C2CC2)cnn(C)c1 C(=O)(CCCCC(=O)NC1CN(C(=O)C=Cc2ccccc2)CC1N=[N+]=[N-])NC c1(C(=O)NC(CNC(Cc2c(C)n(C)nc2)=O)C(C)C)coc2c1COC2 C1(CC(=O)NC2(CF)CCC2)CCN(Cc2cocn2)C1 Cc1cc(C)n(CCc2nc(CCc3ccccc3F)nn2CC(N)=O)c(=O)n1 N1(C(CCC)=O)CCCC(CO)(NC(=O)C=C(C)C)C1.c12cccc(c1)C(=O)N2 N1(C(C2CC(CC)C2)=O)CCCN(C(c2nocc2C2CC2)=O)CC1C(C)C N1(C(C(CSC)O)=O)CC2(NC(c3ccon3)=O)CCC1CC2 c1(OCC)ccc(F)cc1S(=O)(=O)NC1CCN(C(c2n[nH]cc2I)=O)C1 c1(C(=O)NCC2N(C(c3c(C#N)csc3)=O)CC(F)C2)ccc2c(c1)CC2 C(C(=O)NCC(C)(C)NC(c1occc1C)=O)(C(C)C)c1cnc(C)s1 CN1CCC(CC(=O)NC2CC2NC(c2ccoc2Cl)=O)C1=O C(=O)(C(C)(C)CC(C)(C)C)NC1CCN(C(CN(CC)CC)=O)CCC1CO Cn1nc(C(=O)NCc2csc(CNC(c3cnoc3C3CC3)=O)n2)cc1O c1(OC)ccccc1C(C)CC(=O)NC1(CO)CN(C(c2c[nH]c(=N)s2)=O)C1 C1(NC(CN(CCC)C)=O)CN(C(=O)Cn2nc(C)oc2=O)C2CCCCC12 CC1(CNC(=O)C(F)OC(F)(F)F)CCCN1C(=O)CC1CCCNC1=O CN1CCC(C)(C(N2CCC(NC(=O)Cn3ccc(Br)n3)C(O)C2)=O)CC1 C1(CC(=O)NC2CC(C)OC2=O)CC2(C1)CN(C(=O)C(C)S(N)(=O)=O)C2 N1(S(CC(=O)OCC)(=O)=O)CC(CO)C2(CN(C(c3cc(F)c(Cl)nc3Cl)=O)C2)C1 c1(C(=O)NC(CCC)CNC(c2cc(C3CC3)sn2)=O)cnc2cccc(C)n12 C1(O)(CNC(CCCN(C)C)=O)CCN(C(c2ccc(CCF)cc2)=O)C1 C1(C(=O)Nc2ccc(F)cc2)CCCN(N2CCC(n3cccn3)C2)C1 CN1CCN(C(C2CCC(=O)N(C)C2)=O)C(C(=O)NOC2CCCCC2)C1 N1(C(c2n(CCOC)ncc2)=O)CCCCC(CNC(=O)C(F)=C2CCC2)C1 c1(C(N2C(CCNC(CCC(C)OC)=O)COCC2)=O)cc[nH]c(=N)c1[N+](=O)[O-] CN1C(=O)CCC1C(=O)NCCC1CC(NC(c2ncoc2Br)=O)C1 c1(CCC(=O)NC2C(NC(c3c(C)ncn3C)=O)CC2)ccc(F)c(F)c1F c1(COC)cc(C(N2CC3CC2C3CNC(=O)CC2(C#N)CC2)=O)ccc1NC Cc1cccc2c(C(N3CCOCC3CNC(=O)C(C)OCC(C)C)=O)coc12 C(=O)(CCS(N)(=O)=O)NC(C)CCNC(=O)C(c1ccccc1F)(C)F N1(C(CC2C(C)C2(F)F)=O)CCCN(C(=O)C=CC(=O)N(C)C)CC1 c1(NC(c2c(-n3cccn3)cccc2F)C)cccn2nccc12 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCC2CN(C(=O)CN(c3ccncc3)C)C2C1 C1(NC(c2n[nH]c(CC)c2C)=O)CCCC(C(=O)N(C)Cc2n[nH]c(C)n2)CC1 C(C)(C)(CCCCC(=O)N1CCCC(CN(C)C(c2cccc(O)n2)=O)C1)OC CC12CCC(C(N3CC4CCCC3(CNC(c3cccnc3)=O)C4)=O)(CC1)CO2 C(=O)(C(CNC(C1(C)CCCC1O)=O)CC1CC1)NCC1(C)CCC1 C(=O)(CC(C)C(=O)OC)NCCC(=C)CNC(C1(COC)CCC1)=O c1(-c2occ(CC(CNC(NCC3N(CC)CCC3)=S)C)n2)cc(C)cc(F)c1 c1(SCC(N2CCN(C(C3CC(C(C)C)OC3)=O)CC2)=O)cc([N+](=O)[O-])n[nH]1 C#CC1CC2CCC1N(C(=O)CC13CCC1CN(C(c1cc(OC)no1)=O)C3)C2 Cc1coc(C(N2CCCC2CN(C)C(C2CCCC(C(F)(F)F)C2)=O)=O)c1C c1(N2CC(NC(C3(OC)CCOCC3)=O)C(C)CC2)ncc([N+](=O)[O-])cc1Br c1(OC)nc(C)ccc1C(=O)NC1CC(F)(CNC(=O)CNS(N)(=O)=O)C1 O=C(C1Cc2c(Cl)cccc21)N1CC(C(=O)OCCC2CCCCC2)OCC1=O C1(C(c2n(CC=C)nnn2)NC2(CCOC)CCC2)CC2(C1)CC(O)C2 C(CCS(N)(=O)=O)NC(C1CC(CNC(C(C2CC2)OC)=O)OC1)=O N1(C(c2ccc(C)nn2)=O)CCC(CNC(c2nnc(O)cc2O)=O)C1(C)C N1(CC(=O)NCC2(NC(CNC(=O)NC)=O)CCCC2)CCS(=O)CC1 N1(C(C2C(=C)C2)=O)CCc2c(c(CNC(=O)CCc3cccnc3)nn2C)C1 c1(C(=O)NCC2CC(NC(Cc3nc(C)oc3)=O)C2(C)C)cc(C#N)ccc1Cl c1(C(=O)NCCC2CC(NC(C=C(C)C(C)(C)C)=O)C2)csc2c1CCC(C)C2 N1(C(CNC(CCCCC)=O)=O)CC(NC(c2ncn(C(C)C)n2)=O)CCC1C Cc1oc(Br)cc1C(=O)NC1CCN(C(C23COC(CF)(C2)C3)=O)C1C1CC1 CCCN=C(NCc1cn(C)nc1-c1ccccc1)NC1CSC1(C)C C1(CCNC(c2ccc(C#C)cn2)=O)CN(C(=O)C=C2CCCC2)CCS1(=O)=O N1(C(c2ccc(=N)[nH]c2Cl)=O)CC23CCCCC2(C1)CN(C(=O)CCF)C3 CCC(C(=O)N1CC(CC(=O)NC(C)CN=[N+]=[N-])(OC)C1)n1cncn1 Cn1nc(C(=O)NCCc2cc(C(=O)NCC3CCCCCC3)no2)cc1O N1(C(Cc2c(C)cco2)=O)CCCCC(NC(=O)CCCC(F)F)C1 c1(CC)cccn2nccc12.C(=O)(C(C(=O)N1CCC(C=O)C1CC)OC)OCC C(CC(=O)NCC1CC1NC(C1(C(N)=O)CC1)=O)(C(C)C)OCC c1(OC)ccc(F)cc1CC(=O)NCC1CC(NC(=O)C(C)(C)O)CCO1 CCC(C(=O)NCCNC(=O)NC)NC(=O)C=Cc1ccsc1 c1(CC)nnc2cc(NC3CC(NC(=O)CC4CC(C)(C)CO4)C3)ncn12 C1(C(=O)NC2(C)CC=CC2)CCN(C(=O)C(O)C(F)(F)F)C(C)(C)C1 C1(C(N2CCCC2CCNC(C2(CCF)CCC2)=O)=O)CC2C=CC1O2 C(CC(=O)N1CC(C)(CO)CC1(C)C)(C(C)(C)C)NC(CN(C(COC)=O)C)=O CN(CCCC(=O)NCCC1(CNC(c2cncc(Br)c2)=O)CC1)N=O c1(N(CC=C)C)cc(NCC)nc(NC(C)Cn2cccn2)n1 C1(N(C)C(C2CC23CCCC3)=O)CN(C(c2cnc(C3CCC3)o2)=O)CC1(C)C C(CN=c1[nH]cncc1I)C1CCC(NC(c2ccoc2Cl)=O)C1 C1(C=C)(C(=O)NC(C#C)CC2CCCC2)CCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(C(N2C3CN(C(Cc4nc(C)[nH]n4)=O)C(CC3)C2)=O)cnc2onc(C)c2c1 N1(C(C(C)n2cccn2)=O)CCN(C(=O)C2=COCC2)CC1c1ccccc1Cl Cc1cc(C(=O)NC(C)C(CO)NC(c2csc(=N)[nH]2)=O)c(C)o1 C1(C(C)O)COCCN1C(=O)C(O)CNC(c1ccnc(CO)c1)=O CCCCCC(CC)C(=O)NC1(C2(COC)CCCCC2)CC1 C(=O)(C(F)C(C)CNC(c1cccc(F)c1)=O)N1CC(c2c(C)con2)C1 N1(C(C(CC(C)C)F)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 C(=O)(CC(C)(C)CCOC)N1CCC(N2CCN(C(CCCCOC)=O)CC2)C1 c1(OC)ccc(CC(C)C(=O)NC(CNC(=O)CNC(N)=O)C(C)C)cc1OC CS(C)(=O)=NCC(=O)NC1(C(=O)NC2CC(=O)NC2=O)CC1 c1(C(=O)NCC(C)NC(=O)C2Cc3c(Cl)cccc32)nnc(O)c2ccccc12 c1(C(=O)OCC)ccc(S(=O)(=O)NCCN2CCOC(C)C2)cc1[N+](=O)[O-] c1(C(=O)NCCN(C(=O)CC2CCC3(CCC3)CO2)C)csc(N=S(C)(C)=O)n1 C1(NC(COc2ccc(C)cc2Br)=O)CCCCN(C(=O)C#CC2CC2)CC1 CCCCC(C(=O)NCCCCCCCNC(=O)CC)ON=C(C)C n1(CCNC(C=CC(C)C)=O)cc(C(=O)NC2(CO)CC(F)C2)nn1 C(=O)(C1=CCCN(C(=O)CNC(=O)OC)C1)NC(CCSCC)C N1(C(C(C=C)O)=O)CCC(C)(C)C(NC(C2CCCC2)=O)C1 c1(C(=O)OCC(CSCC)(C)C)c(OC)cccc1O Cc1cc(F)cc(C)c1C(=O)N(C)C(c1cn(-c2cccc(Br)c2Cl)nn1)C C(=O)(C(CO)C(C)(C)C)NCC(C)NC(c1c(C)nsc1)=O N1(C(C(CC)C)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC12CCC2 c1(C2C(C(=O)NC(CC)CN(C)C(C3CCCO3)=O)C2)c(C)cc(C)nc1O C(=O)(C(F)CC1CC1)N1CC(C(C(=O)NC2(CC3CC3)CC2)O)C1 C(=O)(CS(=O)(=O)CC(F)(F)F)NCCC1(NC(COCCC#C)=O)CC1 N1(C(Cc2nnc(C)o2)=O)CCC(O)(CNC(=O)C(C)Cn2ccnc2)C1 CC(=O)CCN=C(NCc1nnc2n1CCCCC2)N1CCC(c2nncs2)C1 C#CC1CN(C(c2cnc(O)o2)=O)CCN1C(c1ccc(C)c(C)c1)=O C12(CNC(Cc3cc(C)no3)=O)CC(NC(c3csc(C(C)C)n3)=O)(C1)C(C)O2 c1(C(=O)NC2CC(C)(NC(c3oc(C)c(CSC)c3)=O)C2)cn2cnnc2cn1 C=C(C)C1OCCC1C(=O)NC1CC2(C(=O)NC(c3ccco3)CO)COC1C2 C(=O)(C(C)C(F)(F)F)N1CC(OC)C(NC(c2cnsc2C)=O)C1 N1(C(C(CCC)C(=O)OC)=O)CC(NC(C2CCCC2F)=O)CC12CCOC2 Cc1ccc(C2CC2C(=O)NCCOC(C)(C)CNC(=O)CC2CC=CC2)s1 Cc1cc(C(=O)N(C)CC2(CNC(=O)CN(C)S(N)(=O)=O)CC2)ccc1[N+](=O)[O-] N1(C(C=CC(C)C)=O)CCC=C(c2ccccc2O)C1 N1(C(CNC(=O)OC)=O)CC2CCCC1CN(C(c1csc3nnsc13)=O)C2 c1(C(N2CCCC(NC(CC3(C)CCCCC3)=O)CC2)=O)cnc2n1CCCC2 c1(CC)cccc(C(N2CC(NC(C3CCC(CC(F)(F)F)CC3)=O)C2)=O)c1N C1(F)(CNC(C=NOC)=O)CCC(NC(c2c[nH]nc2-c2cccc(Cl)c2)=O)C1 S(=O)(=O)(c1cc(Cl)c(Cl)s1)N1C2CN(C(CN3C(=O)CCCC3)=O)C(C2)C1 c1(C(=O)NCCCC(C)NC(c2scnc2Cl)=O)ccc(=O)n(O)c1 c1(N2CCC(c3c(C)con3)C2)nc2c(F)c(Br)cnc2[nH]1 C(c1cccc(Cl)c1)=CC(N1CC(NC(=O)Nc2ccc(CC)cc2)C1)=O N1(C(CCc2ccc(C)o2)=O)CC(C(=O)NCc2ncccc2Cl)CC1(C)C C1(NC(c2c(C)nc(Cl)s2)=O)CN(C(c2c(F)cncc2F)=O)CC(F)(F)C1 C1(C(=O)NC(C2N(C(C(CC3CC3)OC)=O)CCC2)C)CCC(F)(F)C1 c1(OC)nc(C)c(C(N2CCCC2C(C)NC(c2c(C)cnn2C)=O)=O)s1 N1(C(Cc2c(COC)cccc2)=O)CCCC2CN(C(=O)CS(=O)(=O)N(C)C)CC12 c1(C(=O)NCC(N(C(=O)C(C2CCOCC2)O)C)C2CC2)nn(C)cc1Cl N1(C(c2ccc(OC)c(C(C)(C)C)c2)C(=O)NC)CC(C)C(N=[N+]=[N-])C1 C(CC(C(=O)NC(c1ccccc1F)C)NC(=O)CCCOC)=CC N1(C(c2c(C)ncnc2O)=O)CCCC(O)(CNC(=O)C(F)(F)C(C)C)CC1 CCCC(CC(C)C)C(=O)N1CC(F)CC1C(=O)N(CCC(=O)NC)C N1(C(C(CC)CC)=O)CCCC1C1CCCN1C(=O)COc1ccc(C)cc1 C1(CC(=O)NC2CCC(CNC(c3c(CC)noc3)=O)C2)CN(C)CC1O c1(NC(=O)NC2CCC(C)C2)ccc2c(Br)nn(C)c2c1 C1(CCNC(CCCOC)=O)CCCCN1C(=O)C(C)Cn1ccnc1 C1(C2CCN(C(C3NC(=O)CC3C)=O)C2)(NC(CC2C(C)C2)=O)CC1 c1(C(=O)NC2(C)CCN(C(c3sccc3C#N)=O)C2)cc2ccc(F)cc2s1 Cc1csc(Cl)c1C(=O)NCc1cccc(NC(=O)COCCF)c1 N1(C(C2(N(C)C)CCCSC2)=O)C2CCC1C(NC(=O)C(F)(F)F)C2 C(=O)(C1=C(Cl)CCC1)N(CC)CC1CCN(C(=O)C(c2ccc(F)cc2)F)C1 CC(C)CCCC(=O)NC(CC1CC1)C(=O)NCC(C)(C)C(F)F C(=O)(C(C)(C)C(=O)NCCn1ccc(C(=O)NCC(=O)Nc2cnn(C)c2)c1)OC C1(NCCC(=O)OC(C)(C)C)CCCCC1CNC(=O)CCCn1ccnc1 N1(C(c2c(C)nsc2N)=O)CCC(C)C(NC(=O)CC2(C)CC2(Cl)Cl)C1 C1(NC(C=C(C)Cl)=O)CC(CO)N(C(=O)CCC=CBr)C1 N1(S(CC(=O)NC(=O)NCC(F)F)(=O)=O)CCNC(=O)C1c1cccs1 C1(NC(c2cc(=O)cc[nH]2)=O)CC2C1CCN2C(c1cc(C(F)(F)F)no1)=O c1(C(=O)NC2CCN(C(CC#N)=O)C2)cc(Br)cc([N+](=O)[O-])c1F C1(C(N(CCCN(C)C)CCNC(C2CCCCO2)=O)=O)COC2(CCC2)CO1 CC1CCN(C(=O)C(=O)N(CCCNC(C2CC2Cl)=O)C(C)C)CC1 N1(C(c2c(CCC)n[nH]c2)=O)CC2(CCC2NC(c2csc(C(F)F)c2)=O)C1 C1(C(N2CCC(CN(C(c3cc(C)sc3C)=O)C)C2)=O)CCCNS1(=O)=O CCC(O)CC(=O)N1CC2CC1C2NC(=O)C=C=C(C)C N1(C(c2n(C)ncn2)=O)CCC(NC(=O)CC(C)(C)C2CC2)C12CCC2 C(=O)(CC(O)C(C)CC)NC(CCC=C)C(=O)N1CC(C(C)O)C1 c1(OC)cc(OC)cc(C=CC(N2CCN(C(=O)CC3(C)CC3)CC2CF)=O)c1 C1(C(=O)NCCOC2CCN(C(C=CCC)=O)C2)CCS(=O)(=O)N1 N1(C(c2ccnc(C(C)C)n2)=O)CC(NC(=O)C2=NOCC2)CC2(CC2)C1 C(=O)(CN=S(C)(C)=O)NCC(C1CCC1)NC(CC(c1c(OC)cccc1)C)=O C1(CC(=O)N(CC(C)NC(=O)C=Cc2ccnn2C)CC)CCOC(C)(C)C1 Cc1cccc(O)c1C(=O)NC(C1CCN(C(C2CCCCC2O)=O)C1)C c1(C(=O)NCC(C(C)(C)C)NC(c2cnc(CC)[nH]2)=O)cc(C)c(Cl)cc1F C(=O)(CC(C(F)(F)F)NC(C1CCC(=O)N1)=O)NCCc1c(C)nn(C)c1 CC1=C(CNC(=O)C(c2cccs2)NC(=O)CC2C=CCC2)COCC1 N1(C(C(CC)CCOC)=O)CC2CCCC(C1)N2C(=O)CC(C1CC1)C1CC1 c1(OC)cc(S(=O)(=O)NOC2CCOC2)ccc1F C1(CC(N2CC(N(C)CC)C2)=O)CN(C(c2cc[nH]c2C)=O)CCC1C N1(C(C=COCC)=O)CCC(O)(CCNC(C2CC3CC3C2)=O)C1 N1(C(C(=O)NCC)=O)CCN(C(=O)CCc2ccnn2C)CC1C1CCC1 C1(C)(CC)CCN(C(=NC)NCC2(Sc3ccc(N(C)C)cc3)CC2)C1 c1(C(N2CCCC(CCNC(CC(CC)C)=O)C2)=O)cn2cc[nH]c(=O)c2n1 C1(C(N2C(C3(NC(=O)Cc4csc(S)n4)CC3)CCCC2)=O)CC2(C1)CC21CC1 CCCCCCC(C)C(=O)NC1CCC(C)(NC(=O)C2=NNC(=O)CC2)CC1 c1(NCC(=O)NC(C)(CNC(=O)CCN2CCCC2)C2CC2)ccccc1Cl Cc1cc(CN2CCC(O)C(C(=O)NCc3ccccc3CBr)C2)c(O)c(Br)c1 N1(C(CC2C(C)(C)C2)=O)CC2(C1)CN(C(C13CCCC(CO1)C3)=O)CCO2 c1(C(N2CCN3CC(O)CC3C2)=O)cc(O)nc2ccc(Cl)cc12 C1(O)(C(C)NC(=O)CCc2cnn(C)c2)CN(C(c2coc(CO)c2)=O)C1 C(CCCCC(=O)NCC1OCC2CCC1C2)N(C(=O)C(CN(C)C)N(C)C)C C1(C(=O)NC(C)CCCCNC(=O)CCc2ccccc2)CCOCC12CCC2 C12(NC(=O)C(F)F)CCOCC1CN(C(c1cc(F)ccc1C(F)F)=O)C2 O=C1CCCC(C(N2CCC(NC(c3cnncc3O)=O)CC2)=O)CC1 C(=O)(C(F)(CNC(=O)C(C)NC(=O)OC)C(C)C)Nc1ccc(CC)s1 CCC(C)(C(=O)N1CC(NC(c2ccc(Cl)c(C)c2O)=O)C2(CC2)C1)C(N)=O C1(NC(C(C)O)=O)CCC(C(=O)NCCC(O)CO)OC1 CCCCCC(O)C(=O)N1CCCCC1CCCNC(c1cnc(N(C)C)s1)=O N(C1CC2(CN(C(=O)CCc3cnccn3)C2)n2ccnc21)C(COCC#C)=O N1(C(c2c(C)onc2-c2ccccc2)=O)C2CCC1CC(NC(=O)CC(C)O)C2 N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(=O)C=C3CCC(C)C3)CC2C1 n1(CC)ccc(C(N2CC(NC(=O)C(N3CCCC3CO)=O)C(O)C2)=O)cc1=O Cc1c(C(N2CCC(C(C)NC(=O)C(C)(C)CF)C2)=O)cnn1Cc1ccco1 N1(C(C2C(C(=O)OC)C2)=O)CC2(C1)CN(C(=O)CCc1ccc(C)o1)CCO2 C1(C(=O)NCc2ocnc2C(=O)NCC23CCC(CC2)C3)CCS(=O)(=O)C1 N1(C(c2ccc(OC)nn2)=O)CC(NC(=O)CC(C)SC)CC(F)C1 C1(C(=O)NCCCC(c2ccccc2)NC(COC(C)C)=O)CC2CCC2C1 C1(NC(C2CC(OCC)C2)=O)CC2CCC(C1)N2C(C1CCS(=O)(=O)C1(C)C)=O C(=O)(C1=CCCCO1)N1CC(N(C(COCCCC)=O)CC2CC2)C1 c1(OC)ncc(F)cc1C(N1CCC(CC(=O)Nc2ncc(CO)cc2Br)C1)=O c1(C(=O)NCCCC2(NC(C3C(CC)OCC3)=O)CC2)cc2cc(Cl)cnc2o1 N1(C(C2C(OCC)C2C)=O)CCC2(CCN(C(c3csc4nnsc34)=O)C2)C1 c1(C(N2CC(F)(CNC(CCCCCOCC)=O)C2)=O)onc2cc(C)ccc12 c1(CNC(=O)NC(c2ncoc2-c2cccs2)C(C)C)cccc(C(F)F)c1 C(=O)(C1=CC2C=CC(C1)C2)N1C(CCCNC(CCSC)=O)CCCC1 C1(C2CCCN(C(C3(C#N)CCCOC3)=O)C2)(NC(C(CC)C(C)C)=O)CC1 O=S(=O)(c1ccc(OC(F)(F)F)c(F)c1)NC(CC(F)(F)F)C(=O)O C1(NC(CCCCC#C)=O)CCN(C(c2cncc(N)c2)=O)CCC1CO c1(NC(CN(c2ccccc2)CCC=C)=O)ccc(C(=O)OC)c(OC)c1 C1(C)(C(N(CCN(C(CS(CC)=O)=O)C)C)=O)CCC(C(=O)OC)C1(C)C C1(CN(C(=O)C(C)NC=O)CC)CCN(C(C2CCCOC2C)=O)CC1 CCC(CC)C(C(=O)N1CCS(=O)(=O)C(CCNC(=O)CC(C)(C)OC)C1)OC C1(C(=O)NC(c2ccccc2F)C(C)C)NC(=O)OC1C c1(OC)cc(C(=O)NC(C(N2CCCC2C(=O)N(C)C)=O)C2(O)CCC2)on1 C(=O)(CCC(=O)NN(C)C)N1CCCC(CCC)(NC(=O)C(C2CCC2)OC)C1 N1(C(CCNC(C2C(C)C2)=O)=O)CCCC(CNC(=O)CC2CCC(O)C2)CC1 O=C(C1SCc2cccnc21)N1CCC(CF)C1 N1(C(c2c(C)nn(CC)c2C)=O)CCC(C)N(C(c2cnc(C)cn2)=O)CC1 c1(CC(=O)NCC2(CNC(C(c3ccn(C)c3)C)=O)CCC2)cccnc1 C(N=c1nc2scnc2c(NCc2onc3c2CCCC3)[nH]1)c1c(Cl)cccc1 N1(C(c2cccc(C)n2)C(=O)NC2CCOC2)Cc2cncnc2C1 C12(NC(c3cnc(O)c(Cl)c3)=O)CCC1CN(C(=O)C(F)(F)c1ccccn1)C2 C12CC(C1)CCC(=O)O2.N1(C(=O)OC(C)(C)C)CCC1C(=O)NC1CCOC1 C(c1ccc(Cl)cc1F)=CC(N1CC2(CCN(C(C34CC(F)C3C4)=O)C2)C1)=O c1(C(N2CCCN(C(=O)CC3CC(F)C3)C(CO)C2)=O)cccc2scnc12 c1(CC(=O)NC(CNC(C2N(CC)CC2)=O)(C)CO)ccn2cncc2c1 Cc1nc(N2CCCC(C)(CNC(c3cc(CF)on3)=O)C2)cc(C#N)n1 N1(C(c2ncn(C)n2)=O)CC2CCCC(NC(c3[nH]nc([N+](=O)[O-])c3Cl)=O)C2C1 c1(C(=O)NC2COC3(C2)CN(C(=O)CCn2ccnn2)C3)ccc2c(c1)COC2 c1(C(=O)NC(CC(C)NC(=O)CCc2n[nH]c(=N)s2)C)ncn2c1COCC2 N1(C(C(C=C)O)=O)CCN(CC2CN(C(=O)C=Cc3ccco3)C2)CC1 CC(C)C(O)C(C)C(=O)NC(C1(O)CCCCC1)C(=O)NCCCOCC1CC1 N1(C(C(c2ccccc2)OC)=O)CCN(Cc2ccncc2)C2CC12 c1(OC)c(C(N2CC(CNC(=O)C(C)C(C)(C)O)C2)=O)ccc2c1CCC2 c1(CC(COC(N2CCCCC2CC(=O)CCC)=O)OC)cccc(Br)c1 c1(CC)ccc(C(C(=O)NC)N(CCOCCO)CCN(C)C)s1 CCCCC(CNC(c1ccc(COC)[nH]1)=O)NC(c1cc(Cl)ccn1)=O CON(CCC(=O)N1CC(C2CCC(C)(C)C2)C1)C(=O)C(F)n1ccnc1 N1(C(CC(C=C)CC)=O)CCOC2(C1)CN(C(=O)C1=CCCCO1)C2 Cc1ccc(NCC(=O)NCC2C(C)CCCN2C(=O)CC2=CCCC2)c(Cl)n1 S(=O)(=O)(c1cccc(N2CCOC(C)(CCO)C2)n1)N1C(C)CCCC1 Cc1c[nH]cc(C(=O)NCC(O)CNC(=O)CCn2ccnn2)c1=O C1(C)(C(N2CCC(CC)CC2)=O)CCCN(Cc2ccc(C(C)(C)C)cc2Br)C1 c1(C(C)(C(=O)N(C)CCN(C(=O)COCC(C)C)C(C)C)OC)ccccc1F c1(C(N(C)CC2CCCN2C(=O)CC(C)(C)O)=O)c2c(nn1C)CCS(=O)(=O)C2 c1(C(=O)NC(CN(C(C(C)NC(C)(C)C)=O)C)C)cc(O)nn1C C1(NC(Cc2cn(C)nc2)=O)COCCC1C(N1CCC(F)C1)=O c1(CC)cnc(O)c(NC(=O)NCC2(O)CCCOC2)c1 C1(C(=O)NCC2C(CNC(C3(OC)CCOCC3)=O)C2)CCc2nc(C)cn2C1 C(C(F)C(=O)N1CCC(CN2CCC2)C1)C1CN(C(=O)CC2CC(F)C2)C1 c1(-c2nnc(CC(=O)NON3CCOCC3)o2)ccc(Cl)cc1Cl C1(NC(Cn2c(CCC)ncc2)=O)CC(C)CN(C(=O)CCCC(N)=O)C1 CC1(C)CCC(CC(N2CC(NC(C3CC(=O)NC3(C)C)=O)C(O)C2)=O)CC1 CCC(O)C(CC)NC(=O)CC1CC1CNC(=O)C(C)(F)F N1(C(CN(CC(=O)Nc2cnn(C)c2)C)=O)CCSC2CCCC12 c1(C(=O)NCC(CNC(C(C)(C)N2CCCCC2)=O)F)cc(F)ccc1Cl N1(C(CCC(=C)C)C(=O)NCC)CC23CCCCC2(C1)CS(=O)(=O)C3 C12(C(=O)NC(C=C)C3CCC3)CCCC1CCN2C(=O)C=CC(F)(F)F c1(C(C(=O)NCCCC(C)(C)NC(=O)C=CSC)OC)ccc(Br)cc1 C(=O)(C1c2c[nH]nc2CCC1C)N(CCCNC(c1n(CCC)ncc1)=O)CC Cc1cc(Cl)ccc1CC(=O)NCc1cc(Br)ccc1F C1(O)(CCN2CCCC(NC(N3CCC(COC(C)(C)C)C3)=O)C2)CCCNC1 N1(C(C(C(=O)OCC)C2CC2)=O)CC(NC(C2(OCC)CCC2)=O)C(C)(C)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CC(C2CN(C(=O)C(C)Cc3ccco3)C2)C1 N1(C(COCCC=C)=O)CCN(C)C(C(=O)NC2(C)CCCC2(F)F)C1 C1(NC(=O)C(C2CCOCC2)O)CCN(C(=O)NC2CC2c2ccc(Cl)s2)CC1 C1(CCC)CN(C(c2cc(OC)n(C)n2)=O)CCN1C(c1cnncc1OC)=O C1(CNC(=O)CN2CCOC2=O)C(C2CC2)CCN1C(=O)CC1CN2CCC1CC2 C(CCCCC(=O)NCCc1cc(C(F)(F)F)co1)n1cc(C(C=C)(C)O)nn1 c1(C2N3CCC(C3)NC2=O)nc(F)ccc1Br.C#CC(C1CCC1)OCC c1(C(=O)NC2(CNC(C(CC)C#N)=O)CCCC2)c(F)cccc1[N+](=O)[O-] O=C(CS(=O)C(F)(F)F)NC1CCC(CNC(c2ccc(C3CC3)nc2O)=O)C1 C=C(Cl)C(C)(C)C(=O)N1CC2CC(C1)C2NC(c1[nH]c(C2CC2)nc1C)=O C(=O)(CCC(=O)NN(C)C)NC1C(C=C)CN(C(C2(CSC)CC(F)(F)C2)=O)C1 c1(CC(C(=O)OC)N(C)C)ccc2c(c1)CCN2.C12(OC(C)(C)C)CN(C1)C2=O Cc1nc(NC(c2ccc(O)nc2)=O)sc1CNc1cc(OC(C)C)ncn1 CC(CC(C)(C)C)C(=O)N(C(C)(C)CC(=O)N1CC(O)C(F)C1)C O=C1CCC(CC(N2CCC(Cc3cn(Cc4ccccc4)nn3)C2)=O)O1 c1(C(=O)NCCn2cc(Cn3nccc3C(=O)O)nn2)ccnc2ncnn12 C1(OC)CN(C(=O)OC(C)(C)C)C(C(N)=O)C1Nc1cn(CCN(C)C)nn1 c1(C(=O)NC2C(CNC(c3ccc(C(F)F)cc3)=O)C2)cc(O)cc(F)c1 Cc1ccc(NC(c2ccc(F)cc2NC(=O)OC(C)(C)C)=O)n2ncnc12 c1(C(N(C2CCN(C(=O)C(C)O)C2)CCC)=O)cc(F)c(OC)c(Cl)c1 N1(C(C2N(C(CNC(C)=O)=O)CCC2)=O)CCN(C(C2CC(=O)N(O)C2)=O)CC1 c1(OCCCC(=O)Nc2ccnc(N3CCN(C)CC3)n2)ccc(Cl)c(Cl)c1 N1(C(C23CCC(C(C)=O)(C2)C3)=O)CCCCC(NC(C2(C)CC(C)=NO2)=O)C1 C1(NC(C(C)N(C)C(c2cc[nH]c(=N)n2)=O)=O)CCC(O)C(O)C1 C1(C(=O)NCC(=C)CCNC(=O)CC(C)n2cccn2)CC(=O)N(C(C)C)C1 C(=O)(CCCC(=O)OC)N(C)CCN(c1ccccc1)C(=O)COCCCF Cc1c(F)ccc(Br)c1C(N1CC(NC(c2n[nH]cc2N(C)C)=O)C(O)C1)=O N1(C(c2c(CC)ncs2)=O)CCCC(C)C1CNC(=O)CSCc1cscn1 N1(C(CCC(=O)NC)=O)CCOC2(C1)CN(CC(=O)NCCC1CCOC1)C2 c1(C(C(=O)NC)N(CCN(C)C)C2CC2)ccc(CC(C)C)s1 Cc1n[nH]c(=NC2CC3CC(C2)N(C(c2cnc(C)n2C)=O)C3)s1 c1(CC)ccccc1C(N1CCC(CCNC(=O)CCc2cncn2C)CC1)=O c1(C(N(CCCCNC(CCN(C)CCO)=O)C2CC2)=O)ccc2cnoc2c1 N1(C(c2c(C)nc(COCC)s2)=O)CCCCC(CNC(=O)C2=COCCO2)C1 C(C(C)(CO)NC(c1cc(Br)c[nH]1)=O)NC(C(c1cnccn1)C)=O CCC(COC)C(=O)NCC1CC(NC(C2(C)CCCCO2)=O)C1 C1(C(N2CC(NC(C(C)SC)=O)C(c3ccnn3C)C2)=O)CC(=O)NC(=O)C1 C1(C(C)(C)NC(c2cnn[nH]2)=O)CCN(C(=O)C(F)C2CCC2)C1 CCCC(C)C(=O)NC1CCCC(CC(=O)NCc2ncccc2OC)C1 C#CC1(C(=O)Nc2ccc(OC)cc2)CCN(C(=O)CCc2ccc(C)o2)C1 N1(C(CCOCCOCC)=O)CC2(CCC2)CC1C(=O)NC1(C)CCC1 C#Cc1c[nH]nc1C(=O)NC(C)(CO)C(=O)NC1CN(C)NC1=O C1(CN(c2cccc(OC)c2)CCC)Cc2ccccc2C1C c1(C(N2CCN(C(CCc3ccc(C)nc3)=O)CC2)=O)ccc(F)c2occc12 N1(C(C2CCC(NC(C(CCC)O)=O)C2)=O)CCCC2(C=CCO2)C1 Cc1coc(C(=O)N(C(C)CNC(c2cn(C(C)C)nn2)=O)C)c1C CC1CN(C(C2(C(F)F)CCCO2)=O)CCC1CN=c1ccnc[nH]1 C(=O)(C(F)C(=O)N1CC(n2cc(C3CC3)nn2)C(O)C1)OCC c1(C(c2ccc(OCC)nn2)Nc2ccccc2Cl)c(C(F)(F)F)cccc1F C1(C#N)(CC(=O)NC2CC(C)N(C(=O)CSc3cccc[n+]3[O-])C2)CCOCC1 C1(NC(=O)OC(C)(C)C)CCCCCC1NC(=O)Cc1cc(O)cc(Br)c1 c1(C(=O)NC(C2CCOC2)CO)nc(Cl)sc1Cl C1(c2n(C(CC)(C)C)nnn2)(NCC(C)CC2CCCC2)COCC1CN(C)C c1(C(C)=O)cc(C(=O)N(C2CCN(C(=O)CN3CC=CC3)CC2)CCO)oc1C CCC(C(=O)NCC1(NC(C2CC2COC)=O)CCC1)c1ccccc1 C1(CNC(C(C)(C)NC(=O)OC)=O)C2CN(C(C3(c4ccccc4)CC3)=O)CC12 c1(C2(OC)CN(C(c3sccc3C3CC3)=O)C2)ccccc1F Cc1c(NCCCCCC2CC2)ncnc1NC1CCSC(C)(C)C1 C12(C(=O)NCCNC(=O)NC)CC(CO1)N(C(C1CC3C(C1)C3(F)F)=O)C2 C1(OCC(=O)NC(C)Cn2cc(-c3cnn(CCF)c3)nn2)C#CCCCCC1 C(N=c1[nH]c2c(c(=NCc3nc(C4CC4)n[nH]3)[nH]1)COCC2)c1ncsc1 CC1NC(=O)OC12CN(C(C1C=CC(NC(=O)C=C3CCOCC3)C1)=O)C2 Nc1cnnc(NNC(=O)C2CCCCC23CCC3)c1Cl c1(C(=O)NCCC(C)N(CCC)C)cc(CNC(C2CC2Cl)=O)on1 N1(C(Cc2c(C)cnn2C)=O)CC2(CC(NC(C3(N=[N+]=[N-])CC3)=O)CO2)C1 C1(N2C(NC(=O)CCc3nc(-c4cccc(F)c4)no3)CCC2)CCCCCC1 C1(OC)CN(c2nnc(CC(C)(C)O)n2CC(=O)OC(C)(C)C)C1(C)C Cc1cccc(C(=O)NCC2COCCN2C(=O)Cc2cc(F)cc(F)c2)c1Cl C1(C(=O)Nc2cnc(C)c(Cl)c2)CC2(CCC2)CN1C(C1COCC(C)O1)=O c1(C(=O)NCC2C(CNC(C(CC(C)C)(C)C)=O)C2)cccc2c1CCC(=O)N2 c1(NC(C2CC(F)CN2C(c2cncs2)=O)=O)cccc(-n2cccc2)c1 c1(NC(C2(C=C)CCC2)=O)ccc(NC(C2CC2C2CC2)=O)c(C)c1 CS(=O)(=O)C1CC(C(c2nnnn2C2COC2)NCCCN2CCCC2=O)C1 N1(C(c2cc(C)c(C)s2)C(=O)NCC(F)F)CCOC2(CCCCC2)C1 C1(C(N2C3CN(C(CCC=CC(C)C)=O)C(C3)C2)=O)COc2ccc(O)cc2O1 C1(NC(c2ccc(CC(N3CCCCC3)=O)o2)=O)CCN(C(C2CC2Cl)=O)CC1 C1(COC)(NC(c2cnn[nH]2)=O)CCCN(C(=O)CC2CCC2C2CC2)C1 CC(CN=c1cccc(S(=O)(=O)NCCCSCCO)[nH]1)c1nccs1 c1(NCCOCCC=C)nc(C)cc(=NCC(C)c2ccc(F)cc2)[nH]1 C(CC(C)(C)C)(c1n(CC=C)nnn1)(C1CC1)NC1CCCC(C)(C)C1 c1(C(C)(C)C)cccc2c1OCC2C(=O)NCc1sccc1Br C1(O)(CCNC(C(CCO)N(C)C)=O)CCCN(C(c2cscc2C#N)=O)C1 CC(=O)C(C)(C)CC(=O)NC1CN(C(C2CC3CC3C2)=O)CC1CC1CC1 C1(c2n(CCSC)nnn2)(NCc2cccc(Cl)c2Cl)CCCN(C(C)(C)C)C1 C=C=CCCC(=O)N1CCCC(CN(C(C2(N3CCCC3)CC2)=O)CC)C1 c1(-n2nc(C(N(CC(=C)C)C)=O)c(CCO)c2)ccc(F)cc1F O=S(=O)(c1ccc(Br)cc1NCCS)N1CCC2C(F)(F)C2(c2ccccc2)C1 C(CC1CC1)(C(=O)NCCN1CCCCC1)NC(CN(CC(C)C)CC)=O C1(C)(CNC(C2CCN(CC)C2)=O)CCCN1C(C1CCSCC1)=O C1(CNC(COCCC(C)C)=O)(NC(=O)CC2CCCSC2)CC(F)(F)C1 C(=O)(C1CCCc2nncn21)N(CC(C)O)CCNC(=O)CC(C)(C)C C1(N(C(C(CC)(C)C)=O)C)CCN(C(=O)CNC(c2cccc(C)c2)=O)CC1C c1(C(=O)NC(C2CN(C(=O)CC#N)C2)C)ccc(S2(=O)=NCCC2)cc1 Cc1[nH]c2c(F)cccc2c1CCNC(C1CCCCC1C)=O c1(CC)ncsc1C(=O)NC1CCCC1CN(C)C(C1CC(OC)C1)=O N1(C(c2c(C)nc(C(C)C)s2)=O)CCC(CO)C(NC(c2nn(C)cc2Cl)=O)C1 C1(CC(=O)NC(C(C)NC(=O)Cc2cn(C)nn2)(C)C)CCC(=O)NC1 C(=O)(C(C)(C)C(N)=O)NC(CCN(C(CN1CCC(C)C1)=O)C)C(C)C c1(C(C(=O)NC2CN(C(CC(C=C)C)=O)C2)O)ccc([N+](=O)[O-])cc1 c1(C(N(C2CNCCC2(F)F)c2cc(COC)ncn2)=O)cc(F)c(F)c(F)c1 c1(OCCC=C(C)C)ccccc1Cc1cccc(N2CCC2=O)c1 CCCCC(C)(F)C(=O)N1CCC(NC(C2CCC(C)(C)O2)=O)C(F)C1 C(CC1(C)c2nnnn2NCCN1)SC.c1(CC2CCOC2)scnc1C N1(C(Cc2ccc(SC)cc2)=O)CC2(CCCCC2NC(=O)CNC(=N)N)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C2OCCN(C(CC(=O)OCC)=O)C2)C1 N1(C(CC(CC)(C)C)=O)C2CCC1CN(C(C13CCC1C3)=O)C2 n1(CCCNC2C(CC)COCC2)c(C)cc(O)cc1=O N1(C(c2c(CNC(CC3C(=O)NCCC3)=O)ccs2)=O)CCOC2(CCC2)CC1 CN1CCN(C(c2cc(C(F)(F)F)no2)=O)C(CNC(c2ccc(=O)oc2)=O)C1 c1(CN2CCC(C(C)(C)C)(NC(N)=O)C2)ccsc1S(C)(=O)=O.C1(=O)CCCN1 c1(C(=O)NCC(C)CN(C)C(c2cnnn2C)=O)cnccc1N(C)C c1(OC)nc2cc(N(C(=O)CC(C)c3ccccc3)C)ccc2o1 C(=O)(C1Cc2ccc(F)cc21)NC1CCN(C(C(C)NC(N)=O)=O)C12CCCC2 c1(C(=O)NC2C(NC(C3(OC)CCSC3)=O)CCC2)ccc(C2CC2)cc1Cl c1(C(N2CCCC(C)(NC(c3cnc(C)n3C)=O)C2)=O)cccc(S(C)(=O)=O)c1 c1(N(C)Cc2n(CC)cnn2)[nH]c(=NC2CCOCC(C)C2)nc2scnc12 CCCC(C)C(C)Nc1ncccc1C(F)C(F)(F)F CP(C)(=O)C(O)C(=O)NCCN1CCC(NC(=O)CC2CC(F)(F)C2)CC1 c1(CC(=O)NC(C(=O)NC)C2(O)CCC2)ccc(Cl)cn1 c1(C(=O)NC(CC)(CNC(=O)CC2CCCCCCC2)CC)cnc2[nH]cnc2c1 C1(C(=O)NCc2c(C(C)C)noc2)CN(C)CCN1C(C1C2CCC(F)(F)C12)=O c1(C(=O)NCC(C)(CNC(=O)COCc2ccncc2)OC)cccn(C)c1=O Cc1cc(C(=O)NCCNC(C2CC2C)=O)c(C)n1C1CCCCC1 N1(C2CCN(c3nc(=N)[nH]c(=N)[nH]3)C2)C(=O)C2CCCCC2C1=O c1(OC)cccc(C(=O)N(C)CC2CCN(C(=O)Cn3cc(Cl)c(C)n3)C2)n1 N1(C(C(C)N2CCCC2)=O)CC2CC1(C(N1CCC(OCC3CC3)C1)=O)C2 c1(C(=O)NCCC2(CNC(CSC)=O)CC2)cnc2c[nH]nc2c1 c1(C(N2C(C)CN(C(c3c(C)onc3)=O)C(C)C2)=O)cccc(P(C)(C)=O)c1 C1(CCC)(NC(=O)CC(C)(C)O)CCCN(C(c2cnncc2OC)=O)C1 N1(C(c2cc(OC)nc(Cl)c2)=O)CCC2(NC(=O)C=Cc3cnc[nH]3)CCCC12 N1(C(=O)OC(C)(C)C)CC2CC2(NCc2snnc2C2CC2)C1 c1(C(N2CCC(NC(=O)Cn3cc(Cl)cn3)C(O)C2)=O)ccc2sccc2c1O Cn1cc(-c2ccc(C3CC(C)(Cc4ccccc4)C(=O)O3)cc2)n(C)c1=O C1(C(N2CC(NC(c3ccnc4c3CCO4)=O)C(O)C2)=O)CCCC2(CCC2)C1 C(CC(=O)NC1CC2CC(NC(=O)CCSC3CCCC3)C1C2)(C(C)C)OCC C1(C)(COC)CC(NC(=O)C(C)(C)C)CN1C(=O)Cc1ccc(C)nc1Cl N1(C(C(C)Cc2ccccc2F)=O)CC2CCC(C1)N2C(=O)CC1COC(=O)C1 N1(C(c2c(C)csn2)=O)CCCCCC1C(=O)NCc1ccncn1 C1(C(N2CC(N(C(C(CC)C#N)=O)C)C2)=O)CS(=O)(=O)CC12CC2 C1(CC(=O)N(CCCNC(c2ccccc2O)=O)CCO)CCCCC12CC2 Cc1ccc(Cl)c(N)c1C(N1CCC(NC(=O)C(C)NC=O)C(F)C1)=O CCCCC(O)CC(=O)N(C(C(N1CC2CCC(CO)(C2)C1)=O)C1CC1)C N1(C(c2c(C)nsc2-c2ccccc2)=O)CCOC(C)(CNC(=O)OC(C)(C)C)C1 N1(C(c2c(SCC)cc(Cl)cc2)=O)CCC(N(C)C(c2ccon2)=O)C2(CC2)C1 C(=O)(C1=C(C)OCC1)NC(C(=O)NC(CC)CN1CCOCC1)C CCCCCCC(C)CC(=O)NC1CCC(O)CN(C(c2ccoc2CC)=O)C1 Cc1nn(C)c(C)c1CC(N1CCSCC1CCNC(c1cncn1C)=O)=O c1(C(C(=O)Nc2ccccc2)N(C)Cc2c(C)nc[nH]2)csc(S(N)(=O)=O)c1 S(=O)(=O)(c1cc(C(F)(F)F)cc(O)c1)NC(c1c(C)ccc(SC)c1)=O C(CC1CCCC1)(C(=O)N(CCCNC(=O)Cc1cnc(C)[nH]1)C(C)C)OC c1(C(N2C(CNC(C3CCC4CCC3O4)=O)COCC2)=O)ccc2sccc2c1 N1(C(CS(CC)=O)=O)CCCC(C)(NC(c2cnn(C3CC3)c2C2CC2)=O)C1 Cc1cc(F)c(CC(N2CCC3CC3(NC(=O)CN(C)C3CC3)CC2)=O)cc1F Cc1ncc(C(=O)NCCCNC(=O)C(c2ccc(F)cc2F)C)cc1N Cc1ccc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CC2(C)C)=O)nc1 C(C(C)(C(=O)NC1CCCCC1)NC(C1CCCO1)=O)SC Cc1ccc(C(=O)NCC2CC2NC(c2c[nH]nc2-c2cccnc2)=O)c(N)c1 C(=O)(C1Cc2c(Cl)cccc21)N1C(C2(NC(CCCCOC)=O)CC2)CCCC1 C(=O)(CC(C)N(C(c1cc(Br)cs1)=O)C1CC1)NCCCOC c1(C(=O)NC2CC(C(=O)OC)C2)c(OCCCOC(C)C)cccc1NC(C)=O N1(CN(c2ncccn2)CCOC)CCC2(CCCCN(C(=O)OC(C)(C)C)C2)C1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NCC=CCNC(=O)C1=CCCCC1 c1(NCCCCCCNC(C2(C)ON=C(C)C2)=O)ccc(C)cc1[N+](=O)[O-] C=CCC(CNC(=O)C(F)=CCC)C(=O)NCC(C)(O)CC(C)C c1(SCC=C)ccc(C(=O)NCC2CC2C)cc1.N12CC3CC1C3C2=O CCC(=O)CCC(=O)NC(CC1CCC1)C(=O)NC1CN(C)CCC1O C1(NC(C(C2CCCC2)OC)=O)CN(C(=O)CCS(C)=O)CC1(C)C Cc1cc(C)c2onc(CC(=O)NNC(=S)NCC(O)CC(F)(F)F)c2c1 C1(C(C(=O)N(CC(=O)NC)C)C)CCCN(C(=O)C=Cc2cocn2)C1 c1(-c2scc(C(=O)OCC(CO)Oc3ccccc3)n2)ccc(OC)cc1 c1(C(N2CC(N(C(c3c(CC)c[nH]c3)=O)C)C2)=O)cc(O)c2ccccc2c1 Cc1c(F)ccc(C(=O)NC2CCC(N(C(=O)CC3OCCO3)C)CC2)c1C CCC(CC)CCCNC(=O)C(Cc1cc[nH]n1)NC(c1ccc(CO)o1)=O C1(CNC(=O)OCC)CCC(CNC(C2CC2)=O)CC1.C(=O)(C(F)=CCCF)N c1(OC)ccccc1C(=O)NCC(CO)NC(=O)CC1CCC1C c1(CC)c(C(=O)NC2CC(O)(CNC(=O)C(C)(C)OC)C2)[nH]c(C)c1C(C)=O N1(C(CC(CC=C)NC(c2nccs2)=O)=O)C2CCC1CC(CO)C2 c1(C(C(=O)NCC2CCCO2)N(CC)Cc2cnn(C)c2)cccc(COC)c1 Cc1c(CCNC(N2CCCCC(C)(F)C2)=O)ccc(Cl)c1Cl N1(C(C(CC)C(C)O)=O)CCc2nc(NC(=O)C(=O)NCCNC(C)=O)sc2C1 N1(CC(=O)N(CC(C)(C)CNC(c2cn(CC)cn2)=O)CC)CCS(=O)(=O)CC1 C1(NC(C(CCN(C)C)O)=O)C2CCC(C2)C1C(=O)NC1(C(C)(F)F)CC1 C#Cc1ccc(CNC(C2CN(C(C3CC4C=CC3C4)=O)CCO2)=O)cc1 N1(C(CCCOC(C)C)=O)CCOCC(NC(=O)C(c2ccc(Cl)cc2)O)C1 C=C(C)C1CN(C(=O)CC2CN(C(c3cn(C)c(C)n3)=O)C2)CCO1 C1(OC(C)C)CCCCC1NC(C1CCC(=O)N1)=O.N12CCC(CC1)NC2=O C=CC1(C(=O)N(C)CC2(COC)CCC2)CCN(C(=O)CC2CCCNC2=O)C1 C1(OC)CN(C(c2c(Br)noc2C2CC2)=O)CC1NC(c1ccoc1)=O CN1CC=C(C(=O)NC2CC(CNC(=O)CCn3cnc(=N)[nH]3)C2(C)C)C1 c1(-n2ncc(C(=O)NCC(CC)NC(=O)CC3CNC(=O)C3)n2)ccc(F)cc1 C(=O)(C(F)(F)c1cscn1)NCCN(C1CCCC1)C(COCC=C)=O c1(CC(=O)NCCCCC2CN(C(C)=O)C2)cnc(N(C)C)cn1 c1(C(=O)OC)ccc(F)c(Cl)c1.c1(OCCN2C(=O)C2)ccc(Cl)cc1 N1(C(C2C3CN(C(c4c(CC)ncs4)=O)CC32)=O)CCc2ccc(C#N)cc2C1 C(=O)(C(C)(CO)OC)NCC1C(C(=O)NCC(=C)Cl)CC1 CCS(=O)CC(=O)NC(C1(CNC(c2ocnc2CO)=O)CC1)C c1(OC)cc(C)ccc1CNC1CCC(C(=O)NC(c2ccc(Cl)cc2)C)OC1 N1(C(c2nn(CC)c(C)c2)=O)CCC(CNC(c2cc(C)c(C)o2)=O)C12CC2 c1(C(N(CC(CC)NC(c2csc(C)c2)=O)C)=O)cn2ccsc2n1 CN1CC(O)CC1C(=O)NC(C(=O)NCC(F)(F)C(F)F)C1(O)CCC1 C(c1ccccc1Cl)=CC(N1CCC(NC(CC2CN(CC(C)C)C2)=O)C1C)=O C1(C)(NC(C2OCC(C)C2)=O)CCCN(c2ccncn2)C1 c1(C(=O)NC2(C)CN(C(=O)C(c3ccccc3)NC(N)=O)C2)cncc(N)n1 c1(C(N2CCOCC(NC(C=CCC)=O)C2)=O)c(CCC)sc2c1CCC2 C(CC(C(=O)NC(CC1CC1)CC(=O)NCCCC1CCC1)OC)OC N#Cc1cc2cc(-c3cccc(CN4CCCC4CO)c3)cnc2cn1 c1(OC)cccc(Cn2cc(CCCN(C(C3CC3OC)=O)C3CC3)nn2)c1 n1(C(C(=O)Nc2ccc(C)c(Br)c2)C)cnc2ccccc12 C1(CC(=O)N(C)CC2(N(C)C)CC2)N(C(c2cccs2)=O)CCC1(C)C N1(C(=O)C=Cc2cnc[nH]2)CCCC2C1CCCN2C(=O)Cn1ccccc1=O c1(CC)ccc(C(N2CCC(F)(CNC(C3CCCSC3C)=O)CC2)=O)c(F)c1 Cc1ccc(C2CC2C(=O)NC2(CNC(=O)CC3CCCCO3)CCOC2)cn1 C1(C(N(c2ccc(F)cc2)CC)=O)C2CN(C(=O)C(C)(C)CF)CC12 C1(NC(c2cccc(OC)c2)=O)C2CC3C1C3C2C(=O)NOCC(N)=O c1(SC)ccc(N)cc1C(N1CC2CC(NC(C3(C)CCC(=O)NC3)=O)C1C2)=O C1(C)(C(N2CCC(C=C)C2)=O)CN(C(c2cccnc2)=O)CC1C C1(CC=C)(C(=O)N(CC(C)(C)NC(C2CC2C(C)O)=O)C)CCC1 c1(C(=O)OC)ccc(C)nc1NC(C)(CNC(C1CCCN1C1CC1)=O)CC C1(NC(C(CCC)CC)=O)CC2(CCN(C(C3(OCC)CCC3)=O)CC2)C1 N1(C(C(C=C)O)=O)CCOCC12COCCN(C(C1Cc3cccnc3C1)=O)C2 CC(C)CCCCC(=O)N(C(=O)CC(C)C(F)F)CC1CCCOC1c1cn[nH]c1 c1(C(=O)NCC2CCC(NC(C3CC(C#C)(O)C3)=O)C2)nccc(Cl)c1C N1(C(c2cc(CNC(C(C(C)C)O)=O)on2)=O)CCCC2(CCC2)C1 N1(C(c2cc[nH]n2)=O)CC2(CCOCC2)CC1CNC(C1CC(CF)C1)=O c1(CNC(=O)NCC2(CO)CC(C)C2)ccc(O)cc1Br C=C(CC)CN=c1[nH]c(=NCC(CCO)c2cccnc2)c2cc(Cl)ccc2[nH]1 C1(CNC(c2ncn(CCC)c2)=O)CCCCC1NC(=O)C(c1csc(C)n1)=O N1(C(C2OCCN(C)C2)=O)CC2CC(F)(F)CCC2(N)C1 CCC(CSC)(c1nnnn1C1CCOC1)NCC=Cc1ccco1 c1(C(=O)NCC(C)N(C(C(n2ncc(C)c2)C)=O)C)noc2c1CC(C)(C)CC2 c1(C(=O)NCCCCCN(CC=C)C)c(CNC(=O)C=C2CC2)cnn1C n1(CC)cc(Cl)c(C(=O)NCC(C)(O)CNC(=O)C(F)(F)c2cncs2)n1 c1(C(N2CCCC(NC(C=C3CCC(C)C3)=O)C2)=O)ccc2c(c1)COC2(C)C C1(C)(NC(CC2CC(C(=O)OC)C2)=O)CCN(C(c2cc(C)c(CO)s2)=O)C1 C(=O)(C1=CCC(NC(c2c(Cl)cnn2C)=O)C1)NC(CC)C1CC1 N1(C(c2cc(OC)n[nH]2)=O)CCCC(CCNC(C2(O)CCSCC2)=O)C1 C1(NC(c2cccc(C(F)(F)F)c2)=O)CCCCC1NC(C1(F)CC2(CC2)C1)=O c1(C(=O)Nc2cccc3ccc(Br)nc23)cc(C2=CCNCC2)c2[nH]ncc2c1 CC1CCC(CC(=O)NCCOC2CN(C(=O)CSc3cccs3)C2)CC1C C1(O)(C(C)NC(C23CC(C2)C3)=O)CCN(C(C2CCCN2C)=O)CC1 C1(C(=O)NC2(C)CN(C(=O)CC3(C)OCCO3)C2)CC2CCC1C2 C=CC1CN(C(c2cc(F)ccc2F)=O)CC1NC(c1ccccc1SC)=O c1(C(=O)NC2CCCN(C(=O)Cc3ncc(Cl)s3)CC2)cc2ncccc2[nH]1 c1(CC(=O)N(C2CCCC(N(C(C=C(C)C)=O)C)C2)C)c[nH]c2cccc(C)c12 c1(CC)cc(Br)ccc1NC(C1CCCN(C(C2CC2(F)F)=O)CC1)=O c1(SC(C(N2C(CNC(Cc3scc(C)n3)=O)CC2)=O)C)ccc(F)cc1 C=CCC(CNC(C1(CC(=O)OC)CC1)=O)NC(=O)CC(C)n1cccn1 C1(CC(N2CC(C(C)NC(C3CC34CCCC4)=O)C2)=O)NC(=O)NC1=O C1(NC(C2(OC)CC2)=O)CCC(C(=O)N(CCCN=[N+]=[N-])C)C1 C(CCC(O)C(=O)NCc1ccc(CO)cc1)NC(C1(C)CCN(C)C1)=O C(=O)(CC(C)(C)C(F)F)N1C2C(NC(c3c(C)cncn3)=O)CC(C2)C1 C=CC1CN(C(=O)C(C)Cc2ccc(O)cc2)CC1NC(c1cnc(Cl)s1)=O c1(C(N2C(C)CN(C(C3COCCO3)=O)CC2)=O)ccc2nc(CO)[nH]c2c1 C1(NC(c2c(CCC)occ2)=O)CN(C(=O)Cc2nc(C)sc2C)CC(C)(C)C1 N1(C(COC)=O)CCc2ccccc2C(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(C(=O)NC2CC(C)(NC(=O)CCN3CCC3)C2)ccc2ccoc2c1 C12(C(=O)NCC3(SC)CC3)CCN(C(C3CCC3C(F)F)=O)CCC1C2 c1(C(N2CCC(C)(C(=O)NCC3ON=C(C)C3)C2)=O)cc(C)cc(C)c1 c1(-c2ccc(CO)cc2)csc(=Nc2cccc(O)c2)n1Cc1ccccc1Br CCC(CC1CCCC1)C(=O)N(CCCN(C)C(C1CC1c1cnn(C)c1)=O)C C1(NC(CNC=O)=O)CC(C(=O)NC2CC(OCCO)C2)C12CCC2 C1(C)(OC)CCCN(C(C2CC(O)CN2C(=O)C=CC(F)(F)F)=O)CC1 Cc1cc(C(=O)NCC(=O)NCCNC(=O)CC2CCCC2O)c(C)o1 C1(C(=O)NC2CC(NC(=O)C(C3CCOCC3)O)C2)CCCCC(F)(F)C1 C1(NC(=O)COc2ccsc2)CC2CC(NC(c3nc(Cl)cs3)=O)CC2C1 C1(N(C(C(CC)F)=O)CCO)CCN(C(=O)Cc2ccsc2C)CC1 C1(C(=O)NCC2(COC)CCCN2C(=O)COCCC(C)C)CCCS(=O)(=O)N1 c1(C(N2CCC(N(C(=O)C=Cc3cnccn3)CC)C2)=O)c[nH]nc1[N+](=O)[O-] Cc1cc(N(C)C(c2ccccc2F)C)ccc1NC(N)=O N1(C(CC2CCCN(C(C3CN(C)C(=O)CC3)=O)C2)=O)CCOCC(F)(F)C1 C(=O)(C(CC(C)SC)N1CCN(CC(C)C)CC1)NC(C(=O)OC)C CCC(CN(C)C)C(=O)N1CCCC(CCC(=O)NCC(O)COC(C)C)C1 NC1CCN(C(=O)C(=O)NCc2ccncc2)CC1CO C1(c2nc(C(CC)SC)n(-c3cccc(C)n3)n2)CCC(F)(F)CC1 c1(OC)c(C(=O)NC2(C)CN(C(c3c(F)ccnc3F)=O)C2)cccc1F Cc1sncc1C(=O)NC1CCC1NC(=O)CCc1cnc(Br)s1 C1(NC(C(C)C#N)=O)C=CCN(C(=O)CN(C)Cc2cccc(Cl)c2)C1 N1(C(CC(C)OC)=O)CCN(C(=O)C(=Cc2cccn2C)F)CC1C1CCCC1 N1(C(C2(C)CC2(Br)Br)=O)CC(n2cc(CNC=O)nn2)C(O)C1 Cc1cc(C(N2CCN(C3CN(C(=O)C4=COCCC4)C3)CC2)=O)cc(N)c1Cl CC1(C)CCOC(C(=O)NCC2(C)CCCC2NC(C2CCS2(=O)=O)=O)C1 C1(NC(c2cc3occc3s2)=O)CCN(C(=O)CCCC2CCC2)CC1F N1(C(c2ncc(CC)cn2)=O)CCCC2CN(C(=O)CC(C)C(C)(C)C)CCC12 C=Cc1ccc(C(=O)N(C2CN(C(C3(C)CCOC3)=O)CC23CC3)C)cc1 C1(NC(Cn2ncc(C#N)c2)=O)CCCC(NC(=O)C2=NOCC2)CC1 c1(N2CC(C)N(Cc3cccn3C)CC2)ncnc2c1CCC2 C1(C(=O)NC2CCN(C)C2=O)CC(F)(F)CN1C(=O)CCc1c(N)cnn1C C(=O)(C1=CCCC1C)N1CCCC(Cc2cc(N3CCC(OC)CC3)ncn2)C1 N1(C(CC(=C)Br)=O)CCCN(C(=O)CC(C)C(=O)c2cccc(CO)c2)CC1 C(=O)(C1CCCc2nncn21)N(CCC(C(C)C)NC(=O)C=CCF)C C12(C(=O)NCCC(C)(C)N(C)CC)CC(CN1C(C1CCCCN1CC)=O)C2 S(=O)(=O)(c1cc(C(N2CC3CC2CCC3O)=O)n(C)c1)NC(C)C C(=O)(C1SCCc2ccccc21)NCC1C(C)CCN(C(c2coc(Br)n2)=O)C1 C1(C(=O)NCCNC(C2C=CCC2)=O)(CC)CCCN1C(=O)CCOC C1(CNC(c2n(CC)cc(Cl)c2)=O)CCCC2CN(C(=O)C#CC(C)(C)O)CC12 C#Cc1ccc(C(=O)NC2CCCC(NC(C3CC34CC4)=O)C2)c(C)c1 c1(C(N2CCN(S(c3ncn(C)c3)(=O)=O)CC2)=O)ccc2c(c1Cl)OCCO2 C1(CN(C)C(c2ccccc2)=O)CCCCN1C(c1ccncc1F)=O CCC(C(=O)NCCN(C(=O)CC(O)C1CC1)C1CC1)C(C)(C)CC C12(CC(=O)NCC(C)(C)Cn3cc(CO)nn3)COC(CF)(C1)C2 c1(C(=O)NC2C(NC(=O)C3=NOCC3)C2)ccc2c(=O)c3ccccc3sc2c1 C1(C(=O)OCC)Cc2c(F)cc(OC)cc2N1.C123CCC1CN(C2)C3=O N1(CCN(C)C(C2COCCO2)=O)CCN(C(c2ccoc2C(F)(F)F)=O)CC1 c1(C(N(CCOC)Cc2ccccc2C)=O)coc2c1CNC2 c1(OC)cc(C=CC(=O)NC2CN(C(=O)C3CC3)CC23CC3)ccc1O C(CC(C(C)C)NC(C1CCCC1C(C)C)=O)NC(CC1CC(SC)C1)=O C1(CNC(C(CCC)(C)O)=O)CC2CCC(C1)N2C(C1CCCCC1O)=O Cc1cccc(CN(C(=O)C(C2CCOC2)NC(c2cc(C(C)C)on2)=O)C)n1 c1(OCC)ccc(NC(=O)C(=O)Nc2cnn(C)c2C)cc1F N1(C(C2(COCC)CCCC2)=O)CCC(O)(CCN2CCC(C(N)=O)C2)CC1 CCS(=O)(=O)c1cc(F)ccc1CNC(N1CCCC(c2nnc(S)n2C)C1)=O CCC(C)C(O)C(C)C(=O)NC1(C)CCN(CC(O)CC(C)(C)C)C1 C(C(C)(C)CCS(C)(=O)=O)NC(c1ccccc1)(C)C C(=O)(CS(=O)(=O)C(C)(C)C)NC(CCCCNC(C1C(OC)CCCC1)=O)C N1(C(C(C)(C)N(C)C)=O)CCCC12CCCOC2 C1(C(N(C(C)C(=O)NCC(C2CC2)N(C)C)C)=O)CCCCNC1=O N1(C(C(c2ccoc2)NC(CN(C2CC2)CC)=O)=O)CCC(C(F)F)C1 C(C(C)(C)C(=O)NCCC1CCCCN1C(=O)CC1(C#N)CC1)OC c1(C(N(C(=O)Nc2c(C)cco2)C)C2CC2)cccc(F)c1 C(=O)(C(=O)CC(C)CC)NCCN(c1cccc(Cl)c1)C(CN(CC#C)C)=O c1(C(=O)NC(C2CCOC2)CNC(c2cnc(CC)o2)=O)cnc(OC)c(F)c1 C1(C(N(CC(c2ccc(Br)cc2)O)C)=O)NC(=O)C2CCC12 CC1(C)CN(C(C2C3COCC23)=O)CCC1NC(=O)C=Cc1cncnc1O Nc1c(C(=O)NCC2CCCN2C(=O)Cc2ccsn2)cc(F)cc1[N+](=O)[O-] Cc1ccc(Cl)c(C(=O)NCC2COCC2NC(c2cc(C3CC3)nn2C)=O)c1 Nc1c(Cl)c(C(N2CCC(O)(CNC(=O)C(O)CF)C2)=O)nc(Cl)c1Cl N1(C(CN2CC(C)(OC)C2)=O)CCC(C(=O)NC2CC(C)(O)C2)CC1(C)C C1(C)(NC(C(c2ccc(C)cc2)F)=O)CCCN(C(=O)C=C2CCCC2)C1 c1(C(=O)NCCN(C(C2(C)CCCS2)=O)C2CC2)cccc(OCC(F)F)c1 N1(C(C2(C#N)CCCCCC2)=O)CCC(C2(NC(C3CCC4CC34)=O)CC2)CC1 C1(NC(C2C(C(C)C)C2)=O)CC2CCC1N2C(=O)Cc1cccc(F)c1 CC1(CC#N)CCCN(N2CC(Cc3ccc([N+](=O)[O-])cc3)C2)C1 CCC(CNC(=O)CC1CCCC2CC12)(CC)C(=O)N1CCC(C)(C2CC2)C1 Cc1cc(N)c(C(=O)NCCc2ocnc2CNC(=O)CCc2nccs2)cc1C C1(CNC(CC2(CC(=O)OC)CC2)=O)CN(C(C2CCC=CO2)=O)C(C)(C)C1 c1(C(=O)NC2CN(C(COC)=O)CC2SC)cc2n(n1)CCCCC2=O C1(C(=O)NC(C)Cc2ccncc2)CC=CCN1C(c1scnc1Cl)=O N1(C(C2(C)CCN2S(=O)(=O)CCCCl)=O)CCc2cc(Br)ccc2C1 c1(CNC(C(C2CC2)OCC)=O)cccc2c1CCN(C(c1sccc1F)=O)C2 C1(O)(C(C)NC(C(C)OCCCC)=O)CCN(C(=O)C(C)=C2CCC2)CC1 c1(CCN(C(C)C)CC2(C)CC2)cn(CCCO)nn1 N1(CC)C(=O)CCC1C(=O)NCC(C1CCCN1C(c1ccc(O)cn1)=O)(C)C N1(C(C(C)NC=O)=O)CCCC1CC(=O)N(C(C)(C)C)CC1CC(C#N)C1 c1(SC)cc(C(=O)N(CCCCNC(c2[nH]cnc2C#N)=O)C)oc1C C(=O)(C(C)CC(C)(C)C)NCCC1N(C(c2sc(C)c(O)n2)=O)CCCC1 c1(C(N2C(C)CC(NC(c3cccc(OC)c3)=O)C2)=O)cnccc1C#N CC1CCN(C(=O)CC2CCN(C(C3COC4CNCC4C3)=O)CC2)CCC1O C1(C)(OC)CC(NC(C2(NC(C3CC3(C)C)=O)CCC(C)(C)C2)=O)C1(C)C CCCCCCN(CC(=O)NC1(C2CCCN2C(=O)CSC2CCC2)CC1)C.C c1(OC)ccnc(F)c1C(=O)NCC1CC(NC(C2CC(C)OC2=O)=O)C1 C(CC(=O)NCC(=O)N(C(C)CF)C(C)C)NC(C)=O c1(C(C)C)ccc(C(=O)NC2(CNC(c3ccc(C#N)s3)=O)CCC2)c(O)n1 C(CC(CNC(c1snnc1C(C)C)=O)NC(=O)CCc1cscn1)OC CC1CCC2(CO1)CN(C(C1(CNC(=O)CC3CCCC3)CC=CC1)=O)C2 N1(C(c2ccc(C)nc2C)C(=O)NC(C(=O)OC)C)CCC2(CCN(C)C2=O)C1 c1(C(=O)NCC2C(NC(C(CC=C)OC)=O)C2)c(Cl)ccc(OC)c1N Cc1ccc(OCC(=O)NC(C)(C)CCNC(C2(CN(C)C)CC2)=O)cc1 N1(C(c2c(C)nns2)=O)CCc2sccc2C1CNC(C1CC12CC2)=O c1(C(=O)NCC2CCN(C(c3ccc(OC)s3)=O)C2)cc2c(Cl)cncc2s1 Cc1cc(C(=O)NC(CNC(=O)C=Cc2nc(C)cs2)C(C)C(C)C)c(C)cn1 c1(C(N2C3C(CNC(C(=O)N(C)C)=O)C(CCC3)C2)=O)cnc2ccnn2c1 C1(NC(C2CC(C(C)C)C2)=O)COCC1NC(c1cc(-c2ccccc2)[nH]n1)=O c1(C(N(C2CCCN(C(C(CC)(C)C)=O)CC2)C)=O)ccccc1S(C)=O C1(NC(CCC=CC)=O)CN(C(=O)CC(O)CCC)CCC1C Cc1ncc(Br)cc1C(=O)NCC1CC1NC(=O)Cc1ccc(C(F)F)o1 C(=O)(CC(C)CNC(=O)CCC1CCCCO1)NCCn1ncc(C)c1 c1(CC)nc(C)[nH]c1C(=O)NC(C)(C)CNC(=O)CN1CCS(=O)CC1 Cc1cncc(C(=O)NCC2CC2CNC(c2cn(CC(F)(F)F)nc2C)=O)c1 c1(C(=O)NC23CC(NC(C4(NC(C)=O)CC4)=O)(C2)C3)nnn2c1CCCC2 c1(C(=O)NCC(C)(C)OCC(=O)NCC2(F)CC=CCC2)cccc2occc12 CC(C(O)C(F)F)NC(=O)CCOC1CN(C(C2(C)COC(=O)N2)=O)C1 CCCC(CCCNC(c1cccc(CC)n1)=O)NC(c1cnc(C)c(N)c1)=O CC1(C(=O)NC2CCC2N2CCCC2)CCN(C(=O)C(CO)N(C)C)CC1 c12cccc(c1)OC2.c1(C(=O)NC2(CO)CN(C(COC)=O)C2)ccccc1C C1(F)(CNC(C(C=C)n2cccn2)=O)CCN(C(=O)COCC(=O)OC)C1 Nc1c(Cl)cc(C(=O)NCC2CCN2C(=O)CSC2CCCCO2)cc1Cl C(=O)(CC1NC(=O)c2ccccc21)N1CC(CNC(c2cc(F)c[nH]2)=O)C1 C1(F)(CNC(C(C2CCC2)OC)=O)CCCN(C(C2CCC(C)O2)=O)C1 c1(C(C)C(=O)N2CC(NC(C3C=CCCC3)=O)C2)ccccc1F c1(N2C(=O)CC(C(=O)NCCNC(C3(C)CC=CCC3)=O)C2)ccc(F)c(F)c1 Cc1[nH]c(C#N)cc1C(=O)NC1CCCC1CNC(=O)C(C)(C)c1ccnn1C CCC(C)C(C(=O)N(CC(O)CF)C)N(C)C(c1cnn(C)n1)=O C(C(CC(C)C)C(=O)N1CCOC(C(C)C)C1)NC(c1cccc(C)c1N)=O c1(C(=O)NC2CN(C(c3cc(C)nnc3)=O)CC23CC3)c(F)cc(Cl)cc1F CC1OCCC1C(=O)NCC1(NC(=O)COCC2CCCO2)CCC1 c1(C2(CC(=O)NCC3CCC3NC(=O)CCC=CBr)CC2)ccc(F)cc1 N1(C(C(=O)NCCC(=O)OCC)CC2CCOCC2)CC2(CC=CC2)C1 c1(OC(c2c(OC)c(C)ncn2)=O)c(Cl)cccc1[N+](=O)[O-] CCCCC(CNC(=O)C(C)O)NC(C1CCCC2CC12)=O c1(C(N2CCCC(C(C)NC(c3c[nH]c(=O)cn3)=O)C2)=O)cn(C)c(=O)n1C CC(CC(F)F)C(=O)NCC=CCNC(c1ccc(CSC(F)F)o1)=O C1(CN(CCCNC(COc2c(C)occc2=O)=O)C)CCc2nccn2C1 c1(CCC)cc(C(=O)NCCC(C)CCNC(=O)C(C)(C)c2cscn2)ccn1 Cn1nc2c(cc1=O)CC(C(=O)OCCn1cnnc1)CC2 C1(C(=O)NC(CCC)CO)(C(C)C)CCCN1C(=O)C(CC)NC(C)=O c1(OC)cc(=NC(=O)C2(CNC(c3cc(O)ncc3F)=O)CCCC2)[nH]n1C c1(C(=O)NCC(CNC(=O)C=CC2CCOCC2)O)c(Cl)ccc2ccoc12 c1(C(=O)NCC23CCC(CC2)N3C(C2(O)CC(F)(F)C2)=O)cccc(F)c1F N1(C(c2c(C)c(C3CC3)ncn2)=O)CCC(N=c2[nH]nco2)(c2ccccc2)C1 C(C(=O)N(C)CCN(C(C1(C(F)(F)F)CCCCO1)=O)CC)(C(C)C)SCC CC1(CNC(=O)C(C)(C)NC(c2cnncc2O)=O)CCOCC1 CC1(C)CCOC1C(=O)NC1CCCC1n1cc(CCC(N)=O)nn1 Cc1nn2cc(C(N3CCCC3C(C)NC(C3CCC(C)CC3)=O)=O)nc2s1 C(=O)(C(C)(C)CC1CC1)NC1CCC(CCC(=O)N(CC(=C)C)CC)C1 c1(C(=O)NC(C(=O)NCCCC(=O)N(CCC)CCC)C)ccc(C)c(Cl)c1 C1(C2CCC2)(C(=O)NCC2(O)CN(C(CSCC(C)C)=O)C2)CC1(F)F Cc1c[nH]nc1C(=O)NCCCCN(C(=O)C(C)(C)c1cc[nH]n1)C Cc1cc(C(=O)NCC2CC2NCCNC(c2cc(Cl)ccc2F)=O)cc(C)c1 C(=O)(CC(C)(C)C(F)F)NCC1N(C(C(C(C)C)n2ccc(C)c2)=O)CC1 C1(CCNC(c2cc[nH]c2)=O)CCCN(C(=O)C(c2ccc(Cl)cc2)O)C1 CCN=c1[nH]c(C(N2CCC(NC(=O)C=CC3CCOCC3)C2)=O)cs1 c1(C(=O)NC2CC(C)CN(C(c3c[nH]nc3C3CC3)=O)C2)cc2cnccc2[nH]1 c1(OCCC(=O)NCC(C)NC(c2cn(C)nn2)=O)ccc(F)cc1 c1(C(N(C2CCC(NC(=O)CCN3CCCC3=O)C2)C)=O)cnc2[nH]ccc2n1 c1(C(=O)NCC(CNC(c2cncc(C#C)c2)=O)C)cc2sccc2n1C CC1CN(C(C2C3CCCCC23)=O)CC1NC(c1cnc(O)s1)=O CC(C)CC(CNC(=O)CC1CCCOC1)C(=O)NC1(C)CCOCC1 c1(NC(c2ccccc2Cl)C)[nH]c(=NCC(C)CN2CCCC2)nc2sccc12 N1(CC(=O)NC2CC(NC(C3(S(C)(=O)=O)CC3)=O)CC2O)CCS(=O)(=O)CC1 c1(OC)ncc(C(N2CC=CC(NC(c3ccc(C(C)(C)C)s3)=O)C2)=O)cc1C CCS(=O)(=O)c1ccccc1C(=O)NC(C1CN(C(C2CC3(CSC3)C2)=O)C1)C c1(CCCN(C)C)nc(-c2cncc(-n3ccnn3)c2)n(-c2cccnc2)n1 C1(C2(NC(=O)C(CSC)NC(=O)C(O)CC(C)C)CC2)(OC)CCC1 N1(C(Cn2ccc(C)c2)=O)CCC(C)(C)C1C(=O)N(C)CC1COC(=O)N1 C1(NC(c2cc(C)ns2)=O)C=CCC(C(=O)NC(c2cncnc2)C)C1 C1(CCC(=O)NCCN=[N+]=[N-])CCN(C(C2(C(=O)O)CCCN2)=O)CC1 C1(N(C(c2c(Br)cnn2C)=O)CC)CCCN(C(=O)CS(C)(=O)=O)CC1 CC(C)CS(=O)(=O)NC(c1cc(CF)on1)=O Cc1cncc(-c2cn(CC3CCCN(C(C4CCC4)=O)C3)nn2)c1 C1(C(N2C(C(=O)OC)CC2)=O)CCN(C(c2ccoc2C2CC2)=O)C(C)C1 CC1C(NC(c2coc(C3CCCC3)n2)=O)CCN1C(c1ncccc1N)=O C(=O)(C#Cc1ccccc1)N1CC(NC(=O)CCc2cccnc2)C(F)(F)C1 C1(CCN(C(C(CC)O)=O)C)CCCCN1C(=O)C=Cc1cncn1C N1(C(c2ncc(Cl)cc2Br)C(=O)NCC2CCOC2)CCCC2(C=CCO2)C1 c1(CC(C)NC(Cc2ccc(CC)cc2)=O)ccc(F)cc1F C1(NC(c2c(OC)n[nH]c2)=O)C=CCN(C(=O)Cc2csnc2C)C1 CC1(C)CCc2onc(C(=O)NCC(C)(C)NC(=O)C(F)CC3CC3)c2C1 c1(C(N2CC(OCCNC(C(CC)C#N)=O)C2)=O)c[nH]c2nccc(Br)c12 c1(C(=O)NCC2(CNC(=O)CO)CCCC2)ccc(Br)c(F)c1 C1(CN(C(c2cc(CC)on2)=O)C)C2CN(C(=O)CC3COC(=O)N3)CC12 S(=O)(=O)(c1csc(C(N(CCC)Cc2ccc(F)cc2)=O)n1)NC C(=O)(C1CCCc2ccccc21)N(CCCNC(c1ccc(F)cc1N)=O)C N1(C(C(CCC)NCc2cnc3n2CCOC3)=O)CCC2(CC1)CCS2(=O)=O C1(NC(C2C=CCC2)=O)CC2(CCN(C(c3ccc(CC4CC4)s3)=O)CC2)C1 c1(-c2onc(-c3cccc(CC4C5CCC(F)(F)C54)c3)n2)cnc2cc[nH]c2c1 N1(C(c2ccncc2O)=O)CC(C2CN(C(C3CC3C3CCC3)=O)C2)C1 N1(C(C2C(C)CCC2)=O)CCC(C)(NC(=O)COCCO)C1 N1(C(c2cc(Cl)ccn2)=O)CC2(C1)CN(C(C13CCC(F)(CC1)CC3)=O)CCO2 N1(C(CCc2ccc(C)nc2)=O)CC2CCC2(CC(=O)NCCCCN(C)C)C1 c1(C2C(C(=O)NCc3cc(CNC(C4C=C(C)CS4)=O)no3)C2)cccc(Cl)c1 c1(N(CC(OC)OC)CCCO)nnn2c1N(C)CC2 c1(C(=O)NC(CNC(c2n(CC=C)ccn2)=O)C)ccc2c(c1)COCCN2 Cn1cnc(C=C(F)C(N2CC(C(=O)NC3CC4CCC3O4)(N(C)C)C2)=O)c1 CC(C)CCC(=O)N1CCC(CN(C)C(c2ccnc(N(C)C)c2)=O)C1 CCC(C)(F)C(=O)N1CCC(F)(CNC(=O)Cn2nnnc2C(C)C)C1 c1(C(=O)NCC2C(NC(c3cc(NC)no3)=O)CCC2)nnn(C)c1C(F)F C1(NC(c2ccc(OC)nc2)=O)C(C)CN(C(=O)CN2CCS(=O)CC2)CC1C c1(C(N2CC(NC(C(C)OCCC#C)=O)C2)=O)cnn(CC2CCCC2)c1 CC1CCN(C(c2csc(Cl)c2)=O)CC1NC(C1(C(F)F)CCCC1)=O c1(C(=O)NC2CC3(C(C(=O)NCCC4CC(C)C4)C3)C2)cc(C#N)cn1C C1(CNC(CCOC)=O)COC(CNC(c2cn(CCC(C)(C)C)nn2)=O)C1 CCCCC(CC)(c1nnnn1CC1CCOC1)NC(C)COCC c1(CNC(c2n(CCSC)nnn2)C2CCSCC2)nnc2n1CCNC2=O C1(CNC(C(CC)CC)=O)CCN(C(=O)CSc2ccc(O)cc2)C12CC2 C(C(N=c1nc(C2CC2)[nH]s1)C1CCCCC1)NC(c1ccn2ncnc2c1)=O c1(CN(CCNC(=O)NC2CCCN2C)CC)ccccc1C C1(C)(C(=O)NCCC2CC(NC(C3N(CC)CC3)=O)C2)CCN(C)C1 Cc1c(Br)noc1C(=O)NCCCC1CCCN1C(=O)C=C1CCC1 CC12CCC(C(N3CC4CN(C(=O)CCc5nc[nH]n5)CCC34)=O)(CC1)CO2 c1(C(N2CCN(c3nc(OC(C)C)c(Br)cn3)CC2)=O)cnn2cc(F)cc(F)c12 c1(C(N2CC(NC(CCC3CC(OC)C3)=O)C(O)C2)=O)sc(Cl)c(Cl)c1C O=C1COCCN1C1(C(=O)NC2CCCCC2n2cccn2)CC1 C(c1c(Cl)nc2sccn12)=CC(N1CCC(C(C)NC(=O)COCC(F)F)C1)=O c1(CCC(=O)OCc2c(OCC#C)cccc2F)cnc2n1CCCC2 C(=O)(C#CC1(CCc2cn(-c3ccc(O)cc3)nn2)CC1)NCC1(C)CCCO1 C1(C(=O)NCCCN2CCN(CC)CC2)CN(C(c2ccncc2)=O)CCN1C c1(C(=O)NC(CCNC(C2C(=C)C2)=O)C)ccnc(OC)c1 N1(C(CCc2cccc(OC)c2)=O)CCCC2CN(C(=O)CC=C(Cl)Cl)CCC12 C12(CNC(CC=C)=O)CC(NC(C3CCC3C)=O)(CO1)C2 O=C(C1=NOC2(CCN(Cc3cc(O)ccc3Br)C2)C1)NCc1ccc(F)nc1 c1(C(=O)NCC2CN(C(C(C=CC)O)=O)CC2O)cnc2c(c1)OCC(=O)N2 CC1(CNC(=O)COC(F)F)CCN(C(=O)Cc2cccc(OC(F)F)c2)C1 c1(CNC(C2CC(=C)CN2c2cc(Br)cnc2C(N)=O)=O)cnc2cc[nH]c2c1 CC1CN(C(=O)CC2CC2)C(C)CN1CC1CC=CCC1 N1(C=O)CC2CC1(C)CO2.N1(CCOC)CC(OC)CC1=O.C(C)(C)(C)OC(C)=O C12(COCC)C3CCC(CC13)C2(F)F.C123CCC(CC1)(CO2)CNC3=O Cc1cc(-c2cn(CC3CCN(C4CCC4C(=O)O)CC3)nn2)ccn1 C#CCCC(C(=O)N1CC(F)(F)C1)NC(c1cccc(F)c1N)=O c1(-n2cc(C3CCCN(C(C4C(CC)CC4)=O)C3)nn2)ccccc1C(F)(F)F C(=O)(C1Cc2ccccc21)N1CCC(C(=O)NCc2nn(C)c(=O)o2)C12CCC2 C1(C(=O)NC(CNC(c2cc(C)ncn2)=O)CC(F)(F)F)CCc2nccn2C1 Cc1c(C(=O)NC2(C(C)NC(=O)Cc3cnn(C(C)C)c3)CC2)nnn1C(C)C Cc1cc(CNC(C2CC2CNC(=O)C=Cc2ccccc2)=O)ccc1F C(=O)(C(F)C(=O)NCC1(CC(=O)NCCC2(C)CC2)CC1)OCC Cc1cc(OCCC(=O)NCC2COCC2NC(c2cc[nH]c2)=O)c(C)c(C)c1 c1(OC)cc(C(N2CCCN(Cc3ccccc3F)CC2)=O)cc(Br)c1O C1(CC(=O)Nc2cc(C(C)(C)C)[nH]n2)CC(N=c2ccn3nccc3[nH]2)C1 C1(CC)CN(C(C2CCC(C#N)C2)=O)CC1NC(=O)CCOCCOC Cc1cc2cccc(C(N3CCOCC3CC3CCC3)=O)c2o1 c1(N2CC3C(N(C)C)C3C2)ncnc(NC(=O)C2=CC3CCCC23)c1[N+](=O)[O-] C(=O)(C1=CC2C=CC1C2)N1CCC(CC(N2CCC(C(C)O)C2)=O)C1(C)C c1(C(N2CCCC2CN(C(C23CCCN(CC2)C3)=O)CC)=O)nccc2ccsc12 C1(CNC(C2CC(=C)C2)=O)C(C)CCN1C(c1c(OC)nsc1OC)=O C1(NC(CNS(C)(=O)=O)=O)CC(=O)N(C2CCCCCC2)C1 N1(C(CC2CN(C(c3c(C)n[nH]c3)=O)CC2C)=O)CCCCCC1C C1(NC(c2cnc(CC)s2)=O)CCCC(NC(=O)C(C)(C)c2ccnn2C)C1 N1(C(c2ccc(C(C)=O)o2)=O)CCOCC1C(=O)Nc1ccsc1C(C)C C#CC(CC(C)(C)C)NC(C1CC2CC2N1C(C12CCC(C1)C2(C)C)=O)=O C=C(CNC(N1CCN(CCn2cncn2)CC1)=O)c1ccccc1 N1(C(C(COC)(C)C)=O)CCC(C)C(NC(=O)CN2CCOCC2=O)C1 C1(CNC(C(CC)C2CCOC2)=O)CC(F)(F)CN1C(c1cc(F)ccc1Cl)=O c1(CN(C)C(c2coc(-c3ccccc3F)n2)=O)nnc2n1CCNC2 c1(OC)ccc(C(=O)NCCC2CCN(C(=O)C(C)OCCN(C)C)C2)c(Cl)c1 c1(C(N2CC(C(=O)Nc3c(C(C)=O)cnn3C)C2)=O)ccc2c(c1)OCCN2C c1(COCC(=O)NCC(n2cc(Cn3nccn3)nn2)C)ncnn1C c1(NC(c2ccc(NCC(C)C)nc2)C)ccccc1CCO CCC(C)CC(C(=O)NC(CO)C1CC1)NC(C1CC(=O)N(CC)C1)=O c1(C2C(C(=O)NCC(CC)NC(=O)CC(C)C(=O)OC)C2)c(Cl)cccc1Cl c1(C(c2nnnn2CCSC)NCC(C)CCO)ncnc2c1OCCO2 C1(NC(c2c(CC)cncc2)=O)C2CCC1N(C(=O)C(C)CC)C2 c1(CC)ccc(S(=O)(=O)N2CCCC(C(N3CCOC(C)C3)=O)C2)s1 c1(CNC(C2OCCN(C(C3(C)CNC(=O)C3)=O)C2)=O)ccc(F)cc1Cl c1(C(N(CC(CN(C(C(C2CC2)OC)=O)C)O)C)=O)c(C)cc(Cl)cc1N c1(C(N2CCCC(NC(c3cnc(C)s3)=O)C2)=O)cnn2c1OCCCC2 c1(C(c2n(CC=C)nnn2)NCCc2cccc(F)c2C)ccc(O)c(F)c1F C1(CNC(C2C(OCC)CC2)=O)(NC(C2CN(C3CCOC3)C2)=O)CCCCC1 N1(C(C2CCC(NCc3ccc(O)c(O)c3O)CC2)=O)CCC2(CCOC2)CC1 C1(CNC(C(=O)NCCn2c(C)nc(C)n2)=O)OCCOC1(C)C N1(C(C2CCCS2(=O)=O)=O)CCN(C(c2ccc(O)nc2)=O)C2CCCC12 CN1CCCCC1C(c1cn(CC(=O)NOC(C)(C)C(=O)O)nn1)NC(C)(C)C c1(CC)ccc(C#N)cc1F.c12cccc(c1)CNC(=O)C1CC(O)CN1C2=O Cn1ncc2c(C(N3CC(NC(c4ccc[nH]4)=O)C(CO)C3)=O)cccc12 C1(NC(c2c(C)nc[nH]2)=O)CC2C(NC(C3CCC3C)=O)C2C1 CCN=c1ccc(C(=O)NC2CC2NC(c2ccsc2)=O)c[nH]1 C1(C(N2C(CC#C)CCC2)=O)(CNC(c2ccc(CC#N)cc2)=O)CC(F)(F)C1 CC1CC2=C(C(=O)N1)C(c1c(Cl)cccc1Br)NC(=S)N2CCC1CC1 c1(C(N2C(CNC(=O)CNC(C3CCC3)=O)C=CC2)=O)csc2c1CCCC2 N1(S(Cc2cccc(C)c2F)(=O)=O)CCOC2(CCS(=O)(=O)C2)C1 N1(C(CC2C(C)(C)C(=O)C2)=O)CC(C(=O)NCC(N2CCOCC2)=O)C(F)(F)C1 c1(C(=O)CN(C2(CNC(c3ncn(CN(C)C)n3)=O)CC2)C)cc2sccc2[nH]1 CC(CF)CC(=O)NC1CCCCC1NC(C1(Oc2ccccc2F)CC1)=O CC1CCS(=O)(=O)CCN1C(c1ccn(C(F)F)n1)C(=O)NC1CCC1 C12(C(=O)NCC#CCNC(Cc3cccc(OC(C)C)c3)=O)CCC(C)(C1)OC2 c1(C(=O)OC)ccc(N(C2CN(C(=O)C(O)CSc3ccccc3)C2)C)cc1 CCC(CC)CC(=O)NC1CCCCC1C(=O)NCCN1CCCC(O)C1 N1(C(C(COC)OC)=O)CCC(NC(=O)Cc2cccc(F)c2Cl)C1CCO c1(C(N2C3(CNC(CN(C(C)C)C)=O)CCC2CC3)=O)cccc2c1CCOC2 Cc1nc(NC(=O)NCC2CCC(=O)NC2)sc1F C1(CNC(CCC)=O)C2CCCC1N(C(=O)C(c1cc(C)cc(F)c1)C)C2 CC1(O)CCN(CC(=O)NC2(CCNC(C3CC(CF)C3)=O)CCC2)C1 CC1CC(C(N2CCC(CCCNC(=O)C#CC(=O)N(C)C)CC2)=O)CC(C)O1 c1(C(=O)OC(c2cccn2C)C)cc2c(cnn2C)nc1O C12CN(CCO1)C2=O.c1(COCC(=O)NC2C(CN(C(C)=O)C)C2)cccnc1 N1(C(C=CC)=O)C(CNC(c2ncccc2OCC)=O)CC2CCCC12 CC1(C)CCCC(CC(N2CC(O)(CNC(=O)CC34CNC(=O)C(C3)C4)C2)=O)C1 c1(C(N2CC(CNC(C(C=CC)O)=O)C2)=O)cc(F)ccc1C N1(C(CCc2cc(C)[nH]n2)=O)CC2(C=C(C(=O)N3CCOCC(C)C3)CO2)C1 N1(C(C2(Cl)C(C)(C)C2)=O)CCCC(CCNC(=O)CCCC2CC2)CC1 c1(C(N(CCN(C(c2cc(CC)c(C)cc2)=O)C)C)=O)nccn2cnnc12 c1(Cc2[nH]nc(C(=O)Nc3ccc(Cl)cn3)n2)c(F)cccc1F c1(OC)ccnc(C(N2CCC(O)(CN(C)C(c3nc(C)nn3C)=O)C2)=O)c1O CCCCC(C(=O)NCC(=O)OCC)NC(C1CCN(CCC)C1=O)=O C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(c2c(C)cnnc2)=O)C(C)(C)C1 C(c1ccccc1[N+](=O)[O-])=CC(=O)NCC1OCCN(C(C(COC)OC)=O)C1 C(=O)(C(C#N)C(C)(C)C)NC(CN(C)C(c1ccc(-c2ccco2)[nH]1)=O)(C)C C1(C)(C(=O)OCC(c2c(C)noc2)=O)CCC(Cc2ccccc2Cl)CC1 Cc1nnccc1C(=O)NC(C)CCN(C)C(C1CCC(CN(C)C)O1)=O C(=O)(C(C)C(O)C(C)C)NCCn1ccc(C(NOCCOC)=O)c1 C(=O)(CC(C)CC(C)C)NCc1nc(C(N(CC=C)CCC)=O)sc1 c1(-c2scc(C(N3CC(O)(C(C(=O)OCC)F)C3)=O)n2)ccc(Cl)cc1 c1(OC)ccc2c(n1)NC(C(=O)NC(C)CN(C(=O)C=Cc1cnn(C)c1)C)C2 Cc1nc(NCC(=O)Nc2ccc(F)cc2F)cc(=NCCOC2CCCC2)[nH]1 C1CN(N2C3CN(C)C(C3)C2)CCC1(F)F.c1(C)cc(O)cc(O)c1 c1(OC)c(Cl)ccc(Cl)c1CC(=O)Nc1ccsc1OC N1(CC(=O)NC2CCC(N(C)C(C3CCNC3=O)=O)CC2)CCCNS1(=O)=O Cc1ccc(NC(C2OCCC2CNC(c2ccc(F)cn2)=O)=O)c(C)c1O C1(NC(c2scc(C)c2)=O)CC12CC(NC(=O)CC1C=NN(C)C1=O)C2 C(=O)(C1=CC2CCCC12)NCC(C)(C)CNC(c1ccc(N)cc1O)=O c1(NC(C=C(C)CNC(=O)C=CCN2CCC2)=O)ccc(O)nc1 c1(C(N2CCC(NC(C3CC34CCSCC4)=O)C2)=O)cc2c(cn1)CCCC2 N1(C(c2c(CC)cccc2)=O)CCCC2(NC(c3cnsc3)=O)CCCC12 N1(C(C2(CC)CN(C(=O)CC3CCCOC3)C2)=O)CC2CC2C2CC12 C#CC1CN(C(=O)C(C)=C2CCC2)CCN1C(=O)C(C)OC N1(C(C(C)SC)=O)CCCC2(CCCCC2NC(c2cn(C3CCC3)nn2)=O)C1 N1(CC(CC)C)CC(CNC(=O)CC2CCCOC2)CC1=O C1(NC(c2c(OCCC)cccc2)=O)CCCC2CN(C(C3CC3OC)=O)CC12 N1(C(c2c(OCC)ccc(Br)c2)=O)CC2C(N(C)C)CS(=O)(=O)C2C1 C1(C(=O)NCCN2CCCC2)C2CC2CN1C(c1csc(O)n1)=O c1(C(CCC)C)nc(-c2cc(C(C)C)nn2CCOC)n(CC(N)=O)n1 Cc1ccc(CN2CCCC(C(N3CC4CCCC4C3)=O)CC2)c([N+](=O)[O-])c1 CC1CCn2cc(C(=O)NCC34CC(NC(c5nc(COC)cc(N)n5)=O)(C3)C4)nc2C1 Cc1nn(C(C)C)c(C)c1C(=O)N(C)CCNC(=O)C(C)CS(C)=O C1(NC(CC(=C=C)C)=O)CC2CC(NC(=O)Cn3cc(C4CC4)nn3)CC12 c1(C(N2CCC(C)(CCNC(CC(CC)C)=O)C2)=O)nc(C)c(C)[nH]c1=O N1(C(c2cnc(NC(C)=O)o2)=O)CC2(C1)CN(C(=O)C(C#N)C(C)(C)C)CCO2 C(=O)(C1CCN(C(N)=O)c2ccccc21)OCCC1CCC(C)(C)CC1 C1(C2CCCCN2C(C2CCC2)=O)(CNC(=O)CCc2nccs2)CCOCC1 c1(C(C)=O)cc(C(N2CCC(CO)(NC(C3CC34CC4)=O)CC2)=O)c(C)nc1C C1(C(=O)NC(CCCC)C)N(C(=O)CN(CCCCCC)C)CCC1(C)C C12(NC(c3cccc(CO)c3)=O)CC(C1)N(C(=O)Cc1cncc(O)c1)C2 c1(COC)cc(C(=O)NC2CCC(NC(=O)C(c3cscc3Br)=O)C2)on1 C(C(C)S(C)(=O)=O)(c1ccc(C)cc1)N1CCC(CO)(NC(=O)OC(C)(C)C)C1 c1(CN2CC3(CCC(CNS(C(COC)(C)C)(=O)=O)O3)C2)cccc(B(O)O)c1 c1(OCCC)cccnc1C(=O)NCC1CCN1C(c1ccn(C)c1)=O Cc1ccnc(O)c1C(=O)NC(CNC(=O)C(C(C)C)n1cnnc1)C1CC1 C1(CCC(=O)NCCN(C(=O)C(CO)N(C)C)CCOC)CC(F)(F)C1 C1(NC(COCCC#C)=O)CN(C(c2cc(C)c(CC)nc2O)=O)CC1N=[N+]=[N-] c1(CC(=O)NC(C)CN(C(=O)Cc2cnco2)C)ccc(C2CC2)cc1 C#CC(C)(C)C(=O)NC1CCCCC1CNC(C1CN(C2COC2)C1)=O N1(C(CC(=O)OC)=O)CCOCC2(C1)CN(C(=O)COC1CCCC1)CCCO2 C(CC(CC)C(=O)NCC1(CNC(c2cnc(Cl)s2)=O)CC12CCC2)=CCCC C1(C(=O)NC2C=C(C)CS2)CC2CCC1CN2C(C1CCCN(C(N)=O)C1)=O C123CCCC1N(CCC2)C(=O)CCOCC(=O)NC3.C(C(C)(C)C)OC(C)C C(N=c1nc2c(cnn2C)c(N2CCN3C(=O)NCCC3C2)[nH]1)C1CC(OC)C1 Cc1ccc(C(N2C3CCC2CN(C(C2CCN(C)C2C)=O)C3)=O)c(N)c1Cl C(=O)(C1CN(C(=O)OC(C)(C)C)Cc2n[nH]cc21)OC=Cc1cc(Cl)cc(Br)c1 c1(N(CCCCN(C)C(c2cc([N+](=O)[O-])n[nH]2)=O)C)cc2c(s1)CCC2=O C1(CC(=O)NCC(C#C)C(C)C)C2CCCC2N1C(C1CC(=O)CC(=O)C1)=O CC(c1cnn(C)c1)=CC(N1CCN(C(C2CSCCS2)=O)C(C2CCC2)C1)=O c1(C(C(=O)NC(CNC(Cc2cnc(C)s2)=O)CC(C)C)O)ccc(Cl)c(F)c1 c1(C(=O)NCCCN(C(C2CC(C)=C(C)CC2)=O)C)ccc2n[nH]cc2n1 c1(NC(C)=O)cccc(F)c1C(N1CC(O)(CN(C)C(C2CCSC2)=O)C1)=O C1(NC(c2c(C)nco2)=O)CC2CC(NC(=O)CC3CC(=O)NC3=O)C1C2 N1(C(c2snc(O)c2Cl)=O)CCC2CCN(C(c3cc4ccccc4o3)=O)C2C1 N1(C(C2CN(Cc3ccc(COC)o3)CC(F)(F)C2)=O)CCN2CCOCC2C1 N1(C(c2c(C)ncnc2)=O)CCC(CNC(c2ccncc2)=O)C(C)C1 c1(N(C)C)ccc(C(=O)NC2CCCC2NC(c2c(C)nn(C)c2Cl)=O)c(F)c1 c1(OC)ccnc(F)c1C(=O)NCC1(F)CCN(C(=O)CCC(C)(C)C)C1 c1(C(=O)NCC(C)N(C(=O)COCCSC(C)C)CC)cc(Cl)c2cn[nH]c2c1 C1(C)(CNC(CC(CC)SC)=O)CN(C(=O)CCC2(C)CC2(F)F)CC1C Cc1ccc(Cl)c(NC(=O)C(C)NC(=O)CN2CCC(C(=O)O)CC2)c1 N1(C(C2CC(C#C)(O)C2)=O)C(C(=O)NC2COCC2O)CCC12CC2 C12(NCCn3ccc(C(N4CCC(C(C)(C)O)C4)=O)n3)CC=CC(C1)OC2 CCC(O)C(C)(C)C(=O)NC1CN(C(=O)Cc2ccnc(F)c2F)CC1SC C(C1CN(C(C2C(C)C2C)=O)CC1C(N1CC(=O)NCC1C(C)C)=O)=CC N1(C(c2c(CNC(=O)C=Cc3cc[nH]n3)n[nH]c2)=O)CC2(CNC(=O)N2)C1 N1(C(C(C)CCN2CCOCC2)=O)CC(c2ccccc2)CCC1C c1(C(C)NCC(C(=O)OC)Cc2ccccc2)ccc(Cl)c(Cl)c1C c1(NC(N(C)C)=O)cc(NC(=O)Nc2ccc(-c3ncn(C)n3)cc2)cc(Br)c1 CC1(CNC(=O)C(F)=C2CCC2)CCCN(C(=O)C(c2cccc(F)c2)O)C1 C1(CNC(c2cc(OC)n[nH]2)=O)CCCC2CN(C(=O)Cc3cc[nH]n3)CC12 C1(O)(CN(C(=O)C(c2ccco2)NC(=O)CCC2CC2(C)C)CC)CCC1 c1(C(N2CCCC(CC(=O)Nc3ccc(C4CC4)nc3)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CS(=O)(=O)CCC(=O)N1CC2CC(NC(=O)C(=O)NC3CC3)CC(C2)C1 c1(C(=O)NCC(C)N(C(C(C)NC(CC)(C)C)=O)C)cc2ccccc2c(O)n1 c1(NC(C(=O)Nc2c(C3(C)OCCO3)cccc2)=O)cccc2c1OCCC2=O C1(N(C(C(C=C)C)=O)CC=CCCCCC)CCN(C(=O)COCCCC)CC1 N12CCCC(C1)C(C)C(=O)NC1(CCC1)C2=O.C(C(C)(C)C1CCC1)SCC c1(N(C)CC2(OC)CCC2)nnc(C(C)C)n1CC(C)C(C)C CCC(C(=O)NC1CCCCC1NC(=O)Cn1ccnn1)C(C)O c1(C(N(C(C(N2CCC(C(CC)CC)C2)=O)CC)CC)=O)ncccc1O C1(NC(c2c(C)ncn2O)=O)CCOC2(CCC2)C1 C1(CNC(C2(C#N)C(C)C2)=O)(CNC(=O)Cc2c(Cl)cnn2C)CCCCC1 C1(NC(c2cnc(C)s2)=O)CC2CCC(C1)N2C(=O)CCCc1cccc(F)c1 N1(C(c2nc(CC)oc2C)=O)CCCCC(NC(c2csc3nnsc23)=O)C1 c1(C(N2CC(CC(C(=O)NCC(C(=O)OCC)C)F)C2)=O)cc(C)c(C)o1 N1(C(C2CC3(C(OC)CC3)C2)=O)CC2CCN(C(c3[nH]c(=N)sc3C)=O)CC2C1 N1(C(Cc2c(C)ocn2)=O)CCCC(F)(CNC(=O)CCN2CCCC2=O)C1 C1(NC(Cc2c(C)scc2)=O)CN(C(=O)CC2CCN(C)C2)C2(CCC2)C1 N1(C(C2C3CN(C(C(CC)COC)=O)C2C3)=O)CC2CN(C)CC2C1 C1(NC(C=C(COC)C)=O)CCN(C(=O)CN2CC(=O)N(C)C2=O)C12CC2 C1(C(N2CCC(CS(=O)(=O)Nc3scc(C)n3)CC2)=O)CCc2nc(C)cn2C1 c1(C(C)=O)ncc(C(=O)NCCC(O)CNC(=O)C(C)CC2CCC2)s1 N1(C(CC(C)C)=O)CCC2CN(C(=O)CCCc3ccc([N+](=O)[O-])cc3)CC2C1 C12CCCC(CC1)C(=O)N2.CC1CCC(C(=O)NNC[Si](C)(C)C)CC1 C#CCCCCC(=O)NCC12CC(CN1C(c1ccc(N)c(O)c1)=O)C2 C=CC1CCN(C(=O)CC2(C=C)CN(C(=O)CC3CCCC3C)C2)CC1 C(=O)(CC(F)(F)C(C)C)NCCN(CCC)C(C1CCOCC12CCC2)=O C(CCCC(=O)N1CCCC1C(C)NC(c1cnn(C)c1C(C)C)=O)SC c1(CC)cc(NC(C2CCN2C(=O)Cc2ccc(O)cn2)=O)cc(C)c1 c1(CC(=O)NCC2C(NC(Cc3nc(C)sc3)=O)C2)cccc(C(C)C)c1 n1(CC(=O)NCC2COCCN2Cc2ccsc2Br)ccc2c(F)cccc12 C1(C(=O)NC(C2CCCN2C(=O)CC(=O)NC2CC2)C)CC(C)(C)SC(C)(C)C1 C1(C(=O)NC(C)(C)CC2CCCC2)C(C2CC2)CCN1C(C1CS(=O)(=O)C1)=O C(=O)(C1CCc2cccc(O)c21)NCCN(C(c1ccc(C(C)C)s1)=O)CC C1(CNC(c2nc(CCC)oc2)=O)(NC(=O)Cc2cncnc2O)CCCOC1 c1(C(C(=O)NC2CN(C(CCCN(C(C)=O)C)=O)C(C)C2)C)ccc(C#N)cc1 c1(N2CC(CC(C)NC(C3CCCN(C(C)=O)C3)=O)C2)ncc(C)c(C)n1 C12(C(=O)OC)CC1CN(C(C1CN(C(c3cncc(OC)n3)=O)CCO1)=O)C2 CCCC(CC)C(=O)NC12COC(C1)C(NC(=O)COCc1nccn1C)C2 c1(C(=O)NC2C=CC(CNC(Cc3nc(CC)sc3)=O)C2)ccc(C#N)[nH]1 C(C(=O)NCC1CCC(NC(=O)C(C)Cc2cccnc2)CC1)(C(C)C)SC c1(NC(C(CC#C)(C)NC(=O)C(C)OCC2CC2)=O)cc(C)cn(C)c1=O N1(C(C2(C)CCC(=O)NC2)=O)CCN(C(c2ccc(N)c(Cl)c2O)=O)C2CCC12 CON1CC(C(=O)NCC(C)(C)OCCNC(=O)C(C)(C)C(=O)OC)CC1=O N1(C(=O)CCc2cncnc2)CCN(C(C2C3CCCOC23)=O)C2CCCC12 c1(C(=O)NCC2C(NC(C3N(C(C)C)C(=O)CC3)=O)C2)cc(=O)c(Br)c[nH]1 C1(C)(CC)CC(NC(=O)CC=CCNC(C2CCCN2C)=O)C1 N1(C(C(c2ccccn2)C)=O)CCC(C)(CNC(C2CN(CC(F)(F)F)C2)=O)C1 C(CS(=O)c1ccccc1)NC(N1CC2CC=CCC2C1)=O C=C(C)CCC(=O)NCC1(CNC(c2csc(CCCCC)n2)=O)CCC1 C1(N(C(=O)CCC2CC2(C)C)C)C2CN(C(c3csnc3Br)=O)CC12 N1(C(c2nc(C)nn2C)=O)CCC2CCCC(C1)N2C(c1c(C)cncc1C)=O c1(-n2ncc(C(=O)NC(CNC(Cc3c(C)n[nH]c3)=O)C)c2)ncc(Cl)cn1 C(=O)(CC(C)(O)CC(=O)O)N1CCOCC(NC(c2c(F)ccc(C)c2Cl)=O)C1 C(=O)(C(O)CC(F)(F)F)NC1C(CC)CN(C(=O)C(COC)OC)CC1 C1(NC(C(C(C)C)NC(C)=O)=O)CC2CC1CC2C(=O)NC1CCOCC1F c1(C(=O)NC(CC=C)CNC(C2(NC(C)=O)C=CCC2)=O)c(C)nn(C)c1Cl C1(C(=O)NC(C)CSCCOC)(CC)CN(C(=O)Cc2ccccc2)C1 C1(N(C(c2cc(CCNC(CCOCC(C)C)=O)on2)=O)C)CCC(=O)N(C)C1 CC(O)C(C(=O)NCC1(F)CC(NC(c2cc[nH]c2)=O)C1)NC(=O)C(F)(F)F Cc1[nH]nc2ccc(C(N3CC4(NC(c5c[nH]ccc5=N)=O)CCC3C4)=O)cc12 C(=O)(CC(C)C(F)F)NCCC1(NC(c2occ(C)c2)=O)CCCC1 c1(C(C(=O)NC(C)C(C)NC(C2(n3cncn3)CC2)=O)C)ccc(F)cn1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(CNC(C2(OC)CC2)=O)C(C)C1 c1(C(N(C2CC(NC(C3CC(C4CC4)C3)=O)C2)C)=O)ccn(CCO)c(=O)c1 C1(C(=O)NC2C(C(N)=O)CCC2)CCCN(C(=O)CC2CCOC2)CC1 c1(C(=O)NC2CCCC23CN(C(C2CC=CCC2)=O)C3)ccc2c(c1)CCOC2 C1(CC=C)(NC(=O)Cc2ncoc2C)CCN(C(C2(n3cccn3)CCC2)=O)C1 C(=O)(C(F)C(C)C(F)(F)F)Nc1c(C)nc(Cl)cc1I c1(C(=O)NC(C(C(C)C)C)CNC(c2cnns2)=O)cccc2c1CCN2 C1(C(N(C)CC2CCCN2C(=O)CCC2CC2(Cl)Cl)=O)CCCN1N=O N1(C(c2ccc(CC)o2)=O)CC(N=c2[nH]nc(C(F)F)s2)C2(CCC2)C1 c1(C(=O)NC2C(NC(C(c3cccc(OC)c3)O)=O)C2)cccc2ncsc12 Cc1ccc(C2(C(N3CCC(CF)(NC(C4C(C)C4(F)F)=O)C3)=O)CCC2)cc1 N1(C(CCN(C)CC)=O)CC(CNC(c2ccc(CNC(N)=O)cc2)=O)C2CC12 CCCC(COc1c[nH]nc1NC(C)=O)C(=O)N(CCO)CCOC Cc1nc(C2CCCO2)ccc1C(N1CCCC(C(F)F)C1)=O N1(C(C(C)(CO)OC)=O)CC2CCC(C1)N2C(c1cccnc1OCCO)=O N1(C(c2ncc(OC)cn2)=O)CCCCC(NC(=O)C=C(F)c2ccccc2)C1 C1(NC(C2CC(O)(CC#C)C2)=O)CCCC1(C)CNC(=O)C(C)(C1CC1)OC C(=O)(C(C(C1CC1)C1CC1)N(C)CCc1nc(C)cs1)NCCC c1(OCC=C)ccccc1C(=O)NCC1CC(C)N(C(C2C3CC4C(C3)C24)=O)C1 S(=O)(=O)(c1cnc(NCC2(C3CC3)CC2)c(Cl)c1)NC(c1ccn(C)n1)CC N1(C(c2c(C(C)O)cccc2)=O)CC2CCC2(CNC(C2(C(F)F)CC2)=O)C1 c1(C(N2CC(C(c3ccccc3)=O)C(CO)C2)=O)cc(F)ccc1-c1nn[nH]n1 N1(C(c2oc(CC)c(C)c2)=O)CCCC(C)(C)C1C(=O)NC(CC)C(C)(C)O c1(C(N(CCCn2cc(CSC)nn2)C2CC2)=O)c(C)cnc2ccccc12 c1(OC)cc(CN2CCNCC(C(=O)O)C2)ccc1C#N c1(SC)cncc(C(=O)N(CCCNC(=O)CSc2nncs2)C)c1 Cc1ccc2ncnc(N3C4CCC(C4)C3C(N3CCCCC(C)(F)C3)=O)c2c1 c1(C(=O)NC23CC(CNC(C(C(CC)C)C)=O)(C2)C3)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NCCC(C)NC(C2(NC(=O)NC)CCCCC2)=O)cc2c(s1)CCC2 CCC(CC(F)F)C(=O)NC1CCN(C(=O)Cc2cc(C3CC3)on2)CC1F Cc1cc2cccc(NC(c3csc(NS(=O)(=O)c4ccccn4)n3)=O)c2cn1 c1(C(=O)NCCN(C(CCC(C)SC)=O)CC(C)O)cnc(C)c(N)c1 CC(C)C(C(=O)NC(C)C(CO)NC(C1(O)CC(F)(F)C1)=O)n1cnnc1 C1(C(=O)NC(C2CN(C(=O)CS(=O)(=O)N3CCCCC3)C2)C)(CO)CCCCC1 CC12CN(C(C3(C4CC4)CC3)=O)C(C(N3CCC(C)(F)C3)=O)(C1)C2 C(=O)(CC(C)C(C)(C)C)N1CCCC(N(C(c2c(C)n[nH]c2)=O)C2CC2)C1 c1(OC)c(C(N2CCC(NC(=O)CCC(C)(C)O)C(C)C2)=O)cccc1F c1(C(c2nnnn2Cc2ccccc2)NC(c2ccccc2)CC)coc(C)n1 Cc1oc2cc(C(N3CC(C)(NC(C4CCCCS4)=O)C3)=O)[nH]c2c1C Cc1nnc(C(=O)NC2CC(F)(CNC(c3ccoc3Cl)=O)C2)s1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(O)(CCNC(C(=O)N(C)C)=O)CC1 Cc1cc(Cl)c(F)cc1CNCCCN1CCN(Cc2ccc(I)c(O)c2)CC1 C1(C(=O)OC)CCC2(CCC2)C1C(N1CCN(C(=O)CSCC(C)C)CC1)=O c1(C(N(C(CN(C(CSCCCC)=O)C)C)C)=O)ccc([N+](=O)[O-])c(SC)c1 C1(NC(C=C(CC)CC)=O)COCCN(C(=O)C(F)=C(C)C)C1 c1(-c2n(C)cnn2)cn2cccnc2n1.C123CCCN(C1C2)OC(=O)C3.C(C)(C)C C1(NC(c2cn(CC)nn2)=O)CC(C(=O)NC2CC(CN(C)C)C2)CC1O CN1CCC2CN(C(C3CCCN3C(=O)CCNC(=O)N(C)C)=O)CCC12 c1(C(N2C(CNC(C(COC)C)=O)C(C)CCC2)=O)cc2c(C)cc(F)cc2[nH]1 c1(C(C(=O)NC(C(CO)NC(=O)OC(C)(C)C)C)N(C)CC)cccc(F)c1Br C(=O)(C1=C(CCCCl)N(c2ccc(F)c(F)c2)C(=S)NC1c1cnc[nH]1)OCC C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1C(NC(c2c(C)cccc2Cl)=O)C1 N1(C(COC)=O)CCC(O)(C(C)CNC(=O)C=C(Cl)Cl)C1 C(CC(O)C(=O)NCCOC(F)F)NC(CCc1ccn(C)n1)=O C1(C(=O)OCC)CN(C(=O)C(=O)N(C)Cc2nc(=O)n(C)[nH]2)c2ccnn2C1 N1(CC2CCN(C(c3nn(CC)c(C)c3)=O)CC2)CC(=O)CC12CCCC2 O=C(N=c1cco[nH]1)C1CCCN1c1ncc(-c2cc(F)cc(F)c2)s1 Cc1nc(C(N2CC(NC(c3cc(C(N)=O)co3)=O)C(O)C2)=O)ccc1[N+](=O)[O-] c1(C(N(C2CCCN(C(CCCNC(C)=O)=O)C2)C)=O)cnc2ccnn2c1 C1(NC(c2n(C=C)nnc2)=O)CCC12CN(C(c1ccc(OC(C)C)nc1)=O)C2 C#Cc1cnc(C(=O)N(CC(=O)NC2C(C)C2(C)C)C)c(C)c1 c1(OC)ccc(CCCCC(=O)N2CCC(CCN(C(=O)C(C)O)C)CC2)cc1 c1(C(N(CC(C)NC(CCCC(C)O)=O)C)=O)cc(Cl)cc2c1NCCC2 S(=O)(=O)(c1cc(C#N)ccc1Cl)NCCNC(=O)Nc1cc(OC)c(F)c(F)c1 c1(C(N2CC(CNC(=O)C(F)OC(F)(F)F)C(O)C2)=O)cc2c(s1)CCC2 C1(C(=O)NC)(C=O)CCOCC1.C1(F)(C(=O)NCC2(n3nccn3)CC2)CCC1 c1(C(=O)NC23CC(CNC(=O)C=C4CCCCC4)(C2)C3)ccc(F)c(Br)c1 C(=O)(CCC(F)F)NC(CN(C)C(C1CCCC1(C)C)=O)(C)C C(CNC(c1cc(C2CC2)[nH]n1)=O)(CC(=O)NCCc1csnn1)OC c1(C(=O)NC2C(NC(C3CC(C)OC(C)C3)=O)COC2)c(Cl)ccc(F)c1F Cc1cc(F)ccc1NC(=O)C(c1scc(C)c1C)N(C)Cc1ccc(F)c(Br)c1 C1(C2CCCCO2)(C(N(CC(F)F)CCC)=O)CCCO1 c1(C(=O)NCC(c2cc(F)cc(Cl)c2)NC(C(C(C)C)C)=O)cccc2ncnn12 C(=O)(C(C)c1cc[nH]n1)NCCSCC(=O)N(CCCC)CCCO n1(CC)cc(C(N2CCC(C(F)C(N3CC(C)(O)C3)=O)C2)=O)nn1 c1(C2(C(=O)NC3C(CNC(Cc4nnc(C)o4)=O)C3)CC2)cccc(F)c1F N1(c2ncc(OCCOC)cn2)CC2CN(c3ncncc3F)CC2C1 c1(C(C)=O)ccc(C(=O)N(C2CCC(NC(=O)CSCc3ccco3)C2)C)cc1 C(C(N=[N+]=[N-])C(=O)NCC1C2CCCOC12)OCC.C1(CC2CC2)CC(=O)N1 CC(C)C(O)C(C)NC(C1(CNC(=O)C(F)F)CCC1)=O C1(C(N(C(C)CNC(=O)Cn2c(C)ccc2C)CC)=O)COC(C)(C)CO1 Cc1sc(C(N2CCN(C(=O)Cc3ncn(C)c3C)C3CC23)=O)cc1[N+](=O)[O-] C1(CCNC(C(C)SC)=O)CCCN(Cc2ccc(-c3ccc(F)cc3)s2)C1 N1(C(c2n(CCC)ncc2)=O)CC2CC1CC2NC(c1cc[nH]c1)=O C1(CC)CN(C(=O)C(=O)N(c2ccc(Cl)cc2)CC2CC2)CCC1=O c1(CC(=O)NC2CN(C(c3ccncc3C(F)(F)F)=O)CC2O)cccc(Cl)c1 C1(C(=O)NCC2CCN(C(=O)Cn3cc(CO)nn3)C2)Cc2cscc2C1 CCCC(C)C(=O)NCC1(C(N)=O)CN(C(c2cn(CC(F)(F)F)nn2)=O)C1 N1(Cc2cnc(OCC)nc2)CCC(F)(C(=O)Nc2ccnc(F)c2)CC1 N1(CC)CCCCC1C(=O)NCC1CC(CNC(=O)COC2CC=CC2)C1 C1(NC(COc2ccn(C)n2)=O)CC(NC(C2(C3CCCO3)CC2)=O)C12CCC2 C(N1CCC(S(=O)(=O)N2CCOCC2)C1)n1nc(C)n(CCOC)c1=S C(=O)(CN=c1cc[nH]cc1)N1C(CC)CN(C(c2cccc(Br)c2)=O)CC1 c1(OC)cc(Cl)c(Br)cc1C(=O)NCC(CO)NC(C1(Br)CC1)=O Cc1noc(C2CC2)c1C(=O)NC1CCC1NC(=O)CC(O)CN(C)C CC1CC(=O)CCN1C(c1c(-n2cc(C3(CO)CC3)nn2)cccc1N)=O C1(C)(CC)C=C(C(=O)N2CC(C(C)NC(=O)C(C)C3(O)CCC3)C2)C1 N1(C(CC2CC(=C)C2)=O)CC(CC(=O)NCCC(C)N(C)C)C2(CC2)C1 c1(OC)cc(C(N2CC(NC(=O)Cc3cccc(Br)c3)C(C)C2)=O)cc(Cl)c1O C1(C(N2CCC(C)(NC(C3C=CC=CC=C3)=O)CC2)=O)CC2CCCCC2O1 C(C1(O)CCCc2ccccc21)NC(=O)NC12OCC(CF)(C1)C2 c1(CNC(C2(NC(C3CN(C(C)=O)C3)=O)CC(F)(F)C2)=O)nccc(C)c1F CC1(C(=O)NCCOCCC(=O)NC2CCCSC2)CCC(=O)C1 Cn1nc(CC(=O)NC2(C)CCN(C(=O)Cc3cncs3)C2)cc1C(F)(F)F N1(C(C(C)CF)=O)CC(NC(c2cc(O)cnc2N)=O)CC12CCC2 c1(CC)cccc(C(N2CCC(CN(C(=O)C(CCOC)OC)C)C2)=O)n1 C1(C(=O)NCC2N(C(C(CC)C)=O)CCCC2(C)C)CC(c2cnn(C)c2)=NO1 c1(C(=O)NC2CN(C(c3ccnc(C)n3)=O)C(C)C2)cc2ccc(Cl)c(F)c2o1 Cc1nc(Cl)nc(N2CCCC2(C)CNC(c2ccc(O)nc2)=O)c1Cl C(=O)(CCCCCN=[N+]=[N-])NC(C1(O)CN(C(c2cc3ncccc3[nH]2)=O)C1)C c1(CNC(=O)CCc2ccncc2)cc(O)nc(CNC(C2(N(C)C)CC2)=O)n1 C(=O)(C1=Cc2cccc(OC)c2OC1)N1CCC(CN(C(CCSCC)=O)C)C1 C1(NC(CCOCCOC)=O)CC2CCC1CC2NC(=O)C1=C(Cl)CCC1 Cc1ncnc(NCC(O)CNC(C2CN(C)CC2C(F)(F)F)=O)c1Br C(=O)(C1Cc2c(Cl)cccc21)N(CCN(C(c1c(C(=O)OC)scc1)=O)C)C Cn1c(=N)[nH]c2cc(C(=O)NC3COC4(CCCN(C(=O)CNC=O)C4)C3)ccc12 c1(C(N2CCC3(CC(NC(c4cnn[nH]4)=O)C3)C2)=O)ccnc2ccccc12 N1(C(C(C(C)C)O)=O)CCC2(CCCN(C(C3(C4CCCO4)CCC3)=O)C2)C1 C1(NC(c2ccc(NC(C3CCCO3)=O)c(Cl)c2)=O)CNCC2(CCC2)C1 C1(N(C)C(c2cocn2)=O)CCC(NC(C23CCCC2C3Br)=O)CC1 c1(C(=O)NC2CC(C)N(C(=O)Cn3cnnc3O)C2)ccc2ccc(Br)cc2n1 N1(C(c2cccc(C)c2F)=O)CC(NC(C2CN3CCCC2C3)=O)C2(CCC2)C1 c1(C(=O)NC(C2CCN(C(=O)CCC3CCCOC3)C2)C)ccc(C(F)F)o1 C(=O)(C(C)(O)C(C)(C)C)N1CC(COC)N(C(c2ccc(F)c(SC)c2)=O)CC1 CCC(C)(C)C(O)C(=O)N1CCN(C(=O)C=C2CCC2)CC1C1CC1 CCCC(C)CC(=O)N1CCC(F)(CNC(c2ccc(COC)[nH]2)=O)C1 c1(C(N(CCNC(c2c(C)onc2)=O)C2CC2)=O)nccc(N)c1Cl N1(CC(=O)NC(=O)NCCC)CCC(CNC(C2(C)CC(C#N)C2)=O)CC1 N1(C(C)=O)CSCC1C(=O)NC1CCC(CNC(=O)COC(F)F)C1 Cc1noc(C)c1S(=O)(=O)N1CCC(O)(CN2CCCC2c2ccc(Cl)cc2)C1 C(=O)(C#CC1(C)CCCO1)N(CC(=O)NC1CCC(C)C1)CC1CC1 CC1CCC(N2CCC(CC(C)NC(=O)C(=O)N)CC2)CC1.C1(C)CCCC(C)C1 c1(C(N(CCNC(CC2CC(=C)C2)=O)C(C)C)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 N1(C(=O)NC)CCN(N2CC(N(C)C(=O)OCc3ccccc3)C3(CC3)C2)C1 N1(C(c2ncn(C)c(=O)c2)=O)CCCCCC(NC(C2CC3C=CC2O3)=O)C1 C1(C)(NC(=O)NCC(CC)(C)OC(C)(C)C)CN(C(=O)OCC)CCO1 C1(C(=O)NC(C)CN(C)C(C2CN(C(N)=O)C2)=O)CCCN1c1nccs1 N1(C(c2c(C)ccc(=N)[nH]2)=O)CCC2(CCCN2C(C2CCCCC2(C)C)=O)C1 c1(C(=O)NC2(CC=C)CCN(C(c3ccnnc3)=O)C2)cnc(Br)c(OC)c1 c1(CC)cc(C(N2CC(F)CC2CNC(C2(C)CCCCO2)=O)=O)ccc1F N=c1ncc(C(=O)NC2CCCCC2NC(c2cocc2Br)=O)c[nH]1 C(=O)(C(CNC(=O)OC)CO)NCC(CNC(CC(C)C)=O)F.C(C)(C)(C)O c1(C(=O)NC2(C3N(C(CN(CCC#C)C)=O)CCC3)CC2)ccc(C(N)=O)nc1 C(=O)(CC(C)(C)C(C)=O)NC(C(=O)N(CCCOCC)C)C(C)CC N1(C(C(CCC(C)C)NC(C2CN(CC)C(=O)C2)=O)=O)CCCC2CCCCC12 c1(C(N2CC(CC(C)NC(C(CCSC)OC)=O)C2)=O)cc2ccccn2n1 C1(NC(C2CC(n3cccn3)C2)=O)CCN(C(c2cnco2)=O)CC12CCC2 c1(NC(C(N2CC3CCC2C(O)C3)c2nc(C)sc2C)=O)ccc2c(c1)CCC2 C1(C)(NC(C2C(=C)C2)=O)CCN(C(=O)C(C2CCCCC2)OC)C1 C1(C(=O)NCCCCCCN(C(C(C)NC(C)=O)=O)C)NC(=O)C2CCC12 C1(CNC(c2c(C)cncn2)=O)CC2(CCC2)CN1C(=O)CSCC#N Cc1nccc(C(=O)NC(C(=O)NCCC(=O)NC(C)C)C2(O)CCC2)c1N C1(NC(c2c(C)nccn2)=O)CC=C(C(=O)NCC2(C)CCOC2)C1 N1(C(CC=C)=O)CC2CCN(C(c3cc(-c4ccn(C)n4)on3)=O)C(C2)C1 C1(CC(=O)Nc2ccc(SCC)cc2)CCCN(C(=O)C(C(C)CC)OC)CC1 C(CCC=C(C)C)(C(=O)NCc1ccc(F)cc1)N(CC)Cc1cccs1 N1(C(CS(CC)(=O)=O)=O)CCN(C(=O)Cc2ccc(C)cc2Cl)C(C)CC1C CC1(C)C2CC(C(=O)N3CCC(C(=O)NCCn4ccnn4)O3)CC12 c1(C(=O)NCC23C(CN(C(CCc4c(C)ncs4)=O)C2)C3)cnc(N)c(Cl)c1 C(=O)(CCCCC(=O)NC(C1CCN(C(c2ccnn(C)c2=O)=O)C1)C)NC C(=O)(C1=NOC2COCC12)NC(CC(C)NC(c1ccc(C(=O)OC)o1)=O)C c1(C(=O)NCC2C(C)CN(C(=O)C(O)C3CCCC3)CC2)cccc(N=[N+]=[N-])c1 C1(CCC)(NC(=O)CC2CC=CC2)CCCN(C(C2CC(CN(C)C)C2)=O)C1 CC(C)(C)CC(O)C(=O)NCC(C)(CO)NC(=O)C#CC1(C)CC1 C1(NC(Cc2c(C)ocn2)=O)CC(O)CN(C(=O)C(C2CCCCCCC2)O)C1 c1(OC)cncc(C(=O)NC(C)C(C)NC(=O)CCCn2cncn2)n1 N#CC1CCCC1NC(=O)CC(CC1CC1)NC(=O)CC1CC(F)C1 Cc1noc(N)c1C(=O)NCCCCCN(C)C(C1CCC1n1ccnc1)=O c1(N(CC)CC2CCCN2C(c2cnc(C(C)(C)C)s2)=O)cnc(C#N)cn1 Cc1ccc2cc(C(N3CC4CC3CN4C(C3(O)CC(C)(C)C3)=O)=O)[nH]c2c1 C1(OCC(=O)N(C(CSCC=CCCC(C)=O)=O)C)CCOCC1 c1(C(=O)NC2C(O)CCN(C(c3cccc(C)c3)=O)C2)nc2ccc(F)cn2n1 c1(C(N2CCC(Oc3ccc(C)cn3)C2)=O)cncc(P(C)(C)=O)c1 C(=O)(C1SCCc2ccccc21)N1C(CNC(=O)Cc2ccc(F)c(Cl)c2)CC1 N1(C(C2CC(=C)C2)=O)CCCCC1C1(NC(=O)C(C)NC(=O)NC)CC1 C(=O)(C1=CCN(C(C2CCCOC2)=O)C1)N1C(C(=O)NC)CCC1 Cc1ncn(C)c(=O)c1C(N1CC2CC2(NC(=O)CC2CC3(CC3)C2)C1)=O n1(CC(=O)N(C2CCN(C(=O)CCCn3cccn3)C2)CC)cccc(C)c1=O CC(C)CC(CNC(C1(c2cc[nH]n2)CCC1)=O)NC(=O)Cc1cscn1 c1(NC(CCOC)c2nn[nH]n2)cc([N+](=O)[O-])cc(Cl)c1OC N1(C(C2(CC)CCC2)=O)CC2CN(C(C3CCSCC3)=O)CC(F)(F)C2C1 C(=O)(CCC(C)(C)NC(=O)C=CC(C)C)NC1(CCOC)CCC1 C1(C(C)C)CN(C(=O)CCC(C)C#N)CCCN1C(=O)C=Cc1cccc(Cl)c1 n1(CC(N2CCC3C(NC(CC4N(CC)CCC4)=O)C32)=O)cccc(N)c1=O N=c1[nH]c(C(N2CCC(CS(N)(=O)=O)C2)=O)nc2ccc(Br)cc12 C(=O)(CN=c1ccc(C#N)c[nH]1)NCC1C(CNC(c2c(C)cc(C)nc2)=O)C1 C1(NC(c2ccc(C#C)cc2)=O)C(CNC(=O)C(C)(C)CF)CCC12CCC2 Cc1cc(=NCC2CCCC(F)C2)[nH]cc1S(=O)(=O)NCCCn1cccn1 Cc1cc(F)ncc1NC(=O)C1=CCC(NC(c2ocnc2C(C)C)=O)C1 Cc1cc(Br)cc2cc(C(=O)N(C(C)CNC(=O)CC(C)(C)C#N)C)[nH]c12 CC1Oc2ccc(C(N3CCC4(CCC4)C3)C(=O)NC3CCCC3)cc2NC1=O c1(C(C(=O)NCCNC(C(CC)NC(=O)OC)=O)N(C)C)ccc(F)c(F)c1 N1(C(C(c2ccc(F)cc2)N(C)C2CC2)=O)CCCc2c(C(F)(F)F)cccc21 c1(CC(N2CCCCC2CN2CCCC2)=O)cccc2ccncc12 N1(C(C(=O)Nc2c(CC)cccc2)c2csnn2)CCC2(CC1)CNC(=O)N2 c1(CCCC(N2CCC(C(C)(C)NC(CCCC#N)=O)C2)=O)c(F)cccc1F N1(C(CCn2c(C)nc(C)n2)=O)CC(F)(F)CC1CNC(C1CCN(C)C1C)=O c1(CCC(=O)NC(C2CCCN(C(COC)=O)C2)C)cc(OC)ccc1OC C1(CNC(C2(SC)CN(C(C3CC(=C4CCC4)C3)=O)C2)=O)CCCCN1C C1(c2nc(C)[nH]n2)CN(CC(=O)N(C)CC2CCC(O)CC2)CCO1 c1(C(=O)NCC(C)(C)NC(Cc2cc(OC)no2)=O)cc2c(C)noc2cc1C C(=O)(C1CC(=O)C(=O)N1)NCCNC(CCSC)=O.C(C)(C)(C)OC(C)C.N(C)C S(=O)(=O)(c1c[nH]ccc1=NC(CO)C1CC1)NC(CCOC)c1ccco1 c1(SC(c2ccccc2)C(=O)NC(CC)C2CCC2)ccccc1O c1(CCC(=O)NCCCN(C(c2occc2F)=O)CC)cccc([N+](=O)[O-])c1 C1(NC(CC(C(C)C)O)=O)C2COCC1CC(NC(=O)C#CC1CCOCC1)C2 CN1CC(C)(C(=O)NCCCC2CN(C(C3CCC(O)CC3)=O)CCO2)CC1=O C1(N(C(=O)CCc2ccsc2)CC)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 Cc1cccc(OCc2ccc(-c3nnc(N4CCC(C)(CO)C4)n3C)cc2)c1 c1(C(N(CCNC(C(c2cccc(C)c2)C)=O)C2CC2)=O)ccc(N)c(C)c1C N1(CC)C(=O)CCC1CC(=O)NC1C2CC1N(C(=O)CNC(=O)CN(C)C)C2 C1(CNC(C(CSC)C)=O)(NC(c2cn(CCF)nn2)=O)CC2CCC1CC2 c1(C(N2CC(C)C(NC(=O)CC3CCCCCC3)CC2)=O)nccc2n[nH]cc12 C1(C(N(C2CCN(C(c3sc(O)nc3C)=O)CC2)CC#C)=O)CCC(N=[N+]=[N-])C1 C(=O)(C1=NOC(C)C1)NCCN1CCN(C(c2c(C)sc(O)n2)=O)CC1 N1(C(Cc2nc(C)sc2)=O)CCCC(CCCCNC(=O)Cc2cnccn2)C1 C1(O)(CNC(c2n(CC)ncn2)=O)CCN(C(C2(C)CCCC2(F)F)=O)CC1 N1(C(C(C)OCC#C)=O)CCN(C(c2ccc(CC)c(F)c2)=O)C(CF)C1 C1(C(NOCCC)=O)CC(C)CCN1C(C1CC=C(C)CC1)=O C1(C(=O)NCC2CC(NC(c3ncn(C(C)(C)C)n3)=O)C2)CCC2C(C1)C2(F)F C(=O)(C#CC1(CC)COC1)NC(CNC(COCCCOC)=O)CC c1(C(N(C(CCNC(CCOCCOC)=O)C)C)=O)ccc(F)c(C)c1C N1(C(Cc2scc(C)c2)=O)CCC2(CCN(c3nnc(CO)s3)C2)C1 N1(C(c2nccc(SC)n2)=O)CC2CC(Nc3cc(O)nc(O)n3)CC1C2 c1(C(=O)NC2C(NC(c3cnn(C(C)C)c3F)=O)COC2)cc(F)ncc1NC N1(C(c2c(C)nc[nH]2)=O)CC(C(=O)NC2COCC2CO)C(C)(C)C1 C(C(=O)N(C(CNC(=O)CCCCC1CC1)C1CC1)C)(C(C)C)SC Oc1ccnc(C2CCN(CC(F)C3CNC3)CC2)n1 C1(N(C(C(C)c2ccco2)=O)CCO)CCN(C(=O)CCCc2ncco2)C1 C1(C(=O)NCCCc2c(C)n[nH]c2)CN(C(=O)CCCC2CC2)CC12CC2 c1(C(=O)OC)cccc(N(C(=O)CC2CCN(C(c3cc(C)[nH]n3)=O)C2)C)c1 C1(C(N2C(C3CCN(C(CC4COC(C)(C)O4)=O)C3)CCC2)=O)Cc2cscc2C1 C1(C(=O)NC(C)CN(C)C)(CO)CCN(C(c2cscn2)=O)C1 N1(C(C(CC)(C)C)=O)CCN(C2CCNC2=O)C(C)C1 O=C1CC(C(=O)NC(C(=O)N2CC(SC(F)F)C2)C2CCC2)CC(=O)N1 N1(C(CCOCC#C)=O)CC2CC(C)N(C(c3cncc4nc(C)[nH]c34)=O)C2C1 c1(C(=O)NCC2(O)CCN(C(=O)C=C3CCCC3)C2)cccc2[nH]cc(Cl)c12 Cc1cnc(CC(=O)NCCC2CC(NC(=O)C=C3CCC(C)C3)C2)o1 c1(C(N(C2CCN(C(c3cccn3C)=O)CC2)C)=O)c(C#N)cnn1C Oc1c(CC2CN(c3ncc(F)cn3)CC23CC3)cccc1F c1(C(=O)NC2(CNC(c3occc3Cl)=O)CC2)ccnnc1O Cc1cc(C(N2CCC(NC(c3ccc(O)nn3)=O)C23CC3)=O)c(O)nn1 CN=c1[nH]c(C(N2CC(NC(=O)CCCNC(N)=O)C(n3cccn3)C2)=O)cs1 C1(C)(C(N(CC(CN(C(=O)Cc2ccon2)C)O)C)=O)CCC(F)(F)C1 c1(C(=O)NCCC2(O)CCCN(C(C(COC)OC)=O)C2)ccn2ccnc2c1 c1(CC(=O)NCCC(C)NC(C2CCO2)=O)c(F)cccc1F C1(CC(=O)N(C2CC2)CC2CCCN2C(c2cc[nH]n2)=O)CCCCO1 c1(C(=O)NCC(CNC(C(CCC)OCC)=O)(C)OC)c[nH]c(=N)c2[nH]ccc12 c1(C(N2C(C(N3CC(=O)NC(C)C3)=O)CC(=C)C2)=O)ccc([N+](=O)[O-])c(O)c1 N1(C(C2CC=C(C)CC2)=O)CCN(C(=O)CC2C=CCC2)CC1CCO CC(C)(C)C(=O)CCC(=O)N1C(C(N2CCOCC2CC2CC2)=O)CCC12CC2 CN1CCN(C)C(CNC(=O)C(CC(F)F)N(C)C(C2CCCNC2=O)=O)C1 C1(O)(CN(C)C(C2C3COCC23)=O)CN(C(=O)CC23CCCC2C3)C1 c1(-c2n(CC=C)c(N(C)CC3(OC)CCC3)nn2)cc(=O)c(O)co1 c1(CNC(C(C)NC(C)=O)=O)cc(C(=O)NCC(C)OC(F)F)n(C)n1 c1(C=O)ccncn1.C(=O)(C(C)N(C(C1CC1CF)=O)C1CC1)OCC c1(OCCOC)ccc([N+](=O)[O-])c(C(=O)NC2CCC3CCCCC3C2)c1 c1(C(=O)NC2C(C(C)NC(=O)OC(C)(C)C)C2)cc(S(=O)(=O)NC(C)C)c(C)o1 C(=O)(C1SCc2cccnc21)N1CCC(NC(c2cc(O)ccc2F)=O)C(O)C1 N1(C(CC2CC(CC)C2)=O)CC2CCC1CC2NC(c1cnn[nH]1)=O C(=O)(C(C)(C)CCCCC)N1CC(NC(=O)C(C)OC2CCCC2)CC(OC)C1 N1(C(C2(OCC)CCOCC2)=O)CC2CC(C1)N(c1cc(C)nc(SC)n1)C2 N1(CC)CC2(C1)CN(CC1C=CC(N(C)CC3(NC(C)C)CCC3)C1)C2 c1(C(N2CCC(NC(Cc3cc(C)on3)=O)(CF)C2)=O)ncnc(O)c1Br CC1CC(C(=O)N2CCC(NC(c3c(C(F)(F)F)cnn3C)=O)C2)=NO1 c1(C(=O)NCC(C2N(C(C=CC(CC)=CC)=O)CCC2)(C)C)ccc(C)c(O)n1 C(=O)(C1=C(C)CCCC1(C)C)NCC(C(C)(C)C)NC(CC(CC)(C)C)=O c1(CC)cc(Br)ccc1C(=O)NCC1CN(Cc2ccc(C(F)(F)F)c(O)c2)C1 n1(CC)nc(C)cc1C(=O)NC1CCCC(NC(C2CC(C(F)(F)F)C2)=O)C1 C1(C(=O)NC(C)CCNC(C2(C)CSC2)=O)CCc2cnn(C)c2C1 c1(CCC(=O)N(CC(CNC(C2C(CCOC)C2)=O)C)C)cccn1C N1(C(=O)CC(C(N2CCC(CCO)C2)=O)c2ccoc2)CCC2(C=CCO2)CC1 C(=O)(C(F)CCC(C)C)NCC(CCOC)NC(c1ccncc1N)=O c1(NC)ccc(F)cc1C(=O)NCCC1CCN(C(=O)C(C)CSC)C1 O(NC(=O)CC(C)(C)N(C)C(C1(O)CCSCC1)=O)C1CCCN(CC)C1 Cc1cc(C(N2CC(CNC(C3COC(=O)N3C)=O)C(C)C2)=O)n(C2CCC2)n1 CCC(Cc1nc(-c2cccs2)nn1Cc1cc(C)nc(C)c1)CC(F)F C1(CNC(CCNC(C)=O)=O)CN(C(=O)C(C)c2ccsc2)CC1C CC12CCOC(C(N3CCC(NC(c4ccc(F)s4)=O)C3(C)C)=O)(C1)C2 N1(C(c2cc3ccc(Br)cc3o2)=O)CCC2CCN(C(=O)C3CC3)CC2C1 c1(C(=O)Nc2ccc(C(=O)Nc3cncc(Cl)n3)cn2)onc2ccccc12 C(=O)(CCCC(C)(F)F)NC(CNC(CN(C(C)C)C)=O)C(C)C(C)C c1(CCC(N2CCCN(C(C(CC)C#N)=O)C(C)C2)=O)cccc2c1OCCO2 C1(OC)CC2CN(C(C3C(C)(C)C3(F)F)=O)Cc3cccnc3N2C1 C(CCC)(C(=O)N1CCC(C)(NC(c2cc(OC)no2)=O)C1)=CCC C1(O)(CN(C(Cc2c(C)noc2Cl)=O)C)CCCN(C(C2C=CCC2)=O)C1 C(=O)(C(CC(=O)OC)OC(C)(C)C)NC(CN(C(C=COCC)=O)CC)C c1(OCC)ncc(C(=O)O)cc1NC1CCCC1c1ccc(Br)cc1 c1(N2CC3(C(NC(=O)COC4CCOCC4)CCC3)C2)ccc([N+](=O)[O-])c(O)n1 CC(C)C(F)C(=O)N(C)CC1(C)CCCC1NC(=O)CSc1ccc(O)cc1 C(c1ccn(C)c1)=CC(=O)NC1C(NC(CCc2scc(C)n2)=O)CC1 N1(C(c2c(C)c(F)cnc2)=O)CC(C)N(C(=O)C(C)C(C)C)C(C)C1 N1(C(CCCSC)=O)CCC2CCCC12CNC(c1cn(C)c(C)n1)=O c1(C(=O)NC(CC)CNC(=O)C(C)(F)C(C)(C)F)cc([N+](=O)[O-])ccc1SC CCC1=NOC(C(N2CC(CNC(c3ccccc3Br)=O)C2)=O)C1 N1(C(CC(C)O)=O)CC(CNC(=O)Cc2csc(C3CCCC3)n2)CC(C)(C)C1 C1(F)(CNC(c2c(CC)n(CC)nn2)=O)CCN(C(=O)C(C)=CC2CC2)CC1 N1(C(C2CC(C(=O)OC)C2)=O)CC2CC3CC2C1C3NC(C1CC(O)C(F)C1)=O N1(C(c2nc(OCC)oc2)=O)CCN(C(C2CC(C)CO2)=O)CC1CCO CC1CN(C(=O)CCN2CCN(C)CC2)CCC1NC(=O)C(C1CCC1)C1CC1 C(C)(CO)(C(=O)N1CC(C(C)(C)C#N)C1)NC(c1nc(CC)oc1)=O N1(C(=O)CCF)CC2CC(C1)N(C(=O)C(Cc1ccccc1)C1CCCC1)C2 N1(CCC(=O)NC(C(C)NC(c2cn(C)c(O)n2)=O)C)CCc2ccccc2C1 C1(NC(CC(CNC(CCCCSC)=O)O)=O)C(O)C2CCCC12 C(=O)(CC(C)(C)C(=O)N1CC2=C(C1)CN(C(=O)C(=O)NCC(F)F)C2)OCC N1(C(CSC)=O)CCC2(CC1)CC2(CO)CNC(=O)Cc1sccc1Cl c1(N)cccc(S(=O)(=O)N2CCCC2)c1.C(=O)(CP(C)(C)=O)NC(C)CCSC c1(OC)c(C)cc(C(=O)NCC#CCNC(=O)CSSC)cc1C C1(NC(CC2C(C)CCC2)=O)CN(C(=O)CN(C(=O)C2CC2)CCC)CCC1(C)C c1(C(N2CCC3(CCOC3)C2)=O)n[nH]c2c1CN(Cc1c(F)cc(Cl)cc1Cl)C2 C1(CC(=O)NCC(C)CNC(C2CC(N(C)C)C2)=O)CCC2(CCC2)O1 c1(C(=O)NC2C(C)(C)N(C(C3CC(F)(CO)C3)=O)CC2)ccnc2c1CCO2 c1(CN(C)Cc2cccc(C)c2)cc(Cl)c(Cl)n1C Cn1cc(NCC2CC(NC(C34CCC3C4)=O)C2)c(OCC(F)F)n1 C(CN=c1[nH]c(=NCc2cnc[nH]2)[nH]c2cccc(F)c12)OCC(C)C N1(C(C2(CC(=O)NCN)CC2)C)CCC(C)C2(CCC2)C1.n1(CC=O)ncccc1=O c1(C(CNC(=O)CCOCC(F)F)NC(C(C)SC)=O)ccccc1F C(=O)(C(C)(C)C1=CCN(C(C2CC2C(F)F)=O)C1)NCc1c(C)cn(C)n1 C1(NC(C2CC(C(C)C)C2)=O)C2CC(NC(=O)C(F)(F)CO)CC12 C1(NC(c2nc(CC)oc2)=O)CCN(C(C23CC(F)(C2)C3)=O)C(C2CC2)C1 C1(CNC(CC(C)(C)NC(Cc2c(C)ocn2)=O)=O)CC2(CC2)C(=O)O1 c1(C(=O)NCC2(O)CCN(C(c3cc(C)c(C#N)[nH]3)=O)C2)ncnc2ccsc12 C1(C)(CC)CN(C(C2CC(N(C)C(c3cncs3)=O)C2)=O)CCO1 C(=O)(CC1C(=O)Nc2ccccc21)NCCCN(C(C)=O)Cc1nnc(C)o1 C1(C(=O)NC2(C(=O)NCC3CCN3C(C)(C)C)C(C)C2)CN(C)CCN1C Cc1oc(-c2ccccc2)nc1CC(=O)NCC1(O)CN(C(=O)C=CC2CC2)C1 c1(CNC(c2c(C)cccc2)C2CCC(C(=O)N(C)C)CC2)cncc(C#N)c1 c1(CNC(CC2CCCC(OCC)C2)=O)cnn2c1CN(c1nncs1)CC2 c1(NC(C(F)=C(C)C)=O)cccc(NC(=O)C(F)Cc2ccccc2)c1 c1(C(=O)NCCCC2N(C(C=CC=CCC)=O)CCC2)cc(=O)c(OC)cn1C c1(-c2n(CCCCCC)nnn2)c(C)nn(CCNCC)c1CC N1(C(C(C)N(CCOCC)CC)=O)CCC(C(C)(C)O)CC1.C(C)(C(=O)OC)N c1(C(C(=O)NC2CCC2)N(CCC(C)C)C)cc(Cl)cc(Cl)c1 c1(N(C)CC2(C)CCCC2)ccncc1S(=O)(=O)N1CCOC(C(C)(C)C)CC1 c1(C(=O)NC(C2CCCN(Cc3cccc(C#N)n3)C2)C)ccc(F)c(Cl)c1F c1(CC(=O)NC2C(CNC(C(CCC)OC)=O)CC2)ccc(C)cc1Br N1(C(c2c(C)nn[nH]2)=O)CCCCC(NC(=O)CCSC(F)(F)F)CC1 c1(CNC(c2ccc(C)o2)=O)ccc(CCNC(=O)Cc2cnc[nH]2)cc1 N1(C(C2(CCC=C)CN(C(c3ncncc3C)=O)C2)=O)CCOC2CCCC12 C1(COC)(CNC(=O)CCCC2CCC2)CCCN1C(=O)Cn1nc(C)nc1C N1(C(c2ccc(COC)o2)=O)CCOC(C)(CNC(c2cc(SC)c(C)o2)=O)C1 Cc1cc(F)ccc1N(C)C(=O)N(C1CC1)CC1(c2ccc(Br)cc2)CCCC1 C1(C(N2C(C)(CC(=O)NCc3n(C(C)C)ncc3)CC2)=O)COCCC1C C1(C(=O)OCc2ccc(COC)s2)CC12CC(S(=O)(=O)N1CCCC1)C2 CC1CCN(C(C2CC(O)CCN2C(c2cnnc(O)c2)=O)=O)C1(C)C C1(CNC(c2c(C)nc(CCC)s2)=O)CN(C(C2CCCCO2)=O)CCN1C c1(OC)ccc(N)c(C(N2CC(CNC(C3(C)CC=CCO3)=O)CC2(C)C)=O)c1 C1(NC(C2(SCC)CC2)=O)CCN(C(c2c(C)[nH]c(C)c2C)=O)CC1C(C)C N1(C(CCCC(=O)NCC)=O)CCC(C2(NC(c3nnc(CC)s3)=O)CC2)C1 Cc1cc(=NC(CC2CC2)C2CC2)[nH]c(=NCc2nc3ccc(F)c(F)c3[nH]2)[nH]1 C1(C)(NC(CCCCOCC)=O)CCCCC1C.C1C(=O)N1 c1(C(N(C(c2ccncc2)CC)CC)=O)ccc(Br)cc1-n1cncn1 CC1(C)CN(C(=O)C(c2ccc(F)cc2F)(C)C)CCC1NC(=O)C1=NOCC1 N1(C(CN(C)C)=O)CCOC(c2cc(C(=O)NC(C)(C)C)n(-c3ccncc3)n2)C1 C1(NC(=O)C(C2CCCO2)C2CC2)CC2CN(C(=O)C=C3CCCCC3)CC12 c1(CCC(C)C)ccc(CNS(=O)(=O)CC2CCCC(C(F)(F)F)C2)cc1 c1(C(N(CCC(=O)NC2CCC2C)CC=C)=O)cn(C)c(C)n1 C(=O)(C#CC1CCCO1)N1CCC(NC(c2nccc(OC)c2)=O)C1C(C)(C)C N1(C(C=CCC2(NC(=O)CC3C=CCC3)CC2)=O)CCC(F)(F)C(F)C1 CN1C(=O)CCC1C(=O)NCC(C1CCCN1c1nc(C(C)(C)C)ns1)(C)C C1CCOC(C)(C)C1.c1(C(=O)OC)ccc(CNC(=O)Cn2cc(CN)nn2)s1 N1(C(CNC=O)=O)CC2(CC(CNC(c3ccc(F)c(C(F)F)c3)=O)C2)C1 C1(C(=O)NCC2(O)CCC(C)C2)CC2(CCN1C(c1cn(C)c(=O)n1C)=O)CC2 c1(C(=O)OCc2cccc(SCC)c2)ccc(Cl)c(Br)c1 c1(SCC(=O)NCc2csc(CNC(C3CCC(F)C3)=O)n2)ccc(F)cc1 c1(NC(N(CC(CC)NC(=O)C(F)C(C)C)C)=O)cn(-c2cnn(C)c2)[nH]c1=N C1(C)(C(=O)NC(C)CCN(C)C(c2ccon2)=O)CCCCC1(F)F C(=O)(CCCCC(=O)N1CC(O)(CNC(C2CCCC2(C)OC)=O)C1)OC c1(CC)ccc(C(=O)NCC23CC2CN(C(=O)CC(C)n2ccc(C)n2)C3)cn1 CC(C)C(C(C)NC(c1cccc(N2CC=CC2)c1)=O)NC(=O)COC(F)F N1(C(=O)COCCF)CCN(C(=O)C=Cc2ccccn2)C(CF)C1 c1(OC)cc(C(N2CCC(C)(NC(c3ccc(=N)[nH]c3)=O)CC2)=O)cc(F)c1F O=C(C1=NOC(C2COC2)C1)NCC1CCN1C(c1ncoc1C1CCCO1)=O c1(C(=O)NC2CN(C(=O)CCN3CCCCC3=O)C2)cc(F)cc2nccnc12 c1(C(N2CCC(NC(C=C(C)C3CC3)=O)C2)=O)ccncc1-n1cccn1 c1(C(C)CC(N2CC3CC2C3NC(=O)CN2CCNC2=O)=O)ccc(F)cc1F C1(C(=O)NC2(CC(=O)NCc3cccnc3F)CCC2)Cc2nccn2C1 n1(CC(=O)N(CCOC)CCNC(=O)C(CO)N(C)C)cc(C)c(O)nc1=O C1(CNC(CCCCOC)=O)(NC(=O)C(C)c2cccs2)CC2CCC1CC2 CC1CC(CNC(C2(F)CCOCC2)=O)CN(C(C23CC(C)(CCO2)C3)=O)C1 C(C1=CCCN(C)C1)NC(C1(CNC(C(CSC)OC)=O)CCC1)=O N1(C(c2ncc(C)nc2)=O)CCN(C)CC1CNC(C1CCOC1C)=O CCCCC(CNC(c1csc(COC)n1)=O)NC(c1ccccc1Cl)=O N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CCC1C CC1(C)CNCCN1C(C1CC1NCc1ccc(Br)c(CO)c1)=O N1(C(CCNC(C)=O)=O)CC2CCN(C(C3CCOC3c3ccccc3)=O)CC12 N1(C(C(c2ccc(Cl)cc2F)CC)=O)CC(Cn2cc(CSCC)nn2)C2(CC2)C1 S(=O)(=O)(c1cc(C)c(-c2ccc(OC)cc2)cc1C)NC(C(CC)CC)C(=O)OC C(CC(C)(C)C(=O)NCCc1cc(C(=O)NCC2(CCO)CCC2)no1)OC N1(C(COCCC(C)C)=O)CCC(CNC(=O)COc2ccsn2)C(F)(F)CC1 c1(C(N2CC(CN(C(C3(CCC)CC3)=O)C)OCC2)=O)cc(OC)ncc1F c1(C(N2C(C3(C(=O)OCC)CC3)CCCC2)=O)cc2cc(Cl)ccc2o1 C1(CNC(COCC(=O)OC)=O)C(O)C(O)CN1C(N1CC(N)C1)=O.C(C)(C)C CC(C)(C)C#CC(=O)NCC1(F)CCN(C(=O)CSc2ccccc2)C1 N1(C(C(C)OCCC#C)=O)CCCC(n2cc(CNC(=O)CCC3CC3)nn2)C1 n1(CC(=O)NC(C)CCCNC(=O)CC2CCCCN2C)ccc(=O)n(C)c1=O N1(C(C2COCCN(C(C(CC(C)(C)C)O)=O)C2)=O)CCc2nccnc2C1 C1(N(C(c2c(SC)scc2)=O)C)CCN(C(=O)C#CC2(C(F)(F)F)CC2)CC1C c1(CCCC(=O)NC2C(NC(C(CC)=CC)=O)COCC2)c[nH]c2ccccc12 C12(C(N(CCCN(C(c3cc(COC)cn3C)=O)C)C)=O)CC(C)(C1)OC2C c1(NC2CCCCN(C(C(C=C)(C)O)=O)C2)ncc(S(C)(=O)=O)cc1Cl N1(C(C2C=CCN(C(CC=CCC)=O)C2)=O)CCN2CCOCC2C1 C1(C)(CNC(c2nnn(C)n2)=O)CN(C(=O)CCSC(F)(F)F)C(C)(C)C1 C1(C(=O)NC(CN(C(c2cnsn2)=O)CC)C)CCCN(c2cnccn2)C1 C1(C(=O)OCC)Cc2cccc(NC(=O)N(CC(C)C)CCO)c2C1 Brc1ccc2nc(CN3CCN4CCCCC4C3)cn2c1 C1(NC(CCC)=O)CN(C(=O)C(O)Cc2c(F)cccc2Cl)CC(C)(C)C1 c1(C(N2CC(c3cn(C(C(=O)OC)C)nn3)C2)=O)cc2c(s1)CCCC2 Cc1c(NC(=O)C(C)(C2CC2)N(C)C(C2CCOC2(C)C)=O)cccc1C#N c1(C(C(=O)NCC2CCCN2C(C2COC2)=O)O)ccc(Cl)cc1 c1(C(=O)NCCC2CCN(CCCC(=C)C)C2)c(C)noc1C(F)F c1(C(N2CCC(COC)(NC(=O)CSC)C2)=O)cnc2n1C(C)CCC2 C1(SC(C(=O)NCCCC)CC)CNCC1(C)C CC1(C)CC(=O)NCC1C(N1CCN(C(c2c[nH]nc2F)=O)CC1CC(F)F)=O c1(C(C)(C)C)ccc(C(=O)NC2CCC2NC(c2ccccc2)=O)[nH]1 c1(OC2CC(=O)N(C3CC3)C2)ccc2c(c1)COC2 CC1CC=C(C(=O)N2CC(C(=O)NC3CC(CCC(N)=O)C3)C(F)C2)CC1 c1(CC)ccc(C(N2CCC(CN(C)C(C3CN(C(N)=O)C3)=O)C2)=O)cc1 N1(c2ccnc(C)n2)CCN(C2CCCN(C(c3cnoc3C)=O)C2)C(=O)C1 N1(C(c2c(CC)ccc(Br)c2)=O)CCCN(C(=O)C(O)C(C)C)CCC1 N1(C(CC)=O)C(CNC(=O)C(F)(F)c2ccncc2)CC2CCCCC12 C(CC(N=c1[nH]c(=NCC(C)(C)C2OCCO2)[nH]c2c1CCC2)C(C)C)OCC Cc1cc(CNC(=O)C(C(C)O)NC(C2CCCN2C)=O)nn1C C1(CC)CCCC1(C)C(N1CC(C(C)NC(c2cnc(C(F)(F)F)nc2)=O)C1)=O C1(C(=O)NCC(CC)NC(c2ccc(C(F)F)c(F)c2)=O)CCn2ccnc2C1 C12CC(n3cc(CCCSC4CC4)nn3)CN1C2=O.C1(C(=O)O)(COC)CCC1 c1(C(=O)NCC=CCNC(Cc2nc(C)sc2C)=O)ccnc(O)c1Br C(=O)(N=c1cc(-c2ccsc2)[nH][nH]1)C1C2CN(C(=O)CN3CCCC3=O)CC21 C1(NC(C=Cc2nc(C)sc2)=O)CCC12CCN(C(C1CC1(C)C)=O)CC2 C1(C(=O)NC2CCC(NC(CNC(=O)OCC)=O)C2)NC(=O)CC1C C1(C(N(CCN(C(C(C)=CC)=O)C)C)=O)CCN(C2CCS(=O)(=O)C2)CC1 c1(C(=O)NC2(C)CCN(C(c3cc(Br)no3)=O)C2)ccc(C2CC2)c(F)c1 N1(C(C(C)(C)OCC)=O)C2CCC1CN(C(c1oc(C)nc1C(F)(F)F)=O)C2 CC1(C)COCC(CC(=O)NCC2CCN2C(c2sccc2F)=O)O1 c1(C(=O)NCC2CC(NC(C3CS(=O)(=O)N3)=O)C2)coc2ccc(Cl)cc12 C=CCCC(C(=O)OC)Sc1c(C(=O)OC)cnn1-c1cccc(C)c1 c1(NC(C2(CC=C)CN(C(C3CC(=O)N(CC)C3)=O)C2)=O)ccnc(OCC)c1 C1(C(=O)NCCN(C(c2c(C)noc2C(F)F)=O)C)CCCC2(CCOCC2)O1 Cc1ccc(Cl)c(OCC(=O)NCCCCNC(c2csc(S)n2)=O)c1 C=CC1CCN(C(=O)C(C2CCCOC2)NC(=O)OC(C)(C)C)CC1 N1(CC(N2CC=CC2CNC(C2(F)CC=CC2)=O)=O)CCCCC(O)C1=O C1(C(C)(F)F)(C(=O)NC2CCC(CNC(C3CCC(=O)N3C)=O)C2)CCOCC1 C1(C(N2C(CCNC(C)=O)COCC2)=O)CC2OC(C)(C)OC2C1 c1(CO)cnn2c1CN(Cc1cccc(C(=O)Nc3ccc(O)cc3Cl)c1)CC2 c1(CC)[nH]ccc1C(N1CC(O)(C2CCCN2C(C2CNC(=O)C2)=O)C1)=O c1(C(=O)NCCC(CC)(C)NC(=O)C(F)C(F)(F)F)ccc(C)cc1C CN1CCN(C(=O)CC2(C(F)(F)F)CC2)C(CNC(=O)CN2CCOC2=O)C1 Cc1coc(C=CC(N2CCN(c3ncc(Br)cn3)CC2)=O)n1.C(=O)(CC(C)C)N C1(OC)(CNC(=O)C=C2CCC2)CCN(C(c2ncccc2CC2CCC2)=O)C1 c1(CC2CC2)ccc2c(c1)OCO2.Cc1cccc(O)c1C1C2CC2C(=O)N1 CCCCCC(=O)NCC1CN(C(C2CCCC2NC(=O)C(C)C(C)C)=O)C1 N1(C(C(C)CN(C)C)=O)CC(C(=O)NC2(C(N)=O)CC2)CC12CCC2 N1(C(C(CC(=C)C)OC)=O)CCC2(CCCC2NC(c2nc(Cl)cs2)=O)CC1 Cc1cccc2oc(C(=O)N(C3CCN(CC(C)CC(C)C)C3)C)cc12 C1(CNC(C(CC)Oc2ccccc2Cl)=O)(CO)CCCN(C(=O)CC(C)C)C1 S(=O)(=O)(c1ccccc1Br)NC(C(=O)NCCC=CCCCCC)C(C)O Cc1nn(C)c(F)c1C(=O)NCC1CCCCN1C(=O)CC1COCC1O C12(CNC(C(C)(C)F)=O)CN(C(=O)Cn3ccccc3=O)CC1CCO2 N1(C(CCC(=O)NC)=O)CCC(CNC(=O)COCC2CCCC2)C12CC2 N1(C(C(C)O)=O)CC2CC(NC(=O)COc3ccc(F)cc3Br)CC(C2)C1 Cc1ccnc2nc(C(N3CCC(NC(=O)CCOCC(F)F)C(F)C3)=O)nn12 C(=O)(CC1=CCN(C(c2ccc(C)c(F)c2)=O)CC1)NCC1CC(C(=O)OC)C1 C1(C(=O)NC2CC(C(C(=O)NCc3c(C)ncs3)F)C2)CCCCC(=O)N1 c1(OC)cc(F)c(C(N2CCC(NC(=O)C(O)C(C)C)C2)=O)cc1N S(=O)(=O)(c1cccc(=NCCn2cncn2)[nH]1)N1C(CNC(N)=O)CCC1 c1(CCC(=O)NCC(CNC(C2(O)CCOC2)=O)OC)cscc1Br CCC(O)(CNC(=O)C(C)N(C(c1cnn(C)c1OC)=O)C1CC1)CC N1(C(c2ccc(COC)o2)=O)CC(NC(=O)CC2CCOCC2)C(C)C1 c1(C(N(C)CCN(c2ccnc(C#N)n2)C)=O)cc(F)cc2nccnc12 S(=O)(=O)(c1cnccc1N1CCC2(C1)OCCO2)NCc1ncc(C)nc1 Cc1nc(SC(F)F)sc1C(=O)N(CCCNC(=O)CNC(N)=O)CCO C1(NC(C2CC(C(C)=O)C2(C)C)=O)CN(C(=O)C=C2CCN(C)C2)CC1(C)C C(=O)(C(CN(C(=O)C=CCF)C(C)C)N(C(=O)CC(C)n1cccn1)C)OC C1(CNC(c2scc(OC)c2)=O)CN(C(C2(C)CC2(Cl)Cl)=O)CCO1 C(C(=O)N=c1ccn(CCO)[nH]1)(C1CCCC1)NC(CC1CCC(=O)CC1)=O N1(C(CC(=C)C)=O)CC2(CCCC(CNC(c3cc(O)nc(C4CC4)n3)=O)O2)C1 CC(C)C(C(C)NC(=O)CO)NC(=O)CCNC(c1cc(-c2ccco2)[nH]n1)=O c1(OCC(=O)N(CCCN(C(C2(C)C(C)CCC2)=O)C)C)cccc(C#N)c1 N1(C(c2cc(CCC)[nH]n2)=O)CCN(C)C(C(=O)NC2CC=CCC2)C1 C1(NC(CC(=C)I)=O)CC12CC(NC(=O)C(O)C1CC1)C2 C1(NC(c2ccc(C)nc2)=O)CC2CN(C(c3cnco3)=O)CCN2C1=O c1(C(=O)NCC2CCC(NC(C(C(C)C)N(C)C)=O)C2)ccc(=O)n(O)c1 C1(NC(C2C(C(C)C)OCC2)=O)CC=CCC1C(N1CCCCC1CCO)=O C(C(C)C(C)C(=O)NCC1=CCN(C(c2cc(O)nc(OC)n2)=O)CC1)OC N1(Cc2c(C)n[nH]c2C)CCC2(CC1)C(O)CC(C(=O)O)C2 C1(NC(C2ON=C(C)C2)=O)CCC(C)(NC(C2CCCCCC2)=O)CC1 Cc1ccc(N2CC(NC(C3CC4OC3C3CC43)=O)CCC2=O)cc1C C(=O)(C(F)CCC(C)(C)C)NCC(C(=O)NCc1nn(CC)nc1C)(C)C N1(C(C(F)=CC)=O)CC(C)(C)OCC1CNC(=O)COc1cc(F)ccc1F N1(C(C(C)CC(N)=O)=O)CC(NC(=O)C(C)N2CCCC2)CC12CCCCC2 CC1CN(C(c2cc(Br)cc(N)n2)=O)CC(C)C1NC(c1ccon1)=O O=C(CCCC(F)C(=O)O)N1CCC2CC(C(=O)NCC(O)C(F)(F)F)C2C1 c1(C(N)=O)cccc2c1CN(C(=O)CC1CCN(C(C3CCC(=O)O3)=O)CC1)C2 CCC(C)CC(C)C(=O)N1CCC(C)(C)C(Nc2ccccc2[N+](=O)[O-])C1 C1(CNC(C(C)O)=O)CCC2(CN(C(c3ccc(F)cc3O)=O)C2)O1 C12(NC(C#CC3(C)CC3)=O)CCOCC1CN(C(=O)Cc1ccns1)C2 c1(C(=O)NCC(CNC(c2cnc(OCC)s2)=O)C)nc(O)nc(O)c1N N1(C(C(N)=O)=O)CC2(CCN(C(=O)COCCCF)C2)C1.c12ccc(Cl)c(c1)O2 N1(C(C2(C)CC2C(F)(F)F)=O)CCCC1(C)C(=O)NCC1CCCOC1 C1(NC(Cc2n(C(C)C)cnn2)=O)CCOC2(C1)CC(C(=O)O)C2 c1(C(=O)NC2(C)CC(NC(C(COC)OC)=O)C2)ccccc1-c1ccccc1 C1(CNC(C(C)NC(C)=O)=O)CN(C(C2CC2C2(C)COC2)=O)CCC12CCC2 C1(C2(O)CCOCC2)(C(N2C3CCC(NC(CC(C(C)C)O)=O)(CC3)C2)=O)CC1 c1(CNCc2cnn(C)c2Cl)c[nH]c2ncccc12.N12CC3CC1C3C2=O C1(CC)CN(C(c2cn(C)c(C)n2)=O)CCC1NC(c1ccc(O)c(C)c1)=O c1(C(=O)NCCN(C(c2c(CC)nccc2)=O)C(C)C)ccn2c(C)ncc2c1 N1(C(c2ccc(CC(=O)OCC)o2)C(=O)NCC)CCOC2(COC(C)(C)C2)C1 c1(C(=O)NCC2(COC)CCCN2C(=O)CCF)cc(Br)c(F)cc1N CC1(C)CN(C(=O)Cc2cncnc2)CC(C)(C)C1NC(=O)CCCCC#N CCC(CN(C)C)C(=O)NCC(CC(=O)NC(C)(CO)CO)C1CCC1 N1(C(CCC(CCC)CC)=O)CCOC2(CCSCC2)CC1 CCS(=O)(=O)NC(C)C(=O)N(CC(C)(C)NC(=O)C(C)c1ccco1)C C1(NC(c2n(CC)nc(C(C)C)c2)=O)CCCN(C(=O)C2=CCCO2)CC1 CC(C)(C)CCC(F)C(=O)N1CCCC1C1(NC(=O)CCCF)CC1 c1(CC)nn(C)c(CC)c1C(=O)N(CC(C)(C)NC(=O)C(CC)CC)C C(C1CCOc2ccc(Br)cc21)NCc1n[nH]c(C)c1C c1(C(=O)NCC(C)(CO)NC(C2CC3CC3C2)=O)nc2n(c1Cl)CCCC2 C12(CNC(=O)C3=NOCC3)CN(C(=O)C=Cc3cccnc3)CC1CS(=O)(=O)C2 Cc1cc(C)c(C(=O)N(CC(C)(C)CNC(c2cc(C(F)F)no2)=O)C)cn1 N1(C(C(C)CC2CC2)=O)CC2(CC(CNC(=O)Cn3cnnn3)C2)C1 C1(NC(CCSCC)=O)CCCCCN(C(=O)Cc2csc3cc(C)sc23)C1 C1(N(C(C2C(=C)C2)=O)CC)CCN(C(=O)C=Cc2ncc[nH]2)CC1 N1(C(c2c(CN(C)C)cco2)=O)CCN(C(C2(CC(F)F)CCC2)=O)CC1CO CC1CC(F)(F)CN1C(C1CSCCN1C(=O)C=CC(F)F)=O Cc1cc(C(=O)NCC2CN(C(C3Cc4nccn4C3)=O)CC2O)c(C)cc1Cl c1(OC)cc(C(N2CC(=C(F)C(=O)OCC3CC3)C2)=O)cc([N+](=O)[O-])c1OC C1(C(N2CCN(C(C(CC)CC)=O)C(CF)C2)=O)CC2CC1CC2(F)F C1(OC)(CNC(=O)CCF)CCN(C(=O)CC(O)CNC(=O)OC(C)(C)C)CC1 c1(C(=O)NC(CCNC(CCC2C(C)C2)=O)c2cccs2)cc2cn[nH]c2cn1 CCC(C(=O)N(C)CC1CCN(C(c2sc(C3CC3)nc2C)=O)C1)C(C)(C)CC c1(C(=O)NC2CCCCC2C(N2CCS(=O)CC2)=O)cc(O)nc(O)c1 C12(C(=O)Nc3c(NC(C)=O)cn(C)n3)CCCC(CO1)C2.C1C(=O)NCC(C)O1 C(=O)(CCCCCNC(C1CC2COCC2C1)=O)N(CC(COC)(C)C)C N1(C(Cc2ccc(C#C)cc2)=O)CCN(C(=O)CSCC)C2COCC12 CC(C)(F)CCC(=O)NC1CCCC(C(N2CCC3C(O)CC23)=O)C1 CC(C)CCCCC(C)NCCCc1ccncc1 c1(CNC(N2CCN(S(=O)(=O)C3CC3)CC2)=O)cccc2cncn12 C1(N(C(c2ccn(CCC)n2)=O)C)CCN(C(C2CCCN2C=O)=O)CC1 C1(CC)CN(C(=O)C=Cc2cccc(CO)c2)CCC1NC(c1ccc(C)[nH]1)=O C12(C(N3CCCC(CCC#C)C3)=O)CCCC1CCN2C(C1CCCC(=O)C1)=O N1(C(C(CC)CC2CCCC2)=O)CC(NC(c2ccon2)=O)CC12CCOCC2 C1(C)(C(=O)NCC2(CO)C(C=C)C2)C=CCN1C(C1OCCC1(C)C)=O C1(C(=O)NC2CC(N(C(C=Cc3n(CC)ncc3)=O)C)C2)CN(CP(C)(C)=O)C1 C1(CCC)C(O)CCCN1C(CCCc1ccccc1)C(=O)NC(C)(C)CC CCCCCC(=O)N1CCC(C(C)C(=O)Nc2cnn(C(C)(C)C)c2)C1 c1(N(C(N(OC)C)=O)C(c2ccc(Cl)cc2)C)cnn2c1C(=O)N(C)CC2 C1(CC(=O)NC2CCC(C)(CNC(c3cnco3)=O)C2)CCC2(CCC2)CO1 C(CC(=O)NC(C)CNC(c1ccc[nH]1)=O)OCC C(CC(C)(C)CC(=O)NC(C(=O)Nc1cc(C)cnc1O)C1CCC1)OC Cc1cnc2c(C(=O)NC3CC(CNC(=O)CC(C)C(C)C(C)C)C3)cccn12 CC1CN(C(=O)CC2(C)CC2)CC1(C)C(=O)NCC12CC=CC(C1)OC2 C1(CC)(CC)CC(O)CN1C(=O)CC(O)CNC(=O)CCN(C)CCO Cc1cnncc1C(=O)NCCC1CSCCN1C(c1cc(Cl)ccn1)=O C1(C(=O)NC(CNC(c2c(CC)nc(C)o2)=O)CO)CC2(CO1)CC(F)(F)C2 n1(CC(=O)NC2CN(C(C3ON=C(C)C3)=O)CC(O)C2)c([N+](=O)[O-])cnc1C Cc1c(C(N2CCC(C)N(C(=O)C(F)C(C)C)CC2)=O)oc2c(Cl)cccc12 c1(OC(CC)C)ccccc1C(N1CCC(CNC(c2cc(C)c(C)[nH]2)=O)C1)=O C1(C)(C(=O)NCC#CC(=O)NCCCCOC(C)C)CCCOC1 C(=O)(C(CCC1CC1)OC)N(C1CCN(C(=O)CN(C)C2CC2)C1)CC#C N1(C(c2nc(OCC)sn2)=O)CCC(NC(=O)CC(C)(C)O)CC1C N1(C(CCC2C(C)C2)=O)CCC(O)(CNC(c2cnc(C3CC3)[nH]2)=O)C1 CC(F)(F)C(F)C(=O)N1CCCC1CCNC(C1(C)CCCNC1=O)=O N1(C(C(COCC)n2cc(-c3csc(C)c3)nn2)=O)CC2COCC2(C)C1 c1(C(N(C)CC2CCN(C(COC(C)=O)=O)C2)=O)cc([N+](=O)[O-])c2nsnc2c1 N1(C(c2c(N)ccc(C)c2)=O)CCCC2(CC(NC(C3CC(Cl)(Cl)C3)=O)CO2)C1 c1(NC(=O)OC(C)(C)C)ccc(C(=O)Nc2ccn(C3CCCCO3)n2)cc1I C12(C(N(CCCN(C)C(c3ccns3)=O)C)=O)CCC(CF)(C1)OC2 C(=O)(CC(C)CC(=O)NCC1(C(=O)N(C(C)C(C)SC)C)CCC1)OC CCC(C)C(O)CC(=O)N(CC)CC1(O)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 S(=O)(=O)(c1ccc(NCCC2CCC2)c(C#N)c1)N1CC(C)CC(C(=O)NC)C1 N1(C(C(C(CC)C)N(C)C(c2cnncc2O)=O)=O)CCCN(CC)C(=O)C1 Cc1cc(C(F)(F)F)nc(C(=O)NC2CCC(NC(C3CC=CCC3)=O)CC2)n1 C1(C2CN(C(C3CCCSC3)=O)C2)(Nc2cc(OCC)ncn2)CC1 N1(C(C2CC(CC)N(C(c3cc(C)nc(C)n3)=O)CC2)=O)CCC12CCCSC2 c1(C(N2CC3CC(NC(C(=O)NC4CC4)=O)C3C2)=O)cnc2c(c1)CCCC2 C1(OC)CCCN(C(=NCCC(=O)Nc2ccccc2)NCC(F)F)C1 CC(CC(N)=O)C(=O)N(C1CCCN(C(=O)CN2CCCNC2=O)C1)CCF c1(CNC2OCCCN(C(C(=O)NCc3cnn(C)n3)=O)C2)ccc2[nH]ccc2c1 C1(NC(c2cccc(C)n2)=O)CCN(C(=O)CC2CCC(C)(C)CO2)CC1C CC(C(F)C(=O)NC(C1CCCC1)CNC(=O)C1=CSCS1)C(F)(F)F c1(C(N(CC(N2CC(O)(C(C)NC(c3csnn3)=O)C2)=O)C)=O)ccc(Cl)cc1 c1(C(N2CCC(C)C2CNC(=O)COC(F)F)=O)cc(O)cc(Br)c1 C=CCC(C(=O)N1CCC(C(N2CCOC(C(C)(C)C)C2)=O)CC1)C(C)C c1(CCC(N2CCCC(CN(C(C(C)c3cc[nH]n3)=O)CC)C2)=O)cccc(O)c1F c1(CC(N2CCC(C(CNC(C(CC)O)=O)F)CC2)=O)ccc(O)c(C(N)=O)c1 N1(C(CCCn2cc(C(N3CCNC3=O)C)nn2)=O)CCC(C)(CC#N)C1 c1(C(C)(F)F)n[nH]cc1C(N1CC(CCNC(=O)CN2CCCCC2)C1)=O S(=O)(=O)(c1ccc(C(=O)O)c(F)c1)Nc1cccc(N(C)C)c1 c1(C(=O)NC2(C3N(C(C4C(C=C)CC4)=O)CCCC3)CC2)ccc(Cl)c(OC)c1 C1(OC)Cc2cc(F)ccc2N(C(C2CC3C=CC2C3)=O)C1 c1(CNc2ccc(C(N3C(C(=O)OC)CCCC3)=O)cc2)ccnc(Cl)c1Br N1(C(c2ccc(SCC)c(N)c2)=O)CCC(C2CC2)C1CNC(c1nccs1)=O C1(CC(=O)NCC(c2ccc(F)cc2)OC)CN(C(C2CCCC2)=O)CCO1 Cc1cc(C(=O)NCC(C2CC2)NC(=O)C(C)(F)c2ccon2)c(F)cc1N Cc1c(C(=O)N(CCN(C(=O)C(C)O)C)C(C)C)noc1C1CC1.C1CC1 c1(CC(C)C)cc(C(=O)NC(C)C(C)NC(c2ccco2)=O)ccc1N.C1CC1 CCCC(CCC)C(=O)NCCC(O)CNC(c1cc(Cl)nc(Cl)c1)=O c1(C(=O)NCC(c2cccc(OC)c2)C)cnn2c1SCC2 CCC(C(=O)NC(C)(C)CC(=O)NC(C)CCC1CCCC1)C(C)C C1(C(=O)NCCc2ncc(C)o2)N(C(=O)Cc2cnoc2)CCCC1(C)C CC1CN(C(=O)C(C)C(C)O)CC(C)N(C(=O)C=Cc2ccccn2)C1 C1(NC(=O)OC(C)(C)C)CC2C=CC1N(C(=O)CCCCF)C2 C(C)(CC(C)NC(c1cn(-c2ccn(C)n2)cn1)=O)NC(C=C(C)C(C)C)=O C1(CNC(Cc2cc(C)sc2)=O)(CO)CCCN(C(=O)CCc2ccon2)C1 c1(C(=O)NCc2cc(C(NOCC#C)=O)n[nH]2)oc(C)cc1C C(=O)(C1=NOC2COCC12)NCC1CC(Nc2ncnc(OC)c2OC)C1 c1(C(=O)NCC2C=CCN2C(=O)CCC2CC2(F)F)ccc2ccoc2c1 C1(C(N(CCNC(c2cnc(NC(C)=O)o2)=O)C)=O)Cc2nn[nH]c2C(C)C1 Cc1ccc2cc(C(=O)NC3CCC(N(C(=O)C(C(C)C)C(C)C)C)C3)[nH]c2c1 C1(C(N2CCCC2C2CCN(C(c3cccnc3)=O)C2)=O)(C(F)F)CCCCC1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(C(C)NC(=O)C2=NOC(C)C2)OCC1 N1(C(CCCOCCC)=O)CC(CNC(c2oc(C3CC3)nc2C)=O)CC1C CC1CC2CCC(C(=O)NC3CCN(C(=O)C(C)(C)O)CC3F)CN2C1 C1(C(N(C)CC2(CNC(c3nncc(OC)c3)=O)CC2)=O)CN2CCN1CC2C c1(C(C)CC(=O)NCCCOC(F)(F)F)ccc(OC(C2CCCNC2)=O)cc1 C1(C(=O)NCCCCNC(c2cnc(C3CC3)s2)=O)CC1C1CCCCC1 Cc1cc(F)cc(C)c1C(N1CCC(CF)(NC(C2CC(=O)N(O)C2)=O)C1)=O c1(OC)ccc(Cl)cc1CC(=O)NCC12CC(CN1C(C1(C)CNC(=O)C1)=O)C2 CN1CC(C)(C)CC1C(=O)NCC1CCN(C(=O)CCc2ccnn2C)CC1 C1(C(N(CCCCCNC(C(Cc2c(C)nc[nH]2)O)=O)C)=O)CC12CCCC2 c12ccccc1CNc1csc(n1)C2.S(=O)(=O)(CCc1ccon1)N(C)C CCCCCCCNC(=O)COC1CCN(C(C2CN(C(C)C)C2)=O)CC1 c1(CC)n[nH]cc1CNC(=O)C(C)NC(c1csnc1OC)=O C=CC1CN(C(=O)C(C)CNC(=O)CCC(C)N(C)C)CC1O C1(C(=O)O)CC(C2CCC2)CN1S(=O)(=O)c1cnn(C2CCC2)c1 Cc1cn2cc(CC(=O)NOCc3cn(C4COCC4O)nn3)nc2s1 C1(C(=O)NC(C(=O)NC)CC2CC2)CCN(C(=O)C2CC3(CCC3O)C2)O1 CC12CN(C(CC(=O)OC)=O)CC(CNc3nc(C4CC4)ncc3C#N)(C1)C2 C1(OCC)CC2(C1)CC2C(=O)NC1CCN(C(=O)CC2(OCC)CCCCC2)C1 CC1(C)CN(C(c2cccnc2)=O)C(CNC(c2nc(Cl)sc2Cl)=O)CO1 CC(C)CCCCN(C)C(C1(NC(=O)Cc2ccc(O)nc2)CSC1)=O c1(CNC(C=C)Cc2ccc(F)cc2)cc2n(n1)CCCCO2 N1(C(=O)C2CC2)CCC2(CCCN2C(c2c(Cl)csc2Cl)=O)C1 c1(C(=O)NCC2OCC(C(=O)NCc3cc(C)n(C)n3)C2)ccnc(C)c1C C1(CNC(C(CCC)C)=O)(OC)CCN(C(c2cnc(O)cc2OC)=O)CC1 CCC(C(O)C(F)F)NC(=O)Cn1ncnc1C C1(C)(CNC(COC(C)(C)C)=O)CCN(C(=O)CCN2CCCCCC2)CC1 C1(CC(N2CC(C)(OCC)C2)=O)CN(C(C2CCC2)=O)CCO1 N1(c2c(F)ccc(C#N)c2)CCC2C(C1)NC(=O)N2C1CN(C(=O)NCCCl)C1 n1(CC(=O)NCC2(O)CN(C(C3C(C)CC=CC3)=O)C2)nc2c(n1)CCCC2 c1(CNC(C(C)N(CC)CC)=O)ccc(CN(C)C(C2CC2(F)Cl)=O)cc1 C1(CC(=O)NCC(C)NC(=O)C=CBr)CC(C)OC1C C1(C2CCN(C(=O)C=Cc3cccs3)C2)(NC(C2CC3CCCCC23)=O)CC1 C1(C(NOCC(CC)C)=O)CCOCCN1C(=O)C(C)NC(=O)CC c1(SCCC(=O)NC2CN(C(CCCCSC)=O)CC2O)ncnc2[nH]cnc12 N1(C(CN(C(C)C)C)=O)CCCC(N2CCN(C(=O)CCC3CC3(F)F)CC2)C1 C#Cc1cccc(C(=O)NCC(C2CCOC2)NC(=O)C2=CC(C)(C)C2)c1Cl C=CC(CC)C(=O)NCC(C1CCC1)NC(c1cnn(C)c1)=O C(=O)(CC(C(F)F)C(C)(C)C)N1CCC(CNC(CCC=C)=O)C(F)(F)C1 CCC(F)(F)CC(=O)N1CCCN(CCNC(=O)CCC2CCCCO2)CC1 C1(CCN(C)C(=O)NC2CN(C3COC3)C2)CCOCC1 C1(C(CC)NCc2coc(-c3ccccc3F)n2)CCCCC1C N1(C(c2[nH]cc(S(N)(=O)=O)c2)=O)CCC2CCC(C1)N2C(=O)CC1CCOCC1 c1(C(=O)Nc2c(C)cc(NC(C3(Cl)CCC3)=O)cc2)ccn2ccnc2n1 C(=O)(CC1OCCc2ccccc21)N1C(CNC(c2nc(C)oc2)=O)CC2CC21 Cc1nc(CNC(C2CC2C)=O)oc1C(=O)NCCCCCCF CC1CC(=O)NC(C(=O)NCCCC(=O)NCC2CCC(C3CC3)O2)C1 c1(C(N2CCCC(CN(C(CC=C)=O)C)C2)=O)c(C)cc(OC)cc1F C1(CNC(c2ccc(NC)cn2)=O)COC(C)(C)CN1C(c1cccnc1S)=O C1(C(=O)NCC2(OCC)CN(C(C(CC=CCC)C)=O)C2)CC2C(C1)C2(C)C c1(CC)cc(C)ccc1C(=O)NCCC(C)N(C)C(c1cnc(Cl)c(N)c1)=O Cc1ncc(C=CC(=O)NC2CCCC2n2cc(C3CC3)nn2)s1 c1(C(=O)NCCC2CCN(C(c3ccc(C(C)C)o3)=O)C2)ccnc(C2CC2)c1 C1(CC(N2CC(F)(CC)C2)=O)CC(NC(=O)CN2CCNC2=O)C1(C)C C1(NC(c2cc(O)cc(Cl)c2Cl)=O)CN(C(=O)C#CC2CC2)CC1C1CC1 C1(COC)(CO)CCCN1C(=O)Cn1cc(C2CCCCC2)nn1.C(=O)(C(C)O)N C(=O)(C1=NOC(C)C1)N(CCCNC(c1sc(CC)c(C)c1)=O)CC1CCCC1 N1(C(C=CC(N)=O)=O)CCOCC1CN(C(c1cccc(-n2cnnn2)c1)=O)CC c1(COCC)noc(C)c1C(=O)NCC1(NC(C2CC(C#N)(CSC)C2)=O)CC1 c1(C(C(=O)NC(C)Cn2cc(C(C)(C)CO)nn2)N(C)C)ccc(F)c(F)c1 C1(C(=O)NC2(c3ncon3)CCCCC2)C2CC2C2CC12 N1(C(CC2(OC)CC2)=O)CCCC(CO)(NC(C2CCCC(C)(C)C2)=O)C1 c1(C(=O)NC(C)CCCCNC(c2nocc2Cl)=O)cn2ccnc2s1 N1(C(CCCCCCSC)=O)CC2CCCC(C1)N(C(=O)Cc1cc[nH]c1)C2 c1(CC(N2C(C(C)NC(CCNC(C)=O)=O)CCC2)=O)ccc2c(c1)CCCC2 C=CCC(C(=O)NC(C(=O)NCCc1csnn1)C1(C)CC1)C(C)C C1(C(=O)NCCC2CC(NC(=O)COC3CC(F)(F)C3)C2)Cc2ccccc2S1 C1(CNC(c2cnn[nH]2)=O)COC(CNC(c2nc(Br)c[nH]2)=O)C1 N(C(=NCCC(F)(F)F)NC1CCCCC1)Cc1cccc(N(C)C)c1 C1(CCC(C)(C)NC(CC(C)n2cccc2)=O)CCCCN1C(C1CCC1)=O N1(C(c2ncn(C)c2)=O)CCC(O)C1C(N1CCC1c1ccccc1)=O C=CCC(C)C(=O)NC(C)Cn1cc(CNC(c2csc(CC)n2)=O)nn1 c1(C(=O)NC2CN(C(c3c(OCC)nsc3)=O)CC2C)ccc(Br)c(C)c1F N1(C(CSCCC)=O)CC(CNC(c2c[nH]c(=N)cc2C)=O)C(C)(C)C1 C(=O)(C1CCCc2n[nH]cc21)N1CCCC(N(C(=O)C(F)(F)CN2CCCC2)C)C1 c1(C(N(C)Cc2ccc(CNC(=O)CC(C)(C)F)cc2)=O)cc2n(n1)CCO2 c1(OCC)cc[nH]c1CNCC1(CCO)CCOC1 N1(C(C(C)SCCCC)=O)CC(NC(c2cn(CCO)nn2)=O)C(CC)C1 N1(C(c2c(F)ccc(N)c2)=O)CC2(CCCC2NC(C2CCS2(=O)=O)=O)C1 Cc1ccnc(-c2cccc(NC(C3CCC3C(F)(F)F)=O)c2)n1 CCC(CC(=O)NCCCN(CCCCNC(c1cnn(C)c1Cl)=O)C)C1CC1 Cc1n[nH]c(C)c1C(=O)NC1CC(CCNC(C2C3CC4C(C3)C24)=O)C1 C1(c2nnc(C(C)C)o2)CNCCC1Nc1cccc(OCC(F)F)c1 c1(OC)csc(C(=O)NCCn2cc(CNC(=O)C(C3CC3)OC)nn2)c1 N1(C(CCN(C)C)=O)CCN(Cc2ccc(Br)cc2C(F)(F)F)CC1C#N C1(NC(c2c(OC)ccs2)=O)COCCC1NC(=O)C(C)CN(C)C CCC1=C(C(=O)NC2(C)CCN(C(C3(C)CC(F)C3)=O)CC2)CCCO1 C1(NC(CC)=O)CCC(C(=O)NCC(F)CNC(=O)CCOC2CC2)C1 C1(NC(CC(C(=O)O)NC)=O)CC2CCC(C1F)N2C(=O)OC(C)(C)C CC1CN(C(c2c(CNC(=O)C=CCF)nnn2C)=O)CCC1O CC(C)(C)CC(C(=O)NCc1ccc(CO)o1)NC(C1CCSC1)=O CC1(C(=O)NCC2COCC2NC(=O)CNC(c2ccccc2)=O)CCOCC1 CCC(C)(O)CCNC(=O)C(C1CCN(C(=O)Cc2ccnn2C)C1)C N1(C(c2c(C)nc[nH]2)=O)CC2(CC2)CC1C(N1CC2CC1CO2)=O c1(C(=O)NC(C)C(CO)NC(c2ccc(F)c(N)c2)=O)cc2c(cn1)OCCO2 c1(CC(=O)NC(C2CCN(C(c3cc(F)cs3)=O)C2)C)cc(Cl)ccc1O C1(C(=O)NC(c2cccc(F)c2F)C)CCN(C(=O)COCc2ccncc2)CC1C c1(C(=O)NCC2(NC(c3cc(F)cc(N)c3F)=O)CC2)cc2c(=O)[nH]ccn2n1 C1(C(=O)NCC(O)CC2CCCC2)(CC)CCN(C(C2CN(C(C)=O)C2)=O)C1 c1(CC(N2CCC(N(C(=O)CNC=O)CC)C2)=O)cc(C)nn1C N1(C(C2(COC)CCCO2)=O)CCC(N(C)C(c2ccc(C)cn2)=O)CC1 C1(NC(CN(C(=O)Cc2cncn2C)C(C)C)=O)CCCCC1C C(C)(CC(C)NC(=O)CC1(C2CC2)CC1)NC(C=CC(C)C)=O C(c1cncn1C)=CC(=O)N(C1CC(NC(CCc2onc(CSC)n2)=O)C1)C C(c1cn(C)cn1)=CC(N1CCC(C(=O)NCCCn2c(C)ncc2)C1)=O c1(C(N2CCC(CC=C)(NC(=O)C(C3CCC3)OC)C2)=O)ccc(C#C)cc1C c1(NC(C23C(CN(Cc4cn(CCC)nc4)C2)C3)=O)cnc(C(F)(F)F)cc1Cl c1(C(=O)NCC(C)(C2CC2)NC(C(CC=C)N(C)C)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(c2c(C)scc2)=O)C(C(N2CCOC(C(N)=O)C2)=O)CC2CC12 C1(NC(c2cc(SC)c(F)cc2)=O)CCC2CCN(C(=O)CC3(C)CCC3)C1C2 c1(OC)cc(COC(N2CCC(C(=O)NC(C)(C)C)C2)=O)ccc1OC CC(C(=O)NCC(F)CO)(C1CCC1)NC(=O)Cc1ccsc1 c1(CCC)cc(C(N2CCC(CCNC(=O)CSCC(C)C)C2)=O)c(C)o1 N1(C(=O)COC2CCOC2)CCC2(CC1)CCN(C(=O)Cc1ccc(Cl)nc1)C2 c1(C(=O)NC2CCC(C(=O)Nc3ccno3)C2)cc(Cl)cc([N+](=O)[O-])c1Cl C1(C(=O)NC2(CC=C)CCN(C(=O)CCC(C)(C)C)C2)CCn2nnnc2C1 c1(CN(C(C(C)N(C(=O)Cc2ccco2)C2CC2)=O)C)ccnn1C N1(C(c2c(C)c[nH]c2)=O)CC2CCC1CN2C(c1ccc2occc2n1)=O c1(OC)cccc(OC)c1-c1ncccc1C(=O)NCc1ccc(Br)nc1 C1(C(N(CC(O)C2CCC2)C)=O)CCCCCCN1C(=O)CCCNC(N)=O N1(c2nnc(C(=O)OCC)s2)CC(F)(F)CC1(C)CNC(=O)CSC(F)F c1(C(=O)NCC(CC(=O)NC(CCC)(C)CO)OC)coc2ccccc12 C1(NC(C(=O)N(C)C)=O)CC2CN(C(=O)C(C)(C)N3CCOCC3)CC2C1 N1(C(c2c(C)oc(CNC(=O)C3=NOC(C)C3)n2)=O)CC2C3C=CC(O3)C2C1 N1(c2ncc(OCCOC)cn2)CC2(CCCC2NC(c2nccnc2N)=O)C1 c1(NC(C)=O)ccccc1-c1cc(CN2CCCC2C(=O)NC2CC2(F)F)n[nH]1 c1(C(N2C(C(=O)NCC3C(C(C)C)C3)CSC2)=O)ccc(Br)cc1 c1(NC)ncccc1C(=O)NCC1C(CNC(C2CC(N(C)C)C2)=O)C1(F)F C1(N(C(C2C(C(=O)OC)C2)=O)CCO)CCN(C(=O)Cc2ccncc2F)CC1 c1(C(C)C)ncc(C(N2CC(O)(CCNC(=O)CCC3CCC(=O)N3)C2)=O)o1 c1(OC)cccc(F)c1CC(N1CCC(O)C(C(=O)NC2CCC2)C1)=O N1(C(=O)NC2CCN(CC(=O)N(CC)Cc3ccccc3)C2)CCSC(C)(C)C1 C(=O)(C(C)CCNCC(O)COC(C)(C)C)OC C1(NC(Cc2c(C)scc2)=O)CC=C(C(=O)N2CCCCC2CC(C)C)C1 CC1CN(C(C2(C3CC3)CC2)=O)CC(C)N(C(c2ccc(OC(F)F)cc2)=O)C1 CC(C(=O)N(C1CCN(C(C2CCC(F)CC2)=O)CC1)CCO)C(F)F c1(CN(C(c2ccccn2)C)C)ccc(S(=O)(=O)N2CCC(C(F)(F)F)C2)cn1 C#CCC(C)C(=O)N1CC2C(CN(C)C(c3ccncc3F)=O)C2C1 c1(C(=O)NCC2(CNC(C3C(CC)OCC3)=O)CCC2)cccc(C2CC2)n1 Cc1c(Cl)cc(C(=O)N(c2ncc3sccc3n2)C2CC(N)C2)cc1[N+](=O)[O-] Cc1cc2cccc(C(=O)NCC34CC3CN(C(C3CNC(=O)C3)=O)C4)c2[nH]1 Nc1ncc(C(F)(F)F)cc1C(=O)NCCCNC(=O)C(F)CC1CCCC1 C1(CC(=O)NCCC(C)(C)NC(Cc2c(C)cco2)=O)CCCC(=O)C1 NC(=O)CCCNC(N1CC(CC(=O)OCCCCCl)C1)=O Cc1cc(CCC(=O)NCC=CCNC(=O)COc2ccc(O)cc2)nn1C CC(CC(=O)NCC1CN(C(=O)CN2CCC(F)CC2)CC1C)C(F)F c1(C(=O)NC(C2(O)CCN(C(C3CCC(C)CC3)=O)C2)C)cnc2ccsc2c1 N1(C(C=C(C)C)=O)CCC(NC(=O)Cn2nnnc2-c2ccsc2)C(CO)C1 C1(C)(CC)CC(NC(c2nnn(C)c2N)=O)CN1C(c1ccc(OC)cn1)=O c1(-c2nc(C(CCCC)ON=C(C)C)n(C3CCOC3)n2)ccc(F)c(C)c1 C(CCCCC(=O)NCC=CCC(N1CCC(CN=[N+]=[N-])C1)=O)N(C)C c1(CNC(C2(C)COC2)=O)nocc1C(=O)NC1COC(C2CC2)C1 C(c1ccc(C(F)F)o1)=CC(N1C(CNC(C(C)C2CC2)=O)CCC1)=O c1(C(N(C(C(C)SC)C)C)=O)cccnc1CNC(C1CCOC1C1CC1)=O c1(C(N2CC=CC(NC(C3(COCC)CC3)=O)C2)=O)cc2ccc(C)cc2[nH]1 Cc1nc2n(c1C)CCN(C(=O)C(F)CC1CC(F)C1)C2 Cc1cc(C#N)sc1C(N1CC(F)(CNC(=O)C2=CCSC2)C1)=O N1(C(C(COCC)n2cc(-c3ncoc3C)nn2)=O)CC2(COC(C)C2)C1 c1(CCC)c(C(N2CC(NC(=O)C(C)O)C(C)C2)=O)cnn1-c1ccc(F)cc1 c1(SCC)nccnc1C(=O)N(CC)CC1CCCN1C(c1cnn(C)n1)=O C(CC(C(=O)NC1CC(NC(=O)CC2CS(=O)(=O)C2)C1)N(C)C)SC.C(C)N C(N=c1[nH]c(=N)[nH]c(=NCCCNC(=O)C2CC2)[nH]1)c1nn(C)c(Cl)c1 C(=O)(CCCCC#N)NCC(CN(C(C(c1ccc(C(F)(F)F)cc1)C)=O)C)O Cc1ncc(CCC(=O)OCC23CC(F)C2C3)o1 C(=O)(C(F)(F)CCn1ccnn1)NC(C(C)C)CNC(c1ccno1)=O N1(c2nc(SC)nc(N)c2)CCC2(CC1)CC2C(N1CCC(O)(C(N)=O)CC1)=O c1(C(C)=O)cc(C(=O)N(C2CCN(C(=O)CN3CCC(C)CC3)CC2)C)c(C)o1 C12(NC(c3c(CC)cno3)=O)CCCC1CN(C(c1scc(OC)c1OC)=O)C2 C1(C(N2CCOCC2c2cn(CCCCF)nn2)=O)CC(=O)C12CCCCC2 N1(C(C2(C)CC2)=O)CCC2(CC1)CC2CNC(=O)C(C)(C)C(F)c1ccccc1 N1(C(C2C3CN(C(C(C(CC)O)(F)F)=O)CC32)=O)CCCC(C2CCCCC2)C1 C1(CC(=O)NCC(=C)CCNC(c2c[nH]c(Br)c2)=O)CCC(C)(C)C1 CC1CN(C(=O)C(C)(F)C(C)(C)F)CCC1N=c1[nH]c(C(C)(C)C)nc(=N)[nH]1 C(C)(C)(C(O)C(F)F)NC(C1CC(CNC(c2cnn(C)c2N)=O)OC1)=O C(=O)(CC1OCCc2ccsc21)N1C(COC)(CNC(=O)C2=C(Cl)CC2)CCC1 N1(C(C=C(CC)CC)=O)CCOCC(C(=O)Nc2cn(CCF)nc2C)C1 N1(C(C)=O)CCC(C)(C(=O)N(C2CCN(C(=O)CC3(C#N)CCC3)CC2)CCO)C1 c1(C(=O)NC2CN(C(c3c(OC)ccs3)=O)C(C)C2)ccc(F)c2cnccc12 c1(C(=O)OC)ccc(NC(=O)CCCCNC(N)=O)cc1O C=C=C(C)CC(=O)N(C1CCN(C(=O)CN(C2CCS(=O)(=O)C2)C)CC1)C C(CNC(=O)C1=NNC(=O)CC1)(N=c1[nH]c(Cl)c(C#N)s1)C1CCC(C)CC1 C(C)(C(C)(C)CC)NC(C1(C(C)C)N(C(C(C)OCCCC)=O)CCC1)=O N1(C(CCSCCC)=O)CCC(O)(CNC(=O)C(c2cnn(C)c2)O)C1 O=C1CN(CCCN(C2CCCCC2)C(=O)C(=O)NC2CNCCO2)CCN1 c1(C(=O)NCC(C)(C)OC(=O)CNC2C(OC)(OC)CC2)cc(I)ccc1O C(=O)(C(F)(F)C(C)(C)O)NCC(COC)NC(c1ccc(C)c(C#N)c1)=O CC(C)CC(C)(C)C(=O)N1CCOC(CCNC(=O)C=CC(F)F)C1 C12(C(N(CCCCN(C(=O)CC3CCC(=O)N3)C)C)=O)CCC(C1)C2 O=C(CCCCC1CC1)NC1CC(CNC(=O)C(C2(O)CCCCC2)(F)F)C1 c1(C(=O)NCCNC(c2c(CCC)nco2)=O)ccc(=O)n(CCF)n1 C(=O)(C(C)(F)C(C)C)NCC(CCCC)NC(=O)C(CCC)N(C)C N(C1c2ccccc2CC1NC(=O)C=Cc1cscn1)C(CCC=C)=O C12(CNC(C(C=C)N(C)C)=O)CC(CO1)N(C(=O)C(C)CNC(=O)OC(C)(C)C)C2 c1(C(N2CC(C(N(CCCC=C)CC(=C)C)=O)OCC2)=O)ccc(C)nc1C CC(CCC(C)(C)C)C(=O)NC(C(=O)NCC#Cc1cccnc1)C(C)(C)C Cc1[nH]nc(C(N2CC(NC(=O)CCc3cncn3C)C(C)C2)=O)c1O N1(C(CCc2cc(C)no2)=O)CCC(NC(=O)CCC#N)C(C(C)C)C1 N1(C(CC2CC(CC)C2)=O)CCOCC1CN(C)C(c1nnsc1C)=O C1(CC=C)(CNC(=O)COC2CCOC2)CCCN1C(=O)C(COCC)N(C)C C1(CC(N2CC(OCC(C#C)C)C2)=O)CN(C(C)=O)CC12CC2 c1(CC)nnc(C)cc1C(N1CCN(C(=O)C#CC(C)C)C(CO)C1)=O C(=O)(CC(O)CC1CC1)NCC(C)NC(=O)COc1ccsn1 c1(C(=O)NC(C2C(C(=O)NC3(C(=O)NC)CC3)C2)C)coc(N(C)C)n1 CCCC(CCCNC(=O)CCNC(C)=O)NC(c1ccc(F)c(N)c1)=O C=CC(F)(F)C(=O)N(C)CC1CCCN1C(=O)CN(C)CCOC C(c1ccccc1Cl)=CC(=O)NC1C(NC(=O)C=CC2CCOC2)CCCC1 C1(NC(c2c(F)cccc2F)=O)CC2(CCN(C(C3C4CCN3CC4)=O)CC2)C1 Cc1cc(Br)cnc1C(N1CC(N(C)C(C2CC3(C2)CC(CO)C3)=O)C1)=O c1(OC)cc(C(N2CCOC(CCNC(C3CCC3)=O)C2)=O)cc(Br)c1O C(=O)(C(C)(Cc1ccccc1)C(C)C)NCCC1CCN(C(C(C)CF)=O)CC1 CCCCC(CC)CCC(=O)NCc1cccc(CNC(=O)CCC(CC)OC)c1 c1(C(N2CC(NC(C(C)OCC=C)=O)CC23CCC3)=O)cncc(P(C)(C)=O)c1 c1(C(=O)NC2(CN(C(c3cc(CC)c(C)o3)=O)C)CC2)ccc(Br)nc1N c1(C(=O)NC2CCN(C(CCCC(C)O)=O)C2)cc(S(N)(=O)=O)co1 C(C(=O)N1CC(NC(C2CC3(CC3)C2)=O)C1)(C(C)C)NC(=O)OCC C1(C(=O)Nc2cnc(C)nc2)CCCC12CCN(S(=O)(=O)c1ccccc1Cl)C2 CC1CN(C(C2CCN(C(=O)Cc3ccsc3)CC2)=O)CC(=O)N1 C(=O)(N1OC2C=CC1CC2)C1CC(C)N1C(c1cnc(O)c(F)c1)=O C1(CNC(Cc2ncc(C)o2)=O)CCN(C(C2CCCC2C)=O)CC1 CCCCCCCCC(C)C(=O)NC(C)(CNC(c1cnnn1C(C)C)=O)CC c1(OC)cccc2c(C(=O)NCCOCCNC(C3COC(=O)C3)=O)coc12 C=CCC(C(=O)N1CC(CNC(C2CNC(=O)O2)=O)C1)OC N1(C(c2c(NC)nccc2)=O)CCC(C)(C(=O)NC(C)COC(F)(F)F)CC1 CN1CC(=O)N(CCCC(=O)NC2CN(C(=O)CCc3cnc(O)[nH]3)C2)C1=O Cc1ccc(C(=O)NC(CNC(c2ccc(C(O)CF)cc2)=O)CC(C)C)cc1 C1(CCNC(c2ccn(CCOC)n2)=O)CN(C(=O)Cc2cnns2)CC(C)O1 C12(C(c3nnnn3C3CCOCC3)NCC(C)OCCO)CCC(CC1)OC2 N1(C(CSC)=O)CCCCC2(CCN(C(C34CC5CC3(CSC)CC5C4)=O)C2)C1 C1(NC(CC2(C=C)CCC2)=O)CN(C(C2(C(C)C)COC2)=O)Cc2nccn2C1 c1(CNC(C(=O)N(C)CC2CCCCO2)=O)sc(Cl)cc1Br N1(C(COCCCCC)=O)CCC(C)(CNC(c2c(CC)nnn2C)=O)CC1 C1(NC(=O)CNC(=O)C(F)(F)F)CCCCCN(C(c2ccc(F)o2)=O)C1 C1(COC)(NC(=O)C=C2CCCCC2)CCN(C(C2(C3CCCO3)CC2)=O)CC1 N1(C(C(CCN(C)C)N(C)C)=O)CC2CCN(C(c3ccsc3Cl)=O)CC2C1 c1(CC)ccc(C(N2CC(NC(=O)C=CCO)CC2(C)C)=O)cc1F CC(Cn1ccnc1)C(=O)NCCN(C1CCCC1)C(=O)CC1CCCO1 C1(NC(COCCOCC)=O)CC2CCC1CN2C(c1cccc(CSC)c1Cl)=O N1(C(CN)=O)CCC2C(C1)OCCN2C(C1CC(O)C1)=O CCC(CCOC)C(=O)NCC1(F)CC(NC(=O)Cc2ccsc2)C1 c1(N2CCC(=CC(=O)NC3CCCCC3)CC2)cccc([N+](=O)[O-])c1 C(C(C(=O)NOCCCC1CC1)C(C)(C)C)NC(C(CC)n1ccnc1)=O C1(CNC(C(CO)N(C)C)=O)CC2CCC1N(C(=O)C=Cc1cccc(O)c1)C2 c1(N2CCOCC(NC(C(CCSC)O)=O)C2)ccn2c(Br)cnc2n1 C(=O)(C(C)(C)C1=CCN(C(=O)C2=C(Cl)CCCC2)C1)NC1C(O)CCN(C)C1 C12CCN(CC1)c1ccnc(n1)C2.C1(C(C)(C)C)COC(C(=O)O)C1 Cc1cc(C(N2CC(CNC(=O)Cn3c(C)ccc3C)C(C)C2)=O)c(Cl)cc1F CC(N=c1[nH]c(=NC(C)c2ccc3nc(O)[nH]c3c2)c2[nH]ccc2[nH]1)C1CCC1 C(CN=c1[nH]c(C)nc(C)c1F)(C1(c2ccccc2)CC1)Nc1ccn(CC)n1 c1(N2CCC(OC(F)F)C2)nccc(-c2ccccc2)n1 Cc1cc(C)c(CNCC2CCCCN2C(c2cc(F)c[nH]2)=O)c(C)c1 c1(C(=O)NC2(C)CC(NC(C(CCC)OCC)=O)C2)c(F)cncc1Cl C=CCC(C)(CC)C(=O)NC1CC(C(=O)NC2CC3C=CCC(C2)C3)C1 CC1(C)CC(NC(=O)Cn2cc(C(F)(F)F)cn2)CN1C(=O)C#CC(=O)N(C)C Cc1c(Br)ccnc1C(N1CCN(C)CC1CNC(=O)COCC(F)F)=O C1(NC(C2C=CC(NC(=O)CCCCN3CCCC3)C2)=O)CC12CCCCCC2 N1(C(C2(OC)CCS(=O)(=O)C2)=O)CCC(C2(NC(C3CC(F)C3)=O)CC2)C1 N1(C(C(CC(F)F)NC(C=CC2(C)COC2)=O)=O)CC(O)C2(CCCC2)C1 C1(C)(C(N2CCC(N(C(=O)CC(C)C)CC#C)CC2)=O)CCC(C)(C)CC1 c1(CN2CC(CNC(C34CC(CF)(C3)C4)=O)C2)cc(OC(F)(F)F)cc(Cl)c1 Cc1nc(C(=O)NC2CN(Cc3ncccc3O)CC2F)ccc1F c1(C(=O)NCCC(C)N(C)C(C2(CCF)CCC2)=O)ccc(-c2cnn(C)c2)o1 CC(C)C(CCN(C)C(=O)Nc1cc(C2CCOCC2)no1)N(C)C c1(OC)ncc(Cl)c(=NC2CCCC23CN(C(=O)Cc2csnn2)C3)[nH]1 C1(CC(=O)NCc2c(C)c[nH]n2)COCCN1C(C1C=CCCC1)=O N1(C(Cc2c(C)noc2)=O)C2CCC1C(C)C(NC(C1(F)CCS(=O)(=O)C1)=O)C2 Cc1cc(Cl)c(C(N2CC3CCCC3(NC(C3CC3C(C)(F)F)=O)C2)=O)cc1F N1(C(C2C(NC(C(C)c3cccs3)=O)C2(C)C)=O)CCC(C2(C)CC2)C1 C#CC1(C(=O)N(C(CO)C(C)C)C)CCN(C(c2oc(C)nc2C)=O)C1 c1(C(=O)NC2CCN(C(C3C(OC)(OC)CC3)=O)C2)cnc2nccn2c1.C(C)(=O)N N1(c2n(CC)c(CCc3ccc(-c4nc[nH]n4)cc3)nn2)CC(C)CC(C)C1 C1(C(=O)NC)CCC(NC(C2CC(N)CN2C)=O)CC1 Cn1c(O)nc2cc3ccc2cccc1C1(CCC1C)C(=O)N1C(CC1)CNC3=O N1(C(CC(CC)CC)=O)CCN(C(=O)CSCCN(C)C)CC(O)C1 N1(C(CC(CCSC)O)=O)CC2CC3CC2C1C3NC(c1cocn1)=O N1(C(C(C(CC)O)C)=O)CC2CCC1CN2C(c1sc(F)cc1Cl)=O CC1CC(CNC(c2ccc(C(F)(F)F)nc2)=O)CN1C(c1ccc(O)cn1)=O N1(C(CC2(C)CCN2C(=O)C=Cc2cocn2)=O)CC2C(C1)C2(F)F C1(NC(C2(C(N(CCC#C)CCO)=O)CC2)=O)CN(C(C)C)CC1C C1(N(C(CSCCN(C)C)=O)C)CCCN(C(=O)Cn2cc([N+](=O)[O-])cn2)CC1 C1(Cc2onc(C3(COC)CCCC3)n2)CC(N)CC(C)(C)C1 C(=O)(CC(C)(C)C#N)N(C(C)C(=O)NC1(C)CC(F)(F)C1)C CN=c1[nH]c(SC)ncc1CN1CC2CC1C2C(N1CCC(CC#N)CC1)=O c1(C(N2C3CN(C(c4c[nH]c(=NC)o4)=O)C(CC3)C2)=O)cc2nn[nH]c2cc1F C(=O)(C(O)CC(F)F)NCC(c1cccc(Cl)c1)NC(CN(C)CC)=O C1(COC)(NC(C2COCC(C)(C)O2)=O)CCCN(C(c2ccco2)=O)C1 c1(CCC(=O)NC2C(NC(Cc3nc(CC)sc3)=O)CC2)cnn(C)c1C N1(C(C2N(C(c3c(OC)cccc3Br)=O)CC(C)C2)=O)CCCC2(CCOC2)C1 C1(C(N2CCC(C(C)C)C2)=O)CCCCN(C(=O)Cn2cncn2)C1 c1(NC(C2C(NC(c3ccc(C)cc3Br)=O)C2)=O)ccc(Br)c(F)c1CO N1(C(c2sccc2C(=O)C(F)(F)F)=O)CC2(CCCCC2)CC1CO C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CCN(C(CCSCC)=O)C12CC2 Cc1cccc(OCCC(=O)N2CC(CC(C)(C)CNC(=O)CCC=CBr)C2)c1 c1(C(=O)NC2COCCN(C(C3C(C)C3)=O)C2)nn(C)c2ccccc12 C1(CNC(CC(CC)C)=O)CC12CCN(C(c1cc(C(C)(C)C)oc1C)=O)CC2 N1(c2nnc(CCC)s2)CCC(O)(C2(C(=O)O)CCC2)CC1 C1(NC(COC(C)=O)=O)CCCC1(C)NC(=O)CCOCC(F)F c1(OC)ccc(-c2nc(CP(C)(C)=O)n(CC3COC(C)(C)C3)n2)nc1 C1(C(=O)NC(C)CCO)N(C(c2cccc(F)c2F)=O)CCC1(C)C Cc1ccc2nc(N3CCCC(C(F)(F)F)C3C)[nH]c2c1 C1(NC(CCC(=O)NCCC)=O)CC2CCC(C1C)N2C(c1csnn1)=O C1(N(C(=O)C=Cc2ccc(Cl)s2)C)CCCN(C(=O)C(O)C(F)(F)F)CC1 C1(C(=O)NC2C(C)N(C(=O)C=Cc3cnccc3Cl)CC2)CCc2nccn2C1 CP(C)(=O)CCCNC(C1CC(F)CN1C(C1CN(C(N)=O)C1)=O)=O CC1CN(C(=O)CN2CC3CC3C2)CC1(C)C(=O)NCCC=C1CCC(C)CC1 Cn1cc(C(F)(F)F)cc1C(N(C1CCN(Cc2ccccc2)C1)C)=O c1(CC)ccc(NC(C2CC2)=O)cc1Br.C1(CNC(C2(C)CC2)=O)CC(C)=NO1 N#Cc1ccnc(NCC(C2CCCCC2)NC(C2CC(C3CC3)=NO2)=O)n1 C12(NC(CCCC=C)=O)CCCCC1CN(C(c1nccc(OC)c1F)=O)C2 N1(C(=O)OCC)CC(NC(=O)CC(O)CN(C)C)C(C(F)(F)F)C1 C1(C(N(CCCCC=C)C)=O)CCCCC1NC(=O)Cc1scnc1C c1(OC)cccc(CCC(=O)NCC(O)CCNC(c2sncc2C)=O)n1 c1(C(=O)NCCC2CC(OC)CN2C(=O)Cc2cn[nH]c2)ccn(C)c(=O)c1 N1(C(c2cc(C)nnc2C)=O)CCN(C)CC(C)C1 C1(Cn2cc(CNS(C)(=O)=O)nn2)CC2CCCCC2N1C(c1ccoc1Br)=O C12(CNC(C=COCC)=O)CCCC1N(C(c1ccc(CO)cc1F)=O)CCC2 c1(CC)ncc(C(=O)NCC2CN(C(C3CCN(C)C(C)C3)=O)CCO2)c(O)n1 c1(N2CCC(C)C(CO)C2)nc(=NCC(C)c2nncn2C)[nH]c2ccsc12 C1(CC(=O)NCCNC(c2sc(C(=O)OC)c(C)c2)=O)CC(C)(C)CCO1 C1(NC(CCC=CCC=C)=O)CC2(C(=O)NC3CCN(CC)C3)COC1C2 C(CCCC(=O)NCC1CC2CC2N1C(C1CC1c1ccccc1Cl)=O)SC C1(C(=O)NC(C)CN(C)C(c2ccc(CF)cc2)=O)CC2OC1C1CC21 N1(C(C2(c3ccccc3)CCC2)=O)CCOC(C(O)CO)C1 c1(NC(C(CC2CCCC2)NC(c2ccn(CC)n2)=O)=O)cc(C)c(C)c(C)c1 Cc1ccc(C(=O)NC2(CCO)CN(C(=O)C(C(C)C)N(C)C3CC3)C2)nc1 CC1CC(NC(c2cc(N)nc(Cl)c2)=O)CCN1C(C1CC2C=CC1CC2)=O c1(C(=O)NCC2C3CN(C(=O)CC4CCOC4)CC23)cc(Br)cc2nc[nH]c12 c1(C(N2CC(CC=C)(NC(=O)CCc3ccccn3)C2)=O)c(C)nsc1NCC CC(C)(C)CC(C(=O)Nc1cnccc1OCF)NC(C1C2CC3C(C2)C13)=O CCC(=O)CCC(=O)NCC(C(=O)NCC(CC)CCOC)C(C)C c1(C(C2CCCCC2)C(=O)N(CCC(=O)OCC)C2CC2)ccc(F)cc1 N1(C(CCCN2CCN(C=O)CC2)=O)CCN(C(C2CCC2F)=O)CC1.CC(=O)O c1(OC)cccc(Cl)c1C(N1CCCC(C)(NC(=O)C(O)CSC)C1)=O C1(CC(=O)NC2(CC)CC2)CN(C(c2csc(O)n2)=O)CC1C N1(C(C2N(C)CCC2)=O)CCCC1(C)C(N1CCC1CC(C)(C)C)=O C1(C(=O)NCC(CC(C)C)NC(C2N(CC)CCOC2)=O)CNC(=O)CC1C C(C)(C(CC(=O)NCc1ccc(F)c(F)c1)NC(=O)C(C)(C)CCF)OC C(CCCCO)N(C)C(C1(CNC(=O)CC2C=CCC2)CCCO1)=O C1(C)(CNC(C2(C(=O)OCC)CC=CC2)=O)CCCN(C(=O)C(C)CN(C)C)C1 CC(C)CC(C)C(=O)NC(Cc1ccco1)C(=O)Nc1ccc(O)cc1 CC(C)CCCC(C)C(=O)NC1CC(NC(c2cc(O)nc(O)n2)=O)CC1O c1(C(N2CCC(OC)(CNC(C3NC(=O)CC3C)=O)C2)=O)cc2c[nH]cnc-2n1 Cc1cc(C(=O)NC2CCC(N(C)C(c3cscc3C)=O)C2)c(C)s1 c1(C(=O)NCC2(CNC(c3c(CC)ocn3)=O)CCCC2)ccc(C(F)F)cc1 N1(C(C(N2CCOCC2)C)=O)CC(NC(=O)CC2(C3CC3)CC2)C(O)C1 N1(C(C2(C)COC2)=O)CCC(CCC(N2CCC(N3CCOCC3)C2)=O)C1 c1(C(N2CCC(C)(C(=O)NCC3(C)CCCC3)C2)=O)n[nH]cc1[N+](=O)[O-] C1(CCC)CN(C(=O)C=C2CCCCC2)CCN1C(=O)NC12COCC(C1)OC2 c1(CC)[nH]nc(C(N2CCN(C(=O)CC(C)(C)COC)CC2C)=O)c1[N+](=O)[O-] C1(CC(=O)NC2C=CCN(C(CNS(NC)(=O)=O)=O)C2)COC(C)(C)CO1 c1(C(=O)OC)cnc(NCCCOCCCNC(C2(F)CC=CC2)=O)cn1 C1(C(=O)NCC(CNC(C=CCCC)=O)F)CC(c2ccccc2[N+](=O)[O-])=NO1 c1(OC)cccc(C2(NC(=O)NCC(C3CCC(OC)CC3)OC)CCC2)n1 N1(C(C(CC#C)O)=O)CCN(C(=O)C(c2ccc(F)cc2)(C)C)CCC1C C(=O)(C1=CC(O)CCC1)N1CCCC(NC(CCOc2ccc(OC)cc2)=O)C1 N1(C(c2c(C)n(C)nn2)=O)CCC(C(=O)NCC2CCCN(C)C2=O)CC1C c1(C(C)=O)ccc(=NCC2CCN(C(=O)COCc3nc(C)no3)C2)[nH]c1 c1(OC)cc(=O)n(C)cc1C(=O)NC(C)(C)CNC(C1CCN2CCOCC12)=O CC1CCc2[nH]nc(C(=O)NCC3CN(C(=O)C4=CCCO4)CC(C)(C)O3)c2C1 Cc1cc(C(N2CCN(C(=O)C(C#N)C(C)C)CC2C(C)(C)C)=O)nc(C)c1 Cn1nnc2cc(C(N3CCCOC(CCNC(C4CCOC4)=O)C3)=O)ccc12 O=S(=O)(c1ccc(N2CC3CCC(C2)O3)cc1Br)NC1CC2CCCCN2C1 c1(-c2cnc(C(=O)Nc3c(CC)n(C)nc3)nc2)ccc2c(c1)NCC(=O)N2 c1(CCC(=O)NC(C)CCN(C)C(c2cc(CO)[nH]n2)=O)nnc(S)nc1O c1(N2CCC(C)(CNC(=O)COC3CCOC3)CC2)nc(Cl)nc(C)c1[N+](=O)[O-] N1(C(C(CCC)N(C)C)=O)CCC(NC(c2ccc(F)c(C(C)C)c2)=O)CC1C C1(CC(=O)NC2(C(=O)NCC3(C(F)(F)F)CC3)CC2)CCCCC1 CCC(C)C(C)C(=O)NCC12CC1CN(C(=O)Cc1cccnc1C)C2 C12(NC(c3ccccn3)C)CCCC1CN(NCc1cc(C3CC3)no1)C2 c1(C(=O)NCC2(CCNC(C3C(C)C3)=O)CC2)ccc2c(c1)SCCN2 N1(C(c2[nH]cc(C)c2C)=O)CCC(NCC2CCC(F)(F)C2)C(C)C1 C1(NC(c2ccc(C(C)=O)[nH]2)=O)CN(C(=O)CCc2cccnc2Cl)CC1(C)C CCC(C)(C)C(C)NC(=O)CSc1cccs1 c1(CN2CC(F)CC(C(=O)NCc3ccn(CC)n3)C2)ccc(Br)c(Cl)c1Cl C(=O)(C1CCCc2cnc(C)nc21)NC(CC)CNC(c1cc(C)c(C)[nH]1)=O N1(C(CCCC(=O)OC)=O)CC2CC(C)N(C(=O)C(c3ccc(C)cc3)C)C2C1 C=C(C)C(CC(=O)NC1CCCC1CNC(=O)CN(c1ccncc1)C)OCC c1(C(N2C3CC(NC(COC(CC)(C)C)=O)C3CC2)=O)cc2cccc(O)c2[nH]1 c1(C(N2CCN(C(C=CC(C)(C)SC)=O)C(C(C)C)C2)=O)cccc2sccc12 C#CCCCC(=O)N(CC(=O)NCc1ncnn1C)C(C)C c1(NC(CCC)C)ccc(S(=O)(=O)NCCCn2cnnc2C)cc1Cl C1(CCC=C)(C(=O)NCCC(=O)OCC)CN(C(=O)CCc2cnn[nH]2)C1 C(C(C)CC(C)C)NC(C(COC(C)C)NC(=O)C(O)Cn1cncn1)=O N1(C(C(c2cncnc2)C)=O)CCCC(CCC(=O)NCC2(NC(N)=O)CC2)C1 c12c(F)ccc(c1F)CO2.c1(N(CCC)CCC)cc2nncn2cn1 C1(C(N(CCN(C(CC(C)OC)=O)C)C)=O)CN(S(C)(=O)=O)c2ccccc2O1 CCCCC(C)(F)C(=O)NCCCCC1CCN(C(C2CC2CC)=O)CC1 C1(CNC(C2CC(=C)C2)=O)CCCC(NC(c2csc(-c3cccnc3)n2)=O)C1 C1(NC(C(C)NC(C)=O)=O)C2CC3CN(C(=O)C(N4C(C)CCC4C)C)C1C3C2 c1(CNC(C)(C(C)CC)c2n(CCOCC)nnn2)c(C)c(C)cc(C)c1C c1(C(=O)NC2C(N(C)C(C3C=CCCC3)=O)CCCC2)ccc([N+](=O)[O-])cc1Cl N1(C(C2(OC)CCSC2)=O)C2CCC1C(CNC(=O)CC1(C)CCCO1)C2 C1(NC(Cc2c(C)nc[nH]2)=O)CCC(NC(c2coc(C3CCC3)n2)=O)CC1 c1(CCC(=O)NCC2CCCN2C(=O)CC2(O)CCCC2)ccc(Br)cc1F C(CS(=O)CC(F)(F)F)NC(C(C(=C)Cl)(C)C)=O CCS(=O)(=O)CC(=O)NCC1CCCC(NC(c2ccc(C(N)=O)[nH]2)=O)C1 C1(NC(CCc2cn(C)nn2)=O)CC2CCC1(NC(=O)C=Cc1ccc(Cl)s1)C2 CC1(C)CC(CNC(C2CCCO2)=O)CN(C(c2cnn(C(C)(C)C)c2)=O)C1 n1(CC)nc(C)c(CC(=O)N(CC(C)(C)C(=O)OC(C)(C)C)C)c1C N1(C(c2nncc(CCC)c2)=O)CC(NC(C2CNC(=O)C2)=O)CC(C)(C)C1 c1(C(=O)NC(C2CCCN(C(CCC(=C)C)=O)C2)C)cc2c(C)n[nH]c2cn1 c1(OC)ccc2c(C(=O)NC3CCCC3NC(C3CC34CCC4)=O)ccnc2c1 CC(C)C(CCC(=O)N1CC(N(C)C)C2(CC2)C1)NC(=O)C(F)n1ccnc1 c1(CCC)ccc(C(=O)NC23CC(NC(=O)C(C)SC)(C2)C3)cc1[N+](=O)[O-] C(=O)(CCC(=O)NC(C(C)NC(C1COCCO1)=O)C(C)C)OC N1(C(C(C)OCCC=C)=O)CCCC1CN(C(=O)CCNC(C)=O)C N1(C(c2c(OC)nn(C)c2)=O)CCC(NCc2nc(C(=O)O)n[nH]2)C(C)C1 C1(NC(C(C)CO)=O)CCN(C(=O)C(F)=C2CCCC2)C1C1CC1 C1(N2CCN(C(=O)C(C)C#N)CC2)(C(=O)NCC(C)(C2CC2)OC)CCCCC1 C1(F)(CNC(CC2CCCN(C(C(Br)=C(C)C)=O)C2)=O)CCC(C(=O)O)CC1 C1(CNC(CC(C)CNC(C2CC=CCC2)=O)=O)C2CCCCCC12 N1(C(Cn2ncc(C#C)c2)=O)CC(F)(F)CC1CCNC(=O)CCc1ccsc1 c1(C(N2CCCCC23CN(C(=O)C(F)(F)C2CC2)C3)=O)ccc2c(c1)COCC2 c1(SC)c[nH]c(C)c1CCC(=O)NC(CN(C(CCOC)=O)C)C.C=O C1(CNC(C(CC#C)O)=O)CC2CCCC2N1C(=O)CCCCc1cnc[nH]1 C12CCCC3(CN(C3)C1=O)O2.c1(C(C)C(=O)Nc2nn[nH]n2)cccc(Cl)c1 c1(C(N2C(CNC(c3c(CC)ocn3)=O)CC(OC)C2)=O)cc(C)cc(F)c1 CC1(C)CCC2(CC1)CC2C(=O)NCC1C2CN(C(c3cnccn3)=O)CC12 c1(C(=O)NCC2CN(C(=O)CC3CCCCO3)C2)cc2nc[nH]c2cc1[N+](=O)[O-] C(=O)(CC(C)N1CCCC1)NCC(C)N(C)C(C1C2CCCC12)=O CCC(C)CCCC(=O)NCCCN(CCCNC(=O)CCCCCNC(N)=O)C N1(C(C(=O)C2CC2)=O)CC2CCC(C1)N2Cc1ccc(F)c(C(=O)O)c1 c1(-c2nc(-c3scc(C)n3)nn2C)ccc(S(C)(=O)=O)c(-n2nc(C)cc2C)c1 c1(C(=O)NC(C(C)O)CO)cn2c(n1)CN(Cc1ccc(C3CC3)cn1)CC2 N1(C(c2[nH]cc(CC)c2)=O)CCC(C2CC2NC(=O)COCC2CCCO2)CC1 c1(C(=O)NCC2CCCN(C(c3cnc(OC)s3)=O)CC2)ccc2ncccn12 C1(NC(C2(C=C)CCC2)=O)CN(C(=O)CN2CCC2C)CC(C)(C)C1 c1(C(N(C)CC2OCCN(C(C=C(C)C(F)F)=O)C2)=O)cncc(S(N)(=O)=O)c1 C1(N(C(C(CC)OCC)=O)C)CCCCN(C(=O)Cc2cc[nH]c(=N)c2)C1 C1(CNC(C(N2CCOCC2)C)=O)C2CN(C(C3(CO)CCCO3)=O)CC12 C(=O)(C(CC)NC(=O)COc1ccccc1)N1C(NC(C=CC=C(C)C)=O)CC1 Cc1cnn(CC(=O)NCC2(O)CN(C(C3CCN3C(=O)OC(C)(C)C)=O)C2)c1 c1(C(N2C(C3(NC(C(C)=C(C)C)=O)CC3)CCC2)=O)c(Cl)ccc(C)c1O N1(C(C2C(C)CCO2)=O)CC2CCC(C1)N2C(C1CCC2CC1CO2)=O c1(OC2CC(N(C)C(=O)NC3COCC3(C)C)C2)cnn2ccccc12 c1(CCC(=O)NCC(C)N(C(=O)CCC2CCCN2C)C)cccc(Br)c1 n1(CCC(c2nnnn2CC(F)F)NCC(C)C)cc(-c2ccccc2)cn1 c1(C(=O)NC(C2CCOC2)CNC(c2cncs2)=O)c(Cl)ccc2c[nH]nc12 N1(CCNC(Cc2nc(CC)sc2)=O)CCCN(C(C2(C3CCC3)CC2)=O)CC1 C1(C(=O)NCCCN(C(C(C)N(CC(F)(F)F)C)=O)C2CC2)CC(S(C)(=O)=O)C1 c1(C(N(CCOCCCNC(C(C)OC)=O)C)=O)ccc(NC=O)cc1 C12(CNC(C(COCC)C)=O)CC(NC(c3ccsc3SC)=O)(C1)C(C)O2 CCC(C#N)(CC)C(=O)NCC1CN(C(c2ccc(CO)cn2)=O)C(C)(C)C1 C1(NC(c2c(CC)nco2)=O)(CNC(C2CCCCC2OC)=O)CCC(F)(F)CC1 C(=O)(C(CCC(C)C)NC(=O)CNC=O)NCC1C(C(=O)OC)C1 C1(C(=O)NC(C#CC)(C)C)CC=CCN1C(=O)CC(C)N(C)C N1(C(C(CN(C(CN(C)CC)=O)C)C)=O)CC2OC(=O)N(C)C2C1 N1(CCC)CCC(NCc2ccc(NC(C3CC3COC)=O)cc2)CC1 N1(Cc2ncc(C#N)cc2Cl)CC(C2CCCN(C(c3ccco3)=O)C2)C1 N1(C(=O)C=CCN2CCC2)CCC2CN(C(C3CC3(F)F)=O)CC2CC1 Cc1cc(C(=O)Nc2cccc(NC(=O)C(c3cccc(Cl)c3)O)c2)nc(O)n1 N1(C(C(C)N=[N+]=[N-])=O)CCC2(CCC(NC(=O)C=Cc3ccoc3)CC2)C1 c1(NCC)cccnc1C(N1CCCC1CN(C(C12CCCC1C2)=O)C1CC1)=O Cc1cc(CC(=O)NC(C(=O)N(C)C(C2CCCC2)C)C(C)O)n(C)n1 C(=O)(CS(=O)(=O)C1CC1)N1C2(CNC(CN(C3CCCC3)C)=O)CCC1CC2 C(CC(C)C)(C(=O)NCCOCCNC(=O)CC1CCCC1(F)F)NC(C)=O C12(C(N3CC4(CC(NC(CCC(CC)C)=O)C4)C3)=O)CCOC1CC(=O)NC2 c1(C(N2CCC(F)(CNC(C3(C)C=CCC3)=O)C2)=O)cc(F)ccc1O N1(C(CNC(C)=O)=O)CCCC2CN(C(c3cn4cccc(C)c4n3)=O)CCC12 n1(CNC(c2cc(C)sc2)=O)nnc(C(=O)NC2(c3cccs3)CC2)c1C C1(C(=O)NCCN(CCCN(C)C)C(=O)CN2CCC(C)(C)C2)CC1C1CCC1 C12(CNC(CC(C)NC(c3nc(CC)oc3)=O)=O)CCC(CC1)CC2 C1(NC(c2ncc(OC)cc2F)=O)CCN(C(=O)CC2CC=CC2)CC12CCC2 Cc1ncccc1C(N1CC(NC(=O)C(c2ccccc2)C2CC2)C(O)C1)=O C(=O)(C(C(=O)NC(CNC(=O)Cn1nccn1)C1CC1)C(C)C)OCC C1(C(N(CC(CCC=C)O)C)=O)CC(C)CCN1C(=O)C(C)N1CCCC1 N1(C(c2[nH]c(=NC)sc2)=O)CCC(NC(c2ccsn2)=O)C(C)C1 N1(C(C2ON=C(C)C2)=O)CC(NC(=O)Cn2cnc(C(N)=O)n2)CC(F)(F)C1 c1(CC)ccc(OCC(=O)N(CC(C)NC(=O)C(Cl)=CCl)CC)cc1 c1(C(=O)NCCC(C)NC(C2(C)CCCCC2)=O)n[nH]c2c1CCC2 c1(OC)cccc(Cl)c1C(=O)NCC1C2CC1N(C(=O)CC(C)C(F)F)C2 CC(CC(=O)N1CCC(Cn2cc[n+](C)c2)C1)CSC(F)F C1(CNC2CC(=C)C2)CCC(NC(=O)C(CCOC)OC)CC1 CN1CCC(C)(C(=O)NC2C3CC4C2C4C3C(=O)NCC2CCCC23CC3)CC1 CCC(CC)CC(=O)NC1CCN(C(=O)CCCOC(C)C)CC1F c1(OCC)ccc(C(=O)CCC(=O)NC(CNC(=O)C(O)CC)C(C)(C)C)cc1 c1(C(N(C2CC(NC(Cc3cn(C)nc3)=O)C2)C)=O)cc2nccnc2cc1F C1(C)(C(=O)NC(C)CN(C)C(c2ccco2)=O)CCCCC1(F)F N(C(=NC(C)C)NC1CC(S(C)(=O)=O)C1)C(C#C)CCC N1(C(C)=O)CCCCC1C(=O)N(C(=O)C=C(C)c1ccco1)CCNC=O C1(C(N2CCC(C(=O)NC)C2)=O)N(C(=O)C(C)C(O)C(C)C)CCCC1(C)C Cc1ccc(O)cc1C(=O)NC1C2CCCC12.n12cc(cn1)-c1cn(nn1)CC2 Cn1c(=O)oc2cc(-c3cc(CNC4CCCCc5ccccc54)c(=O)n(C)c3)ccc12 c1(N(CCCCC=C)C)cc(S(=O)(=O)N2CCCC(C(C)(F)F)C2)ccc1C#N N1(C(N(c2ncc(C(F)(F)F)s2)C(C)C2CC2)=O)CCOC(c2ccc(Br)s2)C1 CC1CCCCC1(CNC(c1ccc(F)s1)=O)NC(=O)CCn1cncn1 c1(CC(=O)NCCN(CCC)C(C2CCC3CC23)=O)csc(S)n1 C=C=CCC(=O)NCCCOCCNC(C1(C)CCCO1)=O N1(C(CCCOC(C)C)=O)CCCC(CN(C(=O)C=CS(C)=O)C)C1 N1(C(Cc2cc(C)on2)=O)CCN(C(c2cccn(C)c2=O)=O)C(C)C1 CC(C)CCCCC(=O)N1CCN(C(=O)CCCSc2ccccc2)CC1C c1(C(=O)NCCC(=C)CNC(=O)COC2CC2(F)F)cc(C)c(F)cc1F N1(CCN(C(C2(C)C(C)C2)=O)C)CCN(C(=O)COc2ccc(O)cc2)CC1 C1(NC(CNC(C)=O)=O)CCC(N(C(=O)CCCC2CCCO2)C)C1 CCCC(C)C(=O)NCCNC(=O)CCc1ccc(SC)cc1 c1(NC(C2NCCN(C(CCCC=C)=O)C2)=O)ccc(C(N)=S)cc1 C(C1CCCCc2ccccc21)NC(c1ccc(-c2cc(C)c(F)nc2)cc1)C c1(OCC)cc(OC)c(CO)cc1OC.C12(NC(c3sccc3OC)=O)CC(N)(C1)C2 CC1CCn2cc(C(=O)N(C3CN(C(c4cnc5nccn5c4)=O)C3)C)nc2C1 C1(Cn2cc(-c3ccc(C)s3)nn2)CCCN(C(=O)Cc2cnccc2C)C1 c1(CCC(N2CCN(CC(=O)C3(C(F)(F)F)CC3)CC2)=O)c(F)cccc1F O=C(C1=COCCC1)NCC1CN(C(=O)CNC(c2ccncc2)=O)CC1O c1(C(N(CCNC(C2(F)CC(C(=O)OCC)C2)=O)CC)=O)cccc(Cl)c1C c1(C2C(NCc3cccc(OC)c3)C2)c(Cl)cccc1Cl N1(C(C(C)NC(N)=O)=O)CCOCC1CNC(=O)C(F)(F)c1cncs1 C1(C(C)C)N(C(c2cc3c(s2)CCC3)=O)CC12CCN(C(=O)CCCF)CC2 C1(C(=O)NC2(CCNC(CC3(COC)CC3)=O)CC2)COCC1C(N)=O C#CC(C)(C)C(=O)NC(C1CCN(C(c2c(C(F)(F)F)ncn2O)=O)C1)(C)C c1(C(=O)NC(C)CCNC(C2CC(O)CN2C)=O)ccc2nc(O)n(C)c2c1 N1(C(CCC=CC)=O)CCN(C(=O)C(C)Sc2ccccn2)C(CC(=O)NC)C1 C1(C(=O)NC2(CNC(CCCNC(=O)OC)=O)CC2)CCC(=O)N(C)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1(C)CCCN(C(CSSC)=O)C1 N1(C(C(CC)OCC)=O)CCC(NC(=O)C(C)C2CCOC2)C(C)(C)C1 N1(C(CC2OCCN(C(c3c(C)snn3)=O)C2)=O)CC2CCC1C(O)C2O CC(CC(=O)NCC1CCCCN(C(=O)CS(C)(=O)=O)C1)CC(F)(F)F CC(CCCNC(=O)CSc1cn(C)nn1)NC(=O)CCC1CCCCO1 c12cc(C)ccc1C(=O)NCCCC(C)NC(=O)C(CC)S2.C=C1CC(SC)C1 CCN=c1[nH]cc(C(N2CC(NC(=O)CCNC(C3CCC3)=O)C2)=O)s1 C(CN=C(NCc1cc(C(C)(C)C)on1)NCC1CCC(=O)N1)SC Cc1cc(Br)c(C(N2CC(O)(c3cn(-c4ccccc4Br)nn3)C2)=O)s1 n1(C2CC(C(=O)NCC(N3CCSC3)C)C2)cc(C2CC2)nn1 N1(C(CC2(COC)CC2)=O)CC2C(NC(C3CCCOCC3)=O)CS(=O)(=O)C2C1 c1(C(=O)NCCNC(C2(C(F)(F)F)CC(F)C2)=O)cc2cc(F)c(F)cc2[nH]1 N1(c2nnn(C)n2)CCC(C2CC2)(CN(C(C2(C)CCS(=O)(=O)CC2)=O)CCO)C1 N1(C(C2(SC)CCC2)=O)CCC(C(C)NC(=O)CC2CC3(CC3)C2)C1 CCC(CC(=O)N1CC(OCCC(=O)NC2CCOCC2C)C1)C1CCC1 C(=O)(CCCC#N)N1CC(c2c(CNC(C3(C)C(C)(C)C3)=O)c[nH]n2)C1 N1(C(Cc2c(C)ccs2)=O)CCCC(O)(CNC(=O)CCCc2cnccn2)C1 C1(CC=C)(NC(=O)CN2CCC(C)CC2)CCCN(C(C)C(=O)NCC(C)C)C1 C#Cc1cccc(CCC(=O)N(C2CCN(C(=O)CCN(C)CC)C2)C)c1 C12(C(N(C)Cc3ncccn3)=O)CC(CO1)N(C(=O)Cn1ccnn1)C2 C1(CNC(CC(CCC)O)=O)CCC(C)(C)CN1c1nnc(-c2ccon2)s1 c1(OC)ccc(CNC2(n3cc(-c4nccn4C)nn3)CC2)cn1 c1(CC)conc1C(=O)N(C(C)(C(=O)NCC1(CC)CCCO1)C1CC1)C C(=O)(CC(C(C)(C)C)NC(C1CCC(=O)NC1)=O)NCC1(COC)CCCC1 C1(NC(CCC)=O)CC(CNC(c2cnccc2Cl)=O)C12CCC2 C1(C(N2CC(C(CC)CC)C2)=O)CCN(C(C)=O)C1 C1(NC(c2nn(CC)nc2C)=O)CCN(C(=O)CO)CCC1CO C1(NC(C(C)Cc2ccccc2Cl)=O)CC2(CCN(C(=O)Cn3ncnn3)C2)C1 c1(OC)cnc(Cl)cc1C(N1CCCC(C)C1CNC(c1c(C)nsc1N)=O)=O c1(CC(N2CC(N(C(=O)C=CCO)C)C2)=O)ccc(Cl)c(Cl)c1 c1(CC(=O)N(CCC(=O)NCCC2CCCS2)C2CC2)ccc(F)cc1 Cc1ccc(C(=O)NCC2CC3CCC2N3C(c2cnnn2C)=O)c([N+](=O)[O-])c1 C=CCN=C(NCC1(O)CCC(C)C1)N1CCC(O)CC2(CCCC2)C1 N1(CC(=O)N(S(C)(=O)=O)C)CCOC(c2cn(CC3CCCNC3)nn2)C1 C1(CC(N2C(CN(C(=O)C(C3CCOCC3)F)C)CCC2)=O)CC(=O)NC(=O)C1 Cc1ccccc1C(CF)NCc1csnc1C(F)(F)F C12(CC(N3C(CCNC(C)=O)CSCC3)=O)CNC(=O)C(C1)C2 N1(C(CC(C)F)=O)CCN(CCNC(=O)Cc2ccc(F)c(F)c2)C2(CCC2)C1 C1(CNC(COCCC=C)=O)CN(C(c2cc(C)oc2CC)=O)CC1C(F)(F)F CC(C)C(C)C(CNC(=O)C=CCO)NC(C1CC(n2cnnc2)C1)=O N12C=C(Br)CC(C1)C2.c1(NC)ccccc1C(N1CCCC1)=O C1(CNC(C=CC(CC)C)=O)CN(C(c2cc(Cl)ncc2O)=O)CCN1C Cc1cc(C(c2nnnn2CCOCC2CC2)NC2COCCOC2)nc(Cl)c1Br C1(OC)CN(C(C2CC2c2ccccc2C)=O)CC1NC(=O)CC(C)(C)O N1(C(C(OC)OC)=O)CC(CNC(=O)C(C)Cn2ccnc2)CC(C)(C)C1 CC(C)CC(C)CC(=O)NCC1CCN1C(c1ccc(CO)cn1)=O Cc1ccc(C)c(C(=O)NC2CC(F)CN(C(=O)Cn3cccnc3=O)C2)c1 CCCCCC(C)(C)CNC(C1OCCC1NC(=O)C(N1CCNC1=O)C)=O c1(-c2cccc(NC(N3CCN(CC)C(C)C3)=O)c2)cc2cccnc2nc1C N1(CC(=O)NCC2(O)CC(CNC(=O)C(F)CC3CCC3)C2)C(=O)CCC1=O C1(N(C(=O)CCC2CCCCN2C)C)CCCCN(C(C2CCC(F)CC2)=O)C1 C1(NC(=O)Cn2cccc2)CCC(C(N(CCCn2ccnc2)C)=O)CC1 Cc1cc(F)cnc1C(=O)NC(CC(N)=O)C(=O)NC(c1ncccn1)C C1(C(N(CC(N)=O)CC(N)=O)=O)CCN(C(=O)C2CC3(CC(=O)C3)C2)O1 c1(SCC)nc(N2CC3CC(C(F)(F)F)CC23)cc(C)n1 N1(C(Cc2nc(COC)sc2)=O)CC2CC1CCN2C(c1oncc1C)=O c1(OC)cc(SC)ccc1C(=O)NCC1CCC(CNC(=O)C(C)C(C)C)CC1 C(C(CC(=O)NC1CCOC1)C1CCC1)NC(c1c(CCC)[nH]cc1)=O CC1(C)CCN(C(c2ccc(=O)oc2)=O)CC1NC(C1CCCSC1)=O Cc1cccc(C(O)C(N2CCC(O)(C(C)NC(=O)C=Cc3ncc[nH]3)C2)=O)c1 C12(NC(=O)Nc3ncsc3CC3CC3)CC3CC(CC(C3)C1)C2 C(c1cccc(F)c1)=CC(=O)NCCC1(NC(C(CC)O)=O)CC1 c1(N(C)C)ccc(C(=O)NC2CCCC(N(C(=O)C=Cc3cn[nH]c3)C)C2)cc1 CC(C(=O)N1CC(O)(C2CCCN2C(C2CCOCC2)=O)C1)C(C)(C)C c1(C(N2C(C(=O)NC(CSC)C)COCC2)=O)ccc2cc(O)ccc2c1 C1(C(N2CCC(C(=O)NC)C2)=O)CC2(CCN(C(=O)CNc3ncccn3)C2)C1 c1(CNC(=O)COc2ccc(Cl)nc2)ncnc(C2CC2)c1Br N1(C(c2ccc(N(C)C)cn2)=O)CCN(Cc2ccc(Br)cn2)C2CC12 C1(NC(=O)Cc2ccccc2O)CCN(C(=O)CC2CCC(F)(F)CO2)C12CC2 c1(C(N(CC(CC)NC(c2sc(C)nc2C(C)(C)C)=O)C)=O)ccc(C)cc1 c1(CC)cc(C(=O)NC2CC(C(=O)NCc3cc(COC)on3)C2)n[nH]1 C1(CC(=O)NC)CN(C(=O)CCC(N)=O)CCN1C(c1cc(N)nc(Br)c1)=O C(=O)(CCC(C)N(CC(C)O)C)NCC=CCNC(COCC)=O CC(C)(F)CCC(=O)NC1(C(N2CCC(C(F)F)CC2)=O)CC1(C)C Cc1ccn(CC(N2CCC(C(C)(C)NC(c3ccc[n+]([O-])c3)=O)C2)=O)c(=O)c1 C(=O)(C1CCCn2ccnc21)NC(CC)CNC(=O)CC1CC(OC)C1 C(c1cccc(C)c1)=CC(=O)NC(CC)(C)CCNC(c1cncc(C)c1)=O CC1(C)CC(NC(c2[nH]ccc2C2CC2)=O)CN(C(c2cccc(=S)n2O)=O)C1 CC1CCC(C)(NC(C2(C)CCCN2C(=O)CN2CCC(=O)CC2)=O)C1 O=C1CC(=O)CC(C(=O)NC2(C(=O)NC3COCC3N(C)C)CCCC2)C1 Cc1cc(C(=O)NOC2CCC2OC(F)F)c(C)o1 N1(CC(C)C)CCCC1C(=O)N(C)CC1CN(C(C2(O)CCOC2)=O)C1 C1(CNC(CCC2(C)CC2)=O)CN(C(c2ccc3nccn3n2)=O)CC12CCC2 C1(NC(=NCC=C)NCC2(c3cccs3)CCCC2)COC2(CCOCC2)C1O C1(C(N(C2(C(N3CC(SC)C3)=O)CCC2)C2CC2)=O)CCOC(=O)CC1 C1(F)(N)CCS(=O)(=O)C1.Cc1ccccc1C(c1ccccc1Cl)n1cc(C2CC2)nn1 CC1=NOC(=O)C1CCC(=O)NCC(CNC(=O)CCc1ccccn1)CO C1(CNC(C(=Cc2cn[nH]c2)C)=O)CC(C)N(C(=O)CCc2ccccc2)C1 N1(S(CC2(NCc3cnc(C)s3)CCCC2)(=O)=O)CCN(S(C)(=O)=O)CC1.COC CCC(C(=O)NCc1nc(=O)o[nH]1)NC(=O)CCc1cncs1 N1(C(c2cncc(OCC)c2)=O)CCOCC(NC(c2cc(C(F)F)on2)=O)C1 C12(NC(C3CC(OC)C3)=O)COC(C1)C(NC(=O)C(C)c1ccsc1)C2 C(=O)(CCCCN(C)C)NCC(C)C(=O)NCC1CC1c1ccoc1 N1(Cc2ccc(OC)s2)C(=O)CCN(CCSc2ccnc(C(F)(F)F)c2)C1=O C12(COC(C3CN(c4ccc(Br)cc4)C3)=O)COC(CO)(C1)C2 C12(CO)CCN(CC1)C2.N1(C(C(c2ccccc2)N(C)C)=O)CC2C=CC1C2 C#Cc1cc(C(N2C3CCC2CC(NC(C2(O)CC2)=O)C3)=O)cc(F)c1 c1(N(CC=C)CC2CC2)ccnc(SC)n1 N1(C(C=CC=CCC)=O)CC(CC(=O)N(c2ccc(Cl)cc2)CC)CC1C C(=O)(CCCc1csc(=N)[nH]1)NCC(C)CNC(C1C(C)C1(F)F)=O C1(C(C)OC)CCN(C(=O)CN(C2CCCCC2)C(=O)CSC(C)C)C1 C1(O)(CNC(C(C)OCC(F)(F)F)=O)CCCN(C(=O)C2=CCCCO2)C1 c1(C(C)NC(=O)C(=O)Nc2cnc(C3CC3)nc2)ncccc1F CCCCC(C)C(C(=O)NCC1CCOC1)N1CCC(CN2CCCCC2)C1 C(C)(N=c1nc(N2CCC(C(C)C)C2)c2sccc2[nH]1)C1(OC)CCCC1 c1(C(=O)NC(C2N(C(C(C=CCCC)O)=O)CCC2)C)cc(C(C)C)cnc1O c1(C(=O)NCCCN(C(C2(C)C(C)OCC2)=O)C)ccc2cc(Br)ccc2c1 c1(C(N2C(CNC(c3cccc(SCCC)c3)=O)CC2)=O)ccn2ccsc12 c1(C(=O)NCC2C(NC(c3n(CCC)ccc3)=O)C2)ncccc1O N1(C(C(CC)n2cccn2)=O)CCC(C(F)F)(CNC(=O)COCCO)C1 C12(C(=O)NC(c3nc(C)sc3)C)CCCC1CCN2C(=O)CCC1(C#N)CCC1 C1(CC=C)(NC(=O)C(Br)=C(C)C)CCCN(C(c2cc(Cl)ncc2F)=O)C1 C1(C(=O)NCC(C)CNC(=O)CCc2cncs2)CC12CCCC2 c1(C(=O)NCCCCNC(c2cc(F)c(CO)c(F)c2)=O)cc2cn[nH]c2cn1 CC1CCC(=CC(=O)NCC(c2ccccc2)NC(c2scnc2C2CC2)=O)C1 c1(C(=O)NCC2(CC)CN(C(C(CC=C)NC(C)=O)=O)C2)coc2c1CCCC2 C1(COCCN)CCCN(S(=O)(=O)Cc2cccc(Br)c2)C1 CC1(NC(=O)C=Cc2cnc[nH]2)CN(C(=O)Cc2ccccc2)C1 c1(C(=O)NC(CNC(C2(C)CC=CCC2)=O)(C)C2CC2)cnnc2ccccc12 N1(C(CCCc2ncc(C)o2)=O)CCCN(C(=O)Cn2cnc(=N)[nH]2)C(C)C1 C1(C(c2n(CCCOC)nnn2)NCc2sccc2Br)CCCCCC1 c1(C(=O)NC(CNC(c2cc(C)cc(C)n2)=O)C)ccc2c(Br)cccc2c1 c1(C(=O)NCCN(C(C(C)SCCCC)=O)CC(C)O)ncoc1CNCC Cc1ccccc1C(O)C(=O)NCc1nccn1-c1ccccn1 Cc1ccc(CO)c(NC(=O)C(CC(C)C)N2CCCCC2C)n1 N1(C(C2CN(C)C(=O)N2)=O)CCC(C)(C)C1CC(=O)Nc1cnn(C(F)F)c1 N(C1c2cc(Br)ccc2SCC1C)C(=O)NCCc1cc(C)c(F)cc1 Cc1nc(CCN(C(C2OCCC2NC(=O)CCc2ccccn2)=O)C(C)C)n[nH]1 N1(C(C2(C)C(C)C2)=O)CCC2(CCN(C(=O)C(=Cc3c[nH]cn3)F)C2)C1 C(C(=O)NC1CCC(CCC(N2CCCC(CC)C2)=O)C1)(C(C)C)SCC C(N=c1cc(NCCCCC(N)=O)nc(C2CCOCC2)[nH]1)c1c(=N)cc[nH]c1 Cn1ncc2c(C(N3CCN(C(=O)CC4CCC4)CC34CC4)=O)ncnc12 c1(OC)cc(CN2CCCC(NC(c3csc(C(F)(F)F)n3)=O)C2)ccn1 Cc1cc(C(=O)N(C(CNC(C2(O)CC(F)(F)C2)=O)C2CC2)C)n2nccc2n1 c1(C(=O)NCC2C(NC(c3nc(C)sc3C)=O)CCC2)ccc(Cl)c(O)c1N c1(SC)cccc(F)c1C(N1CCCCC(CNC(=O)CCn2ccnc2)C1)=O CC1(CNC(C2CC2c2cccs2)=O)CCN(C(=O)CCN2CCOC2=O)CC1 CC(C)C(CNC(=O)C(C)(C)C)NC(c1ccnn1CC#N)=O N(C(=NCCC(=O)N(C)C)N1CC2C(F)(F)C2(Cl)C1)CC(CC1CC1)N(C)C c1(C(=O)NCC(CC)(CC)NC(=O)Cc2nocc2C)cc2cnccc2o1 Cc1ccn2cc(C(=O)NCC34CCCC(CN3)C4)nc2c1 CC1CN(C(c2ccno2)=O)CC(C(N2CCOCC(C(=O)N(C)C)C2)=O)O1 n1(CC(=O)NC2CCC(NC(c3cc(C(C)C)[nH]n3)=O)C2)cc(P(C)(C)=O)cn1 C1(CC)CN(C(c2csc(-c3ncccn3)n2)=O)CC1NC(c1ccoc1C)=O c1(C(C(=O)NC2CCOC2)N(CC)CC2CC2)ccc(-c2nc(=O)o[nH]2)cc1 c1(NC(=O)CC2CCN(Cc3ccnc(Cl)c3)C2)cccc2ncccc12 CCC(C(=O)N1CCCC(CO)(CNC(=O)C(F)=C(C)C)C1)C(C)C CC(C)CC(C)OCCC(=O)N(CCNC(c1cc(C2CC2)on1)=O)C(C)C N(C(=NCCc1ccncc1)NC1CCCC1)CCN1CC(C)C(C)C1 C(C(=O)NCCCOCCNC(c1onc(C)c1C)=O)(C(C)C)N(C)CC C1(C(N2CC(CC(C#C)C)C2)=O)CNC(=O)CN1C(=O)C(=O)NCC(F)F C1(NC(C2N(C)CCOC2)=O)CN(C(c2cc3scnc3[nH]2)=O)CCC1CO C(N=c1cc[nH]cc1S(=O)(=O)NC1CCN(CC(C)C)C1)c1ccc(CC)cc1 c1(OCCC(=O)NCCOCCNC(C2C(C)CC2)=O)ccc(Br)cc1F N#Cc1ccc(C(N2CC3(NC(C4(F)CCOC4)=O)CC2C3)=O)cc1 NS(=O)(=O)c1ccc(Cl)c(S(=O)(=O)NC(c2cnc3c(c2)CCNC3)=O)c1 CC(CC(C)(F)F)C(=O)N1CC2(C1)CN(C(=O)C(Cc1ccsc1)NC=O)C2 N1(C(C(CC)OC)=O)CCC2(CCCCC2NC(C2CCC3CC2C3(C)C)=O)C1 C(CCC(=O)NC(CNC(=O)CC)Cc1ccccc1)CN(C)CC c1(CN2C(C(=O)Nc3nnc(C(F)F)o3)C3CCC2C3)cc(Cl)cc(Br)c1F c1(OCCCOC)ccc(C(=O)NCCCCN(C(=O)C(C)CF)C)cc1OC CCCCC(C)C(=O)NCC(C)N(C(=O)Cc1ccc(CO)c(C)c1)CC Cc1cc(C(=O)NCC=CCNC(C2(c3ccc(F)cn3)CC2)=O)cc2ccsc12 C1(C(=O)NCc2ccn(C)n2)CC2(CCC2)CN1C(=O)CC1=CCOCC1 C1(NC(COc2cccc(C)c2)=O)CN(C(C2CSCC(=O)N2)=O)CC2(CC2)C1 N1(Cc2ccc(N(C)C)cc2)C(=O)NC(Cc2ccnn2C)C1=O C(C(CC(C)C)C(=O)NCc1cc(C(C)C)no1)NC(c1c(NC)cccc1)=O N1(CCNC(c2snc(Cl)c2Cl)=O)CCCN(C(=O)C(F)n2ccnc2)CC1 C(CCC(C)(C)C(=O)N(C(C)C(=O)NC1CC1)C)NC(CCn1c(C)ncc1)=O CCC(CC(C)C)C(=O)NC1(CC)CCCN(C(c2cn3cc(C)sc3n2)=O)C1 Cc1c(NC(=O)CN2CCCC(C)CC2)ncnc1N1CCOC(C(N)=O)C1 C#Cc1ccc(NC(C2CCN(C(C3CCCCC3)=O)CC2O)=O)cc1Cl N(C(=NCCCOC1CC(c2ccc(F)cc2)C1)NC1CC1)CC(CC)(O)CC Cc1nc2ccc(C(N3CCC(=CCNC(C4(C)CC4(Cl)Cl)=O)CC3)=O)cc2[nH]1 O=C(CCCCC(F)F)NC1CCCN(C(c2nnn3c2COCC3)=O)C1 C1(NC(C(C(C)C)SCC)=O)C2CC3CN(C(=O)C(CC)NC(C)=O)C1C3C2 C1(CNC(c2c(C)cccc2F)=O)CC2(CCOCC2)CN1C(C1(Cl)CC1)=O CC1(C)C2CCC1(C(N1CCCN(CCNC(=O)C=C3CCC3)CC1)=O)C2 Cc1cc(CO)oc1C(N1CCCC1C1CCN(C(C2(C(N)=O)CC2)=O)CC1)=O c1(C(=O)NCC2(CNC(C(C(C)(C)C)SC)=O)CC2)cc2c(C)ccc(F)c2o1 c1(SCC(CO)Cc2cccnc2)ccc2cc(Cl)cnc2n1 c1(SCC(N2CC(C)(NC(C(C)OCCC=C)=O)C2)=O)cccc(F)c1 C1(C(=O)NC2CC(NC(CCCn3c(C)csc3=O)=O)C2)CCC2CC2CC1 S(=O)(=O)(c1ccc(Br)s1)NC1CC(NC(c2cc(C)c(Cl)cc2)=O)C1 CC1CN(C(=O)CC2CCC(C)(C)C2)CCN(C(=O)C(O)CC(F)(F)F)C1 c1(C(N2C(CNC(c3c(C)c[nH]n3)=O)CC2)=O)ccnc(O)c1F CC1=NS(=O)(=O)NC=C1C(=O)N1CCN(C(=O)C(F)n2cccn2)CCC1C c1(C(C)N)nonc1N.C(=O)(C(=O)NCCO)N(CCNC(=O)C(=O)C1CC1)C S(=O)(=O)(c1cccc(NC2CCN3CCC2C3)n1)N1CCN(CC)C(C)C1 c1(OCC#C)ccc(C(=O)NC2(c3ccccc3Br)CC2)cc1Cl CC(C)S(=O)(=O)c1ccc(C(=O)NCCC2(NC(=O)CCC(C)(C)C)CC2)cc1 C1(CC(=O)OC)CN(C(c2cccc(-c3nn[nH]n3)c2)=O)CC(C(F)(F)F)O1 C(=O)(CCC[N+](=O)[O-])N(CC)CC1CCN(C(=O)Cc2ccnn2C)CC1 C1(C(C)NC(COCCOC)=O)CCCN(C(=O)C(c2ccc(O)cc2)=O)C1 CC(C)(C)C(O)C(=O)N1CCC(n2cc(COCC3CCC(F)(F)CC3)nn2)C1 C12(NC(CCC#CC)=O)CCCN(C(c3ccc[nH]3)=O)C1C2 C(N=c1cc(NCC2(C)C=CCCC2)nc[nH]1)c1snc(C)n1 C1(NC(C(C)(C)SC)=O)CCCCN(Cc2ccccc2Cl)C1=O C(CC1CCCC1)(C(=O)NC1CCC(C(N2CC(C(C)OC)C2)=O)C1)OC N1(C(c2c(C)cccc2F)=O)CC2CC(NC(C3(C)CCOC3)=O)CC(C2)C1 c1(C(N2CC(CNC(C(C)OCC3CCCO3)=O)C2)=O)cc(C(F)F)cnc1O c1(C(N2CC(NC(CC3C(C)(C)C3)=O)C(F)CC2)=O)cnn2c1NCCC2 N1(C(C)=O)CCCC(NC(=O)C(=O)NC(C2CC2)C2CC2)C1 c1(C(N2C(C(N(C)C)=O)CC2)=O)ccoc1COCCOC1CCCOC1 c1(C(=O)NCCC2N(C(C(CC)F)=O)CCC2)cnc(C)cc1C C1(NC(C2CCN(C(=O)CC3CCCOCC3)CCO2)=O)C2CCC3C(C2)CC13 c12ccc(cc1)[nH]2.c1(C(N(CCOCC(F)(F)F)CCO)=O)ccc(COC)[nH]1 N1(C(C(C)NC(CC)=O)=O)CCC(O)(CNC(c2cc(C(=O)OC)on2)=O)CC1 CCCC(CC)CC(=O)N(CCC(C)NC(=O)C#CC1CCC1)C C=C=CC(C)C(=O)NCCCCCN(C(=O)CC1OCCC1(C)C)C(C)C C1(COC)(NC(c2cncc(C)c2Cl)=O)CCCCC1C.c12cc([nH]n1)C(=O)N2 N1(C(C(C)OCOC)=O)CCN(CC(=O)N(C2(c3cc[nH]n3)CC2)C)CC1 C(=O)(C(C)CC(C)(F)F)NC1CC(C)(NC(CCCCOC)=O)C1 N(C(=NCc1cc(C2CC2)on1)NC(C1CC1)C1CC1)CC(NOC)=O N1(C(c2cnc(CC)n2C)C(=O)NC(C)CC)CCn2c(C)nnc2C1C C1(C(N2CCC(CCCC)C2)=O)CC2(CC(NC(=O)C=C3CCC3)C2)C1 c1(C(N2CC(N(C(c3cc(C)nnc3)=O)C)C(C)CC2)=O)cccn2cncc12 C(=O)(CP(C)(C)=O)NC1(c2cn(C(C)Cn3ccnc3C(C)C)nn2)CCC1 Cc1nccc(C(=O)NC2CN(C(C3(NC(C)C)CC3)=O)CC2(C)C)c1Cl c1(C2(C(c3nnnn3C(C)C)NC(C=C)C3CC3)CC2)ccc(Cl)cc1 C(CC1CC1)(CC(=O)NCC(C)(O)CO)NC(C1C(C(C)C)(CC)C1)=O n1(C(CC)C)nccc1C(=O)NC1(CNC(c2csc(Br)n2)=O)CCC1 N1(C(C2C(NC(=O)OC(C)(C)C)CC=CC2)=O)CC(C(=O)O)CC1(C)C C1(C#N)(CC)CCN(C(=O)CC(C)(C)NC(=O)CCc2csnn2)CC1 c1(C(=O)NC23C(CN(C(CCC=C=C)=O)C2)CC3)cc2ccc(OC)nc2[nH]1 c1(CC(=O)NC2CN(C(c3c(C)[nH]nc3C(C)C)=O)C2)ccc(Br)cc1C#N c1(OC)ccc(Br)c(C(=O)NC2CCCC(NC(=O)C(C)OC(C)(C)C)C2)c1 C(=O)(CC(C)(C)Cc1cccs1)NCC1N(C(c2cnc(C)[nH]2)=O)CC1 C1(O)(CNC(c2cc(CNC(C(C)N(C(C)=O)C)=O)oc2)=O)CCC(C)C1 NC1CN(C(=O)CC2COCCO2)CC2(CC2)C1 C(=O)(C(CC(C)C)C(N)=O)NC1C2CCN(C(Cc3c(C)cc(Cl)cc3)=O)C2C1 C12(NC(CC(CC)C(C)C)=O)CCCC1(F)CN(C(=O)CCC(=O)NC)C2 N1(C(C(N)=O)=O)CCCN(C(=O)CCSc2ccc(F)cc2)CC1C(=O)O CCC(C)C(O)C(C)C(=O)NCC(CC)(CC)NC(c1cc(Cl)ccn1)=O BrC1=C(CNC2(I)CC2)CC#CCC(I)=C1 C1(C(C(=O)N(CC(CC)NC(=O)CCOC(C)=O)C)F)CCOCC1 c1(C(=O)NCC(CCC)NC(c2n(C=C)nnc2)=O)cc(C)n(C)c(=O)c1 CCC(C)C(C(=O)NC1CCC(CNC(c2ccc(N)cn2)=O)C1)OC C1(C(=O)NCc2c(C)nc(C)s2)CC2(CCN(C(=O)C(C)N(C)C)C2)C1 C1(C(=O)NCc2cnc(C(C)C)[nH]2)COCCC1NC(=O)CCn1ccnc1 C1(NS(NC)(=O)=O)CCCN(C(c2ccccc2F)=O)C1 c1(NCCC)ncccc1S(=O)(=O)NC(c1ccc(Br)cc1)CO c12ccc(cc1)CS(=O)(=O)NC2.n1(CCOC)c(C(C)C)nnc1S N1(C(CNC2(C#C)CCCC2)=O)CC(N(C)C)Cc2ccccc21 C1(CN(C(CC=CC=C)=O)C)CN(C(=O)C=CCO)CCO1 Cc1n[nH]c(C)c1CC(=O)NC(C1CN(C(c2cc(C#N)on2)=O)C1)C c1(C(N(CC(C)NC(c2c(COC)n(C)nc2)=O)C)=O)scc2c1OCCO2 c1(CNC(C2CCCCC2)C(=O)OCC)cccc(OCc2ccccn2)c1 c1(C(=O)NC2(CCNC(c3cc(OC)ncc3)=O)CC2)ccc(P(C)(C)=O)s1 Cn1cncc1C(C1CCCC1)NCC1CCCCO1 N1(C(c2c(CC)c[nH]c2)=O)CC(NC(C2CCCCC(=O)N2)=O)C(S(C)(=O)=O)C1 C(CC(C)C(=O)NCC(O)CCNC(=O)Cc1nc(C)sc1C)=CC c1(C(C)C)cnc(C(N2CCC(N3CCCC3)CC2)C(=O)NCC(F)F)nc1 N1(C(C2(CCNC(c3cccc(C)c3N)=O)CC2)=O)CCOC(C)(C)CC1 CCC(CC(=O)N1CCC(C)(CC(=O)NCC(F)C(C)(C)O)C1)C(C)C CCCC(CC)CC(=O)NC1CN(C(=O)CCC=C(C)C)CC12CC2 C(=O)(C(C(C)(C)C)NC(C)=O)N1C(CNC(C=CSC)=O)CCC1 N1(C(C2(NC(c3ccncc3F)=O)CCCC2)=O)CC2CCC=CC12 N1(C(C2N(C(c3n[nH]c(C)c3O)=O)CC(O)C2)=O)CCC2(CCOC2)C1 Cc1ccc(CCC(=O)NCCN(C(C2CCCC(F)C2)=O)C2CC2)cc1C c1(C(=O)NCc2cn(C3CC(C(=O)OC)C3)nn2)c(C)nc2cccnn12 c1(N2CCC(C)C2)ccc(C(=O)NC2CCOC2C(=O)N(C)C)cc1 C1(CC=C)(C(N2CCCCC2CNC(c2ccncc2C)=O)=O)CCOCC1 CCC(C)CC(=O)N1CC(CNC(c2cnn(-c3ccccc3)c2Cl)=O)C1 c1(NC(c2cc(CNC(CCC(C)OCC)=O)nn2C)=O)cccc(Cl)c1O c1(C(=O)NC2C(C)CN(C(=O)CN3C(=O)CCC3=O)C2)ncccc1N=[N+]=[N-] c1(N2CCC(CNC(c3cnoc3CC)=O)C2)cccc(Cl)c1Cl.Cc1nc(C)cs1 Cc1cc(C(N2CCC2CC(=O)NCC(c2ccco2)O)=O)ccn1 c1(C(=O)NC(CC=C)CNC(C2CC2COC)=O)c(N)c(C(F)(F)F)nn1C c1(N2CC(C)=C(C)CC2)[nH]c(=NCC2(CO)CC=CC2)nc2sccc12 CC1CN(C(c2ncncc2Cl)=O)CC1CNC(C1COCC1(C)C)=O C1(OC)CCCCC1C(=O)N(C1CCN(C(c2ccc(Cl)cn2)=O)C1)CC1CC1 CC(CC(F)F)C(=O)N(C1CN(C(C2C(F)(F)C23CC3)=O)C1)C c1(C(=O)NC(C2CCN(C(C(C=C)(C)C)=O)CC2)C)c(N)sc2c1CCSC2 c1(C(N(CCC(C)NC(=O)CN=S(C)(C)=O)C)=O)cccc2cncn12 c1(CC(=O)NCc2cn(CCN)nn2)ccc2c(c1)OCCO2.N1(C)CC2CC2C1 c1(C(=O)NCC(CN(C)C(C2C=CCC2)=O)(C)C)cc2cc(Cl)ccc2[nH]1 c1(NCC(CNC(c2c(SCC)cccn2)=O)O)ncnc(Cl)c1C(C)=O N1(C(=O)NC(c2onc(C)n2)Cc2ccccc2)CCCC2(CCN(C)C2=O)C1 N1(C(C2CC(NC(CCOC(C)=O)=O)C2)=O)CCCC(CCCO)C1 C(=O)(CCC(=O)c1ccccc1Cl)NC1(CCNC(=O)C=CC(F)(F)F)CCC1 N1(C(C(C(C)C)(C)O)=O)CCCCC2(C1)CN(C(c1cccc(S(C)=O)c1)=O)C2 c1(CC(=O)NC2CN(C(c3ncn(CC)c3)=O)C2)cccc2cnccc12 C1(NC(c2ccnc(OC)n2)=O)CCC2CN(C(=O)CCC(C)SC)CC2C1 Cc1c(C(=O)NNC(=O)C(O)c2ccccc2Br)oc2ccccc12 CN1CC(O)(CN(C)C(C2(CNC(=O)CC3C=CCC3)CCC2)=O)C1 c1(CCC(=O)Oc2ccc(OC)cc2CN)cccc(S(=O)(=O)N(CC#N)CC)c1 N1(C(C2CCN(C(CC)=O)C2)=O)C(CC)CC2CC12 c1(-c2scc(C(N3CC(F)(F)C3)=O)n2)ccc(F)c2ccoc12 C12(NC(c3c(C)n(C)nn3)=O)CCC(NC(c3coc(Cl)n3)=O)(CC1)C2 C1(C(=O)N)CC2(C1)NC(=O)NC2=O.C(C)(C)(C=CC(=O)NC1(CO)CCC1)SC c1(OC)cccc(F)c1CNC(C1CC(c2ccc(-n3ccnc3C)cc2)C1)=O S(=O)(=O)(c1ccc(NC2CCC(n3ccnn3)CC2)nc1)N1CC(CC)SCC1 c1(NC(N2CC(COC)C(OC)C2)=O)ccc2c(c1)CCCO2 C1(NC(CCN2CCN(C)CC2)=O)CCC2CN(C(=O)C3=CCSC3)CCC2C1 CCCCC(C(=O)N(CC(=O)Nc1ccc(F)cc1OCOC)C1CC1)C(C)C C(=O)(C(C)C(=O)NCc1ccc(C(=O)N(C)Cc2cocn2)o1)OC n1(CCC(=O)NC2CC(NC(=O)COCC3CCC3CF)C2)cnc2ccccc12 CC1CC(CNC(C2CCCC2NC(=O)CN(C2CCCC2)C)=O)=NO1 C=CCC(C)(C)CC(=O)NCCC1C(C)CCCN1C(=O)CNC(=O)OC c1(C(=O)NCC2CN(C(CC(CCC)C)=O)C(C)(C)C2)cn(C)c(=O)nc1O N1(C(C(n2cc(CC(=O)NCC(C)C(=O)O)nn2)C)=O)CCc2ccccc21 N1(C(c2cnsn2)=O)CC2CN(C(=O)Cc3cc(Cl)ccc3O)CCC2(CO)C1 C(C(C)(CC)CC)NC(c1ccn(CCNC(C=CC(CC)C)=O)c1)=O c1(C(=O)NCC2C(C)(C)C(NC(=O)COc3ccccc3)C2)cc(F)ccc1Cl c1(CC)oc(C(=O)NC2CCOC(C(=O)N(CCO)CCN(C)C)C2)cc1C c1(C(N2CC(CNC(c3c(C)scc3)=O)OCC2)=O)ccc2c(c1)C(=O)NC2=O c1(C(N2C(CNC(C(CCC)O)=O)CCC2)=O)cc(Br)cc(C)c1C N1(C(C(c2cccc(C)c2)C)=O)CCC(NC(c2cnc(O)s2)=O)C2(CCC2)C1 C(=O)(CCS(C)(=O)=O)N(CCCNC(C(C)=NOCC#N)=O)C Cc1cc(F)cnc1C(=O)N(C(C)(C(N1CCC(F)(CF)C1)=O)C1CC1)C c1(C(N)=O)ccc(O)c(F)c1.C12(F)CCN(C1)C(C1CCOC1)C(=O)N2 C1(N(C(C(C)NC(=O)OC)=O)C)CC2CCC(C1)N2C(C1(OCC)CCCC1)=O C=CC1OCCC1CNC(c1ccc(Nc2nn[nH]n2)cc1)=O C(=O)(C1=NOC(CNC(=O)CCc2cnoc2)C1)N1CC(OC(CC)=O)C1 c1(C(=O)NC(C)CNC(=O)C=Cc2nccs2)ccc(NCC2CC2)cc1 Cc1cc(F)ccc1C(N1CCC(NC(=O)CCn2ccnn2)C1C(C)(C)C)=O C1(C(=O)NCCN2CCCOC2=O)(CC)CCCN1C(=O)Cc1ccon1 C1(C(=O)NCC(=O)NCC(F)F)(NC(=O)CC2CCCSC2)CCSC1 c1(C(N(CC(C)(C)CNC(=O)CC2OCCO2)CC)=O)cccc(C#CCO)c1 n1(CCC#C)c(N(C)CCC2CCCC2)nnc1C(O)C(C)(C)C C(=O)(C1=CCCCO1)N1C(CC(=O)NCC2CCC(C)CC2)CC(O)C1 c1(C(=O)NCCN(C(C2CC=CCO2)=O)CC)cnc(CC(C)C)s1 C12(C(=O)NCC)CCCC1CCN2CC1CC1COC Cc1cccc2c(CC(N3CCN(C(C4CC4(C)C)=O)CC3CO)=O)cccc12 CCC(F)(F)C(C)(C)C(=O)NC1CCCN(C(=O)CCCCc2cnc[nH]2)C1 Cc1ccc(C(=O)NC(CNC(=O)CN(S(C)(=O)=O)C)CC(C)C)c([N+](=O)[O-])c1 Nc1c(C(=O)NCCCOCCNC(C2CCC(F)(F)C2)=O)ccc(F)c1F CCCC(C(=O)N1CC(O)CC1CNC(=O)C(c1ccc(F)cc1)(C)C)OCC c1(C(N2CC(C)(c3cn(-c4cccc(Cl)c4Cl)nn3)C2)=O)c(Br)cccc1Br c1(OC)cc(Cl)c(CNC2COCC3(CCC3)O2)cc1OC c1(OC)ccc(F)c(N)c1C(=O)NC1CCCCC1NC(=O)OC(C)(C)C Cc1c(C(=O)NCC(O)CNC(c2cc(N(C)C)nc(Cl)c2)=O)cccc1N N#CCCCC(=O)N1CCC(OCCNC(=O)C(F)(F)CF)C1 c1(C(C)C)ccccc1-n1nc(C(C)C2CC2)nc1-c1ccsc1 C(=O)(CC(C)C(C)(C)C)NCC(CCOC)NC(C1CC(C2CC2)C1)=O C(CCC(=O)NC(C)CCCNC(=O)C=C1CCC1)=CCC=C C(=O)(C1CCCc2scnc21)NC1C2CN(C(CC3ON=C(CC)C3)=O)CC1C2 CCCC(C)(CCC)C(=O)NCC1COCC1NC(c1[nH]cc2c1CCCC2)=O C1(NC(C(C)(C)OCC)=O)CN(C(=O)CCN2CCC(O)CC2)C(C)(CC)C1 C1(NC(c2c(CC)nco2)=O)CCC2CC1CN2C(c1cnc(C(C)(F)F)s1)=O Cc1cc(C(=O)N(C)CC2CN(C(C3CC(C)(C)C3)=O)CCO2)c(C)n1C1CC1 C1(C(=O)NCC#CCNC(C(c2c(F)cccc2F)C)=O)CCC2(CCC2)C1 c1(CNC(C)C(N)=O)ccc(C#N)cc1Br c1(C(N2CC(NC(C(CC)C(C)C)=O)C(C)C2)=O)cc(F)cc2cc[nH]c12 CC1C2CC(C2NC(=O)C2=COCCC2)N1C(=O)COCCN(C)C c1(-n2cnc(C(=O)NCC(CN(C(C(CC)OCC)=O)C)O)n2)ncccc1F C1(C)(C(N2CC(CN(C(=O)C(=O)Cc3cccc(Cl)c3)C)C2)=O)CC=CCC1 N1(C(c2cc(C(F)F)on2)C(=O)NCC2CC2)CCC2(CCC(O)C2)C1 CN1CCCCC1C(N1CCOC(C(=O)N(CCCF)C)C1)=O CC1CN(C(C2(C3CCC3)CC2(F)F)=O)CC(C)N(C(=O)CCS(C)=O)C1 Cc1ccc(C(=O)N=c2ccn(CCC(F)(F)F)[nH]2)c(=O)n1C Cc1nc(C)c(C(=O)N(CCCNC(c2cc(Br)sn2)=O)C(C)C)o1 C1(CNC(c2ccc(Br)o2)=O)CC(O)CN1C(=O)CCCc1cnccn1 C1(C2CCN(C(=O)CC3CCCOC3)C2)(NC(C(C(C)C)CO)=O)CC1 C1(CNC(C(CC)CN(C)C)=O)CN(C(=O)CCc2cscn2)CC12CCC2 C(C(=O)NNC(=O)c1ncccc1N(C)C(C)C)Oc1c(C)cccc1 c1(CC(=O)NC2(C3CN(C(c4c[nH]c(=NC)o4)=O)C3)CC2)ccc2nsnc2c1 C=CC(O)(C(=O)N1CC(O)(CCNC(=O)CN2CCOCC2=O)C1)C(F)(F)F C(=O)(CCCN(C)N=O)N(CCCNC(C(C(CC)O)C)=O)CC1CCCC1 N1(C(C(c2cccc(Br)c2)C)=O)CC(NC(c2cc(Cl)c[nH]2)=O)C(C)C1 N1(C(C(C)C2CC2)=O)CCCC(O)(CNC(=O)CCSc2cccc(F)c2)CC1 CCC(CC)CC(=O)NC1CN(C(=O)C(C)(C)C2CCCCO2)CCC1C C1(NC(c2ccc(OCCNC(C)=O)cc2)c2n(CC)nnn2)CCC(C)(C)C1 N1(C(CCCC=C)=O)CC2(CCCC(CNC(=O)C(C)(C)SC)O2)C1 C12(C)CCN(CC1)C(=O)c1ccc(o1)C2.c1(C(=O)OC)cc(C(=O)N)on1.CCCO CCCCC(C(=O)NCC(COC)NC(c1ccnc2cc[nH]c12)=O)C(C)C S(=O)(=O)(c1ccnn1-c1ccccc1)NCC(C(=O)OC)C1CCOCC1 C1(NC(C(CC)SC)=O)CC2CCC(C1)N2C(=O)CC1CC(O)C1(C)C N1(C(C2(Br)CC2(F)F)=O)CCC(O)(C(N2CCCC2C(F)(F)F)=O)CC1 C1(CC(=O)NCC2C(NC(c3ncc(OC(C)C)nc3)=O)C2)OCCOC1(C)C CC1CCC(C(NOCC(=O)NC2CCC3(CC3)C2)=O)N1C(=O)OC(C)(C)C C1(C)(CNC(c2[nH]cc(C)c2)=O)CCN(C(c2cnn(C(C)C)c2C2CC2)=O)C1 C=CC(CC)CC(=O)NCC1CN(C(C2(C)CC(C)(C)C2)=O)CC1(C)C Cc1cc(C(=O)NCCN2CCCNC2=O)c2c(C)nn(C)c2n1 c1(CC)nocc1C(N1CCCC1CC(=O)NC(C)C(=O)N(C)CC)=O Cc1ccc(O)cc1C(=O)NCCC1(O)CCN(C(=O)CCC2CC2(F)F)CC1 c1(OCC(=O)NC2C(NC(CC(CC)SC)=O)CCO2)ccc(Cl)c2ccccc12 C1(C(=O)NCC(CC)NC(c2cc(C3CC3)nnc2O)=O)CCCCCCC1 C1(CNC(CCc2ccc(OC)cc2)=O)CN(C(=O)C(C)C(C)(F)F)CC1(C)C c1(N(C)CC2CCCN(C)C2)nc(N(C)CCOC(F)F)c2[nH]ccc2n1 C1(C(N2CC(CC(C)NC(C(CC)O)=O)C2)=O)CC2(C1)CC(C#N)C2 c1(NCC(C)CO)ncccc1S(=O)(=O)NC12CCC(CO)(CC1)C2 C=CCCCC(C)(C)C(=O)NC(C)CC(C)NC(=O)CCc1nccn1CC N1(C(C(C=C)(C)CC)=O)CCc2ccc(C(N3CCOC(C)C3C)=O)nc2C1 c1(C(N(CCCNC(CC(=O)N(C)C)=O)CCO)=O)cnc2c(c1)COCC2 C12(C(N(C3CCOCC3)CCC)=O)CC1CN(C(c1ccccc1SC)=O)C2 c1(NC(CNC(C(N2CCC(C)C2)=O)=O)=O)cnc(O)c(Cl)c1 CCC(C)(CO)C(=O)N1CCC(CNC(=O)CC2NC(=O)CNC2=O)(OC)C1 C(=O)(CC(CCC)CCC)N1C(C(=O)NCCSCC=C)C(C)C1 N1(C(C(C(C)O)NC(C)=O)=O)CCC2(CC(N(C)C)C2)C1.C1(C)CC(=O)N1 C1(CC(=O)NC(c2c(C(=O)NCc3n(CC)cnn3)con2)C)CCN(C)C1=O C1(CC=C)(C(=O)NCC2C=CCCC2)CCN(C(c2cc(C(C)C)on2)=O)C1 c1(N2C3CC(C)CC2CCC3)nc(=N)[nH]c(=NCCC2=CCC3CC2C3(C)C)[nH]1 N1(C(C=C(C)C(F)F)=O)CC(CNC(=O)CNc2nccs2)CC1(C)C C1(C2CCC2)(C(N2CCN(C(COCC(=O)NC)=O)C(CCO)C2)=O)CC1(F)F c1(C(=O)NCCCN(C(=O)CC2CCC2(C)C)C)cc2cc(Cl)ccc2n1C c1(N2CC3C(NC(C(CC)(C)C)=O)C3C2)ncc2ccsc2n1 C1(NC(=O)Cn2cc(C3CC3)nn2)CCN(C(C23CCCC(C2)OC3)=O)CC1F CN1CCC(F)(C(=O)NCCN(C(=O)Cc2ccc(F)c(F)c2)C)CC1 N(C(=NCCCCl)N1CC(F)(F)C(F)(F)C1)CC1C(N(C(=O)OC)C)C1 c12ncc(C)cc1S(=O)(=O)N1CCOCC(C1)CN2C1CC1.N(CC)(CC)CC1CC1 C1(C(=O)NC2(C(=O)NCCCCCOC)CCN(C)C2)CCC(N=[N+]=[N-])C1 c1(C(=O)NCCCOCCNC(C(C2CCC(=O)N2)C)=O)cccc(N)c1F C(=O)(CCCC(C)(C)NC(c1cnn(CCO)c1)=O)NC1C(OC)CC1O N1(C(CC)C(N2CCCOC(CNC(=O)CC3CC3)C2)=O)CCc2ccccc21 c1(C(=O)NCC2C(NC(C=CCC)=O)CC2)ccc(SC)o1 c1(CC)ncc(C(N2CC(CNC(C3CCOC3C)=O)C2)=O)c(C)n1 CN1CCOC(C(=O)NC2CC(F)CN(C(c3cc(C4CC4)nn3C)=O)C2)C1=O c12ccc(c(F)c1)CC(=O)N1CC(N3C(=O)CC(C3)C(=O)O2)C1.CN N1(C(c2cc(C)c(O)cc2)=O)CCC2CCC1C2NC(=O)CCCCCF N1(C(C2(C)C=CCC2)=O)CCCC2(NC(=O)C(F)=CC3CC3)CC2C1 c1(C(N2CC(C)C(NC(C3CCCC(=O)N3C)=O)C2)=O)cc(O)cc(=O)o1 c1(C(=O)NC2CCCC(NC(C(C)(C)O)=O)C2)cn2c(C(F)(F)F)cccc2n1 c1(C(=O)NCCNC(c2cc(CC(C)C)on2)=O)ccccc1Cc1nn[nH]n1 CCC1=C(C(=O)N2CCC(NC(=O)COc3cnn(C)c3)C2)SCCO1 C1(C(N2CC(F)(CNC(c3cnn(CC(F)(F)F)c3)=O)C2)=O)C(F)(F)C12CCC2 C1(C(=O)NCCCN(C(C(C(C)C)c2cnn(C)c2)=O)C)CCn2nccc2C1 C1(CNC(C(C(C)(C)O)F)=O)C(C2CC2)CCN1C(=O)C(=O)Cc1ccccc1 c1(N2CC(NC(C3CCC(C)C3)=O)C(C)(C)C2)ncnc2sccc12 C1(CC=C)(NC(=O)CC2CCCO2)CCN(C(C2(C#N)CC2)=O)C1 C1(C(N2CC(CN(C)C(C3CC=CC3)=O)OCC2)=O)CC2CSCC(C1)C2 N1(C(CCCN(C)C)=O)CC(O)CC1CNC(C1CC1C(C)(F)F)=O CC1(C)C(NC(=O)CCC2CCCC(=O)N2)CCN1C(=O)Cc1cccnc1F C12(CC(=O)NCCCN(C)C(C3CN(C4CCOC4)C3)=O)CCCC1C2 c1(C(C)C)cccc(C(N2CC(CNC(=O)CCC(=O)N(C)C)C3CC23)=O)c1N C(=O)(CC1CCCc2oc(C)nc21)NC1(CC)CN(C(=O)COC2CC=CC2)C1 N1(C(C(C)CC2CCC2)=O)CC(O)(C2(CNC(=O)CC3CCC34CCC4)CC2)C1 C1(CC(=O)NCC(c2ccccc2)CNC(c2c(C)snn2)=O)CCCC(=O)N1 N1(C(c2cc(CC)no2)=O)CCOCC1CNC(c1cnc(C(C)(F)F)s1)=O C=CC1CN(C(c2c(C(F)F)n[nH]c2C)=O)CC1NC(=O)COC1CCOC1 N1(C(c2c(C)onc2C(F)(F)F)=O)CC2(C1)CN(C(C1CCCCC1O)=O)C2 CC1(CNC(C2(C)CCCO2)=O)CCCN(C(=O)C=Cc2ccncn2)C1 c1(C(=O)NC2(c3cc(C)no3)CC2)c(CNC(=O)CC2CC=CC2)cnn1C c1(CNC(NCC2N(CC)CCC2)=NCCSC)ccc2cccnc2c1 CCC(C)CCC(=O)N(C1CCCCN(C(=O)CCOCCOC)C1)C N1(C(CSCCC(C)C)=O)CCCCC1CCNC(=O)C=Cc1ccn(C)c1 c1(C(C)CC(=O)NC(C)(CNC(C2CCCN2C)=O)C2CC2)cccc(Br)c1 c1(C(=O)NCC(CC)NC(=O)Cc2ccno2)cc(O)cc(Cl)c1Cl C(=O)(C1CCCc2nc(C)[nH]c21)N1C(CCCOC(CC)(C)C)CCCC1 c1(C(C(=O)NC2CC(CCNC(CNC(N)=O)=O)C2)O)cc(F)c(F)c(F)c1 CC1(C)CN(C(C2CC(C(F)F)C2)=O)CC(CNC(C2CNC(=O)N2)=O)O1 C1(CNC(C2(C(CC)=O)CC2)=O)CCN(C(C2CCN(c3nc(=N)[nH][nH]3)C2)=O)C1 c1(C(N(C2CCN(C(c3cocc3C)=O)C2)CCC)=O)nn(C)cc1Br N1(C(C(C)OCC#C)=O)CC(C)(CNC(=O)CSC(C)C)CC1(C)C C1(C(=O)NCC(CN(C(CC(=O)NCC)=O)CC)O)Cc2nccn2C1 n1(CC(=O)NCC(C)CN(C)C(c2cn(C)nc2O)=O)sc2ccccc2c1=O CC(CCNC(C1CC(NC(C2CCCN2C)=O)C1)=O)CCO C1(O)(CNC(CC2(NC(c3cc(C)oc3C)=O)CCC2)=O)CCC(C)CC1 Cc1ccc(OCC(N2CC(CO)(CNC(=O)CCCN(C)C(C)C)C2)=O)cc1 C(=O)(CS(=O)(=O)C1CC1)N1CC(C)(NC(c2ccc(NC(N(C)C)=O)cc2)=O)C1 N1(C(=O)CNCP(=O)(O)O)CCCC(NC(c2ccc(C(F)(F)F)nc2)=O)CC1 CCC(O)C(C)(C)C(=O)NC1CCN(C(c2ccc(F)c(C(C)C)c2)=O)C1 C1(OC)CC(C(=O)NCCCNC(C)=O)N(C(C2CC2C)=O)C1 c1(CN(CC=C)C(C2CCN(CC3CCOC3)CC2)=O)cc(Br)ccc1F C(=O)(C1CCCc2ncnn21)NCC1CCCN(C(c2cc(N)nc(Cl)c2)=O)C1 c1(C(N2C(C(=O)NCC(N)=O)CC(O)C2)=O)c[nH]c2nccc(Cl)c12 CC(CC(=O)N1CCC(C)(C2CC2)C1)C(C)(C)NC(c1cc(F)ccc1F)=O C1(N(C(C(C(C)NC(c2nc(=N)cc[nH]2)=O)C)=O)C)CCCC(C)(C)C1 N1(C(C2CC(Cl)(Cl)C2)=O)CCN(C2CN(C(C3(c4cccc(O)c4)CC3)=O)C2)CC1 N1(C(=O)CC2CCCCC2O)CCC2(C1)CN(C(=O)CC1CCCO1)C2 C(=O)(C(C(C)O)NC(=O)NC1CCNC(=O)C1)OC C1(NC(c2ccc(C(F)F)o2)=O)CC2(C1)CC(NC(C1CC3CC1C3)=O)C2 N1(C(C2CN=C3N=CNN3C2)=O)CCN(C(=O)C2=C(Cl)CCCC2)C2(CCC2)C1 C1(NC(C(=O)NCC2C(CC)CCCC2)=O)CCCCC12CC2 C(=O)(C1=CCOCC1)N1C(C(=O)NCC(C)OCCO)CCOCC1 C1(C(=O)NC2(C(=O)NCCC)CC2)CCCC(NC(c2coc(C)c2)=O)C1 C1(C(=O)N(CCO)Cc2cc[nH]c2)CC(F)CN1C(c1ccc(N2CCCC2)cc1)=O N1(C(c2cccc(C)c2)=O)CC2CC(NC(=O)C=CSc3ccccc3)CC2C1 N1(C(CNC(c2c(OC)cccc2)=O)=O)CCC2C1CCN2C(C1(F)CCC1)=O N1(CC)CCC(F)(F)CC1.CC1CCC(C(C(=O)NC)N(C2(C)CC2)C)C1 C1(C)(C(=O)Nc2ccc(C(=O)NC(C(=O)OCC)C)cc2)CC(C)(C)OC1=O Cc1cc(C(=O)NCC2CCOC2C)nn1CCO c1(N(C2CCN(C(C)C(=O)NC3CCCCC3)C2)C(CC)=O)sccc1OC C(Cc1cnc[nH]1)(C(=O)NCC1COCC1NC(=O)Cc1cscn1)NC(C)=O N1(C(=O)CCN(C2CC2)CC2CC2)CCC(F)C1 C1(CN(C(c2cn(CC)nc2)=O)C)CCN(C(c2ccc(OC)s2)=O)CC1 C12(C(N3C(C)CC(CCNC(C4CC4C(N)=O)=O)CC3)=O)C3CC(CC13)C2(F)F N1(C(CCSC)=O)CC(NC(c2ccc(N)cc2Cl)=O)C(C)(C)C1 CC(CC(=O)N(C)CCOCCN(C)C(C1CCS1(=O)=O)=O)C1CCCCC1 CC(C#N)C(=O)NCC1CN(C(c2cn(C3CCN(C)C3)nn2)=O)C1 C#CCC(CC(F)F)C(=O)NC(C)(C)CNC(c1cn(C(C)C)cc1C)=O c1(C(=O)NC(c2cc[nH]c2)C)ccn(CCNC(=O)Cc2cnn(C)c2)c1 c1(C(=O)NCC2N(C(C(=O)NCC)=O)CCN(C)C2)cc2ccccc2c(=O)o1 C12(C(=O)NCC=CC(=O)NC(C)CS(C)=O)CC1CNC2=O S(=O)(=O)(c1ccc(F)c(C)n1)NC(c1ccccc1CSC(F)(F)F)C N1(C(C(CCC)OC)=O)CCOCC(F)(CNC(c2cc(C)[nH]n2)=O)C1 C1(NC(CC(CNC(C2(CC#C)CCCO2)=O)O)=O)CCC(C2CC2)C1 c1(N(CCN(C(C2C(C)CC(=O)NC2)=O)C)C)nnc2c(c1C#N)CCCC2 c1(C(=O)NCCC(=C)CNC(=O)C(CC)CC(F)F)nccc2ccccc12 C(CC(=O)NCC1(OC)CCCCC1)(C(F)F)NC(COCCOC)=O C(CCC(C)C)(C(=O)NC1CCN(C(=O)C2=NNC(=O)CC2)C(C)C1)NC(C)=O C1(C(=O)NC(CC(C)C)CO)CCCC12CCN(Cc1cc(I)ccc1Br)C2 C1(NC(CCCCSC)=O)C(O)C(O)CN1C(=O)C(=O)C(C)C c1(NC(C2N(C(CC)=O)CCCC2)C)ncnc(Cl)c1CO N12CC3(CC(CO3)C(=O)C1)C2.C(=O)(CC(F)(F)F)NC(=O)CC1CCC1C(F)(F)F c1(C(N2C(C)C(NC(C3C4CCCC34)=O)CCC2)=O)ccc2c(c1)OC(C)(C)O2 c1(C(N2C(c3cn(Cc4cnc(C)nc4)nn3)CC2)=O)nc2cc(O)ccc2[nH]1 C(CCCCC(=O)NCc1ccc(C(=O)NCc2cnc(OC)cn2)nc1)=CC Cc1ccc(OC(c2cn(C)nc2C)c2ccc(C)o2)cn1 Cc1cc(Br)ccc1C(=O)NCC(CNC(C1(C)CC=CCO1)=O)CO C(C)(C)(CC(=O)N(C1CCC(NC(c2ccc(C(C)C)nc2)=O)C1)C)OC c1(C(=O)NCC2C(CNC(c3c(CC)n(C)cc3)=O)C2)cc(OC)ccc1OC c1(N2CCCC(N(CCCO)C)(CC)C2)ncnc2c1ncn2CCCOC CC(C)C(CCN(C)C(c1ncn(C(C)(C)C)n1)=O)N=c1[nH]nc(C2CC2)s1 CC12CCN(CC1)CC2NC(C1(C)CN(C(c2cnsc2)=O)C(C)(C)C1)=O c1(C(=O)NCCOCCCNC(c2cc[nH]n2)=O)ccn2c(O)nnc2c1 N1(C(C(CC)NC(C)=O)=O)CC(NC(=O)CC(C)C(C)(C)CC)CC2(CCC2)C1 c1(CC(N2CCC(CCNC(C3(C#C)CCC3)=O)C2)=O)sc(C)nc1C C1(CNC(C(C)N=[N+]=[N-])=O)CC(O)C(O)CC1C(=O)N(C)CCN(C)CCO c1(C(=O)NC2C(C(=O)OC(C)(C)C)CCCCC2)cnc2c(c1)NCC2 c1(C(=O)NC2CN(C(=O)COCC3(F)CC3)CC2CO)cnc2c(c1)CCCC2 N1(C(=O)C=CC(=O)NC=CCBr)CCC2C1CCN2C(c1ccc(F)cc1F)=O C1(C(=O)Nc2cccc(NC(CC3C(C)(C)C3)=O)c2)CCn2nncc2C1 N1(Cc2c(C)ccc(C)c2)Cc2[nH][nH]c(=NC(=O)S(=O)(=O)CCCl)c2C1 Cc1oc(C(N2CCOC(CNC(C3C(C)C3(F)F)=O)C2)=O)cc1Br Cc1nc(CO)ncc1C(N1CCCC(CCNC(C2CC2CF)=O)C1)=O N1(C(Cc2ccc(OCCC)cc2)=O)CCC2(NC(=O)C(C)SC)CCCC12.C.CC c1(C(=O)NC(C)C(C)(C)NC(C2CCN2C2CCCC2)=O)cccn(C)c1=O C(=O)(CCC(=O)NC(C)(C)CNC(C1CC(=O)N(C2CN(C)C2)C1)=O)NC(C)C c1(CC)ccsc1C(=O)NC(C(N1CCC(CC2CCC2)C1)=O)C1(O)CCC1 C1(NC(c2c(C)occ2)=O)C2CCN(C(=O)CN(c3ccc(Cl)cc3)C)CCC12 c1(C(=O)NCC2(OC)CN(C(=O)CC3CCCCC3O)C2)cnn(C(C)C)c1C N1(C(c2cc(CNC(c3c(NC)scn3)=O)ncc2)=O)CCC(C)(CO)CC1 c1(N(C)CC2CN(C)C2)nc(=NCCC(C)(C)C)[nH]c2c1SCC2 C(c1ccc2occc2c1)=CC(N1CCCC(O)(CNC(C(C)(C)CO)=O)C1)=O c1(C(N2CCN(C(CC(C(=C)C)O)=O)CC2C(C)C)=O)ncc(C#N)cc1Cl N1(C(C(C(C)C)N(C)C)=O)CC2(CCN(C(c3cnc4n3CCC4)=O)C2)C1 N1(C(C2C(C)(C)CO2)=O)CCC2(CC1)CN(C(C1CCC(F)CC1)=O)CCO2 C=CCC(CC(F)F)C(=O)NCC=C1CCN(C(=O)CS(=O)(=O)CCO)CC1 c1(C(N2CCCC(CC)(NC(=O)COCCF)C2)=O)c(F)cc(C)cc1Br N1(C(C(c2ccccc2F)(C)C)=O)CCN(C(c2ccc(C#N)s2)=O)C2CC12 CCC(C#N)C(=O)N1CC(C(F)(F)F)C(CNC(c2ncc(C)cn2)=O)C1 N1(C(C2(OC)CCCOC2)=O)CC2CCOCC2(NC(=O)CCCCCOC)C1 c1(NC(C2CCCN(C(C3CCC(C(F)(F)F)CC3)=O)CC2)=O)ccnc(F)c1F C(=O)(CCC(C)(C)C(=O)N1C2CCC1CC(NC(=O)C=CC1CCOC1)C2)OC N1(C(C23CCC(OC)C2C3)=O)CC(C(=O)NCCS(C)(=N)=O)CCC1C c1(C(=O)NC23CCC(CNC(=O)CC(F)(F)Cl)(OC2)C3)cncc2nc[nH]c12 C1(C(N2C(C)(COC)CC2)=O)(C(C)C)CCN(C(c2cc(OC)n[nH]2)=O)C1 C(CCC(C)C)(C(=O)O)N(CCC(C)CCNC(=O)OC(C)(C)C)C(C)(C)C(F)(F)F C1(NC(c2c(CC)ocn2)=O)CCN(C(=O)Cc2cncc(OC)c2)C(C)C1 C(=O)(CC(C)C(F)F)N(CCC(C)NC(c1c(C)oc(C(C)C)n1)=O)C c1(CC(=O)NCc2ccsc2C(N2CCC(O)(CO)C2)=O)cccc(O)c1 C1(c2n(C(CC)C)nnn2)(NCc2ccn(CC(F)(F)F)n2)CC2(C1)OCCO2 CC1(C)CC1(c1ccccc1)C(=O)NCCC1CC(NC(c2ccsn2)=O)C1 C(CCCCC(=O)N1CCCCC1C(C)NC(=O)Cc1ccc(SC)cc1)OC Cc1c(C(=O)NC(C)CC(C)NC(C2CCCC23CCC3)=O)cccc1F c1(C(N(CC(=C)C)C)=O)cc(CCNC(=O)CC2CCC2)on1 Cc1cc(C)c(C(N2CC3CC2CN3C(c2ccc(F)c(CO)c2)=O)=O)cn1 Cc1nc(=NC2CC3CN(C(=O)CCc4cc(Cl)cs4)CC23)s[nH]1 CC(C)C(C(=O)NCC(C)NC(c1nc(-c2ccccc2)on1)=O)n1cnnc1 c1(OC)cc(C(N2C3CCCC2CN(C(C2(C)CC2F)=O)C3)=O)ccc1[N+](=O)[O-] C=CC1(C(=O)NCc2cccnc2NC)CCN(C(C2C=CCC2)=O)CC1 CC(CNC(=O)CNc1ccccn1)C(=O)N(C1CCCCC1)CCC#N C1(C)(OCC)CCCN(C(C2CCCCCN2)=O)C1 C1(NC(C(C)C2CCOC2)=O)CCN(C(C2CC(C)(F)C2)=O)C1(C)C C(CC(C(N)=O)NC(=O)C(C)(C1CCC1)NC(=O)CC1COCCO1)OC C#Cc1ccc(NC(=O)C(=O)NCCc2sc(C)c(C)c2C)cc1 C1(C(=O)NC2CCN(C(CCOC)=O)C2)CNC(=O)CC1(C)C CCCCC(O)C(=O)NC(C)CCC(=O)NC1COCC1SC N#Cc1cn[nH]c1C(=O)NCC1CCC1NC(=O)C=Cc1cn[nH]c1 c1(C(=O)NCC(C2CC2)NC(C(C(C)C)F)=O)nncc2ccccc12 c1(NC(N2CCC(CN(C(C(C(C)C)NC(C)=O)=O)C)C2)=O)cnc(O)c(C)c1 N1(C(c2cc(C)sc2Br)=O)CCC2CCC12CNC(=O)CC(C)(C)C#N C(=O)(C(CO)C(F)(F)F)NC(CC(N1CC(COC)OCC1)=O)C S(=O)(=O)(c1c[nH]c(C(N2CCCCC2CNC(=O)C(F)SC)=O)c1)NC C1(C)(C(N2CCC(NC(C(F)OC)=O)C(CO)CC2)=O)COc2ccccc2O1 N1(C(CCCOCCC)=O)CC(CNC(=O)Cn2[nH]cnc2=N)C(C)C1 N1(C(c2c(C(C)C)onc2)=O)CCCC(CCNC(=O)CCC2CC2(C)C)C1 C1(NC(=O)COCCCF)COC2(CCN(C(=O)CN3CCCC3CO)CC2)C1 c1(CCC)nc(C)cc(=NCCCN(CC)CC2CCCC(C)C2)[nH]1 C(C)(CCC(=O)N1CC=CCO1)NC(C(CCC)C(C)C)=O CC(C)C1=NOC(C(=O)NC2COCCC2C(N2CC3(CO)CC3(CO)C2)=O)C1 C(CC(=O)N=S(C)(=O)CCNC(C)=O)c1ccc(OC)cc1 c1(C(=O)NC2CCCCN(C(c3c[nH]c(=N)s3)=O)C2)cncc2c(F)cccc12 c1(NC(C(CC)NC(=O)C(=O)NCCSc2cccs2)=O)ccnc(OCC)c1 C(=O)(CCCCCS(N)(=O)=O)N1C(CNC(COC)=O)CCC(C)C1 C(C)(CCCC(=O)Nc1cccc(C(C)F)c1)NC(C1(CC#C)CCC1)=O c1(C(N(C2CC(C(=O)NC3CC3Cl)C2)C)=O)ccncc1Cl C12(C(=O)NCCn3cccc(C)c3=O)CCOC1CC(=O)NC2 c1(C(N2CC(C)(NC(C3CC(N(C)C)C3)=O)C2)=O)ccc2c(n1)CCC2 C(=O)(C(C(=O)OC)OC)N1CC(NC(C)=O)C1.N12CCC(C1)CSCC2=O CC(O)C(C(=O)NC(C1CCCC1)CO)NC(C1CC2C=CC1O2)=O Cn1cc(C(N2CCN(C(=O)C=CCn3cncn3)CC2CF)=O)n(C)c1=O C1(CNC(CC2C(C)(C)C2)=O)CC(O)CN1C(c1ncsc1Br)=O c1(C(N2CC(C)N(C)CC2)C(=O)NC2CC(F)(F)C2)cccc2ccnn12 S(=O)(=O)(c1cc(C(=O)O)ccc1Br)NC(Cc1c(C)cc(C)cc1C)C(=O)O S(=O)(=O)(c1cnc(N2CCCC(CO)(CO)C2)c(Cl)c1)NCCCS(C)(=O)=O C1(C(C)C)CCN(C(c2c(Cl)cnn2C)C(=O)NC2COC2)CC1 C1(NC(c2ccc(C(=O)OCC)o2)c2nnnn2C)CC2CCC1CC2OCC c1(C(=O)NC2CCC(CNC(CC=C)=O)C2)cc(OC)ccc1[N+](=O)[O-] C(=O)(C(F)C(CC)CC)N1C2CC(CNC(C=CCN(C)CC)=O)C1CC2 C(=O)(CS(=O)(=O)NC)N(C1CCN(C(c2cc(CN(C)C)c[nH]2)=O)C1)CC C1(C)(C(=O)NC(C)CCNC(c2scnc2C(F)(F)F)=O)CCS(=O)(=O)CC1 Cc1cc(C=CC(N2CCN(C(=O)CC3OCCCO3)CC(O)C2)=O)ccc1F C1(NC(c2c(C(C)C)c[nH]n2)=O)CCC2CC1CN2C(c1cccc(C#N)n1)=O N1(C(C(CCC)C)=O)CCC2(CCC(CNC(=O)Cc3cn(C)nn3)OC2)CC1 C1(C2CCN(c3ncc4c(ccn4C)n3)CC2)(NC(CC(C=C)(C)C)=O)CC1 C1(NC(c2c(CC)ocn2)=O)CN(C(=O)CC(O)C(Cl)(Cl)Cl)CC(C)(C)C1 C1(C2(CC(=O)Nc3ccsc3)CC2)CCCCN1C(=O)CCc1ncccn1.CCC C12(C(=O)NC(CC=C)CNC(c3cccc(C4CC4)n3)=O)CC(C)(C1)OC2C N1(C(C(COC)N(C)C)=O)CC(C(=O)NC(c2nn[nH]n2)CC)C(C)(C)C1 c1(SCC)ccccc1C(N1CC(CNC(c2coc(C(C)=O)c2)=O)CC1C)=O c1(OC)cc(C(O)C(=O)NCC2(C(=O)NCC3CC3(C)C)CCC2)c(F)cc1O C1(C(=O)NCC2C(CNC(CC(CC)(F)F)=O)C2)CC2COCC(C1)C2 C12(NCC(=O)NCC(C)C(F)F)CCCC1N(C(=O)OC(C)(C)C)CCC2 C1(N(C(c2nn(C(F)F)cc2Cl)=O)CC)CCCN(C(=O)CC2CCC2)C1 c1(OC)ccc(C(N2CCC(CNC(c3ncccc3Cl)=O)CC2)=O)cc1F c1(CC(=O)NC2CCC(F)(CNC(C(N)=O)=O)C2)c[nH]c2nccc(Cl)c12 C1(NC(N2CC(CC(F)F)C2)=O)C=CCN1C(=O)CCCC1C(CO)C1 C(=O)(C1=NOCC1)NCC1(NC(C(CC)N(C)C)=O)CCOC1 N1(C(C2CN(C(C)=O)C2)=O)CC=C(C(=O)NCC2CCCC2(C)C)CC1 C(=O)(C(C)(C)c1ccsc1)NCC(CC)NC(=O)CCN1CCC(F)C1 c1(CC(=O)NC(CC)CNC(C2CCOCC2)=O)coc2cc3c(cc12)CCC3 Cc1cc(Cl)ccc1C(N1CCOCC1C(=O)NC(c1cccc(O)c1)(C)C)=O c1(OC)cccc(C(=O)NCCCN(C(=O)CC2CCOC2C)C2CC2)c1 C(c1ccccc1F)=CC(N1C(CN(C)C(C2CC3OC2C2CC32)=O)CCC1)=O N1(C(CCOC)=O)CCCC1(C)C(N1CCC(C(C)O)CC1)=O C=CCCC(CC(C)C)C(=O)NCC12CC(CC)(CN1C(=O)CC1CCOC1)C2 N1(C(C(C)n2ccnc2)=O)CCC(F)(CNC(c2cc(C3CCC3)nn2C)=O)C1 C1(c2nnc(CN3CCC(CC(=O)OC)C(F)(F)C3)o2)CCc2cnc(C)n2C1 C(C1CN(C(c2cnccc2C)=O)Cc2ccccc21)NC(C1CC(OC)C1)=O C1(F)(CNC(CC2(CNC(=O)CCc3nc[nH]n3)CC2)=O)CCCC1 c1(C(=O)NC(CC)CNC(=O)C(F)(F)C2CCCC2)nnn2cc(C)nc(O)c12 C1(NC(=O)CN2CCCS2(=O)=O)CCN(C(c2ccnnc2O)=O)CC1O C(=O)(CC(C)C(F)(F)F)NCC(CC(C)C)NC(c1cn2c(n1)CCC2)=O CCC(C)C(C)NC(=O)C(F)CC1CN(S(=O)(=O)CC2CCC2)C1 c1(CC)c(C(=O)NC2COCC2NC(C2CCS(=O)CC2)=O)cnn1C(C)(C)C CCC(CC(=O)NC(CNC(c1cnco1)=O)CC(F)(F)F)C(F)F C1(C(=O)NC(CC)CN(C(=O)CC(O)C(C)C)CC)CC2(CCOCC2)C1 N1(C(C2(C(C)=O)CCC2)=O)CCOC(C)(CNC(=O)C(F)(F)c2cccnc2)C1 c1(COC(=O)NCC(C(=O)OCC(C)O)O)ccc(CSc2ccccc2)cc1 N1(C(c2ccc(OC)nn2)=O)CCC(NC(c2ccccc2Cl)=O)C(CO)C1 c1(C(C(=O)NC2CCOC2)N(C(COC)(C)C)C)ccc(C(F)F)cn1 C1(C)(C(=O)NCC#CC(=O)N(CCCSC)C)C(C)(C)C1(C)C CCCCC(C)C(=O)N(CCN(C(c1cc(CC)cnc1O)=O)CC)CC C1(C(=O)NC(CCSC)CO)C2CC2CN1C(c1cccc(=O)o1)=O C12(C(=O)NCC3(F)CN(C(c4[nH]cc(C)c4)=O)C3)CCOC1CCOC2 C=CCN=C(NCCc1ccc(C(C)(C)C)o1)NCC1CCCN(C)C1 c1(C(N2C(CNC(c3ccc(SC)s3)=O)CCC2)=O)ccnc2ccc(O)cc12 C1(CNC(CC)=O)CCC12CN(C(=O)C(c1cc(Cl)cc(Cl)c1)O)C2 c1(OC)cc(C(N2CC(CC(C)NC(C3CC(=O)OC3(C)C)=O)C2)=O)ccc1O C1(C(=O)NCC2(C)CC(O)C2)CN(C(=O)CCC2(C#N)CCC2)CC1(F)F CCCC(C#N)C(=O)NC1(CNC(=O)Cn2cc(C3CC3)cn2)CCCCCC1 C(CCCC(=O)N1CCC=CC1C(=O)Nc1cncc(CO)c1)OCC c1(C(C(=O)NC(C2CN(C(=O)C3=COCC3)C2)C)C)cccc(Cl)c1 C1(c2nc(CNC(C(=O)NCC)=O)[nH]n2)CCN(C(=O)C(COC)SC)CC1 CCC(C)C(C)C(=O)N1CCC12CN(C(c1snc(O)c1Cl)=O)C2 Cc1ccnc(CCCNC(=O)C(c2ccns2)NC(C2CCS(=O)(=O)C2)=O)c1 C1(CNC(CC=C=C)=O)(CO)CCN(C(=O)Cc2[nH]cnc2C)CC1 CC1=C(C(=O)NC2C=CC(C(N3CCC(CCO)C3)=O)C2)COCC1 N(C1CCOc2ccc(Br)cc21)C(C1COCCN1S(=O)(=O)C1CCCCC1)=O N1(C(c2c(CC)onc2)=O)CCN(C)C(CNC(=O)CC2CCOCC2OC)C1 c1(C(N2C(CCCNC(C3=C(C)CC3)=O)CCC2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NCC(CC)NC(=O)CCn2ccc(=N)[nH]2)ccccc1F C1(NC(CCCOC)=O)CCN(C(=O)CCC(C)(C)N2CCCC2)C(C)C1 c1(C(=O)NCCc2cc(C(=O)NC3CC(C)OC3)no2)cncc(CCN)c1.C(=O)O C1(C2CC2)(CNC(=O)Cn2cncn2)CCN(C(c2cccc(Cl)c2)=O)C1 C(=O)(CC1CCc2ccccc21)NCC1(OC)CN(C(=O)CCn2cnnn2)C1 N1(C(c2nc(C)sc2)=O)CC2(CCN(C(c3ccc(CCF)cc3)=O)CC2)C1 c1(OC)ccc(NC(c2nnnn2C(C)(C)C)c2ncco2)cc1C(C)C C1(NC(c2cccc(O)c2)=O)CCCCCC1NC(C1CC1c1ccco1)=O C1(NC(C2(CSC)CCC2)=O)CCN(C(c2ncncc2C)=O)C(C)C1 c1(C(=O)NCCC2CCN(c3nccc(OC)n3)C2)c(Cl)sc(C)c1C C(=O)(C(O)C(C)(C)CC)NCC1(OCC)CN(C(c2cnc3sc(C)cn23)=O)C1 c1(C(CC)NC(C2C3CS(=O)(=O)CC23)=O)cc(OC)ccc1OC C#CC(CNC(C1CCCN(C(=O)C(C)N2CC(C)C2)C1C)=O)C(C)C CC1CN(C(c2cc[nH]c2C2CC2)=O)CCC1NC(C1CCC2CC2CC1)=O c1(C(=O)NC(C(C)NC(=O)C=C2CCCC2)(C)C)cc2nn[nH]c2cc1F C1(C(N(CCN(C)Cc2ccc(C)cc2Br)C)=O)CCc2ncnc(C)c2C1 C1(CNC(c2c(C)n(C(C)(C)C)nc2)=O)N(C(=O)C=CC2CC2)CCCC1(C)C c1(OC)ccc(C)c(C(=O)NC(C)(C)CNC(c2ccc(-c3cccs3)s2)=O)n1 C1(CNC(Cn2c(C)cnc2)=O)CC2(C1)CN(C(c1nc(Cl)sc1Cl)=O)C2 C1(CC(=O)NC(c2cccn2C2CC2)(C)C)CCN(C(C2(C)C(C)C2)=O)CC1 C(CCN(C)C(C)C)(CN=c1cc[nH]c(=NCCCOC(C)(C)C)[nH]1)OC c1(C(N2CCN(C(CNS(N)(=O)=O)=O)C(C(F)F)C2)=O)cc2c(F)cccc2[nH]1 C1(NC(CCn2ccc(C)n2)=O)CC2CC(NC(c3nnc(C)s3)=O)C2C1 Cc1nn2c(C)cccc2c1C(=O)NC(C)CNC(C1CC(n2cnnc2)C1)=O Cc1cc([N+](=O)[O-])cc(Cl)c1NC(N1CCC(C(N2CCOCC2)=O)CC1)=O CC(C)(C)CCCC(=O)N1CCC(C(=O)NCCC(Cl)Cl)C12CCC2 CCCCC(C)CCC(=O)NC1CN(C(=O)COCC2CC2)C(C)(C)C1 C(CC(CC)C(=O)NC1CC(C(C)NC(=O)Cc2c(C)nn(CC)c2C)C1)=CC C1(OC)CCCC(CC(=O)NC2(F)CN(C(COCCCCC)=O)C2)C1 CC(C)C(C)C(CNC(=O)COc1ccc(Cl)cc1)NC(=O)CC1(C)CCCC1 C1(NC(=O)CC2CCCN(C(C3CC(O)C(F)C3)=O)CC2)CCCC(O)C1O c1(N2CCCC(COC)C2)nc(N2CCC(S(C)(=O)=O)C2)c2ncn(C)c2n1 N1(C(C(CC=C)(C)C)=O)CCC(NC(c2cnc(O)s2)=O)C2(CCC2)C1 C(=O)(C(C)CCCC(C)C)NC1C=CC(C(=O)NCC2N(CC)CCC2)C1 C1(CCNC(C(F)=CCC)=O)CN(C(=O)Cc2cccc(C(F)(F)F)c2)CC1C c1(NC(C2CCN(c3nc(OC)c(C)cn3)CC2O)=O)cc(Br)cc(Br)c1O c1(C(N2CC(NC(CSC)=O)(CO)C2)=O)ccc(CSc2ccon2)cc1 c1(C(N2CC=CC(NC(=O)COC3CC(F)(F)C3)C2)=O)ccc2c(c1)OCCO2 C(N=c1[nH]cnc(=N)[nH]1)C1CCCC(NC(C(CC)OC2CCCC2)=O)C1 N1(C(CC2(C=C)CC2)=O)CC2(CC(C(=O)NCc3cc(OC)no3)C2)C1 c1(C(N2CCCC(NC(c3c(C)ncnc3)=O)CC2)=O)cnn2c1OCC(O)C2 C(=O)(C(C)(C)CC(C)C)N1CC(NC(CC=C(C)C)=O)C(C)(C)C1 c1(SCC(=O)NC2C(OCC)COC2)cccc(C(F)(F)F)c1.C1(=O)CO1 c1(CN(C(C(c2ccccc2)NC(CC(=O)NCC)=O)=O)C)ccncc1C CC1CCCN(C(c2cc(=O)cc(Cl)[nH]2)=O)C1CNC(c1c(N)ccnc1Cl)=O CCCCCCC(C)(CCC)C(=O)NC1CN(C(c2cc(C)n(C(C)C)n2)=O)C1 N1(C(C2(C(C)(C)OC)CC2)=O)CC2CCN(C(c3occ4c3CCOC4)=O)C2C1 N1(C(C=CC)=O)CC(NC(C2CCCOC2C(C)C)=O)C(c2cnn(C)c2)C1 c1(CC(=O)N(CC(CNC(CNS(CC)(=O)=O)=O)O)C)c[nH]c2cc(Cl)ccc12 C12(CNC(C3=CC(C)C3)=O)CCCC1CN(C(=O)CCN1CCCC1)C2 C(=O)(CS(=O)(=O)CC)NCC(C)N(C(=O)C=Cc1cncn1C)CC c1(C(=O)NCCNC(COCC#C)=O)ccc2occc2c1 N1(C(CSCC)=O)CCC(C(COC)NC(=O)CCC(=O)c2cnn(C)c2)CC1 CC#CCCCC(=O)N1CC(OC)C(NC(=O)CC2CCOCC2(C)C)C1 C1(NCc2ccc(OC(F)F)c(Br)c2)CCc2n[nH]cc2C1 c1(SCC(C(F)(F)F)c2ccccc2)cc(F)ccc1NCCc1ccccc1 N1(C(c2c(CC)c[nH]c2)=O)CC(O)CC1CNC(c1ccc(CO)s1)=O CCC(C(N)=O)n1cc(COC(=O)CC#N)nn1 C1(CC(=O)NCCCSCC)CCCN1C(c1ccn(C2CC2)n1)=O CCCC(CCCNC(c1sccc1CN(C)C)=O)NC(C1CNC(=O)N1)=O C1(NC(c2ccc(OC)cc2C)=O)CC2CC(C1)CN(C(=O)C1=C(Cl)CCC1)C2 Cc1cn(C)c2nc(N(C3CC(N)C3)Cc3nc(C(C)(C)C)cs3)ncc12 c1(C(N(CCCNC(=O)CC(O)C2CC2)CCC)=O)cnc(O)cc1C c1(N(C(CCc2cccc(C)c2)=O)C2CCNC2)ccn2ncc(Br)c2n1 C(=O)(CCCCCSC)NCC(CC(=O)NC(c1ccncc1)C)OC N1(C(c2sccc2Br)C(=O)NCCSC)CCCC2(CC1)CCN(C)CC2 C(=O)(C(CCC1CC1)NC(=O)C(=O)NCC(F)F)NCC1C(C)OCC1 N1(C(CCCC)=O)CC2CCCC1(CNC(c1ccc3ncccn13)=O)C2 C1(C(=O)NC(C2(OC)CCC2)C)CNC(=O)CN1C(c1ccc(O)c(C)c1)=O c1(OC)cc(C(N2CCC(NC(c3ccc(Cl)[nH]3)=O)C2)=O)ccc1Cl C1(NC(C(CCC)NC(C)=O)=O)CN(C(c2ccc(OC)o2)=O)CCC1C N1(C(CCN(CC)CC)=O)CCCC(CC)(NC(=O)CCc2cncs2)C1 c1(C(=O)NCCN(C(C=CC)=O)CCC)ccccc1Sc1ccccc1 c1(C(N2C(CNC(c3nnn(C)n3)=O)CC(C)(C)C2)=O)cc2cc(Cl)ccc2[nH]1 N1(C(C2CCCN2C(C2CCCC2)=O)=O)CC2(CCC2)C12CCC2 c1(CCN(C(c2cc(Cl)no2)C)C)ccccc1F c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)cc(-c2ccncc2)[nH]n1 Cc1ncc2n1CCC(C(=O)NC(C)CNC(=O)C=Cc1ccnn1C)C2 C1(C)(C(=O)NCCOCC)CC(O)CN1C(C1COCC(C)O1)=O N1(C(c2n(C=C)nnc2)=O)CC(C(=O)NC2C=CCC2)CC12CCC2 N(C1CC2(CN(C(=O)C(C)CF)C2)n2ccnc21)C(C(CCC)CCC)=O C(CCCCC(=O)N(C)CC1CCCN1C(=O)CC(C)n1ccnc1)=CC c1(-c2nnc(N(C(C#C)C)C)n2CC(C)C)ccc(C#N)cc1 C(CCF)(C(=O)NCCC1(O)CCCC1)NC(c1c(C)c[nH]c1)=O c1(C(=O)NCCOCCNC(C(N2CCCCC2=O)C)=O)ccc(O)cn1 c1(C(=O)NCC2(C)CN(C(=O)CC3CCCCC3)CCO2)ccn2c1CCCC2 Cn1cc2c(C(N3CCC3CNC(=O)C(O)C3CCC3)=O)cc(F)cc2n1 N1(C(Cn2c(C)nnn2)=O)CCC2(CC1)OCCC2NC(c1ncccc1Cl)=O c1(N(CC(C)OC)C)nc(N2CCC3CCC(C3)C2)c2ncccc2n1 c1(NC(CN(C(c2nc(CC)sc2)=O)C(C)C)=O)cnc2ccnn2c1 Cc1c(C(=O)NC(C2CCOC2)CNC(=O)COCC2CCC2)[nH]ccc1=O c1(CC(N2C(C)(C)C(NC(=O)C=CCN)CC2)=O)ccc2c(c1)CCCS2.CCC N1(CC(=O)NCC23C(CN(C(C=C(C)C(F)F)=O)C2)C3)CCc2ccccc21 N1(C(C=C(CCC)C)=O)CCC2CN(C(c3ccc(C(C)(C)C)o3)=O)CC12 c1(NC(C(C)(C)O)=O)cccc(C(N2CCCC(Nc3ncccn3)C2)=O)c1 CC1CCN(C(=O)C2=COCC2)C1CNC(c1cc(-c2ccco2)[nH]n1)=O CC1CCCCC1(CNC(c1cc[n+]([O-])cc1)=O)NC(C1C2CCC1CC2)=O c1(OC)ccccc1CCC1CCN(CC(=O)NCC(c2ccccc2)O)CC1 CCC(CC(=O)NC(c1ccc(C)cn1)C)NC(c1ccc[nH]1)=O CCCC(C#N)C(=O)N1CCC(C(=O)NCCc2cnn(C)c2C)C12CC2 CCC(F)(F)CC(=O)NC(C(N1CC(S(C)(=N)=O)C1)=O)C1CCOC1 c1(C2C(C(=O)NCC(CNC(CCC#C)=O)O)C2)ccc(C)c(C)c1 CC(CC(=O)N1CC2(NC(=O)CN(C)S(N)(=O)=O)CCCC2(F)C1)CC(F)(F)F c1(C(C)NC)c(O)cccc1F.c1(C2CS(=O)(=O)N2CCC)ccc(Cl)cc1F c1(C(=O)NC(CC=C)CNC(=O)C(CC)NC(C)=O)nn(C)c2c1CCC2 c1(C(N2CC(O)(C(=O)Nc3cc(C(=O)OCC)c(C)s3)C2)=O)cc(F)cnc1Cl O(NC(=O)CCOCCCNC(C1CC(O)C1)=O)C(C(=O)OC)(C)C C(C(C(=O)N1CCC(C)(F)CC1)C(C)C)NC(CC(CC)C1CCC1)=O c1(C(=O)NC2CCC(NC(C=CC)=O)CC2)ncc(F)cc1F c1(C(=O)NC(C)CCNC(=O)CN2C(=O)CCC2=O)nnn2c1CCC2 N1(C(C(C(C)C)CO)=O)CCN(C(=O)Cc2ccccc2F)C(c2cn[nH]c2)C1 C1(C(=O)Nc2cnc(OC)nc2)CC(F)(F)CN1C(=O)CCC(C)N(C)C c1(CC(C)NCc2c(COC)cccc2)ccc2ccccc2c1 N1(C(=O)Cc2cc[nH]n2)CCCC2(C1)CN(C(c1ccc3cc[nH]c3c1)=O)C2 c1(C(=O)NC2C(CNC(CCC=C)=O)COC2)ccc2c(c1)nc(C)n2C1CC1 C(C1=CCN(C(C2CC3C=CC2C3)=O)CC1)NC(COCC(=O)NC)=O C(=O)(CCCC(=O)N(C)C)NC(CNC(C(C)Nc1scc(C)n1)=O)(C)C(C)C C1(N(C(CCOCC#C)=O)C)CCN(C(=O)C(C)(C)NC(=O)OCC)C1 N1(C(C(C)OCCOC)=O)CCC2(CC1)CCN(C(=O)CCC(=O)OC1CC1)C2 C(=O)(C(F)C(C)CNC(c1cc(C)n(C)n1)=O)N(C)Cc1n(CC)ncc1 N1(C(C(=O)NCCCNS(NC)(=O)=O)=O)CCOCC1c1ncnn1C Cc1cc(Cl)cc(N)c1C(=O)NCC1(C)CCCN1C(C1(N2CCCC2)CC1)=O CC1CC(C(=O)N(CC(=O)NCCC(O)C(F)F)C2CC2)CN1C CC(CC(=O)NC1CC2(C1)CC2C(N1CC(S(C)=O)C1)=O)C(F)(F)F CCCC(C(=O)NC(C)(C)C(O)CO)NC(=O)CC(C)CN(C)C Cc1ccc(F)cc1C(=O)NC1CCCC1CNC(c1c(C)ncn1O)=O C1(CC(=O)N(CC=C)CC)CN(C(=O)C(C)c2cc[nH]n2)C(C)(C)C1 C(C(CNC(=O)C=Cc1ccco1)C(F)(F)F)NC(COC(CC)C)=O n1(COCC)nc(C)c(CC(=O)N(CC(C)NC(c2c[nH]c(=N)o2)=O)C)c1C C1(OC)(NC(N2CCC(Oc3nccc(C#N)n3)CC2)=O)CCC(C)(C)CC1 C1(C(=O)NC(C)(C)C(N2CCCC(CCO)C2)=O)CC(=O)CC(=O)C1 Cn1nc(C(=O)NCC(O)C(N2CCCC(CC3CC3)C2)=O)ccc1=O N1(C(CCC(C)C)=O)CC2CC(NC(C3(c4ccc(Cl)nc4)CC3)=O)CC2C1 c1(C(N(C2CCC(NC(c3c(C)cccc3C)=O)C2)C)=O)ccc(C)n(C)c1=O N1(C(C2CCN(C(C(CC(C)C)O)=O)CC2O)=O)CC2OCCOC2C1 C1(C(=O)OCC)C2CC(CN(C(=O)OC(C)(C)C)C2)N1C(=O)C(C)(O)C(C)(C)C CS(=O)(=O)c1cccnc1C(=O)NCC1CN(C(c2cnsc2)=O)C2CC12 c1(C(N(CC(C)N(C(CNC(CC)=O)=O)C)C)=O)ccsc1C(F)F C(=O)(C(C)C(F)(F)F)NC(CCCC)CNC(=O)CCNC(=O)OC(C)(C)C N1(C(C2=NOC(CNC(C(c3ccn(C)c3)C)=O)C2)=O)CC(O)CC1(C)C C(C(C)CC(=O)N(c1nn(C)cc1Br)C1CC1)(C(C)C)OC(C(CC)=CC)=O C(=O)(CC(C(F)F)N1CCOCC1)NCC1(C)CC(NC(=O)CC2(O)CCC2)C1 C1(NC(Cc2nc(COC)sc2)=O)CCN(C(=O)Cn2nc(C)nc2C)C(C)C1 C1(CC)CNC(=O)CN1C(C1(CNC(C2CC(OC)C2)=O)CCCO1)=O Cc1cc(C(=O)N(C)CCOCCN(C)C(c2cc(C)c(C)s2)=O)c(C)o1 C1(NC(CCc2cncc(C)c2)=O)CCN(Cc2ccsc2)C(C)C1 C#CCCCCCCC(=O)NCCC1CCN(C(=O)C=CC2CCC2)C(C)C1 C(=O)(C(C)C(O)C(C)C)NC(C(=O)N1C(CCC=C)CCC1)CC=CC N1(C(CCN(CC)CC)=O)C(CNC(=O)CC(O)CN(C)C)CC2CC12 CC1CCC(C(=O)N(C)CCOCCNC(c2cc[nH]n2)=O)O1 c1(C(=O)NCCNC(C2(CC)CCC2)=O)cc(F)cc(Br)c1O N1(C(C(CC(C)C)C(N)=O)=O)CCCC(C2CN(C(=O)CS(N)(=O)=O)C2)C1 C(CC(=O)N(C)CC1(OC)CCC1)(C(C)OC)NC(CCCOCC)=O C(CNC(=O)CC1=CCCC1)(C(C)C(C)C)NC(C=C(COC)C)=O c1(C(=O)NCCC(CNC(c2cnc(C)nc2)=O)O)cc2ccc(Cl)cn2c1 C1(CCC)(NC(C2CCC3(CC3)C2)=O)CCCN(C(c2cccc(N)c2F)=O)C1 N1(C(C(CC(C)C)ONC(=O)CC2CCOCC2)=O)CCC2(CCCO2)CC1 c1(C(N2C3C(NC(C(CC)OCC)=O)C(C3)C2)=O)cc2ccc(OC)nc2[nH]1 c1(CCC(=O)NC2(CC=C)CCN(C(=O)C(C)(C)OC)C2)cnc(C)nc1O C1(C(=O)NCC2C(NC(c3c(CC)cno3)=O)CCC2)CC1C1CCCC1 c1(OC)cc(C(=O)NC2CC(C)CN(C(=O)Cc3cncn3C)C2)cc(C)n1 N1(C(c2ccn(CC)c2C)=O)C2CCCC1CC(NC(=O)C(F)=CC1CC1)C2 C1(N(C)CCn2cccc2)CC2CCC(C1)N2CC(O)CCl C1(C(N2CCC(NC(c3csc(C)c3N)=O)(CO)C2)=O)CN2CCN1CC2C C(CO)(C(=O)NCC1(C(=O)NCC(C)OC(F)F)CCCC1)OC C1(c2ccccc2)(C(=O)NCC(CC)OC)CCNC1=O.C1(=O)C(C(C)C)N1 CCCCCC(=O)NC1CC(C)(NC(c2nnn(C)c2C)=O)C1 C1(OC)CC2CCC1(NC1CC3(CCC3)C1OC)C2(C)C Cc1ccc2[nH]c(C(=O)NC34CC(NC(C5(F)CCCC5)=O)(C3)C4)cc2c1 c1(N(C(C)C(=O)NC2CCN(CC3CCCCC3)CC2)C(C)=O)cccc2c1OCO2 CC1CN(C(=O)Nc2nc(-c3ccccc3)cs2)CCN1CC(F)F c1(CCC(=O)NC(C)CN(C)C(C2(NC(N)=O)CC2)=O)cccc(Cl)c1 c1(CC(=O)NC2CN(C(C(C)NC(CC)=O)=O)CC2F)csc2nccn12 c1(NC(=O)NCCc2c(OC)cccc2F)nn(C)c2ccccc12 C1(C(N(CCNC(c2c(C)n[nH]c2)=O)C(C)C)=O)CCC(C)CC1 CC1CN(C(=O)CC2CC(C)(C)CO2)CCC1CNC(=O)CN1CCN(C)CC1 CCCCCC(C)(C)C(=O)NCCN(C(=O)C(C)C(C)CC)CCOC c1(C(=O)NC(CC(C)NC(=O)CC#N)C)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 c1(NC2(CNC(C(C)N3CCC3)=O)CCCCC2C)ncnc2sccc12 N1(C(c2c(OC)nn(C)c2)=O)CC2(CCC(NCc3ccnc(Cl)c3)C2)C1 c1(C(=O)NC2C(NC(C3C(CC)CCO3)=O)C2)c(C)ccn1C N1(C(CSS(C)(=O)=O)=O)CCN(C(c2cccc(C3CC3)c2)=O)C(C2CCC2)C1 Cc1ccc(S(=O)(=O)NCC(=O)NC2CC(C(=O)NC3CC3C#N)C2)c(F)c1 CCCC(C#N)C(=O)N1CCC(C(C)(O)CNC(C2(O)CCCCCC2)=O)CC1 C=C1CC(C(F)(F)F)(C(=O)NCC(C)CNC(c2nncn2CC#N)=O)C1 N1(C(c2cc(F)cs2)=O)CCN(C(=O)C(O)C2CCCC2)C(c2cn[nH]c2)C1 CC(C)CC(O)CC(=O)N1CC(NC(c2ccc(C(F)F)o2)=O)C2(CCC2)C1 N1(C(c2c(SC)cccc2)=O)CCCC(C)(CNC(C23CC(N=[N+]=[N-])C2C3)=O)C1 C1(C2CCC2)(C(N2C3C(NC(C4(N(C)C)CC4)=O)CC(C3)C2)=O)CC1(F)F CC1(C)CCOC(CC(N2CC(NC(=O)CCCNC=O)C(O)C2)=O)C1 CC#CC1CCN(C(=O)CC2C3CC2N(C(C2CN4CCC2CC4)=O)C3)C1 C1(NC(C2ON=C(C)C2)=O)CC(C(=O)N(C2CCN(C)C2=O)C)CC1O C(C(C(=O)OCCc1nc(OC)ns1)N(C)C)OC C(CC(C)(C)NC(=O)CN1CCNC1=O)=CC(=O)N(CCCC)CCO c1(C(N2C3CC(CC(NC(C)=O)C3)C2)=O)ccc2nc(S)[nH]c2c1 Cc1cccc(CNC(C2CC(F)CN2Cc2ccc(C(N)=O)nc2)=O)n1 C(=O)(C(CNC(=O)CCc1ccn(C)n1)C(C)C)N1C(CC)CC(O)C1 c1(C2(C(=O)NC3C(OC)CN(C(C4CC5C=CC4O5)=O)C3)CC2)c(F)cccc1Cl C(=O)(C(C)CCCC(C)C)N1CCCC(CCNC(c2n(C=C)ncc2)=O)C1 O=C(C1OCCc2c(F)cccc21)NC1(c2ccc(F)nc2)CC1 CCCCC(O)C(C)C(=O)NC(CCC)C(O)C(=O)NC(C)Cn1cnnc1 N1(C(c2cnn(C)c2N)=O)CCN(C(C2CCOC2)=O)C(C2CCC2)C1 C1(C(N(C(CCCC)CO)CC)=O)CCN(C(=O)COCCC(C)C)CC1(C)C N1(C(c2c(CC)ccc(F)c2)=O)CCC2CCN(C(c3ccc[nH]3)=O)C2C1 c1(C(=O)NCC2(CNC(CC(CC)(F)F)=O)CCOCC2)nccn2nccc12 CC(N=c1[nH]c(=NCC2(CC(N)=O)CC2)[nH]c2cccnc12)c1csc(Br)c1 C1(NC(C(C(CC)C)C)=O)CCN(C(c2ccc(F)c(OC)c2F)=O)CC(O)C1 N1(C(CCSCCC)=O)CCC2(CCC2)C(CNC(=O)CCCC2CCCC2)C1 c1(CNC(CN(C(C2CC(O)(CC#C)C2)=O)CCC)=O)cc(C)cnc1F C1(C(=O)NCC2N(C(c3c(OC)nsc3OC)=O)CC2)CCCC2(C1)CC2(F)F C12(NC(C)C(c3ccccc3Cl)C)CCC(CF)(C1)OC2 c1(C(N2CC(O)(C(C)NC(C3CC(CF)C3)=O)C2)=O)ccnc(O)c1Br C1(C(=O)NC2CC(CNC(c3cc(O)ncn3)=O)C2)CCCC2(C1)CC2(F)F Cc1nn(C)c2c(NCC3CCCN(C)C3=O)nc(=NCCC(C)CO)[nH]c12 Nc1cnc(NCc2nc(Cl)ccc2Br)c(Cl)c1 C1(CNC(CC2CC(OCC)C2)=O)CCCC1NC(c1coc(C(C)OC)n1)=O N1(C(Cn2c(C)ncc2)=O)CCOCC1CN(C)C(c1cc(F)n(C)n1)=O c1(SCC(N2CC3C(NC(C(CSC)C)=O)C(C3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] n1(CC)nc(CN2CCC(N3CCC(N)C3)CC2)c(C)n1 c1(NC)cccc(C(N2CCOCC2CNC(C2CCCC2)=O)=O)n1 C(c1ccc(F)cc1)=CC(=O)NCC1(F)CCC(NC(c2c(C)scc2)=O)C1 c12ccoc1CNC1CC(C1)C(=O)N2.c1(C(=O)O)cnoc1C(F)(F)F C12(C(N(C(C)CNC(=O)COc3ccc(C#N)cc3)C)=O)CCCCC1OCC2 c1(N2CCCC(N(C(CN(C(COC)=O)C)=O)C)C2)cc(C)c(C#N)c(C)n1 c1(CCC(=O)NCC(CN(C(C=CCC)=O)CC)(C)C)cc(F)ccc1F N1(C(Cc2cn(C(C)C)nc2)=O)CCCC1(C)CNC(C1CC1C(C)(F)F)=O C(C1COc2ccccc21)c1n(CCN(C)CP(C)(C)=O)c(C(O)C2CC2)nn1 CC1CC(O)CCN(C(=O)C(Cn2ccnn2)NC(c2ccn(C)c(=O)c2)=O)C1 Cc1nc(N2CCOCC2)c2cc(C(=O)NC3(C)CC4CCC3C4)sc2n1 Nc1c(C(N2CC3C(CNC(C4CNC(=O)C4)=O)C3C2)=O)cnn1CCO Cc1cc(C)n(CCC(=O)N(C23CCC(CC2)C3)C)n1 C12(C(=O)NCc3ccc(C(C)NC(C4C5CCCC45)=O)cc3)CCC(CC1)OC2 c1(OC)cc(C(=O)NCC2(CNC(=O)CCCSC)CCC2)ccc1Cl C12(C(N(C3CCN(C)C3)C)=O)CC1CCN2C(=O)CCCNC(N)=O N1(CC(C)C)CCCC(C(N2CC(C)(NC(c3cnccc3N(C)C)=O)C2)=O)C1 C1(SC)CN(C(=O)Cc2cnns2)CC1NC(=O)C=C(C)C(F)F CC1CN(C(c2cnn(CC(F)F)n2)=O)CCN1C(C12CC1COC2(C)C)=O CC1N(C(=O)C(c2cn(C)nn2)NC(=O)CC23CCC(CC2)C3)CCOC1(C)C C(=O)(CC(CC)C(C)(C)C)N(CCC)CCNC(c1sc(C(F)(F)F)cc1C)=O CC1CCN(CC(N2CC=CC2C(=O)NCCc2ncccn2)=O)C1 C1(C(N2CCC(C)(NC(=O)Cc3cc[nH]n3)CC2)=O)CCn2c(cnc2Br)C1 CCCC(C(=O)OC)C(=O)NCc1ccsc1C(N1CCC(C)(C(N)=O)C1)=O c1(C(=O)NC2CC(C)N(C(c3ccc4occc4n3)=O)C2)ccc2c(c1)CCN2 c1(C(=O)NC(C(=O)NCC(CC)CC)C2CCCO2)ccc(C#N)c(C)n1 CC(CCC(=O)N(C)CC1(C)CCCO1)NC(=O)CCn1ccnn1 C1(NC(c2cc(CCO)on2)=O)CCN(C(c2ncccc2Br)=O)CC1O CCC(CC)CN=c1cc(C)nc(N2CCN3C(=O)CCC3C2)[nH]1 c1(C(=O)NCCCNC(C2CC(OC)CN2C(C)=O)=O)cnn2cccc2c1 N1(CC2CCC(C)O2)CC2CC(NC(c3cnn4c3CCC4)=O)CC1C2 C1(CC)(CO)CCN(c2ccnc(NCc3ccccc3OC(F)(F)F)n2)C1 c1(CC(=O)NC2(O)CN(C(CSCCN(CC)CC)=O)C2)ccc2c(c1)CCC2 c1(COCC2(CC)CC(NC3CCC3(c3nnnn3C)OC)C2)cccnc1C CC1CCOC(C(=O)NC2CCC(NC(=O)C3=CCC3)C2)C1 c1(C(=O)NCC(C2CC2)NC(=O)Cn2cccn2)cnc(CC2CC2)s1 C(C)(C)(CCCNC(C1(C#N)CC=CC1)=O)NC(C(C)Cc1ccco1)=O C1(NC(C(C(C)C)(C)C)=O)CCC2CC1CN2C(c1cc(N)c(Cl)c(O)n1)=O c1(C(=O)NCCCC2CCCN2C(c2ccsn2)=O)cnc(C(F)F)cn1 N1(C(C2(OC)CCOC2)=O)CCC(C(C)NC(=O)CN2CCNC(=O)C2)CC1 C1(CCNC(c2ncn(C(C)C)c2)=O)CN(C(=O)CC(C)n2ccnc2)CCO1 C1(NC(c2c(CC=C)cccc2)=O)CCCCN(C(C2CC(O)CN2C)=O)C1 c1(C(=O)NCCCCC)cc2cc(-c3cc(F)cc(F)c3O)cnc2[nH]1 N1(C(C(C)C)=O)CC(C)C(C)(CNC(=O)COCC2CCOCC2)C1 C1(CNC(C2CN(OC)C(=O)C2)=O)COC(C)(C)CN1C(c1ccncc1)=O C=Cn1nncc1C(N1CCC(C(F)CNC(=O)CCSCCCC)CC1)=O c1(OC(CC)C(=O)N2CCC2CNC(=O)CSC)ccc(CC(=O)OC)cc1 c1(C(N2CC(C)C(NC(=O)CC(F)(F)Cl)C2)=O)c[nH]c2c(F)cccc12 c1(C(N2CCC(CC(C)NC(C3CCC(F)(F)C3)=O)CC2)=O)cccc(N)c1F N1(C(C2C(C)C2)=O)CCC(c2cn[nH]c2)CC1.c1(OCCC(=O)N)ccccc1 c1(-n2c(Cn3nc(C)cc3C)nc(C(C)OC)n2)cc(Cl)nc(Cl)c1 C1(NC(c2ccc(OCC)cc2)=O)C2CCC1N(C(=O)CC1CCCCO1)C2 N1(C(CC2CC(OC)C2)=O)CCC2(CC1)CC2NC(=O)Cc1ccno1 C1(C(=O)NCC2CC(NC(CN(C3CC3)CC)=O)C2)CC1C1CCCCC1 C(=O)(C(C#N)C(C)(C)C)NCC1CCN(C(C(C)CC2CC2)=O)CC1C c1(C(=O)OC(C(=O)NCCC2CCC(C)O2)=O)ccc(C(F)(F)F)cn1 CC1CCCC(C)N1C(C1CC1C(=O)Nc1ccc(C2CCCN2)cc1)=O n1(CC(=O)NCCC2CCN(C(CCCSC)=O)CC2)cccc(O)c1=O C1(C)(C(=O)OC)CCC1(C)C(=O)NCC1CC(C)N(C(c2cn(C)c(C)n2)=O)C1 C12(C(=O)NCc3ccc(S(N)(=O)=O)s3)CN3CN(CN(C3)C1)C2 C#CCC(CC(F)F)NC(=O)C(CNC(c1cnncc1C)=O)CCC N1(C(C(CC)(F)F)=O)CCC2(CCC2)C(CNC(=O)C(CC)NC(N)=O)C1 c1(C(N(c2ccccc2C(=O)O)C(C2C(C)(C)C2)=O)=O)cc(F)cc(F)c1 C1(C(C)(C)NC(CCC)=O)CCCN1C(=O)C(C)OCCC(C)C C1(C)(C(=O)NCC(CN(C(c2c(C)csc2)=O)C)(C)C)CCCCC1C c1(-c2cn(CC(=O)NCC3(OC)CCCOC3)nn2)c(F)cncc1F C(=O)(C1=CCN(C)C1)N1C(CC(N2C(CC)CC(O)C2)=O)CCCC1 N1(C(C2N(C(c3c(C)cccn3)=O)C(C)C2)=O)CCCC(O)(CO)C1 N1(C(CN2C(=O)CC2)=O)CCN(C(c2sncc2Br)=O)C(CO)C1 C(=O)(C(F)(F)CC(C)C)NC1C(NC(C(F)OC)=O)CCCC1 C(C(=O)NC(=O)CCC(C)c1ccccc1)(C(C)C)n1ccc(C)c1 C1(O)(CN(C)C(c2ccnn2-c2ccncc2)=O)CCCN(C(=O)CC2CC2)C1 C(N=c1ccnc(C(C)(C)C)[nH]1)C1CC(NC(C2(CC)CC2)=O)C1 C1(NC(C(CCOC)C)=O)CC2CCC1CN(C(c1ccc(Br)cc1C)=O)C2 c1(CC)nnc(CNC(c2cn(CCNC(=O)Cc3nnnn3C)cn2)=O)s1 C1(NC(CN(C)C)=O)CC2(C1)CC(C(=O)Nc1cccc(Cl)c1Br)C2 C1(C(N(CCCN(C)C(C2CC2CF)=O)C)=O)CCn2c(cnc2Br)C1 c1(OC)ccc(C)c(NC(c2ncccc2-c2ccc(C)nc2OC(C)C)=O)c1 c1(C(=O)NCCN(C(Cc2cn(CC)nc2)=O)C(C)C)cc(OC)cc(Cl)c1O CC(CNCC1CC1)C(=O)NC1(c2ccco2)CC1 CC1(C)CN(C(=O)CCc2ccc(Cl)nc2)CC1NC(=O)CCC1CCCOC1 C(c1ccoc1)=CC(=O)NCC(CNC(CCOCC(C)C)=O)O C1(CC(=O)N(C2CCCC2C#N)C)CN(C(c2cncs2)=O)C(C)(C)C1 c1(Cc2cnc(NC(=O)CCC3CCCOC3)s2)ccc(O)cn1 C1(CNC(C=Cc2ccc(C)s2)=O)CN(C(=O)CCc2ccsc2)CCC1C c1(N2CCC(C)(COC)CC2)cccc(S(=O)(=O)N(CC2=CCCOC2)C)n1 C(=O)(C(F)(F)CCn1ccnn1)NCC(CNC(=O)C(F)OC(F)(F)F)O c1(C(=O)NC2C(NC(CCc3cc(OC)no3)=O)CCC2)ccc2cnnn2c1 C1(CNC(C2C(CNC(CN3CC(C)(C)C3)=O)CCO2)=O)CC2(CCC2O)C1 CC1CCCC(C)N(C(=O)C(=O)NCCCC#N)C1 c1(C(=O)NC(CCOC)CNC(=O)C=C(C)Cl)cc(N)ccc1Cl C#Cc1ccc(NC(C)C(=O)NCCC(C)(C)C)cc1Cl C1(C(=O)NCCOCCC=C)C(C)CN1C(=O)CCCN(C)C N1(C(c2[nH]cc(C#N)c2)=O)C2CCC1CN(C(=O)CC(F)(F)F)C2 N1(C(c2cnc(C(C)C)nc2)=O)CC(NC(=O)CCC2CCCO2)C(C)(C)C1 C1(NC(=O)Cc2csc(Cl)c2)CS(=O)(=O)CC1NC(c1cnoc1C1CC1)=O C1(c2cn(CC(C)O)nn2)N(C(c2ccn3ncnc3c2)=O)CC12CCOCC2 c1(C(N2CCCC(CNC(C(C)C3CCCC3)=O)C2)=O)ccc2c(c1)NCC2 CC(CCO)(C(=O)O)N(C(=O)CCc1cn(-c2cccc(C(F)(F)F)c2)nn1)CCl C1(CNC(CC(C)(C)N(C(=O)C=CC(C)(C)C)C)=O)OC(=O)NC1(C)C C1(C(=O)NCCn2ccc(C)n2)CC(C)CN(C(=O)CCCF)C1 C1(CC)N2C=CN=CC23CC(=O)N(C)C(C)(CNC1=O)CC(CC)CC3 Cc1[nH]c(=N)nc(O)c1CCC(=O)NC1(CNC(C2(C)CCCC2C)=O)CCC1 c1(CC(=O)NCC2C(NC(C3CCC(C)O3)=O)COC2)cc(F)c(F)cc1F C1(CC(=O)NC(CC=C)CC)CN(C(=O)Cn2ccc(C)c2)CCC1(C)C Cc1cc(C)n(C(C)C(=O)NC(CO)C(C)NC(=O)CSc2nncs2)n1 N1(C(C2C(C=C)OCCC2)=O)CC(F)(F)CC1(C)CNC(=O)CC1CCOCC1 C1(NC(C(C)NC(N)=O)=O)CCN(C(C23CCC(C#N)(CC2)CC3)=O)CC1(C)C C1(C(c2nnnn2CCC)NCC(=C)Br)CC12CCC(F)(F)CC2 c1(C(N2CCC(CN(C(=O)C3=NNC(=O)C3)C)C2)=O)ccc2oc(O)nc2c1 c1(SC)nc(=NCC2(C)CCC(NC(c3cc(C(C)C)nc(O)c3)=O)CC2)s[nH]1 C1(CC(N2CCC(C)(NC(c3c(NCC)nccc3)=O)C2)=O)CCC(C)(C)CC1 Cc1scc(C(=O)N(CCCCNC(=O)C(O)C2CC2)C)c1Br c1(CC(c2nc(C3(C)CC3)n[nH]2)C)cnc(CN)nc1 C(=O)(C1CCc2cccc(O)c21)NCC1C(NC(c2cnn(CCF)c2)=O)CC1 c1(CC(=O)NC2CCN(C(C(COCC)C)=O)C2C(C)C)c[nH]c2cccnc12 N1(C(c2cn(C)nc2C(F)F)=O)CC(F)(F)CC1C(=O)Nc1ncc(F)cc1F C1CCC2CCCC2O1.c12cccc(c1)C(=O)N1CC(c3cn-2nn3)C1.C=CC C(CCCCC(=O)NC1CCCCC1N(C)C(c1cc(C2CC2)[nH]n1)=O)=CC c1(C(=O)NC2CC(NC(C(C=C)(C)C)=O)C2)nsc2ccc(OC)cc12 C(CN=c1nc(SC2CCCC2)[nH]s1)C1(NC(C2=C(C)OCC2)=O)CCC1 C1(C(=O)C(CNCCOCCO)OC)(C(=O)N(CCOC)CC)CCOCC1 O=C(C1CCCn2nccc21)N1CC(C2(NC(C3CC(C=C(F)F)C3)=O)CC2)C1 C1(NC(c2c(C)c(Cl)ccc2)=O)COC2(C1)CN(C(=O)CC(C)P(C)(C)=O)C2 CC1CCOC1C(=O)NC(C1(O)CN(C(c2c[nH]c(=N)o2)=O)C1)C C(C(C)(C(N)=O)NC(c1cnn(CCNC(=O)CCn2cc(C)cn2)c1)=O)OC c1(OC)ncc(C(=O)NC2CC(CNC(C3CCS(=O)CC3)=O)C(O)C2)cn1 C1(C(=O)NCCCN(C(c2cn(C3CC3)nc2C)=O)CC)CCC(C)(C)OC1 N1(C(CNC(C)=O)=O)C2CCCC1CN(C(=O)CC(=O)NCC(C)(C)C)C2 N1(c2ccc(C)cn2)CC2(CCC(NC(c3cc(-c4ccsc4)[nH]n3)=O)CC2)C1 c1(C(N2CC(CNC(=O)CC3CC=CC3)C3C2C3)=O)cc(Cl)cc(Br)c1 c12ccc(o1)S(=O)(=O)N2.C#CCCC(=O)NC1(CN(C)C(=O)OC(C)(C)C)CC1 c1(C(=O)NCC2CN(C(c3c(C)onc3)=O)C3C2C3)cccc2ncnn12 C1(C)(C(=O)NCC(NOCC(CC)C)=O)CC(=O)N(C)C1 c1(C(=O)NCC23CC2CN(C(C2CC24CCNCC4)=O)C3)cc(Cl)ccc1O N1(C(c2cn(C)nn2)=O)CC2ON=C(CNC(C34CC(F)(C3)C4)=O)C2C1 Cc1ccc(CC(=O)NCCC(C)NC(c2ccc(=O)n(C)n2)=O)cc1Cl Cc1cnn(CC(=O)N(C)Cc2cnc(SC3CC3)[nH]2)c(=O)c1 C(CCCC(C)NC(=O)CS(N)(=O)=O)NC(Cc1nc(C)sc1)=O C1(CNC(C=C(C)Cl)=O)CN(C(=O)Cc2cnnn2C)CC(C)(C)O1 C1(C(=O)NC(C2CCC2)C)Cc2nccnc2CN1C(=O)C1=NN(C)C(=O)CC1 CC1=CC(F)(NC(=O)CC2(NC(=O)CC3CCOC(C)(C)C3)CCC2)C(F)=C1 Cc1cc([N+](=O)[O-])nn1CC(=O)NCC12CC(CN1C(=O)C=Cc1ccoc1)C2 Cc1ccn(CC(=O)NC2CCC(C)N(C(c3scc(C)c3C)=O)C2)c(=O)c1 N1(C(C(CCOC)C)=O)CC2CCCN(C(C34CCCC3C4(F)F)=O)C2C1 c1(C(=O)NC2CN(C(C(C)OC)=O)CC2C)c(F)c(F)c(F)c(F)c1F Cc1ccc2sc(C(=O)NC34CCCN(C(=O)C=CC(F)(F)F)CC3C4)cc2c1 C(C)(CN=c1cc(Cl)nc(C2CC2)[nH]1)NC(c1cc(C)n(C2CCOCC2)n1)=O N1(C(CCOC)=O)CCCCC1CN(C)C(c1ccc(C2COC2)cc1)=O CC1(F)CN(C(=O)Cc2cccc3c2OCO3)CCN(C(c2n[nH]c(O)n2)=O)C1 N1(Cc2cccc(C(C)(C)C)c2)CCC(F)(F)C(NC(=O)Cn2cccn2)C1 c1(CC(C)C)nc2cccc(C(=O)Nc3ccc(F)cc3CO)c2[nH]1 N1(C(c2c[nH]c(=O)cn2)=O)CCOC2(CCN(C(=O)C3CC3)CC2)C1 C1(C(=O)NC(C(=O)NC2CCC(O)CC2)C2(C)CC2)CC2CCC1CC2 C(=O)(CCCNC(=O)C=CCN(C)C)NCC(CC)NC(=O)Nc1ccccc1 N1(C(c2cncc(SC)c2)=O)CC(O)(C2(CNC(=O)CCOCC(F)F)CC2)C1 c1(C(N2CCC(CC=C)(NC(c3cscn3)=O)C2)=O)nc(C2CC2)ncc1Br CCCC(C(=O)O)N(C)C(C1CCN(Cc2cnn(CCF)c2)CC1)=O N1(C(c2cc(C)[nH]c2C)=O)CC2(CC2)CC1C(=O)NCC(C)(C)N(C)C C1(C(N2C(C)(CCC)CC2)=O)CCCN(C(=O)CC(C)COC)C1CC CC1(C)OC2C3CCC(C2O1)N3C(c1cc(I)ccc1Cl)=O C1(NC(C(C(CC)C)C)=O)C(C)(C)CN(C(=O)Cc2ccoc2)CC1(C)C C1(C(=O)NCC(C2CCC2)NC(CSCCC)=O)CCC1C(C)(C)C C(=O)(C(C)P(C)(C)=O)NCC(CCOC)NC(c1cc(C(=O)N(C)C)on1)=O N1(C(CC2ON=C(C)C2)=O)CCC2(CC1)CCN(C(C1CCCC1CF)=O)CC2 N1(C(c2cc(O)cc(O)c2)=O)CC2CCN(Cc3cc(F)c(Cl)cc3O)C2C1 c1(C(N2CC(N(C)C(C3(C#N)CCOC3)=O)C2)=O)ncc(F)cc1F c1(SC)nc(C(C)C)nc(C)c1C(=O)NCCC1(C)CCC(=O)N1 N1(C(C2C(C(C)C)OCC2)=O)CCC2CC12C(N1CCN(CCF)CC1)=O N1(C(c2cccc(-n3ccc(C)n3)c2)=O)CCCCC(N(C)C(C2CC2C)=O)C1 c1(C(N2CC(C(C(=O)NC(CC(C)C)C)O)C2)=O)cccc(O)n1 N#Cc1c[nH]c2ncnc(Nc3ccc4c(c3)CN(C(c3ccccc3)=O)C4)c12 C1(N(C(C(C2CCOC2)OC)=O)C)CCN(C(C2(C)C=CCC2)=O)CC1 C1(OC)CCCCC1CC(=O)N(C)CCC1CCN(C(=O)C=CC=C(Cl)Cl)CC1 C1(NC(Cc2scc(C)c2)=O)CCN(C(c2cnc(N)cn2)=O)C1C N1(C(c2c(C)cc(C)cc2O)=O)CCN(C(=O)C(C(C)O)N(C)C)CC2(CC2)C1 C1(C(N2CC(NC(=O)NC(C)C(=O)NC3CC3)C2)=O)CC2(C1)OCCO2 CCC(C)CCCCC(=O)NCC1(C)CN(C(C2(C)CS(=O)(=O)C2)=O)CC1C CN1CC(C(=O)NCC2(NC(C3CC4C=CC3C4)=O)CC2)NC1=O c1(OC)ccccc1CNC(=O)C(O)CNC(=O)Cc1cccn1C N1(CC2(NC(C3CCC3)=O)CC2)CCN(C(C2(C3CCCCO3)CC2)=O)CC1 CC1(C(=O)NCCCN(C(=O)Cc2csnn2)CCO)CC2(CC(=O)C2)C1 CC(C)CC(CNC(=O)Cc1ccccc1)NC(c1cnc[nH]1)=O N1(C(c2cc(F)cc(C)c2N)=O)CC2COCCC2(NC(=O)C2=CCCSC2)C1 CC(CC(C)NC(c1cc(C2CCCN2C)[nH]n1)=O)N=c1[nH]nc(C2CC2)o1 Cc1cc(C(=O)NC2CCOCC2NC(C2CCCCC23CC3)=O)c(C)n1C C(CCC)(C(=O)N(CCS(C)(=O)=O)C)NC(c1cn(CCC)nc1)=O c1(C(=O)NC(CN(C(C2C(C)(C(=O)OC)C2)=O)C)C)nccn2c(Br)cnc12 c1(C(=O)NC(CC)CNC(c2cncc(C)c2Cl)=O)coc2c1C(=O)NCCC2 C1(CC(N2CC(C)C(NC(C3CCC(=O)N3C)=O)C2)=O)CCCC(C)(C)O1 CC(=O)C(C)CC(C)C(=O)NCC(CC(C)C)NC(c1cncn1C(C)C)=O C1(CC(=O)NCC2CCC(NC(C(C=C)(C)C)=O)C2)CC2CCC1CC2 C1(C(=O)NC(c2cccnc2)CC)N(C(=O)C(CC2CC2)OC)CCCC1(C)C c1(OC)cc(OC)n2[nH]c(=NC(=O)NC(c3cncnc3)C)nc2n1 c1(C(=O)NCC2CN(C(=O)CCn3ccnc3)CCO2)cnc2ncc(Cl)cn12 c1(C(=O)NCC2(NC(c3n(CCC)ncc3)=O)COC2)ccc(F)cc1OC c1(C(=O)NC2C(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CC2)cnn2c1OCC(O)C2 c1(OC)cnc(C(=O)NCCC2(NC(=O)CCC(N)=O)CC2)nc1 c1(C(N2CCCC(c3cn(CCCOC)nn3)C2)=O)cc(C)nc(Cl)c1 C1(C(N2CCC(NC(COCCCC)=O)(CO)C2)=O)CCC2(CCC2)OC1 N1(C(C2N(C(CC(CC)O)=O)CCC2C)=O)CCCCC(C)(C)C1 C1(Cl)(C(=O)NC(C)CNC(c2ccon2)=O)CC1(C)C c1(CC(=O)NC2CCC(Cn3cc(CCN4CCOCC4)nn3)C2)nc(=O)o[nH]1 c1(C(C)C)ncc(Br)c(N(C2CCCCCC2)CCNC(=O)C2=CCCOC2)n1 c1(C(N2CC(CNC(C3C(C)CCS3)=O)C2)=O)ccnc(-c2ccccn2)c1 CC(CC(=O)NC1CN(C(c2cc3cnn(CCO)c3n2Br)=O)C1)CC(C)(C)C C1(NC(C2C(C)C2)=O)CC12CCN(C(c1c[nH]c(C#N)c1)=O)C2 C(=O)(C1COc2ccc(Cl)cc21)NC1CC(C)(NC(c2cccn2C2CC2)=O)C1 C1(C(=O)NCC2C(OCC)CN(C(C3(OC)CCC3)=O)C2)CCCC(F)(F)C1 c1(Sc2c(C(=O)NCC(CC)NC(C3(OC)CCOC3)=O)scc2)ccccc1Cl c1(CNC(c2c(C)c(F)ccc2)=O)nc2c(s1)CCN(C(=O)CC(C)(C)O)C2 c1(CC)[nH]nc(Cl)c1C(=O)NC1CCN(c2cnc(-c3ccccc3)nc2)C1 C1(CC(=O)NCC#CCNC(c2ccc(C(C)(C)C)s2)=O)CN2CCC1CC2 CC1(C)CCOC1CCNC1CCOC1 c1(-n2cc(C(CCC)NC(=O)CC(C)(C)O)nn2)cc(Br)c(F)cc1F c1(CNC(c2c(Cl)c(C)nn2C)c2n(CCCC)nnn2)cccc(F)c1I C1(CCNS(NC)(=O)=O)CCc2c(OC)cccc2C1CC Cn1cnc2c1CCCC2C(=O)NCC1(F)CCN(C(=O)CCCC2CCC2)C1 c1(CC)ccccc1CN(C(=O)C(=O)NC(C1(Cc2ccccc2F)CC1)C)C N1(C(c2ccc(CC)cn2)=O)CCC(C)(C)C1CC(=O)NC1CN(C)CC1C N12CCC(c3nnnn3C3CC3)(C(C)C1)Nc1cnn(c1)C1CN2C1.CC C1(=O)C(C(C)C)N(C2CC2)CCN1C(C)=O.C(c1ccccc1)=CCNC(C)(C)C C1(C)(N(C2CCCC2)CC(=O)N(C(CSC)=O)C(C)(C)C)CC(C)=NO1.C1CS1 C1(CC#C)CN(N2CCN(C(=O)Cc3ccc(OC)cc3)CC2)C1 C(=O)(C(C)(C)CCC#N)NCC(C)N(C(c1ccc(C(=O)NC)s1)=O)CC CCN=c1[nH]c(C)c(C(N2CCN(C(c3cn(C)cc3C)=O)CC2C2CC2)=O)s1 c1(C(C)NC2CCN(C(=O)C(F)Br)C2)cc(F)c(Cl)cc1Cl S(=O)(=O)(c1cccc(S(=O)(=O)Nc2cc(Cl)cc(I)c2)c1)N(C1CCCC1)C N1(C(=O)CCn2cc(-c3ccc4nc[nH]c4c3)nn2)CCC(=C(F)F)CC1 C1(NC(C=Cc2n(C)ncc2)=O)CC2(C1)CC(NC(C1CC1C(C)(C)C)=O)C2 c1(C(C)(C)C)n[nH]c(=NC2CCCN(C(c3cccn4nnnc34)=O)CC2)s1 C=CC1OCCCC1C(=O)NCc1cn(CCNC(=O)C(CC)C(C)C)nn1 C1(CNC(CCN(CCC)C)=O)CN(C)CCN1C(=O)CC1COC(=O)C1 C1(C(=O)NCC2(NC(C(C)CCO)=O)CC2)CC2CC1C1CC21 C(=O)(CCCCCCC(=O)C(CCCC(=O)O)=O)OC.N1CCC(N2CCC2)CC1 N1(C(C2C(CC)CCC2)=O)CC2(C1)CN(C(C1CCCCS1)=O)C2 C1(OC)CC2CCC1(C(=O)NC1C3CC(NC(c4sccc4CO)=O)CC13)C2 Cn1nc(C(C)(C)C)cc1C(=O)NC1COCCC1NC(=O)CC1CCOC1 N1(CC)CCOC(C(=O)N(C)CCOCCNC(=O)C(c2nc(C)cs2)C)C1 c1(C(N2C(CNC(c3n(CCC)ncc3)=O)C(C)CC2)=O)cc2n(c1)CCSC2 c1(OC)cc(Cl)ccc1CCCNC(c1nc(Cl)sc1Cl)=O c1(OC)nsc(C(N2CCOCC2C2CCOC2)C(=O)NC(C)C)c1Cl CCC(CNC(C1CCSC(C)C1)=O)(CC)C(=O)NCCC1OCCC1(C)C C(=O)(CN=c1cc[nH]cc1)N1CCN(C(c2cccc(C(=O)NC)c2)=O)C2C1C2 C1(NC(C2C(c3n(C)ccn3)C2)=O)CCCC(NC(c2ccoc2)=O)CC1 N1(C(C=CC(C)(C)NC(C(=O)NC(C)C2CC2)=O)=O)CCC(CCO)CC1 C1(CC(=O)NC(C2CC(NC(=O)CN(C3CCSCC3)C)C2)C)CCCC1O CCC(C)C(C(=O)NC1CC(NC(c2nnn(C)c2C(F)F)=O)C1)NC(=O)OC c1(C(c2n(CCC)nnn2)NCC(C)(C)OCC2CC2)nc(F)ccc1Br c1(CC)cc(C(=O)N(CCC(=O)N2CC(C(=O)OC)C2)CC)nn1C C1(NC(C2CC23CCC3)=O)CC2CN(C(=O)CN3CCCNC3=O)CC12 C1(CNC(c2c(C)cc[nH]2)=O)CC(C)(C)CCC1NC(c1cccn(C)c1=O)=O C1(CNC(c2c(CC)onc2C)=O)CCN(C(C2(O)CC(F)(F)C2)=O)CC1(F)F C(=O)(CS(=O)(=O)C1CCCN(C(=O)C(C2(O)CCCCC2)OC)C1)OC CCC(CC)(CO)C(=O)N1CC2CC(NC(=O)CC3CCCC3C)CC2C1 C(C(O)C(=O)NC(C)(C)CCF)NC(C1(OC(C)=O)CC1)=O c1(C(N2CC3C(CNC(CNC(CCCCC)=O)=O)(C3)C2)=O)ccc(N)cc1F N1(C(Cn2ncc(C(N)=O)c2)=O)CCN(Cc2cccc(F)c2)C(=O)C1 c1(C(C)C)cnc(=NNC(=O)CC2CCN(S(N)(=O)=O)CC2)[nH]c1 c1(N(CCC)C)ccc(C(=O)NCCC(C)N(C(=O)CN2CCCC2=O)C)cc1 C12CCCN(CC1)C2=O.c12cnnn1C(C)C(=S)C(C(C(C)C)O)CCN(C)C2=O C1(NC(c2c(C)cc(F)s2)=O)C2CC3C(C2)C13C(=O)NC1(C)CCCCC1 n1(C(C)(C)C)cnc(C(=O)NCC2CC(CNC(C3CC3F)=O)CO2)n1 c1(N(C)C)cnccc1C(=O)N(C(CNC(c1ccc(C2CC2)s1)=O)C1CC1)C c1(OC)c(C(=O)N(C)CCOCCNC(C2CC(F)(F)C2)=O)c(C)nn1C N1(C(C=C(CCC)C)=O)CC2(CCC2)CCC1CNC(=O)CC1CCC(O)C1 N1(C(C2ON=C(CC)C2)=O)CCCC2(CCN(C(=O)Cc3cnn(C)n3)C2)C1 C1(NC(C(C)SCc2ccccc2)=O)CC2CCC1N2 CC1CCC=C1C(=O)NCC1CC(F)(CNC(c2sc(C#N)cc2Cl)=O)C1 C(=O)(C1CC(=O)Nc2cc(F)ccc21)NC1CC(NC(c2onc(C)c2C)=O)C1 c1(C(=O)NCCN(C(CC(CC)C)=O)CC(C)O)cc(NC)nc2ccccc12 C1(C(=O)NC2C(C)(C)C(CC(=O)NCCN3CCCOC3=O)C2)CC2(CCO1)CC2 c1(COC)n[nH]c(=NCC2CC(C)N(C(C3CN4CCC3CC4)=O)C2)s1 C1(NC(CCC2CCC(C)O2)=O)CCN(CCNC(=O)Cc2cccn2C)CC1 CC1CCCC1CC(=O)NC(C)(C)C.N1(C(C2C(C)CC2)=O)CC(C(=O)O)(CF)C1 CCC(C)(C)C(=O)N1CCCC(C(C)(O)CNC(c2ccc(OC)nc2)=O)C1 c1(C(=O)NC2C(C(=O)NCc3cccc(OC)c3)C2)c(F)c(F)c(F)c(F)c1F c1(C(=O)NCCCCCN(C(c2ccc(CC)cc2)=O)C)nccc(Cl)c1Cl C12(C(N3C(C)CC(NC(=O)CCc4cncs4)C3)=O)CC3CC(C1)CC(C)(C3)C2 c1(OC)ccc(F)cc1CC(=O)NC1CC(C)N(C(c2ncc(Cl)cc2F)=O)C1 c1(C(=O)NC2C(CNC(C(C)(C)SC)=O)C2)cc(C)n(-c2ccccc2)n1 C1(CCNC(C(SC)SC)=O)CCN(C(c2nnc(C(C)C)s2)=O)CC1 c1(C(N2C(CNC(C3(OC)CC3)=O)CC3(CC3)C2)=O)ccc(N)c2ccncc12 CC(C)C(C)(CNC(=O)CNC(=O)CN(C)C)NC(=O)C=Cc1nnn(C)n1 N1(C(C(C2CCC2)OC)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)C(C)C1 N1(C(C2N(CCC)CCC2)=O)CCCCC1CC(N1CC2CC1C2)=O n1(C(C(=O)N(CC(CC)NC(C2(C3CCCO3)CC2)=O)C)C)ccc(C)n1 Cc1nc(O)nc(O)c1CC(N1CCOCC(CNC(c2occc2Br)=O)C1)=O C(=O)(C1=CCS(=O)(=O)C1)N1C(CNC(=O)CCN2CCC(O)CC2)CCC(C)C1 c1(C(N2C(C)(c3ccc(Cl)cc3)CCCC2)=O)cnn2c1C(CN)CCC2 N#Cc1[nH]c(=NC2CCC3CN(C(C4Cc5cscc5C4)=O)CC3C2)sc1Cl Cc1ccc(C(=O)NC(C)CCC(=O)NC(c2cccnc2)CO)cc1 C(C(CC(C)C)C(=O)NCC1(CC)CCCCC1)NC(C(CC)=CCCC)=O C1(COC)CN(C(=O)CCC(C)CN(C)C)CCN1C(=O)C=C(C)c1ccsc1 CCC(C)(C(=O)NCCCOCCCOCCO)C(N)=O N1(C(C=CC(C)NC(CSCC=C)=O)=O)CCC1(C)CN(C)C N1(C(c2ccc(C(C)(C)C)s2)=O)CC2COCCC2(NC(=O)Cn2ccnn2)C1 C(=O)(C(C(C)(C)C)OC)NCC1CCCC(NC(CCCOCC=C)=O)C1 C1(NC(C2CC(=C)C2)=O)CS(=O)(=O)CC1NC(=O)COc1cc(F)ccc1F C1(SC(CC(=O)NCCSCCn2cc(C(C=C)O)nn2)C)CCN(C(C)=O)CC1 N1(C(c2c(C)nn[nH]2)=O)CCC(C2CCN(C(=O)C=Cc3ccoc3)C2)C1 N1(C(C(C)(F)F)=O)CC2CCC(NC(=O)CCCCC3CC3)C2C1 c1(C(C(=O)NC2CC(C(=O)OC)C2)N(CCS(C)(=O)=O)C)cc(F)cc(I)c1 CCCCCCC(C)(CCC)C(=O)NC1(CNC(C2CCC3(CCC3)C2)=O)CC1 C1(C(=O)NC(COC)C2(C)CC2)CCN(C(C2CCC(=O)N(C)C2)=O)C(C)C1 c1(C(N(C2CCN(C(c3c(OC)nccc3)=O)C2)C)=O)c(F)ccc(OC)c1N CC(N=c1[nH]c(=NCC2(F)CC(C(C)(C)C)C2)[nH]c2c1COC2)c1cccnc1 C1(NC(C(=O)NC(C)C)=O)C2CCN(C(c3cc(O)ncn3)=O)C12 N1(C(c2nccc(CNC(C(C=C)(F)F)=O)c2)=O)CC2CCCC(O)C2C1 N1(C(c2c(C(C)C)cco2)=O)CCOC2CN(C(C3CC3C(N)=O)=O)CC12 CC1CN(C(C2CCCSC2)=O)CCN1C(=O)CN1CC(=O)NC1=O NS(=O)(=O)c1n[nH]cc1C(N1CC2CCC1C2NC(C1COCCO1)=O)=O c1(CNC(c2nnnn2CC2CCCO2)C2(SC)CCC2)cc(N)ccn1 c1(CNC2C3CN(C(C4CC5C=CC4C5)=O)CC32)ccc(F)c(Br)c1F C12(C(=O)NC(C3CCN(C(C4(C5CCC5)CC4)=O)C3)C)CCCC1CC(=O)CC2 C1(NC(=O)CCNC(=O)CSc2nc[nH]n2)CN2CCCC1C2 C1(NC(C2C(C(C)C)C2)=O)CCN(C(c2csc(-c3nc[nH]n3)n2)=O)C12CC2 CC(O)(C(=O)N1CCC(C)(C(N2CCC(CO)C2)=O)C1)C(F)(F)F C(=O)(CCCC(F)(F)F)NCCC1(C)CCN(C(c2cc(CC)oc2C)=O)C1 C1(CNC(=O)C=Cc2cocn2)CCC2(CN(C(C3(O)CCOC3)=O)C2)O1 C12COC3(CC1C3)CNC2=O.C1(NC(CNC(CN(C)C)=O)=O)CCC(CO)CC1 CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CC2CC1C2NC(=O)CC1CC=CCC1 CCC(C)(CC)C(=O)NCCC(O)C(=O)N(C)CC1CC(O)C1 C(=O)(C1CCCn2c(Br)cnc21)NCCC(C)NC(c1c(C)ccnn1)=O N1(C(C2CC(C(F)(F)F)C2)=O)Cc2n[nH]cc2C1C(=O)NC1(c2nc[nH]n2)CC1 C1(NC(c2occ(C)c2)=O)CCC12CCN(C(c1ccc(N)c(Br)n1)=O)CC2 c1(C(=O)NCC(=O)N(C2(C(=O)Nn3cncn3)CC2)C)occc1C(N)=O C(=O)(CCC(=O)N1CCC(CO)C1)NCC(CO)NC(=O)OC C1(NC(C2N(CC)CCOC2)=O)(CNC(C2CNC(=O)C2)=O)CCC(F)(F)CC1 C=C(C)C(C)(C)C(=O)N1CCCOC(CCNC(C2CC2(Cl)Cl)=O)C1 N12CC3CCN(CC3C1)C(=O)C1C(CCC1)C2=O.C1(O)(OC)CN2CCC1CC2 C1(NC(C(CC#C)C2CC2)=O)CN(C(c2cccc(Cl)c2Cl)=O)CC12CC2 N1(C(CCCCC=C)=O)CC2CCC1C(CNC(=O)CSC(F)F)C2 N1(C2CCN(C(CC)C(N)=O)C2)CCN(C(=O)CC2CCS(=O)(=O)C2)CC1 c1(C(=O)NCC(CC=C)NC(c2ncncc2C)=O)c(Cl)n[nH]c1C N1(C(C=CCC)=O)CCC(NC(c2ncsc2Br)=O)CC(C)(C)C1 N1(C(C2CCN(C)C2=O)=O)CC2CCC(C1)N2C(c1nc(=O)n(C)[nH]1)=O C1(O)(C(CNC(c2c(C)onc2)=O)C)CCN(C(=O)CN2CCCC2=O)C1 c1(C(C2CC2)NC(=O)NCC2(C#N)CC3(CC3)C2)cc2ccc(F)cc2nc1O Cc1cc(Cl)ncc1CNC(C1CCCCCC1NC(C1(C)CC(F)(F)C1)=O)=O c1(C(=O)NC2CC(CNC(CC=C(C)C)=O)C2)ccnnc1O N1(CCC(=O)NCCC(C)NC(C2CC3(C2)CC3F)=O)CCCCCC1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CC(NC(=O)C(CC)C2CCOCC2)CCC1C CC1Cn2nc(C(=O)NCC3CCN3C(c3ccc(Br)o3)=O)cc2C(=O)N1 N1(C(c2cn(C)nc2O)=O)C2COCC1CC(NC(=O)CN1C(=O)CNC1=O)C2 N1(CC=C)CCCN(C(C2(CO)CCN(C(c3c(C)cccc3C)=O)C2)=O)CC1 c1(Sc2ccc(C(C(=O)NC(=O)OC(C)(C)C)=O)cn2)ncnc2c1OCCO2 C12(NC(N(C3CCN(S(=O)(=O)c4cccs4)C3)C)=O)CCC(C#N)(CC1)CC2 C12(NC(=O)C3CC3)CC3CC1C2C3O.C1(=O)CCC(=O)N(CC)CC(CC)N1 Cc1cccc(C(=O)NCCNC(c2[nH]c(C)c(C(=O)N(C)C)c2C)=O)c1Cl C12CN(CC1(C)C)C(=O)C1C(C1)C(=O)N2.c1(C(=O)OC)ccnc(OC)c1 c1(SCC)ccc(C(=O)NCC2C=CC(NC(=O)CN(C)CCF)C2)cn1 C(=O)(C(C)CS(C)(=O)=O)NCc1c(CCNC(c2ccc(C)nc2C)=O)ocn1 Cc1ncccc1CCC(=O)NCC1CCN1C(c1csnn1)=O c1(C(=O)NCC2OCCC(NC(C=C(CC)C)=O)C2)c(C(F)(F)F)cccc1F C(CC(CC)C(=O)NCC=CCNC(c1cnc(O)n1CC)=O)=CC C(=O)(C1COc2ccc(Cl)cc21)NC12CN(C(c3nc(C)sc3)=O)C(C1)C2 N1(C(c2nc(N(C)C)sc2)=O)CCc2sc(CNC(c3cccn3C)=O)nc2C1 C(=O)(C(C)C(F)(F)F)NC1C(SC)CN(C(c2conc2C(C)(C)C)=O)C1 N1(C(C2CC(NC(C(C)CCN(C)C)=O)C2)=O)CCOCC(C)(O)C1 CC1CC(CNC(=O)C(C)(C)C)CN(C(=O)Cc2ccncc2Cl)C1 Cc1cc(-c2nc(C3CCCC3O)n(-c3ccnc(Br)c3)n2)ccc1F c1(C(N(C)CCNC(=O)C(=O)NCC(F)(F)F)=O)ccc2c(c1)OC(F)(F)O2 CCCCN=C(NC1C(C)C1C)NC1CCOC(c2ccccn2)C1 c1(C(=O)NC2CC(CNC(C3(F)CCCOC3)=O)C2)cc2c(nc1O)CCCC2O c1(C(C)(C)C)cc(NC(=O)NC2CCOC2c2ccccc2)n(CCO)n1 CN1CCCCC1CCC(N1CCCC1Cn1cc(CC(C)(C)CO)nn1)=O C1(N(CC=C)C)CN(Cc2ccc(C3CCOCC3)cc2)CC2(CCOCC2)C1 C(=O)(C(CC(C)SC)N1CCCC(N(C)CCO)C1)NC(CC)C CCCCC(C(=O)N1CC(NC(c2ccc(C3CC3)c(OC)c2)=O)C1)N(C)C Cc1cccc(C(C(C)C)N(C(=O)C(=O)NC(c2ccc(C)s2)C)C)c1 C1(C(N(CC(C)NC(c2c(CC)ncs2)=O)C)=O)CCN(S(=O)(=O)N(C)C)C1 CCC(CC(=O)N1CCC(N(C)C(c2cc(OC)cnn2)=O)C1)C(F)F c1(CCC(=O)NCCNC(CC=CCC)=O)cccc(C(=O)OC)c1 N1(C(CN2C(C)CC2)=O)CCCC(NC(c2cc(C3CC3)no2)=O)C1 C1(C(=O)NCC2C(NC(=O)CC(F)(F)F)CCCC2)CC2(CCCC2)CO1 C(=O)(C1CCc2cccnc21)N1CC2CC(NC(=O)CC3CSC3)CC2C1 c1(C(=O)NC2C(NC(COC(CC)C)=O)CCC2)cnnc2ccccc12 C(=O)(C(C)(C1CC1)NC(C1CCOC1C(C)C)=O)N(CC(C1CC1)OCC)C N1(C(CCC(C)=O)=O)CC2(CCCC2NC(=O)Cc2ccc(F)c(Br)c2)C1 c1(C(=O)NCC(C)CN(C)C(C2(C(C)(F)F)CCOCC2)=O)cccc(=S)n1O C1(CNC(=O)CCC2CCCCO2)CC(F)(F)CN1C(c1cccnc1S)=O C1(NC(Cc2cn(CC)nc2)=O)CCC(CNC(C2CC(N(C)C)C2)=O)CC1 O=C1c2ccccc2-c2ccc(NS(=O)(=O)CC3CC4CC4C3)cc21 c1(N(CC(CN(C)C(c2n[nH]c(C3CC3)n2)=O)O)C)ncc2c(ncn2C)n1 C1(COC)(NC(C2CNC(=O)C2)=O)CN(C(=O)CCn2cncn2)C1 O=S1(=O)c2cccc(c2)S(=O)(=O)N1.c1(NCCCC(=O)O)c(F)cccc1Cl C1(CC)CN(C(c2scnc2C)=O)CCN1C(=O)C(C)C1CC1c1ccccc1 c1(OCCNC(=O)NCCC=C=C)ccc(F)c(Cl)c1 CN1CCN(C(=O)CCN(C)C)C(C(N2CCC2(C)CCO)=O)C1 C1(CNC(C(COC)(C)C)=O)COCCN(C(C2CC3(CC3)CO2)=O)C1 Cc1ccnc(C(N2CC(CC(=O)O)C(C)C2)=O)c1Br CC1CCCCC1(CNC(=O)Cc1n[nH]c(=N)s1)NC(=O)C=C1CCCC1 c1(OC)c(C(=O)N(C2CCN(C(C3CCS(=O)CC3)=O)C2)C)ccnc1Cl c1(NCC(CC#C)(C)C)ccc(S(=O)(=O)NCC2CC23CC3(F)F)cc1Cl c1(NC(=O)CCCF)ccc2occc2c1.C12CCC(CC1)NC2=O c1(NC2CCC(CCC)CC2)cc(CC)ccc1O C#CC1CC2(CC2)CN1C(=O)CC1C2CN(C(C3CN4CCC3CC4)=O)CC12 C1(C(N(C(C(=O)NC2(CCC)CC2)C2CC2)C)=O)CCOCC1 N1(C(CCc2cnc(C)s2)=O)CCCC(NC(C2(C(F)F)CCCO2)=O)CC1 C12(NC(c3cc(O)nc(O)n3)=O)CCC(C1)N(C(c1nc(Cl)ccc1Cl)=O)C2 CCC(C)CC(C)C(=O)N(CCC(=O)N(c1ccccc1)C)CC1CC1 c1(CNC(C2C(C(=O)NCC(C#C)C(C)C)CC2)=O)cccn2nccc12 C(CC(C)CC)(C(=O)N(C)CC=C)NC(c1cncc(C#C)c1)=O C#CCCC(O)C(=O)NC1(CCCNC(c2ccc(C3CCOC3)cc2)=O)CC1 C1(C=O)(CO)CCCN1C(C1CCN(N2CC(CC)C2)C1)=O.C(C)(C)(C)NC=O CCC(C(=O)NC(C)CC1CCN(C(=O)Cc2ccc(O)cc2)CC1)C(F)(F)F CC1(C)COCCN(C(=O)COC2CN(C(c3ccc(=N)[nH]c3)=O)C2)C1 C(=O)(CCCN=c1nccc[nH]1)N1CCN(C)C(CNC(C2CC(F)C2)=O)C1 c1(SC(CC)C)nc(C(F)(F)F)c(N)c(O)n1.C1(C(=O)O)CCC12CN(C(C)(C)C)C2 C(=O)(CC(=O)N1CCCC1C1(NC(c2c[nH]cc2CC)=O)CC1)NCC c1(NCC(c2ccccc2)C)sc(CC(=O)O)cc1C#N c1(C(N2CC(F)(CNC(CSCCN(C)C)=O)C2)=O)c(OC)cccc1N(C)C N1(CCC)CC(C(N2CC(N(C(C3C4CC5C(C4)C35)=O)CC)C2)=O)CC1=O c1(C(=O)NCC2(CCNC(C(C)C3CCOC3)=O)CC2)ccc(P(C)(C)=O)o1 c1(CN(CCN(C)C)CCO)cccc(Br)c1.C1(C(=O)O)COCCC1N C(=O)(C(C)(C)CC(C)(C)C)NC1CC(NC(C2(COC)CCCO2)=O)C1 N1(C(C(=Cc2ccco2)C)=O)CCC(C)(C)C(C(=O)NCC(C)(C)CC(C)O)C1 C(=O)(CC(C)C(C)C(C)C)N1CC(O)(CNC(CCSCC)=O)C1 Cc1nnc2n1C(C(=O)N(C1CCN(C(C3CCNC3=O)=O)CC1)C)CC2 c1(C2(N(C(CNC3CC(F)(COC)C3)=O)C3CC3)CC2)cc(OC)ccc1Cl c1(C(=O)NC2C3CN(C(CCCNC(C)=O)=O)C2C3)c(F)cccc1Br C(=O)(C1=CCCC1P(C)(C)=O)N1CCC(CNC(c2c(C)onc2C2CC2)=O)C1 C1(NC(=O)CC2CCCOCC2)C(O)C2CCOC12 N1(C(CN(C(C)=O)C)=O)CCC2CC2(C(=O)NCCCC(C)CO)CC1 N1(C(C(CCC#C)(F)F)=O)CC2CCCN2c2ccc(Cl)cc21 C1(NC(c2c(C)cncc2)=O)CC2C1CCN2C(=O)CN1CCCC1=O N1(C(C(C(C)C)F)=O)CCC2CCC(C1)N2C(C1(C2CCC2)CC1)=O Cc1ncc(C(=O)NCCN2CCCN(C(c3ccn(C)n3)=O)CC2)c(C)n1 C1(NC(CS(CC)=O)=O)CCN(C(c2ccc(Cl)cc2C)=O)CC1F C1(CNC(Cn2nc(C)c3c2ncn3O)=O)CC2CCCC2N1C(C1C2CC12)=O C1(Nc2ncc(C)cn2)CCCN(C(c2cnc(-c3ccco3)s2)=O)CC1 C1(O)(CCNC(C(C=C)C)=O)CCCN(C(=O)C=CCOC)C1 Cc1[nH]nc(C(=O)NC2CN(C(c3cncs3)=O)CC2Cc2ccccc2)c1Cl Cn1c(=O)ccn(CC(=O)NC2CCC(NC(c3csc4cncn34)=O)C2)c1=O c1(C(=O)NCCC(C(=O)NC2C(C(C)(C)C)CC2)O)n[nH]c2c1CCC2 c1(C(N(C(C)CNC(=O)C=CC2CCOCC2)C)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(CC(=O)NC(C2CCCN2C(C2C3CCCC23)=O)C)ccccc1F C1(C(N2CC(CCNC(=O)CSCCC(F)(F)F)C2)=O)CC2(C1)CC1(CC1)C2 C1(C(=O)NCCCC)CCCCCN1C(c1cnns1)=O N1(C(CC2CC(OC)C2)=O)CCCCC(NC(=O)C(F)(F)CO)C1 N1(C(Cc2cccc(OCC)c2)=O)CCN(C(C2(C#N)CC(C)C2)=O)C2(CC2)C1 C1(C(N2C(CN(C(CC(C)(F)F)=O)C3CC3)CCC2)=O)CCCC12CCC2 N1(C(c2c(CC)nc(=N)[nH]c2)=O)CC2(C1)SCCC2NC(c1cnc(C)[nH]1)=O C(C(CC(=O)N=c1cc(C2CC2)n(C)[nH]1)N(C)C)NC(C(C(CC)O)C)=O Cc1nc(C)n(CC(=O)NC(CCC2CCC2)C(=O)NC(C(N)=O)C2CC2)n1 Cc1ccc(OCC(N2CC(NC(=O)C(F)F)CC(O)C2)=O)c(Br)c1 C1(C(N2CC3CC(C)C3C2)=O)CC12CCN(C(C1COCC1(C)C)=O)CC2 c1(CNC(C(C)N(C(=O)Cc2cnc(C)[nH]2)CCC)=O)nc(C)sc1C C12(NC(c3noc4c(F)cccc34)=O)CCCC1(F)CN(C(c1ccc[nH]1)=O)C2 C1(C(N(CCCCC)C(C)CCC)=O)Cc2c(OC)cc(OC)cc2N1 c1(CO)nc(-c2ccsc2C#N)n(CCOc2ccc(Cl)cc2)n1 c1(CCC(=O)N(CCC(C)NC(C2CCC(CCO)CC2)=O)C)ccc(F)nc1 c1(C(=O)OC)cccc2c1OCCN2C(=O)C(c1ccc(Cl)cc1Cl)C c1(C(=O)NC(C(C)NC(=O)CCCN2CCCC2)C)ccc[n+]([O-])c1 C1(NC(CN2C(C)CCCC2)=O)CCN(C(C2CCOC(C)(C)C2)=O)C1(C)C c1(C(N(C)CC2CN(C(COCc3onc(CC)n3)=O)C2)=O)c(C)cccc1Cl C1(CCNC(C2(C)CCOC2)=O)CCCCN1C(C1CC1C1CC1)=O c1(C(N2CCCC(CN(C(C(C)CF)=O)C)C2)=O)cc(Cl)c(F)cc1Cl C(C)(C(=O)NCC1CC1C(=O)NCC(F)Cl)=C(C)C C#Cc1ccc(C(N2CCCC(O)(CNC(c3ccnn3CC)=O)C2)=O)c(C)c1 N1(C(C(CCC)C)=O)CCN(C(=O)NCC2CC2c2ccco2)C2(CCC2)C1 C1(C(N(CCN(C(=O)C=CC2CC2)CC)CC)=O)CC1C(F)(F)F N1(C(=O)CC2CC(O)CN2C(C2CC(F)C(=O)N2)=O)C2CCC1CC1(CC1)C2 N#Cc1ccc(F)c(F)c1NC(C1CCCCN1Cc1cc(CO)ccc1O)=O C#CC1(C(=O)NC(C)Cn2cncn2)CN(C(=O)CCC2CC2C)C1 CC(C)C(CNC(C1CC1c1cn[nH]c1)=O)NC(C1CC12CC2)=O CC(C)CC(C)(O)C(=O)N1CCCC(F)(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C1 N1(C(CN(C(=O)CCc2cscn2)C)=O)CC(CC2CC2)C1 N1(C(=O)NCC(c2ccc(Br)cc2)OC)C2CCCC1CN(C)C2 C(=O)(C(C)(C)C(=O)NCc1ccccc1)NCCCNC(C(Br)=C(C)C)=O C1(C(N(CCN(C(c2c(C(C)C)[nH]cc2)=O)C)C(C)C)=O)CC2CCC1C2 C1(NC(Cc2ccn(CC)n2)=O)CCCCN(C(c2cnnc(C)c2)=O)C1 c1(CC(=O)NCCCCNC(=O)CSC2CCS(=O)(=O)C2)cccc2c1OCO2 N1(CC(=O)NC2(CC(C(CC=C(CN)O)=O)=O)CC2)CCOCC1=O c1(OC)ccc(C(=O)NC2CCCC(N(C)C(c3occ(C)c3C)=O)C2)nc1N N1(C(c2n[nH]cc2CCC(F)(F)F)=O)CCC2(CCCN2C(C2CCCO2)=O)C1 c1(C(C)NC(C2CC2C(=O)NCCNC(N)=O)=O)ccc(F)c(F)c1 C=CC(F)(F)C(=O)N1C(CNC(=O)Cc2cccnc2O)CC2CC12 c1(C(N2CC(CNC(C3(CCCC)CCC3)=O)C(C)C2)=O)ncc(OC)cc1F C=CC1CN(C(C2COC3(CCC3)C2)=O)CC1NC(=O)COC(F)(F)F c1(C(=O)NCC2CC(NC(C3(CCOC)CC3)=O)C2)cccc(C#N)c1 N1(C(C(CC=CC)CC)=O)CCCN(C(=O)COCCF)CC1c1ccccc1 c1(N2CC(N(C(=O)C3=CCCCC3)C(C)C)C2)nc2cccc(F)c2s1 C1(C(=O)NC(COC)C2(C)CC2)CC(O)CN1C(=O)CCC1CCCN1C c1(-c2cn(CC(N3CC(CCC)OCC3)=O)nn2)ccc(N)c(CO)c1 N1(S(C(C)C)(=O)=O)CCc2sc(C(=O)Nc3c(Cl)cccc3I)cc2C1 C(=O)(N1CCC(C(=O)NCCc2ncc[nH]2)O1)C1(C)N(C)CCC1 Cc1cc(-c2c[nH]nc2C(N2CCC(O)C(C)(CO)C2)=O)c(F)cc1Br N1(C(Cn2c(C)ncc2)=O)CCC(C)C(NC(c2cc(C(N)=O)cc(F)c2)=O)C1 c1(C(=O)NCC(CNC(CSc2n(C)ccn2)=O)(C)C)cccc(P(C)(C)=O)c1 N1(C(C(C)=C2CC2)=O)CC(C)(C)CC1C(N1CC(C(C)(C)O)C1)=O CC1CN(C(=O)CN2CCCC(C)(NC(=O)COc3ccccc3)C2)CC(C)O1 C1(C(=O)NC2CN(C(CC=CC=C)=O)C(CO)C2)CCc2cn(C)nc2C1 CCCCCCC(C)(CCC)C(=O)NC1CC(CNC(=O)C(C)OCC)C1 C(=O)(C1=CCCN(C(c2ocnc2C)=O)C1)N1CCN(CC)CC1 n1(CCC(=O)NCC(CCNC(c2cnc(=N)[nH]c2)=O)O)cc([N+](=O)[O-])cn1 c1(C(=O)NC2CN(C(CNC(CCCCC)=O)=O)C(C)C2)cc(C)nc(O)n1 C=CCC(CC=C)C(=O)NCCC1=CCN(C(=O)C=C(C)c2ccco2)CC1 N1(C(C2C(C(=O)OC)CC2)=O)CC2(CC2)CC1CNC(c1cn(C)cc1C)=O N1(C(C=CC2CCN(C(C(CCCC)=O)=O)CC2)=O)CC(C)(C)OCC1(C)C c1(C(=O)NCCc2ccsc2)cnc2c(-c3ccc4nccn4c3)cnn2c1 N#Cc1cc(N2CCC(C3OCC3(F)F)CC2)nc(-c2ccccc2)c1 CCC(C)(C)CCCC(=O)NCC(C(=O)NC(C)CF)C(C)C c1(SC)cn(C)nc1C(=O)NC1CN(C(=O)Cc2cnccn2)CC1O C#CC1CC2CCC1N(C(C1(NC(=O)C(N3CCOC3=O)C)CC(O)C1)=O)C2 Cc1cccc(C(=O)NCC2(NC(CCOCc3cnn[nH]3)=O)CCOCC2)c1 C1(C(N2CCC(N(C(=O)CCSC(F)(F)F)CC#C)C2)=O)CCCC(OC)C1 C12(NC(C3C(CCC)C3)=O)CCOCC1CN(C(=O)Cn1cnc(C#N)n1)C2 C(=O)(CC(C)(C)CC(F)F)NCCOCCN(C)C(C1(F)CCS(=O)(=O)C1)=O CC(C)C(O)C(C)C(=O)NCC1(C)CCCN(C(c2cn3ncccc3n2)=O)C1 N1(C(C=CCN(CC)CC)=O)CCC2(CC(C(N3CCCC3(C)C)=O)C2)C1 c1(C(N2CCN(c3nc(OC)c(C)cn3)C(C)C2)=O)cnc2c(c1)c(C)nn2C C1(O)(CC)CCCN(C(=O)C(C)(CO)NC(C2COCC2C(N)=O)=O)C1 C1(OC)C(OC)CN(C(=O)CCS(C)(=O)=O)C1CNC(C1(C)CCCS1(=O)=O)=O N1(C(CCCN(C(CCC2CC(OC)C2)=O)C)=O)CC(C)(C)C12CCC2 c1(N2CCC(C)(CNC(Cc3n(C)cnc3)=O)CC2)ccc([N+](=O)[O-])cc1C#N N1(C(Cn2c(C)cc(C)n2)=O)CC(NC(=O)CO)CC(O)C1 C(=O)(C(=O)NNC(=O)C1CCCS1)N(C)Cc1ccc(OC)c(OC)c1 c1(C(N(C(c2ccccc2)CNC(=O)Cc2ccc(F)cn2)C)=O)cnn(C)c1N C#CC1(C(N2CCC(CC(C)(C)C)C2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 c1(CC(=O)NC(C(=O)OC)C(C)c2ccccc2)ccc(S(=O)(=O)CCO)cc1 N1(C(CC2ON=C(C)C2)=O)CC2CCN(C(c3ncoc3Br)=O)CC12 N1(C(CCc2cn(C)nn2)=O)CCCC1(C)CNC(C1(C(=O)N(C)C)CC1)=O C(=O)(C(C)(C)CCC(=O)NC1CCCN(C(=O)C(O)CC(F)F)CC1)OC n1(CSC)nccc1CNC(=O)CCN(C(=O)CCCN(C)C(C)C)C c1(CSCC)cccnc1C(=O)NCC1CCC(NC(c2c(C)noc2N)=O)C1 C1(CCNC(c2c(CC)cno2)=O)CC(F)(F)CN1C(=O)C=Cc1ccc(C)o1 N1(C(=O)OCc2cc(OC(C)C)cc(Br)c2)CCC(C2CCCC23OCCO3)C1 N1(C(=O)CCCN2CCOC2=O)CCC(c2ncc[nH]2)CC1 c1(C(=O)NC(CC#C)C)cc(CNC(c2c[nH]c(=N)o2)=O)cs1 Cc1cncc(CNC(=O)NC2CC(=O)N(c3ccc(F)cc3)C2)c1C C1(COC)(NC(c2sccc2C)=O)CCN(C(=O)CC2NC(=O)NC2=O)C1 C1(O)(CCNC(C(CC)=CC)=O)CCCN(C(=O)CC(O)c2ccccc2)C1 N1(C(c2cc(COC)no2)=O)CC2CC(N(C(=O)C=CC3CC3)C)C1C2 Cc1noc(C)c1C(C)C(=O)N(C)CC1CCN(C(=O)COCCN(C)C)C1 CCCCCCC(CC)C(=O)NCC(C1CC1)NC(C1(C(F)F)CC(F)(F)C1)=O c1(OC)cc(OCCOC(C2CCSC2)=O)ccc1[N+](=O)[O-] Cc1scnc1C(=O)NC(C)(C)CCN(C)C(C1(c2cccs2)CC1C)=O c1(C(=O)NC(C)CCNC(c2cnc3sccn23)=O)cc2cccnn2c1 C(=O)(C(C)(C)CC(C)C)N1CCC(NC(C(=Cc2cn[nH]c2)C)=O)C(F)C1 N1(C(C2N(C(c3c(CC)cc[nH]3)=O)CC3(CC3)C2)=O)CCCC(N=[N+]=[N-])CC1 N1(C(C(C)(C)c2ccccn2)=O)CC2CCC(C1)C2NC(c1cscn1)=O N1(CC(N2CCC(OC)(CNC(c3c(C)csc3Cl)=O)C2)=O)CCC(=O)NC1=O c1(C(=O)NC2CN(C(C3(CC)CC3)=O)CC(O)C2)cc(C2CC2)nc2ccnn12 C1(C(N2CC(F)(c3cn(-c4cc(F)ccc4Br)nn3)C2)=O)Cc2ccccc2O1 C1(NC(CCCC)=O)CC2CCC(C1F)N2C(=O)CC1CCC(C)(C)C1 c1(CN2CCC(N(C(=O)CCn3cccn3)CC)C2)ccc(C2CC2)nc1 C1(C(=O)OC)C(NC(=O)Cc2cccc(C)c2Cl)C2CCCC12 c1(C(=O)NC2CCCC(NC(C3CC4(CC4)CO3)=O)C2)cc(Cl)cc(F)c1F N1(C(CC2(C)CCCO2)=O)CC(NC(c2cnc(Cl)[nH]2)=O)C2(CC2)C1 C=C=CCCC(=O)N1CCC(F)(C(=O)NCC(C)(O)CSC)C1 c1(COC)n[nH]c(=NCC(c2ccccc2)NC(C23CCCC2C3(F)F)=O)s1 c1(C(N2C(C)CCC(NC(=O)CCn3ccnc3)C2)=O)cnc2ccncc2c1 C12(CCNC(CCOCCCOC)=O)CCC(C1)N(C(=O)C(C(C)C)OC)C2 C1(C(=O)NC(c2cccn2C)C)CN(C(=O)CCc2cocn2)CCO1 C(CC(=O)NOCC(=O)N(C)C)NC(=O)NCC1C(CC)C1(F)F Cc1ncnc(N(C)CC2CCCN2C(c2ccoc2Cl)=O)c1Br CC1CCC(O)(C(=O)NC(C2CCN(C(C3CC(N=[N+]=[N-])C3)=O)C2)C)CC1 C1(C(C(=O)NC2C(C(N(C(CC)C)C)=O)CC2)C)CCCCC1 C1(C(N(C(c2ccccc2)CNC(C(=O)N(C)C)=O)C)=O)CC=CCO1 c1(C(N(C2CCC(NC(=O)C(F)(F)C3CC3)C2)C)=O)nc(Cl)c(Cl)s1 O(P(=O)(CCNC(C1OCC2CCC1C2)C)OCC)C(C)C C1(C(N(CC(CC)OC)C)=O)CC(N=[N+]=[N-])CN1C(C1CC1C1CCCO1)=O C1(CCOC)(NC(=O)CCOCCN(C)C)CN(C(=O)Cc2cnoc2)C1 C1(C(N(CC(CC)NC(=O)C(CN(C)C)CC)C)=O)CCCCCCC1 C1(NC(c2nc(CC)sc2N)=O)CC2CC1CN(C(=O)COCC(C)(C)C)C2 C1(C(=O)NC2CC(CNC(c3sccc3Br)=O)C2)OCC2CCCC1C2 c1(CC)cc(C(=O)NC2CC3(C2)CC3NC(C2CCCCC2(C)C)=O)cc(Cl)c1 c1(CC(=O)N(C(CNC(CCC(C)OC)=O)C)C)ccc2ccccc2c1 c1(C(N2CC(N(C(=O)C(F)n3ccnc3)C)C3(C2)CC3)=O)c(F)cc(F)cc1F CCCCCCC(=O)N1CCCCCC1C(=O)N(C1CSC1)C N1(C(CSSC)=O)CC2(CCC(CNC(C3CCN(CC(F)(F)F)C3)=O)O2)C1 CC1(C)C(NC(=O)CC2OCCCC2(C)C)CCN1C(c1cc(Cl)ccc1Cl)=O c1(SCC2(COC)COC2)cc(C)c(Br)cc1C CCC(C)(C)C(C)CC(=O)NCCC1CCN(C(c2cccn2C)=O)C1 C1(C(N(C)CC2N(C(c3cn(CC=C)nc3)=O)CCC2)=O)CC=C(C)CC1 C(=O)(C1=NNC(C(F)(F)F)C1)NC(C(C)NC(=O)CCn1cnnn1)(C)C c1(CNC(C2(OCC)CCC2)=O)cnn(C)c1C(=O)N(C1CCC1)C1CC1 C1(NC(C(C2CCC2)OCC)=O)CN(C(c2ccn(C(C)(C)C)n2)=O)CC1SC c1(C(=O)NS(C(CCCC)C)(=O)=O)cc2c(s1)CCC(C(C)(C)C)C2 C1(C(=O)OCC)CCC(NC(=O)N(C(C)(C)C)Cc2cc(C)ccc2O)C(O)C1 Cc1ccc(C=CC(N2CC3CC3(CNC(c3sccc3C#N)=O)C2)=O)o1 N1(C(C(C2CC=CCC2)NC(CN(CCOC)C)=O)=O)CCNC(=O)CC1C N1(C=O)CCCCC1C1CCCN1C(=O)C1=COCCO1.c1(OC(F)F)cnccn1 N1(C(C2(C)CCCN(c3nncc(CCC)c3)C2)=O)CCC(C2CNC(=O)C2)C1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CCN(C(C1CC(CC)C1)=O)C2 c1(C(=O)NC(CNC(CCC2CC(C)C2)=O)(C)Cn2cccn2)ccc(CF)cc1 c1(N(C)C)ccc(Cn2nc(-c3cc[nH]n3)nc2CC2(C(F)F)CCCC2)cc1 c1(C(N2CCC(N(C(=O)CC(C)(C)COC)CC)C2)=O)ccn2cncc2c1 CCC(O)(CC)c1cn(C2CCN(C(=O)CC3(CSC)CC3)C2)nn1 N(C1CC2(CN(C(c3csnn3)=O)C2)n2ccnc21)C(c1c(C)cncc1)=O N1(CC(C(C)c2ccccc2)O)CCN(c2ccc(C(C)O)cc2)CC1 N1(C(CCC2CC(OC)C2)=O)CC(NC(=O)C(C)(C)N=[N+]=[N-])CC(C)C1 C1(CNC(=O)CN2CC=CC2)CCN(C(C2CCC(CN3CCCC3=O)O2)=O)C1 Cc1ccc2c(c1)C(C(=O)NC(CNC(=O)Cc1cccc(F)c1)C1CC1)C2 N1(C(CSC)=O)CCC=C(C(=O)N(c2ccncc2)CCOC)C1 N1(C(C(C(C)C)SCC)=O)CCCC(C)(NC(c2cc(C)ccc2O)=O)C1 c1(-c2cccc(C)c2)csc(=Nc2cccc(Cl)c2)n1C(c1ccn(C)c1)C c1(NCCCOC(=O)NC)[nH]c(=NC(C)CN2CCCC2)nc2scnc12 C=CC(CCC)CC(=O)N1CCC(C(F)C(N2C3COCC2C3)=O)C1 C1(C(N(C2CCCN(C(C(C(C)C)OC)=O)C2)CCO)=O)CC2(CCCC2)CO1 N1(C(c2cc(O)cc(Cl)c2Cl)=O)CCC2C(CCCN2C(=O)CC2(CO)CC2)C1 c1(C(N2CCOCC2c2ncccn2)C(=O)NCC2CC2)cc(F)c(Cl)cc1Cl N1(C(c2cn(C(C)C)nc2C)=O)CC(N(C(=O)CCOCC2CC2)C)C(C)(C)C1 C1(C2CCN(C(c3cccnc3OCC(C)C)=O)C2)(NC(C(C=C)O)=O)CC1 Cc1[nH]c(C(F)(F)F)cc1C(N1CCN(C(c2cccc(N)n2)=O)CC1)=O c1(C(=O)NCCCCOCCCNC(C2(C(=O)OC)CC2C)=O)scc(C)c1C CC1(C(=O)NCCCNC(c2nn[nH]c2Cl)=O)CCC2(CC1)OCCO2 C(=O)(C(C(C)(C)C)OC)OC.C1(=O)CC(C2CC2)CN1C1CCC1 c1(CNC(c2cc(Br)cc(F)c2F)c2n(CC=C)nnn2)cc(F)cc(C#N)c1 C12(C(N(C3CCOC3)CC#C)=O)CCCC1N(C(c1ncn3ccccc13)=O)CC2 O=C(C=CSc1ccccc1)NCC1CC1NC(=O)Cc1ccccc1 N1(C(C2(F)CCN(C(C3CCCN(C)C3)=O)CC2)=O)CCC2(CCCCO2)C1 C(=O)(CCCCCSC)N1C(CNC(C(c2ccccc2)SC)=O)CC(F)C1 C#CCCC(O)C(=O)NC1CCC(NC(c2cc(C(F)(F)F)ccc2F)=O)C1 O=C(C(O)CCc1ccccc1)N1CCC(CCNC(C2(O)CCOC2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC1CCCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 Cc1ccc(CN(C2CCNCC2)C(=O)CCc2ccccc2)cc1 C(=O)(CCCCCCNC(c1cnn2ccccc12)=O)NC(C#C)CC1CCC1 C1(NC(C(C)OCC#C)=O)CCN(C(c2oc(CCC)nc2C)=O)CC(C)(C)C1 c1(CC(=O)NC2CN(C(C(=O)NC(C)=O)=O)CC2C)ccc(OCC(F)F)cc1 c1(NC(C2CCC(n3cc(CCCOC)nn3)CC2)=O)ncc2c(F)cccn12 C=CC(C)(C)CC(=O)NCCn1cnc(C(=O)NC2(C3CCCO3)CCC2)c1 C1(C(=O)NC2(CF)CCN(C(C(C#C)(C)C)=O)C2)CCC2(CCOCC2)O1 C1(NC(c2ccn(CC)n2)=O)CN(C(=O)C(C(C)C)OCC(C)C)CC1C(F)F N1(C(c2c(NC)scn2)=O)CC(O)CCC1C(=O)N(C1CC(CN(C)C)C1)C c1(OCC#C)ccc(C(=O)NC(c2ccccc2F)C(C)C)c(F)c1 N1(C(C2C(C(=O)OC)CC2)=O)CCCN(C(=O)C(C)(Cl)Cl)CCC1 N1(C(C2CCCN(C)C2)=O)CC(C(N2CCC(C3(C)N=N3)C2)=O)CCC1(C)C N(C(=NCCCNC(=O)Nc1ccc(C)cc1)NCC1CC1Cl)CCSC c1(NC(c2cc3ccc(-c4cn[nH]c4)cc3[nH]2)=O)nc2cc(F)ccc2s1 Cc1nc(O)ccc1C(=O)NC1(CNC(=O)CCC2CCOC2)CCCCC1 c1(C(=O)NCC2N(C(C(F)OC)=O)CC3(CC3)C2)sc2cncn2c1C C(C(O)C(C)(C)C)N(C(CCOCCNC(C1(CC)CCOC1)=O)=O)C c1(N2C(C(=O)NCc3ccccc3)CCCCC2)ccc2nnc(C(F)F)n2n1 S(=O)(=O)(c1cccnc1)NCC(=O)N(CCC)CCc1ccnc(Br)c1 N1(C(C2SCCCS2)=O)CC2(CCN(C(C3(Cl)CC3)=O)CC2)C1 CC1CN(C(C2CCC2CNC(=O)C(=Cc2cccnc2)F)=O)CC1C(N)=O C1(CC)CCN(C(=O)C=CC(C)NC(=O)CC23CCCC2C3)C1 N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCC2CN(C(c3nccc4cc[nH]c34)=O)C2C1 c1(OC)cc(CC(=O)N(CCN(C)C(c2ccc[nH]2)=O)C(C)C)cc(Br)c1 CC(CC(F)(F)F)C(=O)N1CCOCCC1C(N1CCC(O)C(O)C1)=O C(=O)(C(CC(N)=O)NC(c1[nH]ccc1C)=O)NC(CC)C C1(C#N)(C(N2CCC(CN(C)CC3CC3)C2)=O)CCCC1 N1(C(c2c(CNC(=O)CC(=O)NC3CC3)c[nH]n2)=O)CCC(O)C(F)(F)C1 c1(C(N(C2CCC(NC(Cc3ccn(C(C)C)n3)=O)C2)C)=O)cc(F)ccc1N c1(C(=O)NCCOCCCNC(=O)CC2CNC(=O)C2)nnn2c1CCCC2 N1(C(N(CCCN2CCOC2=O)CC)=O)CC2(CCC(CC(=O)O)OC2)C1 C1(C(=O)NC(C2CCCN2C(c2cc(Cl)c(Cl)n2C)=O)C)CCOC(=O)CC1 CC(C)(C)C(=O)NCC(=O)NC1(CO)CN(C(=O)Cc2ccsc2Br)C1 c1(C(N(c2ccccc2O)CC)=O)ccc(-c2cccc(OC(F)(F)F)c2)cc1 CC(C)CC(C(=O)N1CCN(C(=O)C(=CC2CCCCC2)F)C(C)C1)N(C)C CCCC(CCC)=CC(=O)NC(CN(C)CC)C(=O)NCC(C)(C)C(=O)OC c1(CC)nnc2c(C(=O)NC(C3CCCCN3C(c3cnns3)=O)C)cccn12 N1(CC(=O)NC2CN(C(c3cnc(CC)s3)=O)CC(O)C2)CCCCCCC1=O c1(NC(C2(CO)CCC2)CC)cc(NCC(c2ccccc2)CO)nc(C)n1 c1(CC(=O)NC(C)CC#N)ccc(O)cc1 N1(C(c2ncn(C)c2Cl)C(=O)NCCCSC)CC(C)OCC12CCC2 c1(CNC(C(C)(C)C2CC2)=O)cnn2c1CN(C(C1C3CC3C3CC13)=O)CC2 C1(NC(CN(C)CC)=O)CCN(C(=O)CC2CN(C)CC2O)CC(C)(C)C1 c1(NCC2CCC(C(N(C)C)=O)CC2)ccc2ccnc(Cl)c2c1 C1(NC(CNC(N)=O)=O)CN(C(=O)C=Cc2ccccc2)C2(CCOC2)C1 CN1CCN(C(C2(NC(C3CCCO3)=O)CC(F)(F)C2)=O)C(CCO)C1 N1(C(C2(CCC)CC2)=O)CC2CCN(C(=O)COCc3nccn3C)C(C2)C1 C(=O)(CC1CC(=O)c2ccccc21)N(CC(CN(C(CCCC(C)=O)=O)C)O)C c1(OC)cncc(C(=O)NCCC(O)CNC(=O)C(C(C)C)N2CCC2)c1 C1(C(N2CCC3CCC(NC(=O)Cn4cncn4)C32)=O)CNC(=O)CC12CCC2 C1(C(=O)NC(CC)CNC(C2(CC(C)C)CCC2)=O)CCOC1c1cnn(C)c1 N1(C(C2C(C)CCO2)=O)CCC(NC(=O)CC23CCC(CC2)C3)C(O)C1 C(=O)(N=c1[nH]nc(Br)s1)C1C(NC(c2ccc(-c3cc(C)[nH]n3)cc2)=O)CCC1 O=C(C1=NN(CCO)C(=O)CC1)N1CC=CC1CCn1cc(-c2nccs2)nn1 C(=O)(C(C)CC(F)(F)F)NCC=CC(=O)NCC1N(CC)CCCC1 c1(OCC)cccc(C(N2CCC(C)(C(=O)NCc3cc(Cl)ccn3)C2)=O)n1 c1(OC(C)C(=O)N2CC(CN(C(=O)CC(O)C3CC3)C)C2)ccccc1 C=CCCCCCC(=O)N1CC(O)(C(F)C(N2CCCCC2CCO)=O)C1 c1(C(=O)NCC(CC)NC(c2cc(N(C)C)ccc2C)=O)cc(OC)cc[n+]1[O-] CCC(C(=O)NCCc1ncon1)N(C)C(C1CCOC1)=O c1(C(=O)NC(C2CC(NC(C3(C)CCNC3=O)=O)C2)C)ccc2nccn2n1 C1(CNC(=O)Nc2cccc(Cl)c2CC2CC2)C(F)(F)C12CCOCC2 CC1(C)CCC(CC(=O)NCc2ccccc2CNC(c2cc(Br)c[nH]2)=O)O1 c1(C(N2CC(NCc3ccc(OCC)cc3)C(C)C2)=O)ccc(Br)c(OC)c1C C1(O)(CNC(COC)=O)CCN(C(=O)C=Cc2csc(Br)c2)C1 c1(C(=O)NCCCCCNC(C2CCC(C)(C)O2)=O)nc[nH]c2nccc1-2 C1(O)(CCNC(c2ncc(C)nc2)=O)CCCN(C(C2CC(F)C2)=O)C1 C1(NC(C(CC)CC(C)C)=O)CCC2(CC1)CN(C(c1ccc(=N)[nH]c1)=O)C2 N1(C(C(C(C)C)SCC)=O)CC2CC(O)C1C2NC(c1cc(C(C)=O)[nH]n1)=O C1(CNCn2c(C)ccc2F)CC2(C1)CN(Cc1ccccc1)C2 C1(C(=O)NCCNC(=O)CC2C=CCCC2)(OC(C)C)CCOC1 c1(OCC)ccccc1C(=O)NC1CCCC(NC(c2c[nH]nc2OC)=O)C1 CCCCC(CNC(C1(OCC)CCOC1)=O)NC(=O)Cc1cccnc1 C(C(C)(C)C#CC(=O)N1CCC(CC(N)=O)C1)NC(CC(C=C)(C)O)=O C(=O)(C(C(C)(C)C)NC(C1CC(C)(C(=O)OC)C1)=O)NC(C#C)CC(C)C C1(C(=O)NC(C)CNC(c2cnoc2)=O)(NC(=O)OC)CCCCC1 C1(NC(c2cnc(C(C)C)o2)=O)CCCCC1N(C(=O)CC(C)(C)C)C C1(O)(CC)CCCN(C(=O)CC2CCCN2C(=O)CCCCCNC(N)=O)C1 c1(CN2C(CC)CCC2C)cnc2sc(C)cn12 Cc1cn2ccnc(C(=O)NCC3COCC3NC(C3C4CCCC34)=O)c2n1 c1(N2CCN(C(=O)NC3CCCCC34CC4(F)F)CC2)ccc([N+](=O)[O-])cc1Br CCCC(C(=O)Nc1cn(CCF)nc1C)NC(c1ccccc1NC)=O N1(C(c2c(CC)nn[nH]2)=O)CCCC(O)(CCNC(=O)C=CBr)C1 N1(C(Cc2cccc(C)c2)=O)CCOCC(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 CC(C)CC(C)C(=O)N1CC(C)(NC(c2cnc(N3CCOCC3)cn2)=O)C1 C(=O)(C1SCCc2ccccc21)N1C2CC(NC(c3cncn(C)c3=O)=O)(C2)C1 C(=O)(C(CNC(c1nscc1C)=O)C(C)(C)C)NCCNC(=O)NCC C1(C(=O)NCC(C(=O)N(C2CN(C(C)C)C2)C)N(C)C(CC)CO)CC2CC(=O)C1O2 N1(C(CCCC)=O)C(CNC(=O)C(O)CC(C)(C)C)CC2CCCC12 C1(C#N)(C(N(CCCCN(C)C(C2CC23CCC3)=O)C)=O)CC1(C)C CCCC(CC(C)C)C(=O)N1CCC2CN(C(=O)CCCC(C)(C)C)CC12 c1(OC)ccc(C(=O)NCC(C)NC(c2nn(C)cc2C(C)=O)=O)c(F)n1 c1(-c2ccc(COCC)s2)ncn(C)c1N(C=O)C1CC1 C1(C(=O)NC2CCC(NC(c3cc(N(C)C)n[nH]3)=O)C2)CN2CCC1CC2 N1(C(CCC2(C)CN(C(C3C4CC5C(C4)C35)=O)C2)=O)CC2CCCC1C2CO CCC(C)CC(=O)NCC1CCC(NC(C2CCC(=O)O2)=O)CC1 N1(CC)CCC(NC(c2sccc2CNC(c2ncc(F)cn2)=O)=O)C1=O C1(C(=O)NC(C(C)(C)C)C(=O)NC2CC3CCC(C2)O3)CC(=O)CC12CCC2 Cc1sc(=O)n(CC(=O)NC23CCC2CN(C(c2ccc(=O)n(C)n2)=O)C3)c1C N1(C(c2c(CC)c[nH]c2)=O)CCCC(C(C)(O)CNC(=O)Cc2c[nH]nc2O)C1 N1(C(Cn2nc(C)oc2=O)=O)CCCN(C(=O)Cc2scnc2C)C(C)C1 C1(C2CC2)(NC(C(CNC(=O)Cc2cn(C)cn2)N(C)C)=O)CCOC1 c1(C(=O)NC2CC(O)CN(C(C3CCCSC3)=O)C2)cnn2c1C(=O)NCC2 c1(CC(C(=O)NCCN(C(=O)CCC(N)=O)CCCCCC)C)c(C)noc1C C1(NC(C(N2CSCSC2)C)=O)CC2CCC(C1)N2C(c1cnco1)=O CS(C)(=O)=NC(=O)C(=O)NC(CNC(=O)CC1CC(F)(F)C1)C1CC1 C1(CNC(=O)CC2CCSCC2)CN(C(C2(Cl)CCC2)=O)CC12CC2 CCC(CC(=O)NCC12CC1CN(C(c1cnc(S)nc1)=O)C2)C(F)F c1(C(=O)OCC)ccc(NC(C2CCCNC2)=O)c(Cl)c1 c1(C(=O)NC2CCC3CCN(C(CCCCOC)=O)C32)cncc(P(C)(C)=O)c1 CC1OC2CCC1(NC(=O)C=CC1=CN(C(=O)OC(C)(C)C)CCO1)C2 C1(c2nnnn2CCCC2CC2)(NCCc2c(OC)cccn2)CCOCC1C N1(C(C(CC)=CCCC)=O)CCCC(N(C(=O)Cc2ccccc2)C)C1 c1(C(N)=O)ccc(CC(=O)NC2(C)CCN(C(=O)C=C3CCC3)C2)cn1 c1(OC)nc(C)ccc1C(=O)NCCC1(NC(=O)C(O)C2CC2)CCC1 N1(C(C)=O)C(C(=O)NN2CCCC2Cc2ccc(F)cc2)CC2CC12 C1(CNC(c2c[nH]c(=NC)s2)=O)CCCCN(C(C2CNC(=O)CC2C)=O)C1 c1(CNC(C2(CC(=O)OC)CC2)=O)nocc1C(=O)NC1CC(N(C)C)C1 C(C)(C)(C(N)C(=O)NNc1cc(Cl)c(Br)cn1)OC c1(NC(=O)NC2(c3ccc(Cl)cc3F)CCCC2)ccc(C(F)(F)F)c(Cl)c1Cl c1(C(N(C(C2CCC(C)(C)C2)C(=O)NCCCSC)C)C)nc2ccccc2[nH]1 c1nc2c(NCCCN3CC=CC3)[nH]c(=NCc3cccc4nsnc34)nc2s1 C1CN=C2N=c3sccc3=C(N2)N1.N1(CC)CCCC1.C(CCCC)NCCC=C C1(CC(=O)NC(CC)(C)CCNC(=O)Cc2cnoc2)CC2CCC1CC2 C(=O)(C(C)(C)CC(C)C)N(C)CC1CCN(C(CSc2ccc(C)cc2)=O)CC1 Cc1[nH]nc(Cl)c1C(N1CCC(CN(C(=O)C=CSCc2ccco2)C)CC1)=O C1(C(N(CCN(C(c2n(CC)ncc2Cl)=O)C)C)=O)CC12CCOC(C)C2 N1(C(c2ccccc2)C(=O)O)CC(C(F)(F)F)CCC1C(=O)OC C1(C(N2CC(NC(C(CSC)C)=O)C2)=O)Cc2c[nH]cc2S1(=O)=O c1(NCC(N2CC(C(=O)Nc3cccnc3)C(O)C2)=O)cccc(C(F)F)c1Cl C1(CNC(C2(C#C)CN(C(C3CCCOC3)=O)C2)=O)CCC2(CC2)CO1 C(CC(C)C)(C(=O)NC1CCN(C(c2cccc(OC)n2)=O)C1(C)C)OC C12(NC(CC(CCC)O)=O)CCCC1N(C(c1cccc3[nH]ccc13)=O)CC2 Cc1cc(CC(=O)NC(CNC(c2cncn2-c2ccccc2)=O)CO)n[nH]1 N1(C(C2(COC)CCC2)=O)CCC(CO)(CNC(C2CC(S(C)(=O)=O)C2)=O)CC1 N1(C(CCCNC(N)=O)=O)CCC(F)(c2cn(Cc3ncoc3C3CC3)nn2)C1 C(=O)(C1=CCC2CCC1N2C(C1COC(=O)N1C)=O)N1CC(C)N(C)CC1 C1(C(=O)NCc2nc(C)c(C)s2)CCN(C(=O)c2cncc(C#N)c2)O1 C1(C2CC2)(C(N2C(C(=O)NC)COCC2)=O)CN(C(=O)CC2CCCC(O)C2)C1 N1(C(CN2C(=O)CCC2=O)=O)CC2CCC2(C(N2CCC(Br)C2)=O)C1 N1(Cc2ccc(C#N)s2)CC2CC1CN2C(C1CCCC1O)=O c1(C(=O)NC(CCCNS(C)(=O)=O)=O)ccc(SCc2cn(C3CNOC3)nn2)cc1 Cn1ccc(C=CC(=O)NCC=CC(=O)NC(C2CCCO2)(C)C)c1 C1(=CC(N2CCC(NC(Cc3cnc(C)o3)=O)C(C)C2)=O)CC2CCC(C1)N2C C(=O)(CS(=O)CCC(F)(F)F)NCC1(CNC(C=Cc2ncn(C)c2)=O)CCC1 C1(C(=O)NCC2CCN(C(c3n(CC#C)ccc3)=O)C2)CCC2(CCCC2)CC1 Cc1nc(C(N2CCCOC(CNC(c3sccc3C(C)=O)=O)C2)=O)cc(O)n1 C1(CC(=O)NCC(CN(C(C(C)OCC=C)=O)C)(C)C)CC(=O)NC1=O c1(C(=O)NC(CC(C)NC(C(C)=C2CCCC2)=O)C)cc2oc(Cl)cc2[nH]1 C1(C(N2CCC(OCC#C)C2)=O)CC=CC(NC(c2ccnc(OC)c2)=O)C1 CC1CN(C(=O)CS(=O)(=O)N(C)C)CC(CCNC(c2ccc(F)cc2F)=O)O1 C1(NC(=O)C=CCN2CCCC2)CN(Cc2cnc(Cl)s2)CC12CC2 C(=O)(C(O)CCCNC(=O)CC1CCCC(=O)C1)NC(C)C(=O)NC1CC1 c1(C(N2C(CNC(=O)C(=O)Nc3ncc[nH]3)CCC2)=O)cccc(Cl)c1C(F)F C1(NC(CCC2(C(=O)OC)CCCC2)=O)COCCN(C(=O)Cc2ccno2)C1 C(CCC(C)(F)F)NC(N1CCC(n2cc(NS(C)(=O)=O)nn2)C1)=O CC1(CNC(=O)C(c2cccnc2)=O)CCN(C(c2cccc(C(F)(F)F)c2)=O)C1 C(=O)(CCCN(C)N=O)NC1CN(C(c2cc(OCC)n[nH]2)=O)CC1(C)C N1(C(C2C(OCC)C2)=O)CCC(NC(c2ncn(C)n2)=O)C(CC)C1 C=CCC(C(=O)N1CC(C)(CC)C1)NC(c1c[nH]c(C)c1)=O C(=O)(C(C)(F)C(C)(C)F)NCC(CNC(CN(C1CCSC1)C)=O)O N1(C(CC)=O)CSCC1C(N1CCC(C(C)NC(=O)CSc2nncn2C)C1)=O C1(NC(COCC#C)=O)CCC2CN(C(C3CCc4n[nH]cc4C3)=O)CCC2C1 C1(C(N(CCCO)CC#C)=O)CCN(C(c2cncnc2)=O)C(C)(C)C1 C(C)(CO)(C(=O)NCCC(C)NC(C1(CO)CC1(F)F)=O)NC(C)=O N1(C(c2c(C)cno2)=O)CCC(C)(CNC(c2cscc2C#N)=O)C1 C(=O)(C1=C(Cl)CCCC1)NC1CCN(C(c2ccc(C(=O)OC)cc2)=O)CC1C C12(C(=O)NCCCN(CCCNC(C(C=C)(C)C)=O)C)CCC(CC1=O)C2(C)C C1(C(n2cc(N(C(=O)C#CC3CCCC3)C(CO)C)nn2)C)CCn2ncnc2C1 C(=O)(C1COc2ccc(Cl)cc21)NC1C2(CN(C(CC(C)OC)=O)C2)SCC1 N1(CC(C)NC(C2(c3ccc(OC)cc3)CC2)=O)CC(C)OC(C)C1 CCC(CC)C(C)C(=O)N1CCCC(CC(N2CCC(O)(CO)C2)=O)CC1 c1(C(N2C(CCCC)CN(C(=O)CC3CC3)CC2)=O)cc2n(n1)CCCC2O C1(CC(N2CC(C)(C(N(C)Cc3ccn(CC)n3)=O)C2)=O)CCCC(C)C1 N1(C(CN(C(=O)OC)C2CC2)=O)CCC(C(=O)NC(C)C(C)n2cncn2)C12CC2 Cn1cc(C(N2CC(NC(=O)COCC3CCCO3)C2)=O)c(O)n1 N1(C(C(C2CC2)OC)=O)CC(CNC(c2ccncc2Cl)=O)CC12CCOCC2 N1(C(C2(CC)CCOCC2)=O)C2COCC1CC(NC(c1cnc(S)nc1)=O)C2 CCC(=O)CCC(=O)N1CCC(CC(=O)NC2CC(C)C2)(OC)C1 C1(C(=O)NCC(C(=O)OC)(F)F)CN(C(c2ccc(C#N)o2)=O)CC1(F)F N1(C(CSCC=C)=O)CCCC(C2(NC(=O)COCC3CCCO3)CC2)CC1 C(=O)(CCCC(=O)NCCC(C)(C)CNC(=O)CC1(C)CC1F)NCC c1(C(=O)NCCN(C(=O)C(O)CC2CCCCC2)C)c(F)cccc1Br Cc1cc2[nH]c(C(N3CCC(CNC(=O)Cc4cc(F)ccc4C)C3)=O)cc2o1 N1(C(C2C(COC)CC2)=O)CC(O)CC1CC(=O)NCCN(C)C1CC1 CC(CCC(=O)NC12CC(CNC(=O)C#CC3CC3)(C1)C2)N(C)C C(=O)(CCS(=O)(=O)N(C)C)N1CCC(N(C(C2C(C(=O)OC)C2)=O)CCO)CC1 c1(C(N(CCNC(C(CC=C)c2ccccc2)=O)CC)=O)cc(C)c(C)c(C)c1 C(=O)(C(CCc1ccncc1)NC(c1cc(Cl)n(C)n1)=O)N1CCC(OC)C1 C(=O)(CCC(C(C)C)NC(=O)Cc1cc[nH]n1)N(CCOC)CC1CCCO1 C1(C(N2C(C)CC(NC(c3cc(C4CC4)no3)=O)CC2)=O)CC12CCC(=O)CC2 c1(C(=O)NCCC2N(C(Cc3nc(C)sc3)=O)CCCC2)c(C)nn(C)c1F C(=O)(CC(C)C(=O)NCC1(F)CC(NC(=O)C(n2ccnc2C)C)C1)OCC C12(CNC(C(CC3CC3)OC)=O)CCC(CC1)N(C(c1n[nH]c3c1CCC3)=O)C2 N1(C(CNC(CCC)=O)=O)CCC(C(F)C(=O)N(CCN=[N+]=[N-])C(C)C)C1 c1(C(=O)NCC2(NC(CC(=C)C)=O)CCOC2)ccc2cc(F)ccc2n1 c1(C(C(N2CC(NC(c3cn(CC)nn3)=O)(COC)C2)=O)=O)cnc(CC)c(C)c1 C1(CCOC)(C(=O)N(CC(C)(CN(C(=O)Cc2ccc(Cl)s2)C(C)C)OC)C)CCC1 C1(C(=O)NCC2(C)CNC(=O)O2)CN(C(=O)Cn2c(O)nnc2O)CC1C1CC1 CC12CN(C(=O)CC3CC4C=CC3C4)C(C(=O)NCC3(O)CCSC3)(C1)C2 N1(C(CCN(C(C)C)C)=O)CCCC1(C(=O)NCC1C2COCC12)C(C)C C1(CC=C)(NC(=O)CC2CC(C(C)(C)C)C2)CCN(C(c2ccc(C)cn2)=O)C1 C1(NC(c2oc(CC)c(C)c2)=O)CC2CC1N(C(C1(CSC)CCC1)=O)C2 c1(C(=O)NC(C2CCN(C(c3c(C)nc(Cl)s3)=O)CC2)C)ccc2c[nH]nc2c1 Cn1ccc2cc(C(=O)NC3CC3NC(=O)CCc3ccc(F)cc3)cnc12 N1(C(C2CCC(NC)CC2)=O)CCC(F)(CNC(c2cc3scnc3[nH]2)=O)CC1 N1(C(c2c(C)c(F)cnc2)=O)CC(C)(C)CCC1CNC(=O)CCC(C)(C)F C1(CCNC(C(C)c2ccsc2)=O)COCCN1C(=O)CCc1ccccc1Cl c1(C(N(C(C(N2CCN(CC)CC2C)=O)CC(F)F)C)=O)ccc2cc[nH]c2c1 CC(=O)CCCC(=O)N1CCC(CNC(c2ccc(C3CC3)nc2)=O)CC1C N1(C(c2c(C)nc(C3CC3)o2)=O)CC2CC(N(C)C(c3cnn(C)n3)=O)C1C2 Cc1ccc(F)cc1C(=O)NC1CC1CNC(C1CC(n2cnnc2)C1)=O CC(C)C(CCNC(C1CCC1)=O)OC(c1ccc(O)cn1)=O c1(C(=O)NC2C(C)(C)C(CNC(C3CC4(CSC4)C3)=O)C2)ccc2ncnn2c1 C=CC(CC)CC(=O)N1CCN(C(C2CSCN2C(C)=O)=O)CC1C c1(C(C)C)cc(C(=O)NCC(O)CCNC(C2C=CC=CC=C2)=O)cc(F)c1 N1(C(C(C=C)(C)C)=O)CCCCC(CNC(=O)C(C)(C)ONC(=O)OC(C)(C)C)C1 n1(CCC)cncc1CNC(C1CCOC1CNC(=O)CSc1cn[nH]c1)=O CC(O)CCCCCC(=O)NCCC(C)(C)NC(c1cc(C2(C)COC2)no1)=O c1(C(=O)NCCOC2CN(C(C3(C)CCCS3)=O)C2)cc2c(cn1)CCCC2 C1(CC)C(NC(c2ccnnc2O)=O)CCCN1C(=O)CNS(N)(=O)=O C(=O)(CC1CN(C)c2ccccc21)NC(CN(C(c1c(C)[nH][nH]c1=N)=O)C)C C1(N(C(c2n(CC)ncn2)=O)C)CN(C(c2cc(C(C)(F)F)n[nH]2)=O)CC1O N#Cc1c(NC(C2CCC(NNCc3cccc(F)c3O)CC2)=O)ccnc1Cl C1(NC(c2c(O)ccc(OC)c2)=O)COC2C(NC(=O)CC(C)CF)COC12 c1(C(=O)NCC(C)(C)OCC(=O)NC(Cc2ncc(C)[nH]2)C)cc2cc[nH]c2cn1 c1(NC(C)=O)ccncc1NC(C1CC(O)CN1C(=O)CNS(C)(=O)=O)=O C(CC(C)C(=O)NC1CC(O)(CNC(c2ccc(N(C)C)nn2)=O)C1)OC c1(N2CCC(O)CC(C)C2)nc(=NCCCCC(N)=O)[nH]c2c1CCC2 N1(C(CCCCCC)=O)CC2CCC1C(CNC(=O)CCCC#N)C2 c1(C(N2CCN(C(c3nncc(OC)c3)=O)CC2)=O)cnc(C)cc1C CN1CCN(c2nccc(C(F)F)c2Br)CC1CS N1(C(C2(F)CC2)=O)CC2(C1)CN(C(=O)C(F)CC1CC1)C2 CC(CCNC(=O)CN(C(C1CNC(=O)C1)=O)C1CC1)CCO C#Cc1ccc(Cl)c(C(N2CC(NC(C3(C)CCC(O)CC3)=O)C2)=O)c1 C1(CNC(CC(C)C)=O)CCCCN(C(=O)C(C)(O)C(C)(C)C)CC1 Cc1cccc(C)c1C(C)NC(c1nnnn1C)(c1nnnn1CCCF)C CCC(CNC(=O)C(=O)NCC1CSCCO1)C(=O)O C(CC1CC1)(C(=O)NC(c1ccnn1C)C(=O)N(C)Cc1csc(C)n1)OC CC1CN(C(=O)CC2(O)CCOCC2)CCC1NC(=O)C=CC1CCCC1 N1(C(Cc2cn(C)nn2)=O)CCCC(F)(CNC(c2cccc(=O)o2)=O)C1 CCC(N=c1[nH]c(=NCC2CC3C=CC2O3)[nH]c2c1SCC2)c1ncc(C)[nH]1 C1(C2CCCN(C(c3ccnc(CO)c3)=O)C2)(NC(c2c(C)occ2)=O)CC1 Cc1cccc(CNc2ncc(-c3cnn(C4CCOC4)c3)s2)c1 Cc1cccnc1CC(=O)NCC(C)(C)NC(c1ccc(C(O)CF)cc1)=O C1(CNC(C(C)N(C)C)=O)CCCC1NC(=O)C(C)(C)C1CCCC1 N1(C(CSCC)=O)CCCCC(NC(=O)CCCCN(C)C(=O)OC)C1 N1(CC(=O)NCC2CCCC2NC(c2cnc[nH]2)=O)CCCc2sccc2C1=O C1(CNC(C2C(C)C2C)=O)CC2COCC2N1C(c1cn(C2COC2)nn1)=O Cc1cc(C)n(C(C)CNC(c2cnn(CCNC(C3COC(=O)N3)=O)c2)=O)n1 C#CCCC(C(=O)NCC(C)CCCO)NC(=O)CC1(C(=C)F)CCC1 C1(NC(=O)CCc2cc[nH]n2)CCN(c2ncnc3scnc23)CC12CCC2 c1(C(=O)NCC(CNC(c2cn(CC=C)nn2)=O)(C)F)nnn(C)c1N c1(OCC)ccc(CCC(=O)NCCCC(C)NC(c2sc(C)nc2C)=O)cc1 C1(C(N2C(C)CC(NC(=O)Cn3nnc(=O)[nH]3)CC2)=O)CCOC2(CCC2)C1 C#CCC(CC#C)n1cc(CC2CCCN2)nn1 C1(CCC)(NC(C2CC3C=CC2C3)=O)CCCN(C(=O)C=Cc2ccco2)C1 c1(C(=O)NC2CC3CN(C(CN(C(C)C)C)=O)CC2C3)ccc(S(C)(=O)=O)cc1 C(C(C)(O)CC(=O)N1CC2(CCC2NC(c2coc(N(C)C)n2)=O)C1)OC C1(O)(CNC(C(CC)NC(=O)CC2CC(C)C2)=O)CCCOC1 n1(CC)ncc(CNC(=O)C(C2(O)CCC2)NC(=O)Cc2cc[nH]n2)c1C N1(C(c2cncc(SC)c2)=O)CC2(CCCN(C(C3CCSC3)=O)C2)C1 c1(C(=O)NCC2(NC(C(=Cc3ccco3)C)=O)CCC2)ccc2c(c1)CCCO2 CCC(Cc1ccc(C(C)(C)C)cc1)C(=O)N1CC(C)(c2ccccc2)C1 CC1CCCN(C(C2(Cc3ccsn3)CC2)=O)C1CNC(C1CCCC(O)C1)=O N1(C(C2CCN(C)C2)=O)CCC2CCN(C(c3ncc(N)cc3Cl)=O)C2C1 c1(N(CCCOC)C(=O)NCCOCCO)ncc(Cl)cn1 N1(C(Cc2cc(OC)no2)=O)C2CCC1CN(C(C1CCCN1CC(C)C)=O)C2 c1(CC(=O)Nc2ncn(CCNC(c3c(CC)n[nH]c3)=O)c2)ccc(F)cc1 c1(COC(C2C(C#C)C2)=O)ccc(S(N)(=O)=O)o1 c1(CC)ncncc1C(=O)NC1CN(C(=O)CCNC(=O)OC)C1 N1(C(=O)CC2CC2)CCCN(C(C2COCC2n2cccn2)=O)CC1 CCC(C)(CC)C(=O)NCC(O)CNC(c1cc(CO)ccc1OC)=O N1(C(c2c(OC)cccn2)=O)CCC2CCCC12CNC(=O)CC1=CCOCC1 c1(C(=O)NC(C(C)NC(CC(=O)OC)=O)CO)c(C)c2ccc(F)cc2oc1=O Cc1cc(C(=O)NC2CCCCN(C(=O)C3=CC(C)CC3)C2)nc(C)c1 c1(C(N2C(C(C)NC(C3(C=C)CCCCC3)=O)CCC2)=O)ccc2c(c1)COC2 c1(OC)ccncc1C(N1CCOC(C(C)NC(=O)CC2(OC)CCC2)C1)=O c1(OC)cc(CC(=O)NCC(C)NC(=O)C(CC#N)c2ccccn2)cc(Cl)c1 C(=O)(CCCNC(C)=O)N(C1CCN(C(=O)CC=CC(C)(C)C)C1)CC#C C1(CCC)CCC(O)(C(=O)NCC2(F)CCN(C(C3CC3C(F)F)=O)CC2)CC1 C(C)(C(C(=O)NCc1sccc1C)C(C)C)NC(c1cc(C)nnc1)=O C1(O)(CC(=O)NC2CC(CNC(C3C(C(C)O)C3)=O)C2)CCOCC1 CC1(C)C2CCC1(C)C2C(=O)NCC1CCC(NC(=O)C(F)F)CC1 C1(=O)C(C)(C)C(C)N1.c1(C(=O)NC2C(CCOC)C2)cc(O)nc(C)n1 Cn1cc(C(N2CC3C(NC(C4CC45CCCC5)=O)C3C2)=O)c(C(F)F)n1 c1(C(=O)OCC)nc(N(C)CCOC(CN2CCCC2)C(C)C)cc(C#N)n1 c1(NC)nc(C)ccc1C(=O)N(CCCOCCN(C(=O)CC(C)F)C)C N1(C(N(C(C)(C)C)C)=O)CC2CCN(C(n3ccn4nccc4c3=O)=O)C2C1 c1(CC(=O)NCC(C)NC(C2CCN(C3CC3)CC2)=O)c[nH]c2c(F)cccc12 CCC(C)C(O)C(C)C(=O)NCC1CCC(C)CN1C(=O)COC c1(OCCOC)ccc(C(=O)NC(C)CNC(C2CS(=O)(=O)C2)=O)cc1 C(=O)(CS(=O)C(F)(F)F)NCC1(OC)CCN(C(C2(F)CC2C)=O)CC1 C(C(C)(C)C(=O)N1C(CO)CC1C)NC(C)=O.c1(C(=O)O)cn(CC)nn1 C1(C(=O)Nc2c(C(C)C)ncnc2)CN(C(C2CCC(C(N)=O)C2)=O)C2(CCC2)C1 c1(C(=O)NC2CC(N(C(COC3CCN(C)CC3)=O)C)C2)c(Cl)cc(Cl)nc1N N1(CCNC(C2(F)CCC2)=O)CCCN(C(=O)Cc2ccccn2)CC1 C(=O)(C1=CC2C=CC1C2)NC(CCOC)C(=O)N1CCCC(N2CCC2)C1 c1(SC)cccc(C(=O)NC2CCN(C(C3CCCO3)=O)C2)c1 Cc1cc(C)c(C(=O)NCCC(C)N(C(=O)CC2CCCOCC2)C)[nH]1 c1(NC(COCCOCC#C)=O)cccc(Sc2ccc(C)cc2)c1 C(C1C(C(=O)NC(C)(CNC(=O)CC2CCOC2C)C2CC2)C1(C)C)=C(C)C N1(C(C(C)(Cl)Cl)=O)CCCCC12CC(NC(=O)Cc1cc3ccccc3o1)C2 c1(C(CNC(COCCC=C)=O)NC(=O)CCc2cnoc2)cc(F)cc(Cl)c1 CCCCC(CC)C(=O)N1CCC(N(C(=O)Cn2ccnn2)CCC)CC1 c1(C(N(C2CN(C(C(CC)N3CCCC3=O)=O)C2)C)=O)nn(C)c(Cl)c1Cl c1(SC(C(N2CCC(CN(CCO)CC)C2)=O)C)ccc(F)cc1 N1(CC(=O)N(CCNC(CCN(C)CCO)=O)C)CCc2ccccc21 c1(CC(=O)NCCOC2CCN(C(C(CC)=CC)=O)C2)ccc2[nH]ccc2c1 CCC(C)(COC)C(=O)N1CCC(C(C)(C)C)(CNC(c2cn(C)[nH]c2=N)=O)C1 C1(CCNC(CCNC(C)=O)=O)(C(=O)NCC2(O)CCCC2)CCCC1 C(=O)(C1=CC2(CCN(C(C3CC3(C)C(F)F)=O)C2)C1)N(CC(=C)Br)C1CC1 C1(O)(CCNC(CCSCC(N)=O)=O)CCN(C(c2cc[nH]c2)=O)C1 CCCC(CNC(=O)CCc1ccncn1)C(=O)NC1(C)CC=CC1 c1(C(=O)NCC(C(C)C)NC(c2ncccc2Cl)=O)nccc2c1CNC2=O C1(NC(c2c(C)nn[nH]2)=O)CCCCN(C(C2CCCN2C(C)C)=O)CC1 C1(C#N)(c2n(-c3c(C)cccc3C)nc(CCO)n2)CC12CCCC2 CCCCC(C(=O)NC1COCCC1NC(=O)C(CC)CC)ON=C(C)C CC(CC(F)(F)F)C(=O)N1CCC(NC(c2n[nH]c(C3CC3)c2Cl)=O)C1 c1(C(=O)NCCCC2N(C(CSCC(N)=O)=O)CCCC2)onc2ccccc12 N#Cc1cc(Cl)c(C(N2CC(F)(CNC(=O)CCN3CCC(O)CC3)C2)=O)s1 C(=O)(C1CC(=O)c2c(F)cccc21)NC(CNC(c1n(CC)nnc1C)=O)CO C1(CC)CCC(C(N2CC(OC)CC2CNC(=O)C(C)CF)=O)CC1 c1(N2CCC(C3N(C(C=CC)=O)CCCCC3)CC2)nc(CCC)ccc1C#N c1(OC)ccc(CCC(=O)NCC(C)NC(=O)C(n2cnc(C#N)n2)C)c(F)c1 c1(N(CCCC)C)nc(N2CCC(C3CCCCC3)C2)c2c(n1)CCS2 c1(C(N2C(CO)CC(NC(CS(C)(=O)=O)=O)C2)=O)cc2cc(F)ccc2[nH]1 C1(C(C)C)(C(N2CCC(CCCO)C2)=O)CCCN1C(=O)CC(C)N(C)C Cc1ncnc(N(C(=O)C(C2CCN(C(C3CC(=C4CC4)C3)=O)C2)F)C)c1C N1(C(C(C)C2CCCC2)=O)CCC(C2CC2)C1CNC(c1ccc(=O)oc1)=O Cc1cc(C(=O)NC(C)(C)COC(C)(C)C)sc1-c1ccccc1Cl N(C(=NCCCCCS(C)(=O)=O)NCc1ccc2[nH]ccc2c1)C(CC)C C(O)(CSC)(CCC(F)(F)F)c1n(CC)ncc1 Fc1ccc2cnc(NC3CN(Cc4ccc(F)c(Cl)c4)CC3(F)F)nc2c1 c1(CC)ccc2c(c1)CCC1C2OCCN1n1cc(-c2cccc(F)n2)nn1.CS C(=O)(C1=C(C)N(C)c2nnnn2C1)NC(CC)(C)CNC(c1ccncc1)=O C1(CNC(c2c(C)nsc2)=O)CCN(C(C23CCC2C3)=O)CC1(F)F C(N=c1nc2c(c[nH]1)C1CCC2C1)c1cc(C(=O)OC)c(Br)cc1 N1(C(CCC#CC)=O)CCCC(C2CCN(C(=O)C(F)(F)CC)CC2)CC1 C1(c2n(C)cnn2)CCCCC1COC(C1(F)CN(C(c2ccco2)=O)C1)=O C1(C(=O)NCCCSCC)CCN(C(=O)C=CCOC)C12CC2 C(=O)(C1CCc2scnc21)N(CC(C)(C)CNC(=O)CCc1ccccc1F)C C1(C(=O)Nc2ccc(CCF)cc2)(NC(=O)C=Cc2ccoc2)CCCCC1 C1(C(=O)NC)CCN(C(=O)CN(C(C2CC3(CC3)C2)=O)C(C)C)C1C c1(C2CCN(NC(N3CCC(C4OCCO4)CC3)=O)C2)ccc2c(c1)OCCO2 C12(NC(c3c(Cl)cn(CC)n3)=O)CCN(C(c3ccc(N)c(F)c3)=O)CC1C2 C1(C(N(CC)CC2CCN(C(c3cc(CO)[nH]n3)=O)CC2)=O)CC2CCC1C21CC1 O=C(C1CCCc2nc[nH]c21)NC1CCN(C(c2cnc3c(c2)COC3)=O)C1 C1(C(C)(C)C)CC(C(=O)N2CCC(c3cn(Cc4ccc(Cl)s4)nn3)C2)=NO1 N1(C(CCOC(C)C)=O)CC2CCC(C1)N2C1CCN(C(C2CCC2C)=O)CC1 N1(C(C(C)(C2(C)CC2)OC)=O)CC2(CCN(C(=O)CCC(C)SC)CC2)C1 C1(NCC(C)OCC2CC2)CN(C(=O)OC(C)(C)C)CC12CC2 C1(C)(C(=O)NC2CCC(NC(c3ccc(CCC)[nH]3)=O)CC2)CCN(C)C1=O CCC(C)CC(=O)C(=O)NCCOC1(CNC(=O)CCSC)CCOCC1 N1(C(c2cccc(C(=O)NC)c2)=O)CCC2CCN(C(C3CCC(=O)N3)=O)C2C1 N1(C(C(C(COC)C)C)=O)CCC(C2(O)CN(C(=O)CCCCSC)C2)CC1 c1(Cc2cn(CC(=O)N(C(C)(C)C)Cc3cncs3)nn2)ccccc1OC(F)F C1(NC(c2c(C(C)NC(C)=O)noc2)=O)CCN(C(C2(C)CC=CCC2)=O)CC1 N1(C(C(CC)SC)=O)C(C(=O)NC2(CO)CCCC2OC)CC2CC12 C=CCCCCCC(=O)NCC1C(O)C(O)CN1C(c1cc(CC)on1)=O c1(OC(CC)C(=O)OC(C)(C)C)cccc(C(=O)OC(C(CCF)OC)=O)c1 c1(C(C(F)(F)F)NC(C(c2ccc(C(=O)O)[nH]2)(F)F)=O)ccc(Cl)cc1F C1(NC(CCc2cc(C)on2)=O)C2CC3CN(C(c4[nH]ncc4C#N)=O)C1C3C2 Cc1cnc2ccccc2c1C(=O)NC1CC2(C1)CN(C(=O)CCC1CCC1)C2 c1(CC(c2cn(C3CN(C(=O)OC(C)(C)C)C3)nn2)C)ccnc(Br)c1O C12CCN(CC1)C(=O)OC2C(=O)OCC.C(C(C)CN(C)C1CC1)OC(C)(C)C N1(C(C(CC)C#N)=O)Cc2nccn2CC(NC(=O)CSc2ccc(C)c(C)c2)C1 c1(OC)nccc(I)c1C(N1CCC(C(N2CCC(C)C2)=O)(OC)CC1)=O O=C1CCC(C(=O)NC(C(N2CCCC2CCCO)=O)C2(O)CC2)C1 Cc1cc(C)nc(-c2ccsc2)n1.c12nc(sc1C)C(C)OC(=O)CC2.C1CS1 c1(C(=O)NCC(C)(C)NC(c2ccc(CO)cn2)=O)cncc(N)c1 N1(C(c2ccc(OC)o2)=O)CCC(C(N2CCC(C)(N(C)C)C2)=O)(C(C)C)C1 N1(C(c2c(NC)cccc2)=O)CCCCC(C(=O)NCCC(C)(C)N(C)C)C1 c1(C(=O)NCC2CCN(C(C3CCC(=O)NC3)=O)CC2)ccc(F)cc1F CCC(C)C(=O)C(=O)N1CCC(C)C1C(=O)NOCCc1ccccc1 C1(C(C)C(=O)N2CCC2C(=O)N(C)C)CCN(C(=O)C=Cc2ccco2)C1 Cc1cnn(C(C)C(=O)NCC2(CN(C(=O)C(C)(C)c3cscc3Cl)CC)CC2)c1 c1(SC)ccnc(NCC2(CNC(=O)C(C(C)C)S(=O)(=O)C3CC3)CC2)n1 C1(C(=O)NC(C#C)C2CCC2)(CNC(C2CNC(=O)C2)=O)CC=CC1 c1(C(N2CC(NC(C3N(C)CCCC3)=O)C3C2C3)=O)cc2c([nH]1)CCCC2=O C(C)(CS(=O)(=O)CC)n1c(CC(CCC)C)nc(-c2ccccn2)n1 C=CCC(CNC(c1cc(CO)n(C)n1)=O)C(=O)N1CC(CO)C1(C)C Cc1cccc(Br)c1C(C(=O)NC1CCNC(=O)C1)NC(C1CC1CC(C)C)=O c1(CN2CC(F)CC(C(=O)Nc3ncc(Br)cc3Cl)C2)ncc2ccccn12 c1(C(=O)NCC2CN(C(C3(CC)CC(F)(F)C3)=O)CC2O)c(C)cccc1Cl C1(NC(c2cc(CC)nnc2C)=O)CCOC2(CCN(C(=O)C(O)CC)CC2)C1 N1(C(c2c(OCC=C)ccc(Cl)n2)=O)CCC(NC(=O)CCCC2CC2)C(O)C1 C1(CC(=O)NC(CN(C(c2cnn(C(C)C)c2Cl)=O)CC)C)C(=O)NN=C1C CC1CNc2c(C(=O)NCC3CCN(S(C)(=O)=O)C3)cnn2C1 CC1(CNC(c2sccc2C(F)F)=O)CC(F)(F)CN1C(=O)CCF CC1(N)C=C(C(=O)NC2CCC(NC(C3CCCC4(CCC4)O3)=O)CC2)C=C1F C12(C(=O)NCC(C)(C3CC3)NC(C=C3CCN(C)CC3)=O)CC(C)(CCO1)C2 N1(C(c2cnc(C3CC3)o2)=O)CCC2CC2(C(=O)N(C2CCC2)CCN(C)C)CC1 N1(C(CN2CCC(C)CC2)=O)CCC(C)N(C(=O)Cc2nn(C)cc2Cl)CC1 C=C(C)CCC(=O)N(C)CC1CN(C(c2sc(COC)nc2C)=O)CCO1 c1(C(=O)NCC(CNC)(F)F)nc2ccccc2n1-c1ccccc1 N(C(=NCC1CCNC(=O)C1)NCC1COCCO1)CC1(S(C)=O)CC1 C1(NC(CC(CC)OC)=O)CCCC(CC(=O)Nc2c(OC)ncnc2C)C1 C1(NC(c2cc(C)oc2C)=O)C(CN=c2nc(C(C)C)[nH]s2)CCC12CCC2 c1(C(N2CCC(N(C)C(c3sccc3CO)=O)CC2)=O)ccc(N)c(O)c1 N1(C(c2cccc(CC)n2)=O)CC2CCC(C(N3CC4CSCC4C3)=O)(C2)C1 Cn1nc2c(c1C(N1CCOCC1CCNC(=O)CN1CC3CC3C1)=O)CCC2 N1(C(Cc2cc(C)cc(C)c2)=O)CCC2CN(C(c3c(Br)cnn3C)=O)CCC12 CC(C)CC(C)(C)C(=O)NCC1CC(O)(CNC(c2cc(Cl)ccc2F)=O)C1 C1(NC(CCC(=C)Cl)=O)CC2CCC(C1C)N2C(c1cc(N)ccn1)=O S(=O)(=O)(c1ccc2c(ccn2C)c1)N1CC(CCOC)C1 c1(OC)cc(C(=O)NCCC(C)N(C)C(C2CC2(F)F)=O)cnc1Br N1(C(C2CC(CC)(CC)C2)=O)CCC(F)(C(=O)NCCSc2ccncc2)C1 CCCC(C(=O)NCCC1(O)CN(C(=O)C=C(C)C)C1)S(N)(=O)=O C(=O)(CC1=CCCCC1)N(C1CCN(C(c2nccc(Cl)c2F)=O)C1)C N1(C(c2cc(CC)c(F)cc2)=O)CCN(C(=O)C(C)(C)CC(F)F)CC12CCC2 Cc1cn2cc(C(=O)NC3CNC(C)C3)nc2c(C)n1 C1(CN(c2cnc(SC)s2)C(C)=O)CC(=O)N(c2ccc(-c3nn[nH]n3)cc2)C1 c1(C2C(C(N3CC(N(C)C(C4C=CCC4)=O)C3)=O)CCO2)cncc(Br)c1 c1(C(N2CCC(C)C(N3CCC(C)C3)CC2)=O)cc2nccn2c(O)n1 C(C(CC(=O)O)CC(C)C)N(C(N=c1ccc(-n2ccc(C)n2)n[nH]1)=O)C(C)C CCC(C)(C(=O)NC1CCC1NC(=O)C=CC1CC1)NC(=O)OC(C)(C)C C(=O)(C(=O)C(C)(C)C)NCC(C1CCCC1)NC(C(CSC)O)=O N1(C(C(C)OCOC)=O)CCCN(C(=O)Cc2csc(Br)c2)CC1C C1(CNC(CC(=C)C)=O)CC2(CO1)CN(C(C1CCCC(C)(C)CC1)=O)C2 C(=O)(C1=CCCCO1)NC1C(OC)CN(C(c2cccc(Br)c2C)=O)C1 Cc1cnc(C(=O)NCC2CC(C(=O)NC3(C(F)(F)F)CC3)C2)c(F)c1 c1(C(=O)NC23CC2CN(C(=O)CCC2CC2(F)F)C3)cccc2c1OCO2 c1(C(N2CC(O)(CN(C)C(c3cc(C4CC4)on3)=O)C2)=O)ccc(=O)n(O)c1 C1(C(=O)NCC2(OC)CN(C(=O)CC(C)C3CCCO3)C2)CC2(C1)CC(C#N)C2 c1(C(N(C)CC)=O)ccc(C(=O)NC(C)CC(C)NC(=O)NCCC(C)C)cc1 C1(CNC(C(CC(C)C)(C)C)=O)CN(C(=O)C2=C(Cl)CCC2)CCC12CCOC2 C1(C(N2C(CNC(c3c(C(=O)OC)coc3)=O)CC2)=O)CN(C)CCO1 N1(CC)CCN(C(C2(NC(=O)C(C)S(N)(=O)=O)CCC2)=O)CC1C.C1CC1 CCCC(C(=O)N1CCN(C(=O)CCC(F)(F)F)C(CF)C1)S(N)(=O)=O c1(NCC(C)C)ccccc1CNC(=O)Cc1ccncc1 C1(C(N2CC3CC(NC(c4c[nH]cc4Br)=O)C3C2)=O)CCc2ccccc2C1 N1(C(c2[nH]cc(CN(C)C)c2)=O)C2CCC1C(NC(=O)Cn1nccn1)C2 O=C(CCCCCC1CC1)N1CCN(C2CCN(C(=O)CC3CC(F)C3)C2)CC1 N1(c2nccc(C)n2)CCOC2(CCN(C(c3nc(F)ccc3Cl)=O)CC2)C1 c1(N2CC3C(C)C3C2)ncnc(=NC2CCN(C)C(C)C2)[nH]1 C(CCCCC(=O)NC1CCC1NC(c1n[nH]c(C)c1Cl)=O)SC N1(C(CCOc2c(OC)cccc2)=O)CCC(C)(CNC(=O)C(O)CSC)CC1 c1(C(=O)NCCCN(C(=O)CC2CCC(=O)NC2=O)CC)ccc(O)c(F)c1 CC1(C)CC(CNC(=O)C(CC2CCOCC2)NC(c2cc(O)cs2)=O)CO1 C(CC(C)C(=O)NCc1cc(C)c(C(=O)N(C)CCOC)o1)=CC C1(CCNC(c2ccoc2Cl)=O)CC2CCC(C1)N2C(=O)CN1CCCNC1=O C(=O)(CCCCC#CC(=O)NC(C)CN(C(=O)C=NOC)C)OCC C(=O)(CCCCCCn1cc(C2CCCN2C)nn1)N1CCCC(OCC)C1 c1(CN2C(C(=O)Nc3ccc(N(C)C)cc3)CC(O)C2)ccc2ccccc2n1 C1(CC(N2CCC(NC(C(COCC)C)=O)CC2)=O)CCC=CCC1 c1(C(N2C(C)CC(CNC(c3ccc(Cl)cc3)=O)CC2)=O)cccc2[nH]ncc12 CC(C)C(O)C(C)(C)C(=O)N1CCOCC(C(=O)NC(c2n[nH]c(CO)n2)C)C1 N1(C(C(CCC)(C)C)=O)CCCC2(CCCN2C(c2ncc(F)c(OC)n2)=O)C1 C1(CCC(=O)NC2(C)CN(C(=O)COCc3nccs3)C2)CCCC(O)C1 c1(C(N2CC(C(C(=O)NC(C#C)CC3CCCC3)OC)C2)=O)cscc1Cl C(CN=c1[nH]cnc(NCCc2ccc(Br)c(C)c2)c1C)(c1ccsc1)OC c1(C(=O)OC)cc(C(=O)NCC2(NC(C3CC3Cl)=O)CCC2)cc(O)c1 C1(CCNC(CCS(C)=O)=O)CN(C(=O)CCN2CCC(O)CC2)CCCO1 CC(CCNC(=O)C(CNC(=O)C#CC(C)(C)O)CC1CCCC1)C(C)(C)C c1(SCC(=O)NCCn2cc(CSC)nn2)cccc(NC(=O)CC2CSC2)c1 N1(CC)CC(C(=O)N(C2CCN(C(c3cc(C)co3)=O)C2)CCO)CCC1=O N1(C(CN(C)C)=O)CCCOC(CC(c2ccc(Cl)nc2)(C)C)C1 C1(O)(CNC(C2C(=C)C2)=O)CN(C(C2(OCC)CCOC2)=O)C1 C1(NC(CC(c2cccs2)NC(C)=O)=O)(CO)CCCN(C(c2cnco2)=O)C1 C1(OC)(OC)CCC1C(=O)NC(C)(C)CN(C)C(C12COCC1C2)=O C12(C(=O)NC3CCC(CCC(N4CCC(OC(C)C)C4)=O)C3)CCC(C1)OC2C c1(C(=O)NC2CC(N(C(CC=CCC)=O)C)C2)c(C(F)F)cccc1F C1(CCNC(C=C(CC)C)=O)CN(C(C23CCC(C2)C3)=O)CC(C)O1 Cc1cn(C)nc1C(=O)NC1CCC(C)(CNC(c2cnc(=N)[nH]c2)=O)C1 N1(C(Cn2c(C(C)C)nnn2)=O)CC2CCC1CN2C(=O)Cc1ccc(Cl)cn1 C1(C)(N(C)CC)CCN(C(C2CCN2C(C2CC3C(C2)C3(F)F)=O)=O)CC1 c1(N(C(c2cn(C)nc2)=O)C(C2C3COCC23)=O)ccc(Br)c2ccccc12 C1(N(C(C(F)(F)C2(CC)CCC2)=O)C)CCCC(N(C(=O)Cc2cnc[nH]2)C)C1 c1(CC)ncsc1C(=O)Nc1nc(C2CC2)cs1 c1(C(N2CCC(NC(c3ncn(CCOC)c3)=O)C2)=O)c(Br)ccc(C)c1N C1(N(C)C(C2CC2(C)C)=O)CC2(CCN(C(C3CC3c3ccccc3)=O)CC2)C1 N1(C(C(CC)N(C)C)=O)CCC2CN(C(c3cccc(C#N)c3)=O)C2C1 C1(NC(C=CCC)=O)CCN(C(c2cnn(-c3nccs3)c2)=O)C(C)C1 N1(C(c2csc(Cl)c2)C(=O)Nc2c(CC)cccc2C)CC(C)OC(C)(C)C1C N(C(=NCCF)NCCN1CCC1)CCC1(OC)CCSCC1 N1(C(C)C)C(=O)COCC1C(N1CCC(CN(C(=O)C(=O)NCC2CC2)C)C1)=O c1(CC)ccc(C(=O)NC(C)CCNC(C2C(C#N)C2(C)C)=O)cc1Cl c1(CN2CC3C(c4ccc(C)cc4)(C3)C2)cn(C)c2cc(F)ccc12 c1(OC)cc(OC)nc(C(N2CC(O)(CNC(=O)COC3CCCCC3)C2)=O)n1 C1(C(C)(C)Nc2cccc(OCCOC)n2)COc2ccccc2C1 C1(C(=O)NC2CN(C(C3ON=C(CC)C3)=O)C2)CC(C)(C)CC(C)(C)C1 c1(NCCCCCC)ccc(S(=O)(=O)NCC2CCSC(C)C2)c(Br)c1 N1(C(c2c(C)ccs2)=O)CCN(C(=O)CC2CCC3(CC2)COC3)C2CCC12 S(=O)(=O)(c1ccc(=NCCCCCCF)[nH]c1)NC(c1ccc(Br)cc1)C1C(C)C1 C1(C(=O)NCCSCC)CN(C(=O)Cc2nn(C)cc2Br)CCC1O c1(C(=O)NC)cccc(S(=O)(=O)NNC(=O)c2ccc(-n3cccn3)cc2)c1 CCC(CC)CCCC(=O)NC(C)C(C)NC(c1occ2c1CCC2)=O N1(C(CC(CN(C)C)O)=O)CCC(NC(=O)CCOc2ccccc2F)CC1C c1(NC(C)=O)cnc(O)c(C(=O)NCC2CCC2NC(=O)C=C2CCC(C)C2)c1 c1(N(C)Cc2ncco2)ccc(Br)c(S(=O)(=O)NCC2=CCCOC2)n1 C(=O)(CC(C)(C)C(F)F)N1CC(OC)C(NC(c2nc(O)c(C)s2)=O)C1 N1(C(C)=O)CCCC1C(=O)NC1CC(C)(C(=O)N(C)CC2CN(C)C2)C1 N1(C(=O)OCC2C(=C)CN2C(=O)OC(C)(C)C)CCCC2(CCSC2)C1 N1(C(CC(=O)OCC)=O)CCSCC1C(=O)NCCC1CCN(C)CC1 C1(CNC(C2CCn3ccnc3C2)=O)CCCC2(CN(c3ncns3)C2)O1 c1(OC)ccc(Br)c(C(=O)NC(C2CN(C(=O)CN(C)C(C)C)CCO2)C)c1F c1(C(=O)NC2CC(CO)N(C(=O)C=C(Cl)Cl)C2)cccn2cncc12 C1(C(N2CC(O)(CCNC(CCC(=O)N(C(C)C)C)=O)C2)=O)CCCC(C)CC1 C1(CC)CN(C(c2c(C)cnn2CC)=O)CCN1C(=O)Cc1cnc(C)s1 CC(C)(C)CCC(=O)NCCC1CN(C(C2(C)CCOC2)=O)CCO1 c1(CC(=O)N(CCNC(COCC=C)=O)C)ccc(NC(=O)NC)cc1 c1(OC)c(C)csc1C(=O)NCCN1CCN(C(=O)C(O)C(C)C)CC1 C(=O)(CC(C)(C)COC)N1CC(CC(N2CC(CC)SCC2)=O)C(C)C1 C1(C(N(CCCC(O)CO)C)=O)C2CCC(C2)N1C(c1cnn2c1CCC2)=O C1(C(=O)NCC(CC=C)NC(=O)CNC(=O)OC)CS(=O)(=O)CC12CC2 CC(C)C(O)CC(=O)N1CCC(F)C(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1 N1(C(Cc2c(C)ncs2)=O)CCC(C)(C)CC1C(=O)NCC1CCOC1(C)C CCCC(C(O)C(=O)NCC1(C(C)(C)OC)CC1)NC(c1cccc(C)c1F)=O N1(C(CCc2cnc(C)o2)=O)CCC(O)(C(C)NC(=O)CSC2CC2)CC1 C1(C(NOC(C(C)C)CO)=O)CCCN(C(=O)CN(c2ccncc2)C)C1 C1(C)(OC)CN(CC(=O)NCCCOCCC(=O)Nc2nn[nH]n2)C1 CC1=C(C(=O)NC2CCC3CC2CN3C(c2ccc(C(N)=O)[nH]2)=O)CCCO1 c1(OCOC)cccc(S(=O)(=O)Nc2cccc(CO)c2COC)c1Br c1(CCC(=O)NC(C2(O)CCN(C(C3CNC(=O)N3C)=O)C2)C)cncnc1O N1(C(c2ccc[n+]([O-])c2)=O)CC2OCCN(C(C3CCC4C(C3)C4(F)F)=O)C2C1 c1(OCCCC)ccc(C(=O)NCC2(O)CCN(C(=O)CCCN(C)C)C2)cc1 Cc1nn(C)cc1CC(=O)NCC12COC(CNC(c3cn(C)c(O)n3)=O)(C1)C2 c1(CC)cc(C(=O)NCCCN(C(=O)CC2CC2(C)C)C)nn1C c1(C(=O)NCC(CNC(CCCc2cnc(C)s2)=O)O)cnn(C2CCC2)c1C c1(C(N2CCC(C(C)Nc3ncccn3)C2)=O)ccnn1CCc1ccccc1 C(CC(C(=O)NC(C)(C)CCOC)NC(C1CC=CC(O)C1)=O)OC c1(CCC(=O)N(CCCNC(C(C)c2cccs2)=O)CCO)nc(C(C)(C)C)no1 c1(C(=O)NCC(C)CNC(=O)C(c2ccccc2Cl)(C)C)cccc(O)c1F N1(C(C(CC)COC)=O)CCN(C(C23CCOC(C)(C2)C3)=O)C(C(C)C)C1 CC1=NOC2(C1)CC(COC(=O)CSCc1ccc(F)c(F)c1)C2 C(CC(=O)NCCCCN(C)C(c1ccccc1CO)=O)(C(F)(F)F)OC CC(C)C(CNC(C1CCC(=O)N1C)=O)C(=O)N1CC(=O)NC(=O)C1 c1cccc2ccccc12.C1(NC(=O)OC(C)(C)C)CC2CC(C(=O)OCO)CC12 c1(CC)noc(C)c1C(=O)NC1CC(NC(C2(CC)CCOC2)=O)C1 C1(C(N2CC(O)(CN(C(CCCOC)=O)C)C2)=O)CCC=CCC1 Cc1nc2c(cc1C(=O)NC(C)C(C)NC(=O)C1CC1)c(C)nn2C C(=O)(C1=CCC(NC(c2cnccn2)=O)C1)NCC(C1CCCC1)C CCCC(O)CC(=O)NC1CC(NC(c2ccc(Cn3cc(C)cn3)cc2)=O)C1 c12cccc(n1)NC(=O)NC1CC(C1)NC2=O.C1(C(=O)OC)CCCSC1 c1(C(N2C(CCNC(C3C(C)(C)CO3)=O)CSCC2)=O)coc(S(N)(=O)=O)c1 C1(C(N2C(C#C)CC2)=O)CC2CC1CN(C(c1c[n+]([O-])c(C)cn1)=O)C2 CCC(C)(CNC(=O)CCCCCNC(c1c(F)cncc1F)=O)C(N)=O c1(C(=O)NCC=CCNC(c2cc(C(=O)OCC)on2)=O)scc(C)c1Cl C1(O)(C(N(CC(CC)NC(c2ccc(-c3ccccc3)o2)=O)C)=O)CCOCC1 C1(CNC(C2N(CC)CCCC2)=O)CC(C)(C)CN1C(c1ccc(CO)cc1)=O c1(C(=O)NCC2(F)CCCN(C(C(C)(C)OC)=O)C2)cccc2occc12 N1(CCc2c(C)cccc2)C(=O)CN(CCCCCc2ccc(F)cc2)C1=O N1(CC(C)(C)NC(C2(O)CC2(C)C)=O)CCN(C(C2CCCCC2O)=O)CC1 C1(NC(C(CC)OC)=O)CC2C1CCN2C(c1cc(F)ccc1O)=O N1(C(c2ccc(N(C)C)cn2)=O)CCN(C(=O)C2=C(Cl)CCC2)C2CC12 c1(N(C)C)ccc(C2C(C(=O)NC3CCCC3NC(=O)CO)C2)cc1 C1(CCNC(CNC(CCC)=O)=O)CSCCN1C(c1ccncc1Cl)=O C1(CC(N2CC(N(C)C(c3cc(C4CC4)ns3)=O)C2)=O)CC2CCC1CC2 C1(NC(c2ccc(-c3cccs3)cc2)=O)CN(C(C2(O)CC2)=O)CCC1F C(=O)(CCCC(=O)NC(CNC(c1cccc(N)c1)=O)C(C)(C)C)N(CC)CC Cc1ncc(CC(N2CCC(C(C)NC(C3COC(C)(C)C3)=O)CC2)=O)c(O)n1 c1(OC)noc(C)c1C(=O)NCC#CC(=O)N1CCC(C(C)O)C1 C(=O)(CCC1CC1C(C)=O)N(CCCC)CC(=O)OCC.C1(=O)CO1 CC#CCCCC(=O)NC(C)CCCNC(C1(C#N)CC1(C)C)=O C(=O)(C(C)CCO)NCC1N(C(C2(C(=O)OCC)CC2)=O)CC1 c1(CCC(N2CC(O)(CNC(c3nnn(CC)c3C)=O)C2)=O)ccc(C)c(C)c1 C1(NC(CC2C(C)(C)C2)=O)CC2CC1CC2C(=O)NC1CCSC1 c1(OC)ncc(C(=O)O)cc1S(=O)(=O)NCC1CC(F)(CN)C1 C1(CN(C(=O)CC2CCCCC2)CC)CCN(C(c2[nH]c(C)nc2CC)=O)CC1 c1(C(N(CC(C)NC(CC2C(CC)C2)=O)CC)=O)cccc(Cl)c1OC(F)(F)F C1(C(=O)NCCCCOC)(NC(c2ccc(C)c(C)c2)=O)Cc2ccccc2C1 Cc1c(CNC(C2CC3CC3N2C(C2CCCCCC2)=O)=O)cccc1Br C1(NC(c2cc(O)nc(Cl)c2)=O)CCCC2CN(C(c3ccco3)=O)CC12 c1(C(=O)NCc2nc(CNC(c3cn[nH]c3)=O)nc(O)c2)cccc2c1COC2 N1(C(CC2(C)CCCC2)=O)CCC2(CCC2NC(c2cscc2Cl)=O)CC1 C(CNC(=O)C(N1CCC(O)CC1)C)(C(C)(C)C)NC(c1c(CSC)scc1)=O c1(C(=O)NCCN(C(c2[nH]c(C3CC3)nc2C)=O)CC)cc2nc(F)ccc2o1 C(=O)(C1=NOC2COCC12)NCC1CC(C)CN(C(C2(C(C)(F)F)CC2)=O)C1 C12(CNC(c3c(C)cc[nH]3)=O)CC(NC(C3CC4CCC3C4)=O)(C1)C(C)(C)O2 C1(C(=O)OCC2(NC(C)=O)CC2)CCCCC1C C(C)(C(=O)NC1CCC(C(=O)NCC(C)CN(C)C)C1)(C(C)C)OC N1(C(C(=O)NC(c2ccco2)C)=O)CCC2(CCC(=O)NC2)C1 C(=O)(C1=CC2CCCCCCC12)N(C1CCN(C(c2snnc2C)=O)CC1)CC c1(C(=O)NCCS(C)(=O)=O)cc2c(-c3cnn4c3CCCC4)cccc2s1 N#Cc1c[nH]c(CN(CCCC2CCCO2)C2CC2)c1 C1(N(C(=O)Cc2cnoc2)C)CCCN(C(=O)Cc2ccsc2Br)C1 N1(C(CC(CNC(CC2(C)CC2)=O)C2CCC2)=O)CCC(C2CCC2)C1 C(C(CC(C)C)C(=O)N1CC(C)(C#N)C1)NC(C1C(=C)C1C(=O)OC)=O c1(C2(C(N(CC(CN(C(=O)CSC(F)(F)F)C)O)C)=O)CCC2)ccccc1F Cc1cc(C=CC(=O)NCC2CC(NC(C3CCCC(C)(C)O3)=O)C2)c[nH]c1=N N1(C(c2cc(C)n(C)n2)=O)CCN(C(=O)CC2(O)CCCCC2)C(CC(N)=O)C1 c1(NC(C)=O)ccc(C)c(C(=O)NC23CC(C2)N(C(C2CCC(C#N)C2)=O)C3)c1 C1(CC(=O)NCC(CC(C)C)NC(CCOC)=O)CCCC2CCCCC12 N1(C(c2c(C)nc(C)n2O)=O)CCOC2(CCC(NC(C3CC3(Cl)Cl)=O)CC2)C1 O(N(CCO)C(=O)Nc1ccc(-c2ccnc(OC)c2)s1)CC N(C(=NC1CCS(=O)(=O)C1)NCC1(CN(C)C)CCCC1)C1CC(C#C)C1 c12cc(ccc1Cl)C(=O)N2.N1(CC)CCC(C(=O)O)C(F)C1 C1(NC2CN(C(c3ncc(C)nc3)=O)C2)CC2CN(C(=O)C(C)SC(F)(F)F)CC12 c1(OC)cc(C)ccc1C(=O)NCCCN(C)C(C1CC1Cl)=O CC1CN(C(c2ccc(Cl)cc2N)=O)CCC1CNC(c1cc2c[nH]nc2s1)=O C(=O)(CC(C)(C)CN(C)C)N(C1CCN(C(C23CC(C(C)C)(C2)C3)=O)C1)CCO N1(C(C(C2CCN(C(Cn3ccc(C)c3)=O)C2)F)=O)CCNC(=O)C1 Cc1c(C(=O)N(C)CC2CCN(C(=O)C=CC(C)C)C2)ccc2c1CCC2 c1(CNC(=NCCc2n(C)ncc2)NC2CCC2)ccc(S(C)=O)cc1 C#Cc1ccc(CC(=O)NC2C3CN(C(=O)CCOC4CCOCC4)CC23)cc1 c1(OC)ccccc1CN(c1cnn(C)c1)CC1COCC1CN c1(C(=O)NCCN(C(=O)COCC(F)F)CC)nccc(Cl)c1O N1(C(C2(COC)CC2)=O)CCN(Cc2cc(Cl)c(Cl)cc2F)CC12CC2 N1(C(CN(c2ccccc2)C(C)=O)=O)CCCC(CO)(NC(c2cccn2C)=O)C1 CC(C)(C)C(CCc1ccccc1)Nc1cc(O)nc(O)n1 c1(NC2CC(CNC(C(CC)C)=O)C2)ncc(Cl)c(O)n1 c1(N(CC(=O)NCCC)C)nc2cc[nH]c2c(=NC(CC)c2nccs2)[nH]1 Cn1nnc(C(=O)NC2CCCN(C(c3ccn(CC#N)n3)=O)C2)c1C(F)(F)F CC1ON=C(C(=O)N2CC(CNC(=O)CCc3c(F)cccc3F)C(C)C2)C1C Cc1nc2ccc(C(N3CCC3CNC(c3csc(C(C)(C)C)n3)=O)=O)cc2[nH]1 c1(OC)ncc(F)cc1C(=O)NCC(C1CCCCC1)NC(=O)C1=COCCO1 c1(C(N2CCC(C)C(NC(=O)Cc3cncnc3)C2)=O)noc2c(F)cccc12 C(=O)(C(Cc1cccc(Br)c1)CC(C)C)NCc1c(C)ncc(F)c1 C1(NC(=O)CC2CCCNC2=O)CN(C(=O)C(C2CCCCC2)F)CC1C1CC1 C#CCC(O)C(=O)NCCCCNC(=O)C(c1ccc(O)cc1)OC c1(C(C)NC)cn(CCCC(=O)NCCCCN2CCCC2=O)nn1 C1(CC(=O)NC)CCN(N2CCN(CCCC(C)(C)C)CC2)CC1 C1(CNC(CN(CC(=O)NC(C)C)C)=O)CCN(C(C2CCCOC2C)=O)CC1 c1(NC(N2C(C(=O)NC(C(=O)OCC)CC)CCC2)=O)cncnc1C CCC(C)CC(C)C(=O)NCc1ccccc1CNC(c1cnn[nH]1)=O c1(CC(N2CC3C(NC(C(C)C4CC4)=O)C(C3)C2)=O)cncc2ccccc12 c1(C(=O)NCC(c2cccs2)OC)nc(C(F)(F)F)ccc1F C(CC(C(=O)NC1(C(=O)NC(c2ncccc2C)C)CC(F)C1)OC)OC C1(CC(=O)NCC2C(CNC(C3(OC(C)=O)CC3)=O)C2)CSCCS1 N1(C(c2n(C)cc(C#N)c2)=O)CCC2C(C1)CN2C(=O)CC1CCCCC1(C)C CC(O)C(C(=O)N1CCC(N(C)C(C2CCCN2C)=O)CC1)N(C)C Cc1ccc(C(=O)NCCCCC(=O)NC2(C(C)C)CCC2)cc1 n1(CC(=O)NC2(CNC(=O)CCc3ccon3)CCCC2)cc2ccccc2n1 Cc1cc(CN2CCOC(CC(N3CCS(=O)(=O)CC3)=O)C2)c(F)cc1Br c1(NC(C)CC2CCCCN2C)cc(N2CCOC(CN(C)C)C2)ncn1 C12(CNC(c3occ(C)c3)=O)CCC(NC(=O)Cc3ccn(C)n3)(CC1)CO2 Cc1sc(N)c(C(N2CCC(C(C)NC(=O)CCOC(C)C)C2)=O)c1C c1(C(N2CCC(NC(c3cc(CCC)oc3C)=O)C2)=O)cccc2c1ncn2C C(N=c1[nH]c(=NCc2ccncc2)[nH]c2cccnc12)c1c(C)scc1 c1(C(N2CC(C)C(NC(=O)CN(C)C)CC2)=O)ccc2c(c1)C=CS2(=O)=O c1(C(=O)NC2CN(C(CC3CC(=C)C3)=O)C3C2C3)c(Br)ccc(F)c1OC c1(C(=O)NCC2OCCN(C(c3ccc(C)[nH]3)=O)C2)c([N+](=O)[O-])c(C)nn1C N1(C(C2CCCO2)COC)CC2C3CCC(C2C1)N(C(c1scnc1C1CC1)=O)C3 N#CC1(CC(N2CCSCC2CCNC(c2occc2F)=O)=O)CCCCC1 c1(-n2cc(CSCCN(C(C3CN4CCN3CC4)=O)CCl)nn2)cccc(Br)c1F N1(C(C2N(C(C3CN(C)C(=O)C3)=O)CC(F)(F)C2)=O)CCC(=C(F)F)CC1 c1(C(N2CCCC(NC(CCCCCC)=O)C2)=O)cc2c(=O)[nH]ccn2n1 N1(C(Cc2c(C)noc2C)=O)CC2CCOCC2(NC(c2coc(Cl)n2)=O)C1 CCC(CCO)C(C)NC(=O)NCCCCCCCCN1CCCC1 C(=O)(C1=NNC(=O)CC1)NC(C1CCCCN1C(C1CCC(=O)N1C)=O)C c1(CC(=O)NCC(CC)NC(=O)CCc2cnco2)cncc(Br)c1 n1(C(C)C(=O)Nc2ccc(OC(F)(F)C(F)F)nc2)cc2ccccc2n1 C(=O)(C1=C(Cl)CCC1)N(C(CNC(c1c(C)nn(CCO)c1)=O)C1CC1)C C1(CNC(C2(CC(=O)NC(C)Cc3ccco3)CCC2)=O)CN(C)CCN1C C1(C)(C(=O)NCC(C)NC(c2c(COC)cco2)=O)CCC(=O)N1 c1(C(=O)NC(CCOC)CNC(=O)CC(C)SC)cc2cccc(Cl)c2[nH]1 C1(NC(=O)Cn2nnc(=O)[nH]2)CCCCCC1NC(c1ccoc1C(F)(F)F)=O C1(NC(c2cc(OCC)no2)=O)CCN(C(=O)C(CO)N(C)C)CC(C)(C)C1 CC12CC(NC(=O)CC3CCCOC3)(C1)C1(CN(C(=O)C(F)(F)C(F)F)C1)O2 C(=O)(C1=NOC(C)C1C)N1CCN(CC(C)NC(Cc2c(C)ocn2)=O)CC1 N1(C(c2c(C)nco2)=O)CCN(C(c2ccncn2)=O)C(C2CCCC2)C1 c1(C(=O)NC2C(NC(C(C(CC)O)(C)C)=O)CCC2)ccnc2c1ncn2C N1(C(Cc2cnc(C)[nH]2)=O)CC2(CCCC2NC(=O)C=Cc2cncs2)C1 C1(C(N2CC(C)(C)C2)C(=O)NCC)CCC(C)(C)N(C=O)C1.C1(C(=O)OC)(C)CC1 C=CCCC(CCC=C)(c1nnnn1CCCF)NCc1cc(C(C)(C)C)no1 C(C(C(=O)NCC=CCl)NC(=O)C=CC(C)C)OC Cc1n[nH]c(C)c1CC(=O)NC1CCC(F)(CNC(=O)CCCc2ccsc2)C1 C(C)(C(=O)N=c1ccn(CCO)[nH]1)N(C(=O)C(C)CCCOC)CCC Cc1ccc(C(N2CCCCC2Cn2cc(-c3ccn(C)c(=O)c3)nn2)=O)c(C)c1Br C1(C(=O)NC2(CCNC(c3ccc(C4CC4)s3)=O)CCC2)CC2CCC1C2 n1(NC(c2cc(Sc3c(Cl)cccc3Cl)ccn2)=O)cnc2ccccc2c1=O N1(C(C(CC(C)C)C)=O)CCCC2CN(C(=O)Cn3ccnc3C(C)C)CCC12 C(C)(C(=O)N(CCC(=O)NCCOC(=N)O)C)SC N(C(=NCCCN1CCOCC1)NCC(C(C)C(C)C)NC(N)=O)c1cc(C)sc1 N1(C(CCC)=O)CCCN(C(c2cccs2)=O)C(Cc2cccc(C(N)=O)c2)C1 CC(C)CC(=O)C(=O)NCC1(NC(=O)CC2(O)CCCC2)CC1 c1(OC)cc(C(=O)NC2CCN(C(C3C=CCC3)=O)C2C)sc1Br c1(OC)ccc(C(F)F)cc1C(N1CCCC(F)(C(=O)N(C)C)C1)=O N1(CC)CCC(C(=O)N(CCCOCCNC(C=CC)=O)C)C1 C=CC1CN(C(=O)C(CC(F)F)NC(c2cncnc2)=O)CC1O Cc1[nH]c(=N)sc1C(=O)NC1(CNC(C2C3CC3C3CC23)=O)CC1 CC1(C)C(=O)CC1C(=O)NCC(N1CCC(N2CCCC2=O)C1)=O CC(C)C1=CCC(C)(C(N2CC(c3cn(CCCO)nn3)C(O)C2)=O)CC1 Cc1sc(C)c(C(N2CC(NC(c3nocc3C(C)C)=O)C(C)C2)=O)c1C#N C1(C(N(CC)Cc2ccccc2)=O)CCC(NC(C2(COC(C)=O)CC2)=O)CC1 C=C(C)C(CC(=O)N(CCCOCC(N1CC(OCC)C1)=O)CCC)OC c1(C(N2CC(CC)N(Cc3ccc(OC)cc3C)CC2)=O)ccc2ccoc2c1 c1(CC)nc2c(C)csc2c(=NC2CCC(NC(c3cc(OC)ns3)=O)CC2)[nH]1 CC#CCC(C(=O)NCCCC(O)CO)NC(=O)C(F)F N1(C(C2=NNC(=O)C2)=O)CC2CN(C(c3cccc(CO)c3)=O)CCC2(CO)C1 Cc1[nH]nc2c1CCC(NC(C1CCNCC1(C)C)=O)C2 c1(C(N2CCCC(CCNC(CC(=O)NCC#C)=O)C2)=O)ccc(NC)c(F)c1 C(=O)(CC(O)C(Cl)(Cl)Cl)N1CC(O)(CNC(c2sccc2C2CC2)=O)C1 CCCCC(O)CC(=O)N1CCCC(C)(C)C1CNC(=O)CC12CCC(CC1)C2 CC1CN(C(c2ccc(Cn3cc(COC4CC4)nn3)o2)=O)CC1N(C)C CC(CC(=O)NC1CC2C1CCN2C(c1cc2ccccn2c1)=O)P(C)(C)=O c1(C(C)NC(c2ccc(C(N)=O)[nH]2)=O)nocc1C(=O)NC1CC1F C1(C2CCOCC2)(C(N2C(CCN3C(=O)CCCC3)CCCC2)=O)CC1 C1(NC(c2cnnc(O)c2)=O)CCN(Cc2ccc(Br)[nH]2)CC1F C1(NC(c2ccc(CCC)s2)=O)CCCC(NC(=O)C=C(C)C)C1 C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(c2cc(C3CCC3)on2)=O)CCC1 C1(NC(c2ccc(SC)cc2Cl)=O)CC2CC(C1)N(C(=O)CCCS(C)(=O)=O)C2 c1(C(=O)NC2CC(NC(c3c(C)n[nH]c3)=O)C2)cc2c(Cl)cncc2s1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)N1C2CN(C(C3CCC(C)O3)=O)CC21 C(C1c2ccsc2CCN1C(c1ccon1)=O)NC(c1ccc(OC)cc1)=O O=C1CC(CC(=O)NC2CN(C(C3CC34CCC4)=O)C3CCCC23)=NN1 CC(C)CN=c1[nH]c(=NC(C)c2ccccc2C#N)c2c(Cl)cccc2[nH]1 C(=O)(C1Cc2ccccc21)NC(C1N(C(c2c(C)cc(N)c(C)n2)=O)CCC1)C C=CCC(CNC(C1CC1C(C)(F)F)=O)NC(=O)C(C)=C(C)C C(CCC(C)C(=O)NC1CN(C(c2ccc(Br)nc2O)=O)CC1O)OC c1(C(=O)NC(C(C)NC(C(C)=C2CCC2)=O)CO)cc2c(nc1O)CCCCC2 C1(CNC(=O)C=Cc2ncc[nH]2)(CO)CCCN(C(C2CCCC23CCC3)=O)C1 CC1(C)CCCC(C(=O)NCC(C2CCCN2C(=O)CCS(N)(=O)=O)(C)C)O1 Cc1cc(CN(C2CCC2)C(C23CC(n4cc(CSC5CC5)nn4)C2C3)=O)n[nH]1 N1(CC(N2C(CCNC(c3c(C)nc(C)s3)=O)CCC2)=O)CCn2ccnc2C1 C=CCC(C(=O)NCC(=C)CCNC(c1c[nH]cc1C1CC1)=O)OC N1(C(CS(N)(=O)=O)=O)CC2CCCC(C1)N2C(C1CC1COc1ccccc1)=O C(CC(C)C(=O)NC(CNC(c1cccc(C(=O)OC)c1)=O)C1CC1)OC C(CC(N)=O)(C(=O)N1CC(NC)C1)NC(C=CC(=O)OCC)=O Cc1c[nH]c2ncc(C(=O)NCC3(C)CCCN3C(=O)CCC(C)C)cc12 c1(OC)cc(C)c(CO)c(C)c1.C12CC(F)CN1C(=O)c1cncc(c1)NC2=O c1(C(=O)NCC2CN(C(c3ccn(C)n3)=O)C(C)(C)C2)ccc2c[nH]nc2n1 N1(CCc2nnc(C)s2)CCC2(NC(=O)CCC3CCCN3C)CCCC12 CC(CC(=O)N1CCC(C(=O)NCc2ccccc2Cl)C(C)(C)C1)C(F)(F)F Cc1noc(C(c2ccccc2)S(=O)Cc2ccn(C3CCNC3)n2)n1 C(=O)(C(O)CC(C)(C)C)NCC1CC(F)(CNC(C(C)NC(CC)=O)=O)C1 Cc1c(C(=O)NC2CCc3nn(CCO)cc3C2)[nH]c2cc(Cl)ccc12 C1(C(N2C(C)CC(NC(c3ncncc3Cl)=O)C2)=O)(CF)CC2(CCC2)C1 CC(C(=O)NNC(=O)c1ccccc1)Sc1cn(CN2CCCC(O)C2)nn1 C1(CCNC(C(C)SCC)=O)CC(F)(F)CN1C(=O)CCC(F)F C1(NC(C2CCCN2C(=O)CCOCCCOC2CC2)=O)CC2CCC(C1)S2(=O)=O Cc1[nH][nH]c2ncnc(=NCCC(C)(C)NC(c3ccc(CN(C)C)[nH]3)=O)c1-2 CCCC(C(=O)OC)C(=O)NCC1(F)CC(NC(C2CCCCC2O)=O)C1 Cc1cc(C)c(C(=O)NCCC2CN(C(c3nocc3C3CC3)=O)CCO2)s1 N1(C(COCC(=C)C)=O)CC=C(CNC(C2CCCCC2F)=O)CC1 N1(C(c2ccn(CCF)n2)=O)CCC2CCN(C(=O)COC3CCOC3)C2C1 c1(-n2cc(C3(NC(=O)C(Br)Br)CC(F)C3)nn2)ccccc1F C12(NC(=O)NCCCn3cc(-c4ccccc4)nn3)CC(OC3CCC3)C1C2 C(=O)(C1CCc2nccn21)N1CCC(C(=O)NC2CC(C)(C)OC2=O)(CF)C1 CC1C(NC(=O)C(C)(C)C(F)F)CC2CCC1N2C(=O)CCN1CCCC1=O C(=O)(CC(C)CN=c1[nH]c(N(C)Cc2cc(OC)ccc2Cl)nc(=N)[nH]1)NC C(=O)(CC(C)C(C)(C)C)N1CC(N(C(c2ccc(CC)cc2F)=O)C)C1 Cc1ccc(C(=O)NCc2nc(CNC(=O)CCC3CC3C)cc(O)n2)c(Cl)c1 CC(C)C(O)CC(=O)N1CCN(C(=O)Cc2cncc(F)c2)CC1C(C)C C(=O)(CCCn1cc(CCC(=O)O)nn1)N1CC(CSC)C1 C12(CNC(C3(C)CN(C(c4cc(C)n(C)n4)=O)C3)=O)CCC(C1)C(=O)N2 C1(CCC(=O)N(CC(C)NC(c2oncc2C)=O)CC)CCCN1C CC(C)CC(CO)N(C(=O)CCN(C(=O)C(C)n1cncn1)CCCO)C N1(C(c2ccc(C(C)=O)o2)=O)CCN(C(=O)C(C)(C)CC(F)F)CC(O)C1 C1(NC(C2CC=CC2)=O)CCN(C(=O)CC2CC3C=CC2CC3)CC1CO C(=O)(C(C)(C)CC(=O)OC)NCC1N(C(c2c(CC)cno2)=O)CCCC1 CC(C)CCC(=O)Nc1ccccc1C1CCN(C(=O)OC(C)(C)C)CC1 c1(OC)ccc(S(=O)(=O)Oc2cc(Br)ccc2Cl)c(C)c1 C=Cn1nncc1C(N1CCCCC1CC(=O)NC(CCOC)C(C)C)=O CN1CCC(C(=O)NCC2CN(C(=O)CC3CCCC(=O)N3)CCN2C)CC1=O C1(CC(=O)NC2C(C(N3CC(OC(CC)=O)C3)=O)CCC2)CCC(C)(C)CC1 CC(C)C(C#N)C(=O)N(CCNC(C1CC12CCSCC2)=O)C1CC1 c1(OC)ccc(C(=O)NC2CCC2NC(=O)Cn2cnnc2O)c2c1CCCC2 c1(C(=O)Oc2ccccc2C)cc2sccc2[nH]1.CCC(CN(C(=O)CSC)C)N C1(NC(CC=C(CC)C)=O)CCN(C(=O)C(C)=C2CC2)CC1C C1(C2CC2)(NC(=O)Cc2ccccn2)CCN(C(C2CCC2c2nc[nH]n2)=O)C1 C1(C(N2C(C(=O)OC)CC2C)=O)CCC2CCC1N2C(c1cnns1)=O N1(C(CC(=O)NC)=O)CCCC(CCNC(c2ccnnc2Cl)=O)CC1 C(=O)(C(F)CCC(C)C)NC1CN(C(C(CCC)CC2CCCC2)=O)C1 CC(C)C(C)CCNC(C1OCCC1CNC(=O)C=Cc1cc[nH]c1)=O C(=O)(CC(C)CC(=O)OC)N(CCCCCC)CCNC(c1cn(CC)cn1)=O Cc1cc(C(=O)NC2CC(NC(c3[nH]nc(C(F)(F)F)c3C)=O)C2)cn(C)c1=O C(c1cc2cnn(C(C)C)c2[nH]c1=O)=CC(=O)NC(CC=C)CN c1(C(=O)NCCC(=C)CNC(C2CCC(C)(CC)O2)=O)c(F)ccc(C#N)c1F N1(C(c2c(C(C)C)n[nH]c2)=O)CC2(C(=O)NCCC3(O)CCOC3)CC1CO2 Cc1cnn(C)c1C(=O)NC(C1CCCCC1)CNC(c1ccc(Cl)cc1)=O N1(CC(O)CC2CCOCC2)CC2CC3CC2C1C3CO c1(SCC(N2C(C(C)NC(C3C(C(C)C)C3)=O)CCC2)=O)cccc(F)c1 c1(C(N2CCC(C(C)NC(c3c(OC)nsc3)=O)C2)=O)ccc(F)c(CO)c1 C1(CC#C)CCN(C(=O)C(C)N(C(=O)CNc2ccccn2)C)C1 Cc1ccc(C(N2CCCC2C2OCCC2NC(C2CCOC(C)C2)=O)=O)nn1 C1(O)(C(N2C3CC(NC(c4c(F)ncc(OC)c4)=O)(C3)C2)=O)CN2CCC1CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CC(C(=O)N(C)CCn2ccnc2C)C(C)(C)C1 C(CC(CNC(c1cc(-c2ccco2)on1)=O)NC(C1(OC)CCC1)=O)OC C1(CNC(CCCC(N)=O)=O)CN(C(c2ccc(Cl)nc2O)=O)CC12CCC2 C(C)(C(C)C(=O)N1CCCC1)NC(CC(=O)OC)=O.C1CC(=O)N1 c1(C(=O)N(CCO)C2CC2)ncccc1NCc1ccc(Br)[nH]1 C1(C)(C(=O)NC2CN(CC)C2)CC(NC(=O)CCCNC(N)=O)C1 Cc1c(NC2CC2)ncnc1N1CCC(C(=O)NCCC2CC2)C1.c1ccc(CO)cc1 C12(CNC(c3n[nH]c(C)c3F)=O)CCC1CN(C(c1ccnn1C(C)(C)C)=O)C2 n1(Cc2n(CC)ncn2)ccc(C)cc1=NC1CCCC1 N1(C(c2cc(C)c(C)[nH]2)=O)CCN(C(=O)CCN2CCN(C(C)C)CC2)C2CC12 C12(C(N(CCCF)CC)=O)CCN(C(c3nonc3C)=O)CCC1C2 C1(CC(N2CC3OCCN(C(=O)C(Cl)=CCl)C3C2)=O)CC2(CCCC2)CO1 C1(NC(c2ccc(OC)nc2C)=O)CCC2(CCN(C(=O)CCNC(N)=O)CC2)C1 C(=O)(C1CCCn2nccc21)NC1CCC(C)N(C(=O)Cc2cccn2C)C1 CCC(CC(=O)NCC1CC(CF)C1)NC(=O)C(CC)N(CC)CC Cn1nc(SCC(=O)NCC2CN(C(C3CC3F)=O)CC2(C)C)c(=O)n(C)c1=O N1(C(C=C(COC)C)=O)CC2CC(NC(c3ncc(C)cc3Br)=O)C1C2 N1(C(CCC(=O)NC)=O)CCC(C2(O)CC(NC(C3CC3C(N)=O)=O)C2)CC1 C1(CC)CN(C(=O)C(=O)Nc2ccccc2)CCN1Cc1sc(OC)nc1Cl C1(C)(NC(c2cncc(NC)c2)=O)CCCCC1NC(=O)COC(C)(C)CC N1(C(C2OCC(C)C2)=O)CCN(C)C(C(N2CCC(CCO)C2)=O)C1 N1(C(C(CC2CCC2)NC(CCNC(=O)NC)=O)=O)CC2CCC1C(O)C2O CC1(C)NC(=O)CC1C(=O)NC1CCC(NC(c2cccc(C3CC3)c2)=O)CC1 N1(C(C2N(C(C)=O)CCOC2)=O)CC2CCC1CN2C(=O)CC(C)(C)C1CC1 C1(NC(CC2(CSC)CC2)=O)CN(C(c2cccc(=O)o2)=O)CC1(C)C C1(C(N2CCC(C(N3CC(F)(COC)C3)=O)CC2)=O)CC2CCCC2C1 Cc1cc(Cl)c(Cl)cc1C(N1CC2(C1)CN(C(=O)C(C)C1CCCO1)C2)=O N1(C(c2cccc(NC)c2)=O)CCC(CNC(C2CCCC2OC)=O)C12CC2 c1(CCC)ncc(NC(C2CC(NC(=O)CN3CC(=O)NC3=O)C2(C)C)=O)cn1 N1(C(CCCOCC)=O)CCC2(CCOCC2)C(NC(c2cn(C)nc2C)=O)C1 C1(C(=O)NC(C2(O)CN(C(C(C=C)O)=O)C2)C)CCCN(CC(F)(F)F)C1 c1(CC)cnc(O)c([N+](=O)[O-])c1.C12CN(CC1O)Cc1ncn(n1)CC2 CC1CC(C(=O)NC(C)CC(C)NC(=O)CCc2cnc(C3CC3)o2)CC(C)C1 CC1CC(C(=O)NC23CC(C2)N(C(c2cncc(F)c2)=O)C3)CCC1=O Fc1cccc2c1OCCC2Nc1cccc2c1OCCC2 C(CCCCCC(=O)O)N1CCC1=O.C=CCNC(=O)OCC Cc1c(C(=O)NC2CCC2CNC(C2(S(N)(=O)=O)CC2)=O)cnn1C C1(C(=O)NC(CCC)CO)(OC)CCN(C(c2cc(C3CC3)on2)=O)C1 C(=O)(C(F)C(C)CNC(=O)Cc1cc[nH]n1)N(CCF)CC C1(C(=O)NCCC2(OC)CN(C(=O)CCSc3n[nH]c(C)n3)C2)CC(=O)NC1=O C1(COC)CC(CNC(c2cc(O)cs2)=O)N(C(C2CNC(=O)N2)=O)C1 C(=O)(C(CCOC)NC(=O)Cc1ccoc1C)N1CC(N(CCOC)C)C1 CCCC(C(O)C(=O)NCC1(CC(C)C)CC1)NC(=O)CCC1CCOC1 CC(C)(C)CC(=O)N1CCC(C(C)(C)NC(C2(CO)CCCCO2)=O)C1 C1(C(N(CCC(F)(F)F)C)=O)CC12CCN(Cc1cc3ccccc3[nH]1)CC2 CCCCCC(O)CC(=O)OC.C1=CCOc2c1cc(Cl)cc2 C#CC1(C(=O)NC2(COC)CCCC2)CN(C(=O)C(CCC)N(C)C)C1 C(=O)(C1=CCCSC1)NC(CC)CN(C(=O)CCC1CCCCO1)CC C(C(C)C(=O)Nn1cncn1)NC(C(CC#C)O)=O c1(C(N2CCC(N(C(CC(C=C)(C)C)=O)C)C(C)C2)=O)ccc2ncncc2c1 CC1CC(CCNC(C2(C)CS(=O)(=O)C2)=O)CCN1C(c1nnsc1N)=O N1(C(c2cn(CC)nc2)=O)CCC(C(C)(C)CNC(=O)C(C)(O)COC)CC1 c1(NCCCc2cccc(OC)c2)nc2c(cc1Br)CCC2O c1(C(N(CCCNC(C2CN3CCC2C3)=O)CC)=O)nccc2n[nH]cc12 N12CC3=C1NC(=N)SC3=NC(=O)C(OC)CCC(CC)C2 C(C(CC(=O)N1CC(CC=C(C)C)C1)NC(=O)C(C)C1CC(C)C1)OC C1(C(=O)NC2(CN(C(C(C)(CO)OC)=O)C)CC2)Cc2ccccc2O1 Cc1cc(C(=O)NCC2CCN(C(=O)C(C)Cc3ccco3)C2)c(N)c(F)c1 c1(C(N2CC(CNC(CCC)=O)OCC2)=O)ccc2c(c1)COB2O c1(C(=O)NC2CC3CC2N(C(=O)C=Cc2ccco2)C3)ccc(Cl)c(F)c1F C(C)(C)(CC(C)N1CCC(C(=O)N(C)Cc2ccnn2C(C)C)CC1)OCC C#CC1(C)CCN(C(=O)CC(C)C(C)(C)NC(=O)C(C)CC(F)F)CC1 c1(C(=O)OCC)cnc(NC(=O)C(=O)NC2CCCC2C#N)c(C)n1 c1(C(N2CC(NC(CSCCC)=O)C(O)C2)=O)c(O)nnc2c1CCC2 c1(C(=O)NCC2(CN(C(C3C(CC(C)C)C3)=O)C)CC2)nnc(S)n1C C1(NC(C2(CSC)CC2)=O)CC2CC(NC(C3CCCCC3)=O)CC12 C=CC(C)(O)CC(=O)NC1CC1CNC(n1nc(Cc2ccccc2)c(C)c1)=O N1(C(C2N(C(C)=O)CCC2)=O)C2CCC1CC(NC(C1(C)CCCCO1)=O)C2 CC1CN(C(C2CCCC3CC23)=O)CCN1C(=O)Cc1ccnc(F)c1 N1(C(c2cc(C(N)=O)[nH]n2)=O)CCCC(NC(C2CCS(=O)(=O)N2)=O)C1 CC(CC(=O)N1CCCC1CCC1CCCCN1C(C1CN(C)C1)=O)C(F)(F)F c1(CNCC2C(C(C)C)=C2)ccccc1CCCC(=O)On1cncn1 C1(C(N(C2CC(O)C2(C)C)C)=O)CCC(C(=O)O)N(C(=O)OC(C)(C)C)C1 C1(C(=O)NCC(CO)NC(c2c(N(C(C)=O)C)cccc2)=O)CN2CCCN1CC2 c1(CC)cccc(C(=O)N(CCCCNC(=O)COCC2CC2)C)c1O C1(CC(=O)N(C)CC2CC2(F)F)CC2(CC2)CN1C(=O)CC1=CCCC1 N1(C(C(C(CC)O)(C)C)=O)CCC2(C1)CN(C(=O)OC(C)(C)C)CCO2 N1(C(C(C(C)NC(C2(C)CCCN(C)C2)=O)C)=O)CCCC(C)(C#N)C1 C(C(=O)N(CCC(C)C)CCO)(C(C)(C)O)NC(c1c(CCC)nco1)=O C1(CC(=O)NCCN(C(=O)CCc2cnc(O)[nH]2)CC(C)O)CC2C=CC1CC2 C(=O)(C(F)(F)CN(C)C)N1CCC(N(C(CC2N(C(C)C)CCC2)=O)C)C1 C1(NC(c2c(OC)scc2)=O)COC2CN(C(c3cc(C)cc(C)n3)=O)CC12 C1(NC(c2c(CC)n[nH]c2)=O)CN(C(C2CC3CC2C2CC32)=O)C2CCCCC12 c1(-c2nc(COC(C3(c4ccccc4F)CC4(CC4)C3)=O)on2)ncc(F)cn1 CCC(CC(=O)NC(C1CCCN1C(c1cnccn1)=O)C)C(F)F N1(C(CC2CC(C)(C)OCC2)=O)CCC2CC1CN(C(c1ccon1)=O)C2 CCC(C(=O)N1CC(CNC(=O)C(C)(C)OC(C)C)C1)OC C1(C(=O)NC(CN(C(c2cc(C(=O)OC)sc2)=O)C)C)CC2(C1)CC21CC1 c1(C(N2CCC(C(N3CC(C)C(=O)CC3)=O)CC2)=O)cccc2c(O)nccc12 N1(C(C2C(C#C)C2)=O)CCCC2(C1)CN(C(c1scc(C)c1Cl)=O)CCO2 N1(C(C(CCCNC(C2CC2C2CC2)=O)O)=O)CCCC12CCOC2=O C1(C)(CNC(C2CN(S(CC)(=O)=O)C2)=O)CCCN(C(c2cnc(CO)s2)=O)C1 N1(C(=O)OC(C)(C)C)CC(C(=O)NCC2(CF)CCOCC2)CC12CCC2 CCC(O)C(C)C(=O)NC12CC(NC(c3cnc(-c4cccs4)s3)=O)(C1)C2 C1(CC)(NC(C2C3CCCOC23)=O)CCN(C(C2CCCC(C(N)=O)C2)=O)CC1 N1(C(C(CO)OC)=O)CCC2CN(C(=O)C(C)(C)OC)CC12 C1(C(=O)NCC2N(C(CCCN=[N+]=[N-])=O)CC(F)C2)CC(=O)C12CCCCC2 c1(C(=O)NC(CC)CNC(C2(C#N)CC(C)C2)=O)c(OC)ccc2ncccc12 c1(C(C(=O)NCC(C)CNC(=O)C(O)C2CCC2)=O)cccn1C C#CCC(CC(=O)NCC(=O)NCC(F)F)NC(c1ccc(CO)cc1)=O N1(C(C(=O)NCCNC(C)=O)=O)CCC2CC2(C(=O)N(C)C)CC1.C1CS1 c1(C(N2CC(CN(C(C(n3ccc(C(F)(F)F)n3)C)=O)C)C2)=O)ccnc(O)c1 Cc1nc(=N)[nH]c(C)c1C(N1CCC(CCNC(=O)Cc2ccc(F)cc2)C1)=O CC(C)(CCC(=O)NCC1CC1CO)NC(=O)CN1CCCC1 c1(OC)c(O)cc(CN2CCC(O)(C(=O)Nc3c(Br)ccnc3C#N)C2)cc1O C1(CN(C=O)Cc2cccc(C(F)(F)F)c2Cl)CCCC2(CCC2)O1 C1(NC(C2CCN(C(C)C)CC2)=O)CC12CCN(C(=O)CSCC(F)F)C2 c1([SH](CC(N2CCN(CC)CC2C2CCC2)=O)C)cc(Cl)c(NC2CCC2)cc1C C1(N(C(=O)CNC(c2cn(C)nc2C(F)F)=O)C)CCCN(C(c2nc[nH]n2)=O)C1 CC1CC(NC(c2cc3c(s2)CCC3)=O)CCN1C(=O)CCc1cncnc1 c1(C(C)NC(C(=O)NCc2cn(CC(C)C)nc2)=O)csc2ccccc12 c1(NC(=O)Cc2nc(-c3ccccc3)co2)cccc(-c2cn[nH]c2)c1Cl N1(C(Cc2cc(C)on2)=O)CC(CNC(c2cccc(O)c2F)=O)CC12CCC2 C1(CC(=O)NC(C(C)C)CNC(C2C(C(C)(C)C)C2)=O)SC(=N)NC1=O c1(N(C)Cc2cnc(CC)s2)ncccc1S(=O)(=O)NC1CC1c1ccco1 c1(NC(C)=O)ccc(C(N2CCC(O)C(C)(CO)C2)=O)c2ccncc12 c1(C(CC(=O)NC2CCCC2NC(c2ccc(F)cc2)=O)O)cccc(F)c1 C1(NC(C(C)SC(C)C)=O)(CNC(c2cc(Br)no2)=O)CCOCC1 C1(NC(c2nc(CC)sc2)=O)CC2CCC1CN2C(=O)C(CC(C)C)N(C)C c1(CNC(=O)NCCN2CCCC(CC)C2)cc(O)nc(O)n1 C1(CC)CN(C(C2CC2CC)=O)CCN1.c1(NC=O)ccnc(OC)n1 C=CCCC(C)N=c1[nH]c(C)cc(=NCC(Br)=Cc2cccs2)[nH]1 c1(OC)nccc(C(N2CC(NC(c3nsnc3O)=O)CC(C)C2)=O)c1F N1(C(c2cnc(CC)s2)=O)C(C(=O)NCC23CCC(CC2)C3)CCC1C(C)C N1(C(Cn2ncc(C#C)c2)=O)CCC(CO)(CNC(C23CCCCC2C3)=O)CC1 N(C)(S(=O)(=O)N(C)C)CC(N1CCC(C(C)NC(C2CC23CCC3)=O)C1)=O N1(C(=O)Nc2cn(CC)nc2C)CCC2CCCCC12 C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCC(NC(C2(C(C)C)CCC2)=O)C1 c1(C(C(=O)NCCCCC2CN(C(C(C3CC3)OC)=O)C2)C)c(C)nn(C)c1C C1(C)(C(=O)NCC(CN(C(C(C)O)=O)C)C)CC2CCC1CC21OCCO1 c1(OC)ccc(S(=O)(=O)NCc2cc3sccc3s2)cn1 CCCCC(C(=O)N1CCC(C2CC2NC(=O)C=C(C)C)CC1)C(C)C c1(C(N2CCC(O)(C(N3CCOCC3CO)=O)CC2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC2CC(NC(C3(C#N)CCC3)=O)C2)cncc2nc[nH]c12 c1(C(N2CCCCC(NC(c3cc(C(N)=O)oc3)=O)C2)=O)cc(S(N)(=O)=O)cs1 CC(c1ccccc1Cl)=CC(=O)NCC1CCC2(CN(C(=O)CO)C2)O1 C1(CC)CN(C(=O)CCCC(F)F)CCN1C(c1ccc(Cl)c(F)c1)=O C(CNC(c1cccn1CC)=O)(C(C)C(C)C)NC(c1c(CC)onc1)=O C1(OC)CN(C(=O)C=CSC)CC1NC(=O)C(C)Sc1cccc(C)c1 N1(C(C=Cc2nc(C)oc2C)=O)CC2CCN(C(=O)CN3CCOCC3)CC12 c1(CC(=O)NC2C(CNC(CSC)=O)C2)cccc(S(C)(=O)=O)c1 N1(C(Cn2c(=N)nc[nH]2)=O)CCC2CN(C(=O)Cc3ccnc(Br)c3)CCC12 CCC(CN(C)C)CC(=O)N(CCNC(C1CC1(F)F)=O)CCc1ccccc1 C1(CN(C(c2cc(C(N)=O)cn2C)=O)CC)CCCN(C(=O)C=CC2CCC2)C1 CC1CCCCC1(CNC(c1sccc1F)=O)NC(C1(n2ccnn2)CC1)=O N1(C(CC(OCC)OCC)=O)CCCC2(C1)CN(C(c1occc1Cl)=O)C2 C1(C(=O)NCCN(C(=O)C(F)n2cccn2)CC)CCCC12CCC2 N1(CC(=O)NCCN(CC#C)C(C)C)CCN(C(=O)COCCCC)CC1 c1(C(C(=O)NC2C(SC)CN(C(=O)C(C)C(F)F)C2)(F)F)cccc([N+](=O)[O-])c1 C1(NC(Cc2ccn(C(C)C)n2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC2(CC2)C1 c1(OC)nccnc1C(C(=O)NC1CCCCC1)N(C1CCC1)CC1CC1 Cc1c(C(=O)NCC(CNC(C2(F)CCC2)=O)C(F)(F)F)oc2ccc(F)cc12 N1(C(C(C)OC)=O)CC2CCC2(NC(c2ncc(C)s2)=O)C1 Cc1cc(C(C)C)nc(=NCC2CC(CNC(c3cc(Cl)c(Cl)s3)=O)CO2)[nH]1 c1(C(=O)NC2CNCC(C)(C)C2)ccc2c(c1)NC(=O)C1CCCN21 C(=O)(C(CC)CC(C)C)N(C(C)C(N1CCC(O)CC1CC)=O)CCC c1(OCC)ccc(CCC(=O)N(CC(C)(C)NC(c2ccc(CC)[nH]2)=O)C)cc1 Cc1nn2cccnc2c1C(N1CC(NC(C2CC(F)(CO)C2)=O)C2(CC2)C1)=O N1(c2cc(NCc3ncc(C)nc3)nc(C)n2)CCc2cccnc2C1 c1(C(=O)NC23CCC(CC2)N(C(C2CCOC2)=O)C3)[nH]cc2c1CCCC2 c1(C(c2n(CCOC)nnn2)NC2COCC2F)cc(C)cc2c1CCC2 c1(CC)ccc(NC(C2CC(=O)CN2C(=O)C(CO)OC)=O)cc1O CC(CCC(=O)N1CC(O)(NC(=O)NC2CCCOC2)C1)N1CCNCC1 C1(C)(C(=O)NC(C)C=CC(=O)NC(CCO)C2CCC2)COC(=O)N1 CCC(CCC(=O)NC1(C(=O)NCCC2CCCC2)CCSC1)OC CCC(C)CCCC(=O)N1CCC(C(=O)NC(C)CSC(F)F)CC1(C)C C1(C(N2CC(C(C)NC(C3OCCO3)=O)C2)=O)(OC)CCSC1 CN1CCC(NC(c2n[nH]c3c2CN(C(C2CC=CC2)=O)C3)=O)C(C)(C)C1 c1(CC(N2CCCC(NC(CCC=C=C)=O)C2C)=O)c(C)cc(OC)cc1C C1(C(=O)NCCN(C(=O)CSc2nc[nH]n2)CCOC)CS(=O)(=O)CN1C(C)=O CC1CCC(O)(C(=O)NC(C)CC(C)NC(c2cn(C)c(=O)cn2)=O)CC1 C(=O)(CCCC(=O)NC1(C)CCCN(C(C2CC23CC3)=O)C1)N(CC)CC Cn1c(Cl)cnc1CN(C(C1CC(F)C1)=O)CC1CCN(C(C)(C)C)C1 c1(CC)ccc(N)c(C(N2CCN(C(=O)C(CO)NC(N)=O)CC2C)=O)c1 N1(C(=O)NCc2c(OC)cc(Br)cc2)CC(CO)C2(CCOCC2)C1 Cn1cc(CC(=O)OCc2ccc(C3CC3)o2)nn1 c1(NC(=O)NC2CCC3CC23)cccc2nc(O)ccc12 c1(OC)cnc(C(=O)NC(C)C(C)(C)NC(C2C=CCN2C(=O)CCF)=O)cn1 C1(CNC(c2ccc(CC)cc2)=O)CC2(CCC2)CN1C(C1CC1F)=O C1(OCC)CC(CNC(c2c(-c3cccnc3)noc2C)=O)N(C)C1 c1(C(=O)NC2CCN(C(C3C(C)CCC3)=O)CC2)cc(C(F)F)cc(Cl)c1 N1(C(C2C(C)(COC)C2)=O)C2CCCC1CN(C(c1ccc(Cl)c(Cl)c1O)=O)C2 C(C(C)(C)C#CC(=O)N1CC(CC(C)C#N)C1)NC(c1c(CC)cccn1)=O c1(C(=O)NC2(CN(C(c3scc(OC)c3)=O)C)CC2)ccc(C)nc1 C#CCCCCCCC(=O)NC1CCCN(C(=O)C(C)C(C)COC)C1 Cc1cc(C(N2CC(NC(c3cnn(C)c3)=O)C3(CC3)C2)=O)cc([N+](=O)[O-])c1 C(=O)(C(CC(C)C)ONC(=O)C(C)SCCCC)NC1CC(OCC=C)C1 Cc1cc(C)c(CC(N2CC(N(C(=O)C=CCCC(C)C)C)C(F)C2)=O)c(C)c1 C1(O)(C(C)NC(C(CC)NC(C)=O)=O)CCN(C(C2(c3cc(C)no3)CC2)=O)C1 N1(C(c2cn(CCC)nn2)=O)CCCC12CCC(NC(=O)CC1CCSC1)CC2 c1(CNC(N2CCC(CN(C)C)(CF)C2)=O)nc(=N)[nH]c(=N)[nH]1 C=CCC(CNC(=O)C=C(C)C(F)F)C(=O)NC(C)CN1CCCC1 C12(CCC(=O)OCc3ncoc3SCC(=O)Nc3c(C)snn3)CCC(CC1)C2 C1(C(C)=O)CCCCC1(C)NC(=O)CCCn1cc(CCC2CCCCO2)nn1 c1(C(=O)NC(CCOC)CO)coc2c1CN(C(=O)CCc1cnco1)C2 C1(C(=O)NC)CCCN(C(C2C=CC(NC(=O)COCCCF)C2)=O)C1C N1(C(c2ccc(C(C)C)o2)=O)CC2CN(C(=O)C(C)(C)N3CCCC3)CCC12 c1(C(N(C2CCN(C(=O)C(C)(C)O)C2)C)=O)nc(C2CC2)n2ccccc12 C1(O)(CC(=O)N(C2CCN(C(=O)Nc3cc(C#N)c[nH]3)C2)CCC)CCCCC1 N1(C(C(C)(C2(C)CC2)OC)=O)CC(CNC(c2cn(C3CCC3)nn2)=O)C(O)C1 c1(C(=O)NCCCCC(CO)NC(CC(C(C)C)C)=O)ncc2ccccn12 c1(C(=O)NC(CC)CNC(=O)CC2CCCN2CC)c(C)cccc1[N+](=O)[O-] N(C(=NCCc1ccncc1)N1CCS(=O)(=O)C(C)(C)C1)CC(=C)C C1(CNC(c2n(CC=C)nnn2)c2cc[nH]n2)CCOC(C)(C)C1 N1(C(C2C(CCC)CCC2)=O)CCC2CCN(C(c3ccc(F)cc3C)=O)C2C1 c1(C(c2nnnn2C)NCc2c(C)n[nH]c2C)cnc(O)c2ccccc12 C(=O)(CC=C(Cl)Cl)NCC(N1CCN(C(=O)CCC2CCCOC2)CC1)C c1(C(N2CC(CNC(C(CC)N(C)C)=O)CC2(C)C)=O)cc(C#N)c(F)cc1F C1(C(=O)NCC(C)N(C)C(c2cccnc2)=O)C2CCC1(c1ccc(F)cc1)C2 Cc1ccnc(C(N2CCC(NC(=O)CC3CC3(C)C)C2)=O)c1Br CC(C)CC(C)(O)C(=O)NCc1ccc(C(=O)NC2CC(C)CC(C)(C)C2)nc1 N1(C(CC=CC=C)=O)CCN(C(c2cnc[nH]2)=O)C(CC#N)C1 c1(NC(=O)CC2CNCCN2)cc(Cl)cc2c1CCC2 Cc1ncc(F)c(NC2CC3CN(C(C4(C)CNC(=O)C4)=O)CC23)n1 n1(CC(N2CCN(C(C(CC)SC)=O)CC2)=O)cc(Br)ccc1=O N1(C(CCCC(C)=O)=O)CC(C(=O)NCc2ncnn2C)C2(CCC2)C1 N1(C(CCc2c(C)noc2C)=O)C2CC1CN(Cc1ccc(CO)cc1)C2 n1(CC)cc(Cl)c(C(=O)NCC(C)(C)OCCNC(C2C=CCCC2)=O)n1 C(CN=C(NC1CC1)NC1CC(=O)N(C2CC2)C1)(C1CCC1)OC c1(C(N2CC(C)(c3cn(C4CC(O)C4)nn3)C2)=O)ccc(F)cc1 C(=O)(CN=c1cc[nH]cc1)NC1CCC(NC(=O)CC(C2CC2)C2CC2)CC1 c1(CCNC(C(C2CN(C(C3COC(=O)N3C)=O)C2)OC)=O)ncccc1C N1(C(C(CC#CC)NC(=O)CCC2CC=CCC2)=O)CCOC(C)(C)C1C C(=O)(CC(C)CC(=O)NCC(C(C)(C)C)NC(c1cnccc1OC)=O)OC C1(C(=O)NC2(COC)CN(C(CN3CC(C)C3)=O)C2)CCCSC1C c12cccc(c1)S(=O)(=O)N1CC3C(C3C1)NC2=O.N1(CC=C)CCc2[nH]ccc2C1 Cc1nc2cnn(C)c2cc1C(N1CC(n2cc(CNC(=O)C=CCO)nn2)C1)=O CCC(C(=O)N(C)Cc1cccc(C(F)(F)F)c1)C(C)O.C1(=O)CCOCCN1 c1(C(=O)NC(CC=C)CNC(C2CCOC2)=O)ccc2[nH]c(=O)cnc2c1 c1(OC)ccc(CC(=O)NC(C2CCN(C(c3ccc(C)s3)=O)C2)C)cc1F C#Cc1ccccc1CC(=O)N(CC(C)(C)NC(C1SC2C=CC1CC2)=O)C N1(C(CC2C(C)CCC2)=O)CC2CCCC(N(C(=O)C3=COCC3)C)C2C1 c1(C(N2CC(NC(Cc3c(C)noc3Cl)=O)C3C2C3)=O)cccc(F)c1F c1(OC)nc(N2CCCC2CCc2cnn(C)c2)c(Cl)cc1Cl C(=O)(C(CN(C)C)NC(C1CNC(=O)C1)=O)NC(c1cnc[nH]1)C C1(C(N(C2CCN(C(C3(CF)CC3)=O)CC2)CC)=O)CCc2c[nH]nc2C1 C1(C(=O)NC2C(CNC(C3CN(C)C3)=O)C2)COCC1(C)C N1(C(C2C3N(C(CN(CC)CC)=O)C(CC3)C2)=O)CCc2c(O)noc2C1 C1(NC(C#CC(C)C)=O)CCC2CC1CN2C(C1CC2(CCOC2)C1)=O C#CCC(O)C(=O)N1CCCC1(C)C(=O)NC(CC)C(=O)N(CC)CC c1(C(=O)NCC2C(NC(c3n(CC)ccc3)=O)CC2)cn2ccc(CO)cc2n1 Cc1nc(CC(=O)NCC(C2CC2)NC(c2sccc2C(C)C)=O)c(C)s1 C=CCC(CC=C)C(=O)N(CCCNC(=O)C(C)NC(=O)CC)CC N1(C(COCCCOC)=O)CC2CCC2(CNC(c2cccc(=S)n2O)=O)C1 C12(C(=O)NC(CC)CO)CCC(C(=O)NCc3cncs3)(CC1)CC2 C(CN=c1cc(NCC2CCN2C2CCCC2)nc[nH]1)c1cc(Br)ncc1 c1(C(N(CCn2cc(CCC3CCCC3)nn2)CC)=O)ccc(Cl)nc1Cl CCCCCC(CC)C(=O)N1CCC(C2(NC(c3csc(CCC)n3)=O)CC2)C1 C1(N(C(=O)CC2CC(C)(C)C2)C)CN(C(=O)CC2(N(C)C)CC2)CC1F C1(NC(c2cc(C)ncc2)=O)CC12CCN(C(c1cnc3n1CCCC3)=O)CC2 c1(SCC2(N(C(=O)NCc3ccccc3)CCCl)COC2)ccc2nn[nH]c2c1 c1(C(C(=O)NCCCOC)N(c2c(C)noc2C)CC)cc(F)c(F)c(F)c1 N1(C(CCCCCSC)=O)CCC2(CC1)CC2NC(=O)COC(=O)CO C1(CC(=O)NCC(c2nncn2C)C)C2CCCC2N1C(C1(Cl)CC1)=O N1(C(c2c(C)scc2)=O)CCN(C(C2OCCOC2(C)C)=O)C(CCO)C1 C=CCCC(C(=O)NCC(=O)NCC=C)NC(=O)C(N1CCOC1=O)C CC(C)(C)CC(C)(C)C(=O)NCC1CC1NC(=O)C(=O)C(C)(C)C c1(C(=O)NC2C(OC)CN(C(c3ccc(O)cc3F)=O)C2)cc([N+](=O)[O-])c(C)s1 c1(C(C)C(C)(C)CO)nc(C2Cc3ccccc32)nn1-c1ncnc(Cl)c1Br O=C(C1CCc2ccccc21)NCC1CN(C(c2ccn3c2CCCC3)=O)C1 c1(C(=O)OC(C)(C)C)ccc2c(c1)CCCC2NCC1COCC2(CCC2)OC1 O=C(NNCc1nccs1)c1ncon1 c1(C(N(C2CCN(C(=O)CCC3CCCO3)C2)CCC)=O)cn(C2CC2)nc1C N1(C(C2CCC(NC(CC3CC(N(C)CC)C3)=O)C2)=O)CCNC(=O)CC1C CC(C)CC(C(C)(C)C)NCC1(Cc2ccc(F)cc2)CCCC1 C(=O)(C(C)S(N)(=O)=O)NCC1(O)CC(C(=O)Nc2cccc(SC)c2)C1 C(CCCCC(=O)NC(CC1CC1)CC(=O)N(C)CCOc1ccccc1)SC c1(N(C(=O)OC)C)cccc(NC2(C)CCOC2)c1 Cn1cc(COC(C2CCc3c[nH]nc3C2)=O)c2ccccc12 c1(C(=O)NC(CCC)C(=O)NC2(C)CCCC2C)cnc2n1CCC2 c1(Nc2c(OC)cncc2)cc(OC)cc(C(=O)NCC(=O)NCCCSC)c1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC23CCCC2(C1)CN(C(=O)C1=CCCC1)C3 Cc1ccc2c(c1)CN(C(=O)CC1CCCN1C(c1cc[nH]c1)=O)CC2 CN(C)NC(=O)CCC(=O)NC1(C2CCCN(C(=O)CCOC3CCC3)C2)CC1 C1(NC(C2N(C)CCC2)=O)C2CN(C(c3cccc(NC(=O)C(C)(C)C)c3)=O)CC12 c1(C(=O)NCC2C(NC(C(=Cc3ccncc3)C)=O)C2)ccc2cnnn2c1 C#CCC(C)(C)CNC(C1CC(OC)CN1C(=O)CCC=C(C)C)=O Cc1ccc(C(=O)NC2CC(C)CN(C(=O)C(c3cn(C)nc3C)O)C2)cc1F N1(C(COCC=C)=O)CC(NC(c2ccc(-c3ccc(F)cc3)s2)=O)CC(O)C1 Cc1c(C(N2CC(NC(=O)C=C3CCC3)C3(CC3)C2)=O)cccc1CO C(=O)(CS(=O)(=O)N(C)C)NCC1C(NC(Cc2n(C)ncc2)=O)C1 N1(C(C(C)CO)=O)CCC2(C1)CN(C(=O)CCOC1CCOC1)C2 C1(C(=O)NC(c2nccs2)(C)C)C(C(F)F)C1(C)C C(=O)(CCC(C)(C)C#N)NC(COC(C)C)C(N1CCC(C2CC2)CC1)=O C1(C(=O)NCCC(C)N(C(c2cn(C(C)C)nn2)=O)C)CCN(CCO)C(=O)C1 N1(C(C2CCC2)=O)CC(C2CC2)(C(=O)NCCc2csnn2)C1 C(=O)(C(C)C(=O)NC1(CNC(c2ccc(OCC(C)C)cc2)=O)CC1)OC c1(C(N2CCC(CNC(C3CCCC(OC)C3)=O)C2C)=O)ccnc2[nH]ncc12 c1(N2CC3C(CO)(C3)C2)nc2c(c(=NCCOc3ccnc(Cl)c3)[nH]1)CCC2 O=C(C1Cc2ccccc21)NCC1COCCN1C(c1cc2ccsc2[nH]1)=O c1(COC)nc(OC)cc(N2CCC(C)(NC(c3c[nH]cc(F)c3=O)=O)C2)n1 C=C(C)C(O)CC(=O)NCc1ccc(CCNC(=O)CN(C)C)cc1 c1(C(N2C(CNC(c3c(C)nc4sccn43)=O)CC2)=O)c(Cl)nc2ccccn12 c1(C(=O)NCCCC(O)C(=O)NCC2CCCS2)ncn2ccccc12 c1(C(N2CC=C(CNC(C3C(CCC)C3)=O)CC2)=O)cc2c(F)c(C)ccc2[nH]1 C1(C(=O)OC)(CSCC(=O)NCCNC(C)(C)C)CC12CC2.C1(O)CN(C=O)C1 N1(C(CC2CC(C)C2)=O)CCN(C(c2ccnn2C(C)(C)C)=O)CC1CCO C(N=c1[nH]c(=NCC(CC)(CC)CCO)c2ccccc2[nH]1)c1n(CC)ccn1 C1(O)(CNC(c2c(C)sc(O)n2)=O)CCCN(C(c2cc(Cl)cc(Cl)n2)=O)C1 N1(C(C(CC(C)C)C)=O)CCC2CN(C(c3cccc4c3COC4)=O)CC2CC1 N1(C(C2CCN(C)C2)=O)CC(N(C)C(c2csc(-c3ccsc3)n2)=O)C(O)C1 c1(C(=O)NC2CCN(C(=O)CCc3cnn[nH]3)C2)cc(Cl)cc2ccncc12 C1(CCC2(N)CC(NC(=O)C3CC3)C2)CN(Cc2ccccc2)CC12CC2.COC N1(C(C2CCC(C(N)=O)O2)=O)CC2CC2(CNC(C2CC(F)(F)C2)=O)C1 CCC(C)(C)C(=O)NCC(C(=O)NC1CC=C(C)CC1)N(C)C C(=O)(C(C)CS(=O)(=O)c1ccc(OC)cc1)NC1(C)CN(C(CC(CC)C)=O)C1 c1(C(N2CC3CN(C(C4CC4F)=O)CC32)=O)cccc2ccnn12 c1(OC)cc(NC(=O)CC2CCN(CC3CC4CCC3O4)C2)cnn1 N1(C(CC(CCC)C)=O)CCC2CCN(C(=O)Cn3ncnn3)CC12 C1(C(N2C(C(=O)NCc3n[nH]c(C)n3)(COC)C=CC2)=O)CN(C)CCN1C N1(C(CCOC2CCN(C)CC2)=O)CC2CCCC(C1)N2C(=O)C=CC(C)(C)C C1(CNC(CS(CCC)(=O)=O)=O)CCC2CN(C(C3CCSCC3)=O)CCC2C1 C1(C(N2CCCC(NC(=O)C(c3cccnc3)O)C2)=O)(NC(N)=O)CCOCC1 c1(C(N2CC(COC)(NC(c3cnn(C)c3)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 N1(C(C2(CCNC(=O)CC3CCCC3)CCCC2)=O)CC(O)(C2CCC2)C1 CN1N=C(CC(=O)N2CCOCC(NC(C3(C4CC4)CCCO3)=O)C2)CC1=O C1(C(C)C)CC(C(=O)N(CCCN(C(=O)Cn2cncn2)C)C)CCO1 c1(C(=O)NCC(C)(CO)NC(C(C=CC)O)=O)ccc2c(c1)COC2 Cc1cc(C(F)(F)F)nc(N2CC3C(NC(c4ccc(F)cc4Cl)=O)C3C2)n1 Nc1c(Cl)cc(C(N2CCCC2CCNC(c2cc(C3CC3)[nH]n2)=O)=O)cc1Cl C1(C(=O)NCC(C2CCCC2)NC(c2csc(C)n2)=O)(CC)CCCC1O Cc1noc(C(C)NC(C2(N(C(=O)C(C)C#N)C)CC2)=O)n1 c1(C(N2CC(O)(CCNC(c3cc(F)ccc3F)=O)C2)=O)cc(F)c(O)c(F)c1 C1(CC(=O)NC(CN(C(=O)C(c2ccccc2)OC(C)C)CC)C)CCC(C)CC1 C(=O)(CC(O)CC(C)C)NC1(CCOC)CCN(C(=O)C(C)=C(C)C)C1 CCN=C(NCC1CC1OC)N1CCC(C(C)C)C1 c1(C(C(=O)N(C2CN(C(C3(C)CC(F)(F)C3)=O)C2)C)O)ccccc1Cl c1(N2CC(C)C(NC(c3cc(Cl)cn3C)=O)CC2)ncc2c(ncn2C)n1 CC1CC(C(=O)NC(C)(C)CNC(=O)COC2CCCCCC2)CC(C)C1 Cc1cc(Cl)c(Br)cc1C(N1CCCC(C(C)NC(=O)C#CC2CC2)C1)=O C#CCCCCC(=O)NC(CCCC)C(=O)NCCc1c(C)n[nH]c1C C(CCCCC(=O)N1C(C(=O)NOCC2CC2)CCC1C)SC c1(OCC(=O)NC(CCNC(CSC)=O)C)ccc2ccc(=O)oc2c1 C1(C(=O)NC(C)(CNC(C2(CS(N)(=O)=O)COC2)=O)C2CC2)SCCCS1 C(C1=NOC2CCCC12)NCC1CCS(=O)(=O)C1 C#CCC(C)C(=O)NCC1CCCCN1C(c1ccc(NC(C)C)cc1)=O c1(C(N2CC(C(C)NC(=O)C(C)(C)C3CC3)OCC2)=O)cc(N)c(F)cc1F C1(C(=O)NCC2CN(C(CC3CC(N(C)C)C3)=O)C2)CC2CCCCN2C1 C1(NC(c2cc(C)c(C)s2)=O)CCN(C(=O)C(C)(C)OC(C)C)CC1C CC1CCC(=CC(=O)NCCC2CCCN2C(=O)CC2(C)OCCO2)C1 C1(C(=O)NC(c2ccc(C#N)s2)C)CCCN(Cc2noc(C3CCCO3)n2)C1 C1(NC(C(C)OCC#C)=O)CCC(C)N(C(=O)Cn2cc(C(=O)OC)nn2)C1 c1(OC)ccc(CCC(=O)N2CC(CC(C)NC(=O)C3=CCCC3)C2)c(F)c1 C12(NC(CCC=C)=O)CCCC1CN(C(c1cccc(F)c1C)=O)C2 C12(CNC(c3cc(O)cs3)=O)CC1CN(C(C1CCO1)=O)C2 C1(C(N2CC(C)(NC(CCOC)=O)C2)=O)C2Cc3c(Br)cccc3C12 C1(NC(C(C(CC)O)C)=O)CC2(CCN(C(C3COC4(CCC4)CO3)=O)CC2)C1 Cc1cccn2cc(C(=O)NCC3CCC3NC(=O)C=CCn3cncn3)cc12 CCC(C(=O)N(C(C(=O)N(C1CCCC1(C)O)C)C1CC1)C)C(F)(F)F C(CC(C)C(C)(C)C)NC(C#C)CCCOc1ccccc1 C(=O)(C1=C(Cl)CCC1)NCc1oc(C(=O)NC(CSC)(C)C)c(C)n1 C1(NC(C2C(C3CN(C(C(C)N)=O)C3)C2)=O)CCC2(CC1)NC(=O)NC2=O C1(NC(C(CCC)NC(CC=C=C)=O)=O)CCOC12CCCC2 N1(C(c2c(N)ccc(Cl)n2)=O)CC2(CCCC2NC(=O)CC2COCCO2)C1 CC1CC(N=c2nc(N3CCCN(C)CC3)c3c([nH]2)COC3)CC(C)(C)C1 C12(CNC(c3n(CCC)ccc3)=O)CCC(C1)N(C(=O)Cc1sc(C)nc1C)C2 Cc1cc2nc(Cl)nc(N(CC(C)NC(=O)CN3CCOCC3)C)c2s1 C1(C(=O)Nc2c(C#N)ccnc2)CCC2(CN(C(c3scc(F)c3Cl)=O)C2)O1 C1(C(=O)NC(c2ccc(C)c(C)c2I)=O)CCC2(CC1)CN(c1ncccn1)C2 c1(C(=O)OC)ncnc(N2CCC(CF)(NC(=O)CC3CCCC3C)C2)c1OC C1(CNC(C2CCC(NC(CCC=CC(C)C)=O)C2)=O)CC2CCC2C1 C1(NC(=O)CCc2ccccc2)CCCCC1NC(C1(O)COC1)=O C1(C(N2CC(N(C(C(C)C#N)=O)C)C2)=O)CCC2(CCCO2)CC1 CC1(C)NC(=O)CC1C(N1CC(C(=O)NCCc2cc[nH]n2)C2(CC2)C1)=O C12(CC(=O)NC)CCCC(CN(C(=O)CNC(=O)C3CC3)C1)C2.NC(=O)C N1(C(CC2C(CC)C2)=O)CCC(F)(CNC(=O)C#CC(=O)N(C)C)C1 CCCC(C(=O)OC)C(=O)N(CCNC(c1cnccc1C(F)(F)F)=O)C1CC1 C(=O)(C(CC)(CC)CO)NC(CCCNC(c1ccc(COC)o1)=O)c1ccco1 c1(-c2ccc(C(C)O)cc2)cc(=O)n(C)c(O)n1 N1(C(c2cc(CC)oc2C)=O)CCCCCC1C(N1CCOC(C2CC2)C1)=O N1(C(c2c(COC)onc2)=O)CC2CC1CN2C(=O)Cc1cc(O)nc(O)n1 CCC(CCNC(C)CS(C)=O)OCC1CC1 Cc1ccc(C(=O)NC2CCC(N3CCN(C(=O)COC(F)F)CC3)C2)c(O)c1 C1(F)(C(N2CCC(CN(C(c3c(C)cno3)=O)C)C2)=O)CC=CCC1 c1(NC(C2CCN2c2ncc(-c3ccc(-c4nn[nH]n4)cc3)cn2)=O)cc(Br)cc([N+](=O)[O-])c1 C1(NC(Cn2ncc(C)cc2=O)=O)CC(C2CCN(C(=O)C=CC(F)(F)F)C2)C1 O=C(CC(F)(F)F)NC1CC12CC(NC(=O)CNC(=O)C1CC1)C2 c1(COC(C)C)ccc(Cl)c(NC(=O)CC2CCC(O)C2)c1 c1(OC)cnc(C(N2CCCCC2CNC(=O)CCCCSC)=O)c(F)c1 N(C(=NCCN1CCCOC1=O)NCC1CCOC1)CC1(COC)CCCC1 Cc1[nH]c(CN2CC(O)CC2C(N2CCC(Br)CC2)=O)c(C)c1C(=O)O CCCC(C(=O)NC12CC(CNC(c3cc(CC)no3)=O)(C1)C2)C(C)C C1(CNC(COC(C)C)=O)(NC(c2ncc(Br)cc2F)=O)CCCCCC1 C1(NC(=O)NC(COC)Cc2cccc(F)c2)COc2ccccc2C1O N1(C(C(CC)OC)=O)CCOCCC1C(=O)Nc1cnc(OC)cc1C C#CCCCCCC(C(=O)NCCCSCCOC)N1CCCC1 c1(SCCN(C(c2ccc(O)cn2)C)CC2CCCO2)cc(C)ccc1F CC(C)C(C)(CNC(C1CC1C(C)NC(C1(C)CCSCC1)=O)=O)C(C)C C1(CC(=O)NC2CN(C(C(C)OC(C)(C)C)=O)C2)CSc2ccccc2O1 c1(C(=O)NCC(CNC(c2scc(OC)c2)=O)OC)cc(SC)c(C)o1 C(=O)(CC(C)C1CCCO1)NCC1CC(NC(C(=O)NC)=O)C1 N1(C(C=C(C)C2CC2)=O)CCOC(CNC(=O)CN2CC(C)C2)C1 N1(C(CC(C(=O)OC)C)=O)CCCC(C2(NC(=O)C(F)C(C)C)CC2)C1 Cc1cn(CC(=O)N(CCCN(C)C(C2C3CC3C3CC23)=O)C)c(=O)nc1O Cc1sc(C(N2CCCCC(C)C2)C(=O)NCCC#N)c(C)c1C CCC(C)(C)C(C)CC(=O)N(C1CN(C(C2CC3C=CC2C32CC2)=O)CC1O)C c1(C(C)C)cc(C(=O)NC2CCN(CCF)C2)ns1.c12cn(nn1)CC(=O)NC2 C1(NC(C(C)CS(C)=O)=O)CCC2(CC1)CN(C(=O)CC(=O)OC(C)(C)C)C2 N1(C(C2(C)CCN(C)C2)=O)C2CCC1CC(NC(c1nnc(S)n1C)=O)C2 Cc1cc(N2CCC(C)(CO)CC2)nc(N(CC(C)(C)C(F)(F)F)C)n1 S(=O)(=O)(c1ccc(F)c(Br)c1)N1CC2(C(C(=O)NCc3ncn(C)c3)C2)C1 c1(C(=O)NCC2CCC(NC(Cc3c(C)noc3)=O)C2)ccc(N)c(O)c1 C(=O)(C1=COCCC1)NCc1occ(C(=O)NCCOC(CC)(C)C)c1 c1(C(N(C(c2ccccc2)CNC(N)=O)C)=O)cccc(CC#N)c1 C12(C(=O)Nc3c(CC)ccc(C)c3)CCCC1N(C(=O)C(C)O)CC2 C1(C)(C(N2CC(COC)(NC(C3COCCO3)=O)C2)=O)COCOC1 C1(CNC(C(CC)n2cncn2)=O)CCCN(C(=O)CCCn2cncn2)CC1 N1(C(C(OC)OC)=O)CCC(NC(C2CCCCN(C)C2=O)=O)C12CCC2 c1(C(N2CCC(O)(CNC(c3n(C)cnc3)=O)C2)=O)ccc2cnnc(O)c2c1 C#CC(C(C)(C)C)NC(C1CC12CC(NC(=O)CC(O)CC)C2)=O C1(C(=O)NCCCC(C)NC(=O)Cc2ccon2)CC1C1CCOCC1 C#Cc1cn(C)nc1C(=O)NCC1(C)CN(C(=O)Cn2cccn2)CCO1 Cc1nn(C)c(Cl)c1-c1cn(-c2cccc(CNC(C3(C)CC3(F)Cl)=O)c2)nn1 C(CC(C(=O)NC(Cc1cn[nH]c1)C(=O)O)NC(C)=O)SC CC1CCC(NC(C2CC(C)(F)C2)=O)CN1C(c1csc([N+](=O)[O-])c1)=O Cn1nc(-c2cnccc2C(N2CC3CCC2CO3)=O)c2ccccc12 C1(C)(C(=O)NCC(C)C(=O)Nc2ccccc2)CCCOC1 C1(NC(C(C)(C)n2cnnn2)=O)CC(F)(F)CC1NC(c1ncc(Cl)cc1F)=O S(=O)(=O)(c1ccc(NC2(CC)CCC(=O)N2)nc1)NC(CCCC)C C1(CC)CC(C(=O)Nc2csc(-c3ccc(Cl)s3)n2)CC(=O)N1 c1(C(=O)NC2(CF)CCN(c3c(C#N)c(Cl)ns3)C2)cc(Br)cc([N+](=O)[O-])c1 C12(C(N(CC)CC3(O)CCC3)=O)CC(CO)(CN1C(c1cc(C)c(CC)o1)=O)C2 Cc1coc(C)c1COCCN(C(C1CCC2CC12)=O)C(C)C c1(C(=O)NCC2C(C)CN(C(c3cccc(O)n3)=O)C2)cc(N)cc(N)c1 c1(C(=O)NC(CC)CNC(=O)C=C(C)C(F)F)ccc2c(c1)OC(C)(C)CS2 N1(C(C(CC=C)(C)N(C)C)=O)CCC2(CC1)CN(C(C1(C)CS(=O)(=O)C1)=O)C2 N1(C(C(C)(C)OC)=O)CCC(N2CCC(CC(=O)NCCN(C)C)CC2)CC1 c1(C(=O)NC(C2CCN(C(c3nccc(C)n3)=O)C2)C)cnn2cc[nH]c12 CCC(C(=O)NC1(C)CN(C(=O)COC(C)=O)C1)n1ccnc1.c1ccsn1 C(=O)(CCC(N)=O)N(C1CCN(C(c2ncn(C)n2)=O)C1)Cc1ccccc1 C(=O)(CCS(C)(=O)=O)N1C(C)(C(=O)NCCNS(N(C)C)(=O)=O)CC1 c1(CCCC(=O)N(CCNC(CC(C)c2cnn(C)c2)=O)C)ccc(CO)cc1 C1(C(NOC(C=C)C)=O)C2CC3C(C2NC(C2CC(=C)C2)=O)C13 N1(CC)CCCC(C(=O)NCC2(NC(=O)Cc3nc(C(C)(C)C)cs3)CC2)C1 C(N=c1[nH]c(C)ncc1C)c1c(C)nn(COCC)c1C c1(C(N2C3CN(C(CCCc4scc(C)n4)=O)CC2C3)=O)cccc2occc12 C1(CCCCNC(C2CC2C(C)O)=O)CCN(C(C2(C(=O)NC)CCC2)=O)CC1 c1(C(N2C(CC)CN(C(=O)C(C)N(C)C)CC2)=O)cc(=O)c2cc(F)ccc2o1 N1(C(C(C2(OC)CCCCC2)(F)F)=O)CC2CC(NC(=O)CC(C)C(C)C)C1C2 c1(C(N2CCC(NC(C3(CC)CCCCC3)=O)CC2)=O)nc(C)ccc1C C1(C(=O)NCCOCCC#C)C2CC2CN1C(C1CC1(Cl)Cl)=O C1(O)(CNC(C2C(=O)NCC2)=O)CCN(C(=O)COC(F)(F)C(F)(F)F)C1 c1(C(=O)NCCC(C)NC(=O)CN2CCC(C)C2)ccc(S(N)(=O)=O)cc1Cl C(=O)(CCS(C)=O)NCC(CNC(c1ccc(COC)s1)=O)O OC1Cc2ccccc2C1NCc1cnc(C(F)F)s1 CN1CCN(C(C2CCCN2C=O)=O)C(CNC(=O)Cn2nnc(C3CC3)n2)C1 CC1(C)OC2CC(C(N3CC4CN(C(C5CC5F)=O)CC4C3)=O)CC2O1 c1(C(=O)NC2CN(C(C(C)OCC)=O)CC2SC)cc(F)cc2ccccc12 CCCCC(O)CC(=O)NC1CCC(NC(c2ccc3[nH]ccc3n2)=O)C1 N1(C(C2C(OCC)C2)=O)CCC2(CCCN(C(c3cncc(SCC)n3)=O)C2)C1 c1(CNC(C(CCC#C)O)=O)nnc2n1CCN(C(=O)CC(C)CF)C2 C1(C(=O)NCCC2CCC(NC(C3(CN(C)C)CC3)=O)C2)(CC)CCCC1 N1(CC(=O)NCC(N(C(Cc2ccn(CC)n2)=O)C)C2CC2)CCC(C)CC1 Cn1ncc2c1CN(C(=O)CCC1CN(Cc3ccc(C(F)(F)F)cc3)C1)C2 C=C(C)CCC(=O)NCCOCCCCCNC(=O)Cc1cnoc1 C=CCC(C)(C)C(=O)N1CCC(NC(c2cc(C3CC3)no2)=O)C(F)C1 N1(C(CN(C(C)=O)C)=O)CCC(CCNC(c2c[nH]nc2C)=O)CC1C CONC(=O)C(=O)NC(CCNC(c1cnc(O)n1C)=O)C(C)C N1(C(c2cnc(CC)s2)=O)CCSCC1CCNC(C1CC(F)C1)=O CCCCCCCCC(F)C(=O)NC1CC2CC1N(C(=O)CNC(=O)CCC)C2 c1(C(=O)NCC2C(NC(c3cn(C(C)(C)C)nn3)=O)C2)c[nH]c2nccc-2c1 C1(C(N)=O)CN(c2nnnn2CC(c2ccccc2)C2CC2)CCO1 C(=O)(C1=NOC(C)C1C)NC1CC1NCCn1ccc(C(NOC(C)C)=O)n1 c1(CNc2c(C(=O)NCCc3ccc(O)cc3)n[nH]c2)cc(Cl)ccc1F C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(NC(C2(C)CC(=C)C2)=O)CC12CCC2 N1(C(CSCC=C)=O)CCN(C(c2csc(C(F)F)n2)=O)C(CCCC)C1 C(C(C)(C)C(=O)NCC(c1cnn(C)c1)C)NC(c1n(CC)ncc1)=O c1(C(N2CCN(CCCOC)CC2)C(=O)NCC)ccnc(P(C)(C)=O)c1 C12CCc3n[nH]cc3N1C(=O)ON(C)C2=O.N1(CCCN(CC(C)C)C)CCCC1 Cc1scc(NC(N2CCN(Cc3nc(C4CC4)no3)CC2)=O)c1N.OC C(C(O)CC(=O)NOC1CC1)NC(=O)CC1CCCOCC1 C(=O)(C(CCC)=CCC)NCCCN(CC(COCCC=C)O)C(C)C C1(NC(C(C=C)(C)C)=O)CCC2CN(C(c3ccncn3)=O)CCC2C1 C1(NC(CCCCC=C)=O)CN(C(c2cc(C)c(C)o2)=O)CC1C1CC1 c1(C(N(C(CNC(=O)C(c2cncn2C)O)C2CC2)C)=O)ccncc1F c1(-c2cn(CC(CC)O)nn2)cn(C)nc1CNC(C1CCCOCC1)=O C(=O)(C(O)CC(N)=O)N1CCC(C(=O)OC)CC1.c12cc([nH]n1)C1CN(C1)C2=O Cc1ccc(NC(C2CC3CC3N2C(c2nc(C(C)C)cs2)=O)=O)cc1Br N1(C(C(CC)(C)COC)=O)CC2CCC(CNC(=O)Cc3cnn(C)c3)C2C1 C1(n2cccn2)(C(=O)NCCCN(C(CSCCOC)=O)CCO)CCC1 N1(C(C(CC#C)C)=O)CC(NC(=O)CCc2ccccc2C)CC12CCC2 Cc1cc(S(N)(=O)=O)sc1C(=O)N(C1C2CN(C(=O)C#CC3CCC3)CC12)C Cc1cccc(C(n2nc(CCCN(C)C)nc2CC2CCCCC2)C)c1 N1(C(C(C2CC(C(=O)NC3CC=CCC3)C2)F)=O)CC(C2CCCC2)C1 c1(C(N(CC(CNC(CC(C)C2CC2)=O)O)C)=O)ccn2c1CSCC2 C1(NC(CSCCCC)=O)CC(F)(F)CC1NC(=O)C(C1CCCN(C)C1)(C)C C=CC(C)(CCOC)C(=O)NCC1(NC(=O)COCCOC)CCCCC1C c1(C(=O)OC)nn(C)cc1C(=O)NC(C)CNC(=O)C(O)CNC(C)=O.C(C)(C)(C)O c1(C(=O)NC(C2CCOCC2)C)cc(-c2ccc(F)cc2O)cc2c[nH]nc12 C1(C(N(C)CC)=O)CCC(F)(CNC(=O)C(C)(C)CN(C)C)CC1 C12(CNC(C(C)O)=O)CCC(CNC(c3occc3C(=O)O)=O)(C1)OC2 N1(C(C2CCC(n3cc(-c4n(CC)ncc4)nn3)C2)=O)CCSC(C)(C)C1 C1(C(=O)OC)CC(n2cc(C3(O)CC(C(=O)O)C3)nn2)CN1C(=O)CCC1CC1 C1(NC(CCOCC#C)=O)CCN(C(c2nc(C)oc2C)=O)CC1CO N1(C(CCC#C)=O)CCN(C)CC1CNC(=O)CO.c1(C)nc(CC)no1 N1(C(c2c(C(C)C)[nH]cc2)=O)CC2CCC(C1)C(NC(=O)CCC1CCCO1)C2 c1(CNC2CN(C(c3n(C(C)C)ncc3)=O)CC2C)cc(Br)cc(F)c1O C1(NC(COC2(C)CCCC2)=O)CCCC2CN(c3nc4cccnc4s3)CC12 C(CN=c1nc2c(cnn2C)c(NCC(C)C(=O)NC)[nH]1)c1ccn(CC)n1 c1(NC(c2n[nH]cc2-c2cc(O)cc(Br)c2)=O)nc(O)c2nc[nH]c2n1 c1(C(N2CC(NC(=O)CC(C)C)CC(OC)C2)=O)cc(O)ccc1[N+](=O)[O-] c1(C(=O)NCC2C(C)(C)CN(C(C3CCC(=O)N3)=O)C2)csc2c(O)ccnc12 C1(F)(CNC(C(C(C)C)N(C)C)=O)COCCN(C(=O)CCc2nccs2)C1 c1(CNC(C(C(=O)OC(C)(C)C)C2CC2)=O)nsc2ccccc12 C(=O)(CCCCCCS(N)(=O)=O)N(C)Cc1ccccc1F Cc1cc(C(=O)N(CC(O)CNC(=O)CCc2nnc(C3CCCC3)o2)C)sn1 C#Cc1cn(C)nc1C(=O)NCC(C)(C)CC1CN(C(=O)CC2CCCCC2C)C1 C(=O)(CC(O)CC(C)(C)C)N1CC2C(NC(Cc3c(C)ncc(Cl)c3)=O)C2C1 c1(C(N2CC(C(C)NC(CSCCC(C)C)=O)C2)=O)cocc1C(N)=O N1(C(C=C(CCC)C)=O)CCCC1C1CCN(C(c2c[nH]nc2C(C)C)=O)C1 C(=O)(CCCC(=O)N(C)C)N1C(CCC(N2C(C)CCCC2)=O)CCC1 c1(C(N(C(C)CCNC(c2cc3occc3s2)=O)C)=O)cnc2ncnn2c1N N1(CCNC(C2NC(=O)OC2)=O)CCN(C(C2CC(CF)C2)=O)CC12CCC2 C12(SC(C)C(c3cccn3C)=O)CCCC1N(C(=O)OC(C)(C)C)CC2 c1(OC)cc(C)c(C(N2CC=C(CNC(C3(CO)CC(F)(F)C3)=O)CC2)=O)cn1 c1(NC(=O)NC(C(CC)O)C)ccc(S(=O)(=O)NC2CCCC2)cc1 C1(C(=O)NC(C2(O)CCN(C(c3ccnn3C)=O)C2)C)CC=CC(O)C1 C=CC1CC1(CO)CNC(=O)CC(C)NC(C1(C)CC=CC1)=O C(C(CC(C)C)C(=O)N1CC2(CC(NC(C3CC(F)CN3C)=O)C2)C1)OC C12(OC)CCC(C(=O)N(C3CCN(C(=O)CC(C)(C)O)CC3)C)(CC1)C2 n1(CC(=O)NCCC2CN(C(c3c(CC)ocn3)=O)CC2C)ccc(C)cc1=O c1(C(=O)NC(CCOC)CNC(=O)CC2CCCCO2)ccc(Br)c(N)c1 C1(C(=O)NCC2C(CNC(c3csnn3)=O)C2)Cc2c[nH]cc2S1(=O)=O C#CC1(C(N2CCC2C(=O)OC)=O)CCN(C(c2ccc(C)cc2)=O)CC1 CS(=O)c1ccc(C(c2nnnn2-c2ccccc2)Sc2ccc(Cl)cc2)cc1 Cc1nn(C)c(C)c1CNC(C1CCCN1C(=O)CCCC1CCCC1)=O c1(OC)ccc(NC(=O)N(C(C)CS(C)(=O)=O)Cc2cccc(F)c2)c(C)c1 c1(C(=O)NCC#CCNC(C2(O)CC(C)(C)C2)=O)cnc2[nH]ncc2c1 c1(CN=C(NC(C#C)C(C)C)NCC2CCCO2)ccc2c(c1)CCNC2=O c1(CC(=O)NC2C(NC(CCc3n(C)cnc3)=O)C2)cc(C(F)(F)F)c(O)nn1 N1(C(c2ccc(C(C)O)cc2)=O)CCC2CN(S(=O)(=O)CCCCCl)CC12 c1(C(=O)NCC(=O)NCC2OCCN(CC)C2)ccc(F)c(F)c1 C(=O)(CC1OCc2ccccc21)NC1C(C)COCC1 C1(c2nc(CSC)[nH]n2)CCN(C(C2(CF)CC2(F)F)=O)CC1.C12(CC1)C(=O)N2 c1(C(N2CCCC(N(C)C(c3sc(F)cc3Cl)=O)C2)=O)c(C#N)cnn1C N1(C(C2N(C(c3c(C)ccc(C)c3O)=O)CCC2)=O)CCc2cccc(Br)c2C1 Cc1cc(C)c(C(=O)NCC2C3CN(C(=O)C#CC(=O)N(C)C)CC23)cc1C C1(NC(=O)CC2CCC(F)(F)CC2)CN(C(=O)C=CBr)C2CCCC12 c1(-c2nc(CC)[nH]n2)cc(OC)c(NC(C2Cc3nnsc3S2)=O)cc1OC c1(OC)cc(C(N2CC(NC(=O)C=C3CCC(C)C3)C(C)(C)C2)=O)c(O)c(Cl)c1 c1(C(=O)OC)c(C(=O)NCC(CO)NC(=O)CN2CC=CC2)noc1C c1(CNC(Cn2ccc(C)n2)=O)cc(C(=O)NCCC(O)C(C)C)ccn1 C1(NC(c2c(O)ccc(OC)c2)=O)CC2(CCCCN2C(=O)C2CC2)C1 C1(C)(C(N2C(CCNC(C(CC)NC(C)=O)=O)CCC2)=O)CCN(C)C1=O C(CCCCC(=O)NC1(COCC)CCN(C(c2ccc(Cl)cc2)=O)CC1)OC N1(C(C2C(C)C2)=O)CCC2(CCCN(C(=O)COc3ccccc3O)C2)C1 N1(C(CN2CC(CC)C2)=O)CC(CNC(=O)C(C)(C)CO)C(F)(F)C1 c1(C(N(C)CC2(O)CN(C(=O)C(C)(C)NS(C)(=O)=O)C2)=O)cc2cccnc2[nH]1 c1(C(N(C(=O)CN2CC3CCCCC3(CN)C2)CC)C)cccc2ncccc12 N1(C(CC2C(C)(C)C2)=O)CCC(CO)(CNC(=O)C(F)CC2CCCCC2)CC1 C(=O)(NN1CCCC1C(=O)NCc1c(C)cnn1C)c1c(C)csn1 C1(CN(C(=O)CCc2ccc(C)cc2)CC)CCN(C(C2COC(=O)O2)=O)CC1 C(=O)(C(C)(C)CCNC(C1C2CCC(F)C12)=O)Nc1c(CC)n(C)nc1 CCC(C)(CO)C(=O)N1CC(CNC(c2cc([N+](=O)[O-])c[nH]2)=O)C(O)C1 N1(C(CN(C(C(CCC)F)=O)C2CCC2)=O)CCN(CCO)C(=O)C1 C1(N(C(C2CN(CCC)C(=O)C2)=O)C)CCC2CN(C(=O)CNS(C)(=O)=O)CC12 C1(C(=O)NC2CN(C(c3cc(C)no3)=O)CC2C(F)F)CN2CCC1CC2 C1(NC(c2c(OC)ccs2)=O)COCCN1C(C)=O S(=O)(=O)(c1ccc(NCC2C=CCCC2)cc1Cl)N1CCN(CCS(C)=O)CC1 C1(NC(CCN(C(C)=O)C)=O)CC12CCN(C(c1cnc(C)cc1Cl)=O)C2 c1(OC)cc(C(=O)NC(C)C)c(-c2cnc(F)cc2C)cn1 N1(C(C(C)OCC(C)C)=O)CCOCC1CC(=O)NCCCCF C1(C(=O)NC2CC(CN)OC2)CCc2cnccc2N1 CC1CCSC1C(N1CC(F)(CNC(=O)CCc2ncc[nH]2)C1)=O c1(CC)oc(C)cc1C(=O)NCCC(C)N(C)C(c1csc(=NC)[nH]1)=O C(=O)(C(C)(C)CNC(=O)CC1CC=CCC1)N(C(C)C)C C(=O)(C1COc2ccc(Cl)cc21)N(CCN(C)C(c1cncc(CO)c1)=O)C C1(S(N)(=O)=O)(C(N2CCC(CCNC(c3c(C)c[nH]n3)=O)C2)=O)CC1 N1(C(C(=O)NCCCC)CC2CCC3CC23)CCC(Oc2cccnc2)C1 c1(NC(CN2C(CNC(C(C3CCCCC3)OC)=O)CC2)=O)ccc(F)cc1F N1(c2c(Cl)ncc(C)c2N)CCCC2(CCN(CC(N)=O)C2)C1 C=CCC(C)C(=O)N1CCCC1C(=O)N(C1COCC1O)C1CC1 C1(OC)CC(C(=O)NC2CCC2NC(c2csnc2C)=O)N(S(C)(=O)=O)C1 O=C(N=c1[nH]nc(Cl)cc1Br)C1C2CN(C(c3ccccc3I)=O)CC12 N1(C(CC(C2CC2)NC(C2(C(N)=O)CCC2)=O)=O)CCC2C(C=O)C2C1 N1(C(Cn2nnc(C)n2)=O)CCC2(CCCN2c2ncnc3c2OCCO3)CC1 N1(C(C=NOC)=O)CCC2(CCN(C(=O)Cc3c(C)cccc3C)C2)C1 C1(C(C)NC(C=CC=CC)=O)CCN(C(=O)Cc2cc(CC)no2)C1 C1(N(c2snc(SC)n2)C)CCN(C(c2oc(C3CCC3)nc2C)=O)CC1 c1(C(N(C)CCNC(c2ccc(CCF)cc2)=O)=O)cn2ccccc2n1 CN(C)NC(=O)CCC(=O)N1CCCC(NC(c2cnn3c2C(C)CCC3)=O)C1 C(=O)(C(O)CCn1cncn1)NCCOCC(N1CC(=C)C1)=O c1(CCC)cn2c(n1)C(C(=O)N(c1ccc(Cl)cc1)CC)CCC2 N1(C(c2c(CC)csc2)=O)CCCC(N(C(=O)Cn2nccc2C)CC)C1 CCCC(CC1CCCC1)C(=O)NCC1CCC(NC(C2CCN(C)C2)=O)CC1 C1(CN(C(=O)C(F)C2CCOC2)CC)CCN(C(=O)CC2(CSC3CC3)CC2)C1 CC1(C(=O)NCc2ccccc2CNC(=O)CN2CC(=O)NC2=O)CCCCO1 N1(CCOC)CCC(C)C1.C12CCN1CC(C)OC(=O)CC1(CC1)N(C)C2=O C1(C(=O)NC(c2nc(CC)[nH]n2)C)CC=CC(NC(=O)CCc2cncnc2)C1 C1(NC(C(C2CC2)SC)=O)CC(C)(CNC(=O)CC2(C3CC3)CC2)C1 Cn1cc(Br)c(CN2CCC2C(=O)NCc2ccc(C(F)F)cc2)n1 N#Cc1nc(=NCC2(F)CCN(C(=O)CCOCC3CCCO3)CC2)c(Cl)c[nH]1 C(CCC(=O)NCC(CO)C(C)C)(C(C)C)NC(c1cc(C)nnc1C)=O CCC(C(=O)N1CCCCC(NC(=O)C(C)(C)N(C)C)C1)C(C)O c1(C(=O)NCC2C=CCN2C(c2cnc(S)[nH]2)=O)cc2nc(=O)ccn2[nH]1 c1(CCC(=O)NC2CC(F)(C(=O)O)C2)cnc2cc(Br)ccn12 C(=O)(C1CCc2cccc(F)c21)NC(CNC(c1cncc2sccc12)=O)CO O=C(CS(=O)(=O)Cc1cccs1)NCC1(O)CN(C(c2cnnc(O)c2)=O)C1 N1(C(c2cnn(C(C)C)c2Cl)=O)CC2CCN(C(C3CCC(=O)N3C)=O)C2C1 C1(C(=O)OCC)CC2(C1)CC21CC1.C1(C2CC(F)(F)C2)CS(=O)(=O)N1 C1(OC)CCN(C(=O)C=CC(C)NC(=O)CC23CCCC2C3)O1 C1(NCC)CCCC(N=c2[nH]c3c(c(=NCC4(C)CC4)[nH]2)CSC3)C1 c1(C(N2CC(C(N(C)C)=O)C(O)C2)=O)ncnc2c1ccn2C c1(CN(C)C(c2ccccc2N2CCNC2=O)=O)ccc(Br)cc1Cl c1(C(N2CCN(C(C(N)=O)=O)C3C2COC3)=O)cc(C2CC2)nc2ccc(Cl)cc12 c1(C(N2C3C(NC(c4cc(C5CC5)on4)=O)C(C3)C2)=O)csc2ncnc(O)c12 CC1(C)CCCC(C(=O)NCc2csc(C(=O)NC3CCCC3C(C)(C)C)c2)C1 C(C1CCCN1C)=Cc1cn(C2CCC(C(N(CCN(C)C)CC)=O)C2)nn1 C(=O)(C(C)(O)C(C)C)Nc1c(C)cc(SCCCc2cn(CCC(=O)OC)nn2)o1 CC1(CCNC(=O)CCC2(NC(c3cccnn3)=O)CCC2)CCOC1 Cn1ccc(C(=O)NCC(O)CNC(c2ccn(CCO)c(=O)c2)=O)c(O)c1=O n1(CC(=O)NC2CN(C(C(COC)(C)C)=O)CC2C)ccc2cc(OC)ccc12 c1(C(=O)NC2CCN(C(C(CCC)c3ccccc3)=O)C2C)cc(F)ccc1Cl C(=O)(C(C(C)(C)C)NC(c1n(C)ncc1C1CC1)=O)NCC1(C)CCC1 C1(C(N(C)CC2CN(C(=O)C3=COCCO3)CCO2)=O)CCn2nncc2C1 c1(C(=O)NCC(C)NC(C(C2CC2)SC)=O)ccc(Cl)c2cccnc12 c1(OCCC(=O)NCC(CNC(C2(CC#C)CC2)=O)F)ccc(C)cc1C N1(C(C2N(CC)CCOC2)=O)CCC(CNC(c2conc2C(C)C)=O)C(O)C1 C1(CC(=O)N(CC(C)NC(c2c(C)nc(CO)nc2)=O)C)CS(=O)(=O)CCN1C N1(C(C(CC)OC)=O)CCOC2(C1)CN(C(=O)CCc1cccc(C#N)c1)C2 C=CCCC(C(=O)NCCC(CO)C(C)C)NC(c1coc2c1COC2)=O CCC(CC(=O)NCCC(C)NC(=O)Cc1ccc(OC)c(OC)c1)C(C)(C)C c1(OC)cnc(C(N2CC3(CC3)CC2CNC(c2ccncc2F)=O)=O)c(F)c1 C1(OC)CC2CC(CO)CC12.c12ccc(cc1)C(=O)N1CCN(CC1)C2=O c1(C(=O)NCCNC(c2c(C)cncc2)=O)ccc(C)c(C#N)c1 C(CCCCOC)(c1n(CCCC)nnn1)NC(C(C)C)c1cncs1 CN1CCC(CN(C(c2sccc2Br)C(=O)NCCC2(C)CC2)C)CC1 CCCC(C#N)C(=O)N1CC(NC(c2cc(OC)nn2C)=O)C(SC)C1 CCC(C)(C)C(O)C(=O)N1CC(NC(c2cccc(C)c2N)=O)C(C)C1 Cc1cc(N)cc(C(=O)NC(C)(CNC(=O)CC2OCCC2(C)C)CO)c1F c1(C(=O)NC2CCN(C(c3cc(C)n(C4CC4)n3)=O)C2)cc(O)c2sccc2c1 c1(C(=O)NC(C(C)C)C)coc2c1CN(C(=O)CC1(O)CCOCC1)C2 c1(SC)cccc(C(=O)NCC(C)(O)CNC(C2CCC(F)(F)C2)=O)c1[N+](=O)[O-] C1(CC=C)(NC(=O)C(C(C)C)OC)CCCN(c2nnc(O)s2)C1 c1(CNC2C(C)COC2)ccnc(S(C)(=O)=O)c1 C1(NC(c2cn(CC(C)C)nc2)=O)CCCN(C(=O)Cc2csc(S)n2)C1C C12(NC(c3cc(C)on3)=O)CCCN(C(=O)C=Cc3cccnc3)CC1C2 C(=O)(C(CCCC)CCCCC)N1CCC(C(C)NC(CC=CC=C)=O)C1 CN1CCC(NC(=O)Nc2ccc(F)c(NC(N)=O)c2)CC12CC2 C(=O)(CCC(=O)N1CCCCC1C1CCCN(C(=O)CN2CCCCC2)C1)NC C(=O)(CC(C(C)(C)C)NC(C1COCCC1C)=O)NCCC(C)(C)OC c1(CC(=O)NCCCC(C)NC(CCC(=O)NC)=O)coc2ccccc12 c1(C(C)C)cccc(OC(C)C(=O)NCC(C)(C)NC(C2COC(=O)N2C)=O)c1 c1(OC)ccc2cnc(N3CCC(NC(=O)C=CC4CC4)C(C)(C)C3)nc2c1 Cc1cc(C)c(C(=O)NC(CNC(c2n[nH]cc2C(C)C)=O)C2CCC2)c(C)c1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CC(CCNC(c2ncccc2O)=O)(OC)C1 c1(CC)cc(NC(=O)CC2CC(NC(=O)C(C)CCOC)C2)cc(C)c1 C12(CNC(c3ccnc(O)c3Br)=O)CCCC1N(C(C1CCC1)=O)CCC2 c1(NCC2CCN(C(C=C(C)C(C)C)=O)CC2C)ncc(C#N)cc1C C=CCC(CC(C)C)C(=O)NCc1occc1C(N1CC(O)CC(C)(C)C1)=O C12(NC(C(N3CCC(S(C)(=N)=O)CC3)c3c(C)n(C)nc3)=O)CC3CC(CC(C3)C1)C2 C1(CC(=O)NCC(CNC(C2(COC)COC2)=O)O)Sc2ccccc2NC1=O N1(C(CCc2n(CC)ccn2)=O)CCC2CN(C(=O)CCCC#N)C(C)C12 C(CCCN=[N+]=[N-])NC(COC1(C)CN(C(C2CCC(N(C)C)C2)=O)C1)=O C1(C(=O)NCC(=O)NCCOC)(C(F)F)CC2(CC2)C1.c12cc([nH]n1)CNC2=O c1(C(C)C(N2CCC(NC(=O)C(Cl)(Cl)Cl)C2)=O)ccc(Cl)c(Cl)c1 c1(CS(N2CC(C(=O)NCc3cnc(Cl)s3)OCC2)(=O)=O)ccc(Br)cc1F Cc1cc(C(N2CC(CNC(=O)CS(=O)(=O)CCO)CC2C)=O)c(Cl)cc1N C(=O)(CC(C(F)F)c1cccc(F)c1)N(CC(C)NC(c1c(C)nccc1)=O)C N1(C(C(C)c2cccs2)=O)CCC(C2CC2)(CNC(=O)C2=CCCCC2)C1 c1(C(=O)NCC(C)(O)CNC(=O)CCN2CCCC2=O)ccc2ncsc2c1 C(=O)(C#CC1CCCCO1)NC(CCNC(c1cn(CC)nc1)=O)(C)C CC1(C2CCN(CCC3SCCS3)CC2)COC(=O)N1 c1(C(N2CCC(NC(C3C4COCC34)=O)CC2)=O)cc2cc(Cl)cc(Cl)c2[nH]1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1CN(C(=O)CC2CCC3COCCC3C2)C1)C N1(C(C2(C)CCNCC2)=O)CCN(CC(=O)NC(=O)C(C)(C)CBr)C(=O)C1 N1(C(NNC(c2c(C)cc(C)cc2F)=O)=O)CCC(S(=O)(=O)C(C)C)C1 C1(CC(=O)NC(CNC(C=C(C)C(F)F)=O)CC(C)C)CN2CCN1CC2 CC(C)CCC(=O)N1CC(C)CC1C(=O)NCC1CC(CN(C)C)C1 C1(NC(c2coc(Cl)n2)=O)CC(F)CN(C(=O)C=Cc2ccncn2)C1 c1(C(=O)NC2CC(C)(NC(c3ccn(CCOC)n3)=O)C2)nncnc1C C(=O)(C1=C(C)N(CC)C(=O)NC1c1cc(C)cc(Br)c1O)OCCN(C)CC c1(C2N(C(C3CCCN(Cc4csc(Cl)n4)C3)=O)CCC2)ccc(F)cc1F c1(CO)cc(N2CC3CC2CN3CC(C2(OC)CCC2)(F)F)nc(C(F)(F)F)n1 CCCC(CCC)CC(=O)N1CC(O)CC1CNC(c1cc2c(s1)CCCC2)=O C1(CC(=O)NCC2C(NC(CCCOC(C)(C)C)=O)C2)NC(=O)CNC1=O C1(C(=O)NC(C#C)C)CCN1C(c1cncs1)=O CC(CC(N)=O)N=c1nc(N2CC3CCC2C(O)C3)c2c([nH]1)CCCC2 C1(C(=O)NCC(C(C)(C)C)O)Cc2nccnc2CN1C(c1cccnc1Cl)=O N1(C(C2N(C(c3c(C)csc3)=O)CC3CC32)=O)CCn2ncnc2C1 C(=O)(CCC(=O)NCC1CC1NC(=O)CS(=O)(=O)NC1CC1)NCC c1(C(=O)NC(CC)CNC(C2CC3CC3CC2C)=O)c(C)nn2cc(C)cnc12 N1(C(CC2CC(=C)C2)=O)CCC2CN(C(=O)C(O)C(F)F)CCC12 Cc1cccc(Br)c1C(C(N1C2CCC1C(CN)C2)=O)C1CCCC1 c1(C(=O)NCCC2CC(C(=O)NC(C(C)(C)OC)C)C2)cc2cccnc2[nH]1 C#CCC(CC(F)F)C(=O)NC(CC(=O)NC1(C(C)C)CC1)C(C)(C)C CC1(CNC(=O)C=Cc2cnc[nH]2)CCN(Cc2ccc(F)cc2)C1 C1(CC(=O)N(C2CCCC2)CC(=O)OC)NC(=O)N(c2ccc(C#N)cc2)C1=O c1(C(N2CC(C)CC(OC)C2)=O)ccc2c(n1)CN(C(=O)CSC)CC2 CC1CCN(C(c2ccnn2C2CCOCC2)=O)CCN1C(=O)CC(C)(C)F N1(C(CCCC(=C)C)=O)CC2CC(C1)CN(C(=O)CCN(CCCCC)C)C2 C(=O)(CC1OCc2cc(Cl)ccc21)NC1CC(NC(C(C)(C)C)=O)CC1O C1(C(=O)NC(CNC(CC(C)OC)=O)Cc2ccccc2)CCCC1(C)C C1(C(=O)NC(CC)C)CN(C(c2cc(C(F)(F)F)nc(Cl)c2)=O)CC1(F)F CC1CCCC1NC(=O)CCN(C(=O)C(C1CCC(=O)N1)C)C1CC1 O=C(C1=C(CC)OCCS1)NC12CCC(CC1NC(C13CC1COC31CCC1)=O)C2 c1(C(=O)NC2CC(C)CN(C(c3cnns3)=O)C2)ccc2c(=O)ccoc2c1 c1(CNc2cncc(C(N3CCn4cccc4C3)=O)c2)c(Cl)cc(Cl)nc1Cl CC(O)(C(=O)N1CCCC1c1cn(Cc2ccc(F)c(F)c2)nn1)C(F)(F)F c1(CC(CC)C)nc(-c2oc(C(F)F)cc2C)n(CCOC(C)C)n1 C(=O)(C(C)CC(F)(F)F)NC1C(C)N(Cc2ccc(C(N)=O)cc2F)CCC1 C(C)(C(C(=O)N(CC(O)COC)C)NC(N)=O)OC C(=O)(CCC(=O)N1CCC(NC(=O)CCC=CC(C)C)C1C(C)C)NCCC c1(C(=O)NCC2(NC(C(=O)NCC)=O)CCCCC2)ccc2c(c1)CCC2(C)C c1(N(C)CC2CCN(C(C3(O)CC(C)(C)C3)=O)C2)nc2ccccc2o1 c1(CNC(C=CCC)=O)ccc(CC(C)NC(C2CCNC2=O)=O)cc1 CC1CCN(N2CCCC2c2cn(-c3cccc(N(C)C)c3)nn2)CC1 C1(NC(C2(CC)COC2)=O)C2CN(C(=O)Cc3cncn3-c3cnn(C)c3)CC12 N1(C(Cc2cn(CC)nc2)=O)CC(NC(=O)CCc2ccn(C)n2)C2(CC2)C1 c1(NC(C)C)nnccc1NC(C1(NC(=O)C(=O)NCC(F)(F)F)CCCC1)=O c1(C(N2C(C)CCC(NC(C3ON=C(CC)C3)=O)C2)=O)cnn2ncccc12 c1(CC)cncc(C(N2CC(NC(=O)COC(CC)CC)CC2CO)=O)c1 Cc1cccc(Br)c1C(C(=O)NCC(C)(C)C1CC1)NC(c1ccc(Cl)cc1)=O C1(CC)CCCC1(C)C(=O)NC1CC(NC(c2ccn(-c3ccncc3)n2)=O)C1 CCCCC(CNC(=O)C(CCOC)OC)NC(=O)C(c1ccc(C)cc1)(C)C CC1(O)CCN(C(C2CC(O)(CNC(C3C4(CC4)C34CC4)=O)C2)=O)CC1 N1(C(C2CCCO2)=O)CCC2(CC1)CC(C(=O)NC1C(O)C3CCCC13)C2 C1(CC)(NC(c2ccc(OC)nc2C)=O)CCN(C(=O)C(O)C(F)(F)F)CC1 C1(C(N2CC(C)N(C(C3CN(S(N)(=O)=O)C3)=O)CC2)=O)CCc2ncccc2C1 N1(C(C(C)=C2CC2)=O)CCC(OC2CCN(C(c3ccc(F)cc3)=O)CC2)CC1 C1(c2n(-c3cc(F)ncc3)nc(CC3CC4CCC3C4)n2)CC2(CO1)CC(F)(F)C2 c1(CNC(CC2CC(=O)NC2=O)=O)cnn2c1CN(CC(O)CC(F)(F)F)CC2 C1(C(=O)NC(C)(C)CNC(c2ccc(Br)cc2N)=O)CCc2cncn2C1 S(=O)(=O)(c1cccc(Cl)c1)N1CCCC(F)(CNC(C(C(C)C)O)=O)C1 CC1CCCN(C(c2ccc(Cn3cc(CN4CCCC4=O)nn3)o2)=O)C1CO C1(C(N(CCOCCNC(C2(C(=O)OC)CC23CC3)=O)C)=O)CCC=CCCC1 Cn1nc(C(N2CCC(CNC(c3nc(C4CC4)cs3)=O)C2)=O)c(C(F)F)c1Cl C(C(O)C(=O)NOC1CC2CCC1C2)=CC.CC(=O)N C1(NC(C(CC)OC)=O)CC2CCCC(C1)N2C(c1[nH]cnc1C#N)=O N1(C(CNC(CC)=O)=O)CC2CCC1CN2C(C1OC2CCCCC2C1C)=O C1(C(=O)NC2C(N=[N+]=[N-])CNC2)CCC2(CC1)C(C(=O)O)C2(F)F c1(NC(C(N2C(C=C)COCC2)c2ccc(CC)cc2)=O)c(C)cc(C)cc1C c1(C(N(C)CCC2CCN(C(C3CNC(=O)C3)=O)CC2)=O)n[nH]c2c1CCC2 c1(OC)nc(C)ncc1C(=O)NCC1(F)CCN(C(=O)C=CSC)CC1 N1(C(C(C)NC(=O)NC)=O)CCN(C(C2CCc3n[nH]cc3C2)=O)CC(C)C1 C1(C(=O)Nc2ccc(N3CCN(C)CC3)nc2)CC12CCN(Cc1cn[nH]c1)C2 C1(CC(=O)N(C2CC(C)C2)C)CCN(C(C23CCC(C2)C3)=O)C1(C)C N1(C(c2cnc(C#N)s2)=O)CCCC2(CCCN2C(=O)CSCc2ncc[nH]2)C1 N1(C(C(C)OCCC#C)=O)CC2(CCCN(C(C3CCCCN3C(C)=O)=O)C2)C1 c1(CC)cc(C(N2CCC(NC(=O)CC3COCCO3)C(O)C2)=O)ccc1F C1(CC(=O)NCCCN(C)C(c2ccnc(OC(F)F)c2)=O)CCOC(C(C)C)C1 C(C(F)(C(=O)NC1CCCCC1(C)C)C(C)C)NC(c1cc(C)oc1C)=O Cc1cc(C)c(C=CC(N2CC(NC(=O)C3=CCCC3)CC(F)C2)=O)cc1C c1(C(=O)NCC(CNC(c2cnc(N(C)C)s2)=O)OC)cc(Cl)c(F)c(Cl)c1 C(=O)(C1=COCCC1)N1C2C(CNC(=O)CC3CCC4CC4C3)C(C2)C1 C1(C(=O)N(C)CC2COCCO2)(NC(c2n(CC)nnc2)=O)CCCC1C C1(NC(=O)NC2C(SC)COC2)CC12CCc1cc(Br)ccc12 c1(OC)c[nH]c(C(=O)NC2CCN(C(c3ccc(C)s3)=O)C(C)C2)cc1=O CCC(C)CCC(=O)N1CCC(NN2CCCS2(=O)=O)C1.C1(C)(C)CCNC(=O)C1 CCCC(C)CC(=O)NCC1CN(C(c2c(C)noc2C(F)F)=O)CCO1 C(=O)(C(C#N)C(C)C)N(CCNC(c1cnc(C(C)O)s1)=O)CC C1(C(N2C(CC=C)(CC=C)CCC2)=O)CCN(C(c2ccncc2N)=O)C1(C)C N1(C(C(C(C)C)F)=O)CCC2(C1)CN(C(c1cnc(CC3CC3)s1)=O)CCO2 C1(CC(=O)NCc2nnnn2-c2ccccc2)CCCCC1O c1(C(C(=O)OC)NC(c2cccc(Cl)c2)C(F)F)cc(C)cc(C)c1 C(=O)(C1=CCC(C)CC1)N1CC(O)(C(=O)NCc2cc(C)ns2)C1 c1(C(N(CC(C)O)CCNC(CSC)=O)=O)snc2ccccc12 CC(CF)CC(=O)N(C)CCNC(=O)Cc1cccc(OC(C)C#N)c1 N1(C(c2ccc(CN(C)C)o2)=O)c2ccncc2CCC1CO CC(CC(=O)NC1(C)CC(NC(C2CCCN(C)C2)=O)C1)C(C)(C)C c1(C(N2CCC(N(C(c3cc(C)cc(C)n3)=O)CC)C2)=O)ccc(S(C)=O)cc1 c1(C(N(C)CC2CCN(C(C(C)NS(CC)(=O)=O)=O)C2)=O)c(Cl)ccc(C)c1N c1(OC)cc(C(C)=O)c(NC(C2CC2C(=O)Nc2cc(Cl)ccc2I)=O)cn1 C(=O)(CS(=O)(=O)c1ccccc1F)NCC1N(C(Cc2cnc(C)[nH]2)=O)CC=C1 c1(C(N2C(C(C)NC(=O)CC3CSCCS3)CCC2)=O)ccc(F)s1 C1(C(=O)NC)C=CC(NC(=O)CNC=O)C1.c1(C(=O)NCC=O)cccs1 Cc1nn(CC(=O)NC(C)CC2CN(C(=O)CC3COCCO3)C2)c(=O)n1C Cc1ncncc1C(=O)NCC(C)N(C(=O)C(C)Sc1ccccc1Cl)C N1(C(C(COC)COC)=O)CCC(CO)C(NC(=O)CCN2CCNC(=O)C2)C1 c1(C(N2CCN(C(c3ccc(C)o3)=O)C(C(C)C)C2)=O)cnn2c1OCC(O)C2 C1(C(=O)NCC#C)CCC2CCC1N2C(=O)CN1CC(=O)NC1=O N1(C(c2c(C)noc2)=O)CC(C(=O)N(C)Cc2nc(C)ns2)C(C)(C)C1 C(=O)(C1=CCCOC1)NC(C)CCNC(=O)CCc1ccnc(Br)c1 CC(CC(F)(F)F)C(=O)NCC1CCCN(C(=O)C(C)(O)c2ccccn2)CC1 N1(C(c2cc(OC)c(O)nc2)=O)CCC(C2CC2NC(c2conc2C)=O)CC1 C=CCC(CC)C(=O)N(C(C)(C(=O)NCCCc1cnn(C)c1)C1CC1)C C1(C(=O)NCC2(OC)CN(C(c3cncc(Cl)c3)=O)C2)CC(C(C)=NO)C1(C)C CC1CC(C(=O)NC(C)CC(N2C3CCC2COC3)=O)=NO1 N1(C(C(C2CC2)OC)=O)CC2CN(C(=O)Cn3cc(C)cn3)CCC12 C1(NC(=O)NCC2CCC(C)(CC)O2)CCC(C2CC2)C1 Cc1c(C(=O)NC23CCC(CC2NC(=O)Cc2csc(S)n2)C3)cccc1Cl c1(-c2cn(COC)nc2)c[nH]c2ccc(C(=O)Nc3cc(F)c(C)cn3)cc12 C1(NC(c2n(CC)cnn2)=O)CCCCCN(C(c2snnc2C)=O)C1 N1(C(C2CC(C)(F)C2)=O)CCC(CO)C(NC(c2csc(Cl)n2)=O)C1 C1(CCSC)C(=O)NCC2CCCCN12.c1(C2CC2)ccco1.CO N1(C(c2cc(SC)oc2)=O)CCOC(C(=O)NC(C)Cc2nn[nH]n2)CC1 c1(OC)cc(C(=O)NCC2COCC2NC(=O)COC(C)(C)C)[nH]n1 C(=O)(C(CCNC(c1cc(C2CC2)[nH]n1)=O)OC)N1CC(CC)C1 c1(C(=O)NCCC(C)(C)NC(c2c(C)ccc(OC)n2)=O)cccc2ccnn12 C=Cc1ccc(C(=O)NC(C)(CO)C(=O)NC(CC(=O)OC)C2CC2)cc1 CCC(C)(CO)C(=O)N1CCC(OC2CN(C(=O)CC3CCC(=O)N3C)C2)CC1 Cc1cnc(CNC(C23CC(CN2C2CC2)C3)=O)nc1 c1(C(=O)NCCCC(C)NC(=O)CC2(C)CC2(F)F)ccnnc1O c1(CN(C)C(c2cccn2C)=O)ccc(CNC(c2ncn(C)n2)=O)cc1 c1(C(=O)NCC(C)(C2CC2)NC(C2C(C)=C2)=O)cnc(Cl)c(C2CC2)c1 N1(C(C2CC(C)OC2)=O)CCC(Nc2ccncn2)CC1C CC(CNC(=O)OC(C)(C)C)CC(=O)N1CCC(N(C(=O)Cc2cn[nH]c2)C)C1 C1(NC(COCCCCCC)=O)CC2(CCC2)CN1C(=O)CCCc1cccs1 N1(C(C(C)CF)=O)CC2CC2(NC(=O)COc2cncc(Cl)n2)C1 c1(C2C(C(=O)NC(CC=C)CNC(=O)C(C)=C(C)C)C2)cccc(OC)c1 c1(C(=O)NCCCNC(C)=O)nn2ccccc2c1C(N1CCCC(Br)CC1)=O c1(C(NNC(CNC(=O)Cc2ncc[nH]2)=O)=O)ccc2c(c1)OCO2 C(CC(C(=O)N(C)CCN(C)C1CC1)NC(=O)CSC(F)(F)F)=CC CC(C)CC(C(=O)N(C1CC2CC2C1)C)ONC(C1C(C#N)C1(C)C)=O CC(C)C(CNC(c1cnn(CCF)c1)=O)NC(C1(C(F)F)CCCC1)=O c1(-c2onc(-c3c(OC)nccc3)n2)nc(C)nc2sc3c(c12)CCCC3 N1(C(CCCc2nc(C)sc2)=O)CCC(C)(NC(C2CCCCCC2)=O)C1 C#CC1(C)CCCN(C(C2C(C3CC3)CCN2C(c2cnn3c2CCC3)=O)=O)C1 C(C(C)(O)CC(=O)NCC1CCCCN1C(=O)CCC(C)(C)O)OC c1(C(=O)NC(CNC(c2nccc(CC)c2)=O)C(C)(C)C)cc(C)n(C)c(=O)c1 Cc1cncc(-c2cn(CC3CN(C(C4(CN)CCOC4)=O)C3)nn2)c1.C1(CC)CC1 c1(C(=O)OC(C)(C)C)ccc(C2CCCN(CC3CC3(C)C)C2)cc1 C(=O)(C1CCCc2nccn21)NC(C)CCNC(=O)CCn1cnnn1 Cc1cc(C#N)c[nH]c1=NCCCC(C)NC(c1cnn2c1CCC2)=O C1(C(N2CC(CNC(C(CCOC)C)=O)OCC2)=O)CN2CCN1C(C)C2 C(c1cn(C)nn1)=CC(=O)NC(C(C)NC(c1csc(-c2cccs2)n1)=O)CO C1(CNC(c2nnc(CC)s2)=O)COCCN1C(=O)C(C)c1cccs1 c1(CC)ncc(C(=O)NCC2(C(F)F)CCN(C(=O)C(C)(O)COC)C2)c(C)n1 C(N=c1ccn(CC2CCOC2)[nH]1)c1c(F)cc(Br)cc1.c1nnnn1C1CC1 CC1CN(C(C2CC(Cl)(Cl)C2)=O)CC(CCNC(=O)Cc2sc(O)nc2O)O1 Cc1nc(=N)[nH]cc1C(=O)NCC1CCN(C(C2CC(=O)N(CC(C)C)C2)=O)C1 c1(CC(N2CCCC(CCNC(CN(C)CCO)=O)C2)=O)cn2ccccc2n1 N1(C(C(C(C)C)CO)=O)CC(NC(=O)C(C)OCC2CCCO2)CC2(CCC2)C1 CCC(c1ccccc1)=CC(=O)N(C(C)CNC(c1ccnn1CCF)=O)C c1(C(N2CCC(CNC(CCC(=O)NCCC)=O)C2)=O)nc(C)ncc1Cl C(=O)(C1=NOC2COCC12)N(C(CNC(c1ccsc1C#N)=O)C1CC1)C c1(CC(=O)Nc2nc(CNC(C(F)=CCC)=O)sc2)cccc(OCC)c1 c1(CC(=O)Nc2c(CCN(C)C)cccc2)csc2cccc(F)c12 C1(S(N)(=O)=O)(C(=O)NCCCC2N(C(CCS(=O)(=O)NC)=O)CCC2)CCCC1 c1(C(N2CC(NC(C(C)CN(C)C)=O)C3(C2)CC3)=O)c(N)cc(Cl)cc1Cl N1(C(CN(CCC)C)=O)CCC(O)(CN(C(=O)Cc2cc[nH]n2)C)CC1 C1(O)(CNC(c2cc(SC)ncc2)=O)CCCN(C(=O)C(F)(F)CC2CC2)C1 Cc1cc(C(=O)NCC(=O)NCC(C)N(C)C(c2coc(C(C)C)n2)=O)n(C)n1 c1(SC)cc(C(N2CCC2CNC(=O)CCn2cc(Cl)cn2)=O)c(C)o1 C(C(C(C)C)C(C)C)NC(C1(C(C)C)N(C(C#CC(C)C)=O)CCC1)=O c1(C(N2CCC(C)(NC(=O)C=Cc3cccc(F)c3)C2)=O)ccc(P(C)(C)=O)o1 C(=O)(CCS(C)(=O)=O)NCCCCC(C)NC(C12CC(CO)(C1)OC2C)=O C1(N(C(C2(CCOC)CC2)=O)C)CCN(C(=O)C=CCN2CCCC2)CC1C CC(C)CCCCCC(=O)N1CCC(C)C1CNC(=O)CCCNC(N)=O S(=O)(=O)(c1c(Br)nc(C)cc1Br)NC(C)CF CN1CCC2CCN(C(C3CC4CN(C(=O)C5=NOCC5)CC4C3)=O)C2C1 c1(C(N2CCC(C(C)NC(C3CCC3C)=O)C2)=O)cccc(C2CC2)c1 c1(CN(C)CC2CCN(C(C3N(C(C)=O)CCC3)=O)CC2)cc2cc[nH]c2cn1 C(=O)(C1=CC2C=CC1C2)NCCC1CN(C(CCN(CC)CC)=O)CC(C)O1 N1(C(c2n(CCN(C)C)ncc2)=O)CCC(NC(=O)CCS(C)=O)C(CO)CC1 C1(CC#C)(C(=O)N(CCCCN(C(=O)Cc2csc(C)c2)C)C)CCOCC1 N1(CC(C)C)N=C(C(=O)NC2CCCC(NC(=O)CO)C2)CCC1=O c1(C(N2CC(F)CC(NC(CC3ON=C(C)C3)=O)C2)=O)cc2c(C)ccc(C)c2[nH]1 Cc1nc(CC(=O)N(C)CC2(NC(=O)COC3CCCC3)CC2)c(Cl)s1 c1(C(=O)OC(C(=O)Nc2c(OC)cccc2)C)cc2n(c(=O)c1)CCS2 C12(NC(=O)C=CC3CCOC3)CCC(CC1)N(C(c1cc(F)c(F)c(F)c1)=O)C2 C1(CNC(C(C)=C2CCCC2)=O)CC2CC(C1)N(C(=O)C=Cc1sccc1C)C2 Cc1ccc(C(=O)NCC2(O)CC(NC(=O)C(C)n3ccnc3)C2)c(Cl)c1 C1(NC(Cn2nnc(C)n2)=O)CC2CCC1CC2NC(C1CCCC(=O)O1)=O Cc1c(Br)noc1C(=O)NCC1CCN1C(C1CC1(F)F)=O CCC(C)C(O)C(=O)NC1(CNC(c2ccc(C(N)=O)c(Cl)c2)=O)CC1 Cc1cnc(CC(=O)NCCC(C)NC(c2c[nH]cc2C(F)(F)F)=O)s1.C1(C)CC1 C1(C(=O)NC(C(=O)NC2(C)C(C)(C)C2)C2CCCC2)C=CC=CC=C1 c1(C(N(CCN(CC)CC)CCN2CCC(C)C2)=O)ccc(N)c(F)n1 C1(NC(CCCCNC(C)=O)=O)CCN(C(c2ncc(C)cc2C)=O)CC1O c1(C2CCC(NC(=O)NCC3(COC(C)C)CCCC3)C2)cccc(Cl)c1 C1(C2CC2)(CNC(c2ccnc(OC3CC3)c2)=O)CCN(C(=O)CC2C=CCC2)C1 C1(C(=O)NCCC2(C(NOCC(C(C)C)O)=O)CC2)OCCOC1C c1(C(N2CCC(NC(C3CN(CC(F)(F)F)C3)=O)C2)=O)cn2ccnc2cn1 N1(C(C(C(CNC(CCNC(=O)NC)=O)C)F)=O)CC2(C1)NC(=O)NC2=O c1(-n2c(C(C3=CCSC3)NC(C)CC3CCC3)nnn2)ccc(F)cc1 C=C(C)CCN=c1nc(N2CC(C(=O)OC(C)(C)C)C(C)C2)c2cnn(C)c2[nH]1 Cc1cc(C(=O)N(CCCNC(C2CC2F)=O)C(C)C)cc(Br)c1 Cn1c(CCNC(=O)C(C)(C)c2ccc(Br)s2)nc2cc(Cl)ccc12 c1(C(=O)NCC(C)(O)C(=O)O)c[nH]c2c(F)cc(F)cc2c1=O n1(CCC(=O)NCCC(C)NC(CC2(N(C)C)COC2)=O)cnc([N+](=O)[O-])c1 c1(C(N2CC(C(C)NC(Cc3nc(CC)sc3)=O)C2)=O)nccc(C)c1O Cc1cc(C(C)(C)C)c(C)cc1NC1(c2nnnn2C2(C)CC2)COCCC1C C1(CNC(C(C)(C)C)=O)CN2CCCCC2CN1C(C1CC2C=CC1CC2)=O Cc1csc2ncnc(NC(C)CC(C)NC(=O)CC(C)(C)C(F)F)c12 c1(C(=O)OC)cc2cc(n1)N1CCC(CC1)CC1N(CC1)C2=O.SC Cn1nc(C(F)(F)F)c(I)c1CNC(C1OC2CCC1CC2)=O c1(C(=O)NC2(c3ncc[nH]3)CC2)cn(C(C2CNC(=O)O2)N(CC=C)CC=C)nn1 C1(CCNC(c2n[nH]cc2Br)=O)(NC(c2ccsn2)=O)CCCC1 N1(C(C(C(C)C)n2cncn2)=O)CCC(C)N(C(=O)C=Cc2ccoc2)CC1 N1(C(c2ncc(NC)nc2)=O)CCC(NC(=O)Cn2nnc(C3CC3)n2)C(O)C1 N1(C(C2C(CNC(C(C)OCC#C)=O)CCCC2)=O)CC2CC3CC2C1C3 c1(C(N2C(CCNC(=O)CC3(CO)CC3)CC(F)(F)C2)=O)ccc2ncnn2c1 CC1(NC(C2CC2(F)Cl)=O)CC(C(=O)NCCn2ccnc2)C1 CC(C)(C(=O)N1C2CCC1CC(NC(C1(F)CCCC1)=O)C2)C1=CCSCC1 C1(CNC(=O)Cc2cscn2)CN(C(C2(C(F)F)CCC2)=O)CCC1C(F)(F)F c1(C(N2CC3CN(Cc4cccc(I)c4F)C3C2)=O)c(F)cc(F)cc1Cl C1(C(C)NC(c2c(C)nc[nH]2)=O)CN(C(C2CC2CN(C)C)=O)CCO1 CC1CN(C(=O)C=C2CCSCC2)CC(C)C1NC(=O)CC12CCC(CC1)C2 C#Cc1cnn(C)c1C(N1CCC(NC(c2cocn2)=O)C1)=O c1(OC)cc(CNc2cc(N(C)CCC3CCCCC3)ncn2)ncn1 C1(C(=O)O)CC2CCN(C(=O)N=c3ccn(CCCc4ccccc4)[nH]3)CC12 CCC(F)(F)CC(=O)N(CCCNC(=O)CCc1cc(OC)no1)C N1(C(C)=O)CCCN(C(=O)C(C)CN(C(=O)CC23CCCC2C3)C)CC1 Cc1sc2ncc(C(=O)N(CCCCN(C(=O)C(O)C(C)C)C)C)n2c1C c1(C(C)C(=O)NC(C)(C)CNC(C2CC=CCO2)=O)ccc(Br)cc1 C(CCC(C(=O)NC(c1cncs1)C)NC(C1CC(C)C1)=O)OC Cc1cc(NC(C2CC2NCc2c(F)cc(F)cc2Br)=O)c([N+](=O)[O-])cc1Br N1(C(C(=O)NC)=O)CC2CC(NC(C3CC4CC4C3)=O)C2C1 O=C1CN(C(=O)C(C2CCCCC2)NC(=O)C2=CC3C=CC2C3)CC2(CC2)N1 C1(CNC(c2c(C)nco2)=O)C2CN(C(C3(O)CCOC3)=O)CC12 O=S(=O)(CCCS(=O)(=O)CCC(O)CC(F)(F)F)c1ccccc1 C1(C(F)(F)F)(C(=O)NC(CCOC)C(=O)N2CC(NC(=O)OC)C2)CC(CC)=NO1 C1(CNC(C2(C(=O)NC)CC2)=O)C2CCC(C2)N1C(=O)CCC(CC)OC c1(C(=O)NCC2(NC(c3ccc[nH]3)=O)C(C)CCCC2)ccn2cncc2c1 C12CCCN(C1)C2=O.CC(C)(C)C(=O)NC1CCCC1NS(C)(=O)=O c1(OC)cc(OC)cc(CN2CCCC2CC(=O)Nc2ccc(C(F)F)cn2)c1 c1(CC)[nH]c(=NC(CC2CC2)c2ccccc2N(C)C)[nH]c(=N)n1 N1(C(C(C(CC)O)(C)C)=O)CC2(CCCN(C(c3cc(C(N)=O)c[nH]3)=O)C2)C1 c1(OC)cccc(C)c1NC(=O)NCC(C)(C)COc1ccccc1Cl N1(C(C=CCN(C)C(C2CC2C2(C)COC2)=O)=O)CCC2(CNC(=O)O2)C1 Cn1cc(CNC(C2CN(C(N)=O)C2)=O)c(C(F)F)n1.C1(=O)C(C)(C)N1 C1(NC(C=CS(CC)(=O)=O)=O)CCC2CN(c3nc(C(C)C)nc(=N)[nH]3)CC2C1 c1(CC)ncnc(CC)c1NC(C12CCC(CN3CC(OC(C)=O)C3)(CC1)C2)=O c1(OC)ccc(CC(N2CC3(CCC3NC(=O)CC(C)(C)O)C2)=O)c(C)c1 C1(C(=O)NC(CN(C(c2cc(SC)oc2C)=O)CC)C)CC2CCC(C1)O2 c1(OC)ccc(COC(C2CC(=O)N(C)C2c2ccccc2)=O)c(C)n1 N1(C(CCNC(=O)OC)=O)CCCCC1CNC(=O)C(C)c1cccs1 CCCC(CCCNC(=O)C(=Cc1c[nH]cn1)F)NC(=O)Cc1ccc(N)cn1 c1(C(=O)NC(C2CC2C(=O)NCC2CC3CCC3C2)C)cc([N+](=O)[O-])n[nH]1 CC(C)CC(C)CC(=O)N1CCC(C(C)(C)NC(c2cncc(F)c2)=O)CC1 c1(C(N(CCC)CCNC(=O)C(O)C(C)OC)=O)c([N+](=O)[O-])ccc(C)c1C c1(OC)cc(F)ccc1S(C)(=O)=O.c1(C(=O)OC)ccc(SC)cc1Cl C1(CNC(C2C(C=C)C2)=O)CN(C(c2ccc(CCC=C)cc2)=O)CC12CCC2 C1(=O)C(CCC(N)=O)N1.C1(c2cccc(Br)c2)(OC(C)(C)C)CCCCC1 C1(C#N)(C(=O)NCC2N(C(Cn3nnc(C)n3)=O)CC(O)C2)CC12CCOCC2 c1(SCC(=O)NCC2C(NC(C3CCC(C)(C)O3)=O)CC2)ncnc2[nH]cnc12 N1(C(C2CC(C)(C(F)F)C2)=O)CC(NC(=O)C(C)(C)C)C(c2ccccc2F)C1 N1(C(c2n(CC)ncc2)=O)CCC2CN(C(=O)CCN(C)C)CC12 Cn1[nH]c(=NC(=O)NCC2CCC(O)(C(F)(F)F)C2)cc1C#N C(=O)(C(C)C(C)(F)F)N(C)CC1(CNC(C(CC)n2nccc2C)=O)CC1 CC1(C)OC2(C(N3CCCC(CCNC(=O)CCCN=[N+]=[N-])CC3)=O)CC1C2 Cc1cccc(C)c1CC(=O)NCCC1CN(C(=O)C(C)N(CC(F)(F)F)C)C1 C(=O)(C(F)CC(C)(C)NC(c1cccnc1O)=O)NCc1cc(C)ncc1 c1(OC)ccc(C(C(=O)NC(C)C)N2CCC2c2ccc(Br)cc2OC)c(C)c1 C1(CNC(C(C)OCOC)=O)(NC(=O)C(C2CC2)SC)CCCC1 Cc1cc(Cl)ncc1NC(=O)C(C)CN(C)C(C1COCOC1)=O N1(C(CC2CN(Cc3c(C(=O)OC)ccc(Br)c3)C2)=O)CCN2CCCC2C1 C1(C(=O)NCC(C(C)C)NC(c2c(CC)n(C)cc2)=O)CCC(N=[N+]=[N-])CC1 N#Cc1cc(C(=O)NCC2CCN2C(=O)Cc2ccc(Cl)cn2)co1 C1(C(=O)NC2CCCC(C)C2)CN(Cc2ccc(-c3ccc(Br)s3)s2)CC1(F)F C(=O)(C1Cc2ccc(Cl)cc21)N(C)CCN c1(-c2nc(C(=O)NCC3CN(c4ncc(F)cn4)CCO3)sc2)cccnc1Cl c1(C(=O)NC(C2CN(C(c3cnsc3)=O)CCO2)C)ccc2c(c1)CC2 C1(C(=O)NCC(c2ccn(C)n2)C)C(NC(c2c[nH]c(=N)o2)=O)CC1O CC1CCN(C(=O)CCCC2CCC2)CC1CNC(C1(CO)CC1)=O c1(CC(N2CC(O)CC(N(C(=O)C=CCO)C)C2)=O)coc2cc(Cl)ccc12 N1(C(C(c2nc(C)sc2)=O)=O)CC2(CCC2NC(c2cnc3sccn23)=O)C1 CC1(C)CCCCC1C(=O)NC1CCC12CN(C(c1c(N)cccc1F)=O)C2 C1(NC(CC(C)C)=O)(CNC(=O)CCc2n[nH]c(=N)s2)CC2CCC1CC2 C1(NC(C2C(C)C2C)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)CC(C)(C)C1 C(C(CC)CC)N(C(=O)C(F)C1CC(NC(=O)C(C)CC2CC2)C1)CCC S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CC2CN(C(CC3C(=O)NC(=O)N3)=O)C2C1 N1(CC2CN(C(C)C)C(=O)C2)CC=C(CNC(c2cn(C(C)C)cn2)=O)CC1 c1(C(N2CCC(n3cc(CNC(c4cnccn4)=O)nn3)C2)=O)cc(Cl)c(Cl)s1 CCC(CN(C)C)CC(=O)NC1CC(F)(CNC(=O)CSc2nncs2)C1 N1(C(C2=CC(O)C(NC(COC(C)=O)=O)C2)=O)CCC2=C(CCCC2)C1 N1(C(C2(CC(C)C)CCC2)=O)CCOC2(C1)CN(C(=O)CC1CCCC(C)C1)C2 S(=O)(=O)(c1cc(C(=O)NCC(C)(C2CCC2)NC(=O)CC=C(C)C)co1)NC c1(C(N(CC(CN(C(=O)Cc2nncn2C)C)O)C)=O)cccnn1 C(=O)(N=S(C)(=O)c1ccccc1C)NC1(c2cc(C)cc(C)c2)CCCC1 CCC(CC(=O)N1CC(CNC(c2cnn(CC(C)C)c2)=O)CC1C)C(C)(C)C C(=O)(CC(C)n1cc(Br)cn1)NCC1CC(NC(CSCCOC)=O)C1 C1(C(N2CCN(C(C(CCC)N(C)C)=O)CC2)=O)CCCN(S(N)(=O)=O)C1 N1(C(C(C2CCC2)OC)=O)CCC(CNC(=O)C(=O)N=S(C)(C)=O)C(F)(F)CC1 Cc1nocc1NC(=O)CC1CCN(C(C2(C(=O)N(C)C)CCC2)=O)C1 c1(C(=O)NC2C(NC(C(CC=C)NC(C)=O)=O)CCC2)cnc2c(C)nsc2c1 C1(NC(C2N(CC)C(=O)CC2)=O)CCN(C(c2cn(C)nc2Cl)=O)C12CCCC2 CCC(CC(=O)NCCOCC(N1CCC(O)C(F)(F)C1)=O)C(C)(C)C C1(C(C)C(=O)NCC(C)N(C)C)CCN(C(C2CCC2C#N)=O)CC1 C1(OC)CC(CNC(=O)C(O)CC2CC2)N(C(c2sccc2CC#N)=O)C1 c1(C(N(CC(C)NC(=O)C(c2cnccn2)C)C)=O)ccc(OC(F)F)cc1F N1(C(c2c(OC)nn(C)c2)=O)CCC(NC(C2CCCCCC2)=O)C(C)C1 C1(NC(c2c(C)cn(C)c2)=O)CC(O)CN(C(c2ccc(C(C)O)cc2)=O)C1 Cc1nc2[nH][nH]cc-2c(=Nc2ccc(NC(=O)C(C)c3cccs3)cn2)n1 C(=O)(C1SCc2cccnc21)NCCOCCN(C)C(C1CCCCC1)=O Cc1n[nH]c(C)c1C(C)CC(=O)NCC(C)(C)CN(C(=O)C1=CCCS1)C N1(C(c2c(OC)cc(F)cc2)=O)C(C)CC2CN(C(=O)CCCCC(C)C)CC12 C1(C(N2CC(c3cn(CC(C4CC4)OC)nn3)C2)=O)CCCC12CC2 C(=O)(C(C)(C)CCNC(C1CN(C(N)=O)C1)=O)NC1C(C)SCC1 N1(C(CN(CCC#C)C)=O)CCC2(C(=O)NCC3OCCCC3(C)C)CCCC12 c1(OC)ccc(C(=O)NCC2(O)CCN(C(=O)CCSC3CCCC3)C2)c(OC)n1 c1(OCC(N2CC(O)(CNC(c3cc(SC)oc3C)=O)C2)=O)ccc(C#N)cc1 c1(CC)cc(C(=O)N(CCC(=O)NCCCN2CCOCC2)CC)n[nH]1 FC(F)(F)CCN=c1nc(N2CC=CCC3(CCOCC3)C2)c2ncccc2[nH]1 C1(NC(C(C=C)CC)=O)COC2(CCN(C(=O)CCC3CCCC3)C2)C1 C1(C(=O)NC2CCCN(C(CCc3n(C)cnc3)=O)C2)Cc2cccc(F)c2O1 C1(CNC(CCCCCN(C)C)=O)CCCC2(CN(C(=O)CC3CC3(C)C)C2)O1 n1(C(C(=O)N(C2CN(C(C(C3CCC3)OC)=O)C2)C)C)ccc(C)n1 C1(NC(C(COC)C)=O)CCCN(C(=O)Cc2c(Br)cnn2C)C1 c1(CC(C(=O)NC(N2CCOCC2)C)NC(C2CCC(=O)N2)=O)ccccc1Br N1(C(COCCOC)=O)CC(O)CCC1c1ccccc1 C1(C(=O)NCC(c2cn[nH]c2)C)(CNC(C2C(C(C)C)C2)=O)CCC1 CC1CN(C(=O)C(C2(O)CN(C(c3cnn4c3CCC4)=O)C2)F)Cc2nncn21 Cc1ccncc1CC(=O)NCC1C=CCN1C(=O)CC1(C)CCC1 Cc1nn(CC(C)C)c(C)c1CC(=O)NCC(O)CNC(=O)CC1(O)CCOC1 N1(C(C(C)N(CC)CC)=O)CC(CO)C2(C1)CN(C(C1CC3(CSC3)C1)=O)C2 N1(C(C(C(C)C)OCC)=O)CCC2(CC(NC(c3csc4nnsc34)=O)C2)C1 c1(CC)ncnc(N2CC3CC3(C(=O)Nc3ccc(OC)cc3Br)C2)c1F c1(NC(C2C(NC(C=Cc3ccc(C)s3)=O)C2)=O)ccc2c(c1)CCCC2=O c1(C(=O)NCC(CNC(C(C)OCOC)=O)O)cccc(C)c1Br C1(C(=O)NCC2CCC(NC(c3nc(C)oc3C)=O)CC2)COC(C)(C)CO1 c1(CC(=O)NC(CNC(CCCOC)=O)C2CCC2)cc(F)ccc1Cl c1(NC(=O)NC(CC#C)COC)cc(-c2ccco2)nn1-c1ccccc1 N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCCC2(CCC2NC(=O)CCCCO)C1 Cc1ncc(C(=O)NCCN(C(=O)CC2CCC2)CCOCCO)n1C(F)F N1(C(C)C(N2CCC(OCCNC(C3CCCSC3)=O)C2)=O)C(=O)CCC1=O CCCC(C#N)C(=O)NCc1occc1C(N1CCCC(CN=[N+]=[N-])C1)=O N(C(=NCC1(C#N)CCOC1)NC1C2(CC2)C12CC2)C(c1ccccc1)C c1(C(=O)OC)ccc(N)c(CO)c1.C12(COC)CN(C1)C2.C(=O)(CS)NCC(=O)OC c1(C(=O)NCC2C3CN(C(C(CC#C)C)=O)CC32)ccc(Cl)c(Cl)c1 c1(C(=O)NC2C3(CN(C(c4c(C)con4)=O)C3)CC2)ccc(F)c(C)c1Cl C#CC1CN(C(=O)Cc2ccc(C)cc2)CCN1C(=O)C(C#N)CC c1(C2N(C(CC3(C)CCOCC3)=O)CCC2)cccc([N+](=O)[O-])c1 C(C(COC)CC(=O)NC(C)CNC(C1(C(F)(F)F)CC1(C)C)=O)OC C(CCCCC(=O)N(C1CCN(C(c2cc(O)cc(O)n2)=O)C1)CCO)OCC Cc1cc(C(=O)NCCCCNC(C23CSCC2C3)=O)ncc1F c1(CC)cccc(C(=O)NCc2ccc(C(=O)NC3(C)CCSC3)cc2)n1 Cc1cc(C(C)C(N2CC(NC(=O)CCc3ncc[nH]3)CC(C)C2)=O)cc(F)c1 c1(C(=O)NC2C(N(C(=O)C(C)(C)N3CCOCC3)C)CCCC2)cc(Cl)ccn1 CCS(=O)(=O)CC(=O)NC1(C(=O)NC(c2ccc(O)nc2)C)CSC1 CCC(C)C(O)C(=O)NCC1CCC(NC(=O)CC2C=CCCC2)C1 O=C1CC(C(N2CCOCC2C(=O)Nc2cncnc2O)=O)C2(CCC2)C1 N1(C(CCCN(C)C)=O)CC2(CCCC(CNC(C3CC3F)=O)O2)C1 C1(n2cc(CCC(C)O)nn2)CC12CCN(C(c1ccc(F)o1)=O)CC2 C1(CC)CCC(C)CN1C(C1(C)C=CCN1C(c1ncsc1NC)=O)=O c1(C(=O)NCC(c2cnn(C)c2)NC(c2ccc(C)s2)C)ccnc(C(F)F)c1 CCC(C)(C)CCCC(=O)NC1(C)CCCN(C(c2ccc(N)c(F)n2)=O)C1 C1(CC(N2C(C(C)(C)NC(=O)Cc3ccc(Cl)s3)CCC2)=O)CC2(CCC2)CO1 C1(C(=O)NC(C(=O)OC)C(C)O)C2CC(O)C(C2)N1C(c1ccc([N+](=O)[O-])o1)=O Cc1nn(C)c(N)c1C(=O)NCC(C)O.C12(CC1)C(=O)NCCO2.C1CN1 CC(O)CCN=c1[nH]c2c(c(=NCC3CCCN3CC(F)F)[nH]1)CSC2 C1(NC(c2c(C)nco2)=O)CCC(C)(CNC(c2cc(F)n[nH]2)=O)C1 N1(Cc2c(C)n[nH]c2)CCC2(CC1)CC(NC(c1ncccc1Cl)=O)CO2 CC(CC(F)(F)F)C(=O)N1CCOCC(NC(c2cc(Cl)ncc2F)=O)C1 C(=O)(C1CCCc2cncn21)N(CCN(C(C(=O)Nc1ccc(C)cc1)=O)C)C C1(NC(=O)C=C2CC2)CN(C(=O)Cc2cccc(F)c2)CC1C(F)F c1(C(=O)NC(C)C(CO)NC(=O)C(C)(C)N(C)C)ccc(C2(C#N)CC2)cc1 CC(C)(C)C(=O)C(=O)N1CC(CNC(=O)CC(c2cccc(F)c2)O)C2CC2C1 C1(CC(=O)N(C2CCN(C(c3ns[nH]c3=O)=O)C2)CC#C)C=NN(C)C1=O N1(C(c2cc(Cl)ccn2)=O)CCC(F)(F)C(NCc2ccc(O)c(O)c2)C1 N1(C(c2c(C)cc(C)o2)=O)CCOC2(C1)CN(C(C13CC4CC1C3C4)=O)C2 C1(C2CCN(C(=O)CCc3ccsc3)CC2)(NC(Cn2ncn(C)c2=O)=O)CC1 CCC(CCC(=O)NCC1(OC)CCCCC1)NC(=O)COC1CC1 N1(C(C2CCCC(NC(c3occ4c3CCC4)=O)CC2)=O)CCc2n[nH]cc2C1 C1(CNC(=NCC)NC2CCN(c3ccccc3Cl)C2)CCC(=O)N(C2CC2)C1 C1(F)(CO)CCCN(c2nc(-c3c(Cl)cccc3Cl)cs2)C1 c1(N(C2CCN(C(=O)CC3CCCN3C)CC2)C)ncnc2ccccc12 c1(-c2cnc(N(C3CCNC3)C)nc2)c(Cl)cccc1Cl.C#CCCCC(=O)NC c1(CC(N2C3CN(C(CC(C)C(F)F)=O)C(C3)C2)=O)c[nH]c2ccc(Cl)cc12 CC1CC(NC(=O)C=Cc2ccc(C(N)=O)o2)CCN1C(c1nc(=O)n(C)[nH]1)=O c1(OCC(=O)NC(CNC(CCC2C(C)=NNC2=O)=O)C)c(C)cc(Cl)cc1Cl CC(C(CO)NC(=O)CCNC(=O)Cc1ccccc1)NC(C1CNC(=O)C1)=O c1(N(CCC#N)C(=O)N(CCC(F)(F)F)C)ccccc1OC C1(C(=O)NC(C(C)(C)NC(c2ccn(C(C)C)c2)=O)C)CCN(C2CC2)S1(=O)=O C1(NC(c2c(CC)csc2)=O)(CNC(=O)C(C#N)C(C)C)CC2CCC1CC2 Cc1cc(C)c(C(N2CCOCC2CN(C(=O)C=C2CCC2)C)=O)cn1 C1(NC(C(C=C=C)C)=O)CCC2(CC1)CC2NC(c1[nH]cnc1C)=O CC(C(=O)N1CCC(O)(C(C)NC(c2coc3c2COC3)=O)C1)C(C)(F)F C1(CN(C(CN(CC)CC)=O)C)CCCN1C(C1CC1F)=O Cc1cc(C(=O)NC2(CF)CN(C(=O)Cc3cnccc3Cl)C2)cc(C)c1N O=C1CC(CNC(=O)C(CC2CCOCC2)NC(=O)Cc2csnn2)CN1 C1(C(=O)NCC2CN(C(C)=O)CC2O)CCC(S(N)(=O)=O)CC1 N1(C(c2c(CC)c[nH]n2)=O)CC2(C1)SCCC2NC(=O)C=CC1CCOC1 c1(C(=O)NCCC2(NC(Cc3c(C)non3)=O)CC2)cncc2c1CCC2 c1(C(=O)NC2C(CNC(CCC(=O)NC)=O)C2)cc2cc(F)c(F)cc2[nH]1 C1(NC(C(C=C)(C)O)=O)CCN(C(=O)COCC(N2CCCC2)C)CCC1(F)F N1(CCOC(C2CCCO2)=O)CCN(C(=O)CCc2ccc(F)cc2F)C(=O)C1 N1(C(C2C(OC(C)=O)C2)=O)CCCCC(C(N2CCC(C#N)CC2)=O)C1 N1(C(CCC=C(C)C)=O)CC2CCN(C(c3cc(Br)ccc3F)=O)C2C1 N1(N(CCNC(C2CCCCC2)=O)C(=O)C2CC2)CCN(C(C2CC2Cl)=O)CC1 C1(C(C)(C)C(=O)NCC(C)(O)C2(C)CC2)CCCN(C(C2CCCS2)=O)C1 C(CN=c1[nH]c2ccc(Cl)cc2s1)C1(OC)CN(C(=O)Cn2cnnn2)C1 C1(NC(Cc2cccc(OCC)c2)=O)CCC2(CC1)CC(NC(C)=O)C2 Cc1cc(Br)c2oc(C(=O)NCC(C(C)(C)C)NC(=O)C3CC3)cc2c1 N1(C(=O)NC(c2ccon2)C)CCC2(CCOC2)C1 c1(C(N2CCC(CCN(C)C(C3C=CCCC3)=O)CC2)=O)cc(F)cc(F)c1 C1(OC)COCC1C(N)=O.C1(C2C(=O)N3CCC3C2)CC(F)(F)C1 N1(C(C2CCC(C)O2)=O)CCCC2(CCCN2C(c2cccc(O)c2F)=O)C1 N12CCOC(C1)C2.C1(c2nn[nH]n2)(C(=O)O)CCCO1 CC1=C(C)CC(C(N2CCCC2(C)CCC(=O)NCCC(C)C(C)(C)C)=O)CC1 c1(CC)ncccc1C(N1CCSCC1C(=O)Nc1cccc(I)c1)=O c1(OC)ccc2c(C(N3CC4(CC(O)C4)C3)=O)n[nH]c2c1F CC(=O)C(C)CC(C)C(=O)NCC(=O)NC(C)(C)CCCF c1(OC)c(C(=O)NC2CC2CNC(c2ccoc2)=O)ccc(Cl)c1C C(CCCCCC(=O)NOC1CCOC1)NC(C(C)n1cccc1)=O c1(C(N2CC3COCC3(C(N3CCC(CO)C3)=O)C2)=O)c(Cl)cc(Cl)cc1Cl C(CCC(C)(C)C(=O)N1CCCC(CC(=O)NCC(C)(C)C(C)C)CC1)OC N1(c2ccnc(NCCn3c(CC)ncc3)n2)CCC2(C)C(F)(F)C2(C)C1 c1(C(C)(C)C)cc(C(=O)N(C2CCN(C(=O)C(O)CF)C2)CCO)[nH]n1 c1(NC)cncc(C(=O)NC(CSC)C(=O)NC(C)C(C2CC2)OC)c1 c1(CC)ccccc1CNC(C1CCC(CNC(C2(COC)CCC2)=O)O1)=O c1(CC(=O)NC2CC(NC(C(C3CC3)OC)=O)C2)ccc(F)cc1 C(C)(C(=O)NC(C)CCSCC)N(CCCNC(C)=O)C.C(C)(C)C CCN=c1[nH]c(C)c(C(=O)NC2CN(C(=O)COc3ccc(F)cc3)CC2C)s1 c1(C(=O)NC(CC2CN(C3CC3)C2)C)nc(C(=O)OC)cs1.C12(CC1)C(=O)N2 N1(CC=C)CCCCC(NC(=O)Cc2ccnn2C)C1 c1(C(N(C2CN(C(C(CC#C)O)=O)C2)C)=O)cnc2n(c1=O)CCS2 C1(NC(=O)CCc2ccccn2)CCOC(CNC(=O)C(F)(F)CC2CC2)C1 c1(C(N2C3CN(c4ncc(OC)c(C)n4)CC32)=O)c(F)ccc2c1CNCC2 C(CCS(=O)(=O)c1ccccc1)NC(CCCC(OC)OC(C)(C)C)=O c1(CC)cccc(C(=O)NC2CCN(C(=O)C(COC)CC)C2(C)C)c1F C(=O)(CCC(C)(C)O)NCC(C1CCCC1)NC(c1cn(CC)nc1C)=O C(=O)(C(F)C(=O)NCC(C(=O)N1CCC(N2CC(O)C2)C1)N(C)C)OCC C1(NC(c2c(C)nccc2)=O)C(C)CN(C(=O)CN(C)CCO)CC1C C1(CCOC)(NC(=O)C(CC2CC2)OC)CCN(C(=O)C=CC=C(Cl)Cl)C1 c1(CC(=O)N(C2CC2)CC2CCCN(C(C(CSC)O)=O)C2)ccc(F)cc1Cl n1(CC)ncnc1C(=O)NC1CC(CCNC(c2scnc2C)=O)C1 c1(CC(=O)NCC2(NC(c3ncoc3Br)=O)CC2)ccc(F)c(F)c1 C#CCC(C(=O)N1CC(O)(CCNC(c2cocc2C(=O)OC)=O)C1)C1CC1 C1(NC(=O)CC2CC23CC3)CC2CCC(C1)N2C(C1(c2nc[nH]n2)CC1)=O N1(C(CC2C(CNC(CC3C(C)CCC3)=O)C2)=O)CCOCC1CO N1(C(C(C)=C2CC2)=O)CCC(CO)C(O)C1.C1(OC)CCOCC1C=O N1(C(c2c(C)cnnc2O)=O)CC2CCCC2(NC(=O)CN2CCCCCC2=O)C1 c1(C(=O)NC2CCC(C)NC2)cc2c([nH]1)CCC2 c1(O)ccc2c(c1)OCO2.c1ccc(N2CCC(c3nn[nH]n3)C2)cc1 CC(C)CCCC(C)C(=O)N1CCCC(C(N2CC(C)OCC(C)(C)C2)=O)C1 C(CC)(CCC(=O)NC1(CO)CCC(C)C1)NC(c1cccc(CC)n1)=O c1(C(=O)NC2C3CC(NC(C(C)=C4CCC4)=O)CC32)cc(C#N)ccc1C C(C1CC1)(C1CC1)=CC(=O)N(CCCOCCN(C(=O)CN1CC2CC2C1)C)C C#Cc1cccc(C(N2CCC(N(C(=O)C(C(C)C)NS(C)(=O)=O)C)C2)=O)c1Cl N1(C(C(CC2CN(C(=O)CC3CSCCO3)C2)F)=O)CCCC(F)(F)C1 c1(CC(N)C(=O)NC(C2CCCCC2)CN2CCCC2=O)ccc(Cl)nc1 CC#CCCCC(=O)N(C)Cc1ccccc1CNC(=O)CC1NC(=O)NC1=O c1(C(N2CCC(OCC(=O)NC3(CO)CC(F)C3)C2)=O)cccnc1C1CC1 Cc1sc(O)nc1C(=O)NCC(C1CC1)NC(c1cc(Cl)c(Cl)s1)=O N1(C(CN(S(CC)(=O)=O)C)=O)CC2CC(NC(=O)CCNC(C)=O)C2C1 c1(CC)c(C(=O)N(CCNC(=O)C(F)F)CC2CC2)cnc2cc(O)nn12 C1(COC)(NC(=O)C(C)C(F)(F)F)CCN(C(=O)Cn2cc(Br)cn2)CC1 c1(C(=O)NC2CC3(CN(C(C4N(C)CC(O)C4)=O)C3)C2)cc2c(cc1Cl)OCO2 c1(C(N2CC3N(C(C4C(C)C4)=O)C(CC3)C2)=O)cc(Br)c2nccnc2c1 c1(C(=O)NCC(CNC(C2C(C)OCCC2)=O)(C)O)cc(C(F)F)ccc1F Cc1cc(CC(=O)NCc2cc(C(=O)NCCCn3cnnn3)on2)ccn1 CC1CN2CCCC2CN1C(=O)CC1(NC(C2C(C)(C)C2(C)C)=O)CCCCC1 c1(C(=O)NCC2CC(NC(C(C=C)(C)C)=O)C2(C)C)cccc(F)c1C#N C1(CNC(c2c(C(=O)OC)csc2)=O)CCCCN1C(c1[nH]cc(C)c1C)=O c1(C(=O)NC(C(=O)NCCc2c(C)n[nH]c2C)C(C)(C)C)cncc2[nH]ccc12 C1(C(N2CC3(CSC3)C2)=O)(CNC(C(c2ccn(C)c2)C)=O)CCCCO1 C1(NC(C(=O)Nc2c(CSC(C)C)cc(Br)cc2)=O)CCC2(CCNCC2)O1 c1(OC)ncnc(C)c1C(N1C2CCC1(CNC(C1CCCC1O)=O)CC2)=O CC1(C)CC(CC(=O)NCC(C)(C)Cn2cc(CCS(N)(=O)=O)nn2)CO1 c1(N2CCCC(c3cc(C)[nH]n3)C2)c(C(=O)O)cccc1[N+](=O)[O-] C1(CNC(=O)CCc2ncccn2)CCCC2(CN(c3nc(Cl)ncc3Cl)C2)O1 N1(CC(N2CC(COC)N(C(c3cnc[nH]3)=O)CC2)=O)CCCC2(CC2)S1(=O)=O C1(C(=O)OC)CC(C(N2CCC(C)(CNC(C3(O)CCOCC3)=O)C2)=O)C1(C)C N1(C(c2c(CC)noc2)=O)CCOC2(CCC(NC(c3cnc(Cl)[nH]3)=O)CC2)C1 c1(C(N2CCC(NC(c3cc(C)n(C(F)F)n3)=O)C2)=O)cc2cc(O)ccc2[nH]1 Cc1[nH]c2ccccc2c1C(=O)NCc1cccc(OCCN=[N+]=[N-])c1 n1(CCC)nc(C)cc1C(=O)N(C(C)CN(C(=O)C(C(C)C)n1ccnc1)C)C c1(C(=O)NCC2(C)N(C(C(C)OC3CCOC3)=O)CCC2)ccc2c(c1)CCO2 c1(C(c2cccnc2)NC(c2ccc(C)s2)=O)nnc2n1CCCC2 N1(C(C2(OC)CC2)=O)CCn2ncc(CN(C(=O)Cc3c(C)noc3C)C)c2C1 CC1=C(C(=O)NC2CCC2NC(C2CC(n3cccn3)C2)=O)SCCO1 CC1=NNC(=O)C1CC(=O)NCCC1CCN(C(=O)C=Cc2ccncn2)C1 C1(C(N(CCNC(c2c(CCC)nns2)=O)CCC)=O)CCC(O)(CC)CC1 c1(C(=O)NC2C(C(=O)Nc3c(C(=O)OC)cc(Br)s3)C2)ccc(F)c(Cl)c1 C(CNC(c1cc(=O)n(C)cn1)=O)(CC(F)(F)F)NC(CSCC(C)C)=O c1(C(N2CCCC(NC(CCN(C)CC)=O)CC2)=O)c(C)c(C)nn(C)c1=O c1(CNC(C=CCCC)=O)ccc(CNC(c2ccc(CN(C)C)cc2)=O)cc1 CC1C2CN(C(C3CCCCC3NC(c3ccon3)=O)=O)CC12 C1(C(=O)OC)CCC(C)(C(=O)NOCC2(C)COC2)C1 Cc1cnc(N2CC(C)(c3nc(-c4cccnc4)no3)C2)nc1 N1(c2ncc(C(=O)OC)nc2)CCC2(CCCCN(C(=O)COCC(F)F)C2)C1 C1(NC(CCCCCNC(C)=O)=O)CCC12CCN(C(c1sccc1F)=O)CC2 c1(C(=O)NCC(C2CCC2)NC(c2cc(F)cs2)=O)cn(CC(F)(F)F)cn1 c1(C(N2CCC(NC(C(C(C)C)N(C)C)=O)C(O)C2)=O)cc2c(s1)CCOC2 N1(C(C=CC(C)(C)NC(CC2(COC)CC2)=O)=O)CC2C(C1)C2(C)C c1(C(=O)OC)cc(C(=O)OC)c(OC(=O)N(C(CO)C(C)C)CC)cc1C c1(C(c2n(CC)nnn2)NCCC2CCSC2)ccc(N(C)C)c(C)c1 C1(C(=O)NCC2(CNC(C3ON=C(C)C3)=O)CC=CC2)CCCCCC1 C1(CN(C(c2cnc(C)s2)=O)C)CCN(C(=O)C(CN(C)C)N(C)C)CC1 CCC(C)CCCCC(=O)N1CC(N2CCN(C(=O)CC(C)(C)C(F)F)CC2)C1 C1(NC(CCC2CCC(C)O2)=O)CC2CCC(C1C)N2C(=O)C(F)OC(F)(F)F N1(C(C(C)C)=O)CCC2(CC1)CC2CNC(C1C2CCC(=O)C12)=O C(C(COC)CC(=O)N1CCCC1CCNC(C1CN(C)C1)=O)OC N1(C(CCCC#C)=O)CC2CC3CC2C1C3NC(c1cnn(C(C)C)c1F)=O N1(C(C2CCN(OC)CC2)=O)CCC2CN(C(=O)CC(C)C)C(C)C12 C(=O)(C(C#N)CC)N1C(C(N(CC#C)CC)=O)CSC1 C(CN=c1[nH]c(=NCCSCCCN(C)C)[nH]c2c1CSC2)c1c(C)nc[nH]1 C1(C(=O)NC(C)CN(C)C(C2COCCN2C)=O)CCCCC1(C)C c1(C(N2C(CNC(C(=O)NC(C)C)=O)CC3CC32)=O)nn(C)c2ccc(F)cc12 c1(C(=O)NCC(CO)NC(C2C(CC)C2)=O)cnn2cc(C)cnc12 c1(-c2cc(C)ncc2)cnn2c1CN(c1cc(C)nc(O)n1)CC2 C(CCCC)(C(=O)NCC(C)CCC)NC(C(CC#C)C1CC1)=O C1(C(N2CCC(C#C)(O)C2)=O)CC(N=[N+]=[N-])CN1C(c1ccnnc1O)=O C(C(C)N=c1[nH]ncs1)(C1CCCC1)NC(C(C)=O)=O C1(C)(CC)C=C(C(=O)N2CCCC2CN(C(=O)C(c2cn(C)nc2C)O)CC)C1 C1(NC2(c3n(CCCF)nnn3)CCCCC2F)CC2CC3CC(C2)C1C3 S(=O)(=O)(c1ccc(Br)cc1NCC(C)Oc1ccccc1Br)NCCC1C(C)C1 c1(OC)cncc(CNC(C2OCCC2NC(c2cnc(S)nc2)=O)=O)c1 c1(CC)nccnc1C(N1CC(OC)CC1CNC(C1(COC)CCC1)=O)=O C=CCC(CC)C(=O)NC1CN(C(=O)CSCCOC)CC1(C)C CCCCC(C(=O)NCC1CCCCN1C(=O)Cc1ccn(CC)n1)N(C)C C1(CNC(C2(C(C)C)CCC2)=O)CC(O)CN1C(=O)CCCCN1CCCC1 C1(C(=O)NCCNC(C2(C#N)CC3CC3C2)=O)CC(c2ccncc2)=NO1 c1(C(=O)NCCc2scc(C)n2)cc(O)nc(C(F)F)n1 C1(=CC(=O)NCCC2(OC)CN(C(=O)CCc3cnn(C)c3)C2)CCN(C)CC1 C1(F)(C(=O)NCC2CC(NC(CCP(C)(C)=O)=O)C2)CS(=O)(=O)CC12CCC2 C(=O)(CCC(F)(F)C(=O)N1CC(OC)C(NC(=O)CC(CC)CC)C1)OCC C1(NC(c2nc(C#C)sc2)=O)CN(C(c2ccc(C)nc2O)=O)C(C)(C)C1 c1(NC(c2nc(C(F)(F)F)no2)C)ccc(S(=O)(=O)NCCCF)cc1Cl N1(C(CC(C)OC)=O)CCCC(C2CCCN(c3cc(Cl)ncn3)C2)C1 C1(COC)(NC(C2(C)CCNC2=O)=O)CCN(C(c2cc(CO)c(C)o2)=O)CC1 N1(C(C(CC=C)(F)F)=O)CCN2CCN(C(=O)C(C3CCCCC3)O)CC2C1 C1(NC(C(CC(C)C)O)=O)CN(C(C2(C)SCCCS2)=O)CC12CCC2 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1(CNC(C2N(C(C)=O)CCOC2)=O)CC1 C1(C(=O)NC(c2cc(C)on2)C)CCOCCN1C(c1cnc(N)cn1)=O c1(C(=O)NCC(C)(O)CNC(C2CC23CCOCC3)=O)cc2ccc(Cl)cc2[nH]1 c1(NC(CS(CC)(=O)=O)C)nc2ccccc2[nH]c1=NC1CCn2nnnc2C1 c1(C(c2n(CCOC)nnn2)NCc2sccc2Br)cccc(OC(C)C)c1Cl N1(C(C(CC)N(C)C)=O)CCC(C)(C)C1C(=O)NC(C)CN=[N+]=[N-] C(C)(C(=O)NCC1CN(C(C2(c3ccc(Cl)nc3)CC2)=O)C1)(C(C)C)OC CCCCCC(CC)C(=O)NC(CNC(c1cccc(C2(CC)CC2)c1)=O)CO C1(C(=O)O)CN(C(C2CCn3c(Br)cnc3C2)=O)C2(CCCC2)C1 C(=O)(NN1CCCC1C(=O)NC)C1CCCN(CCCCCC=C)C1 N1(C(C2(NC(=O)Cn3cncn3)CCC(C)(C)C2)=O)CCc2nnnn2CC1 c1(OCC(=O)NCC(CCNC(c2cncc(C)c2)=O)O)cccc(Cl)c1Cl c1(C(=O)NC(CN(C(=O)CCC2NC(=O)NC2=O)CC)C)coc(S(N)(=O)=O)c1 C(c1cccc(C#N)c1)=CC(=O)NC1CC(N(C(C=C(C)C(F)F)=O)C)C1 CCC(O)C(F)(F)C(=O)N1CCC(C)(NC(c2ccn(C3CC3)c2C)=O)CC1 c1(C(N2CC(N(C(C3CCN(C(C)=O)CC3)=O)C)C(F)C2)=O)ccc(=O)n(C)c1 C(C1Cc2ccccc21)NC(C(CC1CCCC1)NC(c1cncc(C)n1)=O)=O N1(C(c2c(C)cco2)=O)CCCC(C)(NC(C2C(C(F)(F)F)C2[N+](=O)[O-])=O)C1 C(=O)(C1=C(C)CCC1)NC1CC(N(C(c2c(OC)scn2)=O)C)C1 N1(C(CC(C)N(C(=O)C2CC2)CC)=O)CCOCC1c1ccc(C(F)(F)F)[nH]1 c1(C(=O)NC2CCN(C(C(C)O)=O)CC2CO)coc2c1CCCC2 CC(C(C)(C)NC(c1cnc(-c2ccoc2)s1)=O)NC(c1cc(C2CC2)on1)=O c1(CNC(C(C)N(C(C2CCSCC2)=O)C2CC2)=O)ccc(F)cc1 C1(C(=O)OC)CCC2(CCOCC2)N1C(=O)Cc1ccc(Cl)c(OC)c1 c1(CN2CC(c3ccc(C)cc3)OC(C)C2)cccc2c1OCO2 Cc1cc(Cl)c(C(N2CC(NC(C3CC3C(F)(F)F)=O)C3(CC3)C2)=O)cc1N C1(C(C)C)CN(C(=O)Cc2cnc(C3CC3)[nH]2)CCCN1C(C1CCSC1)=O c1(NCCNC(=O)NCC)cc(N2CCCC(C)C2)nc(COC)n1 C1(NC(C2C=CCC2)=O)CCC2(CC1)CN(C(c1cccnc1O)=O)C2 Cc1cc(-c2cn(CC3CCN3C(=O)CN(CC(C)(C)C)C)nn2)cc(C#N)c1 c1(NC(CCC)CNC(=O)C2=NOCC2)ncnc2cc(C)[nH]c12 c1(OC)c(C)ccc(C(=O)N(c2nccn2C)C)c1F CC1(CNC(=O)CN2CC3CC3C2)CCC(NC(=O)C(CO)NS(C)(=O)=O)CC1 CCC(CC(=O)NCC1CCCN1C(c1cn(CC)cn1)=O)C(C)C N1(C(C(C2CCC2)OC)=O)CCCC1C1(O)CN(C(c2ccc(CO)o2)=O)C1 N1(C(C2N(C(CCC)=O)CSC2)=O)CCC(C)(NC(=O)CN(C)C2CC2)C1 N1(C(c2c(CC)n(C)nc2)=O)CC(NC(=O)Cc2ccco2)CC12CCCOC2 N1(C(Cc2cc(C)no2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)C)C2 c1(C(=O)NCC(C)(CO)NC(C(CSC)O)=O)cnn(C2CC2)c1C N1(C(c2nc(C(=O)OCC)sc2)=O)CCN(C(=O)CS(=O)(=O)NC)CC1CF N1(C(c2c(C)c(Cl)cnc2)=O)CC(C)CN(C(=O)CCc2cnoc2)CC1C CC1CCCN(C)N1C(=O)C1CC(O)CN1C(c1nnc(CC2CC2)s1)=O N#CC1(C(N2CCC(O)(CNC(=O)C=Cc3cncc(F)c3)C2)=O)CCCCC1 C=CCCC(O)CN(C(=O)C(c1ccccc1)NC(C1(CO)CC(C)(C)C1)=O)C c1(OC)ccc(C)cc1CN1CCC(NC(C2(C3CCCO3)CC2)=O)C(C)C1 c1(C(N2CC(O)(CNC(CC3(C=C)CCC3)=O)C2)=O)oc(C(C)C)nc1C CC(C)(C)C(CC(=O)N1CCCCC1CF)NC(c1c[nH]c(C#N)c1)=O c1(C(=O)NCC2(C)CCCN2C(C2CC(F)(CO)C2)=O)cccc(=O)n1O N1(C(C2(C(C)C)CCC2)=O)CC(NC(c2cc(F)ccc2F)=O)C2(CCC2)C1 n1(CC(=O)NC2CC(NC(c3cc(CC)ncc3)=O)C2)nc(C)c(Br)c1C CC(C)CC(=O)NCC(=O)NC(Cn1ccnn1)C(=O)NCC(=O)NCCO c1(CN(C(c2cccc(F)c2I)C(=O)NC)C)ccc(Br)cc1OC c1(C(N2CC(C)C(NC(C3CC(=O)CC34CCC4)=O)CC2)=O)ccc2ncsc2c1 Cc1ccc(F)c(C(N2CCN(C(C3CN(C)CC3(C)C)=O)CC2)=O)c1O Cc1cc(F)ccc1C(=O)NC1CCN(C(=O)C(CN(C)C)N(C)C)C1C1CC1 C(=O)(C(C(=O)N(CCCN(C)C(c1ccccc1C(F)F)=O)C)OC)OC CC1CCN(C(C2CCCN(CC(F)F)C2)=O)CC1CNc1nnccc1C#N C(=O)(C1CCCn2cnnc21)NCC(CCNC(c1c(C)cc(O)cc1)=O)O CCC(C)(C)CCCC(=O)N1CCC(C)C(CNC(C2(C(C)=O)CC2)=O)C1 c1(C(=O)NC(C)C(C)NC(C2(C)CCC2)=O)cc(Br)cn2ncnc12 C#CC(CNC(C1(NC(=O)C(C(C)C)NC(N)=O)CSC1)=O)C(C)C C=CCC(F)(F)C(=O)Nc1cc(O)nc(COC(C)C)n1 c1(OC)cc(C(=O)NCCCCCN(C(=O)CC(C)CF)C)cc(N)c1OC C1(C(=O)NC(CNC(C(C(C)C)SCc2ccccc2)=O)C)CC2(CCC2)CO1 CCC(O)C(C)(C)C(=O)NCC(C)(C)CC(=O)N1CCC(O)(CN(C)C)C1 Cc1cc(C)nc(SCC(N2CCN(C(C3C4CCCC34)=O)C(CO)C2)=O)n1 c1(N(C(C2(CC=C)CN(C(=O)C(C)CC)C2)=O)CC)ccc2c(c1)CCC2 C1(NC(c2c(C)onc2CO)=O)CCC2CN(C(C3COC(=O)N3)=O)CCC2C1 C12(NC(CC(C=C)c3ccccc3)=O)CCCC(NC(=O)C(C)(C)O)(C1)C2 N1(C(c2c(OC)nccn2)=O)CC(C(=O)NCCCC2CCOC2=O)C(C)(C)C1 N1(C(c2cc(C)oc2)=O)CC(O)(C2(CNC(=O)C(C#N)C(C)C)CC2)C1 C(=O)(CCCC(CC)NC(=O)CCC1CCCO1)Nc1cnc(CCC)nc1 C1(NC(C23CCC(C)(CC2)OC3)=O)CN(C(=O)Cn2cccn2)C2CCCCC12 Cc1c(C(=O)NCC2CC2NC(=O)COC2CCOC2)[nH]c2ccccc12 C(C)(C(=O)NCC(C1CCOC1)NC(c1cscn1)=O)=C(C)C c1(OC(C(=O)NCC2N(C(C)=O)CC2)C)cccc(Cl)c1 C1(C(N2CC(OCCNC(C3CC(C)OC3=O)=O)C2)=O)(COC)CCCCC1 C1(C(=O)NCC2C(CC)C2)CC=CCC1NC(c1ccoc1C1CC1)=O C1(NC(c2cc(C)n(-c3ccccc3F)n2)=O)CN(C(C2CC2C)=O)C(C)(C)C1 C(C(=O)N=c1ccn(C2CCNC2=O)[nH]1)=CC(c1c[nH]ccc1=O)C C1(NC(C=C(C)C(C)(C)C)=O)CN(C(=O)CCCCC2CCC2)C2(CCOC2)C1 C(=O)(C1=CCC(NC(c2ccc(OC)o2)=O)C1)N(CC(F)Cl)C c1(N(CCNC(C=C(CC)C)=O)C(=O)NC2CCCC2)cc2ncc(C)cn2n1 CC#CCCCC(=O)NCCC1(NC(=O)Cc2c(F)cncc2Cl)CC1 C(CC(CNC(=O)CCc1ccsc1Br)NC(=O)COCCF)OC c1(OC)ccc(N(C)C(C2(NC(=O)C(C)CN(C)C)CC2(C)C)=O)cc1 c1(CSCCC(=O)NC2(F)CCC(NC(=O)CCOC3CC3)C2)ccccc1F c1(Sc2c(C)c[nH]n2)ccc(CC(=O)NC(c2cn(C(C)C)nn2)C)cc1 C1(NC(=O)NCCNc2cc(F)c(Br)cc2Cl)C2Cc3c(Br)cccc3C12 Cc1nccc(C(N2CC(NC(=O)C(C)(C)c3ccno3)C(C)C2)=O)c1C N1(C(C23N(C(c4cnco4)=O)CC(C2)C3)=O)CC2C3C=CC(C3)C2C1 c1(CC)cc([N+](=O)[O-])ccc1C(=O)NCC(C)N(C(=O)C(C)(C)O)CC C(C(C)(C)CC(=O)N1CCOCC1CN(C(=O)C(N1CCN(C)CC1)C)C)OC C1(CNC(CC=C)=O)CC(C(F)(F)F)CN1C(=O)COC1CCN(C)CC1 C12(NC(c3c(C)n(C)cn3)=O)CCC1CN(C(c1ccn(C(C)C)c1C)=O)C2 c1(N2C(C(C)(C)NC(CC(CC)C(C)C)=O)CCC2)ncc([N+](=O)[O-])cc1F C(=O)(C(O)CCC(C)C)N1CCC(C2N(C(c3c(C)noc3)=O)CCC2)CC1 c1(OC)ccc2c(c1)CCC(NC(=O)C1=C(Cl)CCCC1)C2=O C#CC1(O)CC(C(=O)NCc2occc2C(=O)NCC(c2cnn(C)c2)O)C1 CC1CC(CCNC(=O)CC(C)(C)N(C(=O)CCc2ccco2)C)CCO1 CCC(CC(=O)NCCC(C)NC(c1ccc(OCC(F)(F)F)cc1)=O)C(C)C C#Cc1cncc(C(N2CC(NC(=O)CNC(C)=O)CC2(C)COC)=O)c1 CC#CCC(C(=O)N1CCC1(C)C(=O)OC)NC(c1c[nH]cc1C)=O c1(C(=O)NCC2CCC(NC(CC(C)n3cccn3)=O)C2)ccc(F)c(C#N)c1 c1(C(=O)NC(CNC(Cc2cn(CC)nc2)=O)C)ccc(OC(F)F)nc1 c1(OC)ccc(C(=O)NC2CCCC(C(=O)NCC(n3ccnc3)C)C2)cc1 N1(C(Cn2ncn(C)c2=O)=O)CC=C(CCNC(C2COCCO2)=O)CC1 C=CC1(C(N2C3CCC(C3)C2C(=O)NCC2(CCOC)CCC2)=O)CCOCC1 CC(C)C1=NOC(C(=O)NCCCC(O)C(=O)NCC(F)(F)CO)C1 C(N=c1nc2c(c[nH]1)CCC2)C1OCCN(C(c2ccc(C)c(F)c2)C2CC2)C1 N1(C(CS(CCC)(=O)=O)=O)CCOC2CN(C(c3cc(F)cc(F)c3N)=O)CC12 C12(C(N3CCC(CCOCC)C3)=O)CC3CC1C2C3O.C12(CC1)C(=O)NC2 C1(NC(=O)C(C)O)CCC2(CC1)CC2.Cc1nsc(NCC)c1C(=O)NC1CC1 Cc1cc[nH]c(=N)c1C(=O)NCCC1CCN(C(=O)CCCOC(C)C)CC1 c1(C(C)C(=O)N(C)CC2CCCCN2C(=O)CCC(F)F)cc2ccccc2s1 C1(O)(CC(=O)NCC(CC)NC(=O)COC2CCOCC2)CCOCC1 N(C(=NCCCCl)NCc1ccc(C(N)=O)o1)CC1C(C)C1 C1(CNC(C(CCC)O)=O)CCCN(C(=O)CCc2ccc[nH]2)CC1 c1(C(=O)NCC2C(CNC(Cn3ncc(C)c3)=O)C2)ccc(C2CC2)cc1 CC1CCCN(C(=O)C(=O)NCC2C3CC2N(C(=O)C(F)(F)C2CCCC2)C3)C1 C1(NC(c2c(C)cc(F)c(Cl)c2)=O)COC2(CCCN(C(=O)C(C)(C)O)C2)C1 Cc1n[nH]c(C)c1CC(=O)NCCOCC(=O)NCCCCS(C)=O c1(C(=O)NCCCN(C)C(C2CCCN2C(=O)C2CC2)=O)c(F)cncc1F c1(C(=O)NCCCNC(Cc2c(C)non2)=O)cccc2c(O)nncc12 Cc1ncc(C)c(NC2(CNC(C3CC(=O)N(C(C)C4CC4)C3)=O)COC2)n1 N1(C(CN(C)C(C2CC(CC(=O)OC3CC3)C2)=O)=O)CCc2ncsc2C1 N1(C(C(CC)=CC)=O)CC2CCCC2(CNC(C2CC(=C3CCC3)C2)=O)C1 N1(C(CN(C)CC)=O)CCC1(C)CC(=O)NC(C)C(=O)OC(C)C c1(C(=O)NC23CC(C(=O)NCc4cncc(Cl)c4Cl)(C2)C3)ccc2ncnn2c1 C1CCCCC1NC(CN(CC)CC)=O.C(C)CN(C(=O)CN(C)C(N)=O)C c1(C(=O)NC23CC2CN(C(=O)CCCCc2cnn[nH]2)C3)cn2ccccc2n1 C=CCCCCCCCCC(=O)NCC(=O)Nc1nc(C2CC2)c(Br)s1 c1(C(N(CCNC(C(CC)N(C)C)=O)C)=O)sc(C2CCCOC2)nc1C n1(CC(N2CC(O)(CCNC(=O)C3=CCCO3)C2)=O)ccc2ccccc12 Cc1sc(C(N2CCC(C)C2(C)C)C(=O)NC)c(C)c1C N1(C(C2N(C(C)=O)CCOC2)=O)CCCC(O)(CNC(c2ccc(C)nn2)=O)C1 C1(CCC=C)CN(C(c2ncccn2)=O)CCN1C(=O)CC(=O)OC(C)(C)C Cc1ccc(Br)cc1NC(c1nnnn1C1CCC1)(C)Cn1ccnc1C c1(C(=O)N(c2nc(C)c(C(=O)NC3CC3)s2)C2CC2)[nH]nc2c(=O)n(C)cnc12 C12(NC(c3cnc4sccn34)=O)CCCC1N(c1ncccn1)CC2 C=CC1(CC(=O)NCC2(O)CCOC2C)CN(C(c2ccc[n+]([O-])c2)=O)C1 C1(CNC(=O)Cc2cccc(Cl)c2)CN(c2ncncc2Cl)CCCO1 C1(C(=O)NCc2n(C(C)C)cnn2)CC(=O)CN1C(=O)C(C)CC1CC1 c1(C(=O)NCC2(C(=O)NC(C)Cc3nc[nH]n3)CCCO2)cccc2c1CCC2 C#CCCCC(=O)N1CC(NC(=O)CN(C2CC2)CC)CC1C c1(OC)ccc(C(CNC(=O)CC2CCN(C)C2)NC(=O)CC(C)C)cc1 CC1(C(N2CC(NC(c3cnn(C(F)(F)F)c3)=O)C3(CC3)C2)=O)CCC(=O)NC1 C(c1ccccc1)=C(OC)C(=O)NCCCCNC(=O)C(C)(O)C1CCOCC1 c1(C(C)NC(C(C)(C)SC)c2nnnn2C2CCCCC2)cc(Cl)ccc1O c1(C(N2CC(COC)(CNC(=O)C=C(C3CC3)C3CC3)C2)=O)cccc(N)c1F C1(CNC(c2n(CC)nnn2)(C)COC(C)C)CCSC1(C)C c1(NC(=O)CC2CCCN2C(c2cc(F)c[nH]2)=O)cccc(F)c1O N1(C(Cc2n[nH]c(=N)s2)=O)CC2CC(NC(c3ccn(C4CCC4)n3)=O)C2C1 C1(CNC(C(C)C2CCC2)=O)CCCC2(CN(C(c3cccn(O)c3=O)=O)C2)O1 C(=O)(C1COc2ccc([N+](=O)[O-])cc21)N1CC(NC(c2n(CC)ncc2Cl)=O)C1 Cc1oc(C2CCOCC2)nc1C(=O)NCC(F)CNC(C1CC=CCC1)=O C1(C(=O)NC(C)CN(C)C(c2ccc(N)cc2Cl)=O)(OCC)CCC(F)(F)CC1 c1(NCC(=O)NCC2COCC2NC(=O)CN2CCSCC2)cccc(O)c1 N1(C(C2CC(C)C2)=O)CCC2(C1)CN(C(=O)C(C1CCCCC1)N(C)C)C2 C1(C(=O)Nc2c(SC)cccn2)CCC(C)N(C(=O)Cc2scnc2C)C1 CC(C)(F)CCC(=O)NC1(CF)CCN(C(=O)CONC(=O)OC(C)(C)C)C1 C1(C(=O)NC2CCC(CC)CC2)CC(N=[N+]=[N-])CN1C(c1nonc1C)=O C1(CCNC(C(CC)(C)CC)=O)CC2CCC(C1)N2C(C1CNC(=O)N1)=O C1(CCCCNC(CC2C(C)C2)=O)CCN(C(=O)CCc2cnn(C)c2)CC1 C1(C(=O)NCC2CCN(C(=O)CC=C(Cl)Cl)C2)C2C3CC4C1C1C2CC3C41 N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(c2cc3scnc3[nH]2)=O)CC12CCCC2 c1(C(C(C(C2CCC(C)NC2=O)=O)C#N)=O)cccc2cc[nH]c12 CC1(C)CCCCC1=CC(N1CC2CC1CN2C(=O)C(F)(F)CC1CCCO1)=O c1(C(N(CC(CN(C(=O)Cc2ccoc2)C)O)C)=O)cc(C2CC2)on1 CCC(CNC(=O)C(CNC(c1cnn(C)n1)=O)CC1CC1)CCO CC1CC(NC(=O)CCn2ncn(C)c2=O)CCN1C(c1ncccc1N)=O C(=O)(C#CC1CCOCC1)N1C(CN(C(C=CCOC)=O)C)CCCC1 N1(C(C2CCCN2Cc2ccccn2)=O)CC(CO)C(C2CCOCC2)C1 c1(CCNC(N2CCC(n3nncc3I)CC2)=O)cc2ccccc2s1 CCC(C)(C)CC(=O)NCC1CN(C(c2nnn(C(C)(C)C)n2)=O)CCC1C CCCCCCC(C)c1nc(C(C)OCC)nn1-c1cccnc1 C1(C(N2C(CCNC(c3cc(F)n(C)n3)=O)CC(OC)C2)=O)CCCC2(CC2)C1 C1(CC)CCCC(CNC(=O)CC2C=CC(NC(c3coc(C(N)=O)c3)=O)C2)C1 C1(NC(C2CCCC3(C2)CC3(F)F)=O)CC1C1CCCN(c2nc(C3CC3)ns2)C1 c1(CCNc2cc(N3CC4C(C(C)C)(C4)C3)ncn2)ccc2c(c1)CC(C)O2 C1(CNC(C=CC=CCC)=O)COCC2(CCN(C(c3coc(Cl)n3)=O)C2)O1 CCN=c1[nH]c(C)c(C(=O)N(C)CC2CCN(C(=O)C(C)(C)C(C)O)C2)s1 c1(C(N2CC(O)CC2c2ccc(F)cc2)C(=O)NCCC2CC2)ccccc1Br N1(C(c2c(C#N)cn[nH]2)=O)CC2CCCC(C1)N2C(c1ncccc1Cl)=O C1(CC(=O)N(C)CCNC(c2ccc(C(F)(F)F)o2)=O)CC(O)C1(C)C C1(F)(CNC(c2nc(CCC)sc2)=O)CCC(CNC(=O)CC2CC3CC3C2)C1 CC(C)C(C(=O)NC1CCCC1CNC(=O)C(F)(F)c1ccncc1)N(C)C N1(CCNC(c2c(CC)onc2C)=O)CCCN(C(=O)C(O)C(F)F)CC1 c1(CCC(=O)N(CC(C)N(C(c2cnc(OCC)s2)=O)C)C)cccc(F)c1F C1(C(=O)NC2C(NC(c3ccc(C)nc3)=O)CCOC2)CC(C)(C)OC1(C)C c1(C(N(C2CCCN(C(=O)C(F)OC(F)(F)F)C2)C)=O)cccc(-n2cnnn2)c1 CC(C)C(CCC(=O)NCc1c[nH]c2cccnc12)NC(=O)C(O)CC1CC1 c1(C(N2CC(=O)O2)=O)ccc(CCCC#N)cc1.C=CCCSCC C=CCCCCC(=O)NCc1ncoc1C1CN(C(c2cccc(F)c2)=O)C1 C1(CC)(NC(=O)CCOC)CCCN(C(=O)C(C)Sc2ccc(F)cc2)C1 c1(CNC(c2c(CC)ocn2)=O)ccccc1CNC(c1ccn(CCF)n1)=O c1(C(=O)NC2CCCN(C(C)=O)C2)ccc(OC2CC2)cc1Cl N1(C(C2C(=C)C2C(=O)OC)=O)CC2C(CN(C(=O)CN3CCSCC3)C)C2C1 c1(CC)cccc(C(N2CCC(O)(CNC(c3ccnnc3S)=O)C2)=O)c1F CCC(CNC(C1CC(N(C)C(c2ccn(C3CC3)n2)=O)C1)=O)C(C)C C(=O)(C1=CCCCC1C)NC1CCC(C(=O)NC2(CC=C)CC2)CC1 C1(CC(F)(F)F)C(=O)N1.c1(NC(C(=O)NCCCO)=O)cccc(C(F)(F)F)c1 C1(NC(C2(COC)CC2)=O)CN(C(=O)COc2cccc(Br)c2)C2CC12 c1(CC(=O)NC2CCCCC2NC(C2(F)CC=CC2)=O)c(Cl)cccc1Cl Cc1cc(C(N2CCC(C)C(NC(c3ncccc3F)=O)C2)=O)c(O)nc1C C1(NC(C2C(=C)CC2)=O)CCN(C(c2cccc(C(C)(F)F)c2)=O)CC1F CCC(CC(=O)NC1C(C)CCN(C(c2ccc(COC)o2)=O)C1C)C(C)(C)C N1(C(C2CN(CCC)C(=O)C2)=O)CCN(C(=O)C2=NNC(=O)CC2)C(C)CC1C C(=O)(C(F)(CNC(c1[nH]c(C)nc1CC)=O)C(C)C)NC1C(C=C)OCC1 c1(CC)[nH]nc(C(=O)NC23CC(C2)N(C(c2ccccc2C(N)=O)=O)C3)c1C C1(C(CNC(c2nc(C)oc2)=O)(C)C)CCN(C(=O)Cc2cn(C)nn2)CC1 C(CCC(=O)NCC1C=CCN1C(=O)COC1CCOCC1)N(C)C c1(SC)cccc(C(=O)NCCC(O)CNC(=O)COc2ccsc2)c1 c1(C(=O)NCC2N(C(C(C(C)C)SC)=O)CC=C2)cn(C)c(=O)n(C)c1=O N1(C(c2c(-c3n(C)cnc3)csc2)=O)CC2(CC(CO)CO2)C1 c1(CC(N2C(C3(NC(C(CC)N(CC)CC)=O)CC3)CCC2)=O)cccnc1O N1(C(C(c2c(C)nn(C)c2)C)=O)CCC(C)(C)C(NC(=O)C=Cc2cncs2)C1 C(=O)(CCCS(N)(=O)=O)N1CC(C)(CNC(=O)C#CC2CC2)OCC1 C1(CC)C(=O)N(C)CCN1C(=O)C(C)(CSC)NC(C1CC2(CC2)C1)=O c1(C(=O)NC2C(NC(c3c(OC)cncc3)=O)CC2)cc(C)nc(O)c1[N+](=O)[O-] C(C(CC(C)(C)C)C(=O)O)NC(CC1CC(CC)OCC1)=O N1(C(C23OC(C)C(C2)C3)=O)CC2(CCN(C(c3cc(C4CC4)nn3C)=O)C2)C1 c1(C(N(CC(CC)NC(=O)C(O)c2ccsc2)C)=O)c(C)ccc2nsnc12 N1(C(C(C)(C)OCC)=O)CC2C3CCC(C2C1)N(C(=O)CCc1ccccc1)C3 N1(C(C(CC)C)=O)CCOCC(C(=O)NCCCCC(C)(C)C)C1 c1(C(C)NC(=O)C(C)(C)n2cnnn2)ccc(CNC(=O)CC=CC(C)(C)C)cc1 c1(C(=O)NCC2CC3N(C(C(C)C4CC4)=O)C(CC3)C2)c(F)ccc2n[nH]cc12 N1(C(C(C)OCCCC)=O)CC(NC(C23C4CC(CC24)C3(F)F)=O)CC(C)(C)C1 N1(C(c2c(C)c[nH]n2)=O)CC2CCN(C(c3cccc(CF)c3)=O)CCC2C1 N1(C(C(=CC2CCCC2)C)=O)CCC2(CC1)CC2NC(=O)CCc1ccncc1 C(=O)(CC(O)CC(C)C)N1CC(CC(N2CCC(C=C)C2)=O)OCC1 c1(CC(CO)NCCCN(CC(F)(F)F)C(=O)OC(C)(C)C)ccc(O)cc1 C1(C(N(C)CC2(O)CCC2)=O)(NC(c2ccccn2)=O)CC(O)C1 c1(C(=O)NCCN(C(=O)Cn2cc(Br)cn2)CC)ccc2c(c1)N(C)C(=O)CC2 c1(OC)ccc(CN2CCC(CC(=O)NCCc3cccnc3)C2)cc1C c1(CC=C)ccccc1C(=O)NC(C(=O)NCCCOC1CCC1)C(C)C C=C(C)C(C)(C)C(=O)N1CCC(C(=O)NCC2(COC)CC=CCC2)C1 c1(NCCCc2c(C)cccc2)nc(C)nc2sc3c(c12)CCC3 N1(C(=O)Cn2cc(C3CC3)cn2)CCN(C(=O)Cc2nncs2)C2CCCCC12 C=CCC(CC(=O)NC1(C)CCOC1=O)NC(c1cc(=O)n(C)cn1)=O c1(C(=O)NCC2C(CC)C2)ccc(Cn2cc(C3C(C)(C)C3(C)C)nn2)cc1C N1(CCCC)CCCCC1C(=O)NCC(CO)NC(c1ncsc1C1CC1)=O C(CCC(C)C)(C(=O)NC(C)CCSCC)NC(C(C)(C)OCCC)=O CN1CCC(C)(C(N2CCC(C)(CNC(c3cnc(O)o3)=O)C2)=O)C1=O CCCCC(CC(=O)N1CCC(CO)C1(C)C)NC(=O)CC1OCCCO1 C12(CC(N3C(CN(C(=O)C(C4CCCCC4)O)C)CCC3)=O)CNC(=O)C(C1)C2 C1(C(N2CCC(O)(CNC(c3cc(=O)cc[nH]3)=O)C2)=O)CCC2(CCC2)CO1 C1(NC(C(C)(Cl)Cl)=O)CCCC12CN(C(=O)CCCc1ccc(F)cc1)C2 c1(C(=O)NC(CN(C(C(C)OCCCCCC)=O)CC)C)cnc(C)n1C(F)F Cc1cc(Cl)cc(NC(C2CCOC2c2c(C)n[nH]c2C)=O)c1O CC1(C)CCC(CC(=O)NCC23CC2CN(C(c2cc(C(N)=O)c[nH]2)=O)C3)O1 N1(C(CC2C(CC)C2)=O)CC2CC(C1)N(C(c1ccc(Cl)c(C(F)(F)F)c1)=O)C2 C1(COc2ccnc(OCCO)n2)CCCCC12CC2 C1(NC(c2cc(C)n(C)c2)=O)C2CC3C(C2)C13C(=O)NC1CCC(C)(C)C1 CC(C)(C(=O)NCC1CCCN1C(c1cn(CC(N)=O)nn1)=O)n1cnnn1 Cc1cnc2cc(C(N3CC(=C(F)CNC(C4CCCS4)=O)C3)=O)ccn12 N1(C(C2CC(O)(CNC(C3(CC(C)=O)CC3)=O)C2)=O)CCN2CCCC2C1 c1(C(N2C(C)C(NC(=O)C(=O)NCC3CC3)CC2)=O)cc([N+](=O)[O-])c[nH]1 N1(C(c2ccc(CNC(C)=O)o2)=O)CC(C)CN(C(=O)Cn2cnnn2)CC1C c1(C(=O)NCCC2(C)CCN(C(C(CSC)C)=O)C2)ncc(F)cc1F N1(C(C(F)=CCC)=O)CCN(C(=O)CSC(C)C)C(C2CC2)C1 C1(NC(C=CC=CC)=O)CCN(C(c2ccccc2C(F)(F)F)=O)CC1(C)C.C1CC1 C1(NC(c2ccc(OC)s2)=O)CC2CC(NC(=O)Cc3cccc(C)c3)CC2C1 N1(C(c2cccc(OC)c2)=O)CCCC(O)(CC(=O)NC2CCCC2C2CC2)C1 C(=O)(CCCCC(C)(C)C)N1CC(C(C(N2CCC(C#C)(O)C2)=O)O)C1 C1(C(N2CC(NC(c3c(OC)cccc3)=O)C(C)C2)=O)CCC(F)(F)CO1 c1(NC(C(C)NC(c2ccc(N)cc2)=O)=O)cc(C(N)=O)cn1C c1(C(N)=O)ccc(SCC(N2CC(C(O)C(=O)NCc3csc(O)n3)C2)=O)cn1 Nc1cc2c(cc1C(=O)NC1(CCNC(C3CCC(F)CC3)=O)CC1)OCCO2 N1(C(C2CCN(C)C2)=O)CCC2(CC1)CN(C(c1cc3c(cc1O)OCO3)=O)C2 C(C1CCCc2ccccc21)NC(c1c(C)sc(Br)n1)c1nnnn1CCSC N1(C2CCN(C(C(C)N(C)C)=O)C2)CCC(NC(c2ccn(C(F)F)n2)=O)CC1 CC(C)CCC(C)N(C)C(C1CN(C(c2cccc(O)n2)=O)C1)=O.NC c1(SCC(=O)N(CCCC)Cc2ccccn2)ncccc1Cl N1(C(CCOCC)=O)CCC(N(C(=O)C(Cc2ccccc2)C2CC2)C)C1C N1(C(C(c2c(C)noc2C)CC)=O)CCN(C(=O)C=Cc2ccoc2)C(C)C1 C(=O)(C(C)(C)C(C)NC(C1C=CCS1)=O)N(C(c1ccccc1)C)CC N1(C(=O)COc2ccc(F)cn2)CCC2C(CCN2C(c2cnc(Br)s2)=O)C1 N1(C(c2c(C(C)(C)C)con2)=O)CC2(CNC(C3(S(C)(=O)=O)CC3)=O)CCC1C2 Cc1cc(C#N)cnc1N1CCC(NC(=O)CCNC(=O)CO)C(O)C1 CON(CCC(=O)NCC1CC(C)(C)CCO1)C(=O)C1CC(=O)OC1(C)C CC(O)C(C)CN=c1nc(N2CCN(C3CCOCC3)C(=O)C2)c2c([nH]1)CCC2 Cc1csc(C(N2CC3CC2(CNC(c2cnn(C)c2)=O)C3)=O)c1Br CC1(C)COCC(CC(=O)NC2CC3(C2)CC3NC(c2cnccn2)=O)O1 C1(C)(C(=O)NCCCCN(C)C(C2CC(C)(C)C2C(F)(F)F)=O)CNC(=O)C1 C1(C(=O)NC(C(C)C)CN2CCCC2)CNC(=O)CN1C(=O)CN(C)C c1(NC(C2C(NCc3oc(C)c(Br)c3)C2)=O)cnc2ccccc2c1 C1(C(=O)OC)CCCN(C(C2CC(OC)CN2C(c2cc(C3CC3)no2)=O)=O)C1 c1(C(=O)NCC2CN(C(COc3cc(C)on3)=O)C2)nccnc1CC(F)(F)F N1(C(C(CCSC)O)=O)CCC(NC(C2(NC(N)=O)CC2)=O)C2(CCC2)C1 N1(C(c2ncc(C)s2)C(=O)NCCC#N)CCc2ccc(N=[N+]=[N-])cc2C1 c1(C2(C(N3CCC(N(C(c4cc(C)ncc4)=O)C)C3)=O)CC2)ccnc(Cl)c1F C12(C(N3CCC(CNC(C4CCC(=O)NC4)=O)CC3)=O)CCCC1OCC2 c1(C(=O)NCCC2CCCN(C(C(C(C)O)(F)F)=O)C2)cnn2c1NCCC2 CC1=NOC(C)(C(=O)NC2CN(C(c3c[nH]nc3C3CCC3)=O)CC2O)C1 C(CN=c1nc[nH]c2c(C)cccc12)c1nnc(C)n1C N1(C(C2C(OCC)C2C)=O)CCC2(CC1)CN(C(c1nnn(C)c1C)=O)CC(C)O2 Cc1c(C(=O)NC2CCC2NC(=O)Cc2ccccc2CC(N)=O)cncc1Cl c1(CC(=O)NCC2(CNC(CC3(CC(=O)OC)CC3)=O)CCC2)cc(C)no1 C(C#CC(C)NC(C1CCCCC1CNC(=O)OC(C)(C)C)=O)(OC)OC C(C(CO)(CO)N(C)C)N(C(=O)C#CC(=O)N(C)C)C.C1(=O)C(O)CN1 N1(C(CN(C)C=O)=O)CCN(CC2CC2)CC1.N1CC(C=O)C1.C(N)(=O)NC C1(OCCNC(C=CCC)=O)CCN(C(=O)C(c2ccccc2)CN=O)CC1 c1(CNCc2c(OC)cc(OC(F)(F)F)cc2)ccc2sncc2c1 C1(NC(c2cc(-c3ccco3)[nH]n2)=O)C2CCN(C(C3CCCC3)=O)C12 CC(C)C(C)(CNC(C1CC12CCC2)=O)NC(c1ncncc1Cl)=O N1(C(c2c(CCC)nco2)=O)CCC(CF)(NC(=O)C=CC(=O)N(C)C)C1 C1(OC)CN(C(c2cc(C(O)C(F)(F)F)ccn2)=O)CC1NC(=O)C=CSC N1(C(C2(OCC=C)CCNCC2)=O)CC=C(c2ccc(C3CC3)cc2)C1 FC1(F)CCCC(N=c2[nH]c(N3CCC4(CCCO4)CC3)nc3c2SCC3)C1 c1(CSCC)ccc(C(N2CC(NC(=O)CC3(C)CC3(F)F)C2)=O)cc1.C1CO1 C(C(C)C(=O)NC(C1CCCC1)CNC(c1cnc(C(C)C)s1)=O)OC N1(Cc2c(Cl)ccc(OC)c2)CC2CCN(C(c3ccc(CC#N)cc3)=O)C2C1 CCCS(=O)(=O)c1ccccc1C(=O)NC1CCC(C)N(C(=O)C(C)C(=O)OC)C1 C1(CNC(C=C(C)c2ccco2)=O)CC(C(=O)NC2CCCC2CCO)=NO1 C1(C(=O)NCCC2(CNC(C3(CC4CCC4)CC3)=O)CC2)CCS(=O)(=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NC2C3CN(C(=O)CC4CCC(=O)NC4)CC23)n1 c1(SC)nocc1C(=O)NC1(CCCNC(c2sccc2F)=O)CC1 CN1CCCC1C(N1CC(CCCCNC(C2(Cc3cccnc3)CC2)=O)C1)=O c1(C(=O)NC2CC(CNC(C3(C)CC3(F)F)=O)C2)cc(C(F)(F)F)ncc1Cl C(C)(CO)(C(=O)NC1CC1(C)C(F)F)NC(CC1(OCC)CC1)=O C1(CNC(C2(CC)CCCO2)=O)CCN(C(c2cnc(O)n2C)=O)CC1C CC1CN(C(=O)Cc2csc(C3CC3)n2)CCC1CNC(C1(C2CC2)CC1)=O c1(C(=O)NCC(CNC(C2(C)COC2)=O)F)ccc2[nH]c(=N)[nH]c2c1 C(=O)(C(O)CCCNC(C1CN2CCC1C2)=O)NCc1cnc(CSC)[nH]1 c1(CN2C3(CN(CCN(C)C)C)CC3CC2)cc2ncccc2[nH]1 c1(NC(CCN(C(C(CCC)NC(N)=O)=O)C)C)ncnc2c1nnn2C1CC1 Cc1cc(C(N2CCC(CCNC(C3CCCS3)=O)C2)=O)ncc1Cl N1(C(c2c(C)csc2)=O)CCN(C(=O)C(c2ccccc2)C)C(CCO)C1 C1(CC(=O)NC(CNC(c2ncc(OCC)nc2)=O)CO)CCCC2(CC2)C1 O=C1Cc2c(C(=O)NCC(c3ccccc3)NC(=O)CCF)cccc2N1 c1(-c2n(C(COC)C)nc(CC3CC3)n2)cc(Br)cn(CCl)c1=O S(=O)(=O)(c1ccc(N2CC3CC3C2)c(Br)c1)NC(c1cccnc1)COC C1(NC(=O)CN2CCCC2=O)CCC2(CC1)CN(Cc1ccc(Br)cc1O)C2 c1(CCC)cc(C(=O)NC(CNC(c2cnc(Cl)s2)=O)C2CC2)ccn1 N1(C(C(C)OCCOC)=O)CCC(C(C)C)CC1CNC(c1cc(C#N)c[nH]1)=O C1(CC(=O)N(C(C)C)CCNC(C2CC(=C3CC3)C2)=O)SC(=N)NC1=O S(=O)(=O)(c1cc(Cl)cc2cccnc12)N1CCN(CC)C(C)C1 N1(C(c2nc(CCC)oc2)=O)CCCC12CCN(C(=O)C(O)CCC)C2 c1(C(N(CCCNC(=O)C(=O)NC2CCCCC2)C)=O)ccc2c(n1)CCCC2 c1(-c2nccc(C(=O)NC3CC(F)(F)C3(F)F)c2)ccc2c(c1)CNC2.[nH]1cccc1 CCCCCCC(=O)N1CCC(C(C)NC(=O)CCc2ccon2)C1 c1(OC)ccc(Br)cc1C(=O)NC1(F)CCCN(C(c2ncn(C)n2)=O)C1 S(=O)(=O)(c1ccc(NC2CCS(=O)CC2)cc1Br)N(C)Cc1cc(F)ccc1Br C(=O)(C1=C(SC)CCCC1)N1C(CN(C(CN2CCCC(CC)C2)=O)C)CCC1 CC1CN(C(C2(F)CCOCC2)=O)CC(C)C1NC(c1cc(F)cc(F)c1O)=O c1(C(N2C(C(=O)NC(CC)CNC(=O)C=C(C)C)CC(O)C2)=O)c(Cl)cccc1Cl CCC(CC(=O)N1CC2C(CC(=O)NCC(C)(O)CO)C2C1)C(F)F c1(NC2C(C)CN(C(c3ncccn3)=O)C2)ncnc2c1nnn2C c1(C(=O)NCCN(C(=O)C(O)CSC)CC)cc2c(C)c(C)ccc2[nH]1 C=CC(C(=O)NCC1(C(=O)NC(CC)CCOC)CCCC1)OC C(=O)(CC1COc2cc(OC)ccc21)Nc1cc(C(=O)NCC)cc(F)c1 CCCCC(F)C(=O)N(C1CCCC1)CCNC(=O)C(c1ccc(=O)n(C)c1)(F)F C1(CC(=O)NC2CN(C(CCCN(C(C)C)C)=O)C2)CCN(C(C)=O)CC1 c1(N2CCC(C)(CC#N)C2)ccc(Br)c(S(=O)(=O)N2CCC(N3CC(O)C3)C2)n1 c1(CC)ncc(C(=O)NCCn2cc(C(N3CCCC3C3(C)CC3)=O)nn2)cn1 C1(c2onc(C)n2)CN(C(=O)CCc2ccc(Br)cc2Br)CCN1C C#Cc1cccc(CC(N2CCC(C)C2C(N2CCC2(C)C(=O)OC)=O)=O)c1 C1(NC(C23C(CN(C(CCNC(COC)=O)=O)C2)C3)=O)CCN(C)CC1C Cc1cc(Br)ccc1C(=O)NC1CC(NC(=O)Cc2cc(F)ccc2O)C1 C(=O)(CS(=O)CC)N.C=CCC1N(CCO)CCC(=O)C1CC c1(C(N2CCC(C)(NC(=O)Cc3ccccc3O)C2)=O)nnn2c1CCCC2 c1(N2CCC(NC(=O)COCC3CCCCO3)C(O)C2)nc(Cl)nc2c1CCC2 C1(CNC(C(CC=C)(C)C)=O)C2CCCC1N(C(=O)CC1(C)CC1(F)Cl)C2 N1(C(C)=O)CCCC(C(=O)NCCOC2CN(C(=O)C(n3ccnc3C)C)C2)C1 C1(C(=O)NCc2c(C(N(CCC(O)CO)C)=O)[nH]cc2)CC(=O)CC(=O)C1 N1(C(C2C(O)CCN(CC3C4CN(C)CC43)C2)=O)CCN2CCN(C)C(=O)C2C1 C(=O)(C(C(=O)N1CC2C(NC(c3cc(C(C)C)no3)=O)C2C1)C(C)(C)C)OCC N1(C(c2cncc(SC)c2)=O)CC(C)C(C)(CNC(=O)CN2CC(=O)NC2=O)C1 C#CCCCCCC(=O)NCc1nnn(C)c1C(=O)Nc1ccc(N=[N+]=[N-])cc1 N1(C(CCCC)=O)CCCC(O)(CNC(=O)CCCc2ccccc2Cl)CC1 C1(NC(C(C)NC(N)=O)=O)CCCCN(C(=O)C(F)C(F)(F)F)C1 CCC(CCCO)NC(=O)N(C)CC1CC1(F)F Cc1cc(OCCC(=O)NCCCC2(NC(=O)C(C)O)CC2)c(C)c(C)c1 C(=O)(C(F)CC(C)(C)NC(=O)CC(O)C(C)C)N(CC(=O)NC)C C(=Cn1cc(CN)nn1)c1cnn(C)n1 c1(C(N2CC(C)C(NC(=O)COCc3ccccn3)C2)=O)c(O)ccc(Cl)c1O N1(C(Cc2c(C)noc2C)=O)CC(NC(=O)C(C)N(C)C)C2(CCC2)C1 N1(C(C2(C)CCOCC2)=O)CC2COCC(C1)C2NC(=O)C(F)=C1CCCC1 CCC(O)C(=O)NCCN(C(C1CCCC1OC)=O)CC C(=O)(C(F)CCC(C)(C)C)NC(c1cccc(C)c1)CNC(=O)CC1CC1(C)C C1(C(C)NC(Cc2scc(C)c2)=O)CN(C(C2CC(C(C)C)C2)=O)CCO1 c1(NC(C(Cc2cn[nH]c2)NC(C(CC2CCC2)OC)=O)=O)cc(Cl)cnc1O c1(C(N2C(C)CC(NC(C(CC(=C)C)NC(C)=O)=O)C2)=O)cnc2ccccn12 CCCC(C(=O)NC(CC)C(=O)NC)NC(C1CC(C)(O)C1)=O C=CCCCCCC(=O)N1CCC(C(N2CCCC(C#N)C2)=O)C1CC c1(CCC(=O)NCC2CN(Cc3ccc(OC)cc3)C2)ccc(F)c(C(=O)O)c1 c1(OC)ncnc(C(=O)NC2(C)CN(C(C3CCOC3=O)=O)C2)c1F C1(O)(C(C)NCC2C3COCC23)CCN(C(=O)C=C(C)c2cccs2)C1 c1(N2CCN(C(CC(CC)C3CC3)=O)CC(O)C2)nc2cccc(F)c2o1 N1(C(C(C)OCCOCC)=O)CCC(CNC(c2cnc(O)c(F)c2)=O)C12CC2 C1(CNC(C(C)Cc2cnc[nH]2)=O)CC2(CCC2)CN1C(c1c[nH]c(=N)o1)=O C(C(C(=O)N1CCC1CNC(c1c[nH]cc1-c1ccccc1)=O)N(C)C)N(C)C n1(CCCC(=O)NCCCC(C)NC(c2c(CC)n[nH]c2)=O)ccccc1=O C1(C(=O)NC2(C)CCN(C(c3c(C(C)C)scn3)=O)CC2)CC2(C1)CC21CCC1 c1(C(C(=O)NCC#CCNC(C2C(C(=O)OC)CC2)=O)OC(C)C)ccccc1 CC1CN(C(c2nc(O)[nH]c(=O)n2)=O)CCN1C(=O)CCC1CC1(C)C c1(CC)c(C(=O)NCC2CN(C(C3CCCS3)=O)CCCO2)[nH]c(C)c1C(C)=O C(CCCC(C)(C)C)NC(CN(C(=O)CC1CCCOCC1)CCOC)=O C1(CCNC(C(c2nccc(C)c2)(C)C)=O)C(C)CCCN1C(=O)CC1(CO)CC1 C1(CC#C)(C(=O)NC)CCN(C(=O)C=CCN(CCF)CCOC)C1 c1(C(COCC(CNC(C)=O)O)C)cc(Cl)ccc1F CCC(F)(F)CC(=O)NCc1ccc(C(=O)NCc2cnn(C(C)C)c2)nc1 C1(n2cc(CSC)nn2)CC2CCC1(NC(=O)Cc1cncn1CC(=O)O)C2 C1(NC(C(C2CCOC2)OC)=O)CCN(C(=O)CC(C)(C)C#N)C12CCC2 C1(NC(C2(N(C)C)CCCOC2)=O)CN(C(=O)CSc2nc[nH]n2)CC2CC12 CC(C)(C)CCC(C)(c1nnnn1C1CC1)NCc1ncc(Br)s1 c1(C(N2CC(NC(c3ccc(CCC)[nH]3)=O)C(C)C2)=O)nc(O)[nH]c(=O)n1 C1(C(=O)NC2CC23CC(OC)C3)(CC)CCCN1C(=O)COCCCF CC1C(NC(=O)COC2CCC2)CCCN1C(c1ccoc1CC(N)=O)=O Nc1cc(C(=O)NCC=CCNC(c2coc3c2CSC3)=O)cc(O)c1 C#CCCC(O)C(=O)N1CC(NC(=O)CSC(C)C)CC1(C)C CC(C)C(CCC(=O)NCCC1CC(F)C1)NC(C12CCC(CC1)CO2)=O C1(CCC)(NC(C2CCOC(C)C2)=O)CCN(C(=O)CCCCCSC)CC1 C1(NC(c2nc(C)c(C)o2)C)C2CC3CN(C(=O)OC(C)(C)C)C1C3C2 c1(NCC2N(C(c3cccc(C)c3F)=O)CCC2)ncc([N+](=O)[O-])cc1Br C1(C(C(=O)NCC(C)(C)NC(CSCCCC)=O)C)CCCCCC1 C(=O)(CCCC(=O)NC1CCN(C(c2nc(CO)n[nH]2)C)C1)OCC c1(C(C)NC(C2(CC)CN(C(c3cnn(C4CC4)c3)=O)C2)=O)cccnc1F c1(C(=O)NC(CCNC(c2c(C)con2)=O)C)c(S(N)(=O)=O)ncn1C C(=O)(C1=CCC2CCC1N2C(=O)CCc1cccs1)NCCCS(C)=O N1(C(C(C(C)O)N(C)C)=O)C2CC1CN(C(C1(C)CCCCC1C)=O)C2 C1(C)(CNC(N(CC)Cc2cccc(Cl)c2)=O)CS(=O)(=O)CCO1 CCC(CCOC)C(=O)N1CC2(CO)CC1(C(=O)Nc1cncc(F)c1)C2 C(=O)(C(O)CCCNC(c1occ2c1CCC2)=O)N(CC(F)Cl)C CCC(CC1CCCCC1)N=c1cc[nH]cc1NCNC(=O)OC(C)(C)C c1(C(=O)NC2CC(O)(CNC(C(CC)N(CC)CC)=O)C2)cncc(C)c1 C(CS(=O)(=O)c1cccc(NC(=O)NCC2CCN(S(C)(=O)=O)CC2C)c1)OC c1(C(=O)NCCOCCN(C)C(C2SC3C=CC2CC3)=O)nc2ccccc2[nH]1 CCC(C(=O)N(C)CC1CC(NC(=O)CCCOCC)C1)OCC(C)(C)C C1(OC2CN(CC(C(=O)OCC)C)C2)CCN(C2CCOC2)CC1.C1(=O)CO1 C(CCC(O)CO)N(C)C(C1(CNC(=O)COCCN(C)C)CC2(CC2)C1)=O NS(=O)(=O)C1CNC2(CCCC2)C1.C1(NCC2CC2)C2Cc3cc(F)ccc3C12 CC(C(=O)OC(C)(C)C)C(=O)N1CC(F)CC1CNC(c1ccccc1F)=O c1(OCC(=O)NCC2N(C)CCN(C(=O)CC3CC3)C2)c(F)c(F)cc(F)c1F c1(C(=O)NC(CC)(C)CNC(=O)C(C)CC(C)(C)C)cc(S(C)(=O)=O)ccc1O C1(NC(C=CCN(C(c2ncc(OC)nc2)=O)C)=O)CCCCNC1=O CN=c1[nH]cc(C(=O)NCC(C)N(C(=O)Cc2ccc(OCCSC)nc2)C)o1 C1(CNC(C2CC(OC)C2)=O)CCC(NC(C2CCC(=O)C2)=O)CC1 c1(-c2nn(C(C=C)C)c(-c3sc(F)cc3Cl)n2)ccc(Br)c(F)c1 C1(C2CCN(C(=O)Cc3c[nH]nc3O)C2)(NC(C2CCCO2)=O)CC1 c1(C(N2C(CN(C(C(C=C)O)=O)C)CCC2)=O)cc(C)n(-c2ccccc2Cl)n1 CC(C)S(=O)(=O)C(C)C(=O)N1CC(NC(=O)CCc2ccc(O)nc2)CC1(C)C CCC(C)(F)C(=O)NC(CNC(=O)COCc1cccc(C)c1)C1CC1 Cc1c[nH]c(CC(N)=O)c1C(=O)N(C)CC1CC(F)CN1C(C1CSCCS1)=O c1(N(C(C2CCC(CNC(CSCCC)=O)CC2)=O)C)cc(C)ccc1F C1(OC)CCC(C(=O)NCc2ccc(CNC(=O)Cc3csnc3C)cc2)CC1 C12CC3(COC1C3)NC(=O)C1C(C1)C(=O)N2.C1(C2CC2)(CSC)CC1 N1(C(C(C2CCOC2)OCC)=O)CCCC1(CNC(=O)CCOC)COC N1(C(c2cc3c(Br)ccc(OC)c3o2)=O)Cc2ccc(S(C)(=O)=O)cc2C1 c1(C(=O)NCC(C2CC2)NC(C(C)CF)=O)cccc(-c2cccc(Cl)c2)c1 N1(C(C2(C)C(C)CN(C(=O)COCCN(C)C)C2)=O)Cc2cccc(O)c2C1 c1(C(=O)NCC2CC3(C2)CN(C(c2cnco2)=O)C3)ccc2nc(S)oc2c1 C1(CNC(CC=C=C)=O)CCN(C(c2c(C)nn3ncccc23)=O)CC1C1CC1 C1(NC(c2cnn[nH]2)=O)CN(C(=O)CC2COCCO2)CC1C(F)F C1(NC(CNC(CCC)=O)=O)CCCC(NC(=O)CCn2cc(Cl)cn2)CC1 c1(C(=O)NCCCNC(CN(c2ccc(Cl)cn2)C)=O)cc2sccc2s1 C12(COC)CN(C1)C(=O)C1CCC1C2.C1(C(=O)N)CCCCC1.C1(=O)CO1.OC CCC(CCc1ccccc1)C(=O)NC1CCN(C(C2CC(OC)C2)=O)C1 Cc1cc(=NCCC(O)CC)[nH]c(=NCc2ncccc2S(C)(=O)=O)[nH]1 c1(C(=O)NCC(N2CCN(CCN(C)C)CC2)=O)cc(S(C)(=O)=O)ccc1F C1(CCC)CN(C(c2c[nH]c(=NC)s2)=O)CC1NC(c1ccc(C(N)=O)cn1)=O c1(NC(C(=O)NCCSCC#C)=O)ccc(C(F)F)cc1 C12(NC(C(=O)NCC)=O)CC1CN(C(C1(C)CCNC1=O)=O)C2 C1(NC(C(C2CN(C(C3(C)CC=CC3)=O)C2)O)=O)CC2(CNC(=O)O2)C1 c1(CC(C(=O)NC(C)CNC(=O)Cc2cncn2C)C)ccc(F)cc1F C1(C(C)C)CCCC(NCCC2CCCN2C)CC1 N1(C(CNS(NC)(=O)=O)=O)CCCC2(CCCN2C(=O)CCC(N)=O)C1 N1(C(Cc2cc(OC)no2)=O)CCC(CNC(C2CCCN2N=O)=O)C12CCC2 C(=O)(C(CC)C(F)(F)F)NC1C=CC(CC(N2C(CCCC)CCC2)=O)C1 n1(CC)cnc2c(NCC3CNC(=O)C3)[nH]c(=NC3CCCC3C(C)C)nc12 c1(NCC(C)C2CC2)nccc(=NCC(C)Oc2c(F)cccc2F)[nH]1 N1(C(COC(CC)C)=O)CCCC2(C1)CN(C(c1cc(Cl)c(F)cc1Cl)=O)C2 Cc1cnc(O)c(CNC(C2CCC(NC(C3C=CC=CC=C3)=O)C2)=O)c1 c1(C(=O)NCC2C(NC(C(C)CC3CC3)=O)C2)ccc2c(n1)OCC(=O)N2 c1(C(N2CCN(C(C3CC3[N+](=O)[O-])=O)CC(O)C2)=O)c(Cl)cccc1[N+](=O)[O-] Cc1sc(C(N2CCC(C)N(C(C3CCS(=O)(=O)C3)=O)CC2)=O)cc1[N+](=O)[O-] N#Cc1ccc(F)cc1CN1CC(NS(=O)(=O)c2cn[nH]c2)C(F)(F)C1 N1(C(C2(F)CN(C(CC3ON=C(C)C3)=O)C2)=O)CCN(C)CC1C1CC1 c1(CCC)cc(C(N2CCC(CN(C)C(C3CC(OC(F)F)C3)=O)C2)=O)nn1C N1(C(C(C)(C)O)=O)CCC2(CCC(CNC(=O)CC34CC(C3)C4)O2)CC1 CCCCC(C)(F)C(=O)NCC1COCCN(C(=O)C(C)(C)F)C1 N1(C(c2nc(C)[nH]n2)C)CCC(C2CCN(C(c3cc(F)ccc3F)=O)CC2)C1 N1(C(C)=O)Cc2ccc(S(=O)(=O)N3CCOC4COCC34)cc2C1 O=C1Nc2cc(C(=O)NCC=CCNC(=O)C=C(Cl)Cl)ccc2C1=O S(=O)(=O)(c1cc(NC(=O)Nc2cnc3nccnc3c2)ccc1F)N(C)C C12(C(=O)NCCC(C)NC(C3CC(F)(F)C3)=O)COC(CS(C)(=O)=O)(C1)C2 N1(C(C(CC)C(C)C)=O)CCCN(C(=O)CC(C)(C)C)C(c2ccccc2)C1 c1(CCNC(c2snc(OC)c2Br)c2nnnn2CCCF)cccc(Cl)c1F C1(CNC(c2ccc(N(C)C)cc2)=O)(NC(C2CCOCC2)=O)CCCCC1C c1(NC(C)=O)ncc(C(N2CCCC2CNC(C2CN(C(C)C)C2)=O)=O)s1 C1(NC(c2cc(Br)c(C(F)F)o2)=O)CC2(C1)C(C(=O)O)C2(F)F C1(N(C(C=Cc2nc(C)sc2)=O)C)CC2CC1N(C(C1CC(=O)C1)=O)C2 CCCC(C(F)(F)F)NC(=O)C(C)N(C(c1nonc1N)=O)C1CC1 C1(C(N2CC(C)C(NC(c3ccsn3)=O)C2)=O)CCc2ccnn2C1 C(N=c1cc(C(C)(C)C)nc(Cl)[nH]1)C1CC(NC(CN(C)CC)=O)C1 C1(O)(CCNC(CCC2CCC(C)O2)=O)CCN(C(C2CC(CCO)C2)=O)CC1 c1(CC)nnc(CN(C)C(=O)NCCC(O)CSc2ccc(F)cc2)n1C C(c1c(Cl)nc2ccccn12)=CC(=O)NC1CN(C(C=CC(C)(C)C)=O)CC1F n1(CC(=O)N(C(C)C(=O)NC(c2noc(C)n2)C)CC)ncccc1=O c1(CCC(=O)NC2C=CCN(C(CCCOC)=O)C2)nc2cccc(Cl)c2[nH]1 CC1=CCCN(C(=O)CCC2(NC(=O)Cn3cccc3)CCCC2)C1 C(CC(C)(C)C)(C(=O)NC(CC(N)=O)C(=O)NCC(C)Cn1cccn1)OC c1(CC)nn(C)c(CC(=O)N(C)C(c2ccc(Br)cc2)C2CC2)c1Cl c1(C(N2CC(OCCNC(CC3CC(=C)C3)=O)C2)=O)c[nH]c(=N)s1 C1(C(=O)NC2CCC(NC(C3(CC#C)CCCCC3)=O)CC2)CNC(=O)CC1C c1(C(=O)NC2CCCC(N(C(=O)CSC(F)F)C)C2)cccc2nc(O)[nH]c12 C(CCCCCC(=O)NCCc1n[nH]c(C)n1)NC(C1(CC)CCCO1)=O c1(OC)ccc(CC(=O)NCC2CCN2C(c2cc(C)no2)=O)cc1 c1(C(=O)NC2C3CN(C(Cc4n[nH]c(=NC)s4)=O)CC32)c(C)ccc(C)c1C Cc1nc(C(C)(C)C)ncc1C(=O)NC(CO)C(C)NC(=O)CC1C=CCCC1 C#CC(C(=O)NOC(CC(C)C)C(=O)N1CCCC1(C)C(C)(C)C)C(C)C N1(C(C(CCC)OC)=O)CC(NC(=O)C=C(Cl)Cl)CC2(CCC2)C1 c1(C(N2CCC(NC(c3c(C)cno3)=O)C(O)C2)=O)c(F)c(F)c(F)c(F)c1F c1(OC)cc(C(=O)NCC(C)(C)CCNC(c2ccco2)=O)cc(F)c1 CC1CN(C(=O)C(N)=O)CC(C)C1NC(=O)CC1Cc2ccccc2O1 C(C(C)C(=O)NC1CC(CNC(=O)C(C)N(CC(F)(F)F)C2CC2)C1)SC c1(N2CC(C(C)NC(Cc3ccc(OC)cc3C)=O)C2)c(Cl)cccc1[N+](=O)[O-] c1(C(N2CCN(C(C(CC(CC)C)C)=O)C(C)C2)=O)cn2c(n1)CC(C)CC2 C1(CC(=O)NCC2(OC)CN(C(=O)CCC#N)C2)CCCC12CC2 c1(N2CC(C)C(NC(=O)CC3CN(C)C3)CC2)ncc2c(Br)cccc2n1 c1(OC)ccc(F)c(C(=O)NC2CN(C(=O)CCc3nnc(SC(C)C)o3)C2)c1 CCCCC(F)C(=O)NC(CC(=O)N1CCOC(C2CC2)C1)C(C)C CS(=O)(=O)CC(=O)NC1C2CN(Cc3ccccc3)CC12.C12CCN(CC1)C2=O c1(C(N(C(C)CNC(c2ccc(O)cc2F)=O)C)=O)cc2ccc(Cl)nc2s1 CP(C)(=O)CCC(=O)NCC(c1ccccc1)CNC(c1ccsc1C1CC1)=O N1(C(C(n2ccc(C)n2)C)=O)CC2(CCN(C(=O)CC3(C)CCC3)CC2)CC1C C1(N=[N+]=[N-])(C(N2CCC(C#C)(O)C2)=O)CCN(C(=O)CCCCCN(C)C)C1 N1(C(C(=O)NC(C)C)=O)CC2(NC(=O)CC3(C)OCCO3)CCC1C2 CCCC(CNC(=O)CCc1cncs1)C(=O)NC1CN(C)CC1(F)F N1(C(CC)=O)CC(OCC)C(NC(=O)COc2cccc(-n3cnnc3)c2)C1 C=CCC(F)(F)C(=O)NCCOCCC(=O)NCc1ncccc1C C1(C)(CC)CCC(NC(=O)CN(C(C2CCCC3CC23)=O)C2CC2)CC1 N1(C(C2C(c3cncc(C)c3)C2)=O)CC(NC(=O)CCCC#N)C(C)(C)C1 Cc1cc(CCC(=O)NCC(C)NC(c2c(C)nsc2Br)=O)cc(C)c1 Cc1cc(C(=O)NC(C2CCCN2C(=O)C(C)C)C)c(C)n1Cc1ccccn1 CCC(CC)(CC)C(=O)N1CCC2(C(=O)NCC3CCCS3)CCCC12 c1(C(=O)NCC(CNC(Cn2nc(C)n(CC)c2=O)=O)F)cc2ncccc2[nH]1 CS(=O)(=O)C1CCN(C(C2CN(C(=O)OC(C)(C)C)CC2C2CC2)=O)C1 Cc1ccc(Cl)cc1OCC(N1CCCC(CNC(c2cccnc2S)=O)C1)=O CCC(CC(=O)N1CCC(O)(CNC(=O)C(C)=C(C)C)CC1)C(C)C C1(NC(Cc2cnc(C)s2)=O)CC(C(=O)N(C2CC2C2CC2)C)C1(C)C O=C1Cc2cc(C(N3CCCC4(C3)CC4(F)F)=O)ccc2N1 CCC(CC(=O)NCCC1COCCO1)N(C)C(c1cc(CO)c(C)o1)=O C(=O)(C1=NOC(CNC(c2sccc2Cl)=O)C1)N(C(CC)C1CC1)C Cc1ccc(C(=O)NC23CC(C2)N(C(C2SCCC2C)=O)C3)cc1N c1(C(=O)OC)cc(CN2CCCC3(C)CCCCC23)cc([N+](=O)[O-])c1C C12(CNC(=O)Cc3csc(-c4cccs4)n3)CC(CN1C(C1CCSC1)=O)C2 N1(C(c2c(C)ccs2)=O)Cc2occ(C(=O)NCCc3ncc[nH]3)c2C1 CC1=C(C(=O)N(C2CCCN(C(=O)CCc3c(C)noc3Cl)CC2)C)CCC1 c1(CC)nc(C)oc1C(=O)NCC(CC)(CC)NC(=O)C(C1CCCCC1)O CCC(C(=O)N1C(C)C2CC1C2NC(=O)COc1cnn(C)c1)C(F)(F)F c1(OC)ccc(CC(C)Sc2noc(C(=O)C3CC3)n2)c(OC(C)(C)C)c1 CC(C)CC(C(=O)NC1COCCC1NC(c1cnn(CC2CC2)c1)=O)C(C)C Cc1nccc(Cl)c1C(=O)NC1CCN(C(=O)CCCN2CCCC2)C1 CCCC(C(O)C(=O)N1CCC=C(Cl)C1)NC(=O)CC(F)(F)C(F)F C=CC1(C(N2CC(CNC(C3CC(C#N)(OC)C3)=O)(COC)C2)=O)CCOCC1 c1(N(CC(C)NC(=O)C(C2CC2)C2CC2)C)nc(C#N)c(Cl)s1 c1(C(N2CCCCC(CNC(C3(CC(C)C)CC3)=O)C2)=O)ccc2occc2n1 CCCC(CC)C(C(=O)N1CC(c2ccc(F)cc2)C1)N1CCS(=O)CC1C C(C1CN(C(C2CCC(=O)O2)=O)Cc2ccccc21)NC(CCC=C(C)C)=O Cc1c(CC(=O)NCC=CCNC(C2CCN3CCCC3C2)=O)cccc1[N+](=O)[O-] N1(C(=O)NC2C(CC)CCCC2)CCC(COC)C(C)C1 c1(N2CCC(C(F)F)(CNC(c3ccc(F)nc3)=O)C2)c(F)cccc1[N+](=O)[O-] CN1CCC(C(=O)NC2CN(C(c3ccnc(C(C)(F)F)c3)=O)CC2C)CC1 N1(C(C2CC3(C(OC)CC3)C2)=O)CC(NC(c2n[nH]cc2C)=O)CCC(O)C1 c1(CNC(CCN(C)CCO)=O)cn(CCNC(=O)CSCC(F)(F)F)nn1 C1(CCNC(C2(c3cncn3C)CC2)=O)CN(C(CCCC)=O)CC(C)O1 c1(C(=O)NCC2CC(NC(c3c(C)c[nH]n3)=O)C2(C)C)ccc2cncn2c1 Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(c2cccc(=O)o2)=O)CCC(O)C1)=O CC(C(=O)NC(CNC(c1cn(C2CCC2)nn1)=O)C1CCC1)C(C)(C)C CCC(CC(=O)NCC1(CO)CCN(C(C2CN3CCCC2C3)=O)C1)C(C)C N1(C(C(CC(=O)OC)C)=O)CC2CC1CCC2NC(c1ccc(C2CC2)s1)=O Cc1ccc(Br)cc1C(=O)N1CC(n2cc(C3CCCCC3O)nn2)CO1 N1(C(C(C)CC(N)=O)=O)CCCCC12CN(C(=O)C(C)(C)CO)C2 c1(C(=O)NCC2OCCN(C(c3cnc(OC)s3)=O)C2)ccc(Cl)c(F)c1N Cc1nnccc1C(=O)NCC1CN(C(=O)Cn2ccccc2=O)CC1C C1(NC(c2nc(CCCC)sc2)=O)C2CCC1N(C(=O)C=Cc1cnn(C)c1)C2 CCS(=O)(=O)CCOc1ccc(NC(=O)CCn2nc(C)nc2C)cc1 c12cccc(c1)NC(=O)C(=O)NC2C(F)(F)F.C(C)(C)(C)OC(=O)NCC Cc1ccc(C)c(C(N2CC(O)(C(F)C(=O)NCCC3CCCCC3)C2)=O)c1 C(=O)(C(F)C(F)(F)C(F)(F)F)N(c1ccc2c[nH]nc2c1)CC c1(SCC(n2cc(C(C3(C(N4CCCC4)=O)CC3)OC)nn2)C)c(F)cccc1Br c1(C2N(S(CC(C)c3ccccc3)(=O)=O)CCC2)ccc(F)cc1Cl N1(C(=O)CC2CCCO2)CC2OCCN(C(c3cccc(Br)c3F)=O)C2C1 N1(C(C2(NC(C(CC=CC)C)=O)CCCC2)=O)CCn2ncnc2C1 c1(C(=O)NCC2C3CN(C(C(CC)n4nccc4C)=O)CC32)cnc2n1CCS2 C=CCCC(C)(C)C(=O)N1CCN(C(C2CCC(=O)O2)=O)CC1CF C1(C(=O)NC(CC=CC)C(=O)NCCC2CCCN2C)CCCC(C#N)C1 C1(=O)C(C(C)(C)C)CC2CCCCN12.CCCC(=O)NN(C(=O)C(=O)NC)C C(=O)(C1CCCc2c[nH]nc21)NC1(COC)CCN(C(=O)C(O)C2CCC2)CC1 C1(C(NOCC(=O)NC(C2CCC(C)C2)=O)=O)CC2CCC1O2 Cc1cn2cccc(CNC(C3C=CCN(C(C4CCNC45CC5)=O)C3)=O)c2n1 N1(C(c2cc(C3(OC)CCC3)on2)C(=O)NC)CCCCC1C1(O)CC1 Cc1nc(C(N2CCCC2CCNC(=O)Cn2cc(C)ccc2=O)=O)cc(O)n1 C1(C(N(C)CC2(OC)CCC2)=O)CCCC(NC(=O)CCCc2ncco2)C1 CC1CN(C(c2c[nH]nc2F)=O)CCN1C(c1cc(F)ccc1O)=O c12ccccc1CNC2=O.C12(NC(C(C)OCC)=O)CC(C(C)(C)C)(C1)C2 CCC(CC)(CCOC)C(=O)NCC(C1CC2CCC1CC2)(C)O C#CCC(C(=O)NCC1(OC)CC1)NC(=O)CC1CC1CC c1(CNC(C(C)CC2CCN2C(=O)C2=CS(=O)CCC2)=O)ccc([N+](=O)[O-])cc1Cl N1(c2ccnc(C)n2)C(C(=O)Nc2cc(C)ccc2C#N)CC2CCCCC12 c1(-c2c(CN3C(CNC(c4c(C)cno4)=O)CCC3)c[nH]n2)ccc(Cl)cc1 N1(C(CCCSC)=O)CCCC(C2(NC(=O)CC3(C)CC3(F)Cl)CC2)C1 c1(OC)ccc(N)c(C(=O)NCC2CC(NC(C3CC3(C)C(C)C)=O)C2)c1 c1(NC2(CC)CCN(C(C(CC)C(C)O)=O)CC2)cc(C#N)c(F)cc1[N+](=O)[O-] c1(C(N2CCC(NC(C(CC)C3CCOCC3)=O)C2)=O)ccc(O)cc1C c1(NC(CC(CC2CC2)NC(C2C(=C)C2)=O)=O)c(C)cc(O)cc1C C1(N(C(c2ccc(C(C)C)o2)=O)C)CN(C(C2CCCOC2)=O)CC12CC2 CC(CC(F)(F)F)C(=O)NC1CN(C(C2C3CC4C(C3=O)C24)=O)CCC1(C)C C12(C(=O)NCC(CN(C(c3n(C(C)C)cnc3)=O)C)O)CCOC1CC(=O)NC2 C=CCC(CC(C)C)C(=O)NCC(C)(C)CCNC(=O)CCC(=C)Cl c1(CCC)nc(C2CC2OC)n(-c2cncc(Br)c2)n1 C1(C)(NC(CCC2C(C)C2)=O)CCN(C(=O)CCCC2CCC2)C1 CS(=O)CCC(=O)NCCC1CCN(C(=O)C=CS(C)=O)CC1 N1(Cc2cc(OC)cc(C)c2Br)CCN2C(=O)CCC2C1 c1(C(C(=O)NCCC(=O)OC(C)(C)C)NCCN2CCOC2=O)ccccc1 C(=O)(C1=CC2C=CC(C1)C2)N1CCCCC(NC(c2ccc3occc3c2)=O)C1 C1(C#N)(C(=O)NCCC(C)(C)NC(CCCCOC)=O)CC12CCC2 Cc1nnc(C(=O)NCCCC(c2ccccc2)NC(C2CCC(=O)N2)=O)s1 C1(NC(CC=C)=O)CCC(NC(c2sccc2I)=O)CC1 CCC(C)(F)C(=O)N(C)CC1CCN(C(c2c(Cl)cnn2C(C)C)=O)C1 C1(C(=O)NC(c2ccc(C)cc2)C)CN(C(c2csc(C)c2C)=O)CCN1C CC1CC(NC(=O)CC2CC(C)(C)CO2)CCN1C(C1CC2(CSC2)C1)=O c1(OC)ccc(NC(c2c(CO)cccc2C)c2nnnn2C)c(C)c1C c1(C(=O)NCC(CC)(C)NC(c2ccc(C3CC3)c(F)c2)=O)ccc(C)c(O)n1 C1(C(CNC(c2cc(C)on2)=O)(C)C)CCN(C(=O)CC2CCCCCC2)CC1 CC(CN=C(NC1CC1)N1CCC(C2CCC2)C1)N1CCCCC1 C(=O)(CC(C)CNC(=O)Cn1ncccc1=O)N(C(CO)CO)CC N1(C(c2nc(CC)oc2)=O)C2CCC1CN(C(c1[nH]c(C)c(C(C)=O)c1C)=O)C2 CC(C)CS(=O)(=O)CCC(=O)NC(CNC(c1ccccc1N(C)C)=O)C1CC1 c1(CC)ncc2c(n1)CCC(C(=O)NC1CC1NC(C1CC(OC(C)=O)C1)=O)C2 CC(CC(=O)N1C(C(=O)NCC(C)(O)CO)CCC1C)C(F)(F)F CC(C)CCCCC(=O)NC1CCCC(NC(=O)Cn2ncccc2=O)CC1 Cn1cc(C(F)(F)C(=O)NC2(COCCC3CCS(=O)(=O)CC3)CC2)ccc1=O C(=O)(C1(C)Cc2cccc(Cl)c21)NCC(C)NC(C=Cc1cc(OC)ns1)=O CC(O)C(C)C(=O)N1CCC(C(C)(C)CNC(=O)Cc2cc[nH]c2)CC1 c1(C(N2C(CC(=O)Nc3ncc(F)cn3)COCC2)=O)c(O)cccc1[N+](=O)[O-] C1(C(=O)NCCCC(C)NC(c2c(OC)nccc2)=O)CCCCCCC1 CC(C)CC(O)CC(=O)NCC1(NC(c2ccc(-n3cnnn3)cn2)=O)CCC1 c1(C(=O)NCC(CC(=C)C)NC(C2(COC)CC2)=O)ccc2c(c1)C(=O)CCS2 C=C=CCCC(=O)NC(C)C(C(C)C)NC(c1cnc(NC)cn1)=O c1(CCC(=O)NC(CCN(C(C(CC)C)=O)C)C)cc(C)nc(C)c1 C12(NC(c3cncnc3)=O)CC1CN(C(c1ccccc1)=O)C2.C1(=O)CCCO1 n1(CC)nc(C(=O)NCCOCC(=O)N(C(C)CN(C)C)C)cc1O N1(C(c2c(C)ccc(C)c2)=O)CCCN(C(=O)CC2CC2(Cl)Cl)CCC1 C1(NC(CC=CCC)=O)CCN(C(=O)CSc2ccc(C#N)cc2)C(C2CC2)C1 C12(CNC(C3(C(=O)NCCc4ccoc4C4CC4)CCCCO3)=O)CC(CCO1)C2 C1(NC(C(CC(C)C)O)=O)CN(C(=O)Cc2ccc(Cl)cc2Cl)CC2CCCC12 c1(OC)ccc(C(=O)N(CCCCN(C)C(c2ccoc2)=O)C)c(F)c1Cl c1(CNC(C(C(C)C)O)=O)ccc2c(c1)CCCC2NC(=O)CCCCCF CC1CCCC1(O)CN(C(c1cccc(C(=O)O)n1)=O)CCO C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(C)(NC(C2(C)COC(=O)C2)=O)C1 N1(C(CCOC(C)C)=O)CCC2(CC1)COC(CNC(=O)C1=NOC(C)(C)C1)C2 c1(N2CCCC(C)(CNC(C3(COC)CCCO3)=O)C2)ccccc1[N+](=O)[O-] C1(COC(c2c(-c3cn(C)nc3)c[nH]c2)=O)CCC(O)CN1C(=O)OC(C)(C)C CCC(CC)CC(=O)N1C2CC1CN(C(C1CC1C(=O)OCC)=O)C2 C(=O)(C1CCCc2ccccc21)NC1(CNC(=O)CC2(O)CCOCC2)CC1 C(CO)(CCCCNC(C1C2CC3C(C2)C13)=O)NC(C1(CC)CCCC1)=O c1(C(=O)NC2CC3(C(NC(=O)CC4CC5(CCC5)C4)C3)C2)cc(F)cnc1O CC1(NC(c2ccncn2)=O)CCCCC1C(=O)NCC1(CO)CCC1 N1(C(COC(CC)C)=O)CCC(CO)(CNC(c2cnc(C(C)(F)F)s2)=O)CC1 CC1C(=O)N(CC(=O)NCC2(NC(c3cnn[nH]3)=O)CC2)C(=O)C1C N1(C(C(c2c(C)n[nH]c2C)C)=O)CC2(NC(c3cn(C)nc3Cl)=O)CCC1C2 N1(C(c2c(C)oc(CO)c2)=O)CCN(C)C(C(=O)N(C2CCOC2)C)C1 C1(C(=O)NCCC(=O)NCC(C)C)CSCCN1C(=O)Cc1cncnc1 C1(C(=O)NCCC2CCC(NC(CCOC(C)=O)=O)C2)C(C(F)(F)F)C1[N+](=O)[O-] CCC(C(=O)OC)C(=O)N1CC(CCCCNC(C2CS(=O)(=O)CCO2)=O)C1 C1(F)(CNC(=O)CC2CCO2)CCCN(C(=O)CCc2cn[nH]c2)CC1 N1(C(=O)NC(CCC)C)CCC(O)(Cc2ccccc2)C1 Cc1cc2c(C(N3CCC4CN(C(C5CC5(C)C)=O)C4C3)=O)ccc(C)c2[nH]1 C1(C(=O)Nc2ccc(F)cc2O)CCc2nc(-c3ccc(F)cc3)sc2C1 Cc1c(O)c(=O)ccn1CC(=O)NCC(CNC(=O)C(F)C(C)(C)O)C(F)(F)F N(C(=NCC(F)F)N1CCC(F)(C#N)C1)CC(Cc1ccc(C)cn1)CO C=CCCCCCC(=O)N(CC(=O)NC(C1CCCO1)CO)CC1CC1 c1(C(=O)NC2(COC)CN(C(c3cncc(C)c3)=O)C2)ccc(OC)cc1 c1(CC(=O)NC2CCC(CCNC(CS(N)(=O)=O)=O)C2)ccc2nn[nH]c2c1 c1(C(N2CC3C(C(=O)Nc4ccccn4)C3C2)=O)ccnc(OC(F)(F)F)c1 c1(NCC2N(C(=O)C3=CCCS3)CCCC2)ncc2scc(Br)c2n1 c1(C(N(C2CN(C(CC(CCC)O)=O)CC23CC3)C)=O)cc(O)c2ccsc2c1 C(CN=C(NCc1cnc(NC(=O)NC(C)(C)C)s1)N1CCC(F)C1)OCC C(CCCCC(=O)NCC(C)(C)C(=O)Nc1ccc(C(C)=O)cc1)=CC C1(C(=O)NC2C3CN(C(C(=Cc4ccco4)C)=O)C2C3)CCS(=O)(=O)N1C c1(OC)ccccc1C1(C(=O)NCCCCC(C)NC(c2cnc(O)s2)=O)CC1 C1(NC(=O)C=CC2CCCN2C(=O)CC2CN3CCC2C3)CCCC(O)CC1 c1(CCC(=O)NC(CN(C(C2CCC2C)=O)CC)C)ccc(OC)cc1F C1(C(=O)NCC(CNC(CNC(C)=O)=O)O)C=C(C)CS1 C1(C(N(CC=C)CC2CC2)=O)CCN(C(=O)COc2ccn(C)n2)CCO1 N1(C(C2(CCCC)CC2)=O)CC2CC(NC(c3coc(Cl)n3)=O)C1C2 C1(NC(CCC(=O)NC)=O)CCCC2CN(C(C3(C(=O)NC)CCC3)=O)CC12 C1(CNC(CC2C=NN(C)C2=O)=O)CCCCN(C(=O)C=CC2(C)COC2)C1 CCCCC(CNC(=O)CC1(OC)CC1)NC(=O)CCc1ccon1 C(=O)(CC(CC(C)C)NC(c1scc(C)c1C)=O)NC(CC)Cn1cncn1 C(CN=c1[nH]c2ncc(Cl)cc2o1)(C1CC1)NC(C1CC2(CCCO2)C1)=O Cn1cc(C(=O)NCCC(C)(C)CNC(c2cnc(O)c(F)c2)=O)ncc1=O C1(NC(CCC(C)OCC)=O)CC(F)CN(C(C2CC(F)(F)C2(C)C)=O)C1 n1(CC(C)(C)C)nc(-c2cccc(CN3CCCCC3)c2)nc1C1CCOC1 C(=O)(C(C)(C)CS(C)(=O)=O)NCC(C)CNC(c1cc[nH]c(=N)c1)=O c1(C(N(CCOC)CCNC(=O)CCc2ccc(C)o2)=O)ncncc1N Cc1nn(C)cc1C(=O)NC(CNC(c1csc(Br)c1C)=O)C1CCC1 Cn1cc(NCc2ccc(C(F)F)cc2)nc1C(=O)NC1CCS(=O)(=O)C1 c1(C(=O)NC(C2CN(C(C(C=C=C)C)=O)C2)C)coc2c1C(=O)NCCC2 CC1(CCNC(=O)Cc2cn[nH]c2)CCN(C(C2CC(N3CCCC3)C2)=O)C1 N1(C(c2cccc(OC)c2)=O)CC2(C1)CN(C(C)C)C2.c1(N)ccc(OC)c(OC)c1 CCCC(CC1CCCC1)C(=O)NC(CNC(C1(CO)COC1)=O)CCCC C#CCC(C(=O)NCCN1CCC(OC)C1)NC(=O)COCC(C)C C1(N(C)C(c2cc(C(C)(C)C)no2)=O)CCN(C(=O)C=Cc2cn(C)cn2)CC1 c1(C(=O)NCCN(C(=O)C(C(C)C)C(C)C)CC)cc(Br)c(C)cc1O c1(CC)nccnc1C(=O)NCC(c1cccc(Cl)c1)NC(=O)CCC(=O)NC c1(CNC(=O)NC(CC(C)C)C)cnc(S)n1C c1(CC(=O)N(CCC(C)NC(=O)CC2CCCN2C)C)ccc(F)c(Cl)c1 C1(C(=O)NC(c2cccc(C)c2)CNC(=O)CP(C)(C)=O)CC(=O)C12CCC2 C(CN=c1[nH]c2ccccc2o1)N(CC)CC.n1(CC=O)cnnc1 C1(CNC(C(n2ncc(C)c2)C)=O)CC(C(=O)NCCCNC(N)=O)=NO1 C=CC(CC)C(=O)NC1(COC)CN(C(C2(O)CCC2)=O)C1 C(=O)(CC(C)n1ccnc1)N(CC(CC)NC(c1cnc(C2CC2)[nH]1)=O)C C1(CC(N2CCN(C(CC(C)OC)=O)CC2)=O)CCC2CC1C2(C)C N1(C(C(CCOC)C)=O)CC2CC(F)(F)CCC2(NC(c2ncn(C)n2)=O)C1 c1(C(=O)Nc2cccc(NC(C3N(C)CCOC3)=O)c2)c(N)cc(Cl)cc1F N1(CCOC)CCC(N=c2[nH]c(NCc3cn(C)cn3)nc3cc(C)ccc23)C1 c1(C(=O)NCCCN(C(=O)CC2CCC(C)(C)CO2)CC)[nH]nc([N+](=O)[O-])c1Cl N1(C(C2C(C#C)C2)=O)CCOC2(C1)CN(C(=O)C(CC=C)CC(C)C)C2 Cc1nc2ncc(C(=O)NC3CCN(C(c4ccoc4)=O)CC3CO)c(=O)n2[nH]1 C#CCC(O)C(=O)N1CCC(CCC(=O)NCc2cccnn2)C1 N1(C(c2c(COC)ncs2)=O)CC(C)N(C(c2cc(C(N)=O)[nH]n2)=O)CC1C CN1CCN(C(c2cc(C(C)(F)F)n[nH]2)=O)C(CNC(C2CCN(C)C2=O)=O)C1 c1(C(N(C(C)CNC(C2CC=CCC2)=O)CC)=O)csc(COC)c1 C(CC(C)C)(C(=O)NC1CCCCC1F)NC(C(C(=O)OCC)F)=O C(C)(CCC(=O)NCC(c1ccccc1)NC(C1(F)CC1)=O)OC N1(C(CCCOCCOC)=O)CC(O)C(O)C1CNC(=O)CSC(C)C c1(CC)cc(C(=O)NCC(CO)NC(=O)CNCC2CCCCC2)cn(C)c1=O CCCCS(=O)(=O)CC(=O)NC1CCN(C(c2cc(C)c(C#N)cn2)=O)C1 C(CCCCC(=O)NCC(CNC(=O)CC1CCOC1=O)CO)SC C(=O)(CCC(C)(C)C)N1C(C(=O)NC2(C(=O)N(C)C)CC2)(COC)C=CC1 c1(C(=O)NC2C(NC(=O)CCc3nncs3)CCC2)nncc2ccccc12 Cc1ccnc(CNC(=O)CC2CCN(C(=O)Nc3scnc3N(C)C)C2)c1 c1(CC(=O)N(C2CCN(C(=O)CCc3ncnn3C)C2)CC)cccnc1 C1(C(=O)NC2(CF)CCN(C(=O)C=Cc3cn[nH]c3)C2)CC(C2CC2)=NO1 c1(C(=O)NC2(C(=O)NCC(CC)N3CCCC3)CCN(C)C2)cnc(O)c(F)c1 c1(NC23CCCC(NC(C(N4CCOCC4)C)=O)(C2)C3)nccc(S(C)(=O)=O)n1 N1(C(C(C)C)=O)CCN(C(C2(C(F)(F)F)CCOCC2)=O)CC1CS(C)(=O)=O C(=O)(CC(C(F)F)n1cccn1)N1C2C(NC(C(C)SC)=O)C(C2)C1 N1(C(CC=CC)=O)CCC(C2CCC2)(CNC(=O)CC2CCCCC2O)CC1 C1(C(=O)Nc2ccc(OC)cc2OC)CCCC12CCN(C(c1ccon1)=O)C2 CCC(C)(C#N)C(=O)N1CCCOC(CNC(c2cnc(C(C)C)cc2C)=O)C1 c1(C(=O)NCCSCCCn2cc(CCC(=O)OC)nn2)nn(C)cc1Br c1(C(N2CC(CNC(C3(CF)CCC3)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1 Cc1cc(COC(=O)C(CC(F)F)c2ccc(F)cc2)nc(C(F)(F)F)n1 Cc1ccsc1C=CC(=O)NCC1(CO)CCN(C(=O)CCSCC(C)C)C1 c1(-c2cc(CO)cc(OC)c2)cccc2[nH]c(C(N3CCCC3C(N)=O)=O)cc12 C1(OC(c2ccccc2)C)CCN(C(=O)C(C(=O)OC)OC(C)(C)C)CC1 N1(C(C2(N(C)C)CC2)=O)C2CCC1C1CC1(NC(C1(C)CC3CCC1O3)=O)C2 c1(NC(C2CCC(NC(c3cnc(O)c(Br)c3)=O)CC2)=O)ccnc([N+](=O)[O-])c1 c1(C(c2nnnn2C2CCOC2)NCCCO)ccncc1Br C12(NC(CC(C(C)C)O)=O)CCC(CC1)N(C(=O)C(C1CCCCCC1)O)C2 c1(C(N2CCC(C(C)NC(c3ccc[nH]3)=O)CC2)=O)cc(S(N)(=O)=O)ccc1O C1(CNC(CC(C)OC)=O)CN(C(c2cnc(O)s2)=O)CCC1C(F)(F)F c1(C(C(=O)NC2CC(CNC(Cn3c(C)cnc3)=O)C2)=O)ccc(F)cc1 c1(C(N2C(Cn3cc(CCCCC)nn3)CCC2)=O)cc2c(C)c(F)ccc2[nH]1 c1(C(C)C)nc(NCc2cc(Cl)ccn2)cc(=NCc2cc(Br)c[nH]2)[nH]1 C(=O)(C(C)CC(=O)NC1CC(C(=O)NC(C)CCN2CCCC2)C1)OC C(=O)(C(C)CC(=O)NC(C)CC1CCN(C(c2nccc(Cl)c2F)=O)CC1)OC CC1CCN(c2ncc(O)cn2)C1CNC(C1(C)CC=CC1)=O c1(N(C2CCSC2)C)ccc(S(=O)(=O)N(C2CCCC2)C)c(Cl)c1 C(=O)(C(C)CC(C)C(C)=O)N1C(C(N2CC(N(CCC)CC)C2)=O)C=CC1 CCC(CC)CCC(=O)N(CC)CC1CCN1C(=O)Cc1cccnc1OC N1(C(C2CCC(C)C2)=O)CC2(C1)OC1(CO)CC2(NC(=O)CCc2cnco2)C1 c1(C(CC)NCCc2ncc(COC)[nH]2)cc(Cl)ccc1Cl c1(COC)ccc(C(=O)NC2CC(CCNC(=O)CNC(=O)C(C)(C)C)C2)s1 c1(OC(C)C(N2CC3(CC3C(=O)Nc3cncc(Cl)c3)C2)=O)cc(Cl)ccc1Cl CC1CCC(C(=O)NC(Cn2cncn2)C(=O)Nc2cnsc2)CC1 C(CN=c1cc(F)nc[nH]1)NC(C(N1CCNCC1)C)=O C1(C)(C(=O)NC(CN(C(c2ccnc(C3CC3)n2)=O)CC)C)CCCN1C O=C(C1=CC2(CCOC2)C1)NC1CN(C(C2CCC3(CCOCC3)O2)=O)C1 c1(CC(C)C)ccc(S(=O)(=O)NCC(C)NC(C2C3(CC3)C23CC3)=O)s1 C1(C2CCCO2)(C(=O)NC2CN(C(c3c(OC)cc(N)cc3)=O)C2)CCCO1 CCCCC(CC(=O)NCCC(=O)NC1CC1)NC(=O)C(=O)C(C)C c1(C(=O)NCC23C(CN(C(C(CC)OC)=O)C2)C3)ccc(OC(F)F)cc1F c1(N2CC(CCCCNC(c3cc(C)ncc3)=O)C2)ncc2c(c1C#N)CCC2 C1(NC(c2cccc3c[nH]nc23)=O)CCC2(CCN(C(=O)C=CCO)C2)C1 c1(C(N(C2CCN(C(C3CCCC3)=O)C2)CC)=O)cn(C)c(C)c(Br)c1=O N#CCCCC(C(=O)NC(C1CCOCC1)=O)N1CC(CO)OC(C(F)(F)F)C1 CCCN=C(NCc1nc(C(N)=O)cs1)NCC(c1cccc(Cl)c1)CO C#CCC(C(=O)NCCN(C)CCO)NC(=O)COc1cc(C)on1 C1(C(N2CC(CC(=O)OC)C2)=O)CN(C(=O)CC2CCOCC2)CC(C)(C)C1 N1(C(CCN(CC#C)C(c2[nH]ccc2C)=O)=O)CCN(C)C2CC12 CC(CC(=O)N1CCC2(CC1)CC2CNC(C1(O)CC1)=O)C(C)(C)C N1(C(C=C(C)Cl)=O)CCN(C(=O)CC(C)C2CCCC2)CC1CO N1(Cc2cn(C3(NC(C4CNC(=O)C4)=O)CC3)nn2)CCCC(CC(F)(F)F)C1 c1(NC(C2CC3CC3N2C(c2nc(C)oc2)=O)=O)c(OC(C)C)cccc1F N1(C(CN(CC(C)(C)C)C)=O)CC(C)(CCC(=O)NCC(n2cccn2)C)C1 CCC(CCC(=O)NC1(C2CCCO2)CCC1)NC(c1n[nH]cc1C)=O c1(C(N2C(C(CNC(CC=C)=O)(C)C)CCC2)=O)ccccc1OC(C)(C)C c1(C(=O)OC)ccnc(NCC2CN(C(=O)Cc3cc(C)n(C)n3)CC2O)n1 C1(C2CC2)(NC(=O)NCCC(C)CCc2ccccc2)CCCCC1 CN(C)S(=O)(=O)N1CC(C(N2CCC(O)(CNC(c3ccc(=O)oc3)=O)C2)=O)C1 N1(C(C(CC)=CC)=O)CC(CNC(c2cc(CC3CCC3)c[nH]2)=O)C(O)C1 c1(C(N(CCCNC(=O)C(c2cnccn2)C)CC)=O)ccc(F)c(SC)c1 C(=O)(C1=C(Cl)CCC(C)C1)N(C1CCC(NC(c2ccc(C#C)nc2)=O)CC1)C N1(C(=O)CCC2CC2)CCC2CN(C(=O)C=CC3CCC3)CC2C1 C12CC(=O)N(C1)C1CN(C1)CC#CCN2Cc1ccc(C(=O)O)s1.C1CC1.OC N1(CC(=O)NCC(C)(C)CNC(=O)CSC(F)(F)F)Cc2ccccc2C1=O CCC(CC)CC(=O)N1CCCCC(CCC(=O)N(C(C)CSC)C)C1 CC1=C(C(=O)NC(C)CNC(=O)CCc2nc3ncccn3n2)C(=O)OC1(C)C Cc1cc(C(=O)NC(C)CN(C)C(c2cc(C(C)C)oc2C(C)C)=O)nn1C C(CC(O)CNC(=O)CCC1CCOCC1)NC(CSCC=C)=O O=C1CCC(C2=NC3(CCN=C4N(CCCCF)CCC(C)(C4)C3)O2)CN1 CCCCC(CC(=O)Nc1ccc(F)c(CC)c1)NC(c1cn(C(C)C)nn1)=O C1(NC(CSCC#C)=O)C2CCC(C2)C1C(N1CC(N(C)C)C(O)C1)=O c1(C(=O)NCC(CNC(c2c(C)nc[nH]2)=O)O)ccc(OC2CCOCC2)cc1 C(C(=O)NCc1ccc(C(=O)NCC(=O)N(C)O)s1)(C(C)(C)C)OC S(=O)(=O)(c1cccc2c1OC(F)(F)O2)NCc1snc(OC)c1Br N1(C(C(c2ccc(Cl)cc2)C)=O)CC(NC(=O)Cc2cnc[nH]2)C(O)C1 c1(OC)c(C(=O)NC(C)CC2CN(C(C3CCCC3C)=O)C2)nc(O)nc1O C1(C(N(C)CC2(NC(c3cc(C)c(N)cn3)=O)CC2)=O)CN2CCN1CC2C O=C(C=Cc1c(F)cccc1F)NNc1cnnc(O)c1Br c1(C(C(=O)NC(c2ccco2)C)N(CCC)Cc2ccccc2)ccc(I)cc1 c1(OC)ccc(C(N2CCCCCC2CNC(c2ccc(C)o2)=O)=O)c(Br)c1 CC(C)(C(=O)NCCC1CCN(C(=O)C(C)(C)N2CCCC2)C1)c1cscn1 c1(C2(C(=O)NCC3(F)CN(C(c4occc4F)=O)C3)CC2(Cl)Cl)ccccc1Cl c1(C(CC)COc2cccc(OC)c2CC)cccc([N+](=O)[O-])c1 Cc1ccc(C=CC(=O)NC(CCNC(c2cccn2C)=O)C(C)C)cc1Cl N1(C(CCNC(=O)C=CCl)=O)CCN(C(=O)C2=C(Cl)CCCC2)CC2CCCCC12 N(C1CCC(NC(c2csc(COC)n2)=O)c2ccccc21)C(C(=O)NCC)=O c1(OC)cnc(C(=O)NC2CC(CNC(=O)CCP(C)(C)=O)C2)c(F)c1 C12(C(N(C)CC3C(NC(C4C(CSC)C4)=O)CCC3)=O)CC1CNC2=O C12(C(=O)Nc3cncc(NC(CC)=O)c3)CCC(C(=O)NC(C)(C)C)(CC1)OC2 CCC(C)C(O)C(=O)NC1CCN(C(c2ccc(O)cc2)=O)C1C(C)(C)C C1(CCOC)CN(C(=O)CCN2CCSC(C)(C)C2)CCN1C(=O)COC(F)F c1(C(C(=O)NC(CC)C)N(C)Cc2cc(Cl)cc(Cl)c2)cn2cc(Br)ccc2n1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCC(NC(=O)C(F)(F)c2ccccn2)C(F)C1 c1(C(=O)NC2CCCN(C(c3c(C)n(C)nc3)=O)CC2)cc2cccnc2o1 CS(=O)(=O)c1ccc(C(=O)NCCCCC2CN(C(=O)C3=CC4CCCC34)C2)[nH]1 C1(CNC(c2cc(CC)ncc2)=O)CC(C)CN(C(c2cc(C#N)oc2C)=O)C1 CCC(C)(CO)C(=O)NCC12CN(C(c3cncnc3)=O)CC1(C(F)(F)F)C2 c1(C(=O)NC(C(C)NC(=O)CN2CCCC2)(C)C)cnc2n1CCCC2 N1(C(CNC(CC)=O)=O)CC(C(N2CCC(C)(C3CC3)C2)=O)C(C2CC2)C1 O=C1CCC(=O)N1CCS(=O)(=O)NCC(O)CC1OCCO1 N1(C(c2scc(C(=O)OC)c2)=O)CCC(C2CC2)(CNC(=O)C(C)(O)C2CC2)C1 N1(C(c2nc(CCCCC)sc2)=O)CCOC(CCNC(C2CC2C2CC2)=O)C1 c1(C(=O)OC)cc(C)[nH]c1NC(C1CCOC(c2ccc(F)cc2)C1)=O CCC(F)(F)CC(=O)NCCC(O)C(=O)N1CCCC(C(F)F)C1 Cn1cc(C(N2CCCC2CNC(=O)CCNC(N)=O)=O)c(O)n1 C1(C(=O)NCCC2N(C(C3(OC)CC3)=O)CCC2)CCC2C(C1)C2(F)F C1(CNC(c2cc(COC)sc2)=O)CN(C(=O)Cc2ccc(Cl)s2)C2CCN1C2 C(C(=O)NCC1(C)CCCN1C(c1ccc[nH]c1=O)=O)(C(C)C)NC(C)=O C1(NC(C2CC(C)N(C)C2)=O)(CO)CCCN(C(c2coc(O)n2)=O)C1 C1(O)(COC)CCN(C(c2ccncc2)C(=O)NCc2cccc(OC)c2)C1 c1(NC)ccccc1C(N1CC(F)CC1CC(=O)NCCC1C=CCC1)=O CC(C)CCN=C(NCC1(CO)CC2(CCC2)C1)N1CCC(C)(C(=O)N(C)C)C1 C(C(C)C(=O)NC1CN(C(=O)C(Cc2cnc[nH]2)NC(=O)OC(C)(C)C)C1)OC n1(C(C)C)ncc(C(=O)NCCc2ccnc(CO)c2)c1C1CC1 N1(C(C(n2cc(CC(=O)NC(C)(C)C)nn2)C)=O)CCCC2CCCCC12.CO c1(C(=O)NCC(C)N(C(=O)C(C)c2cc[nH]n2)CC)cccc(C)c1Cl O=C(CCOCCNC(c1n[nH]cc1Br)c1nnnn1CC1CCCO1)NO c1(C(=O)NCC(CC=C)NC(=O)C(C)=CCC)ccncc1C=C CC1CN(C(c2cc(C3CC3)on2)=O)CCC1NC(=O)CC1CCC(=O)CC1 C1(CC(=O)NC(C)(CNC(C2(O)CCC2)=O)CO)CSc2ccccc2NC1=O C(=O)(C(CC)CCCCC)NCC1C(NC(C(CC#C)(C)C)=O)CCC1 S(=O)(=O)(c1ccc(Br)cc1NCC1NC(=O)CC1(C)C)NC(CC)CCOC C1(CCNC(C(=O)NC2CC2)=O)CC(F)(F)CN1C(C1CC1F)=O N1(C(C(=O)NC(c2ccccc2-c2ccccc2)C(C)C)=O)CC(N)CCC1C C12(NC(=O)CCOCC(F)(F)F)CC(NC(c3occc3F)=O)(C1)C2 N1(C(c2ccc(N(C)C)cc2)=O)CCc2c(C(=O)NC(CO)C(C)O)n[nH]c2C1 c1(OC)ncccc1C(C(=O)OC)NC(CO)(C(C)OC)c1nnnn1C1CC1 c1(N2CC(NC(c3ccc(N4CCCCC4)cc3)=O)C2)ncnc2c1CCCC2 c1(NC(C(C2C(C)C2C)N(C)Cc2cc(C)on2)=O)ccccc1C N1(C(C=Cc2c(C)ncs2)=O)CC2CC1CCC2NC(=O)Cn1cc(CO)nn1 C1(CC)CN(C(=O)C(c2cn(C)nn2)NC(c2ccc(N)cn2)=O)CCCO1 Cc1nc2cncc(C(=O)NC3CCCN(C(=O)C(F)(F)C(O)C4CC4)C3)c2[nH]1 C1(NC(C(C(C2CC2)OC)(F)F)=O)CCN(C(C)C)C12CCC2 C12(CNC(CC)=O)CC1CN(C(=O)CCCc1ccncc1)C2 Cc1cc(CNC(c2n[nH]cc2CNC(=O)CC2COCCO2)=O)c(C)s1 c1(C(=O)NC(C2CCCCN2C(=O)COC(F)F)C)ccc(OCC(F)F)nn1 C(C(O)C(=O)NCCCC1CCOC1=O)NC(C1C(C#N)C1)=O N1(C(CC2CC(SC)C2)=O)CCC(C(=O)N2CC=CC(O)C2)=C(F)C1 N1(C(CCCC=C)=O)CCC(c2ccc(F)cc2)(NC(=O)C(C)C(F)(F)F)CC1 CCCCCC(CC)C(=O)N1CC2(CC2)CC1C(=O)NCc1nc(C)cs1 C(=O)(CCC(CC)CCC)NCC(=C)CCNC(C1(C)C=CCCC1)=O c1(C(=O)NCC2CCN(C(C3ON=C(CC)C3)=O)C2)cc(O)nc(O)n1 c1(OCC)nccc(C)c1C(=O)NC(C)CC(C)NC(c1c[nH]c(C(N)=O)c1)=O n1(C2CN(C(C(C3CN(C(=O)C(C)N(C)C(C)=O)C3)OC)=O)C2)cc(C)cn1 C1(C(=O)NCC(C)N(C(c2nccc(C)n2)=O)C)CCc2cncn2C1 C1(CNC(CN(C(C)C)C)=O)CCCCN(C(=O)CC2CC(N(C)C)C2)C1 C(=O)(C1=CCC(C)CC1)NCC1OCCN(C(c2c(Cl)ccc(OC)n2)=O)C1 C1(C(=O)NCC#CCNC(Cc2c(C)nn(C)c2)=O)CCc2nc[nH]c2C1 C1(C(N2CCC(n3cc(Cn4c(C)cc(C)n4)nn3)C2)=O)CN2CCCN1CC2 CCCCCCCC(=O)NCC=C1CCN(C(C23CCCCC2OCC3)=O)CC1 N1(C(C=CC(=O)N(C)C)=O)CCC2(CC1)CN(C(c1cnnc(C)c1)=O)CC(C)O2 C1(NC(=O)Cc2c[nH]nc2O)CC2CN(C(C3(C4CC4)CC3)=O)CC2C1 c1(NC(=O)NC(c2ccnc(C)n2)CC)ccc(Br)c([N+](=O)[O-])c1 c1(CCC(=O)NCC(CC)NC(=O)C(C)OCCOCC)ccc(O)c(F)c1 c1(CC(=O)NCC2(F)CCN(C(C3CC3CF)=O)CC2)ccc(Cl)cc1Cl N1(C2(CC3C(OCC)COC3)C(C(=O)OC)(C(=O)OC)C2)CC2(COC)CCC1C2 CC1(NC(c2nnc(C3CC3)s2)c2nnnn2C(C)(C)C)CCC2(CC1)CC2 C1(N(C)C(c2ccco2)=O)CC2CCC(C1)N2C(=O)C(c1ccc(Cl)cc1F)O C(C(CC(=O)N1CCC1Cn1cc(CC(C)(C)C)nn1)C(F)(F)F)N(C)C N1(C(c2c(CC)cco2)=O)CCCC2C1CCCN2C(c1n[nH]cc1Cl)=O N1(c2ncc(OC)c(C)n2)CCC2C(CCN2C(c2cc3cccnc3s2)=O)C1 N1(C(Cc2c(C)nccc2)=O)CC(NC(=O)CC(C)c2ccncc2)CC(F)C1 N1(C(C2C(C(C)C)C2)=O)CCC2CN(C(c3ccc(F)cc3Cl)=O)CC2C1 c1(NCCc2c(OC)cccc2Cl)cc(Br)ccc1S(=O)(=O)NCC1CCCO1 N1(C(C=CCNC(c2nc(C)c(C)s2)=O)=O)CCC(F)(F)CC1C N1(C(C2OCC(C)C2)=O)CCC2(CN(C(=O)C(C)(C)OCC(F)(F)F)C2)C1 c1(SC)cc(C)c(C(=O)NCCC(O)CNC(=O)C(CN(C)C)N(C)C)o1 CCC(C)(C)CC(=O)NC1CCCC(NC(C2CCC(O)C2)=O)C1 C(C(C(C)C)N1CCOCC1)N(CCCN(C)C(=O)OC)C Cn1cnc2sc(C(=O)NC3(C)CN(C(C4CCCCNC4=O)=O)C3)cc12 C(C(CC)(CC)NC(C1CN(C2CCOC2)C1)=O)NC(COCCCCCC)=O C(C(S(C)(=O)=O)c1ccccc1)N(C(Cc1ccc(C)s1)C)C=O N1(C(c2c(N)ccc(Cl)c2)=O)CC2(CCCN(C(=O)C3=CCCOC3)C2)C1 C1(C2CCCC2)(C(=O)NC2CCCN(C(c3cc(C)cc(C)c3)=O)CC2)CCC1 c1(CC(C(=O)NCc2n(C)nc(-c3ccccc3)c2)N)csc2ccccc12 C1(=O)C(C2(C)CC2)CN1CC(C)C.C(=O)CCC.C(COC)SC c1(C(N2CC(CCNC(CCC(C)SC)=O)OCC2)=O)cc2c(cc1O)CCC2 c1(C(=O)O)ccc(CNC2CC(NC(c3ccc(O)cc3Br)=O)C2)c(Br)c1 C12(NC(C(C)Oc3ccccc3)=O)CCCC1N(C(=O)CS(N)(=O)=O)CCC2 c1(OC)ccc(S(C)(=O)=O)cc1C(=O)NC(C)CNC(C1CCC(C)(C)CO1)=O c1(C(=O)NC2C(CNC(Cc3cccc(C)c3Cl)=O)C2)cc2ncccc2cc1Cl C1(NC(CCCCC=C)=O)CCC2(CC1)CCN(C(c1cc(CC)on1)=O)C2 N1(C(c2cc(C)oc2)=O)CC2CC(NC(=O)C(C)(C)C3CCCCO3)C1C2 C1(C(=O)NCC2(F)CN(C(=O)C(F)F)C2)CC1C1CC(F)(F)C1 CCC(C)C(C(=O)N1CCCC(NC(C2CCOCC2(C)C)=O)C1C)OC N1(C(c2c(C)cc(CC)o2)=O)CCC(O)C(NC(=O)C(c2cccc(C)c2)O)C1 CC1=CC(C)CN(C(C2CC(N(C)C)CN2C(=O)CCCC2CCCO2)=O)C1 CC1CCC(O)(C(c2nnnn2-c2cc(Cl)cs2)NC2(c3ccco3)CC2)CC1 c1(OC)ccc(Br)c(CN2CC3C(C2)N3C(c2cccc(Cl)c2O)=O)c1 C#Cc1cccc(C(N2CCCC(CC(=O)N(CCF)C3CC3)C2)=O)c1C CC1(C)CC(NC(c2ccnc3ncnn23)=O)CN(C(C2CC3CCC3C2)=O)C1 c1(OC)ccc2c(C(=O)NC3(C)CCN(C(c4ccc(C)nn4)=O)C3)c[nH]c2c1 c1(OC)ccccc1CCCNCCCC1(O)CCCC1 C1(NC(C2(O)CCCCC2)=O)CN(C(=O)COCC2CCOC2)CC12CC2 C1(C(=O)NC2(C=C)CCOCC2)N(C(C2C(C)(C)C2(F)F)=O)CCCC1(C)C c1(C(=O)NCCCN(CCCNC(C(C2CC2)OCC)=O)C)cccc(C)c1C CC1N(C(c2csc(Cn3cc(CCOC4CCCC4)nn3)c2)=O)CCC1(C)C N(C(=NCC(c1ccccn1)C1CC1)NCCNCCOC)C(COCC)C.C1CC1 N1(C(c2c(C)cc(CC)o2)=O)CC2CC(NC(=O)CCCN(C)C)C(C2)C1 Cc1cc2[nH]c(=O)c(C(=O)NCC34CC3CN(C(C3C5COCC35)=O)C4)cn2n1 N1(C(C2(C(=O)O)CCCC2)=O)CCN(c2cnc(C(C)(C)O)s2)CC1 c1(C(N(C)CCOCCCN)=O)ccc2nccn2n1 Cc1cc(N2Cc3ccc(F)cc3C2)nc(=NCCCCC(F)(F)F)[nH]1 c1(C(N2CC(NC(c3cnc(C)s3)=O)C(F)C2)=O)cccc(I)c1Cl CCCC(CCCNC(c1sccc1C(F)F)=O)NC(c1cc[nH]c1C)=O n1(-c2cn(CC)nc2)nc(-c2ccc(N)cn2)nc1CC1=CCCC1 C1(NC(c2c(C)oc(C(C)(C)C)c2)=O)CN(C(=O)C(C)C(F)F)C2(CCC2)C1 N1(C(C=CS(C)=O)=O)CC2CCN(C(C3CCCCCC3)=O)C(C2)C1 c1(C(CC)(C)C)n[nH]c(=NCCCNC(c2cccc3nccn23)=O)o1 CCCCC(C)C(=O)N(CCCNC(=O)CC1CC(C)C1)C c1(SC)ccc(C(=O)NCC2CC(NC(C3CC4(CC4)CO3)=O)C2)cc1 C1(NC(=O)Cn2cnnc2)CC2CCCC(C1)N2C(C1CC2C=CC1C2)=O N1(C(C2C(COC)C2)=O)CC2CC1CCC2NC(C1CC2C=CC1C21CC1)=O N1(C(C(n2cc(-c3nn(C)cc3C(=O)O)nn2)C)=O)CCC(F)(C(=O)N(C)C)C1 C1(NC(Cc2c(CC)nccc2)=O)(CO)CCCN(C(=O)CC(CC)OC)C1 CCC(C)CC(C)C(=O)NCC1(NC(c2ccccc2[N+](=O)[O-])=O)CC(OC)C1 c1(OC)ccccc1CC(=O)NC(C)CCNC(=O)Cc1cn[nH]c1 C1(NC(=O)C(O)CCCNC(C23CC(CO)(C2)C3)=O)CCCC2(CCC2)C1 CC(C)(C)C(CC(=O)N1CCC(C2(NC(C3C4CCCC34)=O)CC2)C1)C(F)F O(NC(=O)C(C)(C1CC1)N(C(=O)CCCC1CC1)C)CCCC#C CC1CC(F)CN1C(C1(CNC(=O)C(C)CC2CCCC2)CCC1)=O CCC(C)C(CN(C)C)NC(C1(CC)CN(C(C2CC3(CC3)C2)=O)C1)=O n1(CCC)nc(C)c(C(=O)NCCC2CCN(C(=O)C(F)n3cccn3)C2)c1C N1(C(C2CC(CC)OCC2)=O)CCCC(C)(CNC(c2ccnc(OC)c2)=O)C1 N1(C(C(CC(C)C)C)=O)CCC2(CNC(=O)CS(C)(=O)=O)CCCCC12 N1(C(C(COC)(F)F)=O)CCC(NC(c2cc(C(C)C)cnc2O)=O)CC(O)C1 c1(C(=O)NCC(C)NC(=O)Cc2cnn3c2CCCC3)cnc2ccnn2c1N C12(C(=O)NC3(C)CCN(C(=O)CC4CCCOCC4)C3)CCC(CC1)OC2 C1(C(N(C)CC2N(CC)CCC2)=O)CN(C(c2cnc(C)nc2)=O)CC12CC2 C(=O)(C(C)(C)C(=O)NC1CCCCC1CNC(=O)CC1CN(C)CC1O)OC C(CCCCC(=O)NCC1CCN(C(=O)CCC2CCOC2)CC1C)NC(C)=O N1(C(C2OCC(C)C2)=O)CCC(C2CCCN(C(c3csc(C4CC4)n3)=O)C2)CC1 C1(CC)C(C(=O)OC)CCCN1C(=O)NC(C)(C)C.c12nc(n[nH]1)CCS2 N1(C(C=CC2N(C(C(C)OCC=C)=O)CCC2)=O)CCn2nc(C)cc2C1 C12(CNC(=O)CC3CC4CC4C3)CCCC(CN(C(=O)CCc3cccs3)C1)C2 CC(C)C(C(=O)NCC(C)C(F)C(=O)NC1COCC(C)(C)C1)C(C)C CCC(C)(C)NC(=O)CC1CC(CNC(=O)CCOCC(C)C)C1 c1(C(N2CC(CNC(C3(CC(F)(F)F)CC3)=O)OCC2)=O)ccn2c1CSCC2 Cn1cc(CC(=O)NC2(CNC(=O)COC3COC3)CC2)c2ccccc12 CCC(O)C(F)(F)C(=O)NCC(C)(C)OCCNC(=O)C=Cc1nc(C)cs1 CC(CC(=O)NCc1ccon1)C(C)(C)NC(C1C2CCCCCC12)=O C1(NC(CN(C)C(N)=O)=O)CCN(C(=O)C(O)CC2CCCCC2)CCC1(F)F C1(=O)CC(O)(CCOc2ccccc2)C(CCC)C(CC)CC(=O)NCCCN1 N1(C(C(C)C2(O)CCC2)=O)CC=CC1(C)C(=O)NCCCc1nnnn1C N1(C(C2C3CC(=O)OC3C2)=O)C2CCC1CN(CC1CC1)CC2 C(=O)(C(F)CCC(C)(C)C)NC(CCC)CNC(c1cnncc1CC)=O c1(C(N2CC(O)CC(NC(c3c(=N)[nH]cnc3)=O)C2)=O)ccc2ccccc2n1 C1(NC(C2C(C=C)OCC2)=O)C2CC3CN(C(c4cnn5c4OCC5)=O)C1C3C2 n1(CCC=C)cc(C(=O)NC2CCCC2CNC(=O)CC2CC(CF)C2)nn1 c1(C(N(C2CCCN(C(C3(C(=O)N(C)C)CC3)=O)C2)C)=O)cnc2c(F)cccn12 C(=O)(C1=C(Cl)CCCC1)N1CCN(C(CCCC(C)c2ccccc2)=O)C(CO)C1 c1(C(N2CCOCC2CNC(=O)C(F)(F)C(F)F)=O)ccc(Cl)c2ccccc12 C(=O)(C1=CCOC1)N(CCOC)CCNC(=O)C(n1ccc(C(F)(F)F)n1)C c1(CNC(c2cc(SC)nn2C)=O)c(F)ccc(O)c1F CCC(CCCC(=O)NCCCN1CC2CC2C1)NC(C1CCCC1O)=O C(=O)(C(F)C(F)(F)F)NCCC1(NC(c2c(CC(C)(C)C)cccc2)=O)CCC1 CC1CN(C(=O)CC23CC(C2)C3)CCC1N(C(=O)Cc1csc(Br)c1)C O=C(C(F)C(F)(F)C(F)(F)F)NCC1(F)CN(C(c2nccn3nccc23)=O)C1 Cc1cc(C(=O)NCC2CC3CC3N2C(=O)COc2cccc(Cl)c2)c(C)n1C C#Cc1ccc(F)c(C(N2CC(CNC(=O)CC3CC34CC4)OC(C)(C)C2)=O)c1 O(NC(=O)C(C)CN(C)C(C1CC2C=CC1CC2)=O)CCCOCC Cc1c(CC(=O)NCC2CCN(C(=O)CC(C)N(C)C)CC2)ncn1C C(=O)(C#CC1CCCCC1)NC(C(=O)Nc1ccc(OC)nc1C)C Cc1nc(C(=O)NCC(F)CNC(c2cc(C)n(C(C)C3CC3)n2)=O)nn1C c1(OC)cn(CC(N2CC(NC(c3cc(C#N)no3)=O)C(C)C2)=O)c(C)cc1=O C1(CC(=O)Nc2cccc(C(F)(F)F)n2)(NC(C)=O)CCCCC1 O=S(=O)(c1ccc(F)cc1)N1CC2CCN(Cc3cncc(F)c3)CC2C1 c1(CC)cc(CNC(=O)Cn2cc(C3(C)CC3)nn2)n[nH]1.CSC N1(C(c2nc(CC)[nH]n2)=O)CCC(C)C(NC(C2CCC3(C2)CC3(F)F)=O)C1C C12(CNC(=O)CC3COCCN3C(c3ccon3)=O)CCC(CC1)OC2 C12CC13CCN(C3)C(=O)CC(C)(C)n1cc2nn1.c1(C(C)C)nscc1C(=O)O c1(CN(C(C2CCC(NC(CC(C)C3CCCO3)=O)C2)=O)C)cccc(F)c1 c1(C(N2CCN(C(CSCCOC)=O)C(C(C)C)C2)=O)cnc2ncnn2c1O c1(C(=O)NCC2(OC)CN(C(C34OCC(COC)(C3)C4)=O)C2)c(C)ccnc1C c1(C(=O)NC(C)C(CO)NC(=O)Cc2cccc(O)c2)cccc(P(C)(C)=O)n1 CCC(C)(F)C(=O)NCCCCCNC(=O)C(C)Cc1ccc(Br)cc1 C1(CC(=O)NC2(CO)CN(C(=O)CC3(O)CCC3)C2)Oc2ccccc2NC1=O Cc1cc(C)c2cc(C(=O)NC3CN(C(C4CC4F)=O)CCC3F)sc2n1 C#CCC(CC(F)F)NC(=O)C(C)(C)CN(C(=O)C(C)C=C=C)C C1(C(=O)NCCN(C)C(C2CCCN2C2CCCC2)=O)CC(F)(CO)C1 c1(C(C2CCCC2)CNC(CN(C)C)=O)cnn(-c2ccccc2)n1 c1(C(=O)NCCCOCCNC(C23CCCC2CC3)=O)cc2ccccc2cn1 C(=O)(C(C)(C)C(F)(F)F)N(C)CCNC(C1CC12CCC2)=O C1(CNC(C2C(C)N(C)CC2)=O)CCC2CN(C(c3cc(F)ccc3F)=O)CC12 c1(OCCOC)ccc(C(N2CCC3CC23)C(=O)NCCSC)cc1 C(=O)(C1CCCn2nccc21)N1C(COC)CN(C(=O)COC2CCCC2)CC1 C=CC1COCCN1C(C1CCC1CNC(=O)C(=O)C(C)(C)C)=O C(=O)(CCCCC(C)C)NCCC1CCCN(C(Cn2nc(C)oc2=O)=O)C1 c1(C(=O)NCC(C2CCOC2)NC(Cc2n(C)cnc2)=O)cn2cccc(F)c2n1 N1(C(C2CCCCCCN2C(C2C3CC4C(C3)C24)=O)=O)CC=C(C(=O)CCO)CC1 C1(C(N2CCC(NC(=O)Cn3ncnn3)CC2)=O)CC12CCOCC2 Cc1c(C(=O)N(C2CN(C(=O)Cn3c(C)csc3=O)CC2F)C)cncc1Cl C(CC(C(=O)NCC1COCC1O)NC(=O)CCCN(C)C)SC C1(CCOC)(NC(=O)Cc2ccoc2)CCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1 C12(CNC(C3CC4C(C)(C)C4C3)=O)CCC(CC1)N(C(C1CC1CF)=O)C2 Cc1c(C(N2CCCC2(C)C(=O)Nc2cc(O)nc(Cl)n2)=O)cncc1Br c1(C(=O)NCCN(C(=O)C=C2CCCCC2)C(C)C)nocc1Br N1(C(c2c(C)scc2)=O)CC(NC(c2cnc3n2CCC3)=O)C(C)(C)C1 C1(C)(CC)CN(C(=O)CN(C(c2coc(C)c2)=O)C2CC2)CCO1 CN1CCC(n2cc(Nc3ccco3)cn2)CC1.C12CC1N(CCC1CC1)C2=O c12nc-1n(C)n2.c1(COC(C(CC(C)C2CC2)NC(=O)N)=O)ccco1.C(C)(C)(C)O CCC1=NOC(CC(=O)NCc2ocnc2C(=O)NC(c2csnn2)C)C1 C1(N(C(=O)Cn2cnc(C(N)=O)n2)C)CCCN(C(c2cc(Cl)ns2)=O)C1 Cc1cc(O)ncc1C(=O)NCC(c1ccccc1)CNC(=O)C(C)S(N)(=O)=O CC(C)(C)C(C)(O)CNC(=O)CNC(=O)CC1CC(=O)NC1=O c1(C2(C(=O)NC3C(OC)CN(C(CN(CCC)C)=O)C3)CC2)ccc(F)c(Cl)c1 C1(CNC(CSCCC#N)=O)CCCC1CNC(c1c[nH]nc1Cl)=O C1(NC(CN(C)C)=O)CS(=O)(=O)CC1NC(c1cccc(C(N)=O)c1F)=O C1(C#N)(C(=O)NC2CN(C(CCc3ccc(OC)cc3)=O)C2)CCCOC1 C1(NC(C2(CCNC(CCC(=C)Cl)=O)CCCC2)=O)C2CCN(CC2)C1C CCCC(C)(O)CC(=O)N1CCN(C(C2CCN(C)CC2)=O)C(c2cn[nH]c2)C1 C1(CN(C(CC(=O)NCC)=O)C)CCCCN1C(c1cnn(C)c1C)=O C1(CNCc2cn(C3C(C)(O)CCC3)nn2)CCNC(=O)CC1 c1(OC)cc(C(=O)N(CC(C)NC(=O)C(N2CCCC(C)C2)=O)C)nn1C CSC1=C(C(=O)NC2CCC2NC(C2(N(C)C)C=C(F)C(F)=C2)=O)CCCC1 N1(C(C)C)CCCC(C(N2CC(CNC(=O)CN3CCCNC3=O)C(O)C2)=O)C1 c1(CC(N2CCC(NC(C(C)OCC(C)C)=O)C(O)C2)=O)ccccc1[N+](=O)[O-] CC1(C)C(NC(=O)C(=O)NC2CCCC=C2Br)C(C)(C)C1CC(=O)O C1(CNC(C2(COC)CCCC2)=O)(NC(c2cnc(C)[nH]2)=O)CCCCCC1 c1(NC(CC2(C=C)CN(C(c3ccc(F)c(F)c3)=O)C2)=O)cccc2c1CCC2 c1(C(=O)NCC(C)CC2CCC2)cc(CNC(=O)CC2CC2(C)C)no1 C1(NC(CCCCOCCC=C)=O)CCCCCN(C(C2CCS2(=O)=O)=O)C1 C(=O)(C(C)CC#N)N(CC(C)N(C(c1scc(C)c1)=O)C)C C(=O)(C1CCCc2nc[nH]c21)NCCOC1CN(C(c2ccc(OC)nc2)=O)C1 Cc1nn[nH]c1C(=O)NCC1(C(=O)NC(C)C(=O)NO)CCCO1 c1(C(N2C(CNC(C3(C)COC(=O)OC3)=O)CC2)=O)cccc2nc(S)oc12 c1(C(=O)NCC(CN(C(CC2CC(CC)C2)=O)C)O)ncc(C#N)cc1Cl c1(CC(N2CCC3CN(C(C=C(CCC)C)=O)CC32)=O)oc2ccccc2c1C c1(NC(C(c2ccc(Cl)s2)C)=O)ccc(OC(F)F)nc1 c1(C(=O)OCC2(CC(=O)OCC)CCCCC2OC)[nH]c(C)c(S(N)(=O)=O)c1C N1(C(c2scc(OC)c2)=O)CCOCC1CN(C(=O)C(C1CCCCC1)O)C C1(NC(C(N)Cc2ccoc2)=O)CCN(Cc2ccoc2)CC1 c1(C(=O)NC2CC(C)N(C(=O)CCN3CCCCC3=O)C2)cc2c[nH]nc2s1 CC1(C)Cc2ccc(C(N3CC(NC(C4CC4F)=O)C4(CC4)C3)=O)c(O)c2O1 Cc1nn(CC(N2CCN(C(c3cncnc3)=O)CC2CCO)=O)c(=O)n1C C1(CC(=O)NCC(CNC(C2CCN(CC#C)CC2)=O)O)CC(C)CC(C)(C)C1 c1(C(=O)NC(CC=C)CNC(C2CC(C)=NO2)=O)ccc2c(C)cc(Cl)nc2c1 C=Cn1nncc1C(=O)N(C1CCN(C(=O)CN2CCCC2)CC1)C C(C(=O)N(C)CCN(C)C(c1cscc1C1CC1)=O)(C(C)C)OCC(C)C c1(C(N(CC(CNC(CC(CC)C)=O)O)C)=O)cnc2sc(C)c(C)n12 c1(CCC)ccc(C(=O)NCC2CN(C(=O)CC3CCCCO3)C2)cc1 c1(C(=O)NCCCN(CC)CC2C(C(=O)OC)C2)cc(COC(F)(F)F)cs1 Cc1cc(C(c2ccccc2)CNCC2(NS(C)(=O)=O)CC2)ccc1Cl c1(NCCCCC(C)NC(C=C(C)Cl)=O)cc2c(cn1)C(=O)CCC2 c1(NC(N2CCOC(c3ccccn3)C2)=O)cccc(C2CCCC2)c1 C1(CNC(c2c(C)csc2)=O)CC(F)(F)CN1C(=O)CCC1CCC1 C=CC(O)(C(=O)N1CCCN(C(C2CCN(C(C)=O)C2)=O)CC1)C(F)(F)F CC1CN(C(c2ccc(Br)s2)=O)CCN(C(=O)C(F)CC2CCOC2)C1 CC(C)(C)C(C(=O)N1CCC(CCNC(C2(C(C)(F)F)CC2)=O)CC1)C1CCC1 C1(C#N)(C(=O)NCC(CC)NC(C2(Cc3ccccc3)CCC2)=O)CCCO1 CC1(C)CN(C(C2CCCCS2(=O)=O)=O)CCC1NC(=O)C(C1(O)CCCC1)F CC1=C(C(=O)N(C(C)C(=O)Nc2cncc(C(N)=O)c2)C2CC2)CCCO1 c1(CNC(C(c2c(C)cco2)N(C)CC2CCOC2)=O)ccccc1Br c1(CC2(C(N3CCC(CCNC(C(C)(C)F)=O)CC3)=O)CC2)cc(F)ccc1Cl C(C1c2ccccc2CCN1C(=O)C=CCO)NC(C(C)C1CCC1)=O C1(NC(c2ccc(CC)o2)=O)CC(C)CN(C(C23CC4CC2C3C4O)=O)C1 c1(C(N(CC(C)NC(c2cc(CC)n(CCO)n2)=O)C)=O)ccn2nccc2n1 N1(C(C(CSCC)C)=O)C2CCC1CC(CNC(=O)C=CC(=O)OC(C)(C)C)C2 Cc1ccc(C(N2CCC(NC(c3ccc(CN(C)C)[nH]3)=O)C2)=O)n1C C1(NC(C2CCOC2)=O)CCCCCN(C(=O)CN2C(=O)CCC2=O)C1 C(CC(CC)C(=O)NCC(C1CCC1)NC(c1nccnc1SC)=O)=CC c1(C(N2CCN(C(COc3c(C)nn[nH]3)=O)CC2)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(C(CC)(C)CO)=O)CCN(C(C23CCN(CC2)CC3)=O)C2(CCC2)C1 Cc1ccnc(N2CC=CC(NC(C3CCCC3O)=O)C2)n1 N1(C(CC=CC(C)(C)C)=O)CCC(C)(C)C1C(=O)Nc1cc(F)ccc1O c1(C(=O)NC2CN(C(CCc3ncc(C)cn3)=O)C2)cnn2c(N)cc(C)nc12 C=C(C)CC(C(=O)NCC1C=CCOC1)NC(c1cncc(Cl)c1)=O c1(OC)c(Cl)nc[nH]c1=NCC1CCCCN1C(=O)CNc1cc2c[nH]nc2s1 Cc1cn2cc(C(=O)NC3(C)CN(C(c4nn(C)cc4C)=O)C3)sc2n1 C1(C(=O)NC2CCN(C(CCc3[nH]c(=N)sc3)=O)C2)CC2CC1CC2O N=c1nc2ccc(C(N3CCOCC(NC(c4sccc4Cl)=O)C3)=O)cn2[nH]1 Cc1cc(C(=O)C(=O)NC2CCSC2)ccc1F.C12(CC1)CCNC2=O CCC(CC(F)F)C(=O)NC1CC(CNC(c2cnc(O)s2)=O)C(O)C1 Cc1ccc(C(=O)NC2CC3CC(C2)N(C(C24CC(C2)C4)=O)C3)c2cccnc12 c1(C(=O)NC(C)(C)CCNC(=O)CC2CC(F)(F)C2)ccc2c(c1)NC(=O)CC2 C(=O)(C1=C(Cl)CCOC1)N1CC(N(C)C(c2ccncc2N=[N+]=[N-])=O)C1 c1(Cc2nnc(CC)n2C)cc2c(N3CCN(C(=O)NC)CC3)ncnc2n1C Cc1nc(CNC(=O)CC2(C)CCOC2)oc1C(=O)NC1CC(CF)C1 Cc1cc(C(=O)NC2CCC2NC(=O)CC2NC(=O)NC2=O)nc2ccccc12 Cc1nc(CNC(=O)CC2CCCN2C(c2ns[nH]c2=O)=O)sc1C N1(C(CSCC(C)C)=O)CC2(C1)CN(C(c1cncc(Cl)c1)=O)C2 C1(N(C)C(C2(O)COC2)=O)CCCN(C(=O)C(F)(F)c2cnn(C)c2)CC1 C1(C(=O)NC23CC(NC(C(OC)OC)=O)(C2)C3)CC(=O)N(C2CC2)C1 N1(C(C(CN(C(c2cnc(CC)nc2)=O)C)C)=O)CCC(O)CC(C)(C)C1 N1(C(c2c(OC)nccn2)=O)CC2(C1)CN(C(c1cc(Br)ncc1F)=O)CCO2 C=CC1CCCCN1C(=O)C(CCCOC)NC(C1CCC1C#N)=O c1(NC(C(C=C)N)=O)c(P(C)(C)=O)cnn1CCF CCC(C)CC(=O)C(=O)N1CC2CCN(C(=O)CCC3CCCN(C)C3)C2C1 C=CCC(CC(F)F)C(=O)NC(CNC(c1sccc1C(C)C)=O)C(C)C(C)C c1(CC(N2CC(N(C)C(C3CC(C)(O)C3)=O)C2)=O)c[nH]c2cccnc12 CN1CCN(C(=O)C(=O)Nc2ncc[nH]2)C(CNC(=O)CCc2nncn2C)C1 C1(NC(C(c2ccc(Cl)cc2)CC)=O)CCC(S(C)=O)C1 c1(C(C(=O)NCC(C2CC2)SC)NC(=O)CC2OCCC2C)c(C)cccc1Br CCC(C)(C)CCCC(=O)NCC(c1ccc(F)cc1F)NC(=O)C(C)(C)O C1(C)(C(N2CCC(N(C(c3cc(C(N)=O)cn3C)=O)CC)C2)=O)CCCS1(=O)=O C(=O)(C1=CCCNSC1)NCC1N(C(c2ccc(C)nc2O)=O)CC1 Cc1cccc(CNC(C)(CCBr)c2nnnn2C2CCCC2)n1 C1(NC(c2c(CC)cccc2)=O)CN(C(=O)CC2CCCCO2)CC1C1CC1 C(=O)(CC(C)C(C)C(C)C)N(c1cncc(CC)c1)Cc1cn(CC(=O)O)nn1 c1(-c2ccn(C)n2)nc(-c2ccnc(-n3cncn3)c2)nn1C1CCOCC1 C1(NC(C(C=C)(C)C)=O)CN(C(c2cnc3n2CCC3)=O)Cc2ccnn2C1 C1(CC(C)NC(C2C3CC4C(C3)C24)=O)CCNCC1.c1(C(=O)N)cnsc1 C(=O)(CC(O)C(C)C)N1CC(NC(COCC)=O)C(Cc2ccccc2)C1 c1(C(C)C)cccc(N(C)C(c2ccc(C(N)=O)[nH]2)=O)c1 N1(C(CNC2C(C)(C)C2c2ccncc2)=O)CCOC(C)(C(=O)O)C1 c1(C(N2CCC(NC(CN(C)C(N)=O)=O)C23CC3)=O)cccc2ccnn12 C1(NC(CC2CC(OC)C2)=O)CCC(C(c2nnnn2C)SC2CC2)CC1 CC(=O)CCCC(=O)N1CCC(NC(=O)C(C)(C)C2(O)CCOC2)C1C c1(CN(C(CC)C(=O)OC)C)c(F)cc(Cl)cc1Br c1(OC)ccccc1C(C)NC(N1CCCC1CF)=O c1(CCCC(=O)NCC2C(CNC(C(CC)F)=O)C2)ccc(Cl)c(Cl)c1 C=CC1(C(=O)NC(c2ccccc2)CC)CCN(C(c2csc(C)c2)=O)C1 CCC(F)C(=O)NCCN(CCCN(C)C)C(c1ncn(-c2ccccc2)n1)=O CC1(F)CCN(C(C2CCC(CNC(=O)CN3CC4CC4C3)O2)=O)C1 C=CC(C)C(=O)N(CCCC(=O)N(CC(C)(C)O)C)C c1(C(=O)NCC2CN(C(C(CC(=C)C)C)=O)CC2O)cc2c(s1)CCCCCC2 c1(C(=O)NC2CC(C(=O)NCC(O)C(F)(F)F)C2)c(C(F)(F)F)ccc(Cl)c1F Cc1nnc2n1CC(C(=O)NC(C)CNC(c1sccc1SC(F)F)=O)C2 c1(C(=O)NCC2(O)CC(CNC(c3c(C)ocn3)=O)C2)cnccc1OCF C=CC1(C(=O)Nc2ccc(F)c(O)c2)CCN(C(C2CC3(CCC3)CO2)=O)CC1 C1(CCCNC(CC2(NC(C)=O)CC2)=O)CCCCN1C(c1ccnc(C)c1)=O C1(F)(CNC(c2c(COC)cc[nH]2)=O)CCN(C(=O)C=C2CCCC2)CC1 N(S(=O)(=O)N(C)CC(N1CCC(NS(C)(=O)=O)CC1)=O)C(C)Cc1ccccc1 c1(CC(N2CC(CNC(C=COCC)=O)C(C)CC2)=O)c[nH]c2cc(C)ccc12 CC(C)CCC(C(=O)NCCCC(C)CO)NC(C1CC(C)(CF)C1)=O c1(CC(N2C(CNC(CNC(N)=O)=O)CCC2)=O)c(F)cccc1F N1(C(C(CNC(C2(OCC)CCOC2)=O)(C)CC)=O)CCOC(C)(C)C1C C12(CNC(CC3(CSC)CC3)=O)CCCCC1CN(C(c1cncnc1)=O)C2 C1(NC(C(C)OC)=O)CN(C(=O)CC2(n3cnnn3)CCOCC2)CC(C)(C)C1 c1(C(=O)NCCC(C)N(C(C2N(C(CC)=O)CSC2)=O)C)ccc(S(C)(=O)=O)o1 c1(OC)nn(C)cc1C(N1CCC(C)(CNC(=O)C(N2CCCCC2=O)C)C1)=O C1(C2(O)CCCNC2)(C(=O)N(CCN2CCc3ccccc3C2)CCO)CCC1 N1(C(CC2CCCN(C)C2)=O)CC(C(=O)NC(c2ccccn2)CO)CC1(C)C CCC(CC(F)(F)F)C(=O)Nc1cncc(NC(=O)CCSC)c1 c1(C(C2CC2)NC(=O)NC(c2cccc(Cl)c2)CO)cc(Cl)ccc1O C1(NC(C(N2C(CNC(C)=O)COCC2)CC2CC(F)(F)C2)=O)CCC(F)(F)CC1 CCC(CN(C)C)CC(=O)NCCCC(C)(C)C(=O)N(CCCC(C)(F)F)C N1(C(CCNC(COC)=O)=O)CCC(NC(c2coc(C(F)F)c2)=O)C(C)(C)C1 C(=O)(C1CCCc2ncnn21)N1C(C(C)NC(C(C)(C)OC)=O)CCC1 C=CC(CC)CC(=O)NCC1CCCN(C(C2CCCCNC2=O)=O)C1 C=CCCCC(C(=O)N(C)CCOC1CC1)NC(C1CCC(=O)N1)=O C1(NC(C(C2CCC2)NC(c2c(C)cccc2)=O)=O)CC2C(C1)C2(F)F Cc1cnc(C=CC(=O)NCc2ncoc2CCNC(=O)CC(C)C2CC2)[nH]1 c1(C(=O)NC2CC3(C(NC(c4c(C)scc4)=O)C3)C2)cc[nH]c2nccc1-2 NC1C2C=CC(O2)C1C(N1CC(CCc2cn(CCF)nn2)C1)=O CC1(C)C(C)(C)C1(F)C(=O)NCC1CCCCC1NC(c1coc(CO)c1)=O c1(C(=O)NC2C(C)CN(C(=O)CC3=CCCC3)CC2)ccc2c(c1O)CCCC2 N1(C(Cn2ccc(C)n2)=O)CCCC2C1CCN2C(c1csc2c1CCCO2)=O C1(C(N2CC(CC(C#C)C)C2)=O)CCC(NC(c2cc(C#N)c[nH]2)=O)CC1 c1(C(C)CC(=O)NC2(C(=O)O)CCOC2)ccc(F)c(Br)c1 Cc1c(C(N2CC3C(NC(=O)C(F)F)C3C2)=O)cnc2c1c(=O)n(C)c(=O)n2C c1(CC(=O)N(CCCCN(C(C(C2CCC2)OCC)=O)C)C)c[nH]nc1C C1(C(N2CC(N(C(CN(CC(C)(C)C)C)=O)C)C(O)C2)=O)CC(C(C)(C)C)=NO1 N(C)(C1CN(C(C2(C)CC2)=O)CCc2ccccc21)C(c1c(CC)c[nH]n1)=O C1(NC(CC2N(CC)CCOC2)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)C(C)C1 CC1C(NC(C2CCN2C)=O)C(C)CCN1C(C1CCCC2CCCN12)=O C1(NC(C=CCC)=O)CCN(C(=O)CC(C)C2CCC2)CC1C Cc1cc(C)c(CCNC(c2ccc(Cl)cc2Cl)c2nnnn2C2CC2)c(C)c1 N1(C(c2ncn(CC)n2)=O)CCC(C)(C)C(NC(c2ccc(OCF)cc2)=O)C1 C12CC13CCN(C3)C2=O.c1(NCc2scc(C(=O)OC)c2)cncc(C)n1 C(=O)(C1=Cc2ccccc2OC1)N1C(C)CC(NC(C2CC2C)=O)CC1 c1(C(N(C2CCCN(C(C3(C#C)CCCC3)=O)C2)C)=O)cc2n(c1)CCC2 C(CC)(CCCC(=O)N(C1CCNC1=O)C)NC(C(C=C)(F)F)=O c1(C(=O)NCC(CN(C(CC(C)C(C)(C)C)=O)C)(C)C)ccnc2[nH]c(O)nc12 C(=O)(C(C(C)(C)C)NC(=O)CC1CCCC2CC12)NCCC(CCC)F C=C(C)C(C)(C)C(=O)N(C1(C(=O)NCc2ccc(C#N)s2)CC1)C Cc1cc(CN2CCC2CNC(c2cccc(-n3cccn3)n2)=O)ccc1Cl N1(C(C2(C)CC2c2ccccc2)=O)CC(C2CN(C(=O)CN3CCNC3=O)C2)C1 N1(C(c2cncc(C)c2)=O)CCC(CNC(=O)Cn2cccc2)C(C)C1 C(=O)(C1=CCCCC1)NCC1C(C)CCN1C(=O)COCC1CCC1 c1(C(=O)NCC2(C)CCN(C(=O)Cc3cccc(Cl)c3)C2)nccc2[nH]ccc12 N1(C(CN(C(=O)COCCCOC)CC#C)=O)CCC2(CCC(O)C2)C1 Cc1cc(C(=O)NCC(=O)NC2CCCN(C(=O)C(=O)N(C)C)CC2)cc(C)c1 C1(CCNS(=O)(=O)CC(=O)NCC)CC(F)(F)CN1C(=O)CNC(C)=O C(=O)(CC1=CCCCC1)NC(C1CCN(C(=O)CC2CC(C)(C)C2)C1)C C=CC1(CC(=O)NC(C)CC(C)(C)OC)CN(C(=O)C=CC(F)F)C1 c1(C(=O)NC2C(CNC(Cn3ccc(C)n3)=O)C2)ncc(Br)cc1F C1(CNC(=O)NCc2nc(CC)[nH]n2)CCC(=O)NC1C C(CC(C)(C)C(=O)NCC1CCCC(NC(=O)CNC(=O)OC(C)C)C1)OC c1(C(N2C3(CN(C(C(c4cccc(O)c4)C)=O)C3)CC2)=O)noc2c1COCC2 Cc1nncc(C(=O)NC2CC3(C2)CC3C(=O)NCCc2ccnn2C)c1C CCCC(CC(=O)NCCN1CC(CF)C1)NC(C1CC2CCCC2C1)=O CC(O)C1CCCc2ccccc21.O(C1CCOc2ccccc21)c1c(F)cccc1 C1(C(=O)NCC2(F)CN(C(C34CCC(C3)C4)=O)C2)C(C(F)(F)F)CCC12CCC2 C1(C(=O)NCc2cc(C)sc2C)CC(C)CN(C(c2csnc2C)=O)C1 c1(NC(=O)NCCS(NC)(=O)=O)c[nH]c2ccc([N+](=O)[O-])cc12 N1(C(c2cnccn2)C)CCN(C(c2nccnc2C(=O)O)=O)CC1 c1(C(N(C2CN(C(=O)CCc3ccon3)C2)C)=O)ccc(F)c(N)c1 c1(C(N(C)CC2CCN(C(C3(C#N)CCOC3)=O)CC2)=O)c[nH]c2cccnc12 CCC(CCCC(=O)NCC#CC(F)(F)F)NC(C1C2CCCC(=O)C12)=O N1(C(C2N(C)C(=O)OC2)=O)CCCC(C)(CNC(C23CCCCC2C3)=O)C1 N1(C(CCC=CC)=O)CC(C)C(C)(C(=O)NCC2CCN(C(C)C)C2)C1 c1(C(=O)NCC(C)(CC)NC(C(CCCCC)O)=O)cnc2ccc(C)cn12 n1(C(C)C)ncc(Br)c1C(=O)NCC=CCNC(=O)C(F)n1cccn1 CC1(C)CC(CC(=O)NC(C2CCCO2)CO)N(C(=O)C=Cc2cscn2)C1 C(=O)(N=c1cc[nH]c(CCCO)c1)NC(c1ccc2c(c1)CCCC2)C C(=O)(CCCCC(=O)NC1(C(=O)NCCC2=CCCCC2)CCOCC1)OC c1(NCC2(C)CCCN(CC3CCCC(OC(F)F)C3)C2)ccc(Cl)c(Cl)c1F C1(C(=O)N(CC(C)CNC(c2sccc2Cl)=O)C)(COC)CCOCC1 C(=O)(C(C(C)C)C(C)C)N(CCC(C(C)(C)C)NC(C(CSC)OC)=O)C C=CCCCC(C(=O)N1CC(CC)(CC)C1)NC(=O)C=CCO c1(NC(C2CC2C(=O)NCC2CCC=CCC2)=O)ncc(Cl)cc1F C(=O)(CCS(N)(=O)=O)N(C1CCCCCC1)CCNC(Cc1ccn(C)n1)=O c1(C(=O)NCC(CC)NC(c2cc3nc(C)ccc3o2)=O)c(Cl)oc2ccccc12 Cc1cnc2n1CCC(C(=O)NCCCn1cc(C(NS(N)(=O)=O)(C)C)nn1)C2 C1(NC(CCC(=O)NCC)=O)CCN(C(=O)C(C2CCOCC2)C)CCC1CO C(CCF)(C(=O)NCc1ccns1)NC(C=CC(=O)OCC)=O C1(NC(C2C(OC(C)=O)C2)=O)CC=C(C(=O)N2CCN(C)CC2C(N)=O)C1 O(NC(=O)C(CNC(=O)COc1cccnc1)CC1CC1)CC(=C)C c1(N(C(c2cnc(N(C)C)s2)C(=O)NCCOCC)CCSC)ccccc1 C1(NC(C2N(C(C3C(C)(C)COC3)=O)C3(CC2)CC3)=O)CC2(CCCCO2)C1 Cc1cc2c(NC(C3CCC(C)OC3)=O)ncc(I)n2n1 C1(CC(=O)NCCc2cc(C)on2)CC(F)CN1C(=O)C(O)CC1CCCC1 N1(C(C(C)(C)CF)=O)CC2(CCCN(C(c3cc4c(s3)CCC4=O)=O)C2)C1 N1(C(c2c(C)cnnc2)=O)C2CCC1CC(NC(C1CC3(C)CC1CO3)=O)C2 C(=O)(C=CS(F)(F)(F)(F)F)N1CC(NC(CC(C)C(C)(C)C)=O)CC1(C)C N1(c2n(CC3CC(C)OCC3)c(C3CC3)nn2)CCc2ncnc(O)c2CC1 C1(C(=O)NC2CCN(C(=O)CC3CC4(COC4)C3)C2)C2(CCC2)C12CCC2 C(C1CCCn2ccnc21)NC(c1ccc(F)nc1)CC(F)(F)F N1(C(C(C)O)=O)CC(CO)C2(CCN(C(=O)Cc3nccn3C)CC2)C1 C1(c2ccc(-c3n(CCCS(C)=O)ccn3)s2)CCC(=O)CC1(C)C C1(CCNC(=O)C=CC2CCCO2)CC2(CCC2)C1 CN1CC(C(=O)N(C(C2CC(F)(F)C2)=O)Cc2ccco2)C(c2ccnn2C)C1 N1(C(CC(C)OC)=O)CC2CCN(C(=O)C(C)CN(C)C)CC12 C(CNC(=O)CC1CCC(=O)C1)(C(=O)NCCCC1CCOC1)OC CC1=C(C(=O)N2CC(CNC(=O)Cc3conc3C)CC2C)CCS1(=O)=O C12(C(=O)NCCN(C(c3n(C)ncc3Br)=O)C3CC3)CCC(CC1)CO2 C(=O)(C1CS(=O)(=O)c2ccccc21)Nc1c(C)cc(Br)cc1F C1(NC(C2C(OC)CCC2)=O)C2CCN(C(=O)C(C)C3CCC3)CC12 N1(C(C23N(C(C4OCCN(C)C4)=O)CC(C)(C2)C3)=O)CCCN(C)CCC1 C1(C)(C(=O)NCCCN(C(C(C)CC(N)=O)=O)C2CC2)COc2ccccc2O1 C1(C)(C(=O)NC2CC(C)(NC(c3ncccn3)=O)C2)Oc2ccccc2NC1=O C1(CCC)CN(C(=O)CC(C)C)CC1C(=O)NC(C)(C)CCC1CC1 Cn1nc(CNC(C2CCCC(C)(C)C2)=O)c2c1CCN(C(=O)C1=CCOC1)C2 n1(CC(=O)NCCC2(CNC(=O)CC3CCC4CC34)CC2)nnc2ccccc12 O=C(CCCCCBr)N1CCCCC1CCc1cn(-c2ccc(Cl)nc2Cl)nn1 C(=O)(C(C)C(C)(C)C)NCC1(CNC(C(C2CC2)OC)=O)CC1 C(=O)(CC(=O)NCCC1CCCN1C(=O)CC1(O)CCOC1)NCC#C S(=O)(=O)(c1c(Cl)cccc1Cl)N(C1CCN(c2ccccc2)C1)C c1(SC(C)C)ccc(C(=O)NCCOC2CCN(C(c3csnn3)=O)C2)cc1 c1(NC(C2CN(C(c3cn(C(C)(C)C)nn3)=O)CCO2)C)c(Cl)cnnc1Cl N1(C(CCCOC)=O)CCC(NC(=O)C=C2CCCCC2)CC1C C1(CNC(C(C=C)OC)=O)CCC2(CN(C(=O)CCCC3OCCO3)C2)O1 C1(NCc2nc(C)sc2)CCC(CNc2ccccn2)CC1 N1(C(CC(C)N(C)C)=O)CCN(C(=O)CCc2csc(Br)c2)CC(O)C1 Cc1coc(C)c1C(N1CC(C)(NC(=O)CNc2nccs2)C1)=O c1(COC)cc(C(=O)NC2CC2NC(c2ccc(C(=O)OC)s2)=O)no1 C(=O)(C(=O)C(C)C)CC.c12nc(c(C)o1)C(=O)NNC2=O c1(C2(CC(=O)NC3(C4CCCC45CC5)CC3)CC2)cc(C)c(Cl)cn1.CCOC c1(C(=O)NCC(CNC(CNC(CCC)=O)=O)F)nnn(CC)c1C C=CCCC(C)(C)C(=O)N(C)CCNC(=O)C(CC=C)c1ccccc1 S(=O)(=O)(c1cccs1)NCC(N1CC(NC(=O)CC2CC2(Cl)Cl)OCC1)=O c1(C(=O)NC2C(C)CN(C(=O)C(=O)C3CCCC3)CC2)cc2n(n1)CCCO2 Cc1cc(OC(C)C(=O)NC2CC(CNC(c3ccnc(S)c3)=O)C2)ccc1Cl CC(Cc1ccccn1)C(=O)NCC(C)(CO)NC(=O)C=Cc1ncc[nH]1 c1(C(C(CC)C)NC(=O)C(=O)Nc2cnn(C(C)C)c2)ccc(Cl)cc1 c1(C(C)NC(=O)C(c2cnn(C)c2)NC(=O)CCC2CC2C)cnccn1.C1CC1 Cc1c[nH]c2ccc(-c3cnc(CC(=O)Nc4cc(F)c(F)cc4Cl)nc3)cc12 C12CCN(C1)C(=O)C(C)NC(C1CCC1)CN(C)C(=O)CC2.N1(CC)CCC1 N1(c2n(-c3cccc(C(=O)OC)c3)nnn2)CCC2(CN(C(C)=O)C2)C1 N1(C(COC)=O)CCN(C(C2CC2c2ccc(F)cc2)=O)C(CS(C)(=O)=O)C1 c1(C(=O)Nc2ncccc2Br)[nH]nc2c(-c3cncs3)cccc12 C1(NC(C2(CC#C)CCC2)=O)C2CCCC1CC(NC(=O)Cc1c[nH]nc1O)C2 CCC(C(=O)N(CC(C)O)CCNC(=O)C1CC1)Sc1ccccc1 C1(C)(CNC(C2(C)CNC(=O)C2)=O)CC(F)(F)CN1C(c1ccc(Cl)c(O)c1)=O C1(CNC(C(C)(O)C2CC2)=O)CC2(CCOCC2)CN1C(C1CCC2CC2CC1)=O C1(C(=O)NCC(CNC(C2CC(=C)C2)=O)OC)CC(CC)=NO1 C(=O)(C(CC(F)F)N(C)C(C1CCCN1CC)=O)NC(c1ccnn1C)CC C1(NC(CCSC)=O)CCOCC1C(=O)NC1CCN(C2CC2)C1=O c1(C(=O)NC(CC)CNC(C23CCC(OC)C2C3)=O)cccc2nc[nH]c12 C#CC1(O)CCCN(C(=O)CC(CC=C)NC(=O)C(COC)N(C)C)C1 c1(C(N(CCN(C(CN2CCC(C)C2)=O)C)C)=O)cnn2c1OCC(O)C2 CCC(CNC(=O)C(O)CCSC)(CC)C(=O)N(CC(C)(C)C)C C1(C(N2CCC(F)(CF)C2)=O)(CC)CCCN1C(c1cn(C)nn1)=O c1(COC)ccc(C(=O)NC2CCC2NC(c2cc(C3CC3)no2)=O)cc1F C1(NC(N2CC=CC2CO)=O)CCOCCC1(F)F C1(COC)N(C(C2CN(C(=O)C(F)(F)CN3CCCC3)CCO2)=O)CC1(C)C Cc1ncnc(C)c1C(=O)NCC(N1CCC(c2cccnn2)C1)=O C#Cc1ccc(C(=O)NC2(C)CCN(C(=O)Cc3ccc(Br)cc3)C2)nc1 CC1CN(C(c2ccc(C(O)CF)cc2)=O)CC1NC(C1(C)CCOCC1)=O c1(C(=O)NC(C)CNC(=O)C(c2cncn2C)O)cc(O)ccc1N C1(CNC(C(C(C)(C)F)(C)F)=O)CCC2(CCNCC2)CC1 CCCCCCC(=O)NCC(C)(CC)NC(c1ccc(O)nc1C)=O c1(OC)ccc(C(=O)NCC2(O)CC(CNC(=O)CN(S(C)(=O)=O)C)C2)cc1 CCC(C(=O)N1CCC(N(C(C2CNC(=O)N2)=O)Cc2ccccc2)C1)OC C1(C(NOC(C(=O)OC)OC)=O)CC12CC(OCC=CC)C2 CCCCCCCC(=O)N1CCC(C(=O)NCCC2(OC)CCC2)C(C)C1 c1(OC)cnc(C(=O)NCC(CC(C)C)NC(=O)CSc2cccc(Cl)c2)cn1 c1(CNC(c2ccn(C)c2)=O)ccc(C(=O)NC2CCNC2=O)nc1 c1(C(N2CCCC2Cn2cccn2)C(=O)NC)ccc([N+](=O)[O-])s1 N1(C(C)(C)C)CCC(NC(=O)Cc2cc(C3CC3)[nH]n2)CC1 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCCC(NC(C2(C(C)C)CCCO2)=O)CC1 C1(N(C(c2n(C(C)C)ncc2)=O)C)CN(C(C2CCCN2C2CC2)=O)CC1O n1(CC)nc(C(=O)NCC(F)CNC(c2c(C)n[nH]c2C)=O)ccc1=O c1(C(=O)NCC(CN(C)C(C2C3CNC(=O)C23)=O)O)coc2c(F)c(Cl)ccc12 C(=O)(C(C)CS(C)(=O)=O)NCC(COC)NC(C1(C(F)(F)F)CC1)=O C1(C2CC2)(CNC(c2ccc3ccoc3c2)=O)CCN(C(=O)C(F)C2CCC2)C1 CC(C)(C)CCC(F)C(=O)NCC1(O)CC(NC(C2(N(C)C)CCC2)=O)C1 CCCCCCN(CCCCCC)Cc1cn(C)nn1 N=C1Nc2ccccc2S(=O)(=O)N1C(c1n[nH]c2cccc(Br)c12)=O c1(OC)c(C(=O)NC2CCN(C(=O)CCCC(C)(C)C)C2C)cc(Br)cc1F N1(C(COCCOC)=O)CCOC(C(C)NC(c2cnn(C3CC3(F)F)c2)=O)C1 c1(NC(C(CCNC(C(C)=C(CC)C)=O)O)=O)cc(C)cc(C)c1O N1(C(CS(=O)(=O)NC)=O)CCCC(CCNC(=O)C2=CCCC2)CC1 c1(N2CCCC(COCC)C2)nc2ccccc2nc1NCCc1cccs1 C#Cc1cc(Br)ccc1NC(=O)C=Cc1cc(F)cc(F)c1 c1(C(N2CCCC(NCC)C2)=O)ccc([N+](=O)[O-])s1 c1(C(C(=O)N(C(C)CNC(=O)CCn2ccnn2)CC)(C)C)cccc(O)c1 C#Cc1ccc(C(=O)NCC2(F)CCCN(C(c3csnc3Cl)=O)C2)cc1C C(CNC(=O)C(Cl)=CCl)(CCNC(c1ccc(F)s1)=O)OC C(=O)(C#CC1CCCCO1)NC1(CC=C)CCN(C(=O)CNC(=O)CC)C1 C(CC(N)=O)(C(=O)NCC(C1CC1)NC(c1ncccn1)=O)NC(CC(C)C)=O N1(c2nnn(C)n2)CCC2(COC(CNc3ccc(NC(=O)CCF)cc3)C2)C1 N1(C(C(C)O)=O)CC2(CCC(C(=O)Nc3nnccc3C(F)(F)F)O2)C1 C(=O)(C(O)C(F)(F)F)N1CC(C(C)NC(c2cc(Cl)cnn2)=O)OCC1 C1(C(=O)NCc2c(C)occ2)CC(N=[N+]=[N-])CN1C(c1ccoc1)=O N1(C(c2c(OCC)ccs2)=O)CCCN(C(C2CCCC23CC3)=O)C(C)C1 c1(OC)ccccc1CC(C)CC(=O)NC1CC(C)N(C(c2cnc(C)[nH]2)=O)C1 N1(C(CCOCC(C)C)=O)CCC2(C1)c1ncn(C)c1CCN2C(=O)C1=CCC1 Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CC(C)N(C(=O)COCC(C)(C)C)C1 C(=O)(C1=CCCCCC1)NC(CC)C(=O)NOCC1(F)CCC1 C1(NC(C(CCC)OC)=O)CCCOC12CCN(C(c1nc(=O)n(C)[nH]1)=O)CC2 c1(C(=O)NCCN(C(c2ccncc2C(C)C)C)CC)csc2ccccc12 CC1CN(C(=O)Cc2ccc(F)cn2)CCN1c1nnc(C2CC2)s1 CC1CN(C(=O)CC2CC(N(C)C)C2)CCN1C(=O)CCc1ccc(CO)cc1 C1(C2CCN(C(=O)C(F)C(C)(F)F)CC2)(NC(CC(C)CC(C)(C)C)=O)CCC1 N1(C(C)C)N=C(C(=O)NC2(CO)CN(C(=O)C(C)(C)C(C)(C)O)C2)CCC1=O c1(CCC(=O)NCC(C)NC(C2CC3C(C2)C3(F)F)=O)ccc([N+](=O)[O-])cc1 C(C)(N=c1nc(C(C)C)[nH]s1)C1CCN(C(c2c(OCC)scc2)=O)CC1 c1(C(=O)NC(CNC(C(C)OCC=C)=O)C2CCC2)cc(C)nc(C)c1O N1(C(C(C(COC)C)C)=O)CC2(CCC(NC(C3CC(OC4CC4)C3)=O)CC2)C1 C(=O)(C(C#N)C(C)C)NC(CC)(C)CNC(=O)CSc1cccc(F)c1 N1(C(c2cn(CCOC)nn2)=O)CC2CCCC(NC(c3cc(C)sn3)=O)C2C1 c1(C(=O)NCC(CNC(C2CC(CC)C2)=O)O)oc2ccccc2c1COC C1(CNC(C2CCN(C(C(CC)N(C)CC)=O)C2)=O)(CN(C)C)CCCCC1 c1ccc(CCOC2(c3noc(CC4COCCO4)n3)CCCC2)cc1 CC#CCCC(=O)NCC1(CO)CCN(C(C2CC23CCCC3)=O)C1 C12(NC(CC3CCC(C#N)C3)=O)CCC(F)(CC1)C2.C12CCC(C1)C(=O)NCC2 C1(OC)CC(CCNC(=O)C(=O)N(C)C)N(C(c2cncc(C)n2)=O)C1 c1(CCNC(C2(CC=C)CC2)=O)ccc(F)nc1 C(=O)(C1CCCn2c(C)nnc21)N1C2C(NC(CNS(CC)(=O)=O)=O)(CCC2)CC1 C(=O)(C1=CCC2CCC1N2C(C1CC=CC(O)C1)=O)NCC(CC)N(C)C c1(C(=O)NC2CN(Cc3ccc(C)cc3Br)C2)cnn2c1CC(C)CC2 N1(C(C(C=C)(F)F)=O)CCC(F)(C(=O)NC(c2cnccc2C)C)CC1 C1(NC(C2C(OC)C2)=O)CC2CC(NC(=O)COc3ccccc3F)CC2C1 c1(C(N2CCN(C(C(CCC)NC(C)=O)=O)CC2CC)=O)cc2occc2n1C C1(C(N(C(CC(=O)OC)C)C)=O)CCCN(C(=O)CCCSC2CC2)C1 N1(c2nc(Cl)nc(C)c2F)CC(CNC(=O)CC23COC(C)(C2)C3)OC2(CCC2)C1 C12(C(=O)NC3CCCC(NC(c4cc(Cl)cc(Cl)c4)=O)C3)CC3CC1C2C3O c1(C(N2C(CNC(C(C(C)(C)O)F)=O)CC(O)C2)=O)ccc([N+](=O)[O-])c(O)c1 C(=O)(C1=CC2CC(C1)CC2O)NC1C(CNC(CC(C)(F)F)=O)COC1 n1(CCOC)nc(C(=O)N(C)CCN(C)C(c2csc(C(F)F)c2)=O)cc1C c1(CC)ccc(C(N2CC(O)(CNC(C3C4CCCC34)=O)C2)=O)c(C)c1 C(CC(=O)N1CCC(C(=O)OC)O1)=CCNC(C(C=C)(C)CC)=O C#CC1(NC(=O)CCCCCCNC(=O)CC(=O)OCC)CC2CCCC12 C1(C(NOCC(C)C)=O)CCN(C(C2COC(C)C2)=O)CC1 c1(Oc2ccccc2)ncnc2ccccc12.[O-][n+]1cnc2c(c1)N2 C(=O)(C1=CCOCC1)N1C(Cn2cc(C3CN(C(CC(=C=C)C)=O)C3)nn2)CCC1 C1(C)(C(=O)NC2(C(=O)NC(c3cncnc3)C)CCSC2)C=CCCC1 C(=O)(CCC(=O)c1cc(C)sc1C)NCCCNC(C(C)NC(CC)=O)=O c1(C(=O)NCC=CCl)cc(CNC(C2CC3CC3C2)=O)no1 CC1=NOC2(C1)CC(C(=O)NCCCCCCNc1ncc(Cl)cn1)C2 N1(C(c2c(F)ccc(C#C)c2)=O)CCCN(C(=O)CCOCC2CC2)CC1CO c1(N2CCC(NC(CN3C(CCN(C)C)CCC3)=O)C2)ccc(Br)cc1 CC(CC(F)F)C(=O)NC(C(CC#C)O)=O.c12cnn(C)c1C(=O)NOCC2 C1(CNC(CCN(OCC)CC)=O)CCCCN(C(=O)CCC(C)N(C)C)C1 C1(C(=O)OC)CCCC1N(C(CC1CCC2CC12)C(=O)NCCC1CCCC1)C C(N=c1nc(N2Cc3c[nH]nc3C2)c2sccc2[nH]1)C1CC(F)(F)C1 c1(CNC(CCNC(N)=O)=O)cc[nH]c1C(N1CCC(F)C1)=O C1(C)(n2c(COCCC=C)nc(-c3cncc(F)c3)n2)CCS(=O)(=O)C1 c1(N(CCCOC)C)cc(=NCc2ccc(OC)c(Br)c2)cc[nH]1 N1(C(C(CC=C)CNC(c2c[nH]c(=NC)o2)=O)=O)CC(O)(C2CCC2)C1 c1(C(N2CC(NC(COC)=O)C(C(F)(F)F)CC2)=O)cnc2n1CCOC2 N1(C(C(C)=C2CCC2)=O)CCC2(CCN(C(=O)Cn3ncc(C#N)c3N)C2)C1 Cc1nccc(CCC(N2CCC(CO)(NC(=O)COCCO)C2)=O)n1 c1(Cc2onc(-c3ccc(Br)cc3)n2)nc2c(s1)CNC2 C(=O)(C(O)(C(F)(F)F)C1CC1)NCCN(C(c1n(C(C)C)ccn1)=O)C c1(CC(=O)NCC(CC=C)NC(c2cc(Cl)c[nH]2)=O)cccc(C)c1 CN1CCN(C(=O)Cc2ccc(O)c(Cl)c2)CC1CNC(c1nc(Br)c[nH]1)=O C1(C(=O)NCCNC(c2c(N)sc3c2CCC3)=O)Cc2cc(F)cc(F)c2O1 C1(C(=O)NC(COC)CNC(c2cnc(SC)s2)=O)CCCSC1C c1(OC)cc(C(N2CC(CNC(c3coc(SC)n3)=O)C(C)(C)C2)=O)cc(F)c1 O=C1NC2(CCN(C(C3CCC=CO3)C=O)CC2)CO1.C1CCOC1 N1(C(C(C)(C)OC)=O)CCCC(CNC(=O)C(C)(C)C2CCCOC2)C1 N1(c2ncc(C(=O)OC)nc2)CC(NC(c2cnc(C(C)(C)C)o2)=O)C(C)(C)C1 C(=O)(C(COC)CC(C)C)NCC#CC(=O)NCc1c(C)nn(CC)c1C N1(C(c2cc(Cl)sc2Cl)=O)CCN(Cc2c(O)cccc2Cl)C(CO)C1 c1(NC)cncc(C(=O)NC(C)C=CC(=O)N(C(C(N)=O)C2CC2)C)c1 c1(C(=O)NC2CC3CN(C(C4(C)CC=CC4)=O)CC32)ccc2c(c1)C(=O)NCC2 c1(C(=O)NCCCNC(C2CC=CCC2)=O)cnc(C(F)(F)F)cn1 C(=O)(C#CC1CCOCC1)NCCN(C)C(C1CCN(c2nc(=N)[nH][nH]2)C1)=O c1(C(N2CC(N(C(CCC=CCC=C)=O)CC)C2)=O)cnc(Cl)c(C2CC2)c1 N1(C(C2(F)C(C)C2)=O)CC2(C)CN(C(c3cccc4c3NCCC4)=O)CC2(C)C1 C(=O)(C(O)CC[S+](C)C)N1CCC(OC)(CNC(=O)CCC(=O)N(C)C(C)C)C1 c1(C(=O)NCCCC(C)NC(c2cc(O)no2)=O)cc(Cl)cc(Cl)c1 c1(COC)cc(N2CCCC(NC(c3ccnn3C)=O)C2)ncn1 C=C(CNC(=O)CC(CNC(=O)C(C)(F)C(C)(C)F)OC)c1ccccc1 c1(C(=O)NCC2(O)CC(NC(c3cc(C(=O)OC)sc3)=O)C2)cccc(=O)o1 c1(C(N2CC(NC(=O)CC3CCOC3=O)C3(C2)CC3)=O)cc[nH]c2nccc1-2 N1(C(Cc2ccc(OC)cn2)=O)CC=C(CNC(=O)C(C)S(C)(=O)=O)CC1 CN1CCN(C(=O)CSCCC#N)C(C(=O)Nc2ccc(F)cc2C2CC2)C1 C12(NC(c3c(CC)con3)=O)CCN(C(C3CCC(C)=C(C)C3)=O)CC1C2 c1(CC)noc(-n2cc(-c3cccc(C)c3Oc3ccccc3)nn2)c1C#N N1(C(C(CCC#C)O)=O)CCOC2(CCN(C(c3cc(CC)ccn3)=O)C2)C1 C(=O)(C(C)C(=O)NC1CC1)NCC(C1CCC1)NC(CC1(CSC)CC1)=O C=C(C)C(CC(=O)N1CCC(N(C2CCCOCC2)C(=O)OC)CC1)OCC C12(C(N3CCC(N(C(C4(O)CC(C)(C)C4)=O)CC)CC3)=O)OCCCC1C2(F)F c1(C(N(C2CN(C(C(CC)n3cncn3)=O)C2)C)=O)c[nH]c(=N)cc1C c1(C(N2C(CCNC(C3C(=C)CC3)=O)CCC2)=O)cc(F)c(F)c(N)c1Cl C1(CCNC(C2(C)CC(=C)C2)=O)CN(C(C2CC(CC)=NO2)=O)CCS1(=O)=O CCC(C)(C)C(C)NC(=O)C(CN(C)C)NC(c1ccc(C(F)F)o1)=O N1(C(C(=O)OC)=O)CCN(C(=O)CCn2ccnn2)CC1.C1(=O)CSCCN1 C1(NC(c2c(C)nns2)=O)CN(C(=O)C(C2CCCCC2)O)CC1CC1CC1 Cc1cccc2c(C(=O)NC3CCN(C(C45CC(F)(CO4)C5)=O)C3)coc12 C(=O)(C1=CCCC1C)NCC(CC)NC(=O)CCc1ccc(F)c(F)c1 CCN(OC)C(=O)CNC(C1CCC=CC1NC(=O)C(C)CC(N)=O)=O C1(NC(=O)NC(C)(C)C)(CC)CCCNC1.c1(CC)[nH]nc(C(=O)OC)c1Br CC(CCO)N=c1[nH]c(=NCC2(c3ccccc3F)CC2)[nH]c2c1CCCC2 N1(C(C2N(C=O)CCC2)=O)CCCC(CC)C1C(=O)NCC=CCl c1(C(=O)NC(C2(O)CN(C(=O)CC3CC4CCC3O4)C2)C)cccc(Cl)c1F N1(C(c2c(CC)nccn2)=O)CC(NC(C23CCC(CC2)CC3)=O)CC(C)C1 c1(COC)n[nH]c(=NC2CC(NC(=O)C(F)CC3CC3)C23CCC3)s1 c1(-c2c(C)noc2)ccc(NC(C2CCC(CN)C2)=O)cc1 C=CCC(CC)C(=O)N1Cc2ncsc2C1.c12ocnc1C(=O)OC2 c1(OC)c(C(=O)NC2CCC(N(C(=O)C(O)C3CC3)C)CC2)ccnc1F N1(C(CS(CCC)(=O)=O)=O)CCC2(CC1)CC(NC(=O)CSc1cc(C)on1)C2 C1(OCCNC(c2nocc2C2CC2)=O)CCN(C(=O)CCC2CC2(C)C)C1 CN=c1cc(C(N2CCOC(CN(C)C(C3CC4(C3)CC4F)=O)C2)=O)cc[nH]1 CC1(C)CCCC(C(=O)NC2CCCC2NC(C2(c3nn[nH]n3)CC(O)C2)=O)C1 CC1(C(=O)NCC2(NC(C3CC(=O)N(CC(F)(F)F)C3)=O)CC2)CCCC1(F)F C(c1c(F)cccc1F)=CC(=O)NC12CN(C(C(C)NC(C3CCC3)=O)=O)C(C1)C2 N1(C(Cc2c(C)n(C)cn2)=O)CC(C2CC2)(C(=O)NC2CCNC2=O)C1 Cc1ccc(C=CC(=O)NC2CCC2NC(=O)CN(c2ncccn2)C2CC2)s1 Cn1nc(C(N2CC3CC(C2)C3NC(C2CCCO2)=O)=O)c2c1CCCC2 C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NCCN(C(CC=C=C)=O)CCOCCO c1(CC(=O)NC2C3(CN(C(CN4CC(C)C4)=O)C3)CC2)ccc2c(c1)NC(=O)C2 N1(C(CC)=O)CCCC2(CCN(C(C3CC4(F)CC3C4)=O)C2)C1 c1(C(N2CCC(NC(C3C(C)C3)=O)C(CO)CC2)=O)ncc2ccccc2c1N N1(C(=O)CC2CCCC2O)CC2CCN(C(=O)CCCc3ccncc3)CC12 C12CN(CC13CCC3)C(=O)Nc1cc(sn1)C(=O)N2.CC(C)CC1(CC2CC2)CC1 CCCCS(=O)(=O)N1CCCC1C(=O)NC1COCC1CNC(=O)CC(F)F N1(C(C)=O)CCN(C(=O)CCn2cc(-c3cnc(C)o3)nn2)C(C)C1 c1(C(C(=O)NC2CCC2)N(CCCCOC)C)ccc(OC)c(Br)c1 C1(C(N(CCC(=O)OC)CC=C)=O)CCCCN1C(=O)CCC1CCCCO1 S(=O)(=O)(c1ccc(NC(C2CCC3C(CC2)C3(F)F)=O)c(C(F)(F)F)c1)N(C)C c1(CC(C(=O)N(C)CC2CCCC3CC23)NC(c2ccco2)=O)cnn(C)c1O CC(C)C(CC(=O)N1Cc2ncsc2C1)NC(C1CCC2(CCC2)O1)=O C12(C(=O)NC3C(CNC(c4n(CCC)ccc4)=O)CCCC3)CC(C1)S(=O)(=O)C2 CCCC(C(=O)N1C(C(=O)NCc2cc(C)c(C)s2)CCC1C)OC c1(N2CCC(CNC(=O)C(F)CC3CCC3)C2)ccc(N)cc1 c1(OC)[nH]c(=N)nc2sc(C(=O)N(CCC(C)NC(=O)C(C)(C)O)C)cc12 OCC(F)(F)C(c1ccccc1)NC1CC1C(F)F c1(CC(=O)NCC2CN(C(=O)CCc3cnn[nH]3)CC2O)ccc(O)c(Cl)c1 c1(C(=O)OC2CCNC2=O)ccc(N(CC(=O)OC(C)(C)C)C)cc1.C#CCSC c1(COC)cc(S(=O)(=O)N2CC3(CCC(NC(=O)CO)C3)C2)ccc1C N1(C(CCCOCC=C)=O)CCCC(CNC(=O)C=CI)C1 Cn1ccc(=O)c(C(=O)NCC2CCCC(NC(c3ccc(Cl)[nH]3)=O)C2)c1 c1(NC(C(C)N(C)C)=O)ccc(CNC(c2csc(C(C)(F)F)n2)=O)nc1 c1(C(N(C2CN(C(C3C(OCC)C3C)=O)C2)C)=O)ccn2c(C)cc(C)nc12 N1(C(CC(C)(C)C)=O)CCC2CN(C(C3(N4CCCC4)CCC3)=O)CCC2C1 N1(C(C2C(NC(C(C=C=C)C)=O)CCCCC2)=O)CCC2(CCCO2)C1 c1(CC(=O)NC(C)CNC(=O)CC2CCN(C)C2=O)cc(F)ccc1Br CC(C)(O)C(F)(F)CNC(c1ccc(CNC(c2cnnn2C2CC2)=O)o1)=O Cc1cc(C(=O)NCC2CN(C(=O)C=Cc3cc[nH]n3)CCCO2)c(C)c(C)c1 N#Cc1ccc(C(N2CCN(C(C3CC4CCC3O4)=O)CC2CO)=O)c(Cl)c1 c1(C(=O)NC(CC(C)NC(C2(CC)CCC2)=O)C)ccc(C2=CCOCC2)cc1 N1(C(c2cccc(C)c2)=O)CCC(CNC(=O)CC(O)C2CC2)C(F)(F)CC1 C(=O)(C1SCCc2ccccc21)NCC1(O)CC(CNC(CCC)=O)C1 N1(C(C(C)NC(N)=O)=O)CC2CCN(Cc3ccc(Cl)o3)CC2C1 Cc1ccc2c(c1)CN(C(=O)CC1CC1CNC(=O)CC1CCCSC1)C2 c12cc(ccc1C)NC(=O)N2.c1(Cn2c(C)nnn2)cnc(N(C)C)cc1C c1(OC)c(N2CC3CN(C(C4CC4(Cl)Cl)=O)CC3C2)nc(C2CCCC2)nc1C C1(CC(N2C(C3(NC(=O)CCCNC(N)=O)CC3)CCC2)=O)CCC(F)(F)CC1 C#Cc1cc(F)c(C(=O)NC23CCC(NC(c4nnc(C)s4)=O)(CC2)C3)cc1F N1(C(c2c(OC)cc(C)cn2)=O)CC2(C1)SCCC2NC(=O)Cc1ccsc1C c1(OC)ccc2c(C(=O)NCC3C=CC(NC(=O)COCCF)C3)n[nH]c2c1 C1(NC(c2cc(C(C)C)no2)=O)CC2(C1)CC(NC(=O)C=CC(F)(F)F)C2 c1(C(=O)NCCCCCN(C(CSCCCC)=O)C)ccc(C2CC2)nn1 N1(C(=O)C2=COCCO2)CCC(C2CCN(C(c3c[nH]nc3F)=O)C2)C1 C(=O)(C(C)(O)CCN(C)C)N1CC(CNC(C2ON=C(CC)C2)=O)OCC1 N1(C(C(C)NC(N)=O)=O)CCCC(N(C)C(c2cc(=O)cc[nH]2)=O)CC1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCCN(C(CCSCC(N)=O)=O)CC1 C(=O)(C(C)CC(F)(F)F)NC(c1ccccc1)CNC(c1c(CC)c[nH]c1)=O c1(C(N2CCC3(NC(CCSCC(C)C)=O)C(C2)C3)=O)cc([N+](=O)[O-])cn1C C1(CC(=O)NCC)COc2ccc(Br)cc2C1.c12cn(nn1)CC(C)SCC2 C1(CNC(C(CC)(C)O)=O)CC2(CC2)CN1C(=O)Cn1ncnn1 C(=O)(C(C)(O)CC)NCC(CNC(C(CC)C1CCC(=O)N1)=O)C Cc1[nH]nc2c(-c3cc(C(=O)NCC4CCCO4)c4n[nH]cc4c3)cccc12 N1(C(C(c2ccc(F)cc2)OC)=O)CCN(C(C2(C(C)(F)F)CC2)=O)CC1CO CC1CN(C(C2CCC(C)O2)=O)C(C)CN1C(c1cccc(N)c1Br)=O c1(CC(C)C(=O)N(C2CN(C(C3CCN(C(N)=O)CC3)=O)C2)C)ccccc1F n1(COC)nccc1C(=O)NCC1CCCC1NC(=O)C(=O)NC(C)C C1(C(=O)NC2CCN(C(c3cc(OC)n[nH]3)=O)CC2F)CCc2n[nH]cc2C1C Cc1csc2c(COC(c3cnn(C4CCCC4)c3)=O)cccc12 c1(C(N2CC3CCC(C2)N3C(C23COCC2C3)=O)=O)nnn2c1CSCC2 N1(C(CCOC)=O)CCC2(CC1)CCN(C(=O)Cc1cccc(Cl)c1)C2 Cc1ncc([N+](=O)[O-])cc1C(=O)NC(C(C)NC(C1(CC(C)C)CC1)=O)C(C)C C1(N(C(c2nc(C)sc2)=O)C)CC2CC1N(C(C13CC4CC1C3C4O)=O)C2 CCCC(C(=O)NCC(C)NC(=O)C(F)=C1CCCC1)c1ccccc1 c1(NC(=O)CC2CC(NC(c3ccoc3)=O)C2)ccccc1Sc1ccccc1 C1(CNC(c2nc(C)sc2)=O)CCN(C(=O)C2=NOC(C)C2)CC1(F)F N1(C(C(C(C)O)C)=O)CCN(C(c2cc(C(F)(F)F)n(C)n2)=O)C(CO)C1 C(C(=O)NCCCCCCNC(=O)CSC(C)(C)C)(C(C)C)OC C(=O)(C#CC1CCOCC1)N(C)CCNC(C1CCC1)=O c1(OC)cc(NC(C2(F)CN(Cc3ccc(F)cn3)C2)=O)ccc1Cl c1(NC(C2CCCCN2C(c2snc(Cl)c2Cl)=O)=O)cc(Cl)c(O)cc1Cl N1(C(C(F)=CCOC)=O)CC(n2cc(CN3CCCCC3)nn2)C(C)C1 C1(C(=O)NCc2cc(C)on2)CN(C(=O)C(=O)C(C)C)CC12CC2 Cc1cc(N)n2ncc(C(N3CCCCCC3CNC(c3ccon3)=O)=O)c2n1 c1(OC)ccc2c(c1)CC(N)O2.n1(C(N2CCC2Cn2nccn2)=O)cc(C)nn1 C1(NC(CCCC)=O)CCC(N(C(=O)CCC2CC2(F)F)C)CC1 c1(NC(N2CCC(O)(c3ccccc3)C(O)C2)=O)cnc2c(c1)OCO2 N1(C(COCCCOC)=O)CC(CC(=O)NCc2nncn2C)C(C)C1 N1(C(=O)CCc2ncc[nH]2)CCN(C(c2cnc(C(F)(F)F)s2)=O)CC1 c1(C(N2C(CN(C(C(CC3CCCCC3)OC)=O)C)CCC2)=O)ccc(Cl)cc1 C(=O)(CCCC(C)=O)NCC1(O)CCN(C(C2(CCCC)CCC2)=O)C1 N1(C(C2CCC(C)CC2)=O)CCCN(C(C2(F)CCC2)=O)CC1 CC[Si](C)(C)CCCN(S(N)(=O)=O)CCN(C)CC.C(C(C(C)(C)C)OC1CCCC1)N N1(C(c2ccc(O)nc2Cl)=O)CC(CO)C2(C1)CN(C(C13COCC1C3)=O)C2 c1(C(N2CCCCCC(NC(=O)Cc3ccon3)C2)=O)cccc2c1CCO2 N1(C(c2nc(C)oc2C)=O)C2CCC(C2)C1C(N1CCC1CN=[N+]=[N-])=O Cc1nc(N2CC3CC(NC(C4CCC(=O)NC4)=O)C3C2)ccc1[N+](=O)[O-] N1(C(C(C)SC)=O)CCC2(CCCN2C(C2CCC(=O)NC2)=O)C1 c1(C(=O)NCC2(C(=O)NCC3CC3C(C)C)C(C(C)C)C2)cc(C#N)c[nH]1 CCC(CC(=O)NCCC1CCCN1C(c1cccnn1)=O)C1CCC1 C1(C)(CNC(CN(C(=O)OC)C)=O)CCN(C(c2[nH]cnc2C)=O)C1 N1(C(CC2C(C)(C)CCCO2)=O)CC2CCC(C1)N2C(=O)C1=CCSC1 CC(=O)CCCCC(=O)NC(C(=O)NCC1=CCCOC1)c1ccoc1 Cc1cn2c(C(=O)N(CC(O)CNC(C3CCS(=O)(=O)N3)=O)C)cnc2s1 C1(N(C(CC2N(C(c3c(C)nn(C)c3)=O)CCC2)=O)C)CCCC(C)C1C C1(CNC(=O)Cc2cnc[nH]2)C(O)C(O)CN1C(C1CCCCC(=O)N1)=O C(=O)(CC(C)(C)CC(F)(F)F)NC1(C)CCC(NC(c2cn(CC)nc2)=O)CC1 CCCCCCCC(=O)N1CC(CNC(C2SCCCS2)=O)CC1(C)C CC1CN(C(c2cccc(-c3ccsc3)c2)=O)CCN1C(c1cccs1)=O CC(C)C(CCC(=O)NC1CCC(=O)NC1=O)NC(c1cc[nH]c1)=O c1(C(N2CCCCC(C)C2)C(=O)NCCC2CC2)nc2ccccc2s1 c1(CCC(N2CCC(C(C)NC(C3CCCCC3)=O)CC2)=O)cccc(F)c1F C1(CNC(C(=O)N(CC#C)C(C)C)=O)(Cc2ccc(Cl)cc2)CCN(C)CC1 N#Cc1cc(C(=O)NCCCSN2C(Cc3ccc(C(=O)O)s3)CCC2)cs1 c1(CC)ccc2c(C(=O)NC3CN(c4ccccc4)C3)coc2c1 C1(C(=O)OCC)CC(C)CN(C(=O)C(CN)C(C)C)C1 N1(C(C(C(C)C)SC)=O)C(C)CC2CN(C(C3CN(S(C)(=O)=O)C3)=O)CC12 C(CCCCC(=O)NCC1(C)NC(=O)NC1=O)NC(C1(C)CC(C)C1)=O CCC(CN(C)C)CC(=O)N(CCCCNC(c1nn(CC)nc1C)=O)C C#Cc1cc(C(=O)NC(C)(C)C(C)NC(C2COCCO2)=O)ccc1C C(C)(C)(C(F)(F)F)NC(CCC1N(C(c2c(C)nsc2)=O)CCC1)=O N1(C(CC=CCN(C(=O)CC2CSC2)C)=O)CCOC(C2CCC2)C1 c1(NC(C2(CC)CCCN2C(c2cc(C(C)C)[nH]n2)=O)=O)cnc2ncnn2c1 C(=O)(C(C)(C)CCO)N(C(C1CCC1)C)C.n12cc(nn1)-c1c[nH]nc1CC2 C1(OC)CC2(C1)CC2C(=O)NCC1C2CN(Cc3sccc3Br)CC12 c1(CCCC(=O)NC(CN(C(C2CCC23CCC3)=O)CC)C)ccc(O)cc1 c1(OC)cc(F)c(C(=O)NCC(C(C)C)NC(c2cc(C)cnc2N)=O)c(F)c1 N1(C(C2=CCC(C)CC2)=O)CCCC2(CCCN2C(C2CCS(=O)(=O)CC2)=O)C1 CN1C(=O)C(F)CC1C(=O)NC1(CNC(=O)C(c2ccc(F)cc2)(C)F)CC1 c1(C(N2CC(OCCNC(CCc3ccn(C)c3)=O)C2)=O)ccnc2ccsc12 C1(C(N2CC(CCCCNC(CCc3cc(C)no3)=O)C2)=O)CCOC(=O)CC1 S(=O)(=O)(c1ccc(NCC(C)(C)CC(F)(F)F)nc1)NC(CCC)C(C)O c1(CCC(=O)NC(C2N(C(C(C)OC)=O)CCC2)C)ccncc1Br c1(NC)cnccc1C(=O)NCC(C)CNC(C1COCCN1C(C)=O)=O C1(CCC(=O)NCC(CC)C#N)CCCCN(C(C2CC(F)CN2C)=O)C1 c1(C(=O)NCCN(C(C2N(CCC)CCC2)=O)C)ccc(Br)cc1Cl C1(CC(=O)NC(C(C)C)CNC(C2CC3(C2)CC3F)=O)CCCCC1(C)C N#Cc1ccc(C(N2CCCC(O)(CNC(c3ccccc3Cl)=O)C2)=O)cc1F N1(C(=O)NCC(C)C2CC2)CCCC2(CC1)CNC(=O)O2 C(=O)(C(F)Cc1ccccc1)NCCN(C(c1ccsc1Br)=O)CC c1(C(=O)NCCCN(C(=O)CN2CCOCC2)C2CC2)ccc(OC(F)F)cc1 N1(C(CN(C)S(N)(=O)=O)=O)CCc2[nH]nc(CNC(C3(C)CNC(=O)C3)=O)c2C1 N1(C(c2cccc3cnccc23)C(=O)NCC=C)CCC(S(=O)(=O)C(C)C)CC1 C1(NC(CNCC(C)F)=O)CCCC1C CCC(CC)C(F)C(=O)NC(C)(C)C=CC(N1CCCC(CC2CC2)C1)=O CC1CN(C(=O)Cc2cccc(Cl)c2F)CCN1C(c1cc(F)ccc1F)=O c1(-n2ccc(NC(=O)Nc3cc(C(=O)NC)[nH]n3)n2)ccccc1C CC1OC(C)C(C(=O)NCC2CN(C(C3CCCN3C(=O)C3CC3)=O)C2)C1C N1(C(CC2CC(C)OC2C)=O)CCC2(C1)CN(C(C1(C)CCC(=O)NC1)=O)C2 C(C(C(C)(C)C)NC(c1cncc(F)n1)=O)NC(C(C1CCC(=O)N1)C)=O N1(C(CC2C=NN(C)C2=O)=O)CCC2(C)CN(C(c3ncoc3C3CC3)=O)CC12 C(=O)(C1=CCCCC1C)N(CC(CC)NC(c1cnc(OC)c(OC)c1)=O)CC C1(C(=O)NC2CCN(CCCNC(C(CC)(C)O)=O)C2)CC2(CCCC2)CO1 C1(CNC(C(C)CC2CCCO2)=O)CCC(NC(c2cc[nH]c2)=O)CC1 c1(C(=O)NCCNC(c2c(OC)cccc2Br)=O)ccnc2c1CCO2 N1(C(CNC(CC)=O)=O)CC(CNC(C2(c3cc[nH]n3)CC2)=O)C(C)C1 C(C(C)C(=O)NCCN(C(=O)CC1(CO)CC1)C)OCC C1(C(=O)NC(COCC)C(C)C)CC(CC)CCN1C(c1ccnc(O)c1)=O c1(OC)ccc(C#N)cc1CN1CCC(N(C(=O)C(c2ccccc2)C)C)C1 Cc1ccc(-n2nc3nc2C3)cc1Cl.n1(C(C)C2CC2)cc(Br)cn1 c1(C(=O)NCC(O)CNC(C2CCCC2(F)F)=O)c(C(F)F)nc2n1CCCC2 c12ccc3c(c1)CCCC3NC2=O.c1(C(=O)OC)ccc(F)cc1OCC1CC1 C(=O)(C(C(C)(C)O)NC(c1ccn(C(F)F)n1)=O)NC(C=C)C C1(NC(CCCSC)c2nnnn2CCC2(C)CC2)CCOC2(CCOCC2)C1 c1(CC(=O)N(CC(C)NC(c2cncc(CC)c2)=O)C)ccc(C)c(O)c1 N(C1CC(C)(C)Oc2ccc(F)cc21)C(=O)NC12OCC(C#C)(C1)C2 CC1(C)CCC=C1C(=O)NC1CC2CC(NC(=O)CSCCN=O)C2C1 O=S(=O)(c1[nH]c(=NC2CCn3ncnc3C2)ccc1Br)NC1CCN(CC2CC2)C1 C1(CC(=O)NC(CC)CC)CCCN1N(CC(C)C)C(=O)OC C(=O)(C(C)CCCC(C)=O)N1C(CC=C)(C(N2CCC(CCOC)C2)=O)CCC1 C(=O)(C(O)CCc1ccccc1)NC(CNC(c1c(CC)nc[nH]1)=O)C1CCC1 C1(C(=O)NCCN(C(=O)CC2CCCC(=O)C2)CC)CC2OC1C1CC21 C1(C2CCN(C(c3cnns3)=O)CC2)(NC(=O)Cn2cnccc2=O)CCC1 Cc1c(C(=O)NC(C)(C)CNC(=O)C(C)O)[nH]c2c(C)cccc12 N1(C(CCOC)=O)CCOCC1CNC(=O)C(C)(C)Cc1ccccc1 C1(C(=O)NCCCN(CC(C)C)C(c2c(C)nc(CC)o2)=O)CC(=O)OC1(C)C N1(C(C2(COC)CC2)=O)CC(OC)C(NC(=O)CC2CC3CC3C2)C1 C12(NC(=O)COC3CCCCC3)CCCC1N(C(=O)CCc1ccco1)CCC2 N1(C(CC(C)F)=O)CCC(C)(C(=O)NCCN2CC3CC3C2)CC1 N1(C(C(C2CCC2)OCC)=O)CCC2CCCC12C(=O)NC1CC12CCCCC2 Cc1ccc(C(N2CC(CC(=O)Nc3ccc(C)c(Br)n3)C2)=O)c(O)c1 CC1CC(C(=O)NC2CCCC2CNC(C2CN3CCN2CC3)=O)CCS1(=O)=O c1(NCc2c([N+](=O)[O-])cccc2)nc(N2CCC(F)C2)c2ccccc2n1 N1(C(c2cccc(C)c2)=O)CCC2(CCCN(C(c3ccnn3C(C)C)=O)C2)C1 CC1CCC(NC(C23CCN(CC2)C3)=O)CN1C(C1CCN(CC(F)F)CC1)=O c1(C(=O)NC(C2CCN(C(C3C(C)C3C)=O)C2)C)cn(C2CCC2)cn1 CC1CCN(C(C2CNCCN2c2ncnc3occc23)=O)CC1(F)F CCS(=O)(=O)c1ccccc1CN(C(=O)C(N)=O)C Cc1cc2c(C(N3CC(CNC(C4CCC4)=O)OC(C)(C)C3)=O)cccc2o1 C1(CC=C)(NC(=O)Cc2cc(C)sc2C)CCCN(C(=O)CC(C)SC)C1 Cc1nc(CNC(c2ccc[n+]([O-])c2)=O)oc1C(=O)NCC(C1CCCO1)O C1(F)(C(N2C(CNC(C(c3cn(C(C)(C)C)nc3)=O)=O)CC2)=O)CC2(CCC2)C1 C1(N(C(c2c(C)ncs2)=O)C)CCN(C(=O)CC2CC=CCC2)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N1C(CNC(CC(C)(C)C(F)F)=O)CC(F)(F)C1 c1(C(=O)NCC2(CN(C)CC)CC2)cccc(C(N)=O)n1.C12(CCC1)CC(=O)N2 C1(CNC(=O)NCCC(CC)(F)F)CC(OC)C12CCC2 N1(C(c2cnc(C)[nH]2)=O)CCC(CO)(CNC(C2C3CC3C3CC23)=O)CC1 CC(CN(C)C)CC(=O)NC1CCOCC1NC(c1conc1C(C)(C)C)=O C(=O)(C#CC1(C)CCCO1)N1CC2N(C(CC3C=NN(C)C3=O)=O)C(C2)C1 C1(O)(CNC(C2CC(NS(C)(=O)=O)C2)=O)CCCN(C(C2CC23CCC3)=O)C1 Cc1cc(C(N2CCCCC2CN(C(=O)CCC2CCC(=O)NC2)C)=O)n(C)n1 C1(C(=O)NC(CCN(CC)CC)C)CC2(CC2)CN1C(c1oc(C)nc1C)=O C1(C(=O)NC(C(CO)NC(c2c(C)nn[nH]2)=O)C)Cc2cc(Br)ccc2O1 CC1(C)CC(c2ccc(F)cc2)(C(=O)N(CCNC(C2CC2C#N)=O)C2CC2)C1 CC(CNC(=O)CCNC(c1ccc[nH]1)=O)CNC(=O)COc1ccsn1 C1(C(=O)NCC(C2CCC2)NC(C2CCC(=O)N2C)=O)(CC)CC(C)(C)C1 c1(C(CC(=O)NC(CC)(C)CNC(c2csnc2C)=O)O)cccc(F)c1 C(=O)(CC(C)CC(C)(C)C)N1CCN(C(c2c(C)ccc(Cl)c2)=O)CC12CC2 C1(C)(CNC(CCc2c(C(=O)OC(C)(C)C)nco2)=O)CCC(NC2CC2)C1 C1(NC(C(c2cnn(C)c2)NC(c2cnc(OC)s2)=O)=O)CCc2ncnn2C1 Cc1c[nH]nc1C1(C(=O)NCC2CCCC2NC(c2cncn2C)=O)CC1.C1CC1 C(=O)(C(C)(C)CC(C)=O)NCC(CNC(C(CC)SC)=O)(C)C O(S(=O)(=O)c1ccsc1-c1ccccc1)c1ccc(-c2cn(C)nc2)cc1 c1(CN=C(NC(C)C)NC(C)(C)C(F)F)ccc(F)c(F)c1 N1(C(C2C(C)(CC)C2)=O)CCOC2(C1)CN(C(c1c[nH]c3nccc-3c1)=O)C2 C(=O)(CCCCCCNC(C1CCCOC1)=O)NCC(CC)CC N1(C(C2CCC(N(C)C)CC2)=O)C2CCC(C2)C1CNC(C1CC(O)CN1C)=O CCC(C)(CNC(=O)C(C)Cn1cccn1)NC(=O)CNC(c1ccccc1)=O C1(NC(CCn2ncc(C)c2)=O)(CO)CCCN(C(C2CC(F)(CO)C2)=O)C1 N1(C(C2(SC)CN(C(=O)CC=CC(C)(C)C)C2)=O)CCC(=O)N(C)CC1 N1(C(c2c(C)oc(CO)c2)=O)CCC2(C)CN(C(=O)C(C)CN(C)C)CC12 CC1CN(C(C2C3(CC3)C23CC3)=O)CC1NC(=O)C=Cc1cnc[nH]1 C1(C(=O)NCC(C)(C)OCC(=O)NC(c2nnc(C)s2)C)CC(=O)NC(C)C1 C(=O)(C1=C(C)C(C)(C)OC1=O)NCCCC(C)NC(CC(CC)O)=O c1(SC)ccc(C(N2CCSC(C(=O)Nc3nc(O)cs3)C2)=O)c(C)c1 c1(C(N2CC(C(=O)NCCNC(CC)=O)C2)=O)ccc(-n2c(C)ccc2C)cc1 C1(CNC(c2c[nH]c(Br)c2)=O)C(C2CC2)CCN1C(c1ccoc1Cl)=O C1(NC(C2(CC=C)COC2)=O)CCCN(C(C2CC(=O)N(CCOC)C2)=O)CC1 c1(NCC2OCC(CNC(c3cc(CC)n(CCO)n3)=O)C2)nnc(C)c(C)n1 c1(C(N(C2CCC(NC(c3ccc(F)cc3O)=O)C2)C)=O)ccn2cnnc2c1 C1(NC(c2scc(COC)c2)=O)CN(C(c2cc(=O)cc[nH]2)=O)CCC1C n1(CCC(C)C)cccc1C(=O)NCC(c1ccncc1)O C(=O)(C(C)(F)C(C)(C)F)NCC1(NC(c2c(C)scn2)=O)CCCCCC1 C1(CNC(C2(CC)COC2)=O)C2CN(C(=O)C=Cc3ccc(C)o3)CC12 c1(C(N2CCC(=CCNC(=O)Cc3cccc(O)c3)CC2)=O)ccc(Br)cc1F c1(C(N2CC(C)(NC(C(C(CC)C)N(C)C)=O)C2)=O)c(OC)ccc2c1CCC2 N1(C(C2(COC)CC2)=O)CC2CC(O)C1C2NC(c1cc(C(F)F)ccc1Cl)=O C1(C(=O)NCCc2ncc(C)cn2)N(C(C2C3CCCOC23)=O)CC12CCCC2 c1(COC(C(=O)NC2C(CNC(CCSC)=O)CC2)C)ccccc1C c1(C(C2CCCC2)OCC)nc(C2CCCO2)nn1-c1ccc(Cl)nc1 N1(C(C2(COC)CC2)=O)CC=C(CC(=O)NCCC2(C)CCOCC2)CC1 N1(C(C2(C)N(C)CC(OC)C2)=O)CC(C2CN(C(c3cc(C)c(C)cn3)=O)C2)C1 C1(N(C)CC2CCCC2c2ccccc2)CC(=O)N(C(C)(C)C)C1 C1(C(=O)OC)CCC(NC(C2CC2C2CC(F)(F)C2)=O)C(C)C1 c1(C(N(CCN(C(C(C)OCC)=O)C)C)=O)ccc(C(F)(F)F)cc1C#N N1(C(c2c(C)cns2)=O)CC2CCCC(C1)N2C(C1CC(C)CC(C)C1)=O C(CC(C)C)(C(=O)NCCC1CCCN(C(=O)C(n2ccc(C)n2)C)C1)OC C12(NC(c3cc(C)c(C)s3)=O)CCOC(CNC(=O)Cc3ccc(F)nc3)(C1)C2 N1(C(c2cnc(CC)s2)=O)CC2(COC(CNC(=O)C3=CCCOCC3)C2)C1 N1(C(CCC(C)C)=O)CCC(C)(C)CC1C(=O)NCC(C)(O)CC(C)C Cc1cc(C)c2c(c1)CCC2NC1CCCC(N)CC1 CS(=N)(=O)C1CN(C(=O)CN(C(c2csc(Cl)c2)=O)C2CC2)C1 C=CC1CCN(C(=O)C(C)(CO)NC(=O)C(C2CCCCC2)F)CC1 C1(C)(CC)CN(C(C2C3CCC(C3)N2C(=O)C(C)C2CCCC2)=O)CCO1 N1(C(=O)CCCn2cc(-c3ccnc(CO)c3)nn2)CC2CCC1c1ccccc12 CCCC(C)CC(C(=O)NC1COC1)N1CCN(C2CCSC2)CC1 N1(C(c2c(C)cc(N)s2)=O)CCN(C(c2cc3scc(C)c3[nH]2)=O)CC1(C)C C1(C(=O)NC2CC(n3ccnn3)C2)(SC)CCCN(C(C2CCCN(C)C2)=O)C1 c1(C(=O)NC(CCNC(C#CC2(CC)COC2)=O)C)cc2c(cc1N)OCCO2 C(=O)(C1Cc2ccccc21)N1C(NC(=O)C(c2cccnc2)ON)CCCCC1 N1(C(CC(C)C)=O)CCN(C(C2CCC(O)CN2C)=O)C(CCO)C1 c1(C(N2CC(OCCNC(CC(C)SC)=O)C2)=O)ccccc1-n1cccc1 N(C(=NC1CCOCC1)NC1CCN(CC(F)(F)F)C1)C1(OC)CCOCC1 C1(NC(CCCC#CC)=O)CN(C(=O)CCc2nc(C(C)C)no2)CC12CCC2 C1(C2=CCOCC2)(CNC(c2ccc(F)cc2F)CCC=C)CC1 Cn1c(C(N2CCCC2C(c2ccccc2)=O)C(=O)NC2CCC2)cnc1Br c1(OC)ccc(C(N2CC(NCc3ccc(C)o3)C3(CC3)C2)=O)cc1S(N)(=O)=O CN1CCC2(CCCN(C(=O)CC3CCN(Cc4ccccc4)C3)C2)C1 N1(C(C=C(C)C(C)C)=O)CCC(C2(NC(=O)CC3(O)CCCC3)CC2)C1 n1(CC(=O)NC(C)C(C)(C)NC(=O)C=C2CCOCC2)cc(P(C)(C)=O)cn1 c1(N(C)CC2CC2(F)F)nc2ccccc2nc1N1CCN2CCOCC2C1 C12(NC(=O)CC3(O)CC3)CCOCC1CN(C(=O)CCSc1ccccc1)C2 c1(N2CCC(CC=C)(NC(=O)C(C)N(C)C)C2)nc2c(cc1Cl)C(=O)OC2 N1(C(c2cc(C(F)F)no2)=O)CCN(C(=O)C(O)CN2CCCC2)C(C(F)(F)F)C1 C1(C(=O)Nc2nc(Cl)ccc2Br)CCCC12CCN(Cc1cccn(O)c1=O)C2 Cc1nc(C(=O)Nc2ccc(C(F)(F)F)cc2Br)ccc1-c1ccc(F)cc1O C1(NC(c2n(C)ncc2)=O)CC2CC1CN(C(=O)Cc1sccc1Cl)C2 C1(N(C(=O)CCOC2CCC2)C)CCCN(C(=O)CC2CCSC2)C1 C1(C(=O)NC2CC(c3ccccc3)(NC(=O)C=CBr)C2)C(F)(F)C12CCC2 C1(CCNC(c2ccsc2)=O)CN(C(c2ncc3ccccn23)=O)CCS1(=O)=O C1(CNC(c2n(CC)ccc2)=O)CN(C(=O)COC2CC=CC2)C2CCCCC12 Cc1c(C(N2CC3C(CNC(=O)C(O)C(C)C)C3C2)=O)cccc1N C1(C(C)(C)N(C(CC=CC=C)=O)C)CCNC(=O)C1.C1CCN(C(=O)C)C1 N1(CCC)C(=O)NC(c2ccc3c(c2)CCC3)C(C(=O)OC)=C1C1CC1 C1(NC(C(C)Sc2nnnn2C)=O)CCN(c2ccc(Cl)cc2)C1=O CC(CNC(=O)CCn1cccc1)C(F)C(=O)Nc1ccc(O)c(Cl)c1 C(=O)(CCC(F)(F)F)N1CCCC(CN(C(C(CC=C)NC(C)=O)=O)C)C1 N1(CC=C)CC(O)(CNC(c2cn(CCOC)nn2)=O)C1 n1(CC=C)cccc1C(=O)NCC1CC1NC(C1CC(C)=NO1)=O Cc1ccc(C(C)NC(C2CCCN2c2nccs2)=O)cc1[N+](=O)[O-] C1(C(N2CC(CC(C)NC(c3ccc(Cl)s3)=O)C2)=O)CCCN1C C1(C(=O)NC2(COC)CN(C(CC)=O)C2)CCN(C(=O)OC)CC1 c1(C(N2CC3C(NC(C4CCC(C)(C)C4)=O)(C3)C2)=O)cnn2c1SCC2 C1(O)(CN(C(=O)Cc2ccc(O)nc2)C)CCCN(C(=O)CN2CCNC2=O)C1 C(=O)(C1=CC(O)C(N)C1)Nc1cc(-c2c(C)cncc2)c(N2CCCCC2)cc1 C(=O)(CCP(C)(C)=O)N(C(CC)CC(=O)NCc1cccc(O)n1)C c1(COC(c2cc(=N)[nH][nH]2)=O)cc(C)cc(C)n1.C=C1CC2(C1)C(=O)NC2 c1(NC(C(CC)(C)O)=O)ccc(NC(=O)CCn2ccc(C)n2)cc1C CCC(C)(C(=O)NC1CCC(NC(=O)CSCc2ccccn2)C1)C(F)F C1(CC(=O)NC2CC(F)(CNC(c3cccnc3C(N)=O)=O)C2)CCNC(=O)C1 Cc1ccc(CC(=O)NCc2ccccc2CN(C)C(c2nonc2N)=O)cn1 c1(-c2scc(C)n2)cccc(C(=O)NC(Cc2ccc(Br)cc2)C(=O)O)c1 CC(C(=O)NCC(C)CNC(c1cn(C2CCCC2)nn1)=O)S(N)(=O)=O C(=O)(C(C(C)C)c1cccc(Cl)c1)NCCOCCN(C(c1c(C)con1)=O)C C1(COCCOC)CCN(C(=O)CCN(C)CN)CC1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NC1CCC(CNC(CCC#CC)=O)C1 c1(C(=O)NCC(CC)NC(c2cnc(C)n2C(F)F)=O)cncc(N)c1 c1(OC)ccc(C(C(=O)O)NC(=O)NC2CCCCC2C(F)(F)F)cc1Br N1(c2snc(C(C)(C)OC)n2)CCC(C)C(NC(=O)C=CSc2ccccc2)C1 c1(CC)nc(-c2coc(C(C)SC)n2)n(-c2ccc(SC)cc2)n1 N1(C(C(CC=C)NC(C2Cc3nccn3C2)=O)=O)CCC(N(C)OC)CC1 C1(CN(C(c2cnns2)=O)C2CC2)CCCN1C(=O)Cc1cc[nH]n1 C1(C(=O)NCc2ncc(C(N3C(C)CCC3)=O)cn2)CC2CC(=O)C1O2 C(=O)(C1CCCc2cc(C#N)ccc21)NCC1(C(C)(C)O)CCC1 C=CCCC(O)CNC(c1cn(CCNC(C2CC2CC)=O)nn1)=O C1(C(=O)NC(C=C)C)CC12CCN(C(C1CCN(CCO)CC1)=O)CC2 C1(NC(C(C)n2cccn2)=O)CC(C)(NC(=O)CN2CCC(C)C2)C1 c1(OC)ccc(C)cc1NNC(=O)Nc1cc(Cl)ccc1C N1(C(Cc2c(C)ccnc2)=O)C(C(=O)NC2C=CCCC2)CCC12CC2 N1(C(c2cnc(-c3ccsc3)s2)C(=O)NC(C)(C)C)CC2CC1CS2(=O)=O N1(C(C=CCOC)=O)CCOC(CNC(c2cnncc2C(F)(F)F)=O)C1 C1(C)(N(C)C)CCCC1N(C(c1cnc(NC(C2(n3cccc3)CC2)=O)s1)=O)C N1(C(CCc2scc(C)c2)=O)CC(NC(=O)CC2CC3CCC2C3)C(F)(F)C1 c1(C(c2n(CCC(=O)OCC)nnn2)NCc2cn(C)nn2)scc(C)c1C c1(C(C)C)ncc2c(n1)CCC(C(=O)NCCCOCCNC(=O)CC1CC1)C2 Cc1ccc(C(=O)NC(C)CCCNC(C2CC2(C)Br)=O)c(O)c1C c1(SCCc2onc(-c3ccc(C(F)(F)F)cc3)n2)cc2cccc(Cl)c2cn1 c1(C(N2CCN(C(c3cnon3)=O)C(C(F)(F)F)C2)=O)ccc(Br)c(F)c1 N1(C(C(F)=CC)=O)CC(NC(=O)CNC(C)=O)CC(C)(C)C1 C1(CC(=O)NCCOC2CCN(C(=O)C3=CSCS3)CC2)CCS(=O)(=O)C1 C1(C(=O)NC2C(CNC(c3ncccc3F)=O)CCC2)Cc2nccnc2C1 N1(C(c2c(C)n[nH]c2C)=O)CCN(C(C2CCN(C)CC2)=O)CC(CO)C1 N1(C(C(C)OCC)=O)CCC(NC(c2cc3sccc3n2C)=O)C12CCC2 c1(CNC(N2CCC(C3N=N3)C2)=O)cccc(CCn2cncn2)c1 N1(C(C)=O)CCCOC(CNC(c2nc(NCc3ccccc3)ccc2Cl)=O)C1 c1(CNC(C=CC(CC)C)=O)ocnc1C(=O)N(CC(C)(C)O)C C1(NC(CN(C)C)=O)CCN(C(=O)Cc2sccc2Cl)CC1F c1(C(=O)NC(C2CN(C(CCCc3ncc(C)o3)=O)C2)C)cc(Cl)cc(Cl)n1 CC1(C)CC(CNC(C2OC3CCC2CC3)=O)CN(C(c2ccc(Cl)cn2)=O)C1 c1(C(N2C3CC(NC(c4cc(C)n(C)n4)=O)C3CC2)=O)coc2ccc(F)cc12 O=C(C1CCCc2nn[nH]c21)NCC(CO)Nc1ncnc2[nH]cnc12 c1(SC)nc(C)cc(=NCC(C2CC2)NC(=O)CCN2CCCS2(=O)=O)[nH]1 C(=O)(CC(C)N=c1[nH]c(=NCC2CC2C2CCOCC2)c2[nH]ccc2[nH]1)NC C#CCC(C)C(=O)N(CCCCCNC(=O)C(C)CSC)C N1(C(c2sccc2F)=O)CC2CCC(NC(C34CCCC3C4(F)F)=O)C2C1 C12(NC(=O)CSC(F)F)CCC(CNC(C34CCCCC3C4)=O)(CC1)OC2 C(=O)(C(CC(C)C)NC(C)=O)NC(c1ccc(OC)cc1C)C(=O)OC C1(OC)CC(C(=O)NCC2CCCC2N(C)C)N(C(=O)C=Cc2ccco2)C1 N1(C(C(CC=C)NC(C)=O)=O)CCC2CCCC12C(=O)NCCC1CCCO1 c1(NCCN(C(C(CC#C)C)=O)Cc2cc(C)nn2C)c(F)c(F)c(F)c(F)c1F C(c1cnc2ccccc2n1)=CC(=O)NC1CN(C(c2ccc(F)cc2)C)C(=O)C1 c1(C(C(=O)NCCC2CCCN2C(=O)CCc2cn[nH]c2)O)cccc(Cl)c1 N1(C(C2(C)C=CCCC2)=O)CCC2(CCOC2CNC(c2cocn2)=O)CC1 N1(C(C2CCN(CCC)CC2)=O)CC2(CC2)CC1CNC(=O)C(C)CC(F)F Cc1cc(C(=O)NCCC(O)C(=O)N(CC(C)CO)C)nc(O)c1 C1(C2CC2)(C(N(CCN(CCNC(C(C)CN(C)C)=O)C)C)=O)CCC1 CC(C)(C)C#CC(=O)N1CCC1CNC(=O)CC(=O)c1ccccn1 C1(NC(C(C2CCCO2)NC(c2cc(C)nn2C)=O)=O)CCC(C#N)CC1 C1(NC(C(C)N(C(c2cnc(O)c(C)c2)=O)CC)=O)CNC(=O)C1(C)C N1(C(C=CSC)=O)CCOCC(CNC(c2cnnc(C)c2C)=O)C1 CCC(C)CCCC(=O)NCC1CC1NC(=O)COCc1ccccc1 C(=O)(CC(C)CC(C)C)NC1CCC(C(N2CC(C(CC)C)C2)=O)CC1 c1(OC)cccc2cccc(C(=O)N(C3CN(C(=O)CC4OCCO4)C3)C)c12 Nc1cc(C(F)(F)F)ccc1C(N1CCC(NC(=O)C2=CCC2)CC1C1CC1)=O c1(C(=O)NCCCCN(C(C(C2CCCOC2)OCC)=O)C)ccc(O)c(N)n1 c1(C(N2CCCC(NC(c3ccc(N(C)C)nc3)=O)C2)=O)cccc2nsnc12 C1(NC(c2c(N)cn(C)n2)=O)CN(C(=O)CCCN=[N+]=[N-])C2(CCCC2)C1 N1(C(Cc2c(C)nsc2)=O)CCC2(CCCN(C(C3CCOC(=O)N3)=O)C2)C1 C1(C2CCC2)(C(=O)OC)CCN(C(=O)COC2CCC(N)CC2)C1 C1(C(=O)NCC(C)N(C)C(C2CC(C(F)(F)F)C2)=O)CCC(C#N)C1 c1(CC(=O)NC(c2cccnc2)C(=O)NCC2(C)CCCO2)ccc(CO)cc1 C1(C(=O)NC2(c3ccc(C)s3)CC2)CCCN(C(c2ccc(C#N)nc2)=O)CC1 Cc1ccc(C(=O)NC2CN(C(=O)CS(=O)(=O)N(C)C)CCC2F)cc1Cl CC1(C)CCc2cc(C(=O)NC3CC3NC(=O)C(c3ccccc3)=O)ccc2O1 N12CC3CC3C1C2=O.C1(C=O)CC=CCC1.C(CC(=O)OCC)SCC C1(C(=O)NCCc2nc(C)oc2)NCCC12CC2(F)F C1(C2(O)CCN(C)CC2)(C(N2CCN(C(C=NOC)=O)C3(C2)CCC3)=O)CC1 C1(N(C)C(C2CC(F)(F)C2)=O)CC2CCC(C1)N2C(=O)C(C)(C)Cc1cnn[nH]1 N1(C(Cc2n3cc(C)nc3sc2)=O)CCOC2CN(C(c3cnc[nH]3)=O)CC12 CN1CC(C(=O)NCC2CC2NC(=O)CCNc2ccccn2)CC1=O CCCC(O)C(=O)NC1CC(NC(c2cccc(C)n2)=O)C(O)C1 N1(c2cccc(C)n2)CC2CCCCC2OC1 C1(NC(c2cn(CC)nc2)=O)CCN(C(=O)C2=CC(O)CCC2)CC(O)C1 N1(C(CCC(C)OCC)=O)CC(C(=O)Nc2cnn(C(C)C)c2)C2(CC2)C1 Cc1cc(C)n(CC(=O)NCC(C)N(C(=O)CC2COC(=O)C2)C)c(=O)n1 C1(NC(CCCOCCC)=O)CC(N=c2cc[nH]c(OC(C)=O)n2)C1(C)C CCCCC(=O)NC1CCCC1CN(C(=O)CCc1cnn[nH]1)C CN1CC(C)(C(N2CCCC(F)(CNC(=O)CCC3CCC3)C2)=O)CC1=O CCCC(C)CCCC(=O)N1CCC(CCNC(c2nc(Cl)c(Cl)s2)=O)C1 N1(C(C(C)=C(CC)C)=O)CC2(C)CN(C(=O)C3CCc4nccn43)CC2(C)C1 N1(Cc2cn(C(C)C(=O)NCc3ccccc3OC(F)F)nn2)CC(C)CC(C)C1 Cc1nn(C)c(C)c1CC(C)C(=O)N1CCCC1CNC(c1ccncc1)=O C1(NC(=O)Cn2cc(Cl)cn2)COC2(CCN(C(c3cc(O)nc(O)n3)=O)C2)C1 Cc1sc(C(c2nnnn2CCC2(C)CC2)NCCc2nc(CO)cs2)c(Br)c1C C(N=c1[nH]c(=NCc2ncc(C(N)=O)s2)[nH]c2ccsc12)c1cccc(C)n1 C1(C(N(CCCC=C)C)=O)CN(C(=O)CCc2cscn2)CC(C)O1 c1(NC(C2CCCN2C(c2cc(Cl)c(Br)c(Cl)c2)=O)=O)cccc2ccncc12 N1(C(=O)Nc2ccnc(C3(C)NC(=O)NC3=O)n2)CC2CCCC(=O)NC2C1 C1(CNC(CC(C)O)=O)CC2CCCCC2N1C(=O)Cc1csc(NC=O)n1 C12(CNC(c3cn(C)nc3Cl)=O)CCCC1CCC2 C1(CC(=O)NCC(C)(C(C)C)NC(c2c[nH]nc2F)=O)(CC)CCOCC1 Cc1cccc(Br)c1C(=O)NCC1COCCN1C(c1cc(Cl)no1)=O c1(-c2cn(CC3N(C(C=CS(C)=O)=O)CCCC3)nn2)cncc2ccccc12 c1(C(N2C(C(N3C(C)(CC(=O)NC)CC3)=O)CC2)=O)cc(C)cc(C)n1 c1(C(N(c2nnnn2CC(F)F)C)=O)cccc(C(F)(F)F)n1 C(=O)(C1CCSc2ccccc21)N1CCC(C)(O)C(O)C1 N(C1CCCc2ccoc21)C(C(CCCNC(c1cc(CC)no1)=O)O)=O S(=O)(=O)(c1ccc(N2CC3CCC(C2)C3O)c(Cl)c1)N(CC(O)CF)C Cc1c(C(N2CCC(NC(=O)CCc3ccoc3)CC2C)=O)cc(O)cc1N C(=O)(C1CCCc2c[nH]nc21)CCCN1C(=O)NC2(CCCC2)C1=O C1(NC(C2CC23CCSCC3)=O)CCCN(C(c2c(F)cccc2Cl)=O)CC1 N1(c2nc(C)nc(Cl)c2)CC(C)CN(C(C2CC(F)(F)C2)=O)CC1C C(=O)(CC(C)CC(C)(C)C)NCCCCCCC(=O)N(C)Cc1c(C)cco1 c1(CC)nnsc1C(=O)NC(C)(C)C(=O)NC(COC)CC c1(C(N(CCN(C(c2cnc(SC)s2)=O)C)C(C)C)=O)cc(F)ccc1F C(CC(C(C)C)NC(=O)C(O)C1CCCC1)N(C(CCC=C)=O)C C1(NC(C(C)NS(CC)(=O)=O)=O)CC2C1CCN2C(=O)CC1CC(F)(F)C1 Cc1c(C(=O)NC2CN(C(c3c(F)ccnc3Cl)=O)CCC2F)cccc1O N1(C(=O)Nc2cc(N3CCN(C(C)=O)CC3)ncn2)CCC(CO)C2(CCC2)C1 c1(CC(=O)N(C(C)CNC(c2ccc(C)cc2C)=O)CC)ccc(O)c(Cl)c1 c1(N2CC3C(CNC(c4nc(OCC)oc4)=O)C3C2)[nH]cnc2nc(Cl)cc1-2 Cc1n[nH]c(C)c1CC(=O)NC1CC1CNC(=O)C=Cc1cc(C(F)(F)F)co1 c1(SCC(=O)NC(CC(C)NC(C2(C(C)C)COC2)=O)C)ccc(F)cc1 c1(C(=O)N(CCCO)Cc2ccc(Cl)cc2Br)cc2c(C(F)(F)F)cc(O)nc2o1 C(=O)(C1CCCc2c[nH]nc21)N(C1C(NC(c2n[nH]c(C)c2F)=O)CCCC1)C CC1(C)OCCOC1C(=O)NC1CN(C(c2cncc(O)c2)=O)CC12CC2 N1(C(COC)=O)CCC(C)(C)C1CC(=O)NCCNC(=O)N(CC(C)C)CCO C1(N(C(C2CC(C)CO2)=O)CC)CCCN(C(=O)Cc2cccc(Cl)c2F)CC1 N1(C(CC2C(C)=NOC2=O)=O)CCC2CN(C(=O)C(C)(C)C3CC3)CC2C1 c1(OC)ccc(Cl)c(CC(=O)NC2CC(F)CN(C(C3C=CCC3)=O)C2)c1 C1(C(=O)NCC2(O)CCCOC2)(COC)C=CCN1C(c1ccc(C(C)=O)o1)=O c1(C(=O)NC(CCOCC)C(=O)NCCc2c(C)noc2C)nnc(O)nc1O CC1CCCCC1(CNC(=O)CCc1nc(=N)[nH][nH]1)NC(c1ccc(F)cn1)=O c1(CC)ccc(C(=O)NCC(CNC(=O)C(C)Sc2ccc(C)cc2)CO)cn1 N1(C(C=CCC2(NC(C3CC(=C)C3)=O)CCC2)=O)CCC(C(C)SC)CC1 C(=O)(C1(C)CCCc2ccccc21)NC1(CC=C)CN(C(=O)C(C)(C#N)CC)C1 C=CCC(CC)C(=O)NCCC1(C(N2CCCC(F)CC2)=O)CC1 S(=O)(=O)(c1ccc(CC(=O)NC2CN(C(C3(C)CCCCO3)=O)C2)s1)NC C1(C(=O)NCC(C2CCCCC2)C)CC2CN(C(=O)Cn3cnc(C#N)n3)CC2C1 C1(CC(=O)NCC(CC)NC(=O)C(=O)CCC(C)C)CSc2ccccc2NC1=O C1(CNC(C2(C(=O)OC)CCOC2)=O)CC(NC(c2ccc(Cl)s2)=O)CCO1 Cc1ccc(C(N2CCCN(C(c3cnn(C)c3)=O)CCC2)=O)c(N)c1C C1(NC(C(COC)O)=O)CN(C(c2ccc(Cl)cc2Br)=O)CC12CCC2 N1(C(c2nnc(C)o2)=O)CCOC2(CCN(Cc3cc(Br)c(C)c(Br)c3)CC2)C1 Cc1csc(C=CC(=O)N(C)CCN(C)C(c2cncc(OC(C)C)c2)=O)n1 c1(OC)ccc(F)c(C(=O)NCCC2(NC(C3CCOCC3(C)C)=O)CCC2)n1 c1(C(CC)O)nc(-c2cn[nH]c2C)n(CCS(N)(=O)=O)n1 C1(C(F)(F)F)(C(N(CCCn2cc(SCCC)nn2)C)=O)CCCCO1 C(=O)(C(C)CC(N)=O)N(CCN1CCN(C(C(C(C)OC)N(C)C)=O)CC1)C C1(C)(CC)CCN(C(=NCC2CC2)NCC2(CC(=O)OC)CCCCC2)C1 Cc1ccc(C)c(SCC(=O)Nc2cc(Br)ccc2C(=O)Nc2ccccc2)c1 C1(NC(c2c(CC)ocn2)=O)CCCCC1C(=O)NCC(C)C(F)F CC1(C)CCNCC1CNC(=O)C(=O)NC1CC2CC2N1Cc1ccccc1 C1(C)(C(N2CC3C(CNC(CCNC(=O)OC)=O)(C3)C2)=O)CC(C2CC2)=NO1 N1(C(C2C(=C)C2)=O)CCC(CCNC(=O)CC2(CSC)CC2)C(F)(F)C1 c1(C(=O)NCCC2N(C(C3CC(N(C)C)C3)=O)CCC2)cncc2cnccc12 C1(OC)CN(C(=O)CC23CCCC2C3)CC1NC(=O)C(c1ccn(C)n1)C C1(C(=O)NC2C(NC(c3coc(Br)n3)=O)CCCC2)CC12CCOCC2 Cc1cnc(C(=O)NCC2(CC(=O)O)CC2)s1 CCC(CCO)NC(c1ccn(CCNC(=O)CC2CC(F)(F)C2)c1)=O C1(CNC(CN(C)C)=O)CN(C)CCN1C(c1sccc1Cl)=O C1(c2n(CC)nnn2)(NCC(c2nc(C)no2)(C)C)CCC2CN(C)CC12 c1(C(N2C(CC(=O)Nc3c(OC)cccn3)COCC2)=O)c(F)cccc1Cl Fc1cc(-c2cnc(CN3CCOC(c4cccc(Br)c4)C3)nc2)cc(F)c1F c1(C(=O)NC2C(NC(C(CC)NC(N)=O)=O)CCOC2)ccc(C)c(CO)c1 N1(C(C(C)N(C(C)=O)C)=O)CCn2c(CNC(=O)C3=C(C)CCCC3)nnc2C1 c1(CC(=O)OCC)ccnc(Cl)c1NC(c1ccccc1)Cc1cncnc1 n1(CC(N2C(CNC(C=C3CCC(C)C3)=O)CC2)=O)cc(Br)ccc1=O N1(C(c2ccc(CCC=C)cc2)=O)CC2(COC(CNC(=O)COCCF)C2)C1 CC1CC(=O)N(CC(=O)Cc2ccc(F)c(F)c2)C1=O C1(NC(c2cc(COC)[nH]n2)=O)COC2(CCN(C(c3cccc(CO)n3)=O)C2)C1 C1(CNC(C(N2CCCC2=O)C)=O)CCC12CN(C(c1cccc(C#N)c1)=O)C2 c1(C(=O)OC)ccc(NC(C2C(NC(=O)C=C(C)Cl)CC2)=O)cc1C(F)(F)F C(=O)(C(O)CCCCC)N1CC2C(N(C(C3CC(=C)C3)=O)C)C2C1 c1(NC(C(n2cc(-c3ccc(-c4cc[nH]n4)cc3)nn2)C)=O)cccc(F)n1 C1(S(N)(=O)=O)(C(=O)NCC2(NC(C(CN(CC)CC)F)=O)CC2)CCC1 C1(C(=O)NCC2(NC(C3CCCOC3C)=O)CCC2)(CC)CCCC1O C(C(C)(C)C(=O)NC1CC2(C1)CC2NC(c1[nH]ncc1C#N)=O)NC(C)=O C1(CCC(C)NC(C(CF)NC(=O)OC(C)(C)C)=O)CCC(C(C)(C)C)CC1 c1(COC(=O)C=CCOc2cncc(F)c2)cccc2ccccc12 N1(C(C(=O)NCCOC)C2CC(CO)C2)CCC(CNC(C)=O)C1 c1(C(CC)(C)C)ccc(OCC(C2CCC2)OC(=O)C(C)CF)cc1 Cc1ccc(NC(=O)NC(c2ccc(F)c(C(C)O)c2)CN(C)C)cc1Cl c1(C(N2CC3(C(C(N(c4ccnn4C)C)=O)C3)C2)=O)ccc2nccn2c1 c1(C(N2CC(OCC3(C(=O)OC)CC(=C)C3)C2)=O)c(C)cc(F)cc1C c1(CN2C(c3ncc(-c4c(C)cccc4)[nH]3)CCC2)cc(Br)c(F)cc1O c1(C(N2CCCC(C)(NC(C3N(C)CCC3)=O)C2)=O)cnn2c1NCCC2 C1(CC(=O)NC2COCCC2NC(C2(CO)CCC2)=O)CCCCC12CC2 C1(OC(c2c(OC)c(Cl)ccc2Cl)=O)CS(=O)(=O)C12CCOCC2 c1(OC)ccccc1C(C)(C)C(=O)NCC(C)(C1CC1)NC(=O)COC(C)(C)C Cc1cc(C(=O)NCCCC2CCCN2C(c2cocc2Br)=O)oc1C c1(C(=O)NC2CC(CNC(c3c(C)ncc(N)c3)=O)C2)cnn(C)c1S(C)(=O)=O Cc1cccc2[nH]c(=NC(C)CC(C)NC(c3oc4ccccc4c3Cl)=O)sc12 C#CCC(C)(CNC(=O)C(C)(C1CC1)N(C)C(C1CCC(=O)N(C)C1)=O)CO CC(CCC(=O)NCC(=O)N(C)O)NC(=O)CCC1CC(C(=O)O)CO1 N1(C(C2(C=C)CCN(C(c3cccc(C)c3F)=O)C2)=O)CCCC(F)(F)CC1 C(=O)(C(CNC(=O)CCc1nncs1)N(C)C)NC(COC)(C)C1(C)CC1 c1(CCCCC(=O)NCCC2CCN(C(=O)C=CBr)C2)ccc(F)c(F)c1 C#Cc1ccc(C(N2CC(CC)OC(C)C2)=O)c(F)c1 c1(OC)ncc(Cl)c(C)c1C(=O)NCC1CN(C(=O)C(C)C2CC2)CCC1(F)F C=C1CCC(C(=O)NC2C=CCN(C(c3cc(C(C)CC)no3)=O)C2)CC1 C(=O)(C(C)(C)C(=O)NCc1ccc(C(=O)NCc2ccco2)nc1)NC c1(C(C)C(=O)NC2CCN(C(=O)CCC3CCC(=O)N3)CC2)ccc(F)c(F)c1 C12(C(N3CC(CCCNC(C4C(C)CCO4)=O)OCC3)=O)C3C4C1C1C2C3C41C c1(C(N2CC(N(C)C(C3CC3OC(C)(C)C)=O)OCC2)=O)ccc2nccn2n1 C(CCCCC(=O)NCCN1CCN(C(c2cnn(CC3CC3)c2)=O)CC1)OC N1(C(CC(C)OC)=O)CC2CCC(C1)N2C(c1cc(Br)oc1C)=O c1(CCC(N2CCC(C(C)NC(C3CC(C(N)=O)C3)=O)C2)=O)ccc(O)nn1 C(=O)(C(C)(C)S(=O)(=O)c1ccccc1)NCCC(CNC(C1C(C=C)CC1)=O)O c1(CNCC2N(C(C(C(C)C)NC(C)=O)=O)CCCC2)ccc2ncnn2c1 C1(C(N(C)CC2(NC(C3CC3Cl)=O)CC2)=O)C=CC=CC=C1 c1(C(N(CC(N2CCCC3CC23)=O)C)=O)cc2cc[nH]c2cn1 CC1(C)CC(=O)NCC1C(=O)NCCCOCCNC(=O)CC1CCCC1(F)F C(=O)(C(CC)CC(C)C)NCC1(NC(C(C)SCCCC)=O)CC1 C1(NC(C(C)(C2CCC2)NC(=O)C=CC2CCOCC2)=O)CC2(COCCO2)C1 c1(C(C(=O)N(CC(CNC(c2ccn(C(C)C)n2)=O)C)C)C)nc(F)ccc1Cl CCC(F)(F)C(C)(C)NC(C1CN(C(c2ccc(O)cn2)=O)CC(C)O1)=O Cc1cc(Cl)cc(C(N2CC(CCNC(C3(C4CC4)CC3)=O)C2)=O)c1C C(N=c1ccnc(NCC2CCCC2(C)C)[nH]1)c1c(C)c(Br)ccc1 Cc1c(C=CC(N2CC(NC(=O)C(C)(F)F)C(C)(C)C2)=O)cnn1C c1(OC)ccncc1C(=O)N(C1CCC(NC(=O)CC(C)NC(N)=O)CC1)C c1(N2CCC(NC(=O)Cc3ccc(Cl)cc3)C(F)C2)ccc2nccnc2n1 C(CC(O)C(=O)NCC1CC(CNC2C(C)C2(F)F)C1)NC(COC(C)(C)C)=O C(=O)(C(CC(C)C)C(C)C)NCC(CN(C(C=C(CCN(C)C)Cl)=O)C)C Cc1cccc(C(=O)NCC(C)NC(C2(N(C)C)CCCSC2)=O)c1C c1(C(N2C(C)CCC(NC(c3cncn(C)c3=O)=O)C2)=O)cc(O)cc(C#N)c1 N1(C(c2c(C#N)nc[nH]2)=O)CCCN(C(=O)CCSC2CCCC2)CCC1 Cc1nc(C)n(CCC(=O)NC(C)(CNC(=O)Cc2ccsc2Cl)C2CCC2)n1 C1(C(=O)NC2CCC(NC(c3cnc(C(C)=O)s3)=O)CC2)(COC)CCC(=O)N1 N1(C(C(C(=O)OCC)OC)=O)CCC2CCN(C(=O)C(=O)NCC(F)F)CC12 C(=O)(C#CC1(C)COC1)NC1C2(C(=O)NCC(N(C)C)C3CC3)C3CC1CC23 C(CNC(=O)C1=CCCC1)(CC(F)(F)F)NC(=O)C(O)C(F)F C1(C(=O)NCC(C(C)(C)C)OC)C2CC3C(C2NC(=O)C(C(C)C)SC)C13 CC1(CNC(=O)NC2CC2c2ccccc2)CCCN(C(=O)C2=COCCC2)C1 CCCC(C#N)C(=O)NC(C)(C)CCNC(C1CCC(C(F)(F)F)CC1)=O c1(SC)ncc(C(N2CCC3C(NC(c4ccon4)=O)C23)=O)n1C N1(C(CN(C)C)=O)CCC2CN(C(c3cc(Cl)ncc3O)=O)CC2CC1 N1(CC(c2cccc(Br)c2O)=O)CC2CCC1C(O)C2 CN1CC(C(=O)NCC2(F)CN(C(=O)CC3CCOC3(C)C)C2)OCCC1=O Cc1ccc(C(C)OC(C)(C)CN(C)C)c(OCC(F)(F)F)c1 C1(C(N2C(C(=O)OC)C3CC3C2)=O)CN(C(=O)CCC2CC2)CC1(F)F c1(CC)ccc(C(=O)NC2(CNC(C3(SC)CC3)=O)CCCCCC2)c(Cl)c1 N1(C(C(C(C)C)C)=O)CC2(CCCC(CNC(C3CN4CCC3CC4)=O)O2)C1 C1(C(N2CCCC(NC(C(C)CCO)=O)(CO)C2)=O)CCCC(F)(F)CC1 C1(C(N2CCC(C(C)(C)NC(C=CC(=O)N(C)C)=O)C2)=O)CN(C)CCO1 C(=O)(C(C)(O)C(C)(C)C)NCSCC(C)(C)OCCNC(C=CC)=O C1(CC)CN(C(c2cnco2)=O)CCC1NC(c1ccc(SC(F)F)cc1)=O C(CN=c1[nH]c(=NCc2cccnc2N)[nH]c2cc[nH]c12)(C(F)(F)F)OCC C(CCCCC(=O)NCCC(C)(C)NC(=O)C(C1CC1)OC)=CC Cc1nn(C(C)(C)C(N2CCCC(CN3CCCC3)C2)=O)cc1Br C12(C(=O)OC(C)(C)C)CCCC1CN(C(c1cnc(C(F)F)nc1)=O)C2 c1(C(=O)NC2CC(C)(NC(=O)CSc3cn[nH]c3)C2)cccc(C(F)(F)F)n1 C1(NC(COCCC=C)=O)CCCN(C(c2cc(N)ccc2O)=O)CC1 N1(CC)CCC(C)(c2cccc(F)c2)CC1.C12CC(C1(C)C)NC(=O)NC(=O)C2 C(=O)(CCCS(C)(=O)=O)NCC(C)(CO)NC(c1cc(C(C)=O)c(C)nc1)=O Cc1ccc(C(=O)NC2(C(N3CCCOCC3)=O)CC(F)C2)nc1O c1(OC)cccc(CCC(=O)N(C)CCNC(c2cc(OC)nn2C)=O)n1 c1(C(N2CC3CC(NC(c4n(CC)cc(Cl)c4)=O)C3C2)=O)c(C)nc(O)nc1C C1(C)(CNC(C2CCCN(C)C2)=O)CCC(NC(=O)CC2CCCC2)CC1 C1(NC(CN(C(Cc2nc(C)[nH]n2)=O)CC(C)C)=O)CCCC1C#N c1(C(N2CCC(OC)(CNC(c3ccncc3)=O)C2)=O)ccc2nc[nH]c2c1 c1(OC)cc(C(=O)NCC2C(C)CCN2C(c2n[nH]c(C)c2O)=O)nn1C CCCC(C)(C)CC(=O)N1CCC(CCOC)(NC(C2CCOC2C2CC2)=O)C1 c1(C(=O)NCC(CNC(c2cccc(C(N)=O)c2N)=O)O)cc(F)c(F)c(F)c1 c1(C(=O)NCC2C(C(N(C)CC3(C)CCCO3)=O)CC2)cccc(=O)o1 Cc1nc(C)c(C(=O)NC2(CCCNC(c3ccc(C(C)C)o3)=O)CC2)o1 c1(C(C)C)nc(N2CCC(N(C)C(c3ccc(=O)n(CCO)c3)=O)C2)cc(Cl)n1 c1(C(=O)NC2C(C)CN(C(C3(C)CCCCO3)=O)CC2)cc(C#N)ccc1F C(=O)(C(C)=NOCC#N)NCC(CN(C(COCC)=O)C)O C1(C(N2C(CNC(C3CC(n4ccnn4)C3)=O)CC2)=O)NC(=O)C2CC12 N1(C(CNC(C)=O)=O)C(C(=O)NCCCCC(C)(F)F)C2CC(O)C1C2 CC(C)CCCCCNC(C1CCCCN(C(c2ccoc2)=O)C1)=O CCCC(C)(CC)C(=O)N1CC=CC(C(=O)NC(C)CCC(C)(C)C)C1 Cc1cccc(-c2nnc(N(C)Cc3ccns3)n2Cc2cccs2)n1 N1(C(C(COCC)C)=O)CCOC2(CCN(C(C3(C(C)O)CC3)=O)C2)C1 C1(N(C(=O)Cn2ncnn2)C)CN(C(C2(C)COC2)=O)CC12CC2 C(C)(C)(CCCNC(=O)CSCc1cccc(Cl)c1)NC(C1C(C)(C(C)C)C1)=O C(=O)(CC(C)=C=C)NCCOC(CNC(C(C)OCC#C)=O)(C)C c1(-c2n(C(CC)C)nc(Cc3cnn(C)c3)n2)cccn1C(=O)OC CC(=O)CCC(=O)N1CC(OCCC(=O)NCC2(CC(C)C)CCC2)C1 C(CCC(C)C)OCC.N12CC(C1)C(C(=O)OC)NC2=O C(=O)(C(C)CC(C)(C)C)NC(C(=O)NCCc1scc(C)n1)CC(F)F Cc1c(Cl)ccnc1C(N1CCC(NC(C2CC3CC3C2)=O)C(CO)C1)=O C1(NC(C)=O)CCOC12CCN(C(C1CCC3(CCCCCCC3)O1)=O)CC2 C1(C(=O)NC(C2CCN(C(C3(O)CCSCC3)=O)CC2)C)CC(=O)N(C)C1 Cc1cc(=NC2CCC(NC(c3cncs3)=O)CC2)[nH]c(C(C)(C)C)n1 C12(C(=O)OC)CC(CN1C(=O)NCc1cnn(-c3ccccc3)c1C(F)(F)F)C2 C=CC1(O)CN(C(C2CCCC2NC(=O)C(O)CSC)=O)C1 CC(C)(C(=O)N1CC2CCC(C1)N2C(=O)CCCC(=O)c1ccc(Cl)s1)C(F)(F)F c1(CN2CCC(N(C(=O)C=CC3CC3)C)C2)cccc(Br)c1 CN(C)NC(=O)CCC(=O)N1CCCN(C(C2CCCN2C=O)=O)CC1 c1(OC(CC)CC)ccc(OC(CC(N)=O)C2CC2)o1 CC(C)C(O)C(=O)NC(C)CCCNC(=O)OC(C)(C)C C1(NCCN(C)CCN(C(=O)CCOCCC2CCCC2)C)CCCCC1 C12CCN(C1)C2=O.C1(CN(C)C)C(CNC(=O)C(C)(C)C2CC2)C1(C)C N1(C(C(CC)SC)=O)CCCC(NC(c2occc2F)=O)C1 Cn1nc(Br)cc1C(=O)NCC(CC=C)NC(=O)CCC1CCCO1 Cc1cn2cccc(C(=O)NC3CN(C(=O)CCOC4CCCC4)CC3C)c2n1 c1(C(=O)NC2(C)CC(NC(C3(C=C)CCOCC3)=O)C2)cc2nn[nH]c2cc1F C1(NC(C(CCNC(CCSCC)=O)(C)C)=O)CC2CC1CC21CC1 c1(C(N(CCC2CCN(C(C(CC=C)C)=O)CC2)C)=O)nc(O)[nH]c(=O)n1 c1(C2C(C(=O)NC3CC(N(C(CNC(CN(C)C)=O)=O)C)C3)C2)nccn1C Cc1cnsc1C(=O)NCCC1(C(=O)NC(C)C(C)n2cccn2)CCC1 CC1CCNCCC1N(CCCCN(C)C)C(=O)NCc1cccc(O)c1 C#Cc1cncc(C(=O)N(CC(O)CN(C)C(c2c[nH]c(Br)c2)=O)C)c1 C(=O)(CCCCCNC(C1CCCCC1C)=O)NCCCOCC C1(NC(c2cc(C)nc(C)c2)=O)CCSC12CN(C(C1(O)CCCCC1)=O)C2 C(=O)(CCC(=O)c1cc(Br)cs1)N1CC(CNC(C2C(C(C)C)(CC)C2)=O)C1 c1(C(=O)NC2C(CNC(C(C3CCCCC3)OC)=O)COC2)ccc(Cl)cc1F C(C(=O)NCCNC(C1CCCSC1)=O)(c1ccccc1)=CC(C)(C)C c1(CNC(=O)Nc2c(C)ncs2)cc(=O)n2nc(-c3ccc(Cl)cc3)sc2n1 C12CC13CCN(CC3)C2=O.C1(C2(NC(CC3(OC)CCC3)=O)CC2)CCCCO1 C1(NC(C(COC)OC)=O)CC2C(NC(c3cn(C)nc3C(C)C)=O)C2C1 CC1C2C(CCN2C(c2ccc[nH]2)=O)CN1C(c1ccc(O)nn1)=O C1(CC)C(NC(C23CC2COC3(C)C)=O)CCCN1C(=O)C(CSC)OC c1(OCOC)cccc(O)c1C(=O)NCCCN(C1CC1)Cc1cccs1 C12(C(=O)NCC#CC(=O)NC(C=C)C3CC3)C(=O)C3CC1C2C3 C1(CNC(=O)C=C2CCCC2)CN(C(c2cncc(CO)c2)=O)C2CC12 CCC(C(=O)NCC(O)C(=O)Nc1csnc1C)C(C)C c1(C(=O)NC2CCN(C(C3N(CC)CC3)=O)CC2C)cnn2c1CCCN2 c1(C(=O)OC)oc(C)nc1C=CC(N1CCC(Cc2ccccn2)C1)=O c1(CC)cnc(Cl)nc1N(CCCN(C(=O)C1=CCOCC1)C)C O=C(CC(C(F)F)c1ccccc1)NCC1CC(C(=O)NCC23CC(O)C2C3)C1 C(C(C)(C)CC(=O)NC(C)(C)CN(C)C)NC(C1(CCCC)CCCC1)=O c1(C(=O)NC(C2CN(C(C(C)OCCCC)=O)C2)C)coc(C2CCCC2)n1 c1(CNC(=O)CCCC2CC2)nc(CNC(C(n2cc(Cl)cn2)C)=O)cs1 C1(NC(c2ccc(C(F)F)cc2)=O)C2COCC1CN(C(c1ncccn1)=O)C2 N(C1CCCn2nccc21)C(c1cc(CNC(C(C2CC2)OC)=O)[nH]n1)=O c1(C(N2C(CC(=O)NC3C(C(=O)OC)CC3)CCC2)=O)coc2ccc(Cl)cc12 N1(C(C(C)(C)N2CCOCC2)=O)CC(CNC(C2CCSC2)=O)OC2(CCC2)C1 c1(-c2cc(CC3CC3)sc2)ncccc1F.n12cc(cn1)C2C(=O)N(C)CC(C)C.O.C N1(C(C=C(CC)C)=O)CCCC(NC(=O)C(c2ccc(F)cc2)(C)N(C)C)C1 C1(CC)CN(C(=O)C=CCOCCO)CC1CC(=O)N(C)OCc1ccccc1 CCCC(C(=O)NC(C)CC(=O)N1CCCC1CC(C)C)NC(N)=O C(CC1c2ccccc2CCN1C(=O)C(=O)NC(C)C)NC(C(C)NC(C)=O)=O N1(c2nc(C#N)c(Cl)s2)CCC2(COC(CNC(=O)C=CCF)C2)C1 N1(C(CCNC(COC)=O)=O)CCCN(C(C2CC3CCC3C2)=O)CCC1 N1(c2ncc(C#C)cn2)CCC2(CCCCC2NC(C2CNC(=O)CC2C)=O)C1 c1(CC(=O)NCC=CCN2CCN(C(=O)COC(F)F)CC2)cccnc1Cl C(=O)(C1=CC2CCCC12)N1CCN(C(c2n(C(C)C)ccc2)=O)C(CO)C1 C(CC(C)C)(C(=O)NCC(CC(F)(F)F)NC(c1cc(C)[nH]c1C)=O)NC(C)=O c1(CC)ccc(C(=O)NC(C)(CNC(C2(CSC)CCCO2)=O)CO)c(C)c1 CCCCCC(C)CC(=O)NCc1nc(C(N2CCC(O)(CN(C)C)C2)=O)co1 c1(OC(C)C)ccc(C2CCCN2C(=O)C(C)(C)n2cccn2)nn1 N1(CC=C)CCC(N2CCSCC2CCNC(=O)CC2C=CCCC2)C1=O C1(CC(N2CC(O)(C(C)NC(=O)CC3OCCCO3)C2)=O)COCC(C)(C)O1 c1(CN(C)C(c2ccc(-c3ccc(-n4ccnc4)cn3)cc2)=O)ncccc1Cl C1(NC(c2nc(CC)oc2C)=O)C2CCN(C(c3cc(C(C)C)n(C)n3)=O)CC12 N1(C(c2cnn(CC)c2C)=O)CC(O)C(O)C1CNC(=O)C(C)(C)SC CC1(C)CCN(C(=O)C(F)=C2CCC2)CC1NC(C1CCCC1C(F)(F)F)=O CC(C)(C)C1=NOC(C(=O)NC2CCN(C(=O)CC3C=CS(=O)(=O)C3)CC2)C1 c1(CC)cccc(C)c1-n1nc(-c2cc[nH]n2)nc1Cn1ccc(Br)n1 CC(C)CC(C)CC(=O)NC1CCN(C(c2nocc2Br)=O)C1C1CC1 c1(CC)c(C(=O)NC(CNC(=O)CCCn2cncn2)C(C)C)nnn1C Cc1nc2ccc(C(N3CCN(C)CC3CNC(=O)CS(N)(=O)=O)=O)cc2s1 c1(N2CC3CC(CN(Cc4cnn(C)c4Cl)C3)C2)ncnc2c1ccn2C c1(N(C(CCCC(C)C)=O)C2CC3CC2CN3)ccc2c(c1)CC(=O)N2 C(=O)(C(O)C(C)(C)C)NCCC(C(=O)OCC)NC1(COC)C2CCC12 CCC(O)(CC(=O)NCC1(CNC(=O)CP(C)(C)=O)CCC1)c1ccccc1 C1(CNC(C=CCCC)=O)CCCC(NC(c2cccc(-c3cccs3)n2)=O)C1 C1(C(=O)NCC2CCN(C(c3n(C)c(S)nn3)=O)C2)CN2CCC1CC2 C1(NC(C(CCCC)C)=O)CCC2CC1CN2C(C12COC(CCO1)C2)=O Cc1c(C(=O)NCC2(N)CC3CC3C2)cnn1-c1ccccc1Br CCC(=O)CCC(=O)NC1CC2(C1)CC2C(=O)N(CCCO)C CC1(C)CCN(C(=O)C2=COCCO2)CC1NC(c1ncc(Cl)cc1F)=O Cc1nn(CCO)c(C)c1C(=O)NC(C1CCN(C(=O)CCCCC#N)CC1)C c1(C(=O)NCC2N(C(c3c(C)cco3)=O)CC2)cc(C#N)oc1C C=CCC(CC)C(=O)NCC1(CNC(=O)C(C2CCCCCCC2)O)CC1 CC(C(O)C(F)F)NC(C1(NC(=O)CC2CCCNC2=O)CC(O)C1)=O c1(NC(CCN(C(CC2ON=C(CC)C2)=O)C(C)C)=O)cccn2ccnc12 Cc1ccc2c(=O)c(C(N3CCC(C4CCCN4)C3)=O)cn(C)c2n1 C1(C(N(CC(C)(C)NC(c2ccc(C(F)F)s2)=O)C)=O)CCc2nnnn2C1 N1(C(C=C(COC)C)=O)CC(CNC(c2c(C)ccn2C)=O)OC2(CCC2)C1 c1(OC)ccc(CN2CCN(C(=O)CCC(F)(F)F)CC2C)c2ccccc12 CCC(CC)(CO)C(=O)N1CCC1CNC(c1cc(N)c(F)cn1)=O C1(NC(c2ncn(C)n2)=O)CCSC12CN(C(c1ccc([N+](=O)[O-])cc1)=O)C2 N1(C(C(C)CN(C(=O)C2=CCSC2)C)=O)CC(=O)NC(=O)C1 c1(N2CCC(NC(C(C)n3ccnc3)=O)C(C)(C)C2)ncc2c(ncn2C)n1 C1(NC(c2nc(Cl)ccc2C(=O)O)=O)CC2CCC(C1)N2C(=O)CN1CCCC1 C(C)(CCC(=O)NCC1CN(C(=O)CCOC2COC2)C1)SC N1(CC)C(=O)CCC1CC(=O)N(C1CCN(C(=O)C=CSCc2ccco2)C1)C C=CCCCCCC(=O)N1CCCCC(NC(=O)C(F)C(C)C)C1 c1(C(=O)NCC2(F)CCN(C(C3CC3CF)=O)C2)cn2ccsc2n1 O(NC(=O)CC(C)CNC(c1cc(C#N)ccc1C)=O)CC(CC)C c1(C(N2C(C(C)(C)NC(C(C=C)O)=O)CCC2)=O)cc(C(F)(F)F)nn1C Cc1oc(-c2ccco2)nc1C(N1CC(NC(=O)CCCN2CCC2)CC1C)=O N1(C(C(C)N(C(=O)C(C)N2CCCC2)C2CC2)=O)Cc2cccc(F)c2C1 c1(C(N2CCCCC(NC(C3OCC(C)C3)=O)C2)=O)cnc2ccccn12 N1(C(C2CC(F)CN2C(=O)CCN2CCCCC2)=O)C2CCCC1COC2 C1(NC(C(CSC)(C)NC(c2ccc(O)nn2)=O)=O)CC2(CCC2)C1O C1(CC(=O)OCC(F)F)CCCOCC1.C1(c2ccoc2)C(=O)N1C(=O)CO C(=O)(C(C(C)O)NC(c1cc(=O)cc[nH]1)=O)NC(C(C)SC)C c1(SC)nc(N2CCCC(CN(C)C(c3cccnc3O)=O)C2)c(C)c(Cl)n1 CC1=C(C(=O)NC(C2CC2C(=O)NCCc2nncn2C)C)SCCO1 C(CCC(=O)NCC1(CC)CNC(=O)O1)(C(C)C)NC(CCC(C)N(C)C)=O Cc1nccnc1C(=O)NCC(C(C)(C)C)NC(c1cc(Br)no1)=O C(C(CC(=O)N=c1cc2n([nH]1)CCCC2)OC)NC(C(C=C=C)C)=O C=C(C)CC(C(=O)NCCOCCCO)NC(c1ccns1)=O C1(C2CCN(C(=O)C(C)O)C2)(NC(Cn2c(C)ccn2)=O)CC1 c1(C(=O)NCC(C2CCOC2)NC(c2c(CCC)nns2)=O)nccc(Cl)c1F c1(C(=O)NCC=C(C(=O)NC(C=C)C2CCC2)C)ccc(CO)s1 CC(CCC(=O)N1CCC(NC(c2ncn(C)n2)=O)C1C(C)(C)C)N(C)C c1(NC(C2C(NC(CCOC)=O)CCCC2)=O)ccc(C(=O)OC)cc1Br C1(C(=O)NC2CC(Cl)(Cl)C2)CCOC(c2cccc(F)c2)C1 CCCC(C)(CC)C(=O)NC1CC(C)CN(C(C2CCN(C(=O)NC)CC2)=O)C1 C(CCC(=O)NC1CC1CNC(=O)CC1(C)CCOC1)SC C1(CCOC)(NC(=O)C#CC(C)C)CCN(C(C2(C)CCCOC2)=O)CC1 C1(OCC)CCCC1NC(=O)C(Cc1cccnc1)OC(=O)OC C1(NC(C2C(C)OCC2)=O)(CF)CCN(C(=O)CC2COCCOC2)C1 c1(C(=O)NC2C(CNC(=O)C(C3CCOCC3)O)C2)c(F)cccc1Cl C1(C(N(CC(=O)NCCn2ccnn2)CC2CC2)=O)CCOC1C1CC1 C1(C(=O)NCC(C)N(C(CN(CCC#C)C)=O)C)(CSC)CCC1 c1(C(N2C3C(C(=O)Nc4c(OC)c(F)ccc4)C(C3)C2)=O)ccc(C#N)c(C)n1 CC(C)CC(C(=O)NCC1CN(C(C23CSCC2C3)=O)C1)OC(F)(F)F c1(CC)nn(C)c(CC(N2CC3C(CNC(=O)C(O)C4CC4)C3C2)=O)c1Cl c1(C(=O)NCC(CCNC(=O)C(F)C2CCOC2)OC)cc(O)c(F)cc1N n1(CC)ccnc1CNC(=O)CC1(CNC(c2ccc(Cl)s2)=O)CCC1 c1(N2C(CNC(c3ccc(OC)c(C)c3C)=O)CCC2)nccc(S(C)(=O)=O)n1 C1(CC(=O)NCC2CC(O)CN2C(c2cnccn2)=O)NC(=O)CNC1=O c1(C(N2CCC(=CCNC(C3C(C)(Br)C3)=O)CC2)=O)ccc(Cl)nc1N c1(C(N2CC(NC(C(C)SC(C)C)=O)CC2(C)C)=O)cc2c(nn1)CCCC2 C=CCCCCC(=O)NC1CCC(CC(=O)NCc2cc(C(C)C)on2)C1 Cc1c(NC(C2(C)CCN(C(c3sccc3I)=O)CC2)=O)cncc1Br Cc1ccc(C(N2CCCC2C2(NC(=O)CC(Cl)Cl)CC2)=O)nc1C C12(CC)CCC(C(=O)NCCSCCN=c3[nH]nc(C)o3)(CC1)CO2 c1(C(N2CC(C)(CNC(=O)CC3CCC3)OCC2)=O)c(F)cc(C#N)cc1F c1(C(=O)NCCOCCNC(=O)CO)c(Cl)cccc1Br N1(C(CNS(N)(=O)=O)=O)CCn2ncc(CNC(C3(S(N)(=O)=O)CCC3)=O)c2C1 C1(CC)C(C(=O)N(C2CC3CC3C2)C)CCCN1C(=O)CNc1cccnc1 CC(C)(CCC(=O)NCC1(NC(C2CCCS(=O)(=O)C2)=O)CCOC1)[N+](=O)[O-] C1(C(N2CCC3CC23C(=O)NOc2ccccc2)=O)CC2C=CC1O2 c1(C(=O)NCC2CCC(C)CN2C(=O)C(F)=CCCF)c(Cl)oc2ccccc12 CN1CCCC(NC(C2CSCN2C(C2OC3CCC2C3)=O)=O)CC1 C(C(CC(=O)NCC(C)(C)C1CC1)NC(=O)CCc1nccn1C)OC C12CCCN(C1)C2=O.c1(C(N(CCCC)CCO)=O)csc(C(=O)OC(C)(C)C)n1 c1(N2CCCC(C(C)NC(c3c(C)cc(F)s3)=O)C2)cc2nncn2c(C)n1 C1(NC(c2c(CC)nns2)=O)CCCC12CCN(C(=O)CN1CCCC1C)CC2 C(=O)(CCC(=O)N1CCC(NC(C(N2CCCC(C)C2)=O)=O)C1)NCCNC(C)=O c1(C(=O)NC(C)CC2CN(C(=O)CSC3CC3)C2)c(O)nc(=O)n2c1CCC2 c1(C(C(=O)NCC)N(C2CCCCCC2)Cc2ccc(F)cc2)ccc(C#N)o1 C(=O)(CC(C(C)OC)NC(=O)Cc1ccoc1C)NCC(C=C)O c1(CN2C(C(=O)Nc3ccc(F)cc3Br)CCC2)cc(F)c(Br)cc1F c1(C(=O)NC2CCCC(N(C)C(c3ccnnc3O)=O)C2)ccc2nnnn2c1 Cn1nc2c(c1C(=O)NCC1CCN(c3ncc4ccnc-4[nH]3)CC1)CSCC2 CC1C(CNC(=O)CCCNC(C2CSCCS2)=O)C1(F)F Cc1nsc(C(=O)NCCOCCOCCn2cc(C(C)(C)F)nn2)c1N c1(NC(=O)NCC(C2CCCCO2)(C)C)sccc1C1CC1 C1(CCOC)CN(C(=O)C(O)CN(C)C)CCN1C(C1CC(=C2CCC2)C1)=O c1(OC)cnnc(C(=O)NC(C)(CNC(=O)CCC2CCN(C)CC2)C2CC2)c1 CC1CN(C(C2CN(C(=O)CC3COCC3O)CC2(C)C)=O)C12CCOCC2 N1(C(C2(C(=O)OC)CC2)=O)CCC(C)C(CNC(=O)Cc2cc(C3CC3)on2)C1 CC1CCN(C(=O)CCC2CNC(=O)N2)CCN1C(c1sc([N+](=O)[O-])cc1Cl)=O C(=O)(C(C)CC(C)C(C)=O)NC(CC)CCCC(=O)N(CC(F)F)CC1CC1 Cn1nnc(C(=O)NCCC(C)(C)NC(C2CC(C)(C)C2C(F)(F)F)=O)c1N n1(CC)cccc(NC(c2coc(CNC(=O)C(=O)C(C)CC)c2)=O)c1=O N1(C(CCSCC(N)=O)=O)CC2CC1CN2C(c1cnc(CC2CC2)nc1O)=O C(C(C(C)(C)C)NC(=O)Cc1cncc(F)c1)NC(c1c(CC)csc1)=O N1(Cc2n(CC)nnn2)CC=C(CCNC(=O)Cc2ccc3ocnc3c2)CC1 c1(C(N2CC(CN(C)C(c3ccc([N+](=O)[O-])[nH]3)=O)OCC2)=O)cc2n(n1)CCC2 N1(C(CCCCC#C)=O)CC2CN(CC(=O)NC(N)=O)CC2C1 CC1(C)C(=O)CC1C(=O)NC1CCC(CNC(c2ccncn2)=O)CC1 C1(OC)CCC(CC(=O)NCCCN(C(=O)C(C)(F)F)C2CCCCC2)CC1 CN1CCN(C(=O)C=Cc2ccccc2F)C(CNC(c2cncc(Br)c2)=O)C1 Cc1cc(N)cnc1C(=O)N(C(CC(C)C)C(=O)NC1C(C)CCCC1C)C CC1(C)COCC(C(=O)NCC2=CCN(C(=O)CC3CCCO3)CC2)C1 C(=O)(CCCCC(C)(C)C)N1CCC(N2CCN(C(CC(=C=C)C)=O)CC2)CC1 C1(CC=C)(C(=O)NCC2CC(=C3CC3)C2)CCCN1C(=O)C(C)OCCCC C1(C(=O)OC)CCN(C(C2(SC)CCC2)=O)C2CCCCC12 c1(C(N(CCNC(C(CC)c2cccnc2)=O)C)=O)ccc(N)c(SC)c1 c1(N2CCC(COC)(CNC(c3ccc[nH]3)=O)CC2)cc(C#N)ccc1[N+](=O)[O-] N#Cc1cc(C(N2CCCC2CCNC(C23CCCC2(C(N)=O)C3)=O)=O)on1 c1(NC(CCC#C)=O)ccc(NC(=O)CC2CCCC(C3CC3)O2)c(C)c1 N1(C(C(CCC)(C)CC)=O)CCC2(C1)CN(C(c1csc(C(C)=O)n1)=O)CCO2 C(C1=CCN(C(C2CCC(C)O2)=O)CC1)NC(C(C)NS(CC)(=O)=O)=O C1(CNC(CC=C)=O)CN(C(=O)CC2CC23CC3)CC1C(F)(F)F N1(C(CCSC)=O)CC(C(=O)NCCOCCCF)CCC1C CC(C)(CC(=O)N1CC(CCNC(C2CC2Cc2ccccc2)=O)C1)C1CC1 CCC(C)(C)CC(=O)N(CCCNC(=O)C(C)C(C)c1ccccc1Cl)C(C)C c1(CNC(=O)C(N)=O)cc(O)ccc1O.CC1(NC(=O)CN)CCC1 C1(C(=O)NCC23CN(C(CC(CC)(F)F)=O)C(C2)CO3)CC2CCCCN2C1 C(N=c1ccc(C(F)(F)F)n[nH]1)C1CCC(NC(c2ccc(C(N)=O)o2)=O)C1 n1(CC)nnc(C(=O)NC(C)(C)CCCNC(c2oncc2C)=O)c1C C1(CNC(C2CCCSS2)=O)(Nc2cc3nncn3cn2)Cc2ccccc2C1 C(CN=c1[nH]c2c(c(=NCc3nc4c(s3)COCC4)[nH]1)CSC2)=CCOC c1(C(N(C)CC2CCCN2C(=O)C(F)OC(F)(F)F)=O)cc(=N)[nH]c(=N)[nH]1 C12(C(N3CC(O)(CNC(C4CC(N(C)C)C4)=O)C3)=O)CCCC(C1)OC2 c1(C(=O)NCC(CC)C2CCOC2)nc(C2CCOCC2)no1 c1(C(=O)NCCCCC(C)NC(c2ccco2)=O)ccc2ccnn2c1 c1(OC)ccc(C(N2CC(NC(=O)CN3CCN(C)CC3)C3CC23)=O)cn1 N#CC1CN(C(c2ccc3nonc3c2)=O)CCN1C(c1ccc(CO)nc1)=O Cc1cc(Cl)cc(C(=O)NCC(O)CNC(=O)C=Cc2ccoc2)c1N C=Cn1nccc1C(=O)NC1CCC(NC(c2cccc(-n3cccc3)n2)=O)C1 c1(N2CCC(NC(=O)C=CBr)C(F)C2)ncc2c(n1)CCOC2 C1(NC(C(COC)O)=O)CCC2CN(C(=O)C(C)Oc3cccc(C)c3)CC12 Cc1cc(=NC2CC(CN(C)C)C2)[nH]c(N(C)CC2CCC(C3CC3)O2)n1 C(=O)(C(CN=[N+]=[N-])NC(C1OCC2CCCC12)=O)N(C)CC1CCC1 CC(C(=O)N1CCCC1C(C)NC(=O)CN1CCCC1)C(F)(F)C(F)F N1(CC(=O)NCCCN(C(c2csnc2Cl)=O)C2CC2)CC2CC2C1 CC(=O)CCC(=O)NCCCC(=O)NCCC1CCC(=O)N1 CC1COC2(C1)CN(C(=O)COC(C)(C)CNC(C1(CC3CC3)CCC1)=O)C2 c1(C(=O)OCC)no[nH]c1=NC(=O)C(C)C1CCN(Cc2cnn(C)c2)CC1 c1(C(N(C)CC2CCN(C(C3OCC(C)C3)=O)CC2)=O)cnc2ccccc2c1 Cc1nc(O)nc(C)c1C(=O)NC(CNC(C1CC(C(C)(C)C)C1)=O)CC(C)C CCCC(C(=O)N(C(CO)C(C)C)C)NC(C1CC(O)C(F)C1)=O CC1CC(NC(c2ccncn2)=O)CCN1C(c1cnc(F)c(F)c1)=O C1(CC(N(C2(CC(C)(C)C)CC2)C)=O)CCN(C(C2CC2C(C)(F)F)=O)C1(C)C C12(NC(C(C=C)O)=O)CC(C1)N(C(C1CCCCN1C)=O)C2 CCCC(C(=O)N1CC(C)(NC(C2CC(=O)N(C(CC)CC)C2)=O)C1)NC(N)=O Cc1cc(S(=O)(=O)N2CCOCC2CNCc2cccc(F)c2Br)c(F)cc1Cl N1(C(COC2(C#C)COC2)=O)CC2CCCC2(NC(=O)C(C)Cn2cccn2)C1 C1(CNC(C2C3CC4C(C3)C24)=O)C2CN(C(c3cnccn3)=O)CC12 N1(c2ccc(OC)cc2)CCCC(NCCc2nc(Br)c(C)s2)C1=O Cc1ccc(CC(N2CC(CNC(=O)CNC(N)=O)C(C)C2)=O)cc1Cl c1(CCC(C(=O)NCC)N(CCCO)CCC)nc2ccc(F)cc2s1 c1(CCCCCC(=O)NC(CCC#N)CCO)ccc([N+](=O)[O-])cc1 C1(NC(C2CC(OCC)C2)=O)CCN(C(=O)Cc2cc(CC)n(C)n2)C1(C)C C1(C(=O)NCC(C)N(C)C(c2ccc(P(C)(C)=O)o2)=O)CCC2(CC1)CC2(F)F c1(C(N2C3CN(C(c4n(C)nnc4)=O)C(C3)C2)=O)scc2c1CCCC2 N1(C(CC(C)(C)c2ccccc2)=O)CC(NC(=O)C2=COCCC2)CC(F)C1 C=CC(C)CC(=O)NC(CC1CC1)C(=O)N(C)Cc1cccs1 N1(C(c2cc(C(=O)OC)oc2)=O)CCC(NC(C2(SC)CC2)=O)CC1C(C)C N1(C(COCC)=O)CCC(C2CC2NC(=O)C=Cc2cc(C)c(C)cc2C)CC1 C#CCCCCCC(=O)NC1CCC(C)(CNC(c2cc([N+](=O)[O-])cn2C)=O)C1 c1(C=O)cc(C)nn1CCO.C1(CNCC)CCCCN1C(=O)C(C)C1CC1 N#Cc1ncc(NCC2CCCC(NC(=O)CCc3cc(Cl)cs3)C2)nc1C#N C(=O)(C1=C(F)CN(C(=O)COCC(F)F)CC1)N1CC(C)(C#N)C1 C(=O)(C#CC1(C)CCCO1)N(C1CN(C(C(CSC)(C)C)=O)CC12CC2)C C#Cc1cc(C(=O)NCCNC(C2CCCCC2N(C)C)=O)ccc1C c1(C(=O)NC2CCOCC2NC(C2CCC2(F)F)=O)ccc2nc[nH]c2n1 c1(CNC(C(c2ccc(Cl)cc2)OC)C)ccc2c(c1F)OCCO2 c1(C(N2CCC3(C(NC(CN(C)C4CC4)=O)C3)C2)=O)cccc([N+](=O)[O-])c1 c1(OC)ccc2occ(C(=O)N(C3CCN(C(=O)CC4(C)CC4(Cl)Cl)C3)C)c2c1 C=CCCCN(C(C(C)OCC)c1csnn1)CCc1ccco1 C(CCCCC(=O)N1CC(C(=O)NC2CC(=O)NC2=O)OC(C)C1)=CC C1(CCNC(Cn2c(C)nc(C)n2)=O)CN(C(=O)C=CC2CCC2)CC(C)O1 C1(CNC(CC(CC)(F)F)=O)C2CCCC1N(C(=O)C(O)C(C)(C)C)C2 c1(CNC(C(C)C)=O)ccc2c(c1)CCCC2NC(c1cc2n(n1)CCCO2)=O C(=O)(CN=c1[nH]c(=NCc2ccc(C)cc2Cl)[nH]c2c(F)cccc12)NC C=CCC(C)(CC)C(=O)N(CC(O)CNC(=O)CCCOCCC)C N1(C(CCCOC)=O)CCC(N(CCO)C(c2ccc(C)cc2)=O)CC1 C(=O)(C(O)C1=CCCCC1)N1CCC2C(C(=O)Nc3c(C)c(N)ccc3)C2C1 N1(C(C(CC=CC)CC)=O)CCCCC(CNC(C2CCCC2)=O)CC1 C(=O)(C(F)CCC(C)C)NCC1(OCC)CN(C(=O)Cc2nccn2C)C1 C(C(C)(C)C(=O)NC1CN(C(=O)C(C)CN2CCOCC2)CC1O)OC N1(C(C2N(C(c3c(CC)nns3)=O)CC=C2)=O)CC2CCCC(O)C2C1 c1(OC)ccc(-c2nc(C(=O)NC(C)CN(C)C(c3n[nH]cc3C)=O)cs2)cc1 C(C)(C)(CCC(=O)NC(C)CS(C)=O)NC(CC1ON=C(C)C1)=O Cc1cccc(C2CC2C(=O)N(c2ccc(Cl)nn2)CC(=O)O)c1 c1(CC)cccc(C(=O)NCC2(C(C)(C)O)CN(C(C3CCCN3C=O)=O)C2)c1 C1(C(=O)NCCCN(C(=O)C(C)CC2CC2)C(C)C)CN(C)C(=O)N1 c1(CC(=O)N2CCNC(=O)C(C)OCC2)cnc(C)[nH]1.CCCCCCOC c1(C(C(=O)NC(CC)CN(C)C(c2cn[nH]c2)=O)O)cccc(C)c1F Cc1cn2ccc(C(=O)NC(C3CN(C(c4n[nH]c(=N)[nH]4)=O)CCO3)C)cc2n1 c1(CC)ccc(NC(=O)CC2CCCC(NC(C3CCCOC3C)=O)C2)c(C)c1 c1(C(=O)NCCNC(CC)=O)coc2c1CN(C(=O)C(C)(O)C1CC1)C2 CC1(C(=O)NCc2cc(C(N3CCC(CO)C3)=O)no2)CCCC1O C1(O)(CNC(C2C=CCN2)=O)CCCN(C(c2cccs2)=O)C1 C1(C)(C(N2CC(OC)C(O)C2)=O)CC12CCN(C(C1CCOCC1)=O)CC2 N1(C(C(C)OCCC=C)=O)CC(C2CCCN(C(=O)CN(C)S(N)(=O)=O)C2)C1 C=CCC(CC)C(=O)NC(CCC)CC(=O)NC(COC)COC C(=O)(C(O)C(F)(F)F)N1CCC(N(C(c2cn(CC(F)(F)F)cn2)=O)CC)CC1 N1(C(=O)NCC2CCCN(C)C2)CCCSCC1CN(C)C CC1CN(C(=O)C=Cc2ncc[nH]2)CCCN1C(=O)C1=C(Cl)CCCC1 N1(C(C(CC)OC)=O)CCC(NC(=O)Cc2ccn(C)n2)C(CO)C1 C1(COC)(CNC(C2(F)CCOC2C)=O)CCCN1C(=O)Cc1cnsc1 CCC(O)CC(=O)N(C(CNC(=O)CCC1COC(C)(C)O1)C1CC1)C Cc1scc(C(N2CC(CO)(NC(=O)CC3CC(C)OC3C)C2)=O)c1C N(C1CCCc2n[nH]cc21)C(CC(C)NC(c1nc(C)nc(O)c1)=O)=O C(=O)(C(F)CCC(C)(C)C)N1CCC(F)(C(=O)NC(C(C)C)(C)CO)C1 C1(C(C)NC(=O)C(C)(C)c2ccnn2C)CCCN(C(c2cccc(F)c2)=O)C1 c1(C(N2CC(CC(=O)Nc3ccc(C)cc3C)(OC)C2)=O)cc2c([nH]1)CCOC2 C1(C(=O)NC2(CF)CCN(C(=O)CCc3ccc(F)cc3)C2)CC2CCC1CC2 C1(C)(COC)CC(NC(C2(CF)CC2)=O)CN1C(c1nc(O)c(C)s1)=O c1(C(=O)NC)cncc(C=CC(=O)NCC(C2CC2)NC(=O)C2=COCCO2)c1 CCCC(C(=O)NC1CN(C(=O)CC)C1)NC(=O)CCn1cnnn1 c1(OC)ccc(C2C(C(N3CC(C)CCC3C)=O)CCN2C)cc1OC C=CCCCC(=O)NC1CCCC1CNC(c1ccc(O)cn1)=O c1(C(CC)OCC(=O)N(C(c2nnnn2C)CC)C)cccnc1 c1(C(N2CC(OC3CCN(C(c4c(CC)scc4)=O)CC3)C2)=O)cc(C)nc(C)n1 C1(NC(c2ccc(CC)s2)=O)CCN(C(c2cc(C(N)=O)ccc2F)=O)CC1F c1(CN2CC(C(N3CCC(F)C3)=O)SCC2)c(OC(F)F)cccc1Br N1(C(C(C=C)OC)=O)CC(C(=O)NCCc2ccco2)CC(C)C1 C(CC(F)F)(C(=O)NC1CC2(C1)CC(O)C2)N(C)C(c1sccc1CO)=O c1(-c2cncc(NC(c3ccn4ccnc4c3)=O)c2)ccc(C2=CCCC2)cc1 CS(=O)(=O)c1ccc(C(=O)NC2CCN(C(c3cc(F)cc(F)c3Br)=O)C2)nc1 C=CC1OCCC1C(=O)NCc1cnn(C)c1C(=O)N(CC1=CCSC1)C C1(N(C(=O)C=CC(F)(F)F)C)CN(C(c2ccnn2C)=O)CCC1O C(=O)(CCCCCNC(=O)COCC1CCCCO1)N1C(C)(CC)CC1 CCC(C)(C(=O)NC1CCCN(C(=O)CC(c2cccc(F)c2)O)CC1)C(N)=O CC1CCN(C(=O)CCc2cncc(F)c2)C1CNC(c1cccn1C)=O CN(C(=NCCCc1nncs1)NCCCN1CCOCC1)CC1CC1 N1(C(=O)NCCS(CCCCOC)=O)CC2(CCCC2)c2ccccc21 C1(F)(C(=O)NCC(CC=C)NC(=O)Cn2cc(C)cn2)CCCN(C)C1 C1(CNC(C2(CC#C)CC2)=O)COCCN(C(=O)CN2CCC(=O)NC2=O)C1 c1(C(=O)NCC2CC(NC(c3cc(C)cc(C)c3)=O)C2)ccc(F)c2cccnc12 C1(NC(c2ccc(C)cc2)=O)CCN(N2CCC(CCO)CC2C(C)(C)C)CC1 N1(C(C(CCC)OC)=O)CCC2(CC1)CN(C(c1n[nH]c3c1COCC3)=O)C2 CCCC(C(=O)N1CCC(N(C(=O)Cn2cccn2)CCOC)C1)NC(C)=O N1(C(c2c(C)cco2)=O)CCC2(CCOC2)C(CNC(c2cc(CO)[nH]n2)=O)C1 C(CC(C(=O)NCC1CCN(C(C2CCN(CC(C)C)C2)=O)CC1)N(C)C)SC C(c1ccccc1)=CC(=O)NCC1CC(OCC(=O)NC(C)CCC2CC2)C1 Cc1ccc(F)c(N)c1C(=O)NCCN(C(=O)C1=C(Cl)CC1)C1CCCC1 c1(C(N(CCCNC(C(CC#C)C)=O)C2CC2)=O)ccc(Br)c(C)c1N N1(C(CC2(C)CC2)=O)CCCCC1CCNC(=O)C(C)(C)n1cccn1 Cc1nc(C)c(C(=O)NC2CCOC(C(=O)NCCc3ocnc3CO)C2)[nH]1 c1(OC)cc(CN2CC(C)CC2C(=O)NCCC(N2CCCCC2)=O)ccc1Br C1(C(N2CC(C)(NC(=O)CCc3ccc(Cl)s3)C2)=O)CC(F)C(=O)N1 Cc1nc(N2CCCCC(CNC(=O)C(F)(F)CO)C2)cc(C#N)n1 C1(CC(=O)NCc2cnccc2Cl)C2CN(C(C3CCC4(CC4)C3)=O)CC12 C1(CCNC(C2(NC(Cc3cc(C)no3)=O)CCC2)=O)CCOC1(C)C C1(CC(=O)NCC(CN(C)C(c2coc(C3CC3)n2)=O)O)CCC12CCC2 Cc1cc(C(=O)NC23CCC(N=[N+]=[N-])C2C3)cc(N)c1Cl N1(C(N(CC(=O)OC(C)(C)C)C)=O)CCN(CC(c2cc(C(F)(F)F)on2)=O)CC1 c1(C(N2CCC(CC=C)C2)C(=O)NCCC2(C)CC2)ccc2ccn(C)c2c1 N1(C(C(CCC)OC)=O)CCN(C(=O)Cn2nc(C)c(C)c2C)C(CCCC)C1 C(=O)(C(CNC(c1cncn1C1CC1)=O)CC1CC1)NCC1(CC)CCOC1 c1(C(=O)NC2(CCOC)CCN(C(C3(O)CC3)=O)C2)n[nH]c2c1CC1CC21 N1(C(Cc2ncc(CC)[nH]2)=O)CCCC2(CCN(C(=O)CC3CSCCS3)C2)C1 C1(O)(C(=O)NCCC(CNC(CCc2ccc(C)cc2)=O)O)CCOC1(C)C N1(C(C2(F)CN(C(C(C3CC3)OCC)=O)C2)=O)CCCC(C)(CC)CC1 Cc1cc(NC(C2CCC(NC(=O)CN(C)C)CC2)=O)ccc1[N+](=O)[O-] N1(C(c2c(C)occ2)=O)CCC2(CC1)CC(NC(C1CCC(N=[N+]=[N-])C1)=O)C2 C1(O)(CNC(C2(CNC(CSCCC)=O)CC2)=O)CCC(C)CC1 C12(C(=O)NCC3C(NC(c4scc(C)c4C)=O)C3)CCCC1C2(F)F C1(OCCNC(C2N(C(c3c(C)nns3)=O)CCC2)=O)CCN(C)CC1 C12(CC(C)(C)C1)C(=O)NC2.C1(NC(COCC(=O)NC)=O)CCOC1C(C)C CC1CN(C(C2COCC(C)O2)=O)CC(C(=O)NCCSC(C)(C)C)O1 N1(C(C=CC(=O)N(C)C)=O)CC2CC1CCC2NC(C1(C)CCCO1)=O C1(N(C)C)CN(C(=O)CC2CC(C(=O)OC(C)(C)C)C2(C)C)CCC1O Cc1c(NC(=O)C(C2CC=CCC2C)N(C)CCc2nccs2)cccc1Cl N1(C(C(C)(F)F)=O)CC2(C1)CN(C(c1ccnc(Cl)c1Cl)=O)CCO2 O=C1CN(C(=O)Cc2cncnc2)C(C(=O)NCc2cnc(O)c(F)c2)CN1 c1(C(C(=O)NC(CC)C)N(CC(C)(C)N2CCCC2)C)nc(Cl)cc(Cl)c1C c1(C2N(C(CC(C)NCC(F)(F)F)=O)CCC2)cccc(C(F)(F)F)c1 C1(NC(C(C2CCCC2)OC)=O)CC(N=c2[nH]c3cc(Br)cnc3s2)C1(C)C C=CCC(C(=O)NCC12CC(NC(C3CCCCO3)=O)(C1)C2)OC c1(-n2c3nnc2s3)ccc(S(N)(=O)=O)cc1.c1(C(C)CNC(N)=O)nncn1C S(=O)(=O)(CCC(=O)NCC1(Nc2cc(COC)ccc2C)CC1)NC c1(C(=O)NC(CN(C(=O)Cc2ccoc2)CC)C)nn(C)cc1[N+](=O)[O-] c1(C(C(=O)NC)N(C2CCCC2)Cc2ccc(F)cc2)nc(Cl)sc1Cl CCCC(C(=O)N1CCC1CNC(=O)CCc1nc(C)c(C)[nH]1)OCC Cc1ccc(O)cc1C(=O)NC(CC1CC1)C(=O)Nc1cncc(N(C)C)c1 c1(OC)ccc(CNC2CCCC2C(=O)Nc2cncc(C(F)(F)F)c2)c(O)c1 C12(C(=O)NC(CC=C)CNC(c3ccn(C)c3)=O)CCC(C)(CO1)C2 c1(OC)ccc(-c2oc(C)cc2C(=O)NC(C)CN(C)C(c2cncs2)=O)cc1 C1(c2ccccc2Cl)(C(=O)NCC(CCNC(C(CC)C)=O)O)CCCCC1 C(C(C)N=c1[nH]cc(CNC(=O)NCCCN2CCN(C)CC2)s1)OCCC c1(OC)ccc(F)cc1NC(=O)COCCNC(=O)C(C)=C1CCCC1 c1(CC)sc(C(=O)N(CCCN(C(=O)CS(=O)(=O)NC2CCCC2)C)C)cc1C c1(CN(C)C(c2ccn(CC(F)(F)F)c(=O)c2)=O)c2c(nn1C)CCC2 CC1CCCc2c(C(=O)NC3CCCCN(C(=O)CCc4cnn[nH]4)C3)cnn21 C1(SCC)CCCCN1C(=O)CN(CCOC)C(c1cccc(C)c1)=O C1(C(=O)NC2(C3CCCN3C(c3ccc(C4CC4)nc3)=O)CC2)C2CCCCC12 c1(C(C(=O)NCC(Cn2cc(CN(C)C)nn2)OC)C)ccc(C)s1 C1(NC(C(C(C)C)C)=O)CN(C(c2cc(F)ccc2O)=O)C2CCCC12 N1(C(=O)CCc2csc(Br)c2)CCN(C(c2nn[nH]c2Cl)=O)C2CC12 N1(C(c2cc(C)nc(O)c2)=O)CCC2CN(C(=O)C(C)Cc3cnn(C)c3)CC12 Cc1oc2cc(C(=O)N(CC(C)NC(=O)C(N3CCCC3)C3CC3)C)[nH]c2c1C N1(C(COCCOCC#C)=O)CCN(C)C(CNC(C2(CC)CC2)=O)C1 C(N=c1cc(C)nc(NCCn2ncc3cccnc23)[nH]1)c1cncc(C)n1 C1(OC)CC(CNC(=O)C(F)=C2CCC2)N(C(=O)CC(C)C)C1 Cc1cc(O)nnc1C(=O)N(CCCNC(C1CCC(F)C1)=O)CCO C1(CCN(C(CN2C(C)CCC2)=O)C)CCCCN1C(=O)C=Cc1ccsc1 N1(Cc2ccc(C(=O)O)s2)CCC2CN(C(c3ncc(F)cc3F)=O)CC12 c1(NC(CN(C(=O)C=CC(=O)NC2CC2)CC#C)=O)cnn2c1OCCC2 CC(C(C)(C)C(=O)NC1CC1(C)C(F)F)NC(c1c[nH]c(=S)cn1)=O N1(C(COC(CC)(C)C)=O)CCC(C(=O)NC2CCCC2COC)C(O)C1 c1(CNC(C2CC(S(C)(=O)=O)C2)=O)cnn2c1CN(C(C1(CO)COC1)=O)CC2 n1(CC)nnnc1C(c1cncs1)NC(C)Cn1ccnc1C C=CC(C)(O)CC(=O)NCC1CCC(CNC(c2ccsc2COC)=O)CC1 C(=O)(C1=CCN(C(C2COCC(C)O2)=O)C1)N(CC(CC)OC)C c1(C(=O)NCc2cn(CCNC(CCCCSC)=O)nn2)cc2ncccc2s1 Cc1cccc(Br)c1C(=O)NCC1CCCN1Cc1csc(Br)c1 C1(F)(N(C(C(C2CC2)OCC)=O)C)CCN(C(C2(OCC)CCCCC2)=O)CC1 Cn1cccc1C=CC(=O)OCC(=O)N(CC(C1CCCCC1)(C)C)C(C)(C)C N1(C(CC(C)CF)=O)CCCC2CN(C(C3(CO)CC3)=O)CC12 CCCC1C(=O)N2CCC1C2.c1(SCC)ccccc1Br.C1(=O)C(OC)CO1 N1(C(CCC#C)=O)CC(O)CC1CNC(c1ccc(OCC)cc1)=O CCS(=O)c1ccccc1C(=O)NCC(C)NC(=O)Cc1cccc(C#N)c1 c1(C(N(C)CC2CCN(C(c3coc(Cl)n3)=O)C2)=O)ccc(S(=O)(=O)N(C)C)o1 c1(OC)nc(C)ccc1C(=O)NCC1(CNC(=O)CCC2CCOC2)CC1 c1(N(C(=O)CC2CS(=O)(=O)C2)CCO)ccc(C(=O)O)cc1[N+](=O)[O-] c1(C(N2C(C(=O)NC(CC(C)C)C)CCC2C)=O)ccc(OC(F)(F)F)c(F)c1 C=CC1(C(=O)NCC(C)(C)CCNC(c2ccc(C(N)=O)o2)=O)CCOCC1 C=C=CCCC(=O)N1CCCCC1CC(=O)NCC(O)CN(C)C1CC1 N1(CC(COC(C)C)O)CCN(C(=O)NCC2CNC(=O)O2)CC1 C12(C(=O)NCC(C)(CC(C)C)NC(Cc3c(C)nc[nH]3)=O)CCC(C)(CC1)OC2 N1(C(C(c2scc(C)n2)C)=O)CC(C2CN(C(C3CN(C4CCOC4)C3)=O)C2)C1 C1(NC(C(F)=CCC)=O)CCN(C(c2ccc(OC)cc2F)=O)CC(C)(C)C1 c1(C(=O)NCCCNC(C2C(C)C2)=O)ncc(SCC(=O)NC(C)(C)C)cc1C N1(C(C2C(c3ccc(C)cc3)CCC2)=O)CCCCCC1C(=O)N1CCCO1 CCC(CC(=O)N1CC(CNC(=O)C=Cc2ccccc2C)C1)C(C)(C)C c1(C(N2C(C(=O)NC(CC=C)C)CCC2)=O)ccc(C)nn1 Cn1cnc(C(=O)N(CCC(=O)NCC(c2ccsc2)O)C2CC2)n1 c1(C(N2C(C)CCC(NC(CC(=O)OC)=O)C2)=O)nn(C)c2c1CCC2 c1(C(CC)CC)nc(C(COC)C(C)C)nn1-c1cncc(Br)c1 CCCCC(O)CC(=O)N1CCOC(CNC(=O)CC(C)CC)C1 c1(C(=O)NC2C3CN(CC(=O)NCC#C)CC32)cnc(COC)nc1O CC1CN(c2cc(Nc3ccc(NC4CCCC4)cc3)ncn2)CC(CO)O1 C1(C(N(C)CC2CCCC(NC(c3c(C)noc3)=O)C2)=O)CC2(C1)CC(F)(F)C2 N1(C(c2csc(C)c2C2CC2)=O)CC2CCC(NC(C3CCCC3)=O)(C2)C1 c1(C(=O)NC(C)C(=O)NCCN2CCC3CC23)c(Cl)cnn1C N1(CC)CCOCC1CC(N1CCCC1CNC(c1cc(Br)no1)=O)=O C1(CCC)CCCCC1ONC(C1(OC)CCCCC1)=O.c12ncoc1NC2=O C#CC1CCC(NC(C2CCC(NC(=O)Cc3c(C)n[nH]c3C)C2)=O)C1 c1(C(N2C(C3CCN(C(C4(SC)CCC4)=O)CC3)CCC2)=O)cc(F)ccc1F Cc1c(C(N2CC(O)CC2C(=O)NC(C)(CO)CO)=O)cccc1O N1(CCC)CCCCC1C(=O)NC(C)CCN(C(=O)CCC1(C)CC1)C C(=O)(C1=NOC2(CCOC2)C1)NCC(CNC(c1c(F)ccc(C)n1)=O)(C)OC Cc1cc(NC(=O)Nc2nc(-c3c(C)nn(C)c3C)cs2)cc(C)c1 N1(C(c2ccc(C)c(Br)c2C)C(=O)NCC(C)C)CCn2c(CCO)nnc2C1 CC(C)C(C(=O)NCCN(C)C(C1(C)CCCN1C(=O)OC(C)(C)C)=O)C(C)C Cc1ccncc1C=CC(N1CCCC(N(C(=O)CCF)CCn2cncn2)C1)=O C1(C(=O)NC(CCCNC(c2c(C)cnn2C)=O)C)CCN(CCO)C(=O)C1 C1(CC(=O)NC(CC)CCOC)(NC(C(COCC)C)=O)CCCCC1 N1(C(C2(C)COCCO2)=O)CCCCCC(NC(c2cc(C3CCC3)on2)=O)C1 CCC(C)CCCCC(=O)NCCC1(C(=O)NCC(=O)N(CC)OC)CC1 CC1CCN(C(=O)Cc2cccnc2Br)CC1NC(=O)C(F)(F)CO n1(-c2ccc(C#N)cc2)ncc2c1CCCC2NC(c1ccc(F)cc1)=O Cc1cc(C(N2CC3(NC(=O)C(C)SC(F)(F)F)CCC2C3)=O)c(O)c(C)c1 c1(CNC(c2ncccn2)=O)nc2c(s1)CCN(C(C1CC(CF)C1)=O)C2 C12(N)CCCC1C2(F)F.n1(CCCC)nnnc1C(C)(CCSC)Nc1ccccc1 c1(CN2CC(C(=O)OC)CC(CC)C2)cc2cc(Br)ccc2s1 c1(C(C(F)(F)F)OC(C2C(C(=O)OCC)C23CC3)=O)ccccc1OC C1(C(=O)NCCN(C(CC)C)C)CN(C(=O)CN2CCCCCC2)CC1(C)C C(=O)(C1c2ccccc2-c2ccccc21)NCC(C)NC(C=C1CCC(C)C1)=O CCCC(C)CC(=O)N1CCC(C(=O)NCCF)CC1C C1(c2c(C(=O)NCCC=CC)c[nH]n2)CCCCN1C(=O)CC1CCC(F)CC1 Cc1cccc(C)c1OCC(N1CC2CC1CN2C(c1ccncc1Cl)=O)=O N12CCC(C(F)(F)F)C(C1)NC(=O)C2.c1(NCCCl)ccccc1 C12(NC(=O)C(O)CCc3ccccc3)CCCC1CN(C(c1cscc1Cl)=O)C2 C1(C(CO)NC(c2cn(C)nc2)=O)CCCN(C(=O)Cc2cnc(C3CC3)o2)C1 C(=O)(C1=CS(=O)CCC1)NC1C2CCN(C(c3cc(C)cc(C)n3)=O)C21 N1(C(C(C=C)O)=O)CCC(F)(C(=O)NCc2cncn2CCC)CC1 C1(C)(CNC(C(C2CCN(C(CC3CC(OC)C3)=O)C2)C)=O)CCCCC1 C1(C(N2CC(O)(CNC(CN(C(C)C)C)=O)C2)=O)CCc2c[nH]nc2C1 N1(C(C(C)OCC)=O)CC(C)C(N=c2[nH]c(Cl)nc(C(F)(F)F)c2F)C(C)C1 c1(C(=O)OC)cnc(=NC(CCN(C(=O)C=C2CCC2)C)C(C)C)[nH]c1 CC1(c2cn(CC(N3CC(Cc4cccnn4)C3)=O)nn2)CCCC1 c1(OC)ccc(C=CC(=O)N(CCCNC(=O)CC2CCC23CCC3)C)cc1Cl Cn1cc(C(F)=CC(=O)NC2CCC(C(=O)NC34CCC(F)(CC3)C4)C2)cn1 c1(CNC(=O)NCCN(C(C)(C)C)CC)cc(Br)c(F)cc1Cl C=CCCCCC(=O)NCC1C=CC(NC(c2cc(Cl)ccc2NC(C)C)=O)C1 C1(CNC(c2nc(C)c(C)s2)=O)CCC(C)N(C(c2cnn(C)c2F)=O)C1 CONC(=O)C(=O)NC(C1CCN(C(=O)Cc2ccns2)CC1)C N1(C(C(CC)N(C)CC)=O)CCC(C)(C)C1CC(=O)Nc1ccc(F)cc1C Cc1cc(Cl)cc2[nH]c(C(=O)NC3CCN(C(C4CN(C)C4)=O)CC3CO)cc12 C1(C(=O)NCCCN(C(CC2CC(OC)C2)=O)C(C)C)CCN(CC(F)(F)F)C1 N1(C(C(C2CC2)SC)=O)CCN(C(=O)CCC2CC2)C(CCO)C1 C1(NC(c2ncn(CC)n2)=O)CC2C(NC(=O)CSC3CCCCO3)C2C1 N1(C(c2nnn(C)n2)C2CC2)CC2(CCCC2)C1c1ccncc1 N1(C(C2C(C=C)OCCC2)=O)CCC2CN(C(=O)CS(=O)(=O)NCC)C2C1 C1(CNC(c2cncs2)=O)CN(C(c2nc[nH]c3nccc2-3)=O)CC2(CCC2)O1 C1(NC(C2CCC(=C)CC2)=O)CCC(C)N(C(=O)C(F)Cc2ccccc2)C1 N1(C(C(CO)OC)=O)CCC(CC(C)NC(=O)CCc2ncc(C)[nH]2)CC1 N1(C(C(C(=O)OC)C)=O)CC(NC(c2cccc(F)c2OC)=O)CC(F)C1 C1(C(=O)NCCCN(C(Cc2c(C)nsc2)=O)CCO)COCC1(C)C CC1CCN(C(=O)CC2CCCC(=O)N2)C(C)C1NC(C1CN(C)CCO1)=O CC1CC2CC2CC1C(N1CCC(Cc2cn(Cc3ccco3)nn2)CC1)=O n1(CC(=O)NC2C(C)CN(C(C3OCCCO3)=O)C2)ccc2ccccc2c1=O c1(CN(C(=NCCOC)NCc2ccc(COC)o2)C)c[nH]c2ccc(C)cc12 n1(CC(C)C)ccc(=NC(=O)CC2COCCN2C(c2cc(Cl)n(C)n2)=O)[nH]1 C1(CC=CC(=O)NCCCN(CC(N)=O)C)CCCN1C(N)=O.C(C)(C)(C)OC=O N1(C(C(CSC)C)=O)CCC(NC(c2cncc(Cl)c2Cl)=O)C12CC2 C1(C(N2CCC(C3=NOCC3)C2)=O)C2C3CC4C1C1C2CC3C41 N1(C(C(C(C)O)(F)F)=O)CC(O)(C2(CNC(c3nocc3Br)=O)CC2)C1 n1(CC)cc(C(=O)NC(c2cncs2)C)c(C)n1 N1(C(CC2(OC)CC2)=O)CCC2CN(C(C3CC(C(C)(C)C)=NO3)=O)C2C1 C1(C(=O)OC(c2ccccc2Br)C(=O)OC)CCn2nccc2C1 Cc1c(C(=O)N(C)CCNC(c2cc(Cl)c(Cl)[nH]2)=O)cnc2ncnn12 C(N=c1cc(Cl)nc(S(C)(=O)=O)[nH]1)C1OCC(CNC(C2(OC)CC2)=O)C1 N1(C(CCC)=O)CCC(C)(C)C1CNC(=O)C(C1CCOCC1)NC(C)=O C1(CCNC(CCN(C(C2C(C(C)C)CCC2)=O)C)=O)CC2C=CC1C2 C#CC1CCC(CNC(C2CCC(CNC(C3(CCCF)CC3)=O)O2)=O)CC1 C1(C2CCN(C(c3ncn(C4CC4)n3)=O)C2)(NC(C2N(C)C(=O)CC2)=O)CC1 C1(CC)CN(C(c2cc(C(F)F)ccc2F)=O)CCC1NC(=O)C(CC)C(C)C C1(CNC(C2(C(C)C)COC2)=O)C2CC1N(C(=O)Cn1cnnn1)C2 N1(C(COCCC#C)=O)CC2CCC(C1)C(NC(c1sc(C)cc1Cl)=O)C2 C1(C2(O)CN(C(=O)C(C)(C)F)C2)(CNC(C=COc2c(C)occc2=O)=O)CC1 c1(C(=O)NC23CC(NC(=O)C(F)(F)C4CC4)(C2)C3)cc(SCC)cnc1OC c1(C(N2CCOCC(NC(CCCCN(C)C)=O)C2)=O)cc2c(cc1O)OCO2 Cc1sc(=O)n(CC(N2CCC(CNC(=O)C=CCO)CC2C)=O)c1C c1(C(N2CC(OCCNC(CCC=CCC=C)=O)C2)=O)cc2nccn2c(O)n1 N1(C(C(CC)(C)C#N)=O)CCCC(O)(CNC(c2cc([N+](=O)[O-])oc2C)=O)CC1 N1(C(C(COCC)C)=O)CCCOC(CNC(=O)C(CO)OC)C1 C(=O)(C1=COCCO1)NCCC(C)(C)NC(c1cccc(C2CNC(=O)C2)c1)=O c1(OC)cc(C#N)ccc1C(N1CC(NC(=O)C(C)CC(C)(C)C)CC1(C)C)=O Cc1[nH]c2ccccc2c1C(=O)NCC12CC(CN1C(=O)Cn1cccc1)C2 CC(C)(C)CCCCC(=O)NCC1OCCC1C(N1CC(n2cccn2)C1)=O c1(OC)ccc(C)cc1NC(=O)C1=NOC(CNC(=O)C(C)C2CCCC2)C1 c1(C(=O)NCC2(CNC(c3cc[n+]([O-])cc3)=O)CCC2)c(Cl)csc1Cl c1(C(=O)NCC(C2CCC2)NC(C=NOC)=O)cc2ccc(C(F)(F)F)cc2[nH]1 C1(C(=O)NCCCC(=O)NC)C2CCN(C(=O)C(C)C#N)CC12 c1(C(=O)NCC2N(C(C(C=C)O)=O)CCC(C)C2)c(C)ccc2nonc12 N1(C(=O)N)CCCOC2CCCC12.c1(C2CCN(C=O)C2)ccccc1F C1(CNC(CC(CC)SC)=O)CN(C(C2(CO)CC2)=O)C2CCCCC12 C1(C)(CNC(c2n(C(C)C)ncc2)=O)CCCN(C(=O)CC2(C)CC2(F)F)C1 CC(C(C)C(=O)N(C)Cc1cccs1)NC(=O)CC1CCC(C)CC1 c1(OC)ncc(F)cc1S(=O)(=O)N1CCCC(c2cnc[nH]2)C1 C(=O)(C1CNC(=O)c2ccnn21)N1CC(C2(NC(c3cnc(Cl)[nH]3)=O)CC2)C1 C1(C(N2C(CCNC(c3ccnnc3)=O)CCC2)=O)CC(C2CC2)=NO1 CC(C)C(CCC(=O)N(C(C)CO)C1CC1)NC(c1ccc(F)cn1)=O C1(C(C(=O)NCc2cccs2)N(CC)Cc2cn(C)nn2)CC12CCOC2 c1(NCC2CN(C(COC)=O)C2)ncnc2scc(-c3ccccc3)c12 c1(C(=O)NCC2C(NC(=O)C=CCO)CCC2)c(O)cc(O)cc1O c1(C(N2CCCCC2Cn2cc(C3(O)CSC3)nn2)=O)ccn2ccsc12 N1(C(C(CC)SC)=O)CCN(C(=O)CSCC(=O)OC(C)(C)C)CC1CC#N N1(C(CCc2onc(C)n2)=O)CCN(C(=O)CC(C)O)CC1C1CC1 C1(NC(C2C(CC)CCCC2)=O)CN(C(=O)CP(C)(C)=O)CC12CCCC2 c1(C(CC)NC(c2sc(Br)cc2Cl)=O)cc(F)cc(Cl)c1 c1(C(=O)NCCOC2CN(C(C(C(C)(C)C)SC)=O)C2)cc(C)cc2c1OCC2 c1(C(=O)NC(C)CN(C)C(C2(C)CC=CCC2)=O)cc(N)c(F)c(F)c1Cl Cc1cn2ccc(C(=O)NC3CC4CN(C(C5CC(=O)CO5)=O)CC34)cc2n1 C1(OCCNC(C2C(C=C)C2)=O)CCN(C(C2CCOC2)=O)CC1 N1(c2ncc(C)cn2)CCN(C(=O)CCOC(C)C)CC(O)C1 c1(CC=C)ccccc1C(=O)NCC1(F)CN(C(C2C3CCC2CC3)=O)C1 C1(NC(C(C)NC(CC)=O)=O)CCC(NC(=O)C(C)(C)n2cccn2)C1 CCCCCCC(C)C(=O)NCC1CC1NC(=O)CCCn1cc(C)cn1 C1(NC(c2ccc(CC)cc2F)=O)CC2CC(C1)CN(C(C1CC1[N+](=O)[O-])=O)C2 C1(C(N(CCC(=O)N(C)Cc2cc(C)nn2C)CCO)=O)CCOCC1(C)C c1(NC(C2(NC(C3CCCC3)=O)C(C)C2)=O)cc(S(=O)(=O)N(C)C)ccc1Cl Cc1nc2cccc(C(N3C4CCC3CN(C(=O)C=C(Cl)Cl)C4)=O)c2[nH]1 CC1CCn2cc(C(=O)NCCOCCCN(C)C(c3cc(F)n[nH]3)=O)nc2C1 C(=O)(C(C)C(F)(F)F)NCCNC(C1CN(C(c2ccc(C)s2)=O)C1)=O C=C1CCC(C(=O)NCC2CCCCN2C(C2CCCC2CCC)=O)CC1 N1(C(c2cnco2)=O)CCCC(c2cn(Cc3cnns3)nn2)C1 C(CCC)(C(O)C(=O)N1CCCc2nncn21)NC(C(CC#C)(C)C)=O CC1CCc2onc(C(=O)NCCC3(O)CCN(C(C4CC(F)C4)=O)CC3)c2C1 N1(C(C2C(C(=O)OCC)C2)=O)CCCC(NC(c2conc2C)=O)CC1 C(=O)(C=CS(C)=O)NC(C1N(C(COc2cc(C)on2)=O)CCC1)C C(CC(C(=O)N1CCC(C(=O)OC)C1C)NC(C1CCC(=O)C1)=O)=CC C=C(C)CC(C(=O)N1CCC(C(=O)NC2CN(C)CC2(F)F)C1CC)OC c1(CN2C(CCC(=O)NCc3nc(C)c(Br)s3)CCC2)ccc2ncsc2c1 c1(C(=O)NCCC2CN(C(c3cnc(OC)s3)=O)C2)cc(OC)cc[n+]1[O-] c1(OC)ccc(F)cc1CC(=O)NCC(C)CNC(=O)CC1NC(=O)NC1=O CCC(CC)CC(=O)NC(C1CCS(=O)(=O)C1)C(=O)O C(=O)(C1=CCCOC1)NCCOCCN(C(CC1C(C)OC(C)C1)=O)C Nc1cc(C(N2CCOC(CNC(c3cc(O)nc(O)n3)=O)C2)=O)cc(Cl)n1 c1(C(=O)NC2CCC(CCNC(C3C(C)C3C)=O)C2)cncc2ncn(C)c12 N1(C(c2cc(CC)n(C)n2)=O)CCC(C2CCN(C(c3ncccc3C)=O)C2)C1 c1(C(=O)NC2CCCCCN(C(C3C=CCC3)=O)C2)ccc2ccc(O)nc2n1 N1(C(CN(C)CC)=O)Cc2nccn2CC(NC(=O)CNS(C)(=O)=O)C1 N1(C(CC(=C)C)=O)CC(NC(=O)C=CCN(C)C)Cc2ccccc21 c1(OC)cc(Br)cc(C)c1NC(C1CC(NCc2cccc(C)c2F)C1)=O c1(CCC)noc2nc(C)cc(C(N3CCC(O)(CN(C)CC)C3)=O)c12 Cc1[nH]nc2ccc(C(=O)NCCC3C(C)CCCN3C(=O)COC3CC3)cc12 c1(C(C)C)nc(=NC(CNC(=O)C(C)c2ccsc2)c2ccccc2)s[nH]1 c1(C(=O)NCC2(F)CN(C(c3ccc(F)cc3F)=O)C2)cc2n(n1)CC(F)C2 c1(CCC(=O)NC2CN(C(=O)CN3CCC3)C3CC23)c(F)cccc1F C1(CNC(Cc2c(C)nc[nH]2)=O)(NC(C2C(C)C2(F)F)=O)CCCCC1 c1(CC(=O)NC2CC(NC(C=CSC)=O)C2)cccc(F)c1Cl c1(C(=O)NCCCCN(C)C(C2CC(=C3CC3)C2)=O)cc2c(o1)CCCC2 c1(OC)cnc(Br)c(NC(C2CCN(Cc3cc(Br)cnc3F)CC2O)=O)c1 c1(C(N2CC(C)C(NC(=O)Cc3ccsn3)C2)=O)cc2cnn(C)c2s1 CC1=NOC(C(=O)NC2CCN(C(=O)CCc3csc(=N)[nH]3)C2)C1C c1(C(C)=O)ccccc1C(=O)NCCC1(NC(c2csc(Cl)n2)=O)CC1 Cn1ncc2c(N3CCCC(CCCO)C3)nc(=NC3CSCCSC3)[nH]c12 c1(C(N(C)CC2CCCN2C(C2COC(=O)N2)=O)=O)cc2cc(Cl)sc2[nH]1 c1(C(CCC)=O)cnnc(C(N(CC(O)C(=O)OC)CC)=O)c1 N1(C(C(C)OC)=O)CCC(N2CCN(C(c3cc(Cl)c(Cl)s3)=O)CC2)CC1 c1(C(N2CCCC2C(c2ccccc2)O)=O)cnc2ccccn12 Cc1cccc2cc(C(=O)NC(CNC(=O)CN3CCC(C)C3)C3CC3)cnc12 CC1COCCC1(c1nnnn1CC1CC1)NCc1ccc(-c2cc[nH]n2)cc1F c1(C(N)=O)ccc(C(=O)NC2CCOCC2NC(=O)Cn2nnc(=O)[nH]2)cn1 c1(C(N2C(C)CCC2C)=O)cn2c(n1)CCN(Cc1ccc3cncn3c1)CC2 n1(CC)cccc1C(N1CCCC1CN(C(c1cncnc1)=O)C1CC1)=O CC1(CNC(C2CCCN2C2CCCC2)=O)CCN(c2nnc(C(F)F)o2)C1 O=C(C1=CCCCO1)NCC1C2CC1N(C(=O)Cc1ccc(I)c(O)c1)C2 N1(C(C=CCCC)=O)CCCC2(CCCN2C(=O)C(N2CCCC(O)C2)C)C1 C1(N)(CNC(=O)Cc2ccc(O)cn2)CC2CCCC12 CC1CCCC(c2nnnn2CCCF)(NCc2ccc(Cl)cc2)CC1 N1(C(CN2CCC(C)C2)=O)CC(C2CC2C(=O)NC2CN(C(N)=O)C2)C1 c1(-n2c(-c3cnc(CC)s3)nc(-c3cscn3)n2)cc(C)ccc1C C1(S(C)(=O)=O)(C(N2CCC(OCCSC)C2)=O)CC1.C12(CCOC1)C(=O)N2 C(CCCCCCCO)=CC(=O)NC1(CCCNC(CC2CCN(C)CC2)=O)CC1 c1(C(=O)NC)cc2c(Br)cc(C)cc2[nH]1.c1(CCC(C)=O)cc(C)n(-c2ccco2)c1C C(C)(C)(CCCNC(C1CC12CC2(F)F)=O)NC(CCCOCCC)=O c1(C(C(N2CCC(N(C(=O)CCF)CC)C2)=O)(C)C)ccc(C#N)cc1 C1(CNC(C(CCC2CCCC2)NC(C23CCCC2C3)=O)=O)CC2CCCC2C1 C1(C(N(CCNC(=O)CN(C)C2CC2)CC)=O)OC(C)(C)OC1(C)C C(=O)(C(CC=C)OC)NC1(C(N2CC(C)(OCC)C2)=O)CCCC1 c1(C(=O)NC(C)CN(C(=O)CCCC(=O)N(C)C)C)cc2ccc(Cl)nc2s1 C(CC(C(=O)NC)NC(=O)COCC(=O)NCCNC(c1scnc1C)=O)OC N1(C(C(C)NC(c2ccccc2)=O)=O)CC=CC(NC(C2CCCN2N=O)=O)C1 c1(NCc2c(C)cco2)ncnc2c1c(I)cn2C C1(NC(c2n(C)cnc2)=O)CN(C(c2ccc(Cl)c(F)c2F)=O)CCC1(F)F c1(N(CCC)C)nc(=NCCSC(F)(F)F)[nH]c2cc(C(N)=O)ccc12 N1(C(CC2(C)CCC2)=O)CCC(F)CC1C(N1CCC(CCN(C)C)C1)=O N1(S(CCC[Si](C)(C)C)(=O)=O)CCc2cccc(OC(F)(F)F)c2C1 c1(CC)nc(Cl)nc(N(CCCNC(C2COC(C)C2)=O)C(C)C)c1Cl c1(C(=O)NC(c2ccnn2C)C(=O)NCC(CC)(C)OC)c[nH]c2ncccc12 c1(C(=O)NC(C(C)C)C(C)NC(=O)Cn2cccn2)ncc(Br)cc1O N1(CC2(C(F)F)CCOC2)CC2C3COCC3C2C1 c1(NC(=O)NCCCN(C(C)=O)CCO)cccc(C(C)(C)O)c1 Cc1ccc(C)c(OC(C)C(N2CC3(CC(CN)C3)C2)=O)c1 N1(CC)CCC(CNC(=O)C(C)(C)CNC(C2C=CCC2)=O)CC1 CC1CCC(C)(C(=O)NCc2ccc(CN(C)C(c3coc(C#N)c3)=O)cc2)C1 C1(C(N2CC(C)C(CNC(c3sccc3C#N)=O)C2)=O)CCOC(=O)CC1 N1(C(CCOCC#C)=O)CCc2sc(C(=O)Nc3ccc(C)nc3)cc2C1 C1(NC(=O)Cc2cccc(Br)c2)CCCCC12CCN(C(c1cc[nH]c1)=O)C2 Cc1nccn1CCC(=O)NC(CNC(=O)CCCF)C1CC1 C12(CNC(CCCOC)=O)CC3CC(CC(NC(=O)CCC=C(C)C)(C3)C1)C2 C(CCSC)(C(=O)NCCCCC1CN(C(=O)CCC2CCCC(=O)N2)C1)OC CC1CCC(C)N1CC(=O)NCc1ccc(CNC(=O)C2=NOCC2)cc1 c1(CCC(=O)NCCC2(OC)CN(C(=O)C(C)O)C2)cccc(C(F)F)c1 N1(CC)CCOC(C(=O)NC(CC2CC2)CC(=O)NCC(c2ccccn2)C)C1 C(=O)(CCC(=O)NN(C)C)N1C2CC(NC(COCC=C)=O)C1CC2 N1(C(C(CC=C)(C)C)=O)CC(C)OC2(CCN(C(c3cc(CO)[nH]n3)=O)C2)C1 c1(C(=O)NCC2OCCN(C(C(C(C)(C)F)(C)F)=O)C2)c(Cl)oc2ccccc12 C(C(O)CC(=O)NCCCN1CCN(Cc2cc(C(F)F)no2)CC1)N(C)C c1(COC)ccccc1CC(N1CCCCC1C1CCN(C(=O)COC(C)=O)C1)=O C#CCCN=C(NCC1(S(=O)(=O)NC)CC1)N1CCC2(C1)Oc1ccccc1O2 CC(C)C(C)C(CNC(c1csc(S)n1)=O)NC(c1csc(S)n1)=O CC(C)CCCCC(=O)NCC(C1CC1)NC(C1(C(N)=O)CC1)=O c1(OC)ccc(I)c(CN2CCCC(C(=O)NC(C)(C)C(=O)N(C)C)CC2)c1O C(c1ccc2occc2c1)=CC(N1C(CNC(C2C(=C)CC2)=O)CCC1)=O c1(OC)cc(C=CC(=O)NCC(C)NC(=O)CN2CC(C)(C)C2)cc(Cl)c1OC c1(CCC(=O)N(C(C)C)CC2CNC(=O)C2)c(F)cc(Br)cc1F N1(CCNC(n2cc(C3(n4ccnn4)CC3)nn2)=O)C(=O)CNC1=O Cc1onc(C(=O)NCCCN(C(=O)CCN2CCCC2=O)C)c1Br C1(CNC(c2ccc(F)cn2)=O)CC(NC(c2ncc(Cl)cc2O)=O)C12CCC2 C1(NC(C2C(CCC)C2)=O)CC(C)N(C(=O)Cn2cc(C)cn2)C1 N1(CC(c2c(C)nn(C)c2)=O)CC(Sc2nccs2)CCC1=O c1(C(N(CCCN(C)C(c2c[nH]c(C#N)c2)=O)C)=O)ccccc1OCC(N)=O Nc1cc(C(=O)NC2CCCC2NC(=O)CCC=CBr)cc(F)c1 C1(C(=O)NCC)CCCCC2(C1)OCCO2.c12ccc(c(I)n1)oc2=O C=C(Cl)C(C)(C)C(=O)N1CC2C(CN(C(=O)C(C(C)OC)NC(C)=O)C)C2C1 C1(NC(C(C)C(F)F)=O)CN(C(c2cnc(C(N)=O)s2)=O)CC12CCOCC2 N1(C(c2c(C)ccnc2O)=O)CC2(COC(CNC(=O)C(O)c3ccsc3)C2)C1 C1(OC)CN(C(C2CCCN2C(C2CCCSC2C)=O)=O)CC1OC Cc1cccc2c1CC(C(=O)NC(C)(CNC(=O)CC1CC1)C1CC1)O2 C1(CNC(Cn2c(C)nnn2)=O)CN(C(=O)C=CCN2CCCC2)CC1(F)F C(CCO)(C(=O)NCC1CC2CC2N1C(c1ccon1)=O)N(C)C c1(C(N2CCC(CNC(C(C)OC)=O)(CO)CC2)=O)ccc(N)c(Cl)c1O C=CC(C)(O)CC(=O)NCCc1ocnc1CNC(c1cc(O)nc(SC)n1)=O N1(C(CCN(CC)CC)=O)CC2CN(C(C34COC(CO)(C3)C4)=O)CC2C1CO c1(C(C2CCCC2NC=O)=O)nc(=N)cc[nH]1.c1(C(C=C)(C)O)cn(C)nn1 C(=O)(CS(=O)CCC(F)(F)F)N(C)CC1N(C(C#CC(=O)N(C)C)=O)CCC1 CC(C)C#CC(=O)NC1CCC1CNC(=O)CCCNC(c1cccnc1)=O C1(C(=O)NCCCOC2CCN(C(c3cc(C)[nH]n3)=O)CC2)(CC)CCCC1O N#Cc1ccc(O)c(NC(C2CCCC(NC(=O)C=CC3CCOC3)C2)=O)c1 c1(CC)ccnc(C(N2CCC(C(C)NC(=O)CCCC3CCOCC3)C2)=O)c1 CN=c1[nH]c(=NCCCCC#N)[nH]c(=NC2CCC(OC)C2)[nH]1 Cc1nc(C(c2ccccc2)NC(=O)Cn2ccccc2=O)sc1C Cc1cccc(C(=O)NCCCC(C)NC(=O)CC2CCCCC2O)c1C c1(CC(=O)NCC2C(CNC(c3ccc(F)nc3)=O)C2)ccncc1Cl N1(C(c2ccc(CC)cn2)=O)CCC2(NC(c3cnc(Cl)[nH]3)=O)CCCCCC12 C1(C(=O)NCCCC)CC(F)CCN1C(=O)CC1CC2(CC2)C1 c1(C(N(CCN(C(C23CC(OC)C2C3)=O)C)C)=O)cnc2nccnc2c1 N1(C(C23N(C(CCN(C)CC)=O)CCC2CCC3)=O)CCOC2(CCCC2)C1 c1(OC)ccc(NC(=O)CC2CN(Cc3c(C)cccc3C)C2)c(OC)c1 C12(C(N3CC(N4CCC(c5c(N)nccn5)C4)C(F)C3)=O)C3CC(CC13)C2(F)F C1(CNC(Cc2n(C(C)C)cnn2)=O)(CO)CCN(C(=O)C(F)C(C)(F)F)CC1 CN1CCC(C(=O)NCC2CN(C(=O)Cc3csc(-c4ncccn4)n3)C2)C1 c1(C(=O)NCC(CNC(C2CC(C(F)(F)F)(OC)C2)=O)C)cccc(F)c1SC N1(C(c2c(C)ccs2)=O)CCN(C(c2cc3cnccc3[nH]2)=O)CC12CCC2 c1(C(=O)NC(CC(C)NC(c2cnc3nccn3c2)=O)C)nnn2c1CSCC2 C1(NC(c2nccc(C)c2)=O)CN(C(=O)C(C(C)C)N(C)C)CCC1CO C1(NC(C2CCC(OCC)CC2)=O)CN(C(=O)C(COC)OC)CCC1(C)C C1(O)(CCC)CN(C(c2cc(CNC(C3CC3(F)Cl)=O)[nH]n2)=O)C1 C1(NC(c2ccnnc2O)=O)CC2(C1)CN(Cc1ccsc1)C2 c1(C(=O)NCC(C2CCCCC2)NC(CCCC)=O)sc(SC)cc1N c1(C(C(N2CC(Cc3cn(CCCN(C)C)nn3)C2)=O)O)ccc(Br)nc1 CC1ON=C(C(=O)N2CC(O)(CN(C(=O)CC3CC(F)C3)C)C2)C1C C1(CNC(c2c(CCC)occ2)=O)CCCC(NC(c2ccoc2)=O)C1 N1(C(C2C(CC)OCC2)=O)C2CC=C(C(=O)N3CC4(CCC(C)OC4)C3)C1CC2 c1(C(=O)NC(c2ccncc2)CC)cc(F)ncc1NC(=O)Cc1cncnc1 C=CC1(NC(=O)C(C)(C)C2CCN(C(C3CCCC(C#N)C3)=O)C2)CCCCC1 C1(CC=C)(C(=O)O)CCCCN1C(c1cc(C)ns1)=O c1(C(=O)NC2CC(F)(CNC(CC(=C=C)C)=O)C2)cnn2c1NCC(C)C2 C1(C(=O)NCC2N(C(c3cnc(CC)s3)=O)CCOC2)CCc2c[nH]nc2C1 N1(C(C(C)=C2CCC2)=O)CC(NC(c2csc(-c3cnn(C)c3)n2)=O)CC(C)C1 N1(C(CCC(C)(C)C)=O)CCCCC12CCCN(C(=O)Cn1cc(Cl)cn1)C2 C1(C(=O)NCC(CN(C(=O)Cc2ccon2)C)O)CCn2c(O)nnc2C1 Cc1cc(O)c(C(=O)N(CCCNC(c2cccc(C)n2)=O)C)nn1 C(=O)(C(CO)C(C)(C)C)N(CCC(C)NC(c1c(C)c(C(F)(F)F)ccc1)=O)C C(=O)(CCC(CC)OC)N1CC(CCC)C(NC(c2cc(C)nc(O)n2)=O)C1 CC1CCN(C(=O)Cc2cnccn2)CCN1C(C1CCCN1C)=O c1(CCC)nc2ccccc2n1CCC(N1CCCCC1c1nccn1C)=O C1(C(=O)NC(C2CCCN(C(c3c(C(C)C)noc3)=O)C2)C)CC(=O)CC(=O)N1 c1(C(=O)NCCC2CC(N)C2)cn(C(F)F)ccc1=O C1(C(=O)NCC2CC(OC)CN2C(c2ccncn2)=O)CC2(CCCO2)C1 C1(CNC(C(c2c(C)n[nH]c2C)C)=O)CCN(C(=O)C=CC(F)(F)F)C(C)C1 CCCC(C(=O)NC1(CC)CN(C(c2ccccc2SC)=O)C1)NC(C)=O C#CCCCC(C)C(=O)N1CC2CC1CN2CC(=O)NC(C)C N1(C(CC(C)(C)O)=O)CCCC(CO)(NC(c2ccc(O)nn2)=O)C1 c1(OC)ccc(C)c(C(N2CCC(O)(C(C)NC(=O)CC(F)F)C2)=O)c1N Cc1ccc2c(c1)CC(C(=O)NCCCN(C(=O)Cc1ccoc1C)C)S2(=O)=O c1(C(N2CC(CC)N(C(c3sc(Br)cc3Br)=O)CC2)=O)ccc(F)c(F)c1C Cn1cnnc1N(C1CCCC1)C(CC(C(C)(C)C)c1ccco1)=O N1(C(CCC(=C)C)C(=O)NCCC2CC2)CC2(CCCCC2)C1CC(=O)O N1(C(Cc2ccc(C)s2)=O)CCC2CN(C(C3CC3(Cl)Cl)=O)CC2C1 S(=O)(=O)(c1cc(Br)ccc1Br)N1C(C(=O)NCCc2ccc(O)cc2)CC(=C)C1 c1(C(=O)NC(C)CCCOCc2ccccc2)cc(N)c(F)c(O)c1F C12(NC(c3cccc(OC)c3)=O)CCC(CC1n1cc(C3CCCO3)nn1)C2 C1(CC)CN(C(=O)CCC)CC1NC(=O)CCN(C)CCO N=c1[nH]cc(C(N2CCC(F)(CNC(C3CCCSC3)=O)C2)=O)c2cc[nH]c12 C1(C(=O)NCC2CCCO2)(OC)CCN(C(c2coc(C(N)=O)c2)=O)C1 c1(OCC)cccc(C(=O)NCc2ccc(NC(C3(CO)COC3)=O)cc2)c1 CCCCC(C(=O)NCC(C)N(C)C(C1CCC(=O)N1)=O)C(C)C C1(CC)CN(C(=O)C#CC(C)C)CCC1CNC(C1CCCN1CC)=O C#Cc1cccc(NC(=O)C(C2(O)CCC2)NC(C2CC2(C)CC)=O)c1 N1(CC)CCN(CCCNC(c2ccccc2OC(=O)C(CC)OC)=O)CC1 C(=O)(CCCC(C)(F)F)N(C)CC1(NC(c2cc(CC(C)C)[nH]n2)=O)CC1 N1(CC)CCCC(CNC(=O)C(C)(C)C2CCN(C(=O)CCc3ccco3)C2)C1 N1(C(C2COC2)=O)CCN(C(=O)C=CC2CCCO2)CC(CO)C1 CC1c2ccccc2CCN1C(c1cc2c(s1)CCC2)C(=O)NCCC1CC1 C1(S(C)(=O)=O)(C(=O)NCC(C)CNC(=O)C(C)(C)C2CCCO2)CCCC1 c1(C(N2CCC(OC)(CNC(c3cc(CF)on3)=O)C2)=O)cccc2nc(O)oc12 C(c1cccnc1)=CCNC(=O)C(F)n1ccnc1 C1(C(=O)NC2CN(C(C)C)C(=O)C2)CCN(C(=O)C2CCCC(CF)C2)O1 N1(C(CCC2CCCN(C(CCc3cc(C)no3)=O)C2)=O)CCC(F)C(F)C1 CC1(C)CN(C(c2cc(O)cc(O)n2)=O)CC1NC(=O)CC1CCCO1 CC1CCCC1(C)C(=O)NCCN(C(c1cncnc1C1CC1)=O)C1CC1 N1(C(CCC#C)=O)CCN(C(C2COC(=O)O2)=O)CC1CC(F)(F)F c1(CNC2CN(C(c3nccc(OC)c3)=O)CC23CC3)cc(F)c(Cl)cc1F CC1CN(C(c2cncc(N)n2)=O)C(C)CN1C(=O)CCc1cccnc1 c1(C(N2CC3C(NC(C(C)OC)=O)(CCC3)C2)=O)cnc2cc(C)ccc2c1 CC(C)(CC(=O)NC1CCCCCC1NC(=O)CSc1cccc(F)c1)C(F)F c1(C(N2C(CNC(C(COC)C)=O)CC(OC)C2)=O)cc2n(n1)CCO2 N1(C(C2(c3ccccc3)C(C)(C)C2)=O)CCCC(NC(C2CCCCO2)=O)CC1 c1(C(=O)NC2(C(F)F)CCC2)csc(C2CCNCC2)n1 C1(CNC(c2nc(CC)sc2)=O)CCCN(C(C2CC(=O)N(CC)C2)=O)C1 c1(C(N(CC(C)NC(C2(Oc3ccccc3)CC2)=O)C)=O)ncn2ccccc12 c1(C(=O)NC2CN(C(Cc3nnc(C)o3)=O)C3C2C3)c(F)cncc1Cl Cc1nc(C(=O)NCC2(NC(=O)CN3CCC(C)C3)CCC2)c2n1CCCC2 Cc1nc2ccc(C(N3CCOC(C(=O)NC(c4ccccn4)C)C3)=O)cc2[nH]1 N1(C(CC(C)Nc2ccccc2)=O)CC(O)CC2(CCNCC2)C1 c1(C(=O)NC2CCCC(CNC(=O)C(F)n3ccnc3)C2)ccc(Cl)c(F)c1O c1(C(=O)OC)cc(CN(C(C2CCN(CC(C)CS(C)=O)CC2)=O)C)ccn1 C#Cc1cc(C(N2C3CC2CN(C(=O)COc2ccn(C)n2)C3)=O)ccc1C CCCC(C)(C)CN=c1[nH]c(C)cc(=NC2CCCN(C(C)CC)C2)[nH]1 N1(C(C(COCC)C)=O)CC2(COC(CNC(=O)COC3CCC(C)CC3)C2)C1 C12(C(=O)NCC3C(CNC(C(CC)=CC)=O)C3)CCC(CC1)C2 c1(C(=O)NC(C2CN(C(CCCCCNC(C)=O)=O)C2)C)c(F)cc(F)cc1Cl N1(C(c2c(C)ncs2)=O)CC(NC(C2(C#N)CCCCC2)=O)CC12CCCOC2 C12CCCN(C1)C2=O.c1(C(CC)NC(C2(C(=O)C3CC3)CC2)=O)ncc[nH]1 CC1(C)CCCCC1=CC(=O)NC1(CO)CCN(C(=O)C=C2CCCC2)CC1 C1(C(=O)NCC(Cl)Cl)N(C(=O)CCCc2ncco2)CC12CCCC2 CN1CCCC1CC(N1CC(C)(NC(=O)CC2CCNC2=O)C1)=O c1(COC)ccc(C(N2CCOCC2CNC(C2CC2c2nc[nH]n2)=O)=O)cc1 C=C(C)CC(C(=O)NC(C)CCN(C(=O)Cn1cccc(N)c1=O)C)OC C1(OC)CCCC(CC(N2CC3CC3(CNC(C3(N=[N+]=[N-])CC3)=O)C2)=O)C1 C1(CC(=O)NCCCCCC=C)C2CCC(C2)N1C(C1CC(C)N(C)C1)=O C1(C)(C(=O)NCC2N(C(CC=C(C)C)=O)CCC2)CC2CCC1C2 CCC(C)CCC(=O)NCCC(C)N(C(=O)CC(C)(C)O)C C1(C(=O)NC2(CNC(C34CCCC3CCC4)=O)CCC2)CCCC2(C1)CC2(F)F N1(C(C(C)NC(COC)=O)=O)CCC(NC(C2CC(C)(C)C2)=O)CC1C C1(CNC(C(C)CSC(F)(F)F)=O)(CO)CCCN(C(C2CC3CCC3C2)=O)C1 CC(CC(N)=O)C(=O)N1CCCCC1C1(NC(=O)CCCCNC(N)=O)CC1 c1(SC)ccc(C(=O)N(CCNC(=O)CCOC)CC2CC2)s1 CC(C)C(F)(CNC(C1CC12CC2)=O)C(=O)N1CCCC(C)(C#N)C1 C1(C(N2CCC(NC(c3c(C)cc(F)cn3)=O)C23CC3)=O)COC2COCC2O1 C1(C(=O)NC2(CO)CCN(C(C3N(N=O)CCCC3)=O)CC2)CC2COCC(C1)C2 S(=O)(=O)(c1cnc(NC(c2snnc2C)C)cc1C)N1CC(Br)=C(C)CC1 C=CC1(CC(N2CCC23CN(C(c2ccc(C4CC4)cn2)=O)C3)=O)CCOCC1 Cc1cc(C(N2CCOCC2CC(=O)NC2(C)CCCC2(F)F)=O)cc(O)c1 CC1CC(NC(=O)CC2CCC(=O)N2C)CN1c1ccnc(-c2nccs2)n1 N=c1ccnc(C2(NC(=O)CCc3ccccc3Cl)CCCC2)[nH]1 c1(C(N2CCC(CNC(C(C)NC(C)=O)=O)C2)=O)ccc(Br)c(Cl)n1 CCC(CCC(=O)C1C(O)C2C(OCC1)N2)NC(=O)C(C)(C)C(C)O Cc1nc2c(s1)CCCC2C(=O)N(CC(CO)(CO)NC(=O)C(O)C1CC1)C CCS(=O)(=O)CC(=O)N1CCC(O)C(C(=O)Nc2ccc(OC(C)=O)cn2)C1 N1(C(CC2ON=C(C)C2)=O)C(C(=O)Nc2cncc(C(C)C)c2)CC2CCCC12 c1(C(N(CC(CNC(c2nccc(C)c2N)=O)O)C)=O)ccc2c(c1)C=CCC2 Cc1cc(-c2nc(COC(C)(C)C)nn2C2CCOCC2)nc(N(C)C)n1 C1(C(c2n(CC)nnn2)NCC2CC2)CCN(C(=O)CC=C(C)C)CC1 N1(C(c2c(CC)scc2)=O)CCC12CN(C(=O)CSCC(=O)OC(C)(C)C)C2 C1(NC(C(C)(C)NS(C)(=O)=O)=O)CN(C(C2(C)CC=CC2)=O)CC1O N1(C(COC(CC)C)=O)CCC2(CCC(NC(=O)C3CCN(C)CC3)CC2)C1 CCC(C(=O)NCC1CN(C)CCN1C(=O)C(C)C(=O)OC)C(C)O c1(OC)nc(NC2CN(C(C3CCCN3C(C)=O)=O)CC2F)nc2ccccc12 Cc1cc(C(=O)NCC2CC(NC(C3CN(C(C)C)C3)=O)C2)cc2nn[nH]c12 c1(C(=O)NC2CC(CNC(c3cnc(S)nc3)=O)C2)cc2c(o1)CCCC2 c1(CC)ccc(O)c(C(=O)NC2CC(C)(NC(c3ccc(Cl)cn3)=O)C2)c1 C(N=c1[nH]c2c(F)cccc2o1)C1CCCC(NC(C(c2cn(C)nc2)O)=O)C1 C(=O)(CC(C)C1CC1)N(CCC(C)NC(c1ccns1)=O)C Cc1ccccc1C(C)NC(=O)CC1C2CN(C(C3CCSC3)=O)CC12 CN1CCC(CCC(N2CCCC2CCNC(=O)CS(N)(=O)=O)=O)CC1 N1(C(C(CC)C(=O)OC)=O)CC2CC(NC(=O)C=CC(C)C)CC(C2)C1 N1(CCNC(CN(C(c2nnsc2C)=O)CC)=O)CCCCCC1 c1(OC)cccc(C(=O)NCC(CNC(C2(n3nccn3)CC2)=O)OC)c1C n1(CC(=O)N(CCCC(=O)NCC2C(C)CCC2)C)cnc(C#N)n1 O=C(NNc1cccc(Cl)c1Br)NC1C2CCCCCC12 N1(C(c2cnc(CC)[nH]2)=O)CCN(C(c2ccc(C)nc2N)=O)CC1CC(F)F C1(OC)CN(C(=O)COc2cncc(F)n2)CC1NC(C1CN(C)CCO1)=O c1(CC)ncc(Cl)c(C(=O)NCCC2(NC(=O)CCc3ccc(Cl)cc3)CC2)n1 N1(C(C2C(=O)NCC2)=O)CC2(CC(C(=O)Nc3ccc4nccn4c3)CO2)C1 C1(NC(c2c(CC)oc(C)c2)=O)CCSC12CN(C(=O)C(C)(F)C(C)(C)F)C2 c1(C(N2CC(NC(C3CC(C(C)C)C3)=O)C2)=O)cnc(C(C)O)s1 n1(CCOC)nnnc1C(c1ncccn1)(C)NCCC(COC)OC C1(C(N2CC(N(C(=O)Cc3ccc(N(C)C)nc3)C)C2)=O)CCCCCS1(=O)=O C1(OC)(OC)CC(C2CCN(C(C3CCCC4(C3)CC4(F)F)=O)C2)C1 S(=O)(=O)(CC(=O)NC1CC(C(=O)OC(=O)CCCN(C)C(C)C)C1)N(CC)CC N1(C(=O)OC(C)(C)C)CCCC12CCCN(C(c1cc(=O)n3ccsc3n1)=O)C2 C1(C(=O)NC2CC(NC(c3scc(OC)c3)=O)C2)CCn2c(C)cnc2C1 c1(C(=O)NCC2C=CCC2)coc2c1CN(C(c1cnsc1)=O)C2 C#CCCCCC(=O)N1CC(O)(CCNC(=O)COC(F)(F)F)C1 C=CC(C)(C)C(=O)N(CC(C)NC(=O)Cn1nnc(-c2ccsc2)n1)C c1(C(=O)NCCC2CCC(C)C2)cnccn1.CON=CC(=O)OCC1CC1 Cn1cncc1C(=O)NC1CCCC1CNC(=O)CCNC(=O)OC(C)(C)C C1(C(C)C)CN(C(=O)CN2CCN(C)C(=O)C2)CCN1C(=O)CN1CCCC1=O C1(C(=O)NCC2C(C)CCN(C(COC(C)C)=O)C2)CCc2nncn2CC1 C1(C)(C(N(C(C)CO)C)=O)CCCN1C(=O)Cn1cnnn1 C1(n2cc(C(C(C)(C)C)O)nn2)CCC2CC2CC1.C1CN(CC(=O)O)CCO1 N1(c2nc(C)cc(OC)n2)CC(NC(=O)C(O)C2CC2)CC2(CCC2)C1 c1(CCC(=O)NC(C(C)NC(C(Br)=C(C)C)=O)C)c(F)cccc1[N+](=O)[O-] C(C(C)(C)CNC(=O)Cn1cnnn1)N(C(=O)COC)CC C1(NC(CC2OCCN(C(C(CO)OC)=O)C2)=O)CN(C)CCN(C)C1 Cc1c(CN(CCOC)CCO)cnc2ncnn12.C1(C)COCC1(F)F C(=O)(C(C)N=c1ccn(C(C)C(=O)NCc2ccc(Cl)cc2)[nH]1)OCC c1(OC)ncc(Cl)cc1NC(c1cncc(NC(=O)CC#N)c1)=O c1(C(N(CC(C)N(C)C(c2sccc2F)=O)C)=O)ccc2c(c1)CCC2 CC(CC#N)C(=O)N(CC(C)NC(c1ccc(C(=O)NCC2CC2)cc1)=O)C C1(OC)CCC(NC(C2CN(C(=O)COCC(F)(F)C(F)F)CC2OC)=O)CC1 C#Cc1ccc(CC(N2CC(c3ccccc3)CC(O)C2)=O)cc1 C1(C(N2CCC(C)(NC(C3CNC(=O)N3C)=O)C2)=O)(OC)CCCCCCC1 c1(C(=O)OCC)nc(CNC(=O)OCC)ncc1Cl.C1(C2CC2Cl)C(=O)N1 C(=O)(C1Cc2ccccc21)NCCCONC(C1NC(=O)CC(C)C1)=O N1(C(CCCCSC)=O)CCCC(C)(NC(=O)CC2CCCOC2)C1 C(c1cc(Cl)ccc1OC)=CC(=O)NC1(C)CCN(C(CCC(C)SC)=O)CC1 CN1C(=O)CCCC1C(N1C2CC1CN(C(c1cc(Cl)ns1)=O)C2)=O c1(OC)c(CNC(=O)NCCCCC2(C)NC(=O)NC2=O)ccnc1Cl Cc1c2c(-c3cnc(CC(=O)Nc4cnccc4CO)nc3)cccc2nn1C C1(CCC(=O)N(CC(COC)O)C)CCCN(C(c2ccc(Cl)o2)=O)C1 c1(OCC)cc(C(=O)NC(C)(C(=O)NCC(C)N=[N+]=[N-])C2CCC2)on1 c1(CNCC2(NC(C3C(C)(C)C3C(F)F)=O)CCC2)ccc2c(c1)CCO2 c1(-c2c(CCOC)cno2)nc(CCn2cncn2)nn1CC(F)(F)F CC(=Cn1ccnn1)C(=O)NCCCNC(c1cn(C)[nH]c1=N)=O C(=O)(C(C)CCC(C)(C)C)N1CCCC(C(C)C(N2CCN(C)CC2C2CC2)=O)C1 C1(C(=O)NCCC(CC)C)N(C(=O)CCCN(C)C2CC2)CCCC1(C)C C1(C(N2CCC(CCNC(C3(CC=C)CCOC3)=O)C2)=O)CCC(CC)CC1 C1(NC(Cc2c(C)scc2)=O)COC2(C1)CN(C(c1ccc3nc[nH]c3c1)=O)C2 c1(OC)cc(C(N2CCC(C(=O)NCc3cn(C(C)C)nn3)(CF)C2)=O)nn1C c1(C(=O)NC2C(C=C)CN(C(=O)Cc3sccc3C)C2)ccc2c(c1)NCC2 c1(OC)cc(C(=O)N(CC(C)(C)C(=O)NCCc2cn(C)nn2)C)ncn1 c1(C(=O)NCC(C(C)C)(C)NC(=O)CC(F)(F)Cl)ccc(Cl)c(C#N)c1 c1(N2CC(C)C(NS(=O)(=O)c3ccns3)C2)cc(O)nc(O)n1 C1(C(=O)NC(CC(C)NC(c2cc(C)sc2)=O)C)(C(F)F)CCOCC1 N1(C(C(CCF)NC(C=NOC)=O)=O)CCC(CO)C1(C)C CC1(C)CCC(C(=O)CSCCNC(=O)NC2CCC3(CCC3)C2)CC1 C1(CC(=O)NC(CNC(C2(C)COC2)=O)(C)C2CC2)CCC(F)(F)C1 c1(C(C(=O)NC2CCC2)N(C(C2CCC2)C)CC)c(Br)cnn1C c1(C(=O)NC2C(OCC)COCC2)cc(-c2nn[nH]n2)cc(C)c1 c1(SC)cccc(F)c1CNc1nc(-c2cccc(C(=O)N(C)C)c2)oc1C N1(C(N)=O)CCCC(C(=O)NCCCOCCNC(=O)C(O)c2ccsc2)C1 N1(C(=O)Nc2cc(SCC3CCCC3)ccn2)CCOCC1c1cccc(F)c1 c12ccccc1CC(C)N2C(=S)Nc1ccccc1C.N1(CC(=O)OC)CCCC1=O c1(CC(N2CC(NC(Cn3c(C)ccn3)=O)C(O)C2)=O)ccc2c(c1)CC(C)O2 CC(=O)CCCCC(=O)N1CCC(NC(=O)CC2CC2C(F)(F)F)CC1 Cc1nccn1CCCC(=O)N1CC(CC(C)NC(c2cn(C)cn2)=O)C1 c1(C(=O)NC2CN(C(=O)C#CC3CC3)CC23CC3)cc(F)c2c(c1)CCC2 C1(C2(CNC(=O)NCc3nnc(C4(C)CCO4)o3)CCC2)CCCCO1 c1(CC(C)C)nnc2c(C(=O)NCCC3(NC(=O)C(C)O)CC3)cccn12 N1(C(Cn2cc(Cc3cccc(C)c3)nn2)=O)CCNC(=O)C1c1cccc(Cl)c1 c1(OC)ccc(F)c(F)c1C(N1CCCC1(C)C(=O)Nc1ncc(Cl)cc1I)=O c1(CC(N2CCC(OC)C2)=O)ccccc1NC(=O)CC1CC2(CC2)CO1 N1(C(C(CCOC)NC(c2cc[nH]c(=N)n2)=O)=O)CC2CCOC2C1 C1(CNC(C2(COCC)CC2)=O)(CO)CC12CCN(C(=O)C(C)(F)F)CC2 CC(C)C(C)C(=O)N1CCC(OCCNC(c2cnc(S)n2C)=O)C1 N#CC1(C(N2CCC(CNC(c3cnn(C4CC4)c3)=O)C2)=O)CC2C=CC1C2 c1(C(=O)NCC(C)(C)NC(CCC(=O)NCC)=O)ccc2nc(S)[nH]c2c1 N1(C(CC2C(C)CCO2)=O)CC(CO)C2(C1)CN(C(=O)Cc1ccno1)C2 CN1CC(NC(CN2CC(C)(NCC(=O)Nc3nccs3)C2)=O)CC1=O Cc1cnc(C(N2CCN(C(c3cccc(C4CC4)c3)=O)CC2C)=O)c(F)c1 CC1CCCN(C(=O)Cc2csc(S)n2)C1CNC(C1(CCF)CCC1)=O c1(OC)cc(OC)cc(C(N2CCC(=CCNC(=O)CNS(N)(=O)=O)CC2)=O)c1 N1(C(C2(NC(c3cc(C(C)C)no3)=O)CSC2)=O)CCn2cncc2C1 C1(C(=O)NCC2(F)CN(C(=O)C(C)n3cccn3)C2)(OC)CC(C)C1 c1(C(=O)NC2C(NC(Cc3nn(C)c(Cl)c3)=O)CCC2)nc2n(c1Cl)CCCC2 N1(C(c2c(COC)onc2)=O)CC2(CCCN(C(C3CC(O)C3(C)C)=O)C2)C1 C1(NC(c2nnnn2C)C(C2CC2)OCC)CNCC1CO C1(NC(CCC2(NC(C(C)CC3CCC3)=O)CCC2)=O)C2CCN(CC2)C1C C1(NC(Cn2c(C)nnn2)=O)CCC2(CCCN(C(c3cn[nH]c3)=O)C2)C1 C(=O)(CCCCCC(=O)N1CC(NC(=O)C=Cc2cnc(C)nc2O)C1)OC CC(C#N)C(=O)N(CCC(=O)NCCOc1ccccc1)CCCO C1(CNC(C2(C(C)C)CCC2)=O)CN(C(=O)CC2C=CCC2)C(C)(C)C1 C(c1ccc(F)cc1F)=CC(=O)NCC(C)NC(c1ccc(O)cc1O)=O N1(C(C(c2cn(C)nn2)NC(C(C)OCC)=O)=O)CC2(C)CCC2(C)C1 C(=O)(C1COc2ccccc21)N1CCC(NC(C=COCC)=O)C2(C1)CCC2 C#Cc1cnc(C(=O)N(CCCN(C)C(c2ccc(N)cc2Cl)=O)C)c(C)c1 C1(CNC(COCCC=C)=O)CCC2(CCC2)C1NC(C1C2(CC2)C12CC2)=O c1(OCC)ccc(Cl)nc1C(=O)OC.C12CN(CCN1C)C(=O)C(C)n1cc2nn1 N1(C(c2cc(C(N)=O)no2)=O)CCC2CCCC12CNC(C1(F)CCCC1)=O C=CC(CC)C(=O)NC1(CC(=O)OC)CC1.C12CCCN1C(=O)C1CC21 C1(C(=O)NCc2scc(C)n2)C2CC3C(C2NC(=O)CN2CC(C)(C)C2)C13 C1(C)(CNC(C2(NC(=O)NC)CCCC2)=O)CCCN(Cc2ncc[nH]c2=O)C1 Cc1onc(SCC(N2CCCC2C(=O)NC(CO)C(N)=O)=O)c1C c1(C(N2CC(CNC(c3ccc(O)c(F)c3)=O)OCC2)=O)ccc(Cl)nc1Cl CC1(C)CN(C(=O)C2=CCCS2)CC1NC(=O)CC1CC2(CCC2)CO1 C1(C(F)(F)F)(NC(=O)NC2C(SC)CCC2)CC(F)(F)C1 c1(CN2C(C(=O)Nc3c(C)c(I)ccc3)CC(F)C2)c(O)cc(Cl)cc1Cl S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C#N)NC(c1nnc2ncccn12)C CC12CCN(C1)C2.N1(CC(=O)Sc2ccccc2)CCNCC1=O CC(C)(C(=O)NC1CC(OCC(=O)NOCC2CCOC2)C1)C(F)(F)F C1(C(F)F)(CNC(c2n(CC)ccn2)=O)CCN(C(C2COCC2COC)=O)C1 Cc1cc(C(=O)NC(C)C(C)C(=O)N(C)C(C)C2CC2)cn1C C(=O)(C(CC(C)CC)NC(c1c[nH]c(=NC)o1)=O)Nc1cc(CC)cc(O)c1 C1(C(N2C(CC)CN(C(C3CC4(CCC4)C3)=O)CC2)=O)CCCCC12OCCO2 c1(C(C(=O)NCCC2CC2)N(C(c2cccnc2)C)C)nn(C)cc1I C1(C)(OCCN(C)CC)CCCN(C(=O)CCc2ccc(C3CC3C)o2)C1 c1(C(=O)NCC(CNC(C2CC(CCC)C2)=O)(C)C)cc(Br)cc(C)c1C C1(C2CCN(C(C3CC3F)=O)CC2)(NC(COC(CC)C)=O)CC1 N1(C(CC2(C)COC2)=O)CCOC(C(=O)Nc2cn(C3CCCCC3)nn2)C1 c1(C(N(C2(CC(=O)OC)CCC2)C)=O)sc2nc(C)c(C)c(C)c2c1C c1(C(N2CC(CNC(Cc3cc(OC)no3)=O)C(C)C2)=O)cccc(Cl)c1OC N1(c2cc(C(=O)OC)nc(C)n2)CCCC2(NC(C3CCCN3C=O)=O)CC2C1 c1(OC)cc(C(N2CCC(C(=O)Nc3cc(C)no3)C(O)C2)=O)cc(Br)c1Cl N1(C(C2(NC(C3C(C(C)C)OCC3)=O)CC(F)(F)C2)=O)CCCC(C)C1C C1(C(=O)OC)CC2(C1)CC2SCCNc1ncncc1Cl C(CC(C(=O)N1CCCC(NC(N)=O)C1)NC(c1cncc(C)n1)=O)OC C1(C(=O)NCc2cccc(C)c2)N(C(c2ncn(C)n2)=O)CCCC1(C)C c1(OC)nc(C)c(C(=O)NC2CCCC(Oc3ccc(N(C)C)cc3)C2)s1 Cn1cnc(Cl)c1C(c1nnnn1CCCF)NCc1nnc(C(F)F)s1 c1(C(CSC(C)=O)Sc2c(F)cccc2Cl)ccc2c(c1)CC(=O)N2C Cc1ccc(C(=O)NCC2CCC2NC(=O)C(=O)Cc2ccccc2F)c(C)c1 N1(C(c2cc(O)ccc2Br)=O)CCN(C(=O)C#CC2CC2)C2(CC2)C1 N1(C(C2CC(C)N(C)C2)=O)CCC2C1CCCN2C(c1ccc(C(N)=O)cc1)=O CC(C)CC(C)C(=O)NC(c1nocc1C(N1CC([N+](=O)[O-])C1)=O)C C(=O)(C1CCc2cccnc21)N1CC(O)CCC(NC(CCCCOC)=O)C1 N1(C(C2(NC(c3ccc(NC(C)=O)cc3)=O)CCC2)=O)CC(S(C)(=O)=O)C1 c1(C(=O)OC)sc(CN(C(=O)C(F)CCNC(c2ccccc2)=O)C)nc1C C1(CCC(C)C)C(=O)N1.c1(C(=O)OC)cccc(I)c1OC c1(CCNC(=O)NC2(CC)CSC2)cc(C)cnc1C c1(C(=O)NC(C)CC2CN(C(=O)Cn3cc(C(F)(F)F)cn3)C2)ccc(F)cn1 Cc1cn2c(n1)C(C)CC(C(=O)NCCCCCCN(C(=O)C(O)C(C)C)C)C2 N1(C(C2(O)CCN(Cc3c(C)scn3)C2)=O)CC2COCC2C1 C12(COC)CCC(C(=O)NC3CCC(NC(C4CC4Cl)=O)CC3)(CC1)CO2 C1(CN(C(c2c(CC)nco2)=O)CC)CCCN(C(=O)C(C)C(C)O)C1 C1(NC(C(CC)C2CCOCC2)=O)C2CN(C(c3ccc(N(C)C)cc3)=O)CC12 C1(C(=O)NC(C2CCCCO2)(C)C)CCC(n2cc(-c3cncnc3)nn2)CC1 C(C)(C(C(=O)N1CCC2(CSC2)C1)C(C)C)NC(c1c(CC)n[nH]c1)=O c1(CC(=O)NC2CN(C(c3cccnc3S)=O)C2)cnc2ccccc2c1 c1(C(N2CCC(C(C)O)C2)C(=O)NCCCF)ccc2c(ccn2C)c1 N1(C(C#CC(C)C)=O)CCC(CNC(C2C3COCC23)=O)C12CCC2 C#CCC(C(=O)N1CC(O)CC1CO)NC(=O)NCc1ccco1 C=C(CNC(C1(CCN=[N+]=[N-])CC1)=O)CCNC(=O)CSC CS(=O)(=O)CCC(=O)N1CC=CC1Cn1ccnc1 c1(OC)ccc(-c2cc(C(N3CC(C)(NC(=O)CSC)C3)=O)nn2C)cc1F Cc1cn2c(=O)c(C(=O)NC3CC(CNC(C4COC(C)C4)=O)C3)cnc2s1 C(C(=O)NCC(C)(C1CC1)NC(c1noc(C(F)(F)F)c1C)=O)(C(C)C)SC N1(C(C2CC(n3cnnc3)C2)=O)CCC2CCCC(C1)N2C(C1CCCO1)=O c1(NC(=O)NC2(C)CN(C(C(C)(C)NC(=O)NCC)=O)C2)cccc(F)c1O c1(C(=O)NCc2ccc(CN(C(=O)Cn3ccnn3)C)cc2)cncc(Cl)c1Cl C1(OC)CN(C(c2nnn(C)c2CN)=O)CC1C(=O)NC(C)C(=O)N(C)C c1(C(N2CC(CNC(c3cnoc3-c3cccs3)=O)C2)=O)ccc2c(n1)CCO2 CC(CC(=O)NC(c1ccccc1)CCO)N(C(=O)Cn1cnc(=N)[nH]1)C C(C)(C(=O)N1CC(NC(=O)CCC(N)=O)C2CC2C1)(C(C)C)NC(C)=O c1(C(=O)NC2CCC(CCNC(COC)=O)C2)cc(C(C)=O)ccc1N c1(NC2Cc3c([nH]c(=N)s3)CC2)ccc(S(=O)(=O)NCC2CC3CC3C2)cc1Cl n1(CC)nncc1C(N1CCC1CNC(c1cnn(C2CCC2)n1)=O)=O N1(C(c2c(CC)onc2C)=O)C2CCC1C(F)C(NC(=O)CC(C)C1CC1)C2 N1(C(c2c(C)cccc2)=O)CCC(C)(C)C1CNC(=O)C=Cc1c(C)coc1C c1(C(=O)NC2CN(C(c3ccc(C)n3C)=O)CC2O)cn2c(n1)CCC(C)C2 c1(C(=O)NC2CN(C(C3(OC)CCC3)=O)CC2C(F)F)sccc1S(N)(=O)=O C12(CC(=O)NCC3CN(C(C(CC)OC4CCCC4)=O)C3)COC(COC)(C1)C2 CC(CNCC(=O)NC1(O)CCOCC1)CC(=O)NC(C)(C)C C(CCC(=O)NC1CCCC1C(=O)NCC1CC12CC2)SC Cc1cc(C(C)C)ccc1C(=O)NC1COCCN(C(C2C(C)C2C)=O)C1 N1(C(Cc2ccc(C)o2)=O)CCC2CC(CNC(=O)CCF)CCC2C1 c1(OCCOC)cccc(C(=O)NCC(C)(C)CNC(C23CCC(CC2)C3)=O)c1 c1(C(=O)NC(C)CN(C(=O)C(F)C2CCOC2)C)ccnc(SC(C)(C)C)c1 c1(CC)c(OC)cccc1C(=O)NC1CN(C(c2ccc(OC)s2)=O)C1 C(=O)(CC(O)C(C)C)NC(C(=O)NCCSCCC=C)CCN(C)C Cc1cc(C(N2CC3CC2CN3C(C2(F)CC=CCC2)=O)=O)ccc1O C(=O)(C(C)n1ccnn1)NCCN(C(=O)C(C)n1cccn1)CCC Cc1cccc(C(N2CCCC2CNS(=O)(=O)Cc2ccc(Cl)cc2)=O)c1Cl c1(NC(CONC(c2ccc(CC)s2)=O)=O)ccc2n[nH]cc2c1 Cc1noc(C)c1CC(=O)N(C)CC1CCCN1C(=O)C=Cc1cnc[nH]1 CCC(CC)(CCC(=O)N(C)CCNC(C1CNC(=O)C1)=O)[N+](=O)[O-] C(C(F)(F)C(=O)N1CCCC(CCNC(C2COCC2(C)C)=O)C1)OC C=CCCCC(C(=O)NC1(COCC)CC1)NC(c1cc(C)cc(F)c1)=O CCC1=C(C(=O)N2CCCC(NC(C3(CS(N)(=O)=O)COC3)=O)C2)SCCO1 C1(CNC(c2scc(C)c2)=O)CC(NC(c2cc(C)c(C)[nH]2)=O)CCO1 N1(C(CCCCC(CC)C)=O)CCCC(C2CCN(C(c3cscc3C)=O)C2)C1 c1(CC)cc(F)ccc1C(=O)NC1(CO)CCCN(C(=O)Cc2nnc(C)s2)C1 C(C(C)(O)C(F)F)NC(CN(CCOC)C(C1CC=CC(O)C1)=O)=O C(=O)(C1=C(Cl)CCOC1)N1CC(C)CC(C(=O)NC(C2(O)CCC2)C)C1 N1(CC(O)CC2CCCO2)CCOC2C(O)CC12 c1(CC(=O)NC(C2(CNC(C=CSC)=O)CC2)C)ccc(-n2cccn2)cc1 C(C)(CCCCNC(=O)COc1ccsc1)NC(C(C)OCCCC)=O C1(C(=O)NC2C(CNC(C(C(CC)C)OC)=O)CC2)CC2(C1)CC1(CC1)C2 CCCC(CNC(=O)C(F)CCC(=O)OC)C(=O)NCCC(=O)NCC Nc1cc(F)cnc1C(=O)NC(C(=O)NCCc1cocn1)C1CC1 C(C(=O)Nc1ccc(F)c(NC(=O)CCc2cn[nH]c2)c1)(C(C)(C)C)SC N1(C(c2cnc(CS(C)(=O)=O)s2)=O)CC2(C1)CN(C(C1(C(F)F)CC1)=O)C2 N1(C(=O)NCCn2cnc(C)c2C)CCCC2(NC(=O)OC(C)(C)C)CC2C1 N1(C(=O)CC2CCC3CC23)CCC(C2CC2)C1CNC(=O)C(F)(F)C1CC1 C1(=CC(=O)NC2C=CCN(C(C3CC(N(C)C)C3)=O)C2)CN2CCC1CC2 N1(C(C2(OC(C)=O)CC2)=O)CCC(C)(C)C(CNC(=O)CC2(C#N)CC2)C1 CC(C)CC(F)C(=O)N1CCC(CN(C)C(c2cnn(CCO)c2N)=O)C1 C1(CC=C)(NC(=O)CSc2cccs2)CCCN(C(c2ccnc(C)c2C)=O)C1 N1(C(c2nscc2Br)C(=O)Nc2ccc(C(=O)OCC)cc2)CC(C)(C)OCC1C C1(C(N2CC(O)(CNC(C3(C(F)F)CCC3)=O)C2)=O)CCC(F)CC1 CC(C)CC(CNC(C1(C)COCCO1)=O)NC(c1cc(Cl)n(C)n1)=O N1(C(C(CC)OC)=O)CCOC(CCCNC(=O)CCc2ccoc2)C1 N1(C(c2cnc(C)o2)=O)CCN2CCN(C(C3CC(C)CO3)=O)CC2C1 c1(C(N2CCN(CC(=O)NCCC(C)(C)O)C(=O)C2)=O)ccc2[nH]ccc2n1 C1(CC(N2CC(NC(=O)Cc3ncc(Cl)s3)C2)=O)CCCCCC1(F)F Cc1cnncc1C(N1CCC(C2CCCN2C(=O)CCc2ccco2)C1)=O C1(C)(C(=O)NCC2(O)CN(C(C(CC=CCC)C)=O)C2)CCCC1(F)F CC(O)C(C(=O)N1CCOC(CN2CCC2)C1)NC(=O)C(O)Cn1cncn1 S(=O)(=O)(c1cnc(NCCc2nnc3n2CCC3)c(Cl)c1)N(CC(O)CF)C CCC(CC)CCCC(=O)N1CC(CC(=O)NC2CC(C(F)(F)F)C2)CC1C C(=O)(C1=NOC(C)(C)C1)N(C1CCN(C(C2CN(CC)C(=O)N2)=O)CC1)CCO Cc1nc(NCc2conc2C(F)(F)F)cc(=NCC2CC2C)[nH]1 c1(C(N2CCC(CNC(c3ccoc3)=O)CC2)=O)cc(Br)cnc1Br c1(SC)nc(N2CC(F)(F)CC2C(N2CCN(C)C(C)C2)=O)cc(C)n1 C1(O)(CCNC(=O)C2CC2)CCN(C(C2C(c3ccccc3)C2(F)F)=O)C1 C1(CNC(C2(C)CC(C)C2)=O)CCN(C(=O)CCCn2cccc2)C(C)C1 c1(OC)ccc(CO)cc1C(=O)NC(c1ccc(Cl)c(OC)c1)C c1(NC)nc(C)ccc1C(N1CCC(NC(=O)C(C)n2ccnc2)C1)=O CCC(C)CCC(=O)NCCC1CC(NC(c2ncccc2C2CC2)=O)C1 c1(OC)cc(C(=O)N(C)CC2CCN(C(C3CCCC(F)C3)=O)CC2)ccc1F c1(C(=O)NCCC2CC(NC(c3ncn(C)c3)=O)C2)cc2n(c1)CCC2 C(=O)(C1=NNC(=O)CC1)N1CC(NC(=O)CCCN2CCOC2=O)C(O)C1 N1(C(CC2CCCC(C)(C)C2)=O)Cc2nccn2CC(NC(C2CSC2)=O)C1 C1(NC(=O)Cc2nncs2)CC2CC(NC(c3ocnc3C3CC3)=O)C1C2 CC1CC(C)N(C(c2cccc3nsnc23)=O)CCN1C(c1ccccc1Cl)=O c1(C(c2nnnn2CCOCC2CC2)NCC)ncc(C)c(OCC=C=C)c1C N1(C(c2ncn(C)c2)=O)CCN(C(c2scnc2Cl)=O)CC1 C(C(C)(C(=O)NCCCC1CN(C(C)=O)CCO1)OC)OC Cc1cccc(C(=O)NCCNC(C2C3CN(Cc4ccccc4)C2CC3)=O)c1F N1(c2nnc(CCC)o2)CCC2(CC1)N=N2 C(c1cn(C)cn1)=CC(=O)NCC1(CC(=O)N(C(C)C(C)C)CC)CC1 S(=O)(=O)(c1ccccc1Cl)N1CC2C(CNC(c3cc(Br)ccc3F)=O)(C2)C1 c1(C(=O)NC2(CC=C)CCN(C(c3nc(Cl)sc3C)=O)C2)ccn2ncccc12 C(CCCCn1cc(C2(C(=O)O)CC2)nn1)C(N1CCC(c2cccnc2)C1)=O C(=O)(C1=CCC(C)(C)CC1)NC(c1cn(C)nn1)C(N1CCOC2CC12)=O c1(SC)ncc(C(=O)NC2(CO)CN(C(=O)C(C)Cc3ccccc3)C2)s1 C1(NC(C(CC)OCC)=O)CN(C(=O)CN2CC3CC3C2)CC12CC2 N1(C(C2CCC(C)(CC)O2)=O)CC2CCC2(NC(c2ccc(N(C)C)cn2)=O)C1 N1(C(c2c(SC)ccs2)=O)CCCC(C)C1CCNC(=O)C1=NOCC1 c1(C(=O)NC2(C)CC(NC(=O)COCC3CCCO3)C2)ccccc1OOC(F)F c1(C(=O)NC(C)CNC(c2cccc3c2COC3)=O)ccc2nc(O)cn2c1 N1(C(C2CCC3N(C(Cc4c(C)occ4)=O)C2CC3)=O)CCOc2ccccc21 c1(C(=O)NCC(CC)NC(C2CS(=O)(=O)C2)=O)c(C)ccc2nsnc12 c1(C(=O)NCC(N(OC)C)=O)coc2c1CN(C(c1cc(O)ccc1C)=O)C2 C1(OC)CC2CN(C(C3(C(C)C)CCCN3C(=O)C(F)C3CCCC3)=O)CC12 c1(C(C)C)ccc2cc(C(=O)NC3CC(NC(=O)C=C4CC4)C3)[nH]c2c1 c1(C(N(CC(O)CNC(=O)Cc2ccn(C)n2)C)=O)nccc2cc[nH]c12 n1(CC(=O)N(C2CCCN(C(=O)C(=O)OC)C2)C2CC2)ncc(C)cc1=O c1(SC)c(C(N2CCC(NC(=O)C(C)SC)C2C)=O)ccc2c1OC(F)(F)O2 c1(C(=O)NCC2(O)CC(CNC(=O)CCCC3CC3)C2)cc2ncccc2[nH]1 C1(NC(C2CCC(C)N2C(C2CC(=O)C2)=O)=O)CCC(=O)N(C)C1=O N1(C(c2cccc(NC(C)=O)n2)=O)CCOCC(NC(=O)C2=NOCC2)C1 C(=O)(C(C1=NOC2CC12)N(CC(C)C(C)(C)C)C)NCCCCCC c1(NCc2c(Br)cn(CC)n2)ccc(S(=O)(=O)N(C2(CO)CC2)C)cc1Br c1(C(c2nnnn2CCCF)NC2(C=C)CCC2)cccc(OC)c1Cl N1(C(c2cc(CC)nn2C)=O)C2CCC1CC(NC(c1ccnn1C(F)F)=O)C2 C#CCC(C(=O)NCC1CCCCS1)NC(=O)C(=O)NCC c1(CC(N2CC3C(NC(C(N4C(=O)CCC4=O)C)=O)(C3)C2)=O)cc(F)ccc1F c1(OCC)ccc2[nH]cc(C(=O)Nc3ccc(C4NC(=O)NC4=O)cc3)c2c1 C1(C(N(C2(C(=O)NC3(C(=O)NC)CC3)CC2)C)=O)CCN(C)C1C N1(C(c2n[nH]c(C)c2Cl)=O)CCC2(NC(=O)C=CC(=O)NC3CC3)CCCC12 C(CCC(=O)NCCC1CC(NC(=O)Cc2nncn2C(C)C)C1)NC(C)=O Cc1ccc(Br)c(CCC(=O)NC2CC(NC(=O)CCC(C)(F)F)C2)c1 N1(C(CCn2ncn(C)c2=O)=O)CCC2CCC12CNC(=O)C#CC(C)(C)C C1(NC(c2cnc(S)n2-c2ccccc2)=O)CN(C(=O)C2CC2)C2(CCC2)C1 C(=O)(C1SCCc2ccccc21)NC1CC(NC(C(C2CC2)OC)=O)C1 c1(CCC(=O)N(C2CCN(C(C(CC=C)C)=O)C2)C)ccc(Cl)c(OC)c1 Cc1cc(NC(=O)NCC2(Cc3ccccc3)CCOC2)cn2ccnc12 c1(NC)nc(C)ccc1C(N1CCCCC1CNC(=O)Cc1nncs1)=O Cc1cc(C(=O)NCC2(NC(c3ccns3)=O)CCOCC2)[nH]c1C c1(CC(C)C(=O)NC2CC2CNC(C2CCO2)=O)ccc([N+](=O)[O-])cc1 c1(C(N2CCC(CN(C(CCNC(C)=O)=O)C)C2)=O)ccc2c(c1)CCCO2 c1(C(C)C(=O)NCC(=O)NC2(CNC(C3CC3C)=O)CCC2)cnn(C)c1 N1(CCNC(COC)=O)CCC(CC#N)CC1.c12cn(cn1)SC2 c1(C(N2CC(C)N(C(c3sccc3F)=O)CCC2)=O)cnc2ncc(Cl)cn12 N1(C(C2(CO)CC(C)(C)C2)=O)CC(NC(=O)C2=COCCO2)CC(F)C1 C1(C2CCC2)(C(N2CC(CCNC(C(C)CF)=O)OCC2)=O)CCC1 c1(N2C(CNC(CCNC(CNC(C)=O)=O)=O)CC(O)C2)cc(Cl)c(O)nn1 N1(C(C=C(C)C(C)C)=O)CC2CC3CC2C1C3NC(c1sccc1Cl)=O C1(O)(C(C)(C)C)CCN(C(=O)C(=O)NCCNC2CCC2)CC1 C1(C(=O)NC2CC2(Cl)Cl)(CC)CCCN1C(=O)COCc1ccccc1Cl CC1CCN(C(c2cc(=O)cc[nH]2)=O)C(CNC(=O)C(C)n2ccnn2)C1 CC1CC(CCC(=O)C(=O)N)CC(C)(C)C1.c1(N)ccc(C(F)F)nc1 C1(NC(c2c(COC)nn[nH]2)=O)CC(C2CCN(C(C3SCCCS3)=O)C2)C1 CCCCCC(C)(CC)C(=O)NCCN(C(=O)CC(O)CCSC)C(C)C CC(C)(CC(=O)N1CCC(C(F)F)CC1)C1CCCCC1 O=C(C1COc2ccccc21)NCC(c1ccccc1)NC(=O)Cn1ccnn1 C(C1CCOCC1)=CC(=O)NC(C1CCOC1)CNC(CC=C(C)C)=O C1(NC(C(F)=CCC)=O)CCN(C2CCN(C(=O)CCC(C)SC)CC2)CC1 C1(NC(C2CS(=O)(=O)C2)=O)CC1C1CCN(C(c2ccn3ccnc3n2)=O)CC1 N1(C(CC2CCC(=O)O2)=O)CCC2(CCN(C(c3occ4c3CCC4)=O)C2)C1 c1(C2(NC(C(C3(C(F)(F)F)CCC3)N(CC=C)C)=O)CC2)ccc(F)cc1 c1(C(N2CCC(C(C)(C)CNC(C3CC=CCO3)=O)CC2)=O)cccc([N+](=O)[O-])c1 C1(C(=O)NCCC(C)N(C(C(C)(C)OC)=O)C)CC12CCc1ccccc12 c1(N2CC(C)=C(C)CC2)ccncc1S(=O)(=O)NC(c1cc(F)c(F)c(F)c1)C C(C(C)(CO)NC(c1cn(CC)cn1)=O)NC(C1(CC#C)CCC1)=O N1(C(c2cc(COC)on2)=O)CC(NC(C2CCOC2)=O)C2CCCC12 N1(C(c2ccnc(OC)c2)C(=O)NCCOCC)CC2CCCC(O)C2C1 C1(NC(=O)C=Cc2cncnc2O)CC(O)CN(C(=O)CN2CCCCC2)C1 c1(C(=O)NC2CCN(C(c3cn(C)c(=O)n3C)=O)CC2)cc(O)c2sccc2c1 C1(NC(C(CCSC)OC)=O)CN(C(c2ccc3cc[nH]c3n2)=O)C2(CCC2)C1 C1(CN(C(CCNC(=O)NC)=O)C)CCCC1NC(=O)CC(Cl)Cl CC1CCn2cc(C(N3CCOC(CNC(=O)CN4CCOCC4)C3)=O)nc2C1 Cn1cc(Cl)c(C(=O)NCC2CCC(CNC(C3CC(=O)N3)=O)CC2)n1 C1(C(=O)NCC(C(C)C)NC(=O)CNS(N)(=O)=O)CC(C)(C)CCO1 N1(C(CCC=CC)=O)CCC(C)(C)C(C(=O)NC(C)CC(C)(C)OC)C1 N1(C(C(C)OC)=O)CCC2(CC2CNC(=O)Nc2ccc(Cl)cc2Cl)C1 c1(-n2ccc(C)n2)ccccc1C(N1CC2C(C(=O)NC34CC(C)(C3)C4)C2C1)=O N1(CC)CC(C(=O)NCC(C)C(=O)N(C)Cc2ccoc2)CC1=O CC1C(NC(c2ccc(O)nn2)=O)CCN1C(=O)Cc1cnccn1 N1(C(Cn2cnc(=N)[nH]2)=O)CC(=O)CC1C(=O)NC(CO)C1CC1 CC(C)CC(F)C(=O)N(C)CC1COCCN1C(c1ccc(F)cc1Cl)=O N1(C(c2cnc(C)[nH]2)=O)CC2CC1CN2Cc1c(O)cccc1O c1(C(=O)NC2CCC(Nc3nc(C)nc(Cl)c3)CC2)ccc2cncn2c1 C(=O)(C(CN=C(NCc1cnnn1C)NC(C)C1CC1)C(C)(C)C)OC C1(OCC2CC(=C)C2)C(CC)CCN1CC C1(NC(=O)Nc2cc(F)c(F)c(F)c2F)CC[Si]2(CCCC2)CC1 c1(C(=O)NCCC(C)N(C)C(c2cncc(F)c2)=O)cc(S(C)(=O)=O)co1 N1(C(c2c(Cl)cn(CCC)n2)=O)CCC(C)C(NC(c2ncncc2C)=O)C1 c1(-c2n(CC)ncc2)c(CCN(CC)CC2CCS(=O)(=O)C2)sc2ccccc12 C(=O)(CCC(=O)NCCC)NCC1C(C(=O)NCC(=C)Cl)CCC1 C1(C(N2CCC(C(CO)NC(C3CC34CCOC4)=O)CC2)=O)CN2CCN1CC2 CC(C)(C)C1CCNc2c(C(=O)NCC3CC(NC(=O)CCF)C3)cnn21 C1(NC(c2c(C)c[nH]n2)=O)CCN(C(=O)C(Cc2ccsc2)NC=O)C12CC2 CCCCC#CC(C)(C)NC(c1cc(CNC(c2ccc(C)c(F)c2)=O)[nH]n1)=O c1(C(=O)NCC2CC(NC(CSC)=O)C2)cccc(C)c1N(C)C C1(C(=O)NC(CNC(Cc2nc(C)oc2)=O)(C)CC(C)C)CCc2nnnn2C1 c1(C(N2CCC(N(C(C(C(C)(C)C)OC)=O)C)C2)=O)cc2n(c1)CCCC2 O=C(C(F)CC1CCC1)NC1(CO)CN(C(=O)C=CCF)C1 N1(S(=O)(=O)CCC(F)(F)C2CCC2)CCCC(C2CCCCC2)C1 C(=O)(C(F)(CC)C(=O)OC)N1CCC2(C(NC(Cc3cccc(CC)c3)=O)C2)C1 c1(C(=O)OC)cc(C#N)ccc1NC(C1CCN(Cc2cc(Br)co2)CC1)=O C12(CNC(=O)Cc3ccnnc3O)CCCC1N(C(=O)CCN1CCC1)CCC2 C(C(O)C(=O)N(CC(C)C(=O)N1C(CO)CC1C)C)SC C1(CNC(CCCC#N)=O)C2CCC(C2)N1C(=O)CCOCc1ccccc1 C1(COC)CC2(CCN2C(=O)CNC(c2ccc(C(C)=O)o2)=O)C1 N(C1CCCn2nncc21)C(C(=O)NC(C)COc1ccccc1F)=O C1(C(=O)NCC=CC)CCCCN(C(c2c[nH]c(C)c2)=O)C1 c1(C(=O)NCc2ccnc(OC3CCCCC3)c2)cc2ccc(O)nc2s1 C1(NC(C(C(CC)CC)C)=O)CN(C(C2CCCC3CC23)=O)C2CCCCC12 c1(C(N2CCC(CNC(CC(CC)C3CC3)=O)C2)=O)cc([N+](=O)[O-])ccc1OC c1(C(=O)NCCCCNC(c2c(CC)cno2)=O)cnc(OC)cc1OC C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)NC1C=CC(CNC(C(C=C=C)C)=O)C1 C1(N(C(C=CC(C)C)=O)C)CCC(NC(=O)CC(C)N(C)C)CC1 C(=O)(C(CCOCCO)N(C)C)NC(C1CCCN(C(=O)C(C)(C)N(C)C)C1)C CC(C)N(NC(=O)C(c1cn(C)cn1)C(=O)OC(C)(C)C)C(=O)N(C)C C(=O)(C(CC(F)F)N(C(=O)CC(C)(O)C=CC)C)N(CCCC)CCCO.C1CO1 c1(OC)ccc(C(N2CCC(O)C(F)C2)C(=O)NCCCC2CC2)cc1C(C)C c1(CC(=O)NCC2CCC(C)N(C(c3nccn3C)=O)C2)cc2ccccc2s1 N12CCC(C)(C1)CN(C)CC2=O.c1(NC(=O)CC=CC(C)(C)C)cncnc1 C1(NC(C(C(C)C)OCC(C)C)=O)CCN(C(c2csc(=N)[nH]2)=O)CC(C)(C)C1 N1(C(c2cccc(C)n2)=O)CCC(O)C(NC(c2cnn(C(C)(C)C)c2)=O)C1 Cc1nccc(Cl)c1C(=O)NCc1cn(CCNC(c2occc2Br)=O)nn1 N1(C(c2c(CC)n[nH]c2)=O)CCCC(NC(=O)C=Cc2nc(C)c(C)[nH]2)CCC1 N1(CCCC(N2CCCC(CN(C(C3C(C)C3)=O)C)C2)=O)CCc2ccccc21 c1(OC)cc2c(cc1OC)C1(CC1)CN(C(C1CCC(C#N)(OC)CC1)=O)C2 Cc1ncnc2c1CC(C(=O)NC1(CNC(=O)CNC(N)=O)CCOCC1)CC2 N1(C(c2cccc(F)c2F)=O)CC2CCN(C(c3cc[nH]c3)=O)C(C2)C1 C1(NC(C2(C)CCS(=O)(=O)CC2)=O)CC2(CCCN(C(C3CSC3)=O)C2)C1 c1(COC)ccc(C(N2CC(OCCNC(=O)CCC3CCC3)C2)=O)cc1 C1(C(N(CC(O)CF)C)=O)(NC(c2cncc(F)c2)=O)CCCCC1 CCCC(C(=O)N1CC(O)(C(F)C(=O)NCc2ccc(=O)n(C)c2)C1)C(C)C C(=O)(CCS(=O)(=O)Cc1ccccc1)NCCN(C(C1CC(C#N)C1)=O)CC C1(CNC(C2(CCOC)CCC2)=O)CC2(CCN(C(=O)CCC(C)(F)F)C2)CO1 C1(NC(c2cscn2)=O)CCN(C(C2(F)CC=CCC2)=O)CC1F N1(C(CN(C(C)C)C)=O)CCOCC1CCNC(c1cnc(CC(C)(C)C)s1)=O C1(CCN(C)C(C2CSCCS2)=O)CCCCN1C(C1(C2CCC2)CC1)=O c1(C(N2C(CNC(C3C(CCOC)C3)=O)CC(F)C2)=O)cc2ccccc2n1C Cc1cc(C)n2nc(CC(=O)NC3CC3CNC(c3[nH]ncc3C#N)=O)nc2n1 Cc1ccnnc1C(N1CC=CC1CNC(C1CC(C)(C)CO1)=O)=O c1(CC)cc(Cl)ccc1C(=O)NC1(CO)CCCN(C(=O)Cc2n[nH]c(C)n2)C1 CC(C)(C)C(O)C(=O)NC(C1CCN(C(c2cnnc(O)c2)=O)CC1)C(F)(F)F N1(C(CNC(C(CC)C)=O)=O)CC2CCN(C(=O)CC3CC(C)=NO3)CC12 c1(NC(c2cnnc(Cl)c2Cl)=O)csc2c1CCN(C(=O)CN1CCOCC1)C2 c1(C(N(CCN(C(COC(CC)C)=O)CC)CC)=O)cccc2c1CCOC2 c1(C(=O)NC2C(NC(=O)Cc3cnsc3)CCC2)ccc(Cl)cc1O c1(CNC(c2c(OC)ccc(F)c2)c2nnnn2C)csc2cccc(F)c12 C(C(C)C(=O)N(C(C)CN(C(=O)C(C)(C)c1ccnn1C)C)C)OCC CC(C)(O)C(C1CC1)NC(=O)NCC1CCN(C(N)=O)C1 C1(NC(C=CC=CC)=O)CCN(C(=O)Cc2ccccc2C)C1CC C1(C(N2CCC(C(C)C(=O)NCCC3CC=CC3)CC2)=O)CCCC12CCC2 C1(CC)CN(C(C2CC(F)(F)CS2)=O)CCN1C(=O)CNC(C1(C)CC1)=O c1(NC(C2CN(C(=O)C#CC3CC3)C3CC23)=O)ccc(-n2ccnn2)cc1 C1(C(=O)NC2(C3N(C(CCc4c(C)ncs4)=O)CCC3)CC2)CC2(C1)CC(O)C2 C12(CC(=O)NC3C(NC(c4cnc(C(C)OC)s4)=O)C3)CCC(CC1)OC2 O=C(C(O)(C(F)(F)F)c1ccccc1)NC1CC=CCC1 c1(OC)ccc2c(c1)NC(=O)C2CC(=O)Nc1c(-n2cccc2)sc2c1CCC2 c1(OC)ccc(Cl)c(C2CCCN2C(=O)NCCC(C)(C)C)c1 N1(C(C2(NC(=O)CNS(N)(=O)=O)CCN(C)C2)=O)CCC(C2CCCC2)C1 c1(OCCCN)cccc(C(=O)NC(CC(=O)O)C2CC2)c1 c1(CC(=O)OCc2c(OC)ccnc2O)ccc2oc(O)nc2c1 N1(C(C)=O)CC2CC(C1)C2CO.C1(=O)C(C(C)CC)N1Cc1ccc(-c2nn(C)cc2Cl)o1 C12(CNC(c3cccc(C4CC(F)(F)C4)c3)=O)CC1CN(C(=O)CC1CCC1)C2 c1(CCCC)nc(CN(C(=O)C(=O)NC2CCCC(C(F)(F)F)C2)C)c(Cl)[nH]1 C=CCC(CNC(=O)Cc1ccsn1)NC(C1CCCSC1)=O C(CC(F)F)(C(=O)NOC(c1ccccc1)C)NC(c1c(C)cc(F)cc1)=O C1(=O)C(NC(=O)COc2cccnc2)CCN1.CC1CCN(CC(N)=O)C1 C1(NC(C2(CCCC)CC2)=O)CC2CC(C1)N(C(c1c(Cl)n[nH]c1C1CC1)=O)C2 c1(C(=O)NC2(CNC(CN3C(C)CC3)=O)CCOCC2)cc(F)c(CO)c(F)c1 C(C(=O)NC1CCCCC1CNC(=O)CC(C)(C)CN(C)C)(C(C)(C)C)SC N1(C(CCC#CC)=O)CCC2(CC1)COC(CNC(=O)C(C)CN(C)C)C2 C12(Cc3ccc(NC(=O)CCSC(F)(F)F)cc3)CCCN(C(=O)COC)C1C2 N1(C(CC(COC)NC(C2CCCCCN2C)=O)=O)CCOCC2(CC2)C1 C1(NC(CCCc2nnc(C)n2C)=O)CN(C(C2(O)CC(F)(F)C2)=O)CC12CC2 Cc1cccc(C)c1NC(=O)C(c1cnc(Cl)s1)N(CC(N1CCCC1)=O)C1CC1 CN1CCN(C(C2CCOC2(C)C)=O)C(C(=O)N(CC(C)(C)N(C)C)C)C1 C1(C(N(C)Cc2cc(F)c(Br)cc2Cl)=O)Cc2ccccc2N(C)C1 c1(C2(C)CCO2)cccc(C(=O)N(C(c2ccco2)=O)CC2CCCO2)c1 CN1Cc2ccccc2CC1C(N1CCC1C(=O)NC1CC(CO)C(O)C1O)=O C1(NC(c2cccc3ncccc23)=O)CCC2(CCN(C(=O)CO)C2)C1 C1(NC(CCC=C)=O)CC1C1CCCN(C(C2(CF)CC3(CCC3)C2)=O)C1 C1(C(N2C3CC(NC(C4(CC)CC4)=O)C2CC3)=O)CCCCC12OCCO2 C1(CNC(C2N(CCC)CCCC2)=O)CN(C(=O)C=C(C)C)CC2(CCC2)O1 C(C(=O)N1CC(N(C)C)C(C(=O)NC2CC2)C1)(C(C)(C)C)NC(C)=O C1(CNC(COCC#C)=O)CN(C(C23CCCC2C3Br)=O)CCC1(C)C C1(CNC(=O)Cc2cn[nH]c2)CC(NC(C2(Cl)CC2(F)F)=O)CC1O O=C(C1=COCC1)NCC(CO)NC(=O)COc1ccc(Cl)cc1 N1(c2snc(SC)n2)CCOC(C)(CNC(c2ccnc(Cl)c2)=O)C1 C1(C(=O)NC2C(NC(c3cn(CC4CC(=O)C4)nn3)=O)C2)CCn2nnnc2C1 C1(C(=O)NCC(CC)(C)O)(NC(=O)CCc2cncn2C)CCCCC1 C1(C(N(C2(C(=O)OC)CC2)C)=O)CC2CC1CN(C(=O)C(C)(C)C(F)(F)F)C2 C1(NCc2cn(CCCC(=O)NC(c3[nH]cc(C)c3)C)nn2)CC2CCC1CC2 Cc1ncc(C(=O)NC2CCN(C(c3c[nH]c(=N)cc3C)=O)CC2C)c(O)n1 C(C)(CS(C)(=O)=O)NC(c1n(CCCOC)nnn1)c1csnc1C c1(C(=O)NCC(C)(C)NC(CCCN(C(C)=O)C)=O)cc(Cl)cc(C(F)(F)F)n1 C(CC(=O)N1CCC(C(=O)NCC2CCC(C)C2)O1)=C1C(C)CC1 CCCCS(=O)(=O)CC(=O)NC1CCCC2CN(C(=O)CCCC(C)C)CC12 N1(C(C(CC)(C)C)=O)CCC(C2CCN(C(c3cncn3C)=O)CC2)C1 N1(C(CC2CCCN(c3nccc(OC)n3)C2)=O)CC(=O)N(C)CC1C C1(CC)CCCCCCN1C(C1OCCC1NC(=O)CC12CCCC1C2)=O c1(C(=O)NCCCC(C)NC(=O)C(C)(C)C(N)=O)ccc([N+](=O)[O-])s1 c1(C(N2CC(C(C)NC(=O)C(F)Cc3ccccc3)C2)=O)cn(C)nc1Br c1(C(N(C)CC2(O)CCCN(C(COC(C)C)=O)C2)=O)cc2ccnn2cn1 C1(CCC=C)(CNC(=O)C(c2ccccc2)O)CCCN1C(C1COC(=O)C1)=O c1(C(N(CCNC(C2(C#N)CC(C)C2)=O)CC)=O)cccc(F)c1SC CC(CN(C)C)CC(=O)NC(C1CCN(C(C2(O)CCCCC2)=O)CC1)(C)C c1(C(N2CC=C(CNC(C(COC)OC)=O)CC2)=O)cccc2c1C(=O)CCN2 O=C(C#CC1CCOC1)NC1CCC1NC(C1(CCCCO)CC1)=O C1(C(N2CCC(CC=C)C2)=O)CN(C(c2ccsc2OC)=O)CC1F C1(C(=O)OCCCOCC(N)=O)(CC)CCNC1=O c1(OC)cccc(-c2nc(-c3c[nH]c(C#N)c3)n(C34CC(CC(F)F)(C3)C4)n2)n1 Cc1ccnc(C(C)NC(c2ccsc2C)=O)n1 C1(C(=O)NC(C(=O)NC(COC)(C)C2CC2)C)CC2CC(=O)C1O2 C1(C2CCN(C(C3(N(C)C)CC3)=O)C2)(NC(C2C(COC)CC2)=O)CC1 NS(=O)(=O)c1csc(C(=O)NCc2csc(CNC(=O)COCCF)n2)c1 c1(OC)[nH]c(=N)nc2sc(C(=O)NC(C)CC(C)NC(c3cnc(C)[nH]3)=O)cc12 C(C)(C(=O)N1CCCC(F)(C(=O)NOCCC(C)O)C1)(C(C)C)OC CC1CN(N(C)C2CN(C)C(C)(c3ccccc3)CC2)CCC1(F)F CN1CC=C(CC(=O)N2CC(OC3CCN(C(C4CC=CC4)=O)CC3)C2)CC1 C1(CC(=O)NCc2c(F)ccc(NC(CCC)=O)c2)CCC2(CC1)COC2 CC12CCCOC1CN(C(=O)NCC(c1ccncc1)O)C2 C1(C(=O)NCCc2nnc(C)s2)C2CCC(C2)N1C(C1CCCN1C=O)=O c1(OC)ccc(C(=O)NC2CCC(NC(C3CC3C(=O)N(C)C)=O)CC2)cc1O Cn1c(C(=O)NCCOCCNC(C2(Cl)CC2)=O)cccc1=O N1(C(CCC(c2ccc(C)cc2)=O)=O)CC2CC3CC2C1C3NC(C1CC1C)=O c1(CC(=O)NC(COC)(C)C)sc(C(=O)NC2CCCCC2OC)cc1Br C(=O)(C(C(=O)OC)OC)NCC(CN(C(CN(CCC#C)C)=O)C)(C)C C(N(C1CC1)N1CCC(CO)CC1)N(CC(NC1C(C)Oc2ccccc21)=O)C Cc1cc(C)c2nc(N3CCCCC3CCNC(c3c(C)ncn3C)=O)sc2c1 Cc1nccc(C(=O)NCCC2CN(C(C3CC4CC(=O)C3O4)=O)CCO2)c1C c1(C(=O)NCC(CC)NC(C2(SC)CC2)=O)cc(C(=O)NC)n(C)n1 c1(C(=O)NC(C2CCOC2)CNC(C(NOC)=O)=O)ccc([N+](=O)[O-])[nH]1 C1(CC)(NC(C2CCC3(CC2)CC3)=O)CCCN(C(c2cn(C)nc2OC)=O)C1 c1(CC)c[nH]nc1C(=O)NC(C1CCCCC1)C(C)NC(=O)C(=O)NCC(F)F c1(C(N2CC(CCNC(c3c(OCC)n[nH]c3)=O)C2)=O)cccc2nc(C)[nH]c12 C1(NC(c2c(C)cno2)=O)CN(C(C2CN(C)CCO2)=O)C2(CCC2)C1 C1(CCF)(NC(=O)CCn2cc(CCN(S(C)(=O)=O)C)nn2)CCN(CC)CC1 N1(C(C(CO)NC(C(C)C)=O)=O)CCC2CN(C(=O)C=C(C)C3CC3)CC2C1 C1(C)(C(=O)NCC2(NC(c3cnc(CC(C)C)[nH]3)=O)CCOC2)CC(C)(C)C1 c1(C(=O)NC2CC(C(C)NC(C3CC3C(C)(F)F)=O)C2)ncncc1Cl C1(CNC(C(C2CCC2)NC(C=C(C)c2ccco2)=O)=O)Cc2nccn2C1 CCCC(C(N)=O)NC(=S)NC1CCN(c2ccc(Cl)cc2)CC1 C1(NC(=O)NC2CCN(c3cc(Cl)no3)C2)C2CCC(C2)C1CO C=CC1(NC(=O)CN(C)C(c2cc(C)cc(O)c2)=O)CCCCC1 c1(CC)cccc(C(=O)NCCCC(=O)NCC2CCCOC2)n1 N1(C(c2n(C(C)C)ncc2Cl)=O)CCC(C)C(CNC(=O)CCc2nncs2)C1 C1(NC(CN(C(CCC(C)OCC)=O)C(C)C)=O)CN2CCC1(F)CC2 N#Cc1ccc(N)c(C(=O)NCC#CCNC(C2(C3CCC3)CC2(F)F)=O)c1 S(=O)(=O)(c1ccc(Br)cc1N1CC(O)C(C2CC2)C1)N(C(CSC)C)C C(=O)(C(O)CC(F)(F)F)NCC1(CO)CCN(C(C2N(CC)CCOC2)=O)CC1 c1(C(N(CC(CNC(c2cn(CCC)nc2)=O)O)C)=O)cc2scc(C)c2[nH]1 c1(CC)nc(C(N2CCC(CNC(=O)C=Cc3ccco3)C2)=O)c(Br)s1 N1(C(C=CC(CC)C)=O)CCC(=O)N2CCCC12 CC1(C)CCCOC1CC(=O)NC1CC(O)C1CC(=O)NCCc1cncnc1 c1(C(=O)NCC2OCCN(C(C(CCC=C)(F)F)=O)C2)c[nH]c2ccc(O)cc12 c1(C(CC)=O)cc(C(=O)NC2CCC(NC(c3cn(C)nc3O)=O)CC2)ccc1F C1(CN(C2CCCCCC2)CCNC(C)=O)CCCCC1(C)C c1(C(N2CCCC(NC(COCC=C)=O)C2C)=O)ccnc2ncc(C)cc12 C1(C2(O)CCOC2)(C(=O)NC2CN(CCC(F)(F)F)C2)CC1 c1(CN2CCC(C(C)C(=O)NCC3CCCC(O)C3)CC2)ccc(F)cc1Cl c1(C(=O)NC(CNC(c2c(OC)c(C)cs2)=O)C(C)C)nccc(C)c1N C(=O)(C(C)S(N)(=O)=O)N1CC(CC)C(C(=O)N(C)CCC2CCOCC2)C1 C1(NC(c2cccc(C)c2Cl)=O)C(C)CN(C(=O)CCc2cccs2)CC1C c1(CC(=O)NCC2(F)CN(C(C(CC)c3cccnc3)=O)C2)cc(C)cc(F)c1 c1(NC2(c3nnnn3CC3CC3)C(C)CCCC2)ccc2sncc2c1 C(CC)(C(=O)N1CC(C(=O)NCC(C)CC2CCC2)(SC)C1)OCC N1(CCC(C(=O)OC)F)C(=O)CCN(Cc2nnc(CN(CC)CC)s2)C1=O c1(C(=O)NCC2CC(NC(c3cnc(OC)nc3C)=O)C2)cc(Cl)c(F)cc1O c1(CC(N2CCC(NC(CCC3C(C)(C)C3)=O)C23CC3)=O)c(F)cccc1C#N CC1(C(N2CC(OCC(=O)NCCn3ncccc3=O)C2)=O)CCOCC1 N(C(=NCCCF)N1CCC2(CC(C(F)F)=NO2)C1)Cc1ccc(C)cc1 C(N=c1[nH]ccnc1F)C1CCCN(C(C2(C)CCCS2(=O)=O)=O)C1 C(=O)(C(CC(C)C)c1ccccc1)N1CC(N(C(c2cc(C)oc2)=O)C)C(O)C1 C1(NC(c2ncc[nH]c2=O)=O)C2CCC1N(C(=O)C(O)C1CCC1)C2 CCC1=NOC(C(=O)NC2CCCC2NC(=O)C(=O)NCCOC)C1 C12CN(CC(F)(F)C1)C2=O.c1(NC(CN(C)C)=O)cnccn1 C1(C(N)=O)CN(C(=O)C2=COCCO2)CCC1NC(C1(F)CCS(=O)(=O)C1)=O CC(C(=O)N1CCC2(C1)CN(C(=O)CN1CC(F)(F)C1)C2)C(C)C(C)(C)C c1(C(N2CC3C(CNC(C4C(C)(C)CCC4)=O)C3C2)=O)ncc(F)cc1N c1(C(N2CCC(N(C)C(C)C)C2)=O)cc(CO)c(C)s1.C12CN(C1)C2=O.CO c1(C(N2C(CN(C(C3OCCN(C)C3)=O)C)CCC2)=O)n[nH]cc1[N+](=O)[O-] C(=O)(CC(C)(C)O)NC(C1CCC(NC(=O)CSc2nncs2)C1)C c1(C2CN(C(=O)CCN3CCCC3)C2)ccc(S(=O)(=O)N2CCOCC2)cc1 C1(C(N2C(CNC(c3cc(F)cc(F)c3)=O)CC3(CC3)C2)=O)CCCC(F)(F)C1 c1(N(C)C(C2CC(n3ccnn3)C2)=O)ccc2cc(Cl)cnc2n1 C1(C(=O)OC)(C(N2C(C)CC(C(F)(F)F)C2C)=O)CC(O)C(O)C(O)C1O CC1(C)CC(N(C)C)CN(C(C2(N3CCCC3)CCC2)=O)C1 c1(C(N2CC(CNC(C3(Br)CC34CCC4)=O)C2)=O)cnc2ccoc2c1 c1(C(=O)NC2CC(NC(COC3(C)CCCC3)=O)CC2O)nccc2[nH]ccc12 N1(C(C(c2cnccn2)C)=O)CC2CC(NC(=O)Cn3nnc(C4CC4)n3)C1C2 N1(C(c2ccc(CC)s2)=O)CCC2(CCCN2C(c2cc3cnn(C)c3s2)=O)C1 C(=O)(CCCC(C)(C)C)NCC12CC(NC(Cc3nc(C)[nH]n3)=O)(C1)C(C)O2 c1(C(N(CCCN(C(C(CC(C)C)(F)F)=O)C)C)=O)cccc2cc(O)ccc12 C=C(C)C(CC(=O)N1CCC(CC)(OCC)C1)NC(=O)C(C)SCCCC C#CCCCCC(=O)NC1(CCNC(=O)CSCCC)CC1.c1(NCC)ccccc1 C(=O)(C1CCc2cccc(F)c21)N1CCC(CNC(CCc2n(C)ccn2)=O)C1 N1(C(C(C(C)C)SCC)=O)CCN(C(=O)CCSCC(N)=O)CC1CCO c1(NCC2C(NC(=O)OC(C)(C)C)CCC2)ccc(S(C)(=O)=O)nc1 c1(C(N2CC3C(CNC(CCCC)=O)(C3)C2)=O)csc2nnsc12 c1(N(CCCS(N)(=O)=O)C(C(=O)NC)Cc2ccccc2)cccc(OC)c1 N1(C(C(C=C)(F)F)=O)CCOC2(CCCN(C(c3cccnc3S)=O)C2)C1 c1(CNC(C(=O)N(CCC#N)Cc2cnccn2)=O)cc(Br)c(Cl)c(Br)c1 C(=O)(C(C)(C)C1(O)CCOC1)NCCC(C)NC(=O)CC(C)c1cccnc1 C1(CNC(C(CC)O)=O)CC2CCC1N2C(C1CCC(SCC)CC1)=O n1(C(C)C)cc(CNC(=O)CCc2ccon2)nn1 c1(CC(N2CCSCC2c2nn[nH]n2)=O)cc(Cl)cc2ccccc12 CCN=c1[nH]c(C(=O)NCC2(CN(C)C(C3CCC(C)O3)=O)CC2)cs1 C1(CNC(CC2CCC(C)C2)=O)(NC(C2CCC(C)(C)C2)=O)CCOCC1 c1(NC(C(C2CC=CC2)N(C(C)C(=O)OC)CC)=O)ccc(Cl)cc1 Cc1cn2c(n1)CCC(C(N1CC=CC(NC(=O)Cn3ncccc3=O)C1)=O)C2 C1(C(N2CCC(NC(Cc3c(CC#N)cccc3)=O)C2)=O)CCCC12CCC2 C1(COC)(CNC(C2C=CCC2)=O)CCN(C(C2(C)CC2C)=O)C1 c1(C(=O)NC(C(C)C)CNC(=O)COC2CCCOC2)cc2n(n1)CCO2 C(C1CN(C(=O)CO)Cc2ccccc21)NC(C1CCC(CCCC)CC1)=O C1(NC(c2c(OC)c(Cl)ccc2)=O)CCC(O)CN(C(c2cnccn2)=O)C1 c1(C(N(C2CC(NC(c3c(C)ncnc3)=O)C2)C)=O)cc(N)c2ccccc2n1 c1(CCC)nc(-c2sc(Cl)cc2Br)n(-c2ccc(C(C)OC)cc2)n1 N1(C(c2cc(C)cc(Cl)n2)=O)CCC(CNC(C2COC(C)C2)=O)C(F)(F)CC1 c1(C(N(CCCNC(C(COC)C)=O)C)=O)cc(OC)c(Cl)s1 C(CN=c1nc(N(C)CC2CCCO2)c2c([nH]1)CCS2)C1(OC)CC1 C1(C)(C(=O)NC(C)C(CO)NC(=O)COC2(C)CCCC2)CCOCC1 c1(C(=O)NC2CC(NC(c3ccnnc3)=O)CC2O)n[nH]c2ccc(Cl)cc12 N1(C(c2c(OC)cnnc2)=O)CCOC2(CCN(C(=O)C(C3CC3)SC)C2)C1 C(c1nc(C)cs1)=CC(=O)NC1C(NC(C(c2ccccc2)SC)=O)CCC1 CC1CN(C(=O)C(=O)NC2CC2)CCC1N(C(=O)C(O)CN(C)C)C C(CCCCC(=O)NCC1CCC1NC(c1cc(F)ccc1O)=O)OCC CCC(C)C(O)CNC(=O)CC1(NC(C2CCOCC2)=O)CCC1 c1(C(C)C)nnc2n1CCN(C(c1cc(C3CC3)no1)C(=O)NC1(C)CC1)C2C C1(CC(=O)NC(C)CCNC(c2cc(CCCO)on2)=O)CCCS1(=O)=O C1(CNC(C2(NC(c3ncn4c3CCC4)=O)CCC2)=O)CC2CCCC2C1 N1(C(CC2(N(C)C)CC2)=O)C2CCC1CN(C(=O)Nc1ccc(CO)cn1)C2 C1(NC(Cc2ccn(C(C)C)n2)=O)CC2(C1)CN(C(C1(C(F)F)CC1(F)F)=O)C2 Cc1cc(=O)n(C)nc1C(=O)NCC1(CNC(=O)C=Cc2ccsc2)CCCC1 CC1(C)OCCC1(O)C(N1CCC1(C)CC(=O)NC(c1cccnc1)CO)=O C(=O)(C1CCc2cccc(O)c21)NCCCNC(COCCC(C)C)=O c1(CNC(=O)NC(C)CC2CCOC2)ccc(F)cc1[N+](=O)[O-] C(=O)(C(C)(C)CNC(N)=O)NC1C(NC(c2c(C)coc2)=O)CCC1 N12CC3CCC(C1)C(C3)NC2=O.c1(C(C(C)C)N)ccc(Br)cc1.C1CC1 C1(C(=O)NCc2ccc(C(=O)NC(C3CCCO3)C)s2)CCS(=O)CC1 N1(C(CCC(C)(C)C#N)=O)C2CC=C(C(=O)NCc3ccc(Cl)nc3)C1CC2 CCC(C)CCCCC(=O)NCC(CO)NC(c1[nH]ccc1-c1ccccc1)=O C(N=c1nc(N2CCOCC2)[nH]c(=NC2CCCCC2C#N)[nH]1)C1(C)CCOCC1 C(=O)(C1CCCc2c(O)cccc21)N(C)CC1CCCN1C(=O)C(F)=C1CCC1 n1(CC)cc(C(=O)NCCC(O)C(=O)NCCCCN(C)C(C)=O)c(C)n1 CCC(C)(CNC(=O)C=Cc1cnc[nH]1)N.C(C(C)(C)C)C1C(C(=O)NC(=O)CO)C1 c1(NC(C(C)(C)CCNC(c2cc(F)ccc2O)=O)=O)ccc2c(c1)CCO2 N1(CC(N2CC(O)(CNC(C=Cc3cnc(C)s3)=O)C2)=O)CCc2sccc2C1 N1(C(C(C)n2cccc2)=O)CCCC1(C)CNC(=O)Cc1cscc1Br O=C1CCC(NC(=O)C(c2ccc(C(F)(F)F)cc2)NC(C2(Br)CC2)=O)CN1 C(CCCCC(=O)N1CC(OCC(=O)NCC2NC(=O)CC2(C)C)C1)OCC c1(C(=O)NCC2(C)CC(NC(C(C)=C3CCC3)=O)C2)ccccc1SC(F)(F)F C1(C(=O)NCC(C2CCC2)NC(c2cc[nH]n2)=O)CCC2(CCCC2)C1 C1(C)(CCC(=O)NCCNC(CC(C)OCC)=O)CCC(=O)N1 C(=O)(C(C(c1ccc(OC(C)(C)C)cc1)NC(C)=O)N1CCC(CF)C1)OC N1(C(C(C)N(C(C)=O)C)=O)CCC(N(CCN(C)C)C(C2CCCO2)=O)CC1 c1(C(=O)NCC(C)(C)CNC(=O)CC2CC3CCC2O3)c[nH]c2c(Cl)cccc12 c1(C(=O)NCC(=C)CCNC(=O)C(C2CCC(=O)N2)C)ccc(OC)cc1 N1(CCC)CC(NC(C2CCCN2c2cccc(C(N)=O)n2)=O)C(C)(C)C1 C(C#CCCO)NC(C=C(C)CNC(c1sccc1CO)=O)=O c1(C(C)NC(C2(NC(C(C)N3CCCC3)=O)CC2)=O)ccncc1 n1(COC)ccc(C(=O)NCC(C)N(C(=O)CCCn2cncn2)C)n1 c1(C(N2CCCC(NC(C3(C4CCCCO4)CC3)=O)C2)=O)ccnc2ccnn12 N1(C(C(C)C2CCC2)=O)CCCCC1C(C)(C)CNC(=O)Cc1ccccc1 c1(C(N(C2CN(C(C(CC(C)C)O)=O)C2)C)=O)ccc([N+](=O)[O-])cc1 CC1C(NC(c2cccc3c2CCCO3)=O)CC2CCC1N2C(=O)C(C)N(C)C c1(C(N2CCN(C(c3csc(Br)n3)=O)C3CC23)=O)cc(F)c(F)c(F)c1 C(=O)(C1=CCCC1(C)C)NC1C2CN(C(C(CC(C)C)N(C)C)=O)CC21 C1(NC(c2cccc(C3CC3)n2)=O)CCCCN(C(c2n[nH]cc2Cl)=O)CC1 c1(C(=O)NC(C(C)C)CCNC(=O)C=CCN2CCOCC2)nccc(Cl)c1F CC1(C)CCCC1C(=O)NCCC1CCN(C(C2(C(N)=O)CC2)=O)C1 C(=O)(C(C)CSC)NC(C1CCCC1)CNC(CCOCCOC)=O C1(CN(C(=O)C(F)C2CCOC2)C)CCC(CNC(C23CC2CNC3=O)=O)CC1 C1(=O)CC(C)CC(=O)C(=O)C=CC2CCN1CC2.C=CCCC(C1CC1)N.OC c1(CN(C(C)CNC(c2cc(C3(C)COC3)no2)=O)C)nc2ccccc2o1 N1(C(c2cc(OC)n[nH]2)=O)CC(O)CCC1C(N1CC(c2ccon2)C1)=O CCC(CC(=O)NC1(CCCNC(c2cc(CC(C)C)[nH]n2)=O)CC1)C(F)F N12CCN(C3CC13)CC=CCC(=O)C(=O)C(C)C2=O.CCO.OC C1(CNC(C(C)OC(C)(C)C)=O)CCN(C(c2c(Cl)cnn2C)=O)C12CCC2 C1(C(=O)NC(c2cccc(-n3ccnc3)c2)C)CCCCN(c2ncnc(=N)[nH]2)C1 O=C1CCC(S(=O)(=O)N2CCN(CCNCc3cc(I)cc(I)c3O)CC2)CC1 c1(NC(CC(C)(C)NC(C(C=C)OC)=O)=O)c(C)cccc1C c1(C(=O)NCC2OCCN(CC(=O)OC)C2)cc(Br)c(OC)cc1OC c1(OC)c[nH]c(C(N2CCC(CNC(=O)Cn3ccc(C)n3)C2(C)C)=O)cc1=O C=CC1(CC(=O)NCCCCCN(C)C(c2conc2C)=O)CCC1 Cc1[nH]c(C)c(C(N2CC(C(=O)NCc3ncccc3O)C(F)(F)C2)=O)c1C C1(C(N(C(CNC(C(C)c2ccco2)=O)C2CC2)C)=O)CCc2ccnn2C1 S(=O)(=O)(c1cccc(CNc2ccc(NC(=O)C(C)(F)F)c(F)c2)c1)NC C1(CNC(c2cc(C(F)(F)F)ns2)=O)CC(O)CN1C(c1csc(O)n1)=O N1(C(CCC=C(C)C)=O)CCCC2(C1)CN(C(=O)C(C)S)CCO2 C1(NC(C(C2CCC2)NC(C(C)NC(CC)(C)C)=O)=O)CCCCC12CCC2 c1(C(=O)NC(CC#C)C(=O)NCC2(CO)CC2(C)C)cc(C)cc(C#N)c1 C1(C(N(CC(C)NC(c2ccn(C)n2)=O)C)=O)CCCCC1c1ncccn1 N1(C(CC(C)OC)=O)CCC2(CC1)CC(N=c1nc(C(F)(F)F)[nH]s1)CCO2 c1(C(=O)NCC2N(C(CC=C=C)=O)CC=C2)cncc2c(Br)cccc12 C(=O)(CCCC(OC)OC)NCC(C(=O)NC(CC)C1CCC1)CC1CC1 N1(C(CCCOCC=C)=O)CC(NC(=O)Cn2cc(Cl)c(C)n2)CC1(C)C C=CC(C)(CC)C(=O)N1CC(CN(C)C(c2ccc(-c3cc[nH]n3)s2)=O)C1 CC(C)C(C)(CNC(c1cccn1C)=O)NC(=O)CCC1CCCO1 N1(C(CCN(C(c2c(CC=C)cccc2)=O)CCO)=O)CC(=O)N(C)CC1C Cc1cc(C(=O)NC2(CNC(c3ncccc3N(C)C)=O)CCOC2)[nH]c1C c1(C(N2CC(CNC(=O)CC3CC=CC3)C3(C2)CC3)=O)cnn2c1OCC(F)C2 C1(NC(C23C(CN(C(c4cnc(C)o4)=O)C2)C3)=O)CCCOC12CCC2 CCC(C)CCC(=O)N(CCn1cc(C2COCC2O)nn1)CC CCCCC(F)C(=O)NC1CC2CC(NC(c3ccnn3CC#N)=O)C2C1 N1(C(c2ccc(OCC)c(Br)c2)=O)CC2CCC(C1)C2CC(N1CCC1CO)=O CC1(C)CCC(CCNC(C2CC(O)CN2C(C2COCCO2)=O)=O)O1 Cc1ncc(NC(C2(O)CCN(C(c3sccc3Br)=O)C2)=O)nc1C c1(C(=O)NC2CC3CC2N(C(c2ccc[n+]([O-])c2)=O)C3)cc(F)c2[nH]nnc2c1 N1(C(C=CC)=O)CC(C)(C)CCC1CNC(=O)C(O)Cc1cccc(N(C)C)c1 c1(CNC(c2cc(C)c(-n3cnnn3)cc2)=O)ncnc2c1OCCO2 Cc1cc(C(=O)NC(C2(O)CN(C(=O)Cc3ccon3)C2)C)ccc1Cl Cc1cc(C(=O)NCC2CCN2C(C2CC(C)C2)=O)n(CC(F)F)n1 c1(N(CCC(=O)NC)C)nc2c(c(=NCc3nnc(O)n3C)[nH]1)CSC2 C1(CN(c2ccc(OC)c(C(F)(F)F)c2)C)COc2ccccc2C1 c1(C(=O)NC2C(NC(c3ncc(F)cc3F)=O)C2)cc(OC(F)F)ccc1F CC1CCCCC1(CNC(=O)C(F)(F)c1cccnc1)NC(=O)CC(C)C(F)F c1(CN2CC(CNC(c3cnn(-c4ccccn4)c3)=O)C2)ccc([N+](=O)[O-])o1 C(CCC#C)(C(=O)OC)NC(C(CC#C)C)=O CCCC(CCCNC(c1csc(Br)n1)=O)NC(=O)C(O)CC(C)C Cc1nc(O)[nH]c1C(=O)NCC1CCCCN1C(C1C(C)C1(F)F)=O c1(NC(c2n(C)cc(Nc3nc(OC)cc(OC)n3)n2)=O)cc(C)c(C)cc1Br C(=O)CCC(=O)N(CC(=O)NC(COC)C(C)C)C(C)C.CCOCC C1(NC(C(CC=CC)NC(=O)CCC=C(C)C)=O)CN(C)C(=O)C12CC2 C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1C2(CCN(C(c3ccc(CSC)o3)=O)C2)C1 c1(OC)ccc(C(C)(C)C(N2CCC(C)(NC(=O)C(C)CC3CCC3)C2)=O)cc1 C1(CC)(CNC(=O)CCC2CCN(C(c3n[nH]c(C)c3O)=O)CC2)CC(C)(C)C1 N1(C(c2c(OC)cnc(Cl)c2)=O)CCC(C2CC2NC(C2CC2F)=O)CC1 C1(CC)C(CO)CCN1C(=O)NCCCOC(F)(F)F.c1(O)cccnc1 N1(C(C(C)CC(F)F)=O)CCC2(CC(C(N3CCC(c4cc[nH]n4)C3)=O)C2)C1 N1(C(C(CCN(C)C)(C)O)=O)CCC(C)CC1C1CCC(C)O1 N1(C(C(=O)Nc2c(C)ncs2)=O)CCCC(C2CCNCC2)CC1 N1(C(CC(C)N(C)C)=O)CC2CC(C(=O)NCC(O)C(=O)N(C)C)(C2)C1 Fc1ccc(C2CCCN(CC(c3ccccc3)Sc3cccs3)C2)cc1F c1(C(=O)NC(C(C)NC(c2cc(CC)sn2)=O)C)cncn(C)c1=O CC1=C(C(=O)NC2CC(c3ccccc3)(NC(c3ccc(C)s3)=O)C2)CCO1 CC1CCCC(CNC(c2ccc(-c3ccc(F)cc3)[nH]2)=O)O1 C1(C)(C2CC(C(=O)OC)C2)CCC(COC(C)(C)C)C1.c12cc-1on2 c1(NC(C2(C)N(C(CC=CC)=O)CC2)=O)cc(C)cc(C)c1O C1(CNC(c2nnc(CC)s2)=O)C(C)CCN1C(C1OCCCO1)=O Cc1nc(C)c(CNC(=O)CC2COCCN2C(=O)C(C)O)s1 c1(N2C(C)(C(=O)Nc3cnoc3)CCC2)ccn2ncc(I)c2n1 CC1CCC(C(=O)NCC(C2CCC2)NC(c2csc(C(C)C)n2)=O)CC1 c1(C(N2CC(C)N(C(C3CC(C4CC4)C3)=O)CC2)=O)c[nH]c2ncccc12 N(C(=NCCF)N1CCCC(C(=O)OC)C1C)C(CC)CO C1(CC(=O)NCC2CC(OC)CN2C(c2ccsn2)=O)CC2(CC(OC)C2)C1 Cc1[nH]c2ncccc2c1C(=O)NCCNC(=O)C(CC=CCl)c1ccccc1 CC(O)CCCC(=O)NCC1CCN(C(C2(F)CC2c2ccccc2)=O)C1 N1(C(C2N(CC)CC2)=O)CC(NC(=O)Cn2cccc2)CC(O)C1 C12CN(CC1n1ccnn1)CC1CCN1CC(=O)N2.C1(C(=O)OC)(SC)CCC1 C(C)(N=c1[nH]c2c(c(=NCCN(CC(F)F)C)[nH]1)SCC2)c1ccc(C)cc1 C1(NC(C(C=CC)O)=O)CCN(C(c2cscc2Cl)=O)C1c1ccccc1 C(=O)(C1CCCn2cnnc21)NCC=CCNC(c1nc(CC)oc1C)=O c1(C(N2CCC(O)(C(CNC(c3c(CC)ocn3)=O)C)C2)=O)ncc(C)cc1C C1(C(N2CCC(NC(c3c(C)nn(C)c3Cl)=O)C(O)C2)=O)C2CCC1(C)C2(C)C c1(C(N2CCC(CNC(C=CCOC)=O)(OC)C2)=O)cn2ccccc2n1 C1(CN(C(CCN(C)CC)=O)C)CCCN(C(=O)C(O)c2ccsc2)C1 C(=O)(C1=CC2CCC(C1)C2)NC1C(C)(C)CN(C(C2CC(C(F)(F)F)C2)=O)C1 CCC(CC(=O)NC(C)C=CC(=O)NC(CF)C(F)(F)F)C(C)(C)C c1(C(N(CC(N2CCN(C(CCC(C)C)=O)CC2)=O)C)=O)c(N)ccc(F)c1F CCCC(CNC(c1cncn1C)=O)NC(C1CC1Cl)=O C=CCC(C)(CC)C(=O)NCC(O)CCNC(c1ccnc(Cl)c1O)=O C#CCCCC(=O)NC(C1CCN(C(c2cncnc2C2CC2)=O)C1)C C(=O)(C(C)C(C)(C)C)N1CC(CNC(CCC#C)=O)(COC)C1 C1(CCC)CN(C(=O)COc2cc(C)on2)CC1NC(c1sc(F)cc1C)=O C1(C(=O)NCCC2CC(NC(C(c3ccccc3)C)=O)C2)CCCCCC1(F)F Cc1nc2cncc(C(=O)NC(CNC(=O)C(F)C(C)(C)O)C3CC3)c2[nH]1 c1(C(C)(C)C)ccc(C(=O)NCC(C)(O)CNC(=O)C(O)C2CCC2)cc1Cl C1(NC(CN(C)C)=O)COCC1CNC(=O)C(F)Cc1ccccc1 c1(C(=O)NC(CC=C)CNC(C2C(C(F)F)C2(C)C)=O)ccn(C(C)C)c1C C(C)(C)(CCC(=O)N1CCCC(O)C1C)NC(CC=CC)=O C1(C(C)NC(=O)C(C)n2cccn2)CCCN1C(C1CC(n2ccnc2)C1)=O c1(OC)cc(CC(=O)NC(C2CN(C(=O)CN3CSCC3=O)C2)C)ccn1 C(=O)(C(C)CC(F)F)NCC(C(C)(C)C)NC(c1c(C)oc(-c2ccsc2)c1)=O N1(C(c2cc(OCC)n[nH]2)=O)CCC(C(=O)N(C)CCOCC)C12CC2 C1(C(=O)OCCC2(C)CC2)Cn2cnnc2CN1CC(C)(C)C c1(C(=O)NCC(CNC(C2CCN(C(C)C)CC2)=O)CO)cccc2scnc12 C1(O)(CN(C)C(c2cc(Cl)nn2C)=O)CCN(C(C2(C)COC(=O)N2)=O)C1 N1(C(CCCC)C(=O)OC)CC2(NC(=O)OC(C)(C)C)CCC2(C(=O)O)C1 Cc1ccc(CNC2CCOC(C)(C)C2)c(O)n1 C1(C2CCCN(C(C3CC3Cc3cccnc3)=O)C2)(NC(=O)C=CC2CCC2)CC1 n1(CC(N2CC=CC(NC(C(c3c(C)cccc3)C)=O)C2)=O)nc(C)n(C)c1=O c1(N2CCC3(CC(OC)C3)C2)nc2c(c(=NCCS(=O)CC(F)(F)F)[nH]1)CCC2 c1(OC)ccc(-n2nc(CSc3ccco3)nc2CC(C)C2CCC2)cc1C N12CC(C(C)(C)C1)n1cc(nn1)C2.c1(C[SH](c2c(C)c[nH]n2)C)nnc(C)n1C N1(C(C)=O)CCC(C)(C)C(NC(=O)C(Cc2ccc(F)cc2F)N(C)C)C1 N1(C(Cn2ccc(C)n2)=O)CCC2(CC1)CN(C(c1ccc(C(C)O)cc1)=O)C2 O=C(CCCCC(F)(F)F)NCCC1CN(C(C2CCC(F)(F)C2)=O)C1 CC(CCNC(=O)CC(C)F)CCNC(=O)Cc1cc(Br)cs1 C1(C(=O)NC(C(CC)CC)C)CCCN1NC(=O)c1nnsc1N c1(-c2cn(CC(=O)NCc3ccccc3)nc2)cncc(OC2CCCCO2)c1 c1(SC)cscc1C(=O)NCC1(CN(C(=O)CC2CCC(C)C2)C)CC1 c1(NC(C2CC(F)CN2C(c2cc(C(F)(F)F)c[nH]2)=O)=O)cc(F)c(Cl)c(Cl)c1 C1(C(=O)NCCC2(OC)CN(C(C3CCNC3=O)=O)C2)CCCN(S(N)(=O)=O)C1 c1(OC)ccccc1C(=O)NCC(C)CNC(c1cc(C)n(C(C)C)c1)=O N1(C(c2cnc(O)o2)=O)CCC2C(CCN2C(c2cccc3sncc23)=O)C1 C12(NC(c3cc(C(N)=O)sc3)=O)CCCC1(F)CN(C(C1CCCS1)=O)C2 N1(C(COCC(C)(C)C)=O)CCCCCC1CNC(C1(CO)CCCO1)=O C(=O)(C(CC(C)C)N(C(=O)CCCNC(C)=O)C)NCC(=O)OCC N1(CCCNC(COCCCC)=O)CCC(NC(=O)C(C2CCOCC2)F)C1 c1(C2C(N(C(C)(C)C)C(c3c(C)nc[nH]3)c3nnnn3C)CCC2)ccc(F)cc1 C(C)(C(N=c1ccnc(Cl)[nH]1)C(C)C)NC(c1cnc(SC)nc1O)=O C=CCC(F)(F)CNC(=O)C(CC1CCOCC1)NC(=O)C(c1ccn(C)n1)C N1(C(C2(CC=C)CCC2)=O)CC(NC(=O)CCC2CCC(=O)N2)C(CO)C1 c1(SC(C(=O)NCCCCNC(CC(COC)C)=O)C)ccc(C#N)cc1 Cc1c(C(=O)NC2CCN(C(=O)CC(F)F)C2C(C)C)nnn1-c1ccccc1 C1(C(=O)NCc2onc(C)n2)C2CCC(C2)N1C(C1C2CCCCCC12)=O C(=O)(C(CCOC)OC)N(CCCC)CC.c1(C(=O)OCC)ccc(CCOC)o1 Cc1cc(C(=O)N(C(CNC(c2sc(=N)[nH]c2C2CC2)=O)C2CC2)C)nc(C)c1 Cc1nccc(C(=O)NCCC2(C)CCN(C(=O)C(CC(C)C)N(C)C)C2)c1O C1(CC(=O)NCC2CC(F)(F)CN2C(c2cc(O)cs2)=O)CCCCCC1(F)F c1(C(C)C)nccc(C(=O)NCCC2CN(C(=O)CC3COCCO3)C2)n1 CC(=O)CCC(=O)NC1CC(CCC(N2CC3CC3C2)=O)C1 N1(C(C2C(C(C)C)CCC2)=O)CC2(CCN(C(c3ccn(C)c3)=O)CC2)C1 c1(C(N(CCCCNC(=O)C=Cc2cncs2)C)=O)c(O)cccc1F c1(C(N2CCCCC(NC(C3CC4CCC3O4)=O)C2)=O)cccc(O)c1[N+](=O)[O-] C1(C(=O)NC(CSCC)C)CN(C(=O)CSC)CCN1 CC1c2nccn2CCN1C(C1(F)CCN(C(c2cnc3cc[nH]c3c2)=O)C1)=O Cc1cn2ccnc(C(N3CCN(C)C4(CC4)C3)=O)c2n1 C12(NC(c3nc(CC)sc3N)=O)CCCC1CN(C(=O)C(O)c1cnc[nH]1)C2 CCC(CC)CC(F)C(=O)N1CCC(F)(C(=O)NCC2CN(C3CC3)C2)C1 N1(C(c2ccc(OC)o2)=O)CC(C(=O)NCC2(O)CC3CCC2O3)CCC1C C1(C(N2CC(CNC(c3ccc(C(C)C)cn3)=O)(CO)C2)=O)CC2C(C1)C2(C)C C(CCOC)(C(=O)N1c2nsnc21)N1CCC(C(=O)OCC)C1.C(COCC)NC CC(CS(C)(=O)=O)C(=O)NC1CCC12CN(C(c1cccn3cncc13)=O)C2 c1(NCCNC(C2C(CCCC)CCC2)=O)ccc(Br)c(C)c1[N+](=O)[O-] c1(C(C)=O)c(Cl)nc[nH]c1=NCC=CCNC(c1cc(C2CC2)nc(O)c1)=O c1(CC)ncc(C(=O)NC2CCC(CC(=O)NCC(c3ccco3)O)CC2)cn1 c1(C(=O)OCCCCn2cc(CCCC)nn2)oc(OC(C)C)nc1-c1cccs1 C(N=c1nc2c(cnn2C(C)C)c(N2CCS(=O)(=O)C(CO)C2)[nH]1)C1C(C)C1 C1(F)(C(N(CC(C2CCC2)OC)C)=O)CCCN(C(=O)C=C2CCC2)C1 N1(CC(=O)NC(C(=O)NC(C(=O)NC)Cc2ccoc2)CC2CC2)CCN(C)CC1 C(=O)(C1CCCc2cncn21)NC(C(C)NC(C(C(C)C)n1cnnc1)=O)CO Cc1cc(CNCC(c2ccc(Br)c(F)c2)NC(=O)Cc2ccco2)nnc1C S(=O)(=O)(c1cccnc1N1CC2(C)COCC2(C)C1)N(CC)Cc1ccnn1C C(CCCCCCC(=O)NCC1CCCN1C(=O)Cc1ccc(F)c(F)c1)SC c1(CNC(CSCCN(CCN(C)C)C)=O)ccc(F)cc1C1CC1 N1(Cc2nnc(-c3cc(OC)ncc3)o2)C2CCCC1CN(C(C)=O)CC2 C1(NC(=O)OC(C)(C)C)C2CCC(C2)C1C(=O)OC(C)CCC(=O)O C1(C(=O)NCC2(C(=O)NC(CSCC#C)=O)CC2)Cc2ccccc2N1C(C)=O O=S(=O)(c1ccc(N2Cc3cccnc3C2)c(Br)c1)NCCCn1cncn1 n1(CCC)cc(CNCCC2CCOC(C)C2)c(C)n1 N(C(=NCCC(=O)OC(C)C)N1CCCC(C)CC1)C1CC2(CC(OC)C2)C1 c1(N(CC(C)(C)C)CCC#C)[nH]c(=NCCC(C)c2ccccc2)nc2scnc12 CC1CC(NC(c2cc(O)cc(Cl)c2)=O)CCN1C(C1C2CCC12)=O c1(C(=O)NC(C)C(C)NC(c2ccc(O)s2)=O)cc2n(n1)CCNC2=O C#CCCN=C(NCCS(=O)(=O)CC)NC1CCC(C(F)(F)F)CC1 C12CCCC1CCO2.Cc1ccncc1-c1cn(C)nn1.C1(C)(C)CC=CC(=O)N1 C(=O)(CC(C)(C)C(F)F)N1CCN(CCCNC(CC(C)C(F)F)=O)CC1 c1(CC(C(=O)NC(C)CCNC(=O)Cn2ncnn2)C)ccc(Cl)cc1 c1(C(=O)NC(C(C)(C)C)CNC(C2CCCN2C2CC2)=O)ccnc2ccsc12 C1(NC(=O)CC2(C(F)(F)F)CC2)CC(NC(C2CCCCC2)=O)C12CCOCC2 C(c1ccccc1OC(F)F)=CC(=O)NCC(CC)NC(=O)C(C)=C1CCC1 C(=O)(C1CCc2nnc(C)n21)N(CCC(C)NC(CC(C=C)(C)C)=O)C c1(CC)cc(F)ccc1CC(N1CCCCC1CN(C)C(C1CCCCO1)=O)=O c1(C(N(CCNC(=O)C(F)=C2CCC2)C2CC2)=O)cn(-c2ncccn2)cn1 c1(CNC(=O)NCC2CCCC2NC(c2ccccc2)=O)cc2c([nH]1)CCC2 C1(NC(c2cnc(CC3CC3)s2)=O)CN(C(=O)C2=COCC2)C2CCCCC12 c1(CC(N2CC(CNC(c3cccc(OC(C)C)n3)=O)C2)=O)cc(F)ccc1C C1(CNC(C(=O)NCC2N(CCC)CCCC2)=O)CCCC2(CCOCC2)O1 C1(C(=O)NC(C2CC2)C2CC2)CCCCCN1C(c1ncnn1C)=O Cc1cc2cc(CN3CCNC(=O)C3C(N)=O)ccc2s1 c1(OC)ccc(C(CNC(c2cccn2C)=O)NC(C2(C)CCCN2C)=O)cc1 c1(C(N2CC(NC(c3cnc(C(C)C)nc3)=O)C2)=O)c(O)ccc2ccccc12 C(=O)(C1=C(C)OCCC1)N1CC(COC)(NC(=O)CC2CC2C)C1 S(=O)(=O)(C1CN(C(=O)Nc2ccccc2)C1)NC(C)Cn1cnnc1 C(=O)(C1=CC(C)CC1)N(C)CC1N(C(Cc2nc(C)sc2Cl)=O)CCOC1 c1(CNC(=O)COc2ccsn2)ccc(F)cc1.C1(=O)CCCOC2CN1C2 N1(C(C(CCC)NC(N)=O)=O)CCC(C(=O)N(CCF)CCOC)C(C)(C)C1 CC(C)C(C)(CNC1(N2CCOCC2)CCSC1)NC(=O)OC(C)(C)C c1(OC)cccc(C(CNC(=O)C(F)=CCCF)NC(=O)Cc2sccc2C)c1 C1(NC(c2cn(CCCC)nc2C)=O)CCN(C(c2ccsn2)=O)C12CCC2 CCC(C)(C#N)C(=O)NC(CC(=O)NCc1cncc(C)c1)C1CC1 C(c1ccc2occc2c1)=CC(N1CCC(C(C)NC(c2ccns2)=O)CC1)=O c1(CN2CCC3(C(C(=O)Nc4nc(C(F)(F)F)cs4)C3)C2)cc(Br)c(F)cc1O n1(C(C)C)ccc2ccc(C(=O)NC(C)CCNC(c3cnsn3)=O)cc12 c1(C(=O)NCC(C2CCC2)NC(CC(=C)Br)=O)ccc(N(C)C)cc1F C1(NC(c2n(C)ncc2Br)=O)C2CCN(C(=O)CCc3cccs3)CC12 C1(C(CNC(C(CC)C)=O)(C)C)CCN(C(=O)CCC2CC2(C)C)CC1 c1(-c2cn(C3CCC(C(N)=O)CC3)nn2)cc(F)cc(Cl)c1.C12CCCN(C1)C2 c1(OC)cc(CC(=O)NCC(C)N(C(=O)C(c2ccccn2)O)C)on1 CS(=O)C1CN(C(C2CCOCC2NC(c2cc[n+]([O-])cc2)=O)=O)C1 c1(OC2CCC(NC(N3CCN(C)CC3)=O)C2)ccc(C(F)(F)F)c(F)c1 CC(C)CC(=O)C(=O)N1CCC(O)(C(N2CCCC(C(N)=O)C2)=O)C1 CP(C)(=O)C1CCC=C1C(=O)NCC1CCCN1C(=O)Cc1cnoc1 C(CCO)(C(=O)NCCCCn1cc(CCS(N)(=O)=O)nn1)N(C)C C(CC(=O)NCc1cnn(C)c1)(C(F)F)NC(C(CC1CC1)OC)=O N1(C(CCN(C(=O)C(C(=O)OC)OC)CC)=O)CCCC12CCCC2 C1(NC(C23CCC(C)(CC2)OC3)=O)COC2(CCCN(C(C3CC34CC4)=O)C2)C1 CC12CC1CCN2C(=O)NCc1ncccc1CO c1(C(N(C2CCCN(C(C3CCCOC3)=O)C2)CC)=O)cc(OC)cc(F)c1 c1(OC)ccc(Cl)c(C(N2CCCCC2CNC(c2ccc(C)c(F)c2)=O)=O)n1 C1(C(=O)NC(CNC(c2cnn3c2OCC3)=O)C2CC2)CCc2ccccc2O1 C1(C)(CNC(c2c(CC)n(CC)nn2)=O)CC(OC)CN1C(=O)CC(C)C N1(C(c2ccc(CCC)s2)=O)CCC(C(F)F)(CNC(c2c[nH]c(=N)o2)=O)C1 CC1COCCN1C(C1CCOC(CNC(c2cncs2)=O)C1)=O C1(CNC(C(C)(C)SC)=O)CCCN(C(=O)CCOC2CCC2)C1 C(CC(C)(C)C)OCC(=O)N(C)CC=CC(=O)NCCF c1(CC(=O)N(C)CCOCCNC(C2(COC3CC3)CC2)=O)ccncc1 C12(C(=O)NC(CC)CN(C(=O)CSCC(C)C)C)CCC(CC1)C(C)O2 c1(C(N2CC(C3CN(C(C(CC)CC)=O)C3)C2)=O)cc(S(N)(=O)=O)ccc1C C(=O)(CCCCCS(N)(=O)=O)N(C1CCN(C(=O)CC2(OC)CC2)CC1)CCCC C1(NC(c2ccccc2SC2CCOC2)=O)CN(C(C2CCOCC2)=O)CC1O CC1CN(C(c2ccc(CCCNC(=O)C(=O)N(C)C)[nH]2)=O)CC1(C)CO c1(-c2nc(C3CC(N(C)C)C3)n(CCOC(C)(C)C)n2)ccc(F)c(Cl)c1 CC(C)(C)CC(=O)NC1CC(F)(CNC(C2CCCOC2)=O)C1 C(=O)(C(C(C)C)C1CCC1)NC(COC)C(=O)N(C)CCC1CC1 c1(C(=O)NCC(C)(O)CNC(=O)C=CBr)cc2cscc2s1 N1(C(C(N2CCOCC2)C)=O)CC2CC(C1)N(C(C1CCCC(C)(C)CC1)=O)C2 N1(C(CC(CN(C)C)O)=O)CCC(NC(=O)CCCC2CCOCC2)C(O)C1 CCCCC(O)C(=O)NCC#CCNC(C1COCCN1C)=O N1(C(C(CSC)O)=O)CCCC2(C1)CN(C(c1cc(C)n(C3CC3)c1C)=O)C2 c1(CC2(C)CC2(F)Cl)nc(-c2ccccc2Br)nn1CCCCO N1(C(c2ccc(C(=O)OC)c(Br)c2)=O)CCC2CN(C(c3occc3Br)=O)CC12 C1(NC(c2cc(Cl)ncc2Cl)=O)CCCC2CN(C(=O)C=Cc3cnc[nH]3)CC12 N1(C(c2nc(CC)oc2)=O)CCCC(C)(C)C1C(=O)NC1C2CCCOC12 N1(C(C2(C)CC2)=O)CCN(C(C2CC2Sc2ccccc2)=O)CC(O)C1 c1(C(=O)NC(C2CCCN2C(C2CC=CC2)=O)C)cc2cc(Cl)ccc2o1 c1(C(N2CCC(C)(NC(CCN(C(CCC)C)C)=O)C2)=O)ccc(N)c(C)c1 C(C(N=c1[nH]c(C(F)F)nc(=N)[nH]1)C(C)C(C)C)NC(C1N(C(C)=O)CCC1)=O CCCCC(C(=O)N(C(C)CN(C)C(c1csc([N+](=O)[O-])c1)=O)C)N(C)C C(CCC(C)C(=O)NCC1CC2(CC2)CN1C(c1ccoc1C)=O)OC c1(C(=O)NC(CNC(CCCCN(C)C)=O)(C)CO)nn2cccnc2c1Cl c1(N2CC=C(CNC(C3C(C)(Br)C3)=O)CC2)ncc2ncnc-2[nH]1 CC1=NOC2(CCN(C(c3coc4ccc(Cl)cc34)=O)CC2)C1 Cc1ccc2cc(C(=O)NCCOC(=O)C3CC3)cnc2c1 c1(C(=O)NC(C2N(C(CCC=C)=O)CCC2)C)cc2c(cnn2C)nc1O N1(C(CC2(C)CC2)=O)CCC(CCCCCNC(=O)CSc2nncs2)CC1 CC1CCC(CNC(=O)CCOc2cccc(F)c2)N(C(=O)CC2CC2)C1 c1(C(=O)NC2CCC2NC(C23CC(O)C2C3)=O)cnc(O)c(Br)c1 N1(C(C2CN(C(C)=O)C2)=O)CC=CC(C(=O)NC2C(O)CC2O)C1 CCC(N=c1ccnc(CN2CCC(Oc3ccncc3)C2)[nH]1)c1ccncc1 C=CC1(C(=O)NCC2(CNC(=O)CC3CCOC(C)(C)C3)CCC2)CCOCC1 c1(C(=O)NCC(C)(O)CNC(=O)CCC(N)=O)ccccc1O N1(C(CNC(CNC(C)=O)=O)=O)CCCC12CCN(C(C1CCCOCC1)=O)C2 c1(C(N(CCCn2cc(CCN(C)C)nn2)C)=O)c[nH]c2cccc(F)c12 N1(C(CCCCOCC)=O)CCC(NC(c2cc(C3CC3C)on2)=O)C(O)C1 C(=O)(C(C)(CO)NC(=O)COC1CCCCC1)NC(C(=O)NC(C)C)C c1(OC)cccc([N+](=O)[O-])c1C(N1CC(NC(c2cncs2)=O)C(C#N)C1)=O c1(-c2n(CC(=C)C)c(N3CCC(CCCC)C3)nn2)nc2cc(C)ccc2o1 Cc1cc(CN(CC(C)C)C(=O)NCC2CC23CC3)n(C)n1 S(=O)(=O)(c1c(F)cccc1F)N1CCC(C#N)(NC(C2CCC(=O)NC2)=O)C1 C1(NC(C(c2n(CC)ncc2)=O)=O)CN(C(=O)CCSC)CC2(CC2)C1 c1(C(=O)NC2CC(NC(C3C(c4nc(C)[nH]n4)C3(C)C)=O)C2)cnccc1C c1(NCC(=O)NC(C)CN(C)C(c2csc(O)n2)=O)ccc(C(F)(F)F)cn1 c1(CC(=O)N(CCN(C(COCC(=O)OC)=O)C)C)cnc2n1CCCC2C C1(NC(c2ccc(C(F)F)nc2)=O)CCN(C(C2C=CCCC2)=O)C12CCCC2 N1(C(CC(CC)C)=O)CCC(F)C(NC(=O)CCNC(=O)Cc2ccccc2)C1 N1(C(C(CSC)(C)C)=O)C(CNC(=O)C(F)(F)C(C)(C)O)CC2COCC12 C1(O)(CN(C(C(COC)(C)OC)=O)C)CCCN(C(=O)C(=Cc2cnc[nH]2)C)C1 N1(C(C=NOC)=O)CC(=O)NC2CN(C(c3cnn(CCC(F)(F)F)c3)=O)CCC12 c1(C(=O)NC2(CCCNC(C(C)CC(F)F)=O)CC2)cc(O)c2ccoc2c1 CCCCCCC(C)CC(=O)N1CCN(C(=O)CNC(=O)OC)CC1C(C)C C(=O)(C1=CC(C)(CC)C1)N(CC(=O)N(CCC)CCN(C)C)CC1CC1 Cn1nc(Br)c2ncnc(N3CC4CC3CCC4NC(=O)C(C)(C)C)c12 c1(OCCC(=O)N(CCC)CCCN)ccccc1OC.c12cnc(s1)s2 C1(NC(CSCC(C)C)=O)COC2(CCN(C(c3cc(Cl)cc(F)c3N)=O)C2)C1 C1(C#N)(Cn2c(N3CCCC(c4onc(C)n4)C3C)nnn2)CCS(=O)(=O)CC1 Cc1nc2c(C)cc(C(=O)NC(C)CCN(C(=O)C(O)C3CCCC3)C)cn2n1 c1(OC)cc(OC)c(CNc2cn(C)c(C(N3CCC(CO)C3)=O)n2)c(O)c1 N=c1ccc(C(=O)NCC(O)CNC(C2(CC3CCC3)CC2)=O)n[nH]1 c1(NC(=O)Oc2c(Br)ccc(OC)c2)ccc(F)c(Cl)c1C c1(NC(CC2C=CC(NC(C(n3ncc(C)c3)C)=O)C2)=O)cnc(C)nc1C C(CCCCC(=O)NCC1CCCOCC1)N(C)C(c1cc(O)cs1)=O c1(OCC)cc(C(N2CC(NC(=O)C3CC3)C(c3cncn3C)C2)=O)ccn1 c1(C(=O)NC2CC(F)(CNC(c3cnc(O)o3)=O)C2)c[nH]c2nc(Cl)ccc12 CCCCC(O)CC(=O)NCC1(NC(=O)CNC(=O)OCC)CCC1 C1(CCC(=O)N(CC(C)NC(CN2CC(C)C2)=O)C)CCCN(C)C1 c1(N(C(CCSCC)C)C)[nH]c(=NCC(C2CCC2)C2CCC2)nc2sccc12 C1(C(=O)NC2CC3CN(C(C(C)OCCC(C)C)=O)CC32)CCS(=O)(=O)C(C)C1 C1(C(=O)NC2(CNC(C3CCS(=O)(=O)C3)=O)CCOCC2)CN2CCC1CC2 C1(C(=O)NC(CCN(C(=O)Cc2c(C)n[nH]c2C)CC)C)CCc2n[nH]cc2C1 N1(C(C2CC(C)(F)C2)=O)CCCC(F)(CNC(C2CCC3CCC2O3)=O)C1 C12(NC(c3c(Br)c(C)n(C)n3)=O)CCCC1CS(=O)(=O)C2 C(C)(CCCCCO)NC(C(Cn1ccnn1)NC(CSCCOC)=O)=O N1(C(C=CC2N(C(CCCN=[N+]=[N-])=O)CCC2)=O)CC2CCCC2(CO)C1 C#Cc1ccc(CC(=O)N(C(C)CCNC(=O)CC2CCC(C)(C)O2)C)cc1 CCCC(C)(C)CC(=O)NC(C)(C)CNC(c1ccnn1C(F)F)=O c1(CC(=O)NCC(C)NC(C(CCC)C#N)=O)cc(Cl)c2c(c1)OCCCO2 c1(CNC2CC(NC(c3cc(Cl)c(Cl)c(Cl)c3)=O)C2)ccc(F)c(F)c1F c1(Cc2nc(C3N(C)CCOC3)on2)nc2c(s1)COCC2 c1(NCC2(CN)COC2)cc(OC(=O)C2CC2)cc(Br)c1 c1(C(=O)NC(CCCC)CNC(=O)C(C2CCCCC2)O)cc2cn[nH]c2cn1 C1(CCC)CN(C(=O)CCC2CCCC2)CC1NC(C1(n2cnnn2)CC1)=O O=C1NCCN(C(=O)CC2CCCCC2NC(c2ccc(O)cn2)=O)C1CCO CC(CC(=O)N1CCC(CNC(=O)Cc2cccnc2O)CC1)C(C)(C)C C(C(O)C(=O)N1CC(O)(CN(C)C(C2(F)CCOC2)=O)C1)SC C12(CNC(c3c(C)oc(C4CC4)n3)=O)CCC(C1)N(C(C1CC(C(C)C)C1)=O)C2 N1(C(Cn2c(C)cc(C)n2)=O)CC(CNC(c2[nH]c(O)nc2C)=O)C(F)(F)C1 n1(CC(=O)NCC(CC=C)NC(=O)CC2CCN(C)C2)cc(C#N)c(O)nc1=O N1(C(C(CC)O)=O)CCN(C(c2cccc(C)c2Br)=O)CC1CC(C)(C)C CC1CCC(CC(=O)NC2(C)CC(C(=O)NCC(CO)C3CCC3)C2)O1 c1(OCC)ccc(C(=O)NCC(CO)NC(=O)CCCn2ccnc2C)cc1C Cn1nccc(C(=O)NC2(CO)CCN(C(=O)Cn3nnc(=N)[nH]3)CC2)c1=O CC(C)C(F)(CNC(C1CCCC(=O)C1)=O)C(=O)NC1COCC(C)(C)C1 c1(C(=O)NC2C(SCC)C2)cc(F)cc(Br)c1C.C12(CCCC1)C(=O)N2 c1(OC)ncc(F)cc1C(=O)NC1CCN(C(=O)CC(C)C(F)F)C1(C)C C1(C2CC2)(CNC(C2CC(C)OC2)=O)CCN(C(=O)C(F)(F)CC2CC2)C1 N1(Cc2sc(C)c(Br)c2)CC2C(C1C(N1CC(C)C1)=O)C2(C)C C1(NC(CC(C=C)CC)=O)CN(C(=O)Cn2cc(C(C)=O)nn2)CCC12CCC2 S(=O)(=O)(c1cc(C)ccc1-c1ccccc1)N1C(CCCC)CCCC1 c1(C(=O)NCC2(F)CCC(NC(C=CC(C)(C)SC)=O)C2)ccc(O)c(F)c1F c1(OC)cc(F)c2c(C(=O)NCCCC(C)NC(C3CCC(=O)C3)=O)n[nH]c2c1 C(CS(=O)(=O)CC(F)(F)F)NC(NC(CC)C)=NCCNc1ccc(F)cc1Cl S(=O)(=O)(c1ccc(C(N2CCCC2(C)CNC(=O)C2=CCCC2)=O)o1)N(C)C c1(NC)ccc(C(=O)NCC2(CCNC(=O)COCc3scnc3C)CC2)nc1 CC1CCC(C)N(C(=O)NCCN2CC(c3cc(O)n[nH]3)C2)C1 Cc1ccc(C(N2CCCC(CNC(C3CCS3(=O)=O)=O)C2)=O)cc1S(C)(=O)=O C1(C(N(C)CC2CCCCN2C(c2nccs2)=O)=O)COc2ccc(O)cc2O1 c1(C(=O)NC2(C)CC(NC(COC3(C#C)COC3)=O)C2)cnc2ncccc2c1 c1(OC)nc(C)ncc1C(=O)NC1CC1NC(C1OCCCO1)=O c1(OC)ncc(Cl)c(=NCC2CN(C(=O)C(C)(C)CN(C)C)CCCO2)[nH]1 C1(NC(c2c(OC)csc2)=O)CC(CC(=O)N(C)Cc2cc(C)nn2C)C1(C)C c1(NCCc2cnc(NC(C(CCC)C)=O)s2)c(Cl)c[nH]c2nccc1-2 c1(C(=O)NCCNC(c2c(CCC)onc2C)=O)cc(F)c2c(c1)CCC2 C#CCC(O)C(=O)NC1COCC1CNC(c1sc(C)nc1C)=O C1(N(C(C=NOC)=O)C)CN(C(c2cc(Br)c(C)o2)=O)CC1(C)C c1(C(=O)NCC2(O)CN(C(CCSCCCC)=O)C2)ccc2cc(O)ccc2c1 S(=O)(=O)(c1ccc(=NCCC2COC(C)(C)O2)[nH]c1)N(C)CCO CCCCCCCc1cn(C2CN(C(C34CCCCC3C4)=O)C2)nn1 c1(COC)nccc(=NC2CC(NC(C3CC(C)OC3C)=O)C2(C)C)[nH]1 C1(NC(N2CCCN(CC)CC2)=O)CC2CC(C1)CC(F)(F)C2 C1(NC(C2CC(O)CN2Cc2ccc(OCCO)cc2)=O)CCC(F)(F)C1 Cc1cc(=NC2CCCC(C(F)F)CC2)[nH]c(NCc2nccn2C(F)F)n1 C1(CCC(=O)O)(NS(=O)(=O)Cc2ccon2)CCOC1 N1(C(CC2C=NN(C)C2=O)=O)CCC2CCN(C(=O)C=Cc3cn[nH]c3)CC12 C(C)(CCC(=O)NCCC1CN(C(=O)CN2CCC(=O)CC2)C1)SC c1(C(N(CCNC(c2c(OC)cccn2)=O)C2CC2)=O)sc2nccnc2c1N c1(C(=O)NCC(C)(C2CC2)NC(C(CC(C)C)F)=O)occ2c1CCOC2 c1(CC(c2ccn(C)n2)NC(N2CCOCC2CC(F)F)=O)cccc(Br)c1 C1(C)(NC(C(C)(C)CF)=O)CCN(C(C2CC(O)CN2C(N)=O)=O)CC1 N1(C(c2ccc(C)s2)=O)CCCC(N2CCN(C(=O)C(F)(F)C3CC3)CC2)C1 c1(C(=O)NCCCCCN(C(CC(C)OC)=O)C(C)C)c(C)[nH][nH]c1=N C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCC1N(C(CC(=C=C)C)=O)CCC1 c1(C(c2n(CCOC)nnn2)NCCc2ccc(Br)cc2)nc(OC)ccc1F CC(C)C(CC(=O)N=c1cc2c(Br)cccn2[nH]1)c1ccon1 C1(CNC(c2cc(Cl)ns2)=O)CN(C(=O)Cn2cccnc2=O)CC2(CCC2)O1 N1(C(C(CSCCN(CC)CC)F)=O)CCOC2(C1)CN(C(c1ncsc1Br)=O)C2 CC(CCC(C)(C)C)C(=O)NC1CC(CN=c2[nH]nco2)C1 C(=O)(CCCCNC(c1ccccc1OC)=O)N(CCC(=O)OCC)CC c1(C(C)OC)nc(C(=O)NCC2CC(NC(C3CC3(F)Cl)=O)C2)cs1 C1(C)(NC(C(C2CCCCC2)C)=O)CC(NC(C2CCC2(C)C)=O)C1 c1(C(=O)NC(C2CCN(C(=O)C=CSC)C2)CC)cc(-c2ccccc2)[nH]n1 c1(OC)cccc(CC(N2CC(CNC(=O)C=Cc3ccsc3)C3CC23)=O)c1 C1(C(N(C2CCN(C(c3ccc(C)c(O)n3)=O)C2)CCC)=O)CCCCNC1=O Cc1ccc(NC(=O)C(C)OC2COC2)c2nccn12 C=CC(C)N=c1[nH]c(N(CC(C)COCCOC)C)nc2c1CCCC2 c1(C(c2n(CCSC)nnn2)NCCC(F)(F)F)ncc(C)n1C c1(NC(CNC(CN(c2ccnc(CO)n2)CC)=O)=O)ccc(OC)cc1 c1(OC(CN2CCN(CCOC)CC2)=O)ccc(Cl)cc1NC(=O)OC(C)(C)C C1(C(=O)NCC=CCCOC)CN(C(C2C3CC(=O)CC23)=O)C(C)(C)C1 c1(N(C(=O)CC2(NC(=O)C(C)NC(C)=O)CC2)CC#C)ccc(OC)cc1 Cc1sc(C)c(C(=O)N(CC(C)(C)NC(=O)CCc2ccc(C#N)cc2)C)c1C N1(c2cc(N3CCC(CN(CC=C)C)CC3)ncn2)CCC(C)(C2CC2)C1 N1(C(c2c(C)nccn2)=O)C2CCC1CC(CCNC(C1(C)C=CCCC1)=O)C2 C12CCN(CC1C)C(=O)C(=O)N2.n1(C(C)C)cnc(C(N)=O)c1 n12c(nnc1N(C)OC1CCCC1)C2C1CC1.Cc1cc(C)n(CCOCC(C)C)n1 CCC(CC)(CCNC(=O)C(F)C1CCCC1)NC(=O)CCC#N C1(C)(NC(C(CC=C)CNC(c2ccccc2CC#N)=O)=O)CCC(=O)NC1=O c1(C(N(CC(C)N(C(c2c(C)nc(CO)o2)=O)C)C)=O)ccc2occ(C)c2c1 n1(CCCC)cc(C(N2CC(CNC(c3ccn(C)c3)=O)C(O)C2)=O)c(C)n1 n1(CC)nnc2c1C(C(=O)NC1CC(F)C1)CN(C(=O)CCN1CCOC1=O)C2 C(=O)(C1=CC2(CN(C(c3cnnn3C3CC3)=O)C2)OC1)NCC(CC(C)C)OC CCCCCCC(=O)NCCCC(O)C(=O)NC1CN(C)CC(O)C1 Cc1cccc(C)c1C(=O)NC1CCCCN(C(C2CC3CCC(C2)O3)=O)C1 c1(SC)ccc(C)c(C(=O)NCC2CC2CNC(C2CCC(C)C2)=O)c1 CC1=C(C(=O)NC2CCCC2NC(c2cc(C)sn2)=O)C(C)(C)CCC1 N1(C(C2N(C)C(=O)OC2)=O)CC(O)C(O)C1CNC(c1ccnc(C(F)F)c1)=O c1(C(=O)NC(C(C(C)C)NC(=O)CN2CCC(C)(C)C2)C)c[nH]cc(Cl)c1=O C1(C(=O)NCCNC(Cc2c(C)cnn2C)=O)CN(C(=O)OC(C)(C)C)CCN1C C1(C(N(CC(C)C#N)C2CC2)=O)CC(NC(=O)Cc2ccn(C)n2)CCO1 c1(C(=O)NC(C2CN(CC3CCCC4CC34)C2)C)cccc(C2CC2)c1 C1(C(=O)NC(C)(CNC(c2c(F)cccc2Cl)=O)C2CC2)CC(C2CCCC2)C1 N1(C(=O)C(N2CCC(O)(c3ccccc3Cl)C(O)C2)=O)CCCC2(CC2CO)C1 CCC(C)(C(=O)NC1C2CC(NC(=O)C#CC(=O)N(C)C)CC12)C(N)=O C#Cc1cc(C(=O)NC2CC(CNC(=O)CSc3ccc(F)cc3)C2)cc(N)c1 C1(C(C)NC(c2cc(CC)[nH]n2)=O)CN(C(=O)CC2C=CCCC2)CCO1 Cc1cscc1C(=O)NCC(C)(CO)NC(=O)Cn1nnc(C2CC2)n1 c1(OC)ccccc1CN1CC(NCCCN2CCCC2=O)C1 Cc1cc(C(=O)NCCC(C)NC(C2COCCN2C)=O)nn1CCO S(=O)(=O)(c1ccc(OC)cc1OCC1CC1)NC(CC=C)COC C#CC1CCN(C(=O)CCN(C(=O)CCCOCCN(C)C)C2CC2)C1 c1(CC)nc(Cl)[nH]c(=NCCC2CCCCN2C(c2ccc(C)cc2)=O)c1Cl C(c1cnc(C(C)(C)C)s1)=CC(=O)NC1CC(F)(CNC(COCCCC)=O)C1 C1(NC(=O)COCC2CN(C(N3CCCC3)=O)CCCO2)CC2(COCCO2)C1 N1(C(C(C)(C)SC)=O)CCC2CCN(C(C3(C)CC4CCC(C3)S4)=O)CC2C1 N1(C(Cn2ncc(C(C)=O)c2)=O)CCN(C(c2cnc3sccn23)=O)CCC1C C(N=c1[nH]c(=N)[nH]c(=NC2CCOC(C)C2)[nH]1)c1ccc(S(=O)(=O)NC)cc1 Cn1ccc(S(=O)(=O)NC2CC2C(=O)Nc2ncc(Br)cc2F)n1 CCCCCCCCOCC(=O)N(CCNC(C1ON=C(C)C1C)=O)CC N1(C(C(CSC)C)=O)CCCC(N(CCO)C(c2cn(C)[nH]c2=N)=O)C1 C1(C(=O)NCc2c(C(=O)NC(C)Cc3ccoc3)con2)CC2CCC(C1)C2 C1(NC(CCC=C)=O)CC1C1CCN(C(C2CC(c3ccccc3)=NO2)=O)CC1 CCC(O)C(C)(C)C(=O)NC(C)CN1CCN(C(=O)CC2(CC(=O)OC)CC2)CC1 C#CCC(CC(F)F)C(=O)Nc1cccc(C(=O)NCCCCOC)c1.C(CC)=C N1(CC(=O)NC2CC(NC(C3(CCC)CCC3)=O)CC2O)CCc2sccc2C1 Cc1oc([N+](=O)[O-])cc1C(N1CCC(NC(C2CCCS2(=O)=O)=O)C12CC2)=O c1(C(N2CC(CNC(=O)CC3(N4CCCC4)COC3)C2)=O)cncc(F)c1 Nc1ccc(C(=O)NCC2(Cc3cn(CCCF)nn3)CCCCC2)c(F)c1 c1(OC)ccc(F)cc1C(N1CC(NC(C2CCS(=O)(=O)N2)=O)C2(CC2)C1)=O C1(NC(c2cccc(OC(F)(F)F)c2)C)COCCC1c1ccccc1 C1(NC(=O)NCC(COC)COC)C2C3CC4C5CC(C1C35)C4C2 N1(CC(=O)NCC(N(C(C(=O)NCCOC)=O)C)C2CC2)CCCCC(O)C1=O C1(C(=O)NC(C(=O)N(CC)CC)C)COCCC1NC(c1ccnc(OC)c1)=O N1(C(CCC#C)=O)CCC(c2nnc(CNC(=O)Cc3scnc3C)s2)CC1 C1(NC(c2ccc(C(=O)OC)cn2)=O)CC2CC(C1)N(C(c1cn[nH]c1)=O)C2 C(=O)(CCCCCc1ccccc1)N1CCCC(NC(C(C)O)=O)C1 C(N=c1[nH]cncc1I)C1CCCN(C(CCOCC#C)=O)C1 C#CC1(C(=O)NC2CCCC2NC(=O)CNC(=O)NCC(F)(F)F)CCC1 c1(C(=O)NC2CN(C(C(=O)N(C)C)=O)CC(O)C2)ccnc2[nH]c(C(F)F)nc12 C1(NC(=O)C2CC2)CN(C(=O)CCCc2cccc(Br)c2)C2(CCOCC2)C1 C12CCN(CC1)C(=O)N(CCCCO)C(=O)C2.C1(NCC)CS(=O)(=O)C1 n1(CC)cnc2c(N3CCC4(CC(OC)C4)C3)nc(=NCC(C)CN(C)C)[nH]c12 C1(NC(CCC=C)=O)CN(C(C2(CCc3ccccc3)CC2)=O)CC12CCC2 Nc1cc(F)cc(C(N2C3CCC2C(CNC(=O)Cc2cncnc2)C3)=O)c1F CC(c1ccccc1F)=CC(=O)N(c1cc(Cl)ccc1Cl)C1CC1 C(=O)(C1COc2ccccc21)NC(CC=C)CNC(C1CCC(C)CC1)=O C=C(C)CC(C)C(=O)N1CCCCC(CNC(=O)CC(C)(C2CCC2)N(C)C)C1 N1(C(c2n(C)ncc2)C(=O)NCc2ccccc2Br)CCSCC1(C)C c1(NC)cnc(C(N2CCOCC2CNC(c2ncsc2C(C)C)=O)=O)cn1 c1(COC(N2CCC(N(C)C(C3(Nc4ccccc4)CC3)=O)C2)=O)ccccc1 Cc1cc(C(c2nnnn2CCCF)NCCCC(C)(C)C(N)=O)c(C)s1 Cc1cccc(C)c1C(O)C(=O)NC1CCN(C(c2c(C)noc2C)=O)CC1O c1(OC)ccncc1CC(=O)N(C1CN(C(=O)CC(=O)NC2CC2)C1)C C(C(O)C(=O)N1CCCC1CN(C(=O)CN(C)C1CC1)C)OC C1(C(N(C2C(C)C2)C)=O)CCCN1NC(=O)C(=O)C1CCOCC1 C1(C(N2C(C)(c3ccccc3)CC(O)C2)=O)COC2C(O)COC12 CCC(F)(F)C(=O)NCc1ccc(C(=O)NCCCS(N)(=O)=O)s1 C1(C(C)NC(=O)C#CC(C)(C)O)CC2CCC(C1)N2C(=O)CCC(F)(F)F N1(C(COC2C(C)C2)=O)CC2(NC(c3cccc(-c4nccs4)c3)=O)CC1C2 C1(CN(C(C(C)CO)=O)C)CCCN(C(C2(n3cccc3)CCCC2)=O)C1 c1(NC(c2c[nH]nc2OCC(F)F)=O)cccc2nc(-c3cccnc3)[nH]c12 C(=O)(C1=CCCN(C(c2ccc(Cl)s2)=O)C1)N1CCC(O)(C(N)=O)C1 c1(C(C)(C)C)n[nH]c(=NCC2CCCC(NC(c3c(Cl)csc3Cl)=O)C2)s1 N1(C(c2c(CC)cccc2C)=O)CCC(C)(C)C(CNC(=O)CC(O)C(C)C)C1 C12(C(N3CCCC(N(C(c4cncc(C=C)c4)=O)C)C3)=O)CCC(=O)N1CCS2 N1(C(=O)CC2(c3ccccc3)CC2)CCC(C2CCN(C(=O)C=C(Cl)Cl)C2)C1 c1(C(=O)NC(C(C)NC(=O)C2=NNC(=O)CC2)C)ccc2c(c1)CCCCN2 c1(C(=O)NC(C2CCCC2)CNC(=O)CC2CNC(=O)C2)nnc(O)cc1O c1(C(=O)NC(C=CC(=O)NCC(CSC)(C)C)C)cc(C)n(C(C)C)c1 c1(NC(CNC(CCCONC(C=CCC=C)=O)=O)=O)ccc(C)nn1 C1(CNC(c2sc(CC)c(C)c2)=O)(NC(=O)CCCCC#N)CCC(F)(F)CC1 N1(C(C2CC(CNC(C(CC)(C)C)=O)C2)=O)CCCC2(CCOC2)C1 c1(CC(=O)NC2CCC(NC(C(C)n3cncn3)=O)C2)cccc2cccnc12 c1(C(=O)NC2CCC(NC(c3c(C)snc3)=O)CC2)coc([SH](=O)=O)c1 CN1CCC(C2(C(N3CCC(c4ccccc4)(NC(=O)C(N)=O)C3)=O)CC2)CC1 C(CCC(C)(C)C(=O)NCC(C)C(F)C(=O)N(CC(C)(C)O)C)OC C1(COC)(CNC(=O)C=CCCC=C(C)C)CCCN1C(c1coc(C#N)c1)=O c1(-c2c(C)nn(C)c2)cnc2[nH]c(C(=O)Nc3ccc(C(C)C)c(Br)c3)cc2c1 CCC(C)(CO)C(=O)NCC1CCN(C(=O)Cn2ccnc2C)C1(C)C O=C1CC(CC(=O)N2CC(O)CC2CNC(C2CCn3cnnc3C2)=O)=NN1 N1(C(C(C)CNC(c2cccc(CO)c2)=O)=O)CC(CO)C(C)(C)C1 N#Cc1cnc(N2CCC3(CN(C(=O)Cc4cnoc4)CCO3)C2)c2sccc12 c1(OC)nc(Br)ccc1C(N1CCC(O)C1C(=O)NCc1nn[nH]n1)=O c1(C(CNC(=O)Nc2cnn(CC3CC3)c2)C(F)F)c[nH]c2c(Br)cccc12 N1(C(Cc2cc(OC)no2)=O)CCCC(F)(C(=O)NCC2(O)CCOCC2)C1 c1(C(=O)NCC(CC)(C)NC(c2ccc(O)cc2F)=O)c[nH]c(=O)c2ccsc12 Cc1cncc(CC(N2CC(O)CC2CNC(=O)CCC2OCCO2)=O)c1 Cc1cc(NC(c2cnn3c2OCC3)=O)ccc1NC(=O)Cc1ccsc1Cl c1(C(N2CCCC(NC(c3c(F)cc(F)cc3F)=O)C2)=O)scc2c1OCCO2 c1(C(N2CCC(C)C2CNC(C2(O)CC2)=O)=O)ccc2nccnc2n1 c1(CC)cc(C(=O)N(CC(C)NC(C2CC23CCC3)=O)C)c(C)nn1 N1(C(C=C(C)c2ccco2)=O)CCC2(CCC(NC(=O)CO)CC2)CC1 C(=O)(CCS(=O)(=O)C(F)(F)F)NC1CC(O)(CNC(C(CCCC)C(C)C)=O)C1 c1(OC)nc(C)ncc1C(N1CCCC1C(C)NC(c1sccc1C)=O)=O CONC(=O)C(=O)N(CC(=O)N(CC(C)C)CCO)C N1(C(c2cccc(COC)c2)=O)CC(NC(=O)C=CC(C)C)CC(C)C1 C1(C(N2CCC(CC=C)(NC(c3cc(C)oc3C)=O)C2)=O)CC2CC(=O)C1O2 C=CC1(C(=O)N(CC(O)CNC(c2nn(C(F)F)cc2Cl)=O)C)CCCCC1 O(NC(=O)C(C(C)O)NC(c1ccco1)=O)CC(=C)C C1(CC(=O)NCCN(C(=O)C(C)(C)N2CCCCC2)CC)COCC1O CC1(CNC(=O)CC2(C(F)F)CC2)CN(C(=O)CCCCc2cnc[nH]2)CCO1 C(=O)(C#CC1(C)CCCO1)N1CCN(C(C(CC)NC(N)=O)=O)CC1C C1(C(=O)NC(CC)CNC(c2[nH]ccc2C2CC2)=O)CC(=O)N(CC2CC2)C1 c1(OC)ccc2cc(C(=O)NS(=O)(=O)CC(F)(F)Cl)ccc2c1 c1(C(N2CCCN(C(c3cnn(CC)c3C)=O)CC2)=O)n[nH]c2ccc(F)cc12 N#CC1(C(N2CC3(CCN3C(=O)CCc3nc(O)n[nH]3)C2)=O)CC12CCC2 c1(OC)ccc(C=CC(=O)NC(C(C)NC(C2(O)CC2)=O)C(C)C)cc1F N1(C(C(CC=C)OC)=O)CCC(C2CCN(C(=O)CCCC3CCC3)CC2)C1 Cc1c(C(N2CC(F)(C(=O)NOCC(O)C(C)C)C2)=O)ncn1C C1(CC(=O)NCCCN(C(=O)CCc2nc(C(C)(C)C)no2)C)CC2CC2C1 Cc1cc(C(=O)N(C)CC2(O)CCN(C(=O)C(C)(C)N(C)C)CC2)cnc1C c1(C(N2CCC(N(C(C(CC)n3cccn3)=O)CC)C2)=O)ccc(Cl)c(O)c1 Cc1cnn(C)c1C(=O)NCC1C2CN(C(C3CC3c3cccs3)=O)CC12 N1(C(CCC(C)=O)=O)CC2CCC1C(CNC(c1ccoc1C)=O)C2 c1(C(=O)NCC2CC(OC)CN2C(c2cc(O)ncn2)=O)cc(F)cc(F)c1O c1(C(=O)NC2CCN(C(COC)=O)C2)cc(Cc2ccccc2)n(C(C)(C)C)n1 C12(C(N3CCC(O)(CC(C)C)C3)=O)CC(C)(CN1C(=O)CCC1CCCCO1)C2 C12(C(N3CCCC(CN(C(=O)C(F)C4CCCC4)C)C3)=O)CCCN(CC1)C2 CC#CC1CCN(C(c2cnn(CCNC(c3cccc[n+]3[O-])=O)c2)=O)C1 Cc1cc(C(=O)NC(C)CCN(C)C(c2ccnn2C)=O)c(C)cc1Cl Cc1c(N(C)Cc2cc(Cl)ncc2N)cccc1F N1(C(C(C)Cc2cnc[nH]2)=O)CCCC(N(C(=O)C(C)n2cnnn2)C)C1 N1(C(c2c(CC)n(C)cc2)=O)CC(NC(c2ccc(CO)c(F)c2)=O)C(C)(C)C1 Cc1ccc(F)c(C(=O)NC(C)(C)CCC(=O)NCC2CCN2C(C)(C)C)c1 C12(NC(CC3C(CC)C3)=O)CCC(CC1)N(C(=O)C(C)(F)F)C2 N1(CC)CCN(CC(N2CCCC(N(C)C(C3(C4CCCO4)CC3)=O)C2)=O)CC1 c1(CNC(=O)NC2CCC(C)C2)ccc(Cl)nc1 C1(CNC(C)=O)CN(C(C2CC(C)CO2)=O)CC1C Cc1cn2c(n1)C(CNC1(C)CCN(C(=O)CCC(=O)OC(C)(C)C)C1)CCC2 N1(C(c2c[nH]nc2-c2ccc(Cl)cn2)=O)CCCC(C2CC2(F)F)C1 c1(OC)cc(C)ccc1CN=C(NCCOCC(F)(F)F)NCC1CCC(C)O1 c1(N(C)CCc2cccs2)ncccc1S(=O)(=O)N1CCC(C)(CCO)C1 C1(O)(C(=O)NC(C(=O)NCCOCCOC)Cc2cn[nH]c2)CCSCC1 C1(=CC(=O)NC(C2CCN(C(=O)Cc3ccno3)C2)C)CCOCC1 c1(C(=O)NC2(CF)CN(C(CC3CCC(C)C3)=O)C2)cc(O)nc(O)n1 C1(C(=O)NC(C)CNC(c2ccc(CC#N)cc2)=O)Cc2nnsc2S1 C1(C(N(C(C)COC)CC=C)=O)CCCC1CNC(=O)C(C1(O)CCCC1)F c1(CC(=O)N(CCNC(C2CC23CCOC3)=O)CC)c(C)[nH]c2ccccc12 C1(C#CC(=O)NCCC(O)C(N2CCN(C)CC2C(C)C)=O)(CC)COC1 c1(OC)cc(C)cnc1C(=O)NC(C)(C)CCCNC(C1(O)CCSC1)=O C=CC1(C(=O)NCC2CCN2C(c2cc(OC)cs2)=O)CCC1 c1(C(N2C(CN(C)C(C3CC34CCOC4)=O)CCC2)=O)cccc(C#CCO)c1 N1(C(C(C2CC2)OC)=O)CC2(C1)CN(C(=O)CC1CCN(C)C1=O)CC2CO C(=O)(C(C)(C(F)F)c1ccccc1)NC(CC)C.C1(=O)C(C)(COC)CO1 c1(C(=O)NCCOCCCNC(C(COC)COC)=O)cc(C)c(Cl)cc1F c1(C(N(CC(C)(C)NC(=O)CC2CCCC(O)C2)C)=O)cc2c(F)cccc2[nH]1 C1(CN(C(C2COCCN2C)=O)CC)CCCCN1C(=O)CCCCOC c1(C(=O)NC(C)CCNC(c2c[nH]nc2CO)=O)cccc2cnsc12 C12(CNC(c3ccccc3O)=O)CC(NC(C3CC34CCC4)=O)(C1)C1(CCC1)O2 N1(n2cc(C)nn2)CCN(C(=O)Oc2ccccc2C)C(CO)C1.Cc1nnco1 C12(NC(CCC(C)=O)=O)CCC(C(=O)Nc3ccnc(Br)c3)(CC1)C2 N1(C(C(CCC)NC(C)=O)=O)CC(CNC(=O)C(C)C(O)CC)OC(C)(C)C1 c1(CCC(C2C3CCCC23)=O)cc(C(=O)N(C)C)no1.C1(COC)(CN)CC1 C1(C(=O)NCc2ncc(C(=O)NCc3cc(C)c(C)s3)cn2)CCC2(CC1)CC2 C(C(C)(O)CNC(C1(CO)CC1(F)F)=O)NC(COC)=O c1(NC(C2C=CCN2C(c2cnsn2)=O)=O)ccc([N+](=O)[O-])c2ccccc12 c12ccc(c(Cl)c1)S(=O)(=O)N2.C(CC(C)N1CCCC1)NC1C(CC)C1 C1(C(C(=O)OC(C)(C)C)N2CCC2C(N)=O)CCCC(CC(=O)NCC2CC2)C1 N1(C(C(C)=CCC)=O)CC(C(=O)NC(c2nn[nH]n2)C2CC2)C(F)(F)C1 N1(C(C(c2cccnc2)NC(C2C(CCC)C2)=O)=O)CCCc2occc2C1 N1(C(C(Cc2ccccc2)OC)=O)CCC(N(C)C(c2cnn[nH]2)=O)CC1 CC1CCC(CNC(c2cc(N)ccc2F)=O)N(C(C2CCC=CCC2)=O)C1 N1(C(c2c(C)ocn2)=O)CCC2C(NC(c3ccnc4[nH]cnc34)=O)C2CC1 C(N=c1[nH]c(=NC)[nH]c(=NCCCOC)[nH]1)c1ccc(NC(=O)NCC)cc1 C(CN=[N+]=[N-])(C(=O)OC)N(C)CC1(C(=O)NCC2CC3C=CC2CC3)CC(=C)C1 c1(N2CC(CC(C)NC(C3CC(=O)NC3(C)C)=O)C2)ncccc1S(C)(=O)=O C1(CN(C(C=CCCC)=O)C)CN(C(=O)Cc2cnc(C)nc2O)CC12CC2 C(=O)(C(COC)(CC)CC)N(CC(CNC(c1cnc(CC)nc1C)=O)O)C Cn1c(C(=O)NCC2(NC(=O)CCC3CCC(=O)NC3)CCOCC2)nnc1S N1(C(CCCS(N)(=O)=O)=O)CCC2(CC1)OCCC2NC(c1occc1Cl)=O C(=O)(C1=NOC2(CCOC2)C1)N1C2C(NC(c3c(F)cccc3F)=O)C(C2)C1 C1(NC(c2n(C)nc(CO)c2)=O)COC2(C1)CN(C(C1(F)CCOCC1)=O)C2 C12(CC(=O)NC)CCC(CC1)OC2.n12cc(cn1)C(=O)NCC1(CCC1)CC2.CO C(C(C)(O)CC(=O)N1CC=C(C(=O)NC(c2nccs2)C)C1)OC c1(C2(CC(N3CCOCC3)=O)CC2)cc(Cl)cc(Br)c1.C12CN(C1)C2=O C1(CC)COCCN1CC(C1(O)CCN(S(=O)(=O)CCOC)C1)(F)F c1(N(CCS(=O)(=O)NC)C)ccc(S(=O)(=O)N(C)OC(F)(F)C(F)(F)F)cc1F N1(C(c2cnn(CC)n2)=O)CC2CC1CN2CCc1ccc(C)cc1 n1(CC(=O)NC(C(C)NC(CC(=C)C)=O)(C)C)cccc(C)c1=O C12(C(=O)NC3CC(CNC(C(F)=C(C)C)=O)CC3O)CC3CC(CC(C3)C1)C2 Cc1[nH]c(C)c(C(=O)NCC2CCN(C(c3cc(N4CCCC4)ncn3)=O)C2)c1C Cc1ccc(C)c(OCC(N2CCN(C(=O)CC3CCCSC3)C(CO)C2)=O)c1 CC1CCc2nc(C(=O)NC3CN(C(c4cnc(O)o4)=O)C(C)(C)C3)cn2C1 c1(C(N2CC(NC(c3ccc(CN(C)C)[nH]3)=O)C(F)C2)=O)cccc(F)c1F CC(C)S(=O)(=O)CC(=O)N1CC2(CCN(C(=O)CC(c3ccccc3F)C)C2)C1 c1(C(CC)N(C2C3CN(C(=O)CCC(F)F)CC23)C)ccc(C)cc1 C1(C2CC2)(CNC(C(COC)O)=O)CCN(C(c2c(C)ccn2C)=O)C1 O=C(C1CSc2ccccc21)N1CCN(C(C2CC3COCC(C2)C3)=O)CC1 CCC(C)C(O)C(=O)NCCC(=O)NCc1cnn[nH]1 Cc1nn(CC(=O)NCc2cc(C(=O)NCC3(C)CC3(F)F)on2)c(=O)o1 c1(C(N2CCC(O)(C(C)NC(C(CC)N(C)C)=O)C2)=O)cc(O)c2ccoc2c1 c1(CNC(C2C(OC)C2)=O)ccc(C(C)NC(c2cn(C(C)C)cc2C)=O)cc1 S(=O)(=O)(c1ccc(C)cc1)NCC(=O)NCC1CCCN(C(C=CC=CC)=O)C1 C(=O)(C(CO)C(F)(F)F)NC1(C(N2CCN(CCOC)CC2)=O)CC(F)(F)C1 c1(OC)cc(CNCC(c2ccc(Br)cc2)O)c(O)c(Br)c1 c1(C(=O)NCC2C(NC(c3nccc(N)c3)=O)CCC2)cc2cnc(Cl)cc2s1 N1(C(C(C(C)C)N(C)C)=O)CCCCC(CNC(=O)C(F)(F)Oc2ccccc2)C1 N1(C(C(C)SCCCC)=O)CCCC(C)(NC(c2cnn(C)c2F)=O)C1 c1(CNC(c2ccccc2OC(F)(F)F)CC(=O)OC)c(Br)nc(C)n1C N1(C(CN(C2CCSC2)C)=O)CCOCC1CNC(c1cc(Br)n(C)c1)=O C(=O)(CC(c1ccccc1)NC(=O)CN(C(=O)C(C)(C)C)C1CC1)OC c1(OC)ncccc1NC(=O)CC1CCCN1C(C1CC(C)CCO1)=O CCCC(F)C(=O)N1CCSCC1C(N1CCC(N2CCCC2)C1)=O N1(C(c2cc(C)cc(Br)n2)=O)CC(C)Cc2cc(C(F)(F)F)cc(Cl)c21 C(CC1CCOCC1)(C(=O)NCC1(NC(=O)CC2CCCO2)CC1)N(C(C)=O)C N1(C(C(C(C)C)SC(F)F)=O)CCC(C2CC2)C1C(=O)NC1CC(CN(C)C)C1 C[S+](C)CCC(O)C(=O)N1CCCC(C)(CNC(=O)CC2CCOCC2)C1 C1(NC(C2(C)N(C(c3ccc(OC)nn3)=O)CC(O)C2)=O)CC2(C1)CC(C)(C)C2 c1(C(=O)NCCN(C(c2ccccc2N=[N+]=[N-])=O)CC)cc(F)c(F)cc1C C1(C(=O)NC2CN(C(c3ncc(OCC)nc3)=O)CC2O)CC(C)(C)OC1(C)C N1(CC(C2CCOCC2)N(CC)CC)CCCC1CCn1cc(CC2CC2)nn1 n1(CCC#N)c(N2CCOC(n3cncn3)C2)nnc1-c1cccc(Br)c1 Cc1ccc(NC(=O)C(C2CCCO2)NC(c2ccc(C#N)cn2)=O)cc1C N1(C(CCC2(C)CN(C(C(C)C#N)=O)C2)=O)CC(O)CC1(C)C1CCC1 C(CCN=c1[nH]c2ccc(F)cc2s1)NC(CC1(C(=C)F)CCC1)=O c1(NC(=O)NCCCc2c(C)ccnc2)cnc(Cl)c(C(F)(F)F)c1 C12(C(=O)NC3C4CN(C(c5cn(CC)nc5)=O)CC43)CC(C1)C(C)(C)O2 C1(NC(C=CCOC)=O)CCN(C(=O)Cc2cc(-c3ccccc3)oc2C)C(C)C1 C1C(C)(C)CCN=C(NC(C2CC2)C2CC2)N1.C1CCN(S(C)(=O)=O)C1.CO C1(N(C(CS(CC)=O)=O)C)CC2CCC(C1)N2C(=O)CC1CCC2(CC1)COC2 c1(CNC(C(C)=C2CC2)=O)c(C)nn2c1CN(C(=O)Cc1cccnc1Cl)CC2 Cc1cccc(F)c1CC(N1CCC(CF)(NC(=O)CCNC(N)=O)C1)=O N1(C(C(C=C)OC)=O)CCC(C)CC1CNC(=O)C(C)O C=CCCC(C)(C)CNC(C1C=CCCN1C(=O)Cn1cnnn1)=O c1(C(=O)NC(CNC(c2c(C)c(C3CC3)on2)=O)C)c(C(F)(F)F)cc[nH]c1=N c1(CN(C2CCCCC2)C(CC2CC(CC)C2)=O)ncncc1C(=O)OC Cc1oc([N+](=O)[O-])cc1C(=O)NCC(O)CNC(=O)C(C(C)C)N(C)C C(C(C(=O)N1CCCCC(CO)C1)C(C)C)NC(CCCSC)=O c1(OC)cc(C(=O)NC(C(=O)NOCC(C)C)c2ccco2)ncn1 c1(SCC(=O)NCC(Cc2ccccc2)N(C(CC=C)=O)CC)ccccc1O Cc1nnc(CC(=O)NC(C2CCN(C(C3(O)CC3)=O)C2)(C)C)s1 c1(CC)cc(C(N2CCN(CC)CC2)C(=O)NC(C)C(=O)OC)ccn1 C1(OC)CCCC1C(=O)NCc1cn(CCN(C)C)nn1 Cc1cc(C(N2CC3CC(NC(c4cnc5n4CCS5)=O)C2C3)=O)cn(C)c1=O c1(C(N(CCC(C)NC(CC(C=C)CC)=O)C)=O)c(C)ccc2c1CCCN2 N1(C(CCC=CC)=O)CC(NC(c2cc(OC)n(C)n2)=O)C(CCC)C1 c1(C(=O)NCC2CCCN(C(CC(C)(C)O)=O)CC2)cnc2n(c1=O)CCS2 C1(C(N2C(C)C(NC(C3CN4CCC3CC4)=O)CC2)=O)Cc2nn[nH]c2C(C)C1 C(CC(=O)N1CCC(O)(C(C)NC(C2COC(C)(C)C2)=O)CC1)(C(F)(F)F)OC c1(C(=O)NC2C(CNC(CCc3cc(C)no3)=O)C2)c(C)ccn1C c1(C(N2CC3CC(NC(Cc4c(C)ncs4)=O)C3C2)=O)nccc2cccnc12 N1(C(C(CC)(C)O)=O)CCOC2(CCN(C(c3cn(C)nc3SC)=O)C2)C1 CCCCCS(=O)(=O)CC(=O)NC1CCCN(C(c2cc(=O)n(C)o2)=O)CC1 c1(C(=O)NCCCN(C(C2CCC(C)O2)=O)C2CC2)cc(=O)c2ccncc2o1 c1(OC)cc(C(N2CC(CCNC(c3cnc(Cl)[nH]3)=O)OC(C)C2)=O)ccc1Cl C1(C)(C(=O)NCCCC(C)NC(=O)CN(C)S(=O)(=O)N(C)C)CCCCNC1=O C1(CC)CCOC1C(=O)NC1(C)CN(C(C2CN(CC(C)C)C2)=O)C1 C#CC1CC2(CC2)CN1C(c1ccnc(C(F)F)c1)=O c1(C(=O)OC)ccc(O)nc1N1CCC(CF)(NC(=O)CCCCCO)C1 c1(CCC)nc(C(=O)NCC2(NC(C3C=CCCC3)=O)CCCC2)co1 C(C1CCC(C2OC(N)(C)CC(C(=O)NNc3cc(C)ccc3F)C2)O1)=C(C)C C=CC1(C(=O)NCc2[nH]ncc2C)CCN(C(=O)CCn2ccnc2)CC1 C1(C(CC)C)CCN(C(c2cncc(OC)n2)=O)CC1.C12CCCCC1NC2=O c1(CCC(=O)N(C2CCN(C(=O)C(C3CC3)OCC)C2)CC#C)ccc(C)cc1 N1(C(CC(CC#C)NC(c2sccc2OC)=O)=O)CCC2(CC1)CC(O)C2 C1(CNC(c2c(C(C)C)occ2)=O)CC(C(=O)NC(CN(C)C)CCO)=NO1 N1(C(c2cc(SC)oc2C)=O)CCN(C(c2cnc(Cl)s2)=O)CC1CF C(=O)(CC1=NN(C)C(=O)C1)N1C(C)CN(C(c2cc(F)c(F)cc2F)=O)C(C)C1 c1(C(=O)NC2C(C(=O)NCCc3c(OC)cccc3)C2)cn2ccc(Cl)cc2n1 C(=O)(C1NCCc2c1ncn2C)N1CCC(C(C)=O)CC1.CCSC C1(CNC(=O)C(O)Cn2cncn2)CN(C(c2sc(F)cc2Cl)=O)CCO1 N1(C(CCCOC)=O)CCC(C)(C)C1CNC(c1cc(C(F)(F)F)nn1CC)=O CC1CC(NC(=O)CC2OCCC2C)CN1C(=O)Cn1cc(CO)nn1 CN1CC2CCN(C(=O)C(c3cccnc3)NC(c3c[nH]c(=N)o3)=O)CC2C1 c1(-c2ccc(NC(Cc3cc(C(=O)O)on3)=O)cc2)ccc([N+](=O)[O-])cc1 N1(C(c2cc(OC)nc(Cl)c2)=O)C2CCC1CN(C(c1nc(C)c(C)s1)=O)C2 c1(C(=O)NC(C)CCNC(=O)CC2CCC(O)C2)cccc(C(N)=O)c1 c1(C(=O)NCC2CCN(C(c3occ(C)c3)=O)C2)ccc(N)c2ncccc12 N1(C(C2C(C)CC(=O)NC2)=O)CC2CCC(C(=O)NCC=C(Cl)Cl)(C2)C1 CCC1=NOC(C(=O)NC2CC(c3ccccc3)(NC(=O)C=C(C)C)C2)C1 c1(CNC2(COC)CCOC2)cc(Cl)c(C)c(Cl)c1 CC1CCc2ccccc2N1CCN=C(NCC(F)F)NCCc1ccc(Cl)cc1 C1(C(N(C(c2ccccc2)CNC(Cc2c(C)non2)=O)C)=O)CC(F)C(=O)N1 C=C(C)CCCC(=O)N1CCC(C2CCCN2C(=O)CCCNS(C)(=O)=O)C1 c1(C(N(CC(CC)NC(c2cn(CC=C)nc2)=O)C)=O)cc2ccccc2nn1 c1(OC(N(C(C)(C)C)C)=O)ccc(NC(=O)OC(C)(C)C)cc1.C12CCN(C1)C2 CC1(C(N2CCCCC2C(=O)NCC2CC(CF)C2)=O)CCC2CC2C1 C1(C)(CNC(C(C)Oc2cccnc2)=O)COCCN(C(c2cccn2C)=O)C1 C(=O)(C(C)(O)C(C)(C)C)NCC(C(C)(C)C)NC(c1nc(C(F)(F)F)cs1)=O C1(NC(c2nc(C(C)(C)C)sc2)=O)CCCCC1NC(=O)C(F)C1CC1 CCC(C)C(C)CNC(C1COCCN1C(=O)CC(C)OC)=O c1(NC(CCCC=C)(CC)c2nnnn2C2CCCC2)ccc2oc(O)nc2c1 C1(O)(C(C)NC(c2ncsc2C2CC2)=O)CCN(C(c2cscc2C2CC2)=O)C1 c1(N(C)C)ccc2c(c1)OCCN2C(=O)Nc1coc(-c2cnn(C)c2)n1 C1(C(N(CCCCN(C(=O)C=CS(C)=O)C)C)=O)CCCCC1C(N)=O Cc1cc(=NC(=O)CC(C)c2ccc3c(c2)OCO3)[nH]n1C1CCCCC1 C1(NC(c2c(C)nc(O)[nH]2)=O)CCN(C(=O)CC2CC(C)(C)CO2)CCC1(F)F c1(C(=O)NCC(C(C)C)NC(CC=CC)=O)ncnc(O)c1Br CCC(c1cccc(Cl)c1)=CC(=O)NCCC1CC(NC(c2[nH]cnc2C)=O)C1 C(=O)(C(CC)SC)NCCCNC(C1C(C=C)C1)=O C=CCCCC(C(=O)N1CC(OCC)C1)NC(=O)C(C1CCC1)OCC c1(CC)ccc(C=CC(=O)NC2CN(C(=O)Cc3cncn3C3CC3)C2)cc1 N1(C(COCC#C)=O)CC=CC(C(=O)NCCOC2CCC2)C1 Clc1c(NC2CCNC3CC23)cccc1I c1(OC)ccc(C(=O)NCC(=O)N(CCS(C)(=O)=O)Cc2ccccc2)cc1 c1(C(N2CC3(CNC(C4(O)COC4)=O)CC2CO3)=O)cc(C(F)F)cc(Cl)c1 c1(N(CC(C2CC2)OC)C)nc(=NCC2CCCOCC2)[nH]c2c1CCC2 C(=O)(C1=NOC2(CCC2)C1)NCCCCC(C)NC(c1n(CCC)ncc1)=O Cc1cc(C(=O)NCC(c2ccccc2)CNC(=O)C(=O)NC2CC2)c(C)cn1 C1(NC(CC2CC(=C)C2)=O)CN(C(c2cnc[nH]2)=O)CC2CCCC12 C(=O)(C(F)(F)c1cccnc1)NCC(=C)CCN1CCOCC1 C(=O)(CCC(=O)NCC1CCCN1C(=O)CC1CCNC1=O)OC CCCN=C(NCCc1nccnc1C)NCC(C1CCOC1)CC CCCC(C)(O)CNC(=O)C(C1CCCN(C(C2(Cl)CCCCC2)=O)C1)C C1(C(N2C(C)CC(NC(=O)C(C)(O)C3CCC3)C2)=O)CCCC(C)(C)C1 C1(CC)CN(C)CCN1C(=O)NCc1nnc(C(F)(F)F)o1 c1(C(=O)NCCC2CCCN(C(C3N(CC)CC3)=O)CC2)cncc2c1CCC2 C(CCCCC(=O)NC1CNCC(O)C1)SC c1(NC(N(CCC)Cc2cncc(OC3CCCC3)c2)=O)cn(C)c(C)n1 c1(C(=O)NCCC(C)(C)NC(C(C)NC(COC)=O)=O)cn(CCOC)nc1C c1(NC(C(c2ccc(F)cc2Br)N(C)CC2CS(=O)(=O)C2)=O)cccc([N+](=O)[O-])c1 N1(C(CCSCC(N)=O)=O)CC(C2(NC(c3cc(O)cc(Cl)c3)=O)CC2)C1 C1(C2(O)CCN(C(c3cccc(N)n3)=O)CC2)(NC(CC(C)(O)C2CC2)=O)CC1 CC1CN(c2cccc(S(=O)(=O)NC3C(=O)OCC3(C)C)n2)CCC1(F)F N1(C(c2c(C)ccnc2)=O)C(C(=O)Nc2ccnc(O)c2)CC2CCCCC12 C1(N(C(=O)C(O)Cn2cncn2)C)CCN(C(=O)CC2CCCC(=O)N2)CC1 CCCCC(C(=O)NC(c1nnnn1CC)(C)CC1CC1)Nc1cccc(Cl)c1 c1(CNC(CCC#CC)=O)nc2c(s1)CN(C(C1CCCN1C)=O)CC2 c1(CC(N2C3CC(NC(C(C)O)=O)CC2CC3)=O)cn(C)c(=O)c2ccccc12 C1(NC(c2c(CNC(C(C)CC(N)=O)=O)occ2)=O)CC2CC1CC21CC1 c1(C(=O)NCC(CNC(C=CCC)=O)CO)nc(Cl)ccc1OCCOCC c1(NC(C2CCN(C(c3ccoc3)=O)C2)=O)ncccc1C1CC1 N1(C(c2scc(C)n2)=O)CC2COCC2(C(=O)NCC(C)S(C)(=O)=O)C1 CC1(CNC(=O)C(C2CCOC2)NC(=O)CCc2ccsc2)CCCC1 c1(CC(N2CC(CNC(C(CC=C)CC)=O)C3(C2)CC3)=O)c(C)cc(C)nc1O C1(C(=O)NC2CCCN(C(c3nc(C)sc3C)=O)C2)CCC(F)(F)CC1(C)C C1(C(N2CC(CNC(CC3CC(CC)C3)=O)C(N(C)C)C2)=O)CCC2CC1CO2 N1(C(C)=O)CCN(C(=O)NCC2CC3(CCC(SC(C)(C)C)O3)C2)C2(CC2)C1 N1(CC(N2CCC(OCc3ccsc3)C2)=O)CCCCCC1=O.n12cc(nn1)C2 N1(C(CC=CCC)=O)CC2CC1C2NC(C1CC1C(C)(C)C)=O C1(C(N2CC(CC=C)(NC(C3CCNC3=O)=O)C2)=O)CCC2(CCC2)O1 CN=c1[nH]ccc(C(N2CC(C(N)=O)(CNC(=O)C(F)OC(F)(F)F)C2)=O)c1N c1(C(N2C(CNC(c3cn(CC)nn3)=O)CC2)=O)ccc2c(c1)NC(=O)C(C)O2 N#CC1(CC(=O)NCCOCCCNC(C2CSCCS2)=O)CCC1 C1(C2CN(C(C3CC(=O)N(C)C3)=O)C2)(NC(C(C2CCCCCC2)OC)=O)CC1 C1(N(C)CCNC(=O)C(=O)NC(C)(C)C)CC2CCC1N2C1CCc2ncccc21 CCCC(C(=O)NCCC(O)C(=O)NCc1coc(CC)n1)OCC c1(C(=O)NC2CC(F)CN(C(=O)C=Cc3cocn3)C2)ccc2nccn2n1 N1(C(C(F)=CC)=O)CCC(N(C(=O)CCc2ccc(OC)c(OC)c2)C)C(C)C1 C(CC(C)(C)CC(=O)N1CCN(C(c2cccc(CC(C)C)c2)=O)C2CC12)OC C1(CSCC(N2CCC(N(C(=O)CC3CC3)C)C2)=O)CCCCO1 C1(C(N(C23CC(C(=O)O)(C2)C3)C(c2cncs2)=O)=O)CC12CCNCC2 C=C(Cl)CCC(=O)NC(C)CCN(C)C(c1cc(C)n(-c2ccc(F)cc2)n1)=O Cc1cc(C(=O)NC2CC2NC(=O)C(C)(O)Cn2c(C)cccc2=O)cnc1O c1(C(N2CCC(C(=O)NC3CC3C(C)C)(OCC)C2)=O)cccc(F)c1F C1(NC(c2cc(C)nn2C)=O)CN(C(=O)CCC(=O)N2CCOCC2)CC12CC2 c1(CC)ccc(C(=O)NCC2C(C(=O)NCC(CC)(CC)OC)C2(C)C)nc1 N1(C(c2c(CNC(=O)CC3CCCC34CC4)noc2)=O)CC2C3C=CC(C3)C2C1 C12(NC(c3cncnc3)=O)CCN(C(=O)CC3CCC4(CC3)CC4)CC1C2 c1(-c2c(C)occ2)nc(COC(C)C)n(CCCOC(F)(F)C(F)(F)F)n1 c1(N(C)CC2CC2(F)F)cc(S(=O)(=O)NC2CC2C(C)(C)C)ccc1C#N C(=O)(C1CCCn2cnnc21)NC1CCN(C(c2nc(C)n(C)c2C)=O)CC1O C1(CC)CN(C)C(=O)CN1C(=O)C(C1CN(C(c2ccccc2OC)=O)C1)OC C(=O)(CC(C)CCc1nn[nH]n1)N(C1CN(C(C(CCC)NC(C)=O)=O)C1)C c1(C(N2CC(NC(CC(C=C)C)=O)C(F)CC2)=O)cc(C)nc2c(O)cccc12 CN1CCN(C(=O)CC2CSCCO2)C(C(=O)NCc2ccnc(F)c2F)C1 c1(C(=O)NC2CC(C)(C)N(C(c3cccnc3O)=O)C2)ccc2c(c1)OCO2 c1(C(=O)NC(CC)CNC(=O)CCNC(=O)OC(C)C)cccc(OC)n1 c1(C(C)C)cc(C(C(=O)NCCCCCO)N(C(C)C)Cc2ccccc2)[nH]n1 N1(C(C=CC(C)=O)=O)CCC2(CC1)CN(C(c1cnn3cccc(C)c13)=O)C2 C1(NC(CNC(=O)OC)=O)CCCC1NC(=O)COC1CCCOC1 N1(C(C)=O)c2ccccc2CC1C(=O)NC1CC1CNC(c1ccc(C#N)s1)=O Cc1cccc(C)c1C(O)C(=O)N1CC(CCNC(C2CCCC(O)C2)=O)C1 N1(C(C(C)C)=O)CC2(C1)C(CNC(=O)CC1CC1(C)C)CCS2(=O)=O N1(CCC(=O)N(CC(CC)NC(=O)C(O)C(F)F)C)CCN(C)CC1 c1(NC(=O)C(C2CCOCC2)C)ccccc1C.CCC1CNC(=O)CO1 N1(Cc2c(C)ccs2)CCC2CN(c3ncncc3I)CCC12 c1(C(=O)NC(CN(C(C2CC3CCC3C2)=O)CC)C)ccc2c(c1)CN(C)CC2 c1(SC)ccc(C(=O)NCC2(O)CN(C(=O)C3=CCCCC3)C2)c(Cl)c1 CCCC(CCCNC(c1[nH]nnc1C)=O)NC(=O)CCc1c(Cl)cccc1Cl c1(CCNC(=O)NCC(c2cccc(F)c2F)F)nc2cccc(Br)c2[nH]1 O=C(CCCC(F)(F)F)NC1CCN(CC(=O)NCc2ccc(F)cc2)CC1O C(=O)(CC(C)(C(F)F)N(C)C)N1CCCC(O)(CNC(CCCC)=O)C1 C1(CNC(c2c(CC)nccc2)=O)CC(=O)NC(=O)C1.C1=CCNC(=O)C1 C1(C(N(C)CC2CCN(C(c3c(C)scc3)=O)C2)=O)CCNC(=O)C1 c12cc(cnc1O)NC(=O)NNC2=O.C1(c2cn(C)nc2)CC(C(=O)O)CCO1 Cc1cc(C(N2CC(NC(=O)CC3CC4(CCC4)CO3)CC(C)C2)=O)cc(N)c1 Cc1csc(CCNC(=O)C(CC2CC2)NC(C2C=CCCC2)=O)n1 c1(C(=O)NCCCN(c2ncc(C#N)cc2F)CC)cccn2nncc12 C1(NS(CC(C)c2ccc(F)cc2)(=O)=O)CCCc2ccccc2C1 Cc1nncc(C(N2CC(O)CC2C(=O)NCCCN(C(=O)C(C)C)C)=O)c1C N1(C(C(C(=O)OCC)F)=O)CC2(CCCC2NC(C2CCC(C(C)(C)C)O2)=O)C1 CC1(O)CC2(CN(C(C3CNC(=O)CN3C(c3ccc(C#N)o3)=O)=O)C2)C1 CC(C)CN=C(NCC(c1ccccn1)C)NC1CC1 Clc1cc[nH]c1C(c1nnnn1C1CCOC1)NC1CSC1 C1(C(=O)NC(C(C)NC(C(CC)O)=O)C)CCN(c2ncccn2)CC1 c1(SCC(=O)OCC)ccc(NC(=O)NC2CN(C(=O)C=NOC)CC2C)cc1 C1(CNC(c2ccc(C)c(F)c2F)=O)CN(C(c2cccs2)=O)CC2(CCC2)O1 C1(C(=O)NC(CC(C)C)CO)C2CCCC2CN1C(=O)CC(C)O N1(C(C2C(C)CCO2)=O)CCC(CO)(NC(c2cc3[nH]ccc3s2)=O)CC1 C1(CNC(CCn2c(C)ncc2)=O)CN(C(=O)C(F)C(F)(F)F)CC(C)(C)C1 C(CC(C)(C)CC=C)NC(C1N(C(COCC#C)=O)CCC1C)=O n1(CC)nnc2c1CCC(C(=O)N(CCCNC(=O)CC1CCC1)C(C)C)C2 C(=O)(C1CCc2nc(C)cn21)NCC1C(NC(CCCOCC)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CCCC(C(C)NC(c2c(C)c(F)ccc2)=O)C1 C1(NC(c2cn(CC=C)nn2)=O)CCCC12CN(C(c1ccc(C)c(N)c1)=O)C2 C1(CNC(c2nnnn2CCCF)C2(C(=O)OC)CCC2)Cc2nccn2C1 c1(C(N(CC)CC2CCN(C(c3scc(C)c3C)=O)CC2)=O)cc2n(c1)CCC2 c1(C2C(C(=O)NC3C(C)(C)CN(C(c4cocn4)=O)C3)C2)cccc2ccccc12 CC(C)CC(C(=O)NCC1=CCCN(C)C1)ONC(C1CCCOC1)=O C(=O)(C(C1CN(C(=O)C=CCN(C)CC)C1)OC)NC1(OCC#C)CC1 N1(C(C2(C#N)CCCO2)=O)CCOC2(C1)CN(C(C1CCC(=O)NC1)=O)C2 N1(C(CC(C)(C)C2CC2)=O)CCCC(F)(CNC(C2CS(=O)(=O)CCO2)=O)C1 CN1CCC(NC(=O)C=CBr)C12CCCN(C(c1ccc(-c3cc[nH]n3)s1)=O)C2 c1(CN(C2CC(OC)C2(C)C)CCC)cc(=O)oc2cc(O)c(O)cc12 C1(F)(C(N2CCC(NC(C(CSC)(C)C)=O)C2)=O)CCS(=O)(=O)C1 CN1CCCC(C(=O)N(C)CC2(O)CN(C(c3scnc3C(F)F)=O)C2)C1 C1(NC(C(CC)(C)C)=O)Cc2cccnc2C1.C12CCCN(C1)C2=O c1(OC(C)C)ccc(C(=O)NC2CN(C(=O)Cc3cccn3C)C3CC23)cn1 CCCCC(C)C(=O)N1CCCC1CNC(C1CC12CCCC2)=O C(C(=O)N(C)CCNC(=O)C(C)Cn1ccnc1)(C(C)(C)C)N1CCC(C)CC1 C(=O)(CCC(=O)N1CCOCC1CCNC(c1ccc(C(C)F)cc1)=O)NCC c1(C(N2CC(NC(c3c(C)c(Br)cnc3)=O)(CO)C2)=O)cc2c(ncn2C)[nH]1 CCC(CC)C(F)C(=O)N(C)CC1(O)CN(C(C2(C)CCOC2C)=O)C1 Cc1cnnc(C(=O)NC2CC(C)N(C(c3csc(C(F)(F)F)n3)=O)C2)c1 C1(NC(c2c(CNC(C3C(C)OCCO3)=O)noc2)=O)(CO)CCCCC1C N1(C(c2cccc(C#C)c2)=O)CCN(C(=O)C=CSc2nc[nH]n2)C(C)C1C C(=O)(C(O)C(F)(F)F)N1C(CCCNC(Cn2c(CCC)ncc2)=O)CCC1 c1(CC(N2CC(N(C(C(C3CCC3)OCC)=O)C)C2)=O)ccc(S(N)(=O)=O)cc1 CCC(CC)C(C)C(=O)NCCn1cc(CNC(=O)C(C)(C)O)nn1 c1(CC(=O)NCC(C)NC(c2c(NC(C)=O)cncc2)=O)ccccc1S(C)=O C1(N2CC(CNC(=O)C(Cc3ccc(F)cc3)C3CC3)C2)CCC(=O)NC1=O c1(C(C(=O)NCC(CCC)NC(c2ccc(C#N)[nH]2)=O)O)cccc(C)c1F S(=O)(=O)(c1[nH]c(=NCC2CCOC2)ccc1Br)N1C2CC(CC)CC1CCC2 CC1CC2CCC(C1)N2C(C1(F)CCC1)=O.C12C3CCC(C3)C1NC2=O N1(C(c2n(C)ncn2)=O)CC2(CC(C(N3CCC(C#N)C3)=O)CO2)C1 CC1(C#N)CCN(C(C2CC3CC3N2Cc2ccc(O)nc2)=O)CC1 C1(NC(C(C=C)C)=O)CN(C(=O)CCCN(C)C)C2CC12 C#CC(CO)(CO)NC(=O)C(C1CCN(C(c2coc(C(N)=O)c2)=O)CC1)C C1(NC(c2ccc3[nH]ccc3n2)=O)COC2(C1)CN(C(c1ccco1)=O)C2 C=C1CCC(C(=O)NCCC2CC(C(=O)N(C)CC3(O)CCOC3)C2)CC1 C(C(CC(C)C)C(=O)N(CC(=O)NC1CC1)C)NC(c1c(C#C)c[nH]n1)=O C12(CNC(C3CCCC(OC)C3)=O)CCCCC1N(C(=O)OC(C)(C)C)CCC2 C1(C(N(C)Cc2cc(C)no2)=O)CC12CCN(C(=O)CCn1ccnc1)C2 CN1CC(C)(C(N2CC(N(C(=O)CSc3ccc(Cl)s3)C)C2)=O)CCC1=O C(=O)(CCCCC(F)(F)F)N1CC(n2cc(C34C(C)OC(CC3)C4)nn2)OCC1 c1(C(N(CC(N)=O)C(C)C)=O)cccc(-n2ccnc2)c1.N N1(C(CC2C(C)OCC2)=O)CCCC2(C1)CN(C(C13CC(C)(CCO1)C3)=O)C2 C1(CC)C(C(=O)NOCCCCC(=O)OC)CCN1C(=O)CCCC1CCC1 Cc1nccc(Cl)c1C(=O)NCCC(C)N(C)C(c1ccnc(Cl)c1N)=O N1(Cc2cc(C)cc(OC)c2O)CCC2CN(C(c3ccccc3S)=O)CC2C1 c1(SC)cccc(CC(=O)NCC(C)CN(C)C(c2cnc(C)s2)=O)c1 c1(C(=O)NCC(C)NC(=O)Cc2cnn(C)c2)cc2cc(N)ccc2o1 c1(C(=O)NCCC(CC)(C)NC(=O)C2=C(Cl)CCC2)ncc(Cl)cc1F c1(NC2C(F)(F)CCN(C(c3cc(CO)on3)=O)C2)ncnc2ccc(Br)cc12 N1(C(Cc2ccc(C)o2)=O)CC2CCCC(NC(=O)CSc3nnc(S)s3)(C2)C1 C1(C(=O)NCC(CCCC)NC(c2ncsc2C(C)C)=O)CC2CCCC(C1)C2 CC(CC=Cc1ccccc1)C(=O)N(C1CCCN(C(c2ccccc2)=O)C1)C c1(C(=O)NC2CC(C(=O)NCC3SCCS3)C23CCC3)cccn2ccnc12 c1(C(N(CC(CC)NC(C2(COC)CCCO2)=O)C)=O)nc(C)ccc1F C(=O)(C(F)C(C)(C)O)NCCCC1N(C(c2cc(OC)ncc2)=O)CCCC1 C1(C(=O)NCCCCC(C)NC(C23CC(C)(C2)C3)=O)CCCC(F)(F)CC1 c1(OC(C(=O)OC)C)cccc(NCC2CCC(C)(C)C2)c1 c1(C(N(CC(C)N(C(CC(CC)O)=O)C)C)=O)c(OC)cc(OC)cc1CC C1(C(=O)NCCc2c(C)n[nH]c2)(NC(=O)CC2CC(=O)C2)CCOCC1 N1(C(C(c2n(C)cnn2)(C)C)=O)CCC(O)(CCNC(c2csc(Cl)c2)=O)C1 C1(C(=O)NCCC2N(C(c3c(C)n(C)nn3)=O)CCCC2)CCC(=O)C(C)C1 CCC(F)(F)C(C)(C)C(=O)NCCn1cc(CC(C)(C)C(F)(F)F)nn1 c1(C(N2CC3CCN(Cc4c(Br)ccc(NC)c4)C3C2)=O)cccc2[nH]ccc12 c1(OC)c(Cl)cccc1S(=O)(=O)NCc1c(Br)cccc1Br N1(C(C(c2cccc(C(F)(F)F)c2)CC)=O)CCC2(CC1)COC(C)C2 C#CCCCCCC(=O)NC(C)C=CC(=O)NC1CCc2nn[nH]c2C1 CCC(C)CC(C(=O)NCCCc1c[nH]nc1C)NC(=O)CNC(=O)C(C)CC c1(C(N(CC=C)CC=C)=O)c(OC(C2CCCC2C(=O)O)=O)cccc1CC CC(C)S(=O)(=O)C(C)C(=O)N1CCN(C2CCN(C(=O)C(F)=C3CCC3)C2)CC1 CON(C(=O)C1=CCC(NC(=O)C(C)=C(C)C)CC1)C1CCOCC1 c1(N(CC(C2CCCC2)OCC)C)ncnc2c1ncn2CC(O)C(C)O CCCC(CC)C(=O)NC1C2CC1CN(C(=O)CCOc1ccccc1)C2 Cc1ccc(O)c(CC(=O)NCC(C)N(C)C(c2cnc(Cl)[nH]2)=O)c1 Cc1cccc(Br)c1C(C(=O)N1CC(=CC(C)(C)C)C1)NC(=O)C(F)C(C)(C)O CC1CC(C)(C(=O)NCC=C2CCN(C(=O)C(C)OC3CCCC3)CC2)CCO1 c1(CN2CCC(NC(c3ccc(C4CC4)o3)=O)CC2)cc2n(n1)CCSC2 CC(C)CC(O)C(=O)N1CCN(C)C(SCCCS(=O)(=O)Oc2ccccc2)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC(CNC(=O)Cc2ccccc2)C12CCC2 CCC1=C(C(=O)NOCC(N2CC(O)(OC)C2)=O)CCCO1 C(=O)(CC(O)CC(C)C)N1CCC(N(C(=O)C(C)NC(C)=O)CC#C)C1 C1(C(=O)NCc2ncc(C)o2)CC12CCN(C(c1ccn(C(C)C)n1)=O)C2 CCC(C)C(O)CC(=O)NC1CC2(C1)CN(C(C13CC1C3)=O)C2 Cn1nnc(C=CC(N2CCN(CCCCCNC(=O)CCC3CC3)CC2)=O)n1 C(=O)(C(CCC1CC1)NC(=O)Cc1cc(C)on1)NC(c1ncnn1C)CC C(=O)(CCCC(F)(F)CO)NCC1C(C)CCN1C(C1OCCO1)=O c1(C(C)NC(=O)C=CCNC(C2CC2(F)Cl)=O)nnc(O)n1C CC(F)(F)CCC(=O)NCCN1CCSCC1c1cccs1 C1(N(C)C)(C(=O)NC2CCC(CNC(c3cc(Br)n[nH]3)=O)C2)CCCCC1 c1(CC(=O)NCC2N(C(C3(COC)CCC3)=O)CC2)cc(F)ccc1O N1(C(C2(NC(Cn3ccc(C)n3)=O)CCCCC2)=O)CCOCCC1C c1(C(=O)NC2CC3(C(NC(CC(=C)C)=O)C3)C2)cccc2c1OCO2 C1(CCCC)(C(=O)Oc2ncnc3cc[nH]c23)CN(C(=O)COC)C(=O)CO1 C1(C(N(CCCN(C(C[SH](c2ccccc2)CC=C)=O)C)C)=O)CCC(OC)C1 CCCC(CCC)CC(=O)NC1COC2(CCN(C(c3cccnc3N)=O)C2)C1 C(=O)(C1=CC2(CCOC2)C1)NC(CN(C(c1cc(Br)n[nH]1)=O)CC)C C1(NC(CC(C)C2CCCO2)=O)CN(C(c2sccc2C(F)F)=O)CC1(C)C n1(CC(=O)N(C2CC(NC(C3ON=C(CC)C3)=O)C2)C)cc([N+](=O)[O-])ccc1=O c1(C(=O)NCC2CCN(C(CCC)=O)C2)cc2c(Cl)cccc2nc1C C(=O)(C1=CCCOC1)N1CCCC(N(C2CC2F)C(=O)OC(C)(C)C)C1 C(CC(=O)NCC1(F)CCC(NC(c2cscc2OC)=O)C1)(C(F)(F)F)OC C1(CNC(CCCCCNC(C)=O)=O)CC(C(=O)N2OC3CCC2CC3)=NO1 C(=O)(CCC(=O)N(C1CC(NC(=O)C(c2cccc(Cl)c2)N(C)C)C1)C)OC c1(CC(=O)NC(C)CCNC(=O)CN(C)C2CC2)cc(Cl)c(Br)cc1F N1(C(c2ccc(C(C)=O)cc2)=O)CCN(C(C2CCC(=O)O2)=O)CC(C)(F)C1 Cc1nc(CNC(=O)C(CNC(C2COCCN2C(C)C)=O)CC2CC2)sc1C Cc1ccc(CNC(C2CC(C)CN2C(C2CC2[N+](=O)[O-])=O)=O)nc1 c1(C(N2CC(CNC(CC(CC)SC)=O)C(O)C2)=O)cc(C)c(Cl)cc1F Cn1cnc(C(=O)NC2CCC(CNC(C3(c4ccno4)CC3)=O)C2)n1 N1(C(c2cnc(C)cn2)C(=O)NCCOC)CCCC2(C)CCCC12 c1(C(=O)NCC(=C)CCNC(C2(C#N)CC2)=O)nn(CC)c(=O)c2ccccc12 N1(C(CC2(C=C)CN(C(=O)Cc3ccoc3)C2)=O)Cc2cccnc2C1 c1(C(=O)NCC2CCN(C(C3C(F)(F)C34CCC4)=O)C2)ccc(O)cc1[N+](=O)[O-] N1(C(C(C)C2CCCO2)=O)CC(O)(NC(C2(CNC(=O)OC(C)(C)C)CC2)=O)C1 C1(NC(CC(=O)N(C)C)=O)C2CCC1N(C(=O)Cn1cnc(Br)n1)C2 c1(NCCc2n[nH]c(=N)s2)ccc(S(=O)(=O)N2CCC(CO)C2)cc1Cl Cc1cc(S(=O)(=O)N(C)C(C)C)c(C)cc1-c1ccc(C(=O)NCC(C)C)cc1 C1(C(=O)NC(C(C)C)CNC(=O)CC2CC3(CC3)C2)CN(CP(C)(C)=O)C1 N1(C(COC)=O)CCN(C(c2ccc(F)cc2OC)=O)C2CCCCC12 c1(C2(C(=O)NCC(CC)(CC)NC(=O)C(=O)N(C)C)CCC2)ccc(C#N)cc1 c1(C(=O)NCC=CCNC(C2CC3(OC)CC2C3)=O)cccc(S(C)=O)c1 c1(OC)cc(F)cc(C=CC(N2CCN(Cc3cnc(Cl)nc3)CC23CC3)=O)c1 CN1CCN(C(N2CCCC2)=O)CC1c1cn(CCN2CCCCC2)nn1 Cc1cnc(N(C2C3CCC2CNC3)C(=O)C(C)(C)C)cc1Cl.C1(=O)CN1 N1(C(COc2c(C)cccc2)=O)C(C)CC2CN(C(=O)CCc3cscn3)CC12 N1(CCC=CCC)CCn2ncc(CNC(C3CCC4(C3)CC4(F)F)=O)c2C1 N1(CCN(C(Cc2ccccc2)CCO)CC)CSCCSC1 c1(N2CCC(O)(CNC(c3cc(C(C)C)no3)=O)C2)ncc2c(ccn2C)n1 c1(SC)ncc(C(=O)N(C)CCOCCN(C)C(C23CC(F)(C2)C3)=O)[nH]1 N1(C(Cc2scc(CC)n2)=O)CCCC2CN(C(c3ccnc(Cl)c3)=O)CC12 C(=O)(CS(=O)C(F)(F)F)N1CCC(NC(c2ccc(C(=O)OC)cn2)=O)C1 c1(C(=O)NCC=CCNC(C2(C)CCC(=O)C2)=O)c(F)ccc2n[nH]cc12 C(CCN=c1[nH]c(=NCCc2ccn(C)n2)c2[nH]ccc2[nH]1)N(C(C)C)C CC1(C)CCN(C(C2C3CCC2CC3)=O)CC1NC(=O)COCC1CCC1 Cc1c(NCCNCc2ccncc2-c2nn[nH]n2)cnn1C1CCCC1 c1(-c2ncc(C(=O)NC3CC(C)(NC(C(C)CO)=O)C3)s2)c(F)cccc1Cl C1(C(N2CC(OC)(CNC(=O)Cn3cc(C(F)(F)F)nn3)C2)=O)CC1C1CCC1 C1(NC(C2CCN(CC)C2)=O)CCC12CCN(C(=O)CCc1cnoc1)CC2 C1(NC(c2ccc(CC)s2)=O)CCC2(CCN(C(=O)C3=C(C)CCC3)C2)C1 c1(CC(=O)NCC(C)(C2CCC2)NC(=O)COCC(F)F)cccc2sccc12 c1(C(N2CCC(NC(C(CC)(C)COC)=O)C2)=O)c[nH]c2cccc(Cl)c12 C(=O)(C1=CCCCO1)N1C(C)C(CCC(=O)NCC(F)CO)CC1 c1(OC)cc(Br)cc(C(=O)NCC(Cl)(Cl)Cl)c1N Cc1ccc(C(N2CC3CN(C(=O)C=CBr)CC3(C)C2)=O)c2c1CCC2 N1(C(Cc2ncc(C)o2)=O)CCC2(CCC(NC(c3csc(O)n3)=O)C2)CC1 c1(C(=O)NCCCC2CCCC2O)cc(O)nc2c1CCCN2 c1(NC(CC2CCN(C(=O)NC(c3noc(=O)n3C)C)C2)=O)ccc(Cl)cc1 CCC(C(O)C(C)C)Nc1cnn(CC(F)(F)F)c1C1CC1 N1(Cc2ccc(C(C)=O)cc2)CC(=O)N(CC2(COC)CC2)C1=O c1(C(=O)OCC)ncnc(N2CCN(C)C(CNC(=O)CSS(C)(=O)=O)C2)c1OC C1(C(=O)NCC(CN(C(C(CCC)N(C)C)=O)CC)(C)C)CCCCN1N=O CCCC(O)C(=O)N(CCCNC(=O)CC1CSCCO1)CC1CCCC1 c1(C(=O)NC2C(CC)CN(C(=O)CCCOC)C2)c(Cl)ccc2ncccc12 Cc1noc(N)c1C(=O)NC1CC(OCC(=O)NCc2cnccn2)C1 CC(C)C(O)C(C)(C)C(=O)NCC1CCC(C(=O)NCCCC(N)=O)O1 c1(CN2C(C)(C(=O)Nc3c(OC)cccc3Br)CCC2)ccc(C)c(F)c1F C1(C(=O)NC(C=CC(=O)NCc2c(C)n(C)nn2)(C)C)CNC(=O)CC1C c1(N(C2CNCC2(F)F)Cc2c(F)ccc(Br)c2)cc2ncnn2cn1 n1(CCC)ccnc1C=CC(N1CC(C)(N(C(=O)CC2COC(C)(C)C2)CC)C1)=O N1(C(=O)Cc2c(F)cccc2Cl)CCC2CCCN(C(=O)C3=COCCO3)C2C1 N1(C(C(C)CO)=O)CC(C2CCN(C(C3CCC4(CC3)CC4)=O)CC2)C1 C(=O)(C(CN(C)C)NC(c1csc(Cl)n1)=O)NCCNC(CC)=O C1(CNC(c2ncnc(C)c2Br)=O)(CO)COCC2CCCCN12 Cc1cc(C(=O)NCC(O)CN(C)C(c2cccc(C3CC3)c2)=O)n(C)n1 C1(CNC(C2C(OC)CC2)=O)CCN(C(c2ccc(C)nc2O)=O)CC1(F)F C1(CNC(C(c2ccco2)NC(c2ccc(C)nn2)=O)=O)CC2(CCC2)CO1 C(=O)(C(C)(C)CCC(=O)NCC(O)CN(C)C(C1CC=CC1)=O)OC c1(C(C(=O)NCCCN(C(C)C)C(c2cc(C(F)(F)F)cs2)=O)O)cncn1C C1(NC(c2occ(C)c2C)=O)CC2CN(C(c3ccnc(C(N)=O)c3)=O)CC2C1 C(=O)(CC1=CCOCC1)N1CC(CNC(c2n(C)c(-c3ccccc3)nn2)=O)C1 N1(C(CSCCC)=O)CC(NC(=O)C(CC)C2CCOCC2)C(S(C)(=O)=O)C1 c1(OC)ccccc1C(CNC(=O)C(C)C(F)F)NC(=O)CCc1ccn(C)c1 C1(CC)CN(C(C2(COC)CCCO2)=O)CCC1NC(=O)CCC(C)(C)O C1(OC)(CNC(=O)Nc2nc(C(F)(F)F)sc2N)CCN(C(C)=O)CC1 N1(C(c2cn(C)nc2)=O)C(C(=O)N(CC(F)F)CCO)CCC12CC2 c1(OCC)ncc(C(=O)N(CC(C)O)CCNC(C2(F)CCC2)=O)cn1 C1(C2(NC(C3CCCN3C3CCCC3)=O)CC2)CCCCN1C(=O)C=CCF C1(CN(C(C)=O)C)CCN(C(=O)CN2CCNC2=O)C1 c1(C(=O)NCC2CC(NC(c3cccc(=O)o3)=O)C2)cc(Cl)cc2cccnc12 Cc1c(C(=O)NC2CN(C(c3cnc(Br)o3)=O)CCC2(F)F)ccc(Br)c1F c1(SC)ccc(C(=O)NC2CC2CNC(=O)C(c2ccnn2C)O)cn1 Cc1ncc(NC(=O)CC2(CNC(C3CCCC(=O)CC3)=O)CC2)c(C)n1 c1(-c2cn(C3CN(C(=O)Cc4nc(C5CC5)cs4)C3)nn2)cc(F)c(Cl)c(F)c1 N1(C(C(NOC)=O)=O)CCN2CCN(C(c3cnc(N)cn3)=O)CC2C1 N1(C(c2cc(CCC)ncc2)=O)CCC(CNC(c2nccn2CC)=O)C(C)C1 C1(C(N(C)CC2N(C(c3cc(C)sc3)=O)CCC2)=O)CC2(C1)CC21CC1 C1(CNC(c2ccc(SCC)nc2)=O)CN(C(=O)C=Cc2ccco2)CCCO1 N1(C(Cc2cccc(C)c2)=O)CC2CN(C(=O)CCOCC(F)F)CC2(C)C1 C(CCC(=O)NCCCC(C)NC(=O)Cc1sccc1C)=CCC=C c1(CNC(N2CCCC2CSC2CC2)=O)cncc2[nH]ccc12 c1(C(=O)NCCCCCNC(c2c(CC)nn[nH]2)=O)cnc(N)c(CO)c1 C(=O)(C1=C(C)CCCC1(C)C)N1CC(CC)C(NC(c2ccnnc2)=O)CC1 C1(NC(c2cn(CC=C)nc2)=O)CN(C(=O)Cc2ccc(Cl)s2)C(CC)(CC)C1 N1(c2n(CCOCC=C)c(C3(OC)CCOC3)nn2)CC(CCO)OCC1(C)C Cc1ccc2c(c1)SC(C(N1CC3CN(C(=O)C(C)c4cc[nH]n4)CC3C1)=O)C2 N1(C(C(CC=C)C)=O)CCCN(CCNC(c2ccc(F)c(Cl)c2)=O)CC1 C1(NC(CC2C(CNC(CSC(C)(C)C)=O)C2)=O)CCSCC1 C1(C(=O)NC2(CC=C)CCOC2)CCN(C(=O)C=Cc2ccco2)O1 N1(C(C(C(C)C)O)=O)CCCOC(CCNC(C2(F)CCCCC2)=O)C1 C(=O)(CCS(=O)(=O)C1CCCC1)NC12C(CN(C(CCC(=O)NC)=O)C1)CCC2 c1(NC2(CNC(C3(OCC)CCOCC3)=O)CC2)ncnc2c1COC2 C1(C(C)C)CN(C(c2cnc[nH]2)=O)CCN1C(C1CC(OC(F)F)C1)=O c1(C(N(CC(N2CCC(O)(CC#C)CC2)=O)CC(C)C)=O)ccc2cc[nH]c2n1 C1(CNC(c2cc(CCC)oc2C)=O)CN(C(c2ccnc[n+]2[O-])=O)CCN1C C1(C(N2CC(CNC(C3=NNC(=O)CC3)=O)C(O)C2)=O)CCc2nncn2CC1 c1(OC)ccc(NS(=O)(=O)CC2CC3(CCC3)CO2)cc1S(N)(=O)=O C1(NC(c2nc(CC)sc2)=O)CCN(C(=O)C(C)(C)F)CC(C)(C)C1 C(C(=O)NCC1(C(C)NC(c2nn(C)cc2C(C)=O)=O)CC1)(C(C)(C)C)OC c1(NC(C(C)(CO)NC(C(C)=C(CC)C)=O)=O)ccc(Cl)cc1Cl c1(C(N2C(C)(CC(N3CCCCC3CO)=O)CC2)=O)c(O)cccc1[N+](=O)[O-] N1(C(C2CN(C(c3ncnc(C)c3C)=O)CC23CC3)=O)CCc2n[nH]cc2C1 c1(CN2C(C(N3CCCC(C(=O)OCC)C3)=O)CC(F)C2)c(O)ccc(Cl)c1Cl c1(CCCC(=O)N(CCNC(C2(COC)CC=CC2)=O)CC)cccc(OC)c1 C12(C(N3CC(C(N)=O)(CNC(C(C=CCCC)O)=O)C3)=O)CCC(OC)C1C2 CCCCCC(O)CC(=O)N1CCN(C(C)CNC(c2ccccc2C)=O)CC1 CCCCC(C)(F)C(=O)N1CC=C(C(=O)NCC(C)(C)CCO)CC1 CC(=O)CCCC(=O)N1CCC(C(F)F)(CNC(c2nccc(Cl)c2F)=O)C1 CCC(C)(CNC(=O)CC1CCCCC1)C(=O)NC1CC(CO)C12CCC2 C#Cc1cc(NC(C2CC23CC(NC(c2ccc(Cl)o2)=O)C3)=O)ccc1C C12(CN)CC(CC1CN1CCC(O)C1c1ccccc1Cl)C2 N1(C(CCC=C(C)C)=O)CC2CC(C1)N(C(=O)C=Cc1cscn1)C2 C(=O)(C#CC1CCOC1)N(C)CCN(C)C(c1cc(F)cc(Br)c1)=O Cc1nc(CNC(=O)CCCN(C)C)oc1C(=O)NOCCCN(C)C N1(CCNC(C(CC)O)=O)CCN(C(=O)C(F)(F)c2ccsc2Cl)CC1 CC(C)CS(=O)(=O)CC(=O)NC(C1CCCCC1)CNC(C1CCCCO1)=O N1(C(C(C)N(CCC)C(C2CCOC2C2CC2)=O)=O)CC=C(COC)CC1 c1(OC)cc(C(N2C3CN(C(=O)CC4COCCO4)CC23)=O)cc(O)c1O C1(OC)CCN(C(C2CC(C)(C)CN2C(c2cc(O)n(C)n2)=O)=O)CC1C C1(CC(N2CCC(C)(CNC(=O)CS(N)(=O)=O)C2)=O)COc2ccccc2O1 CCC(C)C(C(=O)NCCc1ccccc1)N(C(=O)Cc1coc(C)c1)C CCCC(O)CC(=O)N1CC(NC(c2cccc(Cl)c2N)=O)CCC1C CCCCCCCCCC=CC(N1CC(NC(=O)C(C)C2CCCC2)C(F)C1)=O C1(CNC(=O)C=CCO)CN(C(=O)Cc2ccc3c(c2)CCC3)C2COCC2O1 C1(CNC(CCC(C)OC)=O)(OC)CCN(C(C2CN3CCN2CC3)=O)CC1 C(CC(C)(C)C(=O)NC(CNC(=O)CCN1CCC1)CC(C)C)OC N1(C(c2c(C)nsc2)=O)CCC2(CC1)CC2C(=O)NCc1sccc1Cl N1(CC(CC)C)CCC(c2cccc(NC(C3C4COCC34)=O)c2)CC1 N1(C(c2cccc3cccnc23)=O)CCCC2(CCCN2C(=O)C(F)Cl)C1 c1(OCCC(=O)N(C2CN(C(C3C(SC)CCC3)=O)C2)C)ccc(C)cc1C C1(C(C)(C)NC(C(C)C#N)=O)CCN(C(=O)CCCn2c(O)nnc2O)CC1 C1(NC(C(n2cc(CNC(c3ccccc3)=O)nn2)C)=O)CCN(C(N)=O)C1 N1(C(c2ccc(CC)cc2)=O)CCC(NC(=O)CSC)C(C(C)C)C1 C1(CNC(C(CC=C)(C)CC)=O)CCCC2CN(C(=O)Cc3cc(C)[nH]n3)CC12 C1(C(=O)NCC2C(NC(c3ccn(C4CC4(F)F)n3)=O)CCC2)CC2(C1)CC2F C(=O)(CC1=CCCCC1)N1C(CC)CN(C(c2cn(C)nc2Cl)=O)CC1 C12(CNC(CCCCCSC)=O)CCCC1CN(C(=O)C(C)Cc1cnco1)C2 c1(CC(=O)Nc2nc(-c3cccc(F)c3)cs2)cc(Br)ccc1Br c1(C(N2CCC(CC(=O)NCCCS(N)(=O)=O)C2)=O)ccc(Br)cc1F C1(C(=O)OC)COCCN1C(C1CC(NC(=O)CCc2ccsc2)C1)=O Cc1cc(C(=O)NC2(CC(O)CO)CC2)c(C)n1C1CCOC1 Cc1ccc(CC(=O)N(C)CC2(O)CCCN(C(=O)CC(C)F)C2)cc1Cl Cc1ccc(F)cc1NC(=O)CN(C)C.C12CN(C(=O)CCC(F)F)CCC1N2 c1(C(N(CC(C)O)CCNC(CCCNC(=O)NC)=O)=O)c[nH]c2nccc-2c1 C1(C(N2CC(F)(CNC(C3(C)ON=C(C)C3)=O)C2)=O)CCc2cn(C)nc2C1 N1(C(c2cc(CNC(C3(C=C)CCC3)=O)nn2C)=O)CC2(C1)CC(C)(O)C2 C(=O)(CC(C)CCC(=O)NC1CC(C)CN(C(=O)C2=CCCC2)C1)OC C12(C(=O)NC(C(=O)NC(c3ccc(F)cn3)C)C3(O)CCC3)CC1CNC2=O c1(COC(CC)C(=O)NC2CCCC2NC(C2(CF)CC2)=O)ccc(OC)cc1 C1(C)(CC)CC(NC(=O)C(CC(F)F)N(C(=O)CN=[N+]=[N-])C)CCO1 c1(C(N2CC3C(NC(C(C)SCCCC)=O)C3C2)=O)c(OC)ccnc1OC C1(CN(C(c2n(C)nc(Br)c2)=O)C2CC2)CCC(C)(C)CN1C(=O)OC(C)(C)C CCC(C)CC(=O)C(=O)NCC1CC(NC(C2CCSCC2)=O)C1 c1(OC)cnc(Cl)cc1C(=O)NC1CC2CN(C(c3cnc(Cl)cc3Cl)=O)CC12 c1(NCC(C(C)c2ccccc2)C)nnccc1C#N C1(C(C)NC(c2c(CC)scn2)=O)CCCN(C(=O)Cc2ccncc2Cl)C1 C1(NC(c2cccnc2)C(C)C)C2CN(S(=O)(=O)Cc3ccc(F)cc3)CC12 C(=O)(C(O)CC(F)(F)F)NC1C(n2cc(C(C)NC)nn2)CCC1 C1(C)(CNC(C=C(CCC)C)=O)CCN(C(c2cc(N(C)C)nc(Cl)c2)=O)CC1 N1(C(Cc2ccc(C)o2)=O)CC(C2CN(C(=O)Cc3ccc(Br)cc3)C2)C1 C1(C(N(C2CCN(C(C3CN(C(C)=O)C3)=O)CC2)CC)=O)OC2CCC1CC2 c1(C(=O)NC2C(C(=O)NC(C=C)(C)CC)CC=CC2)cc(N)cc(F)c1 C(=O)(CCCCCO)NCC(C)(C1CC1)NC(C(C)c1cccs1)=O Cc1csc(C(=O)NC2CC(O)C2CC(=O)C2(c3ncccn3)CC2)c1 C1(c2cn(-c3cc(C)c(N)cc3)nn2)CC(C)N(C)CC1C CC(CCNC(=O)C(CO)NC(N)=O)CCNC(c1cnc(CC(C)(C)C)s1)=O C1(NC(CNC(C)=O)=O)CC12CCN(C(C1CCCCC(=O)N1)=O)CC2 CC(C)C(C)(O)CNC(=O)C(CO)NC(=O)CC1CCOCC1 N1(C(c2cc(C(C)C)nn2C)=O)CCN(C(=O)C(C)CSC(F)(F)F)CC(O)C1 N1(C(CC(COC)NC(=O)CCC2CC2(C)C)=O)CCCC2(CCOC2)C1 N1(C(c2c(OC)scc2)=O)CCCC2(CCN(C(=O)C(O)CC(C)C)CC2)C1 C1(C(=O)NCC2(C)CC(NC(Cn3ncc(CC)c3)=O)C2)CC2CCC2C1 c1(C2C(C(N(C3CCC(O)CC3)C)=O)C2)cc(F)cc(Cl)c1 CC(O)C(C)(C)C(=O)NCC1(NC(c2cc(C(C)(C)O)on2)=O)CCCC1 C(C(F)(F)F)(C1CCC1)C(=O)NC1CC(C)C1.c1(C2C(=O)N2)ccccc1 CN1CCCC(F)(C(=O)NCC2CN(C(c3c[nH]c(=S)cn3)=O)C2)C1 c1(OCC)ncc(NC(C2CCC(NC(c3n[nH]cc3I)=O)C2)=O)cc1Cl c1(C(=O)NC2CCC(N(C(CN(C(C)=O)C)=O)C)CC2)c(O)ncc2c1CCC2 c1(CCNC(=O)NC(C(C2CC2)OC)C)ccsc1C N1(C(C2CCc3ccnn3C2)=O)CCC2(CC1)CCN(C(C1SCCS1)=O)CC2 c1(NC(CCc2cc(C)cc(C)c2)=O)nc2cc3c(cc2s1)OCCO3 c1(OC)cc(S(=O)(=O)N(C)C)ccc1C(=O)O.C1(C)C(=O)O1 C1(C(=O)NC(CC)C(=O)NC)C2CCCC2CN1C(=O)C(C#N)C(C)C CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(=O)CCC2CC2(Cl)Cl)CC(C)(F)C1 C=C1CCN(C(=O)CC(O)C(C)C)C(C(=O)N(CCO)CCN(C)C)C1 Cc1c(NCC(c2ccccc2)C)nc[nH]c1=NCC(C)O C(=O)(C(C)(O)C(C)C)N1CC(NC(C(n2c(C)ccn2)C)=O)C(O)C1 C(=O)(CN=S(C)(C)=O)N(C(C)CCNC(c1ccc(C2CCCCO2)cc1)=O)C C1(C(=O)NCC(N(CC)OC)=O)CCCN(C(C2CCCSC2C)=O)CC1 c1(SCCNC(N2CCC(N3CC=CC3)C2)=O)ccc2c(c1)OCO2 O=C1CCc2ccc(SCC3CCCC3NC(=O)CSCCCl)nc2C1 c1(CC2(C(=O)NC)CN(C(C3N(C(C(C)C)=O)CSC3)=O)C2)cccc(F)c1 N1(C(C2(C3CC3)CN(C(C3CCCC4(CC4)C3)=O)C2)=O)Cc2n[nH]cc2C1CO C=CC1CN(C(=O)C(C)C(C)(C)O)CC1NC(=O)CCc1ccc(CC)cc1 C1(C(=O)NCC2(OC)CC2)CCN(C(=O)C(n2ccnc2C)C)C1C c1(OC(C=CC(=O)NCC(C)NC(c2cnn(C(C)(C)C)c2)=O)=O)ccccn1 C(CCC(C(=O)NCc1ccccc1)N1CCOC(CN=[N+]=[N-])C1)OCC=C C(C1CN(C(C2CC2(C)C(C)C)=O)Cc2ccccc21)NC(c1cc(C)ncn1)=O C12(NC(c3ccc(CC)s3)=O)CCOC(CNC(C34CC(C)C3C4)=O)(C1)C2 CC(C)(C(=O)N1CCCC1CNC(=O)CCc1cccs1)C1CCCC1 C1(NC(CN(c2ccccc2)CC)=O)CCCC1NC(C12CCCC1C2)=O c1(C(N2CC(O)(CN(C)C(C3CCOC3)=O)C2)=O)cc(Br)n2c1CCC2 C1(C)(CNC(C(C)(C)c2ccno2)=O)CCN(C(c2ccccc2C2CC2)=O)C1 C1(c2n(CC)nnn2)(NCc2csc(SC)n2)CCCC1CN(C)C Cc1cc(C(N2CCCC2C2(NC(C3CCC(=O)N3)=O)CC2)=O)n[nH]1 C1(NC(C(C=C)O)=O)CN(C(=O)CC2CCCN2C)CC1C(F)F c1(C(=O)NCCC(C)NC(=O)Cc2ccno2)csc(-c2cccnc2)n1 c1(N(C(=O)CC2CN(C(C3C4CCCOC34)=O)CCO2)C)ccccc1O C1(CCC)CCCC1C(=O)NCCOC1CN(C(c2cnc(CC)s2)=O)C1 CCC(O)C(C)(C)C(=O)NCc1ccoc1C(=O)N(C1CC(F)(F)C1)C Cc1nc(C)c(C(=O)NC2COCCN(C(C3(N=[N+]=[N-])CC3)=O)C2)nc1C C(=O)(C(C)CC(N)=O)NC1CN(C(C=Cc2ccc(C)s2)=O)CC1n1cccn1 CN1CCCC2(CCN(Cc3conc3C3CC3)C2)C1=O C1(C(=O)NC)C2CN(C(=O)CCN(CCO)C(c3cn(C)cn3)=O)CC12 CC(C)CC(CC(=O)NCC12CCC(CC1)OC2)NC(=O)CC1OCCO1 C(=O)(C(O)C(C(C)C)NC(CCCONC(c1c(CO)cc[nH]1)=O)=O)N1CC1.CS C1(NC(=O)NC2(c3n(C)ncc3)CC2)CS(=O)(=O)C12CCCCC2 Cc1ccc(C(N2CCC(F)(C(=O)NC(C)C(N)=O)CC2)=O)c(C)c1F c1(C(=O)NC2CC(C)(CC)N(C(=O)COCCOC)C2)cc([N+](=O)[O-])c(C)s1 Cc1c(C(=O)NC(CNC(N)=O)C(C)C(C)C)cn(C)c1Br c1(CC(=O)NCC2CCCC2NC(=O)C2=CCCC2)nc(F)c(F)cc1F CC1(C)CCc2sc(NC(=O)NC34CC3CS(=O)(=O)C4)nc21 C=CC(C(=O)NCC1CCCN1CC(=O)Nc1ccncc1)OC C(C(CC(=O)NC(CC1CC1)CO)NC(c1cnc(N)cn1)=O)OC CC1CCCC1CS(=O)(=O)NCCN(c1cncs1)C c1(C(=O)NCC(CNC(c2ccsc2)=O)CO)ccn2cnnc2c1 C=CC1OCCC1C(=O)N(C(C)CCNC(=O)CNC(=O)NCc1ccco1)C c12ccc(cc1)OC1CC(C1)C(=O)NCCNC2=O.C(C(F)(F)F)OCF Cc1ccc(F)cc1CC(=O)NCC1(NC(C23CC(C2)C3)=O)CCCCC1C c1(C(=O)NCCC2CCN(C(CC(C=C)CC)=O)C2)c(Cl)ccc2c1OCO2 c1(C(=O)NCCCNC(C(c2cn(C)nc2)O)=O)cc(F)cc(Cl)c1 C12(C(=O)NC3CCCC(NC(=O)COc4cn[nH]c4)C3)CC3CC(C(=O)N1)C2C3 CCC(C(=O)N1CCCCC(CCC(=O)NC(C)(CSC)CO)C1)C(C)C C1(NC(CCC2(C)CC2)=O)CN(C(C2CCCS2)=O)CC1CO C1(NC(C=CCCC)=O)CN(C(=O)C(=O)NCc2ccc(C)cc2)CC(C)(C)C1 C(C(=O)NCC(C)NC(C12COCC1C2)=O)(C(C)C)SCC n1(CC(N2CCC(NC(c3c(C)snn3)=O)CC2)=O)ncc(C#N)c1Br C(=O)(C(O)CC[S+](C)C)N(C1CCN(C(c2c(CC)cccn2)=O)C1)CCO Cc1nn(C)c(Cl)c1C=CC(=O)NCC(CNC(=O)C=CC1CCOCC1)CO Cc1ccccc1OCCCC(=O)NC1COCC1NC(=O)CN(C)C(C)C c1(N2CC(C)(NC(CC3C(C(=O)OC)C3(F)F)=O)C2)cc(OC)ncn1 C1(c2n(C)ncc2)CN(C(=O)C(C)(C)c2ccn(C)n2)CCN1C(C1CC1F)=O C(C(=O)NC(C1CCCCC1)CNC(=O)CN1CC(F)(F)C1)(C(C)C)OCC c1(C(N2CC(C)(C(=O)Nc3c(C)n[nH]c3)C2)=O)cccc(C2CC2)c1 c1(OCC#C)cc(CNC(=O)NC2CCCSC2)cc(Br)c1 c1(OC)cc(C)c(NC(C2CC2C2CN(C(c3csc(Cl)c3)=O)C2)=O)cn1 C1(C(=O)NCC2(CC)CCC(=O)N2)CCCN1NC(=O)C1CSC1 c1(C(=O)NCCC2CCN(C(c3cc(SC)oc3)=O)C2)cc(C)n(C(C)C)c1C C1(c2cn(Cc3cccc(C)c3)nn2)CN(C(=O)Cn2nccn2)CCN1C Cc1ccc(F)cc1NC(=O)C(N1CCN(c2nc(C(F)(F)F)cs2)CC1)=O C1(CNC(c2cocn2)=O)CCCN(C(C2CCCN2CC(F)(F)F)=O)CC1 C(=O)(C1=NNC(=O)CC1)NC1C(SC)CN(C(=O)C(F)(F)c2nccs2)C1 N1(C(CCN(CC)CC)=O)CCC(CNC(=O)C(C)N(C)C)(COC)C1 Cc1cc(CCC(=O)NC2CC3CC2N(C(c2csc(CO)n2)=O)C3)cc(C)c1 C1(NC(CC2(C=C)CCC2)=O)CCN(C(c2csc(C(F)(F)F)n2)=O)CC1 N1(C(c2cn(CC)nc2)=O)CCC(F)(CNC(=O)C(C)=CC2CC2)C1 c1(C(=O)NCC2CC(C)N(C(c3ccc(C(F)F)cc3)=O)C2)cc(=O)cc(Cl)[nH]1 C1(C)(C(=O)NC2CCN(CC)CC2)CN(C(=O)CCc2nccn2C)C(C)(C)C1 N1(C(COCC)=O)CCC(CCNC(c2ccsc2C#N)=O)CC1C c1(CC)cc(=NC2CCC(NC(C3CCC(=O)N3C(C)C)=O)CC2)[nH]c(CC)n1 c1(C(C(=O)NC(CC)CNC(c2cn(CC)cn2)=O)(C)C)c[nH]c2ccccc12 C1(C2CC2)(NC(C2CC(NC(C3CC4C=CC3O4)=O)CCO2)=O)CCC1 C#CCCN=C(NCC1(O)CC2CCC1C2)N1CC2CCN(C)C2C1 c1(C(N2C(CCNC(=O)CC34CC(C3)C4)CCC2)=O)cnc2[nH]cncc1-2 c1(C(=O)NC2(C)CCN(C(CCCCC)=O)CC2)cccc2occc12 C12(C(N3CC(OC(=N)O)C3)=O)CC(CCO1)N(C(C1CC(=O)CCO1)=O)C2 N1(C(CN(C)C)=O)CCCC(O)(CCNC(C23CC(C)(CO2)C3)=O)C1 c1(CC(=O)NC(C2CN(C(=O)C(=O)NCC(F)(F)F)C2)C)ccnc(F)c1F c1(C(N(CCCNc2nc(-c3ccccc3)no2)CC)C)ccccc1OC C1(C(=O)Nc2c(SCC)cncc2)CCC2(CC1)CN(C(=O)C(C)(O)C(C)C)C2 N1(C(CC2=C(C)CCC2)=O)CCN(C(c2ccn(C)c2C)=O)CC2CCCCC12 C(C(C)CN=c1cc[nH]c(-c2nccs2)n1)NC(C(CC)CC1CCCC1)=O N1(C(c2cnc(OC)s2)=O)CCCC(C2CN(C(=O)C=C3CCC3)C2)C1 N1(C(C2CC(CCC)C2)=O)CCC=CC1C(=O)N(C(C)C(C)(C)O)C Cn1cc(S(N)(=O)=O)cc1CC(=O)NC1CC1NC(c1c(Cl)ccc(O)c1N)=O c1(C(N2CCN(Cc3c(C)n[nH]c3)C(CC#N)C2)=O)cccc2ccoc12 C1(C(=O)NCC2N(C(CC(C)(C)C3CC3)=O)CC(F)C2)CCOCC12CCC2 C=C=CC(C)C(=O)NCCC1COCCN1C(c1cc(C(=O)OC)co1)=O c1(CC(C(=O)NC(C)CCO)NC(=O)CNC(=O)CN(C)C)cnn(C)c1O c1(C(=O)NCC2CN(C(C3(C)CCCCO3)=O)C2)cc(C(F)(F)F)c(Cl)cn1 C1(NC(c2ccc(CO)cc2)=O)CC12CCC(NC(c1ncccc1C)=O)CC2 CN1CC2(CCN(C(=O)COC3CN(C(C4(O)CC(C(=O)O)C4)=O)C3)CC2)C1 CC1CN2CCN1CC2C(N1CCC(CCNC(=O)CSc2ccncc2)C1)=O C1(C(N2CCC(C(C(=O)NC3CC(CSC)C3)C)C2)=O)C2CCC(C2)C1C C1(CN(C)C)COCC1NC(=O)CC1(NC(C2CNC(=O)C2)=O)CCC1 CC(C)CC(O)C(=O)N1CC2(CC2)CC1C(=O)Nc1c(Cl)cnn1C C1(N(C(c2nc(-c3nc(C)sc3)sc2)=O)CCF)CCCN(C(C2CC2F)=O)C1 N1(C(C2N(CC)CCCC2)=O)CC2CC(NC(C3CC(=O)N(C(C)C)C3)=O)C2C1 C1(C(C#C)NC(C(F)(F)F)C2CCCCC2)CCC(F)(F)CC1 c1(CC(=O)N(C2CCN(c3ncncc3F)C2)C)ccc(F)c(Br)c1 c1(-c2ccc(C)cc2C#N)cc(C(=O)Nc2ncc[nH]2)c2cc[nH]c2c1 C(C(=O)N=c1cc[nH]cc1)OC(CN(C)Cc1ccccc1)(C)C1CC1 C1(C(=O)NCC(C)NC(=O)Cc2ccc(CN(C)C)o2)(CN(C)C)CCCC1 C=Cn1ncc(C(N2CC(O)(C(F)C(=O)NC3CC3C(F)(F)F)C2)=O)c1N C(=O)(C(C)(C)CC(C)C)N1CC(C)CC(CNC(CCN(CCC)C)=O)C1 CC1(C)Cc2ccccc2C1NCc1n[nH]cc1Br CC1CN(C(c2csc(C(F)(F)F)n2)=O)C(C)CN1C(=O)COCCCN=[N+]=[N-] c1(C(=O)NCC(C)(C2CCC2)NC(=O)C2=CCCCC2)nccc2ccsc12 c1(CN(CCNC(C2(CC)CCOC2)=O)C(c2ncoc2C)=O)ccc(Cl)nc1 C(=O)(C(C)C(O)CC(C)C)NCC(N1CCN(C(c2c(C)cncc2)=O)CC1)=O C(=O)(CC1OCc2ccccc21)NCC=CCNC(C(CN(C)C)O)=O C(c1nccs1)=CC(=O)NC1CC(CNC(C2(CF)CCC2)=O)C1 CCCC(C)CN=c1cc[nH]cc1S(=O)(=O)N1CC2C(C1)C2(C)C N1(CC)CC2CN(C(=O)CC3CCCN(C(=O)CCCCN)CC3)CC2C1 N1(C(C(C)(C)SC)=O)CC(C(=O)NCCc2cnc(C)s2)CC(C)(C)C1 c1(C(N(C2CC(NC(C(CC)C(C)(F)F)=O)C2)C)=O)c(F)ccc2c1OCC2 c1(COCC2C(C)C2)ccnc(CO)n1.C12CCN(C1)CCCNC2=O.C(C)(C)C c1(C(N2C(C)CC(CNC(=O)CNS(C)(=O)=O)C2)=O)cccc2cnsc12 c1(OC)c(C(=O)NCCCCN(C)C(C2CC23CC3)=O)occc1=O C1(C(NOC(CC)C)=O)(CC)CN(C(=O)CC2CCCCC2)C1 CCCCC(O)CNC(=O)C(c1cnn(C)c1)NC(c1ncoc1C)=O C1(CNC(C(C)Cc2ccccn2)=O)CC(C)N(C(C2CC(F)(F)C2)=O)C1 S(=O)(=O)(c1cccc(N(C2CC2)CCNc2cn(-c3cccc(Br)c3)nn2)c1)N(C)C C(C(=O)NC1CCC(F)(CNC(c2nc(O)c(C)s2)=O)C1)(C(C)C)SC C1(O)(CNC(C2(N(C(c3cnn(C)n3)=O)C3CC3)CCC2)=O)CCOCC1 C1(NC(C(C)OCCCC)=O)C2COCC1CN(C(=O)CCc1ccn(C)n1)C2 Cn1ncc(C(=O)NCCNC(c2cc(-c3ccccn3)no2)=O)c1N N1(C(c2ccccc2S)=O)CCC2CN(C(=O)Cc3ccc(Br)cc3Br)CC12 c1(CC)cccc(C)c1C(=O)NCC1(COC)CN(C(c2ccn(C)n2)=O)C1 N1(C(CC(=O)NCC)=O)CCOC(C(C)NC(C2(C)CS(=O)(=O)C2)=O)C1 C1(NC(=O)CCNc2ccccn2)CCCN(C(=O)C=CSc2nc[nH]n2)C1 c1(CN2C(C(=O)NCc3ccc(Cl)c(O)c3)CCCC2)c[nH]c2ncccc12 c1(C(=O)NC(C)CCNC(=O)CC2CC(C)(C)CO2)cc(Cl)cc(Br)c1 CC1=C(C(=O)N2CCOC(C(C)NC(C3CC(F)C3)=O)C2)Cn2nnnc2N1C Cc1nc(C(N2CCCC2CNC(C2CC23CCOCC3)=O)=O)c2ccnc-2[nH]1 CC1CCCN(C(C2NC(=O)CC2C)=O)C1CNC(c1nc(=O)cc(N)[nH]1)=O c1(SCC(=O)NCc2scc(CNC(C(CC)(C)O)=O)n2)nc(C)cc(C)n1 Cc1nc(NCc2ncc(C(F)(F)F)[nH]2)cc(=NCC2CN(C)CCN2C)[nH]1 Cc1nc(C(N2CCCN(CCNC(=O)CCC3CC3)CC2)=O)c2ccccn12 Cc1c(NC(=O)N(C)C)cccc1C(N1CCC(Cc2ccccc2)C1)=O c1(N2C(C(=O)N(C)CCOC(C)(C)C)CC(OC)C2)ncnc2cnn(C)c12 N1(C(C(C)C2(O)CCC2)=O)CCC(C)(C(=O)NCC(O)Cn2cccn2)CC1 CC(C)(O)C(C)(C)C(=O)NC1CCC1C(N1CCCC(F)(CO)C1)=O N1(C(CC(N)Cc2cc(Cl)ccc2Cl)=O)CCOC2(CCCC2)C1 C(=O)(CC1=NN(C)C(=O)C1)N(c1cc(Cl)ncc1[N+](=O)[O-])C(C1C(C)CNCC1)=O c1(C(=O)NCC2CN(C(CC(C=C)C)=O)C2)c(F)cc(O)cc1F c1(C(C2(C)CC2)NC(c2n(CC=C)nnn2)C(C)CC)cccc(Cl)c1 c1(CCC(N2CC(CN(C(CN(C)CC)=O)C)C(O)C2)=O)cccc(OC)c1F n1(COC)nc(C)c(NC(C23CC2CN(C(c2ccoc2)=O)C3)=O)c1C N1(C(CCN(C(C)=O)C)=O)CCc2ccc(CC(=O)NCCN(C)C)cc2C1 c1(C(N2CCC(N(C(=O)CCn3ccnn3)CCO)C2)=O)csc2ccccc12 N1(C(c2cnc(C)nc2)=O)CCCCC(CNC(C2CC(C(C)C)C2)=O)C1 N1(CC2OCCCN(C(=O)OC(C)(C)C)C2)CC(=O)N(CCOC=O)C(=O)C1 N1(C(C2CCCC(F)(F)C2)=O)CCC2(CCCN(c3cc4nncn4cn3)C2)C1 C1(C(N(C(c2ccccc2)CNC(C2CCCC2)=O)C)=O)CCC12CCCO2 CC1(C(=O)NCCN2CCC(NC(=O)CCC3CC3(F)F)CC2)CCCS1(=O)=O c1(NC(CNC(=O)NC(c2ccccc2)C)=O)cc(I)c(Br)cc1Cl N1(C(c2n(C=C)ncc2)=O)CCN(C(c2ccc(OC(F)F)cc2F)=O)C2CC12 C1(C)(NC(C2C(COC)C2)=O)CCCN(C(=O)Cc2csc(S)n2)C1 C(=O)(C(C)CCCCCC)N1CCC2(CN(C(CC(C=C)c3ccccc3)=O)C2)C1 c1(OC)ccc(CN2CCOCC2)cc1C(=O)NCCF Cc1ccc(C)c(C(N2CC3CC(O)C2C3NC(=O)CC2(C)CCCC2)=O)c1C O=C1CCC(CCC(=O)NCC2CCN(C(=O)Cc3ccccc3)C2)C1 Cc1cnc(C(N2CC(C)(C(N3CCC3c3cccnc3)=O)C2)=O)c(F)c1 c1(C(=O)NC(CC)(CNC(=O)C(C)(CC)C(N)=O)CC)ccc2nc(C)[nH]c2c1 C1(NCC(CC)C)COCCN1C(=O)C(=O)N(C1CCN(S(=O)(=O)CC)CC1)C CCC(CNC(=O)C=Cc1cc[nH]n1)(CC)C(=O)NCC(O)(CO)CO N1(C(c2nc(CNC(C3(C#N)CC=CC3)=O)oc2)=O)CC2CCCC(C2)C1 Cc1c(Br)c(C(N2CCC2(C)C(N2CCC(F)C2)=O)=O)nn1C C(CS(=O)(=O)Cc1cn(-c2cnn(-c3ccccn3)c2)nn1)C(N)=O N1(c2nnc(SC(c3cnn(C)c3Cl)=O)n2C)CCCC(C)(C)C1CCO O=C(NOCCCO)C(CNC(C1(O)CCC1)=O)CC1CCCC1 N1(C(c2c(CC=C)cccc2)=O)CCC2(CCN(C(C3CC3C)=O)C2)C1 CC1(C)CCC(S(=O)(=O)N2C3CCC(C3)C2C(=O)O)CC1 C1(NC(CCNC(=O)NC)=O)CCC(C)(CNC(=O)Cc2ncoc2C)C1 c1(OC)c(F)cc(F)c(CN2CC3(CC3)CC2C(=O)N=c2[nH][nH]cc2I)c1F C1(C2(NC(=O)CC(C(F)F)NC(c3ccc(F)cc3F)=O)CC2)(OC)CCC1 C=CCCCCCCC(=O)N1CCC(C)(NC(c2cc3n(n2)CCCC3O)=O)C1 C1(NC(c2cccc(OCC)c2)=O)CCN(CC(O)CNC(N)=O)C(C)C1 C12(C(N3CCC(C(C)NC(C4(C(C)(F)F)CC4)=O)CC3)=O)CCCCC1C2(F)F N1(C(C=CCN(C(C(C)CC#N)=O)C)=O)CC2(CCC2(C)C)C1 Cn1c(CNC(c2cc(Cc3ccccc3)[nH]n2)=O)nnc1C1CCC1 C1(CNC(C2C(C(C)C)C2)=O)CCC2(CCN(C(c3cnc[nH]3)=O)CC2)O1 Cc1nnc2ccc(C(=O)N(C(C)CNC(=O)C(F)CC(C)C)C)cc2c1C C1(C(=O)NCC(CN(C(=O)CNC(=O)C(F)(F)F)CC)(C)C)CC(=O)OC1(C)C c1(C(=O)NCCOCCCNC(c2c(CCC)[nH]cc2)=O)cc2cnn(C)c2s1 c1(SC)snnc1C(=O)NC(c1ccccc1)C1CCC1CN N1(CC(=O)NC2CC(CC(=O)N(C)CCN3CCOC3=O)C2)CC(=O)NC1=O CCCC(CCNC(=O)C(C)NC(c1nocc1C(C)C)=O)CCC c1(C(=O)NC2C(NC(C3(C)CCCC3)=O)CS(=O)(=O)C2)cc2n(c1)CCCC2 N1(C(c2cnc(C(C)C)nc2)=O)CCN(C(C2CCCCO2)=O)C(C(F)(F)F)C1 c1(C(N2CC(C(=O)NCc3c(CC(=O)OC)cccc3)C2)=O)cc(Cl)ccc1I c1(NC(C)=O)ccc(C)c(C(N2CC(C)(NC(c3cccc(C)c3F)=O)C2)=O)c1 N1(C(CCc2nc(C)sc2)=O)CCOC(C(C)NC(C2(c3ncco3)CC2)=O)C1 Cc1noc(C)c1CNC(C1(NC(C2CC(=C3CCC3)C2)=O)CCSC1)=O CCC(CC(=O)NCC1CCCN1C(=O)C(c1ccc(F)cc1)C)C12CC(C1)C2 N1(C(C(C)(C(C)C)OC)=O)CC2CCC1C1CN(C(=O)CCC(C)C)CC21 c1(C(N2CCC(NC(C)=O)C2c2ccccc2)=O)ccc2c(c1)CCC2(F)F N1(C(CCc2cc(OC)no2)=O)CCC(N(C(=O)C(CCO)N(C)C)CC)CC1 C1(C(=O)NC2C(OCC)COC2)C2CC(O)C(C2)N1C(=O)C1=CCCC1 C1(C(=O)OC)CC(C)CN(CC(N2CCCC(C(=O)N(C)C(C)C)C2)=O)C1 c1(N(C(C)CNC(CC(OCC)OCC)=O)CC)ccc(F)c(SC(F)(F)F)c1 N1(C(C2CCC(OC)(OC)C2)=O)CCC(NC(=O)CCC2(C)CC2)C(CO)C1 c1(C(N2CCC(CNC(C(C)SCC)=O)C2)=O)cc(Cl)ccc1C(F)F CC(N=c1[nH]c(=NCC2(N(C)C)CC2)[nH]c2c1CSC2)C1CCOC1 c1(C(N2CC(NC(C(CCC)OC)=O)C(C)C2)=O)cc(=O)c2ccccc2n1C c1(SCC(=O)NC(C)C(C)NC(=O)C(C)(C)C2CCCCC2)nnnn1C C1(C(C)C)CCCCC1NC(=O)CCc1cc[nH]n1 CC1CCC(CC(=O)NCC2(F)CC(CNC(c3cn(C4CC4)nn3)=O)C2)O1 C1(CNC(C(C)N(C)C)=O)(NC(C2C3CC4C(C3)C24)=O)CC2CCC1CC2 c1(C(C)C)cc(NC(C)C(C2CCCCC2)NC(C2CN(C)CCO2)=O)ncn1 N1(C(c2c(C)c[nH]n2)C(=O)NC2CCOC2)Cc2ccccc2N(C)CC1C c1(C(N2CCC(CNC(CSC)=O)C2)=O)ccnnc1C Cc1ccc(C(=O)NC2CC(C)CN(C(C3CCOC(C)(C)C3)=O)C2)c(N)c1C C1(OC)(CNC(C2CCN2C(C)C)=O)CCN(C(=O)C(C)(O)C2CCC2)C1 c1(CC(=O)NC2(CNC(C3CCCO3)=O)CCC2)cc(F)c(F)c(F)c1 CC(=NO)C1CC(C(=O)NCCN(C)C(c2ccsc2Br)=O)C1(C)C C1(C(=O)NC(C)C(=O)NCC23CC(F)(C2)C3)CC2OC1C1CC21 C1(CNC(C(c2cncnc2)C)=O)CC2(CC2)CN1C(c1cscn1)=O C1(CC)CN(C(=O)CC2(O)CCC2)CCC1NC(=O)CC1CC=CC1 Cn1nc(Br)cc1C(=O)NC(CNC(=O)CC12COCC(C1)C2)C1CCC1 CCC(CC)C(C)NC(C12CC(CN1C(=O)CN1CSCC1=O)C2)=O c1(C(=O)NCC(C)N(C(CCCCOCCC=C)=O)CC)cc(CC)n(C)c1C C1(NC(c2c(C(C)C)csc2)=O)CC2(CCN(C(=O)CC3(C)CC3)C2)C1 Fc1cccc2nc(NC3C4CCCCC34)nc(N3CC=CCC3)c12 N1(C(c2cc(C(C)(F)F)ccn2)C(=O)NCCSC)CC(O)C2(CCOCC2)C1 C1(NC(C2C(CC)C2)=O)COC2(C1)CN(C(c1ccc(C(=O)OC)cc1)=O)C2 c1(CNC(N(c2ccc(Cl)cc2)C)=O)c[nH]c(=O)c2ccnn12 C(CCC(C(=O)NCCC1CC(C)(C)C1)NC(c1c[nH][nH]c1=N)=O)OC C1(C(=O)NCC(C)(C)NC(C=CC(C)(C)SC)=O)CC2(CCCCC2)CO1 C1(CNC(C2CCCCC2O)=O)CCCC(NC(=O)C(c2cccnc2)O)C1 c1(C(=O)NC2(C)CCN(C(=O)CC3CCC(=O)N3)CC2)csc2ccncc12 C1(CNC(C2(CCCC)CCC2)=O)CCN(C(=O)CCNC(=O)CO)CC1 N1(C(c2c(C)cc(F)s2)=O)CCN(C(=O)C(C)OC(C)(C)C)CC(C)CC1 CCCCCC(F)C(=O)NOC1CCN(C(=O)CCF)CC1 c1(C(=O)NC2C(NC(CSC)=O)CC(F)(F)C2)cc2c(C)cccc2[nH]1 C1(O)(C(C(=O)NCC(CNC(Cc2c(C)noc2)=O)O)O)CCCCC1 C1(NC(C2CCC(C)(C)C2)=O)CC2CC(NC(=O)CCc3ccc(F)cc3)C2C1 CS(=O)C1CN(C(=O)CCC2CCC(NC(=O)C(C)(Cl)Cl)C2)C1 c1(-c2cn(CC(N3CCC(N4CCOCC4)C3)=O)nn2)ccc(F)c(C(=O)O)c1 CC(C)(CC(F)C(=O)N1CCC2CN(C(=O)CS(N)(=O)=O)C2C1)C1CC1 c1(C(C)OCC)nc(C)c(C(=O)NC2CCCC(NC(c3cc(C)ns3)=O)C2)s1 CC1=C(C(=O)NC2CCCC2C(=O)NCC2CCC(=O)N2)CCC1 C1(C(C)C)(c2n(CC=C)nnn2)CC1.C1(CCOC)(CN)CC1 C1(C)(CNC(=O)OC(C)(C)C)CCC(C(=O)Nc2nccc(-c3ccccc3)n2)C1 C1(C(C)C)CN(C(=O)C(C(C)(C)C)N(C)C)CCCN1C(=O)CS(=O)(=O)N(C)C N1(C(Cc2nccc(C)c2)=O)CCC(N)C(F)(F)CC1 N1(C(C#CC(=O)N(C)C)=O)CCC(NC(=O)C=CC(C)(C)SC)C(F)C1 N1(C(c2ccccc2C(F)(F)F)=O)CCC(O)C2(CC2)C1 c1(COCCOc2ccccc2)nc(C)cc(N2CCN(C(=O)OC)CC2)c1C C1(C(=O)NC(CC)C(=O)N2CCC(COC(C)=O)C2)COC(=O)N1C c1(C(C)C)ncc(Br)c(C(=O)NCC2COCCN2C(C2C=CCCC2)=O)n1 N1(C(C(C)C)=O)CCCCCC1C(=O)NCC1CC2CCC2C1 Cc1cc(C)c(CO)cn1.C12(CCOC1)C(=O)N2.C12CC(C1)OCC(=O)N2 c1(C(=O)NC2CCN(C(C3(C4CC4)CCCO3)=O)CC2O)cccc2c1OCO2 C1(C#N)(C(N2CC3N(C(C(CC)(C)COC)=O)C(CC3)C2)=O)CC12CCOCC2 C1(N(C)C(C2CCCNCCC2)=O)CC2CCC(C1)N2C(=O)C(=O)NCC1CC1 c1(C(N(C2CCC(NC(CC=CCC)=O)C2)C)=O)ccc(C(=O)NC)c(F)c1 c1(CN(C)C(C2(N(C)C)CC2)=O)ccc(CNC(c2nscc2Br)=O)cc1 c1(C(N(CCC(C(C)C)NC(C)=O)C)=O)ccc2c(O)nncc2c1 N1(C(CN(C2CC2)CC)=O)CCC(NC(=O)C(C)Oc2ccccn2)C1(C)C C1(NC(CN(C(COCCOCCOC)=O)C)=O)CC(SC(F)F)C1 c1(CC(N2CCC(NC(c3ccoc3C3CC3)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 C1(CCC)(NC(=O)Cn2cncn2)CCCN(C(C2CCC2c2nc[nH]n2)=O)C1 Cc1ccc(Br)cc1C1CC1C(=O)NC1(CNC(=O)C2=CCC2)CCOC1 C1(C(N(CCCNC(C(C)SCC)=O)C)=O)(COCC)CCCCO1 C(CC(C(C)C)NC(C1(C2CC2)CCCO1)=O)N(C(c1cc(C)sc1)=O)C c1(OC(C(=O)NC(C2OCCN(C(C(C)OC)=O)C2)C)(C)C)ccc(F)c(F)c1 C1(C(N(CCCN(C)C)CC)=O)CCCCN(C(=O)C(COC)OC(C)=O)C1 N1(C(C(CC)F)=O)CC2CC2(NC(=O)CCc2c(C)noc2C)C1 C1(C(=O)NC)(NC(=O)CCC23CC2CCN3)CCCCC1 c1(C(N2CCCC3(COC3)C2)=O)cnc2n[nH]c(-c3ccccc3F)c2c1 CCCCS(=O)(=O)CC(=O)NC1CCOCC1NC(=O)Cc1sc(O)nc1O C1(C)(C(=O)NC(CC(=C)C)C(=O)OC)CN(C(C2(SC(C)C)CC2)=O)C(C)(C)C1 C(=O)(C(C)CC(=O)NCCCOCCC(=O)N(c1ccc(O)cc1)C)OC c1(NC(C2CCCN(Cc3cc[nH]n3)C2)=O)c(O)cccc1F C1(CNC(c2c(C(C)NC(c3ccn(C(F)F)n3)=O)n[nH]c2)=O)CCN(C)CC1 N1(C(c2coc(CO)c2)=O)CC(NC(C2CS(=O)(=O)C2)=O)C(c2ccncc2)C1 C1(C(N2C(C)(CC)CCC2)=O)CN(C(=O)CCN(C)C)CC12CCC2 N1(C(C2(S(C)(=O)=O)CC2)=O)CCCC(NC(=O)C(=Cc2cccc(F)c2)F)CC1 c1(CCC(N2C3CC(NC(CCOCCN(C)C)=O)(C3)C2)=O)ccc(N)c(F)c1 C=C=CC(C)C(=O)NCC(C)CN(C(=O)CCC=C=C)C C(=O)(CCCC(C)(C)NC(c1cccnc1O)=O)NC(C)CCN(C)C N1(C(CSC)=O)CCN(NC(=O)CNC(C2CC(CN(C)C)C2(C)C)=O)CC1 C1(CC(=O)N(CC(N2CCC(OCC=C)C2)=O)CC(C)C)CCCOCC1 C(=O)(C(F)(F)C(O)CC)N(C)CC1CCN(C(CS(=O)(=O)N(CC)CC)=O)CC1 c1(C(C)NC(c2c(C(CC)(F)F)cccc2)=O)cccc(F)c1F N1(C(c2c(F)ccc(C#C)c2)=O)CCOC2(CCN(c3nc(SC)ns3)C2)C1 c1(C(=O)NCC2(O)CCCN(C(C(CCSC)O)=O)C2)cccc2c1OCC2 N1(C(C(C)(C)O)=O)CCC2(CC1)CN(S(=O)(=O)CC#N)CCO2 Nc1c(C(=O)NCC2(NC(=O)CC3CCC(O)C3)CCOCC2)cc(F)cc1F c1(-c2cn(CCC(C)C)nn2)ncc(C(N2CCC(O)(C(F)F)C2)=O)n1C c1(OC)ccc(CC(C)C(=O)NC2CCC2NC(=O)CN2CC3CC3C2)cc1 Cc1csc2ncnc(NC3CCC3C(C)C)c12 c1(NC2CC3CN(C(CC4CCC(=O)NC4)=O)CC32)ncc2scc(Br)c2n1 c1(C(N)=O)coc(C(=O)NC23CC(NC(C4CCC(C(N)=O)C4)=O)(C2)C3)c1 c1(OC)ccc2c(CN3C(C(=O)Nc4cccc(C)c4O)CC4CC34)c[nH]c2n1 c1(C(N2C3C(NC(CC(CC)C)=O)CC(CC3)C2)=O)[nH]c2c(c1C)C(=O)CCC2 Cc1cccc2ccc(CNC(c3cccc(F)c3)CCO)nc12 N1(C(CNS(CC)(=O)=O)=O)CCC(CO)(CNC(C2(O)CCCCCC2)=O)CC1 C1(NC(C2CC(=C)C2)=O)(CF)CCN(C(C2(CC)CC2)=O)C1 CC1C(NS(=O)(=O)Cc2ncoc2CN)CC(=O)N1C c1(C(N2CC3C(NC(CCn4c(C)cc(C)n4)=O)C3C2)=O)c(F)cccc1Cl c1(CNC(c2nc(CC)oc2)=O)nc(C)c(C(=O)NCCC2CCCC3CC23)o1 C1(C)(C(=O)NCC(CC)NC(=O)CC23COC(CSC)(C2)C3)CCSCC1 C(CCNC(=O)C(CC1CC1)NC(C1(OC)CCCCC1)=O)(C(C)C)OC C1(CC=C)(NC(=O)C=CCSC)CCN(C(=O)C(C)COc2ccccc2)CC1 c1(CC(=O)NCCC2N(C(C3COC(=O)O3)=O)CCCC2)ccc2n[nH]cc2c1 c1(C(=O)NC2CN(C(c3scc(C)n3)=O)CC2C)ccc2ncn(C)c2c1 c1(CN2CCC(OC(C3(COC)CCCO3)=O)C2=O)cc2cccc(C)c2[nH]1 C1(CCOC)(NC(=O)CCCC(C)O)CCN(C(c2ccncc2SC)=O)CC1 C1(C(=O)OC)CC(COC)CN(C(N2CC3CC3C2)=O)C1 C12(C(N3CC4C(NC(=O)C=CCCc5ccccc5)C4C3)=O)CC3CC1C2C3O N1(CC2(NC(C3(C(=O)NC4CC(CC)C4)CC3)=O)CCOC2)CCCS1(=O)=O c1(C(=O)NCC(C)(C)NC(CC(COC)C)=O)cccc2c[nH]nc12 N1(C(C23CC(C)(C2)C3)=O)CCOC(CNC(c2sc(Br)cc2Cl)=O)C1 Cc1nc2c(o1)CCCC2CC(=O)N1CC2CC2(NC(=O)CC=C(Cl)Cl)C1 C(CCCC(=O)NC(C(=O)N1CC(c2cccs2)C1)c1ccco1)OC Cc1ccc(C(N2CCC(C)(C)C2CNC(C2CCCCO2)=O)=O)nc1O C1(C(=O)NCC2(OC)CCCC2)CCOCCN1C(=O)C(C)C1CCC1 C12(C(N3C(CN(C(C4C(C)OCC4)=O)C)CCC3)=O)CCCC1C2(F)F C1(NC(C(=O)NCC(CC2CC2)C(=O)N2CCC(C(F)F)C2)=O)CC(=O)C12CCC2 C1(NC(CNC(=O)OCC)=O)CN(C(=O)CSc2ccccc2)CC2(CCC2)C1 CC(CCCCNC(C1CCCC(C)C1)=O)NC(=O)CC1COCCO1 C12(CNC(CN(CC)CC)=O)CCCC1CCN2C(=O)C=Cc1ccncn1 N1(C(C(F)=CCC)=O)CCC(NC(C2(COC(C)C)CC2)=O)CC(C)(C)C1 C1(NC(CCOc2ccc(C)cc2)=O)CCN(C(=O)CCOC2CC2)CC1CO c1(C(=O)NC2CN(C(Cn3c(C)cc(C)n3)=O)C(C)C2)ccc(C(C)=O)c(C)c1 c1(CC(=O)NC2CC(C)(CNC(c3nc(C)sc3)=O)C2)cnccc1C C1(O)(C(=O)NCC(C)CN(C(=O)COc2ccon2)C)CCSCC1 C1(NC(C2(C(=O)NCC=CCNC(C3CCCCC3)=O)CC2)=O)C(F)(F)C12CCC2 c1(C(=O)NCC2(CCNC(CC3CC(C)C3)=O)CC2)ccc(F)cc1F N1(C(C2(CSC)CC2)=O)CCC(CCNC(=O)CCc2ccc(O)cc2)CC1 Cc1cnn(C)c1CNC(C1CC(CCNC(=O)C(F)C(C)C)C1)=O N1(C(c2ccc(CC)nc2)=O)C2CCC1CC(NC(C1CCN1CC)=O)C2 c1(COC)cccc(CC(=O)NC2(C)CCC(NC(C3CSCCS3)=O)C2)c1 C1(NC(C2CCCC2)=O)CN(C(c2cn3ccccc3n2)=O)C2(CCCC2)C1 CC(C)(C)C(CNC(C1CC12CCC2)=O)NC(c1cnn(C2CC2)c1Br)=O c1(NCc2c(C(=O)OC)ccc(Cl)c2)nc2ccccn2c1C1=CCCCC1C CC1CCC(NC(=O)CCc2ccsc2)CN1C(=O)Cn1cccc1 N1(C(C(OC)OC)=O)CCN(C(=O)CCc2ccc(C)nc2)C(CF)C1 CCC(CC)C(=O)NCC(=O)NC1(C2CCCCN2C(=O)C=C2CCCC2)CC1 Cc1ccc(C)c(C(=O)CCC(=O)N2CC(NC(c3cncn3C)=O)C(C)C2)c1 C(=O)(CCCS(N)(=O)=O)NCC1CCC(C)N(C(C2CC3C=CCC(C2)C3)=O)C1 C1(OCC)CCCC1CC(=O)N(C(C)C(=O)OCC)CC1CCCO1 C(=O)(C(C(C)C)SC)N1CC(C(C(=O)NCC=CCOC)OC)C1 CC1CCCCC1(CNC(=O)C(C)(C)C(N)=O)NC(=O)C=C1CCCCC1 N1(C(c2ccc(SC)o2)=O)C2CCC1(CNC(C1(C)CCNC(=O)C1)=O)CC2 n1(CC)nc2c(c1C(=O)NC1CN(C(C3(C(N)=O)CC3)=O)CCC1F)CCCC2 N1(C(c2cc(CC)[nH]n2)=O)CCOCC(NC(=O)CN2CC(C)(C)C2)C1 c1(C(N2CC3C(NC(Cc4cnn(C)n4)=O)C3C2)=O)c[nH]c2cccnc2c1=O c1(C(N2CCC(N(C(=O)COc3ccn(C)n3)C)C2)=O)cnc2cccnn12 c1(C(=O)OCC)cc(C)n(CCCNC(c2nccc(C3CC3)n2)C)c1C Cc1csc(=NCC(=O)NC2(C)CN(C(c3cnn(C(C)C(C)C)c3C)=O)C2)[nH]1 C1(NC(C2(CCCC)CCC2)=O)(COC)CCN(C(c2ccncn2)=O)C1 C(=O)(CC(C)(C)C)NCC1C(NC(C(CC2CC2)OC)=O)CC1 C12(C(N(CCCCN(C(=O)CSCc3ccccc3)C)C)=O)CCC(CC1)OC2 C(=O)(C(C)(C)C(C)(C)C)NC1CCCN(C(C(c2cccnc2)N(C)C)=O)CC1 N1(C(C2CC=CC2)=O)CCC(CC2COCCN2C(C2CC=CCC2)=O)CC1 c1(C(N2CCC(NC(C3(CC=C)CC3)=O)C2)=O)ccc2ncccn12 N1(C(C(C(=O)OC)C)=O)CCCC12CCN(C(c1nccnc1C)=O)C2 N1(C(c2n(CC=C)ccc2)=O)CC2CCN(C(=O)C=CCOC)C2C1 CCCCC(C(=O)NC1CCC(C)N(C(C2CCN(CC)CC2)=O)C1)N(C)C CS(=O)(=O)c1ccccc1CNC(=O)C(=O)NCC12CCCC(CC1)N2 c1(C(N2CCCC(C(=O)NC3CC3C3CCC3)C2)=O)cc([N+](=O)[O-])n[nH]1 c1(OC)ccc2cc(C(=O)NCCN(C(C3CC4CC4C3)=O)C3CC3)ncc2c1 C=CCCCCC(C(=O)NC(C)(C)C)N1CCC(c2cccc(OC)c2)C1 C(=O)(CS(=O)(=O)CC(C)C)NC1C(NC(c2c(C)oc(Cl)n2)=O)COCC1 N1(C(c2n(C)nc(Br)c2)=O)CC2CCN(C(=O)CCc3ccon3)CC2C1 CC1(NC(=O)CNC(c2ccc(F)cc2)=O)CCCN(C(=O)CC=C(Cl)Cl)C1 C1(CC)CN(C(=O)C(C)(C)CF)CCN1C(=O)CSc1c(C)n[nH]c1C C#CC1CC2(CC2)CN1C(=O)CCCCCCNC(c1c(F)cccc1F)=O C1(CC(=O)NC2C(NC(=O)CCc3cccnc3F)C2)CCc2sccc2C1=O C(=O)(C1=Cc2ccccc2OC1)NCCCCCCN(C(CCSCCC)=O)C n1(C(C(=O)OC)C)cc(C(C)N(C(=O)C(Cc2ccccn2)NC(C)=O)C)nn1 c1(CCN2CC(O)(CNC(C3N(C(=O)NC)CCCC3)=O)C2)cccc(Cl)c1F c1(CC)ccc(C(=O)NC2(CNC(=O)C(C)=C3CCOC3)CCCC2)o1 N1(C(C2(C#C)CN(C(=O)Cc3ccccn3)C2)=O)CCn2ccnc2C1C C1(NC(C2(N(C)C)CCC2)=O)CCN(C(c2c[nH]c(Br)c2)=O)CC(O)C1 C1(SC)CCC2(CC1)CCN(C(C1N(c3snc(CC)n3)CCC1C)=O)CC2 CC1CCCC1C(=O)NCC1(F)CC(NC(=O)COC2CCOCC2)C1 N1(C(c2cc(C)c(C)o2)=O)CC2CN(C(=O)C(C)c3ncco3)CC2(C)C1 c1(C(=O)NCC2N(C(CCSCC)=O)CC2)cncc2ccccc12 C(=O)(C(CC(C)C)ONC(C1CCN(C)C1)=O)NC(CCCC)(C)C c1(C(=O)NC2C=CCN(C(C3CC3F)=O)C2)cc([N+](=O)[O-])cc2ccccc12 C1(=O)C(C(C)C(C)(C)C)N2CCOC(C2)N1.N1(CCSC)CCOCC1 C=CC1(CC(=O)NC2(COC)CN(C(c3cnc(C4CCCO4)s3)=O)C2)CCC1 c1(CN=C(NC(CC)CC)NCc2nc(C3CC3)n[nH]2)ccc(Cl)c(N)c1 C(=O)(C(F)C(C)(C)O)NCC(C1CCN(C(=O)CC2(c3ccon3)CC2)CC1)C c1(C2(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)CC2)cccc(C#N)c1 c1(SC)cccc(F)c1C(=O)NC1CC(N(C)C(C2CCCN(C)C2)=O)C1 c1(C(=O)NC(CC)CNC(C2(C)COC2)=O)ccnnc1O CC1CCN(C(=O)CC2CCOCC2)C1C(=O)NOC1CCC1 C12(C(=O)NCC(CC)N)CC3CC(C1)CC(O)(C3)C2.c1(C(=O)N)ccc(COC)s1 C1(N(C(c2ccccn2)c2nnnn2CCCSC)CC)C2CCOC2C1(C)C Cc1c(C(=O)N(C)CCN(C)C(C2CC2[N+](=O)[O-])=O)sc2nccn12 c1(-c2cn(-c3ccn(C4CC(C(=O)NCC)C4)n3)nn2)ccnc(F)c1 Cc1nc2ncccn2c1C(=O)N(C1CC2CC1CN2)c1cc(Cl)n[nH]1 C(=O)(C(O)CC(C)C)NCC1(O)CCN(C(c2ncn(CC)c2)=O)C1 O=S(=O)(c1ccc(Br)cc1NCCCC1CC1(Cl)Cl)NCCN1CCC2(CC1)CC2 c1(CNC(c2ccccc2C(F)(F)F)=O)ccc(F)nc1Br C1(CNC(CCC)=O)CN(C(c2nc(Br)c[nH]2)=O)CC12CCC2 N1(C(C2CC(OC)C2)=O)CC(C(=O)NCC(=O)NCC(F)F)CCC1(C)C c1(N2C(=O)CC(C(=O)OC(C)(C)C)C2)ccc2c(c1)OC(F)(F)O2.CC1C(=O)N1 c1(OCC)ccc(CC(=O)NC2CCN(C(=O)CCc3ncccn3)CC2)nc1 CC1CCN(C(=O)C=CC2CC2)C(C(=O)NOCC)C1.c1(C(C=O)O)cccnc1 c1(C2(C(=O)NC3(C)CC(C)C3)CCC2)ccc(-c2nn[nH]n2)cc1F C1(CCC(=O)NCCOC2CN(C(c3csc(-c4cccs4)n3)=O)C2)CCCOC1 c1(CNC(c2ccc(Oc3ccccc3)c(Cl)c2)=O)ccc2c(Br)cccc2c1 c1(C(N(C2CCCC(NC(=O)C3CC3)C2)C)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] C1(C)(CN(C)C(C2CC2CNC(c2csc(Cl)c2)=O)=O)CCCC1 C(=O)(CC1=CCN(C(=O)C(C)n2cccc2)CC1)N.CC1CN(C)CCC1N(C)C S(=O)(=O)(c1cnc(N2CCC3CC3C2)c(Cl)c1)N(CCCc1ccco1)CC C#CCCN=C(NCCc1cn(C)c2ccccc12)NCC1CCNC(=O)C1 C1(OC)(CNC(c2c[nH]nc2C2CCCO2)=O)CN(C(c2cccs2)=O)C1 CC(CC(F)F)C(=O)N1CCC(O)(CNC(=O)CCOc2ccc(F)c(F)c2)C1 c1(COC)nc(CNC(=O)C(C2CCOC2)NC(C2CC(C)(C)C2)=O)no1 c1(CN(C2CCN(C(C)=O)CC2)C2CC2)cnn(CCCOCCC#C)c1C C1(C(N2CC(COC)(CNC(=O)C=CC(C)C)C2)=O)CCc2ncc(C)n2C1 N1(C(C=C)=O)CCC2(CC(NC(=O)CN3Cc4ccccc4C3=O)CO2)C1 Cc1nn(C)c(C)c1C(N1CCOC(C(N2CCC(O)(C(N)=O)C2)=O)CC1)=O n1(CC)nc(C(C)C)cc1C(N1CC2CC1C2CNC(=O)CCC1CCCO1)=O C1(NC(C(CCCC)C)=O)CCC2(CC1)CN(C(C1C3CCN1CC3)=O)C2 c1(NCCC(=O)OC)ccc(OC)c(C(=O)NN(c2c(CC)occ2)C(C)=O)c1 C(=O)(C(N=C1NS(=O)(=O)c2ccccc21)C(C)(C)C)N1C(OCC)(CC)CCCC1 C1(C(=O)NC(C2CC2C)C)CCN(C(=O)CN(C2CCCC2)C)CC1O N1(C(C2(COC)CC=CC2)=O)CCC2CN(C(C3CCc4ccnn4C3)=O)C2C1 c1(NCc2cccc(C(N(C)C)=O)c2)cc(=NCCCNc2ccco2)[nH]cn1 C=CC1(NC(C2(CNC(=O)CC(C)OC)CCC2)=O)CCOCC1 C1(NC(C(CNC(C2CCCOC2)=O)O)=O)CC2(CCC2)C1O C1(C(C)NC(C2(C3CC3)CCCO2)=O)CCN(c2ccnc(CCC#N)n2)CC1 c1(C(=O)NCC(C)(C)Cn2cc(C3CCC3)nn2)ccc(C#N)c(Cl)c1 C12(NC(CSC)=O)CC(CNC(=O)Cc3ccc(C)c(C)c3)(C1)OC2(C)C C=CCCCCCCC(=O)NC(CO)C(=O)NCCNC(=O)COC C(CC(CO)NC(=O)Cc1csc(-c2ccsc2)n1)=CC N1(C(C(C)c2ccco2)=O)CCC(C2(NC(=O)CN3CCSCC3)CC2)C1 c1(CN2C(C(=O)Nc3ccc(C)nc3)CC(F)C2)ccc(C(F)(F)F)nc1Cl c1(C(N2CCC(CNC(C(C)CC3CCCC3)=O)C2)=O)cc(Br)ccc1O c1(C(N2CC(C(N3C(C=C)CC3)=O)OCC2)=O)n[nH]cc1[N+](=O)[O-] C1(CNC(C(Br)=C(C)C)=O)CC2COCC2N1C(c1coc(C(N)=O)c1)=O C1(C(=O)NC2C(NC(C3(C(F)(F)F)CC(=C)C3)=O)C2)CCC(CO)CC1 C(=O)(C1Cc2ccccc21)N1CC(OC2CCN(C(C(C)(C)O)=O)CC2)C1 C1(C(=O)NCCCCNC(CC(=O)N(CC#C)C)=O)C=CC=CC=C1 CCC(C(=O)NCC(C)(C)NC(C1CCC(C)(C)O1)=O)C(C)(C)CC CC(CCC(C)(C)C)C(=O)NCC1(C)CCCN(C(c2cc(C#N)c[nH]2)=O)C1 Cc1ncc(CC(=O)NCCCNC(=O)C=CC(=O)NC2CC2)[nH]1 Cc1nc(C(=O)NC(Cc2cnc[nH]2)C(N2CC3CC3(CO)C2)=O)cn1C c1(C(N(C)Cc2nnc(C)o2)=O)nc(CNC(=O)CCc2nccn2C)oc1C Cn1ccnc1CN1CCC(NC(=O)NCCCn2cccn2)C1 N1(C(COCCC=C)=O)CCOC(CCCNC(=O)CC2CC=CCC2)C1 Nc1ccc(NC(C2CN(C(=O)CNS(=O)(=O)C3CC3)C2)=O)cc1[N+](=O)[O-] c1(CCC(N2CCN(C(=O)C(F)OC(F)(F)F)C(CO)C2)=O)ccc(F)c(F)c1 c1(NC(C2(C(=O)NCCOCCOCCOC)CCC2)=O)ccc(C)c(F)c1F C1(C(C)C)CN(C(c2ccc(N)c(Br)n2)=O)CCCN1C(C1CC1F)=O C1(C)(C(N2C(CN(C(c3cc(C)no3)=O)C)CCC2)=O)CC(C#N)C1 c1(CC(N2CC3C(C(=O)NC4CC(C(N)=O)C4)C3C2)=O)ccc2c(c1)CC2 C(=O)(C(O)C(C)(C)CC)NCc1cccc(NC(c2nncc(CCC)c2)=O)c1 c1(CN(C(c2ccc(C)o2)C(=O)NCC)CCOCCO)ccc(F)cc1Br C1(CC(N2CCC(=CCNC(CCC(=C)Br)=O)CC2)=O)CC(C)CC(C)(C)C1 CC1CN2CCN1C(C(N1CCC(CCNC(C3(CC4CC4)CCC3)=O)C1)=O)C2 CC(C)CC(C)(O)C(=O)N1CC(n2cc(Cn3ccccc3=O)nn2)C(C)C1 N1(C(=O)Nc2nc(CC)c(C)cc2C#N)C2CCC1CC(N(C)C)C2 Cc1cnc(N(C(=O)CC2CCOCC2)CC2(F)CCCNC2)nc1C c1(CCC(=O)NCC2CCN2C(=O)C=CC2CCC2)ccc(Cl)nc1 Cc1ccccc1CCC(=O)NC1CCC(CNC(c2ccccc2Br)=O)CC1 c1(C(N2CCOC3COCC23)C(=O)NCCOC)cc(C)c2occc2c1 CC1CN(C(=O)C=C2CCOCC2)CC1CNC(c1cnc(C2CC2)nc1)=O c1(OC)ccc(-c2cnc(OCC3CC3)c(C(N3CCOC(C)C3)=O)c2)cc1F C#Cc1cccc(C(=O)NC(C)(CSC)C(=O)NCCCC(=O)OC)c1 Cc1nn2cc(NC(C3CC(CNC(=O)C(C)Sc4ccccn4)C3)=O)nc2s1 C(=O)(CC(O)C(C)(C)C)NCCN(C(C)C)C(C1CCc2nc[nH]c2C1)=O CCC(C)(C)C(O)C(=O)NC1CCN(C(=O)Cc2ccc(OC)nc2)C12CCC2 c1(C(=O)NC(C)(C)C)ccc(OCC2CC2(Cl)Cl)c(F)c1 Cc1sc(C(=O)NCC(C)(CO)NC(=O)Cc2ccc(O)cc2)nc1Br CC(CC(C)(C)C)NC(=NCc1cccs1)NCC(C)(C)CC#N n1(CCOC)nc(C(=O)NC(C)CCNC(C23CCC(CC2)OC3)=O)ccc1=O c1(N(CC(C)NC(c2ccc(N3CCCC3=O)cc2)=O)C)snc(Cl)c1C#N N(C1CCc2ccc(Cl)cc21)C(=O)NC(CSC)C(C)(C)C CC1(C)C=C(C(=O)N2CCC(C(C)(C)C(=O)NC3(C)CCCCC3)C2)C1 N1(C(c2cn(CC)nc2C2CC2)=O)CCC(NC(=O)Cc2ncc(C)s2)C12CC2 c1(NC(CCNC(CC(CC)(F)F)=O)C)cc(C)nc2c(C)cnn12 c1(OC)cnc(Cl)[nH]c1=NC(=O)C1(CNCc2ccc(C)cc2OC)CC1 C1(F)(C(N2CCC(C(CC)C)CC2)=O)CCN(C(c2cc(Cl)no2)=O)CC1 N1(Cc2c(OC)cc(C)cc2)CC2CCN(C(c3cc4ncsc4[nH]3)=O)C2C1 c1(NC(C)=O)nc(C(=O)NCC(C)N(C(=O)Cc2cnn(C(C)(C)C)c2)C)cs1 CC(CCCCO)NC(c1ccc(CNC(C2CCC2(F)F)=O)cn1)=O C(=O)(CC(O)CNC(=O)CC(C)n1cccn1)NC(C)CC1CCCC1 C1(C(N(C(CNC(C(C)CS(C)(=O)=O)=O)C2CC2)C)=O)CCC2C(CC1)C2(F)F n1(CC(=O)NC(CC(C)C)CNC(=O)Cc2ccn(C)n2)nc(Cl)ccc1=O C1(C)(CC)CCCC(NC2CCCCC2n2cccn2)C1 c1(CCC)ccc(-n2nc(C(C)O)nc2CCCn2ccnc2)cc1 O=C(CC(C(F)F)N1CCOCC1)NCC1(c2ccccc2F)CC(F)(F)C1 O=S(=O)(c1cncc(Br)c1)NC1CN(CC2(c3cc(Br)ccn3)CC2)CC(F)(F)C1 O=C(CCCCCNC(C1(O)CCSC1)=O)NCc1ccncc1Cl N1(C(CN(C(C)=O)C)=O)CCC(CNC(=O)C(C)CN(C)C(C)C)C(O)C1 c1(CC(N2CCC(CCC(=O)NCC(=O)NC)C2)=O)ccc2ccoc2c1 C(C(C)(C)CC(=O)NCC(CC1CC1)C(=O)N(CC(C)(C)O)C1CC1)N(C)C C(C(F)(F)C(C)(C)O)NC(C(C)NC(C(C)c1cccs1)=O)=O c1(C(=O)NCC2(NC(CN(C)CC)=O)CCOC2)ccn(CC(F)(F)F)c(=O)c1 CN1CCCC(CCC(=O)N(C(CNC(C2(C#N)CCC2)=O)C2CC2)C)C1 N1(C(CC(C)(C)NC(c2ncc(C#C)cc2C)=O)=O)CCC2CCCCC12 N1(C(CCOC(C)=O)=O)CC(NC(=O)C2=C(Cl)CCOC2)Cc2ccccc21 C1(CNC(c2cn(C)[nH]c2=N)=O)CCCCN(C(C2CN3CCC2CC3)=O)C1 c1(C(N2CC(F)(CNC(C(CC=CC)CC)=O)C2)=O)c(C)c2cnccn2c1C c1(C(=O)NCCC2CCN(C(C3(O)COC3)=O)CC2)cncc2c(Cl)cccc12 Cc1nn(C)c(C(N2CCSCC2C(=O)NC(c2ccc(Br)c(F)c2)C)=O)c1F CC1CCN(C(C23CCC(CC2=O)C3)=O)CC1NC(c1coc(Cl)n1)=O Cc1[nH]nc(C(=O)NC(C)(C)C=CC(=O)NCc2ccnn2C)c1O c1(CNC(=NC)NCC(O)COC(C)(C)C)ccc(N2CCOCC2)cc1 N1(C(c2ncn(CC)n2)=O)CC2CC1CN2C(C1(OC(=O)NC(C)C)CC1)=O CC1CC(C)(C)CCC1NC(=O)C(C)(C)CCCNC(=O)C=Cc1cccnc1 N1(Cc2cnc(-c3cc(C)c(F)cc3)s2)CCC2(CC1)OCCO2 C=C=CC(C)C(=O)NC(C1CCCC1)CNC(=O)CCc1cccnc1Br CC1(C)CC(C(=O)NOCc2cn(-c3cccc(Cl)c3)nn2)CC(C)(C)O1 N1(C(C(C)=C(C)C)=O)CCC(C(N2CCC(CO)C2)=O)C1(C)C C1(COCC)CN(CCO)CCO1.c1(C2CC(N)C2)nnnn1C CC(CC(=O)N(CCCCCCNC(C1CC(C)(C)OC1(C)C)=O)C)C(C)(C)C CC(c1ccccc1Cl)=CC(=O)NCCOC1CN(C(C2CC3CC23)=O)C1 c1(C(N(CC(C)NC(=O)Cc2n[nH]c(=N)s2)CC)=O)nnc2ccccc2n1 C1(NC(C(CSC)OC)=O)CCCC(N(C(=O)C=C2CCN(C)CC2)C)C1 CC1(CNC(c2cccc(C#N)c2)=O)CCN(C(C2CCCS(=O)(=O)N2)=O)CC1 Cc1cc(CC(=O)NC2CC(CCNC(=O)Cc3ccoc3C)C2)no1 Cc1nn(C)c(C)c1-c1cn(CC2C=CCN2C(c2occc2Br)=O)nn1 C1(NC(C2(CNC(CC(C)OC)=O)CCCO2)=O)CCCC(O)C1O c1(OC)ncc(F)cc1C(=O)NC(C1CCCN1C(C1CSCC(=O)N1)=O)(C)C c1(C(N2CCC(CN(C(CC(C)SC)=O)C)C2)=O)cnc(C(C)(C)C)nc1 N1(C(C(N2CCSCC2)C)=O)CCC2CN(C(=O)CCNC(C3CCC3)=O)C2C1 c1(CN(C(=O)NCC(CN(C)C)(C)C)C)cc(Br)c(F)cc1F c1(N(C)Cc2ccc(C)c(C)c2)ccc(S(=O)(=O)NC2CCCCC2F)c(Br)c1 c1(C(=O)NC2CN(C(C=CCC)=O)CC2C(F)(F)F)cnc(SC)nc1O CC(C(=O)N(CCNC(=O)CCc1nccs1)CCc1ccccc1)C(F)F N1(C(c2c(CC)cccc2)=O)CCCC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C1C Cc1cc2ncc(C(=O)NCC=CCNC(c3ccnnc3C)=O)cc2[nH]1 CC1(C(=O)NCC2CC(F)CN2C(=O)C=Cc2cnc[nH]2)CCCOC1 C(=O)(CC(C)P(C)(C)=O)N1C(C)CCC1C(=O)N=c1ccn(-c2ccccc2)[nH]1 C1(NC(c2c(SC)ccs2)=O)CC(C2CCN(C(=O)CNC=O)C2)C1 C=CC(CCC)CC(=O)N1CCCC(C(=O)NC(c2ccsc2)C)C1CC Cc1cc(=O)c(C(=O)N(C2CC(=O)CS2)C)c(C)[nH]1.N12CC(C1)NC2=O c1(CC(=O)NC(C(=O)NCc2ccco2)C2(O)CCC2)cnn(CCF)c1 c1(CC(N2C(CN(C(C(C)NS(C)(=O)=O)=O)C)CC(F)C2)=O)cc(O)nc(O)n1 CN1CCN(C(=O)CCc2nccs2)C(CNC(c2cn(C)c(C(F)F)n2)=O)C1 c1(C(=O)NC2C(NC(C(CC)O)=O)C2)cc(F)ccc1NS(C)(=O)=O N1(C(Cc2cn(C(C)C)nc2)=O)CCCC(NC(C23CC=CC(C2)C3)=O)C1 C12(NC(C3CC(C)C3)=O)CCCC1(F)CN(C(=O)CN1CC3CC3C1)C2 FC1(CSCC2CC(=C3CC3)C2)COC1 C1(CN(C(=O)CCc2cnccn2)C)CCCN(C(C2COCCO2)=O)C1 c1(N(C(=O)OC(C)(C)C)CC)cc[nH]c(=NCCNC(=O)C2=COCCC2)n1 Cc1[nH]c(C#N)cc1C(=O)NCC1(C(=O)NCC2CCCC(C)O2)CC1 N1(C(C(CCCC)(C)F)=O)CC2CCCC(C1)N2C(=O)C(CC)CC(F)F c1(CN2CC(CC(N3CCCC(CO)C3)=O)OCC2)c(O)ccc2ncccc12 CCCCCC(C)CC(=O)NCc1cc[nH]c1C(=O)NCCSCCO c1(C(=O)NC2(CNC(c3[nH]cc(CC(C)C)c3)=O)CCC2)cc(O)ncn1 C(CC)(C(=O)NC1CCCC1NC(=O)C(C#N)C1CC1)=CC c1(C(N2CC(CCC)C(NC(=O)Cc3c[nH]nc3C)C2)=O)cc2cn[nH]c2cn1 c1(OC)cccc(NC(C2CCN(C(=O)CCC(C)O)C2)C)c1C C1(NC(C2CC3(C2)CC3F)=O)CN(C(c2c[nH]c3nccc-3c2)=O)CC12CCC2 c1(C(N2CC(NC(c3ccc(C)s3)=O)C(O)C2)=O)c(O)cccc1Br c1(CC)ccc(C(=O)NC2(NC(c3ccncn3)=O)COC2)cc1Br C1(C(C)(C)CNC(C2CCCC2F)=O)CCCN1C(C1(C2CCCO2)CC1)=O CCC(C)(CNC(=O)CN1CCCC1)C(=O)N1CCC(CCN2CCC2)CC1 c1(C(N(CCN(C(c2occc2C)=O)CC)CC)=O)ccc(C)c2c1CCC2 N1(C(CN(C)CCO)=O)CCC(COC(F)(F)F)C1.N12CC(C1)CC2=O Cc1ccncc1CCNC(C12CC1CN(C(c1ccc(CO)o1)=O)C2)=O c1(CN2CC3CN(C(=O)CCc4cnc[nH]4)CC32)nccc2ccccc12 C1(C(C)C)CN(C(c2cccc(Cl)c2F)=O)CCCN1C(=O)C1=NNC(=O)CC1 C1(NC(C2CCC(=C)CC2)=O)CC2(C1)CC(CNC(C1CC3CCC(C1)C3)=O)C2 c1(CN(C2CCCN(C(c3ccncn3)=O)C2)C)nn(C)c(Cl)c1Cl N=c1nc(-c2cccc(F)c2)nc(N2CC(CNC(C34CC(CO3)C4)=O)C2)[nH]1 CCC(C)C(C(=O)N(C1CCCC1OC)C)N(C)C(c1ccc(O)nc1C)=O c1(OC)ccc(Br)c(CN2CC3CN(C(c4c[nH]c(C)c4)=O)CC23)c1O C1(C(=O)NC2C(NC(c3ccccc3Br)=O)CC2)CCc2nncn2CC1 CC1OC(C)CC1C(N1CCCC1CNC(c1cnn(CCO)c1N)=O)=O C(=O)(C(F)(F)C(O)C(C)C)NC1CC(N(C(C2N(C(C)=O)CCOC2)=O)C)C1 CCC(CC(=O)N1CC(F)CC1CNC(=O)Cc1cc(C(C)C)no1)C1CC1 N1(C(c2c(C)con2)=O)CCC(NC(c2ccn(CCF)n2)=O)C(O)C1 C1(CC(=O)NC2C3CCN(C(c4cncc(C)n4)=O)C32)OCCCC1(C)C N1(CC(=O)NCCC(=O)N(CC(C)O)C)C(=O)CCCC1=O C=CCC(C(=O)NCCCCCC(=O)N(CC(O)COC)C)C(C)C CCCCCC(=O)N(C)CC1COCCN1C(C1CC1(CC)CC)=O c1(NC(=O)NC2CC(C(C)(C)C)C2)cccnc1 CC1(C(N2CCC(c3cccs3)CC2)=O)CCCCCCC1 N1(C(C(c2cccc(C)c2)O)=O)CC(C2CCN(C(c3ccc(=N)[nH]n3)=O)C2)C1 C1(NC(COCCC=C)=O)CN(C(=O)Cc2ncsc2Cl)CC2(CC2)C1 C=C1Cn2c(C(=O)NC3CC(C)CN(C(c4cnc(Cl)c(N)c4)=O)C3)nnc2S1 Cc1cc(CC(=O)NC(CN(C(=O)C(Cl)=CCl)C)CCOC)n[nH]1 c1(C(=O)NCCNC(=O)OCC)cc(NC(c2ncn(C3CC3)n2)=O)on1 CN1CCC(C(=O)NCC2(CNC(C3SCCS3)=O)CCCO2)C1=O CC(CC(=O)NC1(CNC(c2conc2C2CCC2)=O)CCOC1)n1ccnc1 N1(C(c2c(C)scn2)=O)CC(NC(=O)CC2C=CS(=O)(=O)C2)C(C)(C)C1 N1(C(CN(C)C(C2CCCC2)=O)=O)CC(NC(=O)C(CO)N(C)C)C(F)C1 C(=O)(CS(=O)(=O)CCO)N(C1CCCN(C(C(F)SC)=O)CC1)CC N1(C(C(C2(C)CC2)NC(CCOCCCOC)=O)=O)CCC(F)CC1 N1(C(c2nnc(C)s2)=O)CCC(NC(c2cncn2C)=O)C(C)C1 N1(CCCOC)CCc2nc[nH]c2C1c1cccnc1CC(=O)NC1CCC1 c1(CC(=O)NCC2CCN(C(C3(c4cc[nH]n4)CCC3)=O)C2)cc(F)cnc1Cl N1(C(COCCOC)=O)CCCC(CNC(=O)CCn2cnnn2)CC1 C1(CNC(C(CC)=CCCC)=O)CC(O)CN1C(C1CC(OC)C1)=O c1(-c2n(C(CC)C)nc(-c3cccc(OC(C)(C)C)n3)n2)cccc2occc12 Cc1nc2ncnn2cc1C(=O)NCCNC(C1Cc2ccccc2S1(=O)=O)=O C=CCN=C(NCC1CCCC1(F)F)NCC(C)(C1CC1)OC N1(C(=O)C=CC=C(Cl)Cl)CCOC2(C1)CN(C(c1ccnc(C(F)(F)F)n1)=O)C2 N1(C(c2nc(C)[nH]n2)=O)CCOC(CNC(C2CCC23CCC3)=O)C1 c1(-c2nnc(C)o2)ccc(Cl)c(OS(=O)(=O)Cc2cccc(F)c2F)c1 c1(OC)cccc2c1OCC(NC(c1nn(-c3ccccc3)c3c1CCCC3)=O)C2 N1(C(C(COC(C)=O)C)=O)C(CC(=O)NCC(O)CC(C)C)C2CCCC12 c1(C(NNC(=O)NCCC(CCCC)O)=O)ccc2cc[nH]c2c1 c1(C(N2CC(NC(c3cnccn3)=O)C(C(F)F)C2)=O)c(Cl)ccc2c[nH]nc12 N1(C(C(C=C)C)=O)CCC(C)(C)C1CNC(C1(CCN=[N+]=[N-])CC1)=O C1(N(CC#C)C(C2CC2[N+](=O)[O-])=O)CCCN(C(C2CCC(C)CC2)=O)C1 C(=O)(C1=NNC(=O)C1)NCc1cn(CCNC(c2cc(C)nn2C)=O)nn1 C1(NC(C(CC)F)=O)CCCC12CN(C(=O)C1=C(C)CCCC1)C2 Cc1cc(C)c(C(N2CCCC(C)(NC(C3CCC(C)(F)CC3)=O)C2)=O)c(S)n1 CC(=O)CCCC(=O)NC1(C(N2CCCC(C)(CO)C2)=O)CC(F)C1 C1(C2(NC(c3c(SC)ccs3)=O)CC2)CCCCN1C(=O)Cc1cnc[nH]1 C1(CC)CC(O)CN1C(=O)CONC(c1nc(OC)sc1C)=O c1(C(C(N2CCC(N(C(C3CC(=C)C3)=O)CCSC)CC2)=O)O)cccc(C)c1F CC(C)(C)CCC(=O)N1CCCC(CO)(NC(C2CC3CC2C3)=O)C1 c1(C(N(CC(CC)NC(=O)COCCC(C)C)C)=O)cccn1C1CCCC1 c1(CN2C(C(=O)Nc3cc(O)ccc3Cl)CC2)nc2ccccc2[nH]1 C(=O)(CCCCCCCC)N1CC2N(C(C3C(=C)C3C(=O)OC)=O)C(C2)C1 C12(C(N(CCN(C(C(n3ccc(C)n3)C)=O)C)C)=O)CC3CC(C1)CC(C)(C3)C2 Cc1ccc(NNC(=O)C2CC(=O)N(C)C2c2cnn(C)c2)cc1C Cc1ccc(S(=O)(=O)NCC(=O)NC(C)CCCCNC(C2CCC2C)=O)cc1 C#Cc1cccc(C(=O)NC2CN(C(C3(C)CC=C(C)CC3)=O)CC2O)c1F N1(C(CNC(CC)=O)=O)CC(C)CCC1C(=O)N(C1CCCC1C)C C(=O)(CC(C)C(F)(F)F)N1CCCC(CN(C(=O)Cc2cccnc2C)CC)C1 N1(C(c2cnc(OCC)s2)=O)CC2CS(=O)(=O)CC2(NC(=O)C(N)=O)C1 N1(C(Cc2nc(NC(c3n[nH]c(C)c3C)=O)sc2)=O)CCC2(CCNC2=O)CC1 C=CC1(C(=O)NC(CC)CC(=O)OC)CCN(C(c2cc(F)c[nH]2)=O)C1 C1(C(N2C(C(=O)Nc3c(OC)nc(Cl)cn3)CC2)=O)CCc2ccccc2C1 C12(NC(C3CN(C)C3)=O)CC1CN(C(=O)CSc1nccn1C)C2 CCC(O)CC(=O)N1CCC(C2CCCCN2C(=O)CCc2cncn2C)CC1 c1(OC)ccc(C(N2CCC(C)(c3nn[nH]n3)CC2)=O)cc1NS(C)(=O)=O c1(C(=O)NCC2C(C(=O)NCC(CCC)CCO)CCO2)cc2cccn2cn1 N1(c2n(CC)c(-c3cc(C4CC4)[nH]n3)nn2)CCC2C(CCCN2C)C1 Cn1ccc(CCC(=O)NCC2CCN(C(=O)C(O)C3CCCC3)C2)n1 C(=O)(CC(C)C(F)F)NCCOCC(=O)NCC(CC(=O)OC)O CC(C)C(C)CS(=O)(=O)NCc1cnn(C)c1C(C)C N1(C(N2CC(CCC(F)(F)F)C2)=O)CCC(=CC(F)(F)F)CC1 n1(CC(N2CC(C(C(=O)NCC(COC)(F)F)OC)C2)=O)cccnc1=O C12(C(N(C)Cc3cc(C)no3)=O)CCC(CC1NC(=O)COc1ccccc1)C2 c1(OC)ncc(C(N2CC(OC)CC2CCNC(c2ccnnc2S)=O)=O)cn1 c1(C(N2CC(CC=C)(NC(=O)C3=CCCS3)C2)=O)c(F)c(F)c(F)c(F)c1F c1(C(N(CCO)CC)=O)ccc2c(C)c(C(=O)Nc3ncc(C#N)s3)[nH]c2c1 N1(C(C(CCC)OC)=O)CCCCC12CC(NC(=O)CCn1cccnc1=O)C2 C#Cc1ccc(C(N2CC(NC(c3ccc(OC)s3)=O)CC2C)=O)c(F)c1 Cc1[nH]c(C#N)cc1C(=O)NCC(C1CCCC1)NC(c1ncc(Cl)nc1Cl)=O CC1c2c(Br)cccc2CCN1Cc1cc2ccc(F)cc2nc1O C1(C(=O)NC2C(C)CN(C(C3CC(C(F)(F)F)C3)=O)C2)Cc2ccccc2O1 CN1CCN(C(=O)C(C2CC2)NC(c2cccc(Cl)c2)=O)C(CO)C1 c1(CC)nc(=N)[nH]cc1C(=O)NCC1CCCN1C(=O)C(F)C(C)(C)O Cc1cc(Cl)c(C(=O)NCC(F)CNC(c2cccc(F)c2)=O)cc1F N1(C(c2c(Cl)cc(C)s2)=O)CCC2CN(C(=O)Cc3nocc3C(C)C)CC12 CC1(C)COCCC1CC(=O)NCCOC1CN(C(=O)CNc2nccs2)C1 C1(NC(C2CCC(=O)O2)=O)CC(F)CN(C(=O)CSC2CCS(=O)(=O)C2)C1 C(=O)(CCC(=O)NCC1(NC(c2ccc(C)nc2)=O)CCC1)NCC C(=O)(C(C)(C)C(C)(F)F)NC1CC(C)CN(C(=O)CCSc2ccccc2Cl)C1 c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)C2CC2)cc(C(F)(F)F)ncn1 c1(OC)ccc(CN(C)CC2CCC2(F)F)cc1 c1(OCC)ccc(C(=O)NCCN(C(=O)CC2CC(C)(C)CO2)C)cn1 C(=O)(C1=NOC(C)C1)NC1CN(C(c2c(C)ncnc2)=O)CC1C CC(CS(C)(=O)=O)NC(=O)CCNC(=O)CC1CCCC(C)O1 C1(C(=O)NCC(CN(C)C(c2cc(-c3cccnc3)on2)=O)O)(CO)CCCO1 C1(C(N2C(CNC(c3ccc(CC)o3)=O)CCC2)=O)(OC)CCS(=O)(=O)C1 c1(C(=O)NC2C(CNC(CCS(=O)(=O)N(C)C)=O)CC2)cc(F)c2[nH]nnc2c1 c1(C(=O)NC2CCC(N(C(C3(F)C(C)C3)=O)C)CC2)cc(N)ccc1O N1(C(C)CN(C2CC(C(=O)OC)C2)C(C)(C)C)CCOCC1.c1(CC)cccs1 CC1CC(NC(=O)COC2CC(NC(C3CCN(C)C(=O)C3)=O)C2)CCC1(C)C C1(NC(C=CC)=O)CN(C(C2CCSC2)=O)CC1O C(=O)(CCCCNC(=O)OC(C)(C)C)NCCCNC(CCSCCCC)=O C1(CC)CN(C(C2CN(C(=O)C(C)n3ccnn3)CC2OC)=O)CC1O CC1(C(=O)NCC2(O)CC(CO)C2)CCN(C(=O)CCOCC2CC2)CC1 N1(S(CCC(=O)OCC)(=O)=O)CC2(CC2)CC1C(=O)N(CC#N)CC#N C1(C(N(CCCNC(c2ccc(N(C)C)cn2)=O)C)=O)CC2C(C1)C2(C)C C1(C(=O)NC2(CN(C)C(C3CCSC3)=O)CC2)CC1C1CC(F)(F)C1 c1(OC)ncnc(NC2CCC(NC(=O)C(C)NC(C)=O)CC2)c1OC C1(N(C(CC=C)=O)C)CN(C(=O)CC(c2cccs2)NC(=O)NC)CC1F C1(C)(CC(=O)N(CCCC)CC)CCN(C(=O)Cn2ccc(C)n2)C1 N1(C(C2(CC=C)CCCN2C(=O)C=C=C(C)C)=O)C2CCC(C2)C1CO Cc1nn(C)c(C)c1CCC(=O)N(C1CC2CC1N(C(c1csnn1)=O)C2)C C(C(O)CC(=O)NCCc1ccncn1)NC(Cc1c(C)ncs1)=O S(=O)(=O)(c1ccc(NC2CCOC(C(C)C)C2)c(Br)c1)N(CCSC)CC c1(C(N(C2CN(C(C3(CC)CC3(F)F)=O)C2)C)=O)cc2cccc(Br)c2o1 C1(NC(=O)OC(C)(C)C)CN(N2CCCCCCNC(=O)CC2)CC1C(F)(F)F c1(NC(=O)COc2ccc(Cl)cc2Cl)cc(Cl)ccc1F CC1CCCCC1CC(=O)NCCCC(C)(C)NC(=O)CCn1ncn(C)c1=O C1(c2cn(C3CN(C(C4(C)CC4(Br)Br)=O)C3)nn2)(N(C)C)CCOC1 c1(C(=O)NCCCCCCNC(=O)CN2CCC2CF)ccc2c(c1)COC(=O)N2 c1(OC)cc(C(=O)NC2CC(C)CN(C(=O)C(C)(C)CO)C2)cc(C)n1 N1(CC(c2cnc(Cl)s2)=O)CC(C(=O)O)C2(CCC2)C1.C1(N)CCOCC1 C(=O)(C1CCCCc2ccccc21)NC(C)(C)CNC(C1CC2C=CC1CC2)=O C1(NC(c2nnc(CC)s2)=O)COC2(C1)CN(C(c1ccc(C)cc1O)=O)C2 Cc1ncc2c(n1)CCC(C(=O)NC1(CNC(=O)C(O)C3=CCCCC3)CC1)C2 Cc1cccc2[nH]c(=NCC(C3CCCCC3)NC(c3ccoc3)=O)oc12 c1(N(C)CC2CCN2N2CCCC2)ncc(Br)cn1 N#CC1CCCC(C(=O)NCC2COCC2NC(c2cc(C(F)F)cs2)=O)C1 Cc1coc(C(=O)NCC2CCCC2C(N2CC(O)(CCO)C2)=O)c1 N1(C(CC2CC(C)C2)=O)CCC(CC(=O)N(CC(C)(C)CO)C)CC1 C12(C(=O)NCC=C3CCN(C(CC(C=C)C)=O)CC3)CCC(CC1F)C2 N1(C(c2ccc(-c3nccn3-c3ccc(F)cn3)cc2)=O)CCOC(CO)CC1 C(=O)(C(C(C)(C)C)NC(C1CCC(NC(C2CCCC(C#N)C2)=O)C1)=O)NC c1(C2CCN(N(C3CCCN(C(=O)C(C)(F)F)CC3)C)C2)cncc2nnnn12 N1(C(C(CC)=CC)=O)CCC(CNC(=O)C(N2CCCCCC2)C)CC1 C12(C(=O)NC3CN(N4C(C)(C)C=CC4)C3)CCC(CC1)N2C(=O)OC(C)(C)C N1(C(C(C(CC)C)O)=O)CC2CN(C(=O)C(C)NC(C)=O)CC2(C)C1 CC1(C)CCC(NC(=O)C=Cc2cccnc2)C(CNC(C23CC(C)(C2)C3)=O)C1 N1(C(c2scc(C(=O)Nc3cc(F)nc(F)c3)n2)=O)CCc2nc[nH]c2C1 C1(C(N2CC(O)(C(C(=O)N(CC(C)C)CC)F)C2)=O)COCCN1C O=C(C1c2ccccc2CN1C(c1ccc(=O)oc1)=O)Nc1cc(Br)ccn1 C1(C)(C(=O)NCC2C(NC(C3CCN(CC)C3)=O)COC2)CC2CC2C1 c1(C(=O)NCCCCC2CN(C(CCOCCOC)=O)C2)occc1Br Cc1nc(C(=O)NC2(CN(C(=O)CCCc3ccccc3)C)CC2)cc(O)n1 C1(OC)CC2(C1)CC(C(=O)N(CC(C)O)CCNC(=O)C(C)(C1CC1)N(C)C)C2 N1(C(COCCC)=O)CCC(CO)(CNC(=O)CSC(C)(C)C)CC1 CC1CN(C)CC(C(=O)NCC2(C)CCCC2NC(c2cc(C3CC3)on2)=O)O1 c1(CN2CCC(Nc3cc(OC)ncn3)C2)ncc(Br)cc1C C(=O)(CCS(=O)(=O)N(C)C)N(C1CN(C(C2CC2C#N)=O)C1)C C1(NC(C(C)SC)=O)CC2(C1)CC1(CC(NC(=O)CC3=CCCCC3)C1)C2 C(=O)(CCCC(F)(F)F)N1C(C2(NC(C(C(C)O)C)=O)CC2)CCC1 C(=O)(C(Cc1ccc(F)cc1)C(C)C)NC1(CNC(CCSC)=O)CCCCC1 Cc1cnc(N(C(=O)C2=CC(C)(C)C2)CC(=O)N(C)C)nc1C(F)(F)F C1(NC(CC(C)(C)C)c2n(CC(=C)C)nnn2)CC2OC(C)(C)OC2C1 c1(OC)cccc2c1C(C(=O)N1CCCC3CN(C(=O)C(C)(C)CO)CC13)CC2 c1(C(=O)NC2C(NC(C(=O)NCC(F)F)=O)CCCC2)cccc2ccncc12 C1(C)(CNC(CSCC=C)=O)CCCN(C(=O)CCCCCOCC)C1 C1(NC(COCC(C)(C)C)=O)CN(C(c2c[nH]c(Br)c2)=O)C2(CCCC2)C1 c1(C(=O)NC2CN(C(C(CC#C)O)=O)CC2C)ccc(=O)n(C2CCOCC2)n1 N1(C(C2(C(C)(F)F)CC2)=O)CCCC(F)(CNC(c2ncc(Cl)cc2F)=O)C1 C12(CNC(C=CCC)=O)CCCC1CCN2C(=O)C1=COCCO1 S(=O)(=O)(c1cnc(NC2CSCC2C)c(Cl)c1)NCc1c(OC)cccc1 c1(C(=O)OCC)ccc(CN2CCCCC2C(=O)NCc2cnccn2)cc1 N1(C(CCCC)=O)CCN(C(=O)C=C2CCC2)CC1c1cccc(Cl)c1 C1(CNC(C2CCN(C)CC2)=O)CCCC12CCN(C(c1c[nH]cc1Br)=O)CC2 C(C(=O)N1CC(OCCC(=O)N(CC(C)O)C2CCC2)C1)(C1CC1)SC CC1CCC(NC(=O)C(F)C2CC2)CN1C(=O)CCc1ccccc1Cl CCC(C)(C)C(O)C(=O)N1CC(COC)(NC(c2sc(N(C)C)nc2Cl)=O)C1 C(CCN=c1nc(NCCCN(C)C)cc[nH]1)c1c(OC)c(F)ccc1 c1(C(=O)NCC2CC2CNC(C2CCCOC2)=O)ccc2ncc(Br)n2c1 N1(C(C(CSC)C)=O)CC(C2CN(C(C3(C(C)C)CC3)=O)C2)C1 c1(C(=O)NC2CN(C(=O)Cc3ccnnc3O)C2)cc2c(nn1)CCC2 C#CCC(O)CC(=O)NC1(C)CCN(Cc2cn(C3(C(=O)O)CC3)nn2)CC1 C(=O)(C1=C(C(C)=O)C(c2ncnn2C)N(C)C(=O)N1C)N(c1cccc(C)c1)CC C=CCCCC(C(=O)NC1CC1)N1CCC(Cc2cnn(C)c2)C1 c1(OC)ncc(C(N2CCC(NC(c3cscc3OC)=O)C(CO)C2)=O)cc1Cl c1(NCC)ncc(C(=O)NCC(C)N(C(=O)C(C(C)C)NS(N)(=O)=O)C)cc1Cl N1(C(C2C=CCN(C(CC=CC)=O)C2)=O)CC2(C1)CC(C)(C)C2 Nc1c(F)cc(C(=O)NCC2CCCCCN2C(=O)C(F)CC2CCC2)cc1F CCCCC(C(=O)NC1CCN(C(c2nc(C)oc2OC)=O)C1)N(C)C N1(C(C(CC#C)O)=O)CCC2CN(C(=O)CCC(=O)c3ccccn3)CC12 C1(CNC(C2(C(C)NC(C(CSC)C)=O)CC2)=O)CCCN(C)C1=O C=CCCC(O)CN(C)C(c1cc(CNC(c2cnc(CC)o2)=O)[nH]n1)=O C1(CNC(C(CC#C)NC(c2snc(C)c2N)=O)=O)CCCCC1(C)C C1(N(C(c2cccc(CC)c2)=O)C)CN(C(c2c[nH]nc2OC)=O)CCC1O Nc1cc(C(N2CCN(C(c3coc(CO)c3)=O)CC2C2CC2)=O)cc(F)c1O C1(C(=O)NCCC2CC(NC(c3nc(CCC)sc3)=O)C2)C2(CC2)C12CC2 C1(C(=O)NCC2(OC)CN(C(=O)C(C)O)C2)Cc2cccc(C)c2O1 C#CC1CC2(CC2)CN1C(C1(NC(=O)CC2COC(=O)C2)CSC1)=O c1(C(=O)NCCN(CCOC)C(C2CCC(=O)N2)=O)cc2cccn2c(O)n1 S(=O)(=O)(c1ccc(NCCCN2CCCC2=O)c(F)c1)N1CCC(OC)(CO)C1 c1(C(=O)NC(CC)CN(C)C(c2ccccn2)=O)cccc(CC2CC2)c1 N1(C(C2CCC(C)(C)C2)=O)CC(NC(=O)CN2CCOCC2)CC(F)C1 c1(N2C(CNC(CCSC)=O)CCC2)cc(C)nc(-c2ccccc2Cl)n1 N1(C(c2cc(OC)c(F)cc2)=O)CCC2C(C1)CN2C(c1cc2n(n1)CCC2)=O C1(CNC(C(C2CCCC2)SC)=O)CCCN(CC2CCCC2C)C1 N1(C(c2nc(C)sc2C)=O)CCCC12CN(C(=O)CSc1cccc(F)c1)C2 C(=O)(C1CCCc2scnc21)N1CCCC(CNC(=O)CS(=O)(=O)C2CC2)C1 c1(OC)nccc(CNC(=O)CC2CCN(C(=O)COCCN(C)C)C2)n1 N1(C(=O)OC(C)(C)C)CC(C(=O)NCC2(C)CN(C(N(C)C)=O)C2)C2(CC2)C1 C12(C(=O)NC(CC=C)CNC(=O)CCCn3cc(C)cn3)CCC(CC1)CC2 N1(CC)CC2(C1)OC(=O)NC2C.C1CC(=O)NC(=O)C(C2(C)CC2)NC(=O)N1 CC(C)(C)S(=O)(=O)CC(=O)NCC1C2CN(Cc3cscn3)CC12 CC1(C)CCCC1CNC(C1CCC(CNC(=O)C(=O)C2CCCC2)C1)=O c1(OC)cc(C(N2CCC(C)(C)C(CNC(=O)C(F)OC)C2)=O)cc([N+](=O)[O-])c1 N1(C(C2CC(=C)CN2C(c2cncn(C)c2=O)=O)=O)CC(C(=O)OC)CC(C)C1 CC(C)C(C#N)C(=O)NC(C(=O)N(C1CC2CC2C1)C)C(C)(C)O Cc1c(C(=O)NC2CN(C(=O)CC3CCS(=O)(=O)C3)CC2C)ccc2cncn12 c1(C(N(C(CC)C(=O)N(C)Cc2nccn2CC)C)=O)nnn(CC)c1C c1(C(N2C(CNC(C(CC(C)(C)C)F)=O)CC2)=O)cccc2ccncc12 C(=O)(C1CCOc2ccc(F)cc21)NCC1(NC(CN(C)C)=O)CCOCC1 C1(NC(C(CC)COC)=O)CC2CC(C1)N(C(C1CCOCC1)=O)C2 C(=O)(CCCC(F)F)N(C(CNC(C(C)NC(=O)C(C)(C)C)=O)C1CC1)C C(CCCC(=O)NC(C1CCOC1)CO)NC(COCCCC(C)C)=O CC1C(C(=O)NCC2CC3CCC(C2)C3)CCCN1C(=O)CN(C1CCCC1)C C=C(C)CCCC(=O)NC1(CNC(=O)CC2CCCOC2)CCCCCC1 c1(CC)c(-c2nc(C(C)CC)nn2CCS(N)(=O)=O)cnn1CC(C)C C1(CC(N2CCC(CN(C(c3cnc(C)nc3)=O)C)C2)=O)CCCCC1(F)F c1(C(N2C(C(=O)NC3(CC(=O)OC)CCC3)CCC2)=O)c(F)cc(C#N)cc1F c1(CC(C(=O)OC)F)ccc(NCC2C3COCC23)cc1 C1(NC(C2C(C)(C)N(C(C3CCC(=O)N3)=O)CC2)=O)CC2COCC(C1)C2 c1(C(=O)NC2C(NC(C3N(CC)CC3)=O)CCCC2)ccc(C)c2c1NCCC2 C(C(C(=O)NC(C1CCCO1)(C)C)NC(C)=O)OC.n12cc(nn1)C(=O)NCC2 c1(C(C)NC(=O)C(=O)NC(c2nccn2C)C2CCOCC2)cnnn1C n1(CCCC)ncc(C(N2CC(CC(C)(C)CNC(C3(F)CC3C)=O)C2)=O)c1C N1(C(c2cc(COCCO)no2)=O)CC2CN(C(=O)Cc3c[nH]nc3C)CC2C1 c1(OC)cc(Br)c(CNC2(CO)CC2C)cc1F N1(C(CCC(=C)Cl)=O)CCC2CN(C(c3nn[nH]c3Cl)=O)CCC2C1 N1(C(CC2(C)N(C(c3ccc(C(C)=O)o3)=O)CC2)=O)CCC2(CCC2)C(O)C1 c1(C(=O)NC2C(NC(CNC(C)=O)=O)CCOC2)c(F)ccc(C)c1F c1(CNC(C(N2C(COC)COCC2)c2cn(C)nc2C)=O)ccc(C)cc1Cl c1(C(=O)NC(CCOC)CNC(=O)CC2(OC)CC2)c(N)cc(F)cc1Cl C1(C#N)(C(=O)NCC2N(C(c3cc(OC)n[nH]3)=O)CC2)CCOCC1 C=CC(CC)CC(=O)NC1CCC(NC(c2ccnc(OC(F)(F)F)c2)=O)CC1 Cc1[nH]c(=NCc2ccc(C(F)(F)F)nc2)sc1C(=O)Nc1c(O)ncnc1O N1(C(C(C)n2ccnc2)=O)CC(NC(=O)C=Cc2c[nH]cn2)C(C)(C)C1 N1(CCN(C2CCCO2)CCN(C)C)CCCC2(CCC2O)C1 C(CCC(=O)NCC(C)(C1CC1)NC(=O)CC1COCCO1)OCCN(C)C c1(CCC(=O)NC2C(CNC(CC(C)(C)C3CC3)=O)CC2)c(F)cccc1Cl c1(OC)nc(Cl)c(C(N2CC(=C(F)CNC(=O)CC(C)C3CC3)C2)=O)s1 c12nc(ncc1Br)S2.Cc1ccccc1OCCN(CC(=O)NC1(CF)CC1)C c1(CC(=O)NCCN(C(C)=O)C)coc2ccc(C)cc12 C(=O)(NNc1ncc(F)cc1F)NCC1(C)COCCO1 S(=O)(=O)(c1ccc(=NCC2CC23CC3(F)F)[nH]c1)NCc1nn(CC)nc1C CC1(C)CC1(Br)C(=O)NCCCN(C(C1CCC(=O)N1)=O)C1CC1 C1(CNC(C=CSC)=O)CN(C(=O)C(C)NC(c2cccs2)=O)CCO1 C(=O)(C(O)(C(F)(F)F)C1CC1)NC1C(NC(c2n[nH]c3c2CCC3)=O)CCCC1 C(CCN(C)C(c1cccn1C)=O)(C(C)C)NC(C(C=C)OC)=O c1(NCc2cnc(Cl)s2)cccc(OC(F)(F)F)c1F.C12CCC(CC1)C(=O)N2 C(=O)(C(CCC(=O)OC)N1CCN(C)CC1)N1C(CN)CCC12CC2 C12(C(N3CCC(NC(CCC(=O)N(C)C)=O)C(F)C3)=O)CCCC1CC(=O)CC2 N1(C(C)=O)CC(N=c2cc(NCC3CC(N(C)C)C3)nc(C(F)(F)F)[nH]2)C1 Cc1nn(C)c2c(NC3CCn4cnnc4C3)nc(N3CCOC(C)(C)C3)nc12 C1(C)(CC#C)CC2CN1C(=O)CCOCC(=O)N2.C(CCCC)NC(=O)C1CC1 CCCCC(C)CCC(=O)NC1CC(O)(CNC(c2cncc(C=C)c2)=O)C1 C1(C(N2C(CC)CC(C)C2)=O)N(C(c2cc(Cl)n(C)n2)=O)CCCC1(C)C c1(C(=O)NCCC2CCN(C(C(CCC)C)=O)CC2)ccc2ccccc2c1C Cc1nc(NC(=O)C(=O)NCC(c2ccsc2Br)(C)O)sc1-c1ccc(F)cc1 CC1C(NC(c2cnco2)=O)CCCN1C(c1ccc(C(N)=O)cn1)=O c1(C(N2C(CCNC(C(CC)(F)F)=O)CCC2)=O)cc(C)c(F)cc1O C1(C(=O)NC2C(NC(COCC=C)=O)C2)CC(F)(CO)C1 c1(C(N2CCC(COC)(NC(=O)Cn3nnc(=O)[nH]3)C2)=O)cc2n(n1)CCCN2 N1(C(c2ccn(CCCC)n2)=O)CCOC(CN(C)C(c2cccc(N)n2)=O)C1 C1(N(C)C(C2CC2CF)=O)CCC(NC(=O)C=Cc2ccc[nH]2)CC1 c1(CCCC(=O)NC2CCC(NC(c3c(C)nc[nH]3)=O)C2)ccc(F)c(F)c1 C(C(F)(F)C(=O)NCC(O)CN(C)C(C1CN(C2CCOCC2)C1)=O)OC O=C1CCC2(CCC(OC(=O)CCCCCc3ccccc3)CC2)N1 c1(C(=O)NCC(C)(O)CNC(C2(c3cc[nH]n3)CCC2)=O)cccc(Cl)c1F C1(C(=O)NCc2c(C(=O)NCCC3CCN(C)CC3)n[nH]c2)CCCC12CCC2 c1(N(CC=C)CC)ccc(S(=O)(=O)NC(COC)C(=O)NCCOC)cc1Br c1(-n2cc(CC3N(C(=O)Nc4ccncc4)CCC3)nn2)ccc(Cl)c([N+](=O)[O-])c1 c1(CC)cc(F)c(NC(c2ccc(C3CCNCC3)o2)=O)cc1F N1(C(c2cc(CC)[nH]n2)=O)CCC(C(C)(C)C)(CNC(=O)COC2CCOC2)C1 C1(C)(C(N2CCCN(C(C)=O)C2)=O)CC(O)CN1C(c1ccn(C)c1)=O c1(C(N(CC(C)CNC(C2(C(F)F)CC3(CC3)C2)=O)C)=O)nn(C)c(Cl)c1Cl C1(=CCNC(C(C)Cc2cnco2)=O)CCN(C(C2COCCN2C)=O)CC1 N1(CC(N2C3CN(Cc4ccc(C)cc4C)C(C3)C2)=O)C(=O)OC(C)(C)C1=O c1(C(C)=O)cc(C(=O)NCCC2CN(C(=O)CC(=O)NC3CC3)CCO2)n(C)c1 C(C(C)(C)CN(C(=O)C(F)(F)c1ccccn1)C)NC(C(C1CCCO1)OC)=O N1(C(C2(F)CCN(C(c3cc(OC)n(C)n3)=O)C2)=O)CCCC(O)C1C C(=O)(CCCC(C)(C)C)N1CCC(C(=O)NCCN(CCO)CC)(CC)C1 c1(OCCCC)ccc(C(C(=O)NCCCF)N(C)CCOC)cc1 CN1CCCC1(C)CC(=O)NCCC1(NC(=O)COCCCF)CC1 n1(CCC=C)c(N(CCc2ccc(Cl)cc2)CC)nnc1CC1CCCOC1 C1(C(N2CC(C(C(=O)NCC(N3CC(CC4CC4)C3)=O)O)C2)=O)CC12CCCC2 N1(C(Cn2c(C)nc(C)n2)=O)CCC(C=CC(=O)NCCC2=CCCCC2)CC1 c1(C(C(=O)NCCC2(C)CC2)N(CCOC)CC#N)ccc(SC)s1 CCCCC(CN(C(CCC1(C)CC1)C(=O)NCC1(C)CCCO1)C1CC1)CC c1(OC)ccc(CC(N2CCN(CCCNC(=O)CS(N)(=O)=O)CC2)=O)c(F)c1 C(=O)(C(C(C)CC)N(C)C(c1cnn2c1OCC2)=O)NC(CC#CC)CO N12CCCC1CN(CC)C(c1cnc(Cl)s1)C2=O.C(C(C)C)SC1CC1 c1(N(C2CN(C(C3CC(F)C3)=O)C2)C)nc(Cl)nc2c1ncn2C CC1(C)C(NC(=O)CCOc2cccc(C#N)c2)CCN1C(=O)COCCCF c1(C(=O)NCC2(O)CC(NC(CCCC)=O)C2)ccc(-n2cccc2)cc1O C1(C(=O)NCC(C)(CNC(c2csnn2)=O)OC)CCCN2CCCC12 c1(CCC(=O)N(CC(c2csc(Br)c2)=O)C)nnc(C2CCCC2)o1 C1(NC(c2c(C)nccn2)=O)CC(O)CN(C(C2C3CCC2(C(F)(F)F)C3)=O)C1 C12(CNC(c3ncc(OC)cn3)=O)CCCCC1N(C(c1ocnc1C)=O)CC2 C1(n2cnnn2)(CC(=O)NCC(CNC(c2c(CC)ncs2)=O)O)CCSCC1 C1(CNC(C2CC(SC)C2)=O)CN(C(=O)CN2CCC(C)(O)C2)CCN1C C=CCC(CNC(c1ccn(C)n1)=O)NC(c1cn(CC2CCCO2)nn1)=O CC1CN(C)CCCN1C(C1C(C)CN1C(=O)C1=CCCCCC1)=O C(C(C)(C)CC(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)C=CCO)CC2)OC c1(C(=O)NCC(CC)NC(=O)C(C)(C)CSC)[nH]cnc1C#N Cc1ccc2nc(CCNC(=NCCCC#CBr)NCC3CCOC3)cn2c1 c1(CC(C(=O)NCC2CN(C(C3CCS3(=O)=O)=O)C2)OC)ccccc1Br C=CC1(C(=O)NCCN(CC(C)O)C(C2(n3ccnn3)CC2)=O)CCC1 C1(C(N2C(CNC(c3c(C)cc(C)s3)=O)CCC2)=O)CC(S(C)(=O)=O)C1 c1(CN(C(C)CO)C(=O)CC2CC(C(=O)O)C2)c(O)ccc(F)c1F c1(CNC(C(N2CCC(NC(CCC)=O)C2)=O)=O)cc(Cl)c2c(c1)OCO2 CCC(C)C(O)CC(=O)N(C1CC(C(=O)NC(C)CSC)C1)C n1(CC)nnnc1CN(C(=O)C(C1CCOC1)NC(=O)C(C)SC(C)C)C C(C)(C)(C(C)c1ccccc1)OC(CN(CC(F)(F)F)CC)=O c1(C(=O)NCC(CC=C)NC(C2CC(F)C(=O)N2)=O)cc(Cl)c(OC)c(Cl)n1 C1(C)(NC(=O)NCC(n2cccn2)NC(CC)C)CC(=O)C1 S(=O)(=O)(c1ccc(C(N2CC(CNC(=O)COC)CC(C)C2)=O)cc1)NCC#C Cc1cn(C)cc1C(=O)NC1CC(N(C(=O)CSC2CCOC2=O)C)C1 C(CC(=O)N1CCC(NC(=O)CNS(N)(=O)=O)C(C)(C)C1)(C(F)(F)F)OC N1(C(CC(COC)(C)C)=O)CCC2(CCCN(C(C3CC3C)=O)C2)CC1 CC1CC(=O)NC(C(N2CCC(C)C2C(=O)NC2CCC(N(C)C)C2)=O)C1 c1(C(=O)NC2CCCN(C(CC(=C)C)=O)C2)c(F)cccc1Br N1(C(CCC=C=C)=O)CC2CC(NC(C3CCN(CC(F)(F)F)CC3)=O)CC1C2 C12(C(=O)NCCC(C)NC(C3CC3F)=O)CC(C(C)(C)C)(C1)C2 C1(NC(C2CCS(=O)(=O)N2)=O)CCN(C(c2cc(C3(O)COC3)on2)=O)CC1O C(=O)(C(C)CC(=O)NC(CCN(C(=O)C1=COCC1)C)C(C)C)OC c1(CC)c(C(N2CC(N(C)C(c3cn(C)nc3C)=O)C(O)C2)=O)csc1C N1(C(C(C)(C)c2cccs2)=O)CCCC2(CC(NC(=O)Cc3cnns3)CO2)C1 c1(OC)ccc(C(=O)NC2CC2NC(=O)CC23CCC(CC2)CC3)cc1Cl c1(C(N2CCC3CCC23)=O)cc2c(cc1F)CNCC2 N1(C(C)=O)CCCC1NC(C1CC(C(=O)N(CCO)CCN(C)C)C1)=O C1(CNC(CSCC)=O)CCC2(CN(C(=O)CC(C)(F)F)C2)O1 c1(C(=O)NC2(C(=O)NCCC#C)CCCC2C)cnn(C)c1C#N c1(C(N2CC(NC(C3C(CCOC)C3)=O)C2)=O)ccnc(N2CCCC2)c1 N1(C(C=CCC=C)=O)CCC(CC(O)CO)C1 CCCC(C)(O)CC(=O)N1CC(NC(c2csnc2C2CC2)=O)C(SC)C1 C1(NC(C2(COC)CC=CC2)=O)CC2CC(NC(=O)CC(O)CN(C)C)C1C2 c1(C(=O)NC(CCCNC(CCOCC#C)=O)C)ccc(-c2cscn2)cc1 N1(C(C2CCC(OC)C2)=O)CC2CC1C2CNC(=O)CCOc1cccnc1 C#CCCC(C(=O)N(C)CCN(C(CC)CC)C)NC(=O)C(C)SC Cc1ccoc1C(=O)NCCC(C)NC(=O)CC1(O)CCC1 C1(CN(C(=O)C(C)(C)CF)C)CCCC(NC(=O)CNC(c2cccs2)=O)C1 C1(C(=O)NC2CN(C(C(CC=C)CC)=O)CC2C)CCC2(CCCC2)CC1 C(N=c1nc2scnc2c(CN2CC(CO)CC2C)[nH]1)C1(OCC)CCCC1 N#CCS(=O)(=O)c1ccc(F)c(C(=O)NCC(C2CC2)NC(=O)Cc2cocn2)c1 c1(C(=O)NC(C2CCCN(C(=O)C=C3CCCCC3)C2)C)cc(N)cc(O)c1 c1(C(=O)NCC(C)CN2CCOCC2)cccc(CNC(C2CCC2(F)F)=O)c1 C1(NC(CCc2ccn(C)n2)=O)CC(C(=O)NC2CC(=O)N(O)C2)C12CCC2 C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC(CN(C(C(C=C)(C)CCOC)=O)C)C CCC(CC(=O)N1CC(OC)CC1CCNC(c1occc1C)=O)C1CC1 C=CC(C)(C)CC(=O)NC1(COC)CCN(C(c2cc(F)cs2)=O)C1 c1(C(=O)NC2CCCC(NC(=O)C=Cc3nccs3)CC2)ccc2cc[nH]c2n1 CC1CN(C(c2cc(C(F)F)[nH]n2)=O)CC1CNC(c1cncc(C(F)F)c1)=O C1(C)(C(=O)NCC(CC)NC(=O)C=Cc2cc[nH]n2)CCCCCC1 c1(CC(=O)NC2(N)C(C)CC2)ccc(C(=O)N(C)C)cc1 C1(NC(C=CCCC)=O)CCC2CCN(C(c3ccoc3Cl)=O)C12 c1(C(N2C(CNC(c3csnn3)=O)CC2)=O)cnn(CC2CC2)c1 CCC(C)C(=O)N(C)CCOCCNC(C1CC(n2ccnn2)C1)=O c1(C(=O)NC2C=CC(CNC(C3(CC#C)CCOC3)=O)C2)cc(Cl)c(N)cc1F CC(C)CC(F)C(=O)NCC(C(C)(C)C)NC(c1cn(CC(F)(F)F)nn1)=O CC1(C)CCC(O)(C(=O)NCC2CC2NC(C2(c3cccs3)CC2)=O)CC1 N1(Cc2c(C#C)cccc2)CCN(C(C2(CC)CCC2)=O)C(C#N)C1 CCC(C)C(O)C(=O)NCC(C)(C(C)C)NC(C1(O)CCCCCC1)=O c1(C(=O)NC(C2(CNC(C(CCC)C)=O)CC2)C)cncc2c[nH]nc12 C1(=CC(=O)NCC(c2c(F)cccc2F)NC(CC)=O)CCCCC1(C)C c1(SC)nc(C(N2CCCN(C(C3CC3(F)F)=O)C(C)C2)=O)c2ccccn12 c1(OC)nc(C(=O)NC2(CNC(=O)CC3CC(SC)C3)CCCCC2)sc1C C(C)(CNC(=O)CCc1cnc(C)s1)(CC)NC(C1C(OC)C1)=O C1(CNC(CC(CC)C)=O)CN(C(=O)COCCCF)CCN1C c1(C(N2C(C(CNC(CS(CC)=O)=O)(C)C)CCC2)=O)cnc(O)c2cncn12 N1(C(C(C)OCCCC)=O)CC2CC2(NC(=O)CNS(=O)(=O)CC)C1 S(=O)(=O)(c1cc(Br)ccc1Cl)N(c1cnn(-c2ccncc2)c1)C(C(C)C)=O c1(NC(C2N(C(CN(C)C)=O)CC(O)C2)=O)cccc(F)c1OC(F)(F)F C1(NC(C2ON=C(CC)C2)=O)CN(C(c2c(Br)n[nH]c2C)=O)CCC1O c1(SCCN(C(C2CCCCC2)=O)Cc2nnnn2-c2ccccc2)ccncc1 N1(C(C(F)=CCC)=O)CCCC(NC(=O)CC2NC(=O)NC2=O)CC1 C1(CNC(c2c(C)nc[nH]2)=O)CN(C(=O)Cc2ccsc2C)C2CC12 C(=O)(CCC(=O)c1ccc[nH]1)N(C1CCCN(C(=O)CCc2cnn(C)n2)C1)C C(=O)(C#CC1CC(F)(F)C1)NCCNC(c1c(C)ncc(Br)c1)=O N1(C(C2(CNC(C(C(C)C)F)=O)CCCO2)=O)CC23CCC2(COC3)C1 C(=O)(C(CCS(C)=O)NC(C)=O)NCc1cccc(OC(COC)C)c1 CON(C)CCCNC(=O)C(c1ccoc1)NC(C1CC=CCO1)=O c1(C(=O)NC2CC(C)(NC(Cc3nnc(C)o3)=O)C2)ccc(N2CC=CC2)cc1 N1(C(C(c2cnn(C)c2)C)=O)CC2CC(NC(=O)CN(C)S(=O)(=O)N(C)C)C2C1 c1(OC)ccc(Cl)c(C(=O)NC2CCN(C(=O)C(N3CCCCCC3)C)C2)c1 N1(C(c2c(C)ccs2)=O)CCCC(CNC(c2coc(C(N)=O)c2)=O)C1 C1(C(=O)NCC(C)CNC(C2(F)CCOC2C)=O)CCC2(CCOCC2)O1 C(C(=O)NCC(c1ccc(C)cc1)NC(C1(C)CC=CC1)=O)(C(C)C)OC c1(CNC(c2c(C)nco2)=O)ccc(CNC(C2CCOC(C)C2)=O)c(F)c1 c1(OCC)cc(OC)cc(NC(C2CCCN2C(C2(O)CC2)=O)=O)c1 N1(C(C(CCC)C)=O)C2CCC1CC(C(=O)NCc1c(Cl)cccc1Cl)C2 N1(C(c2c(CC)noc2C)=O)CC2CC(NC(c3cn(C(C)C)nc3C)=O)C2C1 C12(NC(C(C3CCOC3)OCC)=O)CC(C1)N(C(=O)C=Cc1csc(C)n1)C2 CC1CN(C(c2cccn2C)=O)CC(C)N1C(=O)C1=C(Cl)CCCC1 c1(C(=O)NCC(C)(C)NC(C2CC(C)=C(C)CC2)=O)cc(C)c(C)c(F)c1 C(=O)(C(CNC(c1nonc1N)=O)C(C)(C)C)NCc1cnc(CC)[nH]1 Cc1cc(F)c(S(=O)(=O)N2CCN(c3ccccc3)CCC2C)cc1C(=O)O O=C1NCC2(CCN(c3nc(N4CCC(CCF)CC4)nc4sccc34)C2)O1 CC(C)C(O)C(C)(C)C(=O)NCCCN1CCN(C(c2csc(=N)[nH]2)=O)CC1 CC(C#N)C(=O)N1CCC(CCNC(C2CCC(C(C)(C)C)O2)=O)C1 CC(C)CC(CNC(=O)C(C)CNC(=O)CNC=O)N(C)C N1(C(c2c(C)ncs2)=O)CCC(N=[N+]=[N-])(C(=O)NC(c2nncs2)C)C1 N1(C(C(CCC#C)O)=O)CCCN(C(c2nn(C)cc2Cl)=O)CC1C c1(C(=O)NCC2CC(COC)CN2C(=O)CC2CCOCC2)cccc(C)c1O C1(NC(=O)C(=Cc2c[nH]cn2)F)COCCN(C(=O)CC2CC(O)C23CCC3)C1 N(C1CCc2ccc(Br)cc21)C(C1(C)CCN1C(c1cc(F)cc(Br)c1)=O)=O C1(C(=O)Nc2cc(-c3n(C)ccn3)sc2)C2CC3C(C2=O)C13 c1(C(=O)NC2CC(F)(C(=O)OC)C2)ccc(C2CCNCC2)nc1 c1(CSCC(=O)NCC2(O)CCN(C(=O)CC(F)F)C2)ccc(F)cc1 Cc1nc(Cl)[nH]c(=NC(C)CNC(c2ccc3c(c2)COB3O)=O)c1Cl C(=O)(C(O)P(C)(C)=O)NC(CCOC)C(=O)NCc1cc(F)cc(F)c1 C1(C(N2CC3C(CNC(c4cc(CC)no4)=O)C3C2)=O)CN(CP(C)(C)=O)C1 CCC(O)C(C)C(=O)N(CC(C)(C)C(=O)NC1COCC1F)C O=C(C1=NNC(C(F)(F)F)C1)NC1CC(NC(=O)CC2CS(=O)(=O)C2)C1 C1(NC(c2cn(CC)nc2)=O)CC2CC1N(C(c1nnn(C)c1N)=O)C2 C1(N(C(c2[nH]cc(CC)n2)=O)CC2CC2)CCN(C(=O)CC(=O)OC)CC1 C(c1ccc(F)cc1F)=CN1CCN(C(CSc2ccc(C)cc2)=O)C2C1C2 N1(C(C(C)O)=O)CCCC(O)(CCNC(=O)C(O)c2ccco2)C1 c1(NC(COCCNC(CC2N(CC)CCOC2)=O)=O)cnn2cccc(Cl)c12 c1(OCCC(N2CC(CNC(C3(C)CCCO3)=O)OCC2)=O)ccc(F)c(F)c1 C1(C(=O)NC2CCC(CCNC(c3ccn(C(C)C)n3)=O)C2)CC2C(C1)C2(F)F Cc1oc(C#N)cc1C(N1CCC(CCCNC(=O)C=CCF)CC1)=O C1(C(=O)NC(c2ccncc2)(C)C)CC1C1CN(C(=O)C=C2CCCCC2)C1 n1(CC)nc(C)c(CC(=O)NCCC(C)N(C)C(C2CC2OC)=O)c1C CCC1=C(C(=O)NCC2(F)CN(C(c3ncnc(C)c3C)=O)C2)SCCO1 C1(CC2C3CN(CC)CC32)CCC(C#N)CC1.C1C(n2cc(CCO)nn2)C(=O)N1 CC1(NC(=O)NC2CC2(F)F)CCC(=O)NC1 C1(CC=C)(NC(=O)Cc2cc(F)cc(Cl)c2)CCN(C(C2CCCCO2)=O)CC1 C(=O)(C(C(C)O)SC)NCCN(C(=O)C(c1ccccc1)n1cccn1)CCC C12(C(N3CCC(C(N(C(C)C(N)=O)C)=O)CC3)=O)CCC(C1)OC2C C(c1ccc(C(N)=O)o1)=CC(=O)NCC(CN(C(C(C)=C(C)C)=O)C)C c1(C(N2CC(NC(c3coc(Cl)n3)=O)CC3(C2)CC3)=O)nc2cc(O)ccc2[nH]1 N1(C(c2c(CC)nn[nH]2)=O)CC(C(=O)NC(c2ccoc2)C)C(C)(C)C1 C#CC(C)(C)C(=O)NCCCOCCCNC(=O)CC1CCCN1C c1(C(=O)NC2C=CCN(C(Cn3c(C)nnn3)=O)C2)ccc2ccccc2c1F c1(C(=O)NC2CCCC(N(C(Cc3c(C)nc(C)s3)=O)C)C2)ccc(Cl)nc1O CC(C)CC1C(=O)N1.c1(COC(=O)NC2CCN(C(C)C)C2)ccccc1 c1(C(=O)OC)sc(S(N)(=O)=O)cc1NC1CCOC(c2ccncc2)C1 c1(C(N2CCC(CC=C)(NC(=O)C(C3CC3)OC)C2)=O)cc(OC)cc(F)c1 CC(F)(F)C(F)C(=O)N1CC2CC2(C(=O)NCCCCCCO)C1 c1(C(=O)NCC2=CCN(C(c3cc(C)ns3)=O)CC2)nc[nH]c2nccc1-2 C(C)(CC1CCOCC1)(C(=O)O)NC(CN(C1C2CNC1CO2)C)=O N1(C(COCC#C)=O)CCC(C(=O)NC2(C3CC3)CC2)CC1(C)C N1(c2c(C(C)=O)cc([N+](=O)[O-])cc2)CCC2CC(=O)NC2C1 C1(N(C(=O)CCc2cnc(O)[nH]2)CC#C)CCN(C(=O)CCCOCC=C)CC1 c1(C(=O)NCCCCCN(C(=O)CC2(O)COC(C)(C)C2)C)cccc(=O)n1C c1(NC(c2c(C)noc2)c2nnnn2C2CCCCC2)cncc([N+](=O)[O-])c1 NS(=O)(=O)c1cnn(CC(=O)NC2CCCCC2NC(=O)C(F)(F)CO)c1 C1(C(=O)NCCC#C)C2CCCC1CN(C(c1ccc(C#N)s1)=O)C2 CC1OCCC1CC(=O)N(CCCCNC(=O)COCP(C)(C)=O)C c1(C(N2C(CCC)CCC2)=O)ccc(COC)cc1.C1C(O)CN1CC C(CC(=O)NCc1cccc(C#N)c1)(C(C)(C)C)NC(C(CC=CC)C)=O C1(CC(=O)NC(c2cccc(Br)c2)C)CC(F)CN1C(=O)C(C)(F)F C1(CC(=O)NCc2cn(C)nc2)C2CCCC2N1C(=O)CCCC1CCC1 C1(NC(c2ccco2)=O)CC2CCC(C1)N2C(=O)CCc1cc(F)ccc1F N1(C(C(C)OCCC=C)=O)C2CCC1C(C(=O)NCC1CCCOC1)C2 C1(C(C(=O)NCCC(=O)NC(C)CC)N(C2(C#C)CC2)C)CC=CCC1 C1(C(N2C(C(C)NC(c3ccc(CO)o3)=O)CCC2)=O)CC(C)(C)C12CC2 c1(OC)cccc(CC(=O)NC2CCN(C(=O)CC3(C)OCCO3)C2)c1Cl C(=O)(C1=CCc2ccccc21)N1CCC(NC(C2(C3CCCCO3)CC2)=O)CC1 CS(=O)(=O)c1ccc(C(N2C3CCC2C(CNC(c2coc(CO)c2)=O)C3)=O)[nH]1 N1(C(c2nc(COC)sc2)=O)CCC(CNC(C2CCS(=O)(=O)N2)=O)C12CCC2 n1(CC(=O)NCC(C(C)C)NC(C(CC)F)=O)c(C(F)(F)F)nc2ccccc12 C1(NC(c2ccc(C)cn2)=O)CC(NC(=O)CCCSC(C)(C)C)C12CCC2 C(=O)(C(CN(C)C)NC(c1cc(C)sn1)=O)NCCCC=C CN1CCC(C)(C(=O)NCC2COCCN2C(=O)Cn2ncc(O)nc2=O)CC1 O=C(C1CC(O)c2ccccc21)NC1CCC(CNC(=O)C(F)C2CCCC2)C1 c1(CC(=O)NCC(CC)NC(c2coc(C)n2)=O)sccc1C CC1(CO)CCN(C(c2sccc2NC(c2ccc(Br)nc2F)=O)=O)CC1O C1(c2sc(C)c(O)n2)CC2(CCOCC2)C(=O)N1COCC1CCCO1 C#Cc1ccc(CCC(N2CCC(NC(c3occc3F)=O)C2C(C)C)=O)cc1 C1(NC(c2cn(CC=C)nc2)=O)CC(C)N(C(=O)Cc2csc(C(C)(C)C)n2)C1 c1(C(=O)NCC(C(C)C)NC(=O)CN2CC(=O)N(C)C2=O)cccc2c1COC2 c1(C(N2CCC(CNC(C(C)=CC)=O)CC2)=O)ccc(N)cc1[N+](=O)[O-] c1(CCC(N2CC(C(=O)NCc3ccoc3)C3(CC3)C2)=O)cnc2ccccn12 CON(C)C(=O)Cn1cc(-c2cccc(C(F)F)c2)nn1 N1(C(c2cscc2C2CC2)=O)CCOC(COc2ccccc2)C1 C(=O)(CCCCC(F)F)N1CC(N(C(=O)CC2CC3(CC3)CO2)C)C(C)(C)C1 N1(C(C(C(CC)C)N(C)C(c2cnc(O)c(C)c2)=O)=O)CC2(CCOC2=O)C1 C(c1ccccc1)=CC(=O)NC(C(C1CCCCC1)NC(C(C)=CC)=O)C(C)C C=CC(C)(C)CCN=C(NC(C)CC)N1CCC(O)C(O)(CCC)C1 C1(CNC(C(c2n(C)ncc2)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CC1(Cl)Cl c1(C(=O)OC)ccc(C(N2CCCC2Cc2ccccc2F)=O)n1C C#CCC(O)C(=O)N1CC(N(C)C(c2cccc(CSCOC(F)(F)F)c2)=O)C1 CC(=O)CCCC(=O)NC(C(=O)N(C(C)CC(F)(F)F)C)C1CCCC1 c1(OC)cc(C(=O)NCCC(C)NC(c2ccc(C)c(Cl)c2)=O)cc(Cl)n1 C(c1cncc(F)c1)=CC(=O)NCCC(C)N(C(=O)CCC(=O)N(C)C)C C12(NC(=O)CCn3cnccc3=O)CCC(CN(C(c3cnc(Cl)s3)=O)C1)C2 c1(C(=O)Nc2ccc(Nc3scc(SCC)n3)cc2)cc2c(s1)CCC(CC)C2 CC1OC(C)CC1C(N1CC2CC1(CNC(C1(CO)CCOCC1)=O)C2)=O N1(C(c2cc(COC)oc2C)=O)CC2CCOC2(CNC(c2csnn2)=O)C1 Cc1ncc(C(N2CCOCC(CNC(c3csnc3Cl)=O)C2)=O)cc1N CCCC(C)(C)CC(=O)NC1CC(CCNC(C2(C)CCNC(=O)C2)=O)C1 c1(CNC(C2CC(C(=O)OC)C2)=O)cn(CCNC(c2csc(C)c2)=O)nn1 C(c1ccc(F)cc1)=CCC(=O)N(C1CN(C(CCCNC(C)=O)=O)C1)C C=C(Cl)C(C)(C)C(=O)N1CC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1 c1(CC(=O)NCc2ccc(-n3cc(C4(C)CC4)nn3)cn2)cc(F)cc([N+](=O)[O-])c1 c1(OC)ccc([N+](=O)[O-])cc1-c1ncsc1C(=O)Oc1c(O)ncnc1O CCCCC(C)(F)C(=O)N1CCC2(NC(=O)CC3CC3)CCCC12 C1(C(=O)OC)CCCCN(C(=O)CCCC(C)NC(=O)CC(C)(C)C2CC2)C1 c1(C(N2CC(C(C)NC(Cc3cc(C)[nH]n3)=O)OCC2)=O)cc(N)nc(Cl)c1 N1(CC(C)OC)CC2(C1)C(NC(c1ccsc1C)=O)CCS2(=O)=O C12(NC(c3c(CC)occ3)=O)CCCC1CN(C(C1(CF)CCC1)=O)C2 N1(CCC)CCCCC1C(=O)NC(C)C(CO)NC(=O)C(C)(C)N(C)C N1(C(c2c(C)cc(C)nc2)=O)CCC2(CCC(NC(=O)C(C)C3CCC3)C2)CC1 c1(C(=O)NC(C)(CNC(=O)C(O)c2ccco2)CO)cn2ccnc2s1 C1(NC(CC(C)c2ccccc2)=O)CC2(CCN(c3cncc(Cl)n3)CC2)C1 c1(OC)cnc(C(=O)NCC2CC2CC(=O)NC2COC(=O)C2)cn1 C1(C(N(CC#N)Cc2ccccc2)=O)CCc2ccccc2C1 C1(CNC(=O)CCCC2CCCO2)CCCN(C(C2CC3CCC2CC3)=O)CC1 C1(SCC)CCC(C(=O)N(C2CCC(NC(=O)C3=COCC3)CC2)C)CC1 N1(C(COC(C)C)=O)Cc2ccccc2C(NC(=O)C(C)CS(C)(=O)=O)C1 C1(NC(c2c(C)oc(C#N)c2)=O)CC12CCC(NC(=O)CSC(F)(F)F)CC2 N1(C(C2C(CC)CCO2)=O)CCCC(C)(C)C1CNC(c1nnn(C)c1C)=O C1(C2CC2)(C(N2CCC(C=C)C2)=O)CN(C(=O)C(C)CC2CC2)C1 c1(OCC)cnccc1C(=O)NC(C1CCCN1C(=O)CC1CC(OC)C1)C c1(NCCOC)ncccc1S(=O)(=O)N1CCCC1c1ccc(C)s1.C1(S)CCCO1 C(=O)(C1OCCc2ccccc21)N(CC(O)CNC(=O)CCCC(F)F)C c1(C(N2C(CC=C)CCCC2)=O)cc(Cl)c2ccccc2n1 c1(C(=O)NCCC2(NC(C(CCSC)O)=O)CCC2)cccn2nccc12 N1(C(CCOC)=O)C2CCC1C(C(=O)NCCC(C)(O)C1CC1)C2 C(=O)(C1CCCc2c(OC)cccc21)NCCCCC(=O)OCC C1(c2n(CC)nnn2)(Nc2ccc(C3CC3)c(F)c2)CCC2(CCC(=O)N2)CC1 C1(CNC(C(C)(C)CF)=O)CC12CCN(C(c1cnc3[nH]ccc3n1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NCC(CCOC)NC(C(CC)(C)COC)=O C1(NC(C2CC(C(C)(C)C)C2)=O)CCN(C(c2nnc(O)nc2O)=O)C12CCC2 c1(C(=O)NC(C)C(C)(C)NC(=O)CSCC(=O)Nc2ccco2)cc(O)n(C)n1 N1(CC(=O)NCC2CC3CCCC3C2)C(=O)C2=C(CCCC2)C1=O C1(OC)C(OC)CN(C(c2cnc(C)o2)=O)C1CNC(C1CCOC1C(C)C)=O Cc1cc(CC2CC(COC(C3CC(OC(C)(C)C)C3)=O)C2)nc(S(C)(=O)=O)n1 C1(OC(N2C(C(CC)OC(c3ccccc3)C3CC3)CCC2)=O)C=CC(C)(C)CC1 CC(C)C(C)(CNC(=O)CCNC(c1ccc(Cl)cn1)=O)NC(c1cccs1)=O C(=O)(C1=CCc2ccccc21)NCC1(C)N(C(c2c(=O)ccn(C)c2)=O)CCC1 CN1CCN(C)C(C(=O)NC2(C)CC(C(=O)NCC3CC4CCC3CC4)C2)C1 N1(C(C2N(C(C)=O)C(=O)CC2)=O)CCN(C(c2sc(O)nc2C)=O)C2(CC2)C1 N1(C(=O)Cn2ccnc2)CCC2CC2(C(N2CC(O)(CCO)C2)=O)CC1 C12(NC(CCOc3ccc(C)cc3)=O)CCC(CC1NC(=O)C1=COCC1)C2 c1(SC)nc(N2CCC(NC(=O)CC3(C)CCCCC3)C2)cc(C)n1 CC1(C)CCN(C(C2Cc3nccn3C2)=O)CC1C(=O)NC1C2CCCCC12 c1(C(N2C(CNC(Cn3c(CCC)ncc3)=O)CC(O)C2)=O)c[nH]cc(Cl)c1=O c1(C(N(C)CC2CCCN(C(c3cnsn3)=O)C2)=O)ccc(F)cc1NC(N)=O c1(C(=O)NC2CC(CC)(CC)N(C(=O)C=CC(C)C)C2)ccc(N)c(C)c1F N1(Cc2n(CC)ncn2)CCC(NC(C2CCc3nncn3C2)=O)CC(C)(C)C1 CCC1=NOC(C(N2CCCC2(C)CNC(c2cc(CC(C)C)[nH]n2)=O)=O)C1 N1(C(c2c(C)scc2)=O)CC2CCCC(C(N3CC4CC4C3)=O)C2C1 c1(C(=O)NCC2CN(C(=O)Cc3cocn3)CCO2)nc[nH]c1[N+](=O)[O-] C1(N(C(c2c(C)nco2)=O)C)CCC2CN(C(=O)C(F)C(C)(F)F)CC12 N1(C(CSCC(c2ccncc2)C)=O)CCC(NC(c2c[nH]cc2C2CC2)=O)C1 C1(N(C(CC(C)(C)OC)=O)C)CCCN(C(C2CC2Cc2ccccn2)=O)CC1 C(CCN=c1[nH]nc(C(F)F)o1)N(C(=O)C=C1CCCCCC1(F)F)C C(=O)(C(CC(F)F)c1ccccc1)NCC(CC)NC(c1cccnc1NC)=O CCC(CC(=O)NC1CC2CCC1(C(=O)NCC(C)(C)C(C)O)C2)CC(C)C C1(CNC(=O)CC2C=CCC2)COCCN1C(C1CC=CCO1)=O N1(Cc2cncc(C)c2)Cc2ccccc2CC1C(=O)Nc1nc2c(s1)COCC2 Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)N1CCN(CC(F)(F)F)CC1CF C1(C(=O)NCC2CC(CC)C2)C(C)CCN1C(c1ccc(N)cn1)=O C(C(C)C(=O)N1CCCC1CN(C)C(c1cnc(C2CCC2)s1)=O)OC C(=O)(C(C)(O)C(F)(F)F)NCC(CC=C)NC(c1cc(C)nc(O)c1)=O C(N=c1cc(C)[nH]c(=NCc2cc(C)c(C)nn2)[nH]1)c1cc(OCC)c(C)cc1 c1(C2C(C(N(S(=O)(=O)CC3CC(F)(F)C3)C)=O)C2)cccc(F)c1 Cc1nc(C)c(C(N2CCCC(N(C(=O)CNC(C3CCOCC3)=O)C)C2)=O)s1 Cc1ccc(F)c(C(=O)NCC#CC(=O)N2CC(C(C)(C)C#N)C2)c1 N1(C(c2c(C)csc2)=O)CCC(C2CC2)C1C(N1CCC(C(C)C)CC1)=O c1(C(=O)NC2CCN(C(c3cnc(C)s3)=O)CC2F)cc2c(cc1F)NCCC2 c1(C(=O)NCc2c(C(=O)NCc3n(CC)ncn3)nco2)nnccc1C c1(N2CCCC(C(C)NC(Cc3cn(CC)nn3)=O)C2)cc2nncn2cn1 N1(C(c2nc(CC)oc2C)=O)CC(CNC(=O)Cc2ccsc2)OC2(CCC2)C1 N1(C(C(c2cn(CC)nc2)=O)=O)CC(NC(C2(C)CCCC2)=O)C(O)C1 C(=O)(CC(C)(C)C(F)F)NC1CC(C)N(C(=O)CCc2cc[nH]n2)CC1 C12(C(=O)NCC3CCN(C(CN=S(C)(C)=O)=O)C3)CCCN1S(=O)(=O)CC2 C1(NC(C2(Cl)CCCCC2)=O)CC(C(=O)NCC2CCCC23CC3)=CC1O c1(C(=O)NC(C)C(C)NC(c2coc(Br)n2)=O)ccc2c(c1)OCCNC2=O N1(C2CCN(C(=O)C=Cc3cc[nH]c3)C2)CCN(C(c2cccnc2)=O)CC1 C1(CN(C)C(c2ccsc2Cl)=O)CCCC(CNC(C2CC(C#N)C2)=O)C1 c1(C(CCO)NC(=O)NCC23CC(CC2CO)C3)ccc(F)cc1F c1(NC2CCCN(C(C(C)(C)C3CCCCC3)=O)CC2)ncc2ccsc2n1 C(=O)(C1CCCOC(=O)N1)N1CCN(C(CC)C)CC1.C(C)(C)(C)OC(C)=O C#CC1CC2(CC2)CN1C(C1CC(C)(C)CN1C(=O)Cn1nnc(C)n1)=O N1(C(C=CCN(C)CC)=O)CCC(O)(CNC(C2CCC23CCCO3)=O)CC1 O=C(C1CCCc2nn[nH]c21)N1CCC(CO)C(NC(C2(C(F)(F)F)CC2)=O)C1 N1(C(C(C)SCCCC)=O)CCc2[nH]nc(CNC(=O)C(C)OCOC)c2C1 C(c1ccc(F)c(F)c1)=CC(N1CC(CN(C(=O)C(C)(C)C#N)C)C2(C1)CC2)=O C(=O)(N=c1[nH]oc2ncccc12)C1C(NC(C(c2ccccc2)OC)=O)CCC1 c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C=Cc3cnc[nH]3)C2)c(F)c(Cl)c1 N1(C(CC(=C=C)C)=O)CCN(C(=O)C(c2ccc(Br)c(C)c2)C)CC1CO C1(OC)CC(NC(c2cn(C)c(=O)n2C)=O)CN(C(=O)CC2(C#N)CCC2)C1 N1(C(C(C2CCCCC2)C)=O)CCC(NC(c2nccc(Cl)c2O)=O)C(F)C1 C1(NC(c2ccc(NC)cn2)=O)CCC(C)N(C(=O)CSc2ccc(F)cc2)C1 CC(CC(=O)NC(C1CN(C(C2CCCC3CC23)=O)C1)C)CC(C)(C)C c1(OC)ccc(OC)c(CC(=O)NCC(C)CNC(=O)CC(C)F)c1 c1(C(N2CC(OCc3cn(CCC)nn3)C2)=O)cc(-c2ccccc2)nc(O)c1 Cc1cc(N)cnc1C(=O)NCc1ncc(C(=O)NC(C2CCCO2)C)cn1 C(N=C(NC1CC1)N1CCC2(CCOCC2)CC1)C1CCC(C(F)F)CC1 CN1CCC(O)(C2(C(N3CCC(N(C(=O)C4=CCOCC4)C)C3)=O)CC2)CC1 c1(OC)nccc(I)c1C(N1CCSC(C(=O)Nc2ccc(Br)c(O)c2)C1)=O O=[N+]([O-])c1cc(Cl)c(CN2CCC(CO)(CO)C2)s1 c1(C(N2CC(CC)N(C(=O)CN3CC(C)(C)C3)CC2)=O)ccc(F)cc1C#N Cc1nsc(C)c1-c1noc(C2CCS(=O)(=O)C2)n1 CC(=O)CCCC(=O)N1CC(NC(c2ccc(Br)cc2Cl)=O)C1 c1(CNC(N2CCC(COCCOC)C2)=O)ccc2c(c1)C(=O)CCS2 N1(c2cc(NC3CCN4CCCCC34)nc(C(C)C)n2)CCC2(CCCCO2)C1 c1(C(C(=O)NCCCCCC)N(CCC(C)C)C2CC2)ccc([N+](=O)[O-])cc1OC C1(CNC(C=CSC)=O)CC(C)N(C(c2ccnc(C(C)(C)C)n2)=O)C1 C1(CC(=O)NCC(C)CNC(=O)CCOCC(C)(C)C)CCCCC12CC2 C(=O)(C(C)(C)CNC(=O)CC1(C)CCN(C(c2cc(C)oc2CSC)=O)C1)NC c1(NC2C(OC)CN(C(=O)CN=S(C)(C)=O)C2)ccc([N+](=O)[O-])c(C#N)c1 c12cc(Cl)cnc1NC(=O)C2.C1(CC(=O)OC)(OC)CCOC1 C1(NC(C(CNC(CCC(=C)Cl)=O)OC)=O)CCN(C)CC1C#N c1(C(N2CC=CC(NC(C(C)C3CCCO3)=O)C2)=O)cccc2c1CCCC2 c1(OC)cccc(C(C)(C)C(=O)NC2CN(C(C3C=C3C)=O)CC2C)c1 CC(CC(C)(C)CO)NC(=O)COC1CC(NC(c2ccc(Cl)cc2)=O)C1 c1(C(=O)NCCC2(NC(CNC(=O)OC)=O)CCC2)nc(C)n(C)n1 N1(C2CN(C(C3C(C)CCN3)=O)C2)CCC(C#N)C1 C1(C(N(C(C)CNC(=O)CCCn2ccnc2)C)=O)CC12CC2(F)F C1(C(C)NC(C2CC(Cl)(Cl)C2)=O)CCN(C(c2cnoc2C2CCC2)=O)CC1 C#CCC(C)(C)C(=O)NCC1CN(C(=O)Cc2ccccc2C2CC2)CCN1C C1(C(=O)NC(c2ccc(Sc3ccccc3)cc2)C(=O)OC)C(C)(C)C1(F)F C1(C(N(CCOCC)CC)=O)CCOCC1[NH+](C(=O)C(C)(O)CC)[O-] c1(N2CCC(N)C2)cccc(Cl)c1.C1(COC)(CNC=O)CCC1 N1(C(c2ccc(O)nc2)=O)CC2OCCN(C(=O)CCOCC(F)(F)F)C2C1 N1(C(c2cccc(OC)c2)=O)CC(NC(c2nc(C)nn2C)=O)C2(CC2)C1 C1(N(C(c2ccc(OC)c(C)c2)=O)C)CCC2CN(C(=O)C(C)N(C)C)CC12 c1(CNC(NNC(c2ccc(OCCC(C)C)cc2)=O)=O)nc2ccsc2s1 c1(CN2CCCC(COC)C2)ccc2cc(F)c(F)cc2n1 CC1CN(C(=O)C(c2ccco2)NC(=O)CC2CCN(C)C2=O)CC(=O)N1C c1(CC)ccnc(C(N2CCC(OCCNC(c3nc(Cl)sc3C)=O)C2)=O)c1 c1(C(N2CCC(NC(=O)C(Cl)(Cl)Cl)CC2)=O)ccc2c(C(=O)O)n[nH]c2c1 CC(F)(F)C(F)C(=O)NCC1(F)CCCN(C(=O)C(=C2CCCCC2)F)C1 CC1CCC(C)C1NC(=O)C(Cc1ccoc1)NC(=O)CC1(N(C)C)CC1 C1(NC(CC(CC)C)=O)CCCN(C(C2CCN(C(C)C)CC2)=O)CC1 C=C(C)CC(C(=O)Nc1cscc1Cl)NC(=O)CC1CC(C2CC2)C1 Cc1[nH]cc(C(N2CC(NC(c3nn(C)cc3Cl)=O)C(N=[N+]=[N-])C2)=O)c(=O)c1Cl N1(C(c2n(CC)ncc2)=O)CCC=C(C(=O)NC2CCOC23CCCC3)C1 c1(CC)cc(C(N2CC3(CCC3NC(=O)CC(C)C3CCCC3)C2)=O)ccc1C S(=O)(=O)(c1ccc(F)cc1F)N1C(C(=O)Nc2cnn(C(F)(F)F)c2)CC1 c1(CNCc2cncc(OC(C)C)c2)cccn(Cc2ccccc2)c1=O C1(CNC(CSc2nc(C)[nH]n2)=O)CN(C(=O)C(c2ccccc2)F)C(C)(C)C1 N=c1cc(C(N2CCC(F)C(NC(c3ccc(Cl)s3)=O)C2)=O)nc(Cl)[nH]1 C1(NC(CN(CC)CC)=O)CCN(C(C2CN3CCC2C3)=O)CC1O C1(C(=O)NC2CC(n3cc(C(C4CCCCO4)(C)C)nn3)C2)CNC(=O)C12CC2 CC(CCN(C)C)C(=O)N1CC2CC2C1C(=O)NCCc1cccc(F)c1 CC1(C)CCN(C(=O)Cc2ccsc2)C1C(N1CCOC(CC(N)=O)C1)=O C1(C(=O)NC2(CCC)CCC2)CN(C(C2CCCCN2C(=O)C2CC2)=O)CCO1 c1(OC)ccncc1C(=O)NCC1CCN1C(=O)C(CCO)N(C)C C1(NC(C2N(CCC)CCCC2)=O)CCN(C(C2(C#N)CCCCC2)=O)CC1O c1(OC)c(NC2CC(C)N(C(=O)Cc3ccn(C)n3)C2)ncnc1Cl C12(NC(CCCCOC)=O)CCC(C1)N(C(c1ccc(O)nc1C)=O)C2 Cc1ccc2c(c1Br)CCCN2CC(=O)N(C)Cc1ccc(F)cc1F Cn1ccc(=O)c(C(N2CCC=CC2C(=O)NCC2(CCO)CCCC2)=O)c1 CC(C)(C)CC(O)C(=O)N1CCCC(C)(CNC(c2ccnc3c2CCC3)=O)C1 c1(C(=O)NCC23C(CN(C(C(CN(CC)CC)F)=O)C2)C3)cnc(O)cc1C C1(N(C2(C(O)CO)CC2)C(=O)NCC2CC(=C)C2)CC(C#N)C1 c1(COCC)ccc(C(=O)N(C2CCN(C(=O)CCC3CC3(Cl)Cl)C2)C)cc1 c1(SC)ccc(O)c(C(=O)NC2CCCN(C(=O)C=Cc3nc(C)c(C)[nH]3)C2)c1 c1(C(=O)NCCC2CCN(C(CC(=O)OCC)=O)CC2)cc2nc(=O)ccn2[nH]1 CC(c1ccccc1)=CC(=O)NC1CCCC1NC(C1(C)CC(C#N)C1)=O c1(NC(C2N(C(c3cn(C)cc3C(F)(F)F)=O)CC=C2)=O)ccc(C#N)cc1Cl C(C1=NOC2CN(C(c3c(C)nn(CC)c3C)=O)CC12)NC(C=CC=CCC)=O N1(C(C(C)(C)CCl)=O)CCOCC2(C1)CN(C(C1(F)CCNC1)=O)CCCO2 C#Cc1ccc(C(N2CC(N(C(=O)C(CCC)OCC)C)C2)=O)cc1F C1(CC(N2CCC(COCC3CC3)C2)=O)CCCCN1C(C1COCOC1)=O c1(C(=O)NCCOC)ncncc1OC.C1C(=O)N1CCCN(C)C c1(OC)c(C)cc(C(=O)NC2CC(NC(c3oc(C)cc3C)=O)C2)cc1C C1(OC)CC2(C1)CN(C(=O)C(O)CNC(=O)C(C)C(F)(F)F)C2 N1(C(C(C)CN2CCCCC2)=O)CCCC2(CCN(C(=O)Cc3ccoc3)C2)C1 C(=O)(CCCS(C)(=O)=O)NCC1C(C)(C)CN(C(=O)Cn2cc([N+](=O)[O-])cn2)C1 N1(C(C=CC(C)=O)=O)CC2(C1)SCCC2NC(C1CC12CCSCC2)=O C1(C(=O)NC(CC(C)C)CNC(c2csc(=N)[nH]2)=O)CN2CCCN1CC2 C(=O)(C(F)C(C)C(F)(F)F)NCC1C(C)CCN1C(C1CCCC1(C)C)=O C1(c2nnnn2CCCOC2CC2)(NCCC2(C)COC2)CCCC1C1CC1 CC(Cc1ccccn1)C(=O)Nc1ncc(CCNC(=O)Cc2cc(Br)cs2)s1 c1(CNC(c2ccc(CNC(C(COC)(C)C)=O)o2)=O)cc(C)c(C)nn1 c1(NC(C2CN(Cc3ccccc3)CC2C(F)(F)F)=O)cnc2c(Br)n[nH]c2c1 N1(C(C(n2cc(-c3c(C(=O)OC)cc(F)cc3)nn2)C)=O)CCC2(CC1)CSC2 c1(C(=O)NC2C(NC(CNC(N)=O)=O)CCCC2)cc2cccc(Cl)c2s1 C1(C(=O)NCC2(S(C)(=O)=O)CCC2)C2CCC(C2)N1CCO.S1(=O)(=O)CCN1 C#Cc1cccc(C(=O)NC(CNC(c2cc(C(C)(C)C)no2)=O)C(C)C)c1F C1(NC(CC2C(C)CCC2)=O)CN(C(=O)C(C)CC2CCC2)CC(C)(C)C1 C1(C(=O)NCCC(=C)CNC(=O)CCc2cccnc2Cl)CCCN1N=O c1(N(C(C(C2CC=CCC2)N(CCN(C)C)CC)=O)C(C)CC)ccccc1 C(C)(C(=O)NCC1CC(NC(C2(CF)CC2)=O)C1)OCC=C c1(CN2CCC(=CC(=O)NCc3n(C)cnc3)CC2)cccc2[nH]ncc12 CCC(C)CCCCC(=O)NCC(O)CCNC(=O)C=Cc1cncc(OC)c1 c1(C(=O)NC(CNC(CC=C)=O)C(C)C(C)C)coc2c(C)cc(Br)cc12 C(=O)(C(C)(O)C(C)(C)C)Nc1c(SCC)cc(C(F)(F)F)cc1 Cc1nc(NC(C2CN(C(c3c(F)cc(F)cc3F)=O)C2)=O)c(F)c(Cl)n1 CCCC(O)CC(=O)NC1CN(C(c2cncc(F)c2)=O)CC1c1ccccc1 Cc1cc(C=CCN2CCCC(O)C2C(F)(F)F)ccc1C(=O)O NC(=O)C(CCC(=O)O)OCc1ccc(NC(=O)CCc2cc(F)ccc2F)cc1 Cc1cc2c(cnn2C)cc1C(N1CCC2CN(C(=O)C(C)N)CC12)=O N(C(=NCC1(CC#N)CC1)NC(c1ccco1)C1CC1)CC c1(C(=O)NCC2CN(CC(=O)OC(C)(C)C)C2)cc2cc(Br)cc(Br)c2o1 C1(C(=O)NCCC(=C)CNC(c2ccc(CC)s2)=O)CC(=O)NC(CC)C1 CCC(CC(=O)NCCC(C)O)NC(C1(SC)CC1)=O CC1C(C(=O)NCCS(N)(=O)=O)CCN1C(C1CCSCC1)=O C1(CC(=O)NC2CCC(N(C(C3CCCC3)=O)CC)CC2)CC(C)CC(C)(C)C1 CCC1=NOC(CC(=O)NC(Cc2ccoc2)C(=O)NCC#CCOC)C1 c1(Cn2c(C3OCC4CCC3C4)nc(CCCSCC)n2)cnn2c1NCCC2 N1(C(C)(C)C)CCCCNC(=O)C(F)(F)C1.N1(C(=O)OC(=O)C2CC2)CCCCC1 N1(C(CNS(CCCC)(=O)=O)=O)CC(NC(C2CCCCC2)=O)CC1(C)CSC Cc1cnc(F)cc1C(C(=O)Nc1ccccc1Cl)N(C)Cc1cncn1C CC1(C)CCOC(=O)C1NC(N1CC2CSCC2(C)C1)=O Cc1cc(C(N2CCC(C)(C)C2CNC(C2CCCCC2)=O)=O)cc(N)c1 CC1C(NC(c2c(C#N)cnn2C)=O)CCCN1CC(=O)NC1CCCCC1 c1(CNC(C2CC(C)(NC(C(CC)C#N)=O)C2)=O)ccc2n[nH]cc2c1 C=CCCC(C(=O)NCC12CCC(CC1)C2)NC(=O)Cn1[nH]cnc1=N C1(NC2(Cc3ccc(Br)cc3)CCC2)CCC2COCCC2C1 S(=O)(=O)(c1ccc(NCC2CCS(=O)(=O)N2C)c(F)c1)N1CCC(CCC#N)CC1 C1(F)(CNC(CC(C)C)=O)COCCN(C(C2CCC(C(F)(F)F)CC2)=O)C1 c1(C(N2C(C(C)NC(c3c(COC)noc3)=O)CCCC2)=O)[nH]c(=N)ccc1C c1(C(N2CCC(OCCNC(CN(C(C)=O)C)=O)C2)=O)csc2cnccc12 N1(C(c2n(COC)ncc2)=O)CC(N(C(=O)C(C)C(C)O)C)C(O)C1 N1(C(CCCC=C)C)CCN(C(=O)Oc2ccccc2C(F)(F)F)CC1C C1(c2n(CCCSCC)nnn2)(NCCCCC(F)(F)F)CCCC1(C)C c1(C(=O)NC2CN(C(C3CC(C#N)(OC)C3)=O)C2)cn2nc(C)cc2[nH]c1=O c1(CC)cc(Cl)ccc1C(N1CC(NC(c2cscc2OC)=O)C(C)(C)C1)=O C(CCCCC(=O)N1CCCC(O)(CNC(=O)Cc2nnc(O)s2)C1)N(C)C C(=O)(C(F)CC(C)(C)NC(=O)CCCSC(C)C)N1CCN(C(C#C)C)CC1 C1(c2cccc(F)c2)(NC(=O)C=CC2CCCO2)CCN(C(=O)Cc2ccsn2)C1 N1(C(CS(=O)(=O)NCC)=O)CCC(NC(c2ccsc2-n2cnnn2)=O)C(C)C1 c1(C(=O)NC(C)CCCNC(=O)C#CC2(C)CC2)coc(S(N)(=O)=O)c1 C1(NC(c2c(C)nco2)=O)CN(C(c2cnn3c2SCC3)=O)CCC1CO N1(C(C2C(C)C2)=O)CCC2CCN(C(=O)Cc3ccc(O)nc3)CC2C1 CC(C)C(C(=O)N1CCCC(NC(c2cc(-c3ccccc3)co2)=O)C1)N(C)C N1(C(CC(CC)NC(C2CC2C(N)=O)=O)=O)CCC(=O)N(C)CC1 C(=O)(CC(=O)NCC1CCN1C(C)(C)C)N(CC(C)(C)S(C)(=O)=O)C c1(CN2CCC(O)(C(=O)Nc3cnc(OC)nc3)C2)ccc(OC)c(Cl)c1 CCC(C)(CCNC(=O)CC1CC12CC2)NC(=O)C=Cc1cnn(C)c1 C(=O)(C1=CCCCC1)N1C(CC(=O)NCc2cnc(C)[nH]2)CCCC1 N1(C(C(=O)C(N2CCC(OCCOCCOC)C2)=O)=O)CCCC2C(=O)CCC12 n1(CC(=O)N(C)CC2CN(C(=O)C(O)CC(F)(F)F)C2)c(O)nc2ccccc12 c1(C(=O)NCC(C(C)C)NC(C(CC)OC)=O)cccc(-n2c(O)nnc2O)c1 Cc1cc(Cl)ncc1CC(N1CC2C(C1)N2C(c1ccccc1I)=O)=O N1(C(c2ccc(CC)cc2C)=O)CC2CC(C)N(C(c3cc(C)ncn3)=O)C2C1 C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cnc(N(C)C)o2)=O)C1 C(CC(C)C(=O)NC(c1ccnn1C)C(=O)NCC1CC2CCC1O2)=CCC Cc1csc(C(=O)NCCc2n[nH]cc2C(=O)NCCC2CCC3CC23)c1C c1(C(N2CCC(C(C)NC(C3C(=C)CC3)=O)CC2)=O)csc2cccnc12 CCC(C(=O)NCCN(CCOC)C(C1CSCN1C(C)=O)=O)n1ccnc1 C(=O)(C1Cc2ccc(F)cc21)N1C(CNC(c2ccc(N)c(F)n2)=O)CCC1 C1(C(N(CCCCCC)CCNC(=O)C(C)SC)=O)CC(F)C(=O)N1 C#CCCCC(C)C(=O)NCC12CC(NC(=O)CCC(=O)OCC)(C1)C2 c1(C(C)C)nc2[nH]ccc2c(=Nc2cccc(O)c2)[nH]1 c1(C(=O)NC2(CCOC)CCN(C(=O)CC3CC34CC4)C2)cc2ccccc2o1 C1(CCCNC(C(C)(C)C)=O)CCCCN1C(=O)CCCOc1ccccc1Cl O=C1CC(C(=O)NCCC2(NC(c3ccc(Br)c(O)n3)=O)CCC2)=NN1 C(CCCCCNC(c1cnoc1C1CCOCC1)=O)NC(CC=C)=O C(C)(C)(CC(F)C(=O)N1CC2CCCCC12)NC(C1C(CC)CCC1)=O C(C(C)(CC(C)C)NC(=O)C(C)OC1CCOC1)NC(Cn1nc(C)oc1=O)=O N#Cc1cnc(N2CCCCC(NC(=O)CCn3cc(Cl)cn3)C2)c(Cl)c1 C1(CNC(c2n(CCCSC)nnn2)c2ncco2)(OC)CCC(=O)C(F)(F)C1 C1(NC(CC2(OC)CN(C(CCC(C)OC)=O)C2)=O)COCCC1(F)F N1(C(C(C(CC)C)NC(=O)C=CCF)=O)CC2CCCC(C2)C1 C1(C)(C(=O)NCC2CN(C(C3(CC=C)CC3)=O)CC2C)C(C)(C)C1(C)C C1(C(=O)NC2C3CCCOC23)(CC)CCN(C(c2nonc2N)=O)CC1 C(=O)(CCCCCNC(=O)C1CC1)NC1CCC(NC(COCC)=O)C1 c1(C(N2C(CCc3cn(CCCC)nn3)CCC2)=O)cncc(-n2cccn2)n1 Cc1nc2cc(C(=O)NC3CN(C(=O)CCNC(=O)C=CCl)CCC3C)[nH]c2s1 C1(CCC(=O)N(C2CCCCC2)C)CCCN(C(C23COCC2C3)=O)C1 Cc1c(C(N2CC(O)CC2CNC(=O)C(C)CC2CC2)=O)ccc2c1CCC2 N1(C(C2C(CC)OCC2)=O)CC(C)CN(C(C2CC2C2CCCCC2)=O)C(C)C1 C1(C)(C(=O)NCC2CN(C(c3c(OC)nsc3)=O)C(C)C2)CC2(CCC2)C1 C(C)(C(=O)NC1CCC1CNC(=O)C(=O)NCC(F)F)(c1ccccc1)OC N1(c2nc(C(C)C)cc(C)n2)CCC2(CCCN(C(C3CN(C)C(=O)N3)=O)C2)C1 C(=O)(C(F)CC(C)(C)NC(=O)CCC1CCOC1)NCc1c(C)nn[nH]1 Cc1ncsc1C1CCN(C(c2ncoc2-c2ccon2)=O)C1 C1(C(N(CC(C)(C)NC(C2CC(NCCO)C2)=O)C)=O)CC(F)C(=O)N1 N1(S(CC)(=O)=O)CCC(C(=O)NC2CN(C(=O)CCc3cccc(F)c3)C2)CC1 C(=O)(CC(C)C(C)C)N1CC(C(=O)NCCCOCC=C)C(C)C1 C(N=c1[nH]c(=NCc2nccn2C(F)F)c2ncccc2[nH]1)C1C(F)(F)C12CCC2 CCCCCCCCCCC(=O)NCC1COCC1NC(c1sccc1C)=O c1(NCC(c2ccccc2F)NC(C(C)OC(C)C)=O)ncc2ccccc2n1 c1(C(=O)OCC)nnc(SC)nc1N1CCC(NC(c2ccon2)=O)C(F)C1 N1(C(c2cnc(C)o2)=O)CCC(CCNC(=O)Cc2cn[nH]c2)CC1C C1(CNC(C(CCSC)O)=O)CCCCCN1C(=O)Cn1cccc(C)c1=O C1(C(=O)NCC2(OC)CN(C(C(COC)(C)C)=O)C2)CC1C1CCCC1 c1(C(C)O)ccc(C(=O)N(C)CCN(C)C(C2CC=CC2)=O)cc1 c1(-c2cn(C)nc2)ccc2cc(C(=O)NCC3CCO3)n(C)c2c1 Cc1nc(NCc2cc(C)nc(Cl)c2)c2c(C)c(C)sc2n1 c1(NCC(CC=C)(C)CO)[nH]c(=NCC2(C)CC(C)=NO2)nc2sccc12 CCN=c1[nH]cc(C(=O)NCCCCC(C)NC(c2cnn(C3CCC3)c2)=O)s1 C(=O)(CCC(=O)NC1CCC(Cc2c(C(=O)N)[nH]c(C)n2)C1)OCC c1(C(N2CC(C(C)NC(c3cnc(C(N)=O)s3)=O)C2)=O)cncc2nc[nH]c12 CCC(C)C(CC(=O)N1CCN(CC)CC1)NC(C1CNC(=O)N1)=O N1(C(C2(CC)CCC2)=O)CCC2CC2(C(=O)Nc2ccc(C(C)C)cc2)CC1 Cn1nc(C(F)(F)F)cc1CC(N1CC(O)(CNC(C2CCS(=O)CC2)=O)C1)=O C1(C(=O)NC2CC(CCNC(CC(c3ccccc3F)C)=O)C2)CCN(C)C1=O C1(NC(c2cccc(C(F)F)c2)=O)CN(C(=O)CCC2CC2(F)F)C2CC12 c1(C(C)C)c(C(=O)N(C)CCNC(=O)CC2(O)CCCC2)nc2n1CCCC2 c1(NC(C2CN(C(c3c(OC)scc3)=O)CC(C)C2)=O)cccn2ncnc12 c1(N(C2CNCC2O)C(c2c(C)c(Br)ccc2)=O)ncc2c(ccn2C)n1 C1(NC(C2CCCO2)=O)CCN(C(c2ccnc(C3CCCC3)n2)=O)C12CCC2 c1(C(N2CC(CCC)C(NC(=O)C(C3CC3)OC)C2)=O)cc(F)c(F)c(N)c1Cl C#CC1(C(=O)NC2CCCCC2NC(c2cc[nH]c(=N)c2)=O)CCCC1 c1(CNC(C2CC(CNC(Cc3cc(C)on3)=O)OC2)=O)nn(C)c(=O)n1C c1(C(=O)NCC(CC=C)NC(=O)CCCc2ccc(Br)s2)ncccc1C C1(CSC)CCCCN(C(C)=O)C1.c12nc(cc(C)n1)N1CCC(C1)CC(=O)N2 N1(C(C(C)(C)CC2CC2)=O)CC(CNC(C23CCCC2C3(F)F)=O)C2(CC2)C1 N1(C(CCC2CCN(C(C(C)CC(F)F)=O)C2)=O)CC2(CCOC2=O)C1 Cc1ncc(Br)cc1C(=O)NCC1(O)CCCN(C(=O)CC2(CO)CC2)C1 C(CCN(C(=O)CC1CC(N(C)C)C1)C)(C(C)(C)C)NC(C(COC)OC)=O C(C(C)(C)CNC(=O)Cn1cccn1)N(C(=O)CSCC(=O)OC)C C1(C(N2C(C)(C)C(CNC(c3cnsn3)=O)CC2)=O)Cc2ccc(F)cc2O1 C(=O)(C#CC(C)(C)CNC(C1CC1(C)C(C)C)=O)Nc1c(C)ccc(O)c1C c1(N(C)C)nc(C(N2CCC(C)(NC(c3cc(Cl)nnc3O)=O)C2)=O)cc(O)n1 C1(CNC(c2c(C)ccn2C)=O)CN(C(=O)CC2CCS(=O)(=O)C2)C2(CCC2)C1 C12(CNC(CC)=O)CN(C(c3cc(COC)cs3)=O)CC(F)(C1)C2 N1(C(C2ON=C(C)C2)=O)CC(C2CC2C(=O)NCCn2ncnn2)C1 C=C=CCC(=O)NCC(O)CNC(=O)CCC1CCOC1 N(C1C(=O)Nc2cccnc21)C(C(N)Cc1cc(F)ccc1F)=O c1(NC2CC(NC(c3cnc(C)n3C)=O)C2)nc2ccc(O)cc2s1 N1(C(CCNC(C)=O)=O)CC2CCC(C1)N(C(c1cc([N+](=O)[O-])cs1)=O)C2 N=c1ccc(C(=O)NCC(c2ccccc2)NC(=O)C=Cc2ccsc2)n[nH]1 CC1COCCN1CCNC(=O)CC(C1CC1)NC(=O)CC1CSCCO1 C(C)(C(=O)N(CCC(=O)N1CC(SC)C1)C(C)C)(C1CC1)OC N1(C(C2CNC(=O)O2)=O)CCC(F)(c2cn(-c3cccnc3)nn2)CC1 c1(C(=O)NCCC2(NC(COCCCC)=O)CCC2)cc(F)ccc1CC Cc1c(C(=O)NCCN(C(=O)CSC(F)F)CCOCCO)ccn1CCO C1(C(N2CCC(C)(CNC(=O)C(F)(F)F)C2)=O)CC2(COC(=O)N2)C1 C12(NC(c3c(C)snn3)=O)COCCC1CN(C(C1(C)CSC1)=O)C2 c1(N2CCC(C)C2)ccc(S(=O)(=O)N2CCC(CC3CCCO3)C2)cc1Cl C1(C(=O)NCC(CNC(=O)COc2ccc(Cl)cc2)OC)CCCCC(C)(C)C1 N1(C(c2ccc(CC)c(F)c2)=O)CCC(=O)C(C)C1CC C1(NC(c2c(CC)cco2)=O)CN(C(=O)C=Cc2ccc[nH]2)C2(CCOC2)C1 Cc1nnc2n1CCCC2C(=O)N1CCCC(CN(C(=O)C(O)CF)C)C1 O=C(C#CC1CCCCC1)N1CC2(C1)CN(C(C1(O)CCOCC1)=O)C2 C1(CNC(c2c(C)nco2)=O)C(O)C(O)CN1C(=O)Cn1ccc(C(F)F)n1 C12(NC(CCC)=O)CCCC1CN(C(c1cc(-c3ccccc3Cl)[nH]n1)=O)C2 C1(CC(C)C)CC(C(=O)NCC2CN(C(C3(C)CC3)=O)CCN2C)CC(=O)N1 C(=O)(C1=CCC(F)(F)CC1)NC1CCCCCN(C(C=CC(CC)C)=O)C1 N1(C(C2CCCN(C(=O)Cc3ncccc3F)CC2)=O)CCOCC(F)(F)C1 N1(C(C(c2c(C)nn(C)c2)O)=O)CC2CCCC(C1)N2C(=O)C(F)C(C)(C)O C=CC1CN(C(c2csc(COC3CCC3)n2)=O)CC1NC(=O)C(F)(F)CC Cn1[nH]c(C(N2CCC(CCNC(=O)CSc3cccc(F)c3)CC2)=O)nc1=O S(=O)(=O)(c1ccc(NC2CC2(C)C)c2cnccc12)N(C1CN2CCC1CC2)C CCCC(CCC)C(=O)NCCCCCC(=O)NCc1ccc(F)cc1O C(=O)(C1=CC2CC=CCC12)NC1CC(NC(c2c(O)ccc(C(C)C)c2)=O)C1 c1(C(N2C3CN(C(C(=O)NCC(C)C)C)C(CC3)C2)=O)cccc2c1CCOC2 N1(C(C(COC)O)=O)CCN(C(c2cc(O)nc(Br)c2)=O)C(CO)C1 N(C(=NCCF)NCC1CCOC(C)C1)CC1(COC)CCOCC1 Cn1cncc1C=CC(=O)NC1CCCC1CNC(=O)Cc1coc(C(F)F)n1 C1(C(N(C(CCNC(C2N=C(C)SC2)=O)C)C)=O)CC2(CCC2)C1 c1(SC)cc(C(=O)NC2CCN(C(c3ccnn3C3CC3(F)F)=O)C2)co1 C1(C(=O)NC2CCN(C(c3cn(C)nc3Br)=O)C2)CCn2c(O)nnc2C1 c1(C(N(CCCCO)C)=O)[nH]ccc1CNC(=O)C(C)(F)c1ccon1 N1(C(C(=O)NCCOCCCC)=O)CCC(NC(C2(C)CC2(C)C)=O)C(O)C1 N1(C(CC(C(C)C)C)=O)CCC(C2CCCN(C(=O)Cc3nccn3C)C2)C1 CC1CCN(C(=O)C=CC(=O)NCC2CCCO2)CC1N(C)C(C1CC1(Cl)Cl)=O N1(C(C(C)CC2CCCC2)=O)CC(F)(F)CC1(C)CNC(c1cnn(C)c1)=O CC1(C)CC(CCNC(=O)N(c2cc[nH]n2)Cc2cocn2)CNC1=O C12(C(N3C(CN(C(=O)CN4CCCNC4=O)C)CCC3)=O)CCCC(C1)OC2 c1(C(N(C(C)CN(C(=O)CCc2n[nH]c(=N)s2)C)C)=O)nc(=O)n(C)[nH]1 C1(C(N2CCC(CN(C(=O)CC3CC3(C)C)CC)CC2)=O)(COC)CCOCC1 c1(C(N2CC3CCCC(OC)C3C2)=O)oc2ccc(I)cc2c1C CC1CCc2nc(CNC(=O)CC(C)NC(=O)OC(C)(C)C)sc2C1 Nc1cccc(F)c1C(N1CCCC1CCNC(=O)Cc1c(F)cccc1F)=O c1cc(-n2cc(C3CCOC3)nn2)c2c(c1)COCC2 c1(CC)ccc(C(N2CCC(Nc3ncc4c(n3)COC4)C2)=O)cc1[N+](=O)[O-] CCC(C)CCC(=O)N1CCCCC1CN(C(=O)CCn1cccnc1=O)CC CC1COC(C)(C)CN1C(=O)CCC1(C)CN(C(C2CC(=O)NC2(C)C)=O)C1 Cc1cc(C(=O)NC(C(=O)NCCc2ncoc2C)c2ccoc2)co1 CCC(CC(=O)N1CCCC1(C)CCC(=O)NCCC(C)(O)C1CC1)SC C1(C(=O)NCC2(NC(c3c(CC)nccc3)=O)CC2)CCC(O)CN1C N1(C(COCCOCC)=O)CCC(C(=O)NCCn2cnccc2=O)C1C Cc1cc(-n2cc(C3CN(C(c4cnn(C)c4C(=O)O)=O)C3)nn2)nn1C C1(N(C)Cc2nc(SCC(F)(F)F)no2)CCS(=O)(=O)C1 C1(CCOC)(NC(c2sc(F)cc2C)=O)CCN(C(C2(N(C)C)CC2)=O)CC1 c1(C(N(CC(CN(C(c2ccc(C#C)o2)=O)C)O)C)=O)cnc2sccc2c1 c1(C(N2CC(C)(NC(C3CC(CC)C3)=O)C2)=O)cc(Br)ccc1N Cc1ccnc(N2CCC(CF)(NC(c3cc(Br)co3)=O)C2)n1 C1(NC(C2(CC)CC(C)(C)C2)=O)CC(C)CN(C(=O)C=CCOCCOC)C1 CCC(CC(=O)N1CCOC(CC(=O)NOCCCN(C)C)C1)OC c1(OCC)nc(N2CC(C(=O)Nc3ccc(C)nc3C)C2)ncc1OC CC(C)(C)CCCCCC(=O)N1CCN(C(=O)CC(O)C(C)(C)C)CC1CCO C1(CC(=O)NCC(Cn2cc(CC3(O)CCC3)nn2)OC)CCC(=O)CC1 O=C(NNc1c(F)cccc1Br)c1ccc2ccccc2n1 c1(C(=O)NCC2CCC(NC(CCC(=C)C)=O)C2)cc2cc(OC)ccc2[nH]1 C(=O)(CCN(OC)C(=O)CNC(=O)NCc1ccco1)NC(CCOC)C(N)=O c1(CNC2(c3nnnn3CCCF)C(OC)CCC2)nnc2cccnn12 c1(-c2ccc(CCCCNC(=O)OCC3CCCO3)o2)ccccc1Cl N1(S(CC(C)(C)F)(=O)=O)CCc2c(OC3CCCC3)cccc2C1 C(CNC(C1(Cl)CC1(F)F)=O)(C(=O)N(C)C(c1cccs1)C)OC CC1=C(C(=O)N2CCC(N(C(=O)C=Cc3cscn3)C)C(C)C2)CCO1 c1(OC)cccn2ncc(C3CCCCC3)c12.c12ccc3nc(oc3c1)C(=O)N2 C1(O)(CN(C(=O)CC2CC=CC2)C)CCCN(C(c2nc[nH]c2C(C)(C)C)=O)C1 c1(CCCO)cc(C)ccc1N(C)C.C12(C)C3C4C5C3C1C5C24.C(=O)OCC C1(OC)CC(C(N2CC(C)(NC(=O)CCSc3ccc(C)cc3)C2)=O)CC1OC c1(C(=O)NCC2CCCC2NC(c2cocn2)=O)ccc(F)c(C2CC2)c1 C1(OC)(CNC(=O)Cc2ccns2)CCN(C(=O)COCCCN=[N+]=[N-])C1 Nc1ncc(Br)nc1C(=O)NCC1CC(NC(C2C=CCC2)=O)CCO1 C1(C(=O)NCCN(C(C2CCC(C)(C)C2)=O)CC)OCCCC1(C)C c1(C(N2CCN(C(CC(C)C3CC3)=O)CC2C)=O)ccc2c(n1)NCC2 CCCC(C)(CC)C(=O)N1CC(CNC(C2(C#N)CC2(C)C)=O)C(C)C1 Cc1ccc2cc(C(=O)NCC(C)(C3CCC3)NC(=O)C(C)C3CCC3)oc2c1 C(=O)(C1CNC(=O)c2ccccc21)NCC(C(C)(C)C)NC(COC(CC)C)=O n1(CCOC)nccc1C(=O)NCC(O)CN(C(=O)CCCC1CCCC1)C c1(C(=O)NC2C(CNC(CN3CC(CC)C3)=O)C2)ccc2oc(S)nc2c1 C1(NC(C2CCN(C(C)=O)CC2)=O)CN(C(c2csnn2)=O)C(C)(C)C1 c1(C(=O)NCC2C(NC(CSC(C)(C)C)=O)CCC2)cnc2sccn12 C1(NC(C2N(CC)CCCC2)=O)CCCN(c2cc(Cl)c(O)nn2)C1C c1(OCC)ncccc1C(=O)NC1CN(C(c2cc(C)cc(C)n2)=O)CC2CC12 CC1(C)CCCN(C(c2cncc(Cl)n2)=O)C1CNC(=O)CCNC(=O)CO c1(SCC(=O)NCc2cn(CC(O)COCc3ccccc3)nn2)ccccc1 N1(C(c2ccc(Cl)c(C)c2)C(=O)NCCCCCC)CCC2(CCC3CC2C3)C1 C1(OC)CC2CCC1(NC(C1CC3CC1CC3NC(=O)OC(C)(C)C)=O)C2(C)C C(=O)(C1=CCCN(C(C2CCOC2C=C)=O)C1)NCC(CC=C)(C)C C1(C(C)(C)C)(CNC(c2cc(CCCO)on2)=O)CCN(C(c2cc[nH]n2)=O)C1 C1(CNC(C(CC)O)=O)N(C(c2nccc3[nH]ccc23)=O)CCCC1(C)C C(CC(C)C(=O)NCC1CCN(C(c2c(Br)nnn2C)=O)C1)OC C1(NC(CC2(C(=C)F)CCC2)=O)COC2(C1)CN(C(=O)COCC1CCCC1)C2 c1(N(C)CC2(SC)CCC2)nc2ccccc2c(=NC(C)C2CCC2)[nH]1 C1(NC(COCCCC)=O)COC2(CCCN(C(=O)C3=C(Cl)CCC3)C2)C1 C(=O)(CCCC(F)(F)CO)N(CCCCCCNC(c1ccnc(Cl)c1O)=O)C c1(OC)cc(N)ccc1C(=O)NCC1C2CN(C(C34COC(CCO3)C4)=O)CC12 Cc1cc(=NC2CC(CS(C)(=O)=O)C2)[nH]c(N2CCOC(C3(N(C)C)CC3)C2)n1 CC(C(C)C(=O)NC1C=CCN(C(c2c(Cl)ccnc2Cl)=O)C1)S(C)(=O)=O C1(CNC(c2c(CC)ncs2)=O)CN(C(=O)C(C)(CC)OC)CCC1(C)C Cc1nncc(C(N2CCCC2CN(C(=O)C=CSCc2ccco2)C)=O)c1C N1(C(N2CCC(CO)C2C(F)(F)F)=O)CCC2(CC=CCO2)CC1 N1(C(C2(CSC)CCC2)=O)CC(CNC(=O)C(C)c2ccco2)C(O)C1 c1(C(=O)OC)ccc(CC(C)C(=O)N2CCCC2Cc2cnn(C)c2)cc1F C(=O)(C1=CCCC1C)NC(CSCC)C(=O)NCCCCCCN(C)C C1(CNC(CCC=C)=O)CN(C(=O)C(C)SCCCC)CCC12CCC2 c1(CS(=O)(=O)NCC(CC)(C)c2nn[nH]n2)cc(OC)ccc1F CCCCC(C(=O)N(C)CC1(O)CN(C)C1)NC(=O)CCC1CCCO1 c1(OC)ncccc1C(=O)N(C)CC1CN(C(=O)CC(C)(C)C)CCO1 C1(C(=O)NCCOC(=O)CNCC)CC(C)N1C(=O)C=C(CC)CC Cc1cc(N2CC3CCCN(C(=O)C(F)CC4CC4)C3C2)n2nc(C)nc2n1 c1(COC)nc(N2CCC23CN(C(c2ccc(C)c(I)c2)=O)C3)cc(O)n1 C(=O)(CC(CNC(C1(C)CCCCO1)=O)C1CCC1)NC(c1ccc(F)cc1)C c1(CSC)cccnc1C(=O)NC1CCN(C(C2CCC3(CC3)C2)=O)CC1 C1(N(C(C(C)OCCC=C)=O)C)CN(C(c2cn(C(C)C)nc2C)=O)CC1(C)C Cc1ccc(C(=O)N(C2CCCC2)CCCNC(=O)C2=NOCC2)c(F)c1C C=C=CCCC(=O)NCc1noc(C(C)(C)C)n1 C1(NC(=O)C(C2CCCCC2)NC(C2CC3CCC3C2)=O)CCc2nncn2C1 C(=O)(C1=CS(=O)CCC1)N(CC(C)NC(c1csnn1)=O)CC c1(C(=O)NC(C(=O)NCCNC(N)=O)CC(F)F)cc2cccnc2[nH]1 c1(-c2cn(C(C(=O)N(CCCN(C)C)CC)C)nn2)cnc(C)c(C)c1 C(=O)(C1COc2ccc(Cl)cc21)NC1C2(CC(NC(CC=CC)=O)C2)C1 C1(C(=O)OCC)CN(C(=O)C2=NOC(C3(O)COC3)C2)CC12CCN2 C1(CNC(c2cccn3nncc23)=O)CC12CCN(C(=O)C(O)C1CCC1)CC2 c1(OC)ccncc1NC(=O)COCC(N1CCC(Nc2ccccc2)C1)=O c1(NC(C(c2cccc(OC)c2)C)=O)cc(C(=O)O)c(C)c(C)c1 c1(N2CCC(C)C2)nc(=NC2CC3(CCC3)C2)[nH]c2c1CCC2 C1(NC(c2n(C3CC(SCC)C3)nnn2)c2scnc2Cl)CCCOC12CCC2 c1(C(=O)NC2CN(C(C(CC)C#N)=O)C2)cnn2cc(Br)cnc12 C(=O)(C1=CNC2=NCCCN12)N1CCC(CNC(C(C)(O)C2CC2)=O)C1 C1(CNC(C2(CC#C)CCCO2)=O)CCN(C(=O)CCCC2CC2C)CC1O c1(-n2cc(OCOC)nn2)ccccc1CCC(=O)OC(C)C(C)F c1(C(N2CC(CNC(Cc3cc(C)nn3C)=O)OCC2)=O)cc(Cl)c(Cl)cc1C C(=O)(C1COc2ccccc21)NC1C(C)(CNC(c2c(CC)occ2)=O)CCC1 C1(C(N2CCN(C(CN(CC(=O)NC(C)C)C)=O)CC2)=O)C2C(=O)OCC12Br C(C(C)(C)CC(=O)N1CCC(O)C1C(=O)NCCC1CC1C)OC c1(CC(=O)NCC2N(C(C(CCCC)O)=O)CC(O)C2O)cn2ccccc2n1 C12(NC(C(CCC)OC)=O)CCC(C(=O)NCCc3ccncn3)(CC1)C2 c1(C(N2C(C)(CC(N3CC(CC(=O)OC)C3)=O)CC2)=O)ccc(C)cn1 N1(C(c2cnsc2)=O)CC(F)(F)CC1CNC(=O)C(F)(F)c1ccncc1 c1(C(C)C)cccc(OCC(=O)NCCCC2(NC(=O)C(O)CC#N)CC2)c1.C CCC(CCC(=O)N1CC(N(C)C(c2cc(OC)n[nH]2)=O)C2(CC2)C1)OC CC(C)CC(C)C(=O)NC(CN=[N+]=[N-])C(=O)NCc1cncc(C#N)c1 c1(OC2CC2)cnc(C(=O)NCC2(C)CC(C(=O)Nc3ccc(CO)o3)C2)nc1 Cc1cnc(C)c(C(=O)NCC2CCCCN2C(c2ccnc(O)c2)=O)n1 n1(C(C)(C)C)cc(C(=O)NCC2C=CC(NC(=O)C(F)=CC3CC3)C2)cn1 N1(C(c2c(C)cncn2)=O)CCC2C(CCCN2C(=O)CN(C)C)C1 c1(C(N2CCC2c2cn(Cc3ocnc3C(=O)OC)nn2)=O)occ(C)c1OC C(CC(C)C)(C(=O)NCC1CC1c1ccncc1)ONC(=O)C1C(OC(C)=O)C1 N1(CC(=O)N(C(CNC(c2c(C)[nH]nc2Br)=O)C)C)CCCCCCC1=O C(N=c1[nH]c(Cl)c(C#N)s1)C1(CNC(C2CCC(CC)O2)=O)CC1(F)F C1(Cn2ncc(C)c2)CCN(C(C(=O)NCC(C)C)c2ncco2)CC1 c1(C(C(=O)N(CCCCCNC(=O)Cn2ncn(C)c2=O)C)O)ccc(F)cc1 C1(CN(C(=O)COC2CCOCC2)CC)CCCN(C(=O)CCC(C)OCC)C1 c1(NC(=O)CCCSc2ccn(C)n2)cccc(Cl)c1.C12CC(C1)N(C)C(=O)C2 C1(CNC(CCSCCC)=O)CC2(CCN(c3nc(C(F)(F)F)ns3)C2)CO1 C1(C)(CC)CC(NC(=O)C=Cc2ccsc2)CN1C(=O)Cc1cnn(C(F)F)c1 S(=O)(=O)(c1cc(C(=O)NC2CC3CC(NC(=O)CSC(F)F)C2C3)co1)NC CC1CN(C(c2c(Cl)cncc2Cl)=O)CCCN1C(c1cn(C)nn1)=O Nc1cccc(CC(N2CC(NC(=O)C=Cc3ccc(Cl)cc3)C(O)C2)=O)c1N c1(NCC2(O)CC(OCC)C2(C)C)cc(Br)cc2nn[nH]c12 Cc1cc(C(=O)N(CCCNC(=O)CN(C)C)CCO)nn1-c1ccccn1 C(=O)(C(C)S(C)(=O)=O)N1CCC(N2CCN(C(c3cccc(OC)c3)=O)CC2)C1 c1(N(CCCOC)C)ncccc1S(=O)(=O)NC(C)C(C)CO N1(C(c2c(COC)nn[nH]2)=O)CCC(C2CC2)C1CNC(=O)CC1(COC)CC1 C1(C(=O)NC2CN(C(C=CSC)=O)C2)CC(O)CN1C(C)=O N1(C(C(CCSC)N(C)C)=O)CCCN(C(c2cnn3c2CCC3)=O)CC1 C(=O)(CC(C)CC(=O)N1CC2C(C1)C(=O)N2)OC.C(CCOC(C)=O)OC CCCCC(F)C(=O)NCc1cncc(C(=O)NC(C)CCC2CCCO2)c1 C1(C(=O)N(C2(CC(=O)NC3(CC(C)C)CCC3)CC2)C)(OC)CCC(C)(C)C1 CN1C(=O)CSC1=CC(=O)NC1(CF)CCN(C(C2CN3CCN2C(C)C3)=O)C1 C12C(O)C(O)CN1C2=O.c1(-n2c(C(=O)OC)cnn2)ccc(F)cc1Cl c1(-c2n(C)c(N3CCOC(C(F)(F)F)(C(F)(F)F)C3)nn2)cn2ccsc2n1 Cc1ccnc(C)c1C(N1CCCN(C(=O)CCn2cncn2)CC1)=O C(=O)(CC(O)C(=C)C)NC(CNC(COCCOCC#C)=O)CO c1(C(N(CC(COC)(C)C)C)=O)ccnc(CNC(=O)C(C2CCOCC2)F)c1 C(=O)(C(O)C(C)C)NCCC1CCN(C(C2(C(C)C)C(C(=O)OC)C2)=O)C1 Cc1nc(C)c(C(N2CC(NC(c3sccc3CC#N)=O)C(C)C2)=O)[nH]1 Cc1ccc(C(C)CC(=O)N2CC(NC(=O)CCCc3ccc(C)cc3)C2)cc1 C(CN=[N+]=[N-])(C(=O)NCCN1CC=CCC1)NC(C1CCN(CC)C1)=O c1(C(N2CCC(O)(CCNC(C(c3cnn(C)c3)C)=O)C2)=O)cnc(O)cc1O c1(NC(C(C(=O)N(C(CO)CO)C)NS(C)(=O)=O)=O)cc(Cl)cc(Cl)c1 c1(CC(=O)NC2C3CN(C(c4nc(CCC)sc4)=O)C2C3)ccc([N+](=O)[O-])cc1 C1(NC(C(C2CC2)OCC)=O)CN(C(C2CC3C=CC2C3)=O)CC1C(F)F C(=O)(C1=COCCC1)NC1CCC(N(C(CCN(C(C)=O)C)=O)C)C1 N1(S(CC(C)C)(=O)=O)CCC2(CCCC2C(N2CCN(C3CCCC3)CC2)=O)C1 C(C(O)CC(=O)NCC1(F)CCC(NC(c2csc(Cl)n2)=O)C1)N(C)C C1(CC=CC)CCN(C(=O)C(Cc2ccoc2)NC(c2ocnc2C)=O)CC1 C1(C2CCCN(C(=O)CN3CCS(=O)CC3)C2)(NC(=O)CN2CCCC2=O)CC1 CN1CCCC(C(=O)NC2CCN(CCCO)C2)C1.n12cc(nn1)C(=O)NCC2 c1(C(=O)NC2CCC(N(C(=O)CC3CCCC34CC4)C)CC2)ccc(O)c(Cl)n1 n1(C(CC)CC)nc(C(N2CC(NC(C3CC3(C)CC)=O)C2)=O)cc1C C1(NC(C2C(C)(C(F)(F)F)C2)=O)CC2CC(NC(=O)CN3CCOC3=O)CC12 O=C(CC1=CCOCC1)NCC1CCC(NC(c2ccc[nH]2)=O)C1 C1(NC(c2cc(OC)no2)=O)CC(N=c2ccnc(SC)[nH]2)C12CCOCC2 C(CC(C)(C)C)(c1n(CC(=C)C)nnn1)NCc1c(Cl)cnn1C CCC(CN(C)C)CC(=O)N1CCCCC(C(N2CC(C(C)C)C2)=O)C1 n1(CC)cnc2c(NCC34CCCC3C4(F)F)[nH]c(=NCCC(C)C)nc12 c1(OC)ccc(C(CNC(=O)CC2CC2(C)C)NC(=O)CSC(F)F)cc1 Cc1ccc2c(c1)N(C(C1CCCN(C(=O)C(n3nccc3C)C)CC1)=O)CC2 C(=O)(C1CCCc2ccccc21)NC1CC(CNC(C2(C#N)CC2)=O)CC1O c1(CCC(=O)NC2CN(C(c3c(C)cc[nH]3)=O)C3C2C3)cccc(Cl)c1Cl N1(C(c2c(N)nccn2)=O)CCC2CN(C(C3CC(=O)NC(=O)C3)=O)C2C1 c1(C(=O)NCC(CNC(C(CC(C)C)OC)=O)(C)F)occ2c1CCOC2 C1(NC(c2ccc(Cl)cc2I)=O)CCNC2(CCC2)C1 N=c1[nH]c(-c2c[nH]cc2C(=O)NCCC2CC(NC(=O)C(O)CC3CC3)C2)cs1 Cc1cnc2cc(C(=O)NC(C)CCCNC(c3cn(C)ccc3=O)=O)ccn12 C1(NC(CSCCOC)=O)(CF)CCN(C(=O)C(=Cc2cnn(C)c2)C)C1 Cc1ncnc(C(N2CCC(C(F)CNC(C3(C)CCCS3)=O)CC2)=O)c1C C(=O)(C(CC1CC1)C(C)C)NC(CC(=O)NC(c1ccccc1F)C)(C)C CC1CN(C(C2CCC(C)C2)=O)CC1NC(=O)C(c1ccccn1)O Cc1cccc(CNC(N2CC(CNC(c3n[nH]cc3Cl)=O)CC2C)=O)c1 C(c1ccc(Cl)cc1)=CCN1C(C(=O)Nc2ccnnc2O)CC1 c1(C(=O)NC(C2N(C(CC(=C)C)=O)CCC2)(C)C)cccc2cccc(OC)c12 N1(C(C(=O)NC(c2onc(C)n2)C)=O)CCc2cc(Br)ccc2C1 CC1=NN(C)C(=O)C1CC(=O)NC(C)CCN(C(=O)CCc1ccncc1)C c1(C(N2CC(NC(C3(F)C(C)OCC3)=O)C(C)(C)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C=CC(C)(C)CCNC(c1[nH]ccc1CNC(C1CC=CCC1)=O)=O c1(NCCC(C)N)ccc(S(=O)CCC#N)cc1 c1(C(=O)NC(CN(C(c2ccc(OC)s2)=O)C)C)cc2c(F)cc(F)cc2o1 c1(C(N2CC(C)(NC(CC3N(CC)C(=O)CC3)=O)C2)=O)nccc2cccnc12 Cn1ccc2cc(C(N3CCC4(COC(CNC(=O)C=CCO)C4)C3)=O)cnc12 C1(C)(C(=O)NC2CN(CC)CC2C)CCCN(C(C2CCCN2C(C)C)=O)C1 c1(CC(=O)OC)c(C(N2CCC(F)(Cc3ccccc3)C2)=O)[nH]c2ccccc12 C(=O)(C(C)CC(C)C(C)=O)N1CC(C(N2CCC(COCC)C2)=O)(COCC)C1 n1(CC)cnnc1C(=O)NCCCCN(C(=O)C(O)Cn1cncn1)C C(c1cncs1)=CC(=O)NC(C1(C(=O)NC(c2nncn2C)C)CC1)C CCCC(C(=O)N(CCC)CCNC(c1coc(C(F)F)c1)=O)C(C)C CC(C)CC(C)(C)C(=O)NC1CCN(C(=O)C(C)(C)Br)CCC1CO c1(OC)ccccc1C(C)(C)C(=O)NC1CC(CNC(=O)C2=CCOC2)C1 C1(OC)CN(C)CC1N=c1[nH]c(=N)[nH]c(=NCP(C)(C)=O)[nH]1 c1(C(=O)NCC(CNC(C2C(C)(C)C2(C)C)=O)OC)cc(Cl)cc(C)c1O N1(C(C(C)NS(C)(=O)=O)=O)CC2(COC(CNC(c3cc4n(c3)CCC4)=O)C2)C1 c1(COC)ccc(C(N2CSCC2C(=O)NOCC2CCCO2)=O)o1 C1(C(N(c2csc(N3CCOCC3)n2)C(C)C)=O)C2CCC1(c1ccn(C)n1)C2 O=C(COc1ccccc1Br)NNC(=O)c1ccc(OC(F)(F)F)nc1 C1(C(N(CCC(=O)NC)C)=O)CCCC1CNC(=O)CCCn1ccnc1 c1(C(=O)NC23CCN(C(c4cnc(Cl)[nH]4)=O)CC2C3)ccc2c(c1)COC2=O N1(C(C(CC#C)C2CC2)=O)CCC(C2CC2NC(=O)Cc2sccc2Cl)CC1 C(CC1=CCCCC1)NC(CC1CCN(C(Cc2c(C)ocn2)=O)C1)=O c1(C(N2CCC(NC(C34CC(C)(C3)C4)=O)C(O)C2)=O)cc(O)c(F)cc1N C1(C(N(CCF)CC)=O)(SC)CN(C(=O)C=Cc2cncs2)C1 C=CC1(C(N2CCCN(C)CCC2)=O)CCN(C(=O)C(C)NC(=O)C2CC2)CC1 N1(C(COCC(C)(C)C)=O)CCN(C(c2ncsc2C2CC2)=O)CC(O)C1 N1(C(C(C(CC)C)NC(C)=O)=O)CC2CCC(C1)N2C(C1CC(=O)N(O)C1)=O c1(C(N2CCCN(C(C=C(COC)C)=O)CC2C)=O)coc2c1CS(=O)(=O)C2 c1(C(=O)NCC=CCNC(c2ccc(C(N)=O)s2)=O)ccc2nncn2c1 N1(C(CC(COC)(C)O)=O)Cc2nccn2CC(NC(c2cscc2Cl)=O)C1 C=CC(CCC)CC(=O)NC1COC2(CNC(c3csc(Cl)c3)=O)CC1C2 Cc1sccc1CC(=O)N(CCNC(=O)CSC1CCOC1=O)C1CC1 c1(COC)nc(C(=O)NC(C2CC(NC(=O)Cc3cccnc3)C2)C)cs1 Cc1ccc(F)c(C(=O)NC(C)(C)C)c1S(=O)(=O)NCc1n[nH]c2c1CCCC2 C(=O)(C#CC(C)(C)C)N1CC(n2cc(CNC(c3ccc(CC)[nH]3)=O)nn2)C1 N1(C(C2(C)CCC(F)(F)C2)=O)CCCCC(O)(CNC(=O)CN2CC3CC3C2)C1 N1(C(c2cnc(C(C)C)s2)=O)CCCN(C(=O)CC2(O)CCOC2)C(C(C)C)C1 C=CCN=c1[nH]c(C(N2CCCC(C)(NC(=O)C(C)CC)C2)=O)cs1 C1(CC(C)NC2(C)CC2OC2CC2)CCN(C(=O)CCOC(C)(C)C)C1.C(=O)NCO C1(C(=O)NC(C)(CNC(=O)CCc2ccc(Cl)nc2)C2CC2)CC2(CCCC2)C1 c1(C(N(C(CC)C2CC2)C)=O)sccc1CNC(c1ccc(C)s1)=O c1(C(N2C(CNC(CC(C)C(F)F)=O)CCCC2)=O)n[nH]c2c1COCC2 CC1CCN(C(=O)CCC#N)C1CNC(c1cc(C(F)(F)F)ncn1)=O C(=O)(CC(F)(F)C(C)(F)F)NCCOCCN(C(C=CCN(CC)CC)=O)C C1(NC(Cc2ccc(OC)cn2)=O)CCN(C(=O)Nc2cnnc(O)c2)CC1O CC(F)(F)CCC(=O)NC1CC1CNC(c1ccc(Cl)cc1)=O N(C(=NCCc1nc2c(s1)CCCC2)N1CCC(OC(C)C)C1)C(CC)C C(C(C)C(=O)NC(CN1CCCC1)C(=O)NC(C)(C)CCOC)OCC Cc1oc(C)c(C(=O)NC2CN(C(=O)CC(C)C3CC3)CC2C)c1C Cn1cnc2c(NC(=O)NCc3nc(C#N)cs3)ncnc12 c1(OC)cc(C(=O)OC)ccc1Cl.N1CC(C(F)(F)F)OC1=O.C1C(C)CN1C C1(C(C)C)CCC(C(N2CCOCC2CCNC(=O)CSC(F)F)=O)CC1 CCCCCCC(=O)NCC(C)(CC)C(=O)NCc1ccccc1C c1(CC(=O)NCC(CNC(C(CC)(F)F)=O)C)c[nH]c2cccnc12 c1(CNC(N2C(C#C)CC2)=O)nc2c(s1)C(C)(C)OC(C)(C)C2 C(N=c1nc(N(C2CCOCC2)C)c2c([nH]1)CCCCC2)C1(OC)CC(OC)C1 c1(C(=O)NCC(CC)NC(c2ccc(Cl)cc2)=O)n[nH]c2c1CC(F)(F)CC2 c1(OC)cccc(CN2CC(C(=O)Nc3ccnn3C)CC(F)C2)c1Br C1(C)(CC)CCN(C(=NCCC(=O)NC)NCC2(O)CCSC2)C1 c1(C(=O)Nc2ncc(C(=O)OCC)s2)cnc2c(Br)cc(Br)cc2c1 c1(NC(C(C)C)=O)cccc(C(=O)N(C2CCCCC2N(C(=O)CO)C)C)c1 c12ccccc1S2.N1(CCNC(C2CCCCC2)=O)CCNCC1 C1(CNC(C2(CC=C)CCOCC2)=O)(OC)CCN(C(=O)C(C)OCC)CC1 O=C(CC1CCCCN1C(=O)CN1CCCNC1=O)N1CC=CCO1 C1(C(=O)NCCCN(C(=O)CC2OCCCC2(C)C)CC)CCC(=O)N(C)C1 c1(C(C)C(=O)NC2CN(C(c3ncncc3F)=O)C2)ccc([N+](=O)[O-])cc1F C12(NC(c3c[nH]c(=O)cn3)=O)CCC1CN(C(=O)CCc1ccsc1)C2 C12(NC(C3(COC)CCN(C(COC(CC)CC)=O)C3)=O)CCCN(CC1)C2 c1(C)ccc(C2(C(=O)NON3CCCOCC3)CCCC2)cc1.C1CCCCN1 Cc1cc(Cl)cc(C(N2CC=CC(NC(=O)CC3CCCN(C)C3)C2)=O)c1C c1(C(=O)O)ccc2cc3ccc(-c4cccc5cc[nH]c45)cc3nc2c1 C(=O)(C(O)C(F)(F)F)NCCC1CC(OC)CN1C(c1ccc(C#N)o1)=O c1(SCCC(=O)N(CCNC(C(C)NC(N)=O)=O)CCN(C)C)ccccc1Cl C1(C(N2C(CNC(Cn3nnc(C)n3)=O)COCC2)=O)CCCCC(=O)C1 C1(C)(C(=O)NC(c2cccc(C)c2)CNC(c2cc[nH]n2)=O)CCCCC1(F)F C1(CN(C)CCF)COC(C(=O)O)C1 N1(C(C2(C(N)=O)CCC2)=O)CCN(C(=O)CN2CCCCC2)C(CCO)C1 C(=O)(CCC(=O)N1CCCC(CN(C)C(C)C)C1)N(CC)CC c1(CNC(CC2CCC(C)O2)=O)ccc(CNC(C2(F)CC=CCC2)=O)c(F)c1 N1(C(C(C(CNC(c2cc(C)oc2)=O)C)F)=O)CCC2CN(C)CCC12 C1(OC(C)(C)C)CCN(C(=O)NC(CC2(OC(C)=O)CC2)C)C1 Cc1cn(C(C)C)cc1C(=O)NCC1(F)CCC(CNC(c2cnc[nH]2)=O)C1 C1(NC(c2c(CCC)nco2)=O)CC(C2CCN(C(C3CCC(=O)O3)=O)CC2)C1 CC(CNC(=O)CC1COC(C)(C)C1)CN=c1[nH]c2cc(Cl)ccc2s1 c1(C(=O)NCC2C(C)CCN(C(COCC#C)=O)C2)ncnc2ccsc12 C#CCC(C)C(=O)NCC1C(C)CCN1C(c1cnc(-c2ncccn2)s1)=O c1(C(=O)NCCC(C)NC(=O)CC(C)(C)O)coc2c(F)cc(Cl)cc12 CC(C)S(=O)(=O)CCNC(c1ccncc1)c1nnnn1CCCC1CC1 CC1CN(C(C2(O)CCN(C)CC2)=O)CCN1C(=O)C(c1cncn1C)O N1(C(C2(C)CC(C)C2)=O)CCOCC(NC(=O)Cc2cncc(O)c2)C1 N1(CC(C)C)CCC(C(=O)N(CCCCNC(=O)C(C)c2ccsn2)C)C1 c1(C(C)OCCOC)nc(CO)nn1-c1ccc(-c2ccccc2)cc1 CC(C)S(=O)(=O)C(C)C(=O)N1CCC1CNC(c1ccccc1C(C)(F)F)=O c1(C(NNC(c2cnn3ccncc23)=O)=O)c[nH]c2c(Br)cccc12 N1(C(C(C)SC(C)C)=O)CC(C)C1C(=O)NCC1CCCSC1 N1(C(C(COC)COC)=O)CC2CCN(C(c3c(F)cc(F)cc3Cl)=O)CC12 Cc1[nH]nc2c1CCC(C(=O)NC(CNC(=O)C=CS(F)(F)(F)(F)F)C(C)C)C2 c1(C(CNC(C2(Cl)C(C)(C)C2)=O)NC(=O)CC2CC=CC2)cc(Cl)cc(Cl)c1 C1(NC(CCC(=O)NCC)=O)CCC2CCN(C(C3CCC(C)(C)CC3)=O)C1C2 C(=O)(CC(c1ccccc1)OC(F)(F)F)OC(C)(C)Cn1cncn1 C1(OCCC(=O)NC(C2CN(C(C(CC)F)=O)C2)C)CCN(C)CC1 c1(C(c2n(CCSC)nnn2)NCCCS(C)=O)nc(C)n(C)n1 c1(CC(C2CC2)NC(C(CCC)OCC)=O)nc2ccc(C)cc2[nH]1 C1(OC)(CNC(c2ocnc2C)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1 C1(OC)CN(C(=O)CCCC2CCCO2)CC1C(=O)NC1(CF)CC1 c1(C(C(=O)N(C(CC)CNC(=O)Cc2nncn2C)C)O)cn(C)nc1C O=C1CN(C(=O)C(=O)NCC2CC3(C2)CC3F)CCN1 Cc1ccc(CN2CC(C)(CC(=O)N(C)C)C2)c(Br)c1.c12ccccc1C(=O)N2 Cc1c(N)c(C(N2CC(NC(c3nccc(Cl)c3Cl)=O)CC2C)=O)nn1C c1(NCc2ccc(C(OCC)OCC)cc2C)ccc(C)cc1C C(=O)(C(F)C(C)(C)O)N1CCN(CC2CCN(C(C3(C(C)(F)F)CC3)=O)CC2)CC1 N1(C(c2c(CC)cco2)=O)CCN(C(=O)C(c2cc(C)oc2C)C)CC1CC C1(CNC(c2cncnc2)=O)CC(O)(CNC(c2cc(C3CC3)on2)=O)C1 CN1CCOc2c(C(=O)NC3CCC3NC(c3cncc(C#N)c3)=O)cccc21 c1(C(N2CC(C(N(CCC=C)CC)=O)(CC=C)C2)=O)c[n+]([O-])c(C)cn1 CC(CC1CCCCC1)C(=O)N1CCC(CNC(=O)CC2CC(C)(C)C2)C1 c1(OC)ccnc(F)c1C(=O)NC(C)CCCNC(C1CCCC1SC)=O C(CO)(CCCCNC(c1n[nH]c(C2CC2)c1Cl)=O)NC(C1C(C)(C)CCC1)=O n1(CCC(=O)COCCNCCC)ccc(C(=O)OCCSC)n1.C1(=O)CN1.CC#N CC(C)(C)C(C)(C)C(=O)N1CCC(CNC(=O)C2=COCC2)CC1 C(=O)(C1OC(=O)c2ccccc21)N1C(CNC(C2COC(C)(C)O2)=O)CCC1 c1(C(=O)NCc2c(C)ccs2)ccc(NC(=O)C(C)OCC(C)C)cc1F N1(C(=O)OC)CCCN(Cc2c(Cl)cccc2I)CC1 c1(C(CNC(C2(OC)CC2)=O)NC(C(F)OC)=O)ccccc1OC c1(C(=O)NCC(CC)NC(C(F)=CCC)=O)cc2c(C)cc(C)nc2s1 N1(C(CCC(=O)OCC)=O)CCCC(C2CCCN(C(C3CCN(C)C3)=O)C2)C1 C(=O)(C(CC(C)C)N)NCC(F)(F)Cl.CCC(C)N(C(C)=O)CC CC1CCC(Cl)=C(C(=O)N(CCNC(=O)CC2CCC(F)(F)CC2)C(C)C)C1 n1(C(C)C)ccc(C(=O)NCC(CNC(=O)Cc2cnccn2)CO)cc1=O c1(OC)cc(C)n(OC(F)F)n1.C12CC(F)(C1)C2OCC(C)(C)OC c1(CCCCC)noc(CCNC(c2ccc(Cc3ccccc3)cc2)=O)c1C CC1(C)CCC(C(=O)NC2CN(C(=O)CC3(O)CCCC3)CC2F)C1 N1(C(Cc2c(C)scc2)=O)CCC(N(C)C(C2C3CCCCC23)=O)C2(CC2)C1 C1(C(=O)NCC(CO)NC(C(CC)SC)=O)CC2CCC1O2 N1(C(c2ccc(CC(CC)C)[nH]2)=O)CC2CC(C(=O)NCCO)CC2C1 C1(C(N(C)CC2CCN(C(=O)Cn3nnc(=O)[nH]3)C2)=O)CC2(C1)CC(O)C2 c1(C(C(=O)CCCCn2cc(C(C(C)C)O)nn2)(C)O)cc(F)cc(F)c1 c1(C(=O)NC(C(C)C)CNC(C2(CCF)CCOCC2)=O)cc2ncccc2[nH]1 CCC(C)CCCCC(=O)NC1CCC(CNC(=O)C2=CSCCO2)CC1 c1(CC(C)NC(=O)CCCF)ccc(CNC(=O)CCc2ccc(O)nn2)cc1 c1(OC)cc2c(cc1OC)C(NC(c1ncccc1C)C)CC2 N1(C(C(CC)C)C(=O)O)CC2COCC2(C(N2CCC3(C2)OCCO3)=O)C1 C12(NC(Cc3ncc(C)s3)=O)CCCCCC1N(C(c1cnc[nH]1)=O)CC2 c1(OCCOC)c(C(=O)N(C(C)CN(C(=O)C(C)=C(C)C)C)C)cccc1C C1(C(N2CC3C(CN=c4cc(Cl)nc[nH]4)C3C2)=O)CCc2nncn2CC1 C1(C(C)Nc2nc(C(C)(C)C)no2)CCN(C(=O)CCc2ccc(Cl)cc2)CC1 N1(C(c2ccsc2CO)=O)CCCC2C1CCN2Cc1cc([N+](=O)[O-])ccc1Cl C1(C2CCC2)(C(N(C)CC2CC(F)(F)CN2C(=O)Cc2ccco2)=O)CC1(F)F Cc1nc(C)c(C(=O)NCCC(O)CNC(c2c[nH]cc2-c2ccccc2)=O)s1 C1(C(N(C)CCN2CCOCC2)=O)CC(N=[N+]=[N-])CN1C(=O)CCc1cscn1 N1(Cc2c(OC)cccn2)CCC2CN(C(=O)C(O)CC(C)C)CC12 c1(C(N2CCCN(C(Cn3c(C)ccn3)=O)CC2C)=O)c[nH]c2c(F)cccc12 c1(CN2C(C(=O)Nc3c(C)ccnc3Br)CC(F)C2)c(Cl)cnc(Cl)c1Cl C1(CNc2n(-c3ccccc3C)nc(C)c2Cl)C2CCC3C(C2)CC13.C(C)(C)(C)C=O N1(C(C=Cc2ccc(CC)o2)=O)CC2(C1)SCCC2NC(C1CC2C=CC1C2)=O C(=O)(C(C)CC(C)CC(C)C)N1CC=CC(NC(C(CC)=CCCC)=O)C1 C1(NC(CC2CC(=C)C2)=O)CC2CCC1N2C(c1n[nH]c(C(C)(C)C)n1)=O CCCC(C)(C)C(=O)N(CCNC(c1cccc(C)c1N)=O)CC c1(C(CC)C)ccc(OCC(=O)N(CC(C)NC(=O)C=CC=C(Cl)Cl)C)cc1 CC1CN(C(=O)C2=CCC2)CCCN1C(=O)CC(C)(C)Cc1ccc(Cl)cc1 c1(C(=O)NCCC(C)N(C(CCCCCNC(C)=O)=O)C)ccc(S(C)(=O)=O)o1 N1(C(CCCCOCC)=O)CCC(NC(c2cc(C#N)oc2C)=O)C2(CCC2)C1 c1(C(N2CCOC3CCN(C(C4CSC4)=O)CC32)=O)cnc2ccc(F)cc2c1 CCCC(C(=O)NC1CN(C(c2c(C)noc2C(F)(F)F)=O)C1)C(C)C c1(C(=O)NC(C)CCNC(=O)C=CI)ccc2cc[nH]c2c1 C1(CNC(CC2CC(=C)C2)=O)(OC)CCN(C(=O)C(C)(C)C2CCOC2)CC1 C1(F)(CNC(C(C=C)OC)=O)CCCN(C(=O)C(O)Cc2cnn(C)c2)C1 c1(OC)ccc(CN2CC3CN(C(c4cccc(I)c4C)=O)CC3C2)c(F)c1F C(N=c1nc2scnc2c(NC(C2CCC2)=O)[nH]1)c1cc(C(F)(F)F)on1 C1(OC)CC(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CCC2)N(C(C)=O)C1 O=C(N=c1ncn(Cc2cc(-c3ccncc3)n[nH]2)[nH]1)NCc1cc(F)ccc1F C(CO)(CCCCNC(C1CNC(=O)N1)=O)NC(CC(C)F)=O C1(C(=O)NCC2C(CNC(=O)C=Cc3cnc[nH]3)C2)CCC(CCO)CC1 N1(CCC(CC)O)C(=O)NC(Cc2ccccc2)C1=O N1(C(CCn2c(C)ncc2)=O)CC(F)(F)CC1(C)CNC(=O)C(C)NC(N)=O C1(C(C)C)CCOC1C(N1CC(N(C(=O)C(C)CC2CCCCC2)C)C1)=O c1(C(N2CCN(C(=O)C3=CCCCO3)C(C(F)F)C2)=O)cc2ccsc2s1 c1(C(=O)NCCC2CCCN(C(CC(CC)O)=O)C2)n[nH]c2c1CCCC2 c1(OCC)ccc(CC(=O)N(C(CNC(C2CC2F)=O)C2CC2)C)nc1 c1(CNC2(C)CC(O)(CO)C2)n[nH]c2cc(F)ccc12 C(N=c1[nH]c(C)ncc1C)C1CCC(NC(C(CCC)OC)=O)CC1 N1(C(CCC2C(C)(C)C2)=O)CCC(O)(CNC(=O)Cn2ccc(O)nc2=O)CC1 c1(C(=O)Nc2c(CC)nn(CC)c2)cc2cccc(C(F)(F)F)c2nc1O c1(C(=O)NC2C(C(N(CCC)CCO)=O)CCC2)ccc(C)nn1 C1(N(C)C(c2nsnc2O)=O)CCCC(NC(=O)C(c2ccc(F)cc2)(C)F)C1 c1(C(C)(C)C)ccnc(C(=O)NC2C3CN(C(C4CCCN4C=O)=O)CC23)c1 Cc1ccc(C)c(C(=O)NC(C)CN(C(=O)COCc2ccncc2)C)c1O CC1=C(C(=O)N2CC=CC(NC(C3(N(C)C)CCC3)=O)C2)Cn2ncnc2N1C c1(OC)cccc2c1C(C(=O)NC1CCOC3(CCOCC3)C1)CC2=O C(CCCC(=O)NC1CC(F)(CNC(c2ccc(C(C)(F)F)cc2)=O)C1)N(C)C C1(C(=O)NC(CNC(Cc2ccn(C)c2)=O)C2CC2)CCC(F)(F)C1 C1(C#N)(CNC(c2scc(CNC(c3cc(C)c(C)o3)=O)c2)=O)CC(C)(C)C1 N1(C(C2CC(C)(C)C2)=O)CC(NC(C2(C)CCC(=O)N2)=O)C(n2ccnn2)C1 C12(NC(C(C)NC(C)=O)=O)CC(C)(C1)OC21CN(C(=O)CC2COCC(C)O2)C1 C1(C(=O)NCC(C)N(C)C2CC2)CCC(C2CC2)N1C(=O)Cc1ccsc1 C1(O)(CNC(c2ccnc(C3CC3)n2)=O)CCN(C(C2CC23CCC3)=O)C1 C(=O)(C(CC(N)=O)NC(=O)CCCCN(C)C)NCC(C=C)O CCC(CC(=O)N(CCCNC(c1ccc(OC)s1)=O)C)OC C1(NC(c2cccc3oncc23)=O)CCCCN(C(c2cc(O)nc(O)n2)=O)C1 C1(CNC(C2CC(=C)C2)=O)N(C(=O)C(F)OC(F)(F)F)CCCC1(C)C N1(C(c2c(OC)n[nH]c2)=O)CCCC(C)(C)C1CNC(=O)CSC C1(NC(c2ccc(OC)nn2)=O)CN(C(=O)Cc2cc(C)ns2)CC2(CCC2)C1 Cc1cncc(CC(=O)NC2CCN(C(C3(O)CCOC3)=O)C2)c1 c1(C(CCC)=O)c(CCC)oc(C)c1COC(=O)C(CC)OC CCCCC(CNC(=O)C=Cc1ccco1)NC(=O)CCCCF C1(C2CCC2)(C(=O)NCc2c(CNC(c3ccc(Cl)o3)=O)cccc2)CC1 O=C(CN1C(=O)Cc2cc(Cl)ccc21)NCCOC1CC1c1ccncc1Cl CCCC(C)C(C)N=c1nc2c(cnn2C(C)C)c(N(CCC(C)(C)C)C)[nH]1 C(=O)(C(C)(C)C(=O)NC(C)CNC(c1cccc(-c2ccc(F)cc2)n1)=O)NC C12(NC(c3cc(C)no3)=O)CCCCCC1N(C(C13CCC(C1)C3)=O)CC2 C1(N=[N+]=[N-])(C(=O)NC(c2ccco2)C)CCN(C(c2ccccc2)=O)C1 C(=O)(C1CCCc2nncn21)N1CCC(C(C)NC(C(C)c2cccs2)=O)CC1 c1(C(=O)NC2CN(C(c3c(C)nc(O)[nH]3)=O)C2)cc2cnc(C)nc2nc1O Cc1c[nH]nc1C1(C(=O)NCC2(c3ccnn3C)CC2)CCC1 c1(C(=O)NCC2(O)CCN(C(c3c(CC)csc3)=O)C2)ccc2c(c1)NCCC2 Cc1cc(C(=O)NC2CN(C(=O)CCNC(N)=O)CC2C)cc(O)c1 n1(CC)c(C)nc([N+](=O)[O-])c1NC1C2CCOC2C1(C)C C(=O)(C1=NOC2(CCC2)C1)N1C(c2cn(Cc3cncc(C)c3)nn2)C(C)CC1 C1(C(=O)NC2CC(C)(NC(c3cn(CCOC)nn3)=O)C2)CCN(C)C1C N(C(=NCCCCl)NCC1OCC1(C)C)Cc1cnc(CN(C)C)o1 N1(C(C2C(=C)C2)=O)CCCC(C(=O)NCCC2COCCO2)CC1 N1(C(CCC=C)=O)CCOC2(CCN(C(=O)C(C)(F)C(=O)OC)C2)C1 N1(C(CC=CC)=O)CC2(CCN2C(=O)CCCC2CCCCC2)C1 c1(C(=O)OC)cncn1CC(=O)NCC1CCCN1C(c1sccc1OC)=O C(=O)(NN1CCCC1C(=O)NCC12CCCC(C)(CO1)C2)C1C(C)C1C C1(NC(=O)N(CCC#N)C)(CO)COC(C)(C)OC1.c12ccc(cc1)n2CCC c1(N(CC(CNC(CC2C(C)=NOC2=O)=O)C)C)snc(Cl)c1C#N C(=O)(CCCCC(C)CC)NC(C(=O)NCC(N(OCC)C)=O)COC C1(c2n(CCOC)nc(C3CC3)n2)CC(OC)C12CCC2 N1(Cc2cn(CC3CN(C(CC(C)(C)N4CCCC4)=O)C3)nn2)CC(=O)CCC1=O c1(CC)ccc(CC(=O)NC2CC(CNC(C3(CC4CC4)CCCC3)=O)C2)cn1 C12(CNC(C3N(CC)CC3)=O)CC1CN(C(=O)Cc1c(Cl)cnn1C)C2 CC(N=c1nc2scnc2c(N2CCC2c2cccs2)[nH]1)c1nc(C2CC2)cs1 N1(C(C=CC(C)(C)NC(=O)Cc2ccon2)=O)CCC2CCC(C2)C1 C(=O)(CCC(C)OCC)N(C(CC)CNC(C1CC1CC)=O)C Cc1oc(C#N)cc1C(=O)NC1CCN(C(C2(C3CCCO3)CCC2)=O)C1C c1(CC(=O)NC(CN(C(=O)CC(C)n2cc(Br)cn2)C)(C)C)ccccc1 N(C1COc2cc(F)ccc21)c1nccc(=NC(C)c2n(CC)ncc2)[nH]1 N1(C(CCN(CC#C)C(C2CCCC(F)C2)=O)=O)CCCC(C)(C)CC1 N1(C(CCN(C(c2c(OCC)nn(C)c2)=O)C)=O)CCC(O)(CO)CC1 c1(O)c(Br)cc(Br)cc1Br.c1(OC)cccc(CN2CCCC(N)C2)c1 C1(NC(C(C)SC)=O)CN(C(c2c(O)cccc2O)=O)CCC1C C(=O)(C(F)(F)C(F)F)N1CCC(C2(NC(CC(C)C3CCCCC3)=O)CCC2)C1 n1(CCC)nccc1C(N1CCC(CCC(=O)N(C(C)CS(C)=O)C)C1)=O C(c1cnc(C)nc1O)=CC(N1C(CO)CC(NC(COC(CC)C)=O)C1)=O CN1CC(C)(C)CC1C(=O)NCC12CC(CO1)N(C(C1CCCC3(CC3)C1)=O)C2 N1(C(COCCC)=O)CC2CC2(NC(c2ccccc2C2CCCC2)=O)C1 N1(C(C(N2CC(CC(N3CC(CC(=O)OC)C3)=O)C2)=O)=O)CCCCC1=O C12(C(=O)NC(C)CNC(c3cccnc3N(C)C)=O)CCCC1OCC2 N1(C(CCc2onc(C)n2)=O)CCCC(C)(C)C1CNC(=O)CCC1CC1(F)F O=Cc1cncc(-c2cnn(Cc3ccccc3)c2)c1 C1(N(C(=O)Cc2cc(C3CC3)no2)C)CC(C(=O)Nc2ccsc2)C1(C)C c1(C(N2CCC(C)C2CNC(c2cnc(O)n2C)=O)=O)ccn(CCO)c(=O)c1 C1(NC(C(C)N(CC)CC)=O)CCN(C(=O)CSc2cccc[n+]2[O-])C(C)C1 N1(C(C(C)CCN(C)C)=O)CCC(C2(NC(=O)CC(C)SC(F)(F)F)CC2)C1 c1(C(=O)NCCN(CCOC)C(c2cc(F)n(C)n2)=O)ccc2nc(C)oc2c1 c1(C(=O)NC2CC(CNC(C3ON=C(C)C3)=O)C2)[nH]cc2c1CCC2 c1(C(=O)NC2CC(C(C)NC(C(CC)O)=O)C2)cc(O)ccc1Cl C(C)(CNC(c1cnc(S)n1C)=O)(CC(C)C)NC(CCN(C(CCC)C)C)=O C(=O)(C1=C(C#N)CCC1)N(CCCNC(c1cc(C(F)F)cs1)=O)C(C)C c1(C(N2C(CN(C(C3(C#C)CC3)=O)C)CCC2)=O)ccnc2[nH]nnc12 C#CC1(O)CC(C(=O)NC2CC23CC(NC(=O)C(C)CC=C)C3)C1 C1(C(N2C(CCOC)CN(C(=O)OC(C)(C)C)CC2)=O)CC2(C1)NC(=O)NC2=O C12(C(N(C(C)C(N3CCC(O)(C(C)C)C3)=O)CCC)=O)CCC(CC1)C2(C)C N1(C(c2c(C)[nH]nc2Cl)=O)CC2CCCC(N=c3nc(C(C)C)[nH]s3)C2C1 c1(C(C(=O)NC2C3COCC23)NC(C(C)=CC(C)(C)C)=O)cnn(C)c1 C(=O)(C1=CCN(C(c2ccc[n+]([O-])c2)=O)CC1)N1CC(C)C(N(C)C)C1 N1(C(C(C)(C)CCCO)=O)CCCC(C2CCCN(C(=O)CCC[N+](=O)[O-])C2)C1 C1(NCc2nnc(C)o2)CC(NC(c2cc(Br)c[nH]2)=O)C12CCC2 C=CCC(C)(C)CC(=O)NCC(C)C(F)C(=O)NCc1nnc(C2CC2)o1 C(=O)(CCCCCC(C)C)NC1CN(C(c2cnn(CCCC)c2C)=O)CC1C C(=O)(C1=C(C)CCOC1)N1CCN(C(CNC(COCCOC)=O)=O)CC1 C1(NC(=O)C2=CCSC2)CCCN(C(c2nnc(O)nc2O)=O)CC1 C1(NC(c2c(OC)cc(N(C)C)cc2)=O)CCN(C(c2cnc(C)[nH]2)=O)CC1(C)C C1(NC(CNS(C)(=O)=O)=O)CCC(NC(=O)CCCC2CCC2)C1 c1(CC(=O)NC2CC(F)(CNC(C=C(CC)C)=O)C2)coc2c(C)c(Cl)ccc12 C1(c2ncco2)(C(=O)NC(CNC(C2CC23CC3)=O)C2CCC2)CCC1 C(=O)(C1=CC2CCC=CCCC12)NC(C1CCCN1C(C1CCCCO1)=O)C c1(CNC(c2n(CCCC)nnn2)c2cnc[nH]2)cn2ccc(C)cc2n1 N1(C(CCC(C)(C)C)=O)CC(C2CCCN(C(C3OCC4CCCC34)=O)C2)C1 C(=O)(C1=CCCC1C)NCC1C(C(=O)NCC(CC)C(C)C)CCC1 C1(C(=O)NCC2CC(F)CN2C(=O)C=Cc2ccoc2)CC12CCOCC2 CC1(C)CN(C(=O)Cn2cc(CCNC(N)=O)nn2)Cc2ccc(Br)cc21 C(c1cnn(C)c1)=C(C(=O)N(C(CNC(CN1C(C)CC1)=O)C)C)C#N CC1=C(C(=O)NC(C2CCN(c3nc(C(C)(C)C)nc(=N)[nH]3)C2)C)CCS1(=O)=O C1(C)(NC(CCN(C(CCC)C)C)=O)CC(NC(=O)CCCc2ncc(C)o2)C1 CC1(CNC(c2ccc(NC(N)=O)s2)=O)CCC(NC(C2CC(F)(F)C2)=O)C1 S(=O)(=O)(c1ccc(C#N)cc1)N1CCC(C(=O)NCc2cc(CCC)no2)CC1 N1(C(c2c(OC)noc2C)=O)CCC(CNC(=O)C(C)(C)N2CCCC2)C(C)C1 C=C(C)CC(C(=O)NCCN(CCCC)C)NC(C)=O.c12cn(nn1)CC2 C1(CN(C(C(c2cn(C)nn2)NC(CCSCC)=O)=O)C)CCN(C)CC1 C1(NC(c2nccc(C)n2)=O)CCN(C(=O)CCC2CCCC(O)C2)C12CCC2 CC(C(=O)N1CC(C)(C)CC1CC(=O)NCC(C)(O)C1CCCC1)C(C)(C)C N1(C(C2CCCC(C)(C)C2)=O)CC2CN(C(=O)CC(C)(O)C(F)(F)F)CC(C1)O2 C1(CC)C(NC(=O)C(CSC)OC)CCCN1C(C1CCC2(CCC2)O1)=O c1(OC(CC)C)cc(C)ccc1CNC(C1CCCCC(=O)C1)=O N1(C(c2ccc(C)c(C#N)c2)=O)C(C)CC2CN(C(c3cc(F)n[nH]3)=O)CC12 N1(C(C(C=C)CC)=O)CCC(C=C)(C(N2CCC(CC)CC2)=O)C1 C1(NC(CCOCCOCC)=O)CCSC12CN(C(c1ccsc1CC)=O)C2 c1(C(N2CC3C(C(N4CCC(F)C4)=O)C3C2)=O)cc(Br)cc2cn[nH]c12 C(=CCC(N=[N+]=[N-])C(C=C(Cl)CCCC)C(C)=O)C(C)C.N(C)C N1(C(C2(C)CCN(C(C(C3CCC3)OCC)=O)C2)=O)CCCC(C)C1CO C(=O)(CC(F)(F)C(F)(F)F)N1CCC2(CC(NC(c3c(C)nn[nH]3)=O)C2)C1 c1(C(=O)NC(CC2CN(C(CSCC)=O)C2)C)cccc(F)c1SC C1(CN(C(C2CCN(C(C)=O)C2)=O)C)COCCN1C(=O)CN1CCNC(=O)C1 N1(C(CCOC(C)=O)=O)CCC(C2CCCCN2C(C2CCN(C)C2=O)=O)CC1 N1(C(Cc2c(C)cco2)=O)CC2CCC(NC(=O)C(C)NC=O)(C2)C1 c1(C(=O)NC2CC2NC(c2c(CC)occ2)=O)c(C)nn(-c2ccccc2)c1Cl C1(O)(CCNC(Cc2nc(C)sc2)=O)CCN(C(=O)Cc2ccncc2Cl)C1 Cc1nn(C)c(C(N)=O)c1C(=O)Nc1ccccc1CN1CCOCC1 Cn1ccc(C(=O)NCC(C)(C)CNC(=O)Cc2ccns2)c1C1CCC1 C(=O)(CC(O)CC(C)(C)C)N1C2CN(C(CC(CN(C)C)O)=O)C(CC2)C1 Cn1cnc2sc(C(=O)NCC(C(C)(C)C)NC(=O)Cn3ccccc3=O)cc12 C(C(=O)NC(C)CNC(c1cc(C2CCOC2)[nH]n1)=O)(C(C)C)NC(COC)=O N1(C(CC2CC(CC)OCC2)=O)CCC(C2CC2)C1CNC(=O)CCNS(C)(=O)=O c1(C(N(C2CCC(NC(=O)CN3CC=CC3)C2)C)=O)ccc(Cl)cc1N c1(C(N(CC(C)N(C(=O)C(N)=O)C)C)=O)cc(C2CC2)ccc1F C(=O)(C1CCCc2sc(C)nc21)NC(CCC)CCCNC(=O)CCN1CCC1 C1(C(=O)NCCOCCCNC(c2n(CC)ccn2)=O)CN2CCN1CC2 c1(C(=O)NC(C(C)C)CNC(C2(c3cccnc3)CC2)=O)ccnc2c1CCO2 N1(C(c2c(CCC)n[nH]c2)=O)CCCCC1C1CCN(C(=O)C=CCF)C1 C1(C(=O)NCC(C)OCC)CCN(C(c2nonc2N)=O)C1 CC(N=c1[nH]c2c(c(=NCC3(C)CCS(=O)(=O)N3C)[nH]1)SCC2)c1nncs1 N1(CCCNC(C2C(C)(CC)C2)=O)CCN(C(c2ccccc2C(F)F)=O)CC1 N1(C(C2CC(C)(CC)C2)=O)CC(F)CC1CN(C)C(c1ccnc(N(C)C)c1)=O c1(OC)ccc(C(=O)NC2CCCC2NC(c2cc(Cl)n(C)n2)=O)c(Cl)c1 c1(NCC2C(C)C2C)ccc(S(=O)(=O)N2CC3C4C=CC(O4)C3C2)cc1F c1(C(N2CCC(CNC(CC(CCC)C)=O)C2)=O)noc2c1CN(C(C)C)CC2 N1(C(c2scc(C)c2)=O)CCc2ccccc2C1CNC(c1ccccc1Cl)=O c1(NC)ccc(N(C(C2C=CCN2)=O)Cc2ccc(-c3ccccc3)s2)cc1C c1(C(C(=O)NC(CC)(C)C)N(C2CC(F)(F)C2)CCCO)ccc(Cl)c(Cl)c1Cl C1(CNC(c2c(Cl)ccc(OC)n2)=O)CCN(C(=O)CNS(N)(=O)=O)CC1(F)F c1(Nc2nc3ccc(C(=O)OCC)cc3s2)cc2cc(CC)ccc2o1 C1(CNC(CC=CC=C)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)C12CC2 C1(COCC)CCN(C(C2(NC(c3c[nH]cc3C)=O)CCCC2C)=O)CC1 C(=O)(C(F)(F)C(C)O)N(C(c1cn(-c2cccc(Br)c2)nn1)C)C CCCCCCCCCC(=O)NCC12CCC1CCN2C(=O)C=Cc1cn[nH]c1 c1(C(N2CC(CCNC(C(C3CCC(=O)N3)C)=O)C2)=O)cnn2cccc(Cl)c12 CC(CC(=O)N1CC(N(C)C(c2cnn(C3COC3)c2)=O)C(C)(C)C1)C(F)(F)F CC1COCCN(C(C2CC(NC(=O)C(C)n3cccc3)C2)=O)C1 N1(Cc2c(C)nc(F)cc2)Cc2ccc(C(N3CC4OCCOC4C3)=O)cc2C1 c1(C(C(=O)NCCCC#C)N(CCC)CC)cnc(-c2ccco2)s1 C12(CNC(c3cncc(COC)c3)=O)CCC(CC1)N(C(C1(CCO)CC1)=O)C2 C=CC1CN(C(=O)C(C)(C)C(=O)NC)CC1NC(c1csnc1OC)=O CCC(CCCO)NC(=O)CCCN(C(=O)CC=C(Cl)Cl)C c1(OC)cc(CN2CCN(S(=O)(=O)c3cccc(F)c3)CC2)cc([N+](=O)[O-])c1Cl c1(C(=O)NCC2N(C(C(C=C)O)=O)CC=C2)cccc(C)c1[N+](=O)[O-] CC1CCN(C(=O)CCOC(F)(F)F)CC1NC(c1ccnc(OC(F)F)c1)=O n1(CCCCNC(C2CS(=O)(=O)C2)=O)cc(C(c2ccccc2)C2CC2)nn1 CN1CCC2CCN(C(C3CCN(C(=O)Cc4cnnn4C)C34CC4)=O)C2C1 N(C1CCc2cccnc21)C(C1CCN(C(=O)CCc2ccc(F)nc2)C1)=O C(=O)(C(C)(O)CCN(C)C)N1CC(C(C(=O)NCC(=O)N(C)CC)OC)C1 c1(C(C)C)cnc(Cl)[nH]c1=NCCCC(C)NC(=O)CCn1cncn1 C(=O)(C(F)CCC(C)C)N(CCCNC(=O)Cc1n[nH]c(=NC)s1)CC C(=O)(CCC(=O)N1CCCC(C(C)C(=O)NCCC(=O)NCC(C)C)C1)NCC N1(C(C2(c3ccccc3)CCC2)=O)CCC(CO)(Cc2ccc(F)cc2)C1 c1(CN2CCCC(C(=O)NCc3cncc(Br)c3)C2)cc(Br)ncc1Br C1(C(=O)NCCCCCNC(C2(C)CCNC2=O)=O)Cc2n[nH]cc2C(=O)N1 C=CC(C)(C)CC(=O)N1CCCCC1C(=O)NC(C)C(O)C(F)F C1(C(C)C)N(C(C2CC2C)=O)CC12CCN(C(c1ccc3ncnn3c1)=O)CC2 N1(C(c2ncc(OC)cc2F)=O)CCOC2(C1)CN(CCC(C)(C)F)C2 N1(C(CNC(CCC)=O)=O)CC(NC(c2ccc(CC)o2)=O)C2(CCC2)C1 C1(C(=O)NCC(C)NC(=O)Cc2ccccc2F)COC2(CO)CC1C2 c1(OC)ccc2cc(C(=O)N(CC(C)CNC(=O)C(C)NC(N)=O)C)ncc2c1 Nc1ncccc1C(=O)NCC(C1CC1)NC(C1(c2cc[nH]n2)CC1)=O c1(C(N2CC(CNC(=O)OC(C)(C)C)C(F)C2)=O)cc2ccccc2nn1 C1(C(=O)NC(CNC(c2cc(OC)n[nH]2)=O)C(C)C)C(F)(F)C12CC2 c1(NC(C2CN(Cc3c(N(C)C)nc(F)cc3)C2)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(CC(C)(C)C#N)=O)CCC(C2CC2)C1C(=O)NCc1cc(C2CC2)no1 CN1CCN(C(c2cc(F)cnc2O)=O)C(C(=O)NCCC2(C)N=N2)C1 N1(C(C2CC(=O)NC2)=O)CCCC2(CCN(c3ccnc4ncnn34)C2)C1 c1(NC(C)=O)ccc(CC(=O)NN2CC(CNC(c3cnc(O)[nH]3)=O)OCC2)cc1 CCC(C(=O)NC(C)C=CC(=O)NCC(C)(O)C1CC1)N(C)C CC(C)(C(=O)NCC1(F)CN(C(=O)CCc2ccoc2)C1)C1CCCC1 C(N=c1[nH]c(=NCCCc2cn[nH]c2)[nH]c2c1SCC2)c1cc(CC)no1 C1(NC(C(C)n2ccnc2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC1F Cc1ccc(F)c(C(=O)N(C(CC(F)F)C(=O)N(CC(N2CCCC2)C)C)C)n1 Cc1nc(O)ccc1C(=O)NCC(C)CNC(c1ccnc(-n2cccc2)c1)=O Cc1c(C(N2CC(F)CC2CNC(=O)C=C2CC2)=O)nn2c1OCCC2 c1(CC(=O)NCC(O)CNC(C2CC2[N+](=O)[O-])=O)ccnc(O)c1 C1(F)(CNC(=O)CSc2nncs2)CCCN(C(C2CCCCC23CC3)=O)C1 N1(C(C2(OC(C)=O)CC2)=O)CCN(CCCNC(=O)C=C(C)C(C)(C)C)CC1 N1(C(c2cccc(C)c2)=O)CC2C=CC1C(C(=O)NC(C)(C)C(C)C)C2 C(C(F)(F)CC(O)CO)N(C(c1cc(C)ns1)C(=O)NCCCF)C c1(C(N2CCCC(NC(CC(CC)SC)=O)CC2)=O)cc(OC)c(C)c(OC)c1 CC(CC(=O)NCC1COC(CNC(=O)Cc2csc(S)n2)C1)n1cccn1 N1(C(C2CCC(CCCC)CC2)=O)CCN(C(=O)CC2(CSC)CC2)CC1C Nc1cccc(CC(=O)NC(C)(CNC(=O)CC2CCCCO2)C2CC2)c1N N1(C(c2c(NC)cc(Cl)cc2)=O)CC2(CCCC2NC(=O)CSSC)C1 N1(C(C2(CC#C)CCOCC2)=O)CCC2(C1)CN(C(=O)CCCF)C2 C1(CC)CCCC1C(=O)NC(C)(CNC(C1CN(S(C)(=O)=O)C1)=O)C1CC1 c1(C(C)OC(C2(C)CCN2C(=O)OC(C)(C)C)=O)cc(Br)c(C)c([N+](=O)[O-])c1 N1(C(CN(C(C(C)C)=O)C)=O)CCC(C(=O)NCc2ncn(C(C)(C)C)n2)C1C c1(C(N(CCNC(CCCOCCOC)=O)CCOC)=O)ncccc1C(F)F C(CC(C(=O)NCC(=O)NC(C)(C)C)NC(C12CC(F)(C1)C2)=O)=CC C12(C(N3C4C(CNC(C(N5CCCCCC5)C)=O)C(C4)C3)=O)CCCN1CCC2 Cc1cc(C)cc(C=CC(=O)NCC(C)N(C)C(c2cccn3nccc23)=O)c1 C1(CNC(=O)Cc2ccnc(O)c2)CC2CC1CN2C(C1(F)CC1)=O n1(CC)ncc(C(N2CCC(N(C(=O)CC3CC3C)CC3CC3)CC2)=O)c1Cl C(=O)(C1=COCCC1)N1CC(C(N(C(C)C(F)F)C)=O)C(F)C1 c1(OC)cc(C#N)ccc1C(=O)NCC1CC2(C1)CN(C(C1CC=CCO1)=O)C2 c1(C(=O)NC(C2CCOC2)CNC(c2cn(CC=C)nn2)=O)cc(O)nc(O)c1 CCCCCCCCCC(=O)NCC1CC(NC(=O)CC2CCCOC2)C1 N1(C(CCCc2c(C)ccs2)=O)C2CCC1C(C)C(NC(=O)Cc1ccon1)C2 c1(OC)cccc(C(O)C(N2CC3CC3(NC(=O)CCn3cncn3)C2)=O)c1 C=C(Cl)C(C)(C)C(=O)NC1CCC(CNC(=O)COc2cc(C)ccc2F)C1 Cc1ccc(Cl)c(O)c1C(=O)NC1CCN(C(=O)C2=CCCCC2C)CC1C c1(C(N2CCC(NC(c3c(Br)ccc(C)c3)=O)C(F)C2)=O)ccc(O)c(C#N)c1 C1(NC(C2(CN(CCCC)CC)CC2(F)F)=O)(COC)CCCOC1 c1(N(C2CCCC2O)C)nc2ccsc2c(=NCCOC(C)(C)C)[nH]1 C1(C(N2CC(CCNC(c3cccc4scnc34)=O)C2)=O)CCCCC1C1CC1 C#CC1(C(=O)NC(C)CNC(=O)CCC(C)CN(C)C)CCOCC1 C(=O)(C1=CCCOC1)NC1(C2N(C(c3cccc(CC)c3)=O)CCC2)CC1 C#CCC(CC#C)C(=O)N1CC(N(C(=O)CSc2ccc(C)cc2)C)C(C)(C)C1 c1(CC)cc(C(=O)NC(CNC(=O)CSc2cn[nH]c2)CO)ccc1F CC#CCC(C(=O)NC1CC(C(=O)OC)C1)NC(=O)C(C)C(C)C CC(C)C(CNC(c1cc(C#N)n(C)n1)=O)C(=O)NC1CN(C)NC1=O C(=O)(CC(C1CC1)NC(=O)C(CC1CC1)NC(c1cc(O)cs1)=O)OC N1(C(CCCCC=C)=O)CCC2(CC(NC(c3cnc4n3CCCC4)=O)CO2)C1 c1(CC(=O)NCC(CC)NC(=O)CCCOC)cc(C)on1 N1(C(C)C)CC(NC(C2(CCNC(C3CCC3CF)=O)CCC2)=O)C(C)C1 Cc1cc(CNc2csc(-c3c(Cl)ccnc3Br)n2)ccc1F C1(C)(C(=O)NC2CCC(NC(C3(COC)COC3)=O)CC2)CCN(C)C1=O C#CC1CCCN(C(=O)C(C)(C)CNC(c2cnn(C3CC3)c2)=O)C1 N1(C(CC(C)n2cccn2)=O)CCC(CCN2CCN(C(=O)CO)CC2)CC1 N1(C(c2cn(C)nc2)=O)CC2CCC(CNC(c3cnn(CC(F)F)c3)=O)C2C1 c1(C(C)N(CC(=O)O)C(c2cn(CCCF)nn2)=O)ccc(Br)cc1 C1(C(=O)NC(c2nocc2C(=O)NCCCC2CCCCC2)C)COCOC1 c1(C(c2nnnn2CCCSC)NC2(COC)CCC2)ncc(Cl)cc1Cl C(CCCCCOC(C)=O)NC(=O)C(C)CC=Cc1ccccc1 C1(NC(CCC=C(C)C)=O)CCCN(C(C2CC2c2ccc(F)nc2)=O)C1 c1(-n2cc(Cc3cccc(CNC(CC(CC)C)=O)c3)nn2)ccc2c(c1)CCC2 c1(OC)cc(C)[nH]c(=NCC(=O)NCC2CC3(CCN(C(C4CC4C)=O)C3)CO2)n1 N1(C(CSCC#C)=O)CCN(C(CNC(=O)Nc2ccc(F)cc2)C(F)F)CC1 CC1COc2c(C(N3CC4CCC(C3)N4C(=O)C(C)CF)=O)cccc21 C1(C(=O)NCCOCC#C)C2CN(C(=O)C(C)n3cccc3)CC12 c1(C(=O)NCC(C)NC(c2nc(CCC)oc2)=O)cnc(N)c(N)c1 N1(C(c2cc(CC(C)C)on2)=O)CCCC(CNC(c2cccnn2)=O)C1 CC1CCN(C(=O)CCc2cnn(C)c2)CC1CNC(c1ccc(Cl)c(F)c1)=O CN1CCCC(C(=O)NC2(C(F)C(=O)NOCC3CCOC3)CCCC2)C1 C1(NC(Cc2cc(C)no2)=O)C=CCN(C(c2ccnn2C2CC2)=O)C1 CC(C(=O)NCC1(O)CCN(C(c2ncoc2C(F)(F)F)=O)C1)C(C)(F)F C(C(=O)NCC(C)(C)CC1CN(C(=O)Cn2nnc(C)n2)C1)(C(C)(C)C)OC C1(C(N2CC(CNC(CCc3scc(C)n3)=O)OCC2)=O)CN2CCN1C(C)C2 c1(C(=O)NC2CN(C(COC)=O)CC2c2ccccc2)ccc(F)c(O)c1F c1(C(=O)NCCCN2CCN(Cc3ccc(C)s3)CC2)ccn2cncc2c1 c1(OC)ccc(C(=O)NCC2(C)CCC(NC(=O)CSC(F)(F)F)C2)c(C)c1OC C(=O)(CCCCCCNC(C1CCC1OCC)=O)NC(C(CCC)O)CO.CC N1(C(C(C)(C)F)=O)CCC2(C1)CN(C(c1cnc(O)[nH]1)=O)CCO2 C(=O)(C(C)(C)C(C)(F)F)NCC(CNc1cc(OC(C)C)ncn1)O C1(C(N2CCC(F)(CNC(CC)=O)CC2)=O)CCC2CCC(=O)N12 C1(C(C)C)CN(C(=O)Cc2cscn2)CCN1C(=O)C(O)Cc1cccc(Cl)c1 c1(C(=O)OCC)ccc(-c2cnccc2-c2nccn2C2CCS(=O)(=O)C2)cc1 Nc1ccnc2c(C(=O)NC3CCN(C(C45CC(CN4C4CC4)C5)=O)CC3)cnn12 N1(C(CCCC#C)=O)CCCC1C1CCCCN1C(c1cc(CC)c[nH]1)=O N1(C(CC(CC)SC)=O)CCC(NC(c2cnc(C(F)F)cn2)=O)C(O)C1 C1(NC(CCn2c(C)nc(C)n2)=O)CN(C(C2SCCCS2)=O)CC(F)(F)C1 N1(C(C=CC=CCC)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)C(C)CC1C C1(CC)CC(C(=O)NCC(O)C(C)(C)C)CCN1C(=O)CC1CCCN1C CC(C)(C)C(CNC(=O)C=Cc1ccc(Br)o1)c1nc[nH]n1 C1(NC(C=CC)=O)CCC(NC(C2CCCN(C(=O)OC(C)(C)C)C2)=O)CC1 c1(C(C)C)nccc(=NCC2CN(C(=O)CC3CC(C)OC3C)CC23CCC3)[nH]1 c1(C(=O)NCC(CNC(CSc2ccn(C)n2)=O)O)ccc(NC(=O)C2CC2)nc1 N1(C(C2(CCCC)CCC2)=O)CCOC(CCCNC(=O)C(C)CN(C)C)C1 c1(C(N2C3CN(C(C4CCN(C)C4)=O)C(CC3)C2)=O)ccc2cc(N)ccc2n1 c1(C(=O)NCC2CN(C(C(CN(C)C)O)=O)CC2O)cnn2c1S(=O)(=O)NCC2 Cc1ccc(CC(=O)NCCC2CN(C(=O)CCC3CCC3)C2)cc1O C(=O)(C1=CCCC1C)N(C1(C(=O)OC)CC1)C.C(=O)C=CCNC Cc1nccc(C(=O)N(C2CCCC(NC(=O)CN3C(=O)CNC3=O)C2)C)n1 N1(C(CC(C)F)=O)CCCC(COc2cn(-c3cccc(CCO)n3)nn2)C1 CC(C)C(CN(C)C)C(=O)NCC(C1CCCCC1)NC(=O)C1=CCCOC1 C1(C(N2C(CNC(=O)CC3OCCCO3)CC(COC)C2)=O)COCCN1C=O c1(NC(C2CC(C)CN2C(=O)C2=CC=NC(=O)C2)=O)cc(Cl)nc2ccccc12 c1(C(=O)NC2C(C(=O)NC(C(CC)C)C)OCC2)ccnnc1O N1(C(C(C)OCCCC)=O)CCC(CCOC)(NC(=O)Nc2nnc(C)s2)C1 c1(C(=O)NC2(CC=C)CN(C(C3CC(C(C)C)=NO3)=O)C2)c(C)nc(O)nc1S c1(OC)ccc(C(C(=O)NCCCF)N2CCC2C2CCC2)cc1C N1(C(c2ccc(CC#N)cc2)=O)CCC(C)(CC(=O)NC2CCC(C)O2)C1 c1(COC)cccc(CC(=O)NC(CO)C(C)NC(c2cnc(OC)s2)=O)c1 C(=O)(CS(=O)(=O)CC)NCC(CC)(C)NC(C1CCC(C(F)(F)F)CC1)=O CCCC(C(=O)NCC1CCOC1=O)NC(c1ccccc1O)=O N1(C(CC(C)C)=O)CCC(NC(c2sccc2OC(F)F)=O)CC1C1CC1 c1(C(N(CC(CC)NC(=O)CCc2cnoc2)C)=O)ccc(NC(N)=O)cc1 C#CCC(C(=O)NC(c1cn(C)nn1)C)NC(=O)COCc1ccoc1 N1(C(Cc2c(CC)con2)=O)CCC2CC12C(=O)NCCC1(C)CCOCC1 C(=O)(CC(C)P(C)(C)=O)N1CC(NC(Cc2cc(C)sc2C)=O)C(C)C1 C=CC1(CC(=O)NCC2CCCC(C)O2)CN(C(c2ccc(C)s2)=O)C1 C1(CCOC)(NC(c2cncc(Cl)c2C)=O)CCN(C(C2(O)CCC2)=O)CC1 c1(C(N2CCCC(C(C)NC(c3c(C)sc(O)n3)=O)C2)=O)c(F)ccnc1Cl Cc1cc(NC(=O)NC2(c3ccncc3)CNC2)c(F)c(Br)c1 CCC(CC)(C(=O)N(C1CCN(C(=O)C(C)=C(C)C)C1)CCO)c1cccc(Cl)c1 c1(OC)ccnc(OC)c1C(=O)NCC1CCCN1C(C1CC=CC1)=O C1(NC(C2N(CC)CC2)=O)CN(C(=O)Cn2ccc(C3CC3)n2)CC1O c1(C(N2CC(C(C)C)C(NC(C3(C)CCOC3)=O)CC2)=O)ccnc2ccnn12 CC(C)(CNC(=O)C(=O)NC1(C(c2csc(C(C)(F)F)n2)=O)CC1)CCN CCC(C)(C(=O)N1CCc2sccc2C1CNC(C1(O)CC1)=O)C(F)F CCC(C)C(CC(=O)NCC1CCC2(CC2)C1)NC(C1(CO)CCOCC1)=O C1(NC(C2(CC)CCCC2O)=O)C2CCN(C(=O)C=CC(F)(F)F)CC12 N1(C(COCCC=C)=O)CCN(C(=O)C2=CCOC2)C(C2CCC2)C1 N1(C(c2c(CC)n(C)nc2)=O)CC2CCC2(CCNC(C2(C#N)CC=CC2)=O)C1 c1(CC(=O)NC2(C(=O)NCC3(O)CCCCC3)COC2)ccccc1[N+](=O)[O-] N1(C(CCN(C)CC)=O)CCC(=O)NC2CN(C(c3nc(=N)cc[nH]3)=O)CCC12 Cc1nc(O)nc(C)c1C(=O)NCC1CN(C(=O)C(C)(Cl)Cl)CCC1C Cn1cc(C(=O)NCC2(CNC(=O)C(O)CN3CCCC3)CCC2)c(C2CC2)n1 c1(-c2c(C)nn(C)c2)cccc2[nH]nc(C(=O)Nc3ncc(I)cc3Br)c12 c1(NC(CCSCC)C)ccc(S(=O)(=O)N2CC3OCOC3C2)c(Cl)c1 C=CC1CN(C(C2CC(CF)C2)=O)CC1NC(c1cc(Cl)cnc1C)=O C1(NC(C(=O)NCC(C(=O)OCC)C(C)C)=O)CCCc2ccccc2C1 N1(C(C(C=C)O)=O)CCC(C(=O)NCC(C)(C)COC)(CC)C1 C12(CNC(C=CCN(CC)CC)=O)CCC1CN(C(C1(C)CC1(Cl)Cl)=O)C2 C1(NC(c2cc(CC)oc2C)=O)CCC2CN(C(=O)C(CC)(CC)OC)CC2C1 c1(C(N2CC(NC(C#C)=O)CC(F)(F)C2)=O)ccnc2ccc(O)cc12 c1(OC)ccc(C(=O)NCCCC2CN(C(C3CC=CC3)=O)CCO2)c(Cl)c1 C(C)(C)(CN=c1cc(C(F)(F)F)nc[nH]1)NC(C1=NOC(C)C1)=O c1(SCC(=O)NCCCN(C(CC2C(C)CCCC2)=O)CCO)ccc(Cl)cc1Cl C1(NC(C2CC2(C)C)=O)CCN(CCSCc2cn(Cc3ccccc3)nn2)C1 c1(C(=O)NCc2c(C(=O)NC(CCCC)CC)occ2)ccc(C)nc1O c1(CCC(N2CC(CN3CCN(C(C(C)O)=O)CC3)C2)=O)nc2ncccn2n1 c1(C(=O)NC(CC)CNC(C2CC23CC(C)(C)C3)=O)cc(Cl)cc(F)c1F N1(C(CCN(C)CC)=O)CCC2(CCC2NC(c2cc(C3CC3)[nH]n2)=O)CC1 N1(C(=O)CC2CCCNC2=O)CC2=C(C1)CN(C(C1COCCC1(F)F)=O)C2 N1(C(C(=O)NCCC(=O)OCC)c2cn[nH]c2)CC(CF)C2(CCCCC2)C1 c1(CCCSCC)nc(-c2ccnc(C(F)(F)F)n2)n(-c2ccnc(Cl)c2)n1 CN1CCOC(CN(C(C(=O)NC2COC2)c2nccs2)CC2CC2)C1 C1(CN(CC(F)(F)F)C(Cc2c(C)nsc2)=O)CCCN(C(=O)OC(C)(C)C)C1 C1(CN(C)C(C2CCCN2C=O)=O)CC(F)CN1C(c1c[nH]c(=N)s1)=O c1(C(N2CCCC(N(C(c3cc(C)sc3C)=O)CCF)C2)=O)ncn2c1CCC2 C1(NCc2cn(C)nn2)CC(NC(C2(C)CCCCCC2)=O)C12CCC2 Cc1nn(C)cc1C(C)C(N1CCCC1CNC(=O)CC1COC(C)(C)C1)=O N1(C(C(CCC)OC)=O)CC(CNC(c2c[nH]cc(Cl)c2=O)=O)CC1(C)C c1(C(=O)NCCc2c(CNC(CCC(=C)C)=O)nco2)cn(C)c2ncccc12 N1(C(C2(N(C)C)CCC2)=O)CC2CCC2(CC(=O)NCC(O)CO)C1 c1(CCC)c(C(=O)NCC2CN(C(c3c(SC)cnn3C)=O)CC2O)cnn1C C12(C(N3CC(C)C(F)C3)=O)CCC(NC(c3cncnc3)=O)(CC1)CC2 c1(OC)ccc(C(C(=O)O)NC(C2CC2c2cccnc2)=O)cc1 C1(NC(C2CC(C)(CC)C2)=O)CC2(CCN(C(C34CCCC3CCC4)=O)C2)C1 N1(C(c2ccc(COC)o2)=O)CC2CC(C1)N(C(=O)CNC(=O)C(C)CC)C2 N1(C(c2n(CC)ncc2Cl)=O)CCC(O)(CNC(c2cc(C)nn2C)=O)CC1 CC(CN(C)C(c1cnn(-c2ccncc2)c1)=O)N=c1[nH]nc(O)s1 c1(SCC)ccccc1C(=O)NCC1CC(NC(C23CC(OC)C2C3)=O)C1 C1(CNC(c2ccc(F)c(F)c2)=O)CCCCCN1C(=O)C(CO)c1ccccc1 CC(CS(C)(=O)=O)C(=O)NC12CC(NC(=O)Cn3ncc4ncccc34)(C1)C2 c1(COC)cccc(C(=O)NCc2ccc(C)cc2)c1.C12CC1C(=O)O2 c1(C(=O)NC2CCC(NC(c3ncc[nH]c3=O)=O)C2)cccc(F)c1C(F)F O=C(CC1=CCCC1)NC1CN(C(=O)CCCc2ccc(F)c(F)c2)CC1O N#CC1(C(N2CC3(CCN3C(c3ccc(CN4CCCC4)o3)=O)C2)=O)CCCOC1 NS(=O)(=O)c1ccc(C(=O)NCC2CC(NC(c3cscc3F)=O)C2)cc1 C(=O)(C(C)C(C)S(C)(=O)=O)NCCC1CCN(C(c2c(C)cnn2C)=O)CC1 c1(C(N2CC(CNC(c3n(CC)cnn3)=O)C(F)(F)C2)=O)cnn2c1OCCC2 Cn1nc(C(N2CC=CC2CNC(C2CCC(C(F)F)CC2)=O)=O)cc1Br CN1CCOC(C(=O)NC2(C(=O)N(C3CC(F)(F)C3)C)CCOCC2)C1 C1(C(N2CC3CC(C2)N(C(=O)CCC(F)F)C3)=O)Cc2cccnc2C1 N1(C(CCCNC(C)=O)=O)CC2CCC1CC2NC(c1nccc2cc[nH]c12)=O CC(C(C)(C)C(=O)N1C(CO)CC1C)NC(c1cncn1C)=O C12(CC(=O)NC3CC(C)(NC(C(C)Cc4ccccc4)=O)C3)COC(CF)(C1)C2 C1(CN)CCN(C(=O)Nc2cccc(C(=O)NC(N)=O)c2)CC1(F)F C#Cc1ccc(C(N2CC(NC(c3cn(C)nc3OC)=O)CC(O)C2)=O)c(F)c1 N1(C(c2c(C)nc(CC(C)C)s2)=O)CC2=C(C1)CN(C(c1nn(C)cc1N)=O)C2 C=C(C)C(CC(=O)N(CC(C)O)CCNC(c1cc2occc2s1)=O)OCC C1(C(N2CCN(C(CCC)=O)CC2)=O)CC12CCN(Cc1nc(Cl)ccc1F)C2 C(=O)(CC(C(F)(F)F)NC(c1cc(C)sc1N)=O)N1C(CSC)CCC1 C1(NC(COC(C)C)=O)CC(F)CN(C(c2ccc(Cn3cc(Cl)cn3)s2)=O)C1 c1(C(=O)NC(C2(O)CCN(C(=O)C3=CCCC3)CC2)C)ccc(Cl)c([N+](=O)[O-])c1 C1(CNC(c2ccoc2)=O)C2CN(C(c3cc(C(F)F)[nH]n3)=O)CC12 C1(OCc2c(OCCCOC)cccc2)CCCN(c2ccccn2)CC1 CC1CCC(NC(C2CC2C#N)=O)CN1C(=O)Cn1nc(C(F)F)cc1C(F)F C1(CNC(C(C)OC(Cn2ncc(C(C)C)c2)=O)=O)COc2ccccc2O1 C1(NC(c2c(CC)nn(C)c2)=O)CCCN(C(=O)CC(C)C(=O)OC)C1C N1(C(C(C)CSC(F)(F)F)=O)CCN(C(c2cn(C)nn2)=O)C(c2cn[nH]c2)C1 O=C(C1=CCCCO1)Nc1ccc(C2CCN(Cc3ccc(Br)c(Br)c3)C2)cc1 Cc1ncn2ccc(C(N3CC4C(CNC(c5ccc(CO)o5)=O)C4C3)=O)cc12 C1(C(=O)NC2CC3(CC(NC(CCC)=O)C3)C2)CCc2nn(C)cc2C1 C1(C(N(CCCF)C)=O)CCCC(NC(c2c[nH]c(C#N)c2)=O)C1 N1(C(=O)C(F)C2CCOC2)CCC2(C1)CN(C(c1ccnc(Cl)c1F)=O)C2 c1(N2Cc3c(=N)[nH][nH]c3C2)nc(=NCc2ncc[nH]c2=O)[nH]c2c1SCC2 C(=O)(CC(C)(C)CC(F)(F)F)N(CCCNC(c1ncc(F)cn1)=O)C N1(C(c2cnn(CCCC)c2C)=O)CCC(CNC(c2cc(Cl)on2)=O)C12CC2 N1(C(CC2N(C(c3ccc(SCC)nc3)=O)CCCC2)=O)CC(OC)CCC1C c1(CC(=O)NC2CCN(C(C3C(C)(C)OCC3)=O)C2(C)C)cn2c(n1)CCCC2 N(C(=NCC(=O)N(C(C)C)CC)NCc1cccc(Cl)n1)C(C=C)C C1(OC)CC(NC(=O)C(C)(C)C)CN(C(=O)Cc2cnc(COC(C)=O)[nH]2)C1 N1(C(CC(C)F)=O)CC2(C1)SCCC2NC(=O)Cn1cnc([N+](=O)[O-])n1 N1(C(C=Cc2ncc(C)[nH]2)=O)CCC2(CC(NC(=O)C#CC(=O)N(C)C)C2)C1 N1(C(CCS(N)(=O)=O)=O)CCCCCC(NC(c2cc3cc(Cl)sc3[nH]2)=O)C1 N1(C(CCN(C(C)=O)C)=O)CCCCC1CNC(C1(C(F)(F)F)CCCCO1)=O CC(C)CC(CC(=O)O)NC(C1CCCN(Cc2cncc(N(C)C)c2)CC1)=O c1(OC)ccc(C=CC(=O)NCC(CNC(=O)C=CC2CC2)CO)cc1 C=C1CC2(C1)CC(C(=O)NCC1CCCN1C(=O)CCC(=O)c1ccccn1)C2 c1(OCC)c[nH]c(=NC(=O)c2nc3cccc(CC)c3o2)cn1 N1(C(C=C(C)Cl)=O)CCCCC(CNC(=O)C(C)Sc2ccccc2Cl)C1 c1(CNC(NOCC(=O)NCC(=O)OC)=O)cn(CCn2cncn2)nn1 C(C1CCc2nccn21)NC(C1CC(C)CN(C(c2cc(=O)cc[nH]2)=O)C1)=O Cc1cc(C(N2CCC2CC(=O)NCC2CN(C(C)C)C2)=O)cnc1C O(P(=O)(CCCNC(Cn1cccn1)CC)OCC)CC C1(CC)C(NC(=O)Cn2cncn2)CCN1C(c1cc(C(C)C)nn1C)=O c1(CC(=O)N(C)CCNC(c2cnccn2)=O)c(F)cccc1Cl O=C1CC2CC(C(N3CCN(C(=O)CCc4ncco4)CC3)=O)C1C2 C(c1cc(F)cc(F)c1)=CC(=O)N(C1C2CN(C(C3(CCF)CCC3)=O)CC12)C N(C(=NCC1CCOC1)N1CCC(C2CCC2)C1)Cc1cc(C(F)(F)F)no1 Cc1cccc(F)c1C(=O)NC1CCC(CC(=O)NCC2CCCNC2=O)C1 c1(N2CCC(C(C)NC(CCc3c(C)cccc3)=O)CC2)ccccc1[N+](=O)[O-] C12(CN3CCOCC(CC)C3)CCC(C1)C(=O)NC2 c1(CC2c3cn(nn3)CC3(CC3)CO2)[nH]c(O)nc1C.C1(NC(C)=O)CCCC1 c1(CC(=O)N(C(C)CN(C(=O)CC2CCOC2)C)C)cncc2ccccc12 N1(C(C2C(=C)CC2)=O)CCCC(C)(CNC(=O)C=CCN(C)CC)C1 c1(C(N2CC(CNC(c3[nH]cc(CC)c3)=O)C2)=O)ccc2ccc(Br)c(F)c2n1 C#Cc1cc(C(=O)OC2CCN(CCO)CC2)ccc1Cl c1(C(=O)NC(CNC(CC(C=C)C)=O)C2CC2)ccc(OC)c(OC)c1C N1(C(C(Cn2cncn2)NC(CCN(CCC)C)=O)=O)CC(C)(C)OCC1C CC1(CNC(c2cnc(C3CCC3)s2)=O)CCOC1C1CC1 CC1CCN(C(=O)C(N)=O)C1CNC(C1(c2ccccc2F)CCC1)=O N1(C(COC2(C)CN(C(C34CC(F)(C3)C4)=O)C2)=O)CCC(C)(C#N)C1 N1(C(c2ccc(CNC(c3n(C=C)nnc3)=O)s2)=O)CC(O)C(C)(C)C1 c1(C(=O)NCC(C2CC2)NC(C2CCN(C(=O)OC)CC2)=O)ccc(F)c(F)c1 C1(C(=O)NC2COCC2N=[N+]=[N-])CC2(C1)CC(NC(c1cccn1C1CC1)=O)C2 CCC(C)C(=O)C(=O)NCC(C)NC(c1nnnc(O)c1C)=O c1(C(=O)NC(CCNC(CCCOCCOC)=O)C)cc2c(C)ccc(C)c2[nH]1 C=CCC(C)(C)C(=O)N1CCCCC(CN(C(=O)C(COC)OC)C)C1 C1(CCNC(C=Cc2c(C)ccnc2)=O)CC(F)(F)CN1C(=O)C(C)C(C)(C)C N1(Cc2c(F)ccc(OC)n2)CC2CCCCC2C1.c12cc(ncn1)N2 C1(NC(c2cc(F)c(C(=O)O)cc2F)=O)CCC2(C1)CN(C(=O)NCCCCl)C2 C1(CNC(C(C)(C)C2CCN2C(=O)Cc2cc[nH]n2)=O)CCCCC(=O)N1 CCCC(CCC)C(=O)NC1CCC(NC(c2cc(C3CCC3)no2)=O)C1 c1(C(=O)NCCN(CCC)C(C2CCCC23CC3)=O)cc2c(C)cc(F)cc2[nH]1 C(c1c(F)cccc1F)=CC(=O)NC1CCCC(NC(CCC(C)(F)F)=O)C1 CCCCC(C)CCC(=O)N1CCC(C)(CC(=O)NCCN2CCCCC2)C1 S(=O)(=O)(c1ccc(NCC23CCCC2C3(F)F)c(C#N)c1)N(C)CC1C=CCC1 C(=O)(C(C)C=C=C)N(C1CCN(C(C2CCC=CCC2)=O)C1)CC#C CCC(C(=O)N1CC(N(C)C(c2cn(C)nc2OC)=O)C2(CC2)C1)C(C)C C1(CC=O)(CC2(CN(C(C)C)C)CCOC2)CCOCC1.c1(S)cncc(F)c1 N(C(=S)c1ccccc1)(C(C(=O)O)Cc1ccc2[nH]c(=O)[nH]c2c1)CC(F)F C=Cn1nccc1C(=O)N(C(C)CNC(c1sc(-c2ncc[nH]2)nc1C)=O)C c1(C(N(CC(CNC(c2nc(C(C)C)oc2)=O)O)C)=O)cccc(C2COC2)c1 N1(C(=O)CSn2nccn2)CCCCC1C1CCCN1Cc1ccc(F)cc1Cl C=CCC(CC=C)C(=O)NC1CC2CC(NC(=O)C(COC)COC)CC12 c1(CS(N2CCCCC2C(F)(F)F)(=O)=O)cccc(-c2cn[nH]c2)c1 c1(C(=O)NCC(=O)NC(CC(C)NC(C2(CC)CCC2)=O)C)cncc(Br)c1 N1(C(C(CN(C)C)O)=O)CCC2(CCCN(C(C3CC34CCC(=O)CC4)=O)C2)C1 CC(C)C(CCC(=O)N1CCN(C2(C)CC2)CC1)NC(=O)CN1CCCCC1 C1(CCNC(=O)OC(c2ccccc2)COC)CCC(OC)CC1 C1(NC(CCOCC#C)=O)CCCN(C(c2cnn[nH]2)=O)C1C C(=O)(CC1c2ccccc2C(=O)N1C)N(C1CN(C(c2c(C)nncc2)=O)C1)C N1(C(C(C)=CC)=O)CC(CNC(=O)CCN(CC)CC)CC1(C)C C1(C(=O)NC(C)C(CO)NC(=O)COC2CCCC2)CCS(=O)(=O)N1C N1(C(C(C)C)=O)CCC2(COCC(CNC(=O)CNc3cccnc3)O2)C1 CCCC(C)CC(=O)N1CC=CC(NC(c2ccn(CC3CC3)c2C)=O)C1 C1(O)(CNC(=O)Cc2ccoc2)CCN(C(=O)C(c2ccc(Br)cc2)O)CC1 n1(CC(=O)NC(C2CCN(C(=O)CC3CC=CC3)C2)(C)C)nc2c(n1)CCCC2 N1(C(COC(C)(C)C(F)(F)F)=O)CCCC(C)(c2cn(-c3cnc(Cl)nc3)nn2)C1 c1(C(=O)NC23C(CN(C(c4c(C)[nH]c(=N)s4)=O)C2)C3)csc2c1CCCC2 C1(SCC)COCCC1c1noc(-c2cscc2C(F)(F)F)n1 C1(C(=O)NCCN(C)C(c2ccccc2OC(F)F)=O)CCC(C#N)C1 c1(C(=O)NCCCN(C)C(c2ccc(F)c(F)c2F)=O)ccc(F)c2c1OCC2 C1(NC(CNC(CC)=O)=O)CCCC12CCN(C(=O)COCC(F)F)C2 C(=O)(C1=CCC2CCC1N2C(=O)CCCC1CC1C)NC1(C(N(OC)C)=O)CC1 C1(CC)(NC(=O)CC2CC(F)C2)CCN(C(C2CCCCC2(C)C)=O)CC1 Cc1c(NC(=O)NC(c2ncc[nH]2)C)cc([N+](=O)[O-])cc1C(F)(F)F Cc1c(C(N2CCC(F)C(NC(C3CC3C)=O)C2)=O)ccc2c1OCCO2 C(c1cocn1)=CC(=O)NC1CCC(NC(=O)COCc2nc[nH]n2)C1 C(=O)(C(C(C)NC(C1CC2CC(=O)C1O2)=O)C(C)C)NCCC=CCCC c1(OC)cc(OC)cc(C(=O)NNC(=O)NC2(C)CC3CC3C2)c1 c1(C(N2C(CCNC(C(C(COC)C)C)=O)CCC2)=O)ccc2nnn(C)c2c1 c1(C(=O)NC(CNC(C(C2CC2)SC)=O)C)ccnc(C)c1C CS(=O)(=O)c1ccc(C(=O)NC2CN(C(C3CC3C#N)=O)C3(CCC3)C2)s1 C1(c2ccc(F)cc2)(C(=O)OC)CCN(C(C2CCCN2)=O)C1 C1(C(N2CCC2C(=O)NCCC23CC(CO2)C3)=O)(CC)CCCCO1 CC1(CCCC(=O)NC2CC2CNC(c2ncc(C(F)F)s2)=O)NC(=O)NC1=O N1(C(C2C(OC)CCC2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)CC1CO N12CC3(C1)CN(C3)C(=O)Cn1nccc1C=CC(=O)C(=O)C(C)C2=O.CO c1(C(N(CCCNC(C2CCCO2)=O)CC)=O)cccc(C(F)F)c1F c1(C(=O)NC2CC3C(NC(C(C=CC)O)=O)C3C2)n[nH]c(C)c1[N+](=O)[O-] C1(C2CC2)(NC(CNC(C)=O)=O)CCN(C(=O)CN2CCS(=O)(=O)CC2)C1 c1(CC(=O)N(C2CCN(C(C3COCC(C)(C)O3)=O)C2)CC)cc(C)ccc1F c1(C(C)(C(F)(F)F)NC(C(C2CCNCC2)C)=O)ccc(C#N)cc1 C1(C(=O)NCc2cc(C(N(CC(COC)(C)C)C)=O)n(C)n2)CCCC2(CC2)C1 C(CCC(O)CO)NC(C(C)(C)C1CCCN1C(=O)Cc1ccsc1)=O n1(CCCC)cc(C2(C(=O)OC)CN(C(=O)C(n3cc(Br)cn3)C)C2)nn1 c1(C(N2C(CN(C(=O)C(C)C3CCCO3)CC)CCC2)=O)cc(O)cc(O)n1 C1(NC(c2cnc(OC)s2)=O)CCN(C(C2CC2c2ccn(C)n2)=O)CC1(C)C C12(C(=O)NCC(C)(C)NC(C3CCC4(CC3)CC4)=O)CC3CC(C1)CC(O)(C3)C2 CC1CCC(=CC(=O)NCC2CC2NC(c2n[nH]cc2-c2ccncc2)=O)CC1 C(=O)(CC(C)P(C)(C)=O)N1C(CNC(=O)C(C)(C)C)CC(OC)C1 N1(C(C2(CC(C)C)CC2)=O)CC(NC(C2CC(=C3CC3)C2)=O)C(O)C1 C(C(=O)N1CC(NC(=O)CC2OCCCO2)C1)(C(C)C)NC(C(C)OC)=O N1(C(c2c(C)[nH]cc2)=O)CC2(CCC2)CC1CNC(c1cc2ccccn2c1)=O N1(C(C2(NC(C)=O)CCC2)=O)CCCN(C(C2CCC(=O)NC2)=O)C(C)C1 c1(CNC(COC2CN(C(CC(CC)OC)=O)C2)=O)cnc(F)c(C)c1 c1(NC(C(=O)N(C2CCN(Cc3cn(C4CC4)cn3)CC2)C)=O)ccc(F)cc1 C1(CC)C(C(=O)NCCCOC(F)(F)F)CCCN1C(c1ncc(N)cc1C)=O c1(C(=O)NC2C(CNC(=O)CCc3cc(Cl)no3)CCC2)cc2sccc2[nH]1 C(=O)(C1=CC(C)(C)C1)NCC1(OC)CN(C(=O)CC2CCCOCC2)C1 c1(CC(N2C(CCCNC(C3C(C)OCC3)=O)CCC2)=O)ccc(O)cc1 CCC(C)C(O)CNC(=O)CCN(C(=O)CCc1cncs1)CCO N1(CC(=O)NNC(=O)c2ccccc2Br)CC(O)CC2(CC2)C1 C1(C)(N(C)CC)CCN(C(=O)CCN2C(=O)C3CCC3S2)C1.CCS.C(C#N)C CC1(C)CN(C(=O)CC2=CCOCC2)CCC1NC(=O)C1=CC2CCC1C2 CN1CCCC(NC(=O)C(Cc2ccco2)NC(c2ccc(C#N)n2C)=O)C1=O Nc1c(C(=O)NC2CCCCC2NC(C2C3COCC23)=O)ccc(F)c1F c1(NC(=O)NCc2cc(C)c(I)cc2)ccc2c(c1)CC(N)C2 C1(O)(C(=O)NCCSCC(=O)NCC2(C(C)(C)O)CC2)CCCC1 c1(CCC)nc(C)c(C(=O)NCC2(C)CCN(C(c3cnoc3C3CC3)=O)C2)o1 C#CCCCC(=O)NC12CC1CN(C(=O)C(C)(F)c1ccccc1)C2 c1(C(=O)NCCCNC(C2C(OC)CCCC2)=O)ccc(C(F)(F)F)c(F)c1C N1(C(C(=O)NC(CC)(C)C)c2cccs2)CCc2c(F)ccc(C#N)c2C1 c1(CC(=O)NC2CCN(C(C(CC#C)C)=O)C23CC3)cc(Cl)cc2c1OCC2 C1(CCC)CCCCC1NC(=O)C(CNC(=O)C1=CCC1)OC c1(C(=O)NCC2N(C(Cc3c(C)ccs3)=O)CCC2C)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC(NC(c3n(CC)cc(Cl)c3)=O)C(F)CC2)=O)cnn2ccn(C)c12 CC1CN(C(=O)C(F)Br)CC1n1cc(-c2ccsc2)nn1 C=CC(C)(CCOC)C(=O)N1CCN(CC(C)(C)NC(C2(C)CCCO2)=O)CC1 C1(CNC(C(C)C(C)(F)F)=O)CC(C)(C)OC1(C)C C(=O)(CC(=O)NC1CC1)N(CC(CNC(CC=C)=O)O)C n1(CC(=O)N(C)Cc2cn(CCCF)nn2)ncc2ccccc12 C(C(COC)N=c1nc(N2CCCC(CCC#N)CC2)cc(C)[nH]1)OC N1(C(C=CC(c2ncccc2F)(C)C)=O)CC(NC(=O)CC(=O)C2CC2)C(F)C1 C1(CC(=O)N(C)CC2(C)CCCC2)COCCN1C(=O)CC1CCC(=O)N1C C1(NC(=O)CC(F)(F)F)CC2CC1CN(C(=O)CCc1cccc(F)c1F)C2 c1(C(N2CCC(COC)(NC(=O)CC3OCCCO3)C2)=O)cc(F)ccc1Cl N#Cc1ccccc1OCCS(=O)(=O)NCC(=O)Nc1cccc(F)c1 c1(COCCCN2CCC(CCCCC(=O)OC)CC2)ccc(Cl)c(F)c1 CCCC(C)CC(=O)N1CCC(CCC(=O)NC23CC2CN(C)C3)C1 C1(O)(CNC(CCSC)=O)CN(C(c2coc(N(C)C)n2)=O)C1 C1(NC(C(c2c(C)cccc2C)O)=O)COC2(C1)CN(C(=O)CCS(N)(=O)=O)C2 CCC(CC(=O)N1CCC(C)(C)C1CC(=O)NCc1sc(C)nc1C)CC(C)C C1(C)(C(=O)NC(C(=O)N(CC)CC)C)CC(O)CN1C(=O)CC1CCOC1=O C(=O)(CCCC(C)(C)C#N)NC1C(C(N(CC(CC)O)CC)=O)CC1 C#CC1(C(=O)N(CC(CO)(CO)NC(=O)C(C)C(F)F)C)CCCCC1 CCCCCC(O)CC(=O)N(C(C)C(N1CC(C)(C)CC1C)=O)CCC CCS(=O)c1ccccc1C(=O)NC1CCC(NC(c2cnc(O)o2)=O)CC1 N1(C(C2(CCCC)CCCC2)=O)CC(NC(=O)C(C)(C)CF)C(F)C1 Cc1cncc(C(=O)NCC(CC2CC2)C(=O)N2CCCCC2CF)n1 Cc1cc(=O)ccn1CC(=O)NCC1CC1CNC(c1cncc(C#N)c1)=O c1(NC2CCC(NC(C(=O)NC3(C)CC(=C)C3)=O)CC2)ccc(Cl)cc1Cl Cc1cc(C(=O)NCCC#N)ncc1-c1ccccc1CC1CC1 Cc1csc(CC(=O)NC2CC(CNC(=O)C(C)Cn3ccnc3)C2)n1 N1(C(C(CSC)OC)=O)CCCCC1CNC(c1cc(-c2cnn(C)c2)on1)=O c1(C(N(CCCN(C(C(C)Oc2cccc(F)c2)=O)C)C)=O)cncc(F)c1Cl CCC(C)(CCNC(c1cnn[nH]1)=O)NC(=O)CCCOC(C)C N1(C(CC(CC)C)=O)CC(C(=O)Nc2ccc(OC)c(C)c2)CC(C)(C)C1 c1(NCC2CC3CCC2C3)cccc(N2CCOCC2)c1.N12CC(C1)NC2=O C1(CNC(C2CN(C(c3ccn(C4CC4(F)F)n3)=O)C2)=O)(CO)CC1(F)F N1(C(C(=O)NC2CC2)=O)CCC2CN(C(=O)CC3OCCCO3)CC12 c1(C(N2CC3(CCNC3=O)C2)C(=O)NC)nnc2n1CCCCC2 c1(C(N(CCCNC(CNC(CCC)=O)=O)CCC)=O)sc(O)nc1C C1(NC(C2CN(C)CC(C)O2)=O)CC2(CCN(C(=O)CC(C)(C)C#N)C2)C1 c1(SC)ccccc1CC(=O)N(CCCCNC(C1CC1(F)Cl)=O)C c1(C(=O)NC(CN(C(c2occc2C2CC2)=O)CC)C)nccn2nccc12 c1(C(N2C(C(=O)NCC3N(CC)CCCC3)CCCC2)=O)occ2c1CCC2 N1(C(C2CCCC(OC)C2)=O)CCOC2CN(C(=O)C(N)=O)CC12 Cc1cc2ncn(CC(=O)NC3CC(O)CN(C(C4CC(O)C4)=O)C3)c2cc1C c1(CC)cc(F)ccc1-c1ccc(C(=O)Nc2c(C(N)=O)ccnc2Cl)c(C)n1 C=C1CC2(C1)CC(C(N1CCC(NC(=O)Cn3ncnn3)C1C)=O)C2 c1(C(=O)NC(C(C)NC(CCc2cc(C)no2)=O)C)ccc(-c2ccsc2)cc1 N1(C(CCc2ncc(C)[nH]2)=O)CC2CCCC1(CNC(C1CCCCC1O)=O)C2 c1(C(N(C2CCN(C(=O)COCC(F)F)C2)CC)=O)cccc2nc[nH]c12 CC1CN(C(=O)C2CC2)CCC1NC(c1c(-c2ccccc2)noc1C1CC1)=O c1(NC(C2N(Cc3cc(C)oc3C)CCC2)=O)ccc(Br)cc1C(C)(C)C C1(C(N(C)CCOCCNC(c2ccc(CF)cc2)=O)=O)CCc2cncn2C1 N1(C(C(C(C)C)C#N)=O)CCN(C(=O)CCc2ccc(F)nc2)CCC1C c1(C(=O)NCC(C)NC(c2c(OCC)ccc(C)c2)=O)ccc2c(C)[nH]nc2c1 N1(C(C(Cc2cn[nH]c2)NC(=O)CC=C(Cl)Cl)=O)CCC(C2CCC2)C1 C1(OCC)CN(C(=O)C(C2CN(C(c3cscc3OC)=O)C2)OC)CC1C C1(CC(N2CCCCC(NC(c3cnoc3)=O)C2)=O)CCC2(CCC2)CO1 c1(C(=O)NC23C(CN(C(c4ccc(C)o4)=O)C2)C3)cc2sc(C)cc2s1 C(=O)(C1=C(C)OCCS1)N1CCC(C=C)(C(N2CCOCC2CO)=O)C1 c1(C(N2CCCC(NC(C3CCS(=O)(=O)C3)=O)C2)=O)cc(Cl)ccc1Cl C(=O)(CCCCCCN=[N+]=[N-])N1C(CNC(=O)C(C)C2CC2)CC(OC)C1 c1(N(C)C(c2cnc(-c3ccccc3)o2)=O)ccc(NS(=O)(=O)C2CC2)cc1 c1(Cn2c(C)c(NC(=O)NC(C)(C)C)cn2)ccc(=O)n(-c2cnn(C)c2)c1 Cn1cc([N+](=O)[O-])c(C(=O)NC2CCCN(C(=O)Cc3ccns3)CC2)n1 C(=O)(CCCN=[N+]=[N-])NC1C(NC(C2C(C)(C)CCC2)=O)CCCC1 Cc1ccc2c(ccn2CC(N2CC3CCC2CNC3)=O)c1 c1(C2CCN(C(c3nc(C(=O)O)nn3C)C)CC2)ccc(Cl)cc1Cl N1(C(CCc2cc(C)[nH]n2)=O)CCOC(CC(=O)NCCn2cnnn2)C1 N1(C(CC2N(C(CC3CC(=C)C3)=O)CC2)=O)CC(F)(F)CC1C c1(C(N2CC(C)C(CNC(=O)C(N)=O)C2)=O)ccc(O)cc1F CC1(C)CC(CNC(=O)CCOCC(F)(F)C(F)F)CN(C(c2cnn[nH]2)=O)C1 C(=O)(C(C)C(O)CCCC)N1CCC(n2cc(CC3(SC)CNC(=O)C3)nn2)CC1 N1(C(c2n(CC=C)ccn2)=O)CC2C(CNC(=O)CCC(C)C)C2C1 C1(CNC(c2ccc(F)cc2Cl)=O)C(O)C(O)CN1C(C1CC2C=CC1O2)=O S(=O)(=O)(c1ccc(NCCC23CCC(C2)C(=O)N3)cc1Br)N(CC(C(C)C)C)C C(=O)(CC(CC(C)C)NC(=O)Cc1cn(C)cn1)NC(CC=C)(C)CC=C C1(O)(C(C(=O)OCC)(F)F)CCN(C(CCCNC=O)C(=O)NC)CC1 O=C(CC1=CCCCC1)NCC12CCC(CN(C(C3CCCN3C3CC3)=O)C1)C2 CCCCC(C(=O)NC(CNC(c1occ2c1CCOC2)=O)C1CC1)C(C)C C1(NC(c2c(SCC)nccn2)=O)CN(C(=O)CCOCC(F)(F)F)CC1(C)C C12(NC(C3C(SC)CCC3)=O)CC(C1)N(C(=O)COCc1cc(C)on1)C2 c1(CC)cc(C(=O)NCc2ccoc2C(=O)NOC2CCC2)c(C)o1 c1(CC(=O)NCC2(C)CC(NC(C3CSCCS3)=O)C2)c(Cl)cccc1Cl C1(NC(c2c(CNC(CC3(C)CCCCC3)=O)cc[nH]2)=O)C(=O)OCC1(C)C C(=O)(C(O)C(F)(F)c1ccccc1)NC1C(C)CN(C(=O)C=Cc2cocn2)C1 N1(C(CSCC#C)=O)CC2CN(C(=O)C(C(C)C)n3cc(C)cn3)CC2(C)C1 C(C(CC(C)C)C(=O)NOCCC(C)O)NC(c1ccnc(C)c1C)=O N1(CC)CC(CNC(=O)C(CC2CCCC2)NC(=O)CC(Cl)Cl)CC1=O c1(C(N2CCC(NC(C=CCOC)=O)(CO)CC2)=O)c[nH]c2ncccc12 c1(C(=O)NCCC2N(C(CC(C=C)(C)O)=O)CCC2)cc2cnn(C)c2s1 c1(C(=O)OCC(CCCC(=O)OC)=O)cc2ccccc2cc1Br N1(C(COCCN(C)C)=O)C2CCCC1CN(C(=O)CCCCC1CC1)CC2 C1(C(=O)NC(C(C)O)C(=O)N(C)C)(C(=O)O)CC2(C1)CC(F)(F)C2 Cc1nn(CC(N2CCC(NC(c3ncccc3F)=O)C(F)C2)=O)cc1[N+](=O)[O-] c1(C(=O)NC2C(CNC(c3c(OCC)ccs3)=O)CC2)c(OC)ccnc1F CC1c2nccn2CCN1C(c1sc([N+](=O)[O-])cc1Br)C(=O)NC1COC1 C1(NC(C(CCC)CCC)=O)CC1C1CCCN(C(=O)CCCOC(C)C)C1 CN1CCCCCC1C(N1CCC(CC(N2CCOC(CF)C2)=O)C1(C)C)=O c1(C(=O)NC(CCC)CC(=O)NCCN2CC3CC3C2)ccc2n[nH]cc2c1 c1(COC)ccccc1C(=O)N(CCC(C(C)C)NC(=O)CC1CC1C)C C1(CC)(CC)CC(C(=O)N(C2(C(=O)NCCCCOC(C)=O)CC2)C)C1 C1(C(N2CCN(C(c3c(C)n(C(C)C)cc3)=O)CC2)=O)CCCC1S(C)(=O)=O c1(CC)nc(C)oc1C(=O)N(CC(C)N(C(=O)C(C)SCc1ccccc1)C)C c1(OC(C)CCOCCS(=O)(=O)NCC2CCC2)ccc(I)cc1 N1(C(C(CO)NC(C(C)C)=O)=O)CC(C2(NC(C3CCCS3)=O)CC2)C1.C(C)(C)(C)O C1(CNC(c2cnc(CC)s2)=O)CN(C(c2ccc(F)s2)=O)C2(CCOCC2)C1 N1(CC(CC)C(=O)O)CC2COCC2(C(=O)N(CC(CC)CC)C)C1 c1(C(N2C(CNC(c3c(OCC)cncc3)=O)C=CC2)=O)occ2c1CCC2 c1(C(=O)NC(C2CCCN(C(c3ncc(Cl)n3C)=O)C2)C)cccc(F)c1F CCCCCC(CC)C(=O)NC1CC(C(F)C(=O)NCCCCF)C1 C1(CNC(c2c(C)coc2)=O)CC2CCC1N2C(C1CCCN(S(C)(=O)=O)C1)=O C1(NC(CC(=O)OCC)=O)CC(C)N(C(c2scc(OC)c2Cl)=O)C1 C(C)(C(=O)NCC(C1CCC1)OC(C)CCC)SCCCC c1(C(=O)NCC=CCNC(C2(CC(C)C)CC2)=O)cc(F)c(Br)c(F)c1N c1(C(=O)NC(C(C)NC(=O)CCc2ccoc2)CO)ccc(O)c([N+](=O)[O-])c1 c1(OC)c(Br)cc(C(=O)O)cc1S(=O)(=O)NCCC(O)C(=O)O CCC(CC(=O)N1CCN(CC2CCN(C(c3ccccc3)=O)C2)CC1)SC C1(C(N(CC(C)NC(C2CC(=O)N(C3CC3)C2)=O)C)=O)CCCN1N=O N1(C(CC(C)O)=O)CC(N(C)C)C(CNC(c2csc(Cl)n2)=O)C1 c1(C(=O)NCCNC(c2cc(Cl)cnn2)=O)cc(F)c(F)cc1O CCCCCC(C)(C)C(=O)NC(C)CCNC(C1(C)CCCS1)=O C(=O)(C#CC(C)(C)C)N1C(C(=O)NCc2cc(C3CC3)n[nH]2)(COC)C=CC1 N1(C(C2(CC=C)CCCC2)=O)CCOC(CN(C(=O)Cc2cnn(CC)c2)C)C1 C1(NC(c2ccc(-c3nc[nH]n3)nc2)=O)CC2CC(NC(c3cccs3)=O)C1C2 Cc1cccc2c(C(=O)NC3CCCC3NC(=O)CC=C(Cl)Cl)n[nH]c12 Cc1[nH]ccc(=NC(=O)CC2CN(C3CCN(C)C3)C2)c1F C1(CNC(c2c(C)nsc2)=O)CC2CN(C(=O)CCc3ccc[nH]3)CC12 C1(OCC)CC2CN(C(=O)CCN(C(=O)Cc3cc[nH]c3)C)CC12 Fc1ccc(Cl)c(I)c1CN1CC2(C1)CCC(C(F)(F)F)C2 CC1(C)CCC(C(=O)NCC2CC2NC(=O)C(Cl)=CCl)O1 C1(C(=O)NCCC(=C)CNC(C2(O)COC2)=O)CCC(CC)CC1 C1(C(=O)NC(C(=O)NCC2CCCN(C)C2)CCC2CC2)CC12CCCCC2 CC1=CCC(C(N2CC=CC(NC(=O)CN3CCCC3=O)C2)=O)CC1 c1(SC(C2CN(C)CCO2)C)ccc(NC(=O)C=CC2CCC2)cc1O c1(C(c2n(CCC)nnn2)NCCc2cccc(Cl)c2F)cc(Br)ccc1F c1(Cc2cn(CCNC(C(C(C)O)NC(=O)C3CC3)=O)nn2)cc(F)cc(Cl)c1 C(=O)(CCC1=NNC(=O)CC1)NCCCC(C)NC(=O)Cc1cncnc1 C=C(Cl)CC(C(=O)NC(CO)C(=O)OC)NC(=O)CCCCOCC C1(NC(C2ON=C(CC)C2)=O)CN(C(c2csc(S)n2)=O)CCC1C(F)(F)F CC(O)CCCCCC(=O)N1CCC2CN(C(=O)COC3CCCC3)CC2C1 c1(C(=O)NCC2N(c3c(F)cnc(C)n3)CCC2)cccc2c1ccn2C c1(CC)ccc(C(=O)NC(C)(CNC(=O)CC2CCC23CCC3)C(C)C)cc1 CC(C)CC(CNC(C1CCOC1CNC(=O)CC1OCCO1)=O)N(C)C c1(C(=O)NCC2CN(C(c3nc(C)oc3)=O)C(C)C2)ccc2nnn(C)c2c1 N1(C(C)C)CCCC1C(N1CCCC1C(C)NC(c1cnnn1C1CC1)=O)=O N1(C(CC(=O)NC2CC2)=O)CC(NC(c2ccc(-c3nccs3)cc2)=O)C(O)C1 c1(SC)cc(NC(c2cnc(CNC(C3CCCN3C(N)=O)=O)nc2)=O)ccn1 N1(C(C(CSC)(C)C)=O)CC(C)(C(=O)NCCC(=O)NC(C)C)CC1(C)C N1(C(c2n[nH]c(=N)[nH]2)=O)CC2(CC2)CC1CNC(c1cnoc1C1CC1)=O c1(C(=O)NC(C2CCC(C)(C)CN2C(=O)CC(C)(C)C)C)cc(F)c(N)cc1F c1(OC(CC)C(=O)N(n2cc(-c3ccc[nH]3)nn2)C)ccccc1C(F)(F)F N1(C(c2cc(C)nc(Cl)c2N)=O)CCC2(CC1)OCCC2NC(C1CCSC1)=O c1(C(N(CCOCCNC(c2c(N)sc(C)c2C)=O)C)=O)cn2ncccc2n1 c1(N2CCC(C3N(C(c4cn(CC)nn4)=O)CCC3)C2)cc(C)c(C#N)c(C)n1 C1(OC)CC(CNC(=O)C=C2CCCCC2)(NC(=O)CCN2CCCC2=O)C1 N1(c2ccnc(C(C)C)n2)CC2CC(NC(C3CCC4CCCCN34)=O)CC1C2 O=C1COC2(CCN(C(=O)Nc3cccn4nccc34)CC2)CN1 C(=O)(CS(=O)(=O)c1ccccc1F)N1CC2CC(NC(C3(CC)CC3)=O)CC2C1 N1(C(c2c(C)nn(C)c2)=O)CCC2CC2(NC(=O)CC2CCC(F)(F)CC2)CC1 C1(C(N2CC(C(=O)OC)OC3(C2)CCC3)=O)CSC(c2ccccc2)=N1 C(c1ccc(NC)cc1)=CC=C(C(=O)NCC=CC(=O)NC)F c1(C(=O)NCC2(NC(C(C)N(C)C)=O)CCOCC2)cc(Cl)ccc1O c1(OC)cccc(C(C)=CC(=O)NC23CCCN(C(=O)CC4CC4)C2C3)c1 CC1(C)C(C)(C(N2CCCCC(NC(C3CC(Cl)(Cl)C3)=O)C2)=O)C1(C)C c1(CC)ccc(C(C)CC(=O)NCCCCCCNC(=O)Cc2cnsc2)cc1 C=CCC(C)(C)CC(=O)NCCC(C)NC(C1CCC(=O)N1)=O CC(F)(F)CCC(=O)NN1CCCCC1C(=O)N(C(C)(C)C)C1CC1 C12(NC(c3scc(C(N)=O)c3)=O)CCC(CC1NC(c1ccc(F)cc1)=O)C2 c1(C(N(C(C(=O)NCc2ccc(CC)cn2)C)CC)=O)cc(C)c(C)cn1 N1(C(c2n(C)nc(Br)c2)C(=O)NCCCF)CCOc2ccc(Cl)cc2C1 C1(CNC(=O)CCCF)CCCCN(C(C2CCCC2C2CC2)=O)C1 S(=O)(=O)(c1ccc(NC2CNC(=O)C2)c(C#N)c1)NCC(CN(CC)CC)O C1(n2cc(C=CC)nn2)CC2CCC1(NC(c1cnc(C(F)(F)F)cn1)=O)C2 S(=O)(=O)(c1cccc(Br)c1C#N)N1CCC(C(N2CC(C)OCC2)=O)CC1 C(=O)(CC(C)(C)CC(F)F)NC(CC(C)NC(c1[nH]nc(OC)c1Cl)=O)C C(C(CC(=O)N1CCC(N(C)C)C1C)C1CCC1)NC(c1c(C)ccs1)=O C1(N(C(C(C)NC(CC)=O)=O)CCC(=O)N2CCCC2)CCC(C)(C)C1 C1(NC(C2(SC)CC2)=O)CCCC1(C)CNC(=O)C(C)(C)C1CCOC1 CC1(NC(=O)CCc2cnco2)CCCN(C(C2COC(=O)N2)=O)C1 N1(C(C(C)OCC2CC2)=O)C(C(=O)N(C)CCC2CCOCC2)CCC12CC2 C(CCCCC(=O)NC(C)CC1CN(C(=O)CSc2cccc(C)c2)C1)=CC c1(NC(=O)NC(c2ccccc2NS(C)(=O)=O)C)c(F)ccc(Br)c1F C1(C(N2CCCC(CCNC(C3(C)COC3)=O)C2)=O)CCc2ccccc2O1 C=CC1OCCC1C(=O)N(CCC(=O)Nc1ccc(CO)nc1)CC1CC1 Cc1cccc(C)c1C(O)C(=O)NC(CC(C)SC)c1nnnn1C1COC1 C1(CCCN(C(C=C(C)C)=O)C2CC2)CCCCN1C(=O)CC1(C)CCC1 N1(C(C2C3N(C(CN(C)C)=O)C(CC3)C2)=O)CCC12CCC(C)CC2 Cc1nc(C)c(C(N2CCC(OCC(=O)Nc3cc[n+]([O-])cc3)C2)=O)s1 Cc1ccc(C(=O)NC(C)CNC(=O)C(F)(F)c2nccs2)cc1N C1(NC(c2cc(Cl)ccc2Cl)=O)CCCC12CCN(C(C1CCS1(=O)=O)=O)CC2 C=CCCCCCCC(=O)N1CCSCC1CCNC(c1cnc(O)s1)=O n1(CC)c(C(=O)N(CC(=O)N(C2CC3(CCC3)C2)C)C2CCC2)cnc1O c1(C(=O)NC2(C3N(C(CC(CC)O)=O)CCCC3)CC2)c(Cl)ccc(F)c1C c1(C(C(=O)NC(CC)CN(C)C(C2(CF)CC2)=O)=O)cnn(C)c1 C#Cc1ccc(C(N2CCC(O)(CNC(C3(c4oncc4C)CC3)=O)C2)=O)nc1 C1(CC)CN(C(c2cncc(C)n2)=O)CCN1C(c1ccc(CC(C)C)cc1)=O N1(C(c2cc(CNC(CC(CSC)O)=O)[nH]n2)=O)CCCC(CCO)CC1 C1(NC(c2cnnc(C3CC3)c2)=O)CN(C(=O)Cc2cncs2)CC2(CCC2)C1 c1(OCC)ccc(OCC(=O)NC2CN(C(=O)CC3CC34CC4)C2)cc1 c1(-c2ccccc2)c[nH]c2ccc(F)cc12.CCN=C(NCCC1(C#N)CC1)N c1(C(=O)NCC(C)NC(CC(C=C)C)=O)cc(OC)c2occc2c1 CCC(CCCC(=O)N1CCC(N(C)C)C(C)C1)NC(C1CCC(C#N)CC1)=O C#Cc1cc(C(N2CC(CC(N3CCC(OC)C3(C)C)=O)C(C)C2)=O)ccc1C N1(C(C(CC)Sc2ccccc2)=O)CC2(CCC(NC(=O)COCCF)CC2)C1 C1(SC)CN(C(c2c(C)ncn2O)=O)CC1NC(c1cnn(CCF)c1)=O c1(C(=O)NCCCCCNC(C(C)c2ccco2)=O)ccsc1S(N)(=O)=O C(=O)(C1=COCCC1)N1C(C(=O)NCCC(C)O)CCC1C C1(C(N2CC(CNC(c3c(CC)occ3)=O)(OC)C2)=O)CC(F)CN1C CCC(O)C(F)(F)C(=O)OCc1cccc(SC(F)(F)F)c1 C1(NC(=O)CN2CCCC2CO)CC2CC1CN(C(c1ncc[nH]c1=O)=O)C2 O=C1CC(=O)NC(C(=O)NC2(C(=O)NCCOCC(F)(F)C(F)F)CCCCC2)C1 c1(CNC(c2c(Br)ncc(C)c2)c2nnnn2C2(C)CC2)cc2cnccc2o1 C1(O)(CN(C(C(CC)C)=O)C)CCN(C(c2ccccc2-n2cccn2)=O)CC1 c1(C(N2CC(C)C(CNC(=O)C=C(Cl)Cl)CC2)=O)ccc2nc(O)oc2c1 N1(C(c2cnc(C)o2)=O)CC(C(=O)NCCC(F)(F)CO)CC(C)(C)C1 c1(C(=O)NC2CCC(NC(c3nc(C)n(C)c3)=O)CC2)cccc(N)c1C(F)F Cc1[nH]nc(C(F)(F)F)c1C(=O)NCC(CO)NC(=O)Cc1cnn(C(F)F)c1 c1(OC)cc(C(N2CCCC2C(C)NC(=O)C(C)CF)=O)ncc1Br c1(C(=O)NCC2(OC)CCN(C(=O)CCCC(C)O)C2)ccc2n[nH]cc2c1 C1(CN(C(c2ccc(C)n2C)=O)C)CN(C(c2ncsc2C2CC2)=O)CC12CC2 c1(C(N2CCCC(n3cc(C4(O)CCOC4)nn3)C2)=O)ccc2cncn2c1 c1(N(C)C)nc(C(=O)NC23CC(C2)N(C(c2ccnn2C(F)F)=O)C3)cc(O)n1 c1(CNC(C(CO)NC(=O)CCC2CCCOC2)=O)ccc(F)cc1 C(=O)(CC(O)CC1CC1)NCC1C(NC(CCc2cn(C)nc2)=O)C1 C(=O)(C1CCc2nccn21)N1C(CCNC(C=CC(=O)N(C)C)=O)COCC1 CC1CCOCC1C(=O)NCC(C1CC1)NC(=O)CC1(O)CCCCC1 CCCC(C(=O)OC)C(=O)N(CCCNC(c1cccc(C(C)(C)C)n1)=O)C1CC1 C(=O)(CS(=O)(=O)CCCc1ccccc1)NCC(C)NC(C1CCN1S(C)(=O)=O)=O c1(OC)ccc(C=CC(N2CCCN(C(C3CNC(=O)N3)=O)C(C)C2)=O)cc1F CC(C)CCCC(=O)NC1CCN(C(=O)CCc2cnn(C)n2)C(C)C1 C1(C(N2C(C)CC(Nc3nc(C)nc(C#N)c3)C2)=O)CCCC2(C1)CC2(F)F c1(C(=O)NCCCOCCNC(=O)Cc2cc[nH]n2)cncc(C(F)(F)F)n1 c1(NC(CC(C)O)C)ccncc1S(=O)(=O)NCC(C1CCCCC1)(C)C C1(C)(C(N2CCC(N(C)C(c3cc(Br)co3)=O)CC2)=O)CCC(=O)NC1 C=CC1CCCC(N=c2[nH]c3cccc(N(CC)CC)c3s2)C1 c1(C(N(C)CCNC(C2(C)COCCO2)=O)=O)cnc(O)c(F)c1 c1(C(N2CC(C)(NC(CCC(C)SC)=O)C2)=O)[nH]c2c(F)cc(F)cc2c1C S(=O)(=O)(c1ccc(Cn2cc(Br)cn2)cc1)C(=O)NC(CCSC)CCO c1(C(=O)NCC=CCNC(c2ncc(F)cn2)=O)ccc(-c2ccco2)nc1O Cc1cc2c(C(=O)NCCC3CCCCN3C(=O)C(C)N3CCC3)cccc2o1 CC1=C(C(=O)NCC#CCNC(c2occ3c2CCCC3)=O)SCCO1 c1(OC)ccccc1CC(=O)N(CCNC(c1cnn(C)c1C1CC1)=O)C(C)C c1(Sc2n(CC)cnn2)nn(C)c(C(=O)NOCCC(C)O)c1Cl S(=O)(=O)(c1ccc(C(=O)NCCCNC(=O)C(C#N)C(C)C)o1)NC N1(C(CCC(C)C)=O)CCCC12CCCN(C(=O)CC1=NNC(=O)C1)C2 CC(C)C(O)CC(=O)N(C1CCN(C(c2cc(F)ccc2C(F)(F)F)=O)C1)C Cc1cc2[nH]c(=O)c(C(N3CCN(C(C)C(=O)NC4CCCC4)CC3C)=O)cn2n1 c1(OCC)ccccc1NCC1(F)CC1.C1(=O)C(C)N1C1CC1 CCC(CO)(C(=O)NC(CNC(=O)CCC1CC1(Cl)Cl)C1CCC1)OC C1(NC(c2c(OCC)ccc(C)c2)=O)CC2CN(C(=O)COCC(C)(C)C)CC12 C1(C(=O)NCc2c(C)snn2)CC(O)CN1C(=O)CCCN1CCCC1 C1(NC(C2C(C)C2C)=O)(CF)CCN(C(=O)C(Cc2ccccc2F)N(C)C)C1 C(=O)(CC(C)(C)N(C(=O)CSCCN(C)CCO)C)OCC.C12(CN(C)C1)CN2 N1(C(CCCC(C)NC(C(COC)(C)O)=O)=O)Cc2cccc(O)c2C1 C(CC(O)C(F)F)NC(CCNC(C(C)(C)C)=O)=O.C12CC1C(=O)NC2 c1(NC(C)=O)sc(Cl)cc1C(=O)NC1CCC1NC(c1cncnc1C)=O C(Cn1cccn1)(C(=O)N1OC2CCC1CC2)NC(c1ccc2nccn2c1)=O c1(C(C)=O)ccc(C(N2CCC2(C)C2CC2)C(=O)NCC2CC2)c(F)c1 C1(F)(CNC(Cc2c(CC)cccc2)=O)CCCN(C(=O)Cc2cnc(C)[nH]2)C1 C1(NC(C2N(CC)CCOC2)=O)CCCC2CN(C(C3(O)CCCC3)=O)CC12 C(CC(C(C)C)N(C)C)NC(c1c(OCC)scc1)=O.C12CC(C)N(C1)C(=O)C2 C12(C(N3CC(C)C(C(=O)NCC(C)(C)C4CC4)C3)=O)CCC(CC1F)C2 N1(C(COC)=O)CCC(C2CCCN(C(=O)CC(C)CC(C)(C)C)C2)CC1 c1(N(C)CC2C(OC)CC2)ccnc2c1CCO2 C12(CNC(CCn3ncc(C)c3)=O)CCC1CCN2C(=O)Cn1cccnc1=O C1(O)(CNC(C(c2c(C)noc2C)C)=O)CCN(C(=O)C2=CCCS2)CC1 C(=O)(C1=CCC(C)(C)CC1)NC(CNC(C(C(C)C)OCC(C)C)=O)C c1(C(=O)NCC2C(NC(C3(C)CC=CCO3)=O)C2)cncc(N)n1 N1(C(c2scc(OC)c2)=O)CCC(CCCCCNC(c2cscc2C)=O)CC1 Cc1cc(C(=O)NCCCN(C)C(c2ccn(C)n2)=O)[nH]c1C#N c1(C(C(N2C(CNCc3c(C)cccc3)COCC2)=O)=O)ccc(F)c(C)c1 c1(C(=O)NC)ccc(C(=O)NC2CN(C(c3ccnc(S)c3)=O)CC2C)cc1F c1(C(C)=O)cc(C(=O)N(C2CC(NC(=O)CC3CC4CC4C3)C2)C)c(C)o1 C1(C(N2CCC(C)(c3cn(C4C=CCCC4)nn3)C2)=O)CCn2nnnc2C1 c1(C2(C(=O)NCCNC(C3CC34CC4(F)F)=O)CC2)cncc(Br)c1 C1(C(=O)OC)CCCCCCN1C(=O)C(C)(C)C N1(C(C(=O)NCC)=O)CCCC(C(C)NC(C2(COC)CCCO2)=O)C1 c1(CNC(c2c(C)c(Br)cnc2O)=O)cc2c(F)c(F)ccc2s1 CC#CCC(C(=O)N(CC1=CCSC1)C)NC(c1cc(C(C)=O)c[nH]1)=O N1(C(C(COCC)NC(=O)C=NOC)=O)CCN(C)CC1CO O=C1CC(=O)CC(C(=O)NC(C2CCOC2)CNC(c2ccoc2Cl)=O)C1 c1(C(N2CCC(O)(CNC(CC=C=C)=O)C2)=O)cc(C)c(C#N)c(C)c1 C1(CCNC(C2CC=C(C)CC2)=O)CN(C(=O)C#CC(C)(C)C)CCS1(=O)=O c12ccc(cc1F)S(=O)(=O)N1CCc3sc(cc3C1)C(=O)N2.S(C(F)(F)F)CC c1(CNC(c2c(C)cc(C)o2)=O)nc(CNC(=O)C(C)(C)N2CCC2)cc(O)n1 c1(N(c2ccccc2)C2CN(C(CCc3cnn(C)n3)=O)C2)ncnc(Cl)c1F O=C(N=c1nc(-c2cccc(Cl)c2)[nH]s1)NCC(F)C(F)(F)F C(=O)(CCCN=[N+]=[N-])N1C(C2CCN(C(c3c(CCC)nns3)=O)C2)CCC1 N1(C(Cc2scc(C)n2)=O)CCC(CF)(NC(=O)CCSCc2ccccn2)C1 c1(C(=O)NCC(CO)NC(C(C)c2cccs2)=O)cc(Cl)ccc1N CC1CC(C(N2CC=CC(NC(=O)C(C(C)(C)C)C3CCC3)C2)=O)CC(C)O1 Cn1ncc2ncnc(N3CCCC34CN(C(c3ncsc3Br)=O)C4)c12 CC(CCC(=O)NC1C=CCC1)NC(=O)Cc1ccn(C)c1 c1(-c2nc(CO)nn2C2CCC2)cc2ccc(I)cc2[nH]1 C12(C(=O)OCC)CCC(NC(c3cc(Br)ccc3F)=O)(CC1)CC2 c1(N2CCC(C)CC2C)nc(NCc2cccc3ccsc23)c2ncn(C)c2n1 c1(OC)cccnc1C(=O)NC1CN(Cc2cccc(C(C)(C)C)c2)CC1O c1(CNC(C(C)(C)OC)=O)cccc(CN(C)Cc2nncs2)c1 c1(NC(C)=O)cc(C(=O)NCC2CC(NC(c3c(C)ccn3C)=O)C2)ccc1C C(=O)(CCS(=O)(=O)NC)NC1C(NC(Cc2cccc(OC)n2)=O)C1 N1(C(c2nc(C(=O)OC)oc2)=O)CC(CNC(c2ccnc(O)c2)=O)C(O)C1 CC(CNC(C1CCS1(=O)=O)=O)CC(=O)NCC1(C)CC(F)(F)C1 C(=O)(CC1=CCN(C(c2ccc(C)c(O)n2)=O)CC1)NC1CCN(CCC)C1 n1(CC(=O)NC(CC=C)CNC(=O)C(C)CC=CC)cccc(N)c1=O C1(CCOC)(NC(c2cn(CCC)nc2)=O)CCN(C(c2cccs2)=O)C1 c1(-c2c(N)non2)nc(Cl)nc2cccc(Cl)c12 N1(C(CCC(C)O)=O)CC2CC1CN(C(c1n[nH]cc1Br)=O)C2 c1(C(N2CC(NC(=O)CC3(O)CCCC3)C(F)CC2)=O)c(F)cccc1[N+](=O)[O-] N1(C(c2cccc(OCC)c2)=O)CC2(C1)CN(C(c1cncc(C)n1)=O)C2 N1(CC)CC(C(N2CC3CC3(CNC(c3csc(C(=O)OC)c3)=O)C2)=O)CC1=O CCC(C)(C)C(O)C(=O)NCC(C(N1CC(CO)CC(C)(C)C1)=O)OC CC1CC(CNC(=O)CCC2(C)CN(C(=O)CP(C)(C)=O)C2)CCN1C c1(CC)oc2ccccc2c1C(=O)NC1CC2CN(C(=O)C=C(C)Cl)CC2C1 c1(C(N2CCC(O)(CNC(C3CC(CC)C3)=O)C2)=O)cc2ncccc2o1 N1(CC(=O)N(C)C(C2CCC(CN)C2)=O)CC2OCCN(C)C2C1 c1(CNC(=O)NC(C#C)(C)CC)nnc2n1CCCC2C(F)(F)F C1(C(=O)NCC(CN(C(=O)C(C)C(C)C)CC)(C)C)CCCC(C#N)C1 C(=O)(CCCC(=O)NC(C)CN(C(=O)C(C)C1(O)CCC1)CC)NCCC N1(C(CC(COC)C)=O)CCOCC(CNC(c2cnoc2)=O)C1 N1(C(COCC(=O)OC)=O)CCC2(CC2)CC1C(=O)NC1CCc2nn[nH]c2C1 c1(C(N2CCC(C)(NC(C(Br)=C(C)C)=O)CC2)=O)cc(Cl)c(F)cc1O CC1(C(=O)Nc2ncc(C(N)=O)s2)CCN(C(=O)Cc2cccnc2)C1 N1(C(C(CC(C)C)O)=O)CC2CCC1C(CNC(C1C(F)(F)C13CCC3)=O)C2 C1(NC(C2(C)ON=C(C)C2)=O)CCN(C(c2sccc2C#N)=O)CC1(C)C C1(NC(COCCC=C)=O)CC12CCN(C(=O)C=CCOC)CC2.C1CO1 C1(C(=O)NC(C(C)NC(CC2CCN(C(C)C)CC2)=O)(C)C)CC2(CCCC2)C1 C#Cc1ccc(CNC2CCN(C(c3c(O)cccc3Br)=O)C2)cc1 c1(NCC)nc(C)ccc1C(=O)NCC1CN(C(C2CC2C2CCCC2)=O)C1 N1(C(CCOCC(C)C)=O)CC2CC1CC2NC(c1ccc(Cl)s1)=O Cc1c(Br)ccc(N(CCCCN(C)C(c2cnn3cccnc23)=O)C)c1[N+](=O)[O-] C1(CC=C)(C(=O)NC2(CC=C)CC=CC2)CCN(C(=O)CCc2ccnn2C)C1 C1(CC)(CC)CCCN1C(c1ncoc1CNC(=O)C(O)CN1CCCC1)=O c1(C(=O)NCC2CC(NC(C3C(=C)CC3)=O)C2)cccc2c(C)cccc12 N1(C(c2ccc(C)c(CO)c2)C(=O)NCCC2(C)CC2)CCC2(CCCN2C)C1 c1(C(C)C(=O)NC2(C)CCN(C(=O)Cc3ccn(C)n3)C2)ccc(O)c(O)c1 N1(C(c2n(C)nnc2)=O)CC2CC1CCC2NC(C1CCS(=O)(=O)N1)=O C1CC(O)C(=O)N1.n12cc(nn1)C1CN(C1)C(=O)C21CC1.CC(=O)NC C1(C(=O)NC(c2c(C)ccnc2)C)CC(C)CN(C(=O)CC2CCSC2)C1 CCC(CC(=O)NCC1(CCNC(=O)COc2cc(C)on2)CCCC1)C(C)C n1(CC)nc(C(=O)NCCCc2csnn2)c(I)c1C C1=C(CN=c2[nH]c3c(c(=NCC45CCN(CC4)C5)[nH]2)CCC3)CCSCC1 N1(C(CN(C(=O)OC)C)=O)CCC1CNC(C1CC1C)=O c1(C(=O)NC(C)CN(C)C(c2ccn[nH]2)=O)ccc(OC2CC2)cc1.C1(C)CC1 CC1(C(=O)NCC(O)C(=O)NCC2CC23CCCCC3)CCC2CC2C1 c1(C(N2CCN(C(CNC=O)=O)C3C2C3)=O)nc2cc(F)ccc2s1 c1(CCCC(=O)NCCC2(O)CN(C(C3CCCC34CC4)=O)C2)ccc(Cl)cc1 C12(CC(=O)NC3CC(C)(NC(Cc4c(C)scc4)=O)C3)COC(CN(C)C)(C1)C2 C1(C(N(CCC(=O)NC(C#C)C(C)C)CCOC)=O)CC2C=CC1C2 CCC(C)(C)CC(=O)N(CC(N1CCC(O)(C(N)=O)C1)=O)CC(C)C N1(C(COCCCC)=O)CC(NC(=O)C2=CCSC2)C(C(F)(F)F)C1 c1(C(=O)NC2C(NC(COC)=O)CC2)cc(F)c2cn[nH]c2c1 c1(C(=O)Nc2cncc(C(=O)OCC)c2C)cc2ccccc2cn1 c1(C(=O)NC(CNC(C(C(C)C)NC(=O)OCC)=O)C)cc([N+](=O)[O-])c(C)s1 C1(C2CC2)(CNC(c2cnc(C)[nH]2)=O)CCN(C(=O)Cn2nnnc2C)C1 S(=O)(=O)(c1ccc(NC(=O)C(O)CCC(C)C)cn1)NC C(=O)(C1=NOC(C)C1)N(CCN(C(C(CCC)c1ccccc1)=O)CC)CC Cc1ncnc(C)c1C(N1CCC(NC(=O)C(c2ccc(Cl)cc2)CO)C1)=O C1(F)(C(=O)NCCCC(C)NC(C2(CC=C)CC2)=O)CCCOC1 c1(C(C(=O)NC2CCOC2)N(C2CCOC2)C)cc(Cl)cs1 CC(CC(=O)N1CCC2(CC1)CC2NC(=O)C(C)(C)N1CCCC1)C(C)(C)C CC1CN(C(=O)Cc2ccns2)CC(CCNC(C2(N(C)C)CCC2)=O)O1 C1(C(=O)NCC2COC2)CC12CCN(C(c1cccc(F)c1Br)=O)CC2 CCCCCC(O)C(=O)N1CC2CCC1CN2C(C1CC2CC2CO1)=O Cc1ccc2nc(C(N3CC(C)(C)CCC3C)C(=O)NCC3CCCO3)cn2c1 N1(C(C(C2CCCC2)OCC)=O)CCOC(CNC(C2(OC)CCCOC2)=O)C1 c1(C(N2CC(NC(COC3C(CC)CCCC3)=O)(CO)C2)=O)cc(O)nc(O)c1 c1(C(=O)NC2C(CNC(CN(C)CC)=O)C2)ccc(Cl)c(Br)c1F C(=O)(C1=CCCCO1)NC1(C2N(C(c3ccc(N(C)C)cn3)=O)CCC2)CC1 C1(N(C(C(C)CC2CCC2)=O)C)CCCCN(C(c2ccccc2C(C)O)=O)C1 C1(CNC(c2n(CC)ncc2)=O)COCCN(C(c2ccc(N)cc2OC)=O)C1 N1(Cc2c(NS(C)(=O)=O)cccc2)CCOC2(CCCNC2)C1 C(C(C(=O)N1CCCC1CCNC(=O)C(C)(F)c1ccon1)OC)OC C1CN=C2N=C(C3=C(N2)CCOC3)N2CCC(C2)S1.C(C)(C)(C)CSC S(=O)(=O)(c1cc(C(=O)NCC2(Cc3ccccc3)CCOC2)ccc1Cl)N(C)C N1(C(C23CC4CC2C3C4O)=O)CC2(CC2)CC1CNC(C1CCC(=O)N1)=O c1(CCCCC(N2CC=CC(NC(=O)COCCF)C2)=O)ccc(O)c(F)c1 C(=O)(C1=COCCO1)N1CC(C2OCCN(C(CCSCC(N)=O)=O)C2)C1 C1(C(=O)OC)CCN(C(C(=O)N(C2CCCCC2)CC#N)C2CC(O)C2)CCO1 C(=O)(C(C)(C)CC(F)F)N1CCC(NC(c2c(OC)scc2)=O)CC1C c1(COCC(CNC(=O)CN2CSCC2=O)O)ccccc1 c1(C(C(=O)NC(CN(C(COCCOCC)=O)CC)C)C)c(C)n[nH]c1C c1(C(N2CCC23CCC3)C(=O)NC(CC)(C)C)ccc(F)c2c1CCC2 N1(CC(N2CCN(S(C)(=O)=O)CC2)=O)CCNCC1c1cccc(Br)c1 c1(OCC)nc(Cl)ccc1C(=O)NC1CCCN(C(=O)C(C)(F)F)C1 c1(NC(=O)CCC2CC2(Cl)Cl)cccc(CNC(C2CNC(=O)N2)=O)c1 CC1(CCNC(=O)CO)CCN1CCNC(=O)C(F)=CC1CC1 c1(C(N2C3(CNC(C4C(C)N(C)CC4)=O)CCC2CC3)=O)ccc([N+](=O)[O-])cc1 N1(C(C(C(C)NC(C2C(C(C)C)CCO2)=O)C)=O)CCCCCCC1 c1(OC(C)C)cccnc1C(=O)NCC(O)CCNC(c1ocnc1C1CC1)=O C(C(=O)NC(C1CCCN1C(=O)CS(=O)(=O)CC)C)(C(C)(C)C)SC Cc1ncc(C(N2CC(NC(C3CCC34CCC4)=O)CC2CO)=O)c(=N)[nH]1 C(C)(CCCCNC(=O)Cc1cccc(C(C)(C)C)c1)NC(C(C)OCC#C)=O Cc1cc(C(N2CCCCC(NC(C3C(C)C3C)=O)C2)=O)cc(C)c1OC(F)F C=C(C)CC(C(=O)NCCC1(C)CC1(F)F)NC(=O)CCn1ccnc1 c1(C(=O)NC2C3CN(C(CC(C=C)(C)O)=O)CC2C3)ccc(S(=O)(=O)CC)cc1 N1(C(C(N2CCCC(O)C2)C)=O)CCC(F)(CNC(=O)CC2CSC2)C1 CN1CCOCC1C(=O)NCCC1CC(NC(=O)C(N2CCCC2)C2CC2)C1 C1(F)(C(N(CCN(C(c2cc(O)n(CC)n2)=O)CC)CC)=O)C(C)(C)C1(C)C N1(C(CN(C)S(N)(=O)=O)=O)CCC(C2CC(NC(c3nn(C)c(Cl)c3Cl)=O)C2)C1 Cc1ccc(C)c(NCC(N2CCCCC2C(C)NC(c2ccccn2)=O)=O)c1 C=CC(C(F)(F)F)NC(=O)C(c1ccccc1)NC(c1c(C)n[nH]c1C)=O C(=O)(CN=S(C)(C)=O)N1CCC(CCNC(C2N(C)CCOC2)=O)C1 c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CCCC1CNc1ccccn1 C1(CC(=O)N(C2(C(=O)NC(C)Cc3cnn(C)c3)CC2)C)CC(C)(C)CO1 c1(NC(N2CCC(c3nnco3)CC2)=O)cccc(C2CCOC2)c1 N(C(=NCCn1cccn1)NCC1CCS1(=O)=O)CC(c1ccc(C)cc1)(C)C Cc1nn(C)c(-c2ccsc2)c1C(=O)NC(C)CC(C)NC(C1CC(O)C1)=O CC(CC(=O)NCc1c[nH]nc1C(N1CCC(c2nc[nH]n2)C1)=O)C1CCCO1 N1(CCCc2onc(C)n2)Cc2ccccc2CC1CNC(C1CCS(=O)(=O)N1)=O c1(C(N(C2CN(C(C=CC(C)(C)SC)=O)C2)C)=O)cc(F)c2[nH]nnc2c1 C#Cc1ccc(C(=O)NC(CNC(c2ccc(Br)cc2N)=O)CO)nc1 Cc1nn(CC(N2CCC(Cn3cc(C4CCCCO4)nn3)C2)=O)cc1[N+](=O)[O-] c1(C(N2CC(NC(C(C)(C)CC#N)=O)C(C)(C)C2)=O)nccc2cccnc12 C(=O)(C1CCCc2nn(C)cc21)N1CC2CC(CN(C(C(CCC)C#N)=O)C2)C1 c1(C(=O)NC(CN(C(=O)C(F)n2cccn2)CC)C)cc(-c2cccnc2)no1 C(=O)(C#CC(C)(C)C(F)F)N1C(C)C(c2ccccc2)CCC1 c1(NC(C)CNC(c2cnn(CC(=O)OC(C)(C)C)c2)=O)cc([N+](=O)[O-])n[nH]1 c1(SC)ccsc1C(=O)NCC(C1CCCCC1)NC(=O)Cc1ccoc1C C1(CCCCNC(C23CC(C)(C2)C3)=O)CCCN(C(=O)CCn2ccnc2)C1 C1(CCNC2CCN(C(C(=O)NC(C)C)=O)C2)CCCC1(F)F c1(SC)ccsc1C(=O)NC1CC(N(C(=O)C=Cc2ccsc2)C)C1 N1(C(c2cc(OC)ns2)=O)CCN(C(c2ccc3cccnn23)=O)CC2(CC2)C1 C1(C(=O)NC(CCNC(CCCCCC=C)=O)(C)C)CCc2cn(C)nc2C1 c1(C(CC)NC(=O)CCCCn2cc(CN(CC)CC)nn2)ncc(F)cc1F N12CCc3cc(ccc3C1)C2.c1(C(=O)O)ccc(O)c(CN2CCSCC2)c1 N1(C(c2c(CCC)n(Cc3ccccc3)nc2)=O)CCN(C(=O)C(C)O)C(C)C1 N1(C(C(C)C(C)(F)F)=O)C2CCC1C(C)C(NC(=O)CNC(=O)CC(C)(C)C)C2 CC(F)(F)CC(=O)N1CCCCC1CC(=O)NCC1CCCOCC1 c1(C(N2C3CC(NC(CCC)=O)CC2CC3)=O)cc2cc(O)ccc2nc1C c1(C(N2CCC(Cc3c(C)cccc3)C2)=O)cc(F)cc2ccoc12 C1(=O)CC1=O.C1(C2CCCO2)C(=O)N1.CO C1(NC(C(C)SCCCC)=O)CCN(C(c2scc(C)c2C)=O)C1C c1(C(=O)NCC(=C2CN(C(c3cc(CCC)on3)=O)C2)F)ccc(OC)c(C)c1 c1(CC(=O)NC(C(C)OC)C)c(C)nc2nc(=N)[nH]n2c1C N1(S(CCOC)(=O)=O)CCN(C(=O)C(c2cc(Cl)cc(Cl)c2)O)C2(CC2)C1 CC(CCCC(=O)NC1CC2CC2C1)NC(C1CC1(F)F)=O N1(C(c2c(N(C)C)cccn2)=O)CCCCC(NC(c2c(O)cccc2Cl)=O)C1 c1(C(C2C(C#N)C2)NCC2(NC(=O)CCC3CCOCC3)CC2)ccccc1F C1(C#N)(C(=O)NC2CCN(C(c3c(C)c(Br)sc3)=O)C2)CC2(CCC2)C1 C1(CNC(c2n(CC)ncc2)=O)CC2CN(C(=O)C(C)(C)C(C)C)CC12 c1(CC(=O)NCCCCCNC(c2c(SC)csc2)=O)c[nH]c2ccc(Cl)cc12 C1(C(N2CCC(C)(CNC(c3cc(C)oc3)=O)C2)=O)CCC(C2CC2)C1 Cc1cc(C(=O)NCC(F)CNC(=O)CNC(=O)C=Cc2ccco2)ncc1Cl C1(C)(CCC(=O)NCCC(=O)N(CC)CC)CCCN1C(C1CCOC1CC)=O N1(C(C(=O)NCC=C)CCc2cccc(Cl)c2)CCc2ccncc2C1 C1(CCCC(=O)NCC2(F)CC(CNC(COCC#C)=O)C2)CCCC(=O)N1 C(C(O)CC(=O)NCC12CCC(CC1)O2)NC(CC(C)N(C)C)=O C1(C(N(CCC=C)CC)=O)CN(C(c2cc(C(=O)OC)ccn2)=O)CCC1(C)C c1(C(=O)NC(C2(O)CN(C(C3(C#N)CCC3)=O)C2)C)[nH]nc([N+](=O)[O-])c1Cl N1(C(CCCC2(C)N=N2)=O)CCC(O)C(NC(=O)CCC2CCC2)C1 C1(CC(=O)NCCCNC(c2cc3[nH]ccc3s2)=O)CC2(CCC2)CO1 c1(NC(C(C)(C)CF)=O)cnc2c(c1)C(=O)NCC2 n1(CC(N2C(CCCNC(C3CCCC(C)C3)=O)CCC2)=O)ccc([N+](=O)[O-])n1 N1(C(c2cnc(Cl)s2)=O)CCCC2(C1)CN(C(C1CCC3(C1)N=N3)=O)CCO2 Cc1nnc2n1C(C(=O)NCC(C)NC(C1(n3cnnn3)CCCCC1)=O)CC2 C(=O)(C1CCc2c[nH]nc21)N1CCN(C(=O)Cn2cncn2)CC1C1CC1 C1(CNC(c2ccc(-c3nc(C)sc3)s2)=O)CC(F)CN1C(=O)C=CCN(C)C N1(C(C(CC)N(C)C)=O)CCC(CNC(c2ncn(C)n2)=O)(COC)C1 c1(C(=O)NCCOCCN(C(CC(=O)NCC#C)=O)C)nc(Cl)c(CC)[nH]1 c1(OC)sc(C(=O)NC2CC(c3ccccc3)(NC(=O)C3CC3)C2)cc1Br C1(NC(=O)C=Cc2ccc(Br)s2)CCC12CN(C(C1CC13CCC3)=O)C2 c1(C(N(CCN(C(C)C)C(c2ncc(CO)[nH]2)=O)C)=O)c(Cl)cnn1C C(CC(C)C)(C(=O)NCC1CCCCC1C(N1CC(F)CC1CO)=O)OC c1(C(=O)NCCn2ncc(C(=O)NC(CC(C)C)(C)C)c2)cnc2n1CCC2 C1(OC)CCC(CC(N2CCC2CNC(c2[nH]c(C)cc2C)=O)=O)CC1 C1(CNC(c2ccoc2Cl)=O)CCCN(C(=O)C=Cc2ccc[nH]2)C1 N1(C(C2CCN(C)C2=O)=O)CCN(C(=O)CCCNC(N)=O)CC1CC(F)(F)F CCCCC(C(=O)N1CC(F)(CNC(C2CCCSC2)=O)C1)C(C)C N1(C(CCNS(CC)(=O)=O)=O)CCC(CNC(=O)C(=CC2CCCCC2)F)CC1 C12(CCCC1)C(=O)N2.C1(NC(CN(CCOC)C)=O)CCC1COC Cc1cn2cc(C(=O)NCC3CN(C(=O)CCC4CCOC4)C(C)(C)C3)sc2n1 C(=O)(CN=c1cc[nH]cc1)NCc1nccc(C(N2CCOCC(C)C2)=O)c1 CC1=CCC(NC(=O)C(C)(C)C2CCCN2C(=O)CC2CCC(C#N)C2)CC1 N1(C(CC2N(CC)C(=O)CC2)=O)CCC2(C1)CN(C(=O)CCc1cn(C)cn1)C2 N1(C(c2c(C)noc2)=O)CCCC2(CCCN(Cc3cc(F)ccc3F)C2)C1 C12(C(=O)NCC3(NC(Cc4cc(COC)on4)=O)CCC3)CC(CC(C)O1)C2 C(C#CCN=c1nc(N2CCCC(C(=O)OC)C2)c2c(ncn2CC)[nH]1)OC c1(CC)nn(C)c(CC)c1C(=O)NC(C)CN(C)C(c1ccn(C)c1)=O N1(C(C(CC)OCC)=O)CCC(CO)(CNC(C2CCCCC(=O)N2)=O)CC1 C1(NC(C(CCOCC)NC(C2CCN(C)CC2)=O)=O)CN(C)CC1(F)F C1(C)(C(N(C2CCN(C(C(C)OCC#C)=O)CC2)CC)=O)COC(C)(C)CO1 N1(Cc2c(NC(c3c(C(=O)OC)cccc3)=O)ccs2)CC2C(C1)C2(F)F Cc1ncsc1CCNC(c1cc(OC)ns1)c1nnnn1CCOCC1CC1 C=CCC(CNC(=O)CCCCCNC(=O)C(C)CC1CC1)CC(C)C c1(CS(=O)(=O)NC(C2CCCOC2)CC)cccc(OC2CCCC2)c1 N1(C(CC2(OC)CCC2)=O)CC2CCC1C1CN(C(c3ccccc3O)=O)CC21 c1(C(N(C)CCOCCCNC(=O)CCCN(C)C)=O)nccc2ncccc12 C1(CCC(=O)NC(C(=O)OC)(C)C2CC2)CCN(C(=O)C(C(C)C)SC)CC1 N1(C(CCCC(C)NC(C(CC=C)CC)=O)=O)CCC12CCOCC2 N1(C(C(C)NC(c2ccoc2)=O)=O)CCOC2(CCN(C(=O)C(F)F)C2)C1 N1(C(C(C)NS(CC)(=O)=O)=O)CC(O)(CCNC(c2ncnn2C)=O)C1 CN1CCC(NC(=O)C=C2CCSCC2)C12CCCN(C(c1cnns1)=O)C2 N1(Cc2sc(C(=O)OC)c(C)c2)CC2CCC1CN(C(C(C)(C)C)=O)C2 C#CCC(C)(C)C(=O)NCC(C1CC1)N(C)C(c1cc2sccc2s1)=O N1(C(c2c(CC)nco2)=O)CC(N(C)C(c2cc(OC)no2)=O)C(O)C1 c1(C(=O)NC23C(C)OC(CNC(=O)Cn4cnnc4)(C2)C3)c(F)ccc(F)c1F c1(CC)ccnc(C(=O)NC(CC2CC2)CC(=O)NCC2(Cl)CCC2)c1 C#CC1(C(=O)N(CC(CC)NC(=O)CCCNC(=O)C2CC2)C)CCCC1 C(=O)(C1Cc2ccccc21)N1CC=C(CNC(c2c(C(C)C)occ2)=O)CC1 Cc1nn(C2CC2)c(Cl)c1C(=O)NC1CCCC1NC(c1ccc(N)c(N)n1)=O N1(C(CNC(CC)=O)=O)CC2(CCC2NC(=O)C(=O)Nc2c(F)cccc2F)C1 C1(CNC(C(CC)OC)=O)CC(F)CN1C(c1cccnc1)=O Cc1cc(Cl)c(C(=O)NC2(C)CCN(C(c3ncccc3F)=O)CC2)cc1C C1(CNC(C(C2CC2)SC)=O)CCN(C(=O)CNC(=O)CN(C)C)C12CC2 C1(N(C(=O)CC2CCC(C)CC2)C)CN(C(c2cnnn2C)=O)CC12CC2 N1(C(C(c2ccco2)SC)=O)CCC(CCC(=O)NCCc2nc(C)cs2)C1 CC1=NOC(C)(CNC(=O)C(C)N(C(=O)Cc2ccon2)C)C1 Cn1nc(C(=O)Nc2cc(I)ccc2-n2cccc2)c(Cl)c1Cl C1(NC(CSCC(=O)OC)=O)COCCC1NC(=O)C(F)CC1CCC1 C1(CNC(CCS(C)=O)=O)CN(C(=O)CC2CC2)C2COCC2O1 CCC(CC(=O)N(C)CC1(C)CCCO1)NC(=O)C(F)F CCCCC(O)CC(=O)NC(CN(C)C)C(=O)NCc1ccncc1OC C1(CNC(c2cc(CNC(C3C(C)CCO3)=O)sc2)=O)CCC(=O)NC1 S(=O)(=O)(c1cccc(Cl)c1Cl)NC12CC(C(=O)NCc3ncc(Br)s3)(C1)C2 c1(OC)nc(Cl)ccc1C(N1CCC(C(C)NC(C2CCN(OC)CC2)=O)C1)=O Nc1cccc(Cl)c1CNCC(O)Cn1ccnn1 CCC(C(=O)Nc1ccc(NC(c2ccc(OC)cn2)=O)cc1C)C(C)C N1(C(CCOCCOC)=O)CC2C3CCC(C(NC(=O)C(O)P(C)(C)=O)C3)C2C1 Cc1cccnc1C=CC(=O)NCCC1C(C)CCCN1C(c1coc(O)n1)=O N1(C(C(C)OCCC(C)C)=O)CC(C)(C(=O)NCC2(CF)CC2)CC1(C)C CC(C)(C)C(O)C(=O)N1CC(O)C(O)C1CNC(=O)C(F)=C1CCCC1 C1(N(C(c2c(C)snn2)=O)C)CCC2CN(C(C3CC(O)C3)=O)CC12 C(=O)(C(CCC(N(C(C)C(O)C(F)F)C)=O)C(C)(C)C)OC(C)(C)C C=CC(CC)CC(=O)NC(C1CC(NC(C2CCOC(C)(C)C2)=O)C1)C CC1(C)Cc2cc(CN(c3cccc(-c4ccncc4)c3)C=O)ccc2O1 C1(NC(C(F)=C(C)C)=O)CCCN(C(c2ccc(-c3ccco3)[nH]2)=O)C1 C1(C(N2CCC(C(C)(C)NC(C3COC(=O)C3)=O)C2)=O)CCN(S(N)(=O)=O)CC1 C(=O)(C(CC(C)(C)C)OC)NCCn1ccc(C(N2C(C(CC)C)CCC2)=O)c1 N1(CC(=O)NC(C2CCCCN2C(=O)C=CBr)C)CCCCCCC1=O C1(NC(C2(NC(C3CC34CCCC4)=O)CCSC2)=O)CCN(C2CCC2)CC1 N1(C(c2ccc(CNC(C3CC(OC)C3)=O)cc2)=O)CCCN(C(C)=O)CC1C c1(COC)ccc(C(N2CC(CNC(=O)Cc3ccco3)C(C)C2)=O)cc1 c1(C(N2CCC(F)(C(=O)NCC3CN(C)C(=O)C3)CC2)=O)ccc(Br)c(F)c1F N1(C(C2(C#N)CC(=O)C2)=O)CCCC2(CC(NC(c3cccnc3Cl)=O)C2)C1 c1(C(=O)NCCC(C)NC(c2conc2C2(C)COC2)=O)ccc(C(F)F)cn1 C1(NC(CCn2c(C)ncc2)=O)CC2(C1)CC2C(=O)N(CCCO)C1CCC1 N#Cc1cc(C(N2CCC(NC(=O)CCCC(F)(F)F)CC2)=O)cc2[nH]ccc12 C1(C(=O)OC)(NC(COCCC=C)=O)CCOCC1.C1C(F)C(=O)N1 C1(CNC(C2ON=C(CC)C2)=O)COCCN(C(=O)CCc2cncc(O)c2)C1 c1(C(=O)NCC2CC(NC(C3C4CCCOC34)=O)CC2O)cc(Cl)nnc1O N1(C(C(CN(C(COC(CC)C)=O)C)C)=O)CC(O)(C2CC2)C1 Cc1onc(Cl)c1C(=O)NC(C)CCCNC(c1cc(C2(C)COC2)no1)=O C1(OC)CC2(C(=O)NC3CC3NC(=O)C(c3cncn3C)N(C)C)CC12 Cc1cccc(C(=O)NCCCCC2CN(C(C3CCCC34CC4)=O)C2)c1N CC(C)C(CO)CCNC(=O)CC(C)(C)NC(=O)CNC(=O)CN(C)C C1(C)(C(=O)OC)CC(OC)(OC(C2(C(=O)O)CCCCC2)=O)C1 C1(NC(c2c(C)nncc2)=O)CCC2(CCCN(C(c3cc(F)n(C)n3)=O)C2)C1 O=C(C#CC1CCCO1)NCCCOCCCNC(=O)C(c1cccc(F)c1)O N1(CCNC(C(CC)O)=O)CCC(NC(=O)CCC2(C#N)CCC2)CC1 c1(C(N2CCC(C(NOCCN=[N+]=[N-])=O)CC2)=O)cc(F)cc(F)c1 C12(NC(COCCC(C)C)=O)CCC(C(=O)NC3CCN4CCC3C4)(CC1)C2 c1(Cn2c(C(C(CC)C)NCCCC(=O)OC)nnn2)ccc(C)cc1Cl C#CC(CNC(=O)C(C1CCCO1)NC(=O)CC1CCN(C)CC1)C(C)C c1(OC)sccc1C(=O)NC1CCCC1NC(=O)CCN(S(C)(=O)=O)C c1(C(N(C)CC2CN(C(=O)C=CI)CCO2)=O)c(F)cccc1[N+](=O)[O-] c1(C(=O)NCC2(F)CC(CNC(c3c(C)coc3C)=O)C2)cc(O)cc(F)c1F C(=O)(C1=CC2C=CC(C1)C2)N(C1CCN(C(c2cc(C)cc(N)c2)=O)C1)CCO CCC(CC)C(C(=O)NCCc1cccc(F)c1)N1CC(CC)CC(C)C1 C=CC1OCCCC1C(=O)NCCC(C)NC(c1cc(Br)sc1C)=O C1(NC(C(C)(C2CCC2)NC(c2c(Cl)cn(C)n2)=O)=O)CCCC(O)CC1 Cc1cc(Cl)c(C(=O)NC2(CF)CCN(C(C3CCC4(CCC4)C3)=O)C2)cc1F CCC(Cc1cn(C(c2nnc(C3CCCC3)o2)C)nn1)C(=O)O Cc1ncccc1C(=O)NC(C1CCN(C(C2CCCSS2)=O)C1)C c1(CCC=O)c[nH]c2cc(Cl)ccc12.C12(C(N(CCCN)C)=O)CC3CC1C2C3 N1(C(CCC(C)N(C)C)=O)CCC(NC(C2(CF)CCC2)=O)C(C)(C)C1 c1(C(N2CC(C)(NC(c3cn(C)nc3)=O)C2)=O)ccc(NC(=O)C2CC2)cc1 c1(COC)nc(C)ncc1C(=O)NCc1cn(C(C)C(=O)NC(C)(C)C)nn1 c1(C(=O)NCC2(NC(CCCC3C(C)C3)=O)CCC2)cc2n(n1)CC(C)NC2=O c1(C(=O)NCC(CNC(C(CC)CC)=O)(C)O)ccnc2cc(F)cnc12 C=CCCCC(C1CC1)NC(c1coc(C(C)NC(=O)C=Cc2ccco2)n1)=O C1(N(C(=O)C(=O)C(C)(C)C)C)CC2CCC(C1)N2C(=O)C=Cc1ccnn1C Cc1ccc(F)cc1C(N1CCCC(CNC(=O)Cc2ncc(C(F)(F)F)[nH]2)C1)=O CN1CC(NC(=O)CCNC(=O)CC(C)(F)F)C(F)(F)C1 C1(NC(C(CC=CC)NC(C2CN(C)CCO2)=O)=O)CCCCC1(C)C C1(NC(c2scc(CNC(c3c(C)con3)=O)c2)=O)CCC(C#N)CC1 N1(C(C2OCCN(C)C2=O)=O)CC(NC(C2(S(N)(=O)=O)CC2)=O)CC(C)(C)C1 N1(c2nnc(CCC)s2)CCC(C)C(NC(=O)CCc2cn(C)nn2)C1C C1(C(C)C)CCC(C)CC1C(N1CCCC(N(C(=O)C(C)CC2CC2)C)C1)=O C(=O)(CCS(C)(=O)=O)NCC1C(NC(CCc2cccc(OC)c2)=O)C1 C12(NC(c3cc(OC)no3)=O)CCCC1CN(C(=O)C1=COCCC1)C2 S(=O)(=O)(c1ccc(NCC2CCCC(F)C2)c(F)c1)NCc1c(C)nns1 C1(CCN(C(CN2CC=C(C)CC2)=O)C(C)C)CN(C(=O)OC(C)(C)C)CC(C)O1 c1(CC(=O)NCCNC(=O)CC2=CCCCC2)ccc(F)cc1[N+](=O)[O-] CC1(C)C(C(=O)NC(C(N2CCCC(C)(CO)C2)=O)c2ccco2)CC1(F)F CCC(C)C1CC(=O)N1CC(C)C.C(=O)(C(O)Cn1cncn1)N1CCCC1 C(CN=c1[nH]c2c(c(=NCC3CC3(Cl)Cl)[nH]1)CC(C)CC2)c1ccc(C)cc1C CC(C)(C)C1=NOC(C(=O)NCC2CCN(C(=O)Cn3cncn3)C2(C)C)C1 S(=O)(=O)(c1ccc(=NCC(CCS(C)(=O)=O)OC)[nH]c1)NCCN(C(CC)C)C c1(OC)cc(C(=O)Nc2ccc(-n3cncn3)c(C)c2)c(N)c(Br)c1 c1(C(=O)NC2C(NC(C(CC)Nc3ccccc3)=O)C2)cc(C)c(C)cc1C N1(C(c2ccnc(C)c2O)=O)CCC(C2(NC(=O)CS(N)(=O)=O)CC2)C1 c1(C(=O)NC2C3CC(NC(CCC(CC)OC)=O)CC32)ccc2c(c1)OCO2 N1(C(c2c(=N)cc[nH]c2)=O)CCC2CN(C(=O)CC3=NNC(=O)C3)CCC2C1 CCC(C)CC(C(=O)N(C)Cc1scnc1C)NC(=O)CCCC1CC1 c1(C(C(=O)NCC2(NC(C3C(C(N)=O)C3)=O)CCCC2)(F)F)cc(F)ccc1F c1(C2C(NC(C(C)OCC=C)=O)C2)ncnc2c1cnn2-c1ccccn1 c1(C(=O)NC(CC)CNC(=O)C(c2ccc(F)c(Cl)c2)C)cccc2c1OCC2 c1(C(=O)NCCN(C(c2c(C)ccc(F)c2N)=O)C)c(F)ccc2ccncc12 Cc1cc2cccc(C(N3CCN(C)C(CN(C)C)C3)C(=O)NCC3CC3)c2o1 S(=O)(=O)(c1cc(C)c(-c2ccno2)cc1C)N1CC(COC)OCC1 c1(C(N2CCC3CN(C(CNC(CCC)=O)=O)CC32)=O)cc2cc(F)ccc2o1 CCCC(CCC)CC(=O)NCC(C1(O)CN(C(c2coc(CC)n2)=O)C1)(C)C C1(CNC(CCOCC(C)C)=O)COCCN(C(C2CN3CCC2CC3)=O)C1 S(=O)(=O)(c1ccc(C#N)c(NCC2CCC3CCCC3O2)c1)N(C1CCCC1)C C1(C(N(CCCC(=O)NC(CC#C)C(=O)NC)C)=O)CC2(C1)CC(C)C2 N1(C(CC(C)C)=O)CCCC1(C)C(=O)N(CCCNC(C1CCCCC1O)=O)C c1(C(N2CC(F)CC(NC(C(C)=C3CC3)=O)C2)=O)cccc(C2=CCOCC2)c1 C(=O)(C(C)S(C)(=O)=O)N(C1CCCN(C(C2CCC(=C)CC2)=O)C1)C C1(NC(CNS(NC)(=O)=O)=O)CC(O)CN(C(c2nc(C(F)(F)F)sc2C)=O)C1 c1(C(=O)OC)ccnc(C(=O)NC2CCC(NC(=O)CC3COCC3O)CC2)c1 C12(C(N(C(CC)CC)C3CC3)=O)CC(C)(CN1C(c1ccc(Cl)cn1)=O)C2 CC1(c2cn(CC3C4CCCC34)nn2)CCCN1C(=O)CC(Br)Br C1(C#N)(C(=O)NCC2(CO)CCN(C(c3ccc(CC)s3)=O)C2)CC12CCCC2 N1(C(c2c(C)c(N)cnc2)=O)CCC(NC(=O)CC2CNC(=O)C2)C(C)(C)C1 N1(C(C(n2ccc(C)n2)C)=O)CCC2(CCN(C(c3conc3C)=O)CC2)C1 N(C1CN(C(c2ccoc2)=O)Cc2ccccc21)C(C1CCc2ncnn2C1)=O c1(C(=O)NC(C(=O)OC)CC2CCCCC2)cccc(-c2cn[nH]c2)n1 S(=O)(=O)(c1cccc(NCC2CCCC(=O)C2)c1)NC(CC(C)C)C N1(C(CC2C(C)C2)=O)CCCC(C)(CNC(=O)CC(C)(C)C)C1 Cc1ccc(C=CC(=O)NCC(C)N(C)C(C2(C)CCCS2(=O)=O)=O)nc1 C1(CNC(c2cn(CC(F)F)cn2)=O)CC(O)CN1C(=O)COCC1CCCC1 N1(C(CN(CCC)C)=O)CC2CC1CN2C(c1cncc(SC)c1)=O C#CCCCCC(=O)NCC1CCCN(C(C2CC3(CC3)CO2)=O)CC1 c1(C(=O)NCCCCCNC(C23CCC(OC)C2CC3)=O)c(N)ccc(C)c1F CC(CC(=O)N1CCC(CNC(=O)Cc2cn(C)nn2)C12CC2)P(C)(C)=O C12CCCN(C1)C(=O)C(C(=O)OC)N2C(C)=O.c1(C2(CC)COC2)cccnc1 Cc1nc2c(s1)CCCC2CN(CCO)C(=O)Nc1nc2n(c1Br)CCC2 C(=O)(CC(C)N(C(=O)CCc1cc(C)on1)C)NC(C#C)CC1CC1 N1(C(c2n(CC)nnc2C)=O)CC(C)C(NC(c2cc(F)c[nH]2)=O)C(C)C1 c1(C(N2CC(CCNC(C3ON=C(C)C3)=O)OCC2)=O)ccc2cc[nH]c2c1F N1(C(CN(CCOC)C(c2cccc(OC)n2)=O)=O)CC(C)OCCC1C C(CCCC(=O)N1CCC(c2nnc(Br)n2C)CC1)N(C(C)=O)C C1(NC(CCC(CC)C)=O)CC2CCC1CC2NC(c1c(CC)cccc1N)=O N1(C(C(C)(C)OCC)=O)CCC2(CCC(NC(c3ccc(C)n3C)=O)C2)CC1 C(=O)(C#CC1CCC1)N1CC(NC(CCCc2ccc(CC)cc2)=O)C(OC)C1 N1(C(C=CCCC=C(C)C)=O)CC2CCC2(NC(c2cc(C#N)c[nH]2)=O)C1 c1(NC(C2CCCN(C(c3cc(O)ncn3)=O)C2)=O)cnncc1Br C#CCCCCC(=O)N1CC(F)CC1CNC(C1OCCOC1C)=O c1(C(N2CCC(C(CNC(c3ccn(C)n3)=O)F)CC2)=O)c(F)ccc(F)c1F C=CCCC(C)C(C(=O)NCC1CC2CC(OC)C2C1)N1CC2CCCCC12 c1(C(N2C(CNC(c3conc3C3CCC3)=O)CC2)=O)cccc2c[nH]nc12 N1(C(C2N(C(C=CC(C)(C)SC)=O)CC(=O)NC2)=O)CC(C)(C)OC(C)(C)C1 C1(C(N2CC(C)(NC(CN3CCC(C)(C)C3)=O)C2)=O)CCC2C(C1)C2(F)F C(=O)(C1OC(C)Cc2ccccc21)NCc1c(C)cccc1Br C1(C(F)(F)F)(C(N2CCC(CN(C)C(c3nn(C)cc3Cl)=O)C2)=O)CCOCC1 N1(C(c2c(OC)c(F)ncc2)=O)CC2CCCC(NC(c3cc(C)cs3)=O)C2C1 C1(C#N)(C(=O)NC2C(N(C(COCCOC)=O)C)CCCC2)CC12CCCC2 C1(NC(CCn2cc(COCP(C)(C)=O)nn2)=O)CC2CC(C1)CC(F)(F)C2 C1(NC(c2nnn(C(C)(C)C)n2)=O)CC2(C1)CN(C(C1(C3CC3)CC=CC1)=O)C2 C1(NC(C(c2ccc(-c3nn[nH]n3)cc2)C)=O)CCCC(C(N)=O)C1 C1(CC(=O)NC2(CNC(C3C(C)(C)C3)=O)CCCC2)CCCC(C)(C)O1 c1(CC)cc(Br)c(C(C(=O)Nc2ccccc2)N(CC(Cl)Cl)C)s1 N1(C(C(CCC)NC(C)=O)=O)CCC(CC(N)=O)(NC(=O)CCCCF)CC1 c1(C(=O)OC)ccc2c(SCc3cccc(NCC4CCCO4)c3)csc2c1 C=C(Cl)C(C)(C)C(=O)NC1CN(C(C2(F)CC2c2ccccc2)=O)CC1C C1(CNC(C(C2CCCC2)OC)=O)CN(C(c2cc(O)ccc2F)=O)C(C)(C)C1 c1(C(N2CCS(=N)(=O)C(C)C2)C(=O)NCC=C)cc(OC(F)F)c(OC)cc1Br c1(C(=O)NCC2CC(F)CN2C(C2CC23CCC3)=O)nccn2nccc12 N1(C(CSCC(C)C)=O)CCC2CN(C(=O)Cn3nnnc3C3CC3)CC2C1 c1(C(=O)NC(CCN(C(=O)CCC(N)=O)C)C(C)(C)C)cccc(N=[N+]=[N-])c1 N1(C(COCCOCC)=O)CC(OC)CC(NC(=O)CN2CCCC2=O)C1 c1(C(N2CCC(NC(Cc3ncc(C)s3)=O)CC2C)=O)occ2c1CCOC2 CC(CCC(=O)NOCCOCCF)C1=CC2CCC1C2 c1(NC(=O)C(C2CCC2)OC)cc(F)ccc1OC.C12(COC)CCN(C1)C2=O C#Cc1ccc(C(N2CC(NC(c3ccc(Cl)nc3N)=O)CCC2C)=O)cc1 c1(C(=O)NCCCC(C)NC(Cc2c(C)cco2)=O)ccn(C)c(=O)c1O N1(C(C2CCN(CC(C)C)C2)=O)CCCC(CN(C)C(c2ccns2)=O)C1 C1(=O)C(C(C)(C)C)N1.c1(OC)cnnc(C(=O)NCC(F)C(C)(C)O)c1 C=C(Cl)CC(C(=O)N1CC(C#N)C1)NC(=O)CCC(=O)NCC C#Cc1ccc(F)c(C(=O)NCC(CC(F)(F)F)NC(C2CC(C(F)F)C2)=O)c1 C1(NC(n2cnnn2)=O)CCN(C(=O)Cc2cncnc2)CCC1(F)F CCCCCC(CNC(=O)Cc1ncc(C)s1)NC(=O)CN1CCCC1=O C(c1cccc(F)c1Cl)=CC(N1C2C(NC(CC(C)C3CCCO3)=O)C(C2)C1)=O c1(C(=O)NCC(CC)NC(=O)C=C2CN3CCC2CC3)cnc(O)c(C)c1 C(=O)(CCCCOCC1CCCC(C)O1)OC N1(C(C2CC(OC)CN2C(c2cc(C#N)cs2)=O)=O)CCCC(C)(O)C1 C1(CC(=O)NCC(CC)(CC)NC(=O)C(C)CSC)CC2CCC(C1)N2C C1(O)(C(=O)OC)CCCN(C(C2COC(C)C2)C(=O)NCCCF)C1 c1(-c2c(C(N3CC(NC(=O)CN4CC5CC5C4)C3)=O)c[nH]n2)cccc(Br)c1 c1(OC2CCCC(NC(=O)OCC)C2)ccc(F)c(C(C)(C)F)c1 Cc1cc(CCC(=O)NCC2CC(F)(CNC(=O)C(C)(O)C3CC3)C2)no1 N1(C(C2(CC)CC2(F)F)=O)CC2(C1)CN(C(c1cccnc1C1CC1)=O)CCO2 c1(CC(=O)NC(C2CCCCC2)CNCCCC(=O)NC)ccccc1[N+](=O)[O-] c1(CC)nncn1NC(=O)C1CC(NC(c2ccc(C)cc2O)=O)C1(C)C O=C(C1=C(Cl)CCCC1)NCC1(F)CCC(NC(=O)C=C2CN3CCC2CC3)C1 c1(OC)ccc(Cl)cc1C(=O)NCCC1CCN(C(c2cc(O)nc(O)n2)=O)C1 C(=O)(C1=CC2CCC=CCCC12)N(C(C)CCNC(=O)CCc1ncccn1)C CCC(CC(C)C)C(=O)NCc1nc(C(=O)N(C2CSC2)C)c(C)o1 C1(NC(C(C)CCO)=O)CC2(CCCN(C(C3CCS(=O)(=O)C3(C)C)=O)C2)C1 c1(C(=O)NC2C(F)CCN(C(CC3C(=O)NC(=O)N3)=O)C2)ccc2nc[nH]c2c1 c1(C(=O)NC2CCCN(C(CCc3n(C)ccc3)=O)C2)scc2c1OCCO2 CC1CN(C(=O)CCC2CC2(C)C)CCC1NC(C1CCC(N(C)C)CC1)=O N1(C(C(C(C)C)(C)C)=O)CC2(NC(c3cccc(O)c3Cl)=O)CCCC2(F)C1 c1(NC(Cn2[nH]c(=N)c(Br)c2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 c1(C(=O)NCCC(C)CCNC(=O)C=CS(C)=O)cc(N)cc2c1OCCO2 C(CNC(=NCc1ccccc1)NCC1CN(CC)C(=O)O1)(C(F)(F)F)OCC c1(CCC)cc(C(=O)NCC2CCCN2c2nc(COC)ns2)nn1C N12CC(C(C)(C)C1)C(=O)NOCC2=O.C1(C(=O)N(C)C)(OC)CCOCC1 c1(NCC(N2CCN(C(C=CSC)=O)C3C2C3)=O)ccccc1[N+](=O)[O-] C1(NC(C2(CCC)CC(=O)C2)=O)CC(C)CN(C(C2CC(=O)NC(=O)N2)=O)C1 C1(c2ccccc2)(NC(c2csc(C#N)c2)C)CCN(CC2SC(=N)NC2=O)C1 c1(C(=O)NC2(C)CCN(C(c3cccc(O)c3F)=O)C2)cccc(Br)c1F N1(Cc2c(C)noc2C)CC2COCC2(C(=O)N(C2CC2)Cc2nc(O)n[nH]2)C1 C1(OCC(=O)NCC(O)CNC(c2cn(C(F)(F)CO)nn2)=O)CCOCC1 CC(C)C(C(=O)NC(C1CCCN1C(c1cc[nH]n1)=O)(C)C)n1ccnc1 c1(Cc2n(CC(=C)C)c(N3CCC(C)OC(C)C3)nn2)nc2ccc(O)cc2o1 C1(CC(=O)NCc2cc(OC)no2)CCCCN1C(c1cn(C2CC2)cn1)=O C1(N(C(CCOCC(C)C)=O)C)CCCC(NC(c2cc(CO)[nH]n2)=O)C1 N1(C(C(CC)C(C)C)=O)C(CNC(c2cc(F)n(C)n2)=O)CC2COCC12 C1(NC(CSC(C)C)=O)C2CCCC1CC(NC(C1CCCCS1)=O)C2 N1(C(C=Cc2c(C)ncs2)=O)C2CCC1CC(CNC(=O)CCc1nc[nH]n1)C2 C(=O)(CCCCCCN=[N+]=[N-])NC1C(C)CN(C(c2c(Cl)cccc2Cl)=O)CC1 O=C(C#CC1CCCCC1)NC1(CNC(=O)CC2CCOC2)CCC(F)(F)CC1 c1(C(N2CCC(C3(C)CC3)C2)C(=O)NC(CC)C)cc(Cl)c2c(c1)OCCO2 c1(OC(C)C)ccc(NC(=O)NC(c2ccc(Cl)cc2)CC2CC2)cc1 C1(F)(C(N2C(C(=O)NCC)CCC2)=O)CCCN(C(=O)C(C)c2ccco2)C1 C1(NC(c2cn(CC=C)nc2)=O)CN(C(c2ccc(C)n2C)=O)CC1C1CC1 c1(OC)cc(C(N2CCCC2C(C)NC(=O)C(n2nc(C)cc2C)C)=O)ncn1 N1(C(c2c(C)nccc2)=O)CC2CCN(Cc3cc4ccccc4s3)CC2C1 c1(C(=O)NC(C)C=CC(=O)NCC(F)(F)CO)ncncc1Cl c1(C(N2C(CCc3cn(CCOC)nn3)CCC2)=O)ccc(O)c(CO)c1 c1(CC)ccc(C(=O)NCCOC2CCN(C(=O)C=CCO)C2)cc1 CCC1=NOC(C(=O)NC2CCC(CC3CC3CC(C3(CC)COC3)=O)CC2)C1 C(=O)(C1=C(C#N)CCC1)N1CC(C)(CCC(=O)N2CC(N3CCC3)C2)C1 C1(C)(NC(CC2CCCC(C)C2)=O)CCN(C(c2cc(C3CC3)ccn2)=O)CC1 c1(CC(=O)OC(c2ncc[nH]2)C)cccc(NCCN2CCCCCC2)c1 C#CCCC(C(=O)NCc1ccc(C)c(O)c1)NC(C1CCNC1=O)=O C1(OC)CC(NC(C2CN3CCN2CC3)=O)CN(C(c2nccc(Cl)c2F)=O)C1 c1(C(=O)NCCN(C(=O)C=Cc2ccco2)C2CC2)cc2n(n1)CCNS2(=O)=O C1(CNC(CC(C)(C)OC)=O)CN(C(=O)C2=COCCC2)CCC1C(F)(F)F C(C1=CCN(C(C2CC(C#N)C2)=O)CC1)NC(c1c(OC)scc1)=O Cc1nn(C)cc1C(O)C(=O)N(C)CC1CCCN(C(=O)CC(F)(F)C2CC2)C1 CC(C)CCC(C)(C1CC1)NC(C)(C)C.C(C(C)(C)OCCO)NC(=O)NCC N1(C(c2n(C)c(Cl)cn2)=O)CCC2CN(C(c3cc(=O)n(C)cn3)=O)CC12 C(=O)(CCC(C(C)C)NC(c1cccc2occc12)=O)Nc1c(C)cccc1 C1(NC(c2c(C)noc2)=O)CCN(CC(=O)NCC2CCCC2)CC1C CC1CCCC(CNC(C2(NC(c3nccnc3N)=O)CSC2)=O)O1 C1(COC)(CNC(c2nc(Cl)sc2C)=O)CCCN1C(=O)C#CC(=O)N(C)C O=C1C(C(=O)NC2CN(S(=O)(=O)c3ccccc3OC(F)F)C2)c2cc(Br)ccc2N1 c1(C(N2CCC(C)(N(C)CC)C2)C(=O)NCCCSC)ccc(N=[N+]=[N-])cc1 C1(C(N(CCO)CC)=O)CN(C(=O)CCc2cccc(Cl)c2)CCO1 C1(CC(=O)NC2(COC)CC=CC2)C=NN(C)C1=O.C12CC1C(C)NC2=O C#CCCC(C(=O)N1CC2CC1C2)NC(=O)C(F)C(C)C O=C1CCCCC(C(=O)NCC2CC(NC(c3occ4c3CCC4)=O)C2)N1 Cc1ccc(N)cc1C(N1CC(N(C(=O)CCn2cnnn2)C)C(F)C1)=O C(=O)(CCCS(N)(=O)=O)NCC1C(CNC(c2c(N)cc(F)cn2)=O)C1 CN1CCCC1C=CC(=O)NCC1CC1NC(c1coc(Cl)c1)=O c1(CC(=O)NCCC(C)NC(c2cncc3nc[nH]c23)=O)cc(F)c(F)cc1F C12(O)CCN(CC1)NCc1c(cccc1)C(CC)NC2=O.c1(SC)cccnc1 c1(C(N(C2CCCC(N(C(CC(=O)OC)=O)C)C2)C)=O)ncn2c1CCCC2 N1CC(C)CCC1CNC(=O)CC(CC)CC.n1(CCCC)nccc1C=O C(=O)(C#CC1CCCOC1)NC(CNC(c1c(=O)cc(C)n(C)c1)=O)C CCCCCCC(=O)N1CCCC(C)(CNC(C2CN(C)CCO2)=O)C1 n1(C(C)C)ccc2cc(C(N3CCCC(CCNC(C4CCC4)=O)C3)=O)ccc12 c1(C(N2CC3CC2CN3C(=O)C(Cl)(Cl)Cl)=O)ccc2nc[nH]c2n1 N1(C(C(C(CC)C)O)=O)CCC(C)N(C(=O)Cc2cc(C3CC3)no2)CC1 c1(C(c2nnnn2N)C(C2CCOC2)C2CC(=CC)C2)csc(Cl)c1Cl.FC=CBr C12(CNC(C3(S(N)(=O)=O)CC3)=O)CCCC1CN(C(=O)Cc1ccc(O)nc1)C2 c1(C(=O)NCCN(C(=O)CSc2ccccc2)C)cc(F)c(F)cc1N N1(C(c2c[nH]c(=N)s2)=O)CC2=C(C1)CN(C(C1CCc3cncn3C1)=O)C2 C(=O)(C(CC)C(C)(C)CC)NCC(=C)CCNC(=O)Cc1nc[nH]n1 c1(C(=O)NCCCCCCNC(C(C=CCCC)O)=O)c(C)cccc1Cl C12(NC(C=C3CCC(C)C3)=O)CCCCC1N(C(=O)C(C)SC(F)(F)F)CC2 CN1CCN(C(=O)CSc2cn[nH]c2)C(C(N2CC(F)(C#N)C2)=O)C1 N1(C(C2CCC3(C(C)(C)C)C2C3)=O)CCCCCC1CNC(=O)Cn1cncn1 N1(C(c2c(F)cc(OCF)cc2Cl)c2n(C)nnn2)CCS(=O)(=O)N2CCCCC12 c1(NC(=O)NCC(N2CCC(C)CC2)C(C)C)ccc(=O)n(CC(F)(F)F)c1 S(=O)(=O)(c1cc(C(=O)OCC)ccc1F)NC(CC#C)C(=O)OC(C)(C)C C1(C)(CNC(=O)NC(c2c(C)noc2C)CC)CC2CC2C1 Cc1c(C(N2CCC(C)(CNC(C3CCCS3)=O)C2)=O)csc1Br c1(CC)cccc(NC(C2(CNC(=O)CN3CCC(C)(C)C3)CC=CC2)=O)c1 C1(C(N2C(CC)CN(C(=O)CCS(=O)(=O)NC)CC2)=O)CN2CCC1(C)CC2 C1(C(=O)NCC(COC)O)CCC(NC(=O)C=CC(C)C)CC1 c1(C(=O)OCC)nc(C(=O)N(C)CCNC(c2cnc(C(C)(F)F)s2)=O)c(C)s1 C1(C)(C(=O)NCC(CNC(=O)CCSC)OC)Cc2ccc(C)cc2C(=O)O1 c1(NC(C(C)=C(CC)C)=O)cnn(C)c1-c1ncc[nH]1 c1(C(=O)NCC(C)N(C(=O)C2=COCCC2)C)ccc2nc[nH]c2c1F C(=O)(C(CC(N)=O)NC(=O)C=Cc1cc[nH]c1)N(C)CCN1CCCC1 c1(-c2cc(NC)c(F)cc2)cc(C(N2CC3CN(C)CC3C2)=O)cc2[nH]ncc12 CCC(CC(C)C)C(=O)N1CC(NC(=O)Cn2ncnn2)C2(CCC2)C1 N1(C(=O)C=Cc2ccncc2)CCC=C(C(=O)N2CCC3CC23)C1 C(=O)(C(=O)N=c1[nH]n(C(C)C)cc1C)c1ccc(CCCCC)cc1 C1(C(=O)NC(C(N2CC(C)(OC)C2)=O)(C)C)CCCOC1C C(CC)(CCC)(c1n(CCSC)nnn1)NCc1sccc1C c1(C(N2CCC(N(C(c3cncc(COC)c3)=O)C)C2)=O)cnc(Cl)cc1N C1(CNC(CC=C)=O)CC2(CCN(C(=O)C(c3ccc(C)cn3)(F)F)CC2)CO1 CCCC(C(=O)N(CCCNC(C1(CO)CCOC1)=O)C1CC1)OC c1(C(=O)NCCN(C(C2(C#N)CC3CC3C2)=O)CC)ccc2sc(O)nc2c1 c1(N2CC3N(C(C(C=C)(C)C)=O)C(CC3)CC2)ncnc2sc([N+](=O)[O-])cc12 N1(C(COCC(=C)C)=O)CCC2CN(C(=O)Cc3cn4ccsc4n3)CC2C1 c1(CC(C)C)nc(C(=O)NCC2CCC2C)cs1 C1(NC(c2ccc(OC)nc2)=O)CC2CC(C1)CN(C(C1CCSC1)=O)C2 c1(C(=O)NC23CC2CN(C(c2cc(F)n[nH]2)=O)C3)c[nH]c2cccc(Br)c12 C1(CNC(C(=O)N(C(C)C)CC2CCCO2)=O)CC(C)(C)C1 C(=O)(C(CNC(C1CNC(=O)N1)=O)CC(C)C)Nc1cccc(C)c1 C1(CNC(C23CCC(OC)C2C3)=O)(CO)CCN(C(=O)C=Cc2c[nH]cn2)CC1 C(C)(C(C)C(=O)NCC(C)(Cl)CC)NC(C(C)(C)OCCC)=O C12(C(=O)NCC(C)N(C)C(c3cc(-c4ccco4)on3)=O)CC(C1)C(C)(C)O2 C(=O)(CCCS(N)(=O)=O)NC(C1(O)CN(C(c2cc(O)cc(N)c2Cl)=O)C1)C N1(C(CC(C)F)=O)CC2C(CN(C(=O)Cn3nnnc3C3CC3)C)C2C1 c1(C(N2CC(CC)(NC(=O)CCc3ccccn3)C2)=O)ccc(=O)oc1 C(=O)(C1=NOC(C)C1)N(C1CC(C(N2C(C)(CC)CC2)=O)C1)C C(CCCC(CO)NC(c1ccnc(C(N)=O)c1)=O)NC(CCC=CCC=C)=O N1(C(CC(CC)OC)=O)CC2(CCCC2)C1C(=O)NC(c1snnc1C)C C=CC1(C(=O)Nc2cnsc2)CCN(C(C2CC(F)C(=O)N2)=O)C1 C1(NC(C2CCCO2)=O)CN(C(c2cc(Cl)no2)=O)CC2(CCC2)C1 c1(C(N2C(C)(C(=O)Nc3cnc(C)nc3)CCC2)=O)cc(F)c(Br)c(F)c1 c1(-c2c(C(=O)NCCC(C)NC(C3C(C(=O)OC)C3)=O)c[nH]n2)cccc(Cl)c1 n1(CC)nc(C)c(S(=O)(=O)NCCn2ccc(C(=O)NC)n2)c1C C1(O)(CCNC(C=CC)=O)CCCN(C(c2ncc(C(F)(F)F)cc2O)=O)C1 C(=O)(C1CCCc2nc[nH]c21)N1CC(NC(c2nc(CC)sc2)=O)C(C)C1 N(C1c2ccccc2CC1NC1CCC2C=CC12)C(=O)OC(C)(C)C c1(CC)ccc(OC)cc1.C1(NC(C2(CC)CC2)=O)CC(C)(OC)C(C)NC1=O.SC c1(C(=O)NCC2(F)CC(NC(c3nc(CCC)oc3)=O)C2)cccc(O)n1 C1(CCC)CN(C(=O)C(C)CCC)CCN1C(=O)CSC(=N)N N1(C(C2(COC)CC=CC2)=O)CC2(COC(CNC(=O)C3=C(Cl)CC3)C2)C1 c1(CC(=O)NCC2C(C)CCCN2C(C2CCOC2)=O)ccc2nonc2c1 c1(C(=O)NC)ccc(F)c(CN2CCOCC(CCCO)C2)c1 n1(CCCC)ncc(C(=O)N(C)CCN(C(=O)C(COC)NC(C)=O)C)c1CC C(CC1CC1)(C(=O)NCCOCC1CCOC1=O)NC(=O)CC1CCC1 N1(C(C(CC)OCC)=O)CC=C(CCNC(=O)C2=NOC(C)C2C)CC1 C1(NC(C)CCN2CCN(C(C)(C)C)CC2)CCCN(C(=O)OC(C)(C)C)C1C C1(CC(=O)NCCC(CNC(c2cccc(OC)n2)=O)O)CCOC(C)(C)C1 C1(C(=O)NCCN(C(=O)CC2OC(C)(C)OC2=O)C(C)C)CC2(CCCCC2)C1 N1(C(C23OCCC(C)(C2)C3)=O)CCC2(NC(=O)C=Cc3cc[nH]n3)CCCC12 C#Cc1cnc(O)nc1NC(=O)C(=O)Nc1ccc(CCF)cc1 C1(C(=O)NCC2CCC(NC(=O)C=Cc3ccncn3)CC2)(OC)CCCOC1 c1(-c2nc(OC)sn2)cccc2nc(C(N3CCC(N(C)C)CC3)=O)cn12 c1(CC(=O)NCC2CCN(C(COCCC(C)C)=O)C2)ccc2nsnc2c1 c1(C(=O)NC2(CN(C)C(C3CCCC(F)C3)=O)CC2)cc2ncccn2n1 CC1CCCCC1(CNC(C12COC(CCO1)C2)=O)NC(=O)CC(C)(C)C c1(C(C)NC(=O)NC(C(=O)NCC(CC)OC)C(C)(C)C)c(Cl)ccc(F)c1C c1(SC)nn(C)cc1-c1noc(CC(c2cccc(Cl)c2)(C)C)n1 c1(C(N(C2CN(C(c3c(CC)cno3)=O)CC2F)C)=O)cc2ncccn2n1 c12cccc(c1)NC2=O.C(C)(CCn1cccn1)OC(C1C(C)C1)=O C(=O)(C(C(C)C)n1cncn1)N(CCNC(CC1(OC)COC1)=O)CCOC(C)=O c1(C(N2C(C)CC(Nc3ncc(C(=O)OC)nc3)C2)=O)cc(O)cc(O)n1 C1(C(=O)NCCN2CC3CC3C2)CCN(C(=O)CC2CCCO2)CC1 Cc1ccc(C(C(=O)NC2CC2)N(C(C)CC#N)C)cc1OC(F)F C1(CC)CN(C(=O)CCc2cc(Cl)cs2)CCC1NC(=O)C(C)n1cccc1 N1(C(c2c(C)nc(C)o2)=O)CCN(C(c2ccccc2)=O)C2CC12.C1C(=O)O1 Cc1ccc(Cl)c(O)c1C(N1CC(CCNC(c2ccc(C3CC3)cc2)=O)C1)=O N1(C(CCOCCOCC)=O)CC2CC(NC(=O)CCC3CC3)CC1C2 c12noc(n1)C1CCCN1N(CC(C)C)C2C1CC1.C(C(=O)OCCl)CC.C(C)(C)C C1(CNC(C(F)=CC)=O)C(C)CCCN1C(=O)CNC(c1ccoc1)=O C1(C)(NC(CN(CCC)C)=O)CCCCC1C(=O)NCCCN(CC(C)C)C c1(C(N(C)CC2CCCC(NC(CC=C(C)C)=O)C2)=O)ccc([N+](=O)[O-])c(N)n1 N1(C(C(=O)NC)=O)CC(NC(=O)COc2ccccc2C(C)(C)C)CC1C C(C)(C)(CCC(=O)NCC(c1ccccc1)CNC(=O)C(O)P(C)(C)=O)N(C)C c1(OC)coc(C(=O)NC2CCN(C(c3ncc(F)cn3)=O)C(C)C2)cc1=O C=CC(C)(C)C(=O)NC(c1ccc(C)cc1)CNC(c1c(C)n[nH]c1C)=O C1(C(C)CNC(=O)CCC2CCCO2)CCN(C(=O)CCc2cn(C)nn2)CC1 C(=O)(C1=COCCC1)N(C1CCCN(C(c2nnn(COCC)c2N)=O)C1)C C(=O)(CCC(C)(C)C#N)N(C(C(CC)C)C(=O)NCCC(O)C(F)(F)F)C C(C)(CO)(C(=O)NCc1ccc(C(=O)NC2CCCC(O)C2)nc1)OC CC(C)CCC(C)(c1nnnn1C(C)C)NCCCS(C)(=O)=O C12(SCCOC(=O)C(N3CCCC34CCNC4=O)=O)COCCN1C(=O)OC2 C#CC(CNC(c1ccc(CNC(c2ccc(CC)o2)=O)o1)=O)CC1CC1 c1(C(=O)NC2C(CNC(C(C3CC3)SC)=O)COC2)cc2sccc2[nH]1 N1(C(c2c(CC)nn(C)c2)=O)CCC(CO)C(NC(c2c(C)noc2CC)=O)C1 C(=O)(C1=NOC(C)C1)NC(CNC(Cc1c(CC)noc1CC)=O)C(C)(C)C N1(C(C(C(=O)OC)OC)=O)CCOCCC1C(=O)NCC1CN(C(C)C)C1 C1(CNC(C)=O)CCN(Cc2cnn(-c3ccc(F)cc3)c2)CC1 c1(C2CN(C(C3Cc4nccn4C3)=O)C2)cc2ccccc2s1 C(=O)(C1=CCCC(C)(C)C1)N1CC(O)(C(C)NC(c2cn(CCC=C)nn2)=O)C1 Cc1nc2nc(C)ccc2c(=O)n1CCCC(N1CC(O)CC1(C)CO)=O C1(O)(CNC(C2CCCO2)=O)CCCN(C(=O)Cc2cncc(O)c2)CC1 C1(C(N2CC(n3cc(C(CC)CC)nn3)C(C)C2)=O)Cc2cccc(F)c2C(=O)O1 N1(C(CCC)=O)CC2(CCC(C(=O)Nc3ccnc(OC(F)F)c3)O2)C1 C(=O)(C#CC(C)(C)C)N(C(C)CCNC(c1sccc1Cl)=O)C C(=O)(C1=NOC2COCC12)NCCCCC(C)NC(Cc1ncc(C)o1)=O N1(C(C=C(C)C(C)(C)C)=O)CC(C(=O)N(C)Cc2nnc(C)s2)CCC1(C)C N1(C(=O)C=Cc2ncco2)CC2(C1)CN(C(C1CCCCCC1)=O)C2 c1(C(=O)OC)cc(OC)cc(OC)c1Cl.N1C(NC2CC2C)=NCC12CC2 C(=O)(C(CC(F)F)NC(c1ncccc1N)=O)N1CC(CC(C)C)OCC1 C#Cc1cc(C(N2CC(CCNC(c3ccccc3C)=O)(OC)C2)=O)ccc1C C1(CC(=O)OC)CC2(CCOCC2)CN1C(=O)Cc1cccc2c1CCOC2 C1(OCCNC(C(C)c2ccsc2)=O)CCN(C(C2CC=CC2)=O)CC1 Cc1cc(C(=O)N(CCCCCNC(=O)CC(C)O)C)c2nc(C)n(C)c2n1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CC2(C1)CN(C(c1sccc1Cl)=O)CCO2 CCCC(F)C(=O)NCC(C)(C)OCC(=O)NC(c1nc[nH]n1)C C(=O)(CC(C)C(F)F)N1CCC(C(N(CC(F)F)CCOC)=O)CC1 Cc1c(C(N2CC(NC(C3CC34CC(C)(C)C4)=O)C(O)C2)=O)cncc1N c1(CCC(=O)NC(COC)CNC(=O)C(C)C2CCCC2)ccnc(C)n1 N1(C(CCCOCC=C)=O)CCN(C(c2cnn(CC(C)C)c2)=O)C(CF)C1 N1(C(C(=O)NCC)=O)CCCC2(C1)CN(C(=O)C(C)CN1CCCC1)C2 C(CC(C)(C)C)(C(=O)NCCC(C)N(C)C(c1cc(C#N)[nH]c1C)=O)OC C(c1nc(C)cs1)=CC(N1CC(C(C)(C)O)(CNC(CC(C)OC)=O)C1)=O CC(C)C(C(=O)N(CC(C)NC(C1(CF)CCC1)=O)C)SCc1ccccc1 c1(C(=O)NCC2CN(C(C)=O)C2)cc(Nc2cccc(C(C)C)c2)nc(C)c1 c1(C(N2C(CC(=O)NOCCN3CCOCC3)CCC2)=O)cccc(F)c1 Cn1cc(CNC(C23CC(F)C2C3)=O)c(C(F)F)n1 N#CC1CN(C(c2occc2CNC(=O)COc2ccsn2)=O)CC12CCC2 C1(CC)(CC)CCCN(C(=O)COC2CCN(C(C3CCCC(O)C3)=O)C2)C1 n1(C(C)C(=O)NC(C)CN(C)C(c2cnco2)=O)cnc2ccccc12 C1(CNC(C(c2ccccc2)OCC)=O)COCC1NC(=O)CSCC(N)=O C(C)(CO)(C(=O)NC1CCN(SC)CC1)C(C)NC(=O)OC(C)(C)C C1(C(N2CC(CCNC(C(N3CCC(C)C3)=O)=O)C2)=O)CN(C)C(=O)N1 C12(NC(CCCCC=C)=O)CCCCC1N(C(=O)C=Cc1ccnn1C)CC2 C(=O)(C(O)CCCNC(C1CCC2(CC1)CC2)=O)NC1C(c2n(C)ncc2)C1 Cc1nc(Cl)nc(N2CC3CC2CCC3NC(C2(C)CCS(=O)(=O)CC2)=O)c1F N1(C(C(CCC)C)=O)CCC(NC(=O)CCC2CCCN2C)C(CO)CC1 CCC(CC(=O)NC(C(=O)NCc1nc[nH]n1)C1CCC1)C(F)F C(=O)(CCCNC(=O)CCc1cn[nH]c1)N(c1ccncc1)C C(=O)(C(CC(C)C)C(C)C)NCC1CCCC(NC(CCc2cc(C)no2)=O)C1 c1(C(=O)NCC(CNC(C(CC=C)(C)CC)=O)OC)cc(C)c2occc2c1 c1(OC)nsc(OC)c1C=O.N1CCOC(CNc2cc(N)c(C(=O)O)s2)C1 N1(CC(=O)NC(C(=O)N(CCS(N)(=O)=O)C)CC2CC2)CCC(F)CC1 c1(C(=O)NC2CCN(C(C3CC3C3CC3)=O)CC2)cc(F)c(OCCF)c(F)c1 c1(C(=O)NCC(CC=C)NC(CC=C=C)=O)cc(F)c(Br)c(F)c1N c1(-c2n(C(C)C)nc(CCN(C)C3CC3)n2)cc(OCc2ccccc2)ncc1Cl c1(-n2cc(C3C(C(N(C)Cc4cccs4)=O)C3)nn2)cncc(Br)c1.C1(=O)CN1 C(=O)(C(C(C)(C)C)n1cc(-c2ccnn2C)nn1)N(C)Cc1cnnn1C C1(NC(C2CCN(CC)C2)=O)CC2CCC(C1)N2C(c1cc(C)c(F)cc1O)=O C(C(C)(C)CC(=O)N1CCC(NC(=O)COC(C)C)C2CC12)OC c1(OC)ccc(Br)cc1CCN=C(NCCc1ccccc1C)NCC(F)F c1(SCC(C=C)C(C)C)nc(Cl)c(C)cc1F N12CCN(CC1)C(=O)C1(CC1)C2.C1(C(=O)OC)CC1OC(C)(C)C Cc1nn(C)cc1C(N1CC(F)CC1C(=O)Nc1cn(C)nc1-c1ccoc1)=O Cn1ncc2c3nc(nc12)N1CCC2(CC1)NC(=O)C(C2)N3CCOCC(C)CO c1(C(N2CCC(C3N(C(C4C(C)C4)=O)CCC3)C2)=O)nn2c(c1Br)OCCC2 C1(CC)CN(C(=O)C(C2CCCO2)NC(c2cn(C(C)C)nn2)=O)CC(=O)N1 c1(OC)ccc(CC(N2CCCC3CN(C(=O)C(F)CC)CC23)=O)cc1[N+](=O)[O-] N1(C(c2ccsn2)=O)CC2CC1C2C(=O)N(CCCF)C1CC1 C1(CCC)CN(C(C2(C)CCCCO2)=O)CCN1C(=O)CCN1CCCCC1=O C1(NC(=O)Cc2cccc(Br)c2)COCCN(C(C2(C3CC3)CCC2)=O)C1 c1(OC)cc(C(=O)NCC(C)NC(=O)Cc2ccc(Cl)nc2)c2ccccc2n1 N1(C(CCC2CCN(C(C(CCOC)OC)=O)CC2)=O)CC(C(N)=O)CC(C)C1 N1(C(c2c(CC)nccn2)=O)CC(NC(=O)C=Cc2ccccc2)C2(CCC2)C1 c1(CN(CCOC)CCN2CC2)cc(C(=O)OC)cs1 c1(C(N(C(c2ccc(Br)s2)C(=O)OC)C)C)nc2ccccc2s1 O=C1CCC(C(=O)CC23CC(NC(=O)C(=O)NCC4CC4)(C2)C3)C(C(F)(F)F)C1 N1(C(c2c[nH]c(=N)o2)=O)CCc2ccc(C(F)(F)F)cc2C1 c1(-c2nc(NC(=O)CC3C=CS(=O)(=O)C3)sc2)cc(Br)c2c(c1)OCCO2 C1(CC(N2CCCC(OCC(N)=O)C2)=O)C2CCCC2N1C(c1cccnn1)=O c1(NCc2ccc(C)cc2C)cc(=NCCc2ccc(S(C)(=O)=O)s2)[nH]c(C)n1 C1(NC(C=CC)=O)CCN(C(C2CC2(COC)CC)=O)CC1C C(=O)(C1=CS(=O)CCC1)N(CC(CC)NC(c1ccn(CCC)n1)=O)C C(=O)(C(C)(F)C(C)(C)F)N1CCC(NC(COc2c(CC)cccc2)=O)CC1C CC(O)(CC(=O)NCCCCNC(=O)CCc1ccc(F)cc1)C1CC1 C1(C(C(=O)NC2C(CCCC)CCC2)C)CCN(C(c2cc[nH]n2)=O)CC1 C=CC(CCC)CC(=O)NCCCOCCNC(=O)CCC(=O)c1cnn(C)c1 C12(NC(c3c(C#C)c[nH]n3)=O)CC(CNC(C3CC4CCC3CC4)=O)(C1)OC2C c1(-c2cn(CCC)nc2)ncc(Cl)cc1C(=O)NC(C1CCC1)C CC(C)(C)CC(O)C(=O)N1CCCCC(NC(=O)CN2OC(C)(C)CC2=O)C1 C(=O)(C(C#N)=c1sc(=Cc2ncc(Cl)cn2)c(=O)n1C)NCCSCC C1(C(N2CCC(C(C(=O)NCc3ccc(CO)o3)F)C2)=O)CC2(CCC2=O)C1 CCC(CNC(=O)CCCc1cccc(Cl)c1)(CC)NC(c1ccnc(S)c1)=O C1(C(N2C(C(=O)Nc3ncccc3Br)CCC2)=O)CCCC2CCCCC12 N1(C(C2CCN(c3n(C)ccn3)C2)=O)CC2CC(NC(=O)C(C)(C)CF)C(C2)C1 c1(C(N2CCCC2CNC(=O)C(F)(Cl)c2ccccc2)=O)ccc([N+](=O)[O-])o1 C1(CNC(=O)CC2CCCN2C(C2(C(F)F)CC3(CC3)C2)=O)CCC2(CCC2)O1 C(C)(CN=c1cccc(S(=O)(=O)NCc2ncc(C)s2)[nH]1)OCC N1(C(CCC=C=C)=O)CC2CCCC1CN(C(=O)C=CC(C)(C)C)C2 N1(C(C(CC)C2CCOCC2)=O)CCC(NC(=O)CC2(C)CCCC2)CC1C C1(CNC(CC(CC)C)=O)CN(C(c2ccnc(C)c2)=O)CCC12CCC2 N1(C(CC(CC)OC)=O)CCC2C(C1)CN2C(C1(n2cccn2)CC1)=O O=C1CCC(CC(=O)NC2C3CCN(C(c4ccsc4Cl)=O)C23)CN1 C1(C)(NC(C2(CC)N(C(c3c(CC)nn[nH]3)=O)CC=C2)=O)CCC(=O)N(C)C1 C1(CCNC(=O)Nc2ncc(-c3ccccc3)s2)CCCCCC1 c1(OC)ccc(CCCN(C)C(=O)NC(C)C(C)(C)OC)cc1 CC(C)C(C#N)C(=O)N1CCC(C(N2CC(OC(F)F)C2)=O)C1(C)C c1(CC)ncoc1C(=O)NC(C(N1CCC(CN2CCCC2)C1)=O)C1CCCO1 c1(C(=O)OC)ccc(C)c(C(=O)NC(CNC(C2CCCS2(=O)=O)=O)C2CC2)c1 N#Cc1c(N2CC3CCCCNC3C2)nnc2c1OCCCC2 C12(CNC(c3cc(F)n[nH]3)=O)CCCC1N(C(C1CC=CC1)=O)CC2 CC(c1cccc(Br)c1)=CC(N1CCC(CNC(=O)C2CC2)C12CC2)=O N1(C(C2C(CCC)C2)=O)Cc2ccccc2C(NC(c2ccc(O)c(F)c2)=O)C1 [N-]=[N+]=NC1CN(C(C2(C(F)(F)F)CC2)=O)CC1NC(C1CC12CCOCC2)=O c1(C(N(C(C)CNC(C2CCN(C)C2)=O)CC)=O)sc(Br)cc1Cl c1(C(N(C2CC(NC(CC=C(C)C)=O)C2)C)=O)ccc(Br)cc1C#N C(=O)(CCCCCCCCn1cc(CO)nn1)N1C(C)(C(=O)OC)CC(F)(F)C1 CN1CC(n2cc(C3CCNC(=O)C3)nn2)CC1c1ccc(F)cc1 C1(C(=O)NC2CC3(CC(NC(c4cnccn4)=O)C3)C2)CCn2ccnc2C1 C1(C(=O)NCC(CO)NC(=O)CC(C)N2CCCC2=O)(COC)CCCCC1 Cc1cccc(C(N2CC(NC(c3ccccc3C(C)C)=O)C3CC23)=O)n1 c1(CCC(N2C(CNC(c3cc(CC)no3)=O)CC2)=O)ccc(C)c(C)c1 C(C1CN(C(C2CCC(=O)N2)=O)Cc2ccccc21)NC(CN(CCC#C)C)=O c1(C(=O)NC2CCCN(C(C3CC(C)(O)C3)=O)C2)c(F)cccc1Cl c1(OC)ccc(C(=O)NC2CN(C(=O)C(F)OC)CC2c2cnn(C)c2)cc1N N1(C(C2COC(=O)N2)=O)CCC(C)(NC(C(COCC)N(C)C)=O)CC1 c1(OC)cc(C(=O)NCC2(NC(c3cccnc3C)=O)CC2)c2c(c1)CCO2 C1(NC(c2scc(CC)n2)=O)CN(C(c2ccc(C#N)c(F)c2)=O)CCC1(F)F c1(C(=O)NC(C)C(C)NC(c2ccc(Cl)o2)=O)csc(C(F)F)n1 CCCCCCC(C)CC(=O)NCC1CN(c2ncncc2C#N)CCN1C Cc1cc(C)c(C(=O)NC2CC2CNC(c2ccc(C(F)(F)F)o2)=O)[nH]1 c1(C(=O)NC2C(C)(C)N(C(C3CCSC3)=O)CC2)nc2cccnc2s1 Cc1noc(C)c1C(C)(C)C(=O)NCC1(F)CN(C(=O)CCC#N)C1 CCCCC(C(=O)Nc1cnc(F)c(C)c1)NC(c1ncsc1NC)=O CC(C)(C#N)CC(=O)NC1CCCC1C(=O)NC1CC(C)(C)C12CC2 C1(O)(C(=O)NC2(CC=C)CCN(C(C3CC3CCOC)=O)C2)CCC(C)(C)CC1 C12(C(=O)NC(CC)(CNC(C3CC3(C)C(F)F)=O)CC)CCCN1CCC2 n1(CC)ncc(Cl)c1C(=O)N(C)CC1(CNC(=O)Cc2cccc(F)c2)CC1 CN1CC(C(=O)NC2(CNC(C3CCS3(=O)=O)=O)CCCC2)OCCC1=O C1(OC)COCCC1CC(=O)N(C1CCC1)CC1(OC=O)CC1.C1CCC1 C1(C(=O)NC(CC)CNC(=O)C(c2ccc(F)cc2)CO)Cc2ccccc2N1 N1(C(c2ccc(C#C)cn2)=O)CCC2(CCCN2C(c2nccnc2Cl)=O)C1 c1(C(N(C2(C(=O)NC(C)CCN3CCCC3)CC2)C)=O)cc(F)c[nH]1 C12(C(N3C4CCC3CC4)=O)CC(C)(C1)OC2C.c1(C(=O)OC)cc(Cl)ncc1F C12(CNC(C3C4CN(C(=O)CC5C=CCC5)CC34)=O)CCC(CC1O)C2 C(CCC(O)C(=O)NCCCc1nncs1)NC(c1c(C)ocn1)=O C1(NC(C(C)Oc2cccnc2)=O)CCC12CCN(C(C13CC(F)(C1)C3)=O)CC2 CC(C)C(C#N)C(=O)NCC1CN(C(C2CCC3CC3CC2)=O)C1 CC(C)(O)CC(=O)NCC1CCN(C(=O)Cc2ccc(OC(F)F)cn2)C1 N1(C(C(c2ccccc2)=O)=O)CCOCC(NC(c2sccc2SC(F)F)=O)C1 N1(C(CCC#C)=O)CC2CC1C2CNC(=O)CC1CCC1 c1(OC)cc(C(N2CCC(NC(c3n[nH]cc3Br)=O)C23CC3)=O)ccc1F C1(NC(CC)=O)CN(c2ncc(C#N)cc2C)CC(C)(C)C1 C1(C#N)(OC)CC(C(=O)N(CC(O)CN(C)C(c2cc(C(N)=O)[nH]n2)=O)C)C1 N1(C(Cc2ccc(CCC)cc2)=O)CC2CCC1C2S(C(C(=O)NCC)C)(C)CC N1(C(c2cnn(CC)c2C2CC2)=O)CCOC(C)(CNC(=O)C(C)(C)OC)C1 c1(NC(C(Cc2c(C)nc[nH]2)O)=O)cccc(F)c1 c1(C(=O)NC2C(NC(CNC(=O)OCC)=O)CCCCC2)cnc2occc2c1 c1(C(N(CCCCNC(C2(C)CCN(C)CC2)=O)C)=O)cc2cccnn2c1 c1(CC)ncc2c(n1)CCC(C(=O)NCC1CCN1C(=O)C(O)CSC)C2 c1(C(=O)NC2(CN(C(=O)C3=CC4CCCC34)C)CC2)ccc2c(n1)CCCC2 Cc1nccc(C(=O)NC(CCN(C(=O)CC(O)c2ccccc2)C)C(C)C)n1 C1(C)(NC(C2C(CC)OCC2)=O)CCN(C(=O)Cc2ccc(C)s2)CC1 C1(N(c2ccc(C)cc2)C(=O)NCCc2ccccc2)CCC(C2CC2)C1 C(C(CC)(CC)NC(c1cncn1C)=O)NC(C1C(CC)OCC1)=O C12(NC(C(C)C)=O)CCCCC1CN(C(=O)CC13COC(C)(C1)C3)C2 C1(CNC(C2(C(F)F)CC(=C)C2)=O)CN(C(c2cc(C)n(C3CC3)n2)=O)CCO1 c1(OC)nccc(C(N2CCC(OCCNC(C3CC34CCCC4)=O)C2)=O)c1F c1(OC)cnc(SC#N)[nH]c1=NC1CCC(CC(=O)ON2CCC(F)C2)CC1 C(=O)(C(C)(C)C(F)F)NCC1(N(C(CC(C=C)C)=O)C2CC2)CCOC1 C12(C(=O)NC3(CO)C(C)CCCC3)CCCC1N(C(c1ccccc1O)=O)CC2 N1(C(c2cnc(C(C)C)[nH]2)=O)CC(F)CC1CNC(c1cc(C(F)(F)F)on1)=O CCC(O)C(C)C(=O)NCCOC1CN(C(c2cc(C(F)(F)F)cs2)=O)C1 N1(C(C(CCN(C)C)NC(c2c(C)cccn2)=O)=O)CC(O)CC(O)C1 N1(C(c2c(COC)cccn2)=O)CCN(C(c2ccc(C(F)F)cn2)=O)C(C)C1 C1(NC(C2N(C)CCC2)=O)CC2CC(NC(c3sccc3CN(C)C)=O)C1C2 CC(C(=O)NOCCOCCO)N(C(=O)Cc1ccsc1)C N1(C(CC=CC)=O)CCC2(COC(CNC(=O)CS(=O)(=O)N(C)C)C2)C1 C1(COC)CC(CNC(=O)C(C)OC)N(C(c2cc(C(N)=O)co2)=O)C1 Cn1nccc1C(C(N1CC(O)(c2nn[nH]n2)C1)=O)NC(=O)CO C(CC(C)(C)CNC(=O)CC(CC1CC1)NC(C1(CO)CCCCO1)=O)OC N1(C(CC2C(C)CCO2)=O)CCN(C(=O)COCc2ccncc2)CC(C)(C)C1 N1(C(C2C(C=C)C2)=O)CCOC(CCNC(=O)CCC(C)N(C)C)C1 c1(CC(=O)NCC(CO)NC(CCOC)=O)csc(SCCN(C)C)n1 C(CC1CCCC1)(C(=O)NC1COCC1CO)NC(=O)Cn1cnnn1 c1(C(=O)NCCCN(C)C(c2cn(CC3(C)COC3)nn2)=O)ncnc2c1CCC2 c1(SC)cc(C(N2CC3C(CN(C)C(c4cccn4C)=O)C3C2)=O)c(C)o1 C1(CCC(=O)NCCN(C)C)CCCN(C(=O)Cn2cnnn2)C1 CCCCCC(O)CC(=O)N1CC(NC(=O)Cc2cccc(OC)c2)C(F)C1 c1(C(=O)NCC(CC)NC(C2(F)CCC(=O)CC2)=O)cn(C)c(C)cc1=O C(=O)(CCC(C)C(C(=O)NCCCSC)N1CCCC1C(=O)OC)OC c1(CC)ccc(S(=O)(=O)N(C2CN(C)CC2C)CC)cc1C(=O)OC Cc1nc(C(=O)NCC23CC2CN(C(C2C(CN=[N+]=[N-])C2(C)C)=O)C3)c(C)n1C c1(OC)cc(N)ccc1C(=O)NCC#CCNC(c1sccc1F)=O N1(C(c2cc(CC)on2)=O)CCC(CCC(=O)N(C(C)C(C)(C)O)C)CC1 [N-]=[N+]=NC1CCC(C(=O)OCc2cnnn2-c2ccccc2Br)CC1 CC1CCC(Cl)=C(C(=O)NCC2CC2NC(c2ccc(-c3ccccn3)s2)=O)C1 C1(C(C(=O)NC(c2cn(-c3ccccc3)nn2)C)O)CCOCC1 C1(C(=O)NCC=CCNC(C2CCC(=O)O2)=O)CS(=O)(=O)CC12CCC2 C1(C(=O)NCc2c(C(N(C)Cc3ncco3)=O)occ2)CC2(CC(=O)C2)C1 c1(N2CC(C)OC(C)C2)nc2ccc(Cl)cc2c(=NC2CC(CO)C2)[nH]1 C1(NC(C(CC(=C)C)NC(=O)CC(C)F)=O)C2CCN(CC2)C1C c1(C(N(CCOC)CCNC(C2C=CS(=O)(=O)C2)=O)=O)cc(F)ccc1C CC1(CCNC(C2CCC3CC23)=O)CCN(C(c2ccncc2F)=O)C1 Cc1cc(CNC(C(c2ccc(F)cc2)(C)C)c2nnnn2C)nnc1C c1(C(N2C(CNC(C(C)OCC)=O)CC3CC32)=O)ncc2c(F)cccn12 CCCCC(CC)CC(=O)N1CCCC1(C(=O)NCc1ncsc1C)CC C1(NC(c2c(C)ccnc2)=O)CN(C(=O)CCS(C)(=O)=O)CC2(CCC2)C1 N1(C(Cc2ncc(CC)s2)=O)CCC(C)C1c1cn(-c2ccccn2)nn1 c1(C(n2nccc2-c2nc(N3CCN(C)CC3)no2)C)cc(S(N)(=O)=O)cn1C c1(C(=O)NC2CCC(N(C(c3ccc(OC)s3)=O)C)C2)nc(C)c(C)[nH]c1=O C#CCC(O)C(=O)N(CCCNC(=O)C(C)=C1CC1)C1CC1 N1(C(c2c(C)nn[nH]2)=O)CCN(C)CC1CNC(C1CCCC(C)C1)=O c1(C(N2CCC(NC(C=C(C)C)=O)C(F)C2)=O)ccn2c1CSCC2 C#Cc1cc(C(=O)NC2CCCC2NC(C2CCC(C)(O)CC2)=O)ccc1Cl c1(OC)ccc(C)c(C(=O)NC(CNC(=O)C2=CCSC2)CO)c1 C1(C)(CNC(COC(CC)(C)C)=O)CN(C(C2CCCC(=O)N2C)=O)CC1C CCCC(O)C(=O)N1CCN(C2CCN(C(=O)CC3CCC3)C2)CC1 c1(CC)nnc(C)cc1C(N1CCC(C)C(NC(=O)CS(=O)(=O)NC)C1)=O c1(C(=O)NC(C(C)NC(c2onc(CC)c2C)=O)C)n[nH]c2cc(Cl)ccc12 C(=O)(C(C)(C)S(C)(=O)=O)NC(CC1CN(C(CC2C(C)=NOC2=O)=O)C1)C c1(C(N(CC(C)NC(C(CC)NC(C)=O)=O)CC)=O)cc(Cl)cnc1OC C(c1ccc(F)cc1F)=CC(N1CCCC(CNC(=O)CC2CC(F)C2)CC1)=O C(=O)(CC(C(C)(C)C)NC(=O)C=Cc1ccc[nH]1)NCc1ccc(C#C)cc1 N1(C(CCCOC)=O)CC2CC1(C(N1CCCC(C(C)C)C1)=O)C2 C(=O)(C1=CCC(C)(C)CC1)NCC1N(C(c2cc(CC)oc2C)=O)CC(OC)C1 c1(CC(=O)NC2CCC(NC(CCOCCC)=O)C2)coc2ccccc12 c1(C(=O)NCCC(=C)CNC(C)=O)cncc(OCCC)c1.C(CF)O c1(OCC)ccc(NNC(=O)c2cc(OC)cc(C(=O)OC)n2)nc1 Nc1ccc(Cl)nc1C(=O)NCC(CNC(c1ccncc1Cl)=O)CO C1(C(=O)NC(CC=C)CNC(=O)C(C)(C)n2cc(Cl)cn2)CC2C=CC1O2 C1(NC(=O)CCc2nc[nH]n2)CN(C(c2cnn3c2CCC3)=O)CC2CC12 c1(C(N2CC(C(C(=O)NCCCCN=[N+]=[N-])O)C2)=O)cc(F)ccc1F C(=O)(CCCCCS(N)(=O)=O)N1C(CNC(C(C)Oc2cccnc2)=O)CC1 Cc1ccc(OCC(=O)NC2CCC(F)(CNC(=O)C=Cc3cscn3)C2)cc1 C(=O)(C(F)(F)COC)N(CCNC(C1C(C)C1C)=O)CC c1(C(=O)NCCCCCNC(c2ccc(C)cc2Cl)=O)c(F)ccc2occc12 CCCC(C)C(=O)NCCC(O)CNC(c1nc(-c2ccc(Cl)cc2)oc1C)=O CC1Oc2ccc(C(=O)NC3C4CC3N(C(c3csc(Cl)n3)=O)C4)cc2C1C c1(C(=O)OC)cc(NC(N2CCCC(C(F)(F)F)CC2)=O)cc(Cl)c1 N1(C(c2c(C)[nH]cc2)=O)Cc2occ(C(=O)NCc3ncc(F)cc3F)c2C1 C1(C(=O)NCc2cc[nH]c2C(=O)NCc2ccc(C)o2)(CC)CCCO1 C1(NCC(=O)NC(c2ccccc2)C(C)C)CNC2(CCCOC2)C1 C1(C(=O)NCC(C)(CO)NC(=O)CC2CSCCS2)(CC)CCCCC1 Cc1ccc(C(C)C)cc1-c1nc(C(=O)Nc2ccc(Br)nc2F)ccc1F N1(C(CCCN(C)N=O)=O)CC2C3CCC(C2C1)N(C(C1CC=CCO1)=O)C3 C(=O)(C1=CC2(CCN(C(C3CC4C(C3)C4(F)F)=O)C2)C1)N(C1CSC1)C C1(C(N(CCN(C)C(c2ccn3ccsc23)=O)C)=O)Cc2ccccc2CO1 c1(OC)cc(C)nc(N2CCCC(NC(=O)Cc3ccc(O)cn3)C2)n1 Nc1ccc(CCC(=O)NCCNC(c2cccc(N(C)C)n2)=O)cc1F c1(C(=O)NCC2C(C)CN(C(=O)C=CS(C)(=O)=O)C2)cc2ccc(O)nc2s1 c1(N2CCC(CNC(=O)Cn3cccn3)C2)ccnc(Cc2ccccc2F)n1 c1(C(=O)NC(C2CCCCC2)C(C)NC(=O)Cn2cccn2)cc[nH]c1C1CC1 c1(C(N2CCC(C)C2CNC(=O)COC2CCOC2)=O)nnc(O)nc1O c1(CC(N2C(C(=O)NCC(=C)C(F)(F)F)C(C)CC2)=O)ccc2c(c1)CC2 C1(O)(C(N2CC(NC(=O)NC)C2)=O)CCN(C(=O)CCC(=O)N(C)C)C1 N1(C(CCN(C(=O)CC2CCOC2=O)C)=O)CC(=O)NCC1C(N1CCCC1)=O Cc1cc(Br)cnc1C(=O)NCC(C)(C)CN(C)C(c1nc(=O)n(C)[nH]1)=O Cc1cc(C2CC2NC(N2CCN(CCO)CC2C)=O)cc(O)c1 c1(C(N(C)CCN(C(=O)C(C)(Cl)Cl)C)=O)cc2n(c1)CCOC2 Cc1ccc(C(=O)NC(C)CNC(=O)C(C)(C)CN2CCOCC2)c(C)n1 c1(C2CC(C(N(CCC)CC)=O)C2)cn(C2CCc3c(Cl)cccc32)nn1 O=C(NN1CCCCC1)C1CC(=O)N(C2(C(=O)O)CCOC2)C1 Cc1nc2ccccc2cc1C(=O)N(C1CCCN(C(C2(C(C)C)CC2)=O)C1)C c1(C(=O)NCC2CCC(NC(=O)Cn3ccnn3)CC2)cn2c(n1)COCC2 Cn1ccc2cc(NC(C34CC(NCc5cc(Br)c(F)cc5Cl)(C3)C4)=O)ccc12 C1(CC(=O)NC2CCCC(NC(=O)CC3(C)CC(F)(F)C3)C2)(OC)CCCCC1 c1(OC)ccc(F)cc1C(=O)NCC1CCC(C)CN1C(=O)CSCC(N)=O C1(C(=O)NC2CCC(C3CC3)C2)(CC)CCN(C(c2cn[nH]c2)=O)CC1 C1(C)(CNC(C2CC(O)(CC)C2)=O)CCN(C(=O)CSCc2c(C)noc2C)C1 N1(C(c2cc(C)c(Br)s2)=O)CCN(C(=O)CN(C)C)CC12CC2 C=Cn1nncc1C(N1CCC(C)(CNC(=O)C(C2CCOCC2)OCC)C1)=O O=S(=O)(c1ccc(NCc2cccc(F)c2Br)c(F)c1)N1C2CCCC1COC2 N#CC1=C(C(=O)NC2CCCC(NC(c3onc4c3CCCC4)=O)C2)CCC1 c1(CN2CCC(c3noc(C)n3)(NC(C)=O)C2)cccc(Cl)c1O C1(F)(CNC(Cc2cccc(C)c2)=O)CCCN(C(C2CN(C)CCO2)=O)C1 CC1CCN(C(=O)C=Cc2cn(C)cn2)CC1CC(=O)NCCN1CC(CF)C1 CC1(C(N2CC(CO)(NC(c3cnc(C(C)(C)C)[nH]3)=O)C2)=O)CC2(CC2)C1 CC1CCCN(C(=O)C(=O)NC2(C)CC(NC(=O)C(C)SC3CCCC3)C2)C1 C1(NC(c2cnn(C)c2Cl)=O)CCCCN(C(=O)CN2CC3C=CC2C3)C1 C1(NC(C=CCC)=O)CCC2CCN(Cc3ncc(C(C)=O)cc3C)C1C2 Cc1cc(CCC(=O)N(CC)CC2CCCN(C(=O)Cc3ccno3)C2)c(C)s1 c12ccc3cc(ccc3n1)CNC2=O.C(=O)(C1=CCOC1)N1CC(SC)C1 c1(NC(N(C(CO)CC(C)(C)C)C)=O)cc(Br)cc([N+](=O)[O-])c1N CC(C)(C)C(CC(=O)N1CCC(OC(F)F)C1)NC(=O)CC1(CO)CCCCC1 c1(C(=O)NC(CC)CN(C(=O)C(C)OCCOCCO)C)cccc(C)n1 C(C)(C(O)C(=O)NCCNC(=O)CCc1cccc(OC)c1)OC CCCC(CCO)N=c1[nH]c(=NC2CN(Cc3ccccc3)C2)[nH]c2c1CSC2 c1(C(C)=O)ccc2c(c1)CCN(c1nnc(C3CCSCC3)n1CC(C)C)C2 CCCCC(C)(CO)NC(=O)C(O)C1CN(C(=O)CCCC(C)C)C1 C1(C(=O)NCc2noc(C)n2)(SC)CN(C(=O)CCc2n[nH]c(C)n2)C1 c1(C2(C(=O)NCC3C(NC(C4CC45CC5)=O)COC3)CC2)ccc(O)cc1 N1(C(CCCCC#C)=O)CCCCC2(CCN(C(C3(O)CC(F)(F)C3)=O)C2)C1 C(C)(CCN=c1[nH]c(Cl)ncc1[N+](=O)[O-])NC(C1(CC#C)CCCCO1)=O c1(C(=O)NC(CCC)CC(=O)N2CCC=C(Cl)C2)ccc2ccoc2c1 c1(C(=O)NCC(C)NC(c2cc(CC)oc2C)=O)ccc(S(=O)(=O)NOC)cc1 N1(C(c2c(NC)cccc2)=O)CC2CCC(C1)N2C(C1CN2CCCN1CC2)=O CC(C)S(=O)(=O)c1ccc(Cl)c(C(N2CC(C)CN(C(=O)CO)C(C)C2)=O)c1 N1(CC)CC(C(=O)NCC2(O)CCN(C(=O)CN3CSCC3=O)C2)CC1=O c1(C(N2CCN(C(=O)CC3CCC4(CCC4)CO3)CC2)=O)ccc2n[nH]cc2c1 N1(C(c2c(CCC)occ2)=O)CC(NC(C2CN(C(C)C)C2)=O)C(C)C1 c1(C(=O)NCc2scnc2Cc2nn[nH]n2)ccc(-c2nc(=O)o[nH]2)cc1 Cc1ccccc1OCC(=O)NC1(O)CN(C(=O)C(F)CC2CCC2)C1 c1(C(CC(=O)OCC)NC(c2cn(NC(CC#C)=O)nc2)=O)ccc(C#N)cc1.OC C(=O)(C(=O)C(C)C)NC(c1cn(C)nn1)C(=O)NC(c1c(C)ncs1)C C1(C(=O)NC(C)C(C)(C)NC(c2cccc(C3CC3)c2)=O)COCCC1(F)F c1(C(N2CC3(CN(C(CCCCC=C)=O)C3)C2)=O)cc2cccc(Cl)c2o1 C1(CN(C(C23CC(n4cc(CC(C(C)C)O)nn4)C2C3)=O)C)CCCCCC1 c1(OC)n[nH]c(C(=O)N(C2CCN(C(c3cnc(C(F)F)nc3)=O)C2)C)c1Cl c1(C(=O)NCCCCCCNC(C2CC(F)C2)=O)cn2ncccc2n1 N1(c2nccc(OC)n2)CCCCC(NC(c2sc(Cl)nc2C)=O)C1 C(=O)(C(F)(F)CC=C)N1C2(CNC(C3(OCC)CCC3)=O)CC(C1)C2 c1(NC(N2C(C)(CC3CN4CCN3CC4)CCC2)=O)ccc2c(c1)OCCO2 CC(F)(F)CCC(=O)NC1CCC(NC(C2(c3ccc(Cl)cc3F)CCC2)=O)C1 N1(C(C2C(=C)CC2)=O)CC2C3CCC(C2C1)N(C(=O)C1CCCc2cncn21)C3 c1(NC(C2CC(NS(=O)(=O)C3CCC3)C2)=O)nc(Cl)c2ccnc-2[nH]1 N1(C(Cc2c(C)ccnc2)=O)CCC2CC1CN2C(c1[nH]ncc1C#N)=O CC(Cc1cnn(C)c1)C(=O)NCCOCCCNC(C1(F)CC1)=O Cc1cccc(OC(C)C(=O)NC2CCOCC2NC(C2(n3cnnn3)CC2)=O)c1 N1(C(CC=C)=O)CCCC1C(C)NC(c1ccoc1CC)=O C(=O)(CCCS(C)(=O)=O)NCC1CC(F)(CNC(c2c(C)nc(C3CC3)o2)=O)C1 Cc1cccc(C(N2CCC(NC(c3cn(C)c(=O)n3C)=O)C(C)C2)=O)c1Br CC1(O)CCN(C(C2CC(NC(=O)C=CC3CCOC3)C2)=O)C1 c1(C(=O)NCC(CC)NC(C2CC2C2CCCC2)=O)cccc2c(C)c(C)[nH]c12 c1(NC(C2CCN(C(CCC)=O)CC2O)=O)cccc2c1CNC2=O N1(C(C2(CCC=C)CC2)=O)CCCC(O)(CNC(C2CC(C)CC(=O)N2)=O)C1 c1(C(=O)NCC(CC=C)NC(c2ccc(C=C)cc2)=O)cc(F)ccc1C(C)C c12cc(C)c(o1)C(=O)N(CC1CC1)C2.C1(C(=O)Nc2cnn(C)c2)(OC)CCOC1 c1(NC(C2C(CC)CCN2C(=O)Cc2cnns2)=O)cc(O)cc(F)c1 CC(C)CCC(O)C(=O)N1CC(C(C)C)CC1CNC(c1ncoc1C(C)C)=O C(=O)(C(C)(C)CCC#N)NCC1C2CN(C(C(C)n3ccnn3)=O)CC21 C1(CNC(CC(C(C)C)O)=O)N(C(c2ccc3c(c2)CC3)=O)CCCC1(C)C N1(C(c2n(CC=C)ccc2)=O)CCC(C)(C)C(NC(=O)Cc2cnns2)C1 N1(C(Cc2nnc(C)o2)=O)CCC(CNC(c2cnc(C3CC3)o2)=O)C(C)C1 N1(C(C(C)NC(=O)NC)=O)CC2CCC(CNC(C3CC4(C3)CC(O)C4)=O)(C2)C1 S(=O)(=O)(c1ccc(C#N)c(NCc2cc(F)ccc2Cl)c1)N(C(C)CO)C N1(C(CCC=C)=O)CCCC(NS(=O)(=O)CCCOCC2CC2)C1.OCC N1(C(CCOC)=O)CCCCC1C(C)NC(=O)COc1ccc(F)cn1 N1(C(CC(C)(C)N(C(COC)=O)C)=O)CC2CC(C)C2C1 c1(CC)c(C(=O)NC2CC2CNC(c2ccc(C(F)(F)F)nc2)=O)nnn1C.COC N1(C(CC2(OCC)CCC2)=O)CCCCCC1CNC(=O)C(CCOC)OC c1(C2C(NC(N(CC(CC)C)CC)=O)C2)c(Cl)cccc1Cl CC(C)(C)CC(F)C(=O)N(CCC(=O)N(CC(F)F)CCO)CCCO.OC CC1=NN(C)C(=O)C1CC(=O)NC1CCCC1CNC(=O)C(=O)C(C)(C)C C1(C(N2CC3C(NC(c4c(OC)scc4)=O)(C3)C2)=O)CCCC(F)(F)CC1 C1(C(=O)NCCCN(C(=O)CCC2CC2(Cl)Cl)C)CCCCO1 c1(N(C(=O)C(C)(C)C2CC2)CCCNCC)c([N+](=O)[O-])c(C)nn1CC1CC1 CC1CCn2cc(C(=O)NCCC3CC(NC(C4CCCNC4=O)=O)C3)nc2C1 C1(NC(C(C)CN(C)C)=O)CN(C(c2ccc(OC(F)F)cc2)=O)CC12CC2 C1(C(N2CCCC(OCC(F)(F)C(F)F)C2)=O)CCCC12CCOCC2 c1(OCC)cncc(C(=O)NCC(C2CCOC2)NC(C2(COC)CC2)=O)c1 c1(CCCCSC)nc(-c2cc(SCC)ccn2)nn1C1CCOC1(C)C C12(NC(Cc3ncn(C)n3)=O)CCC1CN(C(=O)CSc1nnnn1C1CC1)C2 CC(C(=O)NC1(CNC(=O)CCNS(C)(=O)=O)CCOCC1)P(C)(C)=O N1(C(c2cc(CC)[nH]n2)=O)C2CCC1C(NC(=O)CC(C)(C)c1ccccc1)C2 N1(C(C2(CCOC)CCC2)=O)CC2(C1)CN(C(=O)C=CC1(C)CCOCC1)C2 C(=O)(C1=CC(O)CCC1)NC1COCCN(C(C(=O)N(C)C)=O)C1 FC1(CN=C(NC2CCCC2)NC2CC23CCCC3)COCCOC1 N1(C(C2C(C)CC(=O)N2)=O)CCCC2CN(Cc3nnnn3C)CCC12 N1(CCC(=O)NCC(CCCC)NC(c2cc[nH]n2)=O)Cc2ccccc2C1=O c1(C(N2CCC(NC(C(CC)(C)CC)=O)CC2C)=O)ccc2c(c1)OCO2 CC1(C(=O)NC2CCN(C(c3cncc(Cl)c3Cl)=O)CC2F)CCNC(=O)C1 C1(C#N)(C(=O)NCC(CC(C)C)NC(c2[nH]cc(CC(C)C)c2)=O)CCOCC1 N1(CC)CCC(NC(=O)C=C(C)CNC(=O)C(C(C)(C)C)OC)C(C)C1 C12C(O)CCN1C2=O.C1(CC(N2C(CN=[N+]=[N-])CC2)=O)CCOC1=O CC1C(NC(c2cccc(=O)n2C)=O)CCCN1CCOc1ccccc1 c1(N2CCC(C)(C(C)C)CC2)ccc(S(=O)(=O)NCC2CCCOC2)cc1C#N CC1(C)CCC(C(N2CCCCC2CC(N)=O)=O)(NC(=O)CN2CCOCC2=O)C1 C(=O)(C1OC(=O)c2ccccc21)N1CC2CC(CN(C(C(C)O)=O)C2)C1 c1(C(C(=O)NC2COC2)N(C)Cc2ccc(CF)cc2)ccnc(Br)c1 CC1CCCn2ncc(C(=O)NC3CN(C(C4CC5(CC5)C4)=O)CCC3C)c21 N1(C(CN(CCC)C)=O)C2CCC1CN(C(c1cccc(C)c1O)=O)C2 C1(C(=O)NC(CC)C(=O)N2CCSCC2)(C(=O)OC)CC(C)=C(C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NC(CCNC(Cn1nnc(C)n1)=O)C(C)C C1(C(=O)NCC(CC)(C)CC)CC(C)(C)CN1C(=O)CC(C)(C)OC C12(NC(c3c(Cl)cc(C)c(C)c3)=O)COCCC1CN(C(c1cccnn1)=O)C2 c1(C(N2C(CCC(=O)Nc3nccc(I)n3)CCC2)=O)cn2ccc(Cl)cc2n1 C#Cc1ccc(Cl)c(C(=O)NCC2COCCN(C(=O)C#CC3CCCO3)C2)c1 Cc1cc(NC2CCN(C3CC3)C2)nc(NC2CC2c2ccccc2Br)n1 CCCCCC(O)CC(=O)N1CCC(CNC(=O)C(C)CC2CCCC2)CC1 CCCCCCCCC(F)C(=O)NCC1(NC(=O)C(O)C(C)C)CC1 N1(C(CNC(C2CCCSC2)=O)C(F)F)CCN(C(=O)Cc2ccsc2)CC1 c1(OC)c(C(N2CCC(N(C(=O)C=CC(F)(F)F)C)CC2)=O)c(C)nn1C C=C1CCC(C(=O)NC(C)(C)CCCNC(c2ccncc2C(F)(F)F)=O)CC1 CC(C)CCCC(=O)N1CCC12CN(C(=O)CC1(O)CCC1)C2 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC23CC3)=O)ccc2[nH]ccc2c1F S(=O)(=O)(c1nc(N2CCOC(CC)C2)ccc1Br)N(C(CSCC)C)C N1(CC(CNC(C2CCN(C)C2=O)=O)O)CC(=O)Nc2ccccc21 c1(COC)nc(C(=O)NC(C(=O)NCc2nccn2C)C2CCOC2)co1 c1(N(CCc2n(C(CC)C)nc(-c3ccc(Cl)nc3)n2)C)cc(C)ccc1C C1(C)(c2cn(-c3n(C)nnc3)nn2)CCN(C(=O)CCc2cccc(O)n2)CC1 C(=O)(C(C(=O)NCC(O)CNC(c1cc2cnn(C)c2s1)=O)C(C)(C)C)OCC CCCC(O)C(=O)NCCCCCN(C)C(C1COC(C)(C)C1)=O Cc1c(F)ccc(CN2CC(C)(C(=O)NC(CO)C(C)O)C2)c1Cl N1(C(c2c(Cl)n[nH]c2C2CC2)=O)CCC2CCCN(C(=O)Cc3cnc[nH]3)C2C1 c1(C(=O)NCC(CN(C(C(c2scc(C)n2)(F)F)=O)C)O)c[nH]c(C#N)c1 N1(C(CCN(CC)CC)=O)CC2(CC(NC(=O)CCc3cc(C)nc(C)c3)C2)C1 CCC(CC(=O)NCCC1CC(NC(=O)Cn2ccnn2)C1)C1CC1 C(=O)(CCC(C)S(C)(=O)=O)NC(C1CCN(C(=O)CSS(C)(=O)=O)C1)C N1(C(C2(C#C)CCN(C(=O)CCOC3CCC3)C2)=O)CC2CCCC(C1)N2C CC(C)C(C#N)C(=O)NCc1nnn(C)c1C(=O)NCC1CCCOC1 C1(CC)CN(C(=O)CCS(C)=O)CCN1C(C1C2CCC1(c1ccncc1)C2)=O c1(C(N2CCN(C(CC(=O)NCC#C)=O)CC2)=O)ccc2c(c1)ncn2C c1(CS(N2CCN(CC(=O)OC)CC2)(=O)=O)cccc(C#N)c1 c1(C(=O)NCC2CN(C(CC3CC(OC)C3)=O)CC2(C)C)cn2ccnc2cn1 C(CCCCCNC(=O)CN(C)CCO)N(C(c1c(C)n[nH]c1)=O)C CCCCC(C(=O)NC1CC2(C1)CC2NC(C1CC(C)C1)=O)NC(N)=O C1(C(=O)NCC2CCN(C(C3ON=C(CC)C3)=O)C2(C)C)CC2(CCCC2)CO1 CC1CN(C(=O)C(c2ccn(C)n2)N)CCS1(=O)=O N1(C(CC2=NNC(=O)C2)=O)CC(C2CCCCN(C(c3scnc3Cl)=O)C2)C1 C(=O)(C#CC(C)(C)CNC(=O)C(C)(C1CC1)OC)N1CC(C(=O)NC)C1 C1(CNC(Cc2c(C)scc2)=O)CCCCC1NC(c1cnn(C)c1F)=O C#CC1(NC(=O)C(=O)NCc2sccc2C(=O)O)CCCCC1.C(C(=O)OC)N C1(C(=O)NC(C(C)(C)NC(CCCC(=O)NCC)=O)C)CCn2cc(C)nc2C1 C(c1ccccc1F)=CC(N1CC(C(C)NC(C2CC2c2cccs2)=O)C1)=O C(=O)(C1=CCC(F)(F)CC1)NC1C(NC(C2C(=C)C2C(=O)OC)=O)CCC1 c1(C(N2C(C)(CNC(C3CN(C)C(=O)N3)=O)CCC2)=O)coc2c(Cl)cccc12 CC1CN(C(=O)CCNC(=O)C(=O)NC2CCOCC2)CC(C)(C(F)F)O1 C1(CNC(=O)Cn2cccn2)CN(C(=O)Cc2ccc(C(F)F)cc2)CCO1 N1(c2nc(C)nc3c2c[nH]n3)CC2CCC1C1CN(C(c3ncc[nH]3)=O)CC21 c1(COC)ncc(C(=O)NCC(CC(C)C)NC(=O)Cc2cccs2)c(O)n1 C1(C(=O)NC(CCC=C)C2CC2)CN(C(C2CC(=O)N(C)C2)=O)CC1C CC(C)CC(C)CC(=O)NCCn1cc(C(=O)NC(C)CCC(C)(C)C)nn1 c1(C(N2CC(N(C(C(C)n3cnnn3)=O)C)C2)=O)ccnc(N2CCC(C)C2)c1 N1(C(C(C)NC(=O)NC)=O)C2CCCC1CN(C(C1(C#N)CCOCC1)=O)CC2 C(CC(O)CO)NC(=O)C(O)CN1CCCC1.CC(C)(CNC(=O)CC1CC1)ON c1(C(=O)NC2CCN(C(=O)C(c3ccccc3Cl)O)C2)cccc(C(F)(F)F)n1 O=C(C1=CCS(=O)(=O)C1)NC1CCCC1(c1ccccc1)C(F)(F)F C1(CNC(CN(S(C)(=O)=O)C)=O)(CO)CCN(C(C2OCCC2C)=O)CC1 C1(CCN2CCOCC2)CCCC1S(C)(=O)=O.C1(=O)C(=O)NC(C)CN1C n1(CC(=O)N(C2C(C)CCN(C(C3(CO)COC3)=O)C2)C)cnc2ccccc12 CC1(C#CC(=O)N2CCCCC2CCCNC(C2CCC3CC23)=O)CC1 N1(C(C2(CC(=O)OC)CC2)=O)CCCC(NC(=O)C=Cc2ccc(C(N)=O)o2)C1 c1(C(=O)NC2C(CNC(Cc3c(C)occ3)=O)COC2)ccn2nnnc2c1 N1(C(c2c(Cl)cn(C)n2)=O)CCCN(C(C2(O)CC2)=O)CC1 Cc1[nH]nc2ccc(C(=O)NC3CC4CCC3C(NC(c3cnn[nH]3)=O)C4)cc12 c1(NC(C2(SC)CN(C(=O)Cc3ccccn3)C2)=O)c[nH]ccc1=O C1(c2cccnn2)(OCCCN(C)C2CC2)CCC(P(C)(C)=O)C1 c1(SC)cn(C)nc1C(N1CCCC(c2cn(-c3cccnc3)nn2)C1)=O c1(C(N2CCC(CN(C)C(c3nn(C)cc3N)=O)C2)=O)ccc2nn[nH]c2n1 CC1(C)CCC(CNC(C2(C)CC2(C)C)=O)N(C(c2cnc(S)nc2)=O)C1 C(CCC(=O)NCC(CNC(=O)C(c1cnn(C)c1)OC)CO)NC(=O)OC C(c1ccccc1)=[SH]C(C(=O)NCCNC(C1C(C(=O)OCC)CC1)=O)C1CC1 c1(NC(c2cn(CCN(C)C)nc2)=O)ccccc1C1CCCCC1 c1(OC)c(Br)ccc(CN2CCCC2CNC(c2cc3nccn3cn2)=O)c1F N1(C(=O)Nc2n[nH]c(C)c2C)CCC(C)(NC(=O)CS(N)(=O)=O)CC1 C1(C2CCC2)(C(=O)NCC(CNC(c2csc(C(C)C)n2)=O)OC)CCC1 c1(C(=O)NCC(CNC(C(C)(c2cccs2)N(C)C)=O)(C)O)ccc(F)cc1F N1(C(CCCN(CCC)CCC)=O)CCC(C)C(CNC(=O)CC2=CCCC2)C1 c1(NC)ccc(C(N2CCC(N3CCN(C(C4(OC)CCCC4)=O)CC3)C2)=O)nc1 Cc1cc(C(N2CC(F)CC2CNC(=O)C(C)(C)Cc2cnn[nH]2)=O)ccn1 c1(NC)cccc(C2(C(=O)NCC3CC3NC(=O)CC3CCCC3)CC2)c1 N1(C(c2cn(C(C)C)c(=O)cc2)=O)CC(NC(=O)CCC2CCC2)C(C2CC2)C1 C1(C(=O)NCC(C2CCCC2)NC(C(COC)C)=O)C(C(F)(F)F)C1[N+](=O)[O-] c1(C(C(=O)N(CCN(C(CC(C)SC)=O)C)C)O)cc(F)c(F)c(F)c1 N1(C(C=C(CC)C)=O)CCC(CNC(c2cc(-c3ccccc3)cs2)=O)C(C)C1 c1(CCCC(=O)NCC2C(NC(C3(C(C)(F)F)CC3)=O)C2)ccc(Br)cn1 C1(NC(C(C)NC(CC)=O)=O)CN(C(C2CC(N3CCOCC3)C2)=O)CC1F N1(C(C2N(C(c3c(OC)nsc3)=O)CC3CCCC32)=O)CC2CCC1C(O)C2O Cc1cnc(CN2CC3C(NC(=O)CCC(C)C)C3C2)cn1 C1(OC)CC(C(=O)O)CN(C(c2ccc(I)cc2Br)=O)C1 c1(C(=O)NC2(CC(=O)NC(C#C)(CC)CC)CCCCC2)ncc2ccccn12 c1(C(=O)O)cc(-c2ccc(=O)n(C(F)F)c2)cnc1O N1(C(C(CC(C)C)NC(C)=O)=O)CCCC(C2CN(c3cncc(Cl)n3)C2)C1 N1(C(C2CN(C)C(=O)N2)=O)CCCC(CCNC(C2C3COCC23)=O)CC1 C1(NC(c2c(C)n(C)cn2)=O)CN(C(=O)C2=NNC(=O)C2)C2CCCC12 C1(NC(CSCC#N)=O)CN(C(=O)CCSC)CCC1c1ccc(F)c(F)c1 c1(-n2cc(CN3CCN(C(C(CC)CO)=O)CC3)nn2)cc(Cl)ccc1CO N1(C(C=C(CCC)C)=O)CC2(CCCCN2C(c2cc(C)co2)=O)C1 C1(CNC(Cc2cc(C)nn2C)=O)CN(C(C2CCC(=O)N2C)=O)CC(C)(C)C1 C1(C(=O)NC2CCSC2)CN(C(=O)COc2ccsc2)CCCO1 C#Cc1cc(C(=O)NCCCn2cc(CCNC(N)=O)nn2)ccc1Cl CC1(C)CCCC(C(N2CCC(OCC(N3Cc4c[nH]nc4C3)=O)C2)=O)C1 c1(C(=O)NCCC(C)NC(CC2(CC=C)CCCC2)=O)n[nH]c2ccc(O)cc12 C1(CC(=O)NCCN(C(C)C)CC)CC(O)CN1C(=O)CCc1ccco1 c1(C(=O)NCC2(C(C)NC(c3c(CC)nco3)=O)CC2)ncnc(OC)c1F c1(C(C)C)ccsc1C(=O)NCC1COCC1NC(C1COCCO1)=O C1(C(=O)NCC2C(CNC(c3ccc4nn[nH]c4n3)=O)C2)CCc2nn[nH]c2C1 C1(C)(C(N(C2CCCC2)C)=O)CCCN(C(=O)Cc2c(Cl)cccc2Cl)C1 C1(NC(CC(n2c(C)cc(C)n2)C)=O)CCN(C(c2cc[nH]c2C)=O)C(C)C1 CCC(C)(C#N)C(=O)NCC1CN(C(=O)C(C2CCCCC2)O)CCO1 CC1CCOCC1C(N1CCC(NC(c2cn[nH]c2)=O)C1)=O C1(CCNC(c2ccc(F)s2)=O)CC(F)(F)CN1C(=O)COc1ccc(O)cc1 Cc1c(C(N2CC(N(C)C(C3CC(F)C(=O)N3)=O)C2)=O)[nH]c2cc(F)cc(F)c12 Cc1cccc(OC(=O)CC(C)(C)C)c1C.N12CCC(C1)Cn1cc(nn1)C(=O)C2 S(=O)(=O)(c1ccc(NC2COC2)c(Cl)c1)NC(c1nc(C(F)(F)F)cs1)C C1(NC(c2cn3ccnc3s2)c2n(C(CC)(C)C)nnn2)Cc2ccccc2C1 C1(C(N(CC(=O)N(CC(=C)C)C)CC#C)=O)C2(CC2)C12CC2 c1(C(N2CC3(CC(CNC(COCC#C)=O)OC3)C2)=O)cn2ccc(C)cc2n1 c1(NCc2c(C)ccc(C)c2)nc[nH]c(=NCc2cc(N)ccc2F)c1C CC(C)CCC(F)C(=O)NC(C)CCC(N1CC(CO)C(C)(C)C1)=O Cc1oc(C)c(C(=O)NC2CCCC2NC(=O)CCc2cnco2)c1C c1(NC(=O)C(C2CCN(C(c3ccc(F)cn3)=O)C2)F)ccc2cc[nH]c2c1 C1(CC(=O)NC)CCN(C(=O)C(=O)NCc2ccsc2C(=O)OC)C1 C1(CC(C)NC(c2scc(COC)c2)=O)CCN(C(C2(C#N)CC=CC2)=O)CC1 N1(C(C(C)N(C(c2cn(C)ccc2=O)=O)CC)=O)CC(C2=NOC(C)C2)C1 N1(C(C(C)CC(F)F)=O)CCN(C(=O)C(C)(C)COC2CCCC2)C2(CC2)C1 c1(CNc2nnc(C)s2)nccc(N2CCC(c3ccc(F)cc3)C2)n1 N1(C(CCCCC)=O)CC(C(=O)NCc2ccccc2CO)C2(CC2)C1 Cc1coc2ccc(C(=O)NC3CCCC3(C)CNC(=O)C(F)(F)C(C)O)cc12 c1(C(=O)NC2(C)CCN(C(CCCCN(C)C)=O)CC2)cnc2n1CCCCC2 N1(C(CCCN(C)C)=O)CCC2CC2(NC(=O)CSc2nncs2)CC1 C1(CNC(Cc2onc(C)n2)=O)CCN(C(c2ccc(N(C)C)c(F)c2)=O)CC1 C1(NC(c2cccc(C(C)=O)c2)=O)CN(C(c2cscc2C)=O)CC12CC2 CCCCCCCC(=O)N1CCC(CNC(=O)COc2ccc(Cl)c(Cl)c2)C1 c1(NC(CN2C(C)CC2)=O)ccccc1OCC1CC1 c1(C(=O)NC2C=CCN(C(C3CCCCO3)=O)C2)c[nH]c2nc(F)ccc12 Cc1ccc2c(=NCc3cnc(O)nc3O)[nH]c(=NCc3ccc(Br)o3)[nH]c2c1 C1(N(C(C2N(C)CCCC2)=O)C)CCCCN(C(c2ccc(N)cc2Cl)=O)C1 c1(C(N2CCN(C(C=CC(CC)=CC)=O)C3C2C3)=O)nc(Cl)c(=O)[nH]c1N c1(C(=O)NC(C(C)C)CN2CCCC2)cc(C(C)(C)C)nn1C C1(NC(C(CCCC)C)=O)CN(C(=O)COC2(C)CCC2)C2(CCCCC2)C1 c1(C(N(C2CCC(NC(COCC(=C)C)=O)C2)C)=O)cc2n(n1)CCCNC2=O N1(C(CCc2c(C)noc2C)=O)CCCC(F)(CNC(C2CC(F)C(=O)N2)=O)C1 C(C#Cc1cn(CCn2cccn2)nn1)NC(C1CCCC1C1CC1)=O C(=O)(C(CC)C(=O)NCCOCC(=O)N(C1CC1)Cc1cccs1)OC C(=O)(C(C(=O)N1CC(CNC(c2coc(C(N)=O)c2)=O)C1)OC)OC C=CC1(C(=O)Nc2cccc(C)c2)CCN(C(=O)C(F)CC(C)(C)C)CC1 C1(C(=O)NCCOCCN(C)C(c2ccnn2CC2CC2)=O)C2(CC2)C12CC2 c1(C(=O)NC(CCCNC(CC2ON=C(CC)C2)=O)C)nnc2n1CCCCC2 C1(C(N2C3(C(N(CC(O)CO)C)=O)CC3CC2)=O)CCCCC(=O)CC1 c1(C(=O)NC2C(NC(C3=C(C)CCC3)=O)CCC2)ccc2nn[nH]c2c1 C#Cc1cc(NC(C2CC(NC(c3sccc3F)=O)C23CCC3)=O)ccc1C C=CCCCCCCCC(=O)NCC(C(C)C)NC(=O)C=CC=CCC N1(C(C)=O)CCCC1C1CCCN1C(c1ccc(C#N)c(C(F)(F)F)c1)=O C1(C(=O)NCC2(CN(C)C(C34CC(C)(C3)C4)=O)CC2)CCCN1C1CC1 C12CN(CC1(C)C)C(CCCC1CC1)C(=O)N2.CC(C)(C)OCCC#N c1(C(=O)NCC(C(C)C)NC(C(CC=C)CC)=O)ccc2nnn(O)c2c1 CCC1=NOC(C(=O)N(CCC(=O)NCC(C2CCCO2)OC)CCCO)C1 Cc1cc(F)c(C(=O)NC(CNC(c2cnc(-c3cccs3)o2)=O)CO)c(Cl)c1 C(=O)(CC(C)C(=O)OC)NCCOC1CCN(C(CNC(CNC(C)=O)=O)=O)C1 C#Cc1cnc(C(N2CCC(N(C)C(C34COCC3C4(F)F)=O)C2)=O)c(C)c1 C(=O)(C1CCCc2c[nH]nc21)NC1CCC(NC(C(CCC)C)=O)CC1 N1(C(CCSC)=O)CCCC2(CCCCC2NC(=O)CC2CCCCC2(C)C)C1 CC(C)(C#N)CCC(=O)NC1CC2CC(NC(C3(C)CCCCO3)=O)CC2C1 C#CCC(CC(=O)Nn1cnnc1)NC(=O)CN1CCOCC1 CCCCCCC(C)(C)C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CC(F)F C(=O)(C(C)CCC(C)(C)C)N(CCCCC(=O)NCc1cc(C)sc1)C c1(CN(C)C)cccnc1C(=O)NCCOC1CN(C(C2CC(C)(C)CO2)=O)C1 C(c1ccco1)=CC(=O)NC(C(=O)NCCC(=O)NC(N)=O)C1(O)CCC1 c1(NC(N2CC(C)(C(=O)OCC)OCC2)=O)coc2ccc(OC)cc12 N1(C(COC(CC)CC)=O)CCCC(NC(C2CC2C(C)(F)F)=O)C1C c1(CN(C(CC(C)c2cccnc2)=O)CC(=O)O)ccc(Cl)cc1 N1(C(C=C(CCC)C)=O)CCCC(C(=O)N(CCC(=O)OC)CCOC)C1 C(=O)(C(F)(F)C(F)F)NCC(C)(CNC(c1cncn1C)=O)OC C12(C(=O)OC)C3C4C1C1C2C3C41C.C12(O)CCN(CC1)C(=O)CC(=O)N(C)C2 C(=O)(CC(F)(F)Cl)NCCC(=C)CNC(=O)C(c1ccc(OC)cc1)C C1(CNC(C(C)CNC(=O)C(C)(C)C2(O)CCC2)=O)CC(C2CC2)=NO1 C12(C(N3CC(NC(c4n(C=C)ncc4)=O)C(F)C3)=O)CCCCCC1OCC2 C1(CC(=O)N(C(CNC(C(C2CCCCC2)C)=O)C)C)C=NN(C)C1=O C1(NC(C(c2ccccc2)NC(C2CC(OC)C2)=O)=O)CCCSC1 C1(C(N(CCOC)CCNC(=O)CCc2nc(O)n[nH]2)=O)CCCCN(C)C1=O C(=O)(C1=C(C2CCOC2)N(C2CC2)C(=S)NC1c1cn(C)c2c(Br)cccc12)OC N1(C(c2c(C)cc(C#N)cc2)=O)CCC2OCCN(C(C3CCCOC3)=O)C2C1 c1(C(N(C(CC)CNC(=O)C(C)n2cccc2)C)=O)cncnc1 N1(C(C(C)C#N)=O)CCCC(N(C(=O)CCOc2cccnc2)C)C1 C1(n2cc(C(N(C)C)C3CC3)nn2)CC2CCC1(NC(c1cccc(Cl)c1F)=O)C2 c1(C(=O)NCC(CNC(c2cn(CCF)nn2)=O)OC)cc(C)c(F)cc1Cl C(=O)(C(C)(C)CF)N1CC(OCCNC(C=COCC)=O)C1 c1(OC)cc(C(=O)NCC(C)NC(c2n[nH]c(C3CC3)c2Cl)=O)cc(Cl)c1 C1(C(=O)NCCC(C(C)C)OC)CCCCCCN1C(c1cccc(F)c1C)=O C1(=CC(=O)NCC(=C2CN(C(c3cccnc3F)=O)C2)F)CN2CCC1CC2 Cc1cc(O)c(C(N2CCC(NC(C3CC(C)CO3)=O)C2(C)C)=O)nn1 C1(NC(C2CC(C)N2C(=O)C(=C2CCCCC2)F)=O)CC(C)(C)C12CC2 c1(SC(C)Cn2cccn2)nnc(C2CC2)n1CCCN c1(C(=O)NCCCCNC(c2nc(CC)[nH]n2)=O)cnn(CC)c1C(F)(F)F C1(CNC(CC2C(C)CCO2)=O)CC(NC(=O)Cc2ccccc2)CCO1 N1(C(CC(C(C)C)OCC)=O)CCN(C(=O)C(C)(C)CC(=O)OC)CC(C)(C)C1 C(CN(Cc1cccs1)N(C)CC1CC1C)SC N1(C(C2CC(C)CN(C(c3ccccc3)=O)C2)=O)CCC2(CC1)CC(CO)C2 N1(C(C2CN(C(C)C3CC3)C(=O)C2)=O)CCC(C)N(C(=O)Cc2ccoc2)CC1 [N-]=[N+]=NCCCCC(=O)NCC1CCCC1NC(c1ccc(C(F)(F)F)[nH]1)=O CON1CCC(CC(=O)NC(CO)C(C)NC(c2cc(CN(C)C)on2)=O)CC1 c1(C(C)(C)OC)nc(C)c(C(=O)NC2CCCN2C(=O)CC2CC2)s1 c1(C(N2CC(C)(NC(C=CC(CC)=CC)=O)C2)=O)ncn2ccccc12 c1(C(=O)OC)ncccc1C(=O)NCC1CCN(C(c2cc(F)c[nH]2)=O)C1 C(=O)(C(C)(O)CC(C)C)N1CCN(C(CNC(CC2C(C)=NNC2=O)=O)=O)CC1 c1(OC)cc(C#N)ccc1NC(=O)CN(C(=O)C(C)ON)C1CC1 c1(C(N2CC(NC(C3C4COCC34)=O)C(F)CC2)=O)cccc2nc[nH]c12 Cc1ccn(CC(C)C(=O)NC2CCC2CNC(c2cnc(C(C)O)s2)=O)n1 C1(NC(c2nccc(OC)c2F)=O)CN(C(=O)CC2(CO)CCC2)CC12CCC2 CN(C)S(=O)(=O)N(C)CC(=O)NC1CC1NC(c1cc2c(s1)CCC2)=O CC(C)CC(O)CNC(C1CCC(CNC(=O)COC(C)C)O1)=O CC(C)C(C(=O)NC(C)C(C1CCCCC1)NC(=O)CCCC#N)NC(N)=O C(CCCC(=O)NC(C1CCCC1)CNC(C1(Cl)CC1C(C)=O)=O)N(C(C)=O)C C1(C)(C(=O)NCCCCN(CCCNC(=O)CCc2ccon2)C)CCCS1 N1(C(C(C)(F)F)=O)CC2CCCC(NC(c3cc(Cl)cc(Cl)c3N)=O)C2C1 C(=O)(C1=CCCOC1)N(C1CN(C(C2C(C(=O)OC)C=C2)=O)CC1O)C N1(C(=O)CC2CCC(O)C2)CCC2(CC1)CN(C(c1ccoc1)=O)CCO2 c1(C(N2CCC(CCC(=O)NCc3ncn(C)c3)C2)=O)ccsc1C#N N1(C(C=CCCC(C)C)=O)CCC(CNC(=O)C(c2cncn2C)O)CC1 CCC(C)CCCC(=O)NCC1(C)CCCN1C(c1cc(C(C)C)oc1C)=O CCC1=C(C(=O)NCCCNC(c2nccc(OC)c2N)=O)SCCO1 CCS(=O)CC(=O)NCC1CN(C(c2ccnc(F)c2)=O)C1 CC1(C)C(CC(N2CCC(C(=O)NCC3(F)CC3)(CO)C2)=O)CC1O N1(C(c2c(C)ncn2O)=O)CCC(NC(c2ccsc2Cl)=O)C(F)(F)CC1 n1(CC(=O)NC2C(F)CCN(C(C(CC)(C)C)=O)C2)cc([N+](=O)[O-])c(C)n1 c1(NC(c2ccc(C)cc2)=O)ccc2c(c1)CN(Cc1c(Br)ccc(F)c1F)C2 Cc1cc(Br)ccc1C(=O)NC1CCN(C(C2CC2(F)F)=O)C1(C)C c1(C(=O)NCC2C(NC(=O)CSCc3ccccc3Cl)C2)cc2cccn2cn1 N1(C(C(CC#C)C2CC2)=O)CCC2C(C1)CN2C(c1csc(C(C)(F)F)n1)=O C1(C(N2CCC(C(=O)NCC(NOCC)=O)C2)=O)CC=CC(O)C1 C(C(C(=O)NCCn1cc(CO)nn1)NC(=O)C(O)CC1CCCC1)SC N1(C(c2n(C(C)C)cc(Br)c2)=O)CC2CC(C1)N(C(=O)C=C1CCCC1)C2 N1(c2n(CCOc3cccc(C)c3C)nnn2)CCN(C)c2ncccc2C1 C1(OC)CCCC1C(N1CC(CN(C)C(c2cscn2)=O)C1)=O CC1CN(C(C2C(CNC(c3cnsn3)=O)C2(C)C)=O)CC(C)(C)C1 C(CC(C)(C)CC(=O)NCCC1(NC(C2SCC=C2C)=O)CCCC1)OC CCCS(=O)(=O)NC(C)C(=O)N(C1CC(NC(=O)COCC)C1)C c1(C(=O)NC2CN(C(C(CC)C#N)=O)CC2C)cnc2ncnn2c1O C1(NC(c2ccns2)=O)CC2CCC(C1)N2C(C1CCC(O)CC1)=O c1(C(=O)NCC2(F)CCCN(C(CCCC3C(C)C3)=O)C2)cncc2ccccc12 CCC(CC)(C(C)C)NC(=O)C(C1CC=CCC1)NC(c1sccc1C)=O C1(NC(C=CCCC)=O)CN(C(=O)CCCCCOC)C2(CCCCC2)C1 CCC(C)C(CC(=O)NC1CN(C)C(C)(C)C1)NC(=O)C(C)(CO)OC S(=O)(=O)(c1cccnc1)N(C(=O)COc1ccccc1C(F)(F)F)CC=CCO N#CC1(C(N2CCC(O)(CNC(=O)Cc3ccco3)C2)=O)CC2CCC1CC2 c1(C(=O)NCCNC(c2nn(C)c(Br)c2)=O)ccc2c(c1)COC(=O)N2 c1(CC(=O)NCC(C)(C)NC(c2nc(C(C)OC)sc2)=O)cccc(C#N)c1 c1(NC(c2cc(C(F)F)ncn2)=O)nc2ccc(Cl)cc2[nH]1 c1(C(N2CCC(NC(CC=C=C)=O)CC2C2CC2)=O)cncc2c[nH]nc12 C#CCCC(C(=O)NC1CC1(C)CC)NC(C12CCC(OC)C1C2)=O C12(CC)CN(C(=O)Cc3cccc(C)c3F)C(CNC(c3cnnn3C)=O)(C1)C2 C1(C(N2C(C)CCC(NC(C3CC(n4cnnc4)C3)=O)C2)=O)CCCC(F)(F)CC1 C(=O)(CCC(F)F)N(C1CCN(C(=O)C(c2ccc(Cl)cc2)CO)C1)C c1(C(N2CC(CNC(c3ccoc3)=O)C3C2C3)=O)occ2c1CCC2 N1(C(=O)C=Cc2cc[nH]c2)CCN(C(C23CCCC2C3(F)F)=O)CC1CCO c1(NC2C3CN(C(CCCOCC)=O)C2CC3)nc(C(C)(C)C)ccc1C#N C1(OC)(CNC(C2(C)CC(C)=NO2)=O)CCN(C(=O)CCc2ncccn2)C1 CC1CC2(CO1)CN(C(=O)CC1CC(NC(c3cc(CO)ccn3)=O)C1)C2 N1(C(C2(COCC)CC2)=O)CC2(CC(NC(=O)C(c3cccc(C)c3)C)C2)C1 C(CCCCCNC(=O)Cn1ccnn1)N(C(=O)C=CC(c1ccc(F)cc1)=O)C N1(C(c2c(C)coc2)=O)CCN(C(=O)CSC(C)(C)C)CCC1C C1(C)(C(=O)NC(c2ccncc2)C)CCN1Cc1cnc(-c2ccccc2)[nH]1 c1(CC)nc(C)c(CC(N2CCC(C)(CNC(=O)C(C)CC)CC2)=O)c(C)n1 C1(C(C)C)(CC)CN(C(c2cn(C)nn2)C(=O)NCC2CCOC2)CCO1 c1(C(N2C(C(N3CC(COC)C3)=O)CC(O)C2)=O)ccc(S(=O)(=O)CC)cc1 C=CCC(C)C(=O)NCC(C1CC1)NC(c1oc(-c2cnn(C)c2)nc1C)=O c1(CC)noc(C)c1C(N1CC(CNC(c2ccncc2OC)=O)C(O)C1)=O C1(CNC(C(F)=C(C)C)=O)CN(C(c2csc(C)c2N)=O)CCC12CCC2 c1(C(N2CC(NC(CN3CC(C)C3)=O)C(F)C2)=O)cccc([N+](=O)[O-])c1Br c1(C(C(=O)N(C2CN(C(=O)CC3CCCC3)C2)C)O)ccccc1 C(N=c1[nH]c2c(c(=NCC3CC(F)(F)C(=O)N3)[nH]1)CCCC2)c1c(CC)con1 C(=O)(CCCC(=O)NCC1(OC)CN(C(c2cccnc2Cl)=O)C1)NC C1(NC(CC=C=C)=O)CCN(C(C2CC(C3CCC3)C2)=O)CC1(C)C C1(F)(c2cn(CCC(=O)NC(c3ccc(Cl)cc3)C3CCCC3)nn2)CCOCC1 C=CC1CN(C(=O)C(F)C(C)(C)O)CC1NC(c1ccc(OC)cn1)=O C(=O)(CCCCCCn1cc(CCCCO)nn1)Nc1c(C)cc(O)cc1 N1(C(CN(c2c(C)[nH]c3ccccc32)C)=O)CC(C(=O)O)CC1C1CCCC1 C1(NCc2c(OC)cc(Cl)nc2)CCC2(C1)CN(S(=O)(=O)c1cnn(C)c1)C2 C1(F)(CNC(c2cccc(F)c2Cl)=O)CCCN(C(c2cscn2)=O)C1 C(C)(N=c1[nH]c(=NC2CCCC2)[nH]c2c1CCCCC2)c1nnc(C)s1 C1(NC(CC(C(C)C)O)=O)CCN(C(C2CCC3CC3C2)=O)C12CCCC2 c1(OC)n[nH]cc1C(N1CCCC1CNC(=O)Cc1ccc(Br)o1)=O C1(CNC(c2cc(COC)sc2)=O)CN(C(c2csc(C)n2)=O)CC1C(F)(F)F c1(OC(C)C(=O)N(C(CNC(C2CC(C#N)C2)=O)C2CC2)C)cccnc1 c12nc(cc(C#N)n1)N2C(=O)CCS(=O)(=O)N(C)C.C12(SCC)CC(N)(C1)C2 C1(C(=O)NCC(CSC)O)(CNCC(=O)NC(N)=O)CCCCC1 C#CCCCCCCC(=O)NC1(CF)CCN(C(c2ncnc3c2CCC3)=O)C1 Cn1cnc2nc(Nc3cc4n(n3)CC(O)CO4)ncc12 c1(C(CNC(C(C)(C)OC)=O)NC(c2ccc(CO)s2)=O)cccc(C)c1 C(=O)(CC1C(=O)Nc2ccccc21)N1CC(CNC(C(CC)(C)CC)=O)C(O)C1 c1(C(=O)NC2(CN(C)C(C3CC4C=CC3C4)=O)CC2)ccc2c(c1O)CCCC2 Cc1nn(-c2cccc(C(F)(F)F)c2)c(Cl)c1CNCC12CC(F)(C1)C2 CS(=O)(=O)CC(=O)NC12CC(CNC(=O)CCNC(c3ccco3)=O)(C1)C2 N#CC1CN(C(c2cccc(-c3cn(-c4ccccc4)nn3)c2)=O)CC12CCC2 c1(CC(N2CC(C)C(NC(=O)CC3CCCC34CC4)C2)=O)c(O)ncnc1O C1(CCC(N2CCC(CCC)C2)=O)CCCCN(C(C2CCCC(C)(C)C2)=O)C1 N1(CC)CC2CN(C(C3CN(C(=O)CC(O)CC(C)C)CC3F)=O)CC2C1 C(=O)(C1=C(C)OCCS1)N(C1CCCN(C(C2CSCN2C(C)=O)=O)C1)CC c1(C(=O)NC2CC3C(NC(c4c(C)ccc(O)c4)=O)C3C2)cc2n(c1)CCCC2 C1(CCCNC(c2cscn2)=O)COCCN1C(=O)C(C1(O)CCCC1)F c1(C(=O)NCC2(F)CC(NC(c3c(C)ncnc3)=O)C2)cnc(O)c([N+](=O)[O-])c1 C1(CNC(CC(=C)C)=O)CN(C(c2cc(C(CC)CC)no2)=O)CC12CC2 CC(C)(C(=O)N1CC(CNC(=O)CNc2ccccc2)C1)C(F)(F)F C1(C(C)NC(C2CCOCC2)=O)CCN(C(c2cnc(C(C)(C)CF)o2)=O)CC1 CC(=O)CCC(=O)N(CC(=O)NCCC1OCCC1(C)C)C(C)C C=CCCCCC(C(=O)NCCC(F)F)N(C)Cc1ccc(F)c(F)c1 C(=O)(C1CCCn2nccc21)NC1C(N(C(=O)CN2CC(C)(C)C2)C)CCC1 N1(C(CSCCCC)=O)CC=CC(C(N2C(CO)CC2C)=O)C1 N1(C(C(C)NCCS(C)(=O)=O)=O)CCC2CN(C(=O)Cc3ncc[nH]3)CC12 c1(-c2cc(C(=O)NCCN(C(=O)C(C)CSC)CC)on2)ccc(Cl)cc1 C1(C(N(C(C#C)C)C2CC2)=O)CC(NC(=O)CCSCCCC)C(O)C1 CC(C)C1=CCC(NC(=O)CC23CCC2CN(C(=O)C2=CCSC2)C3)CC1 N1(C(c2cn(CC(C)C)nc2)=O)CC(N(C)C(C2CC2C(N)=O)=O)C2(CC2)C1 N1(C(Cc2cn(C(C)C)nn2)=O)CCC(NC(c2cnn[nH]2)=O)C(CO)C1 c1(C(C)=O)cc(C(C)NC(=O)OC(C)(C)C)cnc1C.C1(=O)COC(=O)CN1 C1(NC(C(C(C)C)c2ccccc2)=O)CC2CCC1CN2C(c1cncn1C)=O C1(NC(C2(O)CN(C(N3CC(C)C3)=O)C2)=O)CCC(=O)NC1 N1(C(C2(CC=C)COC2)=O)CC(NC(c2coc(C3CC3)n2)=O)CC(C)C1 c1(OC)cccnc1C(F)(F)C(=O)NCCN(C(=O)Cn1cc(C)cn1)C c1(C(=O)NC(C)CCNC(=O)C(C(C)O)N(C)C)ccc2cnsc2c1 CC(CC(C)(C)C)C(=O)N1CCN(C(c2ccnc(C3CC3)n2)=O)CC1CO C#CC1CCCN(C(=O)C(C(C)(C)O)NC(=O)CCCCCOCC)CC1 c1(SCCC(=O)NC(C2CCCN2c2nnc(CO)s2)(C)C)ccccc1Cl C(C)(C(=O)NCC(C)N(C)C(c1cc2sccc2[nH]1)=O)(C(C)C)NC(C)=O Cc1ccc(C(=O)NC(CNC(=O)C(O)C(C)(C)C)CO)c(Br)c1 c1(CC)nc(NCCc2cnn(C)c2)cc(=NC(C)CCC2CCCC2)[nH]1 N1(C(c2cn(CCC)nn2)=O)CCC(C(=O)NCCCNC(=O)COC)CC1C c1(CC)cc(Cl)ccc1C(N1CCCC1CNC(c1cnc(CO)nc1C)=O)=O C1(C(=O)NCCN(C(=O)C(C2CCCCC2)O)C)CC2OC(=O)OC2C1 Cc1nc(C)c(C(=O)NCC2CCCC2C(N2CCCCC2CF)=O)s1 N1(C(C(CC)SC)=O)CCCC(F)(CNC(=O)Cc2ccc(Br)cn2)C1 c1(C2(C(N(C)CCNC(=O)Cc3ccc(Cl)cc3)=O)CCC2)ccc(Cl)c(F)c1 Cc1occc(=O)c1OCC(=O)Nc1cc[nH]c1C(C)C C(c1cncc(F)c1)=CC(N1C(C(C)(C)NC(CCOCCC#C)=O)CCC1)=O N1(C(C2C(CC)C2)=O)CCC2CN(C(c3ccc(O)cc3C)=O)CCC12 CC1CC2(CO1)CN(C(=O)CC(C)C(C)(C)NC(=O)C1=CC3CCCC13)C2 C(=O)(C(O)CC1CC1)NCCCC1(NC(=O)C(O)C2CCCC2)CC1 N1(C(CCOCC)=O)CCC2(CC1)CN(C(C13CC(C1)C3)=O)CC2CO CC(C)CC(C(=O)NC1CCC1CNC(c1cnc(N)cn1)=O)C(C)C N1(C(c2cc(COC)no2)=O)CC2CC(C1)N2C(c1ccc[nH]1)=O C(CC(C)(C)C(=O)N1CCN(C(=O)C(O)C(F)F)C(c2cccc(F)c2)C1)OC Cc1nc(C)c(C(C)NC(=O)CC2CCC(NC(C3(CC(C)C)CC3)=O)CC2)[nH]1 c1(OC)cc(C)c(CN2C(C(=O)Nc3cccc(OC)c3F)CC3CC23)c(C)c1 C=C(C)C1CCC(C)=CC1CC(=O)N(CCNC(=O)Cc1ccn(C)c1)C(C)C c1(CC)ccc(C(N2CCCC(NC(=O)C(C)(O)CC)C2)=O)cc1OC C(=O)(C1=C(Cl)CCCC1)NC1CC(C(N(C)Cc2ccccc2F)=O)C1(C)C c1(CCC)onc(C)c1C(=O)NCCNC(=O)C(c1ccc(F)cc1)(C)O Cc1ccc(OCC2CCCO2)c(NC(=O)NCc2cccn(C)c2=O)c1 C(=O)(C(CCCC(C)(F)F)N1CCC(C2=NCCC2)C1)NC C(c1ncccc1C)=CC(=O)NC1CCN(C(c2cnc(CCC)s2)=O)C1 c1(C(C)C)[nH]nc(C(=O)NCCC(C)NC(C2(C#N)CCCO2)=O)c1Br N1(C(C(COCC)n2cc(CNC3CCC3)nn2)=O)CCC2(CC2)CC1C c1(C(=O)NCCCCNC(=O)CC23COC(CF)(C2)C3)nnn2c1CCC2 C(CC)(C(=O)NCC(C)(CO)NC(=O)COCc1nc(C)no1)=CC C(=O)(C1COc2ccccc21)NCCCCN(C(=O)COC1CC(F)(F)C1)CC C1(C(=O)NCCN(CCCN(C)C)C(c2n(C=C)ncc2)=O)CC2CCCN(C1)C2 c1(C2C(C(=O)OCc3nc(C)oc3)C2)ccc(Br)nc1 c1(N2CCC(C)SC2)nc(NCC(F)(F)C(F)(F)Br)c2ncsc2n1 c1(C(N2C(C(C)(C)NC(Cc3c(C)ncs3)=O)CCC2)=O)cc(Cl)cc(Cl)c1F N1(C(C2C(NC(C3(CC)COC3)=O)CCOC2)=O)CC2(CCOC2=O)C1 c1(N2C3CCN(C)C3CCC2)nc(=NCCC=CBr)[nH]c2cc[nH]c12 c1(CC)cc(F)ccc1C(=O)NC1CCC(N(C(=O)CCN2CCC2)C)C1 c1(C(=O)NC(C2CCN(C(c3cc(F)n[nH]3)=O)C2)C)cc(Cl)c(Cl)c(Cl)c1 CC1CC(CNC(C2CC2C)=O)CCN1C(=O)CNC(c1ccsc1)=O C(C(CC(C)C)NC(C1CN(C(=O)NC)C1)=O)NC(CCC#C)=O N1(C(Cc2cn(C)nc2)=O)CCN(C(c2cn(C)cn2)=O)CC1c1cccnc1 C(CCCCCCCl)c1onc(-c2cc(OC(C)C)ncc2)n1 C(=O)(CCC(C(=O)NCC(C(C)(C)C)NC(c1csc(C)c1)=O)N(C)C)OC c1(C(=O)NCC(C)CNC(=O)Cc2ccccc2CC#N)ccc2c(n1)CCO2 N1(Cn2c(-c3cccc(C(C)(F)F)n3)nc(CCSC)n2)C(=O)CCCC1=O C1(NC(C(C2CCC2)NC(C2(C)CCCCO2)=O)=O)CC2CCCCCC12 N1(C(C2(OCC)CCOC2)=O)CC2CC(C1)N(C(c1ccc(CC)nc1C)=O)C2 CCCC(C(C)(C)C)NC(=O)C(Cn1cccn1)NC(=O)CCC(C)(F)F c1(OC)ccc(OC)c(-c2ccnc(CNC(=O)Cc3cncc(C)c3)c2)c1 N1(C(CNC(CC)=O)=O)CCC(CNC(C23CC(CN2C2CC2)C3)=O)C1(C)C CN1C(=O)CSC1=CC(=O)NC1CN(C(=O)Cc2nnc(O)s2)CCC12CCC2 C1(CNC(c2c(C)ocn2)=O)C2CCC(C2)N1C(=O)C(C)(C)N(C)C c1(C(N2CCC(N(C(=O)C(C)NS(C)(=O)=O)CC)CC2)=O)cccc(=O)n1C C(=O)(C(O)CCCNC(c1cc(C(F)F)[nH]n1)=O)NCCC(=O)NO C(=O)(CC(C)C(=O)N1CC(O)(C(F)C(N2CC3CCC3(C)C2)=O)C1)OCC c1(C(N(CC(=O)NCC2(CO)CCCC2)CC#C)=O)ccc(C#N)cn1 N1(C(CCCc2cc(C)sc2C)=O)CCCN(C(c2coc(Cl)n2)=O)CC1CO S(=O)(=O)(c1cccnc1)N(CC(=O)NC1CCN(C(c2cnccn2)=O)CC1F)C CCC(C(=O)OC)C(=O)NC(C)C=CC(N1CC(C)(O)C1)=O c1(C(=O)NCC(CN(C(C2(CC=C)CC2)=O)C)C)ccc2c(c1)CCCC2 C(CNC(c1sccc1Cl)=O)(CC(=O)NCCN1CCC(C)C1)OC c1(C(N2CC(OCCNC(c3cnncc3O)=O)C2)=O)ccncc1N1CCCC1 c1(C(=O)NCC2(NC(CSCCC#N)=O)CCC2)cccn2cnnc12 N1(C(CCC(C)SC)=O)CC2CCC(C1)N2C(C12CCCCN1CCC2)=O C=CC1(NCC2CC2F)CCNCC1 N1(C(c2n(C)cnc2)=O)CCC(C(N2CCCC(CC3CC3)C2)=O)C1(C)C Cc1cnc(CC(c2ccccc2)N(C)C(=O)NC2(n3cnnn3)CC2)s1 c1(C(=O)NCCC2(OC)CN(C(C3(C)CC3(F)Cl)=O)C2)cc(OC)ccc1O c1(OC)cnc(C(=O)NC2CCCCC2NC(c2cc[nH]c2C(C)C)=O)c(F)c1 C(=O)(CCC(C)S(C)(=O)=O)NCCC1CN(C(c2cc(CC(C)C)[nH]n2)=O)C1 C(CC(=O)N1CCC(C(=O)NCC(c2ccncc2)O)C(O)C1)(C(C)C)OCC COn1cnc(C)c1C(N1CCC(C(C)NC(=O)CCc2ccc(C)s2)C1)=O c1(CC)ccc(C(N2CCCC2C2(NC(=O)Cc3csnn3)CC2)=O)cn1 CN1CCN(C(C2(c3cnn(C)c3)CCCO2)=O)CC1CNC(=O)CCC1CC1 CN1CCN(c2ncc(C#N)cc2F)CCC1C(C)(C)CNC(=O)C(C)(C)C(N)=O N1(C(c2n[nH]cc2Br)=O)CCN(C(c2ncc(F)cc2F)=O)C(C(F)F)C1 C(N=c1[nH]c(=NCCc2cocn2)c2ccccc2[nH]1)c1nc(CC(C)C)sc1 C#CCCCCCC(=O)N1CCCC(NC(=O)C(=O)C(C)(C)C)C1 C1(CC(=O)NCC(C2CCC2)NC(C2(C(F)(F)F)CC2)=O)(CC)CCC1 C(=O)(C1=CC(C)(C)C1)NC12CC(NC(c3c(CC)nco3)=O)(C1)C2 C(=O)(C1c2ccccc2C2CC1C2)NCCOCCNC(c1cnc[nH]1)=O c1(COC)ccc(-c2nc(C)c(NCC3CCCN(C)C3)s2)cc1 N1(C(C(COC)(F)F)=O)CCN(C(c2cn(C)c(C)n2)=O)C(C(C)C)C1 c1(CN(C(c2c(CC)nn(C3CC3)c2)=O)CC)ccc(Cl)cc1Br N1(CCN(C(CSCCC)=O)C)CCN(C(c2ncncc2F)=O)CC1 C1(CC(=O)NC2CC(CCNC(c3nc(OC)c(C)s3)=O)C2)COCC(C)(C)O1 N(C1=NCCC(=O)N(C)N1)C(C=C)C.C1(CC2CC2)CCN(C(=O)C(C)(C)C)CC1 c1(OC(C)C)cnc(NC(C)CNC(=O)C(O)Cc2cnc[nH]2)nc1 CCC(CNC(=O)CCC1CC1(Cl)Cl)NC(=O)CCOCC1CC1 C(C(C)(C)CN=[N+]=[N-])NC(C1N(C(C2(c3cccs3)C(C)C2)=O)CC(CO)C1)=O C(=O)(CCCCCSC)NC(CC(=O)NC1(CCOC)CCC1)C CC1CN(C(C2(C(F)F)CCC2)=O)CCN1C(c1cc(Cl)c(Br)[nH]1)=O C1(C(N2C(C(C(N3CC(C#C)(O)C3)=O)(C)C)CCC2)=O)CC2(CC(=O)C2)C1 N1(C(c2ccc(OC)nn2)=O)CCC(C)CC1CNC(=O)CCc1cnn(C)n1 C1(NC(=O)NC(CC)C(C)CN(C)C)CC2(CCN(C(=O)OC(C)(C)C)CC2)C1 c1(C(N2CCC(CNC(C=CC=CCC)=O)C(C)C2)=O)ccc2c(c1)CC(C)O2 c1(C(=O)NC23C(CN(C(CC=C=C)=O)C2)COCC3)cccc(S(=O)(=O)CC)c1 C1(CC(=O)NC(C(C)C)(C)CNC(C2CC=CC2)=O)Cc2cc(F)ccc2O1 c1(NC(C2(c3c(-c4c(OC)nccc4)cccc3)CC2)=O)nc(C)c(Cl)cc1Cl N1(C(C2CC(F)(F)CN2Cc2ccc(Cl)o2)=O)CCN2C(=O)OCC2C1 c1(NCC2(C(c3n(CC=C)nnn3)CC)CCC2)cc(OCCC)cc(Cl)c1 c1(CC(C)C)ccc(C(=O)NCC2CC(C)N(C(=O)CSCC(N)=O)C2)cn1 CC(C)CC(C(=O)NC1CC12CCC2)ONC(c1cccc(=O)n1C)=O Cc1cc2c(SCCC(=O)N3CC(c4ncccn4)C3)ncnc2s1 CC(C)C(N)CC(=O)N(C)Cc1ccc(I)cc1 c1(OC)cccc2c1N(C(c1cn(Cc3cccc(C)c3)cn1)C(=O)O)CC2 Cc1cccc(C(C)(C)C(=O)NCC(C)NC(=O)C(c2cn(C)nc2C)C)c1 C(N=c1[nH]cnc(Cl)c1C#N)C1(C)CCC(NC(C(C)SC)=O)CC1 N1(C(C2N(C)CC(O)C2)=O)CC2CC1CN(C(C1CC1c1cccc(O)c1)=O)C2 c1(OC)ccc(C=CC(=O)N(C(C)CNC(=O)Cc2cc(C)ccc2C)C)cc1 C#CCCCCC(C(=O)NC)N(CCC1CCCN1C)Cc1ccc(OC)cc1 N1(C(C(C2CCOCC2)C)=O)CC2CC(CNC(=O)CCc3nc[nH]n3)C2C1 C1(CNC(c2nc(CC)oc2)=O)CCCCN1C(C1CC=CC1)=O C12(NC(c3c(CC)c(C)sc3)=O)CCCC1N(C(c1ccc(F)c(C)c1)=O)CC2 N1(C(C2CC(F)CN2Cc2cccnc2Cl)=O)CCN2C(=O)OCC2C1 c1(OCC)ccc(C(N2CCC(NC(=O)CC3CCC3)CC2)=O)cc1OC Cc1ccoc1CC(N1CCC1Cn1cc(CCC2CCOCC2)nn1)=O N1(C(c2cc(CCC)on2)=O)C(CNC(c2cccc(C3CC3)c2)=O)CC2CC12 C1(CC(=O)NC(CCOC)COC)CC(C)N(C(=O)CCn2ccnn2)C1 C12(C(=O)NC3CCN(C(C4CCS(=O)(=O)C4)=O)CC3F)CC3CC(CC1C3)C2 C#CC1(O)CC(C(=O)NC(C(C)NC(c2cccc(COC)c2)=O)C(C)C)C1 C1(CC)CN(C(=O)CC2(CSCCN=[N+]=[N-])CC2)CCN1C(=O)Cc1n[nH]c(C)n1 c1(-c2cn(CC3OCCN(C(c4ncc(C)o4)=O)C3)nn2)ccnc(Cl)c1N c1(C(C(=O)NC(C)CO)N(C(C)=O)CC2CC(C(F)F)C2)ccc(Cl)c(Cl)c1 N1(C(C2CC(=C)C2)=O)CC2CC1CCN2C(=O)CSc1nc[nH]n1 c1(C(N2CCC(CCNC(C(C)OCCC=C)=O)C2)=O)ccc(C#N)o1 c1(CN2CC(C(C)NC(CCC)=O)C2)c[nH]c2cccc(F)c12 N1(C(c2ccc(CSC)cc2)=O)CC2CC1CN2C(=O)C(F)OC(F)(F)F CCCC(C)(CC)C(=O)N1CCC(OCCNC(c2cc(OC)n(C)n2)=O)CC1 CC1CCC(CNC(=O)CCF)CN1C(=O)CNc1ccc(O)cc1 C1(OC)(CNC(=O)C(O)CC(C)C)CCN(C(c2c(Cl)sc(C)c2C)=O)CC1 n1(CC)nnc(C(N2CC3CC3(CNC(c3ccccc3C)=O)C2)=O)c1C N1(C(C2CCC(=O)O2)=O)CCOC2(CCN(C(c3ccc(CCO)cc3)=O)C2)C1 N#Cc1cccc(CNC(=O)C(N2CC3CC(F)(F)CC3C2)=O)c1Br c1(C(C)NCC(C)(C)NC(C2CCS(=O)(=O)C2)=O)cccc2ccccc12 C(CC(C)C(=O)N1CCC(CCOC)(NC(=O)CCCN(C)C)C1)=CCC C1(C)(NC(CC(=C)C)=O)CCCN(C(=O)Cc2ccnc(Cl)c2F)C1 c1(NC2C(CC)CCCC2)ccc(S(=O)(=O)N2CCc3c[nH]nc3C2)cn1 c1(C(=O)NCC(c2cnccn2)=O)nscc1Br CN1CCOC(CN(C)C(C2C3CC2N(C(C2C4CC(=O)CC24)=O)C3)=O)C1 CC(C)(O)C#CC(=O)NC(C(=O)NCC1(C)CCCC1)C1CCCC1 c1(CCC(=O)NC(CC=C)CNC(c2ccsc2C)=O)cc(C)nc(C)c1 C(C)(CC(=O)N1CCCC(O)(CCNC(c2cnsn2)=O)C1)(C(F)F)N(C)C C(CC(C)(C)C(=O)N1CCC(N2CCN(c3ccnc(C(C)C)n3)CC2)C1)OC C(=O)(CC1CCc2ccc(O)cc21)NC(CCCC)CNC(c1nc(C)c[nH]1)=O C(=O)(C(CC=CCl)c1ccccc1)NC(C)CCNC(c1[nH]ccc1C1CC1)=O CC1C2C(CCN2C(=O)CCS(C)=O)CN1C(c1cc(CO)on1)=O c1(CN2CCC(CC(=O)Nc3nc(Br)cs3)C2)cc(Br)cc(F)c1F C(=O)(N=c1nc[nH]n1C(C)(C)C)NC1C(c2n(C)ncc2)C1 C1(C(N(CC(C)O)C)=O)CC(NC(=O)CN(C)C)C(O)C1.C1(=O)CN1C CC(C)C(C(=O)N1CCC(O)CO1)c1cc[nH]n1 c1(CCC(=O)NC(C)CN(C(=O)CC(C)C2CCCO2)C)cccc(O)c1 c1(C(=O)NC2C=CCN(C(c3c(C)cncc3)=O)C2)ccc(N=NC(N)=O)cc1 c1(CC(C)NC(c2cccc(C(=O)OC)n2)C)ccc(C(F)(F)F)c(F)c1 N1(C(CC(C)n2cccc2)=O)CCC2CN(C(c3ccc(CO)c(Cl)c3)=O)CC12 N1(C(Cc2c(N)cccc2)=O)CCCC(NC(=O)C(c2cccc(Cl)c2)O)CC1 Cc1nnc2n1CCC(C(N1CC(NC(=O)CC3CN4CCN3CC4)C1)=O)C2 CCC(CC)CCC(=O)NCCNC(c1ncoc1CCC(F)(F)F)=O CC1(C)CC(NC(C2CC3C=CC2C3)=O)CCN(C(=O)COC2CC(F)(F)C2)C1 CC1CN(C(c2c[nH]c(Br)c2)=O)CCC1NC(=O)C(C1CCCCC1)O C1(C(N2C3CC(NC(C4CNC(=O)O4)=O)CC2CC3)=O)CCc2ccccc2C1O CC1(C)C2CN(C(=NCC(F)(F)CC3CC3)NCC(=O)NCCC(C)(C)C)CC12 N1(C(c2nc(OC)oc2)=O)CC(C)N(C(=O)Cc2ccc(Cl)cc2Cl)CC1C N1(C(C(CCc2ccc(CC)cc2)C)=O)CC2CCN(C3CCNC3=O)C2C1 c1(C(=O)NCC2CCN(C(CCC=CC)=O)C2)ccc(C2(C)CC2)cc1 CC(CC(=O)NCCOCCNC(c1cc(O)cc(F)c1)=O)CC(C)(C)C c1(C(=O)NC2CCC(NC(C3(CCC=C)CC3)=O)CC2)c(C)cncc1C c1(C(N2CCCC(NC(CCC(C)OCC)=O)C2)=O)cc2c(o1)CCCC2 N1(C(C(CC)C)=O)CC(NC(=O)Cc2cnsc2)CC2(CCOCC2)C1 c1(CCC(=O)NC2(CC=C)CN(C(C3CCNC3=O)=O)C2)cnc(C)nc1O C(CCC(O)C(=O)NC)NC(C1CC(N(C)C)C1)=O.c1(C2CCC2)cc[nH]n1 c1(OC)cc(C)ccc1NC(=O)NC1CCC(C)N(C(=O)CCc2cnoc2)C1 C(=O)(CCS(=O)(=O)c1ccccc1)N.C=CC(O)C(C)(C)C=O C1(c2ccccc2)CC(C(=O)NCC2C(CC)C2(F)F)CCN1C(=O)NC Cc1cc(Br)c(S(=O)(=O)NC2CCN(CC(F)F)C2)cc1Br O=C(CCC(F)(F)F)NCC1CCCC1NC(=O)CC1CCCC1 CC(C)(C)C(C#N)C(=O)N1CCCC(NC(=O)C(=O)Nc2ccccc2)CC1 Nc1ccc(CCC(=O)N(CCCNC(C2CCCCC2O)=O)C2CC2)cc1F CCC(C)(C#N)C(=O)N1CC(C(N2CC3CC2(C(F)F)C3)=O)C(F)C1 N1(C(COC)=O)CC(C)(CNC(C2CC(S(N)(=O)=O)C2)=O)CC1(C)C C1(OC)CC(CNC(c2ccc(F)cc2)=O)N(C(=O)CCc2ccon2)C1 c1(CNC(=O)NC2C(OC(C)(C)C)COC2)cncc(-c2ccccc2F)c1 CC(CCC(=O)NC1CCCC(CNC(=O)CN(C)CCO)C1)N(C)C c1(C(=O)OC)ccc(Br)cc1NC(C1CCCCN1Cc1cc(F)cc(Cl)c1)=O c1(C(=O)NC2CN(C(C(CC)=CC)=O)C2)cc(Cl)ccc1SC1CCCC1 c1(CC)ccnc(C(=O)NC(CCNC(=O)C(F)n2cccn2)C(C)C)c1 C(=O)(C1CCc2ccccc21)NC(C1CCCN1C(=O)COCCOCCO)C C1(NC(CCC(C)C)=O)CN(C(=O)CCCNC(c2ccco2)=O)CC(F)(F)C1 N1(C(C(COC)N(C)C)=O)CCC(C(C)C(=O)N(C(C)COC(F)(F)F)C2CC2)CC1 c1(OC)c(C(=O)NCC2CC2NC(c2ccc(C3(O)COC3)cc2)=O)cnn1C C1(=CC(N2CCC(C(C)NC(=O)C(C#N)C3CC3)C2)=O)CCC(C)(C)CC1 C(=O)(CCC1=CCCCC1)N1CCCC(CNC(CC(=O)NCCOC)=O)CC1 N1(C(c2ccc(C)cc2Cl)C(=O)NCC=C)CCCCCCC1CC n1(CC)ccnc1C(=O)NCC(C)(C)CC1CN(C(=O)COCC(=O)OC)C1 Cn1cnn(CC(=O)NC2CCCC2C(N2C(CO)CC2CO)=O)c1=O N1(C(c2cc(=N)[nH]cc2)=O)CCC(NC(C2CCCS(=O)(=O)C2)=O)CC(O)C1 C1(NC(Cc2nc(C)[nH]n2)=O)CCN(C(=O)Cc2c(F)cccc2F)CC1O C1(NC(c2ccc(CCC)[nH]2)=O)(COC)CCN(C(=O)C(c2ccnn2C)C)C1 c1(OC)ccc(F)c(C(=O)NC2CC(N(C)C(C3(OC)CCC(C)(C)C3)=O)C2)n1 c1(NC(=O)C(N2CC(CF)OC(CF)C2)=O)cccc2c1OCC2 c1(NC)cc(Cl)ccc1C(=O)NC1CCC(CNC(=O)C(C)(C)CF)C1 S(=O)(=O)(c1ccc(Cl)c(C(=O)O)c1)N1C(C)(C(=O)NCC(C)C)CC1 C1(NC(CCCCCC)=O)CC2(C1)CC(C(N1CCC(C)(COC)CC1)=O)C2 C1(NC(c2occc2CNC(=O)C(O)C2CC2)=O)CCCC12CC2 N(C1CC2(CN(C(c3ccsc3C#N)=O)C2)n2ccnc21)C(C1CCC(C)O1)=O n1(CC)cc2ccc(C(=O)NC3CN(C(=O)C(C)COC)C3)cc2n1 c1(C(=O)NC2(CF)CCN(C(C=CC=CCCCCC)=O)C2)ncc(C)cc1F c1(C(=O)NCc2cn(CCNC(CCC(=C)C)=O)nn2)cc([N+](=O)[O-])n[nH]1 N1(C(C(=O)NCC)COc2ccccc2)CC(CC(F)(F)F)OC(C)C1 C1(CC(N2CCC(NC(c3c[nH]c(=NC)o3)=O)C2)=O)COC(C)(C)CO1 c12cc-1ccc2S(C)(=O)=O.C(C(O)CF)N(C)C(C1CCCC1)=O C(CCNC(c1ccc(=O)oc1)=O)(C(C)C)NC(C1N(C(CCC)=O)CSC1)=O c1(C(=O)NC2CN(C(C(C)n3cccc3)=O)CC(O)C2)cc2cccnc2[nH]1 N1(C(CC(CCC)C)=O)CC2CC(C1)N(C(c1nc(F)ccc1Cl)=O)C2 N1(C(C=Cc2nnn(C)n2)=O)C2CCC1C(F)C(NC(=O)CC1C=CCC1)C2 Cc1nc(C(=O)NCCCCCC2CCN(C(c3nccs3)=O)CC2)c(C)o1 C(=O)(CC(C(C)C)NC(=O)CCCNC(=O)OC)N(CCCC=C)C c1(CCC)cc(C(=O)N(C(C)CCNC(=O)C(C)N2CCC2)CCOCCO)n[nH]1 C1(C2(C=C)CCC2)(C(N2CC(CC=C)(NC(=O)CCC(=O)N(C)C)C2)=O)CCC1 c1(CN2C(CCC(N3C(C(C)(C)C)CCC3)=O)CCC2)cccc(Cl)c1O C1(CC(N2CC(CNC(c3n(C)ccn3)=O)C(C(F)(F)F)C2)=O)OC(C)(C)OC1=O C(=O)(CC(C)(C)C(F)(F)F)NCC12CC(NC(CCC(=O)NC)=O)(C1)C2 c1(CC(C)N(C(c2cn(CCN)nn2)=O)CC)ccc(OC)cc1 CC(C)CC(C(=O)N1CCN(C(=O)CCCCC(N)=O)C(CO)C1)C(N)=O c1(C(=O)OCCOC(N(C)C(c2nn(C)cc2N)=O)=O)cc2ccncc2cc1F Cc1nn(C)c(C)c1OCC(N1CCN(C(C2CC2CF)=O)C(C2CC2)C1)=O c1(NCC)cccnc1C(N1CC(CCNC(=O)CCOC2CCOCC2)C1)=O c1(C(=O)NCC2(CC(=O)NCC(C)C#N)CC2)c[nH]c(=S)cn1 c1(C(=O)NC2C3CN(C(c4c(OC)c(C)ccc4)=O)CC32)sc2ccccc2c1C C12(c3n(CCCSCC)cnn3)CCCCC=C1OCC2.C(CCC(C)C)OCC c1(C(N2CCN(C(CSCC=C)=O)CC2CC)=O)ccc(Br)c(C)c1F N1(C(CCCS(C)(=O)=O)=O)CC(CO)C2(C1)CN(C(=O)CCc1nc(=N)[nH][nH]1)C2 N1(CC(=O)N(C)C)CCN(C(=O)NCc2cc(-c3ccccc3)ns2)CC1 c1(C(N2CCC(OCCNC(C=CC(N)=O)=O)C2)=O)ccc(F)cc1F c1(C(N2C(CNCc3ccc(C#N)cn3)CCC2)=O)cc2ccccc2nc1O Cc1cc(C(=O)NC2CC(C)N(c3ncc(C(C)(C)O)cn3)C2)ncc1C(F)F N1(C(c2cccn2CC)C(=O)NCCOCC)CC(C(N)=O)CC(C)C1 c1(CC)ccc(C(=O)NC(C2CCCC2)CNC(=O)CN2CCC(C)C2)c(O)c1 c1(OC)ccc(F)cc1S(=O)(=O)N1CC(C)(C(=O)Nc2oncc2C#N)C1 C1(CNC(CSCC=C)=O)(CO)CC12CCN(C(C1CCS(=O)(=O)N1)=O)CC2 C(=O)(C1CCCc2n[nH]cc21)NC1C2CC(NC(C3CC(C)(F)C3)=O)C(CC2)C1 c1(C(CC)C)nc(-c2cc(Br)n(C)n2)n(Cc2ccc(OC)cc2)n1 Cn1nc(C(=O)NC2CCN(Cc3coc(-c4ccccc4)n3)C2)ccc1=O N1(C(C2(OC)CCC2)=O)CCCC(N(C)C(c2coc(Cl)n2)=O)CC1 Cc1ccc(C(=O)NCC2(CNC(=O)CCCC(C)C)CC2(F)F)c(N)c1 N1(C(c2n(C)ncc2C2CC2)=O)CC2(CC2)CC1C(=O)NOCC1CCOCC1 c1(OC)cc(C(=O)NCC2C(C)CCN2C(=O)C2CC2)cc(OC)c1C N1(C(c2ccc(OCC)cc2)=O)CC(O)C(O)C1CNC(=O)Cc1c[nH]nc1O C1(C(=O)Nc2cn(CC)nc2C)CC(NC(=O)C(C)CC2CCC2)C12CCC2 c1(C(N(CCCF)CC)=O)cc(CCNC(=O)CC2CCCCO2)on1 C1(C)(C(N2CCC(CCC(=O)NCC(C(C)C)O)C2)=O)CCCOC1 CCC(C)CCC(=O)N1CC(NC(=O)CS(=O)(=O)NC(C)(C)C)CC1COC CCCCC(C)CCC(=O)NC1(CC)CCCN(C(=O)Cc2ccc(F)cc2)C1 C12(C(=O)NCc3cn(C(c4cccc(C)c4)CC)nn3)CCC(C)(C1)OC2 c1(C(=O)NC(CNC(CCC#C)=O)C(C)C)cnc2ccc(Br)cc2c1 c1(NC(CN(C(C)CC)CCC)=O)ccc(OCC)c(OC)c1Cl CCC(C)C(O)CC(=O)N(C1CCN(C(=O)CN(C)C)C1)CC c1(NC2C3CC(CCNC(C(c4ccc(C)cc4)O)=O)CC32)nc(C)cc(C)n1 C12(CNC(C(C)C3CC3)=O)CC(NC(=O)CC3NC(=O)NC3=O)(C1)C1(CCC1)O2 c1(CCC(=O)NC2(C)CCN(C(C3(C)CCOCC3)=O)C2)cnc2ncccn12 c1(C(CN(C(c2ccc(N3CCNC3=O)cc2)C)C)=O)cnc(N(C)C)nc1 C(=O)(CC(C(C)C)c1ccon1)N1CCCC(C(NOC(C(C)C)CO)=O)C1 N1(Cc2scc(C)n2)CCN(C(c2cnc(Br)o2)=O)C(C#N)C1 N1(C(Cc2nc(C)oc2)=O)CCC(C)CC1CNC(=O)C(C)S(C)(=O)=O N1(C(C2CC(C)OC2)=O)CC2(CCN2C(c2ccc(CO)c(F)c2)=O)C1 C1(CNC(C(C2CC2)SC)=O)CC(C(=O)N2CCSCC2C2CC2)=NO1 CC(C)CC(Cn1cc(-c2cnn(C)c2)nn1)NC(=O)Cc1ccno1 N1(C(CCS(C)(=O)=O)=O)CCCC2(CCCN2C(=O)Cc2ccc(Cl)s2)C1 Cc1ccc2c(=O)c(C(N3CCN(CCC4CCS(=O)(=O)C4)CC3)=O)c[nH]c2c1 N1(C(c2c(OC)scc2)C(=O)Nc2ccc(Cl)cc2F)CCC2C(C1)C2(F)F c1(C(=O)NC(CCCC)CCCC)cc(F)cc(C)c1[N+](=O)[O-] C(=O)(CC(O)CNC(=O)Cc1cn[nH]c1)NCC1CC(C)(O)C1 C=CCC(C)(C)CC(=O)N1CC(O)CCC1C(N1CC(S(N)(=O)=O)C1)=O c1(C(N2CCC(=CCNC(C(CCSC)OC)=O)CC2)=O)cc2ccccc2[nH]1 C1(NC(=O)CCc2ccnc(Cl)c2)CC2CCC1N(C(=O)C=Cc1ncc[nH]1)C2 c1(CC(=O)NC(C2CC(C(F)(F)F)C2)C)nc2ccccc2n1CC(F)F CC(C)CS(=O)(=O)CC(=O)NC(C1CN(C(c2cc(F)ccc2O)=O)C1)C c1(C(=O)NC2CC(CC(N3CCCC(CC)C3)=O)C2)ccc2[nH]ccc2c1 CC(=O)C(C)CC(C)C(=O)NC(CCC(C)C)C(=O)NC(c1ccc(C)cn1)C Cc1cccc(C(=O)NC2CC2C2CCCC2)c1I c1(NC)cccc(C(F)(F)F)n1.c1(NC(CN)=O)ccccc1Cl CCC(C)CCCC(=O)NCCOCCOCCNC(c1ccsn1)=O C(C(C)(C)NC(=O)C(C)c1cccs1)NC(C=C(C)Cl)=O c1(C(N2CC(C)C(NC(=O)C(C)NS(C)(=O)=O)C2)=O)ccc(C(F)F)c(F)c1 C1(NC(CC=CCNC(CCn2c(C)ncc2)=O)=O)C(C)(C)C1(C)C CC(C(=O)NC12CC(C1)N(C(=O)COCCc1ccccc1)C2)S(C)(=O)=O CC(CCNC(=O)Cc1csc(C(F)(F)F)n1)CCNC(=O)CS(N)(=O)=O C1(C(=O)NCC(F)CNC(C2(F)CC2)=O)CCN(c2ccccc2)C1 C1(CNC(c2cn(CCOC)nc2)=O)CN(C(=O)C=C(C)Cl)C2CCCCC12 c1(C(=O)NC2CCC(N(C(c3c(C)ncn3C)=O)C)CC2)cc(Cl)ccc1F C1(C(=O)NC2CCC(CNC(C=CC(=O)N(C)C)=O)O2)CCC2(CCC2)C1 N#Cc1ccc(S(=O)(=O)NCC2CC3CCCCN3C2)cc1NCCS(=O)(=O)NC c1(CC)nccn1C(C)CC(=O)N1CC=CC1CNC(=O)CC1CC2(CC2)C1 C12(CNC(C(c3ccc(Cl)cc3)C)=O)CCC(CC1)N2C(c1scnc1Cl)=O Cc1c(NC(C2CCCCN2C(=O)CCCCCCBr)=O)cc(Br)cc1[N+](=O)[O-] c1(C(N(CC(C)NC(=O)COC(C)(C)CC)CC)=O)ccc(C(=O)N(C)C)cc1 c1(Cc2nnc(Cc3n(C)cc(Br)c3)o2)ccc2c(c1)COCC2 CC(C)(C(=O)NCCC1(O)CCC1)C1=CCN(C(C2CC=CCO2)=O)C1 c1(C(=O)NCC(CCNC(=O)CCC2CCN(C)C2)OC)ccc(C)cc1O C1(NC(c2ccc(C(=O)OC)o2)=O)CS(=O)(=O)CC1NC(=O)CCCF CCCCC(C)C(=O)NCCN(C(=O)CCc1cnn(C)n1)Cc1cccnc1 C(=O)(C(F)(F)CCn1ccnn1)N1CC2C(CNC(=O)Cc3ccsn3)(C2)C1 C1(O)(C(C)NC(CN(C(C)=O)C)=O)CCN(C(=O)CC2(C)CCC2)C1 C1(n2cc(C(CC(N)=O)CC)nn2)CN(C(=O)C(C)N(C)C)CCC1C(F)(F)F C1(C(=O)NC(C(=O)NC(CC)COC)CCC2CCC2)CC(=O)CC12CCC2 N1(C(=O)CC2CCCOC2)CC2(CCN2C(c2cn3ccnc3s2)=O)C1 Cc1ncc(NC(=O)NCc2csc(C(F)(F)F)c2)c(C(C)C)n1 N1(C(CN2CC(C)C2)=O)CCC2(CC1)CC2NC(=O)C(c1cc(F)ccc1F)C N1(C(C(C(=O)OCC)F)=O)CC2(CCC2)CC1CNC(c1coc(Br)n1)=O C1(NC(c2cc(C(C)C)no2)=O)CCOCC1NC(c1ccc(C(C)O)cc1)=O c1(C(C)C(=O)NCC(C)(O)CNC(C2(CC3CC3)CCC2)=O)ccc(Br)cc1 C12(CNC(C3C(C)OCCO3)=O)CCC(CC1)N2C(C1(CC2CC2)CCC1)=O Cc1cccc(C(=O)NC2CCCC2NC(C2CC2C)=O)c1C#N C1(CNC(C(C)OCC)=O)CCC2CN(C(c3ncccc3N)=O)CC12 Cn1ncc(C(=O)NC2CC(O)(Cn3cc(C4CCCCC4)nn3)C2)c1F N1(C(C2CC=CC(NC(=O)C=CCO)C2)=O)CC2COCC(C2)C1 C(=O)(CCCCCCCO)N1C(C(=O)NCc2nccnc2Cl)CC2(CC2)C1 Cc1nc2nccc(C(=O)NCC3CCN3C(c3csc4cccnc34)=O)n2n1 Cc1ccc(C)c(C(=O)NC2CC(CNC(=O)CS(N)(=O)=O)C23CCC3)c1 C1(CC(=O)NC2CN(C(c3c(C)cnnc3)=O)C2)CCCC(F)(F)C1 N1(C(C(CC)=CCCC)=O)CCC2CCCC12C(=O)NOC(c1n[nH]c(C)n1)C C(=O)(C1=CC2(CCOCC2)C1)NC(C1CCN(C(c2c(SC)cn(C)n2)=O)C1)C CCS(=O)(=O)C=CC(=O)NC1CC(C)N(C(=O)CCc2nnc(C(C)C)o2)C1 C(CC(O)C(=O)NCCCc1ccccn1)NC1(C)CCCC1 N1(C(=O)OC(C)(C)C)CC2CN(C(=O)CC34CCC3CN(C(C)=O)C4)CC2C1 C1(CNC(c2c(C)nc(O)[nH]2)=O)CC(C)(C)CN1C(c1nn(C)c(N)c1C)=O FC1(F)C(CN=c2ccnc(N3CCC(C4CC4)C3)[nH]2)C12CCOCC2 C1(CCNC(C(=O)Nc2ccc(C(=O)NC(C)C)cc2)=O)COCC2(CCC2)O1 C=C(Cl)CC(C(=O)NCC1(F)CCOC1)NC(=O)C(C)NC(=O)C1CC1 C1(C(N(OCC(=O)OC)C)=O)CCC2(CC2)N1C(=O)CC1CC2C=CC1C2 C1(NC(C2(S(C)(=O)=O)CC2)=O)CC2CCC1CC2NC(C1CC=CCC1)=O c1(N2CC3CC(NC(c4c(SC)nccn4)=O)C3C2)c(C)c(C)nc2ncnn12 C(=O)(C1=CCC(NC(=O)CC2C=CCC2)C1)N(C(C#C)C)C N1(C(C2(CC=C)CN(C(=O)C(c3ccn(C)n3)C)C2)=O)CC(C)SC(C)C1 c1(-c2nc(-c3ccc(C)cn3)on2)nc(-c2ccc(OCCBr)cc2)cc(O)n1 CC(C)CC(O)C(C)C(=O)NCC1(CC(N2CC(N=[N+]=[N-])C2)=O)CC1 c1(CNC(CSC)=O)ccc2c(c1)CCC2NC(c1nsc2ccc(C)cc12)=O N1(C(C)=O)C2CCC1CN(C(=O)Cn1cc(-c3c(O)nnc(C)c3C)nn1)CC2 c1(OC)ccc(C(=O)NCCCN(C(=O)C(C)OC)C(C)C)c(OC)c1 C1(CC(=O)NCC2(CSC)CC2)CCCN1C(c1cnn(C(F)F)c1)=O Cc1nn(-c2ccccc2F)c(C)c1NC(C1C(C)C1(F)F)=O c1(CCC(=O)NC(CCNC(C2(F)C(C)OCC2)=O)(C)C)ccc(Cl)cc1Cl N1(C(c2c(NC)scn2)=O)CCC(C=CC(=O)NC2CCC23CCCC3)CC1 n1(CC(=O)NCC(C)CN(C)C(C2(C#N)CC2(C)C)=O)cc2ccccc2n1 C(c1c(F)cccc1F)=CC(=O)NCc1cccc(CNC(c2cncs2)=O)c1 c1(OC)ccc(C(=O)NCC(C)(CC(C)C)NC(c2cc(C)c[nH]2)=O)cc1Cl CON(CCC(=O)Nc1ccc(F)c(C#N)c1)C(=O)c1ncc(C)cc1F N1(C(c2cn(CCOCC)nc2)=O)CCCC1(C)CNC(C1CCCN1C)=O C1(OC)CCC(CO)CC1.C12CN(CCO1)C(=O)C(C1CC1)NC(=O)C21CC1 N1(C(Cc2c(C)ocn2)=O)CCC(C2CC2)C1Cn1cc(COCCO)nn1 C1(NC(=O)CCCN2CCCCC2)CCN(C(=O)CC2COCC2O)CC1O Cc1cncc(CC(=O)NC(C)(CNC(c2cnccc2N(C)C)=O)CO)c1 S(=O)(=O)(c1ccc(C#N)c(N2CCCN(C)CC2)c1)NCCC(CC)(C)C N1(C(CC2(C)CCOCC2)=O)CC(CC(=O)NC(CO)CCF)C2(CC2)C1 C1(CCOC)(NC(=O)C(N2CCC(C)C2)=O)CCN(C(c2cnns2)=O)C1 Cc1nc(C)c(C(=O)NC(C)(CNC(C2CCOC2(C)C)=O)C2CC2)s1 c1(C(=O)NCCN(C(c2cnc(C(F)(F)F)s2)=O)CC)ccnnc1S C1(CNC(C(CC)(C)C)=O)CCC2CN(C(C3CS(=O)C3)=O)CC12 C12(CNC(C(C)OCCCC)=O)CN(C(=O)C(=O)N(C)C)CC1CS(=O)(=O)C2 N1(C(c2sc(C(=O)OC)c(N)c2)=O)CCC(F)C(NC(c2ccnc(S)c2)=O)C1 C1(CNC(c2c(NCC=C)cccc2)=O)CCN(C(C2C3CCCC23)=O)C1(C)C Cc1cccc2c1OC(C(N1CCN(C(C3CCCC3)=O)CC(C)(C)C1)=O)C2 C(=O)(C(C)(C)C(=C)Cl)NC1CC(OCC(N2C(CC#C)CCC2)=O)C1 C=CCCCC(=O)N1CCC(N(C(=O)C=C(C)c2ccco2)C)CC1 C1(CC(=O)NCC(C2CCN(C(C(C)NC(C)=O)=O)CC2)O)CCCC(F)(F)C1 CCCC(CC(=O)NOCC(O)CO)NC(c1cccc(F)c1)=O Cc1noc(C)c1C(=O)NC1CN(C(=O)CCOC2CC2)CC1n1ccnn1 C1(CCOC)(NC(C(CCC)N(C)C)=O)CCN(C(C2NC(=O)OC2C)=O)CC1 CCCCC(C(=O)N1CCCC(C)C1CNC(=O)C(C)(C)n1cnnn1)C(C)C C(CC(O)CO)N(CC)CSC1(C)COC1 C1(C(=O)NCC23OCCC(NC(=O)CC4CCC4)(C2)C3)CCC(=C(F)F)CC1 C(=O)(CC(C)(O)C=C)N1CC(CC=C)(NC(C2CC2C2CCC2)=O)C1 C1(C)(NC(C(C)NC(c2ccco2)=O)=O)CCCN(C(=O)Cc2ccns2)C1 N1(C(C2(CC#C)CCOCC2)=O)CCC(C(F)(F)F)C(NC(c2cnsn2)=O)C1 CC(C)(F)C(C)(F)C(=O)NCC1(F)CCCN(C(c2ccc(C#N)s2)=O)C1 O=C(C(c1cccs1)C1CCCC1)N(CCCNC(=O)C1CC1)CC1(Cl)CC1 C(=O)(CC(=O)NC1CCN(C(=O)C2CC2)C1)OC.C12COCC1N2 C(=O)(C(C)CCOC)N(CC(C)NC(C1(CC#C)CCC1)=O)C C(CCC(C(=O)NC1CC(CO)(CO)C1)NC(C1CCC(O)CC1)=O)OC CN1CCCC1(C)CCN=c1ccn2ncc(S(=O)(=O)NCCCSC(F)F)c2[nH]1 N1(C(C2CC(F)(F)C2)=O)CC2OCCN(C(c3cc(O)n[nH]3)=O)C2C1 CCC1=C(C(=O)NC(CC(=O)N2CCC(O)CC2C2CC2)C(F)F)CCCO1 c1(C(=O)NCCNC(Cc2c(C)ccnc2)=O)cc2c(F)c(F)ccc2[nH]1 CC1C(NC(=O)C=Cc2cocn2)CC2CCC1N2C(c1cccc(N)c1F)=O Cc1c(F)ccc(CNc2cn(C)c(C(=O)NCc3ccc(O)nc3)n2)c1Cl Cc1cc(N2CCOC(C)(C)C2)ncc1S(=O)(=O)NCC1CCC=CCCC1 N1(C(c2c(C)scc2)=O)C2CCC1C(NC(c1cnc(Br)c(O)c1)=O)C2 N1(C(c2n(C=C)nnc2)=O)CC2(CO)CC1(C(=O)NC1(COC)CC1)C2 CCN=C(NCc1conc1CC)NCC(c1ccsc1)C C(=O)(C1=NNC(C(F)(F)F)C1)NCC1C(C)CN(C(c2ccsc2Cl)=O)C1 CCC(C)(C(=O)NC1CCCCC1NC(=O)C(O)C(C)C)C(N)=O C1(NC(C(C(C)O)C)=O)CC2CN(C(c3cnn(CC4CC4)c3)=O)CC12 c1(OC)cc(F)c(Br)cc1-n1cc(C2(C)CN(C(=O)C(C(C)C)OC)C2)nn1 C1(CCC(=O)N(CC(C)CNC(C2(n3cnnn3)CC2)=O)CC)CC(F)(F)C1 c1(NC)ccc(S(=O)(=O)N2CCCC(CCN(C(C)COC)C)C2)cn1 c1(CC(=O)NC2C(C)CN(C(c3coc(Br)c3)=O)C2)cccc(N=[N+]=[N-])c1 C1(CN(C2CN(CC)C2)CC)CCCC(C)C1.c12nccc(n1)N(C)C2 C(=O)(C(C)(C)C1CCC1)N(CCCOCCNC(CCOC(C)=O)=O)C C=CC1OCCC1C(=O)NCC(CCC)NC(c1ccc(CO)cn1)=O N1(CCOCC)CCN(C(c2cc(C3CCCC3)no2)=O)CC1 C(=O)(C=CS(C)(=O)=O)NC(C1CCN(C(C2C(CC)C2)=O)C1)C CC1CN(C(=O)Cn2ccc([N+](=O)[O-])n2)CC(C)CN1C(C12CC(F)(C1)C2)=O CCCC(CCCO)C(=O)N1CCC(CNC(c2cc(O)n(CC)n2)=O)C(C)C1 c1(C(N(CCNC(C2(F)CC2C)=O)CC)=O)scc(Cl)c1Cl C1(CNC(CC=CC=C)=O)CCCCCN1C(=O)CC1(OC)CC1 CC(CC(N)=O)C(=O)NCCCCCNC(C1(C)COCCO1)=O C(=O)(C1=CCCCC1C)NCC1(O)CCN(C(c2cnc(CC)nc2)=O)C1 N1(C(c2cc(CC)on2)=O)CCN(C)C(CNC(=O)Cc2cnns2)C1 c1(C(=O)NC(C)C(C)(C)NC(=O)C=CC2CCOCC2)ccc2c(c1)CCC2 Cc1cc(C(=O)N(C)C)ncn1.C1(=O)C(C)C(C)NC(=O)C2(CC2)CN1 S(=O)(=O)(c1ccc(C)c(C(N2CCN(C(=O)CCCCOC)CC2)=O)c1)NC C1(CNC(CC=C)=O)CCN(C(C2CC2C(=O)NCCO)=O)C12CC2 CC1CN(C(=O)C2=CSCS2)CC1NC(=O)CCCOc1ccc(Cl)cc1 C1(CNC(C2N(C(CC)=O)CSC2)=O)C(C)CCN1C(=O)Cc1cnoc1 N1(C(C2=CCCC2C)=O)CCCC2(C1)CN(C(c1cc3scnc3[nH]1)=O)CCO2 C12(NC(CC3CCN(C)C3=O)=O)CCC(CC1)N(C(C1(F)CCCOC1)=O)C2 O=C(C1=CCCCC1)NC1(C2CCCN2C(=O)C=Cc2cncs2)CC1 C1(C(=O)NC2(C)CCN(C(CNS(CC)(=O)=O)=O)C2)CC(=O)N(C)C(=O)N1 N1(C(CCCC#C)=O)CCC2(CC1)CC(NC(C1(C)CCC(=O)NC1)=O)C2 CC1OC2(C)CC1(C(=O)NCCCCCCNC(=O)Cn1nnnc1C1CC1)C2 C1(C(=O)NCC(C2CCC2)NC(c2c(C)noc2C2CC2)=O)CC12CCSCC2 N1(C(CCCC)=O)CC(C(F)(F)F)CC1CNC(c1ccnc(C(F)(F)F)n1)=O O(NS(=O)(=O)c1cc(Br)ccc1C#N)CC(=O)NCCN(CCCC(=O)NC)C c1(NC(CSC)C)ncc(C(=O)O)cn1.c12nc(co1)C(=O)NC2 c1(C(N2CC3C(NC(CC(C)C4CC4)=O)(C3)C2)=O)ccnc2ccc(O)cc12 n1(C(CC)CC)ncc(C(N2CCC(C)C2CNC(=O)C2=CCCO2)=O)c1C c1(C(N(C2CCN(C(CCC(C)SC)=O)C2)C)=O)cccn2c(C)nnc12 CC1CCC(NC(c2nnc(S)n2C)=O)CN1C(c1ccc(N)cc1Cl)=O N1(C(CCCN(C)C)=O)CCC2(CC1)C(N(C)C(c1n[nH]cc1Cl)=O)CS2(=O)=O N1(C(=O)Nc2cc(-c3ncccn3)ncn2)Cc2n[nH]cc2C1CO C12(CNC(Cn3c(C(C)C)nnn3)=O)CCC(CN(C(C3(C)CC(C)C3)=O)C1)C2 C1(C(N2CCC(CC(=O)N(CC=CC)CC)C2)=O)CN(C)C(=O)N1 c1(C(=O)NC2CC3CC2N(C(=O)CCCc2cccs2)C3)cc2cnccc2o1 C=CCC(F)(F)C(=O)N1CCC(c2cn(C(C)(CSC)C(=O)O)nn2)(OC)CC1 c1(OC)ccccc1CC(=O)NC1CC(CNC(=O)C(O)C(C)SC)C1 S(=O)(=O)(C1CS(=O)(=O)c2ccccc21)N(CC(F)F)CC C12(C(N(CC)CC3CCCCN3C(=O)CC3CCC3)=O)CCC(F)C1CC2 C=C(Cl)CC(C(=O)NC(CCCOC)C(=O)OC)N(C1(C)CCC1)C C=CC(C)(CC)C(=O)NCC(=O)NCC(N1CCC(COC)CC1)=O N1(C(C(CCCC)C)C(=O)NC(C)C)CCC2(CC1)CCN(C)C2 C(=O)(CCCC(C)(F)F)N1CC2(CC(NC(C(N3CCN(C)CC3)C)=O)C2)C1 c1(C(=O)NCC(C(=O)N(CC(=O)N(C)C)CCC)O)ncnc(O)c1F C1(N(C(=O)CC2CCCOC2)CC#C)CCN(C(=O)CCCOCC=C)CC1 c1(C(N2C(C(=O)NC(C(C)C)c3cccs3)CC(F)C2)=O)cc(Cl)cc(Cl)c1 c1(C(N2CCC3C(C(=O)NCC(CC)(C)CO)C3C2)=O)cnn2ccc(Cl)c(F)c12 c1(C(N(C2CCC(NC(c3c(C)noc3C)=O)CC2)C)=O)ccc(F)c(F)c1N N1(C(C(C)CN(C)C)=O)CCC2(CC1)CCN(C(C1Cc3cccnc3C1)=O)C2 c1(OCC)ncccc1NC(c1nc(C)sc1OC)=O N(C1CS(=O)(=O)c2cc([N+](=O)[O-])ccc21)C(=O)NC(C1CCC1)C1CC1 CC(C)C(C(C)NC(c1nn(Cc2ccccc2)cc1Cl)=O)NC(C1(C)CC1)=O c1(C(N(C(CCNC(C(CC(C)C)O)=O)C)C)=O)cn(C)c2c(Cl)cccc12 CC(C)(C)C(C)(C)C(=O)N1CC(CNC(=O)C(F)(F)CCn2ccnn2)C1 N1(C(CCN(C(C)=O)C)=O)CC(CO)C2(CCN(C(=O)C(C)C(C)(F)F)CC2)C1 N1(C(C(C)(C)OC)=O)CCCC(C(=O)Nc2ncn(C)n2)C1 CC1(C)Cc2cc(S(=O)(=O)Nc3cccc(CO)c3C#N)sc2C1 C1(NC(c2ccon2)=O)CN(C(=O)COCC2CCOC2)C2(CCC2)C1 c1(C(=O)NC2C(CNC(C(c3ccccc3)C)=O)C2)cnc2scnc2c1 c1(OC)ccc2nc(N3CC(CO)C(C)C3)[nH]c(=NCC(C)S(N)(=O)=O)c2c1 c1(CNC(C(=O)NCCNC(C2CC2(F)F)=O)=O)cc(-c2ccccc2)cs1 c1(N(C)C2CC2)nc(N2CC3CC=CCC3C2)nc2c1CCC2 c1(C(=O)NC2CC(CNC(C3C(C(C)(C)C)CC3)=O)C2)cccc2c1C(=O)NC2 C1(CNC(C2C(SC)CCC2)=O)(NC(=O)CC2CCCCCC2)CCCCC1 C(CCCC(C)NC(=O)C=Cc1cnn(C)c1)NC(C1(CCC=C)CCCC1)=O c1(NC(=O)NCC2(Sc3ccncc3)CC2)c(F)cccc1[N+](=O)[O-] CC1CN(C(=O)CCS(C)(=O)=O)CCCN1C(c1c(N)cc(Cl)nc1Cl)=O N1(C(c2c(CC)cccc2)=O)CC2CCN(C(c3cc(F)cn3C)=O)C2C1 c1(CCC(=O)NCC(C)(C2CC2)NC(COCCOCC#C)=O)cccc(C)c1 N1(C(CC(CC)(F)F)=O)CC(C)N(C(c2c3c(nn2C)CCC3)=O)CC1C C1(NC(Cc2cc(OC)no2)=O)CCCCN(C(c2csc(Br)c2)=O)C1 CCC(CC)CCC(=O)NC(C)CCNC(=O)CSCCOC Cc1[nH]c2ccccc2c1C(N1CCC(NC(c2cc[nH]c2C)=O)C(C)C1)=O c1(C(=O)NCC2C(CCC)C2)n[nH]cc1CNC(c1cnco1)=O Cc1nc2ccccc2nc1C(=O)NC1CCC2CC1CN2C(C1CCC1)=O Cc1nc(C2CCC2)[nH]c1C(=O)NC(C)(C)C(C)NC(=O)CSCC(C)C C1(NC(C2N(C(COC)=O)CCC2)=O)CCCC12CN(C(=O)OC(C)(C)C)C2 c1(N2CCC(OC)C(C)(O)C2)ccc(S(=O)(=O)NCCc2cc(Br)cs2)cc1Cl C1(CCNC(C2(C=C)CCCCC2)=O)CN(C(=O)C(C)(C)COC)CCS1(=O)=O Cc1ncnc(C)c1CC(N1CC(N(C(=O)C(c2ncccc2F)(F)F)C)C1)=O CCCN=C(NCC1(C)CCCOC1)NC1CCCN(C(=O)CN2CCCC2)C1 N1(C(=O)OC(C)(C)C)CCCC2C1CCCN2C(c1cncc(F)c1C(=O)O)=O Cc1noc(C)c1CC(N1CCC1CNC(=O)CC1CCC(=O)N1C)=O CC1OC2(C(N3CCCC(CN(C)C(C4CC4C(N)=O)=O)C3)=O)CC1C2 C(=O)(C1CCCc2ccnn21)NCC1CC(NC(c2cnc(C)[nH]2)=O)C1(C)C C(=O)(CCCS(N)(=O)=O)NCCc1[nH]c(=NCc2cn(C(C)(C)C)nc2)sc1 C1(CN(C(C(CSC)C)=O)C2CC2)CC(F)CN1C(=O)CCCN1CCCCC1 C1(CNC(CNC(CNC(C)=O)=O)=O)CCN(C(=O)Cc2csnn2)C1(C)C CC(CC(N)=O)C(=O)NC1C=CCN(C(=O)CC2COC(C)(C)C2)C1 c1(C(=O)NCCN(C(=O)CCc2cscn2)CCOC)cc(C(F)F)[nH]n1 C=CC1(C(=O)NCCOCCCO)CCN(C(C2(OC)CCC(C)C2)=O)C1 CCC(CCC(=O)N1CCC(NC(C)=O)C1)NC(c1cc(COC)[nH]n1)=O CCCCCC(O)CC(=O)N1CC(C)CN(C(C2CN(CC(C)C)C2)=O)C(C)C1 CC1(C)CC(CNC(c2cncc(Cl)c2Cl)=O)N(C(=O)CC2CC3CCC2O3)C1 c1(CC)nn[nH]c1C(=O)N(C(C)CCNC(C1CCCC1C)=O)C c1(C(=O)NCCN(C)C(c2nc(Cl)cc(N)c2Cl)=O)cc(Cl)c(F)cc1F Cc1cc(C(F)F)oc1C(=O)NCC1(O)CCN(C(=O)C(C)c2ccsc2)C1 N1(CCCOC)C(=O)CCN(CCC2CCC(C)CN2C(=O)OC(C)(C)C)C1=O c1(C(N2CC=C(CNC(c3cn(C)nc3)=O)CC2)=O)ccc2cnoc2c1 N1(C(C2C(C)(C)CC=CC2)=O)CCCc2nc(O)ccc2C1 c1(C(C(=O)NCCCF)N(C(C)COC)CC)ccc2nc[nH]c2c1 C1(NC(c2nc(CCC)sc2)=O)CCCC(N(C)C(c2nocc2C(C)C)=O)C1 C1(NC(C2(CCC)CCC2)=O)CN(C(=O)CCS(=O)(=O)NC)CCC1(C)C C(CC1=CCN(C(c2ccnnc2C)=O)CC1)NC(c1cc(OC)ncc1Cl)=O CC(=O)CC(C)(C)C(=O)N1CCC(C)N(C(=O)C#CC(C)C)CC1 N1(C(c2n(C)nc(CNC(C3CC=CCO3)=O)c2)=O)CC(O)C(C)(C)C1 Cc1ncc(CNC(C2(C)CC(NC(=O)C(c3cncnc3)C)C2)=O)o1 c1(CC)onc(C)c1C(=O)NCc1ccc(C(=O)NCc2cc(OC)n[nH]2)cn1 c1(SCC(CC)O)cc(-c2cccn2CC)cc(-c2ccccc2)c1 Cn1cc(C(=O)NCC2CCCN2C(C2CC(C)(C)C2)=O)c(C(F)F)n1 c1(NC(=O)NCCCC2CC(N)C2)cnccc1-c1cccc(F)c1 CCC(CNC(C1C2CCCCC12)=O)(CC)NC(=O)CCOC1CC1 N(C(=NCC(C)C)NCC(c1cccc(F)c1)SC)Cc1nnc(COCC)s1 C1(NC(CCC(C)OCC)=O)CCN(C(c2ccc(CC)c(F)c2)=O)C12CC2 C(=O)(CC1OCCc2ccsc21)NC(CC)CNC(c1cnc(Cl)s1)=O C(=O)(CCCC(F)F)NCC1CC(NC(COCP(C)(C)=O)=O)C1 C#CCC(C)(CNC(c1ncccc1OCC(F)F)=O)CO N1(C(Cc2c(C)con2)=O)CCCC1C1CCCN1C(=O)C1=CCSC1 C1(C(N(C2C(C)C2)C)=O)CCC=CC1NC(=O)C(F)CC1CCOC1 CC1(C)OCCC1C(=O)NC1CCCC(C(N2CCCCC2CCO)=O)C1 C1(C(=O)NC2C=CC(CNC(C(C)=CC)=O)C2)CCc2nc(C(F)(F)F)cn2C1 CCC(CC)C(=O)N(C1CN(C(=O)C=Cc2cnn(C)c2)CC1F)C Cc1cc(C(=O)N(C)CCN(C)C(C2CCOC2C(F)(F)F)=O)ncc1N C1(NCCNC(c2cn(CCC)nc2)=O)CNCC(C)C1 c1(C(=O)NC2(CN(C)C(C34CC3COC4(C)C)=O)CC2)ccc(F)cc1[N+](=O)[O-] C(CCCC(=O)NC)(c1ccccc1)C(C)Nc1nnnn1C1CCC(F)(F)CC1 c1(CNC(CN(C(CC2C(C)=NNC2=O)=O)C2CC2)=O)ccc(F)c(O)c1 Cc1ccccc1OCC(=O)NCC1CCN1C(=O)C(F)C1CCOC1 N1(C(C(c2c(C)noc2C)C)=O)CCCN(C(=O)Cc2ccsc2C)C(CO)C1 N1(C(C2CC(C)OC2)=O)CC2CCCN(C(c3cnc4c(c3)nnn4C)=O)C2C1 C1(S(N)(=O)=O)(C(N2CCC(CN(C)C(c3coc(N(C)C)n3)=O)C2)=O)CCC1 c1(C(N2CCC(N(C(C=CC)=O)CCO)C2)=O)nc(Br)n2c1COCC2 N1(C(C(CC=CC)CC)=O)CC(CO)C2(C1)CN(C(=O)CC(=O)NC1CC1)C2 C(=O)(C(C(C)C)c1cnn(C)c1)N1CC(N(C(CCC=CCC=C)=O)C)C1 c1(C(N2CC(OC)C(NC(=O)Cc3ccns3)C2)=O)c[nH]c2ccc(F)cc12 C(=O)(C(O)C(C)CC)N(CC(CC)NC(C1(CC)CC(F)(F)C1)=O)C C#CC1(C)CCCN(C(=O)CC(C)(C)NC(=O)CC(C)(C)OC)C1 c1(C(N2CC(O)(CNC(c3cc4ccnn4cn3)=O)C2)=O)ccc2c(c1)OCC2 c1(C(=O)NC(c2cccc([N+](=O)[O-])c2)C(=O)O)csc2c(Br)ncn12 c1(C(=O)NCCCCOC)ccc(CNC(C2COC(C)C2)=O)s1 C1(CNC(CCC)=O)CN(C(=O)CCOCC2CC2)CC1c1cncn1C Cc1cc(C(=O)NC2CCCN(C(c3cccc(NS(C)(=O)=O)c3)=O)C2)ccn1 C1(CN(C(=O)CCOCCCN)CC(OCC)OC)CCC(=O)N1C c1(C(=O)NCc2occ(C(=O)NC(c3cnn[nH]3)C)n2)ccnnc1O c1(C(C(=O)N(C2CCN(C(C)C)CC2)C)C)ccc(Cl)c(Cl)c1 C1(C(N(C)CC2(O)CN(C(c3cc(C#N)cs3)=O)C2)=O)CCCCC12CCC2 c1(CC(N2CC(N(C)C(c3csc(O)n3)=O)C2)=O)ccc(F)c(F)c1 c1(NC(C2(OC)CCN(C(C(CCSC)O)=O)C2)=O)cc(CO)cc(F)c1 N1(C(=O)Cc2cnoc2)CCN(C(=O)CNS(=O)(=O)c2cccs2)C2CC12 N1(C(CC(CC)C)=O)CCC2(C1)c1ncn(C)c1CCN2C(c1ccsn1)=O C1(C(=O)NCCC2CC(NC(=O)C(OC)OC)C2)(OCC)CCCCCC1 N1(C(C)=O)CCOCC1C(=O)NCCCN(C)C(c1sccc1C)=O c1(OC)nc(Nc2ccc(NC(=O)Cn3nc(C)c(Cl)c3C)cc2)ncc1Br C1(C(=O)NC2CNC(=O)C2)(CC)CCCN(C(=O)CCSC)C1 N1(C(C(C)NC(=O)OC)=O)CC(NC(=O)CCS(C)(=O)=O)CC12CCC2 C(=O)(CC1=CCN(C)CC1)N(CCCNC(c1c(CC)cccc1F)=O)C C(C(CC)n1cccn1)N(CCC#C)C(=O)OCC.C(C)(C)(C)O N1(C(CCC(=O)OCC)C)CCOCC(C(=O)NCC(C2CCCC2)OC)C1 C(=O)(CC1COc2ccccc21)N1CCCN(C(Cc2c(C)cccc2)=O)CC1 CCCC(C)CN(C(=O)CC1C=CC(NC(=O)C(C2CCOCC2)=O)C1)C n1(CC)cc(Cl)c(C(C(=O)NC2(C)CC2)N(C(COC)C2(CC)CC2)C)n1 c1(OC)cc(C(=O)NC2(C3CCN(C(c4ccccc4F)=O)C3)CC2)c(F)cn1 c1(CNC(=NCc2cncc(OCC)n2)NC2CCC2)cc(I)ccc1Br N1(C(CCCC(=O)N(C)C)=O)CCC2(NC(C3CCCC34CC4)=O)CCCC12 c1(-n2c(C)cc(C)n2)cccc(O)c1NC1CCC(C)C(C)C1=O C=CCCC(C(=O)NC1CC(C)(C)OC1=O)NC(=O)CC1CCC=CCC1 C(=O)(C(COC)CC(C)C)N1CCC(O)(CNC(CN(CCC)C)=O)C1 C1(CC(=O)NC2(CNC(=O)OC3CCCCCC3)CCOC2)CCC2(CCC2)O1 S(=O)(=O)(c1ccc(N2CCCC(N3CC(O)C3)C2)c(Cl)c1)N(CC=C)CCO c1(OCC)ccc2cc(C(N3CCC4C(NC(c5csnn5)=O)CC34)=O)[nH]c2c1 N1(C(c2c(OC)ccs2)=O)CC2CCN(C(c3cnn(-c4nccs4)c3)=O)CC12 N1(C(C2=CC(C)(C)C2)=O)Cc2n[nH]cc2C1C(=O)NC1CC(C2CC2)C1 C(=O)(CC(C)C(=O)N1C(CC(=O)N(C)Cc2ccn(C)n2)C2CCCC12)OC c1(OCC(N2CCCC(C#C)CC2)=O)c(C)sc2nc(C(C)C)nc(O)c12 Cn1c(=N)[nH]c2cc(C(=O)NC3CC4(C3)CC(NC(C3CC3F)=O)C4)ccc12 C1(NC(C=CS(C)=O)=O)CS(=O)(=O)C2CN(C(c3ccnc(O)c3)=O)CC12 c1(C(=O)NCC(C)N(C(C(n2ncc(C)c2)C)=O)C)ccc2snnc2c1 C1(COC)CCCCN(C(=O)CCC2CCCCN2C(c2cccc(=O)o2)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)NC(CC=C)CNC(C1CCCCCCC1)=O c1(C(N2CC(NC(c3c(OC)ccnc3)=O)C2)=O)ccc(C#N)c(F)c1Br N(C(=NCCC(=O)N1CCN(CC(C)C)CC1)NC1CC2CCC1O2)C(CC)C CC1CN(C(c2cc(CN(C)C)on2)=O)CC1(C)CNC(=O)CSc1nc[nH]n1 c1(CC(=O)NC(C(C)(C)C)CNC(C2(CO)CCC2)=O)ccc2nonc2c1 C1(CNC(c2nc(C)n(C)n2)=O)COCCN(C(=O)CCc2ccsc2)C1 c1(C(N2CC(C3CCN(C(C(CC)(F)F)=O)C3)OCC2)=O)cccc2cnnn12 C1(NC(c2cccc(C#C)c2)=O)CCC12CCN(C(=O)CC1C=CCC1)CC2 C(=O)(C(C)N=c1cc[nH]cc1)NC1CC(O)(CNC(C(C)OCC)=O)C1 C(=O)(CCCCC(=O)NC(C1CCN(CCCOC)CC1)CC(=O)O)NC c1(NCC(N(C(=O)CCc2csc(=N)[nH]2)CC)C2CC2)cc(OC)ccc1OCC C1(NC(C=C2CCC(C)CC2)=O)CN(C(C2(C#N)CC(C)C2)=O)CC1(C)C c1(C(N(C)CCN2CCN(C(C34CC5CC3C4C5)=O)CC2)=O)coc2c1CCCC2 c1(CNC(CSCCCC)=O)cn(C2CCN(C(=O)C(C)CF)C2)nn1 N1(C(Cn2c(C)nnn2)=O)CCN(CC(C)NC(=O)CC2(C)CCCO2)CC1 C1(C(C)C)(C(=O)NC2(CC3CCC3)CC2)CCN(C(=O)Cn2cnc(=N)[nH]2)C1 C12(NC(C(C)CF)=O)COC(C1)C(NC(c1csc(-c3ncccc3F)n1)=O)C2 N1(C(C2(CC)CCCN2C(c2cccc(C)c2O)=O)=O)CC2(CNC(=O)C2)C1 Cc1cc(F)cnc1C(=O)NCc1nc(C(=O)N(C)CC2CC2C)co1 c1(C(=O)NC2(c3ccccc3)CCN(C(COC(C)=O)=O)C2)cncc(C)c1Cl C1(NC(c2c(CC)con2)=O)CN(C(=O)CNC(=O)OC)CC2(CCC2)C1 N1(C(C(C)C2CC2)=O)CCC(O)(C(C)NC(=O)Cc2cncnc2O)CC1 C(=O)(C(C)CC(C)(C)C)NCC(C(N1C(CC)(CO)CCC1)=O)C C1(C(=O)NC(CN(C(c2c(SC)scc2)=O)C)(C)C)Cc2ccccc2O1 C1(C(N2CCCC(NC(c3cnnc(O)c3)=O)C2)=O)CC(C2CC2)=NO1 c1(SCC(N2CC(CC=C)(NC(=O)CC(C)C)C2)=O)ccc(C)c(C)c1 N1(CC(=O)N(C(CC(C)C)C)C)CC(NC(=O)C(C)(C)C2CC2)CCC1C C(=O)(CC1=NN(C)C(=O)C1)NC1C(C(N2C3CC(CC(OC)C3)C2)=O)CCCC1 CC1CC(C(=O)Nc2ccccc2O)CCN1C(C1CCCCCCC1)=O C1(NC(CC2ON=C(C)C2)=O)CCN(C(c2c[nH]c(=N)c(C)c2)=O)CC1O N1(C(c2ccn(CCC)n2)=O)CC(NC(=O)C(C)CCO)C(C)(C)C1 N1(CC)CCC(ONC(C2C=CCN2C(=O)CCc2cnn[nH]2)=O)CC1 C1(NC(COCC#C)=O)CC(C(=O)N(C2CN(C3CC3)C2)C)C1(C)C C1(O)(C(=O)NC(CC(C)NC(c2c(C)n(C(C)C)nn2)=O)C)CCCCCC1 C1(C(=O)NCCC(=C)CNC(=O)C(F)(F)c2cnn(C)c2)CCCC(O)C1 Cc1cccc2c(C(=O)NC3C4CC3N(C(C3(C(F)(F)F)CC3)=O)C4)cccc12 c1(OC)cc(C(N2CCC(C(C)NC(c3cc(C)nn3C)=O)CC2)=O)cc(F)n1 C(=O)(C1=CCSC1)NC(CNC(=O)CC1(C(F)F)CC1)CO c1(C(N(CCOCC)C)=O)c(F)cc(NC2CC(CN)C23CCC3)cc1F c1(C(=O)NC(CCCNC(c2cc(CC)cc(Cl)c2)=O)C)cc(N)c(C)cc1C C1(CC=C)CCCCN1c1cc(N2CCC(C(F)(F)F)(CO)C2)ncn1 CC1CCCC(CC(=O)NC2(CF)CCN(C(=O)CCn3cccn3)C2)O1 Cc1cc(Br)ccc1NC(N(C1CN(c2nncs2)C1)C(C)(C)C)=O C1(CC(=O)NCCCC(C)NC(C(C)N(CC)CC)=O)C(C)(C)C1(C)C C1(C(=O)NCC(c2ccccc2)NC(Cc2cnc(C)s2)=O)CCC(=O)N(C)C1 Cc1ncc(C(=O)NC2CCC2CNC(=O)CCC2OCCO2)c(C(C)C)n1 Cc1ncc(C(N2CC(C(C)NC(=O)CC3COCCO3)C2)=O)cc1N C=C1C2C1N(CCNC1CC1)C2=O.C(=O)(CCC1CC1C(=O)OC)NC.C=O c1(C(N(CC(C)CNC(c2cc(C(C)(C)C)n[nH]2)=O)C)=O)cnc(N(C)C)nc1 Cc1cc(C(=O)NC(C2CCN(C(C3CC3C3CCCC3)=O)C2)C)cc(O)n1 C1(C(N(CC(O)CN(C)C(C2(C#N)CC3(CC3)C2)=O)C)=O)CCC2CCCCN12 Cc1cc(=NCc2ccc(F)c(F)c2C)[nH]c(=NCC(C)(C)C2CC2)[nH]1 c1(C(C(F)(F)F)Nc2nc(SC)nc(C)c2)ccc(Cl)cc1Cl Cc1c(C(=O)NCCN(C(=O)C(n2nccc2C)C)C(C)C)cccc1C1CC1 N12CCC(F)(C1)CNC(=O)c1nc(cs1)CC2=O.C(=O)(C(C)(C)F)OC(C)(C)C CCC(F)(C(=O)OC)C(=O)NCC(O)CNC(=O)C(C)(C)C1CCC1 C1(NC(CC(C)(C)C)=O)CC2CN(CC(O)COCc3cccs3)CC2C1 C(=O)(CCCN=[N+]=[N-])NC(C(=O)N(CCC(O)CO)C)Cc1cc[nH]n1 C12(C(=O)NC(C)CNC(=O)CC3(O)CCN(C)CC3)CC3CC(C1)CC(O)(C3)C2 N1(C(COC(CC)(C)C)=O)CCN(C(c2nocc2C)=O)CC1C C1(CC=C)(NC(=O)C=COCC)CCCN(C(c2cncc(Cl)c2C)=O)C1 c1(CCCNC(C2N(C(C(C)NC(C)=O)=O)CCCC2)=O)ccc(F)cc1F c1(C(=O)NCC2N(C(c3nc(C)nc(O)c3)=O)CC(F)C2)ccc2c(c1)OCC2 c1(C(N2CCC(C)(NC(C3CCC(C)(C)O3)=O)CC2)=O)cncc2ccccc12 N1(C(C(C)N(C)C)=O)CC(C)(C)CC1CNC(c1coc(N(C)C)n1)=O CC1(C)CC(NC(C2CCCC23CC3)=O)CN1C(=O)CCCN1CCCC1 CC(C)(C)C(O)C(=O)N1CCC(OCCNC(c2ccn(C(F)F)n2)=O)C1 N1(C(=O)NCCc2cc(O)cc(F)c2)CCOc2cc(F)ccc2C1 N1(C(c2scc(OC)c2OC)=O)CCCC(NC(c2cc(N)ccc2O)=O)C1C C1(NC(C2C(CN(C)C)C2)=O)CCC2(CC1)CN(C(c1ccc(F)o1)=O)CCO2 C(=O)(NN1CCCC1C(=O)NC1CC2(CCOC2)C1)C1CC2(CC(OC)C2)C1 c1(NC(C(CC2CCOCC2)NC(c2c(C)ccs2)=O)=O)ccc2occc2c1 C1(C(=O)NCCC2(CNC(c3n(CC)ncn3)=O)CC2)CCCC1P(C)(C)=O C1(C(=O)OC)CCN(C(C)C(=O)NCc2ccc(Br)cc2OC(C)C)CC1C C1(C(=O)OC)CC(F)(F)CN1C(C1CN(C(c2ccc(Br)nc2C)=O)CCN1)=O Cc1cnc(C(C2CC2)NC(=O)NCC(C(C)C)c2ccnn2C)[nH]1 n1(N(C)C)cc(CNC(=O)C(=O)N2CC(SCCC(N)=O)C2)nn1 c1(C(=O)NCCC2(CNC(C(S(C)(=O)=O)C3CC3)=O)CC2)csc2c1CCCC2 N1(C(c2c(=N)cc[nH]c2)=O)CCC2(CCOCC2)C(NC(=O)Cc2ccco2)C1 c1(OC)ccc(CCCC(=O)NC2CC2NC(c2c(C)noc2C)=O)cc1 C(c1ccc(Cl)nc1)=CC(=O)NC1(CNC(C2(C(F)(F)F)CCCC2)=O)COC1 C1(C(=O)N(c2cccc(=O)n2CC(F)(F)F)c2ccccc2F)CCC(F)(F)CC1 CCCCCC(F)C(=O)N(C)CC1CCC(NC(C2(CC)CCCO2)=O)CC1 N1(C(c2ccc(OCC(N)=O)cc2)=O)CC2CC(C1)N(C(=O)CNC=O)C2 Cc1nc2cc(C(=O)NC(CNC(c3occc3C)=O)C(C)C)cc(O)c2[nH]1 N1(C(CCc2ccnc(C)n2)=O)CCC(C)C(NC(c2sc(O)nc2C)=O)C1 Cc1cc(N)c(C(N2C3CCC2C(NC(=O)CCC=CC(C)C)C3)=O)cc1F C(=O)(CCC(=O)N1CCC(CCNC(=O)CCN2CCCS2(=O)=O)CC1)OCC N1(C(C2C(C)(C)C2)=O)CCC(Cn2cc(C3(O)CCCC3)nn2)CC1 C1(NC(C(C2(O)CCCCC2)CC)=O)CN(C(=O)Cn2cnnc2O)C(C)(C)C1 CC(CCc1ccc(F)cc1)C(=O)NC1CC(CNC(C2CCC(O)C2)=O)C1 c1(OC)cc(C)cc(CNCC2CCCN(C(c3ccccc3Br)=O)C2)c1O N1(C(C(COC)OC)=O)CCCC(O)(CN(C)C(c2cnn3c2OCC3)=O)C1 C1(NC(C2(CO)COC2)=O)CC(O)CN(C(C2(F)CC=CCC2)=O)C1 Cc1cc([N+](=O)[O-])ccc1C(N1CCCC(NC(=O)C(N)=O)CC1)=O C1(C(=O)NC(C)CCCNC(C2CC3CC2C2CC32)=O)C2CCC(C2)C1(C)C C1(NC(C=CC=CC)=O)CCN(C(c2cc(C(F)(F)F)cc(O)c2)=O)CC1C c1(C(=O)NC2CCN(C(CCCOCC)=O)CC2(C)C)csc2c(F)cccc12 C1(CC=C)(NC(c2nc(C(F)(F)F)cs2)=O)CCCN(C(=O)C(O)C(F)F)C1 C1(F)(C(=O)NC(C)CN(C)C(C2CCCO2)=O)CCS(=O)(=O)C1 N1(C(C(CC)(C)COC)=O)CCC2CC2(C(N2CC3COCC(C3)C2)=O)CC1 Cc1ccc(NC(c2cccc(NC(=O)Cc3ccc(Cl)c(F)c3)c2)=O)cc1I c1(C(=O)NCCCCCCNC(C(CC#C)C2CC2)=O)ccn2c(C)cnc2c1 c1(NC(CC2C(C)CN(C(C3C=CCC3)=O)C2)=O)ccc(O)c(CO)c1 C(=O)(CC(C(C)(C)C)NC(c1ncc(CC)cn1)=O)N(CCCO)CC#C c1(C(N2C(C)CN(C(C=CC(C)C)=O)C(C)C2)=O)[nH]c2ccc(Cl)cc2c1Cl c1(C(N)=O)cc(=NC2CCCN(C(=O)C3=CCCC3)C2)[nH]c(Cl)n1 C1(C(=O)NCC2OCCC(C)(C)C2)CCN(C(=O)C(Cl)Cl)C(C)(C)C1 O=C(C(O)C(F)F)N1CCCCC1CNC(C1(F)CC=CC1)=O CC1CC(CNC(=O)C(O)CN(C)C)CN(C(c2ccc(C3CC3)nc2)=O)C1 c1(C(=O)NCCC2(O)CCN(C(C34CC(C)(C3)C4)=O)C2)c(F)ccc2occc12 C1(C(C)NC(C2CC(F)C2)=O)CCCCN1C(c1nncn1C)=O CCCCCC(C)NC(c1cccnc1CNC(c1ccncc1F)=O)=O N1(C(C2N(C(C=Cc3n(C)ncc3)=O)C(CO)CC2)=O)CCCC2CCCCC12 c1(C(N2C3CN(C(CCCNC(=O)OC)=O)C(C3)C2)=O)nn(C)cc1S(N)(=O)=O Cc1cc(N2CC3CC2CN3C(c2c(F)cccc2F)=O)nc(-c2cccs2)n1 C=CCC(CNC(c1cnnc(C)c1)=O)C(=O)NC(CC1CC1)C1CC1 N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(c2cn[nH]c2)=O)CC12CCCC2 C1(c2cc(C)no2)COCCC1NC(c1ccsc1)=O C(=O)(C(O)CCCNC(c1ccc(O)c(F)c1)=O)NCC(C1CC1)SC c1(C(=O)NC(CNC(CCOCCC)=O)C(C)C(C)C)cccc2c1CNC2=O c1(C(=O)NC(C2N(C(c3cnc(CC)s3)=O)CCC2)C)cc([N+](=O)[O-])n[nH]1 C1(=O)CCCCCN1.c1(C(N2CC(N(CC)CC)C2)=O)cc[nH]c1C(C)C c1(C(=O)NCC(C(=O)NC(COCC)C)N(C)C)ccn(C)c(=O)c1 c1(C(C)=O)c(N2CC3CC(NC(=O)Cn4cnnn4)C3C2)nc(C2CCC2)nc1Cl N1(C(CCCC(C)NC(CC(CC)(C)C)=O)=O)CC2COC(=O)C2C1 c1(C(N(C2CN(C(CC=C(C)C)=O)CC2F)C)=O)cn2cnnc2cn1 C(CCC(C)CC(=O)OCCCN1CCCC1)=C(C)C Cn1cc(CC(=O)NCCCOCCNC(C2CC2c2ccncc2)=O)nn1 C1(NC(Cc2cc(C)no2)=O)CCC(C(N2CCN(C(=O)C3CC3)CC2)=O)CC1 N1(C(Cc2cnc(C)s2)=O)CCOCC1CC(N1CC(F)C(F)C1)=O C1(C(N2CC(CC(C(=O)N(C)Cc3c(C)ccs3)F)C2)=O)CCC=CCC1 c1(C(=O)NCC2CCCC(CNc3cc(OCC)ncn3)C2)cc(Cl)ccc1F c1(NC(C2(F)CN(Cc3ccc(C)cc3C)C2)=O)cc([N+](=O)[O-])ccc1Br C#Cc1cc(C(=O)NC2(CNC(c3cncc4c3CCC4)=O)CCC2)cc(N)c1 c1(N2C(C)(C(=O)Nc3ccnn4cccc34)CCN2)ncnc2c(F)cccc12 c1(C(N2CC3(CC(CNC(=O)Cc4ccon4)C3)C2)=O)ccc([N+](=O)[O-])c(O)c1 c1(OC)ccc(C(=O)NC(CNC(c2cc(C)n(C(F)F)n2)=O)CO)c(F)c1Cl C(=O)(C#CC1CCCO1)N1CCC(CN(C(=O)C(C(C)(C)C)NS(C)(=O)=O)C)CC1 c1(C(=O)NCCN(C(=O)CCc2cc(F)c(F)c(F)c2)C)c(F)cccc1[N+](=O)[O-] Cc1cc(Cl)ccc1C(=O)NCC(O)CNC(=O)C(C)(C)C12CC(C1)C2 S(=O)(=O)(CCC(=O)NCC1CCCCN(C(=O)C(F)=C(C)C2CC2)C1)NC C1(NC(C(=CC2CCCC2)C)=O)CC(O)CN(C(=O)Cc2n[nH]c(C)n2)C1 C1(NC(C(C)=CC2CC2)=O)C2CCN(C(c3csc(=N)[nH]3)=O)CCC12 N1(c2ncc(CC)s2)C(=S)NC(c2cccc3nccnc23)C2=C1C(C)NC2=O c1(NC2(C)CN(Cc3onc(C)c3-c3nn[nH]n3)C2)ncnc(Cl)c1C N1(C(C(C=C=C)C)=O)CCCC(NC(c2ncn(C)n2)=O)CC1 O(NC(=O)C(c1ccc(C)cc1)NC)CC(=O)NC(C#C)C Cc1[nH]c(C(=O)NCC2CCN(C(c3ccc(C(C)C)s3)=O)C2(C)C)c(C)c1C N1(C(=O)NCC(CC)C(C)C)CCC12CC(C(F)F)C2 Cc1cnc2nc(C(=O)NC3CC(CNC(c4sccc4CC#N)=O)C3)nn2c1 Cc1c[nH]c(C(=O)NCCC2(NC(C3CC(C)(F)C3)=O)CCCC2)c1 NS(=O)(=O)c1ccc(C(=O)Nc2ncc(-c3c(F)cc(O)cc3F)cc2O)cc1 C1(CC(=O)NCCC(C)NC(C(CC=C)CC)=O)CCC2(CC1)OCCO2 C1(C)(C(C)(C)C)CC(=O)N(CN2CCC(N3CCCC3=O)C2)C1=O C1(C(N2C(COC)CN(C(=O)Cn3nccc3C)CC2)=O)Cc2nnc(C)n2C1 CCCC(C(=O)N1CC=CC1C(N1CCC(CCC)C1)=O)N(C)C Cc1ccc(F)c(-c2ccc(C(=O)NCC3CCOC3)cc2)n1 Cc1scc(C(N2CC3CC3(NC(=O)CC3CCOC3)C2)=O)c1Br CCCCCCC(F)C(=O)N1CCN(C(=O)COCC)C(CS(C)(=O)=O)C1 C(N=c1cc(C)nc(C)[nH]1)C1OCCCN(C(CCCSC)=O)C1 S(=O)(=O)(c1csc(C(=O)N(C)Cc2ccccc2)c1)NC(COC)CC(=O)O c1(C(=O)Nc2c(OC)ccc(C)c2)cnc2c(C3=CCN(C)CC3)cnn2c1 N1(C(c2c(OC)nccn2)=O)CC(O)CC1(C)C(N1CC(C)OCC1C)=O C1(CCNC(c2cnn(CC)c2Br)=O)CCCN(C(=O)CN(C)CCO)CC1 N1(C(C(CC=C)CNC(c2[nH]cc(C)c2C)=O)=O)CCC(C)(O)C(O)C1 Cc1nn2cccnc2c1C(=O)NCCC1CN(C(C2(C(N)=O)CC2)=O)CC1C N1(C(C(C)(C)C2CC2)=O)C(CNC(C2(F)CCOC2)=O)CC2CC12 Cc1ccc2[nH]c(C(N3CCOCC(NC(=O)C(CO)N(C)C)C3)=O)cc2c1 c1(NC(C(=O)NCC(CN(C)C)(C)C)=O)nnc2n1CCNC2 N1(C(CC)=O)CCCC(C(=O)NCc2cccnc2)C1.c12cccc(c1)NC2C c1(CN2CC(NC(c3ncccc3Cl)=O)C(F)(F)C2)cc(Cl)c(O)c(Cl)c1 C(=O)(CC(C)(C)COC)N(C1CN(C(c2c(SCC)cccc2)=O)CC1O)C N1(CC(C)C)N=C(C(=O)N2CC3CC2CN3C(c2ccccc2Cl)=O)CCC1=O C(C(C(F)(F)F)OC)NC(C1(CNC(c2cncc(CC)c2)=O)CC(=C)C1)=O c1(NC(C(=O)NCC2CCC3(COC3)OC2)=O)cccc2cc(F)ccc12 c1(C(=O)NC2CCC(NC(CN(C)C)=O)C2)ccc2ncc(=O)n(C)c2c1 N1(C(Cc2c(C)cccn2)=O)CCC(NC(c2ccoc2)=O)C(F)(F)CC1 c1(-n2cc(C3(O)CN(C(=O)CC4CCCS4(=O)=O)C3)nn2)cc(Cl)nc(Cl)c1 N1(C(C(c2ccc(F)cn2)C)=O)CC(NC(C2CCC(F)CC2)=O)C(C)(C)C1 C1(NC(C=C(CNC(C(C)OCC=C)=O)C)=O)CCOC(C)(C)C1 Cc1cccc(NC(=O)C=CC(=O)N(C(C)CCNC(C2(OC(C)C)CC2)=O)C)c1 c1(C(=O)NCC=CCC(=O)Nc2cn(CC)nc2C)cccc(O)c1C Cn1ccc2nc(NC3CC(C(N4CCCC4c4ccc(Cl)s4)=O)C3)ncc12 c1(C(=O)NCC(O)C(F)(F)F)cc2c(s1)CCN(C(c1c(I)ccnc1F)=O)C2 c1(COC)ncc(C(N2CC3CC3(NC(=O)CC3CCCOC3)C2)=O)c(O)n1 C(=O)(CCCCCNC(=O)CC(C)n1ccnc1)NCc1ncc(C)o1 c1(C(=O)NCCC2(CNC(=O)C#CC3CC3)CC2)ccc([N+](=O)[O-])cc1Br Cc1cn2c(n1)CN(C(=O)C(O)CCNC(c1cc(C)c(F)cn1)=O)CC2 c1(SC)ccccc1C1CC1NC(c1cnn(CC2CCC2)c1)=O.C12(CC1)C(=O)N2 N1(C(C23C(C)(C)C(CC2)CC3)=O)CCC2CCN(C(C3CC(F)C3)=O)CC12 C(C(CC(F)(F)F)NC(=O)C(c1ccc(Cl)s1)=O)NC(C=Cc1ccc(C)o1)=O CCCCCCC(=O)NCCN(C(=O)Cc1scnc1-c1cccs1)CCOC NS(=O)(=O)c1ccc(C(=O)NCC2C3CN(C(=O)Cc4cnsc4)CC23)c(Cl)c1 N1(CCC(=O)NCC(CC)NC(C2(CCF)CCC2)=O)CCCC1=O c1(C(C)(C)C)cc(C(N2CCC(NC(C3CCOCC3)=O)C2)=O)cs1 C(=O)(CC(COC)NC(=O)Cc1ccc(F)cc1)N(CCC)CCO C1(C(=O)NCC(C(C)C)NC(=O)C=CSc2ccccc2)CN(C(N)=O)CCO1 C12(COC)CCC(C(=O)NCC(C)(C)CN(C(=O)C(C)(C)C)C)(CO1)C2 C1(C(N2CC(CC(C(=O)N(C3CCCC3)C)F)C2)=O)CC(C)(C)CO1 c1(CCC(=O)NCC2CN(C(CC(=C=C)C)=O)C(C)(C)C2)cc2ccccc2o1 N1(C(CC(C)(C)N(C)C(C2CC3CCC(C2)O3)=O)=O)CCC2(COC(=O)N2)C1 C1(CC)CCCN(CC(=O)NC2CC(NC(C3CCC4CC34)=O)C2)C1 C1(C(N(C2CCN(C(=O)C(O)Cc3ccccc3)CC2)C)=O)CC(C)(C)CN1C N1(C(C2(C)CCNC2=O)=O)CC2C3CCC(C2C1)N(C(=O)CCCC1CCC1)C3 c1(CNC(=O)CCCn2cccc2)ncccc1C(=O)NCC(O)(C1CC1)C1CC1 C1(C(N(C2CCN(C(c3cccc(OC)c3F)=O)C2)C)=O)CCCCC12CCC2 c1(CSCC)ncc(C(C)NC(C(C)(C)C)c2nnnn2CCCOC)s1 N1(CC(=O)NCC2CC(CNC(c3cn[nH]c3)=O)CO2)CCCC1CO CC1=C(C)CC(C)(C(=O)NC2CCC2NC(c2cccc(C)c2)=O)CC1 c1(NC(C(NOC)=O)=O)cc(C)ccc1C N1(C(Cc2c(C)nsc2)=O)CCN(C(C2CCOC2C)=O)CC1CC(C)(C)C c1(-c2ccc(C)o2)csc(=Nc2ccnc(Cl)c2)n1CC(C)C(C)C N1(C(Cc2cn(CC)nc2C)=O)CC(NC(=O)CN(C)C(C)=O)C(C2CC2)C1 C=CC(F)(F)C(=O)NCC1CC1CC(=O)NCCC#CCO CC(C)C(C)C(=O)N(C(C)CCC(=O)N(C1CC1)C(C)C1CC1)C C1(CCNC(=O)CC(C2CC2)C2CC2)CCCCN1C(=O)COc1cccnc1 N1(C(c2n(C)ccn2)=O)CCCC(O)(CNC(c2cccc(F)c2Cl)=O)C1 C1(CN(CCNC(c2c(C(N)=O)cc(F)cc2)=O)C(N)=O)COc2ccccc2O1 c1(OC)ccc(S(=O)(=O)NCC2CC3CC3N2)cc1C(C)C c1(C(=O)NCC2C(NC(C(C=C)O)=O)CC2)ccc(Br)c2c1OCCC2 CS(=O)(=O)c1cccc(S(=O)(=O)N2CCN(C(c3cnc(Br)s3)=O)CC23CC3)c1 c1(N(CCCC=C)C)nc(=NCC2(C)CCS2)[nH]c2c(C)nn(C)c12 C1(NC(c2cccc(NC)n2)=O)CN(C(c2sccc2CO)=O)C(C)(C)C1 CC(F)CC(=O)N1CC(CNC(C2(C)CCCO2)=O)C1 c1(C(N2CCC(O)(C(C)NC(C(C)=CC)=O)C2)=O)cc(C)cc([N+](=O)[O-])c1 CCC(C)(C(=O)NCC(C)CN(C)C(c1ccncc1-n1cccn1)=O)OC C(=O)(CC1=NN(C)C(=O)C1)N(C1CCC(NC(c2cccc3c2COC3)=O)C1)C CC(N=c1cc(C(F)(F)F)nc(-c2ccccc2)[nH]1)c1c(F)cccc1F CCC1=C(C(=O)NC2(C)CC(NC(=O)CC(COC)COC)C2)CCCO1 CC1C(NC(=O)C(F)C(F)(F)F)CC2CCC1N2C(=O)CC1C=CS(=O)(=O)C1 c1(C(=O)NC(C)C(C)NC(c2cc(Cl)ccc2Cl)=O)ccc2sncc2c1 C1(C(C(=O)NCC)N(C(C)C)CC2CC2)CCOC1(C)C C12(CO)CCN(C1)C2=O.C1(CO)CC1(C)C.CC1CC1N(C(CO)=O)C N1(C(c2c(C)cns2)=O)CC2=C(C1)CN(C(c1cc(O)ncc1F)=O)C2 c1(CCCCC)ccc(NC(C2CCC(NC(=O)C(C)SCCOC)CC2)=O)cc1 C1(C(=O)NCC(CC)O)CC2CCN(C(c3cccc(F)c3N)=O)CC12 N1(C(CN(CCC)C(c2cn(CCC)nn2)=O)=O)CC2COCC(C2)C1 CCC(CC(=O)NC1(CNC(=O)CCC2CCCCN2C)CC1)C(C)(C)C N1(C(COCC)=O)CC2CCC(C1CO)N2C(=O)C(c1ccccc1)NC(N)=O c1(NC(C2(CC)CCCN2C(=O)CCn2cccn2)=O)cc(CO)cc(F)c1 C1(C(=O)OC(C)(C)C)CN(c2nc(-c3ccc(Cl)cc3)no2)CC1C(C)(C)C C1(CC(c2ccc(Br)cc2)=O)CC2CC1CN2Cc1cc(Cl)ccn1 C1(C(C(=O)NC2(C)CC2)N(C)Cc2ccc(Cl)o2)CC2C(C1)C2(F)F CC1CCN(C(=O)C2=CCCSC2)CC1N(C)C(c1ccc(=O)n(C)c1)=O n1(CC(N)=O)cc(C(=O)NC2CC2CNC(C2C=CCC2)=O)nn1 C(CNC(C1CC1(F)F)=O)(CC(F)(F)F)NC(c1c(CC)cno1)=O C1(CC(N2CC(CCNC(=O)Cn3nnc(C)n3)C(C)C2)=O)(OC)CCOCC1 C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CC=CC(NC(CCc2onc(C)n2)=O)C1 Oc1cccc2cc(CN(c3nccc(Br)n3)C3CCCNC3)ccc12 C1(NC(CNC=O)=O)CCCC(CNC(C23COCC2C3)=O)C1 c1(C(=O)NC(CC=C)CNC(c2sccc2C)=O)c(C)nnn1C N1(C(=O)Cc2ccsc2Cl)CCC2CN(C(C3CCN(C4CC4)C3=O)=O)C2C1 C(=O)(C1=CCN(C)C1)N1C(C(=O)NCC2(CC)CCOC2)CCCC1 Cc1noc(CCCNC(=O)C=CC(C)NC(c2cc(Cl)c[nH]2)=O)n1 c1(C(N2CCN(C(=O)Cc3cnoc3)CC2CF)=O)sc2sccc2c1Cl CC1(CNC(C2CCN2CC2C3COCC23)=O)CCOCC1 C1(NC(c2cccc(C)c2Cl)=O)CCN(C(=O)C=Cc2cccs2)CC1(C)C CN1CCN(C(=O)C=Cc2cncn2C)C(C(=O)NCC(c2ccccn2)O)C1 c1(C(=O)NCC(CNC(Cc2ccc(OC)cn2)=O)O)cccc2c1nnn2C N1(C(C(=Cc2cn[nH]c2)C)=O)CCCC(CNC(=O)C(C)N2CCC2)C1 CCC(C(=O)NCC(C)CNC(c1ccnc(OCCCOC)c1)=O)C(F)(F)F N1(C(c2cc(C)nnc2O)=O)CCC2CN(C(=O)CCC3CCCOC3)CC12 c1(CC(C(=O)OC)CNCc2ccc(NS(=O)(=O)CC3CC3)o2)ccc(C)cc1F c1(C(=O)NCC2CCC(NC(c3c(C)nsc3)=O)C2)nccc(Cl)c1F c1(C(=O)NC2CC3CN(C(COCCN(C)C)=O)C2C3)cc2cccn2c(O)n1 N1(c2ccc(S(=O)(=O)NCC(C)F)cc2Br)Cc2ccccc2OC2(CCC2)C1 CCCC(F)C(=O)NC1(C(N2CCC2(C)CCC)=O)CCCC1 C1(CNC(COC2(C)CCCC2)=O)CN(C(=O)C2=NNC(=O)CC2)CCC1(C)C Cn1c(CN2CCS(=O)(=O)C(CC(=O)OC)C2)nc2cccc(Br)c12 C12CC(C1)CC(=O)N2.C1(CCOC)(C(=O)N(CCOC)C)CC1 N1(C(C(C)CF)=O)CCC2(CCC2)C(NC(C2C=CC=CC=C2)=O)C1 c1(OC)cccc(CCC(=O)NC2CC2NC(=O)C=Cc2cn(C)nn2)c1F C1(C(CO)NC(=O)CC(Cl)Cl)CCN(C(C2CC2F)=O)CC1 C1(C(=O)NC(C2(O)CCCCC2)C(=O)NCCOCC(=O)NC)CCN(C)C1=O c1(C(N(CCC(C)NC(C2CCC(O)C2)=O)C)=O)ccc2ccnn2c1 C(=O)(CCCCCCn1cc(COC)nn1)NC(C)CCC(NOC(CC)C)=O C(CC(=O)NC1(CO)CCC(C)C1)(C(F)F)NC(c1ccc(CC)nc1)=O c1(NCC2C(NC(c3c(OC(C)C)cccc3)=O)CCC2)ncnc2c1CCO2 CC1CCC(C)N1CC(N1CC(O)(CCNC(=O)CCc2cncs2)C1)=O N1(C(c2cc(C)sc2C)=O)CCC2CN(C(c3c(C)cccc3O)=O)CC2CC1 CC1(NC(C2CCCC2O)=O)CC(NC(=O)Cc2nc[nH]n2)C1 C1(C(=O)NCC(CC(C)C)NC(C(c2ccc(C)s2)C)=O)CC2(COC(=O)N2)C1 C(C)(C(C(=O)NC1(C)CSC1)NC(=O)COCCN(C)C)OC c1(CC)cc(C(N2CCC(CNC(=O)CCNC(N)=O)C(O)C2)=O)ccc1O Cn1nccc1COC1CN(C(C2N(C)CC2)=O)C1.C(=O)(C(O)Cc1cnc[nH]1)N C1(C)(NC(C(c2scc(C)n2)C)=O)CCN(C(C2CCC(C(N)=O)CC2)=O)C1 c1(C(=O)NCC(c2ccc(C(=O)O)cc2)(F)F)cc(-c2nn[nH]n2)cnc1O C(=O)(C1CCc2cccc(Cl)c21)N1C(C(=O)Nc2c(C)ccc(C)n2)CSCC1 c1(-c2nn(CCS(C)(=O)=O)c(C3CCOCC3)n2)ccc(F)c(Cl)c1 C1(C2(O)CCOC2)(C(N2C(C(C)C)CN(C(=O)Cc3cnns3)CC2)=O)CC1 C1(C)(NC(CC2N(C(CC=CCC)=O)CC2)=O)CCCC1O N1(c2nc(Cl)nc(C)c2F)CCOCC12COCCN(C(=O)C1=COCCO1)C2 c1(C(=O)OCC)ccccc1C.C1(C(=O)NCC(=O)OCC)CC1COC C1(C2CN(C(C3(C)CCN(C)C3)=O)C2)(NC(C2C(C#C)C2)=O)CC1 C1(O)(CNC(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC1 C1(CN(C(CCNC(COC)=O)=O)C)CCCCN1C(c1cc(F)c[nH]1)=O C1(CC(=O)NC(CC)CN(C(=O)CN2CCC(C)(O)C2)CC)OCCCC1(C)C N1(C(c2cc(C)cc(C)n2)=O)CC(NC(=O)C(C)(C)CO)CC12CCCOC2 Cc1ncc2ccc(C(=O)NC)cn12.C1(C(N2CCC2CC=O)=O)OCC1(C)C C1(C(=O)NC(C2CCOCC2)CC)CCN(C(=O)CNC(C)=O)C1CC CS(=O)(=O)C(C(=O)NCC12CC(CN1C(=O)C(=O)NCCC(N)=O)C2)C1CC1 c1(NC)nc(C)ccc1C(N1CCCC1CNC(=O)C=Cc1cn[nH]c1)=O C(=O)(CN=c1cc[nH]cc1)NCc1cc(C(=O)NC2CCN3CCCC23)n[nH]1 C1(C(=O)NC(C(=O)NCC)C)CCN(C(C2CC23CCC3)=O)C1(C)C N1(C(CCCOC)=O)CCC2(CCCC2NC(C2CC(C(C)(C)C)=NO2)=O)CC1 c1(C(C(=O)NCC2CCOC2)N(C)Cc2c(C)ccs2)cc(F)cc(I)c1 C(=O)(C(C)(C)CC(=O)N(CCNC(c1c(Cl)c(C)nn1C)=O)CC)OCC c1(CNC(CCNC(C2CCC(CCOC)C2)=O)=O)cc2c([nH]1)CCCC2=O c1(C(=O)NC2CCCN(C(CCCNC(C)=O)=O)CC2)cncc2cnccc12 N1(C(c2c(C)csn2)=O)CCCC(C(=O)NCCc2ccco2)CC1 C1(NC(C(CC(C)C)O)=O)CC12CCN(C(=O)CC1(C)CCCCC1)CC2 C1(NC(C(CC=C)C)=O)CCCCC12CCCN(C(=O)CC1CCCC1(F)F)C2 N1(C(CCCC=C)=O)CCCCC(CNC(c2ccc(C#N)n2C)=O)C1 c1(C(=O)NCC2(O)CCN(C(c3ccc(=NC)[nH]c3)=O)C2)ccc([N+](=O)[O-])cc1 CC(C)C#CC(=O)NC(C1(O)CCN(C(=O)Cc2ccc(Cl)cc2)C1)C C1(CCNC(CC(C)F)=O)CSCCN1C(c1cnc(C(N)=O)s1)=O c1(OC)ncc(C(=O)NCC2(F)CCCN(C(=O)CCC(C)(C)OC)C2)cc1Cl C1(CC(=O)NCC2(C)CCCN2C(c2cc(O)cs2)=O)CC(O)C12CCC2 N1(C(C(COC)C)=O)CCCC(C)(C(=O)N(CCCO)C2CCC2)C1 c1(C(=O)NC2CCCN(C(c3nccc(CC)c3)=O)C2)c(C)cc(C)cc1N c1(N2CCC(COC)(CO)C2)ncnc2ccccc12 C1(C(C)NC(c2cn(C)cn2)=O)CCCN(C(C2(CF)CCC2)=O)CC1 N1(C(CCCOCC)=O)CCC(O)C1C(N1CCC(N2CC(O)C2)C1)=O N1(C(CC(C)(C)NC(C(CC#C)C2CC2)=O)=O)CCC12CCN(C)C2 C(=O)(C(O)CCNC(c1nccnc1C)=O)N(CC=C)C C(=O)(CN1C(=O)C(F)(F)Oc2ccccc21)NC1CN(C(CSC)=O)C2C1C2 C(=O)(C1CCc2cccc(O)c21)N(C(C)CNC(C1C=CCC1)=O)C C1(CC)C(NC(=O)CCCCOC)CCN1C(=O)CCC(=O)c1ccc[nH]1 CC1CCN(CC(=O)N(C)CCN2CCN(C(=O)C(C)(C)C3CCC3)CC2)CC1 c1(C(N(CC(CC)NC(c2c(Cl)cnn2C(C)C)=O)C)=O)cccc(C(C)C)c1 N1(C(c2cnc(COC)s2)=O)CCC(NC(C2CN(C3COC3)C2)=O)CC1C n1(CC)cc(Cl)cc1C(=O)NCC1(C)CCCN1C(=O)C(C)Cn1ccc(C)n1 c1(OC)cccc(C(F)(F)F)c1.C12COCC1n1cc(nn1)CCOC(=O)N2C C1(C(=O)NCC(CN(C(=O)COOC(F)F)C)(C)C)C2CC2C2CC12 c1(C(=O)OCC)ccc(NC(=O)COCC2(CC(C(C(CO)C)=O)=O)CC2)cc1 CCN=C(NCC)NCC(C)(C)C(=O)OC(C)(C)C.c12cccc(c1)NC2 O=C(CCC1=CCCCC1)NC1CCN(C(c2ccnc(OC(F)F)c2)=O)C1 c1(NC(C2N(C(COCCOC)=O)CCC(F)C2)=O)c(C)cc(O)nc1C N1(C(C(n2cc(Br)cn2)C)=O)CCC2(CCC(NC(=O)CC3CC3)C2)CC1 Cc1ccc(C(=O)NCCC(O)CNC(=O)CC2(O)CCCCCC2)cc1N N1(Cc2n(CCC)ncn2)CCCC(CO)(NC(c2ccc(Cl)nc2OC)=O)C1 CCC(CC)CCC(=O)NCC1CC2(CC2)CN1C(=O)CC1CC2(CCC2)CO1 C1(NC(c2cnc(Cl)s2)=O)CC2CN(C(=O)COC3CC3)CCN2C1=O N1(C(c2ccc(OC)nc2Cl)=O)CCN(C(C2OCCCO2)=O)C(C)C1C N1(C(c2cscc2F)=O)CCC2CN(C(=O)CSc3ccc([N+](=O)[O-])cc3)C2C1 c1(C(=O)NC23CC(C2)N(C(=O)C=Cc2cnc[nH]2)C3)ccn2nncc2c1 c1(-c2c(OC)cncc2)ccc2c(C(N3CCN4CCCCC4C3)=O)c[nH]c2c1 c1(COCCN(C2CCN(C(=O)CC(O)C3CCCC3)C2)C)ccc(F)c(F)c1 CC(CO)(C(=O)NCCN1CCC2CC12)NC(=O)CC1OCCC1(C)C C(=O)(C(C)CC(=O)OC)N1CC(CCC)C(NC(C2(C3CCC3)CCC2)=O)C1 C1(OC)CC(NC(=O)CCNC(C)=O)CN(C(=O)CCOC)C1 C1(C(N2CCC(NC(C(OC)OC)=O)CC2C)=O)CC2(C1)CC1(CC1)C2 c1(C(C)OCC)nc(CC(N2CC(O)(CNC(=O)Cc3n[nH]c(C)n3)C2)=O)cs1 C1(C(=O)NCCC2(NC(c3cnc(CCCC)s3)=O)CC2)CN2CCN1C(C)C2 C(N=c1c(Br)c[nH]cc1[N+](=O)[O-])C1N(C(=O)C(c2cccc(F)c2)O)CCC1 C1(C(=O)NCCC2CCCN(C(c3c[nH]nc3C(F)F)=O)C2)CCCCC(=O)N1 c1(C(=O)NCC#CCNC(c2c(C)ccnc2C)=O)nccc2c1NCCC2 N1(C(COC)=O)CC2CCCC2C1CNC(c1cscc1OCCOCC)=O c1(OCC)ncc(C(=O)NCC2CCCCN2C(=O)CC(C)(C)SC)cc1Cl c1(C(N2CCCN(C(CCN(CCC)C)=O)C(C)C2)=O)ccc2cnc(C)n2c1 C1(CC(=O)NCCC2C(C)N(C(=O)CCn3cccn3)CC2)CCCCC12CC2 c1(CCC)cc(C(=O)NC2CCN(CCNC(=O)Cn3cnnn3)CC2)sc1C C=CC(C)(CCOC)C(=O)NCC1CCCCN1C(=O)Cc1cccnc1 C(=O)(C(C)C(F)(F)C(F)F)NC1CC(NC(C2CCC(OC(C)C)CC2)=O)C1 c1(CC(=O)N(CC(C)NC(C(CCC)O)=O)CC)cc2ccccc2c(O)n1 c1(NC2C(C(F)(F)F)CCN(C(C=CCOC)=O)C2)ccc(C#N)c(C)n1 c1(CC(N2CC(CNC(c3n(C)ncc3)=O)C2)=O)cn2c(nc1=O)SCC2 C(=O)(C1CCc2cccc(O)c21)N1CC(NC(C(c2cnccn2)C)=O)C(C)C1 C(=O)(C(CC(F)F)NC(=O)C1=NOCC1)N1CC(CC)C1 c1(CC)cc(C(=O)NC(C)CCCCNC(=O)C=Cc2ccccn2)ccc1C C1(F)(C(N2CC3C(NCc4ccc(C)cc4C)C3C2)=O)CCCCC1(F)F c1(CNC(=O)COC2(C(=O)NC3CCC(CN(C)C)C3)CCC2)nnc(S)n1C N1(C(CSC)=O)CC(NC(=O)CC(C)c2ccccc2)C(F)C1 c1(OC)c(C(=O)NC2CC(NC(=O)COc3cc(F)ccc3F)C2)cccc1F C1(NC(CNC(CNC(C)=O)=O)=O)CCN(C(c2cccc(C3CC3)c2)=O)CC1 C(=O)(CCS(C)(=O)=O)NCC1CCN(C(C(C=C)O)=O)C1 C1(C(=O)NCCCC2CCCN2C(C2CCCO2)=O)CC(=O)N(C2CCCC2)C1 C(C(C)(C)CS(=O)(=O)CC)NC(c1ncc(Cl)cc1F)c1n(CC)nnn1 N1(C(C2CC(=C)C2)=O)CC(NC(=O)CCn2ccnc2)Cc2ccccc21 C(=O)(CC(C)(C)C(C)(F)F)NC(C1(O)CN(C(=O)Cn2cc(Br)cn2)C1)C Fc1cc(CN2CCOC(C3CC4CC3C4)C2)c2c(c1)CCC2 CC(C)C1=NOC(C(N2CC(O)CC2CC(=O)NCCS(C)(=N)=O)=O)C1 c1(NC(CCCC=C)C)ncc(S(=O)(=O)N2CCCC2COC)cc1Cl CCC(C)CCCCC(=O)NCCC1CC(C(N2CC3(CCC(=O)O3)C2)=O)C1 c1(C(NOC(C(=O)NCC(C(=O)OC)OC)CC(C)C)=O)cccc(C#N)c1C C1(F)(C(=O)NC2CC2NC(C2CCOC2)=O)CCCCC1 C(=O)(C1=CNC2=NCCC2=C1)NCC(CCOC)NC(=O)C(C)CCC(C)(C)C N1(C(C2(C)CC(=C)C2)=O)CCCCC1CCNC(c1ncccc1OCC)=O Cc1cc(C(N2CCC(C)C(CNC(=O)CC3CC3)C2)=O)ccc1C(N)=O c1(C(N(C2CC(NC(c3cc(CO)on3)=O)C2)C)=O)ccc(O)c(CO)c1 N1(C(=O)CC2CN3CCC2CC3)CCC2(CC1)CN(C(C13CSCC1C3)=O)C2 C1(NC(CN2CC=C(C)CC2)=O)CCCN(C(c2cocc2C)=O)C1C CCC(O)C(C)(C)C(=O)N1CCCC(N(C(=O)Cc2cncc(C)c2)C)CC1 C(CCCC(CO)NC(=O)Cc1csc(C)c1)NC(C(C(C)C)OC)=O C#CC1CCCCN1C(C1(C(C)C)CCCN1C(=O)CSCC(=O)NC)=O O=C(C1=COCCC1)NC1(CCCNC(=O)C2=CCCCC2)CC1 N1(C(C2CCCN(C(CC=CCC)=O)C2)=O)CCOC(C2CC2)CC1 c1(C(N(CCCN(C(C(C)N(CC(F)(F)F)C)=O)C)C)=O)coc(C(F)F)c1 c1(NC(C2CC23CN(C(c2cncc(F)c2)=O)C3)=O)nccc2cccnc12 N1(C(c2cc(C(C)C)n[nH]2)=O)CCN(C(C2CS(=O)(=O)C2)=O)C2CS(=O)(=O)CC12 C1(C(=O)NC(CCC)C)CCCC12CCN(C(=O)Cc1cccn1C)C2 c1(C(=O)NCC2(C)N(C(c3c(C)sc(O)n3)=O)CCC2)cc2c[nH]nc2s1 N1(C(c2oc(CC)c(C)c2)=O)CC2(CNC(=O)C(C)=C(C)C)CC1CO2 c1(C(N2C(CN(C(C3C(OC)CC3)=O)C)CCC2)=O)cc(O)nc2c1CCCC2 c1(N2CCC(NC(c3cnc(OC)nc3)=O)C(O)C2)ncnc2c1COC2 Cc1cc(C(N2CC(NC(=O)C3=CCSC3)CC23CCCC3)=O)cc2nc[nH]c12 C=C(C)C1CN(C(=O)CCN(C)C(C2CC2OC)=O)CCO1 N1(C(c2cc(Cl)cs2)=O)CCCC(N(CCO)C(c2cc(CCO)on2)=O)C1 C12(NC(CCCOc3ccc(C)cc3)=O)CCCC1CN(C(c1ccon1)=O)C2 c1(C(=O)NCC2OCCN(C(CN3C(C)CC3)=O)C2)ncc(F)cc1F c1(C(CNC(C(C)C23CC(C2)C3)=O)(F)F)nnc2ccccn12 C=CC1(CC(=O)N(CC(C)N(C)C(c2c(C)coc2C)=O)C)CCCCC1 CCCCCC(F)C(=O)N1CC(=O)CC1C(=O)NCC(C)N(CC)CC c1(N(C(C(CC2CCCC2)NC(C(C2CC2)OC)=O)=O)C)cc(C)cc(C)c1 C(CNC(=O)CCCC1CCCCC1)(C(C)C(C)C)NC(C(C)(C)OC)=O C1(C(=O)NCC2N(C(c3n[nH]c(C)c3Cl)=O)C3C(C2)C3)CCC(C)(C)CC1 c1(C(N2CC(OC)C(C)(C)C2)C(=O)NCC(=C)C)ccc2ncc(Br)cc2c1 C1(CNC(c2nc(CC)sc2)=O)CC(NC(c2ccncc2)=O)C1(C)C C1(C(=O)NCCCN(C(=O)COc2ccccc2Cl)C)Cc2ccccc2S1 c1(N2C(C(=O)OC)CC2C)cc(Br)c(C(c2ccc(CC(C)C)cn2)=O)cc1C CC(O)C(C)C(=O)N(C)CCOCCCN(C(=O)C(C)(C)c1ccns1)C C1(NC(c2n(CC(C)C)ncc2)=O)CC(C)N(C(=O)COc2ccccc2Cl)C1 C1(C(N2C(C)C(NC(c3cc(Cl)cs3)=O)CC2)=O)CCc2ccccc2N1 C=CCCCCCC(=O)NC(CCCNC(C1C=CS(=O)(=O)C1)=O)c1cccs1 C1(C(=O)NCCC(CC)O)(CC)CCCN(C(=O)CCOC(C)=O)C1 N1(C(C(C)N(C)C)=O)CC2CCC(C1)C(NC(=O)Cc1cc(Br)cs1)C2 N1(C(C(C)C(C)O)=O)CC2(CCN(C(C3SCCS3)=O)CC2)CC1C C1(NC(CN(C(C)=O)C)=O)CC2CN(C(=O)CC3C=CCCC3)CC12 N(C1CC2(CN(C(c3cccnc3N)=O)C2)n2ccnc21)C(CCC(C)(C)F)=O CC1=C(C(=O)NC2CC2NC(=O)C=Cc2cscn2)Cn2nnnc2N1C N1(C(c2ncc(C)nc2)=O)CC2CC1CN2C(C1(Cc2cccnc2)CC1)=O C1(CC=CCCOC)CCCCN1C(=O)NCc1ncc[nH]c1=O C1(C(N2CC(CCC)C(C(=O)N(CC(C)C#N)CC)C2)=O)CC(C)CC(C)C1 c1(C2(C(N(CCCNC(=O)CCOCCN(C)C)C)=O)CC2)ccc(F)cn1 c1(OCCC)ccc(C)cc1-c1cnc(NC(=O)Cc2ccn(C)n2)s1 c1(C(=O)OCC2CCC(F)(F)C2)ccc2c(n1)OCCO2 c1(C(N(C2CCC(C)(C)CC2)CCC)=O)nc2ccc(NC(C)=O)cc2s1 C1(CCCNC(CC=C)=O)CCCN1C(C1CCNC1=O)=O CCC(C)(C(=O)NCC(C)(C)NC(=O)C(C)(c1ccccc1)OC(C)C)C(F)F C1(C(=O)NC2C(NC(C3C(OCC)CC3)=O)COC2)CN2CCN1C(C)C2 S(=O)(=O)(c1ccc(C#N)c(NCCOc2cccc(C(F)(F)F)n2)c1)NCC=CC C(=O)(C(C)CC(F)(F)F)NCC1(O)CCN(C(COC2(C#C)COC2)=O)C1 CCCC(CC)C(=O)N1CCN(C(=O)CCN2CCSC(C)(C)C2)CC1C(C)C C1(CCC)CN(C(c2ccc(CC)c(Cl)c2)=O)CCN1C(=O)CCn1cccn1 Cc1ccc(S(=O)(=O)N2CC=CC2C(=O)Nc2cncnc2I)cc1C C1(C(N2CC(OCC#C)C2)=O)CC(C)CN(C(=O)C(C(C)C)NC(C)=O)C1 Cc1nc(N(C2CC(=O)N(C)C2c2cccnc2)C)c(C)c(Cl)n1 C(CN=c1nn[nH]n1C)C1CCN(C(c2c(C)snc2)=O)C1 C1(CCNC(Cc2cc(C)no2)=O)COCCN1C(=O)C(O)CN1CCCC1 C1(NC(CCCC)=O)CCN(C(=O)Cc2ccnc(F)c2)C1(C)C N1(C(CC2(CNC(c3cc(COC)[nH]n3)=O)CC2)=O)CCC2CCNC(=O)C12 CC1CCN(C(C2CSC2)=O)C(C(=O)NCC(F)(F)Cl)C1 c1(CCC(=O)NC2CCCC2NC(C2CCCC2O)=O)cnc2n1CCCC2 C(=O)(C(C)CCC(C)(C)C)N1CCC(CCOC)(NC(=O)C(CO)C(C)(C)C)C1 N1(C(=O)NCC2(C#N)CCCC2)CCN2C3CCC(C3)C2C1 N1(C(C(CCOC)NC(Cc2c(CC)con2)=O)=O)CCC(F)(CF)CC1 C(=O)(CCCCCCCCC1CC1)N1CCC(O)(CNC(C(F)=CCC)=O)C1 CC1(C)CCC(C(=O)NC2CCC(C#N)CC2)CN1C(C1(C)COCCO1)=O N1(C(C23OC(C)C(C2)C3)=O)CCC2(CC1)CCN(C(C1CC1(F)F)=O)CC2 C1(C(=O)NCC2(F)CC(CNC(CCCC3C(C)C3)=O)C2)CC2(C1)CC2F C1(NC2CCCC2)CC(F)CN1C(=O)CN1CCSCC1.O=C1COCCN1 C1(C(=O)NC2(CC3CC3)CCC2)(NC(C(COC)C)=O)CCN(C)C1 c1(CCNC(C2N(C(C(C(C)C)OC)=O)CCOC2)=O)cn(C)c2cccc(C)c12 c1(CC(=O)NCC(CC)NC(c2sccc2-n2ccnn2)=O)cncn1C C#Cc1cn(C)nc1C(=O)NCCCCN(C)C(C1CCC(OC)C1)=O C1(C)(CNC(c2cn(CCCOC)nc2)=O)CCN(C(=O)COC2COC2)CC1 C1(NC(C=CC(C)NC(=O)Cc2ccco2)=O)CCCCCC1 c1(C(C(=O)N(c2ccccc2)C)O)ccc(NC(c2ccsc2Cl)=O)cc1 C1(CCNC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)C(F)CC2CC2)CC1 C1(OCC)COCCC1CC(=O)N(C)CC1CCCCN1C(=O)C(F)CC N#CCS(=O)(=O)c1ccc(C(N2CCN(C(c3nc(Cl)cs3)=O)CC2)=O)cc1 Cc1ncccc1-c1cn(C2CN(C(c3ccccc3C(C)(F)F)=O)C2)nn1 CC(O)C(C)(C)C(=O)N1CC(CO)(CNC(c2cc(C(F)(F)F)cc(O)n2)=O)C1 C1(NC(c2c(C)cns2)=O)CCN(C(=O)CC(O)C2CC2)CC1F C1(N(C(=O)C2=CCOC2)C)CCCCN(C(C2CC2c2ccccc2)=O)C1 c1(C(=O)NC(C)CNC(=O)CCCCC(F)F)cc(P(C)(C)=O)ccn1 CC(C)C(F)(CNC(=O)CCC(C)N(C)C)C(=O)NCCn1cnccc1=O C1(C(N2CC(C)C(NC(c3cscc3C(F)(F)F)=O)C2)=O)CCc2nncn2C1 O=C1Nc2ccc(C(=O)OCCOC34CC(CC(C(=O)O)O3)C4)cc2C12CC2 N1(C(c2[nH]cc(C(N)=O)c2)=O)CC2CC(NC(=O)C(F)CC3CCC3)C(C2)C1 C(=O)(CC(C)CC(C)(C)C)N1C(NCc2ccc(CCCC)cc2)COCC1 C1(C)(C(N(CC(C)N(C(c2c(CC)c[nH]c2)=O)C)C)=O)CCCCNC1=O c1(C(=O)NCCC(=C)CNC(C2CCCCN2C)=O)cncc(N)n1 c1(C(N2CC(=O)N(O)C2=O)c2ccccc2)nn(-c2ccccc2Cl)c2c1CCC2 C(=O)(CC(O)CC(C)(C)C)N1CC(CCC)C(C(=O)NCc2ccc(C)nc2)C1 C1(NC(C(C)CO)=O)CC2C1CCN2C(c1cn(CC2CCCOC2)nn1)=O C(=O)(C(O)C(C)(C)C)NCC12CC(F)(C1)C2.C12(SC)CN(C1)C2=O C1(C(N2C(C(CNC(C=CCCC)=O)(C)C)CCC2)=O)CCC2(CCOCC2)O1 C(C1C(C)C1(Cl)Cl)=CC(=O)N(C(C)C)CCNC(c1ccc(C2CC2)nc1)=O C1(C(=O)NCCCCC)C(=O)OCC1(C)C.C12(CC1)CC(=O)NC2 C=C(Cl)C(C)(C)C(=O)N1C2CCC1C(CNC(c1cccc(C(F)(F)F)c1)=O)C2 CCCC(CC)C(=O)N1CCC(CC(C)NC(c2c(C)cnnc2O)=O)CC1 c1(CC(=O)NC2CCN(C(=O)Cc3csc(C4CC4)n3)C2)cccc(Cl)c1F C1(CNC(c2ccn(CCNC(C3C(C)CC=CC3)=O)c2)=O)CC(=O)N(C)C1=O C1(CC)CCC1(c1nnnn1C1CCOCC1)NCc1ccsc1Cl N#Cc1cc(F)c(NC(C2CCCN2C(c2cc(C3CC3)no2)=O)=O)cc1Cl c1(C(=O)NC2C(CNC(C(C)C)=O)CCC2)cc2scc(Br)c2[nH]1 C(=O)(CC1=NN(C)C(=O)C1)NCC(CC)N(C(=O)CC1COC(C(F)(F)F)C1)CC N1(C(C(CCC)N(C)C)=O)CCCC12CCN(C(c1cc(C3(C)CC3)on1)=O)C2 N1(CC)CC(C(=O)NCCN(C(=O)C=CC2CCOC2)CCOC)CC1=O c1(C(=O)NCCOC(CNC(C(CC)N(C)C)=O)(C)C)ncccc1F Cc1cc(C(N2CCC(c3ccnn3C)C2)C(=O)NCCC2(C)CC2)sc1Cl C=CCC(C(=O)NCCN(C(=O)C(C)n1cncn1)C1CC1)C(C)C N1(Cc2ccc(OC)nn2)CCCC(NC(c2cccc(Br)n2)=O)CC1 C(C(=O)N1CCC(C(C)NC(C2(c3ccccc3F)CCC2)=O)C1)(C(C)C)OC C1(CNC(=O)NCCCCC(OC)OC)C2Cc3c(Br)cccc3C12 N1(C(=O)CCc2nc(O)n[nH]2)CCC2CCC(NC(C3(Cl)CC3)=O)C1C2 C1(NC(C(C)(C)F)=O)CCCCC12CCN(C(c1ccc(O)c(F)c1)=O)C2 CC1(CNC(=O)CC2(C)CCCO2)CCCN(C(=O)CCCC2CCCCC2)C1 C1(CNC(CC2OCC(C)(C)C2)=O)CCN(C(c2cnnn2C2CC2)=O)C1(C)C N1(C(C(C)S(C)(=O)=O)=O)CCC2(CCN(C(C3(O)CCSCC3)=O)C2)C1 C(c1cn(C)cn1)=CC(=O)NC(C(=O)N(CC(CC)NC(C)=O)C)C c1(C(N2CCC(C)(CNC(c3scc(OC)c3)=O)C2)=O)cn(C)c(C)cc1=O N12CCC(CC1)NC2=O.c1(C(N)=O)ccc(CCn2ccnn2)s1 c1(C(=O)NCC2N(C(C#CC(C)C)=O)CCC2C)oc2ccccc2c1CO Nc1nc(Br)ccc1C(=O)NC1CC(F)CN(C(=O)Cn2ncnn2)C1 C1(NC(c2c(Cl)ncc(C)c2)=O)CCN(C(c2c[nH]c(=N)o2)=O)C12CCCC2 c1(C(=O)NC2C(CC)CN(C(c3csc(O)n3)=O)CC2)ncnc2c1CCC2 Cc1cccc(C(O)C(=O)NC2CCCCN(C(c3cc(N)ccn3)=O)C2)c1F c1(NCC2CC(O)(C(C)C)C2)nccc(=NC(C)c2nccc(=N)[nH]2)[nH]1 C1(O)(CNC(CCCOCC=C)=O)CCCN(C(c2cnoc2C2CC2)=O)C1 c1(NC(C)=O)ccc(C(=O)NC(CNC(C2CC(C)(C)C2)=O)CO)cc1O N1(C(C(CCOC)C)=O)CCN(C(c2cc(C)ccc2Br)=O)CC1CO CCCCC(C)C(=O)NCCCC1CCN(C(=O)CCC(=O)N(C)C)CC1 C1(CNC(C2(OC)CCSC2)=O)CN(C(C2(CC(C)C)COC2)=O)CC(C)(C)C1 c1(C(=O)NC2CN(C(c3ccc(OC)c(O)c3)=O)CC2F)cc2ccccc2[nH]1 N1(C(c2nc(NC(c3c(N(C)C)n[nH]c3)=O)sc2)=O)CCNC(=O)C1 CC1CCN(C(=O)COCCF)C1CNC(=O)Cc1csc(C2CCCCC2)n1 C1(NC2CC(c3ccccc3)(NC(C3C(C)CC=CC3)=O)C2)CCCC(=O)N1C N1(C(C2ON=C(C)C2)=O)CC(NC(=O)Cc2ccc3n[nH]cc3c2)CC(C)(C)C1 C1(NC(CN(C(COC)=O)C)=O)CCN(C(c2c(Cl)cnn2CC)=O)CC1CO C(=O)(CS(C)(=O)=O)NCC1(C(=O)NCCC2CCC(C)O2)CC(=C)C1 C12CCN(CC1)C2=O.C1(C(=O)NC(C)C)CCCC(C2CC2)O1 c1(C(=O)NCCC2N(C(CC3(C)CCCO3)=O)CCC2)ccc(F)cc1[N+](=O)[O-] C1(NC(C(C)NC(c2ccc(C3CC3)cc2)=O)=O)CCCC(C)(C)CC1 CCCC(C(=O)NCCc1ccccc1O)NC(C1CCCN1CCC)=O C(C1Cc2ccccc21)NC(c1cocc1C(N)=O)=O.CC1(C)C2C1CNC2=O CC(=O)C(C)CC(C)C(=O)N1CC(C)CCC1CNC(=O)Cc1ccc(O)cn1 C1(O)(C(N2CC(CNC(c3cc(CC)on3)=O)OCC2)=O)CCC(C)CC1 C(=O)(C1=C(C)CCCC1(C)C)N1CC(F)CC(NC(CC2CC(OCC)C2)=O)C1 N1(C(C(CC)NC(N)=O)=O)CCCC(C)(C(N2CCC(O)C(C)C2)=O)C1 C1(C2CCOCC2)(CNC(CCCOC)=O)CCN(C(C2CCN(C)C2C)=O)C1 C1(CNC(CC=CC=C)=O)CC(F)CN1C(=O)COc1ccc(C(F)(F)F)nc1 c1(C(=O)NCC(CC=C)NC(=O)C2=C(C)OCCS2)n[nH]c2c1CCOC2 c1(C(N2CCC(NC(c3ncn(C(C)C)c3)=O)C2)=O)ncc2n1CCCC2 C(=O)(C(O)C(C)(C)CC)N1CC(n2cc(SCC)nn2)C1.N12CCCC1CC2=O c1(C(N2C(c3cn(CCC(C)(C)O)nn3)CCC2)=O)ccc(CS(C)(=O)=O)cc1 CC(C)(C)CC(O)CNC(C1(CCNC(=O)CCc2cccnc2)CC1)=O Cn1[nH]c(-c2ccc(F)cc2)nc1=NC(=O)NC1(c2nnc3n2CCCC3)CC1 c1(CC(N2CCN(CCCF)CC2)C(=O)NC(C)C)cc(CC2CC2)cc(F)c1 N1(c2c(Cl)cnc(OC)n2)CCN(C(c2cccc3cnsc23)=O)CCC1C C1(NC(C(C)Cc2cnc[nH]2)=O)CN(C(=O)Cc2cccc(Cl)c2Cl)CCC1C c1(C(CNC(c2c(CC)occ2)=O)NC(C2CCCO2)=O)cccc(C)c1 N1(C(C2CC2CC)=O)CCOC2(C1)CN(C(=O)Cc1ccccc1C1CC1)C2 Cc1cc(F)c(F)cc1NC(C1CCCN1C(=O)Nc1ccc(Cl)cc1C)=O O=C(C1=CC2CCC=CCCC12)NCCC1CN(c2ncns2)C1 C1(C(C(=O)NC(C#C)C2CCC2)NC(=O)CC2(CSC)CC2)CCCC1 C12(NC(c3c(CC)occ3)=O)CC3CCC(C1C2)N3C(c1nocc1C1CC1)=O c1(OC)cccc(NCC(=O)NCC#CCNC(=O)C(C)n2cccn2)c1 N1(C(CCCCOC)=O)CCCC12CCC(NC(=O)C(C)Cn1ccnc1)CC2 C1(CC(=O)Nc2ccc(C)nc2)CCCC12CN(C(c1cc(C)n(C)c1C)=O)C2 c1(C(N2C(CCNC(C(CSC)C)=O)CCCC2)=O)occ2c1CCCC2 c1(NCC(C)CN(C)C)nccc(-c2ccoc2)n1 C1(OC)C(OC)CN(C(=O)CCS(N)(=O)=O)C1CNC(=O)C(c1cnn(C)c1)O CC1Oc2ccc(C(N3CC4C(CNC(=O)CC(C)N(C)C)C4C3)=O)cc2C1C c1(C(N(C2CN(C(C(C)C#N)=O)CC23CC3)C)=O)n[nH]c2ccccc12 C1(C(=O)NCC2N(C(CCC(=C)C)=O)CCC2C)CCN(S(=O)(=O)NC)CC1 c1(NCC2CC(C)SCC2)ccc(S(=O)(=O)N2CCC(C)(C)CC2)cc1Cl N1(Cc2cnc(C)o2)CCC2(CCCN(C(C3CCCCCC3)=O)C2)C1 c1(C(=O)NCCCN(C(C(CC)n2cccn2)=O)C)nc(C(C)C)oc1C c1(C2N(C(c3csc(Br)c3)C(=O)NCC=C)CCCC2)cccc(C)c1F N1(C(c2c(C)cc[nH]2)=O)CCOCC1CCNC(C1CCC(F)(F)C1)=O C#CC1(NC(=O)CC(C)(C)CNC(=O)C(C)CO)CCCCCC1 C1(NC(c2c(Cl)nc(N(C)C)s2)=O)CC2CCC1N2C(=O)CC1CCC(=O)N1C c12cccc(c1)NC2=O.c1(CC(=O)OCC)nnc(N(CC(C)C)C)s1 c1(N(C)CC2CCCO2)nc(N2CCC(F)(F)C(C#N)C2)c2ncsc2n1 O=C(CCCCC(F)(F)F)NC(CNC(=O)CC1CCC2(CCC2)CO1)CO N1(C(c2cc(C)ns2)=O)CCC(C)N(C(C2CC3C=CC2C3)=O)CC1 CC(C)C(CN=c1nc(N(CC(C)C#N)C)c2c(F)cccc2[nH]1)OCCO C=C=CCCC(=O)N1CCCC1C(C)(C)NC(=O)C(O)Cc1ccc(F)cc1 C1(O)(C(=O)NC2CCCC(NC(=O)CC3(C(F)F)CC3)CC2)CN2CCC1CC2 c1(C(=O)NCCC(C)NC(=O)C(O)CN(C)C)cc(Cl)cs1 Cn1cnc(C(=O)NC(C)C=CC(N2CC(C(C)(C)C)C2)=O)c1 N1(C(Cc2n(C)nnc2)=O)C(C(N2CCCC2(C)CO)=O)C2CC(O)C1C2 CCCCCCC(=O)NCCc1cc(C(=O)NCC2CCC(C)N2C)no1 O=C(C1=CC2C=CC1C2)NCC1CCC2(CC2)N1C(=O)COc1cccnc1 Cc1cccc2ncnc(N3CC4CC3CN4C(C3CC(=O)N(C)C3)=O)c12 N1(C(C2N(C(C)=O)CCC2)=O)CCOC2CN(C(c3ccnnc3C)=O)CC12 c1(CC(=O)NC(C2CCCN2C(c2ccc(O)c(O)c2)=O)C)ccc(F)cc1Cl c1(CNC(C2(CC=C)CC2)=O)ccc(C(=O)N(C)Cc2ccccn2)s1 N1(C(=O)OC(C)(C)C)Cc2ccccc2OC2(C1)CN(C(C1(Cl)CC1)=O)C2 CC(CC(=O)N1CCC1(C)CC(N1CCOCC1CO)=O)C(C)(C)C c1(C(=O)NCC2CCC(NC(c3cn(C(C)(C)C)nn3)=O)C2)ccc(O)nn1 c1(C(N(C)CC2CCCN2C(C2(O)CC(F)(F)C2)=O)=O)cncc2sccc12 Cc1nn(C)c(Cl)c1CC(N1CC(NC(c2cnnc(O)c2)=O)CC1C)=O N1(C(C2(C#N)C(C)(C)C2)=O)CC2CN(C(c3cc(O)c(F)cc3N)=O)CC2C1 O=C(CCS(=O)(=O)c1cccc(Br)c1)N1CCC(O)CC1 c1(C(N2C(C)CC(NC(C3CCS3(=O)=O)=O)CC2)=O)ccc2c(O)nncc2c1 C(C(C)(C)CNC(C1C2COCC12)=O)NC(CCNC(C1C(C)C1)=O)=O N1(C(c2c(C)scn2)=O)CCC(O)(C(C)CNC(c2ccnc(N(C)C)c2)=O)C1 c1(C(c2n(CCCC)nnn2)NC(c2csc(C)n2)C)cc(C2CC2)ccc1F c1(C(=O)NCC2(CNC(CC3OCC(C)(C)C3)=O)CCC2)cccc2cncn12 C1(CC(=O)OC)C(=O)NCCN1C(=O)C(N1CCN(c2cnccn2)CC1)=O CCC(O)C(C)C(=O)NCCN(C(c1nc(F)ccc1Cl)=O)Cc1cccc(Cl)c1 Cc1cc([N+](=O)[O-])ccc1CN(C)Cc1c(F)ccc(F)c1F N1(C(CCN(C(C)=O)C)=O)CCC(N(C)C(c2cc(-c3ccco3)cs2)=O)C1 N1(C(c2ccc(COC)s2)=O)CC2(C1)SCCC2NC(c1csc(C)c1)=O c1(OCC(=O)NC2(C3CCC3)CC(NC(C=C(COC)C)=O)C2)cccc(C)c1 N1(C(c2c(C)ccc(Cl)c2)=O)Cc2ccc(C(=O)Nc3cnn(C)c3)cc2C1 C(=O)(C(C)(COC)OC)N.C(CC(=O)N(CC(=O)N(CC(C)C1CC1)C)C)OC O=C1C(NC(c2nnnn2CC(F)F)c2nccs2)CCN1O N1(C(C(C2CCCCC2)OC)=O)CCN(C(c2cnccc2Cl)=O)C2CCC12 Cc1ccc(C(N2CCN(C(=O)Cc3cc(Cl)sc3Cl)C(C)C2)=O)c(C(C)C)n1 c1(C(=O)NC(C(C)C)CO)nc(NC(c2ccc(OCF)cc2)=O)cn1C CCC#CCCN(C(=O)CC(O)C1CCCC1)CONC(=O)Cc1nc[nH]n1 c1(Oc2c(Cc3cc(NC(N4CCOCC4)=O)no3)cccc2)ccc(F)cc1F N1(C(C(n2cc(C(C)(C)F)nn2)C)=O)CCOCC2(CCC2)C1 CC(CCC(C)(C)C)C(=O)NCC1(CC(=O)N(C2CC2)Cc2ccco2)CC1 S(=O)(=O)(c1ccc(NCC2CCCO2)nc1)NC1C2(CC(OCC)C2)C1 C1(NC(C(n2ncc(C)c2)C)=O)CCC(NC(C2CC2CF)=O)CC1 O=C(C1=CC2CC=CCC12)NCC1=CCN(c2nnc(C3CCC3)o2)CC1 c1(C(C)C(=O)NCC#CCNC(=O)CNC(=O)CN(C)C)ccc(Br)cc1 C(=O)(C1CCCn2ccnc21)NC1(CNC(C2(C)CC(F)(F)C2)=O)CCC1 C1(CCNC(=O)CCN2CCCC2)CSCCN1C(=O)COc1ccc(O)cc1 Cc1nc(N(C)C(=O)NCC2CCN(C(C)C)C2)sc1C N1(C(C2=CC(C)(CC)C2)=O)CCN(C(c2c(O)noc2C)=O)C2(CCC2)C1 Cn1cncc1C=CC(N1CCCC(CC(=O)NC(C)(C)CC2CCOC2)C1)=O C(CCC)(CC(=O)N1CCN(C)C(=O)C1)NC(C(CC=C)OC)=O N(C1COc2ccccc21)C(C1C(C)(C)C1NC(c1cc(Cl)c[nH]1)=O)=O C=C1CCN(C(=O)C(C(C)C)OCC)C(C(N2CCCOCC2C)=O)C1 C1(C(N2CC(C(=O)NCCC=CC)(CC)C2)=O)CCCC(CC)C1 CCC(O)C(C)(C)C(=O)N1CCC(NC(=O)CC2(C)CCC2)C(C)(C)C1 Cc1c(C(=O)NC(CO)C(C)NC(C2CCC3(CCC3)C2)=O)[nH]c2ccccc12 N1(CC(=O)OCC)CCC2NC(=O)OCC2C1 CCC(C)(CNC(c1c(CNC(=O)C(F)(F)C(C)O)cnn1C)=O)C(N)=O N1(C(CCn2ncc(C)c2)=O)CCN(C(c2nc(C)ncc2Cl)=O)C(C)C1C n1(CC)c(CNC(=O)CCC2CCC(NC(c3cnsc3)=O)C2)nnc1O C1(CN(C(COCc2nnc(C)s2)=O)C)CCC(NC(=O)C(C)(C)CO)CC1 N1(c2c(C)c(NC3CC3c3cc(S(C)(=O)=O)cs3)ncn2)CCC(C2=NOCC2)C1 C(C(CO)C(C)CC)NC(C1(NC(C2C(=C)C2)=O)CSC1)=O N1(C(c2cc(OC)no2)=O)CCC(C)C1CNC(C1CCCSC1)=O C(=O)(C1CCc2ccccc21)NCCC(CC)(CC)NC(c1ccncc1F)=O N1(CC(C)CC2CC2)CCOC2CCC12 C1(C)(C(=O)NC2CC(C)(NC(CC=CC)=O)C2)CCCCNC1=O CC1(C)CN(C(c2ncsc2C(F)(F)F)=O)CCC1NC(C1C(C)(C)C1(F)F)=O c1(C(N(C(C)CNC(c2cncc(Cl)c2Cl)=O)C)=O)ccc(O)cc1[N+](=O)[O-] Cc1cc(C#N)ccc1C(=O)NC1CN(C(=O)CCc2ccon2)CC1F c1(C(=O)NCC=CCNC(CN(C)CCO)=O)cc(C(N)=O)cc(F)c1 c1(C(=O)NCCC23CN(C(C(=O)NCC)=O)C(CC2)C3)coc2c1CCCC2 C1(NC(C(C)=C(C)C)=O)CCC(NC(c2ccsn2)=O)CC1 N1(C(C(C)OC)=O)CCC(CCC2CCCN(C(c3cn(CC)cn3)=O)C2)CC1 n1(C(C)C)cc(NC(=O)C(=O)N(C)C(c2ccccc2)C)nn1 c1(NCC2CCCN(CC(F)(F)F)C2)c(Cl)ccnc1Br Cc1ccc2c(=NC3CCC(C)C3)[nH]c(=NCc3cc4ccccc4o3)[nH]c2c1 C1(C)(CNC(C(CC)(C)C)=O)CCCN1C(c1nn(C(C)C)nc1Br)=O N1(C(C(CC)=CCCC)=O)CCN(C(=O)C(N2CCOCC2=O)C)CC1CF C1(C2CC2)(NC(CC2(C=C)CC2)=O)CCN(C(=O)C(C)OCc2ccccc2)C1 C1(CNC(CCCC(C)O)=O)C(C2CC2)CCN1C(=O)CCc1ccncc1 O=[N+]([O-])c1ccc(Cl)cc1Nc1ccc(-c2ccccn2)cc1 Cc1ccc(Br)c(C(N2CC(N(C(=O)C=Cc3ccn(C)c3)C)C2)=O)c1 c1(-c2cccc(C)n2)c(F)c(F)c(F)c(F)c1F Cc1ccc(C(=O)NCC2(O)CN(C(c3sccc3Br)=O)C2)c(C)c1Br CC1(C)C2CCC1(C)C2C(=O)NC1CCC(NC(c2ccncc2N)=O)C1 Cc1cc(C(=O)NC2CC(NC(=O)C(O)C3CC3)CC2O)nn1CCO O=C1CN(CC(=O)NCC23COC(CNS(=O)(=O)CC4CCOC4)(C2)C3)CCN1 C1(C(=O)NC(C)C(=O)NCC2(Cl)CCC2)CCCN1C1CC1 N1(C(C2C(OC)CN(C(C(NOC)=O)=O)C2)=O)CCC(CO)C(C)C1 C(=O)(CCCn1cccn1)OCCOCCOCCN=[N+]=[N-] C1(NC(C2CC(OCC)C2)=O)(CNC(C23CSCC2C3)=O)CCCCCC1 c1(OC(COCCCC)C)ccccc1.C(COC(C)(C)C)(CO)NCCNC c1(OCC(=O)NC2(C)CC(NC(CC3ON=C(C)C3)=O)C2)ccccc1C(C)C CCC(CC(=O)N1CCN(C(=O)C2=NOC3(CCC3)C2)CC1CCO)CC(C)C C1(CNC(C(CC)N(CC)CC)=O)CN(C(=O)C=CCN(C)CC)CCC1O C1(C(N2CCCCC(CO)C2)=O)CN(C(=O)CN2CC(=O)NC2=O)CC12CCC2 N1(C(c2ccc(C)o2)=O)CCC(C)C(CC(=O)NC(C)(C)C(=O)N(C)C)C1 O=C(CS(=O)CCC(F)(F)F)NCC1CCN(C(c2ncn3ccccc23)=O)C1 C#CCCCCC(=O)N1CCN(C(c2cc(OC)ns2)=O)C(CO)C1 C#CCC(C)(C(=O)N1CC(O)(CCO)C1)NC(=O)CCC1(C)CC1 C(C)(C(=O)NCC(C)(C)OCCNC(=O)C(=O)NCC(C)O)OC C1(F)(CNC(c2c(C)onc2)=O)CCC(NC(C2CCC(C)(C)C2)=O)C1 c1(C(N2C(CNC(c3c(C)ncc(Cl)c3)=O)CCC2)=O)cnc2c(c1)NCC2 C1(CCC)(NC(=O)CC2CCCC2)CCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 c1(C(=O)OC)cc(OC)cc(CN2CC(CO)C(F)C2)c1 c1(N(C)Cc2n(CC)ccn2)nc(N2CC(C(N)=O)OC(C)C2)c2c(n1)COC2 c1(C(N(C(CNC(CC(CC)c2ccccc2)=O)C)C)=O)cn2nc(C)sc2n1 C1(NC(=O)CSC(F)F)CCCCN(C(c2ccncc2N2CCCC2)=O)C1 CN1CCN(C)C(C(=O)NCC2CCC(NC(=O)CC3CC34CC4)CC2)C1 Cc1nc(NC(C2COC(C)C2)=O)sc1Br Cn1cc(CNC2CC3(C2)CC(NC(=O)C2=COCCC2)C3)c2cccnc12 N1(C(C(CC)SC)=O)CCn2nc(CNC(c3nc(O)sc3C)=O)cc2C1 CC(c1ccccc1C)=CC(=O)N(C1CCC(NC(=O)C(O)CC(C)C)CC1)C N1(C(CCC)=O)CC(CNC(=O)CN2CCCC(CC)C2)CC12CCC2 c1(C(=O)Nc2scc(-c3cn(C(C)(C)C)nc3)n2)ccc(Br)c(Cl)c1 C12(C(N3C(C(N4CCOCC4)=O)CC4CC43)=O)CC3CC(C1)CC(O)(C3)C2 C1(NC(CCN(C)CCSCCO)=O)C=CCCCC1 N1(CCC(N2CCN(Cc3cccc(C)c3C)CC2)=O)Cc2ccccc2C1 N1(c2cc(OC(C)C)ncn2)CCC2(CCCN(C(=O)C(C)(F)F)C2)C1 c1(C(=O)NCCC)cccc(NC(=O)CCOC(=O)C(C)OC)c1 c1(C(=O)NC2(CCNC(CC(C)(C)C)=O)CC2)cccc(F)c1SCCO C(C(O)CC(=O)NC1(CC#C)CCCC1)NC(C1(CO)CCCC1)=O C1(C2CCN(C(=O)CC3(O)CCCC3)C2)(NC(=O)C=CC2CCCC2)CC1 C=CC1(C(N2C(C(N3CCC3(C)C(C)C)=O)CC2C)=O)CCCCC1 C(=O)(CCC(CC)CCC)NC(CC(=C)C)C(=O)NCCCC=CC c1(CS(=O)(=O)NCC(=O)NC(c2cccnc2)CSC)ccc(Cl)cc1[N+](=O)[O-] c1(OC)cnc(F)cc1C(N1CCC(CO)(CNC(C2CC3CC3C2)=O)CC1)=O C1(NC(c2cnoc2)=O)CCCCC12CCCN(c1nc3ccc(Br)cc3o1)C2 c1(C(=O)NCCN(C(c2c(CC)nnc(C)c2)=O)C(C)C)ccc(C#N)cc1O CCS(=O)(=O)c1cccnc1C(=O)NCC1CC(NC(C2C3CCC2CC3)=O)C1 N1(C(COCCOCC)=O)CCN(C(=O)Cc2cc(Cl)cs2)CC2CCCCC12 c1(C(N2C(CN(C)C)CC(O)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C1(C(=O)NC2CN(C(c3cc(CCC)n(C)n3)=O)CC2O)CC(C)OC(C)C1 c1(OCCNC(C2NCCN(C(CC(=O)OC)=O)C2)=O)ccc(F)c(C(F)(F)F)c1 Cc1c(C(N2C(CC(C)C)CCC2C)=O)cccc1Br O=C(CC(Cl)Cl)NCC1(CNC(=O)COc2ccsn2)CC1(F)F N1(C(Cc2n(C)ccn2)=O)CCC(C)(CC(=O)Nc2ccc(Cl)cc2)C1 c1(C(N2CCC(N(C(=O)C(O)C3CC3)CC)C2)=O)ccn2cc(C3CC3)nc2c1 Cc1n[nH]c(C)c1CCC(=O)NCCN1CCN(C(C2CCCOCC2)=O)CC1 C1(OCC(=O)NCC(CN(C)C(c2cc(C3CC3)[nH]n2)=O)(C)C)CCC(C)CC1 FC1(F)CC(N2CCC(Nc3nccnc3I)CC2)CC1 C1(NC(C(C2CC(F)(F)C2)OCC)=O)(COC)CN(C(C2CC2C)=O)C1 C#CC1(C(N2CCCC3(CCO3)C2)=O)CCN(C(c2ccccc2C)=O)CC1 CCCC(O)C(=O)N1CC=CC1(C(=O)NCc1cncn1C)COC C#Cc1cc(C(=O)NCC2CC2CNC(c2[nH]c(C3CC3)nc2C)=O)cc(N)c1 c1(C(=O)NC(CC(C)NC(Cn2c(C)c(Cl)cn2)=O)C)n[nH]c2c1COC2 c1(NC(C2C(C(=O)NCc3ccc(O)nc3)C2)=O)cccc2c1OCO2 CC1CN(C(=O)C=CCN2CCNC(=O)C2)CC1CNC(C1(Br)CC1)=O C1(NC(C(CC=C)C)=O)CCN(C(=O)CSc2ccc(O)cc2)C12CC2 C1(O)(C(C(=O)NC2CC(C(=O)OC)C2)NC(C2SCCS2)=O)CCCCC1 c1(C(=O)OC)ccc(NC2CC(SC(C)C)C2(C)C)c(N)c1 c1(NC(C2CC(C)NC2)=O)nc(Cl)c(Cl)s1.N12CCC1CNC(=O)CNC(=O)C2 c1(C(N2CC3CC(NC(=O)Cn4cnnn4)CC3C2)=O)cncc2cnccc12 Cc1cn(C(C)(C)C(=O)NC2CC(N(C(=O)CC3CC3(Cl)Cl)C)C2)cn1 c1(C(=O)NC2CC(C)N(C(c3ncn4c3CCC4)=O)C2)c(Cl)cc(Cl)nc1N C1(CNC(CN(C)CC)=O)CC(C)(C)CN1C(C1CCN(CC)C1)=O CC#CC1CCN(C(C2CN(C(=O)COCc3nc[nH]n3)CCO2)=O)C1 c1(OCC)c(C(=O)NC(C2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)C)cccc1F N1(C(=O)OC(C)(C)C)CCCN(C(=O)CNc2n(CC)nc(C)c2)C(COC)C1 C1(C(=O)NC2(CCC(=O)NC3CCN(N=O)C3)CCCC2)CCCC1C1CC1 CCCCC(C)C(=O)NCCc1n[nH]cc1C(=O)NCC1CCC(O)C1 c1(NC23CCN(C(C(C)NS(CC)(=O)=O)=O)C2CCC3)cc(C)nc2ncnn12 C1(C(N(CC(=O)OC(C)(C)C)CC(F)F)=O)CN(C(=O)OC(C)(C)C)CCS(=O)(=O)C1 c1(C(=O)NCCOCCOC)oc(CNC(c2cnc(C)n2C)=O)nc1C Cc1c(C(=O)NC2CCSC2)nn(C)c1C1CC1 c1(C(=O)NC2C3(CC(NC(c4cnccn4)=O)C3)C2)ccc(Br)cc1F c1(NC)cncc(C(=O)NCCC2CN(C(C3CCCN3S(C)(=O)=O)=O)C2)c1 CC1CCCCC1(CNC(=O)CSc1ccncc1)NC(C1CCS(=O)(=O)C1)=O C1(C(N(CC(C)SC)C)=O)CCC2(CC2)N1C(=O)CC(C1CC1)C1CC1 CCC(O)C(C)(C)C(=O)N1CC(CNC(C2(CF)CCOCC2)=O)C(F)(CO)C1 CC1CN(C(=O)C2CC2)CC1(C)CNC(C1CC2(CSC2)C1)=O C(CCC(C)C(=O)NC(C)CCCNC(=O)Cc1cncn1C1CC1)OC N1(C(Cc2cc(C)on2)=O)CCCC(C2CCCCN2C(=O)CN(C)C(N)=O)C1 c1(OC)ccc(OC(F)(F)F)c(CNC(C2CC2NC(C2CC=CC2)=O)=O)c1 N1(C(CC2(OC)CCCC2)=O)CC(NC(=O)CSc2n[nH]c(O)n2)C(F)C1 c1(NC(NOC(C(=O)OC)(C)C)=O)c[nH]c2cc(Cl)cc(Cl)c12 CC1CCC=C1C(=O)N1CCC2(CC2NC(C2C=CCS2)=O)C1 C1(NC(=O)C2=CCCSC2)CC2(CCN(C(=O)CCSc3ccccc3Cl)C2)C1 c1(C(=O)NC(C2C(C(N(C3CCC3)CC#C)=O)C2)C)cc(C2CC2)on1 c1(OC)nccnc1C(=O)NC1CN(C(=O)Cc2csc(=N)[nH]2)CC1OC N1(C(c2cnc(COC)s2)=O)CC2CC1CN(C(C1CCC(OC)CC1)=O)C2 C(C(C)CN=c1[nH]cc(Br)cc1C#N)NC(c1c(CC)nns1)=O C(=O)(CC(F)(F)C(F)(F)F)N1CCCC(NC(CC2CCN(C)CC2)=O)C1 C(=O)(CC(C)CC(=O)NC1CCC(CCNC(=O)C2=CCOC2)C1)OC C#CC1(C(=O)NCCS(C)(=O)=O)CCN(C(c2ccsc2Cl)=O)C1 Cc1nn2c(c1C(N1C3CCC1CN(C(C14COCC(C1)C4)=O)C3)=O)CCCC2 C(C1=NOC2COCC12)NC1C(CCC)CCCC1 C1(NC(C(c2ccccc2)C)=O)COCCN(C(c2c(C3CC3)noc2C)=O)C1 c1(C(N2CCC(C(=O)NC3CC3)C2)=O)cnc2cc[nH]c2c1.C1(C2CC2)C(=O)N1 N1(C(=O)OC(C)(C)C)CCCCC1CC(C(F)(F)F)C(=O)NC(C)(C)C N1(C(C2C(C=C)C2)=O)CCC2(C1)CN(C(=O)C(C1CC1)SC)C2 Cc1nc(CCC(=O)NCc2nc(C)n(C)n2)[nH]c1C CC(CC(N)=O)C(=O)NC1CC(NC(c2cnc(C(C)C)[nH]2)=O)C1 C1(CNC(c2c(C)nco2)=O)CN(C(=O)Cn2c(C)c(C)sc2=O)CCN1C c1(C(N(CC(CNC(C(C)OC2CCCC2)=O)O)C)=O)cnc(S)[nH]1 c1(C(=O)NCCC(C)NC(c2nc[nH]c2C(C)(C)C)=O)ccc(N)cc1 C(=O)(C(O)C1=CCCCC1)NCC(C)N(C(CN(C(=O)OCC)C)=O)C C12(CNC(C3N(C)C(=O)CC3)=O)CC(CCO1)N(C(=O)CP(C)(C)=O)C2 c1(C(=O)OCC(N2CCCC(c3nnc(C)o3)C2)=O)nncc2ccccc12 c1(CC(=O)NCC(C2CCOC2)NC(C(=O)NC)=O)cc(OC)cc(Cl)c1 CC(=O)CCCC(=O)NCc1n[nH]cc1C(N1CCOC(C)(C)C1)=O c1(NC(C(CN(C(c2n(C(C)C)ccc2)=O)C)C)=O)cccc(Cl)n1 C(=O)(CC(O)CNC(=O)C(C)OCCN(C)C)NCCOCCC(C)C Cc1nn(C)c(C)c1C(C)C(=O)NCC1CCC(NC(=O)CS(N)(=O)=O)CC1 c1(SC)ccc(O)c(C(N2CCC(NC(c3ocnc3C(F)F)=O)C(F)C2)=O)c1 N1(C(c2cc(C)ns2)=O)CC(C2CC2C(=O)NC(c2nc(=O)o[nH]2)C)C1 C(=O)(C(O)C1=CCCCC1)NC1CCN(C(CC2(C#N)CC2)=O)CC1F CCC(CNC(=O)CC1CCC(=O)N1C)(CC)C(=O)N1CC(CO)(CF)C1 C1(NC(c2c(CC)nns2)=O)COC2(C1)CN(C(C1CCC1(C)C)=O)C2 CC1(C(=O)NCCC2(NC(C3CN(S(C)(=O)=O)C3)=O)CCC2)CCOC1 N1(C(CC)=O)CCCC1(C)CNC(C1CCC(C(C)(C)CC)CC1)=O CC(C(C)(C)C(=O)N1CCOCC1C(N)=O)NC(C1C2CC3C(C2=O)C13)=O CC1(C)CN(C(C23CCCC2C3Br)=O)CCC1NC(c1cn[nH]c1)=O c1(NC(C(C2CCN(C(c3cnc(O)[nH]3)=O)CC2)C)=O)ncc([N+](=O)[O-])cc1I C1(C(=O)NC(C(CO)NC(c2c(C)nsc2N)=O)C)CN(C)CCN1C CC1CN(C(C2CC(N)C2)=O)CC(C)N(C2CC2)C1 C12(CNC(C(C(C)C)F)=O)CN(C(c3cncs3)=O)CC1CCO2 C1(C(=O)NCCCOCCOC)CC2CCN(C(=O)C(C)(O)C(C)C)CC12 N1(C(C)=O)CCOC(C(=O)NCCC23CC(CCO2)C3)C1 c1(COC)ccccc1OCCN(C(=O)CN1CCCC(OC)C1)C C1(O)(C(N(CCNC(C(c2cccs2)SC)=O)C(C)C)=O)CCOCC1 N1(C(CNC(C(CC)C)=O)=O)CC(C2(NC(C3OCCCO3)=O)CC2)C1 c1(NC)cnccc1C(N1CCC1CNC(c1ccnc(OC)c1)=O)=O CC(CCCCNC(=O)C(C)c1cccs1)NC(=O)Cn1cnnc1O CC(C1CCCCC1)=CC(=O)NC(c1ccccc1)CNC(c1[nH]ccc1C)=O C1(NC(c2cnc(CC)s2)=O)CCCC(NC(c2cn(C3CCC3)nc2C)=O)C1 C=CCCCC(C(=O)NC(C1CCCC1)C)NC(C1CCOC1)=O C(c1ccsc1)=CC(=O)NCCC1CC(NC(=O)CCOC2CCC2)C1 C1(C(C)C)CN(C(c2ccc(F)c(CO)c2)=O)CCN1C(c1cn(C)[nH]c1=N)=O C(=O)(C(O)(C(C)C)C(F)(F)F)NC1(CNC(c2c(C)snn2)=O)CCCCC1C C(=O)(C(F)(F)CC1CC1)NCCCN(C(c1nc(Cl)sc1C)=O)CC c1(C(=O)NCC2C(NC(c3occc3Br)=O)CC2)cccc2ccnn12 C1(CNC(C2CCC=CCC2)=O)CC12CCN(C(C1CC3(CCCC3)C1)=O)CC2 Cc1cccc(C(=O)NC2CC3(C2)CC3NC(c2cc(C3CCC3)[nH]n2)=O)c1Cl CCCC(CNC(C1(OC)CCN(C(c2cc(C)nn2CC)=O)C1)=O)CCO Nc1cc(Cl)ccc1C(=O)NC1CC1CNC(=O)CCc1ccc(Br)cc1 C1(CC=C)CCN(C(C2C=CCN(C(=O)C(C)NC(=O)NC)C2)=O)CC1 C1(C(N2CCC(C(=O)NC)C2)=O)(COC)CCN(C(c2cncc(C)n2)=O)C1 C(=O)(C1CCCc2ccnn21)N1C(CNC(C(C)(C2CC2)NC(C)=O)=O)CC1 CC1C2CC(C2NC(=O)CCc2cn(C)nn2)N1C(=O)C(C)(C)C(=O)OC(C)(C)C C1(NC(C(C)O)=O)CN(c2nccc(C(F)(F)F)n2)CC1F Cc1ccc(C=CC(N2CC(C(O)C(N3CCC(N(C)C)CC3)=O)C2)=O)o1 N(C(=NCC1(CO)CCC1)NC(C1CCOC1)C)CC(=O)NC(C)C N1(C(CCC=CCC=C)=O)CCN(C(=O)Cc2ccnn2C)CC1CC(=O)NC C(=O)(CC(C)CC(F)(F)F)NCC12CCN(C(CCCC(=O)OC)=O)C1CCC2 N1(C(COC(CC)C)=O)CCCC1CCCNC(c1n[nH]cc1C(C)(C)C)=O c1(C(=O)OC)cscc1-c1c[nH]c(=N)s1 c1(CNC(c2c(C)cccc2)c2ccc(F)cc2)nn2ccccc2c1Br C1(N(C(C(CC)(C)C)=O)C)CCCN(C(=O)CC2CCC(=O)O2)CC1 C(=O)(C(O)CC(F)(F)F)NC(C(=O)NCc1cnn(CCF)c1)Cn1cncn1 C=C1CCN(C(c2ccc[nH]2)=O)C(C(=O)NCC(C)N=[N+]=[N-])C1 C1(C(F)(F)F)(C(N2C(CNC(=O)Cc3csc(Cl)n3)CC2)=O)CCCCCC1 CC1C(NC(C2C(C)C2C)=O)CCN1C(c1ncoc1C1CC1)=O C1(C)(C(=O)OC)CC(C(=O)NCC2CCCN2C(C2CC(O)C2)=O)C1 C1(N=[N+]=[N-])(NC(C2COCCN(C)C2)=O)CCN(C(C2CN3CCC2C3)=O)C1 Cc1ccc(=O)n(CC(=O)NCC2CN(C(C3CCCN(C)C3)=O)CC23CC3)n1 CCCC(CCC)C(=O)N1CCCC(NC(c2ccc(C)o2)=O)CC1 c1(NC2CCN(Cc3c([N+](=O)[O-])ccc(O)c3)C2)c(F)c(F)c(F)c(F)c1F c1(C(=O)NCCN(C(=O)C(C2CC2)OC)CC)cc(Cl)cc(Br)c1N n1(CC)nc(C)c(CN2C(C(=O)Nc3ccccc3CC#N)CC3CC23)c1C C1(C(=O)NCC2CC2(Cl)Cl)CN(C(=O)CN2CC3CC3C2)C2(CCC2)C1 C1(NC(c2ccc(C)c(CO)c2)=O)CCN(C(C2CCC2C)=O)CC(C)(C)C1 C12(NC(=O)CNC(C3C(C)C3)=O)CC3CC(C1)CC(CNc1nccs1)(C3)C2 N#CC1CCC(C(=O)NC2CCC(NC(c3ccc(OCCO)nc3)=O)CC2)C1 c1(C2C(C(=O)NCC3NCC(C)(C)C3)C2)cc(Br)ccc1F C1(C(=O)NCC(CC)N(C)CC)CCCN(C(=O)C2=C(Cl)CC2)CC1 C1(CNC(C(CC=CC)NC(c2ccc(CN(C)C)o2)=O)=O)CCC(=O)NC1C N1(C(CCCNC(C)=O)=O)CC(CNC(C2CC(C)(O)C2)=O)C(C)(C)C1 C1(C(N(C2CCN(C(c3n(COC)ncc3)=O)C2)C)=O)CC(F)(F)CCC1(C)C C1(C(=O)NCC2(CC(C)C)CCC2)(NC(C2CCCO2)=O)CCN(C)C1 c1(C(N2CC(CC)C(NC(=O)CC(CC)CC)CC2)=O)ccc(C)c([N+](=O)[O-])c1 c1(C(N2CCC(CNC(C(F)OC)=O)C2)=O)cc(C#N)c(C)cn1 c1(C(=O)NCCCNC(c2c(C(C)(C)C)noc2)=O)ccnc2ccc(F)nc12 C1(F)(C(N(CCC(=O)NCCn2c(CC)nnc2)C2CC2)=O)CCOC1C c1(SCC(=O)NCCC2CC(NC(CC3(OC)CC3)=O)C2)cc2ncccc2s1 c1(C(=O)NCCC2CC(NC(C3CCC(F)C3)=O)C2)nccc2occc12 c1(OC)ncnc(NC(C2CC3CC3N2Cc2cccnc2)=O)c1OC N1(C(CC(C)(C)OC)=O)CC(C)(C)CCC1CNC(=O)CC1CCC(C)(O)CC1 O=C(N1CCCc2ccnn21)c1snc(Cl)c1Br c1(NC(C)=O)cccc(-c2cn(C(=O)CCNC3C(C)C3(F)F)nn2)c1 c1(OC)cc(C(=O)NCC(N2CC(C)OC(C)C2)C)sc1S(N)(=O)=O C1(C#CC(=O)N2CC(C)(C(=O)NCCC(C)O)C2)(CC)COC1 Cc1ccc(C(N2CCN(C(=O)CSC(C)(C)C)CC2CF)=O)c(N)c1C Cc1cc(NC(n2cnnc2)=O)sc1C(=O)N(C(C)CNC(=O)CC(F)(F)F)C O=C(N=c1ccnc(N2CCC3OCC(=O)NC3C2)[nH]1)C1CC2(CCC2)C1 Cc1cccc(=O)n1CC(C)(O)C(=O)NCCCCC(C)NC(=O)CP(C)(C)=O CCCCC(C)(F)C(=O)N(C1(C(=O)NCCCC(=O)NO)CC1)C c1(C(N2CC(C(=O)Nc3cnccc3Br)OCC2)=O)cc2ccccc2[nH]1 c1(OC)cc(F)c(F)cc1NC(=O)NCc1cc(F)c(F)c(F)c1 c1(NC(CC2(OC)CN(C(C3(OC)CCOC3)=O)C2)=O)ncc(C(N)=O)cn1 c1(NCCc2c(C)cc(Br)cc2C)cc(C)c(S(=O)(=O)N(C)CC2CC2C)cn1 C=Cc1cnn(C)c1C(=O)NC1COCCC1NC(C1CN(C(N)=O)C1)=O c1(C(=O)NC(C(C)(C)C)CNC(=O)CC2(C)CCCC2)cc2cccc(F)c2o1 C(=O)(C#CC1CCOCC1)N1CC2(CNC(CCC(=O)N(C)C)=O)C(C1)CCO2 N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)CCc2nc(C(F)(F)F)n[nH]2)C2CCC12 CCCCCC(O)CC(=O)N1CCC(CNC(c2coc(CO)c2)=O)(OC)CC1 C(c1cncc(O)c1)=CC(=O)OCCSCC(N1CCCCC1c1ccc(Cl)nc1)=O c1(NC(=O)NCC2N(C(c3nc(CCCCC)sc3)=O)CCC2)nc(=O)n(C)[nH]1 C(CC)(C(=O)NC(C)CCCNC(c1ccc(Cn2cccn2)o1)=O)OCC c1(OC)ccc(Cl)cc1N1CCC(NC(C2CC(OC)C2)=O)C1 N1(C(CCCC=C)=O)CCC(O)C(NC(c2cc(Cl)cnc2OC)=O)C1 N1(C(CC=C(C)C)=O)CC=C(CCNC(c2nocc2C2CC2)=O)CC1 c1(SCC(=O)NCC(CNC(C(CC)Nc2ccccn2)=O)F)cccc(C)c1 C1(C)(NC(c2cc(C)sn2)=O)CCCN(C(c2ccncc2C2CC2)=O)C1 c1(C(=O)NCC(C)NC(C(CC)n2cncn2)=O)c(C(F)(F)F)cc[nH]c1=N c1(C(=O)NCC(CC)NC(c2nc[nH]c2C(C)(C)C)=O)ccc2c(c1)CCO2 CCC(C#N)C(=O)N1CCN(C(=O)C(n2cc(-c3ccccc3)nn2)C)CC1 C12(C(NOCC(C)O)=O)CCCC1CN(C(C13CCCN1CCC3)=O)C2 c1(C(=O)NCCCCC(C)NC(c2cn(CC=C)nn2)=O)ccccc1S(C)=O n1(CCC(=O)NC2CC3CCC2(C(=O)O)C3)c(=O)oc2cc(Cl)ccc12 c1(C(N2CC(NC(C(=O)NCCNC(C)=O)=O)C(C)C2)=O)cnc2nccn2c1 Cc1cnc(C(C)NC(=O)NC2CCOC2C2CC2c2ccccc2)s1 C1(C(=O)NC2C(NC(c3n(CC#C)ccc3)=O)CC2)CCC2CC1C2(C)C c1(N2CCN(C(c3ccc(OCC#C)cc3)=O)CC2)ncnc(OC)c1[N+](=O)[O-] Cc1c(C(=O)NCC2CN(C(C3CCC(C(N)=O)CC3)=O)C2)nn2c1CCCC2 Cc1cccc(C(C)C(N2CCC(O)(CCNC(c3ncccc3Cl)=O)C2)=O)c1 C(C)(C)(CC(F)C(=O)NCCC(C)N(C)C)NC(c1cccc(C)c1C)=O c1(C(=O)NC2(CCNC(C(COC)N(C)C)=O)CCC2)cnc(O)cc1C c1(CN(c2c(C)cc(F)cc2)C)ccc2c(C)c[nH]c2c1.c12cnn(C)c1c2=O c1(C(N2C(CC)C(NC(C3CC=CC3)=O)CC2)=O)ccc(S(C)=O)cc1 CCC(C)(C(=O)NCC#CCNC(C1COC(=O)C1)=O)C(N)=O c1(C(N(C2CN(C(CC3CCCN(C)C3)=O)C2)C)=O)cccc(P(C)(C)=O)n1 Cc1cc(F)ccc1C(=O)NCC1CCCN(C(C2CCCCS2(=O)=O)=O)CC1 C1(NC(C(c2ccccc2)OC(C)C)=O)CC2(C1)CC2NC(=O)CC(C)C1CC1 c1(C(=O)NCC2N(C(C(C)CC(F)F)=O)CC2)coc(C#Cc2ccccc2)c1 c1(NC(C(N2CCN(CCOCC)C(=O)C2)=O)=O)ccc2c(c1)CCC(O)C2 C12(NC(C(C)=C(CC)C)=O)CCCC1N(C(c1c(C)cnn1C)=O)CC2 CC(C)CCCC(=O)N1CCCCC1(C)c1ccccc1 C1(NC(C(CC=CC)NC(=O)C2=C(C)CC2)=O)CC2C=CCC(C1)C2 N1(C(CC(=C)Br)=O)CC(C)C(NC(=O)CN2C(=O)NC(C)(C)C2=O)C(C)C1 C(C(C)(C)C(=O)NC1CCN(C)CC1)N(C)C(=O)NCC(F)(F)CC1CC1 c1(C(=O)NC(c2cccnc2)C#N)cc(Cl)c2[nH]c(O)nc2c1 N1(CC=C)CC2(CCC(C(=O)NCc3ccc(CNC(=O)CC(=O)OC)o3)O2)C1 c1(NC(c2n(CCC(=O)OCC)nnn2)c2cn(C)nn2)ccc(Br)cc1Cl C1(C(=O)NCC2CC(NC(C3CC3C3CC3)=O)C2)CC2(CCC2)C1 N1(C(c2c(NC)snc2C)=O)CC2=C(C1)CN(C(c1ccccc1Br)=O)C2 c1(C(=O)NC2C(NC(C(C)(C)C#N)=O)CC2)nnn2c1CCCC2 C=CCC(CNC(=O)CNC=O)NC(=O)CC1CS(=O)(=O)C1 c1(C(=O)NCCN(C(=O)CC2(C)CC2(F)Cl)CC)ccc2cc(O)ccc2c1 N1(C(CCC(=C)Cl)=O)CC2CCC2(NC(=O)C=Cc2nnn(C)n2)C1 N1(C(C2(C)CC2(F)Cl)=O)CC2CC(C1)C2NC(=O)CC1CC1 C(=O)(CCCN(C(c1cc(C2CC2)[nH]n1)C(=O)NC1CC1)C(C)C)OC C12(CCN(CCC(=O)NC3CC3)CC1)C(=O)N2.C1(COC)CC12CCSCC2 C1(C2(O)CCC2)(C(=O)NC(C2CCN(C(c3cn(CC=C)nc3)=O)C2)C)CC1 N1(C(=O)OC(C)(C)C)CCCN(CCC#N)CC1.C12CCC3(CC13)CCNC2=O c1(OC)nc(N2CCC(C(=O)NCc3cnco3)C(O)C2)ncc1Br CC(CC(F)(F)F)C(=O)NC1CC(C)(NC(=O)C(C)Oc2ccccc2F)C1 N1(C(=O)NCc2c(C)ocn2)CCC12CCCCC2 c1(C(=O)NCC(C2CCN(C(=O)OCCl)CC2)C)cccc(I)n1.C(C)(C)C Cc1ccc2oc(C(N3CC4CCC4(NC(c4ccc(Cl)cn4)=O)C3)=O)cc2n1 C12(n3cc(CN(C(C4CCC(CC)O4)=O)C4CC4)nn3)CCC(C(=O)OC)(CC1)C2 C(=O)(C#CC(C)(C)CNC(C1CCSC1)=O)N1CC(N(C)C)C1 C1(C(=O)NCC(CSC)(C)C)CC12CCN(C(c1ccn(CCF)n1)=O)C2 c1(-c2cncnc2)c[nH]c2nccc-2c1.Oc1ccc(CCn2ccnn2)cn1 N1(C(CCCSC)C(=O)NCC(F)F)CCC2(CC1)CN(C)C(=O)O2 N1(C(C23CC(NC(CCC#C)=O)(C2)C3)=O)CCc2ccc(O)cc2C1 N1(C(C(C2CCC2)OCC)=O)CC2CCC2(C(=O)NCC2(C)CC(F)(F)C2)C1 c1(OCC)cc(C(=O)NCC2(CO)CN(C(c3cscc3OC)=O)C2)ccc1C CC(C)(C)CC(C)(C)C(=O)NCC1(NC(=O)Cc2ccccc2Br)CC1 C1(NC(c2c(C)noc2C)=O)C2CCN(C(=O)C(C)(C)c3ccccc3)CC12 c1(C(=O)NC2C(CNC(CC3(COC)CC3)=O)C2)cc(Cl)ccc1SC1CCCC1 c1(C(N(C2CCC(NC(=O)CCC3(C)CC3)C2)C)=O)cc(C(F)F)no1 c1(NC(N2CCN(C)C(c3nccn3C)C2)=O)cc(F)c(F)c(F)c1O CC1(C)CC2(CC2C(N2CCC(NC(c3ncnc4sccc34)=O)C2)=O)C1 Cn1nnc(C(=O)NC2CCN(C(C3CC=CCC3)=O)C2C2CC2)c1C(F)F C1(NC(CNC(=O)CNC(c2ccc(CF)cc2)=O)=O)CCC2(CC2)CO1 Cc1cn2c(n1)CCC(C(=O)NCC1CCN1C(C1CC(=O)NC(=O)C1)=O)C2 C12(C(N(C3CN(C(C=Cc4c(C)n[nH]c4)=O)C3)C)=O)CCC(C(=O)O)(CC1)CC2 C1(NC(C(C)(C)n2cncn2)=O)CCOCC1C(=O)N(C1CCC1)CCO C1(CNC(C(=O)OC)Cc2cn(C)cn2)CC(C)(C)CN1 C1(N(C(C(C(=O)OC)OC)=O)C)CCCCN(C(=O)CCN2CCC(C)CC2)C1 CCCC(C)(C)CC(=O)NCC1C(C)CCN1C(c1ncccn1)=O N1(C(N(CC)CC)=O)CCC2(C(N3CCC3(C)C(=O)OC(C)(C)C)=O)CC2C1 O=C(CC1NC(=O)c2ccccc21)NC1CCCC1CNC(=O)C1=NOCC1 c12cccc(F)c1C(=O)N2.Cc1ncc(CN2CCC(C)(N(C)C)C2)cn1 c1(C(NCCC)=O)cccc2c1nnn2C.C1(CC)CCN(C(=O)CN(C)CC)C1 C(CS(=O)(=O)C1CCN(c2nc(N3CCC(C)C3)nc3c2CCCC3)CC1)OC N#Cc1c[nH]c(=NC2CCC(C(N3CC4C(C3)C4(F)F)=O)OC2)c2sccc12 N1(C(C(c2c(C)n[nH]c2C)C)=O)CCC(O)(C2(NC(C3CCOC3)=O)CC2)CC1 O=C(C#CC1CCCCO1)NCC1CC1CNC(c1cc([N+](=O)[O-])c[nH]1)=O c1(CNC(C(CC)C)=O)cccc(NC(=O)C(C)CN2CCCCC2)c1 C1(CNC(C(CC)SC)=O)CC2(CCN(C(=O)Cc3cc(C)on3)C2)CO1 c1(OC)cc(C(N2CC3CC2CN3S(=O)(=O)CC2CCC2)=O)cnc1Cl C1(NC(C2CCOCC2)=O)CC2CN(C(c3ccnc(Cl)c3F)=O)CC12 C(CCC(=O)NCCOCCC(C)C)NC(CC1CC(=C)C1)=O C(C(CC(F)(F)F)NC(C1CCCS1)=O)NC(CCNC(=O)CO)=O c1(C(=O)NC(CN(C(c2ccc(OC)cc2N)=O)C)C)ccc2nc(Cl)nn2c1 c1(C(=O)NC2CCC(N(C(C(C(C)O)C)=O)C)CC2)cnn2ccnc(N)c12 CC1CCN(CC(=O)NC2CCC(CC(=O)N(C)CC3CC3(F)F)C2)C1 C(CN=c1cc(-c2cncc(Cl)c2)nc[nH]1)NC(CN(C1CC1)CC)=O c1(CC)conc1COCCNC1COCC1F CC1CN(C(=O)COC2CCOC2)CC1NC(c1cncc(N(C)C)c1)=O c1(OC)cc(C(=O)NCC2CC(C)(C)CN2C(=O)C(C)=CC(C)(C)C)ccc1Cl C1(C(N2CC(C(N(C)C)=O)C2)=O)CC12CCCOC2 C1(C(=O)NC(C)C(=O)N(C)C)CC2CCC(C1)N2C(=O)C(F)C(C)(C)O C1(OC)CCC2(CCN(C(C3CC=CCN3C(c3cnc(Cl)s3)=O)=O)C2)C1 c1(C(COCCOCCOCC)NC(N2CCCC2)=O)ccc(F)cc1.C1CC1 c1(OC)cccc(-n2cc(-c3csc(OC(C4CCN(CC)CC4)=O)c3)nn2)c1 c1(OC)ccc(-c2nc(CC3CCOC3=O)n(-c3ccc(=O)n(C)n3)n2)cc1F C(=O)(C#CC1CCOC1)NC1CC2(C(NC(=O)CCNC(c3ccoc3)=O)C2)C1 C(N=c1nc(C)nc2[nH][nH]cc1-2)C1(OC)CN(C(c2nnn(C(C)C)c2C)=O)C1 c1(C(N2CCC(C(=O)NCc3cn(C)nc3C)(CC)C2)=O)nccc(C)c1N N1(C(CCC(C)NC(C(CC(=O)OC)C)=O)=O)CCN2CC(C)CC2C1 Cc1cc(C(N)=O)cs1.c12nnnn1C1CC(CC2(C)N)C1.C(C)(C)C N1(C(CC2(CC)CCOCC2)=O)C2CCC1(CNC(c1csc(C)n1)=O)CC2 N1(C(c2c(C)cno2)=O)CCN(CCN(C(=O)C(N2CCCC(O)C2)C)C)CC1 C1(C(=O)NCCc2n(C)ncn2)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CCO1 N1(C(C(c2c(C)noc2C)(C)C)=O)CC(NC(C2CCCC2O)=O)CC2(CC2)C1 c1(CC(=O)N(CCC(C2CCCC2)NC(C=CC)=O)C)ccncc1 c1(CC(C)NC(=O)C2=COCC2)ccc(CNC(=O)Cc2cnc[nH]2)cc1 Cc1ccc2c(c1)CN(C(=O)C1=NOC(CNC(C3CC(F)C3)=O)C1)C2 N1(C(c2ccsc2C(=O)OC)C(=O)NC)CCN(CC2CC2)C(CC)C1.COC c1(CC(C2(O)CN(C(=O)OC(C)(C)C)C2)NC(C2(C)CCC2)=O)ccccn1 c1(C(=O)NCC(=O)NC(C2CCOC2)CNC(CCC=CC)=O)ccccc1Cl CCCC(CC)CCC(=O)NCC1CN(C(c2cc(Cl)ncc2O)=O)CCCO1 CCC(C)CC(C(=O)NC(C)C(=O)N(C)CC)NC(=O)Cc1ccco1 CC(C)C(O)CNC(=O)C(C1CC=CCC1)NC(=O)CCC1(C)CC1 N1(Cc2c(OCC(=O)O)cccc2)CCCC(C(=O)NCCCCCCO)CC1 Cc1cnccc1CCNC(=O)NC(c1nncs1)C1CC1 C1(C)(NC(C(C)SCC)=O)CCCN(C(C23CC4CC2C3C4)=O)C1 c1(C(N(C(C)C(=O)NCc2ncsc2C)CC)=O)cnn(CCF)c1 N1(C(C2(CC(=O)OC)CC2)=O)CC2CCC(CNC(C3CC(C)(C)CO3)=O)(C2)C1 c1(C(=O)NCC2C(C)CCN2C(c2ccc(=O)oc2)=O)nn(C)c2c1CCC2 C(CCCC(CO)NC(c1ccn(C(F)F)n1)=O)NC(c1c(SC)scc1)=O C12(C(=O)NC(CCC)C)CCC(NC(C3CCC(=O)O3)=O)(CC1)C2 c1(C(=O)NCC(CNC(C2C(OC)CCCC2)=O)(C)C)c(Cl)ccc(Cl)c1O C1(NC(C(C)n2cncn2)=O)CCC(NC(=O)C(=O)Nc2ccccc2)C1 C1(CC(=O)NC2(C3CCCCN3C(c3cc(F)cs3)=O)CC2)(OC)CCOCC1 c1(C(=O)NC(C)C(N2CCC(F)(Cc3nn[nH]n3)C2)=O)cccc(Br)c1 N1(C2C(=O)NCC2)CCC(NC(c2cc3sccc3s2)=O)C(O)C1 N1(C(c2n(CC)ccn2)=O)CCC(O)(C(C)NC(=O)C=CI)CC1 N1(C(CC2(OCC)CCC2)=O)CCCOC(CCNC(=O)Cc2cnns2)C1 C#CCCCCCC(=O)NCC(C)CC(=O)N(C)CC1CC1 c1(NC(=O)NCC2CCCOC2)c(I)cc(Br)c2ccccc12 c1(C(N2CC3C(NC(C4CC(C)C4)=O)(C3)C2)=O)ccc(O)c([N+](=O)[O-])c1 Cc1nn(C)cc1C(=O)NC1CN(C(c2cc(C(F)(F)F)ns2)=O)C1 c1(CC)cccc(C(N2CCC(C(N3CCC3(C)C)=O)C2C)=O)c1 N1(c2ncc(C)s2)CC2C(C(=O)NC(c3cccc(C(C)C)c3)C)C2C1 CC(CCC(F)F)NC(=O)NCC(c1cnn(C)c1)C Cc1nccc(C(=O)NC2CCC(CNC(c3c(C)noc3C(F)F)=O)C2)c1C C1(NC(Cc2cc(OC)c(O)cc2)=O)COC2(CCN(C(=O)C(S)C(C)C)C2)C1 N1(C(=O)NCC2CCCCO2)CCC(O)C2CCCCC12 C(=O)(C(C(C)C)n1cc(Br)nn1)NCCC#C.C12(CC1)COC2 C1(C(C)(C)O)CCC(C(=O)NC2CCC(C(=O)N(C)C)CC2)CC1 N1(C(CC2C(C)(C)C2(C)C)=O)CC2CCC1C(NC(c1cnn(C(F)F)c1)=O)C2 N1(C(CC(C)C(F)(F)F)=O)CC2CCC1C1CN(C(c3cc(O)ncn3)=O)CC21 C=CCCC(F)(F)C(=O)N1CCC(F)(CNC(c2cncc(F)c2Cl)=O)CC1 N1(C(=O)OC)C(C(=O)NCC2CCC2C(=O)NCC(C)O)C1C C1(NC(CC(C)N2CCCC2=O)=O)CC2CN(C(c3ccc(O)nn3)=O)CC2C1 C(=O)(C1=CC2(CCOC2)C1)NCCC1CCCN(C(c2c(C)cnnc2O)=O)C1 C1(CNC(c2cc(C(C)C)[nH]n2)=O)CCC12CCN(C(c1cncnc1)=O)CC2 c1(SC)cc(C(=O)NCC2(NC(=O)CCC(C)N(C)C)CCCCC2)ccc1F c1(C(=O)NCC(C)NC(C(CCSC)O)=O)cc(F)cc2ccoc12 C1(CNC(=O)COCC2CCOCC2)CCCN(C(c2n[nH]cc2C2CC2)=O)C1 c1(OC)ccc(OC)c(CC(=O)NC(C2CN(C(=O)CCc3ccon3)C2)C)c1 N1(C(CNC(Cn2c(C)ncc2)=O)=O)CC2CC2(CNC(c2ccoc2C)=O)C1 c1(CC(=O)N(CCCNC(=O)CC2CC3CC3C2)C2CC2)ccnc(O)c1 C12(C(=O)NCC(CCNC(c3c(C)nsc3N)=O)O)CC3CC(C(=O)N1)C2C3 C1(n2cc(CNC(c3cc(C(=O)O)cc(O)n3)C)nn2)CCC(F)(F)CC1 c1(C(N2CC(F)(CNC(C34CSC(C3)C4)=O)C2)=O)cc2c(Cl)nccc2s1 c1(C(N(C2CCCN(C(C3(C4CC4)CC3)=O)C2)C)=O)cccc2c1NCC2 C1(CSc2c(OC)cncc2)CN(C(=O)OC(C)(C)C)CC1(F)C(=O)O c1(OC)cc(N)c(F)cc1C(=O)NC1(C)CC(NC(=O)Cc2ccoc2)C1 C(C)(C)(CC(=O)NCC1CN(C(c2cnns2)=O)CC1C)OC S(=O)(=O)(c1ccc(Br)cc1NCC1(C)CCC(=O)N1C)NC(c1cc(Br)cs1)C c1(OC)cc(C)ccc1C(=O)NC1CCCC1NC(=O)CC1CC1C(F)(F)F C1(NC(Cc2ccc(-c3cn(C(C)C(=O)O)nn3)cc2)=O)COC2COCC12 c1(C(=O)NCC2C(CC)CCN2C(=O)Cc2ccsc2C)cc(C)c(F)c(C)c1 C1(C)(C(=O)NCC=CC(=O)N(CCN(CC)CC)C)CCNC1=O C1(CN(C(COC(CC)(C)C)=O)C)CCC(NC(c2cccc(Cl)c2)=O)CC1 c1(C(CNC(CN(C(=O)CC2CC3C=CC2C3)CCC)=O)=O)cccc(C)c1 CC1CN(C2CC2)CC1NC(C1(C)CCC1)=O.C1(C(=O)N)CC(=C2CCC2)C1 N1(C(c2cccc(C(=O)OC)n2)=O)CCC2(CCN(Cc3cccc(N)c3)CC2)C1 CC(C)CC(=O)N(CCCC(=O)NC1CC(NC(=O)CCNS(C)(=O)=O)C1)C C1(NC(CN(CC)CC)=O)CCCCC1NC(=O)C=Cc1cscn1 c1(C(N2C(C)C(NC(=O)CC3CC(F)C3)C(C)CC2)=O)cc2c(cn1)OCCC2 CC1CC(=O)NC1C(=O)NCc1ccc(C(=O)NC2CC(CO)N(C)C2)cc1 c1(N2C(C(=O)Nc3ncc(F)cc3F)CC(F)(F)C2)ncnc2ccc(Br)cc12 N1(C(C2CCC(C)CC2)=O)Cc2occ(C(=O)NCCC3CC3C)c2C1 C(N=c1[nH]cncc1Cl)C1CC(NC(c2ccc(OC)c(Cl)n2)=O)C1 C1(OC)CN(C(=O)CC2(C)CCCO2)CC1NC(C1(c2cccc(Cl)c2)CC1)=O c1(C(N2C(CNC(C3(CC=C)CCC3)=O)CCC2)=O)cccc2ncc(C)cc12 CC(C(=O)NCC#CCNC(=O)CCNC(=O)C=C1CCCC1)=CC1CC1 N1(C(CC(CCOC)(C)C)=O)CCCC12CCN(C(=O)CC1(C)CCOC1)C2 CC1CCCC=C1C(=O)NCC1C2CCC(C2)N1C(c1ccnc(O)c1)=O C1(CC(N2CCC(N(C(C3CC(F)(F)C3)=O)CC)C2)=O)CC(C)(C)OC1=O c1(C(=O)NC(C)CN(C)C(c2ccnc(C(C)(F)F)c2)=O)ccc(Cl)cc1N C(=O)(C(F)CC(CC)CC)NCc1occ(C(=O)NC(C(CC)C)CO)c1 CN=c1[nH]c(=NCc2cc(Br)ccc2F)[nH]c(=NC(C)Cc2ccccc2C)[nH]1 c1(C(=O)O)nc2cc(Cl)c(S(=O)(=O)N3CCC(CO)C(O)C3)cc2s1 C1(C)(NC(=O)OC(C)(C)C)CCCCC1NC(=O)NCCc1cccc(O)n1 c1(C(=O)NCCNC(C2(C)CS(=O)(=O)C2)=O)ccc([N+](=O)[O-])o1 N1(C(N2CCCC(C(=O)Nc3ccccn3)C2)=O)CCCC2CCNCC12 C1(=CC(=O)NCCC2CN(C(C3CC3F)=O)C2)CCCCC1 c1(C(C)C)cccc(C(N2CC(C(N)=O)(CNC(C3CC(F)(F)C3)=O)C2)=O)n1 C1(C(=O)NC2(C)CC(NC(c3ccc(F)cc3N)=O)C2)CCC2(CC1)CC2(F)F C1(N(C(=O)C(F)OC(F)(F)F)CCC)CCN(C(C2(Br)CC2)=O)CC1 c1(OC)cc(CNC(c2ccc(F)cc2OC)c2nnnn2C(C)C)cc(Br)c1 C1(N(C(C(COCC)NC(=O)C=CCO)=O)C)CCC(=O)N(C)C1 CC(C)CC(C(=O)NCC1CC12CCC2)N(C)C(C1CCC(C)(O)CC1)=O C12(NC(c3c(COC)ccs3)=O)COC(CNC(c3cc[nH]c3)=O)(C1)C2 c1(CCCC(=O)NC2CCC(F)(CNC(C(CC)(C)O)=O)C2)cc(C)ccc1C C1(NC(CC2C(C)C2)=O)CC2CC(C1)N(C(c1cccc3[nH]ncc13)=O)C2 C=CCCCC(=O)NCCCCC(C)NC(=O)C(c1ccc(C(F)(F)F)s1)=O c1(N(CCCOC)C)nc(=N)[nH]c(=NC(C)CC2CCCO2)[nH]1 C1(C(N2C(C)(CO)CCC2)=O)CCN(C(=O)C2CCOC(=O)CC2)O1 c1(C2CCN(C(C(C)CC3CCC3)C(=O)NC3COC3)C2)ccc(Br)c(F)c1F CC1CCCC=C1C(=O)N1CCC1(C)CC(N1CC(=O)NC(=O)C1C)=O c1(OC)ccc(Cl)cc1C(=O)NCC1(CNC(CNC(=O)OCC)=O)CCCC1 C1(NC(C2(C=C)CCC2)=O)CC2CC1N(C(C1CCC(F)(F)C1)=O)C2 N1(C(C(C)(C)C#N)=O)CCC2(CCCCC2NC(c2cccc(Cl)n2)=O)CC1 C1(F)(CNC(C2N(C)CCOC2)=O)CCN(C(=O)COCC2CCOC2)CC1 Cc1c(C(=O)NCC2CC(NC(=O)C(C3CCOCC3)F)C2)sc2ccccc12 c1(OC)ccc(OC(C)C(=O)NCC(C)CN(C(=O)C=CCF)C)cc1 N1(C(c2nccnc2Cl)=O)CC(C2CCCCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 CC1CN(C(c2cnccc2Br)=O)CCN1C(C1CCCNS1(=O)=O)=O C1(C(=O)OC)C(NC(C2(CC3CCC3)CC2)=O)CCCN1C(=O)C1=CCCC1C C1(NC(CCc2nc(C)sc2)=O)CCC(Nc2ncc(I)cn2)CC1 C1(CNC(C2(CC)CC(C)(C)C2)=O)COC(C)(C)CN1C(C1CCC1(C)C)=O N1(C(Cc2c(C)nn(C)c2)=O)CC(NC(=O)CCC(C)(C)N(C)C)C2CCCC12 CC(C)(CC(=O)N1CCCC2C1CCN2C(=O)CCCC1CC1)CC(F)(F)F C12(C(=O)NCC3(CC)CCC3)COCC1CN(Cc1ncccn1)C2 N1(C(Cc2nc(C)c(C)[nH]2)=O)CCC(NC(=O)CCNC(=O)CC(C)C)C(F)C1 N1(CC)CCCC(ONC(=O)C(C)N(C(=O)C(F)CC2CCCC2)CC)C1 CC1CC(NC(c2cncc(C#N)c2)=O)CCN1C(=O)C=CC(C)(C)C C1(NC(CCSC)=O)CCC2CN(C(c3cnc4[nH]cnc4c3)=O)CCC2C1 N1(C(CC2C(NC(C(N)=O)=O)CCCC2)=O)CCC(O)CC12CC2 C1(COC)(NC(C2(C#N)CC2)=O)CCN(C(=O)C(C)Sc2ccccn2)C1 C1(C(C)C)CC(C(=O)Nc2c(CO)cccc2Cl)NC(=O)N1 C(=O)(CS(=O)(=O)Nc1cc(C2CCCCC2)sc1C)NC1CC(C(=O)OCC)C1 C(=O)(C(F)(F)c1nccs1)NC1(CN(C)C(C2(C)CC2(F)F)=O)CC1 CC(C(F)C(=O)NCCN(C(=O)C(=O)Nc1ccc(Cl)c(F)c1)C)C(F)(F)F C1(N(C(C(CC)OC)=O)C)CCCN(C(=O)C(F)(F)c2ccccc2)C1 C1(CNC(CCOCC#C)=O)(OC)CN(C(c2ncsc2Br)=O)C1 N1(c2nc(N(CCOC)C)nc3c2n(C)cn3)CCc2c(Cl)cccc2C1 C1(C(=O)NC2CCCN(C(CCC(C)C)=O)CC2)CCc2cc(F)ccc2O1 N1(C(CNC(=O)Nc2cc(Cl)ns2)=O)CCC2CN(C(=O)CCF)CCC2C1 C1(NC(c2c(CC)cco2)=O)CC2CC1CC2C(=O)N(C)CC1CCN(C)C1 c1(C(N2CCN(C)CC2CNC(=O)CC2CCC2)=O)ccc2[nH]ccc2c1F C(=O)(CCCS(N)(=O)=O)NC1CCCN(C(CCSCC)=O)C1C C1(CNC(C(C)(C)OC)=O)CC2CC(C1)N(C(=O)Cc1cccnc1Cl)C2 CCCCCCCC(=O)NCC(F)(C(=O)NC1CC1(C)COC)C(C)C N1(CC(=O)NCCC2N(C(C3C(C)C3)=O)CCC2)CCCNS1(=O)=O C1(CN(C)C(c2ocnc2C(F)(F)F)=O)CN(C(=O)CC2CCCO2)CCO1 C1(NC(c2c(OC)cccc2C)=O)COC2(CCCN(C(=O)C3=NOCC3)C2)C1 N1(c2nnc(SC)s2)CC2C(C(=O)NCC(c3cnn(C)c3)=O)C2C1 CCCC(C(=O)OC)C(=O)N1CC=CC1(C)C(=O)NCC1=NOC(C)C1 c1(CNC(COCCC(C)C)=O)cc(O)nc(CNC(C2COC(C)(C)C2)=O)n1 CC1(C)C(C(=O)NC2C3CCCOC23)CCN1C(=O)C=Cc1cscn1 C(=O)(C(CO)C(C)(C)C)N1C2CC(CNC(c3c(C)c(Cl)ccn3)=O)(OC2)C1 c1(C(N(C)CC2(NC(=O)CCn3cnnn3)CC2)=O)ccn2cccc2c1 c1(C(N2C(CCCNC(c3cnn(CC)n3)=O)CCC2)=O)ccc(=O)n(CC)n1 C1(C(=O)NC2C(C(N(C)Cc3ncco3)=O)CC2)CCCC12CC2 C(=O)(C1=CC2(CCOC2)C1)N1CC(OC(C)C)C1.N12CC3CCC1C(C3)CC2=O Cc1ccc(C(=O)NC(C)CN(C)C(C2(CF)CC2)=O)c2ncccc12 C1(CC(N2CC3C(N(C)C(c4ccsn4)=O)C3C2)=O)COC2(CCC2)CO1 CC1=C(C)CC(C)(C(=O)N(CCCCCCNC(=O)CCN2CCCC2)C)CC1 c1(C(=O)NC2CC(F)(CNC(CC=C)=O)C2)cnc2n(c1=O)CCS2 c1(OC)cc(CCC(=O)NCc2cn(CCOC3CC3)nn2)cc(Br)c1OC C1(C(c2nn[nH]n2)=O)CN(C(C2CC23CC3)=O)CCO1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(CC#C)CC(=O)Nc1ccc(Cl)nc1 c1(C(=O)NCC2N(C(c3c(C)cco3)=O)CC2)nc2ncc(CCO)cn2n1 C=CCC(C(=O)NCCCN(C)C(c1cn(C(C)C)cn1)=O)N(C)C CS(=O)(=O)C(CNC(c1cc2sccc2[nH]1)=O)CNC(C12CC(F)C1C2)=O C1(C(=O)NCCC(=C)CNC(C2(CC3CC3)CC2)=O)Cc2ccccc2C1(C)C n1(CC(N2CCC(NC(Cc3nc(C)sc3Cl)=O)C2C)=O)nc(C)c(C)c1C N1(c2cc(OC(C)C)ncn2)CCC(NC(C2(F)CCOC2)=O)C2(CCC2)C1 CC1(CC(=O)NCC(c2ccccc2F)O)CCCN1C(=O)Cc1cnoc1 c1(CC(=O)N(C(C)CCNC(C2CCC(=O)NC2=O)=O)C)ccc2c(c1)CCC2 c1(C(=O)OCC)nsc(=NCCCNC(=O)COC2CCCOC2)[nH]1 C1(NC(c2cc(OC)n(C)n2)=O)CCC(C)(C)CC1CNC(c1csc(=N)[nH]1)=O CC(C)C(CNC(=O)C(C)C1CCOC1)NC(c1cn(CCN(C)C)nn1)=O Cc1nc(S)sc1CC(=O)N(C(C)CCNC(=O)C(C)OC1CCCC1)C C(=O)(C(CN(C)C)c1ccccc1)NCCN(C(CC=CC=C)=O)CCOC C1(c2c(OC)nc(Br)cc2)NC(=O)N(CCF)C2=C1C(=O)N(C)CC2 c1(NCC(c2ccc3c(c2)OCO3)C)ncnc2c1ccn2C S(=O)(=O)(c1ccc2c(c1)CC(C)(C)O2)N(C)CC1CCCCO1 c1(CNC(C2(OC)CCC2)=O)nc(CNC(C2C=CCC2)=O)cc(O)n1 Cc1cc(C(=O)NCCC2C(C)CCCN2C(=O)Cc2cnsc2)nc(O)n1 N1(CCN(C(=O)NC(C)Cc2ccccn2)CC)CCOCC12CCC2 CC#CCCCC(=O)N1CCC(CC(C)NC(C2CCC2OCC)=O)CC1 C(CCCCCC(=O)N1CCCC1CCC(=O)NCCC(C)N1CCCC1)SC O=C1NCN(Cc2ccc(F)cc2)CCN1c1ccc2cc(O)ccc2n1 O=C(CCCCCF)N1CCCC1CCCNC(=O)C1=COCC1 C(=O)(C(CCc1ccccc1)NC(=O)OC(C)(C)C)N(C(CC#C)C)C c1(N2CCN(C(=O)C=Cc3ccccc3)CC2)nc(Cl)c(Cl)cc1Cl C1(C(N2CCC(CNC(c3occc3CO)=O)C(C)C2)=O)(OC)CCCCCC1 c1(C(=O)NCC(CC(=O)N2CCC(OC(C)C)C2)C2CC2)cn2ccccc2n1 C1(CC(=O)Nc2ccc(F)nc2)CC2(C1)CN(C(=O)C=CC1CCOCC1)C2 N1(C(C2(CC)CCCC2)=O)CC2CCCC2(CNC(c2ccc(F)cc2F)=O)C1 N1(C(C(C)S(N)(=O)=O)=O)CC(NC(c2cc(CO)on2)=O)C(S(C)(=O)=O)C1 c1(C(N2C3CCN(C(C(c4n(C)ccc4)=O)=O)C3CC2)=O)c[nH]c2cc(Cl)ccc12 c1(CNC(C(C2CCN(C(C3(C#N)CC(=O)C3)=O)C2)F)=O)n[nH]c2c1CCC2 C1(CC)CN(C(=O)CC2CCC(O)C2)CCC1NC(=O)CCNC(N)=O c1(N2CCC(O)(C(N3CCn4ncnc4C3)=O)C2)ncc2cc(Br)ccc2n1 C1(NC(C2SC3C=CC2CC3)=O)CN(C(=O)CCc2nncs2)CCC1O N(C=CC(=O)C(F)(F)F)C(CC1N(Cc2c(C(C)C)n[nH]c2)CCOC1)=O C1(C(=O)NC(C)C(N)=O)CC12CCN(C(C1CC1c1cncn1C)=O)CC2 N1(C(C(C2CCC2)OC)=O)CC2CC(NC(C3CCCN3C)=O)C2C1 C1(C(=O)NC2COCCN(C(C(CC(C)C)O)=O)C2)CCC2CC1C2(C)C N1(C(CCN(C)C(c2cnc(Cl)s2)=O)=O)CC(C)(C)CC1CC(N)=O c1(C(N2CCCCC(N(C(C=CSC)=O)C)C2)=O)cn(C)c2ccccc12 c1(C(=O)NCC(CC=C)NC(=O)CCCC(F)(F)F)ncnc2cc[nH]c12 C1(C)(CC)CC(NC(=O)C=Cc2cnc[nH]2)CN1C(=O)CC1CCSCC1 c1(OCC#C)cccc(C(=O)NC2COCC2NC(=O)C(C(C)C)C2CCC2)c1 N1(C(C=CSC)=O)CC(CNC(C2(CO)CC(C)(C)C2)=O)C2(CCC2)C1 N1(C(C(CC)c2ccccc2)=O)CC2CN(C(c3ccc(O)cc3O)=O)CC12 C=C1CN2C(=O)CCC2(C(=O)NCCN(C(=O)C2CCOc3ccccc32)CC)C1 CC(C)CCC(O)C(=O)N1CCC(CN(C(=O)CC2(N(C)C)COC2)C)C1 Cc1c(F)ccc(-c2ccccc2CNC(Cc2cccc(Br)c2)C(=O)O)c1O N1(C(c2n(CC)ccc2)=O)CCCCC2(CCN(C(=O)C(C3CC3)C3CC3)C2)C1 C1(C)(CNC(C2N(C)CCC2)=O)CCN(C(=O)CC2CCCCCC2)C1 c1(C(N2CC(CCC)C(CO)C2)C(=O)NC2CCC2)cnc2c(F)cccc2c1 N1(C(C2C(C)(C(C)C)C2)=O)CCN(CC(C)NC(=O)CCc2nncn2C)CC1 C1(C(N2CC(F)(CNC(COC3(C)CCOCC3)=O)C2)=O)CCC2(CCC2)O1 CC(C)(CCNC(=O)COC1COC1)C(=O)NC12CC(C1)C2 c1(CCN)cc(C(=O)NCC2CC(F)(F)CO2)ccn1 c1(OCC=C)cccnc1C(N1CCCCC1CNC(=O)C(C(C)C)OC)=O CC=C=CCCN=c1nc(N2CCC(CN3CCOCC3)C2)c2c([nH]1)COC2 c1(C(=O)NC2(C)CC(CNC(CN(C(COC)=O)C)=O)C2)ccc(N)c(C)c1F N1(C(CC(CCC(=O)OC)C)=O)CCCC2(C1)CN(C(=O)CSC1CC1)CCO2 N1(C(C(F)OC)=O)CC(NC(=O)CCc2ncc[nH]2)C(CN(C)C)C1 CC1(CNC(=O)CC2CCCS2)CN(C(=O)Cn2cncn2)CCO1 C1(NC(C=CCOC)=O)C=CCC(C(N2CCN(CC3CC3)CC2)=O)C1 c1(C(=O)NCC(CC=C)NC(=O)CC2(C)CCCCC2)ccc2c(c1)C=CCC2 c1(C(=O)NC(CC(C)NC(CCNC(=O)OCC)=O)C)cc(C(C)(C)C)[nH]c1C C1(CCNC(C2CCSC2)=O)CCN(C(c2cc(-c3ccco3)[nH]n2)=O)CC1 C(c1cccnc1)=CC(=O)NCC(C)CNC(=O)C(C)(O)c1ccccn1 C1(C(=O)NCCCN(C(c2nc(C(=O)OC)oc2)=O)C)CC(C(C)C)=NO1 c1(C(=O)NCCN(CCC)C(c2nscc2C)=O)ccc2nsnc2c1 Cc1cc(C(=O)NCC(C2CCCCC2)NC(C2COC(C)C2)=O)c[nH]1 C(C(=O)NCc1ccc(C(N2CCC(OC(F)F)C2)=O)s1)(C(C)C)OCC c1(CC(=O)NC(CNC(C(C=CC)O)=O)C(C)C)ccc(Cl)cn1 c1(C(C#N)ON2CCN(C3CC3(F)F)CC2)ccccc1C(F)(F)F C(=O)(CC(=O)NCC1(CCCNC(=O)C(O)Cc2cnc[nH]2)CCCC1)NCC C(=O)(C(F)(F)C(F)(F)F)N1CC(CC(N2CCC(Oc3cccnc3)CC2)=O)C1 C1(C(N2CCC(N3CCC(N)CC3)C2)=O)CC2(CCOCC2)C1 N1(C(Cc2c(C)con2)=O)CCCCC1CNC(c1cn(C)nc1Cl)=O C(c1cnccc1C)=CC(=O)NCC1(CNC(CCC(C)SC)=O)CCCC1 CCC(CC)CC(F)C(=O)N(C1CCN(C(C2(F)CC=CC2)=O)CC1)C S(=O)(=O)(c1cnccc1N(C)Cc1cncnc1)NCC1(OC)CCSC1 c1(C(N2CCn3nccc3C2)=O)cc2cc(F)ccc2o1.C12CCCCN1NC2=O C1(CC(N2Cc3c(SC)cnn3CC2)=O)CCN(C(=O)OC(C)(C)C)CCC1(F)F C1(c2ccc(-c3cccs3)s2)CCC(F)(F)CC1.C#CC1(CNC(=O)N)CCC1 C1(NC(C2CCC(=C)CC2)=O)COCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1 c1(C(=O)NC(CN(C)C(C2CCC(O)C2)=O)(C)C)ccc(CNS(C)(=O)=O)cc1 C=CCC(C(=O)N1CC=C(C)CC1)NC(c1cccc(CC)n1)=O N1(C(c2c(CC)n(C)nn2)=O)CCOCC(NC(c2cn(C)c(C)n2)=O)C1 C1(C(N2CCC(C(C)(C)NC(c3c(C#C)c[nH]n3)=O)C2)=O)CC2CCC(C1)N2C Cc1cc(C)c(C(=O)NC(c2ccccc2)CNC(C2CCN2S(C)(=O)=O)=O)o1 C1(O)(CN(C(=O)C(c2ccccc2)O)C)CCN(C(=O)CN(C2CCCC2)C)C1 c1(CNC(C(n2cc(-c3ccc(F)cn3)nn2)C)=O)ccc(O)cc1F CC1(C)CN(Cc2ccc(O)c(F)c2)CCC1NC(c1ccncc1F)=O CC(C)(CO)CCNC(=O)C(CCC1CC1)NC(c1ccsc1)=O Cn1cc(C(=O)NC2CN(Cc3cnnn3C)CC2O)c(C(F)(F)F)n1 C(=O)(C1=CC(C)(C)C1)NCCC(CNC(c1ncc(OC)nc1)=O)O C1(CCC(=O)NC2(C3N(C(CCC4C(C)(C)C4)=O)CCC3)CC2)CCCCCC1 c1(CNC(C2CC(C)CN2Cc2ccc(O)cc2)=O)ccc2c(c1)OCO2 C1(O)(CC(=O)NCC2N(C(CCNC(C)=O)=O)CCC2C)CCCN(C)C1 CC1CN(C(=O)CC2(n3cccn3)CC2)C(C)CN1C(=O)CC(C)C(F)(F)F N1(C(C2CC(CC)C2)=O)CCC(CNC(C2CCCN2C2CCCC2)=O)C1 N1(C(C(=O)Nc2c(C)nc(-c3ccc(Cl)cc3)s2)=O)CCC(O)(CO)C(O)C1 N#CC1(C(N2CCN(C(=O)Cc3nnc(O)s3)CC2)=O)CC2CC2C1 c1(SC)cc(C(=O)Nc2c(Cl)cc(C)cc2Cl)cc(SC)c1 Cc1ccc(C(N2CC(N(C)C)C(CNC(=O)CC3CC(C)(C)CO3)C2)=O)cc1 c1(CNC(C(n2cc(CCCC(C)O)nn2)C)=O)ccc2[nH]nc(Cl)c2c1 N1(C(CCCOCCC)=O)CCC(C)(C(=O)NCc2coc(C)c2)C1 C=CCCC(=O)NC(C1CCN(C(c2cnn(CC3CCCC3)c2)=O)C1)C CCCCS(=O)(=O)CC(=O)NCC(O)CNC(c1cnc2[nH]nnc2c1)=O CC1(C(N2CC(NC(c3coc(C(F)(F)F)c3)=O)C3(CC3)C2)=O)CCNC(=O)C1 c1(C(N2CCC(NC(C(C(=O)OCC)F)=O)CC2C)=O)c[nH]c2cccc(C)c12 C1(CC(=O)NCC(CCCC)O)CN(C(=O)CC=C(C)C)CC12CC2 N1(C(C=CC(CC)=CC)=O)CC(NC(c2c[nH]nc2CC)=O)CC12CCOC2 C1(NC(C2N(CC)CCCC2)=O)CCC2CN(C(c3c[nH]nc3F)=O)CCC2C1 Cc1cccc2sc(NC(N3CCOC(CCO)C3)=O)nc12 c1(C(=O)NCC(CC)(C)NC(C2(CCF)CCOCC2)=O)cc(C)oc1C C(=O)(C(C)(C)CCCF)N1CCC(CC=C)(NC(C2C3CCCCCC23)=O)C1 N1(C(C(F)=CCC)=O)CC(NC(c2cc(C(N)=O)cs2)=O)CCC1C C1(C(=O)NCCC(=O)OC(C)C)CCN(C(=O)C(C2CC2)C2CC2)CCO1 c1(OC)ccc(C(C)=CC(=O)NCCN(C2CCCC2)C(=O)COC)cc1 C1(NC(CCC(C)SC)=O)COCCN(C(=O)CSc2ccc(O)cc2)C1 c1(N(C)C)cccc(CNCC(N2CCC(C(CO)NC(C(C)(C)C)=O)CC2)=O)c1 c1(C(=O)NC23CCN(C(C=C4CCC(C)C4)=O)CC2C3)ccc2nc(S)oc2c1 C1(C)(C(=O)NCC(Cn2cc(-c3ccnn3C(C)C)nn2)OC)CCCC1O c1(C(=O)NC2C(NC(=O)C=CC=C(Cl)Cl)CCOC2)cc2ccncc2c(O)n1 C(CNC(c1cc(C2(C)COC2)no1)=O)(C(C)C)NC(C(C)OCCC#C)=O C(=O)(C(C(C)C1CCCC1)N(C1CCOC1)CCN1CCCC1)NCC Cc1ccnc(O)c1C(=O)NC.C12CC(C1)C(=O)NC(=O)CNC2=O.CCC1CC1 Cn1ccc2ccnc(C(=O)NCCCCCNC(=O)C#CC3(C)COC3)c12 N1(C(c2n(C)cnc2Br)=O)CC2CC1CN2C(=O)CN1CC(=O)NC1=O O=S(=O)(c1ncccc1Cl)NCc1cc2c(F)cccc2s1 C(=O)(CC(O)CNC(c1nccn1CC)=O)NCCN(C(CC)C)C CC(C)C(O)CC(=O)N1CC2(CCN2C(c2ccoc2C(F)(F)F)=O)C1 c1(CC)ncccc1C(=O)NC1CCCN(C(=O)CC2C=CCCC2)C1 c1(OCC(N2CCCC(CCNC(C(CCC)O)=O)C2)=O)ccc(Cl)cc1Cl c1(NC)cnccc1C(=O)NC1CC(CNC(=O)CCCc2ccsc2)C1 N1(CC(=O)NCCC2(O)CCCN(C(CC(C)C)=O)C2)CCCCCCC1=O CC(C)C(F)C(=O)N1CCCC1(C)CNC(=O)C=Cc1ccoc1 CC1CCC(C(=O)NCCOCCOCCNC(c2nocc2Cl)=O)C1 C1(C(=O)NCC(C)N(C(c2nc(C)sc2)=O)C)Cc2nn(C)cc2C(=O)N1 CC1CN(C(c2cc(CO)on2)=O)C1C(=O)NCC(N)=O CC1CCN(C(C2(Cc3ccc(O)cc3)CC2)=O)CCN1C(C1CC1F)=O CN1C(=O)NC2(CCC(NC(c3cncn3C)=O)CC2)C1=O C1(OC(C)=O)CC(c2nc(C)no2)N(C(=O)NC2(C3CCCO3)CCC2)C1 Cc1c(C(=O)NCC2CCCCN(C)C2)cccc1-n1cnnc1 C1(C)(CNC(CC(=C)C)=O)CCN(C(C2(NC(C)=O)CCCC2)=O)C1 C=CCC(C)(CNC(C1CC(N(C(=O)C(CO)OC)C)C1)=O)CO N1(C(C2CC(SC)C2)=O)CC(NC(=O)C(n2ccnc2C)C)C(F)C1 N1(C(C(=O)Nc2c(OCC)cccc2)CC2(C)CC2)CC2CC3CC(C2)CC1C3 CCC(C)(O)C(=O)N(CC(C)NC(=O)CC(C)NC(=O)OC(C)(C)C)C N1(C(C)=O)CCC(C(N2CC(C(C)Nc3ccc(N)cc3)OCC2)=O)CC1 N1(C(c2cncc(SC)c2)=O)CCCC(C)(CNC(C2CCC(=O)NC2)=O)C1 c1(C(=O)NCC2C(NC(Cc3n(C)cnc3)=O)CC2)cccc2c[nH]nc12 N1(C(=O)CNc2ccc(Cl)c(Br)c2)CC2(CC=CC2)C1c1ccccc1 C1(C(N(CCC)C)=O)CN(C(C2COCOC2)=O)CC1C1CC1 c1(OC)ccc(CCC(N2CCC(NC(c3ncccc3OC)=O)C2C)=O)cn1 C(=O)(C1CCCc2nc[nH]c21)NCC1N(C(Cc2cn(CC)nn2)=O)CC(O)C1 N1(C(c2c(OC)cncc2)=O)CCC(C)(C)C1C(N1CCC2CCCC12)=O C1(C(C)NC(C(SC)SC)=O)CCCN(C(C2(CF)CCOCC2)=O)C1 c1(C(=O)NCC(C)NC(C2CC(SC)C2)=O)cccc(Br)c1 C1(NC(C(C)S(C)(=O)=O)=O)C(C)(C)CN(C(c2cccc(CO)c2)=O)CC1(C)C CC1CN(C(c2[nH]nnc2-c2ccnn2C)=O)CCC1NC(c1cc(Cl)ns1)=O CCC(C)CC(C)C(=O)N1CC(F)(CNC(C2(CC3CCC3)CC2)=O)C1 c1(OC)cccc(S(=O)(=O)NC(c2ccc(Cl)cc2)CN(C)C)n1 CC(=O)CCCC(C)(C)C(=O)N1CCCN(c2nc(C)cs2)CC1 C(C1c2ccsc2CCN1C(C1CC(C#N)C1)=O)NC(C(C)c1ccco1)=O C(=O)(C1=NOC(C)(C)C1)NC1C=CC(C(=O)Nc2cc(C)c(C)nc2)C1 c1(C(=O)NCC2OCC(CNC(C(C3CC3)OCC)=O)C2)nnc2n1CCOC2 C12(C(=O)NCCCC(=O)NC)CC(CN(C(=O)CCC(C)CN(C)C)C1)C2 C(=O)(C(CNC(C1CCC(=O)N1C)=O)C(C)C)NC1CN(CCC)C1 N1(C(C(CCC)OCC)=O)Cc2[nH]nc(C(N3CC(S(C)(=O)=O)C3)=O)c2C1 Cc1cc(C(=O)C(=O)NCC2CN(C(C3CC(F)(CO)C3)=O)CC2C)ccc1F c1(C(N(C)C)=O)c(NC(=O)NCCC(C)(C)CO)cccc1F c1(C(=O)NCCN(C(C2(C)CCC2)=O)CC)cnc(N)c(Cl)c1 N1(C(C(C)N(C)C)=O)CCC2(CCCC2NC(C2CCC(C3CC3)CC2)=O)CC1 n1(CCC)nc(C)c(C(N2CCC(O)(CNC(=O)C(O)C(C)(C)C)C2)=O)c1C C1(C(=O)NCCOCC(C)C)CCC(C)(C)N(C(=O)C2=C(C)CC2)C1 CC1(C)COCC(CC(=O)NCC2CCCN2C(C2(O)COC2)=O)O1 N#CC1(C(N2CC3CC3(NC(=O)C=Cc3cccs3)C2)=O)CCOCC1 CC1CN(C(c2ccccc2CC(C)(C)C)=O)CC1NC(=O)CSC1CC1 n1(CCCC)nc(-c2cccc(C(F)(F)F)c2)nc1CCC1CCC1 c1(CNC(c2c(CCNC(c3n(CC)nnc3)=O)n[nH]c2)=O)cc(O)ccc1F N1(c2n(CCOC)c(C(C)[N+](=O)[O-])nn2)CC(=O)N2CCCC2C1 C(CCCCC(=O)N(C1CCCC1)CCNC(C1CC(O)CN1C(C)=O)=O)=CC CCC(C(=O)NCCC1CCCN1C(=O)C(c1cccnc1)C)NC(N)=O c1(C(=O)NC2(C(C)NC(CCCOC)=O)CCCCC2)cc(C)n(C)c1C N1(C(CNC(CC)=O)=O)CCCC(C)(C)C1CNC(c1cscc1OC)=O C1(NC(c2cc(C)n(C(C)C)n2)=O)C2CC(O)C1N(C(C1C(C)(C)C1(C)C)=O)C2 N1(C(c2c(OC)n[nH]c2)=O)CC(C)C(C)(CNC(C2(C)SCCCS2)=O)C1 C1(NC(C=CCOC)=O)CCn2ccnc2C1.c1(CC2C(=O)N2)cnn(C)c1O C(c1ccco1)=CC(=O)NCC1C=CCN1C(=O)COCC(F)F C(=O)(CCCS(C)(=O)=O)N(CCOCCN(C(=O)C(=O)NCC(F)F)C)C c1(N2CC(CC=C)(NC(C(N3CCCC(C)C3)=O)=O)C2)ncc2c(n1)CCCC2 C1(C(C(=O)N(CCCNC(C(C)OC)=O)C2CC2)OCCOC)CCCCC1 C1(NC(c2c(C)nsc2)=O)CC2CC(C1)N(C(c1ccc(C#N)s1)=O)C2 C=CC1(CC(=O)NC(C)COCCOC)CN(C(=O)Cc2cc(C)no2)C1 c1(CN(C)C)ccc(C(=O)NCCOCCN(C(=O)CCc2ncnn2C)C)s1 c1(C(C(=O)NCCC#N)N(CC(F)Cl)C)cc(-c2ccccc2)on1 CCC(CC)CCCC(=O)NC1(C(=O)NOCC(=O)OCC)CCSC1 C1(NC(C2(CC(C)=O)CC2)=O)CC(C)(CNC(=O)Cc2cnc(C)s2)C1 C1(C(=O)NCCCNC(=O)NCCCl)COC2(C1)CN(C(c1scnc1Cl)=O)C2 c1(C(N(CCN(C(c2c(CC)nn[nH]2)=O)C)C)=O)ccc(C2CCC2)nc1 C(c1ccco1)=C(C)C(=O)NCCC1CCCN1C(C1CC(CC(F)(F)F)C1)=O C1(CCNC(C(C)O)=O)CCN(C(c2cnccc2C2OCCO2)=O)CC1(F)F c1(C(C)=O)ccc2cccc(C(C)C)c2c1.c12ccc(cc1)OCC(=O)OC2C Cc1[nH]nc(C(N2CC3CC2C3C(=O)N(CC(C)(CO)N(C)C)C)=O)c1O N1(C(COC)=O)C(C)CC2CN(C(c3c(C)sc4ccccc34)=O)CC12 c1(C(=O)NC2CCC2CNC(=O)C(F)n2cccn2)cnc[nH]1 c1(CCC(=O)NC2C(NC(CN(C)C)=O)CCCC2)ccc2c(c1)OCO2 N1(C(Cc2c(C#C)cccc2)=O)C2CCC1CN(C(c1cc(C)[nH]c1C)=O)CC2 c1(N2CCN(CC(c3ccccn3)C)CC2)nc(Cl)nc2ccn(C)c12 C1(C(=O)NCCCNC(=O)C(F)(F)CCn2cccn2)CCC2C(C1)C2(F)F c1(OC)ccc(F)c(C(=O)NCC2CCCCCN2C(C2(OC)CCC2)=O)n1 C(=O)(C(C)(C)CCCNC(=O)C=CC1(C)COC1)NCC1ON=C(C)C1 C1(N(C(=O)CC2(C(F)F)CC2)CC)CCN(C(=O)CN(C2CC2)CC)C1 C#Cc1ccc(CC(N)C(=O)NC2CC(NC(N)=O)C2)cc1 C1(NC(C2CC(F)(F)C2)=O)COC2CN(C(c3c(F)cccc3F)=O)CC12 CCCCCC(O)CC(=O)N1CC(CC(F)C(N2CCNC(=O)C2)=O)C1 C(=O)(CS(=O)(=O)CC1CCCO1)N1CCC(Cn2cc(CN(C)C)nn2)C1 c1(-c2ccc(CCN(C)C)o2)nc(CCO)nn1Cc1cnn(C)c1 C1(CN(C)C(c2nc(=O)n(C)[nH]2)=O)CCN(C(C2CC3CCC2C3)=O)CC1 C(CCNC(c1ccc[nH]1)=O)(C(=O)NCCn1cnnc1)OC c1(C(C)(C)C)cc2n(n1)CCN(C(C1CCN(CC3CCCC3)C1)=O)C2 c1(OC)c(C)csc1C(=O)NCC1CCC(NC(=O)CCn2c(C)ccc2C)C1 C1(C(N2CC(CCCCNC(=O)CN3CCCCCC3)C2)=O)CC(=C(F)F)C1 C(=O)(CCCC(C)O)Nc1cccc(NC(C(C)NC(=O)NC)=O)c1 c1(C(N(CC(=O)NC(c2ncc(C)[nH]2)CC)CCC)=O)cn(C)nn1 O=C(CCC(F)(F)F)NC1CC2CC1CN2C(=O)C(c1ccccc1)C1CC1 N1(C(C=CC)=O)CC(C(=O)NCC2OCCC2(C)C)CC12CCC2 c1(OC)ccc2c(c1)CCC(C(=O)OC1CCC1)C2.c12cccn1c2=O C1(CNC(c2cn(C)c(=O)cc2)=O)COC(C)(C)CN1C(C1CC2CCC1O2)=O C1(C(=O)NCC2C3CN(C(=O)Cn4cnc(C(F)F)c4)C2C3)CCc2nccn2C1 C=CC(CC)CC(=O)NCC1CC1CC(=O)NCC1CCCCS1 N1(C(CCN(C)C)=O)CCCCC1C(=O)Nc1ncc(-c2ccccn2)cn1 c1(COC(CCCNC(=O)NC2CCOC2)=O)cc(F)cc([N+](=O)[O-])c1 C(=O)(CCC(C)(C)NC(c1csc(Cl)n1)=O)NC1C2CN(C)CC21 c1(C(N2C(CNC(c3c(C#N)cccc3)=O)CCC2)=O)ccc2ocnc2c1 C=C(C)CC(C(=O)N1CCC(n2cc(-c3ccccc3OC)nn2)CC1)OC c1(C(=O)NC2C3CN(C(CN4C(=O)CN(C)C4=O)=O)CC32)cc(O)cc(N)c1Cl c1(CC(=O)NC(C(C)NC(C2CCS(=O)(=O)C2)=O)CO)ccc2c(c1)CCOC2 C1(F)(C(=O)NCCC(O)CO)CCN(Cc2scnc2Cl)CC1 C(C(=O)NCc1cnn(C)c1C(=O)NCC(C)(COC)CC)(C(C)C)OCC c1(OC)ncc(Br)cc1S(=O)(=O)NC(C)CCN(C)C C(=O)(C1CCCc2scnc21)NCC1(C)CC(NC(c2cn3ccsc3n2)=O)C1 C12(CNC(=O)C=CCF)CCCC1N(C(C1CC1c1ccoc1)=O)CCC2 N1(C(C(C)C2CC2)=O)CCCC2(C1)CN(C(C1(CO)COC1)=O)CCO2 c1(-n2cc(C(C(C)C)NC(c3nc(Cl)c(Cl)s3)=O)nn2)ccccc1OCCF N1(C(c2oc(C)c(CO)c2)=O)CCC(C2CC2)C1C(=O)NC1CC(C)(O)C1 N1(C(C2CC3(CCC3O)C2)=O)CCC2(CC1)CN(C(C1CCCO1)=O)C2 c1(C(=O)NC2C(O)CCN(C(c3c(C)ccc(N)c3)=O)C2)n[nH]c2c1CCSC2 C1(C(=O)NCCC2CCN(C(c3nc(C)n(C)c3C)=O)C2)CN(CP(C)(C)=O)C1 N1(C(CC(C)SC)=O)CC23CCCC2(C1)CN(C(C1CCC2(CCOC2)O1)=O)C3 c1(C(N2CCC(OC)(CNC(=O)CC3CCCCO3)C2)=O)ccc(C)c(C)c1Cl CCCC(CCC)CC(=O)N1CC(CC(F)C(N2CCC(O)(CC)CC2)=O)C1 C(C(C)(C)C(=O)NCCc1cc(C(=O)N(C)Cc2cscn2)no1)SC c1(OC)cccc(OCC(=O)NCCN(C)C(C2CCCC(C)O2)=O)c1 O=C(CC1=CCCC1)NCC(CNC(C12CCC(CO)(CC1)C2)=O)CO N1(C(CCOC)=O)CCC(CNC(=O)Cc2sccc2C)(OC)C1 C(=O)(CCCC(=O)c1ccccc1)N(C)CC1CCN(C(=O)Cn2ccnn2)C1 C1(NC(c2c(=O)cc(C)[nH]c2)=O)CCCC2CN(C(c3cn[nH]c3)=O)CC12 N1(C(C2(C)CCOCC2)=O)CCCCC(CCC(=O)NCC2(F)CC(CO)C2)C1 CCCC(C)(C)CC(=O)NC1COC2C(NC(=O)C(F)(F)CC)COC12 C(=O)(CCC1=NNC(=O)CC1)N(C)CC1CCC(CNC(C2C(CC)C2)=O)CC1 c1(C(N2CC(CC(CNC(C(C)C3CC3)=O)(C)C)C2)=O)ccncc1Br C1(C(=O)OC)CN(C)CC1NC(=O)C(N)C1(C)CC1 Cc1cccc2cc(C(N3CCCN(C(c4cc(Cl)cn4C)=O)CC3C)=O)nn12 Cc1nc(C(=O)NC2CC(C)N(C(=O)CCc3cnc[nH]3)C2)c2ccccn12 C(=O)(C(C)C(C)(C)C)NCC(CCNC(C(C)(C)OC(C)=O)=O)O c1(NC(C2N(C(COC)=O)CC(O)C2)=O)c(F)ccc(Br)c1F c1(C(N2C(C)(CCC(=O)NCC(F)C3CCC3)CCC2)=O)c[nH]c2ncccc12 C(C(C)(C)C#CC(=O)NC1CCC12CCCC2)NC(CC1(CC)CCC1)=O N1(C(c2ccc(OCC)c(C)c2)=O)CC2(CCCC2NC(=O)CN(C)C(N)=O)C1 c1(CC)ccc(F)cc1.c1(CN(CC(O)COCC)CCN2CCC2)ncc[nH]1 C1(NC(C2CCN(C3CC3)CC2)=O)CC2(C1)CN(C(=O)CC1(O)CCOC1)C2 N1(C(C2CCC(CC)O2)=O)CCC(CC(C)(C)N)CC1 c1(CNCC2CCCCN2C(C2C(C(N)=O)C2)=O)ccc(Cl)cc1Br C1(C)(C(=O)NCCC(C)NC(=O)CCNC(=O)C=CCl)CCNC(=O)C1 C1(CNC(C(C2CCC2)NC(c2c(C)cco2)=O)=O)(CO)CC2CC2C1 C1(NC(CCC=C)=O)CN(C(c2cc(C)c(C)nn2)=O)C(CC)(CC)C1 C(=O)(C(CCC1CC1)NC(=O)Cc1cn(C)cn1)NCCC1CC(C(=O)OC)C1 CC(C)C(C)C(=O)N(CC(C)(C)CNC(=O)C(C(=O)OC(C)(C)C)C1CC1)C C1(NC(c2n(C)c(O)nc2)=O)C2CC(O)C1N(C(c1ccc(O)nc1Cl)=O)C2 CC1=NOC(C)(CNC(=O)C#CCNC(C2CCCN2C(C)C)=O)C1 N1(C(c2[nH]cc(C#N)c2)=O)CCC2CCC12CNC(=O)CCN1CCCC1=O N1(CC)CCCC(C(=O)NCC(C)NC(=O)C(c2ccc(F)cc2)OC)C1 N1(C(Cc2nc(C)sc2Cl)=O)CCC(CNC(=O)C(=O)N(C)C)C(C)C1 Cc1cccc(F)c1C(=O)NCC1CC(NC(C2OCCN(C)C2=O)=O)CCO1 CC(C(C)(O)C(=O)NC1CC(NC(c2cc(O)cc(Cl)c2)=O)C1)c1ccccc1 CCC(C)(CC(=O)NCCC(O)CNC(=O)CCNC(=O)C(C)(C)C)C(=O)OC O=S(=O)(c1ccncc1Br)NC1CC2(CCC2)C1 c1(OC)ccc(C(=O)NC2CCN(Cc3nc(C)cs3)C2)cc1 N1(C(c2scc(OC)c2OC)=O)CCN(C(c2cc(OC)nc(C)c2)=O)CC1CF C1(C)(C(=O)NCC(CC)C)CN(C(C2(OC)CCOC2)=O)C1 C(CC1CC1)(C(=O)N1CC(O)(C(C)NC(=O)CCCn2ccnn2)C1)OC C(CC(C)C)(C(=O)N1CC(C)(O)CO1)NC(C(CC(C)=O)(C)C)=O N1(C(c2cn(C(C)C)nc2)=O)CCC(NC(C2CCCC3(CC3)C2)=O)C1(C)C C1(C(=O)NC2CCCN(CCO)C2)(COC)C=CCN1C(=O)CC(C)=C(C)C C12(NC(CCOCCOC)=O)CCN(C(=O)C[SH]=Cc3ccccc3)CCC1C2 N1(C(C(c2ccccc2)NC(CCOCC)=O)=O)CCC(=C(F)F)CC1 CCCC(C)CC(=O)N1CC(C(=O)N(CCC(=O)NC)C)C(C)(C)C1 c1(C(=O)NCC2(NC(c3c(C)ocn3)=O)CCOCC2)n[nH]c2c1CCCCC2 CCC(C(=O)NCC(C)NC(=O)C(C)(O)c1ccccn1)OC c1(C(=O)OCC)ccc(C(=O)NCCc2ccc(Br)cc2)cc1[N+](=O)[O-] C1(NC(COCC)=O)C=CC(CC(=O)NCCn2cnnn2)C1 C12(C(N(C)C)=O)CCN(Cc3cccc(C(=O)OCC(=O)NC(C)(C)C)c3)CC1C2 C1(C2(O)CCOC2)(C(=O)NCC2CCN(C(c3c(C)[nH]nc3CO)=O)CC2)CC1 c1(N2C3CN(C(c4ccc5c(c4)CC5)=O)CC2CC3)ncc2c(Br)cccc2n1 c1(C(=O)NC2CCC(NC(CNS(N)(=O)=O)=O)C2)coc2c1CS(=O)(=O)C2 CCC1C(=O)Nc2ccc(C(=O)NCC(C3CC3)NC(=O)C3=CCCS3)cc21 N1(C(CCCCC)=O)C2CCC1C1CC1(NC(C1CCc3nncn3CC1)=O)C2 c1(C(N(C2CCN(C(C3(C(F)F)CCCC3)=O)C2)CC)=O)ccc(C2CC2)cc1 c1(C(=O)NC2C(NC(C(CCC)=CCC)=O)CCCCC2)cc2cccnc2s1 CCC(C)C(=O)C(=O)N1CCC2C(NC(C3(CC)CC(O)C3)=O)C2C1 C(C(CNC(C1(C)CCC1)=O)C(F)(F)F)NC(CCc1onc(CSC)n1)=O N1(C(C(C)(C2CCC2)OC)=O)CC2CCCCC2(CN=c2nn[nH]n2C)C1 c1(C2C(C(=O)NCCCNC(c3cc(F)n[nH]3)=O)C2)cc(F)ccc1F C(COC)(CCCC)(c1n(CCOC)nnn1)NCCOC1CCCCC1 c1(C(=O)NC(CN(C(=O)C(C)C#N)CC)C)nn(C)c(-c2ccccc2)c1Cl N=c1ncn(CC(N2CC(F)(C(=O)NCC3CC34CC4)C2)=O)[nH]1 C1(C)(C(=O)NC(C(C)C)CNC(C2(NC(N)=O)CC2)=O)CCC(F)(F)CC1 N1(C(c2cc(OCC)no2)=O)CCN(C(=O)C(C2CC2)SC(C)(C)C)C(C)C1 N1(C(C=CC(C)(C)SC)=O)CC(C)CN(C(=O)Cc2csc(N)n2)CC1C C1(CC(C)NC(C2CCCCS2)=O)CCN(C(=O)Cc2cncn2C)CC1 C(C1CCC(C)CC1)=C(C)C(N1CC(N(C(=O)COCCN(C)C)C)C(F)C1)=O C(CN=C(NC1CC1)N1CCC(Oc2ccccn2)C1)NC1(OC(C)C)CCOC1 N1(C(c2ccc(C(C)(C)C)cc2)C(=O)NC(C)C)CCCC(C)(O)C1 c1(CC(=O)NCC2(CO)CCN(C(C3(CCN=[N+]=[N-])CC3)=O)C2)ccncc1C(F)F Cc1cc(F)cc(C)c1C(=O)NC1CC(CNC(=O)CC2(N(C)C)CCC2)C1 N1(C(c2ccc(CC)cn2)=O)CCC(CNC(c2cc(C)sc2C)=O)C1(C)C N1(C(C2(C#C)CCN(C(=O)CCC(C)C)C2)=O)CC2CN(C)CC2C1 O=C(C1=CC2C=CC1C2)NC1CCN(C(=O)COCc2ccnc(O)c2)CC1O N1(C(C=CSC)=O)CCC2(CC1)OCCCC2NC(=O)CC1OCCC1C C(CN=c1[nH]cnc2cc(C)ccc12)(C1CC1)NC(CC(CCC)O)=O C1(O)(CNC(=O)C=Cc2cocn2)CCCN(C(C2(C)CCCS2)=O)C1 N12Cc3n[nH]cc3C1C(=O)NCCC2=O.c1(OCCSC)cccc(O)c1 N1(C(CC(C(C)C)NC(c2c(CCC)[nH]cc2)=O)=O)Cc2cncnc2C1 Cn1cc(-c2nc(C(=O)NC3CN(C(=O)CCSc4ccccc4)C3)co2)cn1 C1(CNCC2N(C(CCCNC(c3ccccc3)=O)=O)CC=C2)(CO)CC(F)(F)C1 c1(CN(C(C(CCC)O)=O)C)cnn2c1CN(C(C1CCCS1(=O)=O)=O)CC2 Cc1c(C(N2CCCC2CN(C(=O)C=C2CCCC2)C)=O)[nH]c2c(C)cccc12 CC1=C(C(=O)N2CC(NC(C3CC(C)CCO3)=O)C(F)C2)C(=O)OC1(C)C C1(NC(C(c2ccccc2)OC(C)C)=O)CCCC1NC(=O)Cc1cocn1 C1(C(C)C(=O)N(C)CC2CCCN2C(=O)C=CC(=O)NC2CC2)CCCCCC1 Cc1nc(C2CC2)nc(O)c1C(=O)NCCOCCNC(C1CC(C)(F)C1)=O c1(N2C3CC(NC(c4scc(OC)c4)=O)CC2CC3)nc(Cl)nc2[nH]ccc12 c1(C(=O)NC2CCC(NC(C3(CCC)CC3)=O)C2)nnn(-c2ccccc2)c1C c1(C(=O)NC2(CO)CCN(C(CC(CCSC)O)=O)C2)cccc2c1CCC2=O CC1COCCN1C(C1CCC(CN(C)C)CC1)C(=O)NC(c1ccccc1)C c1(CC)nnsc1C(=O)NCC(C(=O)NC(Cc1ccco1)CO)N(C)C C(=O)(N=c1cc[nH]cc1O)C(c1ccnc(-c2ccc(OC(F)F)cc2)c1)=O N1(C(c2cc(F)c[nH]2)=O)CCC(C2CCN(C(c3ccc(F)cc3Br)=O)C2)C1 c1(SC)ncc(C)c(N2CCC(NC(c3c(OC)cccc3C(F)(F)F)=O)C2)n1 C1(CNC(c2c(C)ccnc2)=O)C2CCC1CN(C(c1cc(Cl)ccc1C)=O)C2 c1(C(=O)NC2CC(NC(COC3CCC(C)CC3)=O)C2)cc([N+](=O)[O-])ccc1N c1(N2C(C)(C)C(CNC(=O)C(F)CC3CCCC3)CC2)nc2cccnc2s1 C(=O)(C(C)(CC)C(N)=O)NC1C(C(C)NC(=O)C=C(C2CC2)C2CC2)CCCC1 c1(-c2c(C)nn(C)c2C)ccc2c(c1NC(=O)CCCCCBr)OCO2 C1(C(=O)NC2CC(O)(CNC(C3(C=C)CCC3)=O)C2)CC2CC1CC2O c1(N(C)CC2CCCN(C(CC3CC(OC)C3)=O)C2)ncc2scc(Br)c2n1 c1(CC(=O)NC(CC=C)CNC(c2ccn(C3CCC3)n2)=O)ccc(F)cc1Cl c1(C(=O)NC(CNC(C(C=C)(C)CC)=O)(CC)CC)ccc2snnc2c1 N1(C(C(C(C)C)SC)=O)CCCC(C)(C)C1CNC(=O)Cn1cnccc1=O CCC(C(=O)N1CC(C)(NC(c2cccc(N3CC=CC3)c2)=O)C1)C(C)O c1(C(=O)NCC2N(C(C)=O)CC2)ccccc1S(N)(=O)=O N1(C(c2cccc(C)c2)=O)CC(NC(=O)CC2CCC(=O)O2)CC(C)C1 C1(NC(COCC(=O)NC)=O)CN(C(=O)C(C)OCC(F)(F)F)C(CC)(CC)C1 CC1CN(C(C2CCC(NC(c3ccc(Br)cc3I)=O)CO2)=O)CC(C)O1 N1(C(c2nc(CC)sc2)=O)CCOC(CCNC(=O)C(C2CCOCC2)O)C1 CCCCC(O)C(C)C(=O)NOCC(N1CC2CCC(O)C2C1)=O Cc1ncc(C(=O)NCC2(O)CN(C(=O)CCc3nc[nH]n3)C2)cc1C#N CON1CCC(C(N2CC=CC(NC(C3CC4(CC4)CO3)=O)C2)=O)CC1 N1(C(c2n(CC#C)ccn2)C(=O)NC(C)(C)CC)CCCN(C)CCC1 c1(OC(=O)Nc2n(CC)nc(C)c2)ccc(OC(C)(C)C)cc1I c1(C(N2CC3(CN(C(C4C(C(=O)OC)C4)=O)C3)C2)=O)cnc([N+](=O)[O-])n1C N1(C(C2C3(CC(NC(C4(COCC)CCC4)=O)C3)C2)=O)CCC2CCN(C)CC12 c1(CC(=O)NCCN2CCN(C(C(C(C)C)OC)=O)CC2)ccc([N+](=O)[O-])cc1 c1(COC)cnc(OC)c(C(=O)NCC#CCNC(C2CCC(N(C)C)C2)=O)c1 c1(NC(=O)C(=O)Nc2ccc(F)c(Cl)c2)cc(Br)cc(C(N2CCCC2)=O)c1Cl C(=O)(C1=C2CCCN=C2NN1)NCCCN(C)C(C12CCC1C2)=O C1(C(=O)NC2C(C)CCN(C(=O)CSC(C)(C)C)C2)CCOCC12CCC2 CC1CCCCC1(C)n1cc(CN(C(=O)C(C)Cc2ccc(F)cc2)C)nn1 N1(C(C=CC(C)C2(C(N(C)C)N(C)C)CC2)=O)CC(F)(F)CC1(C)C1CC1 CCC(C)C(C(=O)N1CC=CC1Cn1cc(CN2CCOCC2)nn1)NC(C)=O C1(OC)CCN(c2ncccn2)CC1.c12cn(nn1)CCC(=O)N(C1CC1)CC2 c1(SC)cncc(C(=O)NCC2CC(NC(=O)C(C)C)C2)c1 CCCC(CCC)C(CC)NC(c1nnnn1C1CCCCC1)c1cnoc1 c1(NC(C(C2CC2Cl)N(CCC)C)=O)cc([N+](=O)[O-])ccc1C CCC(C(=O)NCC(CNC(=O)C(C)(C)CF)OC)C(C)C c1(C(C(=O)NCC(C)CNC(=O)CCOC2CCCCC2)(C)C)cccc(F)c1 C1(C(=O)NC(CCC2CCC2)C(=O)NCC(F)(F)Cl)CC2CCC(C1)O2 N1(C(C2C(C)(CC)C2)=O)CCC(CCN(c2nnnn2C)C)CC1 C1(C(=O)NCC(C)NC(c2csc(Cl)n2)=O)CC(=O)CC(=O)N1 c1(C(=O)OC)cc(CCC(=O)NC(C2C(Oc3ncc(C(=O)NC)s3)C2)=O)c[nH]1 c1(C(N2CC(C)CCC2CO)C(=O)NCCCSC)ccc2c(ccn2C)c1 C1(C(N(CC(CNC(c2ccc(SC)s2)=O)O)C)=O)CN2CCN1C(C)C2 c1(OC)ccc2c(c1NC(c1cnn(C3CCCCC3)c1)=O)CN(C(C)=O)CC2 C(CC(CC)CO)NC(C(Cc1cc[nH]n1)NC(CCOCCOC)=O)=O C1(C(C)NC(=O)C=CC2CCC2)CN(C(C2C3CC4C(C3)C24)=O)CCO1 c1(C(=O)NC2C(CCC)CN(C(C3CC3C#N)=O)C2)ncc(C)cc1Br C1(CNC(C(CC)NC(C)=O)=O)CCCCN(C(=O)CC2(O)CCCOC2)C1 C1(CSC)CC(c2nnnn2CSc2ccccc2)(NCCC(Cl)Cl)C1 C1(C(N2CCC(C)C(NC(=O)CCCCC#N)C2)=O)CC1C1CCCCC1 CC(C)CC(=O)NCC(C)(C)OCCNC(=O)C(CO)N(C)C N1(C(c2nc(C)oc2)=O)CCCC(C)C1CNC(=O)CNC(=O)NC1CCCC1 c1(C(=O)NC2C3CN(Cc4c(OC(C)C)cccc4)CC32)cc(F)c2cn[nH]c2c1 N1(C(CC(CC)C(C)C)=O)CCCC2(CNC(=O)Cc3ccc(Cl)s3)CCCC12 c1(CNC(c2ccc(OC)cc2)C)[nH]c(=NCC(=O)NC2CC2)nc2sccc12 c1(CCC)cc(=NCC2(C3CC3)CCN(C(=O)CC(O)C3CC3)C2)[nH]c(Cl)n1 C1(COC)CC(CNC(=O)Cc2cnoc2)N(C(c2nocc2C(C)C)=O)C1 Cn1cnc2nc(=NCC(C)(CC)C(N)=O)[nH]c(NCCCCCCF)c12 Cc1cc(C(=O)NC(C2(O)CN(C(C3(F)CCCOC3)=O)C2)C)cn1C N1(C(CCC)CC2CCCCC2)CC(C#N)(c2cccc(F)c2)C1 C1(C(N2CC3C(NC(C(COC)COC)=O)C3C2)=O)CN2CCN1C(C)C2 N1(C(Cn2ncc(C#N)c2)=O)C2CCC1C(CNC(=O)CN1CCNC(=O)C1)C2 c1(C(N2C(C(=O)NC(C#C)C(C)OC)(CC)CCC2)=O)cc(O)nc(O)n1 c1(C2C(C(=O)NCc3cc(C4CC4)nc(O)c3)C2)ccc2ccccc2c1 c1(N2CC(CNC(CCCC#CC)=O)N(C)CC2)ncnc2sc(CC)cc12 C(c1cccc(Br)c1)=CC(=O)NC1CCC(CCNC(C2(C=C)CC2)=O)C1 Cc1ccc(CN2CC3CCC(C2)N3C(C2CC2C)=O)cc1C#N c1(C(=O)NC(C)COc2cn(C)nc2C(F)(F)F)ccccc1O C1(Nc2cn(CCC(=O)N(C)C)nc2)CCC(F)(F)CC1 N1(C(C2C(CCC)C2)=O)CCCC1C(=O)NCc1conc1C Cc1ccc2c(CC(=O)NC3CCCC3NC(C3CCC(=O)C3)=O)c[nH]c2c1 c1(CNC(c2nnnn2NCC2CCCO2)C2CC(=C)C2)nncn1CC CCCCCCCCC(=O)NC(C)(C)CNC(c1cnn(C2CCCC2)c1)=O Cc1ncc(C(N2CC3CC(NC(=O)C(C)Sc4ncccn4)C3C2)=O)c(=N)[nH]1 C1(C2CCOCC2)(C(=O)NC2CCN(C(C=CS(C)=O)=O)CC2)CCOCC1 c1(-c2cn(CCCC)nc2)c(C(N2CCCC3C(O)CC23)=O)nn2c1CCCC2 c1(C(C)=O)c[nH]c(C(=O)NC(Cc2cn[nH]c2)C(=O)N2CC(OCF)C2)c1 c1(C(=O)NC(CCOC)CNC(C2(C(F)(F)F)CCC2)=O)cccc(N)c1C C(N=c1[nH]nc(C(F)F)o1)C1C(NC(Cc2ccc(SC)cc2)=O)CCC1 C1(O)(C(N(CCC(=O)NCC2CCOC2)CCO)=O)CCSC1 C(=O)(CCCCCC(C)C)N(CCCC)C(c1ccc(OC)cc1)C N1(C(C2C(CCC)CCC2)=O)CCC2CN(C(c3cnn(C)c3C)=O)CC2CC1 c1(OC)cc(OC(F)(F)F)ccc1NC(=O)NCC1CC2C=CC1O2 C1(NC(CC=CCC)=O)CC(CNC(C2(CCN3CCOCC3)CC2)=O)C(O)C1 Cc1ccc(C(N2CC(C3NC(=O)NC3=O)C2)=O)cc1Br C(=O)(C(C)(CC)C(=O)N1CC(CNC(c2cn(C)nc2O)=O)C2(CC2)C1)OCC CCC(O)C(C)C(=O)N1CCC(NC(=O)CC(C2CCC2)C2CCC2)C1C c1(C(=O)NCCCC)ccc(F)c(-c2csc(C(=O)Nc3onc(C)c3C)n2)c1 C(CCC(=O)N(C(C)C(N1CCCC1CC1CC1)=O)C1CC1)OCCC N1(C(C(CCC=C)(C)C)=O)CCOC2(CCCN(C(=O)CNC(=O)C(C)C)C2)C1 N1(C(c2ccc(OC)c(N)c2)=O)CCCC(C2CC2NC(c2cc(Br)co2)=O)C1 S(=O)(=O)(c1ccc(NC(CCO)C2CCC2)c(Br)c1)N(CC(O)CC(F)(F)F)C c1(OC)c(C)cc(C(=O)N(CC(C)NC(C2CCCCC(=O)N2)=O)C)cc1Cl O=C(O)C(CCOCCl)Nc1nnnn1-c1ccc(-c2ccccn2)cc1 C1(O)(C(N2CC(c3cn(Cc4scc(C(=O)OC)n4)nn3)C2)=O)CC(C)(C)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(C)N(C(c2cc(Cl)cc(F)c2F)=O)CC1 C1(NC(c2csc(O)n2)=O)CN(C(=O)C=Cc2cnccn2)CC1C1CC1 N1(C(c2ccn(CC)c2C)=O)CCC2(C=C(C(=O)NC3CN(CC)CC3C)C2)C1 C#Cc1ccc(OC(=O)C(CC(C)C)OC2(C(=O)CC)CC2)cc1 N1(C(c2c(C)ccs2)=O)CC(C)(C)OCC1CNC(=O)CCS(C)(=O)=O c1(C(=O)NCCC2CC(NC(c3snnc3C3CC3)=O)C2)cc(O)cs1 C1(CC=C)(NC(=O)C(C)CCOC)CCN(C(=O)Cn2ccnn2)CC1 N1(C(C2(CCC=C)CC2)=O)CC2CS(=O)(=O)CC2(NC(=O)C#CC(C)(C)C)C1 N1(CC2CC(CSCCC3(CS(C)(=O)=O)CC3)C2)CCCNC1=O Cc1ccnc(C)c1C(=O)NCC1(C)CCCN(C(c2ccccn2)=O)C1 C1(C(=O)NC2CCC(N(C(=O)C=CCN3CCCC3)C)C2)CCC12CCOCC2 c1(OCCCC(=O)NCC(CC)NC(=O)C=Cc2cscn2)ccc(SC)cc1 C1(O)(C(N2CC(O)(CCNC(CC3(C)CC3)=O)C2)=O)CCSCC1 c1(C(N(CCNC(C2CCCCC2C2CC2)=O)CC)=O)cc2ccc(Cl)cc2[nH]1 CC(CC(=O)NC1CN(C(C2CNC(=O)C2)=O)C1)NC(C1CCCC1)=O c1(C(=O)OC)ccc(C(N2CCC(NC(=O)C(O)C(F)(F)F)CC2)=O)c(F)c1 C1(CC(=O)NCC(C)N(C(=O)CN2CC3CC3C2)CC)COCC(C)(C)O1 C1(NC(CC=CC)=O)CN(C(=O)CC(O)CN(C)C)CC2(CCC2)C1 C1(NC(N(C(c2ccccc2)C)C)=O)CCCC2(CC2)C1 C1(N2CCC(Oc3ccc(Cl)cn3)CC2)Cc2ccccc2O1 C1(OC)CC(c2nnnn2C(C)(C)C)(NCCC(c2ccccc2)O)C1 C1(C(N(c2cccc(C)c2)C)=O)CN(C(c2ccc(C3CC3)o2)=O)CC(C)(C)C1 c1(C(N(CCCNC(C(C)N(C(C)=O)C)=O)CCO)=O)ccn2ccnc2c1 Cc1cccc2c(C(=O)NCCCCC3CN(C(=O)C(C)(C)C4CC4)C3)coc12 C12(C(C(=O)OC(CC(=O)OC)C)C)CC3CC(CC(C3)C1)C2 Cn1ncc2ccc(CNC(c3cccnc3-c3ccc(F)nc3)=O)cc12 C(=O)(C1=CCC(F)(F)CC1)NC1CN(C(C2CC(C)C2(C)C)=O)C1 CC1CN(C)CCCN1C(C1CC1CNC(c1cc2cccn2cn1)=O)=O C1(C(N2CCC(CCOC)(NC(=O)CCC=C(C)C)C2)=O)OCC2CCCCC12 c1(C(N2C(CCNC(C(C)(C)C(N)=O)=O)CCCC2)=O)cccc2c1NCC2 c1(C(=O)OC)ccnc(N2CCC(NC(c3cc(Br)co3)=O)C2)c1[N+](=O)[O-] N1(C(c2c(C)[nH]c(C)c2C)=O)CC(NC(=O)Cc2c[nH]nc2O)CC(C)(C)C1 C1(C(=O)NC2C=CCN(C(C(C)c3ccco3)=O)C2)CCCCC12CCC2 C(=O)(C(O)C(F)(F)F)NC1CN(C(c2ccc(COC)s2)=O)C1 C1(C(=O)NC2C(C)CCC2C)C2CCCC2CN1C(C1CC2CC2C1)=O n1(CC(=O)NCCN(C(C2(C)CCC2)=O)C2CC2)nnc2ccccc2c1=O N1(C(CC2C(C(=O)OC(C)(C)C)C2)=O)CCC12CC1CCC2C1 C(=O)(C(C)(C)CC(F)(F)F)N1CC(CCC)N(C(=O)CC2CCCCN2C)CC1 C1(CNC(CCOCCCOC)=O)C2CN(C(c3scnc3C)=O)CC12 C1(NC(CCC(C)OCC)=O)CCC2CN(CC(C3CC3)OC)CC2C1 C1(C(N2CC(C)(C(=O)NC(C)COCC3CC3)C2)=O)CCCCC1F C1(CC(=O)NC(CC)CN(C(=O)C=CC(C)CC)C)CCC(F)(F)CC1 c1(N2C(CCNC(c3ccc(Cl)s3)=O)CCCC2)[nH]cnc2nc(Cl)cc1-2 Cc1ncoc1C(=O)NCC=CCC(=O)NCCC(O)C1CCCC1 c1(C(N2CCC(COC)(NC(=O)CSC(F)F)C2)=O)ccc2cc(C)ccc2n1 c1(CC)c(-c2nc(-c3cccc(C)c3)nn2-c2ncnn2C)cnn1CC c1(C(=O)NCC(C(C)(C)C)NC(C2C(C)C2C)=O)cnn2cc(C(N)=O)cnc12 C(=O)(C1=CC2(CCOCC2)C1)NC1N(S(C)(=O)=O)CCCC1 c1(N(C)C)ccc(N)c(C(N2CC3CCC3(NC(C3CC4C=CC3C4)=O)C2)=O)c1 N1(C(CCC2CCC(=O)C2)=O)CCC2CCN(C(=O)Cn3cccn3)CC12 CC1CN(C(C2(NC(N)=O)CC2)=O)CCC1NC(=O)CC1(C(F)(F)F)CCCC1 c1(CC(=O)N(CCC2N(C(C)=O)CCCC2)C(C)C)cc(F)ccc1Br C1(C(N2CC(C(N(CC(=C)C)CC)=O)(COC)C2)=O)CC=C(C)CC1 C1(C(N2C(C)CCC(CNC(c3cc(CO)on3)=O)C2)=O)CCc2nncn2C1 c1(C(c2n(CCCSCC)nnn2)NCC2CCCS2)n[nH]c2ccc(C)cc12 CCC1=C(C(=O)N2CCC(NC(c3cscn3)=O)CC2C2CC2)SCCO1 N1(C(C2(CC)CCOC2)=O)CC(CO)C2(C1)CN(C(=O)C(SC)SC)C2 C(=O)(C(F)(F)C(C)(C)O)N1CC(CN(C(C(CCC)NC(N)=O)=O)C)OCC1 CC1(C(N2CC(OC3CCN(C(=O)CSC4CCCO4)CC3)C2)=O)CCCOC1 C12(NC(C3CNC(=O)O3)=O)CCC(CN(C(c3cccc(C4CC4)n3)=O)C1)C2 c1(C(N2CC(NC(C(=O)NC(C)C)=O)C3C2C3)=O)cc(C#N)ccc1O Cc1nc(C(=O)NCC2CC3CC3N2C(=O)CC(C)C(F)F)c2ccccn12 CC(CNC(=O)CN(C(=O)Cn1cc(Cl)cn1)C1CC1)(CO)CO N1(C(C(F)=CC)=O)CCC(n2cccn2)(C(=O)NCCN2C(=O)CNC2=O)CC1 c1(N2CCN(S(=O)(=O)CCF)CC2)ccc(C2CCCCC2)c(Cl)c1 N1(C(CN(C)Cc2cccnc2)=O)CC(F)(F)CC1(C)CNC(C1CNC(=O)C1)=O c1(C(=O)NC(c2cn(C)nn2)C(=O)NCCCOC)c[nH]c(C)c1 c1(OCC)cccc(CN2CC(C)(C(=O)NCc3cscn3)C2)c1 C(=O)(CCS(=O)(=O)NCC1CN(C(c2ccc(Br)cn2)=O)CCO1)OC c1(C(N(CCNC(C(C2CCOCC2)OCC)=O)C)=O)nnn(C(C)(C)C)n1 C1(C2CC2)(CNC(C(CN(C)C)N(C)C)=O)CCN(C(C2(C)COC2)=O)C1 C1(C(=O)NCC(n2c(C)cc(=N)[nH]2)C)CC12CCOCC2 C1(NC(C(CCC)NC(N)=O)=O)CC2CN(C(=O)C=C(C)Cl)CC2C1 c1(C(=O)NC(C2OCCN(C(c3c(C)csc3C)=O)C2)C)ncc2[nH]ncc2n1 C12(CNC(C(CO)NC(c3c(N)cncc3)=O)=O)CC=CC(C1)OC2 N(C1CC2(CN(C(=O)CC(C)n3ccnc3CC)C2)n2ccnc21)C(C=CC)=O C1(OCC(=O)NC(CC)CN(C(=O)C(=Cc2ccco2)C)C)CCCCC1C N1(C(Cc2ccc(C(=O)OC)s2)=O)CC(NC(c2nnc(S)n2C)=O)CC(F)C1 N1(C(C(CCC)F)=O)CC2CCN(C(C3CCC(=O)NC3)=O)C(C2)C1 C1(CNC(c2cnc(C)o2)=O)CN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC1(C)C C12(C(N(CC(C)O)Cc3c(OC)ccs3)=O)CCCC1CC(C)CC2 c1(N(C(C(C)(C)C(F)F)=O)CCCN)ncnc2c1CCO2.C1(N)CCC1(F)F N1(C(C=C2CCC(C)C2)=O)CCCC(N(C)C(c2cnn(C)c2N)=O)CC1 C1(OCCC)CCC(n2cc(C(C)(C)CC3CC3)nn2)CC1 C12(CCNC(Cc3c(C)con3)=O)CCC(C1)N(C(=O)CCSCC(N)=O)C2 C1(C(C)C)(C(N2CCC(n3cccn3)C2)=O)CCN(C(=O)C(C)N2CC(C)C2)C1 c1(OC)cc(C(=O)NC(C)(C(=O)OC(C)(C)C)C2CCC2)nc(C)c1 c1(CS(N2CCC(NCCC(=O)N(CC#C)CC)CC2)(=O)=O)cc(F)c(F)c(F)c1 c1(OC)nc(Cl)ccc1C(=O)NCC(CNC(=O)CC1CCCCC1O)CO N1(C(C=NOC)=O)CC(CNC(C2(Cc3cnn[nH]3)CCC2)=O)C2CC12 CC(C)C(C(=O)N(C)Cc1ncccn1)C(C)NC(C1CCCS1)=O c1(CC(=O)NC2(COC)CCCC2)cn(C)nc1C.C1(=O)CC2(CC2)CN1 C1(C(=O)NCC2C3CN(C(c4cc(SC)nn4C)=O)CC32)CN(C)CC(C)O1 N1(C(C2CCC(C)CC2)=O)C2CCC(C2)C1C(N1CCOCC(C(C)C)C1)=O N1(C(CC(=O)NCC(CC)NC(C2CC3CC2C3)=O)C)CCCCC1=O c1(CC)cc(C(=O)NCC2(NC(=O)CN3CCCCC3C)CC2)c(C)nn1 CCC(O)C(C)C(=O)N(C1CCN(C(c2ncoc2C2CCC2)=O)C1)CC C1(C(N2CCCCC2C(C)(C)NC(C2(CO)CC2)=O)=O)CC2(CCN(OC)C2)C1 C(C(C(=O)NCCC(O)C1CCC1)NC(c1ccnn1C)=O)SCC C#CCC(C)(C)C(=O)NCc1cn(C2CN(C(=O)CN3CC(=O)NC3=O)C2)nn1 C(CCCCC(=O)N1CC2CC2(NC(=O)C=CCCC=C(C)C)C1)NC(C)=O C1(NC(c2cc(CCC)on2)=O)CCCN(C(=O)C(CC)CCC)CC1 C1(CNC(Cc2c(C)ocn2)=O)CCC(CNC(=O)CC2CC(C)(C)CO2)CC1 c1(-c2scc(O)n2)cccc(-c2ccc3sccn23)c1.C(CCC(C)(F)F)N(C)CC c1(OC)noc(C)c1C(N1CCN(C(=O)C(c2cccc(Cl)c2)O)CC1)=O C1(NCc2ccc(C)cn2)CCN(C(c2ccc(Br)nc2Br)=O)CC1F C1(C(=O)NC2CC(NC(C3(C)CCCC3)=O)C2)C2CC3C(C2=O)C13 CCCC(F)C(=O)NC1C=CC(C(=O)NCc2cccc(OC)c2)C1 C1(C(N(CC(CC)NC(c2ccccc2Cl)=O)C)=O)CC2C=CC1CCC2 c1(CC)ccc(C(=O)NC2CN(C(=O)CC3(N(C)C)CCCC3)CC2F)cc1Cl CCC(CCOC)C(=O)N1CC(O)CC1CC(=O)N(C)Cc1cn(C)nc1C C(CC(C)(C)C(=O)N1CCC1CNC(C12CC(CC(F)(F)F)(C1)C2)=O)SC C1(NC(CC(COC)C)=O)CC2CCC(C1)N2C(C1(C)CCCO1)=O c1(N(C(C(=O)NCC2CCCO2)C2CCSC2)CC=C)ccccc1 Cc1cc(=O)n(C)nc1C(=O)NC(CNC(=O)CCc1cc(F)ccc1F)CO C1(CN(C)C(C2COC(=O)N2C)=O)COCCN1C(=O)CC1(C)CC1(F)F CC1CC(NCC(F)(F)F)CN1C(=O)C(C)(F)F.c12cccc(c1)COC2=O C12(NC(=O)C=Cc3ccc(Cl)cc3)CCCN(C(=O)CC3CC=CCC3)CC1C2 c1(CC(=O)NCCC2CCCN(C(c3cnc(Cl)s3)=O)C2)cnn2c1CCCC2 C(=O)(C1CCc2cc(F)ccc21)N(C(C)CNC(=O)C(C)(C)n1cncn1)CC c1(CC(=O)NCC(C(C)(C)C)NC(c2cncc(F)c2Cl)=O)c(F)cccc1F c1(CNC(=O)CC2(NC(C3CSCCN3)=O)CCC2)cnc(Cl)cc1Br C1(C(N(C(CNC(C2CCC(O)C2)=O)Cc2ccccc2)C)=O)CCCC12CC2 CC(C)C(C)(C(=O)NCC1CC(n2cc(CCC(C)(C)O)nn2)C1)S(C)(=O)=O C1(NC(C(CNC(CC(=O)NCC)=O)N(C)C)=O)CCN(C)CC1 N1(C(C(CC)(C)O)=O)CCN(c2cc(-c3cccc(Cl)c3)ncn2)C(C)C1 c1(C(N(CC(O)C2CC2)C)=O)cnc(N)cn1.C12CCC(C1)C(=O)N2 N1(C(COC2CCN(C)CC2)=O)CCC(O)(C2CCN(C(C34CCC3C4)=O)CC2)C1 N1(C(CC(C)(C)CC2CN(C(C3CC(C)(F)C3)=O)C2)=O)CCOC(C(C)(C)C)C1 C1(C2(NC(C=CC=CC)=O)CC2)CCCN1C(c1cnn(C(C)(C)C)c1)=O C(=O)(CCCCCC(C)C)NC1(C(=O)NC(c2c(C)ccnc2)C)CC(F)(F)C1 N=c1[nH]ccc(C(=O)NCC2CN(C(=O)C3=CCSC3)CCO2)c1[N+](=O)[O-] Cc1nccnc1CNC(C1C2CC1N(C(=O)CN1CCOCC1=O)C2)=O N1(C(C(C)n2ccnc2)=O)CCCC12CCN(C(=O)CC1CN(C3CC3)C1)CC2 C1(CCNC(C(C=C)(F)F)=O)CCN(C(=O)C(CC)N(CC)CC)CC1(F)F C1(N(C(=O)CCc2cn(C)cn2)C)CC2CCC(C1)N2C(C1CCCCO1)=O c1(C(=O)NC(C)CNC(C2CCC3(CCC3)O2)=O)cnn2ccn(C)c12 O=CN1CCCN(Cc2ccc(N3CCCC3)o2)CC1 CCCC(O)C(=O)N(C)CC=CC(=O)NCC1(CCO)CCCC1 CCC(CC(=O)NC1CC(NC(c2nccc(Br)c2C)=O)C1)C(C)C C1(CNC(C(c2ccco2)NC(C2CCCCO2)=O)=O)(CO)CC2CC2C1 N1(C(C2ON=C(C)C2)=O)CC(NC(C2CN3CCN2CC3C)=O)C(C2CC2)C1 C1(C)(CNC(C(C2(O)CCC2)NC(C(CC=CCC)C)=O)=O)CCCCCC1 CC1CN(C(c2sccc2-n2cccc2)=O)CC1NC(c1cc(C(F)F)on1)=O C(C(C)(O)CNC(c1nnc(C(C)(C)C)s1)=O)NC(C(C)=CC1CC1)=O C(C)(C(=O)NCC1CCN(C(C2CC(SC)C2)=O)CC1)(C(C)C)OC C(C(C(=O)NCc1coc(C)n1)NC(=O)CCNC(=O)CO)SCC N1(CC(=O)NC(c2nc(CC)sc2)C)CCN(C(=O)C(C)NC(N)=O)CC1C N1(C(c2c(C)cccc2)=O)CC(NC(=O)C(C)Cc2ccco2)C(C#N)C1 C1(C(=O)NCC(C)(C)OCCNC(C2C(C)C2)=O)COCCO1 N1(C(C(CSC)OC)=O)CCN(C(=O)Cc2ccc(F)cc2)CC(C)(F)C1 C(=O)(C(C)(C)CC(C)(C)C)N(C)Cc1c(CNC(C(C)S(C)(=O)=O)=O)cccc1 CCCCC(C(=O)N1CC2(C(=O)O)CC2(C(F)(F)F)C1)NC(=O)OC(C)(C)C CC(CC(C)(F)F)C(=O)N(C1CCCCC1NC(c1cnn2c1N(C)CC2)=O)C c1(C(=O)NC2C(NC(c3cncn3C3CC3)=O)CC2)[nH]ccc1C1CC1 C1(C(N2C3C(NC(=O)Cc4cc(C5CC5)on4)C(C3)C2)=O)CC12CCCOC2 c1(NC(C)=O)cnccc1C(=O)NC1CC(O)(CNC(c2sccc2F)=O)C1 N1(C(=O)NC(CC)C(C)C)CCC2(CC1)OCc1ccccc12 n1(CCOC)ncc2c1C(N=c1ccc(C3CC3)n[nH]1)CCC2 c1(COC)cccc(C(=O)N(C2CCC(NC(=O)C(=O)NC3CC3)C2)C)c1C CC1(C)OCCC1NC(=O)C=CC1CCCN1C(=O)CCN1CCC1 CCCCC(CC)C(=O)NC1CN(C(c2cc(C)ccc2Cl)=O)CC1OC c1(C(=O)NCC2(NC(c3c(C)ncs3)=O)CCCCC2)occ2c1CCOC2 Cn1ncc2ccc(NC(C3CN(C(=O)Cc4ccc(Br)nc4)C3)=O)cc12 CN1CCN(C2CCCN(C(c3cccc(C4CCC(=O)N4)c3)=O)C2)CC1 Cc1cc(NC(=O)NC2CCC3CCC2C3)cc(C#N)c1 c1(C(=O)NC2C(NC(CC3N(C)CC=CC3)=O)C2)cc([N+](=O)[O-])c2nsnc2c1 N1(C(CC2N(C(C(CCC)N(C)C)=O)CCC2)=O)CCCC2CCCCC12 Cc1cncc(CCC(=O)NCCCN2C(=O)CNC2=O)c1 c1(C(=O)Nc2cn(CCS(CC)(=O)=O)nc2)cccc(F)c1C#N Cc1cn2c(C(=O)NC(CNC(c3cnc4ccccn34)=O)CO)c(Cl)nc2s1 C(=O)(C#CC(=O)NC1CCCC1)N(C1CCN(C(c2cc(C)oc2)=O)C1)C N1(C(c2cnc(C)nc2C)=O)CC2(CCCC2NC(=O)CCN2CCCC2=O)C1 CC(CNC(C12CCC(C)(CO1)C2)=O)CN=c1[nH]c2ccccc2s1 C1(C)(NC(CN2C(C)CCC2)=O)CCCN(C(=O)Cn2cc(C(F)(F)F)nn2)C1 c1(C(=O)NCC(C2CCCCC2)NC(C(CC)F)=O)nccn2nc(C)cc12 CC1CCN(C(C2(C)CCOC2)=O)CCN1C(c1nc(Cl)sc1Cl)=O CCCC(O)CC(=O)NCC(O)CNC(=O)C(c1ccc(Br)s1)=O C1(O)(C(C)NC(=O)Cn2cccc2)CCN(C(=O)C(C2CCCCC2)O)CC1 C(=O)(C(C)(C)C#N)NCC1(NC(=O)CCc2cccc(Cl)c2)CC(OC)C1 Cc1ccc(CN2CCC(F)(C(=O)NC(c3ccccc3)C3CC3)C2)c(Cl)n1 N1(C(Cc2ccn(CCc3cn(CC)nn3)n2)=O)Cc2ccccc2CC1CO C1(C(C)C)CN(C)CCN1C(C1(C)CC(NC(C2CN(C(N)=O)C2)=O)C1)=O N1(C(CCNS(CC)(=O)=O)=O)C(C)C2CC1C2NC(c1nn(C)cc1C)=O C1(NC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC2CC23CC3)CC1O c1(C(N2CC(C)N(C(c3cscn3)=O)CCC2)=O)cc(N)c(O)cc1Br N1(C(c2sc(Br)nc2Cl)C(=O)N(CC(C)C)C)CCOCC1c1nncn1C N1(C(c2cc(CC)nn2C)=O)CCC2(CCCC2C(=O)NCc2cncnc2)C1 Nc1ncnc2c1ncn2Cc1cccc(NCc2cc3c(s2)CCCC3)c1 C(=O)(C#CC1CCCC1)N1CC(NC(c2c(C)c(N)n(C)n2)=O)C(C)C1 N1(C(c2cc(C(C)C)ncc2)=O)CC2CCC(C1)N(C(=O)COCC(F)(F)F)C2 C12(CC)CN(C(c3ccc(OC)c(C)c3)=O)C(CNC(C34CC(C)C3C4)=O)(C1)C2 C1(CC)(CC)CC(NC(c2cc(C)nn2C2CC2)=O)CN1C(=O)CC(C)(C)C c1(C(N2CC3CCN(C(C4C(C)CC4)=O)CC32)=O)ccc(O)c2ccccc12 c1(C(=O)NC2C=CCN(C(C(COC)OC)=O)C2)[nH]c2cc(F)cc(F)c2c1C C(CC(C)C)(C(=O)NC1CN(C(=O)CN2CCSCC2)CCC1F)OC n1(CC)nc(C)cc1C(=O)N(CCC(=O)NC(C)CC(C)O)C C(=O)(C(CNC(C1CCC(C)(C)OC1)=O)C(C)(C)C)N(C)C1CC1 C(CCCCC(=O)NC(c1ccc(C)s1)C)NC(C(C)NC(C)=O)=O C=CC1(NC(=O)CN(CC(C)C)C(=O)CC2CC=CCC2)CCOCC1 CC1CN(C(C2CCC2(C)C)=O)CC1N(C)C.c12ccc(nc1)[nH]c2=O c1(OC)cnc(C(=O)N(C2C3CN(C(C45CCCC4C5(F)F)=O)CC23)C)c(F)c1 C=C(C)CN=C(NCC1(CCNC(C)=O)CC1(F)F)N1CCc2n[nH]cc2C1 N1(C(C(C)O)=O)CC2CCC(C1)C(NC(c1cccc(C3CCOC3)c1)=O)C2 c1(C(=O)NC23C(CN(C(c4c(C)ccnc4C)=O)C2)C3)c(F)ccc2c1OCC2 C=CCC(CC)C(=O)N(CCCNC(C1CC(F)C(=O)N1)=O)C(C)C C12(NC(c3ccc(COC)cn3)=O)COC(C1)C(NC(=O)C(C(C)O)N(C)C)C2 N1(C(Cc2ccnc(C)n2)=O)CCCC(O)(CCNC(=O)CNC(=O)C2CC2)C1 c1(C(=O)NCC(n2cc(C3C4COCC34)nn2)C)cc(Cl)ccc1Br C1(C(=O)OCC)(COC)C=CCN1C(=O)NC1CC(O)(C(F)(F)F)C1 c1(C(=O)NC(C)CC(C)NC(=O)COCCN(C)C)cccc2ncsc12 N1(C(CC2(C)CCN(C(=O)CC3COCCO3)C2)=O)CC2CCC(C1)O2 C=CCCCC(=O)N1CCC(CO)(NC(=O)Cn2cc(C(=O)OC(C)=O)cn2)C1 C1(C2CCN(C(c3cc(C#N)ccc3F)=O)C2)(NC(CC(C)CF)=O)CC1 c1(C(=O)NCC)cccc2c(Br)cccc12.C12CCC(CC1)C(=O)OC2 n1(C(C)C)cnc2c(NCC(CO)C(C)(C)C)[nH]c(=NCCc3cocn3)nc12 C(c1ccc([N+](=O)[O-])s1)=CC(=O)N(CCNC(=O)C(C(C)O)N(C)CC)CC C1(CNC(COC)=O)CCCCN(C(C2(Cc3cccnc3)CC2)=O)C1 C(=O)(CCCCC(C)(C)C)NC(c1ccccc1)C(=O)N(C)CC1(OC)CCC1 c1(C(N(C2CCCN(C(=O)C(C)(O)C3CC3)C2)CC)=O)cc(O)nc(N(C)C)n1 CC(CNC(c1cc2cccc(F)c2o1)=O)CN=c1ccn2nccc2[nH]1 c1(C(=O)N)cccn2nccc12.c1(C(=O)NC2CCC(OC)CC2)cc(O)nc(Cl)c1 C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NCC1C(NC(C2(C=C)CC2)=O)COC1 Cc1nc(Cl)[nH]c(=NCC2CCCC2NC(C2(C(F)F)CCC2)=O)c1Cl C(CCCCC(=O)N1CC(NC(=O)C(C)C(O)CC)C(CO)C1)=CC C1(NC(C(F)=CC)=O)CN(C(=O)C(C)c2ccco2)CCC1c1cccc(F)c1 c1(CC)cccc(F)c1C(N1CCC(CN(C(=O)CN2CC(C)C2)C)C1)=O C1(NC(C(C)C2CCC2)=O)CCN(C(C2CN3CCCN2CC3)=O)CCC1CO C12(CNC(CC(CC)O)=O)CCCC1N(C(c1nccnc1OC)=O)CCC2 CC(C)CC(C)(O)C(=O)OCCNCC(C)(C)CCC=C(Cl)Cl C(c1ccncc1)=CC(N1CCC(OCC(N2C(CC)(CC)CC2)=O)C1)=O c1(C(N2CCC(NC(=O)Cc3cccc(O)c3)C23CC3)=O)ccc2c(c1)OCO2 CCC(CC(=O)NCc1nocc1C(N1CCOC(C2(C)CC2)C1)=O)OC c1(C(C)C)nc(NCCC(F)(F)Cl)cc(=NCC2(C)CCCCC2)[nH]1.CO c1(NC(C)=O)cnc(C(=O)NC2CC(NC(=O)C(O)Cn3cncn3)C2)c(Cl)c1 C1(C(NOC(C2CCOCC2)CC)=O)CN(C(c2csnc2C)=O)CCO1 N1(C(CCNC(C)=O)=O)CC(C)C(NC(C2CCC2c2ccn(C)c2)=O)C(C)C1 Cc1cc(C(=O)NCC2CCC(NC(=O)CC3(O)CCC3)CC2)cc(C)c1Br c1(OCC)cc(CN2CCCC(CC(=O)NCCC3CCCC3)C2)c(Br)cn1 c1(C(C)=O)cc(Cl)nc(Cl)c1NC(C1CC1NC(C1CCNC1=O)=O)=O N1(C(N2CCCCC(OC(C)(C)C)C2)=O)C2CCC1CN(C(=O)N(C)C)C2 C12(CNC(C=C(C)Cl)=O)CC(NC(=O)C(N3CCP(C)(=O)CC3)C)(C1)C(C)(C)O2 C(CCCCC(=O)NC1CCC(CN(C)C(c2cc(CCO)on2)=O)CC1)SC c1(C(N(C2CCN(C(=O)C(N)=O)CC2)CC#C)=O)cccn2ncc(Br)c12 c1(CC(=O)N(CC(CNC(C2CC(CC)C2)=O)C)C)c(C)nn(C(F)F)c1C N1(C(CN(C)C(N)=O)=O)CCC(CC(=O)NCc2cc[nH]n2)C1 C1(C(N(OC)CC2CCCC2)=O)CC(C)(C)CN1C(=O)COCCSC C(=O)(C#CC1CCC1)NC(C(=O)N(c1ccc(F)cc1)C)CC1CCC1 CC1CCc2n(C(=O)CCC(C)c3ccccc3)ccc21 c1(C(N2C(C)(C)C(CNC(=O)C3=CCOC3)CC2)=O)cc(S(N)(=O)=O)cs1 N1(C(CC2CC(C)(C)OC2)=O)CCC(NC(=O)C(F)C(F)(F)F)C(F)C1 c1(CN2CC(C(=O)Nc3c(OC)ccc(OC)c3)SCC2)cc(F)c(Br)cc1Cl Cc1cc(O)cc(=O)n1CC(N1CCC(CNC(=O)C(C)C(F)(F)F)C1)=O CCCC(O)C(CO)NC(=O)C(C)(C)NC(=O)CC1CCOC1(C)C c1(C(N2CC(CC=C)(NC(c3nccc(C#C)c3)=O)C2)=O)cccc2c1OCC2 c1(C(=O)NC(CN(C(C2CCN(OC)CC2)=O)C)C)cc2c(Cl)cc(F)cc2[nH]1 C1(CNC(C2C(C)(C(F)F)C2)=O)CCC(C(=O)NCCC2CCCO2)CC1 c1(C(=O)NC(C2CC(NC(C3CC=CCC3)=O)C2)C)ccnc2cc[nH]c12 c1(C(N2C(C(=O)Nc3[nH]cnc3C#N)CC(=C)C2)=O)ccc(F)c(I)c1 c1(C(N(CC(CC)NC(C2CC2CF)=O)C)=O)cc2c(OC)c(Cl)ccc2[nH]1 C1(NC(Cc2c(C#C)cccc2)=O)CCC2(CCN(C(C3(C)CCCS3)=O)C2)C1 C1(C)(C(=O)NCC2(OC)CN(C(=O)CCc3ccon3)C2)C2CCC(C2)C1(C)C c1(C(=O)NCC(CC)NC(=O)CC2CCCCCO2)sc(C(C)OC)nc1C C(=O)(C1c2ccccc2CN1C(c1c(OC)ccc(Cl)n1)=O)Nc1c[nH]c(Br)c1 C12(NC(c3scc4c3OCCO4)=O)CCCC1CN(C(=O)Cn1cnnc1)C2 C(=O)(C(F)(F)CCn1cccn1)NCC1(NC(C2CCCCC2O)=O)CCCC1 N1(C(C(CCC)N(C)C)=O)CCCC(C)(C)C1CNC(c1cccc(OC)c1C)=O C(=O)(C(C)(C)C(=O)NC1CCCN(C(=O)CCc2cc(C)[nH]n2)CC1)NC CCC(CO)CN=C(NCCOc1ccc(Br)cc1)NC1CCC(C(F)F)CC1 C(=O)(C1=CCCOCC1)NC1C(C(N2C(C)(C(C)C)CC2)=O)C2CCC1C2 C(C(C(=O)NCCC1(C(=O)NCC2C3COCC23)CC1)N(C)C)N(C)C C1(COC)CCC(C(N2CCCC2CNC(=O)Cc2cc(C)ns2)=O)C1 C12(CCNC(=O)CC3C=CCC3)CCC(C1)N(C(c1cc(O)cc(F)c1)=O)C2 N1(C(C2N(C)CCC2)=O)CC=C(CNC(=O)Cc2cnsc2)CC1 c1(OC)ccc(C(=O)NCCCNC(=O)CC(C)F)c(OC2CC2(F)F)c1 C(=O)(CC(C)(C(F)F)N(C)C)NCC(CNC(c1cn(CC(CC)O)nn1)=O)F CCC(CC(F)(F)F)C(=O)NC(CN(C)C(c1ccc(NC(N)=O)cc1)=O)CC c1(C(N2C(C(N3C(C)CC4(CC4)C3)=O)CC(O)CC2)=O)ncc2ccccn12 C(C1=NOC2CCCC12)NC(C1C(C(C)NC(c2ccc(Cl)o2)=O)C1)=O C1(CNC(C(C)(Cl)Cl)=O)CC2CC2N1C(c1cc(Br)ccn1)=O C(N=c1[nH]c(=NC(C)CC)[nH]c2cccnc12)c1ccc(C(C)C)nc1 N1(C(C(CC)=CC)=O)CCC2CN(C(c3ccccc3CC(C)C)=O)CCC2C1 CC1CN(Cc2ccccc2)CC1NC(=O)NC1CC12CC(O)C2 C1(CNC(C2(SC)CCN(C(c3cc(F)cc(F)c3)=O)C2)=O)CC(=O)NC(C)C1 C(=O)(C(O)C(C(C)C)OC)NC(C(=O)N(CC(CC)OC)C)CCC1CC1 C1(C(N2CC(C(=O)NCC34CCC(CC3)O4)OCC2)=O)CCC2(CCC2)O1 C(CN=c1[nH]cc2ncnc-2[nH]1)N(C(C1CCS(=O)(=O)C1)=O)CC N1(C(C(=O)NC(c2cn(C)nc2)Cc2ccccn2)=O)CCCC2(C=CCO2)CC1 c1(C(N(CC(CNC(c2scc(C)c2)=O)C)C)=O)cc2ccncc2[nH]1 c1(CN(C(=O)C(C2CC3(CNC3)C2)N2CCCC2)CC)cccc(F)c1 N1(C(c2cc(C(C)C)nn2C)=O)CCCN(C(C2CCCC(=O)N2)=O)C(CO)C1 C1(C(=O)NCCOC2CN(C(C3C(C)N(C)CC3)=O)C2)CCc2ncncc2C1 N1(C(C(C(C)(F)F)F)=O)Cc2c[nH]c(=N)nc2C1 Cc1nc(C2CC2)nc(C)c1C(=O)NCC(C)CNC(c1nc(C2CC2)cs1)=O c1(OC)cccc(NC(c2ccc(NC(C3(N)CCC3)=O)cc2)=O)c1 C12(C(N(CC(C)(F)F)C)=O)CCC(CN(C(=O)CC3CCSCC3)C1)C2 C12CC3(CC3)CN1C2=O.c1(NC(CC#N)=O)cc(OC(F)(F)F)ccc1Br C1(NC(c2nncc(OC)c2)=O)CC2CN(C(=O)C=Cc3cc[nH]n3)CC12 N1(C(C(CCC)O)=O)CCCC(O)(CNC(c2ccc(CNS(C)(=O)=O)o2)=O)C1 Cc1nc(C)c(C(=O)NC(CNC(c2cn(CC(F)(F)F)nn2)=O)CO)c(C)n1 C1(C(=O)NC2CCN(C(COCCOC)=O)C2C2CC2)CCc2cnnn2C1 Cc1cc(OC(F)F)c(C(=O)NCC(C(C)C)NC(C2CCO2)=O)s1 c1(OC)n[nH]c(C(=O)N(CC(C)NC(=O)C(c2cccnc2)O)C)c1Cl N1(C(C(c2cnn(C)c2)OC)=O)CCC(C(=O)NC2CCN(C)CC2)C(CO)C1 C1(CSC)CCN(C(=O)NCCC2CCCN2)CC1.N12CCC(C1)C2=O CCC(C(=O)NCC1(OC)CCN(C(c2ncccc2C)=O)CC1)C(C)(F)F CC(C)CC(C)C(=O)N(CC(C)NC(c1ccc(OC(C)C)o1)=O)C N1(CCNC(C2(COC)CCCC2)=O)CCC(NC(c2cc(OC)no2)=O)CC1 N1(C(CNS(C)(=O)=O)=O)CCOC(CNC(c2cccc(CC(F)(F)F)c2)=O)C1 C1(C(C(N2CC(N(CCC)CC)C2)=O)C)CCN(C(C2CCCCCC2)=O)CC1 c1(CC)cc(C(=O)NC2CCCC(NC(c3cncnc3C)=O)C2)cn(C)c1=O c1(OC)cc(CCCN2C(=O)NC(CC(C)(C)C)C2=O)ccc1OCC#N CC1(C)CN(C(=O)CC2=CCOCC2)CC(CNC(c2cc(C(N)=O)cs2)=O)O1 C1(NC(C2CC(=C)C2)=O)CCN(C(=O)C=Cc2ccc(C)c(C)c2)C12CCCC2 c1(C(N2C(C)CCC(NC(C(COC)(F)F)=O)C2)=O)cc(Cl)cc(Cl)c1F N1(C(C2CC3(CCC3)C2)=O)CCC2CN(C(=O)CCc3cc[nH]n3)CC2C1 c1(C(C(=O)NCCSC)N(CCN(C)C)CC2CC2)cccc2c1CC(C)(C)O2 N1(C(C2CCC(CC)O2)=O)CC(O)CC1C(N1CCC(COC)CC1)=O C1(NC(C2N(CC)CC2)=O)(CF)CN(C(=O)Cc2cc(C3CC3)no2)C1 C1(C)(C(N2CC(OC)(CNC(=O)COC3CCCC3)C2)=O)CCCOC1 CCCCC(O)CCC(=O)NCCC1CCN(C(=O)C(c2cccc(O)c2)C)C1 c1(SC)cc(C)ccc1C(N1CCC(OCC=CCNC(=O)C2=CCCS2)C1)=O C1(NC(c2ccc(F)cc2)=O)CCCCCN(C(C2CC3CC2C3)=O)C1 C1(N(C(CN(C)CC)=O)C)CCCN(C(=O)C(=O)NOC)CC1 c1(C(=O)NCCN(C(C(C)OCC)=O)C(C)C)ccc(S(=O)(=O)CC(N)=O)cc1 c1(N(CC)Cc2nc(-c3cccc4nc(C)sc34)cs2)ccc([N+](=O)[O-])cc1F c1(CC(=O)NCC2(NC(CCCC3C(C)C3)=O)CCOC2)ccc(C(N)=O)nc1 c1(C(=O)NC(CNC(c2c(C)occ2)=O)(C)C)cc(C(C)(C)C)oc1C N1(C(CS(=O)(=O)NC2CC(C)C2)=O)CC2CS(=O)(=O)CC2(NC(=O)NC(C)C)C1 Cc1cc(C=CC(=O)NC2CC(=O)N(C3CN(C(=O)C(O)C4CCC4)C3)C2)on1 C(=O)(CCC(=O)NCC1CC1)NC(C=CC(N1CC(SC)C1)=O)C c1(CN2CC(CC#N)N(C(=O)Cc3cccc(Br)c3)CC2)cn2c(Br)cccc2n1 c1(CC(=O)N(CCNC(C2C3COCC23)=O)C2CC2)nc2ncccn2n1 C1(C(N(C(CC)CNC(c2cnc(N(C)C)nc2)=O)C)=O)CCC=CCCC1 c1(OC)ccc(C=NOCC(=O)N(c2ccc(N3CCOCC3)cc2)C)cc1 C(=O)(CCCCCC(C)C)NCCCCC1CN(C(c2cc(C)cc(F)c2)=O)C1 C(=O)(CC(C)NC(N)=O)NCC1CN(C(C(c2ccn(C)c2)C)=O)C1 C(=O)(C1CNC(=O)c2ccnn21)NC(C)CCCNC(=O)CC(C)(C)O C1(COC)CN(C(=O)C=C(C)CNC(=O)Cn2cc(Cl)cn2)C1(C)C C(=O)(C1=NOC(C(=O)NC2CC(CO)N(C(c3cccnc3S)=O)C2)C1)OC N1(C(CNC(C2C(C)(OCC)C2)=O)=O)CC2CCCC2C1C(=O)NCCOC C1(O)(C(=O)OC)CCN(C(C(=O)Nc2ccccc2Cl)c2cnc[nH]2)C1 C12(NC(c3cnc(OCC(F)F)cn3)=O)CCC(CN(C(C3CC3F)=O)C1)C2 c1(N2C(=O)CC(C(N(CCCNC(C(CC)SC)=O)C)=O)C2)c(C)nn(C)c1C N1(C(c2c(C)cc(C)c(C)c2)C(=O)NCC(C)C)CCC2(CC1)CN(C)C(=O)O2 O(NC(=O)C(CN(C)C)NC(=O)C=NOC)CC#C C1(NC(c2c(OC)c[nH]n2)=O)CN(C(c2csc(CO)n2)=O)C2(CCC2)C1 N1(C(CC2(C(=C)F)CCC2)=O)CC=C(C(=O)NC(CC(C)C)C(=O)NC)C1 C12(CNC(CS(N)(=O)=O)=O)CC(CO1)N(c1nnc(C(F)F)s1)C2 C(=O)(C1=NOC(C)C1C)Nc1c(C)cc(NC(c2cncn2C)=O)cc1 C1(C)(NC(Cn2ncc(NC(C(CC)SC)=O)c2)=O)CCC(F)(F)CC1 Cc1c(C(N2CCOC(CC(C)C)C2)C(=O)NCCN(C)C)cccc1C(C)C c1(SCCNC(CCOCCOCC)=O)ccc(C)c(F)c1.c12cn-1nn2 c1(C(=O)NCC2CCC(NC(C(C)SCC)=O)CC2)nccc2ccncc12 c1(C(N2C(CNC(=O)CCNC(c3ccoc3)=O)CC2)=O)ccc2cncn2c1 c1(CCC)n[nH]cc1C(N1CC(F)(CNC(=O)CCOC(C)CC(C)C)C1)=O C12(C(=O)NCC3N(C(C(C(C)C)C#N)=O)CC3)COCC1CS(=O)(=O)C2 C1(CNCc2cc(OCCCOC)c(OC)cc2)CCc2ccccc2C1 C=CC(C)(O)C(=O)N(C)CCNC(c1cc(Br)sc1C)=O Cc1cc(Cl)c(C(N2CCCC2Cc2cn(CC(F)(F)F)nn2)=O)s1 N1(C(=O)CCCCCF)CCCC2(C1)CN(C(=O)CCC1CCCC(O)C1)C2 N1(C(C2C(NC(C(C3CCCC3)OC)=O)CC2)=O)CCCc2ccccc21 c1(C(=O)OCC)ccccc1Cn1cc(CCc2nc(O)n[nH]2)nn1 C(=O)(C1CCc2c[nH]nc21)N(C1CC(NC(C(C(=O)OC)C)=O)C1)C C1(C(=O)NCc2nn(C)c(C(N3CC(CO)C(O)C3)=O)c2)CCC=CCCC1 c1(C(=O)NC2CCC(NC(c3cc(COC)on3)=O)C2)cccc(Cl)c1C c1(C(N2CCC(C(C)NC(c3c(OCC)ccs3)=O)C2)=O)nnn(C)c1N CCCCCS(=O)(=O)CC(=O)N(C)CCOCCN(C)C(c1c[nH]c(C#N)c1)=O CC(C)CC(CNC(C1CCOC1(C)C)=O)C(=O)NCc1ncc(CO)[nH]1 C(=O)(C1(CC)CCCc2ccccc21)N1CC2CN(C(CCCC)=O)CC2C1 c1(CNC(C2C(COC)C2)=O)cc[nH]c1C(=O)NCCC1CCC2CC12 n1(CCCC)ncc(C(=O)N(C(C)CNC(c2cnc(O)s2)=O)C)c1C C(C(C)C)(C(O)C(=O)N1CCN(CC(N2CCN(C(C)=O)CC2)=O)CC1)OC c1(C(=O)NCC(C)(C2CC2)NC(C(CC=CC)C)=O)c[nH]nc1[N+](=O)[O-] n1(CC(=O)N(CCNC(CC(C)SC)=O)C2CC2)cc(C#N)c(O)nc1=O c1(CC)cc(C(=O)NC(C2CCCC2)CNC(C2CCCCO2)=O)ccc1C N1(CCC(=O)NC2C=CCN(C(C=C(C)Cl)=O)C2)C(=O)c2ccccc2S1(=O)=O c1(C(=O)NC2C(C)CN(C(C3CC34CCOCC4)=O)C2)nnn2c1C(=O)NCC2 CC(C)(C#N)CCCC(=O)NCCCC(O)C(=O)NCC1(C)CC=CC1 c1(CSC)ccc2nsnc2c1.N12CCC(C)(CC1)c1cn(nn1)C(C)CCC2=O CCC(C#N)(CC)C(=O)N1CCC(C(=O)NCC2(O)CCCCC2)CC1 c1(C(N(C)CCOCCCN(C(=O)C(F)n2ccnc2)C)=O)ccc2c(c1)CC2 C1(C)(C(=O)NC(C2CCN(C(c3cncnc3)=O)C2)C)CC=CC1 Cc1ccc(O)c(CC(=O)NCCC2CN(C(c3n[nH]c(C)c3Br)=O)C2)c1 C1(C(=O)NCC(C)OC(F)F)CCCC(NC(c2cnsn2)=O)C1 c1(C2C(NC(c3ccc(O)c(C(F)(F)F)c3)=O)C2)cccc2cccnc12 N1(C(C2N(C(CC)=O)CSC2)=O)C2CCC1(CNC(=O)Cn1cnnn1)CC2 C12(CC)CC(C(=O)NCCC3COCCN3C(=O)C(F)F)(CO1)C2 N1(C(C2(C)CC2)=O)CCCCC2(CCN(C(=O)C(CO)NC(=O)C(F)(F)F)C2)C1 CC(C)C1=CCC(NC(=O)CCNC(=O)CCCc2ncco2)CC1 c1(CC(=O)NCC(C(C)C)(C)NC(=O)Cc2sc(O)nc2O)ccc(Cl)c(F)c1 CC(C)C(O)CC(=O)NC(C1CCN(C(=O)C(C)Cc2ccc(F)cc2F)C1)C c1(C(=O)NC2CCN(Cc3c(OC)ccc(Br)c3)C2)ccc2nc(C)oc2c1 C=CC1COCC1NC(=O)C(C)N(C(c1cc(O)n(CC)n1)=O)C1CC1 C1(NC(c2c(CC)scc2)=O)CCN(C(C2COCCN2C(C)=O)=O)CC1(C)C c1(C(=O)NC2CC3(C(NC(c4cc(C(C)=O)sc4)=O)C3)C2)cc(C#N)ccc1N C1(C2CCN(C(=O)CCC3CCC3)CC2)(NC(CCCCOC(C)C)=O)CCC1 c1(N(C)C)cccc(C(N2CCC(C3CCCN3C(c3cccnc3)=O)C2)=O)n1 c1(CC)ccc(C(=O)NCC(C(C)(C)C)NC(=O)CN2CCOCC2)cn1 Cc1nn[nH]c1C(N1CCCC1CC(=O)N(CC(O)CO)CCO)=O CC1CC(NC(c2cccs2)=O)CN(c2nnc(-c3cccn3C)n2C2CC2)C1 N1(CC)C2CCC1CN(C(=O)CCC(C)NC(=O)CC(C)c1ccco1)C2 c1(C(=O)NC2CN(C(C(CC)(C)CO)=O)CC23CC3)ccc(S(N)(=O)=O)nc1 N1(C(CC2(CCC=C)N=N2)=O)CCC2CCN(C)CC12 C1(NC(c2nnc(C)s2)=O)CCN(C(=O)CCc2ccccc2)C1C(C)(C)C Cc1c(O)nc2ccccc2c1C(=O)NCC(C)NC(=O)C(CN(C)C)C(C)C C1(N(C(=O)Cc2nc(C)no2)CC)CCCN(C(=O)CC2CCCCC2C)C1 C1(NC(c2cc(C)nn2C)=O)CC12CCN(C(=O)CC(C)O)CC2 C12(NC(COCCCCC)=O)CC1CN(C(=O)C(CC)C1CCOCC1)C2 c1(OCC)cc(CNc2ccc(C(=O)Nc3ccccc3)nc2)ccn1 N1(CC(=O)NC2C(CNC(c3c(C)nncc3)=O)CCCC2)CC(=O)N(C)C1=O N1(C(c2c(OCC)scc2)=O)CC(NC(=O)C(C(C)O)N(C)C)CC(F)C1 C1(O)(CNC(c2c(OCCC)n[nH]c2)=O)CC2CCC(C1)N2C(=O)CC=C(C)C c1(CC)nnc(C)cc1C(=O)NC(C1CCCN1C(C1CCCOC1)=O)(C)C S(=O)(=O)(c1c[nH]c2c(Cl)cccc12)NC1CC(C(N)=O)C12CCOCC2 C(=O)(C1Cc2c(Cl)cccc21)NC1C(NC(CC(=O)OCC)=O)CC1 N1(C(c2n(C)cnn2)=O)CCC(C)(C)C(CNC(c2cc([N+](=O)[O-])cn2C)=O)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCCC(N(C)C(c2cc[nH]n2)=O)CC1 CN1C(=O)NCC1NC(N1CCCCC1c1cccc(C(F)(F)F)c1)=O C(=O)(CCCC(C)(C)C#N)NC1CC(OC)CN(C(c2cc(C)ns2)=O)C1 N1(C(c2cc(C)sn2)=O)CCCC2(NC(C3CC3(Cl)Cl)=O)CCCC12 C(=O)(C(CCC1(C)CC1)NC(C12CCCC1C2)=O)NCCN(CCCF)C Cc1cnc(F)c(C(N2CCC(=CCNC(=O)CC3CCCCC3)CC2)=O)c1 N1(C(C(CC(F)F)N(C(=O)Cc2ccsn2)C)=O)CCOCC(F)(F)C1 C12(C(=O)NCCN(CCC)C(c3cncs3)=O)CC(C)(C1)OC2C C1(CNC(CC2CCN(C)C2)=O)CCN(C(=O)CCOC2CCCOC2)C12CC2 C1(c2n(CCOC)nnn2)(Nc2ccc(C)nc2OC)COCCC1C C12(CNC(c3sccc3SC(F)F)=O)CC(CN1C(=O)C(F)F)C2 c1(C(N2CC3C(NC(C(CCOC)OC)=O)C3C2)=O)cc(SC)cc(Cl)c1 CC(C)CC(CC(C)C)C(=O)NC(C)CC1CN(C(C2CS(=O)(=O)C2)=O)C1 N1(C(CC=C)=O)CCC2(CCCC2NC(=O)C(CO)NC(N)=O)CC1 C1(NC(C(N2CCOCC2)C)=O)CC2(C1)CC2NC(=O)C(O)Cn1cncn1 C1(C2CC2)(NC(C(c2ccccc2)C)=O)CCN(C(=O)C(C)(C)N(C)C)C1 N1(C(CC=C)=O)CCC(OC2CN(C(C3CC3c3cccnc3)=O)C2)CC1 CCCCC(C(=O)NCC(C)(C)CNC(=O)CC(C)NCC)N1CCCS1(=O)=O Cc1nccc(CCC(N2CCC(C)(NC(=O)CC3CCCCO3)C2)=O)n1 C=C(C)CCCC(=O)N1CCC(NC(c2c[nH]c(C(N)=O)c2)=O)C1 c1(C(=O)NCC2CC(CNC(=O)CC3CCOCC3)OC2)cncnc1C1CC1 Cn1nc(C(N2CCC23CCCC(C)(C)C3)=O)c2cc(Br)ccc12 c1(C(N(CC(C)N(C)C(c2cscc2Br)=O)C)=O)ccc2cc[nH]c2n1 C(N=c1ccc(S(=O)(=O)NCc2[nH]c(C(N)=O)cc2OC)c[nH]1)C1(CC)CCC1 Cn1nc(Br)cc1CC(=O)OCCNC(=O)NC.C(C)(C)(C)OCCS c1(-n2ncc(C(=O)NCC(C)N(C)C(C3CCC(C)(C)O3)=O)c2)ccc(Cl)cc1 C1(NC(C(C2CCN(C(C3CC3C(C)(F)F)=O)CC2)C)=O)CC2CCC1O2 C1(C(N2CC(O)(CNC(CCC=CC)=O)C2)=O)Cc2ccc(F)cc2O1 CC(C)CC(F)C(=O)NCC(C)CNC(=O)C=CC(=O)NC1CC1 N1(C(c2cnc(SC)nc2O)=O)CCC2C(C1)CN2C(c1ccsc1)=O C1(CNC(C(CC#C)C2CC2)=O)COCCN(C(c2cc(C)n(C)c2)=O)C1 CC1CCC=C1C(=O)NC1CCC(CNC(c2ncoc2C2CCC2)=O)CC1 C(=O)(C(Cn1cncn1)NC(c1nnsc1C)=O)NC(CC)C1CCC1 N1(C(C2C=CCN2Cc2ccc(N3CCCCC3)s2)=O)CC2CCCC2C1 C12(CNC(C(CC)(C)C)=O)CCC1CCN2C(=O)CCCc1cccs1 N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)Cc2ccnc(F)c2)C(CCO)C1 c1(CC(N2C(C3(O)CN(C(C(CC)SC)=O)C3)CCC2)=O)cc(Cl)ccc1Cl n1(CC#C)c(C)cc(C(=O)NC(C2CCOC2)CNC(c2cn(C)nn2)=O)c1C Cc1ccc(SCCC(=O)N2CC(CCNC(C3(C)CCCCO3)=O)C2)cc1 C1(NC(C(CCCC#C)C)=O)CC1C1CCN(C(=O)CCc2cnc(C)o2)CC1 c1(C(=O)NC2CCN(C(c3c(C)nc[nH]3)=O)C(C)C2)cc2cc[nH]c(=O)c2s1 c1(C(=O)Nc2cccc(NC(CCCC(CC)C)=O)c2)cnc2n1CCCCC2 c1(NCc2c(C(=O)OCC)scc2)ccc(-c2ncn(C)n2)cc1 c1(N2CCC(CCN(C)C)CC2)nc(Cl)nn2cccc12 C=CCC(C(=O)NCC1CC(CNC(c2cnc(N)cn2)=O)C1)NC(C)=O C(=O)(C1=NNC(=O)CC1)C(C)(C)CNC(=O)CNC(c1ncccn1)=O N1(C(C(=Cc2cccnc2)C)=O)CCC(NC(=O)C2=CCOCC2)C(C)C1 C(=O)(C1=CCCC1C)NC(c1cccc(C)c1)CNC(c1nnn(CC)c1C)=O C#Cc1cc(C(=O)NC2CCOCC2C)cc(I)c1 N1(C(c2c(CC)nco2)=O)CC(CNC(=O)C=Cc2ccc(C)o2)OC(C)(C)C1 c1(NC(C2N(C(c3nc(N(C)C)nc(O)c3)=O)CC2)=O)ccc([N+](=O)[O-])cc1Br C(=O)(C(C)(CNC(=O)C(C)CC(=O)OC)CC)N(CC=C)CCOC C1(C(=O)NCC2(CCNC(C=C(C)C)=O)CC2)CC2CC(C1)CC(F)(F)C2 C1(NC(c2ncc(C)cc2Cl)=O)C(C)(C)C(C(=O)OC(C)(C)C)C1(C)C C#CC1(O)CCN(C(=O)C(CO)NC(=O)C(CC(C)C)NC(C)=O)C1 c1(C(N2C(C3(NC(C(COC)O)=O)CC3)CCC2)=O)cc(N)ccc1Cl C(=O)(CCN(OC)C(=O)C(CNC(C1(C)CC(C)C1)=O)OC)OC C(=O)(C(C(C)(C)C)NC(N)=O)NCC(CNC(Cc1n(C)ncc1)=O)CO N1(C(c2cnc(CC)s2)=O)CCC(CNC(=O)CC(C)C2CCCC2)CC1 N1(C(CCn2c(C)ccc2C)=O)CCC(CNC(=O)C2=C(Cl)CC2)CC1C C1(C(=O)NCCC2CN(C(C=CC(=O)N(C)C)=O)C2)CCc2nnn(C)c2C1 c1(C(=O)OC(COC)Cc2ccccc2)cc(F)c2[nH]nnc2c1 C1(C(N2CC(n3ncc(C)c3)C2)=O)CN(C(C2C3CCC(F)C23)=O)CCN1C N1(C(C23CC(COC)(C2)C3)=O)CC2CC(NC(=O)Nc3nc(C)ccc3F)CC1C2 C(CC(F)(F)F)(c1ccccc1)NC(NCCc1onc(N(C)C)n1)=S N1(C(c2c(C(C)C)n(C)nc2)=O)CCN(C(C2CC(O)C2)=O)C2CCCCC12 c1(N2CC(CC)OC(CC)C2)ccc(S(=O)(=O)N(C)Cc2ncn(C)n2)cc1Cl CCCC(C(F)(F)F)NC(=O)C(CNC(=O)CN(CCOC)CC)CC C1(NC(C2N(C(CSCC=C)=O)C(C)CC2)=O)CC(O)CC(C)(C)C1 C1(OC)CN(C(C2CC(C)(C)CCO2)=O)C(C)(CNC(C2OC3CCC2C3)=O)C1 c1(OCCCC)ccc(-c2ccc(NC(c3nc[nH]n3)=O)cc2F)c(C)n1 c1(C(=O)NCCCC(C)NC(C2CCSC2)=O)ccccc1F C(=O)(C(C)(O)C(F)(F)F)N1CC(N(C(=O)C(c2cnn(C3CC3)c2)=O)C)C1 c1(C(N(C2CCN(C(C3CNC(=O)C3)=O)C2)CCC)=O)coc2c1CCCC2 N1(C(C(c2n(C)ccc2)=O)=O)CC2CC1CN2S(=O)(=O)Cc1ccc(F)cc1F C1(C(=O)NCC#CCNC(Cn2c(C)cc(C(F)(F)F)n2)=O)CCCC(=O)N1C C1(NC(c2c(CC)oc(C)c2)=O)CN(C(C2CC(n3cnnc3)C2)=O)CCC1F c1(N2CC(C)C(NC(=O)CCC(C)(C)F)CC2)nc(CC(F)(F)F)ccc1C#N c1(N(CCCCC)C)nc(=NCCc2ccccc2F)[nH]c2cc(OC)ccc12 NS(=O)(=O)CCC(=O)NCC1CC2CC2N1C(=O)CCc1ccc(C(F)F)cc1 C1(CCCCNC(C(C)(F)F)=O)CCN(C(c2csnc2Br)=O)CC1 c1(OC)ccc(-c2cc(C(=O)NCC3COC(C)(C)C3)no2)cc1 CN=S(C)(=O)CCNC(=O)NC1C=CC=CC=C1 C1(S(N)(=O)=O)(C(=O)NC2CCCC(NC(c3ccc(CCC)[nH]3)=O)C2)CCCC1 C(=O)(CCCS(N)(=O)=O)NCC(C1CC1)NC(c1cc(CSCC)on1)=O C1(NC(COC)C2(C)CC2)CCc2ccc(Br)cc2C1 C1(C#N)(C(N(CCCC(=O)NCCC2ON=C(C)C2)C)=O)CC1(C)C CN1CC(C(=O)NCC2CC2NC(=O)Cc2nncn2C)CC1=O C(=O)(C(=O)NNC(=O)c1ncc(Br)cn1)NC(c1ccc(SC)cc1)CO C1(C(N2CCC3(CCC3)C2)C(=O)NC2CCOC2)CCOC2(CCOCC2)C1 C(c1c(Cl)nc2sccn12)=CC(=O)NCC(CN(C(CCC(C)OCC)=O)C)O C=CCC(C)(C)C(=O)NCc1ccccc1CNC(=O)Cn1cc(C2CC2)cn1 C1(C(=O)NCc2ccc(C(N3CC(C(C)C)C3)=O)s2)CCN(C)C(=O)C1 c1(C(N(CCCNC(C2(CCCC)CC2)=O)C)=O)cnc2n1CC(C)CC2 c1(C(N2CCC(C(=O)NCCCOC(=N)O)(OC)C2)=O)cnc(O)cc1C C1(CNC(=O)CCF)CCCCN1C(c1csc(Cc2ccccc2)c1)=O C1(CCN(C(=O)C(C#N)C2CC2)C)CCCCN1C(c1cnns1)=O c1(C(=O)NCC(C)NC(c2onc3ccccc23)=O)c(Cl)ccc2c[nH]nc12 c1(CCCC)nc(C(=O)NCC=CCNC(C23CC(C2)C3)=O)cs1 C(CC)(C(=O)NCC=C)N(CC(=O)NCCSCC)CC#C C1(CCNC(c2c(CC)nns2)=O)CCCN(C(=O)CS(=O)CC)CC1 c1(OCC(=O)NCC(CNC(C(COC)C)=O)F)c(C)cc(Br)cc1Cl C(C(C)(C)C1=CCCC1)NC(c1n(CCCSCC)nnn1)(C)C(C)C c1(NC(N2C(c3n(CC)ncc3)C(C)(C)CCC2)=O)nc2ccc(O)nc2s1 C(=O)(C(F)C(C)(C)O)NCC(CC)NC(c1cccc(C2(C)CC2)c1)=O c1(CC(=O)NC(CNC(CCC=C=C)=O)(C)CC)cc(C)cc(F)c1 N1(CCCNC(CN(C(C)C)C)=O)CCC(NC(=O)Cc2cnns2)C1 Cc1cnc(N)c(C(=O)NCC2CN(C(c3nncn3C3CC3)=O)CC2C)c1 c1(C2C(C(N)=O)CCC2)ccc(NC(N2CC3CC2(c2ccsc2)C3)=O)cc1 c1(C(=O)NCC2(F)CCN(C(CCC(C)OC)=O)C2)c(C)c(C)cc(C)c1C N1(CC(=O)NCC2(C(C)NC(C(c3nc(C)sc3)=O)=O)CC2)CCN(C)CC1 c1(N2CC(C)CS(=O)CC2)nc(N2CCC3(CCC3)CC2)c2ncn(C)c2n1 c1(OC)nc(C(=O)NCCC2(NC(=O)CNS(N)(=O)=O)CCC2)cc(O)n1 C1(CN(C(=O)CCC2CCCC2)C)CCN(C(c2c[nH]nc2C2CC2)=O)C1 c1(C(N(C2CCCN(C(=O)Cc3ccc(Cl)cc3)C2)CC)=O)cncc(CO)c1 C#Cc1ccc(CC(=O)NC2C3CCN(C(c4ccn(CC)n4)=O)CCC23)cc1 C1(NC(CC2CC(OC)C2)=O)CCN(C(C2CCN(C)CC2)=O)CCC1(F)F c1(C(=O)NCC2N(C(C(CC3CC3)OC)=O)CC2)cccc2c1CCOC2 c1(CNC(c2nnc(Oc3ccccc3)s2)=O)cccc(O)c1[N+](=O)[O-] C1(CNC(c2cnn3c2OCC3)=O)CCCCN(C(=O)Cc2ccsc2)C1 C(CCCOC)(C(=O)N1CCOCC(O)C1)NC(C(F)=CCC)=O C#Cc1cccc(C(=O)NCC2CCCCC2NCc2cc(Br)cnc2OC)c1 CC(C)CC(CNC(c1cccnc1C(F)(F)F)=O)NC(C1CC(C)(C)C1)=O C=C=CCCC(=O)NC1(CNC(=O)C(Br)=C(C)C)CCOCC1 c1(C(=O)NC2CN(C(c3c(C(C)C)[nH]cc3)=O)CC2O)nn(C)c2c1CCC2 C1(C(=O)NCC(CO)OC)(NC(C=CC(CC)C)=O)CCOCC1 c1(C)nc(SC)cc(Cl)n1.C1(C)(C(N(CC(C)C)OCC)C)CC1 N1(C(C(CC)C)=O)CCC2CCN(C(c3ccc(-n4ccnc4)cc3C)=O)C2C1 c1(C(N2C3CN(C(CCCC#C)=O)C(C3)C2)=O)c(OC)ccc(F)c1F C1(C(CC)(C)C)CCC(C(=O)NCCNC(=O)C(C)NC(=O)CC(C)(C)C)CC1 c1(C(C(=O)NCCC2CCCN2C(=O)CCN2CCOCC2)O)ccccc1Cl C1(O)(CNC(C(C2CCC2)OCC)=O)CCN(C(C2CN(C3COC3)C2)=O)CC1 C1(C(=O)NC(C)Cc2cnn(C)c2)(CC)CCCN(C(c2ncccc2C)=O)C1 C12(C(N(CCC)CCNC(=O)C(c3ccccc3Cl)O)=O)CCCC1OCC2 CCCC(CCC)CC(=O)NCC1COCC1NC(=O)CCNS(C)(=O)=O C(C(=O)N=c1cc[nH]cc1)N(c1nnc(C(CC)(C)C)o1)C c1(C(N(CC(C)CNC(=O)C=Cc2ccncc2)C)=O)ccc(N(C)C)c(F)c1 c1(C(N2CC(NC(C(C)(C)OCC)=O)C3(C2)CC3)=O)c(Cl)cccc1[N+](=O)[O-] C(=O)(C1=CC2C=CC1C2)NC1(C2N(C(c3c(CC)cco3)=O)CCCC2)CC1 c1(C(C(=O)NCCC(=O)OCC)N(C2CCNC2=O)C)ncc(Cl)cc1F N1(CCC)CCCCC1C(=O)NCC(C(=O)NC(CO)C(=O)O)N(C)C c1(OC)c(C(=O)NC2CC(CNC(=O)CN(C)C)CC2O)c(C)nn1C N1(C(C(C)NC(CC)(C)C)=O)CC(C)C(C)(CNC(=O)C(C)C)C1 C1(CN(C)C(c2ccoc2C2CC2)=O)CN(C(c2cccc[n+]2[O-])=O)CC12CC2 N1(C(C(=O)Nc2scc(CNC(C(=O)NCC)=O)n2)=O)CCCC(C(=O)OC)C1 n1(CC(=O)NCC2N(C(C(CC)c3ccccc3)=O)CCC2)nc(C)n(C)c1=O C1(C(N2CCC(NC(Cc3c(C)ccs3)=O)C(F)C2)=O)CCc2c[nH]nc2C1 c1(CCC(N2CC(N(C)C(c3csnc3Cl)=O)C2)=O)nnc(S)nc1O c1(C(N2CC(C(C)NC(C3(O)CCCCC3)=O)OCC2)=O)ccnc2[nH]ncc12 c1(OC)ccc(N2CC(C(=O)NCC(F)C(C)(C)O)CC2=O)cc1 C1(n2cc(CCOCCOCCNC(C(CC)C)=O)nn2)CCN(C)C1=O.C1CO1 c1(CCC(=O)NC2(COC)CN(C(C3(O)CCOC3)=O)C2)c(Cl)cccc1Cl c1(C(C(=O)N(CCNC(C2CCN(C)C2C)=O)CC)(F)F)cc(Cl)ccc1OC Cc1cncc(CC(=O)N(C)CC2CN(C(c3cnc(N(C)C)s3)=O)C2)c1 C1(CC)CN(C(C2CCN(C)C(=O)C2)=O)CCN1C(=O)Cc1ccc(Cl)c(F)c1 C1(CC(N2C3CN(C(C4C(COC)C4)=O)C(C3)C2)=O)CCC2(CCC2)CO1 C(CO)(CN=c1ccc(S(=O)(=O)N(C)Cc2csc(Br)c2)c[nH]1)OC S(=O)(=O)(c1c[nH]c(C(=O)NCCCNC(C2COC(C)(C)CO2)=O)c1)N(C)C c1(C(N(C)CCC2CCN(C(C3CC3Br)=O)CC2)=O)cc2ccncc2[nH]1 CC1CN(C(c2cnn(C)c2-c2ccc(F)cc2F)=O)CC(C)C1(F)F Cn1cc(Cl)c(CC(=O)N(CC(F)F)CCC2CC2)n1 N1(c2ncc(C)cn2)CC2COCC2(C(=O)N(C2CC2)Cc2ccncc2)C1 Cc1cc(C(=O)NCCc2cc(C(=O)NC(c3ccnn3C)CO)no2)c(N)s1 N1(C(C(C)n2cnnn2)=O)CCN(C(=O)CC(C)C(F)F)C(c2ccnn2C)C1 Cc1cc(Cl)ccc1CNC(=O)C(=O)NCc1ccc(N2CCOCC2)c(F)c1 C1(NC(C(C)(F)F)=O)CN(C(=O)CS(N)(=O)=O)C2(CCCOC2)C1 CC1CC(C(N2CCC2CNC(=O)Cc2nn(C)cc2Cl)=O)CN1C N1(C(C2CCN(CC)C2)=O)CCC(C(=O)NCC2CC3CCCC3C2)=C(F)C1 N1(C(CCc2c(C)cccn2)=O)CCC2(C1)CN(C(C1(N(C)C)CCCOC1)=O)C2 CCC(CC(=O)N1CCCC(CNC(=O)CCC2CC2)C1)CC(F)(F)F C(=O)(C1=NOCC1)N1CC(C(C(N2CC=CCC2)=O)OC)C1 CC(C)(C)CC(O)CC(=O)NCCCCC(=O)N1CCC(N2CCCC2)C1 c1(C(C)Nc2ccc(-c3nc(=O)o[nH]3)cc2)ccc(O)cc1C N1(C(C2CCC(NC(c3ccc(C)s3)=O)CC2)=O)CCC(O)C(C)C1 N1(C(CC2(C)CNC(=O)C2)=O)CCOCC(C(=O)O)C1 C1(C(N2C(C3(C(=O)NCCc4c(C)n[nH]c4)CC3)CCC2)=O)OCCCC1(C)C CC1Cc2cc(C(N3CCNCC(CO)C3)=O)ccc2N1 Cc1nnc2n1CCCC2C(=O)NC1C2CC1N(C(c1ccc(F)c(O)c1)=O)C2 Cc1nccc(NCCCCC(C)NC(=O)C(C)OCCN(C)C)n1 c1(C(=O)NCCC2CCCCN2c2cc(C(F)F)ncn2)ccnc2[nH]cnc12 N1(C(CCc2ncc(C)[nH]2)=O)CC2CC(C1)N(C(C13CCN(CC1)C3)=O)C2 c1(OC)ccc(C(=O)NC2CC23CC(NC(=O)Cc2cncn2C)C3)c(O)c1F C12(NC(c3c(OC)ccnc3)=O)CCN(C(=O)Cn3nc(C)cc3C)CCC1C2 C=C(Cl)CCC(=O)NC(C1(O)CCCCC1)C(=O)NCC1CC1(C)C Cc1nc(CCC(=O)NCC2CCCN2C(c2ccc(C3CC3)cc2)=O)[nH]c1C C1(C)(C(=O)NCCC(CC)O)CCN(C(C2CC(CF)C2)=O)CC1 CC1C2CC(C2NC(C2CCCCC2(F)F)=O)N1C(=O)C=Cc1ccc[nH]1 N1(C(CC2CCN(C(C(C)OCOC)=O)C2)=O)CC2(CCOC2=O)C1 c1(N(CC#C)C(C)C)ncnc2c1ncn2CC(c1ccc(C)c(F)c1)O c1(OC(C(=O)NC(C2CC(NC(C=CC(C)C)=O)C2)C)C)cccc(Cl)c1 C(=O)(C1CCCc2n[nH]cc21)N1CC(CNC(c2c(C)nns2)=O)C(C)CC1 CC(C)(C)C(O)CC(=O)N1CCC(NC(=O)C(C)(O)C(F)(F)F)C1 CC1CCN(C(C2CC(N=[N+]=[N-])C2)=O)CCN1C(=O)CC1CCC(=O)N1 N1(C(CCC)=O)CC(O)(CNC(=O)Cc2csc(N3CCNC3=O)n2)C1 c1(C(=O)NCC2(C(=O)Nc3c(OC)cccn3)CC2)ccc2cccnc2c1 N1(C(C(C)C2CCC2)=O)CCS(=O)(=O)C(CCNC(c2cccc(O)n2)=O)C1 C1(C(=O)NCCN(C(C)C)C(c2cn(C)nc2C2CC2)=O)CCCOC1C N1(C(C(CC)N(C)C)=O)CC(C)(C)OCC1CNC(=O)C(C)(CC)CC Cc1cncnc1C(N1CC(CNC(C2(C)CS(=O)(=O)C2)=O)C(O)C1)=O c12cc(C#N)cnc1CC2.C1(F)(CNC(C(=O)NC)=O)CCCNC1 c1(C(=O)NCCN(C(c2ccn(C3CC3)n2)=O)CC)cnn2c1OCC(F)C2 C1(C(C(=O)N(C)CC2C3CN(C(c4c(C)scn4)=O)CC32)O)CCS(=O)(=O)CC1 C1(C)(CNC(C2C(C)CCO2)=O)CCC(NC(C2CC(F)(F)C2)=O)CC1 c1(C(=O)NCC2(CNC(C3C(C)(CC)C3)=O)CCCC2)c(Cl)ccc2c[nH]nc12 c1(C(N2C3CC(CC(NC(CCCOC)=O)C3)C2)=O)cc(O)nc2ccccc12 CC1CC(=O)NCCN1C(C1CN(C(=O)C=CC(F)(F)F)CCO1)=O C1(C(=O)NC2(CNC(C(C)(F)F)=O)CCOC2)C2CCCCC12 Cc1c(C=O)[nH]c2cc(C(=O)O)ccc12.N1(N2CCC2CO)CCC(C)C1 C12(CC(=O)NCC(C)(C3CC3)OC)CCC1CN(C(C1CCCN1C)=O)C2 O=C(C(C(F)(F)F)C(F)(F)F)NCCn1cc(-c2ccc(Cl)cc2)nn1 N12CC3(CCN(C3)CC3CN(C3)CC1=O)C2.c1(CC)cc(C(=O)OC)ccc1F C(=O)(C1=CCC(C)CC1)NCc1cc(OC)nc(N(C)C)n1 C1(C(N2CC(CNC(Cc3nc(C)[nH]n3)=O)C2)=O)CC2CCC1CC2(F)F N1(CCC)CCCC1C(=O)NCCCC1CCCN1C(=O)CC1CC1 C(C(F)(C(=O)N1CCC(O)CC(C)C1)C(C)C)NC(C1C(C)CC1)=O CC1(C)CCCCC1=CC(=O)NC1CCCC1NC(=O)COCP(C)(C)=O C1(CC(=O)NCc2ccc(Br)s2)COCCN1Cc1ccco1 C1(NC(=O)Cc2nccs2)CN(C(=O)CCn2cnnn2)CC2(CCC2)C1 N1(C(C2(CC)COC2)=O)CCN(C(=O)CC2CCC(C(F)(F)F)O2)CC1C c1(C(N2CC=CC(NC(C3CCCN3C3CC3)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 CC(C)C(O)CC(=O)NCC1CN(C(c2cncc(C(F)F)c2)=O)C1 c1(-c2nc(NC(c3cncc(-c4cc(SC)ncc4)c3)=O)sc2)ccc(F)c(C)c1 C(CC(C)C)(C(=O)NCc1cnn(CCO)c1)N(C(C(C(=O)OC)C)=O)C C(=O)(C1=C(C)CCOC1)N1CCC(NC(C=CC=CCC)=O)CC1C1CC1 CC1CC(C(=O)NCC2CCN(C(c3cnc(C(F)(F)F)cn3)=O)C2)CC(=O)N1 c1(C(=O)NC2CC(CNC(C34C(C)(C)OCC3C4)=O)C2)ccnc2ncccc12 c1(CC)c(C(=O)NC2(C)CN(C(=O)CN3CCC3C)C2)nnn1C C1(C2CC2)(OC)CN(C(=O)CCCCNC(c2coc(C(=O)OC)c2)=O)C1 c1(C(N2CCC(CNC(C(C)OCOC)=O)C2)=O)ccc(Cl)nc1OC c1(NC(CC2N(C(C(C)OCC=C)=O)CCOC2)=O)cnc(OC)c(C)c1 CCC(C)C(C(=O)N1CCOCC1CO)N(C(=O)Cc1nonc1C)C C(CC)(CCCC(=O)NC1(CN(C)C)CC1)NC(C(CC)NC(C)=O)=O N1(C(c2cn(CCC=C)nn2)=O)CC(NC(C2(C)CCCCC2)=O)CC(O)C1 C1(CC(=O)N(CCN(C(CC2(OC)CCC2)=O)C)C(C)C)CCCC(=O)N1 C(=O)(CC(CC)CCCC)N(CCC(=O)N(CC#C)CCO)CC1CC1 c1(CC)ncc(C(N2CC=CC(C(=O)NC3(C)CC=CCC3)C2)=O)cn1 Cc1cc(COc2cccc(C(F)F)n2)oc1-c1nc(COC(C)(C)C)no1 C1(NC(CC2(CO)CC(=O)NC2)=O)CN(C(C2CCC2)=O)CCC1C(F)(F)F N1(C(C(C=C)(C)C)=O)CCC(C2CC(NC(c3cnn(C(F)F)c3)=O)C2)C1 c1(C(=O)N(C)C)ccnc(F)c1OC.C(C(=O)NCC(O)CN)(C(C)O)NC(C)=O c1(N(c2cc(Cl)c([N+](=O)[O-])[nH]2)C(Cc2ccc(OC)cc2)=O)ccc(Cl)c(C#N)c1 C1(NC(C2CC(OC)(OC)C2)=O)CN(C(c2c(C3CC3)cnn2C)=O)CC1C C1(C2CCN(c3cc(C(C)C)ncn3)C2)(NC(C(CC)NC(C)=O)=O)CC1 C1(C#CC(=O)NC2CC(CNC(=O)CNC(c3cccs3)=O)C2)(CC)CC1 CCC(C)(F)C(=O)NC1CCN(C(=O)CCOc2ccc(SC)cc2)C1 N1(C(CCCCOC)=O)CCN(C(=O)C(C)(C)n2cccn2)CC1CF Cc1oc2ccccc2c1C(=O)NCC1(F)CC(NC(=O)CC(C)C(F)F)C1 N1(c2cncc(C(=O)OCC)n2)CCCC(C)(C(=O)OC)C1 CCC(CC(=O)N1CCN(C)C(C(=O)N(c2cccc(C)c2)CC)C1)C(C)C c1(CNCCC(=O)NC2(c3ccccc3)CCNC2)ccc(F)cc1 c1(C(N2C(C)(C(=O)Nc3cc(Br)ncc3F)CC2)=O)cc(F)c(Cl)c(C#N)c1Cl n1(CCOC)nnc2c(NC3CC(C(=O)NC4CN(C(C)=O)C4)C3)ncnc12 C1(=CN(CCSC(C)C)Oc2cccc(Br)c2)CCC(=O)N(C)C1 N1(C(=O)Nc2c(SC)cccc2)CC(N(C)Cc2ccnc(SC)c2)C2(CC2)C1 C#CCC(C)C(=O)NCC(C)NC(=O)CCCN1CCCC1 C(CCC(=O)NOCC1(c2ccc(F)c(F)c2)CCCC1)OCC=C c1(NC(=O)C(F)OC(F)(F)F)cnc(F)cc1C(=O)Nc1cccc(OC(C)C)c1 C1(CC(=O)NCC(C(CC)C)O)C2CCCC2N1C(C1(C(F)(F)F)CC1)=O c1(NC(C)CC(C)NC(c2coc(CC(C)C)n2)=O)nc(C(F)(F)F)ccc1C#N CC(c1ccsc1)=CC(=O)NCCCN(c1cc(C)on1)C(C)C C(c1c(Cl)cccc1Cl)=CC(=O)NC1C(N(C(CNC(=O)OC)=O)C)CCCC1 c1(C(N2C(C(N3CC(CC(C#C)C)C3)=O)CC2C)=O)cc(O)cc(C)c1 c1(CSCC(=O)NCC(CO)NC(=O)CC2CCCO2)ccccn1 Cc1nn(C)c(C)c1CC(=O)NCCNC(C1CC(N2CCCC(O)C2)C1)=O C1(O)(C(=O)OCC(C(=O)OC)OC(C)(C)C)CCN(C(=O)COC(C)=O)CC1 Cc1ccc(NC(N2CCC(O)(Cc3cccnc3)CC2)=O)cc1Cl C1(c2n(CC3(C)CCC3)nc(-c3ccoc3)n2)CCc2nc[nH]c2C1 CC#CCC(C(=O)NCC(C)C1CC1)NC(=O)C=CC1CCCN1C CC1(NC(c2n[nH]cc2Cl)=O)CCCCC1C(=O)NCC(O)C(N)=O c1(C(=O)NCCC2CCCN(C(c3n(C)ncc3Cl)=O)C2)cc(Cl)c(F)cc1N O(NC(=O)CCCCC(=O)NC1CN(C(=O)Cc2c[nH]nc2O)CC1C)C(C)C C1(C(=O)NCCCC2(N(C)C)CC2)CC(C(F)(F)F)CO1 c1(C(N(CCC)CCNC(c2nn(C)c(C)c2Cl)=O)=O)c(C)cc(C)cc1C N(C(=NCCn1nc(C)cc1C)NCC(C)(C)C)CCc1ccc(OCC)cc1 N(C1CCCc2n[nH]cc21)C(C(C1CN(C(C2(C)CCCS2)=O)C1)OC)=O c1(C(=O)OC)cc(S(=O)(=O)Nc2ccnc(Oc3ccccc3)c2)cc(F)c1F CCCC(C)C(=O)NCCN(C(c1cc(C(=O)OC)n[nH]1)=O)C1CC1 C(=O)(C(O)P(C)(C)=O)NCC(C)CNC(c1ccc(N(C)C)c(F)c1)=O Cc1n[nH]c(C)c1CC(=O)NC1(C(=O)NCCC(=O)N(C)C)CC(CO)C1 C1(C(N2CCN(C(c3ccn(C)n3)=O)C(C3CCC3)C2)=O)OC(C)(C)OC1(C)C C=CC1(CC(=O)NCC2(NC(=O)CN3CC=CC3)CCCCC2)CCCCC1 N1(C(CN(C(c2cc[nH]c2)=O)CC)=O)CCC12CCCSC2 C1(C(N2CCC(CC#C)CC2)=O)CN(C)CCN1C(=O)C(C)C(F)F c1(C(N2CCN(C(C(N)=O)=O)C3C2C3)=O)ccc2c(Br)cccc2c1 N1(C(c2c(OC)cccc2C)=O)CC(C)CN(c2nnc(C(C)C)o2)C(C)C1 N1(C(C(C2CCCC2)OCC)C(=O)NC2COC2)CCC(F)(COC)CC1 N1(C(C)C)CC(NC(=O)CCCc2cccnc2)CCC1=O c1(C(N(CCCNC(C2(C)CCCNC2=O)=O)C)=O)cn(CCO)c(=O)nc1O C1(COC)CC(CNC(c2cn(CCCF)nn2)=O)N(C(c2coc(C)n2)=O)C1 C(=O)(C(C)(C)CCNC(c1ccc(OC)nn1)=O)NCC1(C#C)CCC1 C1(N(C(CN2C(C)CCC2)=O)C)CCCN(C(c2nnsc2C(F)F)=O)C1 N1(CCC(=O)NC2CC(CNC(C=C(CC)C)=O)C2)CCC(F)C1 C(N=c1[nH]c2ncc(Br)cc2o1)c1cc(OC)cc(Cl)c1 CC(CNC(=O)COc1cccc(F)c1)(Cn1cccn1)N=c1[nH]nco1 c1(C(=O)NCC2C(CNC(c3c(C)nn(C)c3)=O)C2)cccc(Cl)c1N n1(CCC)cc(C(=O)NC2(CCO)CN(C(c3ccoc3)=O)C2)c2ccccc12 C1(N(C(C=CCOC)=O)C)CCCN(C(=O)CC(C)(C)OC)CC1 C(CN=c1[nH]c(=N)[nH]c(=NC2c3ccccc3CC2C)[nH]1)C1COCC(C)O1 c1(CNC(c2c(F)cccc2I)=O)ccc(Cl)c(Br)c1 CC1(C)CN(C(c2ccccc2)C(=O)NC2COC2)C12CCC2 c1(OC)ccc(CC(=O)NC2CCCN(C(=O)Cc3cccc(Cl)c3)C2)cc1C CCC(CCOC)C(=O)NCCCONC(=O)Cc1c(C)ncnc1C C(CCCOCCNC(=O)Cc1ccc(Cl)s1)NC(CC1(CC)CCC1)=O C(=O)(CCc1ncc[nH]1)NCCN(C(C1CC1(C)C(F)F)=O)CC N1(C(CC(CC)C(C)C)=O)CCC2C(CCCN2C(=O)Cn2cccc2)C1 C1(C(N(CC(O)CO)CC)=O)CCN(C(=O)CC2(COC)CC2)C1 C12(OC)CCN(C1)C(=O)N2.c1(SCOC)ccc(F)cc1.C12(CCC1)NC2 c1(CC(=O)N(CCCCNC(C2(C)CC(O)CN2C)=O)C)n[nH]c2ccccc12 Cc1occc1CC(=O)NC1CN(C(C2CCN(c3nc(=N)[nH][nH]3)C2)=O)C1 C1(CCC#C)CCN(C(C2CC(NC(=O)C(CC=C)OC(C)=O)C(O)C2)=O)CC1 CCCC(C)CC(=O)N1CC(F)CC1C(=O)N(C)CCC1CCCCC1 CC(C(=O)N1CCCC(CCNC(C2CCCN2C(=O)C(F)(F)F)=O)C1)C(C)O C1(C)(C(=O)NC(CN(C(=O)CNC(c2ccncc2)=O)CC)C)CC2CCC(C1)S2 N1(C(C2OCCC(NC(C(F)=C(C)C)=O)C2)=O)CC2CCCC(O)C2C1 c1(OC(C(=O)NCC(CNC(=O)C2=CCCC2)OC)F)ccc(Cl)c(F)c1 C1(OC(c2cccc3cncn23)=O)CCC2(CCCOC2)C1 c1(-c2cncc(CC)c2)ccc2c(C(=O)Nc3cc(Cl)nn3C)cnn2c1 N1(CCN(C2CCCC2F)C(=O)NC(CC)(C2CC2)C2CC2)CCCOCC1 c1(OC)cccnc1C(=O)NCC1(C(C)N(C(=O)Cc2cc(C)on2)C2CC2)CC1 c1(OC)cccc(CC(F)C(=O)NC(=O)C(=O)Nc2ccccc2C(C)(C)C)c1 C1(C(N(CCC(=O)OC)CC(=O)OCC)=O)CC2(CCC2OC)C1 n1(CC(=O)NC(COC)C)cc(CNCc2cscn2)nn1 C1(NC(C(C(C)C)F)=O)CCN(C(c2ccc(O)cc2)=O)CC1CO C=C(C)CCC(=O)N1CCCC(N(C(=O)Cc2csc(-c3ccc(C)o3)n2)C)C1 c1(C(=O)NCC=CCNC(C2(C)CCCS2(=O)=O)=O)cc2c(s1)CCOC2 CCCCC(C)CC(=O)NC(c1ccc(OC)cc1)CNC(=O)COCC CC(c1ccccc1)=CC(=O)N(CCCOCCNC(=O)C1=CCC1)C Cc1nc(C(=O)NCC2(NC(=O)C=CC3CCOC3)CCC2)c(C)s1 CC(CCC(=O)N1CC2CC2(NC(=O)C(CCC=O)OC(C)(C)C)C1)N(C)C C1(NC(CCOCCCOC)=O)CCCCN(C(c2n[nH]c(=N)s2)=O)C1 Cc1nccc(C(=O)NCCC(C(C)C)NC(=O)C=Cc2ccco2)n1 N#Cc1cn[nH]c1C(=O)NCC1(C(N)=O)CN(C(=O)Cc2ccccn2)C1 Cn1cc(C2=NOC(C(N3CC(NC(C4CSCCS4)=O)C(C)(C)C3)=O)C2)cn1 CC1(C)CC(=O)N(CC(=O)NC2CCC(NC(c3ncccn3)=O)C2)C1=O N1(C(C=CCOC(C)(C)C)=O)CC2C(CNC(=O)C(Cl)=CCl)C2C1 c1(C(N2CC(CNC(C3CCC(F)(F)C3)=O)C2)=O)cnn2c1SCC2 C1(F)(CNC(C(C)(F)c2ccccc2)=O)CCN(C(=O)CCc2ccon2)CC1 N1(C(C2OCC(C)C2)=O)CCCC2(CC(NC(=O)CCC3CC(C)(C)CO3)C2)C1 N1(C(CCC#C)=O)CCCCC1CNC(=O)CCCC1CCOCC1 n1(CC=C)cc(C(=O)NCC2(CCNC(c3nocc3CC)=O)CC2)cn1 CCC1=C(C(=O)NC2(C)CC(NC(c3c(F)cncc3Br)=O)C2)CCCO1 C(=O)(CC(C)(C)CC)N(CC(=O)NC(CCN(CC)CC)C)CC CC(O)CC(=O)OC(C)(C)C.C(=O)(CC(C)C1CCCCC1)N1CC(C)CC1=O C(CCc1ccccc1)(C(=O)O)NC(CCN(CCO)CCCCC#CC)=O N1(C(C2(CC#C)CCCCC2)=O)C2CCC1C(CNC(C1CC(OCC)C1)=O)C2 c1(OC)cc(C)nc(NC(C)=O)n1.c12ccc(c(C)c1)N(C1CNCC1(F)F)C2 N1(C(=O)Cc2ccc(O)cc2)CCN(C(c2cscn2)=O)C2CC12 C(CS(=O)(=O)c1ccc(Br)cc1)NC(N(C)Cc1cnsn1)=O C(=O)(CC1CCc2ccc(O)cc21)NC1CCN(C(C(C)N2CCC2)=O)C1 C(CC1=CCC2CC1C2(C)C)NC(=NCc1c(C=C)cccc1)NC1CC1C C1(CNC(=NCC=C)NCC2CCCO2)Cc2ccccc2O1 N1(C(=O)CCBr)CCOCC2(C1)CN(C(c1cc3ccoc3cn1)=O)CCCO2 CC1(C)C(C(=O)NCC23CCC(NC(=O)CC4(O)CCOC4)(CO2)C3)CC1(F)F N1(C(C(CC)CC2CCCCC2)=O)CC2(CCN(C(=O)C(F)=CC3CC3)CC2)C1 Cn1ncc(S(=O)(=O)N2CCC(Nc3ccc(Br)cc3)CC2)c1F c1(CN(C2(C(N(C3(c4nn[nH]n4)CC3)C)=O)CCC2)C2CC2)cc(C#N)ccc1N C1(NC(c2c[nH]c(=N)o2)=O)CN(C(=O)CN2CCCCC2)CCC1CO C1(NC(CCC2C(C)(C)C2)=O)CN(c2ncc([N+](=O)[O-])cc2F)CCC12CCC2 c1(C(N2CC3(C2)CN(C(C2CCCS2)=O)CCO3)=O)cnc(O)c2ccccc12 CCCC(C(=O)N(C1CC(CCn2cc(-c3ccsc3)nn2)C1)CC)S(N)(=O)=O C(=O)(CCC(C)(C)C)N1C(C2(CNC(C=CC)=O)CCOCC2)CCCC1 c1(C(N2C(CC)CN(C(C3(CC(=O)OC)CC3)=O)CC2)=O)cc(C)c(Cl)cc1F N1(C(c2csc(C)c2C)=O)CCC(CCNC(c2nocc2Cl)=O)CC1C C1(C(N(C)Cc2c(C)noc2C)=O)CN(C(c2cc(C)n(C)c2C)=O)CC1(F)F c1(C(N(C2CCN(C(=O)COC3CCOC3)CC2)CC)=O)cc2cnn(C)c2s1 CC(C)C(C(=O)NC(C1CCCN(C(=O)Cc2ccc(O)cc2)C1)C)C(C)C Cc1c(-c2nc(CCN(C)C)nn2-c2ccc(F)nc2)nn2c1CCCC2 c1(C(N2CCCCC(SC)C2)C(=O)NCC(F)F)cc2n(n1)CCCO2 c1(C(C)=O)ccc(C(=O)NC(CNC(C2CC(=O)N(C)C2)=O)C(C)C)c(F)c1 C1(N(C(COCCC=C)=O)CC)CCCN(C(c2sccc2C(=O)OCC)=O)C1 N1(C(CCN(C)CC)=O)CCCC(CNC(=O)CC(C)F)C1 c1(C(=O)NCC(CCC)NC(c2sc(O)nc2C)=O)cnn2cccc2c1 c1(C(=O)Nc2n(CC)nnn2)csc(=NCc2ccncc2OC)[nH]1 C1(NC(c2c(CC)cco2)=O)CCCC2CN(C(=O)CC3CCCOCC3)CC12 c1(C(=O)NC(c2cccc(Cl)n2)CC)cccc(Cc2cccnc2)c1 C1(N(C)C(C2CC2C(F)(F)F)=O)CCN(Cc2cccs2)CC1 C1(C(N2C3C(NC(Cc4c(C)occ4)=O)CC(C3)C2)=O)CN(S(=O)(=O)N(C)C)C1 N1(C(c2c(C)sc(Cl)n2)=O)CCC(C)N(C(C23CCCC2(C(N)=O)C3)=O)CC1 c1(CNC(Cc2c(C)non2)=O)cc(O)nc(CNC(C2C(C)CC2C)=O)n1 N1(C(c2c(CC)nn[nH]2)=O)CCN(C(=O)C(O)C2CCC2)CC1c1ncc[nH]1 N1(c2c(C)c(NC3CN4CCC3CC4)ncn2)CC2(C)CN(C)CC2(C)C1 Cc1ccncc1CC(=O)N(CCCNC(c1ocnc1C1CC1)=O)CCO N1(C(C2(C)CC2(F)Cl)=O)CCOC(CNC(C2COCC2C(N)=O)=O)C1 C(=O)(C(F)(F)C(C)O)NCC(C)NC(c1ccn(-c2cccnc2)n1)=O CCCC(CC)C(C(=O)NCCSC)N1CCCC(C(F)(F)F)CC1 N1(C(c2c(F)ccc(C)c2F)=O)CC2CCC(NC(=O)CC(=O)N(C)C)CC2C1 c1(N2CC(OC)(CNC(C3(SC)CCCC3C)=O)C2)ncc(C)cc1[N+](=O)[O-] Cc1cn2cc(C(=O)NC3COCC3NC(=O)CSc3ccccc3)sc2n1 C1(CC)CCN(C(=O)CC23CCC(CC2)C3)C1C(=O)NCC1CNC(=O)O1 CCCC(CC)C(=O)N1CC(NC(=O)C2=C(Cl)CC2)C(C)C1 CCCCCCC(CC)C(=O)N1CC2CCC2(CNC(c2cc(OC)cs2)=O)C1 C1(C(=O)NCc2nc(CC)on2)(CC)CCCN(C(C2CC(=O)NC2(C)C)=O)C1 c1(CC(=O)NCC(C2CCC2)NC(CN(CC(=O)NC(C)C)C)=O)ccns1 CC(CCN=c1[nH]nco1)NC(C1(c2cc(Cl)ccc2F)CCC1)=O Cc1cc(N(C)C)ccc1C(=O)NC1CCCC2CC2C1 C1(C(=O)NC(C(C)NC(c2cn(CC)nn2)=O)(C)C)CN(C)C(=O)N1 C1(C(C)NC(C(c2ccccc2)OC)=O)CCN(C(=O)C=Cc2cc[nH]n2)C1 c1(C(N2CC(F)(CNC(COC3(C)CCC3)=O)C2)=O)sc(=N)[nH]c1C(F)F C(CCCN=C(NC1CCCCC1)NC1CCN(C2CC2)CC1)OCC(F)(F)F C1(NC(c2cc3cccnc3s2)=O)C2COCC1CN(C(c1coc(O)n1)=O)C2 C1(C(=O)NCC2CCCC(C#C)C2)C2CC(C(O)C2O)S1(=O)=O N1(C(=O)NC(c2ccn(CC)n2)C)CCC(NC(=O)OC)CC1 c1(OC)ccc2c(c1)CCC(C(=O)NC1CCC(C(=O)Nc3cncnc3)C1)C2 N1(C(c2c(OC)noc2C)=O)CC(N(C)C(C2CC2(C)C)=O)C(C)(C)C1 c1(CC)nn(C)cc1C(=O)NCC1CN(C(=O)CCCc2ccsc2)CC1CC Cn1c(NCC2CCN(C(c3ccc4cccnc4c3)=O)C2)cc(=O)n(C)c1=O CCCCCCC(=O)NC1CC(CCNC(c2ccn(C3CC3(F)F)n2)=O)C1 C=CCCCCCCCCC(=O)NCCN(C(=O)CC1OCCC1C)CCOC C1(CNC(C2(C(=O)NC)CC2)=O)CCCCC1NC(=O)Cc1ccc(Cl)cn1 C1(NC(C(C)c2ccco2)=O)CN(C(C2CCN(C)CC2)=O)C2(CCCC2)C1 C(=O)(C#CC1CCOC1)NCCC(C)(C)NC(c1noc(CC)c1C)=O C(=O)(C(CC(C)C)Oc1cncc(Cl)c1)OC1(CCCC)CC1 C1(C(N(CC(=O)NC(C(C)C)CN(C)C)C)=O)CCCC(C#N)C1 C1(CNC(C23OCC(CC)(C2)C3)=O)CCN(C(c2cn(C(C)C)nn2)=O)C1(C)C C1(C(N2C(CCC(=O)N(CCCF)C)CCC2)=O)(CO)CC(C)(C)C1 N1(C(C(=O)NC2CCCCOC2)=O)CC=C(c2ccccc2Cl)CC1 C#CCCCCC(=O)NC(C1CCN(C(=O)C(C)(C)C)CC1)CO c1(C(N2CCCC(N(C(=O)C=C(C3CC3)C3CC3)C)C2)=O)ccc2cc[nH]c2n1 C1(N(C)C(c2cc(CF)on2)=O)CCCC(NC(c2ccsc2Cl)=O)C1 c12ccc(cc1)CC1CC(OC1)CNC(=O)C2.C1(C(N)=O)(C(=O)NC2CC2)CC1 N#Cc1ncn(CC(=O)N(Cc2ccccc2)Cc2nncs2)n1 C(=O)(C(C)CC(N)=O)N1CC2C(CNC(C3(CC=C)CC=CC3)=O)(C2)C1 CCCC(C#N)C(=O)N1CCOCC(NC(c2cnn(CC3CC3)c2)=O)C1 C1(N(C(C(F)OC)=O)C)CCCC1(C)CNC(=O)CCc1cnc(C2CC2)o1 N1(C(C(CC)(C)O)=O)CC2(CCN(C(=O)C(O)Cc3cn(C)cn3)C2)C1 C#CC1(O)CC(C(N2CC(C)(CCC(=O)NCC3COCC(C)O3)C2)=O)C1 S(=O)(=O)(CC(F)(F)F)Nc1nc(C)c(C(=O)OC(C)C)s1 CCC(C)CN=c1[nH]c(N2CCN(CC(F)F)C(C)C2)nc2cc[nH]c12 N1(C(C(C(C)C)C)=O)CCN(C(=O)CC2CCCC23CC3)C(c2ncc[nH]2)C1 C1(C(=O)NCC2OCCN(C(c3on(C)c(=O)c3)=O)C2)COc2ccccc2C1 Cc1cc(N2CC(F)CC2CNC(C2(C(C)C)CC2)=O)ncc1C#N C(=O)(CC(F)(F)C(F)(F)F)NCCC1CCN(C(c2c(N)ccc(OC)c2)=O)C1 C(=O)(C1CCCc2sc(=N)[nH]c21)N1C(CNC(C(C)(C)SC)=O)C(C)(C)CCC1 C(C)(C(=O)NCCN(C(=O)C(C)NC(=O)Cn1cnnn1)C1CC1)OC c1(CC)ccc(NC(C2CCN(C(c3ccnnc3O)=O)C2)=O)cn1 c1(N(C)C)ccc(CCC(=O)NCC2(C)CCCN2C(=O)CCS(C)=O)cn1 c1(OCC)cc(N(C)CCNC(=O)NCCC(C)(C)C)cc(Br)c1 C1(CNC(C(CC)OCC)=O)C(C)CCCN1C(c1cnc(CC)nc1C)=O N1(C(CC(OCC)OCC)=O)CCC(NC(=O)C=CCN(C)C)C(C)C1 c1(C2(CN3C(COC)C=CC3)CC2)cccc(CN)c1 c1(C(=O)NC(CCSC)C(=O)NCC(C)(CC)C(C)O)cc(C)nc(C)c1 c1(C(=O)NCCCn2cc(CNC(C)=O)nn2)ccc2c(c1)N(C)C(=O)C2 C1(NC(C(C)(C)n2cncn2)=O)CC2CC1CN(C(C1CC1F)=O)C2 Cc1cc(Cl)ccc1CC(N1CCN(C(=O)CC2CCC(=O)N2)C(C(C)C)C1)=O c1(CCC2CCN(CC3C(CC)C3)CC2)nccc(C#N)c1[N+](=O)[O-] C(=O)(CC(C)C(C)C)N(CCC)CCNC(=O)CCc1cc(Br)cs1 N1(C(CNC(Cc2c(C)[nH]cc2)=O)=O)CCN(C(=O)C=C2CCCC2)CC1 N1(C(C2(N(C(=O)Cc3cnn(C)c3)C)CC2)=O)CCCC(F)CC1 CC1(C)CN(C(=O)C2CC2)CC2(CN(C(c3ccc(-c4ccccc4)o3)=O)C2)O1 c1(NC(N2C(NC(Cc3c(C)noc3)=O)C(C)CC2)=O)ccc(F)nc1F c1(C(N2CC(NC(c3cn(C)nc3)=O)C2)=O)cnc(C#N)s1 N1(C(c2n(C)ncc2)=O)CCC12CN(C(c1ccccc1C(C)(F)F)=O)C2 C(=O)(C1=NOC2(CCC2)C1)NC(C(=O)N1CC(C(CC)CC)C1)CC(C)(C)C CCCC(C(=O)NC1C=CCN(C(c2cc(CF)on2)=O)C1)C(C)C C(c1ccc(O)c(O)c1)=CC(=O)NCC(C)CNC(c1cscc1Cl)=O c1(C(N2C(C(=O)NCC3CC3)CC2)=O)cccnc1C(F)F C12CN(CC1O)C(=O)c1cn2nn1.C1(C(=O)N(CCN(C)C)C2CC2)CCC2(CC2)C1 C(=O)(CC(C)(O)c1ccccc1)NC(CC)CNC(c1ccsc1Cl)=O C1(C(=O)NCC2C=CC(NC(C3C(Cl)(Cl)C34CC4)=O)C2)(OC)CCSCC1 c1(C=O)cc[nH]c2nccc1-2.C1(C(=O)NC)C=CC(NC(c2occc2CO)=O)C1 C1(C2CC2)(C(=O)NC(CN(C(Cc2c(C)scc2)=O)C)C)CC=CC1 c1(C(=O)OC)cnn2c1CN(C(c1ccc3c(c1)ncn3C)C(=O)NC(C)C)CC2 Cc1nc(C(=O)NC(C)C2CC2)ccc1-c1ccnc(N2CCNCC2)c1 CCC(C(=O)N(CC(C)(C)CNC(=O)CNc1ccc(C#N)cc1)C)C(F)(F)F N1(C(c2c(C)nsc2)=O)CC(NC(c2csc(Br)c2)=O)C(C)C1 Cn1cnc2nc(N3CCC(CCO)C3)nc(N3CC=CCC3)c12 N1(C(=O)C(O)c2ccco2)CC(C(N2CCOCC2C2CCC2)=O)C(F)(F)C1 N1(C(C2C(CC)CN(C(=O)CCC3CCCN3C)C2)=O)CCNC(=O)CC1C N1(C(c2cn(CC)nc2)=O)CCC(C(=O)NC2CC(N3CCCC3)C2)=C(F)C1 N1(C(C(CC)N(CC(=O)O)C(C)=O)=O)CC2CC2(C)C1.C(c1ccco1)=C(C)C#N C1(NC(c2n(CC)ncn2)=O)CC2CC1CN(C(=O)CCc1ccccc1F)C2 c1(C(N2C(CNC(=O)Cc3ccno3)COCC2)=O)cncc2nc[nH]c12 c1(C(=O)NC2CC(CCC(=O)NCC(C)N(CC)CC)C2)ccc(CSC)o1 C1(C(=O)NC(CC)(CNC(c2cc(C)nnc2O)=O)CC)CC2COCC(C1)C2 C1(NC(C2CCOCC2)=O)CC=CCC1C(=O)NC1CC(O)C(O)C1 N1(C(c2cnc(OC)nc2)=O)CCN(C(=O)CCCCCO)C(C2CC2)C1 c1(C(N2CCC(NC(c3cnc(C)o3)=O)C(F)C2)=O)cncc2ccc(F)cc12 C1(CNC(CC(C)C)=O)CCC(C)(C)CN1C(=O)CCC1CC(C)(C)CO1 Cc1cnc(C(N2CCC(C(N3CC(CO)C3)=O)C2C)=O)cn1 c1(C(=O)NC2CN(C(c3[nH]cc(C)c3)=O)C2)cnn(CC(C)C)c1C C12(C(N3CCC(SC)C3)=O)CCCC1CCN2C(c1cc(C)c[nH]1)=O C1(CC=C)(NC(=O)C(O)C=C)CCCN(C(=O)CCc2cncs2)C1 C(=O)(C1(C)CCCc2ccccc21)NCC1C(NC(c2c(CC)c[nH]c2)=O)CC1 N1(C(C(CCC)CC2CCCC2)=O)CCC(C)(C)C(NC(c2ccc(F)s2)=O)C1 c1(C(N(CC(O)CNC(C2(C)CCCS2(=O)=O)=O)C)=O)c(F)ccc2[nH]ccc12 c1(C(=O)NCC2C(NC(CC(C)F)=O)CCC2)ccccc1C#N C12=NC(=NCCCC(C)NC1=O)SN2.C1(N2CC(CC)C2)CCCCC1 c1(CC=C)ccccc1C(=O)NCC(C)CN(C)C(C1(C)CCN(C)C1)=O CC1CCN(C(=O)CN(C)C)CCN1C(C1CC1c1cccs1)=O C(CCCCCNC(=O)C(F)(F)c1ccncc1)N(C)C(C12CCC1C2)=O C(CC(C(=O)N(C)CC1CN(C(c2cc(C)[nH]n2)=O)C1)OC)OC C1(C(=O)O)CC2(CCCC2)CCN1S(=O)(=O)CC1CCCS(=O)(=O)C1 CC(C)C(C)C(C)CC(=O)N(CCCN(C(=O)C=Cc1ccc(F)cc1Cl)C)C c1(C(N2CCSC(CC)C2)C(=O)NCC(=C)C)ccc(C(F)F)c(F)c1 N1(C(c2nnn(C)n2)=O)C2CCCC1CN(C(=O)CCN1CCC1)C2 C(=O)(CS(=O)(=O)CC(C)C)NC(CCNC(C1(c2c(C)ccc(F)c2)CC1)=O)C c1(NC)ccccc1C(N1C(C(N2CCCCC2C2CCC2)=O)CC1C)=O c1(C(N2CC(NC(C(CSC)C)=O)C(O)C2)=O)ccc2nc[nH]c2c1 C(=O)(C1=CN=C2N=CNN2C1)N1CCOCC(NC(c2coc(C(F)F)c2)=O)C1 C1(CNC(CC(CC)(F)F)=O)CC2CCC(C1)N2C(C1COC(C)(C)C1)=O c12ccc(s1)C(=O)C(=O)NC(C1CCC1)CNC2=O.C1(C(F)F)(CC)CC1 C(CC(F)(F)CO)N(C(=O)CC1CC(NC(c2cnsn2)=O)C1)C C1(C(N(C2CN(C(C(CC=C)NC(C)=O)=O)C2)C)=O)CCN(S(=O)(=O)NC)CC1 CC1CC(C(N2CCN(c3nnc(-c4ccccc4)o3)CC2C)=O)CC(C)C1 c1(C(=O)NCC(=C)CCNC(=O)Cn2nccn2)cnncc1O C(=O)(C1CCCc2ccccc21)N1CCC(NC(=O)CN2CCS(=O)(=O)CC2)C1 N1(CCNC(C(CC)OC)=O)CCC(NC(=O)C(C2(O)CCCCC2)(F)F)CC1 N1(C(C2C(C)(C)COCC2)=O)CC2CCN(C(c3cnncc3O)=O)CC(C2)C1 CCC(CC(=O)N1CC2CC2(CNC(C2(COC)CCOCC2)=O)C1)OC C1(CCOC)(C(=O)NCCCC2(NC(C3CSC3)=O)CC2)CCC1 C1(N(C(=O)C(F)=CC2CC2)C)CCN(C(c2cn(C(C)(C)C)nn2)=O)C1 C1(NC(CCC#C)=O)CN(C(=O)Cc2cncc(Br)c2)CCC12CCC2 c1(C(=O)NCC(C)NC(c2ccnnc2S)=O)ccc(-c2ccon2)cc1 C1(NC(C2(CC)CCC2)=O)CCC2(CC1)CCN(C(=O)CN(C)CC)C2 Cc1ccnc2sc(C(=O)NC3CN(C(=O)Cc4ccno4)CC3(C)C)c(C)c12 C1(C2(O)CCOCC2)(CN2CC3(CN(C(C(C)(C)c4cnsc4)=O)C3)C2)CCC1 c1(C(N(CC(CNC(c2ccc(C=C)cc2)=O)O)C)=O)cc(F)cc2ccoc12 N1(C(c2cc(SC)c(N)cc2)=O)CC2CC(NC(C3(C(C)C)CCC3)=O)C(C2)C1 C(C(C(F)(F)F)NC(c1nc(-c2cccc(C(F)(F)C(F)F)c2)no1)=O)N(C)C C1(C(=O)NC2CN(C(c3n(C=C)ncc3)=O)CC2C)Cc2ccc(OC)nc2N1 c1(C(=O)OC)cc(=NCCCC(C)(C)NC(=O)CCc2ncc(F)cn2)[nH]cn1 C1(Cl)(NC2CCN(C(C3CN(C(C4C=CCS4)=O)C3)=O)CC2)CC2CCC1O2 N1(C(CC(CC)C)=O)CC2(C1)CN(c1nc(C3CCCC3)nc(=N)[nH]1)C2 Cc1cccc(C(=O)NC2CCCN(C(C3CCCO3)=O)C2)c1Br C1(C(N(C)CC2CC(NC(C(CSC)O)=O)C2)=O)OCCC1(C)C C1(NC(C2C(C=C)CC2)=O)CC(CNC(=O)C(CO)N(C)C)CC1O c1(C(=O)NC(CCNC(C=Cc2scc(C)n2)=O)C)ccc(F)c2ncccc12 Cc1ccccc1C(C)C(=O)NC1(CCNC(=O)CN2CCSCC2)CCC1 C1(CN(C(=O)CCOC2CN(C(c3ccnc(S)c3)=O)C2)C)CCCC2(CCC2)O1 C(=O)(CCC(=O)N(CC(N1CCC(CF)C1)=O)CCOC)NCCC N1(CCCSC)CCCC1C(C)NC(C(=O)N(CCCOC)C)=O C1(c2n(CCSC)nnn2)(NCc2c(C)cccc2Cl)CC(C)N(C)C1 c1(OC)c(C)cnc(CC(N2CC(CCn3cc(C4(O)CCC4)nn3)C2)=O)c1C C(CC(C(=O)NC1CC1CC(C)(C)C)NC(=O)C(C(C)C)OC)OCC CCC(C(=O)N1CCC(CNC(=O)CCCSC)(COC)C1)C(C)(C)CC N1(C(CC)=O)CC2CC2(NC(=O)C(CCN)NC(c2ccccc2)COCC)C1 c1(C(=O)NCCCNC(CCCCN(C(C)=O)C)=O)nc(C)c(N)cc1C CC1(C)CC(NC(c2csnn2)=O)CN(C(C2COC3(CO)CC2C3)=O)C1 N1(C(C2(C)CCN(C(C3CC(=C)C3)=O)C2)=O)CCC2(C=CCO2)C1 C(=O)(N=c1[nH]onc1C1CC1)C1(C)CCN(Cc2c(C)nn(C)c2)C1 c1(NC(C(CC#C)NC(c2ccc(C)o2)=O)=O)c(C)ncnc1C NC(=O)CCC(C(=O)N1CCN(C(C2OCCO2)=O)CC1)n1cc(CCCO)nn1 c1(C(=O)NC2(CC=C)CN(C(c3csc(CO)n3)=O)C2)cncc(OC(C)C)c1 c1(C(N2CCN(C(Cc3c(C)cco3)=O)C(C)C2C)=O)oc2ccccc2c1C N1(C(C(C)SC)=O)CC2CCC2(CNC(c2sc(Cl)c(Cl)c2C)=O)C1 C1(NC(c2c(CC)n(C)nn2)=O)CCC2(CCN(C(c3cscc3C)=O)C2)C1 N1(CCNC(=O)CC2CSC2)CCC(NC(C23CC(CC(F)F)(C2)C3)=O)CC1 C1(C(N2CCCC(C(N)=O)C2)=O)(CC)CCN(C(C2CCSCC2)=O)C1 O=C1NCCC2CCN(C(=O)CC3CN(C(C4(F)CCOC4)=O)CC34CC4)C12 c1(CC2C(NC(C3CCN(C(C45CC(F)(C4)C5)=O)CC3)=O)CC2)ccc(O)cc1 CCCCC(CC)CC(=O)N1CCN(C(=O)C(C)=C2CCCC2)CC1C1CCC1 c1(C(=O)NCCN(C(C(C)OCC#C)=O)C2CCCC2)cc(F)c(C#N)c(F)c1 C(=O)(C1CCCn2cncc21)N1CCN(C(C(C(C)O)(C)C)=O)CC1C C1(CNC(C(C=C)(C)C)=O)COCCN(C(c2csc(C(F)F)n2)=O)C1 c1(OC)ccncc1-c1cn(CC(=O)NC(CCN2CCCC2)C(N)=O)nn1 C(=O)(CCC(=O)NCC1CCC(NC(=O)CSCc2cscn2)C1)NCC N1(C(c2nn(C)c(=O)cc2)=O)CCC2CN(C(=O)CCC3CCC(O)CC3)C2C1 CCC(CC)C(=O)NC1CCOC(C(C)C)C1.C12CC(C1)OCC(=O)N2 c1(C(N2CCC(OC)(CNC(=O)Cn3ccnn3)CC2)=O)ccc(N=[N+]=[N-])cc1 Cc1cnn(C(C)C)c1C(=O)NCCC(C)NC(C1CC(F)C(=O)N1)=O C1(C(=O)Nc2ccc(OC)cc2C)CC2(CCN1C(=O)Cn1cnnc1O)CC2 Cc1sc(O)nc1C(=O)NC1CCN(C(C2(n3ccnn3)CC2)=O)CC1 Cc1nc([N+](=O)[O-])cn1CC(N1CC(NC(=O)CCCCCF)CC1C)=O c1(CC(=O)NCC2(NC(c3ccc(O)nn3)=O)CCC2)ccc(Br)c(F)c1 C1(NC(=O)CC=CCN2CCCC2)CCOCC1.c12cnn(c1)CCNC2=O c1(C(=O)NCCOC2CN(C(C#CC(OCC)OC)=O)C2)cc(F)ccc1CC c1(C(=O)NC(c2ccccc2F)CNC(=O)CCC2CC2)c[nH]c2ccccc12 Cc1cc(C)c(C(=O)NC(CNC(c2conc2C(C)(C)C)=O)C2CC2)cc1N C(=O)(C(CC(C)C)NC(=O)CN1CCS(=N)(=O)CC1)OC CCC(CC(F)F)C(=O)N1CCN(C(=O)C(C2CCC2)C2CCC2)CC1CO c1(C(=O)NCC(CCC)NC(c2cc(C3CCC3)[nH]n2)=O)ccccc1C(C)=O N1(C(CCCOCC=C)=O)CCCN(C(=O)C2=CCOCC2)CC1CO c1(-n2cc(C(CCC)NC(c3cc(CC(C)C)on3)=O)nn2)cccc(F)c1Br c1(NC(C2CC(F)CN(Cc3cnccc3Cl)C2)=O)ncc([N+](=O)[O-])cc1I Cc1cccc2c1NC2=O.c1(NC2CCCCC2)nc(Cl)ncc1Br c1(C(=O)NCC(CC=C)NC(=O)CCn2cnc(C)cc2=O)ccc(O)nc1Cl Cc1nccnc1C(=O)NCC1C2CC1N(C(=O)CCCCC1CC1)C2 Cc1ccc(C(=O)NC(C)(C)CCNC(C2CCC(C3CC3)C2)=O)nc1O C1(C(N2CCC(C#CC)C2)=O)CC2CCCC2N1C(c1ncsc1C)=O Cc1cc(C(=O)NCC(C2CC2)NC(c2cnc(C3CCCO3)s2)=O)c(C)cn1 N1(C(CN(C)C(N)=O)=O)CCC2CCC(NC(c3nnc(C(F)(F)F)s3)=O)C1C2 CCCC(C(=O)OC)C(=O)N1CCC(C)(C(=O)Nc2cccc(C)c2C)C1 CCCC(CC(=O)OC)NC(=O)C(C)C(C)OC C1(NC(c2ccc(CSC)cc2)=O)CC2CCC1N2C(c1ccc(F)cc1Cl)=O c1(C(=O)O)nc2n(n1)CC(NC(C(=O)O)C1CC1)CC2 N1(c2snc(C)c2C#N)CC2CC1CC2C(N1CCN(C)CC1C)=O O(NC(=O)C(C)(C)C(C)(C)C)CC(=O)NCCC(C(C)C)(C)C C#Cc1ccccc1NC(c1ccc(F)nc1)c1nnnn1CC1CCOC1 CC(C)(CC1CC1)C(=O)NCC(C1CCC1)NC(=O)CCCCN(C)C c1(C(N2CCc3c(n[nH]c3C)C2)C(=O)NC(CC)C)cccc2cnn(C)c12 CC1(C)COCCC1C(N1CC2CC(NC(C3(O)CCSCC3)=O)C2C1)=O C1(NC(c2cc(Br)no2)=O)CN(C(C2Cc3cscc3C2)=O)CC12CCC2 C1(C(=O)NC(C(C)C)(C)CNC(c2ccc(C#N)s2)=O)CC2(COCCO2)C1 C(C(CC(C)C)C(=O)N1CCCC1C(C)NC(=O)CCc1ccc(F)cc1)OC c1(N2C(C3CCN(C(C4(C)CC4(F)F)=O)C3)CCC2)ncc(O)cn1 CCC(C)(CO)C(=O)NCCOCC(=O)NCC12CC(C)(CCO1)C2 C1(C(=O)NCCc2c(F)cccc2Br)Cn2nc3ccccc3c2N1 c1(C(N2CC(CC(C)NC(CC(=C)Br)=O)C2)=O)nccc2ncccc12 c1(C(=O)NC2CC2NC(C2(c3cccnc3)CCCC2)=O)cnc(O)c(Cl)c1 C1(C)(CCCC)CN(C(=O)CC2CC(NC(=O)Cc3nocc3C)C2)C1 c1(C(N2CCN(C(C(CC(C)C)N(C)C)=O)CC2)=O)[nH]nc2c(=O)n(C)cnc12 C(C)(c1ccccc1Cl)=CC(=O)NC1CCCC(CNC(C(F)=CC)=O)C1 c1(NCC2(O)CN(C(C(c3ccc(C)s3)C)=O)C2)ncnc2c(Cl)cc(Cl)cc12 C(CCCCC(=O)NC(C1CCN(C(C2(C)CCSCC2)=O)C1)C)OCC CC1(C)CCC(CO)N(C(=O)C(C2(O)CCCCC2)NC(=O)CCC(F)(F)F)C1 Cc1ncccc1C(=O)NCCOC1CN(C(=O)C(n2nccc2C)C)C1 N1(C(c2ccc(SC)o2)=O)CC(NC(=O)C(Cl)=CCl)C(N=[N+]=[N-])C1 C1(C(N(C)CC2CCCCN2C(C2(C#N)CCC2)=O)=O)CC(=O)OC1(C)C c1(CCNC(C2(C(=O)NCc3ccccc3Br)CC2)=O)ccc(Cl)cc1[N+](=O)[O-] C#CCCCC(C)C(=O)N1CCC(C(C)(C)C(N2CCC23CCN(C)C3)=O)C1 N1(C(CCc2cccc(C)c2)=O)CCC2(CC1)CC2C(N1CC(F)C1)=O C1(SC)CN(C(c2ccc(C#N)cc2)C(=O)NC2CCC2)C2(CCC2)C1 c1(OC)ccnc(C(=O)NCCC2CCN(c3ncnc(Cl)c3OC)C2)c1F c1(C(=O)NC(CNC(C=CSC)=O)C(C)C(C)C)cc2nc(C)ccc2o1 CC(F)(F)CC(=O)N1CC(F)CC1CNC(=O)CCCc1cnn[nH]1 C12(C(N(CCNC(C3(C4CC4)CC3)=O)CC)=O)CCC(=O)N1CCS2 N1(C(CC(CNC(C2CC2C#N)=O)OC)=O)CCCC(C)(C)CC1 C1(C(N(C(C2CCCC2)CNC(C2(NC(N)=O)CCC2)=O)C)=O)CCCSC1 c1(C(N2CC(NC(C3C(F)(F)C34CCC4)=O)C(O)C2)=O)cc([N+](=O)[O-])cnc1O c1(OCCCC)ccc(CNC(=O)NC(C)CC2CC2(Cl)Cl)c(Cl)c1 c1(OC)ccc(C=CC(N2CC3CC3(CNC(c3coc(O)n3)=O)C2)=O)c(C)c1 C(=O)(C(C)(C)CCNC(c1ccnc(CO)c1)=O)N(CCC(=O)OC)CC O=C(C1CCCn2ccnc21)NCC1CC2(CC2)CN1C(C1CC=CC1)=O Cc1nc(C)c(C(=O)NCCSC2CC2)[nH]1.N12CCCC1C2 C1(C(N2C(C(C(C)C)=O)CC2)=O)CC12CCN(C(C)C(N)=O)CC2 c1(C(N2CC(CC(OC)OC)C2)=O)[nH]nc2c1C(c1ccccc1)CCC2(C)C C(=O)(C1=CC2(CCN(C(=O)C(N3CCNC3=O)C)C2)C1)N1C(C)(C(=O)NC)CC1 Cc1ccc(N(S(=O)(=O)CC2CC(C)(C)C2)Cc2ccccc2)cc1Cl c1(C(=O)NCC(CNC(C2(COC)CC2(F)F)=O)C)cn(C)nc1C N1(CCNC(C(C)N(C(C2C(CC)C2)=O)C)=O)CCCCC1 C#CC1(C(=O)NC2CCCCCC2CO)CCN(C(C2CC=CCC2)=O)C1 C12(C(=O)NCC(C)CN(C(=O)C(c3ccc(F)cc3)O)C)CC(C1)C(C)O2 N1(C(c2c(CC)cco2)=O)CCC2(CCN(C(=O)CC3CCCC(O)C3)CC2)C1 c1(C(CC)N(C(=O)C(N2CCC(n3cc(C(C)O)nn3)C2)=O)C)ccccc1Cl c1(C(C)OC)nc(C(=O)NCC(O)CNC(C2(F)CCCC2)=O)cs1 c1(NC(CN2C(CC)COCC2)=O)cc(N)c(C)cc1C N1(C(c2cncc(OCC)c2)C(=O)NC2CCOC2)CCOCC(C)(C)C1 C(=O)(C(C)(C)C(C)NC(c1cnc[nH]c1=N)=O)N(CCCC=C)CC N1(C(C2(OC)CCSC2)=O)CCC2(CC1)CCN(C(=O)C(C)C(C)O)CC2 c1(C(N2C(CNC(C(C3CCCC(=O)N3)C)=O)CC2)=O)noc2ccc(F)cc12 c1(NC(C23CCN(C(C(C=C)O)=O)C2CCC3)=O)cnc2ccccc2c1 N1(C(c2n(C)ncc2)=O)CC2CCN(C(c3ccc4cc[nH]c4c3)=O)C2C1 c1(C(=O)NCc2c[nH]nc2C(F)(F)F)cc(Br)cc2cn[nH]c12 CCC(C(=O)N1CC(O)(CNC(c2ccn(C)c2C2CCC2)=O)C1)C(C)C N1(C(c2cn(CC)nn2)=O)CC(NC(C2(N(C)C)CC2)=O)C(F)C1 C1(NC(c2scc(CC)c2)c2nnnn2C)COc2ccc(C)cc2C1 c1(NC(C2N(Cc3cnc(SC)nc3Cl)CC2)=O)cc(Br)cc([N+](=O)[O-])c1C N1(C(C=CC=CCC)=O)CC2(COC(CNC(=O)C(CC)OC)C2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1C(CNC(C=C(C)C2CC2)=O)C(C)CC1 C12(CC(N3CC4C(C(N5CC(CN=[N+]=[N-])OCC5)=O)C4C3)=O)CCC(CC1)CC2 C(=O)(C1Cc2ccccc21)N(C(C)CNC(C1CCC2(CCC2)CC1)=O)C C1(CC=C)(C(=O)NC2CN(C(=O)CCc3ccsc3Cl)CC2OC)CCCCC1 c1(OCC=CC(=O)NCC2CC2NC(=O)C=CC2CCCC2)ccccc1 C1(C)(CC)CCN1C(=O)C(C)NC(C1CS(=O)(=O)C1)=O CC(CN(C)C(c1cc(C2CC2)[nH]n1)=O)C(=O)N=c1ccn(C(F)F)[nH]1 C1(CC=C)(NC(=O)C(C)COC)CCN(C(c2sc(C)cc2Cl)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)N(C)CCN(C)C(C1CC1c1cnn(C(C)C)c1)=O C(C1CN(C(C2CC3CSCC(C2)C3)=O)Cc2ccccc21)NC(CC)=O N1(C(c2n[nH]c(C)c2N)=O)CC2CC(C(=O)NCC(c3ccco3)O)CC2C1 c1(C(N2C(C)(CNC(C(C)SCCCC)=O)CCC2)=O)cc2scnc2[nH]1 Cc1c(NC(c2ccc(Cl)nc2)C)ncnc1N(CC(Cl)Cl)C c1(CNC(C(C2CC(NC(=O)C=Cc3cc[nH]n3)C2)F)=O)ncccc1Cl c1(CNC(N2CCCC(C#C)CC2)=O)cc(C)nc2ncnn12 C1(NC(COCP(C)(C)=O)=O)CCCC(NC(=O)CCc2ccc(N)cn2)C1 CC1COC2(C1)CN(C(c1ccc(F)c(N3CCCNC3=O)c1)=O)C2 Cc1ncc(C(=O)NCC(n2cc(CCCN(C)C)nn2)C)n1C c1(CC)[nH]ccc1C(=O)NC1CC(OCC(N2CCC(O)C2)=O)C1 Cn1ncc(C2CC2)c1S(=O)(=O)Nc1ccccc1CN C1(NC(C)=O)CCN(C(c2conc2C(C)NC(c2c(C)n[nH]c2C)=O)=O)CC1 c1(C(=O)NCC2CC(NC(c3ccc(OC)s3)=O)C2)[nH]c(C)cc1C O=C(CCCCCNC(C1CCCN1C1CC1)=O)Nc1ccc(Cl)nc1 c1(C(=O)NC(CC)CNC(=O)CCN2CCC(F)C2)cncnc1C C1(NC(c2cc(C)on2)=O)CN(C(=O)C(N2CCN(C)CC2)C)CCC1CO C1(NC(=O)Cn2cnnn2)CC2(C1)CN(C(=O)Cn1ccc(C(F)F)n1)C2 c1(SC)ccc(CCC(=O)NC(C)CN(C(=O)CC(C)C)C)cc1 c1(C(C)NC(C2CC(NC(c3cnc(C)n3C)=O)C2)=O)cccc(C#N)c1 CCCCC(CC(=O)NCCC(C)N1CCCC1)NC(=O)COC1CCCC1 c1(C(N2CC(C)(C)C2(C)C)C(=O)NCc2ccc(F)cc2)cccc2[nH]ncc12 c1(C(=O)NC2(CCOC)CCN(C(C3C(=C)C3)=O)C2)cnn2c(O)cc(C)nc12 C1(CC=C)(C(=O)NCC(=C2CCCCC2)F)CCCN1C(=O)C(C)NC=O c1(C(n2c(-c3cncnc3C)nc(-c3ccc(C)cc3)n2)C)cccc(Cl)c1Cl N1(C(c2nccc(CNC(c3c(CC)occ3)=O)c2)=O)CCCSCC1C CCC(CCC(=O)N1CC(NC(c2c(Cl)cnn2C)=O)C(O)C1)OC C1(CNC(c2cn(CCCC)nn2)=O)(OC)CCN(C(C2CC23CCC3)=O)C1 C(CC(C(=O)NC1CN(C(C2(C3CCC3)CC2)=O)CC1C)N(C)C)SC Cc1ccc(CC2CCN(C(=O)NCCc3nccnc3C)C2)cc1 CC1(C)COCC1C(=O)NC(C1CC=CCC1)C(=O)Nc1cnc(Cl)nc1 C#Cc1cnn(CC(=O)NCCCC(C)NC(=O)C(C)SCCCC)c1 C(=O)(CS(N)(=O)=O)N(C1CC(C)(C)CO1)CCCc1cn(C(C)CC2CCC2)nn1 CC(CC(F)(F)F)C(=O)NCCn1cc(CCC2CCCCO2)nn1 c1(C(=O)NC(CCNC(CCc2ccn(C)n2)=O)(C)C)ccc2c(c1)OCCN2 c1(CN2C(C(=O)NCC3(O)COC3)CC(=C)C2)cc(Br)ccc1F N1(C(CN(C(=O)C(C)(C)n2cnnn2)CCOC)=O)CCCC1c1cc[nH]n1 C#CCC(CC(=O)N1CCC(OCC(N)=O)C1)NC(=O)CC1CCCC(C)O1 c1(C(C(N)=O)NCC2(O)CCNC2)cccc(OC(F)(F)F)c1 C1(F)(C(N2CC(C3N(C(c4c(C)snc4)=O)CCC3)(O)C2)=O)C2CCCCC12 Cc1ccc(C(=O)NC(C)C(C)C(N2CCS(=O)C(C)C2)=O)c(F)c1 c1(OC)cc(C(N2CCC(C3(NC(=O)C(O)CSC)CC3)C2)=O)cc([N+](=O)[O-])c1 Cc1[nH]nc(CO)c1C(=O)NC1CC2(C1)CC2C(N1CC(N2CCC2)C1)=O C(=O)(C1=C2CCCN=C2NN1)NCC1N(C(c2cccc(C)n2)=O)CC1 C1(C(=O)OCC)CCc2cnccc2N1C(=O)COCCCOC Cc1nn(CC(=O)NCC2CC2CNC(=O)CC=CC(C)(C)C)c(C)c1Br C1(CNC(CCCC#C)=O)CC(NC(=O)Cc2scnc2C)C12CCC2 CC1(C)CN(C(=O)C(O)C2CC2)CC1NC(C1(c2ccno2)CC1)=O c1(C(=O)NCC(CC)NC(C(C=C)(C)O)=O)cnc2onc(CCC)c2c1 c1(C(=O)NC2(CCC)CCCN(C(c3nccn3C)=O)C2)ccc2[nH]ccc2c1 c1(C(=O)NCC2C(NC(CSCCN(C)C)=O)CC2)ccc(-c2cscn2)cc1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC1(NC(c2c(C)ncnc2C)=O)CC1 N1(C(c2n(CC)ncc2)=O)CCC(C)(C)C1CNC(C1(Cl)CC1(F)F)=O c1(C(=O)NCC2C(C(=O)NCC(C)C#N)CCCC2)cccc2cnsc12 N1(c2nc(OC)cc(OC)n2)CCCCC1C1CCCCN1.C1(=O)CN1.C(C)(C)SC C1(NC(C2CC(O)(CNC(c3ccco3)=O)C2)=O)CCN2CCCC12 C12CN(CC(F)(F)C1)C2=O.c1(CN2CC3C(C)(C)C3C2)cc2ncccc2[nH]1 C(=O)(C(CNC(=O)C(c1ccccc1)F)CC1CC1)NCc1n(C(C)C)ccn1 N1(C(C2(CF)CCN(C(c3csc(F)c3)=O)C2)=O)CCN(CCO)C(=O)C1 c1(CC(=O)OC)ccnc(N2CC3CC3(NCc3ccc(SC)cc3)C2)n1 c1(NC(c2cn(C3COCC3O)nn2)=O)cn(CC(F)F)cn1 c1(OC)n[nH]c(=NC(=O)NCC2(c3c(F)cccc3Cl)CCC2)s1 C(=O)(C(F)C(F)(F)F)N(CC(CNC(C1(COC)CCCCO1)=O)(C)C)C CC1CNc2c(C(=O)NC(C)(C)CCCNC(C3CCCC3)=O)cccc2C1 c1(C(=O)NC2CC(NC(C(c3n(C)ncc3)O)=O)C2)cc(F)c(CO)c(F)c1 Cc1cc(Br)cc2c1CN(N1CCN(CC(N3CCN(C)CC3)=O)CC1)CC2 CCCCC(O)C(C)C(=O)NC(CCCC)CC(=O)N1CCC(CO)C(O)C1 Cc1cn2ccc(C(N3CCCN(C(C4C(C)C4(F)F)=O)C(C)C3)=O)cc2n1 c1(C(=O)NCC2(C)CCCN(C(CC(=O)OC)=O)C2)cc(Cl)c([N+](=O)[O-])[nH]1 N1(C(c2c(CNC(=O)C=CC3CCOCC3)noc2)=O)CC2CC=CC1C2 CCC(O)C(=O)NC(CNC(c1nocc1C1CC1)=O)C(C)C C1(C(=O)NC(CC)CO)(SC)CN(C(=O)CC2CCCCO2)C1 N1(C(c2n(CC#N)ncc2)=O)CCCCC(NC(c2coc(Br)n2)=O)C1 C1(C(=O)OCC)OCCNCC1N1CCN(c2ccc(Cl)nn2)CC1 CCC(C)(C)CCCC(=O)NC(C)C(C)(C)NC(=O)CCNC(=O)CO C(=O)(C1CCCc2c1ncn2C)NCCN(C)C(c1ccc(F)c(CO)c1)=O Cc1ccc(C(=O)NCC2CC(N(C)CC(=O)CCCN3CCCC3)C2)c(F)c1 C(=O)(C1=CC2CCCC12)NC12CC(NC(CC(CC)(F)F)=O)(C1)C2 C=C1CCC(C(N2CCC2CNC(=O)CSCCC)=O)CC1 c1(C(=O)NCC(CC)NC(c2ccc(F)c(Cl)c2F)=O)cccc2cc[nH]c12 c1(CC(=O)NC(C)C(N)=O)ccc(O)c(CNC(C23C(CN(C(C)=O)C2)C3)=O)c1 C(C(C)(C)C(=O)NCC1CCC(C)N1C)N(C(c1cc(OC)ns1)=O)C N1(C(c2ccc(C(C)C)nc2)=O)CCCC2(C1)CN(C(=O)C(C)(C)C(C)(F)F)C2 C1(C)(CC)CC(NC(c2cn(C)cc2C)=O)CN1C(c1sccc1C#N)=O c1(N)ncnc2[nH]cc(I)c12.O=C(N=c1cccn[nH]1)c1c(F)cccc1Br N1(C(CN(CCOC)C)=O)CC2CC(NC(c3c(OC)noc3C)=O)C1C2 C1(COC)CN(C(c2cc(Cl)ncc2C)=O)CCN1C(c1ccnc(Cl)c1Cl)=O N1(C2C(C)C2)CCN(N2CCCC2CCCC(F)(F)F)CC1 C1(NC(C=CSC)=O)CC2CCC1(NC(=O)C(C)Cc1ccncc1)C2 Cc1cc(=NCC(C)c2cccc(Br)c2)[nH]cc1Cl c1(C(N2CC(O)(CNC(c3ccc(CC)nc3)=O)C2)=O)cc(F)cc2cc[nH]c12 c1(NS(C)(=O)=O)cccc(C#N)c1.C12CCC(CC1)CNC(=O)C1CN(C1)C2=O N1(C(N2CCCC2c2ncc[nH]2)=O)CCCC(NS(=O)(=O)C2CC2)C1 C1(NC(c2n[nH]c(C)c2C)=O)CCC2(C1)CN(C(=O)CN1CCS(=O)(=O)CC1)C2 C1(CNC(CN2C(C)CCC2C)=O)CC2(CCOCC2)CN1C(=O)CC(C)(C)O c1(C(N(C2(C(=O)NC3CC3(C)C(F)F)CC2)C)=O)ccccn1 c1(C(N(C2CCCN(C(C(c3cccc(O)c3)C)=O)C2)C)=O)cc(F)ccc1F c1(C(=O)NC2CN(C(Cn3ccc(C)n3)=O)C3C2C3)ccc(Cl)c(O)c1 C#CCC(C(=O)OCC)C1CC1.c1(CC=O)ccccc1.C12CCN(C1)C(=O)CC2 O=C1CCC(C(=O)NCCCCC(=O)N2CCOCC2C(F)F)CN1 c1(C(C)=O)ccc(C(=O)NC(CNC(=O)CN2CCCC2C)C(C)(C)C)c(F)c1 C1(C(=O)NCCOC2CCN(C(Cc3n(C)ccc3)=O)CC2)CCC2(CCC2)C1 c1(C(=O)NC2CCCC(NC(C(=O)NCC(F)(F)F)=O)C2)ccc(Cl)cc1O c1(CC)ncoc1C(C(=O)NCCC#N)N(C)C(c1nccs1)C CC(CCCN=c1cc(C(N)=O)nc[nH]1)NC(=O)CC1CC2(CC2)C1 Cc1cc2nc(C(=O)NCCCNC(c3ncc(Cl)cc3O)=O)cn2cc1C c1(C(C(N2CCN(C(=O)NC)CC2)=O)NC(=O)C2=C(Cl)CC2)cc(C)ccc1F N1(C(C=CC(=O)NC2CC2)=O)C2CCC(C(=O)NC3(CF)CCCC3)C1CC2 c1(C(=O)N(C2CCCN(C(=O)C3=CCSC3)C2)CC2CC2)ccc2nc[nH]c2c1 C(C(C)(C)CNC(c1cnn(CC)c1)=O)N(C(c1csnn1)=O)CC c1(C(N2CC3(CC(NC(C4C(CCC)C4)=O)C3)C2)=O)ccnc2c1ccn2C c1(CCCC)cc2nncn2c(NCCCN2CC(C)OC(C)C2C)n1 CCCCC(O)CC(=O)N1CCC(C(=O)NC2(Cc3ccccc3)CCC2)C1C c1(CC(N(C2C(c3n(C)ncc3)OCCC2)C=O)=O)cc(Cl)cc(Cl)c1 CCC(CC)CCC(=O)NC(CO)C(C)NC(C1CCC(c2ccccc2)O1)=O N1(C(C=C(C)C(C)(C)C)=O)CC(C)(C)CC1CC(=O)N(CCO)CC1CC1 Cc1c(Cl)ccc(C(N2CCN(C(=O)CC3CCOC3(C)C)CC2)=O)c1O C1(NC(COC(CC)C)=O)CCN(C(c2ccc(Cl)c(C)c2)=O)C1(C)C c1(C(=O)NCC2N(C(c3nnc(C)s3)=O)CC2)oc(Br)nc1C C1(NC(C=C(C)C(F)F)=O)CCN(c2ncnc3onc(C)c23)C12CCCC2 c1(CN(C(CCSC)=O)C)cnn2c1CN(C(=O)CSCC(C)=O)CC2 C1(NC(CONC(C2(Cl)C(C(C)=O)C2)=O)=O)CCc2nncn2C1 c1(OC)cccc(N(C)C)c1.c12sccc1NC(=O)C2N1CCC(CF)C1 Cc1cccc2[nH]c(C(=O)NCC(F)CNC(c3cn(C)[nH]c3=N)=O)cc12 C1(NC(C2(COC)C=CCN2C(=O)CCN2CCOCC2)=O)CCCN(C)CC1 c1(C(=O)NCC2N(C(Cc3n(C)cnc3)=O)CCCC2)ccc(F)cc1N Cc1ccc(C(N2CCC(NC(=O)C(C(C)C)n3cnc(C)c3)C2)=O)c(N)n1 C1(NC(C2N(C(C)C)C(=O)CC2)=O)COC2(CCCN(C(=O)OC(C)(C)C)C2)C1 C(CN=C(NCc1cnc(OC)cn1)NC1CCC1)N1CCCC(OC)C1 N1(C(c2cc(CNC(CN(C)C(N)=O)=O)no2)=O)CC(F)(F)CC1CO N1(C(c2c(=N)[nH]cnc2)=O)CCC2CC1CN(C(=O)COc1ccc(O)nn1)C2 Cc1nc(C(N2CCCC2CC=CC(N2CCC(c3ccon3)C2)=O)=O)co1 c1(OCC2C(NC(C(C)OC)=O)C2)ccc(Cl)c(Cl)c1.C12(CCC1)CC(=O)N2 Nc1cnc(C(=O)NC(CCC2CC2)C(=O)NC2(c3nn[nH]n3)CC2)cn1 C(=O)(C1=CS(=O)CCC1)N1CCC(C)C1CNC(c1cc(F)ccc1Cl)=O c1(CNC2C(C(=O)Nc3nccc(OC)n3)C2)ccc(C#N)cc1[N+](=O)[O-] C1(C)(NC(C2C(C)CCO2)=O)CCCN(C(c2cccc(N)c2)=O)C1 N1(C(C(c2ccncc2)C)=O)CC2CC(CNC(C3CC(F)C3)=O)C2C1 CN1N=C(C(=O)NC23CC(C2)N(C(c2cc4ccc(Cl)nc4s2)=O)C3)CCC1=O c1(C(N(C2CCCN(C(=O)C#CC3CC3)C2)CC)=O)cc(O)nc(Br)c1 N1(CC)CC(CNC(=O)C(C)(C2CCC2)NC(=O)C(C2CCCCC2)O)CC1=O N1(C(Cn2c(C)ncc2)=O)CCC(C(=O)NCC(C)CCCO)(C(C)C)C1 C1(CNC(C2(CC#C)CCOC2)=O)CC(C)CCN1C(c1ccsc1C#N)=O C(=O)(C1=C(CC)OCCS1)NCC1CN(C(C2CCC(CCC)CC2)=O)C1 Cc1n[nH]c(C)c1C(C)CC(=O)N1CC(CO)(NC(c2c[nH]c(Br)c2)=O)C1 C(=O)(CCCNC(N)=O)NC(C1CN(C(C(C)NC(CC)(C)C)=O)C1)C N1(C(C(CC(=C)Cl)NC(=O)C(C)CC(C)CC)=O)CCC2(CCCC2)CC1 C1(CNC(C(C)OCCOC)=O)CCCCN(C(=O)CCCn2cc(C)cn2)C1 CCN=c1cc(-c2nc(-c3occc3C)n(CCOC)n2)cc[nH]1 CC1(C)CCN(C(=O)NC(CCO)c2cccs2)C1 C1(NC(CCCOC(CCC)=O)=O)CC2(C1)CN(C(C1CCCCC1C)=O)C2 C(C(F)(C(=O)NCC12CCC(CC1)O2)C(C)C)NC(c1c(C#C)cnn1C)=O c1(OC)cccc(C(NC(=O)C(C)Oc2cccc(CN3CCCC3)c2)SC)n1 c1(NCC(=O)NCC(CN(C(CCSCC)=O)C)C)c(F)cccc1F n1(CC)cc(C(=O)NCC2CCCN2C(=O)CC2(C)CC2(F)Cl)c(C(C)C)n1 c1(SC)ccc(CCC(=O)NC2CCC(C)(CNC(=O)CSC(F)F)C2)cc1 N1(C(C(C=C)OC)=O)CCC(C)(C)C1C(=O)NCC1CC(C(C)C)C1 C(c1cccn1C)=CC(=O)N(CC(C)N(C)C(c1ccns1)=O)C C(=O)(CC(C(=O)Nc1cccc(S(=O)(=O)NC(C)(C)C)c1)C(C)C)OC C=CC(O)C(=O)NC1CC1NC(c1cnc(-c2ccco2)s1)=O N1(C(CSCC=C)=O)CCN(C(C2(O)CCOCC2)=O)CC1CO C1(NC(C2(CC#C)CC=CCC2)=O)CN(C(c2n[nH]c(CC)n2)=O)CC1(C)C C1(NC(CN(C)C(C2(C)CC3C=CC2C3)=O)=O)CC12CCCCCC2 Cc1ccc(CN2CCCC(C(=O)Nc3cccnc3I)CC2)cc1[N+](=O)[O-] C(=O)(CCCc1cccs1)NC(C1CN(C(c2cnn(C3CCOC3)n2)=O)C1)C CN1CCCCC1CNC(=O)CC1CCN(C(C2CCC(C(N)=O)CC2)=O)C1 C1(C(=O)NCCc2ccncc2)(CC)CCN(C(C2CCCC2C)=O)CC1 C(C(CC(C)C)C(=O)NC1(C)CCCC1NC(c1cc(C)c(C)[nH]1)=O)OC C1(CCNC(c2c(C)nco2)=O)CN(C(=O)Cc2ncoc2C)CC(C)O1 N1(C(COC(C)C)=O)CCC(CNC(c2cccn(C)c2=O)=O)CC1C N1(C(CC(C)N2CCCC2=O)=O)CC2CC1C2NC(=O)C(c1ccccc1)O CC1(C)CCOC(CC(=O)N(C2CCN(C(C3(C)C=CCC3)=O)CC2)CCO)C1 O=S(=O)(c1ccc(Br)s1)N1CC2CCC(C1)C2NCc1cc(I)c(O)c(I)c1 C1(C)(C(=O)OC)C=CCN1C(=O)CCCn1cc(CNc2cccnc2C)nn1 C1(CN2CCC(N(C(c3cnn(C(C)C)c3)=O)CC)C2)CCC2CC2C1 c1(OC)nc(C)sc1SC.c12cccnc1NC(=O)C1CCC(C1)n1cc-2nn1 c1(OC)ccc(C(=O)NCC2CC(O)CN2C(c2sncc2C)=O)cc1C(F)F O=C(CC(CC(F)F)c1ccccc1)NC1(CF)CCN(C(=O)CO)C1 CCCCCC(O)CC(=O)N1CCN(C)CC1C(=O)N(CCO)OC C(=O)(C1=NOC(C)(C)C1)NC1(CO)CCN(C(COCC#C)=O)C1 C1(S(N)(=O)=O)(C(N(CC(C)NC(c2cccnc2C(F)F)=O)C)=O)CCCC1 c1(C(N)=O)nccnc1C(=O)NC1(CC(N2CCC(CC3CC3)C2)=O)CCC1 C1(C)(C(=O)NCC2(C)CNC(=O)O2)CN(C(C2C3(CC3)C23CC3)=O)C(C)(C)C1 CCN=c1[nH]c(C)c(C(=O)NC(C)C(C)NC(=O)C(F)(F)c2nccs2)s1 C(=O)(C1c2ccccc2CN1C(=O)C(O)CC(F)(F)F)NCCCOC=C c1(N2CCC(Br)=C(C)C2)cc(C)c(S(=O)(=O)NCC(C)CC(F)(F)F)cn1 N1(C(C2CCC(=C)CC2)=O)CC(NC(=O)CCn2cc(C)cn2)CC(O)C1 C1(C(N(C)CCO)=O)Cc2cc(O)ccc2CN1C(=O)COc1ccccc1 C1(F)(C(N2CC(F)(CNC(CNC(C(C)(C)C)=O)=O)C2)=O)CCCOC1 C=CCC(CC=C)C(=O)N(CCC(=O)NCC1(CC)CCOC1)CC=C c1(CN2CCC(CC(=O)Nc3cc(Cl)c(F)cc3Br)CC2)ccc(F)c(F)c1Cl c1(CC)oc(C(=O)OC)cc1S(=O)(=O)NC1(c2ccccc2OC)CCC1 c1(C(=O)O)cc(CNCC2(O)CN(C(C3CCCCO3)=O)C2)cc(Br)c1 c1(C(=O)NC2CC3CC(NC(c4cccnc4)=O)CC23)ccc2occc2c1 C(=O)(C1=CS(=O)CCC1)NC1CCN(C(C(C)(F)F)=O)CC1CO n1(CC(=O)NCCCN(C(C(C)c2cccs2)=O)C2CC2)ccc(=O)n(C)c1=O Cc1ccc(-c2nc(CS(=O)C(C)c3ccccn3)cs2)c(C)c1 c1(C(N2CC(CNC(=O)CC34CCCC3C4)C(O)C2)=O)cccn2nnnc12 CC(C)CC(C(=O)NCCc1cnn[nH]1)ONC(=O)CCc1nc(O)n[nH]1 c1(NC(C2CCN(C(=O)C=Cc3cccnc3)C2)=O)c(F)cc([N+](=O)[O-])cc1Br c1(C(N2CCOC(CNCc3ccc(F)c(O)c3F)C2)=O)ccc(F)c(F)c1F c1(C(N2CC(CCC)N(C(C3CCCS3(=O)=O)=O)CC2)=O)c[nH]c2cccnc12 Cc1nc(C(F)(F)F)ccc1C(N1CCC1C(N1CC(F)CC1CO)=O)=O CC1CCN(C(c2cc(Cl)no2)=O)CC1CC(N1CCC2(CSC2)C1)=O Cc1nc(C=CC(=O)N(C)CC2CCCN2C(=O)CC(Cl)Cl)[nH]c1C C1(NC(C2CCC(=O)NC2)=O)CCCC2CN(C(c3cc(Cl)c[nH]3)=O)CC12 c1(-c2ccc(CC)cc2)ccc(S(=O)(=O)NCCN(C)C)s1 c1(C(N2CC(C(C(=O)NCCN(CCC)C(C)C)O)C2)=O)ccc(O)cc1 Cc1n[nH]c(C)c1SCC(=O)NC1CCCC1NC(=O)Cn1cnnc1 c1(C(C(=O)NC(CNC(C2(C(C)CC3CCC3)CCC2)=O)CO)O)cccc(Cl)c1 CC(C(=O)OC(C)(C)C)C(=O)N1CCCCC1Cn1cc(-c2ccc(Cl)s2)nn1 N1(C(C)CC(=O)NCC(O)CCNC(=O)C(C)(C)O)Cc2ccccc2C1=O CC(CCN=c1[nH]c(=N)[nH]c(=NCc2ccsc2C(F)(F)F)[nH]1)N1CCCCC1 c1(OC)c(C(=O)N(CCCn2cc(C3CCCN3C)nn2)C)cccc1F N1(C(CC2CC(C)(C)OC2)=O)CC(CO)C2(C1)CN(C(C1CS(=O)(=O)C1)=O)C2 CC1(CNC(C2CCCCC2n2cc(SCC(=O)OC)nn2)=O)CCCNC1=O Cc1cccnc1CC(=O)NCC1CCCC1NC(c1cnc(S)nc1)=O CC1Oc2ccccc2OC1C(=O)NCC(C)(C1CC1)NC(=O)COC(F)F C1(C(=O)NCC(C)(CO)NC(c2ccc(N)c(F)c2)=O)CCC2(CCC2)OC1 c1(C(=O)NC2CN(C(c3c(CC)con3)=O)CC(O)C2)ccc2ccsc2c1 N1(C(Cc2c(C)nn(C(C)C)c2C)=O)CCC2(CC1)CC2NC(C1C2COCC12)=O n1(CCC)nc(C)c(C(=O)NCCC2CCN(C(=O)CC3CC=CCC3)C2)c1C CC(C)C(C)C(=O)N1CC(NC(c2ccc(CC(=O)NC(C)C)cc2)=O)C(C)C1 C1(C(=O)NCc2ccc(CCNC(C(CC)C#N)=O)cc2)CN2CCN1CC2 C1(C(C)NC(c2cnn(C3CCCC3)c2)=O)CN(C(C2CCC2)=O)CCO1 Cc1cccc2c(C(=O)NCCN(C(=O)C(F)C3CCC3)C(C)C)cnn12 CCCCC(C(=O)NC12COC(C1)C(NC(C1CC(OC)C1)=O)C2)OC CC(C)CC(CNC(C1CC2(CC2)C1)=O)NC(=O)C(C(C)O)NC(=O)C1CC1 c1(C(N(C2CCN(C(=O)Cn3cnnn3)C2)CC#C)=O)cc(C(F)F)ncn1 C1(C(=O)NC2C3(CCN(C(c4c(C)cno4)=O)C3)C2)CN(C)CCN(C)C1 CC1=NOC(C(=O)NCC(C)N(C(COCCCC)=O)CC)C1 c1(C(N2CCC(CNC(C(CC)Sc3ccccc3)=O)C2)=O)c[nH]c(=O)cn1 C(N=c1[nH]c(C2CC2)nc(C)c1Br)C1(F)CC(NC(C2CC=C(C)CC2)CC)C1 c1(-c2cc(NC(c3nc(C)c(F)cc3)=O)sc2)c(F)cccc1C#N N1(C(C(F)OC)=O)CC(C)CN(C(=O)CN2CCCCCCC2=O)C(C)C1 C1(C(=O)NC2(CSC)CN(C(=O)COc3cccc(C)c3)C2)CC(=O)N(O)C1 C1(C2CN(C(c3ccc(-c4cnco4)cc3)=O)C2)(NC(C=CCC)=O)CC1 C1(CN(C)C(C2CC=CCC2)=O)CCCCN1C(c1cnc(OCC(F)F)s1)=O C1(CC)CCCCC1N(C)C(C1CC(NC(c2sccc2F)=O)C1)=O C1(O)(CNC(C2C(CNC(CNC(CC)=O)=O)C2)=O)CCC(C)(C)C1 C1(C(N2C(C)CC(NC(c3c(C)ncnc3O)=O)C2)=O)CC12CCC(C)(C)CC2 c1(C(=O)NCCN(C(=O)CCc2cncc(F)c2)C(C)C)cnc2nccn2c1 N1(c2cc(C)nc(N3CCC(C(F)F)C3)n2)CCC2(CCN(C)C2=O)C1 N1(C(C(CC(C)C)NC(C)=O)=O)CCCN(C(C2C=CCCC2)=O)CC1C c1(CN(C(C2CCCCC2)C(=O)NC(=O)OC(C)(C)C)C)cccc2c1CCOC2 C1(NC(c2c(SC)csc2)=O)CN(C(c2cc(C(C)(C)C)on2)=O)CC1F CC1CN(C(=O)Cc2ccsc2)CCN1C(=O)CNC(S(=O)(=O)C1CC1)=O N1(C(c2c(C)n[nH]c2)=O)CC2OCC(NC(=O)CC3CCC3)C2C1 c1(OC)ccc2nnc(CC(=O)N(C)CC3(CO)CCC3)n2n1 Cc1[nH]nc(C(=O)NC2C=CCN(C(C3CC4(CC(=O)N4)C3)=O)C2)c1[N+](=O)[O-] C1(C(=O)NC(Cc2c(C)cc(N(C)C)cc2C)C)CC12CCS(=O)(=O)CC2 c1(OC)cc(CCC(=O)N(CC(=O)OC(C(=O)NC2CC2)C)C)ccc1OC N1(C(c2c[nH]c(=NC)s2)=O)CCCC(CNC(C2CCN(C(N)=O)CC2)=O)CC1 N1(C(CCN(C2CC2)CC)=O)CC(CNC(=O)COC2CCCC2)C(O)C1 c1(C(N2CCC(O)(CCNC(=O)C(F)(F)CC3CC3)C2)=O)ccc(F)c(F)c1F c1(C(N2CC(CC(C)NC(=O)C(C)N(C)C)C2)=O)c2ccccc2nn1C C1(=C(NCCCCC(=O)OC)CSC)SC(=S)N(c2ccc(C)cc2)C1=O c1(NC(C2N(c3cc(OC)nc(C)n3)CC(O)C2)=O)ccc(C)c2ncccc12 CC1CC(C(=O)NCC(=O)N(CC(F)F)C)CN(C(=O)C=C2CC2)C1 C12(CC)CN(C(=O)Cc3ccc(F)c(Cl)c3)C(CNC(=O)Cn3ccnn3)(C1)C2 c1(C(=O)NCC(C)N(C)C(C2CC2C2CCOCC2)=O)ccc2oc(=N)[nH]c2c1 N1(C(C(C=C)C)=O)CCN(C(=O)CCCOC(C)(C)C)CC12CC2 n1(CC)ncc(Cl)c1C(N1CCC(C(C)NC(c2cc(C)on2)=O)C1)=O C1(C(CC)(C)C)CCC(NC(c2csc(C(C)(F)F)n2)=O)CC1 C1(C(=O)NC2C(CC(=O)NC(c3cn(C)nn3)C)CCC2)COC(=O)N1C c1(OC)ccc(C(N2CC=CC2CNC(C2CC3CCCCC23)=O)=O)cc1Cl c1(C(=O)NCC2N(C(C(C)OCC=C)=O)CCC2)cc2c(C)cccc2[nH]1 C1(NC(CN2CC(C)C2)=O)CCCC2CN(C(C3CCc4nncn4C3)=O)CC12 Cc1cccc(NC(=O)CCNC(c2c(C)noc2C)C2CC2)n1 c1(CC)ccc(O)c(C(=O)NCCN(C(=O)C(CN(C)C)C(C)C)CCOC)c1 N1(C(Cn2cc(C(C)O)nn2)=O)CCN(C(c2cnn(C)c2N)=O)C(CCO)C1 Cc1cc(C(=O)NCc2ccc(C(=O)NC(C)C(C)O)cn2)[nH]c1C Cc1ccn2cc(C(N3CCOCC(CNC(=O)C(C)C(C)O)C3)=O)nc2c1 c1(OC)nc(C)cc(C)c1C(=O)NC1CN(C(c2ncccn2)=O)CCC1F N1(c2nc(SC)c(Br)cn2)CC(C2CCCN(C(c3cc(F)ccc3Br)=O)C2)C1 CCC(CC)(CCO)NC(c1cc(CNC(C2CC3CC(=O)C2C3)=O)no1)=O CC1(NC(c2cscc2Br)=O)CCN(C(=O)COC2CCC2)C1 c1(CC(=O)NC(C(=O)NCC=C)C2CC2)ccccc1O CC(C)S(=O)(=O)C(C)C(=O)NCC1CC(O)CN1C(c1ccc(C2CC2)nn1)=O C1(NC(C2(CC=C)CC=CC2)=O)CCCCC1NC(=O)C=C(C)c1cccs1 N#Cc1ccccc1C1(C(=O)NC2CC2NC(=O)C2=COCCC2)CC1 C12(NC(C(CC)NC(c3ccc(CC)nc3)=O)=O)CCC(C1)OC2C C1(Cn2cc(C(S)Cc3cccc(C(N)=O)c3)nn2)COC2(CCNCC2)C1 N(C(=NCC1C=CCC1)NCc1ccccc1F)CC(C1CCOCC1)OCC C=CC1OCCCC1C(=O)NC1CC(CCNC(c2cccc(C3CC3)n2)=O)C1 CC1(NC(=O)C=Cc2ccncc2)CCN(C(C2CCCC2C(F)(F)F)=O)C1 c1(OCCOCCCN(C)C)ccccc1C.C12CN(C1)C(=O)N(C)C2.C(C)(C)C C1(NC(C(c2cccnc2)NC(c2ccoc2)=O)=O)CCCN(CC(F)(F)F)C1 C1(NC(=O)CC2C=CCC2)COCCN(C(=O)COc2ccc(Cl)cc2Br)C1 CCC(F)(F)CC(=O)N1CC(C)C(C)(C(=O)NCC2Cc3nccn3C2)C1 CC(C)C(O)CC(=O)NCC1=CCN(C(=O)CCc2ccc(Cl)cc2F)CC1 c1(C(=O)NC(CC)CNC(=O)C(C)NC(=O)OC)ccnc2ccsc12 c1(CSC)cccc(C(N2CCCC2C(C)NC(=O)C=Cc2cnccn2)=O)c1 Cc1ccccc1C(C)CC(=O)NC(C)CNC(c1ncoc1-c1ccon1)=O C1(C)(CC)NC(=O)N(CC(=O)NCC2(NC(c3ccsn3)=O)CCCCC2)C1=O C1(C(=O)NC2(CCCNC(C(C)=C3CC3)=O)CC2)CC(C)=NO1 C1(C(N2CCN(C(=O)C3=CCCCO3)C(CF)C2)=O)CCc2nccn2CC1 C12CCCC1N(C)C2=O.N1(CC)CCC(NC(C2(n3nccn3)CC2)=O)C1 C(=O)(CCCCCS(N)(=O)=O)NC1(CNC(C(CC(C)C)O)=O)CCOCC1 N1(C2CN(CCOCC)C2)CC(NC(=O)C=C(C)c2ccco2)CC1=O C1(NC(C2CC(C)(C)C(=O)NC2)=O)CC2(CCCCN2C(C2CCOCC2)=O)C1 Cc1ccc(C=CCC(N2CCC(O)(CNC(c3ccc(Cl)o3)=O)CC2)=O)cc1 C1(C(=O)NCC(CC=C)NC(C)=O)C2CN(C(c3ccccc3F)=O)CC12 CC1C(NC(=O)Cc2cccs2)CCN1C(=O)CC1CCN(C)C1=O Cc1ccc(C)c(SCC(=O)NC23CCC(C2)N(C(c2ccc(=O)oc2)=O)C3)c1 C1(C)(C(=O)NCCC2CCCC(C)C2)CCCN(C(=O)Cc2n[nH]c(=N)s2)C1 CC1CCC(CC(=O)NC(c2ccnn2C)C(N2CCC(O)(C(N)=O)C2)=O)CC1 N1(C(C2C(CNC(C3(CCCC)CC3)=O)CCC2)=O)CC2(C1)CN(C)C2 C1(NC(C2(C#C)CCC2)=O)CCOCC1NC(C1CCCN1C(=O)NC(C)C)=O N1(C(C(C)OCCCC)=O)CCN(C(=O)COC2CCC2)C(COC)C1 c1(NC(CC2(C)CCN2C(N)=O)=O)cccc(C(C2CC2)C2CC2)c1 N1(C(C(CC#C)NC(c2cccc(OCC)n2)=O)=O)CCN(CC)C(C)C1 C1(CNC(C2CCN(CC)C2)=O)CC(C)(C)CN1C(c1csc(C)c1C)=O c1(C(N2CCCC2C)C(=O)NCCOC)cnn(C(C)CC)c1 Cc1cnc2n1C(C(=O)NCC1CN(C(c3cncn3C)=O)CCO1)CCC2 CC1(CSc2cn(CC(=O)O)nn2)CCCO1.C12CCC1C(=O)N2 c1(N(C(c2ccsc2NC(=O)OC(C)(C)C)C(=O)NC(C)C)C)cccc(Cl)c1 C1(C2CN(C(=O)CCCC3OCCO3)C2)(NC(CC2N(C)CCOC2)=O)CC1 C1(CNC(c2nnnn2C2COC2)(CC)C2CCC2)CC2C(C1)C2(F)F N1(C(=O)CCC2CC(F)(F)C2)CCCN(C(c2csc(C3CC3)n2)=O)C(CO)C1 C#CCCCCCCC(=O)NC(CC#C)CC(=O)N(C)Cc1cn[nH]c1 c1(C(CN2CCC(=C)C2)N(C(=O)CCSC)CC)ccccc1F c1(C(N2CC(F)CC(NC(C(CC)O)=O)C2)=O)noc2c1CC(F)(F)CC2 c1(COC(C(CCCOC)C)=O)csc2cc(Br)ccc12 Cc1c[nH]cc(-c2nc(-c3cccc(C(F)F)c3)nn2CC2CCCCC2)c1=O O=C(C#CC1CCC1)N1CCC(NC(C2(F)CCC2)=O)C(O)C1 CC1C(=O)C2(CC2)CC2(CC2)CS1.C1(NC=O)CCCC1.C(C)(C)C.C1(=O)CN1 CCS(=O)(=O)CC(=O)NC1CCC(NC(c2cnc(C3CCC3)s2)=O)CC1 n1(CC)nc(C(=O)NC2CC2CNC(=O)C(C(C)O)N(C)C)cc1C1CC1 c1(OC)cc(=O)n(C)cc1C(=O)NCC1CC(O)(CNC(c2coc(C)n2)=O)C1 C(=O)(C(C)COC)N(C(C)C(=O)NC(CCO)C1CCCC1)CCC N1(C(C2(OC)CCSC2)=O)CCC2(CC1)OCCC2NC(c1csc(C)n1)=O CCCCC(CNC(C1(CO)CC(C)(C)C1)=O)NC(C1CC2CCC2C1)=O C(CCCCNC(C1CCC1C#N)=O)N(C(=O)C=CC(C)(C)C)C N1(C(c2c(C(=O)OCC)con2)=O)CCN(C(=O)Nc2ccon2)C(C)C1 C1(CC=C)(NC(=O)C(C)c2cccs2)CN(C(c2cn(CCOC)nn2)=O)C1 C1(C(N2CCC(C)C(NC(=O)COCCCF)C2)=O)CCc2nnc(O)cc2C1 CC1=NNC(=O)C1CC(=O)NCC1CN(C(c2[nH]cnc2C(C)(C)C)=O)C1 C1(C(N2C(C)CN(C(c3cccs3)=O)CCC2)=O)COc2cc(Cl)ccc2C1 CC1CCC(NC(=O)CCn2ccnc2)CN1C(C1COC(C)(C)CO1)=O c1(C(=O)NCC2CC(C(=O)NC3CC(OC)C3)C2)ccc2[nH]ccc2c1 C(CC(O)C(=O)OC)OC(Cc1nc(C(=O)OCC)sc1)=O Cc1nc(-n2ccnn2)ncc1C(=O)NCC(N1CCN(C)CC1)=O c1(C(N(C2CCN(C(C(CC)(F)F)=O)C2)C)=O)ccnc2c1nnn2C CC(C)CC(CC(C)C)C(=O)NC1CCN(C(=O)C(C)N2CCCC2)C(C)C1 Cc1nc(O)ccc1C(=O)NC(C1CCOC1)CNC(C1CC2(C1)CC(O)C2)=O c1(C2C(C(N(C)Cc3cncs3)=O)C2)cccc(-c2cncnc2)c1 C1(NC(COCC=C)=O)CCCC2CN(C(=O)C=Cc3ccc(F)c(C)c3)CC12 n1(CC(N2C(CCCNC(c3nc(COC)sc3)=O)CCC2)=O)cnc(C#N)n1 c1(OC)ccc(OC(F)F)c2cc(C(=O)NCC(C)(C)n3ccnc3)[nH]c12 N1(CC(N2CCC(C(C)(C)NC(C3(F)CCOC3)=O)C2)=O)CCCCCC1=O Nc1nc(C(N2CCCC(CCNC(=O)CSc3cccs3)CC2)=O)ccc1O C12(C(=O)NCC3N(C(c4ccc(O)nc4)=O)CC(F)C3)CCCN1S(=O)(=O)CC2 C1(COCC)CCN(C(=O)CCN(CCO)C(c2ncsc2CC)=O)C1 C=CC(C)(CC)C(=O)N(CCCCCC(=O)N1CCC(OC)C1(C)C)C c1(COC(c2c(Cl)cn(CCC)n2)=O)ccncc1C#N C1(OC)CC(NC(c2ccc(F)cc2Cl)=O)CN(C(=O)Cc2ccc(O)nc2)C1 C1(C(N(CCCCN(C(CN2CC(C)C2)=O)C)C)=O)CCC(F)(F)C1 N1(C(COC(CC)C)=O)CCC(NC(c2ccc(C)c(N)c2)=O)C2(CCC2)C1 c1(N2CCN(CCNC(CC(CC)OC)=O)CC2)cc(=O)n2oc(C)cc2n1 c1cc([N+](=O)[O-])ccc1Br.Cc1ccc(-c2nc(C(OCOC)C)c(C)s2)cc1C N1(C(COC)=O)CCC(CCNC(=O)CCc2ccc(Cl)c(Cl)c2)CC1C CC1(C)CCCC(C)(C)C1C(N1CCN(C(=O)C(F)F)C(C2CC2)C1)=O Cn1ncc2c1CCCC2N=c1[nH]ccc(=NCCC2CCN(C)C2=O)[nH]1 CC#CCC(C(=O)N(CCSC)CC)NC(c1cccc(C(=O)OC)c1)=O N=c1cc(C2CN(C3CCC3)C2)cc[nH]1.C12(c3cccc(F)c3)CCN(C1)C2=O C(=O)(C(CC(C)C)OC)NCC(=O)N(CC=C)Cc1ccccc1 C1(NC(Cc2n(C)nnc2)=O)CCC2CN(C(=O)Cc3ccccc3O)CC2C1 Cc1nc([N+](=O)[O-])cn1CCC(=O)NC(C)CNC(c1n[nH]cc1C(C)(C)C)=O c1(NC(C2C(NC(CCOC(C)=O)=O)CCC2)=O)cc(Cl)ccc1C Cc1nc(C(=O)NCC2(C)CCN(C(=O)CC3CCCO3)C2)c(C)s1 N1(C(C2(CC=C)CCC2)=O)CC2C(CC(=O)NC3CC(CC(N)=O)C3)C2C1 c1(C(N2CC(C(=O)Nc3cncc(CO)n3)SCC2)=O)ccc([N+](=O)[O-])cc1F C#CC1(C(=O)NCc2cccc(F)c2)CN(C(=O)CCC(=C)C)C1 CC12CCC(C(=O)NC3COCCC3NC(c3ccncc3Cl)=O)(C1)OC2 C1(CNC(CCN(CCC(C)(C)C)C)=O)COCCN1C(=O)Cc1ccnn1C C=CCCCCCCCC(=O)NC(C1CCCN(C(C2(CSC)CC2)=O)C1)C c1(C(=O)NC(C)CNC(=O)C(F)n2cccn2)nn[nH]c1C(F)(F)F Cc1nc(C(=O)NCC(C)N(C)C(c2ccn(C3CCCC3)n2)=O)c(C)n1C Cc1nc2c(N3CC(NC(c4cc(F)c(F)c(O)c4F)=O)C(O)C3)ncnc2[nH]1 Cc1scc(C(=O)NC2CCC(CCNC(=O)C(F)(F)c3ccncc3)C2)c1C CC(C)CCCCC(=O)N1CCC(C(F)C(=O)NCCC2OCCC2(C)C)C1 C12(CNC(Cc3c(C)non3)=O)CCC1CCN2C(c1cnn(C(C)C)c1N)=O C(N=c1cc(C(C)C)n(CC)[nH]1)(c1cc(F)c(F)c(F)c1)c1n(C(CC)C)nnn1 c1(-c2ccn(C(C(=O)N(CCC(=O)OC)CC)C)n2)ccc(F)cn1 N1(C(Cn2c(C)ncc2)=O)CC(CO)C2(C1)CN(C(C1CCCCC(=O)N1)=O)C2 c1(C(=O)NCCC(CNC(CC(C)C(F)F)=O)O)sc2nccnc2c1N C1(NC(c2c(C)occ2)=O)CC2(C1)CC(CNC(c1cnc(C(C)C)nc1)=O)C2 CCC(CCC(=O)NC(C)(CO)C(=O)N1CC(CC(F)(F)F)C1)OC O=C(CCCC(F)(F)CO)NCC1CC2CCCC2N1C(=O)Cn1cnnc1O N1(C(C(COCC)C)=O)CC2(CC)CC1(CNC(=O)C(c1ccccc1)C)C2 C(=O)(CC(C)CC(=O)NCC1(CNC(=O)CCOCC(C)C)CC1(F)F)OC CC1C(C(=O)Nc2ccncn2)CCCN1C(=O)CCNC(N)=O c1(C(=O)NCCN(C)C(c2cc(-n3cnnc3)ccn2)=O)cc(S(N)(=O)=O)cs1 c1(Nc2scc(-c3sccc3)n2)cccc2occc12 C1(CC(=O)NCC(CNC(C(C)n2ccnc2)=O)O)CC(C)(C)C(=O)N1 C1(C)(C(=O)NCCCCC(=O)NC2(COCC)CC2)CCC(=O)NC1 C1(F)(C(=O)NCC2C(C)CCN2C(=O)CCc2cccs2)CCC(F)(F)CC1 CCCCC(F)(F)C(=O)N1CCN(C(=O)Cc2cc(C3CC3)on2)C(C(C)C)C1 N1(C(C(C)(C)C)=O)CCC(C(F)(F)F)C(CNC(=O)Cn2nnc(=O)[nH]2)C1 c1(OC)ccc2occ(C(N3CC4CC3CN4C3CC3)=O)c2c1 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CC(NC(=O)CCc1cccn1C)C2 N1(c2nc(C)nc(O)c2)CCC2(CCCCN(C(=O)CCOCC(F)(F)F)C2)C1 c1(C(=O)NCC(C)N(C(=O)C=Cc2ccsc2)C)cc(F)cc2c1C(=O)CC2 c1(C(N2CC(C(=O)NCCC3CCCO3)(COC)C2)=O)cncn(C)c1=O c1(C(=O)NCCC2CCCN(C(CN(CCOC)C)=O)C2)cccc(CO)c1C C(=O)(C(F)CC(C)(C)NC(=O)C=C1CCCCC1)NC(C)CN(C)C c1(SC)cc(C)ccc1C(N1CCC(NC(=O)CN2CCC(C)(C)C2)C(O)C1)=O c1(C(=O)NC(CNC(c2cnc(CC)[nH]2)=O)C)cc(Cl)cc([N+](=O)[O-])c1 C1(OC)CC2CC1CN(C(c1occc1CNC(C13CCC(CC1)CC3)=O)=O)C2 C1(F)(CNC(C2C(C)C2C)=O)CCCN(C(=O)C=Cc2ccc(C(N)=O)o2)C1 C1(CC)CC(C(=O)N2CC3CC3(CNC(C3(OC(C)=O)CC3)=O)C2)=NO1 c1(C(CN(C(=O)CC2CCC(NC(C3CNCCO3)=O)C2)C)O)ccc(O)cc1 c1(CN(C(=O)CN2CCS(=N)(=O)C(C)C2)CCC)cccc2ccccc12 C1(C(=O)NC(C2CCN(C(=O)CN3CCOCC3=O)C2)C)CN(S(N)(=O)=O)C1 C1(CNC(c2cncc(Cl)c2)=O)(CO)CCCN(C(=O)C(F)CC2CCOC2)C1 C1(CN(C)C(c2ccn(C)c2)=O)CN(C(=O)CCc2ccc(=N)[nH]c2)CCO1 c1(CC(=O)N(CCO)CC2COC(C)(C)O2)cc(Br)cc(Br)c1 Cc1nc2n(n1)CCCC2NC(=NCCCc1cn[nH]c1)NCC(C)C c1(OC)ccc(CN2CCN(C(=O)NCc3cnc(F)c(C)c3)CC2)cc1OC c1(C(C)=O)cccc(OCCC(=O)NC(C2CCN(C(=O)CSC3CC3)C2)C)c1 CCCC(C(=O)OC)C(=O)N1CC(NC(c2ccc(Cl)s2)=O)CC2(CC2)C1 C1(C(N(CC(CC)NC(=O)CC2(CC)CCC2)CC)=O)CCCCCN1C c1(C(N2CC3CN(C(c4[nH]c(=NC)sc4)=O)CC3C2)=O)cc2ccccc2n1C C1(C2CC2)(NC(=O)Cc2ccno2)CCN(C(C2(C3CCCCO3)CC2)=O)C1 C1(C(=O)NCC(c2cnc[nH]2)C)CCCCN1C(c1cnnn1C)=O C(CC(C)C(=O)NC(C)(CNC(=O)Cc1ccccc1)C1CC1)=CC Cc1sc2ccccc2c1C(N1CCN(C(=O)C(C(C)O)N(C)C)CC1)=O c1(C(C(N2CC(OC)(CNC(c3[nH]ccc3C)=O)C2)=O)=O)ccc(C)cc1 CC1(NC(C2CCNC(=O)C2)=O)CCC(NC(c2cc(F)cnc2O)=O)CC1 c1(C(=O)NC2(C(N3CC(CC(C)OCC)C3)=O)CC2)cc(F)cc(F)c1N N1(C(Cc2c(C(C)C)con2)=O)CCC(NC(=O)CCC(=O)N(C)C)C(O)C1 C1(NC(=O)C(F)=C2CCC2)CCC(N2C(=O)CCC2=O)CC1 C(=O)(C(=O)C(C)C)NC1(CC(=O)N(CCC=CCCC)C)CC1 c1(C(=O)NC2CN(C(CC=CC=C)=O)CC2C)ccn2[nH]c(=N)nc2c1 c1(NCC(CCCC)NC(c2cc[nH]n2)=O)nccc(C(N)=O)c1[N+](=O)[O-] n1(Cc2c(C(=O)NCC3CN(C(C(=O)NC)=O)C3)cno2)nc(C)cc1C Cc1[nH]c(C#N)cc1C(N1CC(NC(=O)C(c2ccc(F)cc2F)(F)F)C1)=O Cc1nn(CC(C)C)c(C)c1CC(=O)NCC(C)NC(C1CCCC(C)(C)C1)=O C1(C(=O)NCCCCOCC)CC(=O)N(c2cccc(C(F)(F)F)c2)C1 c1(C(=O)NC2C(CNC(CCC(C)OC)=O)CCC2)cnn2ccc(O)nc12 CC1CCCN(C(=O)CCn2cncn2)C1CCNC(=O)CCN1CCCC1=O c1(N2CC3N(C(C4CC(=O)NCC4)=O)C(CC3)C2)[nH]cnc2nc(Br)cc1-2 CC12CN(C(C34CCCC3C4(F)F)=O)CC1CN(C(c1cnsc1)=O)C2 N1(C(C(C=C)O)=O)Cc2ccc(CNC(C3(C)CC(=C)C3)=O)cc2C1 c1(C(=O)OCc2n(C(C)C)nnn2)cccc(S(C)(=O)=O)c1C(F)(F)F C(N=c1[nH]c2ccc(S(=O)(=O)NC3CCC3C)cc2s1)C1CC(CC)C1 C1(CNC(c2ncc[nH]c2=O)=O)CN(C(C2CCCC3(CC3)C2)=O)CC12CCC2 Cc1c(C(N2CCN(C(=O)C=C3CCCC3)C3CCC23)=O)oc2c(Cl)cccc12 N1(C(=O)NC2CCCN(C)C2)CCN2C3CCC(C3)C2C1 CC1CN(CC(F)F)CCN1C(c1ccsc1Br)C(=O)NC1(C)CC1 C1(C(=O)NCCC(O)CCO)(NC(C(c2cncnc2)C)=O)CCOCC1 C1(NC(C(CC)=CC)=O)Cc2ccccc2C1NC(c1ccc(Cl)nc1O)=O N1(C(COCC=C)=O)CC(NC(=O)CC2CSC2)CC12CCCCC2 C1(C(=O)NC2CC2c2ccccc2)C2CCC(C2)N1C(c1cccnc1O)=O C1(CC=C)(NC(=O)C(C)(C2CCC2)NC(c2occc2C)=O)CCCC1 c1(OC)ccc(C(N2CCC(O)(CNC(C3(N(C)C)CCC3)=O)C2)=O)cc1C C(CC(CO)N=c1ccn2ncc(C(=O)OC)c2[nH]1)=CC.N12CCN(CC1)NC2=O C1(NCc2c(N3CCN(CC)CC3)cccc2)CNC2(CCCOC2)C1 c1(CC)cc(C)ccc1NC(=O)C(C1CN(C(C2CCS(=O)CC2)=O)C1)OC c1(C(=O)NC(C(C)NC(=O)CC2CCCC2)CO)cc[n+]([O-])cc1 c1(C(N2CC=CC(C(N(CC=C)CC3CC3)=O)C2)=O)ccc(O)cc1F C(=O)(C(C(C)(C)C)N1CCOC1=O)NCCCNC(c1ccc(SCC)cc1)=O C1(C(=O)NCCC(=O)NC)CC2(CC(NC(C3CC3(Cl)Cl)=O)C2)C1 c1(C(c2nnnn2C2CCOC2)NCCOCC(F)(F)F)ccc(C(Cl)Cl)cc1 c1(C(N(C2CCN(C(c3sccc3C#N)=O)C2)C)=O)n[nH]c2c1CS(=O)(=O)CC2 c1(CN(CC#C)C(=O)NCC2(C)CC(C(F)(F)F)C2)ccccn1 N1(C(c2c(C)c(F)c(F)cc2)=O)CC(=O)NCC(C)(C)C1 C1(CC(=O)NC(CC(=O)NCC2(CC)CCC2)C2CC2)CCC(C)(C)O1 CN1CCCCC(NC(=O)C(=O)NCCc2cnc3n2CCOC3)C1=O C=CC1(C(=O)NC2C3CCCOC23)CCN(C(c2cncc(C#N)c2)=O)CC1 c1(C(N2CC(C)(C)C(NC(C3(C)CCC(F)(F)C3)=O)C2)=O)c(N)cc(Cl)cc1F CC1(C)CN(C(C23CCCC2C3(F)F)=O)CC(CNC(=O)CC2CCC2C)O1 c1(OC)ccc(OCC(=O)NC2CCCCC2NC(=O)C(O)C2CC2)cc1 c1(C(N2CC(CCNC(C3C(C#N)C3)=O)C2)=O)occc1F CC(C)CC(C(=O)N(C(C)CC(N)=O)C)ONC(c1ncsc1N(C)C)=O N1(c2c(C(=O)OCC)cncc2)CCC(NC(c2ncc[nH]2)=O)C2(CCC2)C1 c1(C(=O)NC(CCNC(C(C#C)(C)C)=O)C)coc2c1CS(=O)(=O)C2 Cc1cc(C(=O)NC2CN(C(c3cnn4c3OCCC4)=O)CC2F)c(C)nc1C Cc1cc(C)c(N(CCC(=O)NC2(N3CCCCC3)CCOCC2)C)c(Cl)c1 C1(C(F)(F)F)(C(=O)NC(C)CCNC(=O)C(c2ccnn2C)C)CC=CCO1 C12(C(N3CC(O)(CNC(CS(C)(=O)=O)=O)C3)=O)CC=CC(C1)OC2 N1(C(C2CCN(OC)CC2)=O)CCC(C)C(NC(c2nc(C)no2)=O)C1C c1(C(=O)NCCN(C(c2cccc(F)c2Cl)=O)CC)c(N)cccc1F c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cc(C)c(Cl)s2)=O)C(CO)C1)=O N(C)(C1c2ccccc2CC1O)C(=O)NCC(C)SC C1(CNC(=O)CCC2CCOCC2)CCN(C(C2CCOC(=O)CC2)=O)C12CC2 c1(C(=O)NC2CC(C(=O)NCCN(C)C)C2(C)C)ncn2ccccc12 c1(OC)ncc(Cl)c(C)c1C(N1CCOCC(CNC(C2CCCN2C)=O)C1)=O C(=O)(N=c1cc2n([nH]1)CCCC2)C1CCN(C(C2C(C(=O)OC)C=C2)=O)C12CC2 C1(NC(C(N2CCOC2=O)C)=O)C=CCC(C(=O)NCC2(C)CC2CO)C1 C(=O)(C(C)(F)C(C)(C)F)Nc1c(C(=O)OC)c(OC(C)C)n(C)n1 c1(C(=O)NC2(CC)CCCN(C(=O)C3=CCC3)C2)ccnc2c1CCO2 N#Cc1cnn(CC(=O)NC2(CNC(c3cncs3)=O)CCCCC2)c1N C1(CNC(c2c(NC)snc2C)=O)CCN(C(=O)Cc2sc(C)cc2C)C12CC2 C#Cc1ccc(C(N2CCC(O)(C(C)NC(=O)COCCN(C)C)C2)=O)nc1 C1(C(N2CCN(C(CCCC(OC)OCC)=O)CC2)=O)CN2CCCN1CC2 c1(NC(C2CCN(C(c3ccno3)=O)C2)=O)cc(F)c(Br)cc1F C(=O)(C#CC1CCOCC1)N(CCN(C(c1sccc1COC)=O)CC)CC C(=O)(C(C)(C)C(C)(C)O)N1C(CNC(C2(C)CCCS2)=O)CC(O)C1 N1(C(C2(C)CCCNC2=O)=O)CC2(CCOCC2)CC1CNC(=O)CC1(O)CC1 c1(CNC(CCN(C2CCCCC2)C)=O)cnccc1Cl.C12CCN(C1)C2=O c1(OC)ccc(F)c(CN2CCCC2c2ccccc2Cl)c1Cl Cc1cc(CC(=O)NCC2CN(C(=O)CCC3CC3(F)F)CCO2)cc(C)c1 C1(NC(CC(C(=O)O)NC)=O)CC2CCC(C1)N2C(c1ccncc1OC)=O c1(C(=O)NC2(CCOC)CCN(C(=O)CCC3CC3(C)C)C2)ccc(Cl)cc1C Cc1oc(C)c(C(=O)NCCN(C2CCCC2)C(C2(C)CCCO2)=O)c1C c1(NCc2cn(CCOC)nc2)[nH]c(=NCCC2(C)CC2(Cl)Cl)nc2sccc12 CCC(CC)(CO)C(=O)NC1CC(CNC(c2cnc(C3CCC3)o2)=O)C1 C1(CNC(CCN2CCC(C#N)(F)C2)=O)CC2(CCC(F)(F)CC2)CO1 c1(OC)cccc(C(=O)NC2CCC(CNC(C3CC3C(C)(F)F)=O)CC2)c1F c1(CC(=O)NCC2N(C(CC(C)(C)OC)=O)CCC2)n[nH]c2ccccc12 C1(CNC(CCC)=O)CCC(C)CN1C(c1ccc(CN(C)C)nc1)=O N1(c2nccc(OC)n2)CC2(C1)C(NC(=O)CC1CC3(CC3)C1)CCS2(=O)=O N1(C(c2c(OC)nccc2)=O)CC(CNC(C2CC(SC)C2)=O)C2(CC2)C1 Cc1cc(CC(=O)NCC2CCCC(NC(c3ccncc3N)=O)C2)cc(C)c1 C1(NC(C(CC)n2cncn2)=O)CCC2CN(C(=O)Cc3csnn3)CCC2C1 n1(C(C)CN2CCCCC2)nc(-c2ccc(N(C)C)cc2)nc1CC1C=CCCC1 C(=O)(C1=CC2C=CC1C2)N1CC(C(=O)NC(C)C(N)=O)N(C)CC1 C1(N(C(=O)CC2CC2)C)CN(C(=O)CC2CCCNC2=O)CC12CC2 c1(C(=O)NCCCC(C)NC(=O)C(C)(C)c2cscn2)cc(Cl)ccn1 C(=O)(CCC(C)(C)C#N)NCCC(C)N(C)C(C1CCCC2CC12)=O C1(NC(=O)CC2CCOC2)CC12CCN(C(=O)C1=CC3C=CC1C3)CC2 c1(C(=O)NCC(CCNC(CC(CC)C)=O)O)ccc2ncccc2c1F C1(C(C)(C)C)CCC(C(=O)NCCCNC(=O)C(O)CC2CCCCC2)CC1 c1(OC)cc(C=CC(=O)NCCc2cn(C(C)(C)C(=O)O)nn2)cc(OC)c1OC C1(CNC(C(=O)NCCOC)=O)CN(C(c2nn(C(F)F)cc2Cl)=O)CCO1.CSC C1(NC(c2c(C)cns2)=O)CCN(C(=O)CN(S(C)(=O)=O)C)CC1 C1(CC(=O)NCC2C3CN(C(c4sccc4C(F)(F)F)=O)CC23)CCCOCC1 c1(C(=O)NCC(CN(C(=O)Cn2ncnn2)C)O)ncc(C(F)(F)F)cc1Cl Cc1ccn2ncc(C(=O)N(C3CCC(NC(C4(CCF)CCC4)=O)C3)C)c2c1 C1(C(N(CCC(=O)OCC)C)=O)CC(NC(c2ccnc(C)n2)=O)CCO1 C1(CCO)CCCN2N(Cc3cccs3)C1CCc1c(Br)cccc1C2 CCC(F)(F)C(=O)NC1CN(C(=O)Cc2cc(OC)no2)C2CC12 C(C(CC)CCO)NC(c1noc(C)n1)(c1nnnn1CCCSC)COC C(CN=c1[nH]c(=NCc2ncoc2CO)[nH]c2cccnc12)N1CCCC(C)(C)C1 N1(C(c2ccc(OC)nn2)=O)CC2(CCN2C(c2ccc(C(C)(C)C)cc2)=O)C1 C1(CC#C)(C(N2CCN(CCNC(C3(C#N)CC3(C)C)=O)CC2)=O)CC=CCC1 c1(-c2onc(C)n2)cccc(NC(N2CCCC2c2n[nH]c(C(C)C)n2)=O)c1 C=CC(C)(O)C(=O)NCCN(C)C(C1COCC1(C)C)=O C1(CC(N2C(CCNC(c3c(CC)occ3)=O)CCC2)=O)CCC(C#N)C1 Cc1nc(C)c(CCC(N2C3CCC(C3)C2CNC(=O)C=CBr)=O)c(O)n1 CCC(C)C(CO)NC(C1C=CCCN1C(=O)C(C)N(C)C(C)=O)=O C1(NC(=O)CC(F)(F)c2ccccc2)CCN(C(=O)C=C(Cl)Cl)CC1F C=CCCC(C)(C)C(=O)NCC=C1CCN(C(c2ccc(Cl)nc2N)=O)CC1 c1(-n2c(-c3ccc(C(C)O)cc3)nc(C3CCOC3)n2)ccnc2cccnc12 C1(N(C)C)CCCC(C(=O)NCCCN(C(c2csnc2Cl)=O)CC2CCCC2)C1 Cc1noc2cc(C(=O)N(CC(C)NC(=O)COc3ccc(F)cc3)C)ccc12 c1(C(=O)NCCCN(C(CCc2c(C)cccc2)=O)C)cn2cccnc2n1 C(=O)(C(C(F)(F)F)NC(C)=O)NCC(CNC(CC(=O)NCC)=O)OC Cc1ccc(C(=O)NCC2CN(C(c3cscn3)=O)CC2(C)C)cc1S(C)(=O)=O c1(C(N2CCOCC2)=O)ccc2ccoc2c1.N12CCCC(C1)COC2=O c1(CNC(C2N(C(C3(N(C)C)CCCC3)=O)CSC2)=O)ccncc1F CC(C)(CC(F)(F)F)C(=O)NCC1CC(F)CN1C(C1Cc2nccnc2C1)=O N1(C(C2C(NC(CCOCCN(C)C)=O)CCOC2)=O)CC2(COC(=O)N2C)C1 c1(COC(C(C2CCCOC2)OC)=O)ncccc1Cl C12(NC(CCCN=[N+]=[N-])=O)CCCCCC1N(C(c1cnc(F)c(Cl)c1)=O)CC2 C(=O)(CC(C)(C)C(C)(F)F)N1CC(N(C(C(C)=C2CC2)=O)C)C(C)(C)C1 N1(C(c2ccccc2F)=O)CCC2C(CCN2C(=O)CCCC2CCCC2)C1 C1(F)(C(=O)NCc2c(C)ccs2)CCCN(C(=O)CC2CCC(=O)N2C)C1 c1(C(N(CC(C)NC(C(C(CC)CC)C)=O)CC)=O)cccc2ncnc(O)c12 c1(CC)nn(C)c(C(N2CCC3(C(=O)NC(C)(C)C#N)CC3C2)=O)c1Br C(=O)(CCCCC(C)C)N1CC(C)(OCC(=O)NC(C2CCCO2)CC)C1 C1(OC)CCC2(C(=O)NC(C)C(C)(C)NC(c3cnc(O)c(C)c3)=O)CCC12 c1(C(N(CC(O)CN(C)C(C2(C)COCCO2)=O)C)=O)cnc(C2CC2)nc1O C1(CC)CN(C(C2COCCN2C)=O)CCN1C(c1csc(-c2cnc[nH]2)n1)=O C1(C(N2C(CN(C(CNC(CC)=O)=O)C)COCC2)=O)CCn2nncc2C1 c1(C(=O)NC2CC(NC(C34CCCCC3CCC4)=O)C2)coc(=O)c2ccccc12 c1(C(=O)NC(C(C)NC(c2cncc(C#N)c2)=O)C)cc2cnc(Cl)cc2s1 N1(C(c2c(CC)nns2)=O)CCC2(CC2)CC1C(=O)N(C1CCC1)C C(CCCC(=O)NCC(C)(C(C)C)NC(C1CCC(OC(F)(F)F)CC1)=O)OC C1(NC(C2CCSCC2)=O)CC2CN(C(=O)CCCCCF)CC2C1 C(CC(CC)C(=O)NC1(CO)CCN(C(c2cnn3c2OCC3)=O)CC1)=CC C1(CC)CN(C(c2cnc(CO)nc2C)=O)CCN1C(=O)C=C(C)c1ccsc1 CC1(C)CCCC(C(=O)NCC(O)CC(=O)NCC2CCOCC2)C1 CCC(CC(=O)NCC1CCCN(C(c2ncc(Cl)n2C)=O)C1)C(C)C c1(NC(C2CN(C3CN(C(C(C)(F)F)=O)C3)C(=O)C2)=O)cc2ncccc2[nH]1 c1(C(=O)NC2CCCN(C(C3CCCCC3)=O)CC2F)ccc2c(n1)CCOC2 Cc1ccc(C(=O)NCC2(NC(=O)C3=C(Cl)CC3)CCCCC2C)c(N)c1Cl c1(C(=O)NCc2ccc(CNC(C(C)O)=O)cc2F)cccc2c1OCCC2 c1(C(N2C(C(=O)Nc3cc(C)cc(Cl)n3)CC(F)C2)=O)cncc2ccccc12 S(=O)(=O)(c1ccc(C)c(C)c1)NCCC(=O)NC1C(CNC(C(C=C)(C)CC)=O)C1 c1(N(C)C)ccc(NC(c2nc(C(=O)Nc3cccnc3)cs2)=O)cn1 c1(C(C(=O)NCC(C)NC(c2cc(OCC)no2)=O)N(C)C)ccc(Br)cc1 C(CN=c1[nH]cncc1I)OCCN(C(=O)CC(C)(O)C(F)(F)F)C CC1CCN(C(c2ccnn2CCF)=O)CCN1C(=O)CNS(N)(=O)=O C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1CC2C(NC(CNC(=O)NC)=O)C2C1 C1C(C)(C)OCC(=O)N1.c1(C2C(CNCC)C2)ncc[nH]1.C=CCCC(CO)=O c1(CC)ccc(C(C)=CC(=O)NCC2CCCN2C(C2CC2C(C)(C)O)=O)cc1 CC(C)C(C(=O)N1CCC(CNC(c2cnn(C(C)C)n2)=O)CC1)n1cnnn1 C1(C(N(CC(C)(C)CNC(=O)C=CSC)CC)=O)CCc2ccccc2O1 C1(NC(CCCOCCC)=O)CC(C)CN(C(c2ccccc2OCCC)=O)C1 C(=O)(C(F)(F)CC(C)C)NC(CC=C)CNC(=O)Cc1c[nH]ccc1=O C1(NC(N(CC#C)Cc2cccnc2)=O)CCCCC1OC CCC(CC)CCC(=O)NC1CN(C(=O)C(c2ccc(F)cc2)(C)C)CCC1C C1(NC(C(C)N=[N+]=[N-])=O)CC2(CCC(NC(=O)C=C(Cl)Cl)CC2)C1 N#Cc1ccc(-c2ccccc2CN2CCC2Cc2ccc(F)c(F)c2)cc1OC Cn1nnnc1CC(=O)NC1C(NC(CS)=O)C1.C(=O)(CCC1CCCC1)N S(=O)(=O)(CC(C1CC1)N(C)C)N(C)CCc1nnc(-c2ccccc2Cl)o1 c1(C(N2CC=CC(NC(CCCSC)=O)C2)=O)ccc(-c2cccs2)cc1F C1(CNC(Cc2nc(C)c(C)[nH]2)=O)CCN(C(C2C3C4CCC(C4)C23)=O)C12CC2 C1(C(=O)NCC=C=C)C2CN(C(C3(CO)CCOC3)=O)CC12 N1(C(C(N2CCOCC2)C)=O)CCN(C)C(CNC(=O)C)C1.c12ccc(cc1)s2 C1(O)(CNC(=O)CC(=O)NC2CC2)CCN(C(C2CC3(C2)CC(O)C3)=O)CC1 C(C(CNC(c1ccnc(C(=O)OC)c1)=O)S(C)(=O)=O)NC(CC1C(CC)C1)=O Cc1nn(C)c2ccc(C(N3CCN(C(=O)Cc4ccsn4)C(C)C3C)=O)cc12 C1(CNC(Cc2ccc(C)s2)=O)CC(F)(F)CN1C(=O)CCOC1CCC1 c1(C(=O)NC(C)CNC(c2cc3sccc3cn2)=O)cc2n(n1)CCCC2O Cc1ccccc1C(=O)NC1(CF)CCN(C(=O)CCCn2cncn2)C1 N1(C(C)C(=O)NCc2cnccn2)CCCOC(CNC(=O)CC(F)(F)F)C1 C12(C(=O)NCc3ccc(C)nc3)CCN(C(c3c[nH]cc3C)=O)CC1C2 N1(C(CCNC(C)=O)=O)CCC2(C1)CN(C(=O)Cc1ccnc(F)c1F)CC(C)O2 N1(C(CCCN(C)CC2CCCC2)=O)CCCC(C(=O)NC2CCCC(=O)N2)C1 C1(NC(C2C(C)(CC)C2)=O)CC2CN(C(=O)Cc3ccc(Cl)nc3)CC12 N1(C(C=CC(CC)C)=O)CCC(NC(=O)CCc2nc[nH]n2)C1(C)C C(=O)(C1=NNC(=O)CC1)N1C(CN(C(=O)CCCCCC#N)C)COCC1 C1(CCC)C2CN(C(c3ccc(CC)cc3)=O)CC12.C12(CCOCC1)OC2 c1(C(=O)NCC(CNC(c2ncn(CC)n2)=O)C)cc(C2CC2)ccc1F c1(SC)cc(C(=O)NC2CC2CNC(c2ncoc2-c2ccco2)=O)sc1C Cc1csc(=NCC(=O)N2CCCC2CNC(C2CCc3nccn3CC2)=O)[nH]1 CCC(C(=O)NC1CC(C)(NC(c2csc(C(C(Cl)(Cl)Cl)OC)n2)=O)C1)C(C)O N1(C(c2c(C)[nH]c(C)c2C)=O)CC2(CCN(C(C3CCC(=O)N3C3CC3)=O)C2)C1 Cc1ccc2c(=O)c(C(=O)N(CC(O)CNC(C3CC=CC3)=O)C)c[nH]c2c1C N1(CCCC(=O)NCCCC2CCN(C(CC=C=C)=O)CC2)C(=O)CN(C)C1=O c1(NC(=O)OC(C)(C)C)cccc(C(N2CC(C3C(C(=O)O)C3(F)F)C2)=O)c1F c1(C(=O)NC2C(NC(c3c(C)noc3)=O)CC2)cc(C)c2[nH]nnc2c1 c1(C(N(C2CCN(C(=O)C(C3CC=CC3)C)C2)CCC)=O)ccc(N)cn1 C1(CC)CN(C(c2c(C)coc2C)=O)CCN1C(C1OC2CCC1CC2)=O CCCC(C(=O)N1CC(N(CC)CC)C1)NC(=O)C(C)c1ccco1 C(=O)(CC(C)(C)C(=O)N1CC2CCN(C(c3cc(Cl)cnn3)=O)C2C1)OCC c1(C(=O)NCCOC(C)(C)CNC(=O)CNC=O)cc2c(F)c(F)c(F)cc2[nH]1 N1(C(COC(C)(C)C)=O)CCC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C12CCCC2 C(=O)(CCP(C)(C)=O)N(CC(C)CNC(c1cc(-c2cccs2)on1)=O)C C1(C)(C(=O)NC2(CCCC(N(C(CC)=O)C)=O)CC2)CCC(C)C1 Cc1cc(C(C(=O)NCCCF)N(C2CC3CC3C2)C)cnc1C c1(N2C(C)CCC(CC)C2)ccc(S(=O)(=O)NCC2(F)CCOCC2)cc1F C1(CNC(CCc2scc(C)n2)=O)CCN(C(=O)CCc2cnc[nH]2)C1(C)C Cc1c(C(=O)NC2CN(C(c3cc(C(F)F)n(C)n3)=O)CCC2C)cccc1Cl Cc1nocc1C(=O)NCC(C1CCOC1)NC(c1cnoc1C)=O c1(-c2onc(Cc3c(COCCOCC)occ3)n2)ccc(Cl)cc1 c1(C(=O)NCC2C(CNC(C(C)(C)OC)=O)C2)cc2c(s1)CCCNC2=O c1(C(=O)NC(C2(O)CCN(C(=O)CC(C)(C)C)CC2)C)cc2cccc(Cl)c2[nH]1 c1(NC(=O)C(C)OC(=O)C(C)SC)ccccc1.c1(C(CC)C)ccccc1 c1(C(C)C)n[nH]c(=NCC2CCC(NC(c3cccc(NC(N)=O)c3)=O)C2)o1 C1(C(=O)Nc2c(CCC(=O)OCC)nccc2)CCc2n[nH]cc2C1 C1(C(=O)NC2C(C(N3CCC(C(CC)C)CC3)=O)CC2)CC2(CCC2)CO1 c1(C(=O)NCC2C(NC(c3ccn(CC)c3C)=O)CC2)cc2c(s1)CCCC2 Cc1ncc(NC(C2CC2C(C)NC(c2cccnn2)=O)=O)c(C)n1 c1(C(=O)NC(C)C(C)NC(=O)C=Cc2cnc(O)nc2O)ncc(C#N)cc1Cl c1(CN(C)CC)cccc(C#N)c1.C1(=O)CCC(=O)N2CCOC(C2)N1 N1(C(C2CC23CCC3)=O)C2CCC1CC(c1cn(-c3ccccc3F)nn1)C2 C1(C2(N(C(c3ncc(C)o3)C(=O)Nc3ccccc3)C)CC2)NC(=O)NC1=O Cc1ncnc(O)c1C(=O)NC1CC(C)(CNC(C23CCCC2CCC3)=O)C1 C1(F)(C(=O)NCC2N(C)CCCC2)CCCN(C(=O)CC2CCCO2)C1 C1(N(C)C(C2C3CCC2(c2ccnn2C2CCCCO2)C3)=O)CC2(CNC2)C1 N1(CC(C)NC(=O)CC2CCN2C(=O)C(C)c2ccco2)CCOC1=O C1(CN(C(C(OCC)OCC)=O)C)COCCN1C(=O)CCN1CCC1 CC(O)CCCCCC(=O)NC(C)(C)CCNC(c1ccc2nc(S)oc2c1)=O N1(C(c2scc(C)c2C)=O)CC2CCC1CC2NC(C1CC1c1ccccc1)=O C(=O)(C(CSCC)NC(=O)CNC(=O)CC1CC2CC2C1)NCCC C1(C(N)=O)(CNC(=O)CC2(C)CCCC2)CN(C(=O)Cc2nnc(O)s2)C1 C(C(CNC(=O)C(=Cc1cnn(C)c1)C)S(C)(=O)=O)NC(C(CCOC)OC)=O c1(CC)cc(C(N2CCCC(NC(=O)C(O)CC(C)C)CC2)=O)cc(F)c1 c1(CNC(C(CC2CC2(F)F)N(C)CC2(C(=O)OC)CCCC2)=O)ccccc1F C(=O)(C(Cc1cn[nH]c1)NC(=O)C(O)C1CCCC1)NC1(CC#C)CCC1 N1(C(C2N(C)C3C(C2)CCNC3)=O)CCC2CN(C(C34CC(F)(C3)C4)=O)CC2C1 c1(C(=O)NCCCCC(C)NC(=O)Cc2csnn2)cc(N)cc(N)c1 C1(CN(C(Cc2cn(CC)nc2)=O)C)CCCN(C(c2oc(C)nc2C)=O)C1 C(=O)(CC(O)C(C)C)NC1C(OC)CN(C(c2c(C(F)(F)F)cnn2C)=O)C1 C(=O)(C1=C(C)CCC1)N1CC(CCNC(C2(c3c(OC)cccc3)CC2)=O)C1 c1(C(N(C2CN(C(C3C(C)CCC3)=O)C2)C)=O)cnc2c(F)c(F)ccc2c1 C1(NC(C(CC2CCC2)NC(c2coc(CO)c2)=O)=O)C2CCC1CC2 CC(CCC(=O)NC1CCN(C(C2CN(CP(C)(C)=O)C2)=O)C1)S(C)(=O)=O c1(N2CC(C(N3C4COCC3CC(F)C4)=O)OCC2)ncnc2c(F)cccc12 C1(CNC(CC(=O)OC)=O)CCC(NC(=O)C=Cc2cncs2)CC1 c1(C(=O)NC2C(CNC(C3C=C(C)CS3)=O)CCCC2)n[nH]c2c1NCCC2 Cc1cc(Cl)ccc1C(N1CCN(C(C2CCC2(C)C)=O)C(c2cn[nH]c2)C1)=O Cc1c(C(=O)NC2CCN(C(=O)C(C)Sc3ncccn3)C2)cccc1[N+](=O)[O-] C(=O)(CCCCCC)NCCC(CNC(C1CC(CCC)OCC1)=O)OC N1(Cc2ccc(OC)c(O)c2)CC2(CN(C(=O)CCSC)CC2CO)C1 N1(C(CC(CC)C)=O)CCCCC2C1CCCN2C(c1cnc(O)o1)=O C1(=O)C(O)CCN1C.C1(=O)C(CN(C)C)N1C1CC(N(C)C)C1.C1CC1.N(C)C N1(C(=O)CC(C(F)F)n2ccnc2)CC2CCN(C(=O)CCn3cccn3)C2C1 c1(OC)cc(C(=O)NC2CN(CC(C)O)CC2(C)C)ccc1Cl C1(C(=O)NC(COCC)C(C)C)CN(C(c2cnns2)=O)CCO1 Cc1sc(C(=O)NC(C(C)NC(c2cc(O)ncn2)=O)C(C)C)cc1[N+](=O)[O-] c1(C(=O)NCC(C)(O)CNC(C2CN3CCN2CC3)=O)ccc(SCC#N)cc1 CCCCCCCCC(=O)N1CCCN(C(=O)CC2CC23CC3)C(CO)C1 C(C(N=[N+]=[N-])C(=O)N1CCCC(C(=O)N(C)CCc2nccs2)C1)OCC C(=O)(C#CC(=O)NCC1CC1NC(=O)Cc1ccc(OC(F)F)cc1)N(C)C C(C(CC(=O)N1CC(CNC(c2cccc3scnc23)=O)C1)C(F)(F)F)N(C)C C(C)(CCCCN=c1nc2[nH][nH]cc-2c(O)n1)NC(c1cnc(C)o1)=O CN1CCc2nc(O)c(C(=O)NC34COC(C3)C(NC(=O)CNC=O)C4)cc2C1 C1(NC(c2c(OC)csc2)=O)CC(C)N(C(c2cnn(CCF)c2)=O)C1 CCC(C)(CNC(=O)Cc1cnn(C)c1)C(=O)NCC(C)(C)CN(C)C c1(CC(N2CCC(O)(CCNC(CS(CC)=O)=O)C2)=O)nc2ccccc2s1 C1(CNC(CC2CCN(C)CC2)=O)CN(C(C2CCCC2C(F)F)=O)C(C)(C)C1 C1(NC(Cc2ccn(C)n2)=O)CCCCCN(C(C2CC2C(N)=O)=O)C1 c1(C(=O)NC2CCC(NC(C(C#C)(C)C)=O)CC2)cc(C)c(N)c(C)c1 c1(C(=O)NC(C(C)NC(c2c[nH]c(C(N)=O)c2)=O)CO)cnn2ccncc12 C(CCCCC(=O)N(C)CC1COCCN1C(=O)CCc1cnoc1)=CC N1(C(c2cc(Br)cc(Cl)c2O)=O)CC(c2ccccc2)C2(CCC2)C1 Cc1ccc(F)c(CC(=O)NC2CC3CN(C(=O)CCc4nc(C)no4)CC23)c1 CC1CCCCN1CCC(N1CCN(C(=O)C=CC2CCCO2)CC1)=O N1(C(C(C)(C)CCNC(C2SCCS2)=O)=O)CCC12CCCSC2 C1(CC)CCN(C(=O)CCc2nncn2C)C1C(=O)NC(C)CNC(=O)OC(C)C Cc1cc(C(=O)NC(CCN(C(=O)Cc2cncn2C(C)C)C)C(C)C)cnn1 c1(C(N(CCNC(C2CC23CCCC3)=O)C2CC2)=O)ccc(F)c2ccccc12 c1(C(C)C(=O)NCC(C)(C2CC2)NC(C2CN(C)C2)=O)ccc(F)cc1 c1(C(=O)NCC(CCC)NC(=O)C2=C(C)OCC2)cc(C)nc(C)c1O C1(O)(CNC(C2CCC(CNC(c3cc(C)c(C)[nH]3)=O)C2)=O)CCC(C)CC1 C1(C(=O)NC(CCCC)CO)C2CCC(C2)N1Cc1c(C(=O)O)cccc1Cl c1(C(=O)NC2CC2C(=O)Nc2cnccc2Br)ccc(O)c(C(F)(F)F)c1 c1(C(=O)NCC(CC)NC(=O)C(=Cc2ccc(F)cc2)C)ccn2nccc2n1 N1(C(C=CSC)=O)CCCN(C(=O)C(c2c(F)cccc2F)C)CC1C(C)C C(=O)(CC(CNC(=O)C(COC)OC)C1CCC1)NCC(NOC)=O C1(C)(C(=O)NC(C)Cn2cnnc2)CN(C(=O)CC2COCC2O)C1 c1(C(N2CCC(C)C2CNC(=O)CC2(C(F)(F)F)CCC2)=O)c[nH]c2nccc-2c1 c1(CCC(=O)NC2C(C)CN(C(C3(O)CCOC3)=O)C2)nc2cccnc2[nH]1 CC(C(=O)NCC1(F)CC(NC(c2ccnc(S)c2)=O)C1)C(C)(F)F N1(C(c2c(C)occ2)=O)CCN(C(c2cc(O)ccc2Br)=O)CC(O)C1 Cc1cccc2c1CC(C(N1CCCC1CNC(C1C3CCCCC13)=O)=O)O2 c1(C(=O)NCCOCCNC(C2CC2(Cl)Cl)=O)ccc(F)c(CN2CCCC2)c1 c1(C(=O)NC(C(C(=O)NC(C#C)CC(C)C)C)C)cc(O)ccc1F c1(-c2cn(CC(C)NC(C3(CO)CCC(C)C3)=O)nn2)cc(Cl)cc(Cl)c1 c1(C(=O)NCC(CNC(=O)C=CC(C)(C)C)OC)nc2ccc(C)cn2c1N N1(C(CC2C(C(=O)OC)C2)=O)CCN(C(C2CCCCN2C)=O)CC1C1CCC1 Cc1cc(C(N2CC(O)(c3cn(C(C)C(=O)N4CCCC4)nn3)C2)=O)nc(O)c1 c1(C(C(=O)NCCC(CNC(C2(CSC)CCC2)=O)O)=O)cc(F)c(F)cc1F C1(C(=O)NC(CCNC(C(C)c2ccsc2)=O)C)(C2CC2)CCCO1 C1(C(=O)NC(CC)CNC(C2(C)CC2C(F)(F)F)=O)CCCS(=O)(=O)C1 c1(C(N2CCC(CN(C(COC(CC)C)=O)C)C2)=O)ccc(Cl)cc1COC CC(C)CC(C)(C)C(=O)NC(C)CCCNC(=O)C(C)CCc1ccccc1F C1(NC(C(CCC(=O)OC)C2CC2)=O)CCCN(C(c2ncoc2CC2CC2)=O)C1 Cc1ccc2cc(-c3cccc(N4CCN(Cc5ncn(C)n5)CC4)c3)[nH]c2c1 c1(CC)cc(C)ccc1C(=O)N(CCCNC(C1(C)CCCC1)=O)CCO C1(C(C)(C)C)CN(C(C2CCNC2=O)=O)CCN1C(c1ccc(O)nc1Cl)=O C12(C(NOC(C)C)=O)CCC(CC1NC(C1CCCC3(CC3)C1)=O)C2 c1(N2CC(CC=C)(NC(=O)CCCCCF)C2)ncnc2sc3c(c12)CCC(C)C3 c1(CNC(C(CC)n2cc(CC(O)C3CC3)nn2)=O)ccc(C)c(Cl)c1 CCC(CC(=O)NCCC1CC(NC(C2C(C)(C)C2(C)C)=O)C1)C(C)(C)C c1(C(=O)NCC2(OC)CN(C(C(C)=C(CC)C)=O)C2)cn2ccc(F)c(C)c2n1 Cc1cc(C(=O)N(CCC(C)NC(c2cnn(C)n2)=O)C)nn1C(C)C1CC1 C(=O)(CCCCC(C)=O)NC1C(NC(c2ccc(OC)cn2)=O)CCCC1 Cc1cccnc1C(=O)NC(C(C)NC(c1ncccc1F)=O)C(C)C C12(C(=O)NC3C(C)CN(C(=O)COC4CCOC4)C3)CC3CC(C1)CC(C)(C3)C2 C(=O)(C1CCCc2c[nH]nc21)NC(CCNC(c1nc(C)sc1)=O)C(C)C N1(C(C=Cc2c(C)csc2)=O)CC2CCN(C(C3CC4CC3CO4)=O)CC2C1 C1(NC(C2(CC)CCC2)=O)CCCC(CNC(c2cccnc2C)=O)C1 n1(CCN2C(=O)CCC2)ccc2cc(Br)ccc12.C(C)(C(F)(F)F)N(C)CCO.CS C1(CNC(C2C(CC)C2)=O)CC2(CC2)CN1C(c1ccc(C#N)[nH]1)=O c1(C(=O)NC2CCC(CNC(c3occ(C)c3)=O)C2)ccc(F)cc1Cl CC#CCCCCNC(c1ccc(CNC(c2cc(C)ns2)=O)cc1)=O CN1CCC(O)(CNC(=O)CC=CCNC(=O)C(F)C(C)(F)F)CC1 Cc1cc(N)c(C(N2CC(C)(NC(C3CN(C(N)=O)C3)=O)C2)=O)nc1C c1(C(=O)NCC2=CCN(C(C(C(CC)O)(F)F)=O)CC2)ccc2ccn(C)c2c1 N#Cc1ccsc1C(N1CSCC1C(N1CC2CC2C1)=O)=O c1(C(C(=O)N(C)CC2(OC)CCC2)NC(CCOCC)=O)c(C)cccc1Br C1(NC(COCC)=O)CN(C(c2cc(=O)c(OC)c[nH]2)=O)CC2(CCC2)C1 C1(C(=O)NCCC2CCCN2C)(CC)CCN(C(c2cnn(CCF)c2)=O)C1 Cc1nn(C)c2c1CC(NC(N1CCC(c3cccnn3)C1)=O)CN2 c1(C(=O)NC2CCCCC2C(F)F)ccccc1-c1nnnn1C1CC1 CN(C)NC(=O)CCC(=O)NCC(O)CC(=O)N1CCC(O)(CO)C1 C(CCNC(C1CCCSC1C)=O)(C(C)C)NC(C=CC)=O C=C(C)CCC(=O)N1CC(CSc2c(C(N(C)CCO)=O)cccc2)C1 n1(CC(=O)NCC(C)(CC(C)C)NC(C(CCOC)C)=O)c(C)cc(C)nc1=O c1(SCC)c(C(=O)NCC2CCOC2CNC(CC(=O)OC)C2CC2)cnn1C c1(CC)ccsc1C(=O)NCC1CCCN1C(=O)CC1CCCC1C CC1CCCC(C(=O)NCc2ccoc2C(=O)NOC(c2ccncc2)C)CC1 C1(NC(C(CC)F)=O)COC2(C1)CN(C(C1(C(F)(F)F)CC=CCO1)=O)C2 c1(CC(=O)NCC(C)NC(=O)C(C)CF)cc2ccccc2o1 N1(C(CC=CC=C)=O)CC2CCN(C(=O)Cc3ccnc(Cl)c3F)C2C1 CC1CC(NC(c2cnn3c2CCC3)=O)CCN1C(c1ccc(C#N)[nH]1)=O C=CCCC(F)(F)C(=O)N1CC2CC(C(=O)NCCNC(N)=O)CC2C1 N1(C(C2(C(C)(C)F)CCC2)=O)CC2CC1C2NC(=O)CN1CCCCC1 C1(CNC(CN(c2cnccn2)C)=O)CN(C(=O)CC2CCC2)CCN1C c1(OC)c(CN2CCCC(C)(C(=O)N(C(C)C(=O)N)C)C2)c(C)nn1C.N(C)C c1(C(N2C(C(=O)NC(CC)C(=O)NC)CC=CC2)=O)cnc(O)cc1C c1(C(=O)NCCNC(C2CC3C(C)(C)C3C2)=O)cc(Br)cc(Cl)c1F N1(S(C(CC)C)(=O)=O)CC2CN(C(=O)C(C)CC#N)CC(F)(C1)C2 N1(C(C(C)S(C)(=O)=O)=O)CCC(NC(=O)C(F)(F)CC2CC2)C(CO)CC1 N1(C(C2CCC(C)C2)=O)CC2CC(C1)N2C(=O)CCC1CCCC1 c1(NC)scnc1C(=O)N(C(C)CNC(=O)CC1CCC(=O)N1)C C1(C(=O)NC(CNC(=O)OC)C)CCC(O)CN1C(c1ccc(O)cc1)=O N1(C(C2(c3cccc(C)c3)CC2)=O)CCN(C(=O)CC2C=CCCC2)CC(C)C1 N1(C(COCC=C)=O)CC(NC(=O)C=Cc2nonc2C)CC(O)C1 C(=O)(CCS(=O)(=O)CC(C)C)NC(CC)CN(C(=O)C(C)(C)c1cccs1)C c1(C(=O)NC(C(C)C)(C)CNC(C2CCCOCC2)=O)ccc2c(c1)OCC2 N1(C(C2(C)CCC(C)C2)=O)CCC(C(=O)NCC2(C#N)CC2)C(C)C1 c1(C(N2CCC(C)C(N(C(=O)Cc3ccco3)C)C2)=O)cc2cccnc2cn1 N1(C(Cc2c(C)noc2C)=O)CCOC2CN(C(C3CCCC(F)(F)C3)=O)CC12 c1(SCC)ccc(C(=O)NC2CC(CO)N(C(=O)CC3CCCCN3C)C2)cc1 C1(C)(C(N(CCCCCNC(c2cc(CC)sn2)=O)C)=O)CC(OC)CN1C c1(NC(C2CCCN(CCCS(C)(=O)=O)CC2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(C(CC2CCOCC2)NC(CC2CC(=C)C2)=O)=O)CC2(CO)CCC1CC2 N1(CC)CC(C(=O)NC2(C)CC(NC(=O)Cc3ccc(F)cn3)C2)CC1=O N1(CCC)CC(C(=O)NCC=CCNC(=O)CC2CCCC2)CC1=O CN1CCC(NC(=O)C(C)(C)C2CCCN2C(C2CSCCS2)=O)CC1=O c1(OC(C)C)cnc(=NCC2CCC(NC(c3ccc(C(N)=O)o3)=O)C2)[nH]c1 C1(CNC(CSCCC)=O)(CO)CCN(C(=O)CCCCc2ccccc2)CC1 c1(C(=O)NCC(=O)NCC(C)CN(C(=O)COCC(F)F)C)cccnc1 C(CO)(CCCCNC(c1cc(C2CC2)cs1)=O)NC(c1c(SC)cn(C)n1)=O C1(NC(CC2CC(OCC)C2)=O)COCC1CNC(c1ccoc1C)=O N1(C(=O)OC)CCC(C)C(CNC(C2(n3cc(CN)nn3)CCC2)=O)C1 c1(C(=O)NCC(CN(C(=O)C(C)(C)C(F)(F)F)C)(C)C)cn(C)c(=O)nc1O C1(NC(=O)CC2CC(F)(F)C2)COCCN(C(=O)CCCCc2cnn[nH]2)C1 C1(NC(CC2CC(OC)C2)=O)CCCC1CNC(c1ccc(CNC(C)=O)s1)=O C(C(N=c1[nH]c(N2CCCCC(F)(F)C2)nc2c1CCCCC2)C(C)C)OC Cc1cc(C(=O)N(C(CNC(=O)C(=O)NC(C)C)C2CC2)C)nc2[nH]nc(O)c12 c1(CC)cncc(C(=O)NC2CCC(NC(C3CCNC3=O)=O)CC2)c1 N(C(=NCC1CCCCO1)N1CCC(C(N)=O)CC1)C(c1cccc(F)c1)C CCCCC(O)CC(=O)NCC(C)C(F)C(=O)NCc1cnc(C)s1 N1(C(c2cnc(C(=O)OCC)s2)=O)CCC2CN(C(=O)C(F)(F)C(C)O)CCC12 c1(C(=O)NC2CC(NC(C(CC(C)(C)C)O)=O)C2)cc(O)c2ccoc2c1 N1(C(=O)CC2CCSC2)CCC2(CC2C(N2CCC(O)C2)=O)C1 CCC(C(=O)NCC1CN(CC(O)COCC(C)C)CCCO1)C(C)O N1(C(CC2CC(=C)C2)=O)CC(NC(c2cnc(C3CC3)o2)=O)C2CC12 c1(S)ccc(C)c(C)c1.C1(C(=O)NCCCOCCNC(C)=O)CN(CCOC)C1 N1(C(CC(C)NC(=O)C2=CC3CCC(C2)C3)=O)CCN2C(=O)CCC2C1 N1(C(C(C(C)C)NS(N)(=O)=O)=O)CCC(C)N(C(c2cn(C(C)C)nn2)=O)CC1 N1(C(C2N(C(C(CCCC)F)=O)CCC2)=O)CCOCC(C2CC2)C1 C#CC1(O)CC(C(=O)NCC2(C)CCN(C(c3ccnc(OCC)c3)=O)C2)C1 c1(C(N2CCC(CNC(CC3(O)CCCN(C)C3)=O)C2)=O)cnc2c(c1)CCC2 C(=O)(C(F)C(F)(F)F)NC1(CCCNC(C2N(C(CC)=O)CCCC2)=O)CC1 c1(CC(N2CCN(CC(N3C(CC)CCC3)=O)CC2)=O)ccc(F)cc1Cl c1(-n2cc(C(CCC)NC(C3CC(O)C(F)C3)=O)nn2)cccc(Cl)c1 c1(NC2C3N(C(Cc4cccc(C)c4)=O)CC(CC3)C2)nc(C)cc(C)c1C#N C(=O)(CCCCC(=O)NCC1CN(C(c2n[nH]c3c2CC2CC32)=O)CCO1)NC C1(N(C(C(CC)=CC)=O)C)CCC2CN(C(=O)Cc3cccnc3O)CC12 C1(CCNC(c2cc(C)c(C)[nH]2)=O)CCN(C(c2ccsn2)=O)C(C)C1 c1(C(N2CC(C(=O)NC3(CC(=O)OCC)CCCC3)C2)=O)cccc(CO)c1 C1(NC(c2c(C)cc(C)o2)=O)CC2(NC(=O)CCC3CC3(C)C)COC1C2 C1(NC(=O)CC2CC2)CN(C(=O)C=C2CCOCC2)C2(CCOC2)C1 C=CCC(CC)C(=O)NCCN(C(=O)Cc1ccc(OCC)cc1C)C c1(C(N2CC(C)CC(NC(C(CC(C)C)F)=O)C2)=O)cc([N+](=O)[O-])nn1C N1(C(c2c(CCC)nco2)=O)CCCN(C(=O)Cn2nc(C)oc2=O)CC1 C1(C(N(CC(CN(C(C2(CC)COC2)=O)C)O)C)=O)CCC2(C1)CC2(F)F c1(C(=O)NCC(C)N(C(=O)CCNCC(F)F)CC)c(N)sc2c1CCC2 c1(C(=O)NC2(CNC(C3(COC)CCOC3)=O)CC2)ccnc(F)c1OC c1(C(=O)NC(C2CCN(C(=O)Cn3cnnc3)CC2)C)cnn2ncccc12 N1(C(c2cncs2)=O)CCCC2(CCN(C(C3CCC3(F)F)=O)C2)C1 N#Cc1cn(CC(=O)NCC2CCCN2C(=O)CN2CC=CC2)c(=O)nc1O CC(C)(C)C#CC(=O)N1CCCCC(CNC(=O)CCC2CCCC(=O)N2)C1 N1(C(C2CCC(NC(=O)OC)CC2)=O)CC=C(CCNC(C2SCCS2)=O)CC1 C#Cc1cc(C(=O)NCCOCCNC(c2cnc(CO)nc2C)=O)ccc1C C(C(C)(C)C(=O)NC1CC12CC(NC(=O)CCNC(=O)C=CCl)C2)SC Cc1cn2ccnc(C(=O)NCC3CN(C(=O)C(N4CCCCCC4)C)C3)c2n1 N1(C(CC=C)=O)CCCC(NC(c2n[nH]c(O)n2)=O)C1C C(=O)(CCCCN=[N+]=[N-])N1CCC(C2CN(C(CCC(C(C)C)OC)=O)C2)C1 CCC(C)CCCCC(=O)NCC(C)(C)OCC(N1CCC(C)C1(C)C)=O.C(C)(=O)OCC N1(C(=O)OC(C)(C)C)CCCC1(C)CNc1cnn(CCCC2CCCOC2)c1 C(C)(N=c1nc(N2CCSCC2)c2sccc2[nH]1)c1c(OC(C)C)cccc1 N1(C(c2cn(C)nc2Cl)=O)CC2CN(C(C3CC(C)(C)CO3)=O)CC2(C)C1 N1(C(c2nn(C)c(C3CC3)c2)=O)CCN(C(c2ccon2)=O)C2(CCC2)C1 c1(C(N(C2CCN(CC)CC2F)C(c2cc(C#N)cs2)=O)=O)cc2cccnn2n1 N1(C(c2c(C)ocn2)=O)CC(NC(=O)C(F)(F)c2cscc2Cl)C(C)C1 C1(CNC(C(n2cc(Cl)cn2)C)=O)CCN(C(c2csc(Cl)n2)=O)CC1(F)F C1(=CC(=O)NCC=Cc2ccco2)CCN(C(C2CCCOC2)=O)CC1 CCC(O)C(C)C(=O)N1CCCC(CN(C(=O)CC(C)(C)O)C)C1 N1(C(c2ccc(C)c(Br)c2)=O)CCc2ccc(Cl)cc2C1.C1(OC)CC2N(C1)C2=O C#CCCC(O)CCNC(=O)CCCCN(C(=O)C(O)CN1CCCC1)C N(S(=O)(=O)N1CCCc2ccc(Br)cc21)C(c1c(C)cc(Cl)cc1)CO N1(C(CCC)=O)CC2(CC(NC(=O)CC3CSC3)C2)C1 c1(C(=O)NCC2CC(C)N(C(=O)COCC3CCCC3)C2)cn(C)c(=O)nc1O C(N=c1cccc(S(=O)(=O)NC2CCCCC2F)[nH]1)c1snc(N(C)C)n1 Cc1cc(C(=O)NC2CN(C(=O)C(Cl)(Cl)Cl)CC2O)cc(O)c1 C1(CNC(=O)NCC2CCN(Cc3ccccc3)CC2)CCc2ccccc2O1 O=C(C1=CCOC1)NC1(CF)CCN(C(c2ccc(C(N)=O)nc2)=O)C1 C(C(=O)NCCOCCCN(C(=O)C(c1ccn(C)n1)C)C)(C(C)C)OC C1(C(N2CCC(NC(C3C(C)=CCS3)=O)C(C(N)=O)C2)=O)COC2COCC2O1 N1(C(CCCNC(=O)OC)=O)CC(NC(c2snc(Cl)c2Cl)=O)C(C)(C)C1 C12(NC(Cn3c(C)c(Cl)cn3)=O)CCN(C(=O)C=C(Cl)Cl)CCC1C2 C(=O)(C(CC)C(F)(F)F)N1CC(Cn2cc(CNC(CCC(=C)Cl)=O)nn2)C1 CC1CN(C(C2CSCCN2C(=O)CCC2(C)N=N2)=O)CCN1CCO c1(CC(=O)NC2CN(C(c3nncc(CCC)c3)=O)C3C2C3)ccc(F)c(F)c1 C1(NC(C2(CCC=C)CN(C(C3(CC4CC4)CCC3)=O)C2)=O)CC2CCCC2C1 CC(C)CC(O)CC(=O)NCCCCCC(=O)NCCC1(O)CCC1 C(=O)(C(C)C(C)NC(C1CC(=O)C1)=O)NC(C(=O)OC)(C)C C1(C(N(CCC)C(C)C)=O)C2CC(O)C(C2)N1C(C1CC1(C)C(F)F)=O C1(CNC(CC(C=C)C)=O)CN(C(c2nn[nH]c2C(F)(F)F)=O)CCCO1 C1(COC)CN(C(=O)CCn2ccnc2)CCN1C(=O)CCF C(=O)(C(CC#CC)NC(=O)Cc1scnc1C)NC(CC#C)CO c1(C(=O)NC(C(=O)NCC2CC2)C2CCCC2)cccnc1 c1(C2C(C(N3CC(NC(=O)C=Cc4cscn4)C3)=O)C2)c(F)cccc1F Cc1c(C(=O)NCC2CC2NC(c2cc(F)cc(Cl)c2N)=O)sc2ccccc12 c1(CCC)ncoc1C(=O)NC(C)CC(C)NC(=O)C(C)C c1(C(N2CC(O)(CN(C(=O)C3=COCCO3)C)C2)=O)ccc2c(c1)COC2 c1(C(=O)NC2(CCNC(C3CC(C)CC(C)C3)=O)CC2)cc(C#N)ccc1N c1(C(N(C2CCN(C(=O)Cc3nocc3C)C2)CC#C)=O)cc(C(C)=O)c(C)o1 c1(SC)nc(Cl)cc(=NC(=O)c2nccc(CC(=O)N(CC3CCOC3)CC)n2)[nH]1 c1(C(N2CC(CNC(C(C)(C)OC)=O)C(F)(F)C2)=O)c[nH]c2cc(F)c(F)cc12 N1(C(Cc2cnn(C)n2)=O)CC2CC(NC(=O)C=Cc3cncnc3O)CC2C1 C1(CCC)CCCC1(c1nnnn1CCOC)NCCSC1CC1 C1(CNC(C(c2ccc(C)s2)C)=O)CCC(NC(C23CC(C2)C(C)O3)=O)CC1 O=C(C(F)C1=CCCCC1)NCCC1=CCN(C(=O)CSCCO)CC1 C1(NC(COCC#C)=O)CN(C(=O)CCC2CCCN(C)C2)C(CC)(CC)C1 c1(C(N2CCN(c3nc(C#N)cc(C)n3)C3(C2)CC3)=O)ccc2c(C)c[nH]c2c1 N1(C(c2c(C)cc(C)s2)=O)CC(CC(=O)NCCC(C)N(C)C)C2(CC2)C1 Cc1ccc(C)c(N(C)C(C2(C)CC(O)CN2C(=O)C(C)NC(=O)C2CC2)=O)c1 C(c1c(F)ccc(Cl)c1F)=CC(=O)NCC(F)CNC(c1cc[nH]n1)=O CC1Cn2nccc2CN1C(=O)CCCCN(C(=O)CCC1CCC(=O)C1)C c1(C(=O)NC(C2CCN(C(c3c(C)nc(Cl)cc3)=O)C2)C)cccn2ccnc12 C1(NC(c2ccnc(C)n2)=O)CCN(C(=O)CCC(=O)c2ccccc2)CC1F N1(C(CC2(C=C)CN(CC3CC4(C3)CC(O)C4)C2)=O)CC(S(N)(=O)=O)C1 N1(C(=O)CCC2CCCCO2)CCN(C(C2(CO)CCOCC2)=O)C2(CC2)C1 c1(C(=O)OC)cc(C(N(S(CC)(=O)=O)C)C2CC2)n(C)c1C C1(NC(C=CC)=O)CC2CC(NC(C3CC34CC(OCC)C4)=O)C2C1 C1(NC(c2cc(COC)no2)=O)C2CC3CN(C(=O)CS(=O)(=O)N(C)C)C1C3C2 Cc1ccc2nonc2c1C(N1CC(CNC(=O)COC2(C)CCC2)C1)=O c1(CN2CC(C(N(C3CCOCC3)CC)=O)OCC2)cc(C)cc([N+](=O)[O-])c1 C1(CNC(=O)Cc2cnoc2)COCCN(C(c2nocc2Br)=O)C1 CC1CCN(C(=NCCF)NCC2C(F)(F)C23CCC3)CC1 N1(C(C(CCC)OC)=O)C(C(=O)N(C2CCC(O)CC2)C)CC2CCCC12 C1(C(=O)N(CCCOC)C)(OCC)CCCC1.c12cc(c[nH]1)CN(C)C2=O c1(CCC)cc(C(=O)NCCNC(c2c[nH]nc2Br)=O)ccn1 c1(C(=O)NC(c2cn(-c3ccccc3Cl)nn2)C)ccc2c(c1)NC(=O)CCC2 c1(SCC)cncc(NCC2CN(CC#N)CCO2)n1 c1(NC(CNC(CC)=O)C(C)C(C)C)cc2ncnc(O)c2cc1[N+](=O)[O-] c1(C(N2CC=CC2Cn2cc(CC(O)C3CC3)nn2)=O)ncc2c(n1)CNC2 c1(C(=O)NCC(CC)NC(=O)CC(O)CN(C)C)cc(SC)oc1C C1(C(=O)NCC(CCOC)NC(=O)CC2COC(C)(C)C2)CN(C)CC(C)O1 c1(C(=O)NC2(C3N(C(c4nc(N(C)C)oc4)=O)CCC3)CC2)ccc2c(c1)CC2 N1(C(CNC(C)=O)=O)CCCCC1C(=O)N(C)Cc1ccsc1 c1(C(=O)NC2CN(C(COCCOC)=O)CC2O)cc(OC)c2ncccc2c1 N1(C(C2(CF)CCN(C(c3cc(C4CC4)on3)=O)C2)=O)CCN(C2CC2)C(=O)C1 c1(NC(C2CC(NC(c3cc(F)ccc3O)=O)C2)=O)ccc2c(n1)CCC2 Fc1cc(CCNC2CCCC2c2ccccc2Br)ccc1Br C12(CNC(C3(C(N)=O)CC3)=O)CCC(C1)N(C(=O)CC=Cc1ccc(F)cc1)C2 c1(C(=O)NC(CN(C(=O)CCC(C)C)CC)C)cnc(-c2ccncn2)nc1O Cc1ccc(O)cc1NC(=O)C(CC1CC1)NC(C1CCN(C)C1=O)=O N1(C(c2c(C)ccc(=N)[nH]2)=O)CC2CC(NC(c3n[nH]c(C4CC4)n3)=O)CC1C2 c1(OC)cc(Br)ccc1C(N1CCOC(COc2cccc(NC(C)=O)c2)C1)=O N1(C(c2c(CC)nsc2)=O)CC(O)C(O)CC2(CC2)C1 C1(SCC(=O)N(C)Cc2cn(-c3cc(F)cc(Br)c3)nn2)CC(=O)CC12CCC2 c1(C(C)C)c(C(F)(F)F)n[nH]c1C(=O)NC(C)CNC(C1(N(C)C)CC1)=O C(C(C)(O)C(F)(F)F)N(C(=O)C(=O)NCC1(F)CCOC1)C C1(NC2c3c(Br)[nH]nc3CCC2)CCCC2(CC1)OCCO2 C1(C(N2CCCCC(CCCC)C2)=O)CC2(CCN(C(=O)C=CCOCC)C2)C1 c1(SCCCC(=O)OC)ccc(NC(c2ncsc2C(F)(F)F)=O)cc1 C=C(Cl)CCC(=O)N1CC(C(=O)NCCNC(=O)CCc2nc(O)n[nH]2)C1 c1(C(=O)NC(CC)CN(C(=O)CC2CC(C)(C)C2)C)cc(C)cc(Cl)c1 CS(=O)(=O)c1cc(C(=O)NCC2CCCCN2CC(F)F)c(Cl)cn1 Cc1cc(Cl)ccc1C(=O)NCC1CC2CCC1N2C(=O)CC1CC1(Cl)Cl c1(CC(=O)N(C)CC2CCCN2C(=O)CC2CCOCC2)ccc(F)cc1CC#N C1(CCCNC(CC(C)OC)=O)CCCCN1C(c1cccnc1C)=O N1(C(c2c(C)[nH]c(=N)s2)=O)CCCN(C(=O)C(N2CCOCC2=O)C)C(C)C1 C(C(=O)N1CCC(C)(NC(=O)CCc2cccs2)C1)(C(C)C)SC CC(C)(C(=O)O)C(CCO)N1CCC(C(=O)NCCc2n[nH]c(=N)s2)CC1 C1(CNC(C2CCC(C)(C)C2)=O)CCN(C(=O)CCn2ccnc2)CCC1(F)F c1(C(=O)NCC2(F)CC(NC(C3CCC(C)C3)=O)C2)ccc(S(N)(=O)=O)cc1F CCC(CC(=O)N1CCCC(O)(CNC(c2ccc(C(F)F)o2)=O)CC1)C(F)F N1(C(c2cscc2Br)C(=O)NCc2ccc(Cl)cc2F)CCCCc2ccccc21 c1(C(=O)NCCCNC(c2n(CCCC)ncc2)=O)c(F)cc(F)cc1F C1(NC(c2cc(CCC)on2)=O)CCC2CC1CN2C(c1cnccc1SC)=O C(=O)(C(C)CCC(C)(C)C)N(CCN(C(C)C)C(C12CC(CO)(C1)OC2C)=O)C c1(C(=O)NCC(CN(C(Cc2c(C)ocn2)=O)C)C)cc2c(nc1O)CCCC2 C1(NC(c2nn(C)c(=O)cc2)=O)COC2(C1)CN(C(C1(C)COC(=O)C1)=O)C2 c1(C(=O)OC)cncc(CNC(=O)CCC(C)NC(=O)CCOC2CC2)c1 c1(C(=O)NCCCC(C)NC(C(CCCC)C)=O)ccc2c(=N)[nH]cnc2c1 c1(C(=O)NCC2CN(C(=O)CC34CCCC3C4)CCCO2)nc2c(s1)COCC2 Cc1c(F)ccc(C(N2CC3COCC(C2)C3NC(=O)COCCF)=O)c1C#N N1(C(c2nc(C)oc2)=O)CCCCC(C2CN(C(=O)CCCCF)C2)C1 N1(C(CCOC(C)=O)=O)CCC(OC(=O)C(O)C2CN(OC(C)(C)C)C2)CC1 CCCCC(O)CC(=O)N1CCN(C(c2cc(CC)ccn2)=O)C(CF)C1 c1(OC)cc(I)c(CC(c2cc(-c3ccc(NCC)c(F)c3)cs2)=O)cc1N N1(C(CCC=C(C)C)C(=O)NCc2ccccc2Br)Cc2ccccc2C1 N1(C(c2n(C)c(S)nc2)=O)CCC(NC(c2cccc(=O)n2C)=O)C(C(N)=O)C1 C1(NC(C2(CC(C)C)CCCC2)=O)CCN(C(=O)C2CC2)CCC1CO N1(CCC(=O)NC2CC(C)N(C(=O)CN(C)C(N)=O)C2)Cc2ccccc2C1=O C12(CNC(c3c(C)cc[nH]3)=O)CC(C1)C(NC(=O)Cc1cn3ccsc3n1)CO2 c1(C2C(CCC)(CO)C(CCCC#C)N2)ccc(S(=O)(=O)CC)cc1 C1(NC(CC2OCCN(C(CN(C)C(N)=O)=O)C2)=O)CCn2ncnc2C1 O(C=CC(=O)N1CCCC1CCCNC(c1n[nH]cc1-c1ccncc1)=O)CC c1(C(=O)NCC(CC)NC(=O)C(CC)CC(F)F)c(F)cc(Cl)cc1Cl N1(C(C(CC)c2ccccc2)=O)CCCC(CNC(c2cc(F)n[nH]2)=O)CC1 C1(CNC(C(CC)OC)=O)CCC(N(C(=O)CNC(C2CCCCC2)=O)C)CC1 C(=O)(C1CCOc2ccccc21)NC1C(C)CN(C(c2c(F)cncc2Cl)=O)C1 C1(C(=O)NCC(CC(C)C)(C)NC(=O)CC(C)NC(N)=O)CCCCC12CCC2 CC1CCc2nc(C(N3CCC(N(C)C(c4cc(F)c[nH]4)=O)CC3)=O)cn2C1 N1(C(c2ccc(OC)s2)=O)CC(C)CC1C(=O)NCCCCC(N)=O c1(C(N2C(CNC(C3(CSC)CC3)=O)CC2)=O)cnn(CCO)c1C1CC1 C(CCCCNC(=O)CSC(F)(F)F)N(CCc1ccc(-c2ccco2)[nH]1)CC CCC(CC(=O)N1CC(CNC(=O)CCC(N)=O)C(F)(F)C1)CC(F)(F)F c1(C(=O)NC(C)CNC(c2ccc3c(c2)CC3)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(N2C(C)CC(CNC(C3CCC3)=O)C2)=O)cc2oc(Br)cc2[nH]1 C1(C(=O)NC2CN(C(C(CC)(C)C)=O)CC3C2C3)CCc2cn(C)nc2C1 C(=O)(C1=CC2(CN(C(=O)C3=CCCOCC3)C2)OC1)N1CCC(C)(CC)C1 N#CC1(C(=O)NCC2CN(C(=O)Cn3cc(C4CC4)cn3)C2)CC12CCC2 n1(CC(=O)NC(CC2CN(C(C3(COCC)CCC3)=O)C2)C)ccc(C)cc1=O c1(NC(C2CCN2Cc2csc(Br)c2)=O)cc(Cl)ncc1[N+](=O)[O-] Cc1ccc(F)cc1NC(=O)C(=O)NC(c1cscn1)CO C1(O)(CCNC(C2(CC(C)C)CC2)=O)CCN(C(=O)CC2CCC(C)CO2)CC1 C=CC1(CC(=O)NC(Cn2cncn2)CC)CN(NC(C2(C(=O)OC)CC2)=O)C1 c1(C(=O)NCC2N(C(c3nc(C(C)OC)sc3)=O)CC2)c[nH]c(C)c(Cl)c1=O c1(-c2c(C(N3CC(CCNC(CC(=O)N(C)C)=O)C3)=O)cno2)ccc(F)cc1 C(C)(C(=O)NCCN(C(=O)CSCC(C)C)Cc1ccccc1)(C1CC1)OC C#Cc1cccc(CC(=O)NCC2CCC(C)CN2C(=O)C(=O)NC2CC2)c1F C1(C(=O)NCC(CC)NC(=O)CS(=O)(=O)CC)CCc2ncnc(C)c2C1 CC(C)(C)CC(O)C(=O)N1CCC(n2cccn2)(C(=O)NC2C=CC(C)(C)CC2)CC1 C1(C)(CNC(CCCOCC)=O)CCCN1C(=O)C(O)CSC N1(CC(=O)NC)CC2(CN(C(c3ccn4ncnc4c3)=O)CC(C)(C)O2)C1 C1(CC)(NC(c2ns[nH]c2=O)=O)CCCN(C(=O)C(N2CCNC2=O)C)C1 N1(C(Cc2n(C)nnc2)=O)CCC=C(CNC(C2CC3C=CC2C3)=O)C1 C1(NC(c2ccc(C#C)cn2)=O)CN(C(=O)CCCOCC)CC1S(C)(=O)=O C1(N(c2ccn(C)n2)C2CCCC2)CCN(CCC23CCCC2C3)CC1.C1C(=O)N1 N1(C(C=CC(=O)OCC)=O)CCN(CCC2CC2)CC1.C(=O)(CC(C)(F)F)N N1(C(c2cc(CC)ncn2)=O)CCC(C)(C)C1C(N1CCOC(C)C1CO)=O N1(C(C(CC)N(C)C(c2cccs2)=O)=O)CCC(OCCNC(=O)CSC)CC1 c1(OC)cccc(C2CCN(C(C3CC(O)(Cn4cncn4)C3)=O)CC2)c1 c1(C(=O)NCC(C=C)O)cc(OC(C)C)c(OC)cc1C C(=O)(CC(C)(O)CCC)N(C(c1cn(-c2ccc(OCC)cc2)nn1)C)C c1(SC)cc(F)ccc1C(N1CCCC1CNC(C1(F)CCCOC1)=O)=O CCCCC(C)CCC(=O)N1CCC(C2CCCCN2C(=O)C(C)=C2CC2)CC1 C#CCCCCCCC(=O)N1CCC(C(C)NC(=O)C(C)OCCC=C)CC1 c1(C2C(C(=O)NC(CNC(=O)C3=CCSC3)CO)C2)cccc(F)c1Br C1(CNC(CCN(C(C)=O)C)=O)C2CN(C(c3conc3C(C)(C)C)=O)CC12 N1(C(CC2N(C(CC(=O)NCC)=O)CCOC2)=O)CCC(F)CC1C C(CCSC)(C(=O)NCCN(C(C1(C(F)F)CC(F)(F)C1)=O)C1CC1)OC C1(C(=O)NC2C(NC(c3c(C)nc(CC)o3)=O)C2)CCC(=O)N(C(C)C)C1 C1(c2n(C(C3CCC3)C)nnn2)(NC2(C3CC3)CC2=O)CCCN2CCCCC12 Cc1csc(NC(C)C(=O)NC2(C3CCCN3C(=O)C(C)(F)F)CC2)n1 C1(C(=O)NC2CCC(N(C(=O)C=CCOC(C)(C)C)C)CC2)CCn2ncnc2C1 c1(C(=O)OCC)nn(C)c(Cl)c1COC(c1cc(C(C)(C)C)no1)=O C(CC(C(=O)NC(C1CC1(C)C)C)NC(=O)CCSC)OC c1(C(N(C2CCN(C(c3cc(SC)oc3C)=O)C2)C)=O)ccc2[nH]c(C)cc2c1 N1(CC(C)NC(Cn2nnc(C)n2)=O)CCN(C(C2CC(C)C2)=O)CC1 N1(C(=O)CC2CCCC(O)C2)CC2CCC(C1)N2C(C1CCCC1CF)=O C1(C(F)(F)F)(CN(C(C2N(C(CCC)=O)CCOC2)=O)CC)CC2(CCC2)C1 C(C)(C(C(=O)NCC(C)(C)C(C)(C)O)C(C)C)NC(CCCOCCC)=O N1(C(c2csc(O)n2)=O)CCC2CC1CN(C(=O)OCCOc1ccccc1)C2 N1(C(C(C)NS(CC)(=O)=O)=O)CCC(C)N(C(c2nc(COC)oc2C)=O)CC1 C(=O)(C1CNC(=O)c2ccnn21)NC(C)C(C)(C)NC(=O)C=Cc1cccnc1 CN1C(=O)CCCC1C(=O)NC1CCCC1NC(c1cc[n+]([O-])cc1)=O CC1CC(CNC(c2cnsc2)=O)CN1C(=O)C(CC1CCC1)N(C)C C1(CN(C(C2(CCOC)CCC2)=O)C)CCCN1C(c1ccoc1)=O c1(Cn2c(-c3cccnc3O)nc(C(CCC)C)n2)c(Cl)cccc1Cl N1(C(c2cc(C)c(N)cc2F)=O)CCC2(CCC2NC(=O)C(C)C2CC2)CC1 N1(C(CC(CNC(c2cncc(OC)c2)=O)C)=O)C2C=CCC1CCC2 CCC(C)C(=O)NCC#CC(=O)N(CC)Cc1cccnc1 C#CCC(C)C(=O)NCC#CCNC(C1(c2ccn(C)n2)CC1)=O C(=O)(CCCS(N)(=O)=O)NC(CCN(C(C)=O)C)C(C)(C)C N1(C(C2C(C)(C)C2)=O)CCCC2CN(C(c3cc[nH]c3C3CC3)=O)CC12 C1(C)(CC)CCCN(C(C2CCOCC2)C(=O)NCCOCC2CC2)C1 N1(C(CN(C)C)=O)CCCCC(NC(c2ccc(-c3nccs3)cc2)=O)C1 N1(C(c2cccc(COC)c2)=O)CCN(C(=O)COCCCC(C)C)C2CC12 O=C(C1=CCS(=O)(=O)C1)NCC1CC1NC(c1cnc2n1CCOC2)=O c1(SCC(N2CC(COC)(CNC(=O)C(C)CC3CCC3)C2)=O)ccc(F)c(F)c1 c1(C(N(CC(C)NC(C(C)NC(c2ccccc2)=O)=O)C)=O)ccn(C2CC2)n1 c1(CC)cc(C(=O)NCC2CCN(C(=O)CCc3ccn(C)n3)CC2)ccc1O C1(CN(C)C(C23CC(C2)C3)=O)CCCN(C(=O)Cc2ccc(Br)nc2)C1 C1(C(C)C)(C(N2CCC2CF)=O)CCN(C(=O)C(C)OC(C)(C)C)C1 c1(C(=O)NCCNC(=O)CC(=O)NC2CCN(CC)C2)cc(Cl)c(Cl)s1 Cc1ncc(C(=O)NCCC(C)N(C(=O)Cc2ccnn2C)C)cc1N c1(C(=O)OCC(n2cc(C(=O)OC)nn2)C)cc(OC)cc(OC)c1Cl C(=O)(C(C)(F)C(=O)NCCCN(C(=O)C=CC=Cc1ccccc1)CCO)OC C1(OC(C)C)C(c2ccccc2)CCN1C(=O)C(N1CCC(F)C1)=O C1(NC(=O)C2=CCCO2)CC2CCC(C1)N2C(c1c[nH]cc(F)c1=O)=O CC1CN(C(=O)CCCN2CCOCC2)CCCN1C(C1CCCC(=O)CC1)=O N1(C(c2nc(CCC)oc2)=O)CCC2CCCC12C(N1CCC2(CC2)C1)=O C1(OCC)CN(C(=O)CCN(c2cc(C(=O)NC)[nH]n2)CC2CC2)CC2(CC2)C1 C1(CC=C)CC(O)CC(CC(=O)NCC(CO)NC(=O)Cc2csnc2C)O1 N1(C(C2CCN(C(C)=O)C2)=O)CCC(C2CCCN(C(c3ccno3)=O)C2)C1 C12(CNC(CS(=O)(=O)N(CC)CC)=O)CCC(CC1)N(C(c1ocnc1C)=O)C2 C12(C(=O)NC(CN(C(C3CCS(=O)(=O)C3)=O)CC)C)CCC(N(C)C)(CC1)CC2 C#CC1CCCN(C(=O)C(CNC(C2CC3(CSC3)C2)=O)OC)CC1 N1(C(CC(CC)SC)=O)CCC2(CC1)CC2CNC(C12CC(C(F)F)(CO1)C2)=O Cc1ccc2cc(CN3CC4CC3CN4C(=O)Cc3cnn(C)c3)c(Cl)nc2c1 N1(C(Cc2n(C)c(S)nn2)=O)CCC2CN(C(c3ccc4nc[nH]c4c3)=O)C2C1 c1(C(CC)O)nc(C2CN(C(C)=O)C2)n(-c2ccccc2C(F)(F)F)n1 c1(CNC(C(COCC)n2cc(-c3cnc(OC)s3)nn2)=O)ccccc1Cl Cc1nccc(C(=O)NCCCCN(C)C(C2C3CCC(=O)C23)=O)c1C C(=O)(C#CC1CCOC1)NCC1(C(N)=O)CN(C(c2nc(OC)c(C)s2)=O)C1 c1(CC)n[nH]c(=NCC2CC(NC(=O)C(C3CCOCC3)F)C2)s1 C(=O)(CCCC(=O)N(C)C)N1CC(C(C(=O)NCCS(CC)(=O)=O)O)C1 Cc1nn(C2CCC2)cc1NC(=O)C(=O)C(c1ccc(CCC(N)=O)cc1)=O C(C(O)CC(F)(F)F)NC(C(C1CCC1)NC(CC1C(CC)C1)=O)=O C(=O)(CC(C)(C)C(F)(F)F)NC(C(C)NC(CC)=O)(C)C C12(NC(C(c3c(C)noc3C)C)=O)CCCC1(F)CN(C(c1cc[nH]c1)=O)C2 C1(C(N(CC(C)NC(c2cnc(N)cn2)=O)C)=O)CN(C)CCO1 CN1CCOC(C(N2CCCC2(C(=O)N)CC)=O)C1.C(CCS(C)(=O)=O)C1CC1 Cc1ccc(CC(=O)NCC2CC(NC(=O)CCCOCC(C)C)C(O)C2)cc1 C(CN=c1[nH]c2cccc(Br)c2o1)C1N(C(CCNC(N)=O)=O)CCCC1 c1(C(C(=O)N(CCNC(C(=O)NC(C)C)=O)C)N(C)C)ccc(Cl)cc1 C1(COC)CC2(CCN2C(C2CCCC(NC(=O)CC3CCC(C)(C)C3)C2)=O)C1 N1(C(C(CCC)N(C)C)=O)CCCCC(CNC(=O)Cc2ccc(C)cc2F)C1 C=CCCCC(C)(C)CNC(=O)CC(CC)NC(c1cnc(C)[nH]1)=O C(=O)(C1=C(C)OCC1)N1C(CC(=O)NCc2scc(COC)n2)CCC1 CCC(C(=O)N1CCN(C(=O)Cn2ccc([N+](=O)[O-])n2)CC1)C(C)C Cc1cc(N)c(C)nc1C(=O)NCC1=CCN(C(=O)CC2CC2C)CC1 C1(CNC(=O)NC23CC(C(=O)OC)(C2)C3)CC(NC(=O)C(C)C)C1(C)C Cc1cc(C(N2CCC(C)C(CNC(=O)COC3COC3)C2)=O)c(Cl)cc1N c1(CC(=O)NC2CC(NC(c3c(C)cc(Br)o3)=O)C2)c(C)nc(O)nc1C C=CC1(C(=O)NCCCNC(N)=O)CCN(C(=O)NC2CCO2)C1 c1(C(=O)NC(CC=C)CNC(c2ccc(O)c(F)c2)=O)cc(Cl)c(F)cc1F c1(C(N2CCC(NS(CC=C)(=O)=O)(CO)CC2)=O)c[nH]c2cc(F)c(F)cc12 c1(C(=O)NCC(=O)NC(CN(C(c2cscc2F)=O)CC)C)cc2c(s1)CCC2 N1(C(C(CC2CC2)OC)=O)CC(C)(CNC(c2c(F)cccc2Cl)=O)CC1(C)C c1(C(N2CCC(NC(C3CC(=C)C3)=O)C(OC)C2)=O)c(F)cc(C#N)cc1F C1(NC(c2cc(CC)n(C)n2)=O)CN(C(=O)Cc2cc[nH]c2)CC2(CC2)C1 C(=O)(C(C1=NOCC1)N1CCC1c1ccc(Br)cc1C)NCCCSC N1(C(CCCC#C)=O)CC(F)(F)CC1(C)CNC(c1cc(C)cc(O)n1)=O N1(S(CCC)(=O)=O)CCC(C(=O)NCC2(C)CCN(C(C3(C#N)CC3)=O)C2)CC1 c1(CNC(CCC#C)=O)nc2c(s1)CN(C(=O)CCn1ccccc1=O)CC2 C(=O)(N(OC)C1CCCCC1)NC(C(C(=O)OC)(C)C(=O)OC)C N1(C(c2cc(OC)no2)=O)CCCC2(CCN(C(C3CCCCNC3=O)=O)C2)C1 c1(C(=O)NC2C(CNC(C(c3ccc(F)cc3)C)=O)C2)ccc(C#N)cc1O c1(C(=O)NCC2(NC(COCCC=C)=O)CCCC2)cc(F)cc(Cl)c1 CC(C)CCCCCC(=O)NC(C(=O)NC(C1CCC1)C)C(C)(C)C c1(CC(=O)NC(CC=C)CNC(=O)CC2(CC)CCCC2)cn2ccccc2n1 CC(C)CC(C(=O)NC1(CN(C(=O)CN(C)C(=O)C2CC2)C)CC1)N(C)C CC(C)CC(C(=O)NCC(CO)NC(c1c(F)ccc2[nH]ccc12)=O)C(C)C c1(CC)cccc(-n2c(SCC3(CO)COC3)nnc2-c2cnn(C)c2)c1 C1(NC(C2CC(C)NC(=O)C2)=O)CCC12CCN(C(=O)C1=C(Cl)CCOC1)CC2 N1(C(C(C)(C)CO)=O)CCC2(CC1)CC2CNC(=O)COC1CC=CC1 c1(C(=O)NC(c2cnn(C)c2)CNC(C2C(CC)C2)=O)ccc(C(C)(C)C)nc1 CC1(O)CCC(C(=O)NC(C(=O)NC2C=CCCC2)C2CCCC2)CC1 c1(COC)nc(O)c(C(=O)OC)cc1C.c12oc(nc1C)[nH]c2=O Cn1nccc(C(N2CCOCC2CCNC(c2ccc(C(F)F)o2)=O)=O)c1=O N1(C(c2cocn2)=O)CCC2(CC1)CN(C(C1CC1C1CC(F)(F)C1)=O)CCO2 Cc1nnc2n1CC(CNCCOc1ccc(O)cc1)C2 N1(C(C(C)N(C)C)=O)CCC2(CC1)CC2NC(c1cc(C2CCC2)[nH]n1)=O N1(C(C=CC)=O)CCCC12CCCN(C(C1CCCN(C(C)C)C1)=O)C2 C(CC(=O)N1CC2(COC(=O)C2)C1)(C(F)(F)F)NC(C1(C)CCC(=O)C1)=O N1(C(c2c(C(C)C)[nH]cc2)=O)CCOC2(C1)CN(C(=O)CN(C)C(=O)C1CC1)C2 C(CCCC)(CC(=O)NCCC1CCOCC1)NC(C(CCC)CC)=O c1(C(N2CCN(CCNC(C(C=CCCC)O)=O)CC2)=O)ccc(O)c(OC)c1 CC1CCC(C2CCCC2)CN1C(=O)NCc1csc2ccccc12 c1(-c2nc(C)c(NC(c3cnc(O)n(C)c3=O)=O)s2)c(C)cc(N(C)C)cc1C c1(C(N(C2CCN(C(c3c(C)cccc3)=O)C2)CCO)=O)cnc(C2CC2)nc1O c1(CC(=O)NC2(CNC(=O)CC(C)C)CC(OC)C2)coc2cc(C)c(C)cc12 C(N=c1[nH]ccnc1F)C1C(NC(C(C)OCc2ccccn2)=O)CCCC1 C(=O)(C1COc2ccc(F)cc21)NCCNC(CCc1cc(C(C)=O)c(C)o1)=O Cc1ncn(C)c1N(C(c1ccc(N2CCCC2)nc1)=O)C(C1C2CNC1C2)=O C1(NC(C(CN(C)C)NC(c2cccc3nccn23)=O)=O)CCn2nnnc2C1 C1(CNC(c2cc(C(CC)C)no2)=O)CCN(C(=O)Cc2ccsc2C)CC1C N1(C(Cc2ccc(C)cc2)=O)CCN(C(=O)Cc2csc(S)n2)C(C)C1C c1(CNC(C2(CNC(c3nc(CC)sc3)=O)CCCC2)=O)cc(C)ccc1C N12CC(O)(C3CCN(CC3)CC1=O)C2.CC(C)CC(CN1CCOCC1)N(C)C C(C(C)(C)C(=O)NC1COCC1CNC(C1(C)CCNC1=O)=O)N(C)C CC1(C)CCC(C)(C(=O)NCCC2(O)CN(C(c3ccc(F)cc3Cl)=O)C2)CC1 C1(NC(Cc2cccc(COC)c2)=O)COC2(CCN(C(=O)C(C)CN)CC2)C1 CC(=O)CCCC(=O)NCC1CC(C(F)(F)F)CCN1C(C1COCCO1)=O c1(C(N2CC(n3cc(-c4ccc(=N)[nH]c4)nn3)C2)=O)cc2cc(Cl)c(F)cc2[nH]1 c1(NCCC=CC=C)ccc(S(=O)(=O)NC2c3ccccc3CC2C)cc1C#N O=C(CC(C(F)F)NC(C1CC(O)C(F)C1)=O)NCCc1cscn1 C(=O)(C1c2c[nH]nc2CCC1C)N(CCNC(CC(=C=C)C)=O)CC C1(C(=O)NCCC2(NC(c3ncn(CC)n3)=O)CC2)CCCCC12CC2 c1(C(N(C2CN(C(=O)CC3C=CCC3)CC23CC3)C)=O)cc2c(s1)CCC2=O Cc1coc(C)c1C=CC(N1CC(CC(=O)OCC(F)(F)F)C1)=O C1(C(N(C)CC2CCCN2C(=O)CSc2n[nH]c(=N)s2)=O)CCC2CCCCN12 Cc1ccc2cc(C(=O)NC3CCN(C(C4(F)CCCC4)=O)C3C)ccc2n1 c1(OC)nn(C)cc1C(=O)NCc1cc(C)c(C(=O)NC(C2CCOC2)CO)o1 C1(NC(c2c(C)ccnn2)=O)CN(C(C2CCNC2=O)=O)CC12CCC2 c1(C(=O)NC(CNC(c2c(C)ccc(F)c2N)=O)C)[nH]c2ccc(F)cc2c1Cl N(C1CCc2ccccc21)C(CC=CCNC(C1(C)N(C)CCC1)=O)=O CCC(CC)CC(=O)NC(CCSC)C(=O)NCCCCCNC(N)=O C1(NC(C(C)Cc2ccccc2)=O)CC2CC1N(C(c1ccc(Cl)c(O)c1)=O)C2 C1(NC(C2(CC#C)CC2)=O)CC2CC1N(C(=O)CSCC1CCS(=O)(=O)C1)C2 C1(C(N2CC(NC(CC3CC(=O)NC3)=O)C(O)C2)=O)C2C3CC4C1C1C2CC3C41 CC#CCC(C(=O)N1CCC2CC12)NC(=O)CN1CCC(C)CC1 Cn1ncc2c(=O)n(CC(=O)NC3(CF)CCN(C(=O)CC4CC4)C3)cnc12 c1(C(C)C)ncoc1C(=O)NCC1CCN1C(c1cocc1C(N)=O)=O O=C(C1=C(Cl)CCOC1)NC1COCC1NC(c1cc(Br)ccn1)=O C1(C(=O)NCC2CC(NC(CCCCNC(COC)=O)=O)C2)CC2CCC1CC2 c1(OC)cc(C)c(CNCC2CC(F)(F)C23CC3)cn1 c1(CC)nnsc1C(=O)NC1CN(C(C2CCCN2C(C)C)=O)C1 C1(CNC(C(CCCOC)C)=O)CC2(CCC2)CN1C(=O)C(C)(F)F CC1(C)CCC(C(=O)NC2CCN(C(c3ncc(Br)cn3)=O)C2)OC1 c1(C(=O)NC2(CN(C(CC3C(C)CCC3)=O)C)CC2)cncnc1C(C)(C)C C1(NC(CCc2cc(C)n(C)n2)=O)CCN(C(c2nc(=O)cc(N)[nH]2)=O)CC1O N1(C(CCOCCN(C)C)=O)CCC(CNC(c2c[nH]cc(Cl)c2=O)=O)C1(C)C C=CCCCCCCCC(=O)NC(CNC(=O)CSCCC#N)CCC c1(OC)cc(C(N2CC3CC3(C(=O)NCCCc3cc[nH]n3)C2)=O)nn1C c1(CNC(C2CN(Cc3ccc(CC)s3)CC(F)C2)=O)cc(C)c(Cl)c(C)c1 C(=O)(C1CCCc2ccnn21)N1CCCC(Cc2n(CCC)ncc2)C1 C1(C(=O)NC(COCCOC)C)CC2CCCC2N1C(=O)CC1NC(=O)NC1=O N1(C(CN(CCC)C)=O)CCN(C(C23CC(CCC(F)(F)F)(C2)C3)=O)CC1 N1(C(CNC(CCCCC)=O)=O)CCC2CCCC(C1)N2C(C1(CC)COC1)=O C12(CNC(CS(=O)(=O)NCC)=O)CCCC1CCN2C(=O)C(F)=CCCF CC(C)CC(C(=O)NC1(CO)CN(C(c2nnc(S)n2C)=O)C1)c1ccccc1 N1(C(C(CC)(C)CO)=O)CCC2(C=C(C(=O)NC(CN(C)C)CO)C2)C1 CCCC(C(O)C(=O)NC1(C)CCCC(C)(C)C1)NC(C1C2CCCCC12)=O Cc1cc(C(=O)NC2CC(O)CN(C(c3cccc(F)c3Cl)=O)C2)c(C)cn1 N1(C(C(=O)NCc2ccccc2)=O)CCC(CO)(Nc2cncc(Cl)n2)CC1 C1(O)(C(C)NC(=O)CCc2nc[nH]n2)CCN(C(c2ccc(N)cn2)=O)CC1 N1(C(C(CC)N2CCCC2=O)=O)CCOCC1CCNC(c1ccc(C)n1C)=O n1(CC(=O)NCC(C)N(C(c2[nH]cc(C)c2)=O)C)ncc(O)nc1=O CC(CC1CC1)C(=O)NC1CC(NC(C2(N3CCOC3=O)CC2)=O)C1 c1(C(N(C2CN(C(=O)CCn3cccn3)CC2(C)C)C)=O)ccc(N)c(Cl)n1 C(C)(C(C(=O)N(CC1=CCCOC1)C)C(C)C)NC(c1ncnc(C)c1C)=O CC(CCNC(=O)CCN(C)C(C1COC(=O)N1C)=O)CCO Cc1c(NC2CN(C(C3CCC=CCC3)=O)CC2C)ncnc1Cl N1(C(C(CO)NC(C(C)CC#N)=O)=O)CC2CSCC2(C)C1 c1(C(=O)NC(CC)CNC(C2(F)CCC2)=O)nnc(C)cc1O Cc1oc(C)c(C(=O)NCC2(O)CN(C(c3cc(Cl)sc3Cl)=O)C2)c1C c1(OC)ccc([N+](=O)[O-])c(CNCCc2cccc3cc[nH]c23)c1 N1(C(C=C(CC)C)=O)CCC(CCNC(=O)CCCn2cc(C)cn2)C1 C1(CNC(C(CC=C)C)=O)CCN(C(c2ccc(C(F)F)nc2)=O)C1(C)C N1(C(c2nc(COC)sc2)=O)C2CCC1CN(C(=O)C(C)(CO)OC)C2 O=S(=O)(c1cnc(NCC(O)Cn2cccn2)c(Cl)c1)N1CCSC1 N1(C(C(C)(C)C)=O)CCC2CCN(C(=O)NC3CCC4(COC(C)C4C)O3)CC12 N1(C(C2OCCN(C(C(C)(C)CCCF)=O)C2)=O)Cc2cc(O)nnc2C1 c1(C(N2C3CN(C(CCN4C(=O)CCC4)=O)C(C3)C2)=O)nnn2c1COCC2 c1(C(=O)NC2CCCN(C(=O)CC3(CO)CC3)CC2)cnc2ncnc(O)c2c1 C(CCCC(C)(C)C(=O)NNC(=O)C(C)n1cccc1)NC1ON=C(CC)C1 C1(CNC(C2(C(=O)NC)CC2)=O)CCCCCN1C(=O)CC(O)C1CCCC1 C(=O)(C1CCc2c[nH]nc21)N1C(C(=O)NC2CCC(CO)C2)CC=CC1 C1(C(=O)NC2CCN(C(CCC#N)=O)C2C2CC2)CC12CCCCC2 C1(O)(C(C)NC(C2(C(F)(F)F)CC2)=O)CCN(C(C2CCOC2)=O)C1 C1(C(N(CC(CC)CC)CC)=O)CC(C)CN(C(=O)COc2ccccc2)C1 c1(NC(N2CC(N(S(C)(=O)=O)C)C2)=O)cn(C)nc1C(F)(F)F C1(C(N2CC(c3nnc(CC)o3)OCC2)C)C2CCC(C2)C1C C#Cc1ccc(C(N2CCC(CC(=O)NCC(C)(CC)CO)C2(C)C)=O)cn1 C1(CNC(C(C)=CC)=O)CN(C(=O)CSc2ccc(C(C)C)cc2)CC1N(C)C C(CCC(O)C(=O)NCCC(C)CO)NC(CSC)=O C(=O)(C1COc2ccccc21)NCC(CN=c1cc(C)[nH]c(=NCC2CC2)[nH]1)OC c1(OC)ccc(C(N2CCC(CN(C(=O)CC3CC3)C3CC3)C2)=O)cc1OC C(c1ccncn1)=C(C(=O)N(C1CC(OCC)C1)CC(C)=O)NCCCN(C)C C1(NC(c2c(OC)n[nH]c2)=O)CN(C(c2cc(C3CCCC3)[nH]n2)=O)CCC1C C1(C(=O)NC2(C(C)O)CC2)COC(CNC(=O)CCc2cnn(C)c2)C1 N1(C(C2CC(C(F)F)(OC)C2)=O)CCOCC(NC(=O)C=Cc2nccs2)C1 C(C(CNC(=O)Cc1ccnn1C1CCC1)CO)NC(C1(CS(N)(=O)=O)COC1)=O CC1(C)OC2(C(N3CC(NC(=O)CC45CCC(C)(C4)OC5)C3)=O)CC1C2 CN1CCC(C(=O)N(C)CCc2ncon2)(NC(C2CC=CCO2)=O)C1 C(=O)(CCC(C)C)NCCN(C(C=CC=CCC)=O)C1CC1 c1(OC)ccccc1C(=O)N(CC(O)CN(C(=O)CSC(C)C)C)C c1(C(N2C(C)(CNC(C3C(C(C)C)C3)=O)CCC2)=O)ccc(Br)c(F)c1F N1(C(C2N(C(=O)CC3CCCC(=O)C3)CCN(C)C2)=O)CCC2CCCC2CC1 N1(C(C(c2cccc(O)c2)C)=O)CCC(O)C(N(C)C(c2ccncc2)=O)C1 c1(N2CCN(C(c3c(CC)noc3)=O)CC2CCO)nc2cccc(C)c2o1 c1(C(=O)NC(CCN(C(CCCC(C)=O)=O)C)C)cc2c(s1)COCC2 C(=O)(CCCC(=O)NC1CCCC(C(N2CCC(C#N)C2)=O)CC1)OC N1(C(C2(OC)CCCCCC2)=O)CCC(C)N(C(=O)CCCSC)CC1 C12(CC(C)(C)C1)C(=O)NC2.C1(CNC(C2CN(C(C)C)C2)=O)CC(C(F)F)CO1 C(C(C)(O)CC(=O)N(CCNC(=O)C(c1ccc(Cl)cc1)(C)C)C1CC1)OC CC1CC(CNC(=O)C(C)(C)n2cnnn2)CN(C(=O)C(C)(C)C#N)C1 N1(C(CCC2N(C(C)C)CCC2)=O)CCc2n[nH]cc2C1.c12cccc(c1)CN2 c1(C(=O)NCc2occ(C(N(C(CC#C)C)C)=O)n2)cc(O)cc(=O)o1 C1(C(=O)NCC2CCCC(NC(c3c(CC)cno3)=O)C2)CCOC(=O)CC1 C(CCCCCC(=O)NC1CCN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1(C)C)SC c1(C(=O)NC2CC(CNC(C(C)(C)F)=O)C(O)C2)cnc(O)c(C(F)(F)F)c1 c1(CNC(=O)NC(C)C(=O)Oc2ccccc2)cnnc(O)c1.C1(=O)CO1 c1(CSCCC(=O)CCO)ccc(Br)c(Cl)c1 Cc1nc(N)cnc1C(=O)NC1CN(C(c2ccc(C(N)=O)cc2)=O)CC12CC2 C(=O)(CC1=CCCC1)N1C(CCNC(C(C)N(C)CC)=O)COCC1 C#CC1(C(N2CC3(CCC3O)C2)=O)CCN(C(=O)C(C)CCC)CC1 N1C(=NCc2cccnc2)N2CCCC(C2)C1=O.O=C1OCC(CSC2CC2)O1 C(=O)(C(C1CC1)NC(=O)C(C)C)NC(C1CCOC1)CNC(COCC=C)=O c1(NC(C2CCCN2C(=O)CCN2CCCCC2)=O)cc(Cl)ccc1C(F)(F)F O(NC(=O)C(O)CNC(C1CCCC(C)C1)=O)CC=C N1(C(C(c2n(C)ncc2)NC(=O)C(F)C2CCC2)=O)CCC2(CC1)CC(O)C2 N1(C(c2c(CC)oc(C)c2)=O)CC2CCCC1C2CNC(c1cn(C)nc1O)=O N1(C(C(C)(CO)NC(=O)C(C2CC2)C2CC2)=O)CC2(CCOC2)C1 N1(C(CCc2cccc(OC)c2)=O)CCC2C(C1)CN2C(C1CC2(C1)CC2F)=O N1(C(CC=C)=O)C2CCC1CC(F)(CNC(c1cccc3sccc13)=O)C2 Cc1ccnc(C(=O)NC2CC=C(C(=O)NC34CC(F)(C3)C4)C2)c1N N1(CCNC(C(C)NC(CC)=O)=O)CCC(NC(=O)C(CSC)OC)CC1 C1(CNC(C(C)=C2CCC2)=O)CCC(C)(C)CN1C(=O)Cn1ncn(C)c1=O C(=O)(C1=COc2ccccc2O1)N(C1CC(NC(C(CCOC)C)=O)C1)C C(=O)(C(O)CC(C)(C)C)N(C1C=CC(C)(C)CC1)C C1(CC)(NC(C2CC2c2cnccc2C)=O)CCN(CC)CC1.C12CC1C(=O)N2 N1(C(=O)Cc2csc(Br)c2)CCN(C(=O)CN2CC=CC2)C(CO)C1 N1(C(CC(C)(C)SC)=O)CC23CCCC2(C1)CN(C(C1CCC12CCC2)=O)C3 c1(C(=O)NC2CC(NC(C3CCC(=O)C3)=O)CC2O)cccc(F)c1Br N1(C(C(N2CC(C)C2)C)=O)CCC(CC(N2CC(N(C)C)C(C)C2)=O)C1(C)C N1(C(c2c(C)noc2)=O)CCN(C(=O)C=CCO)C2CCCCC12 c1(C2(C(=O)NC(C)CNC(c3cccnc3O)=O)CC2)ccc(Cl)cc1Cl Cc1ccc2snc(C(=O)NCC3CC(NC(C4CC(=O)N4)=O)C3)c2c1 N1(C(C(C(C)C)(C)C)=O)CC(NC(c2cn(CC(N)=O)nn2)=O)C2CCCC2C1 c1(C(=O)NCC2(C(=O)Nc3c(C#C)cccc3)CC2)ccc(C)c(C)c1I C1(C(C(=O)NCc2ccccc2O)N(CCOC)CC)CC2CCC1CC2 C1(C(=O)NC)(OC)CCN(C(=O)CN2CC3CCC2C3)C1 c1(CNC(C2(c3cc[nH]c3)CC2)=O)cnn[nH]1 C1(OC(CC)C)CCN(C(C)CC)C1 CC1C(NC(=O)COC2(C)CCC2)CCCN1C(=O)CCNc1ccccn1 CC1(C(=O)NCC2CCCCC2NC(c2[nH]ccc2C2CC2)=O)COC(=O)OC1 C12(CNC(c3nc(C)oc3)=O)CCC1CCN2C(=O)Cc1ncccc1C c1(C(=O)NCC2(O)CN(C(c3cc(OCC)ncc3)=O)C2)ccc(Cl)c(C#N)c1 C1(C(C)C)CCC(C(N2CCC(CC(F)F)C2)=O)N1C(=O)CC1COCCO1 C1(C(=O)NC(CCCC)(C)C)CN(C(C2CCCN2C)=O)CC1(F)F CCCCC(O)C(=O)NCC1CC(NC(C2(c3ccc(Cl)cc3F)CCC2)=O)C1 Cc1oc(C#N)cc1C(N1CC(C(=O)NCC(c2cn(C)cn2)O)OC(C)C1)=O Cn1cnc(Br)c1C(=O)Nc1ncc(CC2COC2)s1 c1(C(=O)NC(C(C)NC(c2n(C=C)nnc2)=O)C)ccc2c(c1)C(=O)CCS2 N1(C(c2nccc(N(C)C)c2)=O)C2CCC1CN(C(C1CCC(C#N)CC1)=O)C2 C1(C(N2C(CC(C)C)CC2)=O)CCN(C(=O)c2cccn(C)c2=O)O1 C#CC1(C(=O)N(CC(F)Cl)C)CCN(C(=O)C(C2(O)CCC2)C)CC1 c1(C(=O)NC2CCN(C(CN(C(=O)OC)C)=O)C2C)cc(C)c(C)c(Br)c1 c1(CC)nc(CC(=O)NCC(C)NC(=O)CC23CCCC2C3)cs1 S(=O)(=O)(c1ccc(C(=O)NOc2cccnc2C#N)cc1)N(C)C C(CCCCN=[N+]=[N-])c1cn(-c2c(CC(CN(C)CP(C)(C)=O)O)cccc2)nn1 N1(C(CC(=C=C)C)=O)CCC(NC(c2cnn(C(C)C)c2C)=O)C(F)C1 C1(O)(C(=O)NC(CNC(CNC(=O)NC)=O)C)CN2CCC1CC2 C(=O)(CCCC(C)(C)CC)N(C(CCCCn1cc(C(=C)C)nn1)C)C(C)C c1(C(=O)NCC(CO)NC(C(C)OC)=O)cccc(C(C)(C)C)c1 N1(C(C(COC)OC)=O)CC2CCN(C(=O)Cn3c(C)ccc3C)C(C2)C1 C(=O)(CC(O)CC(C)C)N1CCCC(C(=O)N(CC(C)C(=O)OC)C)(CC)C1 c1(C(=O)NC(CC)CNC(c2cccnc2CO)=O)cc(C#N)cc(C)n1 c1(CC)scnc1C(=O)NCC(=C1CN(C(=O)CC(C)c2ccco2)C1)F c1(C(=O)NC23CC(NC(Cc4ccc(OC)cc4)=O)(C2)C3)ncc(Br)cc1C C1(CCNC(CC2CC(OC)C2)=O)CCCCN1C(C1CC(C)(O)C1)=O n1(CCCC)nnnc1C(C(C)C1CCCC1)NCCCC1CCCCC1 C1(F)(C(=O)NC2CC(CNC(CN(c3ccc(F)cc3)C)=O)C2)CCCCC1 CC(C)C(O)C(C)(C)C(=O)NCC(C(=O)N(C)CCOC1CC1)N(C)C N1(C(C2N(C)CCN(C(C3C4CCC(C4)C3C)=O)C2)=O)CC(=O)N(C)C(=O)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCCC(CNC(C(C)(C)C#N)=O)C1 c1(C(C)C)nccc(NC(C2CCN(C(C3CNC(=O)N3)=O)C2C)=O)n1 C1(NC(=O)C=CCN2CCOCC2)CC12CCN(C(C1OCCCO1)=O)CC2 C1(N(C)C)CCC(C(=O)NCCC2CC(NC(c3cc(Cl)n[nH]3)=O)C2)CC1 Cc1oc(CNC(c2cn(C)nc2O)=O)nc1C(=O)NC1(C2CC2)CC1 c1(NC(=O)NCCC2CCCC(C)C2)ccc2c(c1)C(O)CC2(C)C C1(OC)CCC(c2nc(-c3cccc(N)n3)nn2-c2nc(Br)nn2C)CC1 C1(NC(c2c(C3CC(=O)NC3)cccc2)=O)COC2(C1)CN(C(=O)C(F)F)C2 c1(C(=O)NC(C#C)(CC)CC)ccc(OC)c2ccccc12 C1(NC(c2nc(CC)on2)C)CCN(C(=O)CC(c2cccs2)SC)CC1C C1(C(=O)NCC2(CCC)CCC2)CCCN(C(=O)Cc2cc(C)n(C)n2)C1 N1(CC(=O)N(CCCCN(C)C(c2cc(Cl)ns2)=O)C)CCCCS1(=O)=O C1(C(=O)NCC2CCC(NC(C3C(C)CC(=O)N3)=O)C2)Cc2cncn2C(=O)N1 c1(OC)cc(C(=O)NC2CCC(NC(=O)C(C)SC)C2)ccc1C(F)F C1(C(F)(F)F)(C(=O)NC(CC=C)CNC(c2cscn2)=O)CCCCC1 N1(C(CC2(C=C)CC2)=O)CC2CC(NC(=O)C(C)NC(=O)C(C)(C)C)C1C2 CN1C(=O)CCCC1C(N1CCC(C)(C)C1C(=O)Nc1cccc(CO)c1)=O C12(CNC(=O)C(C3(O)CCCC3)F)CCC(CC1)N2C(C1CCCC(CF)C1)=O C1(NC(CN(C2CC2)CC)=O)CC12CC(NC(=O)C(O)c1cnc[nH]1)C2 n1(CC)cnc2c(N3CCCN(C(=O)C(C)O)C(C)C3)ncnc12 C12(CCC)CC(C(=O)NCCC3CC(NC(=O)C(C)CN4CCOCC4)C3)(C1)C2 C12COCCN1C2=O.C1(C(=O)NCc2ccccc2)CCCN1Cc1cn[nH]c1 C(=O)(CCCCCCCCC(=O)N1CCCCC2(CCN(C(=O)C3CC3)C2)C1)OC C1(NC(COC(C)=O)=O)CCC2(C1)CN(C(C1CNC(=O)C1)=O)C2 C(=O)(N=c1[nH]nc(C(=O)NCSc2ccccc2)s1)C1C(N)CCO1 C1(C)(C(N2CCC(O)(C(CNC(C=NOC)=O)C)C2)=O)COC2COCC2O1 Cc1cccn2c(C(N3CC(CNC(c4cccn4C)=O)C(O)C3)=O)cnc12 c1(C(N(CC(C)NC(=O)C(C2CC2)SC)CC)=O)ccc(-c2ccccc2)cc1F Cc1cc(C(=O)NCC23CC2CN(C(C2CC2C(N)=O)=O)C3)nc(C)n1 C1(NC(C=NOC)=O)CCCC(NC(c2c(C3CC3)cnn2C)=O)CC1 C(C)(CCCCNC(=O)CC1(OC)CCC1)NC(c1nc(C(=O)NC)sc1)=O c1(C(=O)NCC(=CC(=O)N(CC(=C)C)C)C)cnnn1CC C1(c2nnnn2C2CCC2)(NC(CC)C)CCN(C(N)=O)CC1 N1(C(c2c(OCC)n[nH]c2)=O)CCC(CNC(C2CCCC(OC)C2)=O)CC1 C1(N(CC(C)CNC(C2CC2c2cccs2)=O)C=O)CC(N(C)C)C1 C1(NC(c2c(C)cncn2)=O)CC(NC(c2ccc(NC=O)cc2)=O)C12CCC2 C1(C2(C(C)O)CC2)CCCN1C(=O)C=CC(C)(C)C.C12CC(C1)NC(=O)C2 N1(C(C(CC)C)=O)CCCC2C(NC(C3CC(C)N(C)C3)=O)C(C)(C)C12 c1(CC(=O)N(CCCNC(C=CC(CC)C)=O)C)cccc(F)c1 c1(CC)noc(C(N2CCC(c3cccc(F)c3)(NC(=O)C(C)CF)C2)=O)c1C c1(CNCCC2CCCC(=O)O2)[nH]c2ccccc2c1Br c1(C(N2CCCN(C(Cc3c(C)ccs3)=O)CCC2)=O)ccc2n[nH]c(C)c2c1 C=CCCC(C(=O)NC1CC(C)(C(N)=O)C1)NC(=O)CC1CCCCO1 C#Cc1cc(C(=O)NCC2(NC(C3CC3C#C)=O)CCCCCC2)cc(Br)c1 N1(C(c2c(C)coc2)=O)CC2CCC(CNC(C3CC4CCC(C3)N4C)=O)(C2)C1 C1(OC)(CNC(c2ccoc2C)=O)CCN(C(C23CC(CCO2)C3)=O)C1 C1(NC(C(CCC)O)=O)CN(C(C2CCC(C(C)(C)C)O2)=O)CC2(CC2)C1 c1(OCC)cncc(C(=O)NC(C)(CNC(=O)Cn2cc(C3CC3)cn2)CO)c1 Cc1ccc(C(=O)N(C)CCC2CCN(C(=O)C(C)(C)F)CC2)c(O)c1 C1(CC=C)(NC(c2ccc(CCC)cc2)=O)CCN(C(c2csc(C)n2)=O)C1 C1(NC(C(C)N2CCCC2)=O)CC2CCC(C1)N2C(=O)CCC1CC(C)(C)CO1 C1(C(=O)NCC2(CNC(C)=O)CC2(F)F)CCc2nn[nH]c2C1 C1(O)(COC(C(C)NC(=O)C2CC2)=O)CCC2CCCC12 C12(CNC(C3CCCN(C(C)C)C3)=O)CCC(NC(=O)CCF)(CC1)CO2 N1(C(c2c(CC)nccc2)=O)C(CC(=O)Nc2ccc(O)cc2C)C2CCCC12 N1(C(c2cncc(NCC)c2)=O)CC(O)C(O)C1CNC(c1nnccc1C)=O c1(OC(C)C)ccc(C(=O)OCc2ccc(C#N)o2)cc1 C#Cc1c[nH]nc1C(=O)NCCN(C)C(c1cccnc1O)=O CCCCCC(=O)NC1CCCC1NC(C1(Sc2ccccc2)CC1)=O c1(C(=O)NC2CC(CCNC(c3n(CC)ccc3)=O)C2)cccc(C)c1O Cc1onc(C(=O)NC(C)(CNC(c2cccnn2)=O)C2CC2)c1Br N1(C(c2c(C)occ2)=O)CCC(NC(=O)CC2CC3(CC3)C2)C1C CC1CCCc2cc(C(N3CCC4(C3)CC4(F)F)=O)nn21 Cc1cc(CCC(=O)NCC2(NC(c3ccn(CC#N)n3)=O)CC2)cc(F)c1 C(=O)(CCCN=[N+]=[N-])NC1(c2ccccc2)CN(C(c2ccc(CC)[nH]2)=O)C1 N12CC(C(C)(C)C1)CN(C)CC2=O.c1(NC(=O)CCN2CCC2)ccc(Cl)cc1 C1(CC(=O)NCC2CCCN(C(=O)CC3CC(F)(F)C3)CC2)CCC(=O)NC1=O C1(COC(C)=O)CN(C(=O)C=C(C)CNC(=O)C(F)C(C)C)C1(C)C C1(c2ccc(F)cc2)(NC(C=C(CC)C)=O)CCN(C(=O)C=CS(C)=O)CC1 N1(C(C(CCC)N(C)C)=O)CCN(C)CC1C(=O)NCC1CC(=O)NC1=O c1(C(=O)NCC2CCN(C(C3CC(OC)C3)=O)C(C)C2)nccc2nn[nH]c12 c1(C(=O)NCCN(CCC)C(C2(NC(C)C)CC2)=O)cccc2ncsc12 C1(NC(C(C)SCCCC)=O)CC2CC(NC(=O)Cc3ccc(CC)cc3)C2C1 N1(C(C(C=CC)O)=O)CCCN(CCCCNC(c2cccc(CC)c2)=O)CC1 CC1CCC(CC(N2CC(F)(CNC(c3cncs3)=O)C2)=O)C1 N1(C(c2cc(C(C)=O)on2)=O)CCC(C(F)F)(CNC(=O)C(C)(C)CF)C1 N1(CCCc2ccc(C)cc2C)CC2CC1CC2(C)O C1(NC(c2ccc(C)c(C)n2)=O)CN(C(=O)Cc2ccno2)C2(CCOC2)C1 c1(CC(=O)NC(CNC(C2N(CCC(C)C)CCC2)=O)C2CC2)ccnc(O)c1 CCC(C)(CO)C(=O)N1CC(C(C(=O)Nc2ccc(CCO)cc2)OC)C1 CC1CC(NC(c2ccsc2F)=O)CN1C(C1CCOC(C)C1)=O c1(C(=O)NC2(COC)CN(C(=O)Cn3ncccc3=O)C2)ccnc(N(C)C)c1 c1(N(CCOCCNC(C2(OCC)CCCC2)=O)C)ncc2scc(Br)c2n1 N1(C(C=CC(CC)=CC)=O)CCC(O)(CNC(=O)COC(CC)CC)C1 C1(NC(C=CSC)=O)CCN(C(=O)C(=O)NCC2CC2)CC1C c1(C(N2CC(C)OCC2)=O)cn2c(n1)CCN(Cc1cc(Br)co1)CC2 c1(CC(=O)NCC(C2CC2)NC(c2n(C=C)nnc2)=O)cccc2c1SCCC2 C(=O)(CC(C)(C)CC(F)F)N(CCC(C(C)C)NC(=O)C=CC1CCOCC1)C c1(CC)cc(C(=O)N(C)CC2CN(C(C3(CC)CCNC3=O)=O)CCO2)c(C)o1 N1(C(c2c(CC)ncs2)=O)CCCC(COC)(NC(=O)C(C)c2ncco2)C1 c1(N2C(CNC(C3CC(=C)C3)=O)CC(C)(C)C2)cc(CCCC)nc2ncnn12 C1(CNC(C2CC(C)(CC(C)C)C2)=O)CCCCN1C(c1cc(O)n(C)n1)=O N1(C(=O)NC(CCSC)C)CCC(CCNC(C)(C)C)CC1 N1(C(C2CC=C(C)CC2)=O)CC(NC(=O)Cc2cnsc2)C(C2CC2)C1 Nc1c(C(=O)NCC2(c3cn(C4CCC4)nn3)CC2)cnn1CCO CCCCCC(C)(C)C(=O)N1C(C(=O)NCCF)CC2CC12 N1(C(C2(C#C)CC2)=O)CCCC(F)(CNC(=O)Cc2ccc(C(=O)NC)nc2)C1 c1(-c2cnc(=NC)[nH]c2)cnc2[nH]cc(C(=O)NCc3cncc(C)c3)c2c1 C1(CNC(C(COC)C)=O)CCC(CN(C(=O)COc2cncc(C)n2)C)CC1 N12CCOC(CC1)C2.N1(Cc2snc(CC)n2)CCC(F)(F)C1c1ccccc1 C1(CCC)C(=O)NCCN1C(=O)CC1CCN(C(c2ccc(Cl)c(Cl)n2)=O)C1 N1(C(C(Cc2cc[nH]n2)NC(c2cccn(C)c2=O)=O)=O)CCOC2C(O)CC12 C1(c2nc(-c3ccc(N(C)C)nc3)nn2C)SCC2C=CC1C2 CC(C)CCC(C)NC(=O)CC1CCCN1C(c1cn[nH]c1)=O C12(CC(N3CC=CC(OC)C3)=O)CCC1CN(C(c1cc(C)ncc1C)=O)C2 C(C)(C(C(=O)NCC1CC(O)CCO1)NC(=O)C(C)OCCN(C)C)OC c1(CNC(C2CCCCCC2)CO)cccc(F)c1Cl c1(C(=O)NCC2(C(N(CCN(CC=C)C)CC)=O)CC=CC2)cncc(O)c1 C1(CNC(CSC)=O)CC2(CCN(C(C3CN(C)C3)=O)CC2)CO1 N1(C(C)C)CCC(N=c2nc(N3CC4C5CCC(C5)C4C3)c3c([nH]2)CCC(C)C3)C1 c1(C(=O)NCCC2CCC(NC(C=Cc3cnc(C)s3)=O)C2)c[nH]c(=N)cc1C Cc1cc(C)n(CCCC(=O)NCCOC2CN(C(=O)Cn3cnc(=N)[nH]3)C2)n1 C1(O)(CNC(Cc2cc(C)sc2)=O)CCCN(C(C2(C#N)CCCCC2)=O)CC1 CN=c1ccc(C(=O)NC2CCC(CNC(=O)CCNC(=O)NC)CC2)c[nH]1 c1(C(=O)NC(C(=O)N(CC(=O)OCC)CCC)C)ccn(C)c1 c1(C(C(=O)NCCS(C)(=O)=O)N(C)Cc2cccs2)ccc(C(N)=O)nc1 c1(N(CC(=C)C)C(N2CCCC(C#C)(O)C2)=O)ccc2ccccc2c1 C1(C(=O)Nc2ccc(C#C)cc2C)CCCN1NC(=O)C(C)C(CC)CC CC(F)(F)C(F)(F)CC(=O)N1CC=CC(NC(c2cc(Cl)sc2Cl)=O)C1 C(=O)(C#CC1CCCCO1)N1CC(CCNC(=O)C(C)N2CC(C)C2)(OC)C1 c1(CC(=O)NCC2(NC(=O)C=CC3CCCCC3)COC2)cccc(Cl)c1F N1(C(C(C(C)OC)O)=O)CCn2ncc(CNC(c3cnoc3C)=O)c2C1 c1(C(=O)NC(C2N(C(CCSCC)=O)CCC2)(C)C)ccc(F)c2[nH]ccc12 CCC(CC)C(C)C(=O)NCC1(C)CCN(C(c2cc(N)c(C)c(N)c2)=O)C1 N1(C(C2N(C(C(CCC)NC(N)=O)=O)CC2)=O)CCCC2(CCOC2)C1 C1(NC(CCc2ccn(C)n2)=O)CN(Cc2cccc(Cl)n2)CC(C)(C)C1 N1(C(CC2CN(C)C2)=O)CCCC(C2CCN(C(=O)C(C)(C)C(C)(F)F)CC2)C1 N1(C(C(=O)NCCc2cnsc2)=O)CCc2c([nH]c3ccc(F)cc23)C1 C1(CNC(CCCOC(C)C)=O)CCN(C(C2CN(C(C)C)C2)=O)C1(C)C C1(N(C(c2scc(CNC(C(CC)C#N)=O)c2)=O)C)CCOC(C)(C)C1 C1(O)(CNC(CC2(C=C)CN(C(c3cc(C)co3)=O)C2)=O)CCC(C)(C)C1 c1(C(=O)NC(CNC(CNC(C)=O)=O)C)cc(C)n(-c2ccc(C(C)C)cc2)n1 Cc1ccccc1CC(=O)NCC1CCCN1C(=O)C(C)Cc1cnn(C)c1 c1(C(=O)OCC(=O)Nc2ccc(Cl)cc2)cc2c(nc1O)CCSC2 C1(C=O)(NC(C(C2CCC2)C(c2snnc2C)C)=O)CC(F)(F)C1.CSCC C(c1ccc(C(C)C)cc1)=CCC(N1CC(N(C(CCN(CCC)C)=O)C)C1)=O c1(C(N2CCCC(C)(CCC)C2)=O)ccc(-c2ccccc2Cl)c2cc[nH]c12 C(Cc1cc[nH]n1)(C(=O)N(C)Cc1cn[nH]c1)NC(C(C1CCC1)OCC)=O C1(C(=O)NCCOC2CCN(C(C(C)SCC)=O)C2)C2CCC(=O)C12 C=CC1(CC(=O)NCCCn2cccn2)CN(C(=O)CC2(C)OCCO2)C1 O=C1NC2(CCOCC2)CC2=C1C(c1cnc3sccn13)NC(=O)N2CCF c1(C(CN(CCOC)C(c2cc(C)[nH]n2)=O)OC)ccc(Cl)cc1 c1(C(=O)NCC2CCCN(C(=O)CC(F)(F)F)CC2)cc2n(c1)CCSC2 CCC(C)C(C)(O)CNC(C1CCCC(NC(=O)C(O)CC(N)=O)C1)=O Cc1cc(N)c(C(N2CC3(CCN(C(C4(n5ccnn5)CC4)=O)C3)C2)=O)cc1F N1(C(C2N(C(C)=O)CCCC2)=O)CCOC(C)(CNC(c2c(C)ccn2C)=O)C1 c1(C(C)C)cc(C(N2CCC(N(C(=O)CSc3ccncc3)C)CC2)=O)n(C)n1 c1(CC)noc(C)c1C(=O)NCC1(NC(C2CS(=O)C2)=O)CCCC1 C1(C(=O)NC2CCC(CN(C)C(C3(C(C)(F)F)CC3)=O)CC2)CCOC(=O)CC1 C12(C(N(C)Cc3cccs3)=O)CCN(C(=O)Cc3cccnc3)CCC1C2 N1(C(c2c(Cl)cnc(C)n2)=O)CC(NC(c2cc(CF)on2)=O)C(N=[N+]=[N-])C1 N1(C(COC)=O)CCOCC1CC(=O)NCCC1CC(=O)N(C)C1 C1(C(N2C(CNC(C3N=C(C)SC3)=O)CC(F)(F)C2)=O)CCc2ncncc2C1 N1(C(C(CC)CC)=O)CC2(NC(=O)C(CC(C)C)OC)CCC1C2 C12(NC(c3ccc(Cl)c(C(F)(F)F)c3)C)CCC(N)(CC1)C2 c1(OC)cc(CC(=O)OCC2CN(C(=O)C3=C(Cl)CC3)C2)c(F)cc1O Cc1nc(O)[nH]c1C(=O)NCC1CCCN1C(C1CCOC1c1ccnn1C)=O c1(C(=O)NCC2(F)CN(C(C3CCCO3)=O)C2)sccc1-n1ccnn1 CCCCCC(C)(C)C(=O)N(CCCCNC(=O)C=Cc1ccc(CC)cc1)C c1(OC)cc(C(=O)NCC2(CN(C)C(C3CC34CCOC4)=O)CC2)c(F)cn1 c1(NCC)cc(Cl)ccc1C(N1CC(NC(c2cccc(C)c2)=O)CC1CO)=O S(=O)(=O)(CC(=O)N1CC(NC(=O)C(C)OCC2CCCO2)C1)NCC C1(O)(CCNC(C2(CC#C)CCCO2)=O)CCN(C(C2CCC2=C)=O)CC1 C(c1cccc(Cl)c1)=CC(=O)NC1CN(C(C(CC#C)O)=O)CC1CC(C)(C)C N1(C(Cc2n(C)ccn2)=O)CC(NC(=O)Cc2ccco2)CCC(O)C1 c1(C(N2C(CC)CN(C(=O)C(F)=CC3CC3)CC2)=O)cc(OC)cc2c1CCC2 c1(OCC)ccc(Cl)c(C(N2CC(NC(=O)CCC(CC)OC)CC(C)C2)=O)n1 c1(CC)cc(NC(=O)CC2(NC(CC(F)(F)F)=O)CC2)sc1C(=O)OC C1(CNC(Cn2c(C(C)C)ncc2)=O)C2CN(C(=O)C=C(C3CC3)C3CC3)CC12 C=C1CC(C(=O)NCCc2ccoc2C(F)(F)F)N(C(=O)Cc2ccncc2)C1 c1(SCC(=O)NCC(Cn2cc(COC3CCOC3)nn2)OC)cnc(C)nc1 CCC(=O)CCC(=O)NCC(C)C(N1CC(CC)C(F)C1)=O c1(CNO)ccc2c(c1)OC(F)(F)O2.C(C(F)Cl)N(C)CCC1CC1 C1(C(=O)NCCOCC(=C)C)(C)CCOC1.C(=O)(C(CN(C)C)N(C)C)N N1(C(c2cncc(OC)c2C)=O)CCOC2(CCN(C(=O)CC(F)(F)F)CC2)C1 CN(C)S(=O)(=O)N1CC(C(=O)NCC2CC2NC(C2CCCS2(=O)=O)=O)C1 c1(COC)cc2c(c(=O)o1)C(c1ccc(OC)nc1)NC(=S)N2CCC(C)=O CC1CCCC=C1C(=O)NC(CN=[N+]=[N-])C(=O)NC1CCC(C(N)=O)C1 C(C(C)(O)CCN=C(NCc1cccc(Cl)c1)NCC1(OC)CCC1)OC CS(=O)c1ccc(C(=O)NC2CCN(c3nnc(C(F)F)s3)CC2F)cc1 N1(C(CNC(N)=O)=O)CC2CCN(C(c3cccc(C4CCC4)c3)=O)CC12 CCCC(CNC(=O)CSC)C(=O)NC1CCOC1(C)C c1(N2CC(c3ccc(C)cc3C)C(C(=O)O)C2)ncc(C#N)cc1C#N c1(CC(N2CCC(C(C)NC(=O)Cc3ccnc(Br)c3)C2)=O)cc(F)ccc1O C(=O)(C1CCCn2nccc21)N(CCN(C)C(c1cnc(=N)[nH]c1)=O)C N1(C(C2C3CC4C(C3)C24)=O)CC2(C=C(C(=O)N3CC4(CCCC4)C3)CO2)C1 C=CC1(C(=O)NC2CC(O)CN(C(=O)Cn3ncccc3=O)C2)CCCCC1 n1(CC)ccc(C(=O)NCC2CCN(C(c3ccns3)=O)C23CC3)cc1=O C=CC1(C(N2CC(N(C)C(c3cc(C)nnc3O)=O)C(F)C2)=O)CCCCC1 C1(F)(CNC(c2ccn(CCOC)n2)=O)CCCN(C(=O)C(C)NS(C)(=O)=O)C1 C1(CNC(=O)CC2CCCC2)COCCN1C(c1cccnc1O)=O N1(C(CC(CNC(C=CC=CCC)=O)OC)=O)CC(=O)NC(=O)C1C N1(C(c2ccoc2CNC(C(C)OCC=C)=O)=O)CC(C)CC1c1ccccc1 C1(CNC(c2c(C)ccnc2C)=O)CCCCN(C(=O)C2=COCCC2)CC1 c1(NCC(COc2c(CCC)cccc2)O)cc(Br)c(C)cn1 C(=O)(C(C)(C)S(C)(=O)=O)N1CC(NC(c2c(OC)nc(Cl)cc2)=O)C(C)(C)C1 CCC(CC(=O)NC(C(=O)NCc1cnco1)C(C)O)CC(C)C N1(C(C(CC)N(C(=O)CCn2cccn2)C)=O)CCCC(C#N)C1 CN(CCC1CCCCC1)N1CCN(C2CC3C=CC2C3)CC1 c1(OC)cc(F)c(C(=O)O)cc1S(=O)(=O)NCc1cc(O)ccc1Cl c1(NC(c2ccc(CCC(=O)O)cc2)=O)ncnc2[nH]cnc12 CCCC(C)(O)CC(=O)NCC1CC(F)CN1C(c1cscc1CC)=O C#Cc1cccc(CC(=O)NCC#CC(N2CCCC(C)C2CCO)=O)c1 C(=O)(C1=CCCN(Cc2cc(Cl)c(O)cc2F)C1)N(CCC(=O)N1CCCC1)C c1(C(N2C(CNC(CCC(C)C)=O)C(C3CC3)CC2)=O)nnc2n1CCCCC2 C1(C(N2CC(C=C)(CC(=O)N(C)Cc3ccns3)C2)=O)CCOC(C)(C)C1 N1(c2nc(-c3coc4ccc(CC)cc43)on2)CCN2CCCC2C1C C(CC(C)(C)CNC(=O)CC1CCCC(C)C1)NC(C(C1CCCC1)OC)=O c1(N(CC(=O)NC2CC2NC(=O)CNC2CNC(=O)C2)C)ccc(C#N)cc1F C1(CC(=O)NCC(CC)NC(C2CCCN2C2CC2)=O)COCCOC1 CC1CCC(C(N2CCC(NC(N)=O)C2)=O)N1C(=O)CCc1ncccn1 N1(C(C(C2(OC)CCCCC2)(F)F)=O)CCC(NC(=O)CN2CC=CC2)C(C)C1 c1(C(=O)NC2CC(CNC(C34CCCCC3OCC4)=O)C2)ccnc2[nH]nnc12 CCC(Cc1ccccc1)C(=O)NC1CCC(NC(c2n[nH]c(C)c2F)=O)C1 C(CCC(C)NC(C1CCC(C)C1)=O)NC(C(C)OCC)=O C1(NC(C(COC)(C)O)=O)CCN(c2ccnc(C3CC3)n2)CC(C)(C)C1 CN1CCNCC1C(N1CC2C(CF)C2C1)=O C1(C(N(C)CC2CCCS2)=O)CC12CCN(C(c1ccc(O)cc1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NC1CC(CC(=O)N(CCCCC)CCO)C1(C)C Cc1ncc(F)c(=NCC2COC(C)C2)[nH]1 O(S(=O)(=O)CCc1cccc(F)c1)CC(=C)CO C(CCN=C(NCC1CCN1C(C)(C)C)NC1CCC(NS(C)(=O)=O)CC1)OCC N1(C(C(CC)CC(C)C)=O)CCC2(CC1)CN(C(c1ccc(Cl)cc1O)=O)C2 c1(C(C(=O)NCC(CC)NC(C23COCC(C2)C3)=O)C)cccc(Br)c1 c1(CNC2CCN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)ccncc1F C1(C(=O)NCCCCCCN(C(CCCC=C)=O)C)C2Cc3ccccc3C12 C12(C(N3CCC(C)(COC)C3)=O)C(NC(c3ccc([N+](=O)[O-])o3)=O)C3CC1C2C3 C1(CC(=O)N(CCCOC)Cc2ccncc2)CCCCC1C n1(CC)cc(C(N2CC(NC(c3cccc(Cc4nccs4)c3)=O)C2)=O)c(C)n1 C1(OC)(CNC(C2(Cl)CCC2)=O)CCN(C(=O)C(O)c2cnc[nH]2)C1 N1(C(COc2cccc(C)c2F)=O)C(CNC(=O)C(C)CO)CC2COCC12 C1(C(N(CCOC)CCNC(c2cccn2CCOC)=O)=O)OCCCC1(C)C C(=O)(C1=CC2(CCOC2)C1)N1CCC(OCCNC(CCC(=O)OC)=O)C1 N1(C(CCC=CC(C)C)=O)CCC2(C1)CN(C(=O)Cc1csc3nccn13)C2 C1(NC(C(CCC)F)=O)CCCCCCC1NC(c1c[nH]c(C#N)c1C)=O c1(C(=O)NC2CCC(NC(C(C)(F)F)=O)C2)ccc(C2(C)CC2(F)F)cc1 C#CCC(CC)NC(=O)CCl c1(C(c2n(C(CC)C)nnn2)N)nc(Br)nn1C.c1(C)cn(-c2ccccc2)nn1 c1(CC)ccc(C(C)CC(=O)NCCN(C(=O)C(C)(COC)OC)C2CC2)cc1 CC(C)(CCNC(C1CC(CC2CC2)C1)=O)NC(=O)C(CO)c1ccccc1 n1(CC)cc(Cl)c(C(N2CCC(C)(NC(=O)Cc3cccc(OC)c3)C2)=O)n1 N1(C(CSCC=C)=O)CCCC(CNC(=O)CC(C)C2CCCC2)C1 C1(NC(c2cn(CC)nn2)=O)CCCC(C(N2CCC(OCCN(C)C)C2)=O)C1 C=CC(C)(O)CC(=O)NC(C1CCN(C(=O)C(c2ccc(C)cc2)C)CC1)(C)C N1(C(CC(C)C)=O)CCOCC1C(=O)NCc1cncc(Cl)c1 Nc1cc(C(N2CC(CNC(=O)CC3CC4(CC4)C3)C2)=O)cnc1Cl CC1(OCC(=O)NC2CC(CC(=O)NC3CNC(=O)C3)C2)CCCC1 N1(C(C(=O)NCc2ncc(-c3c(C)n[nH]c3C)o2)=O)CCC(O)(C2CC2)C1 C1(CN(C2CCN(C)C2)C(C(=O)NCC)=O)CCN(C(C)=O)CC1 c1(C(=O)NC2(C)CC(NC(CC(C)F)=O)C2)cn(C)[nH]c1=N c1(OC(CC)C(=O)NC23CC(CNC(=O)CC4CN(C)C4)(C2)C3)ccccc1C C1(CC)CN(C(=O)CCn2ncn(C)c2=O)CC1C(=O)N(C1CC2CCC1O2)C N1(C(C2CC23CCCC3)=O)CCC2(CCC2)C(CNC(C2(CCF)CC2)=O)C1 C1(CNC(CC(C=C)C)=O)CCC(C)N(C(=O)CC2CN3CCC2CC3)C1 c1(C(=O)OC)cc(C(=O)NCC(CNC(=O)C(C)(C)C2CC2)CO)cc(C)c1 Cc1cc(C(N2CC(NC(=O)C(C)N(CC(F)(F)F)C)C(C)(C)C2)=O)nc(O)n1 N1(C(c2c(C)oc(Cl)n2)=O)CC2CCCC(CNC(C3CCS(=O)(=O)C3)=O)C2C1 C1(NC(Cc2c(C)nn(C)c2C)=O)CCCC12CN(C(=O)Cc1sccc1Cl)C2 C1(NC(C=NOC)=O)CCC2(CC1)CC2NC(=O)CSCc1ccncc1 Cc1cc(P(C)(C)=O)oc1C(=O)NC1CCN(C(=O)C(O)C(C)C)CC12CCC2 C(=O)(C1=C(Cl)CCOC1)NC1CC(C)CN(C(=O)Cc2cnccn2)C1 N1(C(C(COC)C)=O)CC=CC(NC(=O)CCc2nc(-c3ccoc3)no2)C1 C(=O)(C(CC)C(F)(F)F)NCC1(CNC(CC=CCC)=O)CC12CCC2 C1(NC(c2c(C)n(C)nc2)=O)CC2CCC(C1)N2C(c1cc2cccn2cn1)=O c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2)ccc(F)c(SC)c1 N1(C(c2cnn(C(C)C)n2)=O)CCCC1(C)C(=O)NC1(CN(C)C)CCC1 N1(C(c2ncc(OCC)nc2)=O)CCCC(NC(C23COC(CCO2)C3)=O)CC1 N1(CC)CCCCC1C(=O)NC1CCN(c2nnnn2-c2ccccc2)CC1 C1(C(=O)NC2C(NC(c3c(CC)con3)=O)CCOC2)CCCCC1(C)C c1(NC(c2n(CC)nnn2)CCc2ccccn2)cc(Cl)c(C)cc1OC N1(C(c2cc(C)nn2C2CC2)=O)CC2CN(C(=O)CC(O)C(C)C)CC(C1)O2 C(=O)(N1CCCc2nccn21)c1c(CNC(=O)C=C2CCC2)n[nH]c1 N1(C(C(CC(C)C)C)=O)CCC2CCN(C(c3cc(C(F)F)ccc3Cl)=O)C2C1 N(C1CCCc2ccccc21)(C(C(=O)NC1C(CN(C)C)COC1)=O)CC(C)C Cc1cc2ccc(C(N3CC(NC(C4CC4(C)C)=O)C4(CC4)C3)=O)cc2o1 C(=O)(C(C1CCOC1)OC)N(CC(=O)N(CCO)CCO)CCOC c1(C(N2CC(CCC)N(C(C3CCCS3)=O)CC2)=O)cccc2cnsc12 C(C(CC(=O)N1C2CCC(C2)C1CNC(C1(O)COC1)=O)C(F)F)N(C)C c1(C(N(C2CN(C(C(CC)NC(=O)COC)=O)C2)C)=O)cnc2[nH]ncc2c1 CC(C)C(O)C(C)C(=O)NCC1CCN(C(c2nccc3occc23)=O)C12CC2 C(C)(CC(=O)NC1CCOCC1NC(=O)CC1CC=CC1)(C1CCC1)N(C)C C1(NC(=O)C2=COCCO2)CCCCCCC1NC(=O)C1CC1 C(=O)(CCCCC(N)=O)NC1CC(NC(C(C)OCc2ccccc2)=O)C1 CC(C)C(C(C)NC(C1(Br)CC1)=O)NC(=O)Cc1ccc(C(F)(F)F)nc1 c1(OC)ccc(C(C)CC(=O)NCC(C)NC(=O)Cn2nnc(C3CC3)n2)cc1 C1(NC(C#CC(C)(C)C)=O)CCCC2CN(C(C3(C)CCCC3)=O)CC12 c1(C(=O)NC2(CCO)CN(C(CC3CCC(C)O3)=O)C2)cnc(O)c(Cl)c1 C1(NC(C2CCCCN2C(c2ccccc2F)=O)=O)C(O)C2CCOC12 c1(C(N(C(CC)CC)C)=O)nc(CNC(=O)C(F)C2CCOC2)oc1C C1(C(=O)NCC(C)(CNC(c2ccc(CSC)o2)=O)OC)CCC(F)(F)CC1 C1(NC(c2n(CCOC)nnn2)(C)CCC2CC2(Cl)Cl)COc2cc(CO)nn2C1 c1(C(=O)NCC#CCNC(c2cn(CC)nc2C)=O)cc(F)cc2cccnc12 c1(C(N(CC(C)NC(C2(C(C)(F)F)CCC2)=O)C)=O)c(O)cccc1F Cc1ccc(Cn2cc(CCC3CCCN3C(=O)C=CI)nn2)o1 C1(N(C(C(CCCC)O)=O)C)CCC2CN(C(c3cccc(Cl)c3N)=O)CC12 C(C)(N=c1[nH]c2c(F)cccc2o1)C1CCN(C(c2c(C)n(C3CC3)cc2)=O)C1 c1(C(N2CCOCC(NC(C34CC(C)(C3)C4)=O)C2)=O)nc2cc(O)ccc2[nH]1 c1(N2C(C3(NC(c4cc5c(o4)CCCC5)=O)CC3)CCC2)ncnc2scnc12 Cc1cc(C)c(NC(=O)NC(c2c[nH]c3ccccc23)C(Cl)(Cl)Cl)cc1Br C1(NC(c2snc3ccccc23)=O)CS(=O)(=O)CC1N=c1nc[nH]n2cccc12 C12(NC(CS(CC)(=O)=O)=O)CCCC1N(C(c1cnc(N(C)C)nc1)=O)CC2 C1(C(=O)NC2CC(C)N(C(c3c[nH]cc3Br)=O)C2)Cc2nccnc2C1 n1(CC(=O)NC2CCCC2O)cc(Cn2cccc2)nn1.C12CCCN1C2 Cc1cccn2cc(C(N3CC=CC3CNC(=O)C=CC=C(Cl)Cl)=O)cc12 CCC(CC(=O)N(CC(=O)NCc1ccccn1)C1CC1)C1CCC1 Cc1c[nH]c2ncnc(NC3CC(F)CN(C(c4cc(CO)ccc4O)=O)C3)c12 c1(C(=O)NCCNC(CCC(=O)N(CC)CC)=O)ccc(O)c(N)c1 c1(N2CC(c3n(C)nnn3)C2)nc(CSC)c2ccccn12 C1(CNC(CCN(C(C2CC(C)C2)=O)C)=O)CCC=CCC1 C1(F)(C(=O)NCC2C(NC(C3N(C(=O)OC)CCC3)=O)CC2O)CCOCC1 c1(C(N(CCN(C(=O)CCc2c[nH]c(=N)[nH]2)C(C)C)C)=O)c[nH]nc1C(C)(C)C CC1(C)CN(C(=O)CC2CCC(=O)C2)CC1NC(=O)CC1CC(F)C1 C12(CC(=O)N(CC(CC)NC(C3CCN(C)C3)=O)CC)CCC(CC1)CC2 C1(C(N(C2CCN(C(=O)COCc3nc[nH]n3)C2)CC)=O)C2CC3C(C2)C13 N1(C(C2C(C)OCC2)=O)CC2CCC1C2NC(c1cccc(-c2cscn2)c1)=O c1(OC)cnc(Cl)c(C(=O)NCC2CCCN(C(c3cc(Cl)ccc3Cl)=O)C2)c1 C1(CCC(=O)N(CCCCC)CCCC)CNC(C)C1 C(=O)(CC(O)CC(C)(C)C)N1CCC(CC=C)(NC(C2CCC(=O)O2)=O)C1 Cc1onc(-c2cccs2)c1C(=O)N(c1ccccc1)CC(C)C#N C(CNC(=O)COCCOC)(CC(F)(F)F)NC(C(COCC)O)=O c1(C(N2CC(OC)(CNC(C3(C)COC(=O)C3)=O)C2)=O)cc(F)c2[nH]nnc2c1 n1(CCNCc2ccc(C(=O)OC)c(F)c2)cc(C#N)ccc1=O N1(C(CCN2CCN(C)CC2)=O)CCC2CCC(C1)N2C(=O)CC1C=CCC1 C1(C)(CC)CC(NC(c2cc(C(C)C)oc2C)=O)CN1C(c1cccc(O)n1)=O N1(C(c2ccc(C(C)(C)C)o2)=O)CC(CNC(C2CC3CC3C2)=O)C2(CCC2)C1 C1(F)(CNC(C(N2CCSCC2)C)=O)CCN(C(C2CCCC2(C)C)=O)CC1 C12(C(=O)NC3CCN(C(C)=O)C3)COC(C1)C(NC(c1ccc(F)cn1)=O)C2 C1(C(N2CCC(F)(C(=O)N(C)CC3CCCCC3)C2)=O)(OC)CCOCC1 c1(-c2nccc(C(=O)Nc3cc(O)nc(Cl)n3)c2)cccc2ccnn12 C1(CC(=O)N(C2CCN(C(c3cnoc3C)=O)C2)CCC)CCC(=O)NC1 C12(C(N3C(C=C)CCC3)=O)C(NC(c3cnns3)=O)C3CC1C2C3 C1(NC(C(C)C#N)=O)CN(C(C2CC3(CCOCC3)CO2)=O)CC12CCOCC2 C=C=C(C)CC(=O)NCCCC1CN(C(c2conc2COC)=O)CCO1 c1(OC(C)=O)ccc(C=CC(N2CCN(C(=O)CSC(C)(C)C)C(C)C2)=O)cn1 N1(C(c2onc(C)n2)C)CC2(C)CN(C(c3ccnn3CC(C)C)=O)CC2(C)C1 CN=c1[nH]cc(C(=O)NCC2CC(F)CN2C(=O)CNC(c2cscn2)=O)o1 C1(C(=O)OC)(C(=O)NCC2CC2CNC(=O)NC(C)C)CCCC1 c1(CC)cc2c(CC(=O)OCC3(C(F)F)CCOC3)cc(=O)oc2cc1O N1(C(CCC(=C)Cl)=O)C2CCCC1CN(C(c1ccn3nccc3n1)=O)C2 C1(CNC(c2ccc(C(O)CF)cc2)=O)CC(F)CN1C(C1(O)CCCCC1)=O CCC(CNC(c1cc(CC2CC2)on1)=O)(CC)NC(=O)C(F)C1CCC1 C1(C(C)NC(c2cc[nH]n2)=O)CCN(C(=O)C2=CCC2)C1 c1(CC)cccc(C(N2CCC(F)C(NC(=O)COC(C)C)C2)=O)c1O CC(C)(N=[N+]=[N-])C(=O)NC1CC(CC(=O)NCCCCC(F)(F)F)C1 c1(C(=O)NC(C2(O)CCN(C(C(CO)OC)=O)C2)C)cc2ccccc2n1C C(=O)(N1CCC(C(N2CCCC(C)(O)C2)=O)O1)C1CCN(CC)CC1 C(=O)(CCC(=O)N(C)CCNC(C1(c2cncnc2)CCCC1)=O)NC NC(=O)C(N)CCC(=O)NC1CCC2(CN(C(=O)COCCO)C2)O1 C1(CC)CCC(C(=O)N(CC(C)NC(c2cnn(CCOC)c2)=O)C)CC1 Cc1nnn(CC(=O)NCCCCCN(C(=O)C(c2ccncc2)C)C)n1 C1(C(=O)NC(CNC(C(C(C)C)NC=O)=O)(C)C)OCC2CCCC12 N1(C(C2(CCNC(c3cncn(C)c3=O)=O)CCC2)=O)CCC(C2CCOC2)C1 N1(C(C(C=C)(C)C)=O)CC2CCCC2(CNC(=O)CCc2ccc(C)o2)C1 C12(C(N)=O)CC1CN(C(=O)COc1ccc(NC(c3csc(S)n3)=O)cc1)C2 c1(OC)cc(C(=O)Nc2ccc(C)nc2Br)c(-c2cncc(N(C)C)c2)cn1 N1(C(=O)OC(C)(C)C)CC2CC(Sc3cnc(-c4ccccc4F)s3)C1C2 C1(C#N)(C(=O)NCCCCCCN(C)C(c2ccccc2)=O)CCCOC1 c1(NC(CCCC)CCC)ccc2ncnc(O)c2c1 CCCC(CCCNC(=O)Cc1cc(C)ns1)NC(=O)C(C#N)C1CC1 c1(C(=O)NC2CC(C)(NC(=O)CSCc3ccccc3)C2)cc(Br)ccn1 c1(C(=O)O)cc(C(=O)NCC(c2ccc(F)cc2)CO)c2ccccc2c1 CCCCC(CC)C(=O)N1CCC(COC)(NC(c2cc(C(C)(C)C)no2)=O)C1 C#CC1(NC(C2(CNC(C3CCOC3CC)=O)CC2)=O)CCC(C)CC1 Cc1nnc(CC(N2CC(OCCNC(=O)C(N3CCNC3=O)C)C2)=O)s1 c1(CCCC(N2C(CCNC(=O)CC3(O)CC3)CCCC2)=O)cc(F)ccc1F N1(C(C(F)OC)=O)CC(C2CCN(C(c3cc(Cl)ccc3C(C)C)=O)CC2)C1 c1(CCC)[nH]ccc1C(=O)NCCCC(C)NC(=O)CC1CC12CC2 N1(C(C2C(C)(C)C2CNC(=O)CC2(C#N)CC2)=O)CCC2(CC=CCO2)C1 C=CC(CCC)CC(=O)NC1CN(C(=O)CCCc2ccccn2)CC1O O=C(C1Cc2ccc(Cl)cc21)NC1CC(CO)N(C(c2ccc(Cl)nc2Cl)=O)C1 c1(C(=O)NC(CC)(C)CNC(=O)Cn2c(C)c(C)sc2=O)ccc(C)c(C)c1N CC1C(C)N(C(c2cnc3n2CCCC3)=O)CCN1C(c1ccc(Cl)o1)=O c1(C(=O)NC2(CCNC(C(C)(C)OCC)=O)CC2)sc(Cl)cc1Cl C1(C(=O)NC(C)(C)C)CC(=O)N(C2CN(Cc3c(C)scc3)C2)C1.c1(=O)c(=O)[nH]1 C1(c2nnnn2C2COC2)(C(=O)NCCNC(=O)CO)CCC(=O)NC1 c1(C(N(C(CN(C(C2=C(C)OCC2)=O)C)C)C)=O)cccc2c1OC(C)C2 N1(C(C2(C(C)NC(C3CCCCC(=O)N3)=O)CC2)=O)CCc2nc(O)[nH]c2C1 C1(NC(C2(CCCC)CC2)=O)CN(C(=O)CC2(CSC)CC2)CC1OC Cc1cnc(CNC(C2(NC(=O)C(O)C3CCC3)CC2C)=O)o1 C(=O)(C(O)CCNC(=O)CCC1(C)CCCN1C(c1cc(C#N)cs1)=O)OC C1(NC(c2cccc(-n3cnnn3)c2)=O)CCCC2CCNCC12 C1(O)(CNC(c2c(CC)nn[nH]2)=O)CCCN(C(=O)C=CC2(C)COC2)CC1 c1(C(=O)NC2CCN(C(c3c(CC)non3)=O)CC2)cccc(OC)c1N c1(C(=O)Nc2c(C(N(CC)C)=O)scc2)ccc(Br)cc1.c12sc(C)nc1C2 C1(NC(CCc2n(C)ccn2)=O)CCCC(N(C(=O)C=Cc2nnn(C)n2)C)C1 CC(C)C(CCN(C(=O)C(C)C1CCC1)C)NC(=O)C(C)(C)O N1(C(c2ncn(C(C)C)c2)=O)CCC2(C1)C(F)(F)C2(F)F N1(C(c2cc(C)sc2)=O)CCC(C)C1CNC(c1sccc1-n1ccnn1)=O C12(CC)CC(C1)C(=O)NC1CC1C(=O)NC2.C1(CC)CC1C(=O)OCC N1(C(C(CCOC)C)=O)CC=C(C(=O)NCc2ccc(C)c(C)n2)C1 N1(C(c2c(OC)ccs2)=O)CCC(CC(=O)NC2CCC2O)CC1 C1(NC(c2cc(C(F)F)no2)=O)CC2CC(C1)N(C(=O)COc1ccon1)C2 N1(C(C(c2n(C)ncc2)O)=O)CC2CC1CN2C(c1ccc([N+](=O)[O-])o1)=O c1(NCCN(CC)CC)ccc(S(=O)(=O)N2CCCCC2CO)cc1F C(=O)(CC(O)CC(C)(C)C)NCC(CC=C)C(=O)Nc1cccn2ncnc12 c1(N2CCCC(NC(C3CCCC(C(N)=O)C3)=O)C2)ccc([N+](=O)[O-])cc1Br c1(C(=O)NC(C(C)C)CCN(C(=O)CC2CC2C2CC2)C)ccn2cnnc2c1 c1(C(=O)NCC(CO)NC(c2cc(CC)nn2C)=O)nccc2c(C)cccc12 N1(C(C23N(C(C4C(CC)CCC4)=O)CCC2CCC3)=O)CCC(O)(C2CC2)CC1 C1(c2onc(C)n2)CN(C(C2CCN(C)CC2)=O)CC(C)O1 n1(CCCNC(C(C)SC(F)(F)F)=O)cc(CC2CCCC2)nn1 c1(C(N)=O)nccnc1C(=O)NC1CCC1NC(C1CC(F)(CO)C1)=O C1(CCNC(=O)CC(F)(F)C(F)F)CN(C(C2CC3(CSC3)C2)=O)CCS1(=O)=O CCCC(C)(O)CC(=O)N1CCC(C=CC(=O)NC(C)CCCCO)CC1 c1(N2CCCC(C)(C(N(C)C)=O)C2)nccc(=NCc2csc(C3CC3)n2)[nH]1 N1(C(CSCC#C)=O)CCCCCC(NC(c2cc(C(=O)NC)ccc2C)=O)C1 C12(NC(C(c3cn(C)nc3)=O)=O)CC1CN(C(c1ccncc1C1CC1)=O)C2 C=C(C)CC(=O)N1CCC(n2cc(CNC(C3CCCN3C(C)=O)=O)nn2)C1 c1(NCC2(CN(C)C)CCCC2)ccc(S(=O)(=O)NCC2CC23CC3)c(Br)c1 C12CCCN(CC1)CCOC2=O.Cc1sc(-c2ccccc2F)nc1C.C(C)(C)(C)O c1(C(C)(C)CNC(=O)NCc2cnc(CSc3ncccn3)s2)cccc(O)n1 CC(F)(F)C(C)(C)CC(=O)Nc1ncc(C(F)(F)F)cc1Cl c1(CNCC2(C)CCCN(c3ncc(F)cn3)C2)cc(Br)cc([N+](=O)[O-])c1O C#Cc1c[nH]nc1C(=O)NCCC(C)NC(=O)Cc1csc(-c2ccsc2)n1 N1(C(N2CC(Oc3c(C)cc(N)cc3)C2)=O)Cc2nnc(C)n2C(CC(C)C)C1 c1(C(=O)NC(CCN(C(c2c(OC)nn(C)c2)=O)C)C(C)C)cc[nH]c(=N)c1Cl CS(=O)CCC(=O)N1CCC(NC(C2CCCCN2C(=O)CCC(F)F)=O)C1 Cc1ccc(C=CC(=O)NCC(C)(C2CCC2)NC(c2cc(Cl)cn2C)=O)s1 Cc1cc(=O)n(C)nc1C(N1CC(NC(=O)CN2CCCC2CO)CC1CO)=O C(CC(CNC(C1(F)CC=CC1)=O)NC(=O)C(O)CC1CCCCC1)OC CC1=C(c2cc(C(=O)Nc3cnn4ccncc34)c3n[nH]cc3c2)CCCC1 N1(C(=O)COCC2CCCO2)CCN(C(=O)C=Cc2nccs2)C(CCO)C1 c1(OCC)ccc(-c2csc(NC(c3ncc(Br)c(N(C)C)n3)=O)n2)c(F)c1 C#CCC(CC(=O)NCC1(CCO)CC1)NC(c1csc(C)c1C)=O C12(C(N(C)Cc3c(C)ccs3)=O)CC3CC(C1)CC(O)(C3)C2 C1(NC(N(C)CC2(CO)COCCN2C)=O)CC2(CCC2)C12CCC2 N1(CC(=O)NC(C)C(C)NC(=O)C2=C(Cl)CC2)CCCCS1(=O)=O C1(C(=O)NC2(CCCC(N3CC(C=C)C3)=O)CCC2)CCOC(CC)C1 c1(C(CCC)N(C(C2CCCS2)=O)CC2CCN(CC)CC2)ccc(OC)cc1 Cc1c(C(N2CCCOC(CNC(C3(C#N)CC=CC3)=O)C2)=O)nc2sccn12 N1(C(c2c(CCCC)ocn2)=O)CCN(C(C2CCC2C(F)F)=O)C(CCC)C1 N#Cc1ccc(CC(=O)NC(C(=O)NCC(=O)N2CCCO2)C2CCC2)cc1 c1(C(=O)NC2CC(CCNC(CSc3cn(C)nc3)=O)C2)cc2n(c1)CCOC2 N1(C(CNC(CCCCC)=O)=O)CCC(C2(NC(C3C=C3C)=O)CC2)C1 c1(CC(=O)NCC2CCN(Cc3c[nH]c(Br)c3)CC2)cccc(Cl)n1 N1(c2nc(N(CCN(CC)CC)C)c3c(n2)scn3)CCC2(CC1)COC(C)C2 C(=O)(CC(C)(C)C(=O)N1CCCN(C(C2CCC23CCC3)=O)C(CO)C1)OC N1(C(C2C(CCC)C2)=O)CCN(C(c2ccc(CC)o2)=O)CC1CC c1(C(=O)NC2CC(NC(C3CCCCC34CC4)=O)CC2O)cccc2ccnn12 N1(C(c2c(C)onc2Cl)=O)CCC2C(CCCN2C(c2ccnnc2)=O)C1 c1(C(N2C(CC(=O)Nc3c(C)nc(Cl)nc3)CCCC2)=O)cc2ccncc2[nH]1 c1(C(N2C(CNC(C(C3CCOCC3)OC)=O)CC2)=O)cc(C)c(O)c(C)c1 c1(-n2c(-c3c(F)ccc(OC)c3)nc(C3CSC3)n2)cc(O)nc2ncccc12 C1(NC(C2CCC2)=O)CC2(C1)CN(C(C1CCC(C(F)(F)F)OC1)=O)C2 c1(C(=O)NCC(CNC(CSCCOC)=O)O)ccc(NS(C)(=O)=O)nc1 Cc1nc(F)ccc1C(=O)NC1CN(C(=O)C(C)OCCC(C)C)CC1(C)C CCC(CC(=O)N1CCC(C(=O)N2CCOCC2C)=C(F)C1)CC(C)C C12(C(=O)NC(CCC)c3nn[nH]n3)CC(CO1)N(C(=O)C=Cc1cc(C)no1)C2 CC(C)(CCC#N)C(=O)N1CCOCC(NC(C2CCCCC(F)(F)C2)=O)C1 c1(C(C(=O)NC(CNC(c2c(C)ccs2)=O)(C)C)O)ccc(C(F)(F)F)cc1 C1(CNC(C(CC)CC)=O)CCC12CN(C(=O)Cc1ccc(C)cc1)C2 C1(N(C(=O)CCN2CCOC2=O)C)CN(C(=O)CN2CCSCC2)CC1(C)C C(=O)(C(F)(F)C(F)F)N1CC(NC(c2ccn(CC)n2)=O)(COC)C1 N1(CC(=O)NC2(CNC(c3cc(C(C)C)on3)=O)CCOC2)CCCNC1=O n1(CC(=O)NC2CCC2CNC(c2ccc(C3CC3)cn2)=O)cnccc1=O CP(C)(=O)C(O)C(=O)NC(C1CCCC1)CNC(c1cncc(N2CCCC2)c1)=O c1(NCc2cnc(C)[nH]2)nccc(=NC2CC(C3CC3)C2)[nH]1 N1(C(C2C(C(N)=O)CC2)=O)CCN(C(c2ccc(F)cn2)=O)C(CF)C1 CCC(C(=O)N(CCCNC(c1ncc(F)c(OC)n1)=O)C(C)C)C(C)C C1(CN(C(=O)Cc2cccnc2)C)C2CN(C(=O)CCCC3CCCCC3)CC12 C(c1ccc(C(=O)OC(C)(C)C)cc1)=CC(=O)NC(C#CC)(C)C c1(SCCOCCC(=O)N(CC(=O)O)C)ccc(I)cc1 c1(C(N2CC(NC(=O)C(C)C(=O)OC)CC(OC)C2)=O)c(Cl)ccc2c[nH]nc12 Cc1nc2ccc(C(N3CCC(C)C3CNC(C3CCC(C)(C)O3)=O)=O)cc2o1 CC1=NC(C)(CNC(=O)CC2C=CC(NC(C3CCCCN3C3CC3)=O)C2)CS1 CC1CN(C(c2ccc(Cl)c(C(F)F)c2)=O)CCCN1C(=O)C#CC1(C)COC1 c1(CC)ncc(C(=O)N(C)CC=CC(=O)NCCC2CCC(C)C2)cn1 C(C(=O)N1CC2C(NC(=O)CN3CCCS3(=O)=O)C2C1)(C(C)C)OCC c1(C(=O)NCC2(NC(C(CC)SC)=O)CCCC2)scc(C)c1C C(=O)(C(CCC1CCC1)NC(c1cc(CC)n(C)n1)=O)N(CC(=O)NCCC)C CCC(CC(=O)N1C(C(=O)N(CCO)CCN(C)C)CCC1C(C)C)C1CCC1 C(CCCCCN=c1nc(OC)c(F)c(C)[nH]1)NC(C(CCCOC)C)=O N1(C(C(F)=CCC)=O)CCC(C2CCN(C(c3c(F)cc(F)cc3Cl)=O)C2)C1 CC1C(C)N(C(c2cc(C#N)ccc2O)=O)CCN1C(c1ccoc1)=O Cc1nc2cc(NC(C3(C(=O)O)CC4(CC(F)C4)C3)=O)ccc2s1 C=CCCC(C(=O)NC(C)CCOC)NC(c1cc(C)c[nH]1)=O N1(C(CCN(C(C2CC3CC(=O)C2O3)=O)CC)=O)CCC2CCC(C1)S2 N1(C(c2cccc(C#C)c2)=O)CCC2CN(C(=O)CCC(CC)CC)CCC12 C1(NC(c2n(CC#C)cnn2)=O)CN(C(C23CSCC2C3)=O)C2(CCCC2)C1 N1(C(CCSC)=O)CC=C(CNC(=O)CC2CN3CCC2CC3)CC1 Cc1cnccc1C(=O)NCC1CC1NC(c1n[nH]cc1Cl)=O c1([SH](CC(=O)NC2C(CNC(C=CC(=O)OCC)=O)COC2)C2CC2)ccccc1O CC(CNC(=O)C(C)n1cnnn1)CC(=O)NCCOC1CC1 N1(C(CCN(C)CC)=O)CCN(C(C2C(C)C2C)=O)CC(C)(C)C1 Cc1ccc(C(=O)NC(C)C(C(C)C)NC(C2CN(C)C2)=O)cc1NS(C)(=O)=O O=C1CN(C(=O)CCCNC(c2ccco2)=O)c2cc(Br)ccc2N1 C1(NC(C2CCN(C)C2)=O)CN(C(c2conc2C(C)(C)C)=O)CCC1CO N1(C(C(C2CCC2)OCC)=O)CC2CC1C2CNC(=O)CN(C(=O)COC)C N1(C(COCCC=C)=O)CCC(NC(c2c[nH]c(Br)c2)=O)C(F)C1 c1(C(N2CC(CCNC(=O)CCc3ncco3)C2)=O)ccnc2[nH]nnc12 c1(C(=O)NC(C2CCN(C(CCC3C(C)C3)=O)C2)(C)C)cc2occc2n1C C1(NC(C2C(C)CN2C(c2cn(C)c(=O)n2C)=O)=O)CCC=CCCC1 c1(SC)ccc(OC(C)C(N2CCC(C)(NC(=O)CSc3nccs3)C2)=O)cc1 c1(C(C)=O)nc(N2CCC(NC(c3ncoc3C3CC3)=O)C(F)C2)c(C)c(Cl)n1 N1(C(C(C)N(C)C)=O)CC(C)CC1C(=O)NCCC12CC(CO1)C2 C1(C(N(CCCCN(C(c2c(C)cnnc2O)=O)C)C)=O)CCN2CCCC2C1 c1(OC(C)C)cccc(NC(C2(C)CCN2C(=O)C=CC2CC2)=O)c1Cl n1(CC(=O)NC(CCC)CNC(c2ccc(=O)oc2)=O)cc(C)ccc1=O Cc1n[nH]c(C)c1C(C)C(=O)N(C)CC1CCCN1C(=O)C1=NOCC1 C#CC1(C(=O)NCC2(CC)CC2)CN(C(=O)C=Cc2cncn2C)C1 C12(C(=O)OC)CCN(C(=O)Nc3cncc(C#N)c3)CCC1C2 c1(OC)cccc(Cl)c1CN=C(NC1CCCC1)NC1CCCC(F)C1 CC(O)C(C(=O)N1CC(CNC(c2cc(C(F)F)no2)=O)C1)N(C)C c1(C(=O)NC2C(C)CCN(C(=O)CCC3CCC3)C2)cccc2cnnn12 O(NC(=O)CC(C(C)(C)C)NC(C1(O)CCOC1(C)C)=O)CC1(C)CCC1 n1(CC)nc(C)c(C(=O)NC2CN(C(=O)C(O)CC3CC3)CC2SC)c1C C1(NC(c2cnn(C)c2N)=O)CN(C(c2cnc(O)s2)=O)CC2CC12 N1(C(C2C(CNC(c3cccc(O)n3)=O)OCC2)=O)CCCC(F)(CO)C1 C(c1ccc(Cl)cc1Cl)=CC(N1CC(N(C)Cc2ccc(C#N)cn2)C1)=O c1(C(N2CC3CCN(C(C(CC)(C)C)=O)CC32)=O)cccc2[nH]nc(O)c12 C1(CNC(C(C)c2ccco2)=O)C2CCC1CN(C(C1CC13CCSCC3)=O)C2 c1(C(N2C(C)C(NC(c3cn(C)c(=O)cn3)=O)CCC2)=O)cc2sccc2n1C C(=O)(C(C)(C)CCCNC(=O)C(F)C1CCOC1)NC(C#C)CC1CC1 C1(C)(CC(=O)NC(C(C)NC(c2cc(-c3ccco3)c[nH]2)=O)CO)CCCCC1 CCS(=O)CCN=c1[nH][nH]c(=NCCCc2ccnnc2)[nH]1 c1(C(N(C)CC2CCCN2C(=O)C(c2ccnn2C)O)=O)cc(O)ncc1F C(=O)(C1=CCCC1(C)C)NCCC1(C)CCN(C(C(C)C(F)F)=O)C1 C(=O)(CC(CC)C(C)C)N(C1CCN(C(=O)Cc2cc(OC)ccc2F)C1)CC C(=O)(CCCC(F)(F)F)N1CCC(N(C(=O)C(C)(C)CN(C)C)CCOC)C1 Cc1nc(C)n(CC(=O)NCC2CC2NC(C23CC(C)(C2)C3)=O)n1 S(=O)(=O)(c1ccc(Cl)c(F)c1)NC(COC)C(C)C N1(C(CC2OCC(C)(C)C2)=O)CCC2(C=C(C(=O)N3CC4CC3(CO)C4)C2)C1 C1(O)(C(N2CCCC(N(C(CCCCSC)=O)C)C2)=O)CCCCCC1 N1(C(C(COC)C)=O)CCC(CNC(C2CCCC(C)(C)C2)=O)C12CC2 C(=O)(C1=NOCC1)N(CCNC(C1N(C(CCC#C)=O)CCC1)=O)C1CC1 c1(OC)cc(C(=O)N(CCCNC(C2CC(=O)N(C(C)C)C2)=O)C)ccc1C#N C(=O)(C(CC)CCOC)N1CCC(CC)(NC(=O)COCCOC)C1 C1(C)(C(=O)NCC(N(C(c2scc(C)c2C)=O)C)C2CC2)CC(C(F)(F)F)=NO1 N1(C(c2c(OC)nccn2)C(=O)NCC2CC2)CCc2ncsc2C1 Cc1cc(C)n(CC(=O)NCc2cn(CC(N3CCOCC3CC3CC3)=O)nn2)n1 c1(CC)nc(C)ncc1C(=O)N(C)CCN(C)C(c1csc(COC)c1)=O N1(C(c2cncc(OC)c2)C(=O)OC)Cc2cnn(C3CCCC3)c2C1 C1(CCC)CN(C(=O)Cn2cc(C)cn2)CCN1C(c1cnc(C)c(Cl)c1)=O c1(C(=O)NCC2(C(=O)NOCC(F)F)CC23CCC3)cccc2ccoc12 C1(OC)CC2(C1)CC(C(N1CCC(CNC(=O)CCSC(F)(F)F)CC1C)=O)C2 Cc1cnc(NC(C)CNC(c2cc(CO)on2)=O)nc1O c1(N2CC3CC(NC(C(C#C)(C)C)=O)C3C2)ncc2c(n1)CCOC2 C1(CNC(C2CCC(=O)O2)=O)CC(F)CN1C(=O)CC1CCC(C(F)(F)F)O1 c1(-c2ccc(-c3ccc(C(N(CC(=O)O)C)=O)cc3)cc2)cccc(C#N)c1 N#CC1(C(=O)NCCC(O)CNC(=O)CCSc2ccc(F)cc2)CCCOC1 CC1CCN(C(=O)C(F)C(C)(C)O)CC1N(C)C(C1CCC(N=[N+]=[N-])C1)=O C1(NC(CN(CC)CC)=O)CC2CCCC(C1)N2C(c1nccc(Cl)c1Cl)=O c1(C(=O)NC(CC#CC)C(=O)N(CC(O)(C=C(C)C)CO)C(C)C)cccc2[nH]ncc12 C12(C(C)NC(=O)Cn3cc(CNC(C4CS(=O)C4)=O)nn3)CCC(CC1)C2 c1(CCCNC(C(C)(C)OCC)c2ccccc2)ccc(C(=O)O)cc1 c1(CC(=O)NCC(C2CCC2)NC(C2N(C)CCOC2)=O)cccc2cn[nH]c12 c1(C(=O)NC(CCOC)CNC(c2cc(C)c(C)s2)=O)ccc2[nH]c(C)cc2c1 c1(C(N(CCOCCNC(CCOCC)=O)C)=O)cncc2ccc(F)cc12 N1(C(c2c(C)cnnc2)=O)CCC2(CC1)CC2CNC(=O)C(C)c1cccs1 C1(C(N2CCCCC2C(C)C)C(=O)NCC(C)C)CC2C(C1)C2(F)F C(=O)(CCCN=[N+]=[N-])NC1CCC(C(=O)NCc2c(COC)noc2)CC1 c1(C(N2C(C)(CNC(CC3(C(=C)F)CCC3)=O)CCC2)=O)cnc2ccoc2c1 C=C(Cl)CCCN=c1cccc(S(=O)(=O)NCC(c2csc3ccccc23)O)[nH]1 C=CC1(C(=O)NCC2(C)CCOCC2)CCN(C(=O)C(C)CSC)CC1 C1(NC(c2cnc(CC)[nH]2)=O)COC2(C1)CN(C(c1nc3ccccc3[nH]1)=O)C2 CCC(C)(O)C(=O)NCCCCNC(=O)C(C)CCc1cccc(F)c1 c1(C(N2C(C(C)NC(C(C)OC)=O)CCC2)=O)cc(Br)c(C)s1 C1(NC(=O)CNS(=O)(=O)C2CC2)CN(C(C2CC2(F)F)=O)CC1C(F)(F)F N1(C(CS(CC)=O)=O)CC(NC(c2cnc(N(C)C)cn2)=O)CC(F)(F)C1 CC(C)C(C#N)C(=O)NCC1(NC(C2CCC(=C3CCC3)CC2)=O)CCC1 CC1C(=O)NC(=O)CN1C(=O)CC(=O)Nc1cnn(C[Si](C)(C)C)c1 CC(C)CCC(=O)C(=O)NC1CC(n2cc(-c3cccc(CO)c3)nn2)C1 c1(C(=O)NCc2csc(C3CC3)n2)c[nH]c2c(-c3cnoc3)cccc12 c1(-n2c(C3(NCCC(C)OC)CCC(=O)N(C)C3)nnn2)sc2ccccc2c1C O=C(CN1C(=O)COc2ccccc21)NCC1(O)CC(NC(C2CC2(F)F)=O)C1 Cc1cc(C(=O)NC2CCOC2C(N2CCC3CC23C)=O)ccc1C#N CC1Sc2ccccc2N(C(=O)C(=O)NC2CCC2)C1C c1(C(=O)NC2(CN(C(=O)C(O)c3ccsc3)C)CC2)cn2ccccc2n1 C1(NC(C(C(C)C)NC(C(CCSC)OC)=O)=O)CCC2CCCC1O2 CCCCC(F)C(=O)N(C)CCN(C(=O)CC(CC1CCCC1)CC)C c1(C(=O)NC(C(C)OCC(C)C)C)cnc2[nH]c(C3CC3)cc2c1 C(=O)(CCP(C)(C)=O)NCCCN(C(C)C)C(C1CS(=O)(=O)CCO1)=O c1(C(N2CC3C(NC(C4C(C(=O)OC)CC4)=O)(C3)C2)=O)c[nH]c2cccc(C)c12 N1(C(c2c(C)cc(C)o2)=O)CCOCC(CNC(=O)CN2CCCC2CO)C1 c1(OC)cccc(OC)c1C(N1CCC(C)(C(=O)NCC2(O)COC2)CC1)=O C1(CCCCNC(c2cc(CC)on2)=O)CCCN(C(=O)C(C2CC2)C2CC2)C1 c1(CC)cccc2c1N(CC(=O)NC1(CO)CCCCC1)CC2 n1(CC#C)c(C)cc(C(=O)NC2CCC(NC(C3SC4C=CC3C4)=O)CC2)c1C C1(CNC(c2c(CC)c[nH]c2)=O)CC2(C1)CN(C(c1ccc(C(N)=O)cn1)=O)C2 c1(OC)ncc(C(N2CCC2CNC(c2ccc(OC(C)C)cc2)=O)=O)cc1Cl N1(C(CC2C(C)(C)OCC2)=O)CCN(C(c2cnc(Cl)s2)=O)C(C(C)(C)C)C1 N1(C(CCC(=O)NC)=O)CCCCC(CCC(N2CCC(C#N)C2)=O)C1 Cc1ccncc1C(C)(C)C(=O)NCCN(C(=O)C(O)C1CCC1)CCOCCO C(=O)(C1CCCc2ccnn21)NCC(CNC(c1cnn(CC)c1Br)=O)O C1(N(C)C(C2CC2C#N)=O)CCCN(CC23CC(C)(CO2)C3)C1 C(CCCS(=O)(=O)N(C)Cc1ccc(Oc2cncc(Cl)n2)cc1)OC CCS(=O)(=O)CC(=O)N1CCC(c2n[nH]c(CNC(=O)CC(C)(C)O)n2)CC1 Cc1nn(C)c(-n2cncn2)c1C(=O)OC1CCCCC1C O(NC(=O)CCCCCNC(=O)CC(C)CC(C)C)CC(=O)OCC N1(C(C(C)OCCCC)=O)CCC2(CCC(NC(=O)C(C)=CC(C)(C)C)C2)C1 C1(C(N2CCC(NC(C3CC34CC4)=O)CC2)=O)CC2CC(C1)C(=O)N2 C1(C(C(=O)N(CCCn2cc(C(NS(N)(=O)=O)C3CC3)nn2)C)F)CCCCCC1 c1(C(N2C3CC(NC(CCOC)=O)C3CC2)=O)cc2c(C(F)F)nn(C)c2s1 c1(OC)ccc(O)c(C(=O)NCC2COC(CNC(c3cc(CO)on3)=O)C2)c1 c1(C(N2C(CN(C(C(COC)N(C)C)=O)C)COCC2)=O)ccc(C)c(OC)c1 N(C(=NCCSC)N1CCC(C(CC)CC)C1)CC(=C)C.c1(O)ccc(F)c(F)c1 C#CC1CCCN(C(=O)C(C2(O)CN(C(=O)CC3CCC(C)(C)O3)C2)F)C1 CCC(CNC(c1ccccc1OC1CC1)=O)N=c1[nH]nc(CCOC)s1 CC(C)(C)C1=CCN(C(=O)CC(C(C)(C)C)NC(C2CCC3(CCC3)O2)=O)CC1 C1(C(=O)NC2(CNC(c3scc(C(C)=O)c3)=O)CC2)CC1C1CCC1 C1(CNC(=O)C=CC2CCC2)CCCN(C(C2Cc3cscc3C2)=O)CC1 C(=O)(C(CC)C(C)(C)CC)NC1CCCC(NC(c2onc(CC)c2C)=O)C1 c1(C(=O)NC2CCCN(C(C3C4CCCOC34)=O)C2)cccc2nc(O)ccc12 CC1CCCCN(C(C23CC2CN(C(c2cc(Br)ccn2)=O)C3)=O)C1 C1(C(=O)NC(COCCN(C(=O)OC)C2CC2)C)CCCC(C)C1 n1(C(C(=O)N(CCNC(=O)CCN2CCC2)CC)C)cnc(C#N)n1 c1(C(=O)NC2C(C)CCN(C(c3cnc[nH]3)=O)C2)cc2ccccc2c(=O)o1 C(=O)(C(C)CC(F)(F)F)NC(CCNC(c1ccc(CSC)cc1)=O)C c1(C(=O)NCC(CNC(c2c(C)nns2)=O)C)cc2nccnc2[nH]1 N1(CC)CCOC(C(=O)NC(C)CN(C)C(C2(C(=O)OC)CC2Cl)=O)C1 C1(C(=O)NCCCOCC)(CF)CCN(C(=O)CC2(CC)CCCC2)C1 C1(NC(=O)CC2CCCOC2)CCCN(c2ccnc(C3CC3)n2)C1 N1(C(CCOC(C)C)=O)CC(NC(c2cnc3occc3c2)=O)C2(CCC2)C1 C#Cc1cc(C(N2CCOC(CCCNC(C3CCCCS3)=O)C2)=O)cc(F)c1 N1(C(C(CC#C)OC)=O)CCC2(C=C(C(=O)N3CCC(C)(C(N)=O)C3)C2)C1 c1(N2CCC(C3CC3)(CC)C2)cnc(C#N)c(C#N)n1.C(CC(=O)NCC)OCC C(CC(C(=O)Nc1cscc1C)NC(C1CC(C)(C)C1)=O)OCC C1(CC(=O)NC2C(CCC)CCC2)CN(C(=O)COc2ccsn2)CCC1(C)C c1(NCCOCC(=C)C)[nH]c(=NC2CCN(CC)CC2)nc2ccc(OC)cc12 c1(NC(C2N(C(C3(COC)CC3)=O)CCC2)=O)ccc(C2=NCCN2)cc1 N1(C(CNC(=O)CNC(=O)CC2CCCC3CC23)=O)CC2C(C1)C2(F)F CC(C)(CC#N)C(=O)N1CCN(CCNC(C2CCCN2C2CCCC2)=O)CC1 O=S(=O)(C1CCCC(F)(F)CC1)N1CCCC(CN2CCOCC2)C1 CCC(C(=O)NC(CNC(=O)Cc1cn(C)c2ccccc12)C1CC1)C(C)(F)F CCCC(C(=O)NC1CCC(NC(=O)C=Cc2sccc2C)C1)N(C)C O=C(C(CCC1CCCO1)N1CCCCC1c1cc[nH]n1)NN1CCOCC1 C1(NC(C(C)(C)OCC)=O)CC(C2CCN(C(=O)Cc3ccn(CC)n3)C2)C1 N1(C(CC(CC)C)=O)CCOC2CN(C(c3cccc(C4CC4)c3)=O)CC12 C1(CNC(CC2(C(=O)OC)CCCC2)=O)CN(C(=O)CCSCC(C)C)CCO1 CC1OCCN(C(=O)CCn2ccnc2)C1C(=O)NCCC[Si](C)(C)C C1(NC(CCC(C)CN(C)C)=O)CN(C(=O)CCCCC#N)CC1C1CC1 c1(CNC(N(c2cncc(Br)c2)C(C)C)=O)cccc(C#N)n1 C1(CNC(C(F)=C(C)C)=O)CN(C(=O)C(c2cccc(C)c2)C)CC(C)(C)C1 c1(CNC(C(c2ccccc2)N(CC=C)CC)=O)ccc(F)cc1OC N1(C(C(CCC)N(C)C)=O)CCN(C(c2ccc(CO)cc2)=O)C(COC)C1 Cc1cnc(NC(C2CC3CC3N2C(C2CNC(=O)O2)=O)=O)c(C)n1 C1(C)(C(=O)NCC(C)N(C)C(c2ccc(-n3ccnc3)cc2)=O)CCCOC1 N1(C(C(C2(O)CCC2)NC(C(CC(=C)C)OC)=O)=O)CC2CCC(C1)C2O CC1(CCO)CCN(C(C2CCCCC2NC(c2cccc(CC#N)c2)=O)=O)C1 N1(C(=O)Cn2nccn2)CCCC2(CCN(C(=O)C(C3CC3)C3CC3)C2)C1 N(C1CCCc2ccccc21)C(N1Cc2n(C)cnc2CC1)=O c1(NC(CC(CCC)NC(c2cnn(CCN(C)C)c2)=O)=O)ccc2c(c1)OCO2 C1(NC(C(C2CCC2)OC)=O)CN(C(c2occc2C)=O)CC1O C1(N(C(CN2C(C)CC2)=O)CCO)CCN(C(=O)CC(C)F)CC1 C1(O)(CN(C(C=CC(C)NC(=O)C=Cc2cscn2)=O)C)CC(CO)C1.C c1(C(N(C(C)C(=O)N(CC)Cc2ccc(Cl)cc2)CC)=O)ccc(O)c(CC)c1 Nc1cc(C(=O)N(CCCNC(=O)CC(F)(F)F)C2CC2)c(F)c(O)c1 C1(C2(O)CN(C(=O)C(=C3CCCCC3)F)C2)(CNC(C2C3CNC(=O)C32)=O)CC1 C1(NC(C(C)N(C)C)=O)CN(C(c2ccc(Cl)cc2)=O)CC12CCCC2 CC1(C(N2CCC(NC(C3CCCO3)=O)CC2)=O)CCCCCCC1 O=C(C1=CC2(CCOC2)C1)N1CC2CC1CN2C(c1ccc2ncccn12)=O N1(C(C(c2cn(C)nc2)=O)=O)CC2(C)CC1(C(=O)NCC1CC3C=CC1O3)C2 C(C)(N=c1[nH]c(=NCCC(C)c2cn[nH]c2)[nH]c2ccsc12)c1ncc(C)s1 c1(N(C)Cc2c(C)occ2)nc(N2CCC(O)CC(C)C2)c2c(n1)CCCCC2 C1(CC=C)(NC(C2C3COCC23)=O)CCCN(C(C2CC(=C3CC3)C2)=O)C1 C1(CC=C)(NC(C2(C)C=CCN2C(C2CN(C)C2)=O)=O)CCCCC1 C1(CNC(C(N2CCSCC2)C)=O)CN(C)CCN1C(C1CC2(C1)CC(F)C2)=O C#CCCCC(=O)NCC(C(=O)NCCCc1c[nH]nc1C)N(C)C Cc1ccnc(C)c1C(=O)NCCN(C(=O)C1=CCOC1)C(C)C C1(NC(c2ncc(C)c(Cl)c2)=O)C(C)CCN(C(=O)C(C)NC(=O)C2CC2)C1C C1(C)(NC(c2cc(C(C)C)sn2)=O)CCCN(C(c2cnc(Cl)[nH]2)=O)C1 c1(C(N2CCC(CN(C)C(C3(F)CC3)=O)C2)=O)c(F)ccc(Cl)c1F C=CC(CCC)CC(=O)NCCCC1CCCN1C(=O)C(=O)N=S(C)(C)=O C(N=c1[nH]c(=NCCC2CCCS2(=O)=O)[nH]c2c1SCC2)C1(CO)CC1.CCC(F)(F)F c1(C(N2CCC3CN(C(CCC(C)SC)=O)CC32)=O)ccc2nc(C)[nH]c2c1 S(=O)(=O)(c1c[nH]ccc1=NC1CCC2(CCC2)C1)NCCC1(C)CC1(Cl)Cl CC1CCC(CNC(=O)Cn2ncccc2=O)N(C(c2csc(S)n2)=O)C1 C(C(O)(C(=O)N1CCCC(CNC(C2(C(F)(F)F)CC2)=O)C1)C(F)(F)F)N(C)C N1(C(C(C(COC)C)C)=O)CC2CCCC(NC(c3ncccc3N)=O)C2C1 c1(N(CCN(c2ccccc2)C(c2nnnn2CC(=O)NC)C)C)sncc1Br C1(C(=O)NCC(=O)NCC)CCC(O)CN1C(c1ccoc1C)=O c1(C(=O)NCC2(C)CCC(NC(=O)C=C(Cl)Cl)C2)nccc2ccccc12 C1(C(=O)NCCCCC2CN(c3cc(C(=O)OC)ncn3)C2)CCCNS1(=O)=O CC1(C)CC2(CC2C(=O)NCC2C3CN(C(=O)C=Cc4ccc[nH]4)CC23)C1 c1(C(N2C(C3(NC(c4c(C)cno4)=O)CC3)CCC2)=O)sc2cncn2c1C N1(c2cc(C)ncn2)CCCC(C)(C(=O)NC(C(=O)O)C(C)O)C1 C1(NC(C(CC)C2CCC2)=O)CC2(C1)CC(NC(C1OCC3CCCC13)=O)C2 N1(C(CCC(C)OC)=O)CC2(C(=O)NCC=CCl)CC1CCO2 n1(CC)nc(CNC(C2(NC(=O)CCCC3CC3C)CCCC2C)=O)c(C)n1 C#Cc1ccnc(NC(=O)NCC2COC(C)(C)CO2)c1 C1(C(N(C)Cc2ccc(OC(F)F)cc2)=O)CNCC12CCOCC2 C=C(Cl)CCC(=O)NCC1CN(C(c2csc(Br)c2)=O)CC1O CC1C(NC(=O)CC2CCCOC2)CCN1C(=O)CCc1ccc(N(C)C)cc1 C(CC(=O)NC(c1ccoc1)C)(C(C)C)NC(C(=O)NC(C)C)=O N1(c2n(CC)c(-c3cccc(OC(C)C)c3)nn2)CCCC(C)(CCOC)C1 C(c1ccnn1C)=CC(=O)N(C(C)CNC(=O)CN1CCOC1=O)CC C1(C(=O)NCCCCCC)(CC)CCCN(C(c2cccc(C)n2)=O)C1 CN1CCN(CCC(=O)NC2CCN(C(=O)CC3(O)CCCOC3)C2)CC1 C1(C(C)C)CN(C(=O)COc2ccc(F)cn2)CCC1NC(c1nonc1N)=O C(C)(C)(CCC(=O)N(CCCCCC(=O)Nc1cnccc1C)C)OC c1(OCC)ccc(-c2cnc(NC(c3ccc(C)c(O)c3)=O)s2)c(Cl)c1OC N1(C(C(N2CCOCC2)C)=O)CCC2(CC1)CN(C(C1CCC(C#N)CC1)=O)C2 c1(C(=O)NCCCCCNC(c2ncn(CC)c2)=O)nccnc1OC c1(C(N2CC(N(C(C=C(C)C)=O)C)C2)=O)cccc(N2CCOC2=O)c1 c1(OCCC#C)ccc(C(=O)NCC2CCC(NC(=O)C(COC)OC)C2)cc1 C1(C(=O)NC2(CO)CC2c2cccc(Br)c2)CCCC2(CNC2)O1 N1(C(C2C(OCC)C2C)=O)CCC(C)C(CNC(=O)C(C)O)C1 C12(CN(C3CC(C(N4CCCCC4C(C)N)=O)C3)CC)CNCC1COC2 c1(C(C(=O)NCC(CCOC)NC(=O)Cc2cccc(C)c2)C)cc(C)oc1C CC1CN2CC3(CCN(C3)C(=O)CSCC2=O)O1.c1(CNC(N)=O)csc(=N)[nH]1 c1(C(N(CCN(C(Cc2cc(C)sc2C)=O)C)C)=O)cncc(F)c1Cl N1(C(C(CCC)OC)=O)CCN(C(c2sc(=N)[nH]c2C)=O)C(C2CC2)C1 Cc1ccc(N)c(C(=O)NCCOC2CN(C(c3cccc(C(F)F)n3)=O)C2)c1 c1(C2(C(c3ccc(Cl)cc3)C(=O)NC)CCC2)ccc(C(=O)OC)c(F)c1 N1(C(CC(=O)NCC)=O)CCCC(C2CCN(c3snc(Cl)c3C#N)CC2)C1 c1(C(N(C2CCCC(NC(c3ccc(SC)o3)=O)C2)C)=O)cncc2sccc12 C1(C(=O)NCC2CC(N(C)C)C2)CN(C(=O)C(C)(O)C2CC2)CC12CC2 N1(C(C(CNC(C(CC)CN(C)C)=O)O)=O)CCC2(CCC(OC)C2)C1 C(=O)(C(F)(F)C1=CCOCC1)NC1C=CCN(C(c2cncc([N+](=O)[O-])c2)=O)C1 CCC(C)CC(=O)C(=O)NC12CC(C(N3CCSC(C)(C)C3)=O)(C1)C2 C1(NC(c2c(CC)cc[nH]2)=O)CS(=O)(=O)CC1NC(c1cccc(F)c1F)=O N1(Cc2cn(CCCC(=O)OC)nn2)CCN(C(=O)C(C)O)C1=O Cn1c(C(=O)NC2CCN(C(C3CCNC(=O)C3)=O)C2)cc2ccccc12 Cc1cc(C2CC2NC(=O)NCc2cc(C3CC3)no2)no1 c1(C(C)=O)ncc(Br)cc1NC(=O)CC1CCCN1C(c1cc(C)nn1C)=O N1(C(C2C(CCC)C2)=O)CCC2C(C1)CN2C(=O)CCC(CC)CC C(=O)(C1Cc2ccc(Cl)cc21)NC(C1CN(C(c2c(C)ccc(OC)c2)=O)C1)C N1(C(CCC=C)=O)CCCCC1C(=O)NCC1CNC(=O)C1 Cc1cc(C(N2CCC(c3ccccc3)(NC(=O)C(F)C3CC3)C2)=O)ncn1 c1(CNC(C(=O)N(CCCN(C)C)CCN)=O)ccc(N2CCN(C)CC2)nc1 C1(C(=O)OC(c2cc(Br)ccc2F)C(=O)OC)CC2(CCCCN2)C1 C(=O)(CCCS(C)(=O)=O)NC1C(C)(C)N(C(C2CCCC3(CC3)C2)=O)CC1 c1(C(=O)NCC2N(C(CSc3nc(C)[nH]n3)=O)CC=C2)cc(F)ccc1Br CCC(C)C(C(=O)N1CCC(CCc2nn[nH]n2)CC1)c1ccccc1 C1(C(N2CC(O)(CC(C)C)C2)=O)(CC)CN(C(=O)C(n2ccnc2C)C)C1 C1(C(N(CC=C)CC2CC2)=O)CC2(CCC2)CN1C(=O)C(CC=C)C(C)C N1(C(c2c(CSCC)cccc2)=O)CC2CN(Cc3[nH]c(C)cc3C)CC2C1 c1(OC)ncc(C(=O)OCc2cc(N)ccn2)cc1C1CC1 c1(CC)nn(C)c(Cl)c1C(=O)NC(C)CNC(=O)CCc1cccnc1F S(=O)(=O)(c1c[nH]c(C(=O)NC2CC(NC(C3CCC4C3C4(F)F)=O)C2)c1)N(C)C c1(C(=O)NC2C(C)(C)CCN(C(CSC)=O)C2)cc2n(n1)CC(C)NC2=O c1(C(=O)NC(CCC)C(=O)O)ccc(C)c(O)c1O c1(CCC(N2C(c3cn(C(C(=O)OCC)C)nn3)CC2)=O)ccc(Br)c(C)c1 Cc1ccc(C(N2CCC3CN(C(C4CC(=O)NC4(C)C)=O)C3C2)=O)c(F)c1F n1(CCC(=O)N(CC(CC)NC(CCCOCC=C)=O)CC)ccc(O)nc1=O c1(C(=O)NC2CC(C)N(C(c3ccc(=N)[nH]n3)=O)C2)ncc(C2CC2)cc1F N1(C(c2cnc(C)[nH]2)=O)CC2CC(NC(C3NC(=O)CC3C)=O)CC1C2 C12CC(F)CN1CC(=O)NC2.c1(CC)ccsc1C(=O)N(C1CCOCC1)C c1(NC(CC2CCC(Cc3n(C)cnn3)C2)=O)cncnc1Br C1(C(N2CCC(NC(c3nc(CC)oc3)=O)C(CC)C2)=O)CCc2ccnn2C1 Cc1cnc(N(C2CCCCC2)C2CCCCC2)s1 CC1CCN(C(=O)CNC(N2CCCCC2)=O)C1c1cn(N2CCN(C)CC2)nn1 N1(C(C2C=C(C)CS2)=O)CC2(CNC(C3CCC(C)(C)O3)=O)CC1CO2 c1(C(C(=O)OC(C2(C)C(CC)C2)=O)OC)c(F)cccc1F C(C)(CCC(=O)NCC1COCCN1C(=O)CCNC(c1ccsc1)=O)OC [N-]=[N+]=NCCCCCCNC(C1CCC=CC1NC(c1cc(CO)[nH]n1)=O)=O c1(OC)c(CN2CCC2C(=O)NCCCn2cccn2)cccc1Cl c1(CNC(=O)NCC2CCN(C(=O)OC)C2)cn(C)c2ccccc2c1=O CN1CCCC(CC(=O)NCC2=CCN(C(=O)C=Cc3ccncn3)CC2)C1=O c1(C(N2CC(O)(C(C)NC(CSCCOC)=O)C2)=O)cccc(F)c1C1CC1 CN1CC(=O)N(CC(=O)NCCC2CN(C(c3cc(F)cs3)=O)CCO2)C1=O c1(CC)onc(C(N2CCC(O)(CNC(c3ccc(CC4CC4)s3)=O)C2)=O)c1C C12(CNC(c3c(C)nc[nH]3)=O)CCCC1CCN2C(C1CCc2nn[nH]c2C1)=O c1(OC)ccc2c(C)c(C(=O)NCC(C)NC(c3coc(C(F)F)n3)=O)[nH]c2c1 C(=O)(C1=C(SC)CCCC1)N(CCCNC(=O)CC12CCCCC1C2(F)F)CC c1(OCC)oc(C)nc1C(=O)N(CCC(C)NC(c1cccnc1)=O)C N12CC3C(C3C1)N(C)C(=O)COC(C)C2=O.c1(OCC)ccccc1OC C1(C)(C(=O)NC(CC)CNC(c2ccnc(CO)c2)=O)CCCC1(F)F c1(-n2cc(Cn3c(C)ncc3)nn2)cccc(CCNC(=O)C(C)CC#N)c1 C1(C(=O)CC2C(C(N(C3CCN(C4CC4)C3)C)=O)CCC2)CCOC1(C)C C(=O)(C1=CC2CCCCCC12)N1C(CCNC(=O)CCc2ncc[nH]2)CCCC1 c1(C(N(C(C)CCNC(C2CC3(CC3)C2)=O)C)=O)ccc2c(c1)CCCC(=O)N2 c1(C(CNC(C2(C)C(C(=O)OCC)CC2)=O)(C)C)ccc(C(F)(F)F)cc1 C1(NC(c2c(C)nc(CC(C)C)o2)=O)CC2CC1N(C(c1ncc[nH]c1=O)=O)C2 N1(C(c2c(OC)c(C)sc2)=O)CC2CC(NC(=O)CC3CCCO3)C1C2 C1(C(C(=O)NC(c2cn(Cc3cnco3)nn2)C)O)CCCCCC1 C1(NC(C(CC)CC2CCCCC2)=O)CC2(CCN(C(=O)Cc3cnsc3)C2)C1 C1(CC=C)(C(=O)NCCC(=O)NCC)CCN(C(=O)CC2CCCC2)C1 c1(C(N2CCC(N(C(CCCCC#C)=O)C)C2)=O)cccc2occ(Br)c12 C(=O)(C(C)CC(=C)C)NCC(CN(C(Cc1n(CC#C)cnn1)=O)C)O c1(C(=O)NC(CNC(c2[nH]cc(C(C)=O)c2)=O)(C)C)cnc(C(F)F)nc1 C1(C(N(CCCNC(c2ccnc(Br)c2N)=O)C)=O)CCC2CCC(=O)N12 c1(C(=O)NCCN(C(=O)CC2CCCCN2C)CC)ccc2c(c1)CCC(C)N2 c1(C(=O)OC)cc(CNCC(C)CC(N2CC(NC(C)=O)C(O)C2)=O)oc1C CC1CCCN(C(=O)CCc2cnc[nH]2)C1CNC(C1CCCS1)=O C#CCCCCCCC(=O)N(CCC(=O)N(C)CC1(O)CCC(C)CC1)OC N1(C(c2c(C)n(C)c(C3CC3)c2)=O)CC2=C(C1)CN(C(C1C=CCCC1)=O)C2 c1(C(=O)NC2CN(C(Cc3cc(C)no3)=O)CC(O)C2)ccc([N+](=O)[O-])nc1 CN1CCC2CN(C(c3ccc(-c4cnn(C)c4)s3)C(=O)NCCSC)CCC12 C1(C(=O)NC(CC)C(=O)NC)(C(C)C)CCN(C(c2nnccc2C)=O)C1 C1(C(N2CCC(CC=C)C2)=O)CCCCC1CNC(=O)CCCC=C C1(CC(=O)NCC2C(C)CC2)CCC(NC(C2CCC2C(C)(C)C)=O)C1 c1(-c2cn(C3(C)CN(C(=O)C(F)(F)C(F)F)CC3O)nn2)ccc(C#N)c(F)c1 C1(NC(C(C)OCCOCC)=O)CC2C(NC(=O)C(C)(C)Cl)C2C1 Cc1cccc(C)c1C(=O)N(CC(O)CNC(C1COC(=O)O1)=O)C C1(CC(=O)NCCCNC(C(c2cccc(OC)c2)OC)=O)CC(C)(C)CCO1 CC1(C2(C(=O)NC3C=CC(C(=O)NCCCc4cccnc4)C3)CC2)CC1 C1(C(=O)NC(CNC(C2(C=C)CCC2)=O)CC(C)C)CCc2nnnn2CC1 c1(CC)n[nH]c(CC)c1CC(=O)NC(CNC(C1COCCO1)=O)C(C)C O=C1CC2C(CCCN2C(C2(CF)CCN(C(c3ccc([N+](=O)[O-])o3)=O)C2)=O)N1 N1(C(CNC(=O)OCC)=O)CCCN(C(c2c(F)cccc2Br)=O)C(C)C1 c1(C(N2CCOCC2CC2CC2)=O)ccccc1-n1cc(CN2CCCC2)nn1 CC1CCN(C(c2cccnn2)=O)C1C(=O)NCC1(C2CC2)CC1 C(=O)(CCCS(N)(=O)=O)NCC1C(C)CCN1C(=O)C=Cc1scnc1C C1(NC(c2c(N)cc(Cl)cc2F)=O)CN(C(=O)C=CC2CC2)C2(CCCC2)C1 CC(O)C(C)C(=O)NCC1(CNC(c2ncnn2C2CCOCC2)=O)CCC1 O=S(=O)(c1cccc(=NC2CCOC2)[nH]1)N1CCC(c2ccc(Cl)cc2)CC1 C(=O)(C(N)CC(=O)Nc1nnc(C)o1)OC.N12CCC(CC1)C2 N1(C(c2ccc(C(=O)NC)cc2)=O)CC2CN(C(C3CC(O)C3)=O)CC2C1 Cc1nc(C(N2CCC(C(=O)NC(C)CN(C)C(C)C)(C(C)C)C2)=O)cn1C c1(C(=O)NC(C(C(C)C)C)CNC(=O)C=CCO)cc2ccccc2c(=O)n1C C(=O)(C(F)(F)C(C)O)N1CC(C(NOCC(=O)OCC)=O)C(C)C1 c1(N(CC(=O)NCCOC2CN(C(C=CCCC)=O)C2)C)nnc(C)n1C c1(CC(=O)NCC(CCOC)NC(C2(CCC)CC(=O)C2)=O)ccc(OC)cn1 C12(CNC(c3c(C#N)cn[nH]3)=O)CCC(NC(C3CN4CCN3CC4)=O)(CC1)CO2 c1(C(N2CCC(C(N)=O)CC2)C(=O)NC(C(=O)OC)C)cc(Br)nn1COC C1(C(N2C(CCNC(C3CN4CCC3CC4)=O)CCC2)=O)CCCCC1C1CC1 C1(NC(CC2(C=C)CC2)=O)CN(C(c2c(C)cccc2Br)=O)CC12CCC2 C1(C(=O)NC2CC(=O)N(C)C2=O)CCN(C(=O)CC2NC(=O)NC2=O)C12CCC2 C12CCN(CCC1(F)F)C2.c1(-c2cn(C3C(SC)CCC3)nn2)sc(C)nc1C c1(CC(=O)NC2(CNC(C(C(=O)NC)(C)C)=O)CCCC2)cnn2ccccc12 Cc1cccc(C)c1CNC(=O)CC(C(C)C)NC(C1(C)CC1(F)F)=O N1(C(C(C)C(C)(C)C)=O)CCCC12CCN(C(=O)C=CC1CCCC1)C2 c1(C(N2CCN(C(COCCCCCCCC)=O)CC2)=O)ccc(Cl)c(Br)c1F N1(C(CC)=O)CC2CCC(C1)CC2NCc1cccc(C(=O)O)n1 c1(OC)ccc(C(=O)NC2CCN(Cc3ccc(C)nc3F)CC2F)c(C)c1C C(C#Cc1ccccc1)NC(=O)CC1CCCC(=O)N1.C12CCN(C1)CC(=O)N2 CC1(C(=O)Nc2nc(C(N3CCCN(CCO)CC3)=O)co2)CCC2CC2C1 CC(C)C(C)CC(=O)NC1CCN(C(C2CC=CC(O)C2)=O)CC1CO Cc1nn(CC(N2CC(NC(c3nc(Cl)oc3C)=O)C2)=O)c(C)c1Br c1(O)ccc(F)cc1.N1(CC(=O)NC2(C)CN(C(CCOC)=O)C2)CCN(C)CC1 Cn1nc(C(N2CC3CC3(CNC(C3(O)CC3(C)C)=O)C2)=O)cc1Cl c1(-n2c(C(C3CC34CCC4)NCc3ccc(SC)s3)nnn2)ccc(F)cc1 C1(C(=O)NC(C2CCCC2)CC2CCCCC2)CC12CCC2 CCC(CC)CCC(=O)NCC1(NC(=O)C(n2cc(C)cn2)C)CC(OC)C1 c1(CC(C)C)ccc(COCC(=O)NCCNC(C2(N(C)C)CC=CC2)=O)cc1 C1(=CC(=O)NCC(Cc2ccccc2)NC(=O)CC2CC=CC2)CN2CCC1CC2 CC1CCC(CCNC(C2(NC(=O)CN3CC(C)(C)C3)CCCC2)=O)C1 c1(C(C(=O)NC2C(C)CN(C(=O)Cc3cnc[nH]3)C2)=O)ccc(F)c(F)c1 N1(C(Cc2ccc(C)s2)=O)CCC2(CC1)CC(NC(=O)C(Cl)(Cl)Cl)CO2 N1(C(C)=O)CCc2cc(CNC(c3cc4[nH]c(C)cc(=O)n4n3)=O)ccc2C1 C=CC(CC)CC(=O)N(CC(O)CN(C)C(c1cccc(OC)c1)=O)C C(=O)(CCCC(C)(C)C)NCC1CN(C(COCCC#C)=O)CC(C)C1 C#CC(CNC(C1(N(C(=O)C=C(C)C(C)C)C)CC1)=O)CC C(=O)(C1=CCS(=O)(=O)C1)N1CC(CCCCNC(CC(COC(C)=O)(C)C)=O)C1 CC1CC(CNC(C2CNC(=O)N2)=O)CN1C(c1cccnc1F)=O C1(NC(C=C(C)Cl)=O)CCN(C)C12CCCN(C(C1(C(F)(F)F)CC(O)C1)=O)C2 CCCC(C(=O)N(CCNC(c1ccnc(F)c1Cl)=O)CC)C(C)C Cc1cccc2cc(C(N3CC4CC(C3)C4NC(=O)CC(C)C)=O)oc12 Cc1cc(SC2CCCC2)ccc1NC(c1csc(F)c1)=O n1(CC)nnnc1C(c1cccn1C)NCC1(CO)CCCO1 C(=O)(CCN(OC)C(=O)c1ccsc1C)NCCn1ncc(CC)c1 C(=O)(C(N)C(=O)NCCCOc1ccncc1)OC c1(CN(CC(C)C#N)Cc2cc(F)ccc2F)cc2n(n1)CCCO2 c1(C(=O)NC2C(CNC(CC(C=C)C)=O)C2)cnn2c(N)cc(C)nc12 C1(CC)OCCC1C(N1CC(c2ccccc2)(NC(=O)Cc2c[nH]nc2C)C1)=O N1(C(c2nc(C)[nH]n2)NCC(C)(C)CO)CCN(C(=O)OC(C)(C)C)CC1=O N1(C(C2CCCN2CC(F)(F)F)=O)CCN(c2ccc(I)cn2)CC1 CC1c2ccccc2OC1CC(=O)NCCCCNC(C1CCC2(CCC2)O1)=O N1(C(C2C(C)(C)CC2)=O)CC2(CCC(CNC(c3ccnc(C4CC4)c3)=O)O2)C1 C1(C(C)NC(C2CC(N3CCCC3)C2)=O)CCN(C(=O)C=CC2CC2)C1 c1(C(=O)N(CCNC(C23CCC2CC3)=O)C2CC2)cc(Cl)c(Br)s1 N1(CC(=O)NC(CCN(C(C(C)SC(F)(F)F)=O)C)(C)C)CCN(C)CC1 N1(C(Cc2n(C)ccc2)=O)CC(F)CC1C(=O)NCc1ccc(C2CC2)cc1 c1(C(=O)NC(CNC(c2c(OC)cc(C)s2)=O)(C)CO)n[nH]c2cc(C)ccc12 CC1C(C)S(=O)(=O)CCN1CCCCc1cn(C2CCN(C3CNC3)C2=O)nn1 N1(C(c2ccc(OC)cc2O)=O)CC(C(=O)NCCCCCCO)CC(F)(F)C1 C(CCNC(=O)Cc1cn[nH]c1)(C(C)C)NC(C(C)NC(COC)=O)=O C1(C(=O)NCC2(F)CCCN(C(=O)CN3CC4CC4C3)C2)CCCCC12CCC2 C1(C(=O)NC2CCN(C(C3CC(OC4CC4)C3)=O)CC2)CC2COCC(C1)C2 N1(C(=O)CCc2cn[nH]c2)CC2CCN(C(c3cc(Cl)no3)=O)CCC2C1 CCC(CCOC)N=c1nc2c(ncn2C)c(NCc2cc(Br)no2)[nH]1 N1(C(CCC)=O)CC(O)(CNC(C2(N3CCCC3)CC2)=O)C1 N1(C(C=C(C)c2ccsc2)=O)CCN(C(=O)C(c2ccc(F)cc2)=O)CC1CO CC(CCC(=O)N1CC(CNC(=O)Cc2cc[nH]n2)C(C)C1)S(C)(=O)=O c1(C(=O)NCC2CC(OC)CN2C(=O)C2=CCCC2)c[nH]c2ncccc12 C1(NC(C2CC(=C)C2)=O)CCC2CC1CN2C(C1CC(F)(F)C1)=O Cc1cc(C(=O)N(C)CC2CCC(NC(=O)C(C)OC(C)C)CC2)c(O)cc1F CC1CCC(NC(c2ccnc(OCCO)c2)=O)CN1C(c1c[nH]ccc1=N)=O c1(C(C)=O)ccc(S(=O)(=O)NCc2cc3ccccc3n2C)c(C)c1 C1(NC(C(=O)Nc2c(C)nn(CC(F)(F)F)c2)=O)C2CCCCCC12 N1(C(C(CC)C#N)=O)CCC(CNC(c2oc(C)nc2C(F)(F)F)=O)C12CC2 c1(C(=O)NC2C(CC)N(C(=O)C(c3cncnc3)C)CC2)ncc(Br)cc1C CCC(C)C(O)C(C)C(=O)NCC1(C(=O)NCCCC(C)CO)CCCO1 c1(C(=O)NC2(C(=O)NCCC(CC)O)CC2)ccc(O)cc1 N1(C(C2(CC)CC(F)(F)C2)=O)CC2CN(C(=O)C(C#N)CC)CC(F)(F)C2C1 c1(C(=O)NCC=C(C(=O)NC(C2CCOC2)CC)C)cnn(C)c1C#N C1(COC)(CNC(c2cccc(C)n2)=O)CCCN1C(c1csc(O)n1)=O C(=O)(C(C(C)(C)O)NC(C1CCC(C2CC2)C1)=O)NCC(N1CCCC1)C C1(C(N2CCC(OCCNC(c3cc(Cl)ccc3F)=O)C2)=O)CN2CCC1CC2 Cn1nnc(CNC(C2(C)CCOC2)=O)c1C(=O)NCc1ncco1 c1(C(N2CC(C)C(NC(=O)CCC3CCCC3)C2)=O)cc(=O)cc(Cl)[nH]1 C1(C2(O)CCOCC2)(C(=O)NCCN(C(c2cccc(CC)n2)=O)C)CC1 c1(CC)nnc(N2CCC(NC(c3cc4c(s3)CCC4)=O)C(O)C2)nc1CC CCC(CC(C)C)C(=O)N1CCC(NC(c2ccc(Cl)c(O)c2)=O)C1 Cn1cnc2nc(N3CCC(OC(F)F)CC3)nc(NCc3cc(Br)cs3)c12 c1(N(C)C)ccc(C(=O)NC2CNC3CC23)cc1Cl CCC(CC(C)C)C(=O)NCC(C)(C(C)C)NC(=O)CCc1cc(C)no1 Cc1ncc(C=CC(N2CCCC(CNC(=O)COC3(C)CCCCC3)C2)=O)s1 CC(=O)C(C)CC(C)C(=O)N1CC(C)C1C(=O)NCCc1cncs1 Cc1cn2nc(C(=O)N(C(C)CCNC(=O)C(O)CC(C)C)C)cc(C)c2n1 C1(C(N2CCCC2c2ccc(Cl)cc2)=O)CCC2CCC(=O)N12 N1(C(CONC(C(=O)NCC)=O)=O)CC(C)N(C)C(C)C1 N1(C(CCCOC(C)C)=O)CCN(C(C2CCOC2)=O)C2CCC12 Cc1ccc(C(N2CCCC(C(C)NC(C3(c4ncco4)CC3)=O)C2)=O)cc1C C1(NC(C2(C=C)CC2)=O)CCN(C(C2CCC(COC)C2)=O)CC1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCCN(C(=O)CCC2C(=O)NN=C2C)C(C)C1 Cc1cc(NC2CC2)ccc1C(N1CCCC1(C)CNC(=O)C(C)S(C)(=O)=O)=O C1(C(=O)NC2(C)CCC(C)(C)C2)CCN(C(=O)CCC(F)(F)F)CC1(C)C C1(CC(=O)NC)CN(C(c2cnco2)=O)CCN1C(=O)Cc1cncnc1 C=CCC(CC=C)C(=O)NCCC1CN(C(=O)C=C(C)Cl)CC1C N1(C(c2nn(C)c(Cl)c2)=O)CC2CCC(NC(=O)CCOCC(F)F)(C2)C1 N1(CCC)CCCN(C(c2n[nH]cc2Br)C(=O)NCC(C)C)CC1=O C12CC(C1(C)C)CCC(=O)N2.CCC(CC)N(CCC(=O)NC1CC(CO)C1)C c1(N2CCC(COC)(NC(c3cnc(OC)cc3C)=O)C2)cc(C)nc(CO)n1 C1(C(=O)NCCC(C)N(C(C2CCC(C)O2)=O)C)CC2CCC1CC2 C(C(C(C)(C)C)NC(=O)Cc1ccc(C(N)=O)cc1)NC(C1C(OC(C)C)C1)=O CCCCC(C(=O)N1CCCN(CCNC(=O)C(O)C(F)(F)F)CC1)C(C)C Cc1cnc(C(=O)NCCCN(C(=O)C(C)(C)N(S(C)(=O)=O)C)CCO)c(F)c1 C1(C(=O)NCc2c(C)cc(C)s2)CN(C(=O)CCOCCN(C)C)CCC1(C)C C(C(=O)NC1(c2nn[nH]n2)CC1)(c1ccoc1)NC(C1CSC1)=O N1(C(c2cc(C)[nH]c2)=O)CCC(CNC(=O)CC2(O)CCCCCC2)C(O)C1 c1(C(=O)NC)ccc(C(=O)N(C2CCCN(C(C3CC3C(N)=O)=O)C2)C)cc1 C1(C2CCN(C)CC2)(C(N2C(CNC(C3CC(C)NC(=O)C3)=O)CC2)=O)CC1 CCCCC(CNC(c1sc(C)cc1C)=O)NC(=O)C(F)n1ccnc1 c1(C(C2CC2)NC2CN(CCc3ccccc3)CC2O)cccnc1SC(F)(F)F N1(C(CCc2ccc(C)o2)=O)CC2CCCC2(C(N2CC(c3ccon3)C2)=O)C1 CC1(C)CN(CCF)CCN1C(c1cnc(-c2ccc(CO)o2)cn1)=O CC1(C(N2CCOCC2CNC(c2cnc(CC(C)(C)C)o2)=O)=O)CC(F)(F)C1 N1(C(c2ccc(OC)o2)=O)CC(NC(=O)CCc2conc2C)C(C2CC2)C1 c1(C(=O)NC2CN(C(C(CC)C)=O)C(C)C2)ccc(F)c2occc12 C1(CN(C(C(OCC)OCC)=O)C2CC2)(NC(=O)C#CC(C)C)CCC(C)(C)C1 C(=O)(C1CC(=O)c2c(F)cccc21)Nc1c(C)ccc(NC(C)=O)c1 Cc1cccc2c1OC(C(=O)OC1CCCC3(CCCC3)C1)C2 c1(N(CC(C(C)C)O)C)ncc(S(=O)(=O)N2CCC(CO)C(F)(F)C2)cc1Cl c1(C(N2CCCCC(NC(C(C)=CC3CC3)=O)C2)=O)cc(O)nc2ncccc12 CC1(C)CC2(CC2C(=O)NCC(c2ccccc2F)NC(c2coc(Cl)c2)=O)C1 C#Cc1cc(F)c(C(=O)NC(CNC(c2nccc(C(F)F)n2)=O)CO)cc1F Cc1cnccc1C(=O)NCC1CCN1C(=O)CCc1cncc(Br)c1 C12(CNC(=O)C(=O)NCCC3CCCCO3)CC3CC(C1)CC(Cl)(C3)C2 C(Cn1ccnn1)(C(F)(F)F)N(C=O)Cc1cc(-n2cccn2)ccn1 N1(CCC)CCC(NC(=O)NCC(c2ccc(F)cc2)N(C)C)CC1 N1(c2ccc(S(=O)(=O)N(CCCCN(C)C)C)cn2)CCN2C(CNS2(=O)=O)C1 C1(NC(=O)NC(CC)Cc2ccccc2C)CC2CCC(C1)S2(=O)=O c1(C(N2CCC(N(C(=O)Cn3ccnn3)CC)C2)=O)cc(Cl)ncc1NC C=CCCCC(C)(C)C(=O)NCC(O)C(=O)Nc1cn(C)nc1C(N)=O C1(CC=C)(NC(c2ccn(C)c2)=O)CCN(C(=O)C=Cc2cnc[nH]2)C1 C(=O)(C(C)S(N)(=O)=O)N1CC(N(C(Cc2cn(CC)nc2)=O)CCO)C(O)C1 C(=O)(CC(C)CC(C)(C)C)N(CCC(C)NC(Cn1nc(C)oc1=O)=O)C C1(CC)CCN(C(c2ccc(NC)cn2)=O)C1C(=O)NC1(c2n[nH]c(C)n2)CC1 c1(CC)c(N2CC(N(C(=O)OC(C)(C)C)CC)C3(CCSC3)C2)nc(=N)[nH]c1C n1(CCC)nc(C)cc1C(=O)NC1CCCCC1NC(=O)C=CBr c1(C(N(C(CNC(c2c(C)oc(CO)c2)=O)C)C)=O)cc(C(F)(F)F)ncc1Cl Cc1ccc2c(c1)CC(C(=O)NCC1CC(NC(=O)CCCCCO)C1)O2 c1(C(=O)NC2C3CN(C(c4c(SC)nccn4)=O)C2C3)cc2ncccn2n1 C1(NC(C(C)=C2CCC2)=O)CC(C)CN(C(c2ccc(CO)o2)=O)C1 n1(CC)nc(C)cc1C(=O)NCC(C1CC1)N(C)C.C1(C)CC1C(=O)N C1(NC(C(C)N(CC=C)C)=O)CC(Oc2ccccc2)C1(C)C O=C1CCOC(C(=O)NC(C(=O)NCC2(CO)CC=CC2)C2CC2)C1 c1(C(=O)NCCOCC)cnc(OCCC(C)OC)nc1 C(c1ccc2occc2c1)=CC(=O)NC1CC(C)(NC(c2cnc[nH]2)=O)C1 N1(C(CC(CC)SC)=O)CCC2CN(C(c3nc4c(s3)COCC4)=O)CC12 C1(CC)C(NC(=O)C(O)CCSC)CCCN1C(C1CC(=O)NC(C)C1)=O Cc1nc(CNC(c2c[nH]c(C#N)c2)=O)oc1C(N1CCCC(CC(N)=O)C1)=O N1(C(Cn2c(C)ccn2)=O)CC2CCN(C(C3C=CC=CC=C3)=O)C(C2)C1 N1(C(C2CN(C(CC(COC)(C)C)=O)CC2(F)F)=O)CCOCC(C2CC2)C1 CC(CN=c1ccn2nccc2[nH]1)N(C)C(c1coc(C(F)F)c1)=O C(=O)(CC(C)(C)NC(=O)CCCC1CC1)N(C(C)CC(N)=O)C C(=O)(C1=CC(O)C(NC(=O)C(C(C)(C)C)OC)C1)NC(C(CC)(C)C)C N1(C(c2c(C)scn2)=O)CC2CC1C2C(N1CCC(c2ccccn2)C1)=O Cc1cccc2c1OC(C(=O)NC13CCC(C1)N(C(=O)COCCN(C)C)C3)C2 CC(C(=O)N1CCC(NC(=O)CN2CC3CC3C2)C1(C)C)C(F)(F)F CCCCC(C(=O)NCCN(C(=O)CCN(CC)CC)C1CC1)C(C)C N1(C(c2cc(COC)sc2)=O)CCC(NC(=O)CC2CCCN2C(C)=O)CC1 CC(CC(=O)NCC(CNC(c1cc(C2CCC2)on1)=O)CO)n1cccn1 C1(C)(NC(CCN(C(CCc2n(C)ncc2)=O)CC2CC2)=O)CN2CCC1CC2 N1(C(COc2cccc(CC)c2)=O)CCN(C(C2Cc3cscc3C2)=O)C(C)C1 c1(C(=O)NC2C(CNC(C(C)SC)=O)CC2)cnc2ccoc2c1 Cc1nc(F)cc(=NCCc2cccc(C(F)(F)F)n2)[nH]1 S(=O)(=O)(c1cc(C(=O)NCC2CN(C(C3(CC#C)CC3)=O)C2)ccc1OC)NC C1(C(=O)NC2C(CNC(=O)Cc3cnns3)CCC2)CCCC2CCCN12 C(=O)(C(CCCC=C)NC(c1ccc(F)cc1F)=O)N(CC#CC)C c1(CC(=O)NCC(C)CNC(=O)CCC2CCC(=O)N2)cnccc1C(F)(F)F C(=O)(CN=c1cc[nH]cc1)N1C2(C(=O)NC)CC(CO)(C1)C2 N1(C(c2cc(C)c(C)s2)=O)CCN(C(C2CN(C3CCC3)C2)=O)CC1CC1CC1 c1(CCC)ccc(N)c(C(=O)NCCCNC(=O)CCN(C)CCC)c1 c12cc(ccc1Cl)C(=O)O2.N1(CC)CCN(CC#C)C(CC#N)C1 Cc1ccnc(C)c1C(=O)NCc1ccccc1CNC(=O)C(=O)NC1CC1 C(=O)(C(C)CCCOC)NCC(CC)N(C(=O)C(C)Cc1ccncc1)C c1(C(=O)NCCC2N(C(c3c(C)cc(SC)s3)=O)CCC2)cnc(C)c(C)c1 c1(CCC(=O)NCC2CC(NC(C=CCC)=O)C2)nc(C)c(C)o1 c1(N(C(C)=O)CC=CC(N2CC(c3nc(=O)o[nH]3)C2)=O)nscc1N C12(C(=O)NC3CCC(C(=O)OC)C3)CCC(CC1NC(=O)C(C)CSC)C2 C(CNC(c1cnc(C2CC2)[nH]1)=O)(CCNC(C1CNC(=O)O1)=O)OC C1(F)(C(=O)NCc2ncc(C)s2)CCN(C(=O)C(C)CC2CCCC2)CC1 c1(C(=O)NC2CN(C(C=C(CC)CC)=O)CC(O)C2)cc2c(Cl)nccc2s1 c1(C(N2CCC(N3CCN(C(c4c(C)occ4)=O)CC3)C2)=O)cc(N)cc(O)n1 c1(CC(=O)NC2(C3CN(C(=O)C4=CCC4)C3)CC2)c(Br)ccc(F)c1F N1(C(C2C(C)C2)=O)CC2CCC1C(NC(c1ccc(-c3ccccc3Cl)o1)=O)C2 c1(C(F)(F)F)cc(N2CCCC(C3OCCO3)CC2)nc(F)c1 c1(C(CSCC(=O)N(C(=O)CC(F)(F)Cl)CCO)C2CC2)ccc(F)cc1F c1(OC)ccc(C(=O)N(C2CN(C(c3n[nH]cc3Cl)=O)CC2F)C)n2nccc12 C(=O)(C(C(C)C1CCC1)NC(c1cc(C(=O)C(C)C)c[nH]1)=O)OC N1(CC2C(=O)OC(C)(C)O2)C2CCC1CC(CCc1cc(F)ccc1F)C2 C1(C(N(CCOCC=C)C)=O)CCC(C)N1C(c1cnn(C(C)C)n1)=O CC1=C(C)CC(C(=O)NC2C(O)CC2O)CC1.C12CC(CC1O)C(=O)N2C1CC1 Cc1cc(NC(=O)CCc2csc(Br)c2)c(Br)cc1[N+](=O)[O-] C(CCC(C(=O)N1CC(C2CCCO2)C1)NC(c1cc(C)nc(C)n1)=O)OC Cc1cc(N2CCC(C3CCCC3)CC2)nc(=NCCC2CN(C)CCN2C)[nH]1 Cc1cc(N)c(F)c(C(=O)NCC2CC2CNC(=O)CCCC(=O)N(C)C)c1F C(=O)(C#CC1CCCCC1)N1C2C(NC(c3c(SC)nn(C)c3)=O)C(C2)C1 c1(N2CC(F)CC(C(=O)NCCSCC)C2)ncc2ccc(F)cc2n1 c1(C(=O)NCC2N(C(C(C3CCOCC3)OC)=O)CCC2)cnc2nccn2c1 c1(C(=O)NC2C(NC(Cc3nnc(C)o3)=O)COC2)nc(Cl)sc1Br CC1CCN(C(=O)C2=NNC(=O)C2)CC1NC(=O)CNC(c1ccc(F)cc1)=O C(=O)(C(F)Cc1ccccc1)NCC1C(NC(=O)CCC2CCC2)C1 C=C(CNC(c1ccn(C2CC2)n1)=O)CCNC(C1CCC2CC12)=O C(=O)(CC(C)(C)CC(F)F)N1CCC(CN(C(=O)Cn2nnc(=N)[nH]2)C)CC1 c1(C(=O)NCC(CNC(C2C(CC)CCO2)=O)(C)F)occ2c1CCC2 c1(CN2CCC(C(=O)NC(COC)CO)(OC)CC2)nc2cc(Cl)c(F)cc2[nH]1 Cc1cc(CC(N2CC(Cn3cc(CC4CCOCC4)nn3)C2)=O)cc(C)c1 c1(OCC)cccc(OC)c1NC(=O)COC1(Cc2ccc(Cl)cc2C)CCC1 CC(=NO)c1cc(C(=O)NC2(CO)CCCN(C(=O)C#CC3CC3)C2)cnc1O c1(C(N(C)CC2(CNC(=O)CCc3nc[nH]n3)CC2)=O)ccnc(N(C)C)c1 C1(NC(COCc2ccc(C)s2)=O)CCC(C)N(C(C2CCSC2)=O)C1 N1(C(c2ccc(C(C)C)nn2)=O)CCOC(C)(C)C1CO N(C(=NC)N1CCC(Oc2ccccc2OC)C1)CC(=O)N(C(C)C)CC C(=O)(C1=Cc2ccccc2C1)NCC1(C(=O)NC(CC)(CC)CC)CCC1 C12(CNC(CC(C=C)C)=O)CC(NC(C3OCCC3C)=O)(C1)C(C)(C)O2 N1(C(CCC(=C)Cl)=O)CCCCCC1CNC(C1(OC)CCS(=O)(=O)C1)=O c1(C(=O)NCC2C(CNC(C3C(C=C)C3)=O)C2)sc(=N)[nH]c1C C#CCCCC(=O)N(C)CCOCCNC(C1CC1C#C)=O n1(CCNC(=O)CCc2ccccc2)cnc2cccnc12 N1(C(C=CC(CC)=CC)=O)CCC2(CCCC2CNC(=O)C(C(C)O)NC)CC1 C(=O)(C(CN(C)C)C(C)C)NC(CC)C(=O)NCc1ncccc1F CCCCCCC(C)C(=O)N1CC(C(N)=O)(CNC(=O)C(C2CCCO2)C2CC2)C1 C1(NC(C2(OC)CCN(C(c3cscc3C)=O)C2)=O)CCCC1C1CC1 c1(C(N2CC(C(C)NC(=O)CCc3ccc(F)cc3)C2)=O)c(F)ccc(F)c1Cl CN1CCN(C(=O)Cc2ccc(Cl)cc2Cl)C(CNC(C2CC23CC3)=O)C1 C(=O)(C(C(F)(F)F)C(=O)OC(C)(C)C)N1CC(OC)(CNC(=O)CN(C)CCO)C1 C(CC[Si](C)(C)C)S(CC)(=O)=O.N12CCOCC1Cn1nnnc12 N1(C(CCC(=O)N(C(C)C)C)=O)CC(C)CN(C(=O)CCc2cnn(C)c2)CC1C N1(C(c2nc(C)c(C)s2)=O)CCC2(CC2)CC1C(=O)NC(c1ccccc1O)C C1(NC(c2c(C)c[nH]n2)=O)CC2CC1N(C(=O)Cc1ccc(C(N)=O)cc1)C2 N1(C(c2cc(CC)c(C)s2)=O)CCCCC(NC(c2cc(C)ccn2)=O)C1 CC(CC(=O)NCC1(C(=O)NCc2cncc(F)c2)CCCC1)C(F)F C(C(C)(C)CC(=O)NCC1CCN(C(C2CC(=O)N2)=O)CC1C)OC C1(C(N2C(C)CC(CNC(CNC(=O)OC)=O)C2)=O)CC2(CCCCC2)C1 c1(C(N2CC(N(C(COCCCC)=O)C)C(O)C2)=O)noc2c(F)cccc12 c1(OC)cc(C(=O)NCCCNC(c2cnn(C)c2)=O)cc2cccnc12 CC1CCN(C(=O)CCOCCNC(c2nccn2C)=O)C1 C1(NC(C2(CCCC(=O)NCC3(C(C)C)CC3)CCC2)=O)CCC(O)CC1 C12(C(N3CCN(C(C(CCC)NC(N)=O)=O)CC3)=O)CC(CC(C)O1)C2 N1(C(C(c2ccccc2)NC(c2cc(C)nn2C)=O)=O)CC2CC(C)C2C1 N1(C(CC(C)C)=O)CCn2ncc(C(N3CCNCC34CCC4)=O)c2C1 CC1C(NC(=O)C2CC2)CCCN1C(c1ccc(F)s1)=O C(=O)(C(F)C(C)(F)F)NCC(CCOC)C.CCOCCOCCOCC c1(C(=O)OC)ccc(C(=O)NC2(CNC(=O)C=C(C)C)CCC2)s1 N1(C(CN(C)Cc2nnc(C)n2C)=O)CCC(O)(CO)CC1.C1(C=O)OCCCO1 c1(OC)ccc(COCC(=O)NCCC(O)CNC(C2CCCO2)=O)cc1 C1(CC)(CC(=O)NC)CC(O)CN1C(=O)CN1CCN(C(=O)C2=C(C)OCC2)CC1 C(C(=O)NCC1CC1NC(C1CC1)=O)(C1CC1)SCC c1(C(N2CC(NC(c3c(C)ccnc3)=O)C(F)C2)=O)cccc2c1CCCC2 N1(CCNC(Cc2c(C)occ2)=O)C(=O)NC(C)C1=O N1(C(c2cc(N)nc(Cl)c2)=O)CCC2CN(C(=O)CCCNC(N)=O)CC12 c1(CC(CC)OC(=O)C(O)Cc2[nH]cnc2C)ccccc1 c1(C(=O)NCCCCNC(C2C(C)(CC)C2)=O)ccncc1N1CCOCC1 C1(C(=O)NC(CCN(C)C)C(=O)O)CCCC2(CC2)C1 C1(C(=O)NC2(C)CCN2C(C2(C(=O)NC)CC(F)(F)C2)=O)CC12CCCCC2 N12CCC(F)(F)C(C1)C2=O.c1(NCc2c(CC)cccc2)c(C#N)cnn1C C(=O)(C1=CC2(CN(C(=O)Cc3cccnc3C)C2)OC1)Nc1ccc(C#C)nc1 c1(C(=O)NC(C(=O)N2C(COC)CC2)CC2CCC2)ccc(C)nc1 O=C1CN(C(c2cccs2)=O)CC(C(=O)NCCn2cc(C3CCCC3O)nn2)N1 Cc1cc(C(N2CCCC2CCNC(C2CC2c2ccco2)=O)=O)nn1C(C)C c1(NCC(C)N(CC)CC)ncc(C)cc1S(=O)(=O)NCCc1ccns1 CC(C)CCCC(=O)NCC12COC(CNC(=O)C(C)(O)C(C)C)(C1)C2 c1(OC)cccc(C#N)c1NC(C1CC(C)CN1C(=O)CCc1ncc[nH]1)=O C(=O)(C(C)CCCC(C)=O)NCC(C(C)(C)C)NC(COCCCCC)=O Cc1cc(O)c(F)cc1N=c1[nH]cc(C(F)(F)F)nc1OCCCO Cc1cc(C)c(-c2cn(CCCN(C(=O)CC3CCSC3)C)nn2)cn1 N(C(=NCC1COC2(CCCCC2)O1)N1CCC(F)(F)C2(CCC2)C1)CCO C=CC1(C(N2CCC(C)(C#N)C2)=O)CCN(C(=O)C(O)CN2CCCC2)CC1 C#Cc1cc(C(=O)NC2COCCC2NC(=O)C(CC=C)C(C)C)cc(F)c1 N1(C(C(=O)NC(CN)C(F)(F)F)=O)CCc2nncn2CC1 C1(NC(C2N(C(c3nccc(C)c3F)=O)CCSC2)=O)CC2(C1)CC(C)(C)C2 C1(CCNC(C(C2CCC2)OCC)=O)(C(=O)N(C(C)CCO)C)CCCC1 C(N=c1[nH]c(=N)[nH]c(=NC2CC(C)(C)C2)[nH]1)c1ccc(C(=O)NC)cc1 CS(=O)(=O)CCCC(=O)N(C1CC1)CC1CCCN1C(=O)CCC(F)F c1(OC)ccc(C2CCN(C(=O)CSC)CC2)cc1OC C12(CC=CC1)C(=O)NC(C)C1CC1C(=O)C2.N1(c2cccs2)CC(N2CC(O)C2)C1.C N1(C(C(C)c2ncco2)=O)C2CCCC1CN(C(C1CC(F)C(=O)N1)=O)C2 N1(C(c2cc(Cl)n(C)n2)C(=O)NCC(=C)C)CCC(O)(P(C)(C)=O)CC1 C(=O)(CCCN=[N+]=[N-])N.n1(CCCCOC)cc(CNC(C2(C)CCCC2)=O)nn1 c1(C(N(CCOC)CCNC(=O)C(C2CCCCC2)O)=O)noc2c1COCC2 N(C(=NCC(C(C)C)C(C)C)NCC1CCCO1)CC1(OCC)CCCC1 c1(NCCC=C=C)[nH]c(=NCc2conc2C(F)(F)F)nc2scnc12 C12CCN(CC1)C2=O.c1(CCNC(c2csc(Br)n2)=O)ccccc1 c1(N2CCC(OC)(CO)C2)nc(N(CCC#N)C)c2c(n1)CCOC2 Cc1ccc2c(=NCC3CCC(C)(C)O3)[nH]c(=NCC3CCCC(F)C3)[nH]c2c1 c1(NC(C2N(Cc3cnc(C)[nH]3)CC(F)(F)C2)=O)c(Cl)cc(Br)c(C)c1Cl N1(C(Cc2ccc(C(N)=O)nc2)=O)CCCC12CCN(C(=O)CCCC(N)=O)C2 c1(C(N2C(C)CC(CNC(CNC(=O)OC)=O)C2)=O)cc2nccnc2cc1F N1(C(CN(C)CCO)=O)CC(O)C(O)C1CNC(C1CCCN1C)=O N1(C(C(CC)N(C)C)=O)CC(NC(=O)Cc2c(Cl)cccc2Cl)CC2(CCC2)C1 N1(C(CC(C)(C)C)=O)CC(NC(c2ncc3[nH]ncc3n2)=O)C2CCCC2C1 C(c1cccnc1)=C(C(=O)NC1CCN(C(C(C)(F)c2ccccc2)=O)C1)F Cn1c(=O)c2c(nc(Cl)n2C(=O)C2CCC(CN(C)C)C2)n(C)c1=O n1(C(C)C)ncc(C(=O)N(C2CCC(NC(=O)C(C3CC3)C3CC3)CC2)C)c1N c1(OC)cc(C(=O)NC2CCCCC2CCNC(C2(C)CCC2)=O)ccn1.C1CC1 C1(CCN(C(CNC(C(C)NC(CC)=O)=O)C)C)CCOCC1 C1(C(=O)NCc2ccc(F)nc2)(NC(Cn2ncc(CC)c2)=O)CCC(C)(C)C1 N1(C(c2c(C)nns2)=O)CCC(O)(CC(=O)NCc2cccc(O)c2C)CC1 C1(CNC(c2c(C)onc2Cl)=O)C2CCCC1N(C(c1csc(CO)n1)=O)C2 c1(-c2cc(C(=O)NCC=CCNC(CC3C(C)C3)=O)on2)cccc(Cl)c1 C1(C(=O)NCCN(CC#C)CCOCCOC)CCCC1C c1(-c2nc(CCCCC)nn2C2CCS(=O)(=O)C2)cc([N+](=O)[O-])c2nsnc2c1 C1(COC)(OC2(C)CN(C(=O)NCC3CCC3)C2)CCCCCCC1 Fc1cnccc1CC1CCC1ON1CCC(NCCOc2ccccc2)CC1 C(=O)(C1=C(C)NC2=NCCCC2=C1)NCC(C)NC(C1C(CC)CCCC1)=O N1(C(C(F)OC)=O)CC(NC(=O)CCc2cc(C)on2)C(C)C1 C(=O)(C1=C(C)OCC1)NCc1c(CNC(CCCOC)=O)cccn1 c1(C(N2CC(OCCNC(c3nc(C)nn3C)=O)C2)=O)cnc2n1CCCCC2 Cn1ccc2ccnc(C(N3CCC4(CCCN4C(C4C=CCC4)=O)C3)=O)c12 c1(OCC)cc(CC(=O)NCCOCCC2(C)CCOC2C)cc(F)c1 c1(C(=O)NC2CN(C(c3c(C)csc3)=O)C3(C2)CCC3)cccc([N+](=O)[O-])c1N S(=O)(=O)(c1cccnc1NCCc1ccccc1OC)N1CCC(CC)C1 C12(NC(C(CC)NC(C)=O)=O)CCCC1N(C(=O)C=C1CCC1)CCC2 C(C)(C)(CC(=O)NC(C)(C)C)N(C(=O)C(c1cnccn1)=O)C Cn1cc(S(N)(=O)=O)cc1C(=O)NCC1CCN(C(C2(C)CCOC2)=O)CC1 C1(NC(c2cc3ccncc3[nH]2)=O)CCC12CCN(C(=O)CSC1CC1)CC2 N1(C(c2cccc(SC)c2Cl)=O)CCC2CN(C(=O)C3=NOC(C)C3C)CC12 c1(C(=O)NCCCC(C)NC(C2CC23CCSCC3)=O)[nH]nc2c1COC2(C)C C12(CO)CC(CN3CCC(OC4CCCC4)CC3)(CO1)C2 C12(C(=O)NCCOC3CN(C(c4c(CC)con4)=O)C3)CCCC(=O)N1CCC2 CCC(C)CC(=O)NCC(C1CCCN1C(=O)CCc1cccc(OC)n1)(C)C C1(CNC(C(CC)(C)O)=O)CN(C(c2ccc(Br)c(C)c2F)=O)CCC1(C)C N1(C(C(C)c2cc[nH]n2)=O)CC2COCC2(C(=O)N(C(C)C)CC2CC2)C1 C(=O)(C(O)P(C)(C)=O)N1CC(N2CCN(C(C=C(C)c3cccs3)=O)CC2)C1 C1(C(=O)NCC2(CN(C(=O)CC(C)(C)O)C)CC2)CCC2(CCC2)CC1 Cc1nn2ncccc2c1C(=O)NC1CCCC1CNC(=O)Cc1ccsc1 CC(C)CCCCC(=O)N1CCCC1C(=O)NC1(C)CCOC1 c1(C(N2CCC3(NC(C(=O)NCC(F)F)=O)C(C2)C3)=O)cn2cccnc2n1 c1(C(N2CCN(C(Cc3c(C)n(C)nc3)=O)CC2)=O)cnn2ccc(O)nc12 C1(C(=O)NCC2(C(N)=O)CN(C(=O)C=Cc3cc[nH]n3)C2)CC12CCCOC2 C(=O)(C1CCCc2nccn21)N1CCC2CN(C(C(C(=O)OC)(C)C)=O)CC21 c1(C(=O)NCC(C)(C(C)C)NC(C(CC)F)=O)c(F)cncc1Cl C1(NC(c2ccn(CC)n2)=O)CCCCC1CNC(=O)CC(C)c1ccncc1 C1(NC(c2cnc(C3CC3)nc2)=O)CN(C(C2CCCCC2)=O)CCC1CO CCC(C#N)C(=O)NC(C)(C(=O)N(C)Cc1ccccn1)C1CCC1 C1(C(N(C2CCCN(C(c3cncn3C)=O)C2)CC)=O)CCS(=O)(=O)C1(C)C C1(N(C)C(C2SCCS2)=O)CC2CC1N(C(c1cc(F)cc(Cl)c1)=O)C2 C1(NC(c2ccc(N(C)C)cc2)=O)CCN(C(c2cc(C(F)F)no2)=O)CC1O c1(C(=O)NCCCCOC=C)noc2cc(-c3sccc3C)ccc12 C(=O)(CCN=c1ccc(S(=O)(=O)NCCCNCCC2(SCC)CC2)c[nH]1)NC CC12CC(CNC(=O)NCC34CC(C#N)(C3)C4)(C1)OC21CCC1 c1(C(=O)NC2(C)CC(NC(c3cscc3F)=O)C2)cnc2ccccc2n1 C1(C)(NC(CC2CN(C(COc3ccc(C)cc3)=O)C2)=O)CCCCC1C Cc1cc(=O)c(C(=O)NCC(C)(C)NC(=O)Cn2cccn2)cn1C1CC1 c1(C(C(=O)NC(C)C)N(C)C(c2cccc(Cl)c2)C)sc(Cl)cc1Cl c1(NC(C2(C)CCN(C(C(C)NC=O)=O)C2)=O)c(Cl)cc([N+](=O)[O-])cc1Br c1(CCC)nc(C(F)Cc2ccccc2)n(-c2ccc(Cl)cc2)n1 C1(Nc2cc(C)c(C)o2)CC2CCC(C1)N2C(c1cc2nnnn2cn1)=O c1(-c2c(C)n(C)nc2)cnc2[nH]c(C(=O)NCCN3CCCC3)cc2c1 CCC(C)C(CC(=O)N(C(CO)C(C)C)C)NC(=O)CN(c1ccccc1)C CC(C)(C)C(=O)NCCCC(=O)NCCNC(=O)C=CCN1CCOCC1 c1(C(N(C2CCN(C(=O)C=CCOc3ccc(F)cc3)C2)C)=O)cc(Cl)ccn1 c1(CC(=O)NC2COCC2NC(C2CN(C3CCOC3)C2)=O)ccccc1O c1(C2(CNC(=O)CC(=O)N(CCC3C(C)(C)C3)C3CC3)CC2)ccc(F)c(Cl)c1 C#CCC(C(=O)N(CC(C)CO)C)NC(C1CCCC(CF)C1)=O C(=O)(C(F)C(F)(F)F)N1CC(CNC(c2csnn2)=O)OCC1 C(CCOC)(C(C)C)NC(C(n1cc(COC)nn1)C)=O C(C(C)(C)CNC(=O)C(C)(C)N1CCCC1)N(C(CCOCCOCC)=O)C C=C1CC2(C1)CC(C(=O)NCC(CNC(c1ccsc1C)=O)C(F)(F)F)C2 Cc1oc(C(N2CCCC(CNC(=O)C(C#N)C(C)(C)C)C2)=O)cc1S(N)(=O)=O C1(NC(C(CC#C)O)=O)CC2(CCN(C(c3nc(Cl)cs3)=O)C2)C1 C1(C(N)=O)(OC)CN(C(c2ncoc2CNC(=O)C(c2cncn2C)O)=O)C1 N1(C(CC2C(C)CC2)=O)CCC2(NC(=O)CN(C)C3CC3)CCCC12 c1(NC(C2N(Cc3scc(C)c3)CC(F)C2)=O)cccc(C)c1O C(C(=O)NC1CCCC1SC)(C(C)O)NC(C(C1CC1)OC)=O N1(C(=O)NC2CNCCC2F)CCCCC1c1ccc(C(F)(F)F)cc1 C(=O)(C1=CC2C=CC(C1)C2)N1C(C(=O)NCC2C(CC)C2)CNC(=O)C1 C(=O)(CCCCCC(C)(C)C)NCC(C)N(C(=O)C1=CCCCC1C)C C1(C(=O)NC(C)CNC(c2cc(Cl)n(C)n2)=O)CCN(CCO)C(=O)C1 N1(c2ncnc(CC)c2F)CCN(C(c2cc(F)c(Br)c(F)c2)=O)C(C#N)C1 Cc1nc2cc(C(=O)NCCCCNC(=O)CCc3ccc[nH]3)ccc2s1 C1(CNC(CCCC#C)=O)CN(C(=O)C(F)=CC2CC2)CC1(F)F O(NC(=O)CC(CC)C(CC(=O)NCCC(=O)NCCC)C)CCCC C(C(O)CC(F)(F)F)NC(CC(COC)NC(=O)CN1CCCC1)=O c1(OC)ncc(Br)cc1CC(=O)NCC(C)N(C(=O)CC1CC(F)C1)C c1(C(N2C(CC#C)CCC2)=O)cccc(Cl)c1CN1CCCC1 c1(C(=O)NC(CC(C)C)C(=O)N(C)C)n[nH]c2c1CCC(C)(C)C2 c1(C(=O)NCC(C)CNC(c2cscc2F)=O)cnc(N(C)C)s1 c1(SC)cc(C(N2CCC2CNC(C2CCCC23CCC3)=O)=O)ccc1F.C1(C)CC1 C(=O)(C1CCCn2nccc21)NCC1CCCCN(C(C(F)=CCC)=O)C1 Cc1nc(C)c(CC(=O)NC2CCC2NC(c2c[nH]nc2C2CCCCC2)=O)s1 c1(OC)ccc(CC(N2CCCC2CNC(=O)C(C)(C)CSC)=O)cc1F C(CN=c1nc(NC)c2c([nH]1)CCS2)(C1CN(C(c2cnc[nH]2)=O)C1)CCOCC C1(CC(=O)NCCOCCNC(CCN(C)CC)=O)CCCS(=O)(=O)C1 N1(C(c2cc(C(=O)OC)cc(Br)c2)C(=O)NCCC#N)Cc2c[nH]nc2C(C)C1 c1(C(=O)OC)n[nH]c(C)c1Cn1cc(C2CCN2C(c2ccc(Cl)cc2)=O)nn1 N1(C(CC)=O)CCC(CNC(=O)CC2CN(C(C)=O)C2)C1.C12CC1C(=O)N2 N1(C(c2c(SC)snn2)=O)CC(CNC(c2ccc(C(F)F)cc2)=O)CC1C N1(C(C(N)=O)=O)CC2(C1)CN(C(C1CCCN1C=O)=O)C2 N1(C(c2c(CNC(C(C)N=[N+]=[N-])=O)cc[nH]2)=O)CCC2(CCCC2)CC1 CC(CCCCCO)NC(c1csc(CNC(=O)CC2(C)CCCCC2)c1)=O Cc1cc(CC(=O)NCC=CCNC(C2CCCC(C)C2)=O)ccc1O C1(C(N2CC(CCNC(C(C)OCCOCC)=O)C2)=O)CCn2nnnc2C1 CCC(C(=O)NC(C)(C)CN(C(=O)C(c1ccc(OC)cc1C)(C)C)C)C(C)O CC(C)(C)C(O)CCC(=O)NC1COCCN(C(c2cc(Cl)ncc2F)=O)C1 c1(C(N2CCC(CNC(C3CCCN3C3CC3)=O)CC2)=O)c(O)cc(O)cc1O N1(C(c2cccc(C#C)c2)=O)CCC2CCN(C(=O)CC3CC(C)(C)CO3)C2C1 C#CCC(C(=O)NC1(c2noc(C)n2)CC1)NC(C1CC1(F)Cl)=O CC(C)(CC(F)C(=O)NCCCS(N)(=O)=O)NC(C1(n2cccn2)CC1)=O CC1CCc2[nH]nc(C(N3CCOC(CNC(C45CCCCC4C5)=O)C3)=O)c2C1 C1(CNCCCn2ncc([N+](=O)[O-])c2)C(F)CC12CCC2 Cc1ncc(C(N2CC(O)(CNC(=O)CC3CCCCO3)C2)=O)n1C c1(OC)ccc(C(N2CC(C)CC2C(=O)Nc2cc(C(N)=O)ccn2)=O)cc1Br c1(NC2CN(C(C3(C)CCCN3)=O)C2)nc2ccc(Cl)cc2s1 C(C)(C(C(=O)N1C(=O)NC(C)(C)C1=O)C(C)C)c1c(C)noc1C.O c1(CC)cc(F)cc(C(=O)N(C)Cc2cc(F)ccc2Cl)c1C C(=O)(C(CCS(C)(=O)=O)NC(=O)CC(=O)Nc1cccc(Br)c1)OCC N1(C(C2C(C)(CC)C2)=O)CCN(C2CCCN(C(c3ccoc3Br)=O)C2)C(=O)C1 C1(CC)CN(C(=O)C=Cc2ccn(C)c2)CCN1C(c1oc(C)nc1C)=O c1(OC)cc(C)c(NC(c2nnnn2CCCF)(CC)C2COC2)cc1F N1(C(C(N2CCSCC2)C)=O)CC2CN(C(c3ccccc3Cl)=O)CC2C1 C1(NC(C(C=CC)O)=O)CC2CCC1CN2C(=O)C(F)OC(F)(F)F CN1CCCC2CCN(C(=O)NCc3ccc(Br)c(F)c3F)CC12 c1(C(=O)NCCCCCN(C(=O)Cc2cn[nH]c2)C)ccc(Cl)c(F)c1 C1(O)(CNC(C(COCC)C)=O)CCCN(C(=O)Cc2cccc(F)c2)C1 C1(CCNC(C2CNC(=O)N2)=O)CCCCN1C(=O)CC(F)F CC(CN=c1[nH]c2ccc(S(=O)(=O)N3CCS(=O)C(C)(C)CC3)cc2s1)N(C)C N1(C(c2nc(CC)oc2C)=O)CCC(NC(=O)C=Cc2ccc(C)o2)C12CCC2 N1(C(c2sccc2CO)=O)CCC(CO)(CNC(C23COCC2C3)=O)C1 CC1=C(C(=O)NC(c2ccco2)CO)C(C)n2ncnc2N1C C(=O)(CCC(=O)NN(C)C)N1CC(C)C(NC(=O)C(CO)c2ccccc2)C1 c1(NC(CC2N(C(c3c(C)nc(C)s3)=O)CCC2)=O)cc(C)c(F)cn1 Cc1nc2c(s1)CN(C(C(=O)NCc1ccccc1Br)c1csnn1)CC2 c1(OC)cccc(C(CF)NC(=O)NCCCCN2CCCCC2C)c1 CCC(C)(COC)C(=O)NC1CC(OC)CN(C(C2CCC(CO)CC2)=O)C1 c1(-c2cn(CC3CN(C(c4c(CC)cc[nH]4)=O)C3)nn2)ccc(Cl)cc1C c1(CC(=O)N(C)CC2OCCN(C(C3(COC)CC3)=O)C2)ccc(C#N)cc1 c1(C(N2CC(C)C(NC(=O)CCCCCF)C2)=O)ccc(=O)n(C)c1 CCC1=NOC(C(=O)NCC(C23CCC(CC2)C3)NC(c2nn(C)cc2C)=O)C1 c1(C(N2CC3C(NC(=O)CN4CCCC4=O)(C3)C2)=O)cnn2cccnc12 c1(C(=O)NCC(N)C(F)(F)F)ccc(-c2ccccc2)nn1 CCC(CC(=O)N1CC(O)(CO)C1)NC(=O)C=CC1CCOC1 N1(C(Cn2cc(COCCC)nn2)C)CCc2onc(OC(=O)N(C)C)c2C1 C1(NC(C2(N(C)C)CCCC2)=O)CC(NC(=O)CCc2cccnc2Cl)CC1O Cc1sc(C(=O)NCCOCCCNC(=O)C(F)(F)C2CCCC2)cc1[N+](=O)[O-] c1(OC)ccc(O)cc1C(=O)NCC(C)N(C)C(c1cc(C)ccc1OC)=O Cc1cc(F)ccc1CC(N1CCC(CNC(C2CN(C)CCO2)=O)C1(C)C)=O c1(C(=O)NC2CN(C(c3c(CC)occ3C)=O)CC2C)ccc([N+](=O)[O-])c(C)c1 C1(C)(NC(CCCCSC)=O)CCCCC1C(N1CC2CC1CS2=O)=O c1(C(=O)Nc2cccc(OCC)c2)noc2cc(-c3ccsc3CO)ccc12 C(N=c1nc(N2CCC3(CCOC3)C2)c2c([nH]1)CCOC2)c1n(C(C)C)ncn1 C1(CNC(=O)Nc2c(-c3cc(C)no3)cccc2)N(C)CCCC1(C)C c1(CCC(=O)NCC2CN(C(C(C)C3CCOC3)=O)C2)cccnc1 c1(C(=O)NCC(CNC(C(C)CSc2ccccc2)=O)O)cc(N)c(F)cn1 N1(CC(=O)NC2(CO)CN(C(=O)CC3CC=CC3)C2)CCCCC1 N1(CCCN=O)C(CCCC)C(N=[N+]=[N-])CN(C)C(=O)C1 C(c1ccc(F)c(Cl)c1)=CC(=O)NCCOC1CCN(C(C(C)O)=O)CC1 C1(C(=O)NCC2CCCC(NC(C3(NC(C)C)CC3)=O)C2)OCC2COCCC12 C(=O)(C1COc2ccc(Cl)cc21)NCC1CN(C(C(C)c2cc[nH]n2)=O)C1 C(CC(C(=O)NCCC(=O)NC(C)C)NC(=O)CC1(C#N)CC1)OC C1(C(=O)NCC2OCCN(C(c3c(C)ncn3C)=O)C2)C(C)OC(C)C1C c1(C(N2CC(CCNC(C(C)N3CCC3)=O)OCC2)=O)cccc2c1OCCN2 Cn1nc2c(c1C(=O)NCC1COCCN1C(c1cc(F)ccc1O)=O)CCC2 c1(C(=O)NCC(C)(O)CNC(C2CCCCC2O)=O)ccc(S(N)(=O)=O)cn1 N1(C(CN(CC(=O)NCc2ccc(C)o2)C2CC2)=O)C(C)CCCC1C c1(OC)sc(C(=O)NC(C)(C)CNC(c2cnc(S)nc2)=O)cc1Br C1(C)(NC(c2cc(C)c(C)s2)=O)CCCN(C(C2CCC2C#N)=O)C1 O=C1CCC(NC(N2CCN(C(=O)NC3CC(O)C3)CC2)=O)C(=O)N1 c1(C(N(C2CCC(CNC(C3CC(F)C3)=O)CC2)C)=O)cc(F)c(F)c(F)c1F CC(C)C(F)(F)CCN=c1[nH]c(=NC(C)c2nc[nH]n2)c2cccc(F)c2[nH]1 Cc1cc(NC(CN(C)C)CO)ncc1S(=O)(=O)N1CC(C)C(C)C1 C(C)(CNC(=O)C=CC1C(C)C1(Cl)Cl)(CC(C)C)NC(CCC=C)=O C12(C(=O)NC(C3CN(C(c4cnn(C(C)(C)C)c4)=O)C3)C)CC(C(=O)O)C(C1)C2 C1(C(N)=O)CN(C(=O)C(=O)Nc2cc(C3CC3)sn2)CCC1C(=O)O C(=O)CCC[N+](=O)[O-].C1(c2cn(CC3NCCC3)nn2)(SCC)CC=CCC1 C(=O)(CCCC(C)O)NCC1C(NC(c2c(COC)ccs2)=O)CCC1 N1(C(CCSC)=O)CC(CNC(c2ccccc2CO)=O)OC2COCC12 c1(NC(=O)COc2ccncc2-c2cncnc2)ccc(F)cc1Cl C1(CNC(C2CCC(C)C2)=O)CN(c2cc(Cl)ncn2)CCC12CCOCC2 N1(C(c2cc(COC)[nH]n2)=O)CCCC(O)(C(N)=O)C1.C12CCOC(C1)C(=O)N2 c1(CNC(C2CC(NC(C3C(C=C)OCCC3)=O)C2)=O)cc(C)c2[nH]cnc2c1 c1(C(N(CC(=O)NCC2CC2(C)C(C)C)CC#C)=O)cc(CC)no1 N1(CCNC(c2n[nH]cc2Cl)=O)CC2C3C=CC(CC3)C2C1 CC(C)(C(=O)NC1CC(C)(NC(=O)CNC(c2ccsc2)=O)C1)C1CC1 c1(NC)ccc(C(N2CCC(NC(C3(Br)CC3)=O)CC2C)=O)cc1F N1(C(C(CC=C)N(C)C)=O)CCC(C)(CNC(c2cn(C)nc2C)=O)CC1 c1(C(=O)NC(CSC)C)ccc(C2OCC2(C)C)cc1 C1(O)(CNC(C2CNC(=O)N2)=O)CCN(C(C2CCCCS2)=O)C1 C1(C(=O)NC2CCCC(CNC(=O)CCOCC3CC3)C2)(CC)CCCCO1 C1(CC(=O)NCC2(CNC(c3nc(C)oc3)=O)CC23CCC3)CCC(F)(F)CC1 Cc1cccc(Br)c1C(C(=O)NCCC(C)F)NC(C1CC2CC(=O)C1O2)=O c1(C(C(=O)N2CC(NC(C3CC(=O)NC3)=O)C2)(F)F)cccc(F)c1 N1(C(c2c(CC)con2)=O)CC(CC(=O)N(CC(C)C(C)C)C)CC1(C)C C(=O)(C(C(C)OC)NC(c1cc(C#N)cs1)=O)N1CC(COC)C1 c1(SCC(=O)NCC(CC=C)NC(=O)C(O)C=C)cnn(C2CCCC2)c1C c1(C(=O)NCC2C(C(N(CCCCOC)C)=O)C2(C)C)nnc(S)n1C C1(CC=C)(NC(=O)Cc2n[nH]cc2Br)CCN(C(=O)CS(=O)(=O)N(C)C)C1 C1(C(N2CC(c3cn(CC(O)C(F)(F)F)nn3)C2)=O)C2CCCC(=O)C12 c1(CC)n[nH]cc1C(=O)NC(C)CCN(C(C1CCC1COC)=O)CC N1(C(=O)Cn2cc(Br)ccc2=O)CCCN(C(=O)CSC2CC2)C(CO)C1 N12CCN(CC1)CC2=O.c1(C(N2CC(C)C2)=O)coc(C2CCC2)n1.CC(C)O C(C1CC1)(C1CC1)=CC(=O)NC(C(=O)NCCN(CCC)CC)C1CCC1 C1(OCC)CCCC(NC(C23CC(C(=O)N)(C2)C3)=O)C1.C1(COC)CCOCC1 c1(C(=O)NCC2(c3cn(CC(C)NC(=O)C4CC4)nn3)CC2)c[nH]c(C#N)c1 N1(Cc2n(C)nnc2)CCS(=O)(=O)C(CCNC(c2cnc(F)c(Cl)c2)=O)C1 Cc1cc(O)ccc1C(=O)NCC1(C)CCCN1C(=O)CCN1CCOCC1 CCCCCCC(CC)C(=O)N1CC2CC(NC(c3cccc[n+]3[O-])=O)C1C2 C1(O)(C(=O)OCC)CN(C(c2ccccc2)C2CC2)C1.C12CCC1NC2=O c1(OC)ccc(C(=O)NCC(CCOC)NC(=O)C(CC2CCCC2)OC)cn1 N1(C(C(=O)N(CCCN(C(C2C(C(=O)OC)COC2)=O)C)C)C)C(=O)CCC1=O C(=O)(C(O)CCC(C)C)NCCCCCN(C(C1(C)CC=C(C)CC1)=O)C c1(SC)ccnc(C(N2CCCC2CCCN(C)C)C)c1 c1(C(C)C)nc(Br)ccc1C(=O)NCc1csc(Sc2cnc(C(F)(F)F)nc2)n1 C1(C(N2CC(COC)C2(C)C)=O)CCC2CCC1N2C(c1cc(F)cnc1O)=O N1(C(C(C)=C(C)C)=O)CCC(C(=O)NCCC2(C)CC2(F)F)C1(C)C c1(OCCCC)ccc(C(N2CCC2CNC(C2C(C#N)C2(C)C)=O)=O)cc1 c1(NC(=O)NC)ccc(C(=O)NCC2(C)CCN(C(c3ncccn3)=O)C2)cc1 C1(CC(=O)NCCCF)CN(C(=O)C=C(C2CC2)C2CC2)CC12CC2 c1(C(N(CCNC(=O)Cc2cncn2C)CC)=O)c(C)c(O)nc2ccccc12 C1(O)(CN(C(Cn2c(C)ncc2)=O)C)CCCN(C(=O)C(c2cnn(C)c2)C)C1 C1(N(C(=O)CC2CSC2)CCC)CCN(C(=O)CC2CCCOC2)CC1 Cc1cc(C(=O)N(C(C)CNC(C2CN3CCC2CC3)=O)C)cc(F)c1 N1(C(C(C)CC2CCC2)=O)CCOC(CCNC(C2(C(N)=O)CC2)=O)C1 c1(C(=O)NC2CCCC(CNC(C3CCCC3)=O)C2)cccc2occc12 C1(C(=O)OC)CCC(C(N2CCCC2C(C)(C)CNC(c2ccsc2)=O)=O)CC1 c1(C(C)=O)cccc(C(N2CC(NC(=O)C(C)(O)C3CC3)C(C)C2)=O)c1 c1(OC)cccc(C(=O)NCC(C)NC(=O)Cc2cn(C)nn2)c1C c1(C(N2CCCC(C)C2CNC(=O)C2=CSCS2)=O)[nH]nc2ncccc12 C(=O)(CC(C(C)NC(=O)C(CN(C)C)CC)N(C)C)N1CCC(COC)C1 CC(C(=O)NCC12CC(NC(c3cocn3)=O)(CO1)C2)C1=CCCC1 C1(NC(CCN(C(CCC)C)C)=O)CN(C(c2ccc(C)c(C)n2)=O)CC2CC12 C(=O)(C(CC(C)(C)C)NC(=O)C(CC1CCC1)OC)N1CCCC(CCOC)C1 c1(C(=O)NCCOCCN(C(Cn2c(C)c(Cl)cn2)=O)C)occ2c1CCC2 c1(Cc2scc(CN(C3CCC(O)C3O)CC)c2)cnc2cc(C(=O)O)ccn12 N1(Cc2nc(CCCC)[nH]c2Cl)C2CCC1CC(NC(c1ccn(CC)n1)=O)C2 c1(C(=O)NCC(CNC(c2ccc(C#N)cn2)=O)F)c[nH]c2cccc(Cl)c12 N1(C(CC23CC(C(C)(C)C)(C2)C3)=O)CCOC(CCNC(C2CC(C)(O)C2)=O)C1 c1(C(N2CCC(CCOC)(NC(=O)C(C)OC)C2)=O)ncc(F)c2ccccc12 C1(CC(=O)NCC2C(CNC(CC(=O)OC)=O)C2)CCC(C(F)(F)F)N(C)C1 CCCC(O)C(=O)N1CCC(OCC(=O)NCCC23CC(CCO2)C3)C1 N1(CCCCCNC(c2c(CC)nc[nH]2)=O)CCN(C(=O)C(C)=C2CC2)CC1 CC(C)CC(CNC(=O)CNC(N)=O)C(=O)N1CCOC(c2cc[nH]n2)C1 C(CCCCCNC(=O)C1=C(Cl)CC1)NC(COCCCC#C)=O N(C(=NCc1ncccc1OC(F)F)NCC1CCC1)C(CCOC)C C1(C)(CC(=O)NC2(C(F)F)CC(NC(Cc3cnc(C)s3)=O)C2)CCCCC1 C1(N)CC(C)(C(=O)NOCC(O)C(C)C)C1.C=C1CC1C(CCCO)=O C1(NC(C(=O)Nc2c(OCCOC)cccc2)=O)CCN2CCCCC12 CC(F)(F)CCCC(=O)NC(C)(CNC(c1ccccc1[N+](=O)[O-])=O)C1CCC1 N1(C(Cc2cc(OC)no2)=O)CC2(CC2)CC1C(=O)NCC1(CF)CCC1 c1(CC)nc(=N)[nH]c(=NCC(O)CNC(c2cc(OCC)ccc2C)=O)[nH]1 C1(CN(C(CCOCCN(C(C(C=CC)O)=O)C)=O)C)CCCC2CC12 C1(NC(c2nc(C)oc2C)=O)CC2CCC1CN2C(C1CCC(O)CC1)=O C1(C(=O)NCC(CC)NC(c2c(Cl)ccc(C)c2O)=O)COCC2(CCC2)O1 CC1(C)C(NC(C2C(C#N)C2(C)C)=O)CC1C(N1C2CSCC1C2)=O c1(C(C)NC2CC3(C=O)CC23)ccc(-c2cnco2)cc1.C(=O)O C1(C(NOCC(=C)Cl)=O)CCN(C(C2CC23CCC3)=O)C1(C)C c1(CC)cc(C(C)C(=O)N(C)Cc2cn(-c3ccc(F)cc3F)nn2)ccc1C c1(C(N2C3CC(NC(CSCCC)=O)(C3)C2)=O)c(C)ccc(C)c1O Cc1ccc2sc(C(=O)NCCC(C)(C)NC(=O)C(C)C(C)O)c(C)c2c1 c1(C(N(CC(C)(C)NC(C=Cc2cnc(C)s2)=O)C)=O)cc2cc(Cl)ccc2o1 Cc1nc(C(C)C)sc1C(=O)NC1CCCN(C(C2CC3(C2)CC3F)=O)C1 C(=O)(CCCCCCCO)N1CC2(CCN(C(=O)CC3COCCO3)C2)C1 c1(C(=O)NC2C(C(=O)OCC)C2)nccc2c(S(N)(=O)=O)cccc12 c1(NC(C(C)NC(C(C(C)C)(C)O)=O)C(C)C)nc(Cl)nc2c1nnn2C CC(C)C(C)C(C)CC(=O)NCC1(CCNC(C2SCCS2)=O)CC1 C1(C)(CC)CN(C(C2CNC(=O)CN2C(C2CC(OC3CC3)C2)=O)=O)CCO1 N1(C(=O)OC(C)(C)C)CC(C(=O)NCCn2cc(F)ccc2=O)CCC12COC2 Cc1ncc(C(=O)N(CC(C)CNC(=O)Cn2nccc2C)C)cc1N C1(NC(C2C(OC)C2)=O)CCC(O)CN(C(c2cccn3ccnc23)=O)C1 C1(O)(COC)CCOCC1NC(=O)C(N)C1(C(F)(F)F)CC1 Cc1cc(C(N2CCC(N(C)C(c3cnc4n3CCS4)=O)C2)=O)ccc1Br Cc1ccccc1C(C)C(=O)NC(C)Cn1cc(CCc2nn[nH]n2)nn1 C1(C2CC2)(C(=O)NCCN2C(=O)CNC2=O)CN(C(=O)C=C2CCC2)C1 c1(CNC2C(C)CN(C(=O)CC3CCCC(C)C3)CC2)cc2ccccc2cn1 Cc1cc(CC(=O)N(CC(C)NC(C2COCCC2(F)F)=O)C)cc(C)c1 C(C(=O)NC1(CNC(=O)C(O)C(F)F)CCC1)(C(C)C)SCC(C)C N1(CCC(=O)NCCCC(C)NC(=O)CCN(C)CCO)CCSC(C)(C)C1 c1(C(=O)NC2CCC2CNC(C2(CO)COC2)=O)ncsc1-c1ccccc1 C1(O)(CC(N2CC(C(C(=O)NCc3n(CC)ccn3)OC)C2)=O)CCOCC1 C12(NC(CSC)=O)CCCCCC1N(C(=O)CCc1cn(C)nn1)CC2 C1(CNC(C2CC23CCOCC3)=O)C2CCCC1N(C(C1CCCC1O)=O)C2 c1(NC(=O)NCCS(CC)(=O)=O)ccc2c(c1)c(C)nn2C C1(COC)(NC(=O)C(N2CCC2CNC(=O)CS(=O)(=O)N(C)C)=O)CC=CCC1 N1(C(CSc2n(C)ccn2)=O)CCN(CC2CN(C(c3ccc(CO)o3)=O)C2)CC1 c1(C(N(CC(C)NC(C2C(C)(CC)C2)=O)C)=O)cnc2sccc2c1 C1(CNC(C(N2C(CC)CCC2)=O)=O)C2CN(C(=O)CP(C)(C)=O)CC12 C1(C(N(CC(C)C(=O)N2CC(N3CCOC3=O)C2)C)=O)Cc2nccn2C1 c1(C(N2CCC(c3nc(C)cs3)C2)C(=O)NCCCC)nnc(C2CC2)s1 CC(C)CC(C)CC(=O)N1C(CNC(c2cc3ccsc3s2)=O)CC2CC12 C=CC(C)(O)CC(=O)NC1(CC)CN(C(C2Cc3nccn3C2)=O)C1 N1(C(c2c(C)n[nH]c2C)=O)CCC2CN(C(=O)C(C)(C)CNC(N)=O)CCC2C1 C1(NC(C2CC3CCC2O3)=O)CCCCN(C(=O)CC2CSCCS2)C1 C1(C(=O)NCCC(C)OC)(COCC)CN(C(=O)CN2CCCCC2)C1 c1(C(=O)NC2(CC=C)CN(C(=O)C(N3CCCC(C)C3)=O)C2)cccc(NC)n1 c1(CCC2CCCN2C(=O)NC2CN(C)C(=O)C2)cc2ncccc2o1 C12(CNC(c3c(C)nn(C(C)C)c3)=O)CCC1CCN2C(c1ccc(N)cn1)=O C1(C(=O)NCCCC2OCCN(C(c3n(CC)ncn3)=O)C2)(OC)CCCOC1 Cc1nc2ncccc2cc1C(N1CCCN(C(c2coc(Cl)n2)=O)C(C)C1)=O c1(C(=O)NC2C(CNC(=O)C=CC(F)(F)F)CCC2)cncc(Cl)c1Cl CC1CCN(C(=O)CN=S(C)(C)=O)CC1NC(c1c[nH]nc1C1CCCCC1)=O C(=O)(CCCC(=O)N1CC(CC(F)C(N2CCCC(CO)CC2)=O)C1)OC C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCN(C(CCC)=O)C(c2nn[nH]n2)C1 c1(SC)ncc(C(F)(F)F)c(NC2CCCC2C(=O)NC(c2ccsc2)C)n1 c1(C(N2CC(CN(C(=O)OC(C)(C)C)CC)OCC2)=O)cc(OCC)cnc1F C=CC(C(=O)NC(c1cccnc1)C(=O)N(C)CC1COCC1O)OC C1(C(=O)N(CCN(C(CCC#C)=O)CCOCCO)C(C)C)COc2cc(O)ccc2C1 Cc1nc(C)c(C(=O)N(C2CCN(C(=O)C(C)OC3CCCCC3)C2)C)nc1C c1(NCC(c2ccc(F)cc2F)OC)ccc(S(=O)(=O)NCCN(C)C)cc1F C1(CNC(CCN(C(COC2(C)CCCC2)=O)CC2CC2)=O)CC(O)CCO1 n1(CC)nc(CC)cc1C(=O)NC1(C)CCN(C(C2CC(CC)(CC)C2)=O)C1 C1(C2CCCN(C(c3cnn(C4CCC4)c3)=O)C2)(NC(C2CC2F)=O)CC1 C#CCC(O)C(=O)NC(C1CC(NC(=O)CCc2cn[nH]c2)C1)C c1(C(C2CC2)NC(N(C(c2cccs2)C)C)=O)cccc(O)c1 N1(C(C(C2(C)CC2)NC(C=CC(C)(C)C)=O)=O)CCC(O)C(F)(F)C1 c1(N2C(C)CC(NC(CCS(=O)(=O)NC)=O)C2)ccc2cnccc2c1[N+](=O)[O-] c1(C(=O)NCCCC(N2CC(C)SCCC2)=O)ccc(N=[N+]=[N-])cc1 C1(NC(c2ncnc(O)c2F)=O)CC2CC1N(C(C1Cc3cscc3C1)=O)C2 CP(C)(=O)CN1CCCC(C(N2CCC(CNC(c3c[nH]nc3F)=O)C2)=O)C1 C1(C(=O)NC2CCC(N(C(=O)CC(C)(C)O)C)CC2)CC2CCCN(C1)S2(=O)=O CC1CCN(C(=O)CCn2cccc2)CCN1C(=O)CCn1cnccc1=O O=C1CC(C(=O)NC2CN(Cc3ccc(C(F)(F)F)cc3Br)CC2F)NC(=O)N1 c1(CN(C(=O)CN(C2CC(C#N)C2)C(=O)C(F)F)CC)ccccc1 C1(C(N2C(C(C)C)CN(C(=O)CC3(C)CCCO3)CC2)=O)CCC2(CCCC2)C1 C1(C(C)NC(C2(CCO)CC2)=O)CCN(C(C2(c3ccccc3)CCOC2)=O)C1 C12(C(N3C(CNC(c4cccc(OCC)c4)=O)CC(C)C3)=O)CCC(C1)OC2C C(CCCCOC)N(CC=C)C.C(C=CC(=O)NCCCC)(CC)=CC N1(C(c2cc(OCC)ncc2)=O)CC(NC(=O)CC(=O)OC)CC1(CC)CC c1(C(=O)NC(CNC(CNC(CC)=O)=O)(C)C2CCC2)cccn2ccnc12 C1(CS(=O)(=O)NC(C)C(=O)NC(CNSC(F)(F)F)C2CC2)CCCCC1 c1(C(N2CCC(C)(NC(C3(Oc4cccc(C)c4)CC3)=O)C2)=O)cc(C)c(C)cn1 N(C1CCNC(=O)c2[nH]ccc21)C(C(=O)Nc1cccc(F)c1[N+](=O)[O-])=O C=CCC(C(=O)NCC(C(=O)NCCC(=O)N(C)C)C1(C)CC1)OC C1(CNC(C(CC)CCOC)=O)CN(C(=O)CC(=O)OC)CC(C)(C)O1 Cc1nc2ccccc2cc1C=CC(=O)NCCN(C)C(C1CC1F)=O c1(OC)ccc(Cn2nc(-c3ccncc3)nc2CC(C)C(C)C)cc1 C1(CC)CCCC(N=c2cccc(S(=O)(=O)N3CCC(CSC)CC3)[nH]2)C1 c1(C(N(C2(C(=O)NC3CS(=O)(=O)C3)CC2)C)=O)ccc(=O)n(C)n1 CC1(C)CC(C)(C(N2CCC(C3CCCN3C(=O)CCc3cnoc3)C2)=O)C1 CCCC(C)C(=O)N1CC(O)CC1COc1cn(C)nc1-c1ccccc1OC c1(OCC(=O)NCC(C)(CO)NC(C(C)OC)=O)ccc2c(c1)CCCC2 c1(C(=O)NC(CCC)C(F)(F)F)cc2ccc(C(F)(F)F)cc2n1C c1(C(=O)NCCCN(C(CCN(CCCCC)C)=O)C(C)C)oc(C)nc1C N1(C(=O)CCn2ccnc2)CCCC(CCNC(C2(CO)CCOCC2)=O)CC1 c1(CC(=O)N(CCNC(C23CCCN(CC2)C3)=O)CC)ccc2c(c1)CCC2 C1(CC=C)(NC(c2cc(C3(C)CC3)on2)=O)CCN(C(c2ccnnc2C)=O)C1 c1(CCC(=O)NC(C(C)NC(c2sc(CC)c(C)c2)=O)(C)C)ccc(C)c(Cl)c1 CCC(C(=O)NCCOCC(=O)NCC(C)(C)CN(C)C)N(C)C C1(NC(CC2(C=C)CC2)=O)CN(C(c2cc(C3CC3)cc(F)c2)=O)CC1C1CC1 CC1CN(C(C2CCC(=O)NC2)=O)CCN1C(=O)CCc1cccc(N(C)C)c1 CCCCC(CNC(c1ccon1)=O)NC(=O)C(F)(F)CC1CCCO1 N1(C(C2C(CCC)C2)=O)CCCC(N(C(=O)Cc2ccccc2C(F)(F)F)C)C1 C1(C(N(CCCCNC(CCC=CC(C)C)=O)C)=O)CCCCN1C1CCCC1 C1(N(C(C2CCN(C(C(C)CC3CCCC3)=O)C2)=O)C)CC2CCC1O2 N1(C(C2CCC3CC23)=O)CCN(C(c2noc3c2CCCC3)=O)C2(CC2)C1 N1(C(c2ccnn2C2CCOCC2)=O)CCC(NCCOC2CCC2)CC1 N1(C(C(c2ccc(F)cc2)OC)=O)CCC(O)C(NC(=O)C2=CCOCC2)C1 C1(O)(CNC(CN(C(=O)Cc2coc(C)n2)CCC)=O)CC2CCC1O2 C1(O)(CNC(C2(CCCC)CC2)=O)CCN(C(=O)Cc2c(C)cnn2C)C1 C(=O)(C(C)(C)CNC(=O)C(Cc1ccoc1)N(C)C)NC(C=C)CO C1(CC)(NC(c2csc(C3CC3)n2)=O)CCN(C(C2CSCN2C)=O)CC1 c1(-n2c(-c3nccc(SC)c3)nc(C3CCCO3)n2)cccc2nc[nH]c12 CCC(C)C(CC(=O)N1CCC(N2CCCC2)C1)NC(=O)CCN1CCOC1=O c1(CN(C(C2C(C)C2C)=O)C2CC2)nc(Cl)ccc1F n1(CCC(=O)NCC2(CNC(COCC#C)=O)CC2)cnc2ccccc12 c1(C(N(C(C)CNC(C2CCC=CCCC2)=O)C)=O)cc2c(nc1N)CCC2 C1(C(N2CC(CC(=O)NCCNS(N)(=O)=O)(OC)C2)=O)CCCCC1(F)F C1(NC(C(CC=C)NC(C)=O)=O)CCN(C(=O)C(F)CC2CCC2)CC1CC c1(OC)cc(CNC2CN(C(c3cn(C)nc3C(F)(F)F)=O)CC2C)ccc1F C(=O)(C1=CC(C)(CC)C1)NCc1cn(CC(NOC(C(=O)OCC)(C)C)=O)nn1 N1(CC2N(CCCCCC)CCC2)CCC2(CC1)CC2C(N1CCOCCC1C)=O CC1CN(C(=O)C(N)=O)CC(CCNC(c2cccnc2SC(F)(F)F)=O)O1 C#CCC(C)(C)C(=O)NCC1CN(C(c2cnc(C)s2)=O)CC1O c1(C(C(=O)NC(c2ccccc2)CC)N(C)CCc2ccccn2)scnc1Br N1(C(C(=O)NCCCNC(=O)OC(C)(C)C)[Si](C)(C)C)CCC2(CC=CCO2)C1 n1(CC)nc(C(=O)N(C)CCN(C(=O)C(F)CC2CC2)C)c(Cl)c1Br c1(-c2cn(CCCCCC=C)nn2)cnc(OC)c(OC)c1 C1(NC(C2(C(F)(F)F)CC(=C)C2)=O)CN(C(=O)CN2CCCC2=O)CCC1CO c1(C(N2CCC(C(C)NC(C(CC)(F)F)=O)CC2)=O)ccc(P(C)(C)=O)cc1 CC1CCCCC1(CNC(=O)C=CC(N)=O)NC(=O)Cc1ccc(F)nc1 C(CCC)(C(O)C(=O)N1CC(C2=NOCC2)C1)NC(c1c(CCC)n[nH]c1)=O C(=O)(CS(=O)(=O)CC)N1CC2C(CNC(COC3(C#C)COC3)=O)C2C1 C1(NC(C(C2CC2)OC)=O)CC2(C1)CC(NC(C1CC(F)(F)C1(C)C)=O)C2 C(=O)(C(CCF)NC(c1cc(Cl)n(C)n1)=O)N1C(C(N(C)C)=O)CC1 c1(CC)ccc(C(C)CC(=O)NC(C)(C)CNC(=O)C(C)OCCC(C)C)cc1 Cc1cn(C)cc1C(=O)NC(C1CC1C(=O)NC(c1nc[nH]n1)CO)C C1(CC#C)CCCN1C(=O)C(CC1CC1)NC(=O)CC1COCCO1 N1(C(c2cc(C)cc(F)c2)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)C)C2 c1(OC)cnc(Cl)cc1C(=O)NCC1(CNC(C2CCCC(C(C)(C)C)C2)=O)CC1 C12(CNC(COCCCC)=O)CCCC1N(C(=O)C(C(C)C)n1ccnc1)CC2 c1(C(=O)NCCNC2CC(C)N(C3CC3)C2)c[nH]c2cc(F)ccc12 c1(C(=O)NC(CCOC)CNC(c2[nH]cnc2C)=O)cncc(C#N)c1 N1(C(c2cccc(C(C)(C)OCC)c2)=O)CCC(C(F)(F)F)(NC(=O)OC)CC1 CC(C#N)CCC(=O)N(C1CC(NC(=O)CCc2cscc2Br)C1)C C(N=c1[nH]c(N2CCC(=O)N(C)CC2)nc(=N)[nH]1)C1CCC(C)(CO)CC1 N1(CCNC(=O)C(=O)NC2CC(F)(F)C23CCC3)CCc2ccccc2C1 Cc1nc2c([nH]1)C(C(=O)NCCC(O)CNC(=O)CN1CCN(C)CC1)CCC2 N1(C(CC(C)C)=O)CCC(NC(=O)C(CO)NC(N)=O)CC1 S(=O)(=O)(CCCOC(=O)Nc1ccc(NC2CCC2)nc1)NC c1(C(N2C(CNC(c3c(CC)ocn3)=O)CC(O)C2)=O)nc(Br)n2ccccc12 c1(C(N(C)C)=O)cc(NCC2CC2)ccn1.C12CC(C1(C)C)CNC(=O)C(=O)N2 N1(C(c2c(C)nc(N)cn2)=O)CC2CC(NC(c3cc(C4CC4)cs3)=O)C(C2)C1 c1(C(C)NC(C=C(C)CNC(C2C(C)(C)C2(F)F)=O)=O)[nH]c(C)nc1C C(CCC(C)C(=O)N1CCC(C(=O)NCCCn2ccnc2C)(CC)CC1)OC C1(C(=O)NC(C)C(CO)NC(=O)C=Cc2cn(C)cn2)CC(F)(F)CCC1(C)C CCCCCC(O)C(=O)N(C)CC1COCCN1C(=O)CC1CCOC(CC)C1 N1(C(CC2CC(=C)C2)=O)CCSC(C(=O)NC(c2ccccn2)C)C1 C1(NC(C2CC(SC)C2)=O)C2CCCN(C(=O)CN3CC4CC4C3)C2C1(C)C c1(C(=O)NCCCCN(C(=O)CC2COC(=O)C2)C)cc(Cl)ns1 Cc1ccc(C=CC(=O)NC2CC(NC(C3(C)COC(=O)C3)=O)C2)cc1C C1(C(=O)NCc2c(CC)n[nH]c2)(NC(C2CC2(F)Cl)=O)CC(F)(F)C1 C(CC(C)C)(C(=O)NCC1CN(C(C2CC(O)(C(F)(F)F)C2)=O)C(C)(C)C1)OC Cc1ccc(CC(N2CCCC2C(C)NC(c2cnsn2)=O)=O)cc1 C(CCC(=O)NC1CCCC1CNC(c1coc(-c2cccnc2)n1)=O)SC N1(C(C2CCCN(C(C)C)C2)=O)CC2OCCN(C(=O)Cc3cc[nH]n3)C2C1 c1(C(C(C)(C)C)O)nc(-c2cscn2)nn1C1CCc2ccccc21 N1(CC(c2ccccc2)NC(S(C)(=O)=O)=O)CCCC(C2CCCC2)C1 C(=O)(C(O)C(F)(F)F)NC1(CNC(=O)C(=O)N2CCCC2)CCOC1 c1(C(N(C2CCN(C(C(C(CC)O)(F)F)=O)C2)CC)=O)cncc2nc(O)[nH]c12 N1(C(c2c(CC)nco2)=O)CC(C)(C)CC1C(N1CCC(n2ccnn2)C1)=O N1(C(c2c(C)nc(C)[nH]2)=O)CCCCC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)C1 C(CCC(C)C)(C(=O)NC1(C(C(CC2(CNC)CC2)C)=O)CCCC1)NC(C)=O c1(OC)cccc(S(=O)(=O)NC2CN(C(c3cc(Cl)ccc3C)=O)CC2C)c1 C=C(C)C(CC(=O)NC(C)CCN(C)C(C1(CC)CC1)=O)OCC C=CCC(C(=O)OCC)NC(=O)CC1CC1CNC(=O)CCCSC1CC1 c1(CC(N2CCC(c3cn(C(c4ccccc4)(C)C)nn3)C2)=O)ccc(Cl)nc1F N1(C(c2cc(OC)c(Cl)cc2)=O)CC2CCN(Cc3c(C)nn(C)c3C)C2C1 c1(C(=O)NC2(CO)CN(C(C3CCSCC3)=O)C2)onc2c1CCCC2 c1(OC)ccc(NC(=O)C(CCO)NS(=O)(=O)CC(C)F)c(OC)c1 c1(CC)ccc(O)c(C(=O)NCCCC(C)NC(=O)C(C2CCCCC2)F)c1 N1(C(CC2CCC(C)(C)O2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)CC1C1CC1 C1(C(C)=O)CC(CC(=O)NCCNC(=O)C(C)(C)Sc2ccc(C)cc2)C1(C)C N1(C(CCC(=O)NC)=O)CCC2C(CCCN2C(c2nc(C)nn2C)=O)C1 N1(C(C2C(C)CC(=O)N2)=O)CCc2sc(CNC(C3CN(C)C3)=O)nc2C1 c1(C(=O)OCCCOCCOCC)csc(C(=O)OC)n1 c1(C(c2ccc(OC)cc2)NC(=O)CSC(C)C)ncc(C(F)(F)F)cc1Cl C1(C(=O)NCc2c(C)ncs2)CN(C(=O)CCC(N)=O)CC1O C(=O)(CC(C)(O)COC)NC(CC)(C)CNC(=O)C(=O)NCCC(N)=O c1(CNC(CN(C(c2ccnnc2)=O)CC)=O)conc1C N1(C(C(C(CC)C)N(C)C(c2cccn2C)=O)=O)CCOCC(C)(F)C1 Cc1c(C(=O)NCC(CO)NC(=O)C(O)Cn2cncn2)cnn1C(C)C N1(C(Cn2ccc(C(=O)OC)n2)=O)CCCC(N(C)C(C2CCCCO2)=O)C1 c1(CC(=O)NCC(C2(O)CCN(C(CC=C=C)=O)C2)C)ccc2c(c1)CCOC2 O(NC(=O)CC(C)(C)N(C(=O)C=CCCC)C)CC(=C)Cl CCS(=O)(=O)CC(=O)N1CCC(CNC(C2CCCC2OC)=O)(OC)CC1 CC1CN(C(=O)C(C)(C)NC(c2ncn3c2CCC3)=O)CC(C)O1 c1(C2CCC(C)C2)nc(-c2ccccc2)nn1Cc1cccc(Br)c1 N1(C(CC2C(CC)C2)=O)CCN(C(CNC(=O)CO)C(F)(F)F)CC1 CC1(C)CC(C(O)CNC(=O)CCC2CCN(C(c3coc(C4CC4)n3)=O)C2)C1 N1(C(C2(C(=O)OCC)CC2)=O)CCC(C#N)(NCc2ccc(NC(C)=O)o2)C1 c1(-c2cn(CCN(C(C3(C)CCNC3=O)=O)CC)nn2)ccc2cnn(C)c2c1 CCCCC(O)C(=O)N1CCC2C(NC(C3(c4ccno4)CCC3)=O)C2C1 N1(C(C(C=C)(C)C)=O)CCC2CCC(C1)N2C(=O)C(C)=CC C1(CNC(C(C(=O)OC)OCC)=O)CC12CCN(C(c1cc(OC)no1)=O)CC2 N1(C(C2CC2COC)=O)CCCCC12CC(NC(=O)CC1C=CCC1)C2 N1(C(c2c(C)oc(CO)c2)=O)CCCN(C(c2cnn(C3CC3)c2)=O)C(CO)C1 c1(SC)nc(Cl)cc(=NC2CC3CC(C2)N(C(c2ncccc2N(C)C)=O)C3)[nH]1 N1(C(c2cn(-c3c(C)nccc3)nn2)=O)CCCS(=O)(=O)CC1c1cnn(C)c1 S(=O)(=O)(c1cccc2scnc12)N1CC2CN(Cc3cnn(C)c3Cl)CC2C1 C(CCSC)(C(=O)OC)N1CC(CC=C)(C(=O)NC2CCOCC2C)C1 C(=O)(CCCCCNC)N(C(C)C(=O)Nc1cnc(N(C)C)nc1)CC C1(NC(Cc2ncc(C)s2)=O)CCC(CNC(=O)C(c2c(C)noc2C)C)CC1 c1(C(N(C)CC2CCCN2C(C2CC2C(F)(F)F)=O)=O)ccc2c(c1)COC2=O C12(C(=O)NCC(C(=O)N(CC=C)CC3CC3)C)CC1CNC2=O c1(C(N2CC(OCC#C)C2)=O)cnccc1OC1CCCCC1n1cc(Br)cn1 C1(N(CCC(=O)N(CC#N)C2CC2)C(c2ccccc2)=O)CC2CCC1O2 C(=O)(CCC(C)(C)C#N)NCC(C(=O)NCCN(C1CC1)CC)(C)CC C1(NC(C(CC=CCC)C)=O)COC2CN(C(c3ccccc3N)=O)CC12 CC(C)(CC(=O)NCC1COCCO1)n1cc(CN2CCCC2)nn1 c1(NC2CN(c3nc(C)cc(OC)n3)CC2O)nc(C)nc2ccc(Br)cc12 N1(C(c2cccc(C(=O)NC)c2)C(=O)NCC(C)C)CCCCCC1C N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCCC(NC(=O)CNC(C)=O)C1 Cc1nc(CC(=O)NC2CCC(CNC(c3ccon3)=O)C2)cs1 c1(NCC(=O)NCC23C(CN(C(c4c(C)ncn4C)=O)C2)C3)cccc(F)c1F C(=O)(C(C1=Cc2ccc(OC)cc2OC1)N1CCCC1c1ccncn1)NCC C(CC(C(=O)NC(=O)CC1(c2ccccc2)CCCO1)SC)SC(F)(F)F c1(SCC(CC)NC(N2CCC(C(=O)OC)C2(C)C)=O)ccc(O)cc1F Cc1nnc2n1CCCN(C1CCOC(C3(C(F)(F)F)CCC3)C1)C2 c1(C(C(=O)NCC)N(C23CC(C2)C3)CC)cc(Cl)ccc1F C1(NC(Cc2c(CC)con2)=O)CC=C(C(=O)NCC#CCOC)C1 Cc1nc(S)sc1CC(=O)NCC1CC1NC(c1ccccc1C(C)(F)F)=O CCC(O)(CN(C(=O)C(Cc1ccccc1)n1cnnn1)C(C)=O)CC C1(C(N2CCOC3(CC3)C2)=O)C2CC(F)C(C2)N1C(c1ccccc1)=O N1(C(c2cccc(Br)c2O)=O)CCC2(CC1)CC2C(N1CCSCC1)=O N1(C(c2cnc(Cl)s2)C(=O)NC2CC(=O)N(C3CC3)C2)CCC(COCO)CC1 CCC(C)(Cl)CNC(C1COCC1COC)=O.C12(C=O)CSCC1C2 CN1C(=O)CCC1C(=O)NC(c1ccccc1)C(=O)Nc1ccc(OCF)cc1 c1(C(N(CC(O)CN(C2CC=C(C)CC2)C)C(C)=O)=O)c(C)cccc1Br c1(C(=O)NCC(CC)(C)NC(=O)CSc2nc(C)cc(C)n2)c(C)nn(C)c1Cl C(CCCCC(=O)N1CCC(CNC(C2OCCO2)=O)CC1)N(C)C C1(n2cc(-c3c(C(C)NC(C(C)CF)=O)cccc3)nn2)C2CC3C(C2)C13 Cc1cc(N2CCC(c3cc(N)ncn3)CC2)nc(=NCCC2(CO)CCC2)[nH]1 CC(C)C(C(=O)N1CCOC(CNC(c2cc(Br)n(C)n2)=O)C1)C(C)C N1(C(CC(CCC)(C)O)=O)CCCC2CN(C(=O)CCOC3CC3)CCC12 c1(OC)cc(C)c2cc(C(N3CCOC(Cc4ccccc4)C3)=O)[nH]c2c1 C1(C(=O)NC(C2(O)CCN(c3cc(-n4ccnc4)ncn3)C2)C)CCCCN1C n1(CCNC(C2CCC(O)C2)=O)ccc(C(=O)NCC2CC2CO)c1 Cc1ccc(C(=O)N(CC(=O)NCc2cnc(C)c(C)c2)C2CCC2)cc1O c1(C(=O)NC2CC3CC(NC(=O)CSC(F)(F)F)CC32)ccc2c(c1)OCCN2 C1(NC(c2c(C)snc2)=O)CN(C(C2(C(=O)OC(C)(C)C)CCCC2)=O)CC1C N1(C(CC(CC)NC(c2cnc(C)s2)=O)=O)CCCNC(=O)C1CC CC1(C)COCC1C(=O)NC1CC1CNC(=O)CCc1ccc(Br)nc1 Cn1c(NC(C23CC2CN(C(=O)Cc2ccno2)C3)=O)nnc1-c1ccccc1 C(=O)(NNC(=O)Cc1nc(C(O)C2(C3CCCCC3)CC2)no1)C1C(C)OCC1 C1(C(=O)NCC2C(NC(C(N3CCCCC3)C)=O)CCC2)COCCOC1 N1(C(CCC(=O)N(C)C)=O)CC23CCCC2(C1)CN(C(c1nc(=N)cc[nH]1)=O)C3 Cn1nc(-c2ccc(Cl)s2)cc1NC(C1CC1CNC(=O)C=CBr)=O C(=O)(C#CC(C)(C)CNC(=O)C(C)(O)C1CC1)NCC(COC)C(C)C c1(C(N2CC3C(CNC(C=C(CC)CC)=O)C3C2)=O)cc2ccc(Cl)c(F)c2[nH]1 C1(NC(c2cc(C)oc2)=O)CCC(NC(=O)COCc2ncnn2C)CC1 C(=O)(C1=CCC(C)CC1)N(C)CC1CCCN(C(c2c(CC)ccs2)=O)C1 N1(CC(=O)NCC2(OC)CCN(C(=O)C(C)N(C)C(C)=O)C2)CC(=O)N(C)C1=O CC1CCCN2C1CCNC(=O)C2=O.c1(NC(C2(C)CC2)=O)ccccc1Cl c1(NC2(CNC(c3c(Cl)nc(OC)s3)=O)CCC2)cc(C)c([N+](=O)[O-])cc1Br C1(Cc2cn(CC)nn2)CC(CC)CN(CCc2csc(C)n2)C1 C1(NC(c2c(C)csc2)=O)CC(CNC(C2(C)CCC(=O)N2)=O)C(O)C1 c1(CNC(c2cc[nH]c2)=O)ccc2c(c1)CCC2NC(=O)C#CC1CCCOC1 C1(N(C(=O)CSC(C)C)CCC)CCN(C(c2cncnc2C)=O)CC1 N1(C(c2cn(CC(N3CCCC3c3nc(O)n[nH]3)=O)nn2)=O)CCCC(CO)CC1 Cc1nnc(CC(N2CC(O)(CCNC(c3c[nH]cc3C)=O)C2)=O)s1 c1(CN(C(c2c(CC)onc2C)C(=O)NC)CC2CC2)cnc2ccccc2n1 C12C(C3CC3)CCN1C2=O.c1(CCNC(CCC)=O)ccncc1 Cc1nc(C(N2CCC2CNC(C2CCC3CC23)=O)=O)c(C)s1 C1(C(=O)NCC2(Cn3cc(C4CCOC4)nn3)CC23CCC3)CC2CCCC2C1 CC(=O)C(C)CC(C)C(=O)NCC1CCN(C(c2cccc(C)n2)=O)C1 n1(CC(=O)NC2(CC)CCCN(C(=O)COC(F)F)C2)cnc2ccccc12 CC(C)(CC(=O)N1CCCC(NC(C2CC(n3cccn3)C2)=O)C1)C(F)F CC(C)CC(C)C(=O)NC1COCC1NC(=O)COc1cccc(Br)c1 N1(C(CN(CCC)C)=O)CC(OC)C(OC)C1C(=O)NC1CCC(N(C)C)C1 N1(C(C(C)SCC)=O)CCC2CCN(C(=O)C=Cc3cncnc3O)C2C1 C(CCC(=O)NC(C)CNC(C1CC1Cc1ccccc1)=O)OC(C)=O C1(NC(c2n(C=C)ncc2)=O)CC2(CCCCN2C(C2CCN(C)C2C)=O)C1 c1(C(=O)CC2CN(N3CCN(C(CC(C)(C)SC)=O)CC3)C2)cnc2[nH]c(=N)sc2c1.N Cc1cc(N)cnc1C(=O)NCC(C1CC1)NC(=O)Cn1nnc(C(C)(C)C)n1 c1(C(C)C)ccc(C(C2CCN(C(=O)CCN3CCOCC3)CC2)O)cc1 N1(C(C#CC(C)C)=O)CCN(C(=O)CCC2CCC(O)CC2)C2(CC2)C1 c1(OCCC(=O)NC(CNC(C2(CCC=C)CC2)=O)CC)cccc(Cl)c1 C(=O)(C(C)CC(C)C(C)=O)NC(CCC)C(O)C(=O)N1CCCC(C)C1CO C=CC(O)(C(=O)N1CCOCC(NC(=O)CCCN(C)N=O)C1)C(F)(F)F C1(CC(=O)OC)CN(C(C2CCCOC2)C2CC2)C(C)(C)CO1 C1(CC(=O)NCCC(=C)C)CN(C(=O)CNC(C)=O)CCC1C CCCC(C)C(C(=O)Nc1ccccc1Cl)N1CCCC(NC(C)=O)C1 c1(NCC(N(C(=O)CC2CC2(Cl)Cl)C)C2CC2)nc2ccc(N)cc2s1 C1(C2CCCOC2)(NC(c2c(CNC(C3CC(CC)OCC3)=O)occ2)=O)CC1 CCCC(C(=O)NC)NC(C1CC(C)(NC(=O)CC2CCCC(=O)C2)C1)=O C1(NC(=O)C=CCN2CCCCC2)C=CCN(C(=O)C(O)C(F)F)C1 C1(F)(CNC(C2CC(=O)NCC2)=O)CCCN(C(C2(c3cnc[nH]3)CC2)=O)C1 c1(C(N2CCCC(NC(C(=O)N(C)C)=O)C2)=O)cc2n(n1)CC1(CC1)C2 CC(C)C(C(=O)N1CCCC1C1CCN(C(=O)CN2CCSCC2)CC1)C(C)C N1(C(C(C)NC=O)=O)CC(NC(=O)C=CC=Cc2ccccc2)CC(C)C1 c1(C(=O)NC2CC(F)(CNC(CN(C)CCO)=O)C2)ccc(Cl)cc1Cl C(=O)(C(CC(F)(F)F)c1ccc(Cl)cc1)N(C)CCNC(c1cccc(C#N)c1)=O n1(CC(N2C(C(C)NC(=O)CNC=O)CCC2)=O)ncn(C)c1=O C1(NC(C23CC(COC)(OC2)C3)=O)CN(C(=O)CN2CCC(C)CC2)CC1(C)C c1(C(N(CCCN(C(CC(C)C(F)F)=O)C)C)=O)cnc2cc[nH]c2c1 c1(C(N2CCCC(N(C(C(CC)NC(C)=O)=O)C)C2)=O)ccc(OC)cc1F N1(C(C(CC)CN(C)C)=O)CCC2(CC2)CC1C(=O)Nc1cnn2c1CCCC2 c1(C(=O)NCCC2CCN(C(C(CCCOC)C)=O)C2)cc2cnccc2[nH]1 N1(C(CC2N(C(c3ncc(OC)nc3)=O)CCCC2)=O)CC(C)(C)OCC1(C)C C(CCC(=O)NC1(CNC(c2cnn(-c3cccnc3)c2)=O)CCOC1)N(C)C C1(C)(CNC(C(C2CCN(C(c3nccs3)=O)C2)C)=O)CCCOC1 c1(C(N2CC(CNC(C(C)SCC)=O)C(C)C2)=O)c(O)nnc2c1CCC2 c1(C(=O)NC2CN(C(c3c(Br)cn(CC)n3)=O)CC2C)sc(C)c(C)c1C c1(N(CCCNC(=S)NCc2cccnc2)C)ccc(F)c(Cl)c1F C(=O)(CC(C)(C)CC(C)=O)N1C(CN(C(C=CCC)=O)C)COCC1 C(=O)(C#CC1CCOCC1)NCCOC1CN(C(c2ccc(C(N)=O)[nH]2)=O)C1 N1CCCC(O)C1.c1(NC(=O)C(F)F)cccc(C2(C(C(C)(C)C)=O)CCCC2)c1 Cn1cnnc1CCC(=O)N(CCCNC(C1(C(F)(F)F)CCC1)=O)C1CC1 CCC(C)(C(=O)NCCOC1CCN(C(=O)CCC(C)NC(C)C)C1)N(C)C S(=O)(=O)(c1ccsc1C(=O)OC)NCCC(CCC)N c1(C(=O)NC(CC2CN(C(C=COCC)=O)C2)C)nn(C)c2c1CC(F)(F)CC2 c1(C(N2CCC(C(CNC(COC)=O)(C)O)CC2)=O)c(C)cccc1[N+](=O)[O-] N1(C)CCC2CN(OC)CC12.c1(SCC)cc(C(=O)NC)ccc1N N1(C(CSCCCC)=O)CC(CNC(=O)C(C)OC)C2(CCC2)C1 C1(C(N(CCn2cc(C(C)SC)nn2)C)=O)CC(N(C)C)CCN1C(=O)C(C)C CC1(C)CC(NC(=O)COCC(F)(F)F)CN1C(c1cncc(-n2cccc2)c1)=O c1(C2(C(=O)NC3C(CNC(C(C)C#N)=O)CC3)CC2)ccc(Cl)cc1 C1(CNC(c2cnc(C)[nH]2)=O)CC2CCCC2N1C(c1cn(C2CCC2)nn1)=O C1(C(N(CCN(CC)CC)C)=O)CCC(C)N(C(c2csc(Cl)c2)=O)C1 Nc1cc2c(cc1C(=O)NC1CCCCCN(C(C3CCSCC3)=O)C1)CCC2 c1(C(N(C)CCOCc2nccs2)=O)cnc(N(C)C)c(Br)c1 N1(C(c2c(SC)nn(C)c2)=O)CCC2(NC(c3cncc(C)n3)=O)CCCCC12 C1(NC(c2c(C)c(N)ccc2)=O)CCN(C(=O)CCN(C)CCO)CC1(F)F C1(O)(CCNC(CCc2ccc(C)o2)=O)CCN(C(=O)CC2CCC(O)C2)C1 N1(C(C(C)NS(CC)(=O)=O)=O)Cc2ccccc2C(NC(=O)C(N)=O)C1 c1(CC(=O)NCC(CNC(=O)CCc2ncc[nH]2)OC)ccc(F)c(Cl)c1F C1(C(N(CCC)CCCc2ccc(OC)cc2)=O)CCC2C1C2(F)F N1(C(C23N(C(c4c(COC)cco4)=O)CC(C)(C2)C3)=O)CCCC(N=[N+]=[N-])C1 C1(NC(C=CCCC)=O)CCN(C(=O)C(=O)NCC(F)F)C1 C(=O)(NNC(=O)CC(C)(C)n1cnnn1)NC1CC1C(=O)OC(C)(C)C c1(CNC(CSc2nnc(C)o2)=O)cccc(NC(=O)CNC(C2CC2C)=O)c1 N1(CCC(C)(C)NC2C(C)CCCC(C)(C)C2)C(=O)c2ccccc2C1=O N1(C(=O)CN2CC=CC2)CCC2C(CCCN2C(=O)CC2CC2)C1 c1(C(=O)NC(C(=O)N(C)Cc2cccs2)C2CCCC2)cc(CCO)on1 c1(C(=O)NCC(CC(C)C)NC(c2c[nH]cc2Br)=O)ccnc2ccsc12 CC(C)CC(=O)C(=O)NCC1(C(N2CCCCC2C2CC2)=O)CC2(CC2)C1 C1(NC(CS(N)(=O)=O)=O)CCCC(NC(c2ccc(OC(F)F)nc2)=O)CC1 Cc1ccc(C=CC(N2CCC(O)(C(C)CNC(C3(C)C=CCCC3)=O)C2)=O)o1 N1(C(C2CC(C3CC3)C2)=O)CCC2CCCC12C(=O)NCCC1CC1 c1(C(=O)NC(C)CCNC(=O)CC2COCCO2)ccccc1C(C)(C)C c1(NC(C2(C3N(C(CCC(=C)Cl)=O)CCC3)CC2)=O)cc(Cl)ccc1CC CC1C2CCC(C2)C1C(=O)NC1(C(=O)NC2CC2c2cc[nH]n2)CCN(C)C1 N1(c2n(C)c(-c3ccccc3C#N)nn2)CCN(C(=O)NCCSCCO)CC1C C(=O)(CCCC(CC)CC)NC1CCN(C(COCC)=O)CC1 C1(C(C)C(=O)NCc2ccccn2)CN(C)CCN1C(=O)Cn1ccnn1 C=CCCCCCCC(=O)NC(C)(C)CCCNC(C1CCCC(F)C1)=O C12(CCC1)C(=O)N2.CCC(C1CC1)N(C)C(C1CC1C(N)=O)=O C1(NC(C2(C)COC2)=O)CS(=O)(=O)CC1C(=O)NCc1cc(C2(C)CC2)n[nH]1 N1(C(c2c(COC)cco2)=O)CC2CC1C2C(=O)Nc1ccc(C(C)=O)cc1 Cc1cc(=NC(C)c2c(Cl)ccc(F)c2Cl)[nH]c(NCC2C3COCC23)n1 c1(SC)cc(C(N2CC3CC(NC(=O)CC4C=CCC4)C2C3)=O)ccc1N N1(C(c2cc(C)on2)=O)C2CCC1C(C)C(NC(c1ccoc1Br)=O)C2 c1(C(N(C(C(=O)N(C(C=C)C2CC2)C)C)CCC)=O)cnoc1 N(S(=O)(=O)N1CC(C(=O)O)C(C(=O)O)CC1(C)C)(CCCC)CC C(C)(c1ccco1)=CC(=O)NCC(COC)NC(=O)C=CC1CC1 CC1=C(C(=O)NC(C)CN(C(=O)C(C)C)C)Cn2nnnc2N1C C#CC12CCC(C(=O)NCCNC(c3c(F)c(F)cc(F)c3F)=O)(CC1)CC2 c1(OC)cc(S(=O)(=O)NC(=O)C(N)C2CC2)c(Cl)cc1Cl c1(C(=O)NC2C(C)(CNC(C3(OCC)CCC3)=O)CCC2)cc2n(n1)CC(F)C2 C(C)(C(=O)NCC=CC(=O)NC(c1ncc[nH]1)C)NC(C)=O CC1CCN(C(=O)C(=O)NCC(C(C)(C)C)NC(c2nc(Cl)cs2)=O)CC1 C1(NC(c2cc(C(C)=O)[nH]n2)=O)CCC(NC(=O)COC2CCCCC2C)CC1 C#Cc1ccc(C(N2CCCCC2C(=O)NC2C=CCCC2)=O)cn1 C1(CNC(C(C)OCCCC)=O)CN(C(=O)C=CSC)CC12CCC2 c1(C(N2C(CNC(c3ccc(SC)o3)=O)C(C)CC2)=O)nc(O)nc(O)c1N C(CCCC(C)(C)C)NC(CCC(C)NC(=O)C(C)C#N)=O C1(CNC(CC2C(=O)NC(=N)S2)=O)CC2(CCN(C(=O)CC3CC3)CC2)CO1 c1(C(N2CCC(NC(c3ccc(C#N)s3)=O)C2)=O)cc2c(F)cccc2[nH]1 NC1CCN(C(c2cc(C(=O)O)ccc2I)=O)CC12CCC2 C(CCCC(CO)NC(=O)CC1CCC(F)(F)C1)NC(=O)COCC1CCCC1 c1(C(N2CC(C)C(CNC(c3cc(CF)on3)=O)C2)=O)cc(O)nc(Cl)c1 c1(C(N2CCC(C(N3CCCC3)=O)C2)=O)ccc(Cl)cc1.c12ccc(cc1)NC2 c1(C(N2CCC3(NC(C4CC5(C4)CC(F)C5)=O)C(C2)C3)=O)cccc2cncn12 CC(C)C(CCNC(c1cc(CO)[nH]n1)=O)NC(C1(Cl)CC1(C)C)=O CC1=C(C(=O)NCc2cncc(C(N3CC(CNC)C(O)C3)=O)c2)CCO1 CCCCCC(C)CC(=O)N1C2CCC1CC(NC(C1(COC)CCCC1)=O)C2 C(c1ccc(Cl)s1)=CC(=O)NC(CCNC(C1N(C(=O)OC(C)C)CCC1)=O)C C1(C(=O)NC2CN(C(C(c3cncnc3)C)=O)C2)CCC(=O)N1CCC(F)(F)F CON1CCC(C(=O)NCCC2CN(C(c3cc4n(n3)CCC4)=O)C2)CC1 C1(C(N(c2cc(C(F)(F)F)ccn2)CCC)=O)CCc2ccccc2N1C(=O)OC C#Cc1ccc(CC(=O)N(C(CNC(C2CNC(=O)C2)=O)CC)C)c(F)c1 c1(N(C(c2c(CCC)n[nH]c2)=O)C(C2CCOC2=O)=O)ncc(C(F)(F)F)cc1Cl N1(C(C(C(C)C)NC(=O)OC)=O)CCCN(C(c2sc(F)cc2C)=O)CC1 c1(C(=O)NC2CC(NC(C(CC(C)C)O)=O)C2)cc(C(F)(F)F)ccc1[N+](=O)[O-] C1(N(C)C(c2c[nH]ccc2=O)=O)CN(C(=O)C(O)C(F)F)CC12CC2 S(=O)(=O)(c1ccc(C#N)cc1)N1CCCC(NCc2c(C)nn(C)c2Cl)CC1 N1(C(C2(NC(=O)CCCC3CC3C)C(C)CCC2)=O)CCOC2(CC2)C1 c1(C(=O)NCC(CC=C)NC(C2C=CC=CC=C2)=O)cc(C)c(N)cc1F C12(C(=O)NC(CCCC)CO)COCC1CN(Cc1cc(C)no1)C2 C1(C(N(CCCSC)C)=O)CCOCCN1C(C1CC(C)C1)=O c1(OC)cc(C)c(C(=O)NC(C)CCNC(=O)C(c2cccc(C)c2)O)cn1 c1(C(=O)NCC2CC3CC3N2C(c2sccc2F)=O)cc2cc(Cl)ccc2o1 c1(C(=O)NC(C2CN(C(=O)C(C)(C)C(C)O)C2)C)cc(C#N)[nH]c1C C1(C(=O)NC(C)C(C)SC)(SC)CN(C(=O)C(C)OCCC(C)C)C1 c1(NC(c2nnnn2C(C)C(=O)OC)CCSC)nc2c(Cl)c(Cl)ccc2s1 C1(CCNC(=O)CC2CC(F)(F)C2)CCCN(c2nc(C3CCCCC3)ns2)C1 N1(C(CN2CCC(OC)C2)=O)CCC2(C=C(C(=O)N3CC4CC3C4)C2)C1 C1(C2CC2)(NC(Cc2c(C)noc2Cl)=O)CCN(C(=O)CCC(C)OC(C)C)C1 C(c1ccc(Cl)cc1)=C(C(=O)NCCOCCNC(C(CC1CC1)OC)=O)C C1(CNC(N2CCC2C2CC2)=O)CCC1Nc1cccs1 C1(C(=O)OC)CC2OCCC2N(C(c2ccc(NCc3ccccc3)cc2)=O)C1 C1(C(=O)O)(CF)CCN(C(C2CCCC3CC23)=O)C1.c1(C(=O)N)ccc(C(F)F)nc1 C(CC(=O)NCC(C)N(CCC(C)C)C)N(C(CNC(=O)OC)=O)CCO N1(C(CC(C)NC(C2CCCC2)=O)=O)CCN(C(=O)Cn2cnnn2)C2(CCC2)C1 C(=O)(C(O)C(F)(F)F)NC1(CNC(C2CCN(C(C)=O)C2)=O)CCCC1 N1(CC)CCN(C(=O)C(N2CCC(CC)(CN)C2)=O)CC1 C(=O)(C1CCc2nnc(C)n21)N1CC2(C(NC(CC=C)=O)CCC2)C1 C(CCCNC(=O)CC(C)C1CC1)(c1ccccc1)NC(C=CCCC)=O C1(NC(C2CCCC2)=O)COCC1n1cc(-c2ccn(CC(F)F)n2)nn1 N1(C(c2c(C)nccc2)=O)CCC(O)(C2(NC(=O)CSC3CC3)CC2)CC1 C1(NC(C=NOC)=O)CN(C(C2CC(=O)N(C(C)C)C2)=O)CC1n1ccnn1 N1(C(CC(CC)(F)F)=O)CCC2(CCOC2)C(CNC(c2cocc2C)=O)C1 c1(C(N(C(C(C)N(C(CC)(C)C)C(C)(C)C)=O)CC)=O)ncnn1C C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NCC1(O)CN(C(c2c(C)snn2)=O)C1 CC(C)CC(C(=O)N1CCCC1CCC(=O)NC(c1nc(=O)o[nH]1)C)N(C)C CCC(C)C(C)(O)CNC(=O)C(F)C1CC(NC(c2cncc(C)c2)=O)C1 c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC(C)C(C)OC C1(NC(C(C(C)C)C)=O)C(C)(C)CN(C(c2ccc(C(C)(C)C)s2)=O)CC1(C)C CC1CC(CCNc2c(F)cccc2Cl)CC(C)C1 C1(C2CC2)(C(N2CC(CNC(COC(CC)C)=O)C(C)C2)=O)CC=CC1 C1(C(=O)NCc2nc(C(=O)N(C(C)C(=O)N(C)C)C)c(C)o2)(CC)CCCCC1 c1(OC)cccc2cc(C(=O)NCc3ccnn3C(C)C)oc12 c1(OC)ccnc(F)c1C(=O)NCC1CCC(C)N(C(c2ccnc(O)c2)=O)C1 CCCC(C)CC(=O)N1CC=CC(NC(c2c[nH]nc2C(C)(C)C)=O)C1 Cc1cc(C)c(C(N2CCCCC(CCC(=O)NCCOC3CC3)C2)=O)cn1 C1(C(=O)NCC(C)NC(=O)C(C)NC(=O)OC(C)(C)C)C2CCCCCC12 c1(C(=O)NC2C(CNC(C(C(C)(C)C)O)=O)CC2)ccc2nc(O)[nH]c2c1 C12(CNC(c3cc(COC)on3)=O)CCC1CN(C(=O)C(F)(F)c1nccs1)C2 C(=O)(C(C)(F)C(C)(C)F)N1CCCC(N(C(c2ccc(CC)c(Cl)c2)=O)C)CC1 CCC(C)C(C)C(=O)NC1(C(=O)NC(C)(C)CCCN(C)C)CCN(C)C1 n1(CC)cc(CN(C(=O)C(CC2CCC2)NC(C2CCCO2)=O)C)cn1 CC1CCN(C(C2(C)CCSCC2)=O)CCN1C(=O)Cc1ccc2n[nH]cc2c1 O=C1CC(C(=O)NC2CN(C(c3cccnn3)=O)CC2n2ccnn2)CCN1 C(CN=C(NC1(C)CCC1)NC1CC1CC(C)C)c1c(OC)cccc1 CCCCC(C)(c1nnnn1CC(F)F)NC(CC(C)(C)C)c1ccccc1 CN1CCC(C)(C(N2CCC(C)(CCNC(=O)CC3CCC3)C2)=O)C1 C1(CNC(c2ccc(N(C)C)cc2)=O)CC(F)(F)CN1C(=O)C(F)OC(F)(F)F CCCCC(=O)N1CCCC1C(C)NC(=O)C(C)SCC C1(CCNC(C(C2CC2)NC(c2cn(CC)nn2)=O)=O)OCCC1(C)C c1(C(=O)NCCC(C)NC(CC2ON=C(CC)C2)=O)c[nH]c2c(Cl)cccc12 C1(C(C(C=CCN(C)C)=O)=O)CC(CCN)C1.C(=O)C=CI C1(C(N2CCC(NC(CNC(c3c(C)onc3)=O)=O)C2)=O)CCC(C)CC1 C1(NC(C(COCC)NC(C23CCC(CC2)CO3)=O)=O)CCCOC12CCC2 c1(C(N2C(CNC(c3ccc(C)nc3N)=O)CCC2)=O)c[nH]nc1S(N)(=O)=O N1(C(CSCC=C)=O)CCN(C(=O)CSC2CCOC2=O)CC1C1CC1 N1(CCC(CC)SC)CC2CC(C)N(C(=O)C(CC(C)C)C(N)=O)C2C1 c1(OC)cc(CN2CCC(F)(F)C(C(=O)Nc3cnnc(Cl)c3)C2)cc(Cl)c1O C1(CNC(=O)CC(F)(F)F)CC2CCC1N2C(C1(F)CCOCC1)=O c1(C(N2CC(NC(c3c(CC)n(C)nn3)=O)C(C)CC2)=O)cnc2[nH]cnc2c1 c1(C(N2C(CCCNC(C(C)SC)=O)CCC2)=O)nc(SC)n2ccccc12 C(=O)(CC1CCC(C)(C)c2ccccc21)NC(C(C)(C)OC)C C1(NC(CC(C)c2cccnc2)=O)CCCOC12CCN(C(=O)CCC#N)CC2 CCC(C)(F)C(=O)NCCN(C(=O)C(C)SC(C)C)C c1(C(=O)NC23C(CN(C(C(C)OC)=O)C2)CCCC3)ccc(N=S(C)(C)=O)cc1 c1(C(C(=O)NCC(CO)NC(COCC(C)C)=O)F)ccc(F)cc1 Cc1[nH]nc(CNC(=O)CNC(=O)Cn2ccnn2)c1C C1(C(N2CCC(C(C)OC(CCC)C(=O)NCC)CC2)=O)CC2COCC2C1 c1(CC(=O)N(CCC(C)O)CC)c(C)[nH]c2ccc(Br)cc12 N1(C(C2C(CCC)CN(C(=O)CC3OCCO3)C2)=O)CCOCC(C)C1 C1(C(N2CC(NC(c3oc(CC)c(C)c3)=O)C(C)C2)=O)CC2OC(C)(C)OC2C1 CCCC(CC(C)C)C(=O)NCCOCCN(C(=O)C#CC1CCCCC1)C.NCC n1(CC)cnc2nc(N(CCCSC)C)nc(N3CC(C)C(F)(F)C3)c12 c1(-c2cccc(C(C)=O)c2)c(C)nc2c(OCc3ccccc3)cccn12 N12CCC(CO)(CC1)C(c1ccccc1)C1SCCC(C1)C2=O.C1(CO)CC1 c1(NC2C(CC)CCC2)ncc(S(=O)(=O)NC2CCn3ccnc32)cc1Cl C1(C(=O)NCCCOCCC(=O)NCc2onc(CC)n2)CCC(C)CC1 C1(c2cn(CC(C)NC(C3(C)CCCN3C)=O)nn2)CCC=CCCC1 c1(CCC(=O)OCC(=O)N(C(CC)(C)C)C)cc([N+](=O)[O-])n[nH]1 CN1CCCCC(CNC(=O)CC2CC2CNC(=O)CC2C(=O)NN=C2C)C1=O N1(C(c2nc(C)oc2)=O)CCCC2CC(NC(=O)CC3OCCC3(C)C)CCC12 c1(C(=O)OC(C#C)CC2CCCO2)cccc(OCC2CC2)c1 c1(C(N2CCC(N(CCC)C(c3c(C)noc3C)=O)C2)=O)cc(F)c(O)c(F)c1 C12(NC(c3ccc(NC)cc3)=O)CCC(CC1)N(C(=O)CS(=O)(=O)CCO)C2 C(=O)(CCC(C)CC)NCc1c(C(=O)NC(CCCC)CO)n[nH]c1 C(=O)(C(O)C(F)(F)F)N(CC(CC)NC(=O)C(C)(C)c1ccccc1)CC CCC(C(=O)NC(C)(C)CC(=O)NC(CF)C(F)(F)F)C(F)(F)F C1(NC(c2c(CC)noc2)=O)CC2C1CCN2C(=O)COCCOCCO CCCCC(O)CC(=O)NC1CC2CCC(C1)N2C(c1csc(NC(C)=O)n1)=O CC1=C(C(=O)NCC2CCC3CN(C(=O)Cc4csnc4C)CC23)CCCC1 N1(C(c2cnn(CCCC)c2CC)=O)CCC2(CCCN2C(=O)C=CC2CC2)C1 Cc1ccc(C(=O)NC2CCCC(CN=c3[nH]nco3)C2)nc1 C1(N(C)C(=O)C2CC2)(CC)CCN(c2nc(Cl)c(-c3nn[nH]n3)s2)C1 S(=O)(=O)(CC(=O)NC(CNC(C1(F)CCC(C(=O)OC(C)=O)C1)=O)CO)NCC c1(N2CC(NC(C(CCCC)ON=C(C)C)=O)C2)ncccc1S(=O)(=O)CC C1(C(=O)OC)(CC)CCCCN1C(C1C(C)(C)C1(C)C)=O C1(NC(C(C)N(C(C)=O)C)=O)CCC2(CCN(C(=O)C(c3cnn(C)c3)C)C2)C1 C(C(C)(C)C(=O)NCc1ccc(C#N)s1)N(C(C(SC)SC)=O)C CC(CC(C)N(C(=O)C(F)(F)C1CC1)C)NC(=O)C(F)OC(F)(F)F c1(C(=O)NCC(CC=C)NC(c2c(CO)n[nH]c2C)=O)ccc(N)c([N+](=O)[O-])c1 C(=O)(CCC(CC)NC(=O)CC(C)CCC)NCCC=CC=C C1(CC=C)(NC(C2CC2F)=O)CCN(C(c2cnc(OC)c(Br)c2)=O)C1 N1(C(C(C(CC)C)OC)=O)CCC2(CC1)CC(NC(=O)C(C)C)CCO2 N1(C(=O)Cn2ncnn2)CCN(C(C2CC2(Cl)Cl)=O)C2CCC12 Cc1ccc(CSCC(=O)NC2(CO)CN(C(C3CC3C(N)=O)=O)C2)cc1 N1(C(CCN(C(C2CC2C(F)(F)F)=O)CC)=O)CCC(C(=O)OC)C1 C1(C(N(C2CCCNC2=O)C)=O)C2CC3C(C2NC(=O)CCc2cnn(C)c2)C13 C1(C(=O)NCC(=C)CCNC(C2CC(CC(C)(C)C)C2)=O)CCN(C)C(=O)C1 C1(CC(=O)N(C(CC)C(=O)NC(c2nncs2)C)C)COCCOC1 C(=O)(CCCC)N(CCOCCC=C)C.C(=O)(CCC=CC)N N1(C(C2N(C(CC(C)C)=O)CCCC2)=O)CC=C(CNC(=O)C(C)C2CC2)CC1 CC(C)(C)CCCCC(=O)NCC1CC(NC(c2ccnc(OCCO)c2)=O)C1 C(=O)(CC(C)(C)COC)OC.C(=O)(C(C(=O)O)OC)N(c1cccc(C)c1)C1CC1 N1(C(c2c(C)ccnc2O)=O)CC2CCN(C(=O)CC3CC4CC4C3)CCC2C1 CCC(C)(C)C(O)C(=O)N1CCCCC(NC(C2CCOCC2(C)C)=O)C1 C1(C(N2CC(F)(C(=O)OC)C2)=O)C(C)CCN1C(=O)C(C(C)OC)N(C)C CCC(CC)C(CNC(C1(c2nn[nH]n2)CCCOC1)=O)OC N1(C(c2c(CC)n(C)nn2)=O)CC(CNC(=O)CN2CCCNC2=O)CC(C)C1 CCCC(C)CC(=O)NCC1CC(C(F)(F)F)CN1C(C1CC(F)(F)C1)=O CCC1=C(C(=O)NC2CCC2NC(C2CC(C3CCOCC3)=NO2)=O)CCCO1 C1(C(=O)NCc2cccc(C(N(CC(F)(F)F)CC)=O)c2)CC(=O)NC(=O)N1 c1(C(C)C)ccc(C(=O)NCC(C)(C2CC2)NC(=O)C2=CCSC2)cc1[N+](=O)[O-] Cc1c(C(N2CC(CNC(=O)Cn3ccnn3)C(C)C2)=O)sc2ncnc(N)c12 c1(C(=O)NCCN(C)C(C2(C3CC3)CCCO2)=O)cccc(-c2cccnc2)c1 C(=O)(C(C)(C)C(O)CC)N(C1CCN(C(=O)CC=C(Cl)Cl)C1)CC Cc1c(F)cc(C(=O)NCC2CCN(C(c3ccc(C#N)cc3)=O)C2)cc1F N1(C(CNC(CCC)=O)=O)CC2CC(C(N3CC(C)(C#N)C3)=O)C(C2)C1 c1(C(=O)NCC(CN(C(C(C=C)c2ccccc2)=O)C)O)cccc(COC)c1 N1(C(C(C=C)NC(=O)CC(C)N(C)C)=O)CC2CC2(CC)C1 n1(CC)nc(CCCNC(N2CC3COC(C2)C3O)=O)c2ccccc12 C1(C)(C(=O)NCC2(O)CN(C(CN(C)C(=O)OC(C)(C)C)=O)C2)CCCC1C N1(Cc2cccc(OC)c2Cl)CC2CCN(C(c3ccc4cccnn34)=O)C2C1 CCCCC(O)CC(=O)N(C1CCN(C(=O)C=CC2(C)CCOCC2)C1)C CC(C)CC(F)C(=O)NC1CCCCCC1NC(=O)CC(=O)N(C)C C1(C2(NC(CN(C3CCCC3)C)=O)CC2)CCCN1C(=O)CC1(C)CC1(F)Cl C(=O)(C(C)(C)CC(F)F)NC1CC(C)CN(C(C2(C(N)=O)CCC2)=O)C1 c1(C(c2nnnn2-c2ccccc2)NC(c2ccccc2F)CC)cc(C)ccn1 C(=O)(C(O)C(C(C)C)OC)N(C1(c2cn(CCCC)nn2)CCOCC1)C1CC1 C1(COC)(CNC(=O)CC(=O)N(C)C)CN(C(c2ccon2)=O)C1 N1(C(C(CC)=CC)=O)CCC(NC(c2ccc(N3CCOCC3)nc2)=O)C(F)C1 Cc1nccn2ncc(C(=O)NCCCc3cc(F)cc(F)c3)c12 CC1=C(c2ccco2)CN(CC2CCCC2C(F)(F)F)CC1 N1(C(CC(=C)C)=O)CCCC1(C)CNC(c1cn(CCC(C)C)nn1)=O C#CCCCCCC(=O)NCC1CCN(C(c2cnn(CCO)c2)=O)C1 c1(C(=O)NCC2(NC(c3cnn(C)c3N)=O)CCOCC2)cnn2c1CCC2 N#Cc1cccc(S(=O)(=O)N2CCCCC2C(=O)N=c2[nH][nH]cc2C)c1 C1(NS(=O)(=O)CC2CCCC(F)C2)CC2(CCC2)C1 CCC(CC(=O)NC1CCN(C(c2nscc2Br)=O)C1C(C)C)OC N1(C(C2(C)CCSCC2)=O)CC2CCN(C(=O)CCCN3CCOC3=O)C2C1 C1(O)(COC)CCN(C(=O)C(C2CC2)NC(c2cc(F)c[nH]2)=O)C1 CC1C(NC(=O)C(O)CC2CCCCC2)CCCN1C(C1COCCO1)=O N1(C(c2cnc(C)s2)=O)CCCOC(CNC(c2ncccc2C(F)F)=O)C1 CC(N=c1[nH]c2c(c(=NCCN(CC(F)(F)F)C)[nH]1)CCCC2)C1CCOC1 CCC(CC)(C(=O)N(C)CC=CC(N1CC(C)(O)C1)=O)C(C)C c1(NC(C)=O)cccc(CNC(C2CCN(C(=O)CC(F)(F)F)CC2)=O)c1 C(=O)(CCCCCCSCCOCC)N1CCC(NC(C2(OCC)CCC2)=O)C1 c1(C(C)C(=O)NCC2CN(C(=O)COC(N)=O)C(C)(C)C2)ccc2c(c1)OCO2 C1(NC(=O)CC2CC=CC2)CC2CN(C(c3ccc4sncc4c3)=O)CC2C1 c1(C(=O)NCC2C(CNC(c3ccc(O)nc3Cl)=O)C2)cc(Cl)c(F)cc1F c1(C(N2CC(CNC(C=CCN(C)C)=O)C2)=O)cn2c(n1)COCC2 c1(C(=O)NC(CC2CCN(C(c3c(C)ocn3)=O)CC2)C)cc(O)c(F)cc1N N1(C(C2C(C)=C2)=O)CCCCC(CNC(=O)CCn2cc[nH]c(=O)c2=O)C1 CCCC(CCC)C(=O)NC1CCC(N(C(=O)Cc2cc(C)cs2)C)C1 c1(C2N(C(C)C(=O)N(C)C)CC2(C)C)ccnc(Cl)c1 CC1CCN(CC(=O)NC(CNC(=O)CSc2ccc(O)cc2)CO)CC1 C1(NC(C(CC)C)=O)CCCC12CCN(C(c1cc(O)ccc1Br)=O)CC2 C1(NC(CC(C)n2cccn2)=O)CC2CCC(C1)N2C(C1CC2C(C1)C2(F)F)=O Cc1c(NC(C2CN(C(c3cnc(Cl)nc3)=O)C2)=O)cccc1O c1(N(CC(C)NC(C(CCCC)(C)F)=O)C)ncnc2onc(C)c12 C1(NC(C(C)N(C(c2cn(C(C)C)nn2)=O)CC)=O)CCC(OC)CC1 CC1(C)C(C(N2CCC(NC(=O)CNC(c3ccncc3)=O)C2)=O)CCS1(=O)=O CC12CCN(CC1)CC2C(=O)NCC(O)CNC(=O)CSCC(N)=O C1(CNC(=O)Cc2nc[nH]n2)CC(C(F)(F)F)CN1C(c1cnco1)=O C1(NC(C2(SC)CN(C(=O)CNC(C)=O)C2)=O)COCC(C)O1 Cc1cc(C(=O)NC2CCCN(C(C3CCCCO3)=O)C2)c2[nH]cnc2c1 N1(C(c2cc(C)nc(O)n2)=O)CCC(C2CCN(C(=O)CC(O)C3CC3)CC2)C1 C1(CNC(=O)C(F)CC2CCOC2)CN(C(C2CCCSC2)=O)CCCO1 C(=O)(C(c1ccc(F)cc1)=CCN)N(C(C)C(c1ccc(Cl)cc1)=O)C N1(C(CCCNC(=O)CCn2ccnc2)=O)CCOC(C)C1.c1(C=O)ccncc1 C1(C(=O)NCC(C)(O)CNC(C2CN(C3CCC3)C2)=O)(CC)CCNC1=O C1(F)(CNC(c2cc(OC)n[nH]2)=O)CCN(C(=O)CC2CC2(C)C)C1 C1(C(=O)NCCN(C(=O)Cc2c(Br)cnn2C)C(C)C)CCN(C)C(=O)C1 N1(C(C2C(C)C2)=O)CCC(F)(CNC(c2cccc(CC(F)(F)F)c2)=O)CC1 C1(C(=O)NCC2N(C(C3N(C)CC(O)C3)=O)CCOC2)CN2CCC1CC2 CC1(C)COCC(C(=O)NCC2(C)CCN(C(=O)C3=CCCO3)C2)O1 c12c(sc(C)c1C)NCC1CCCN1C2=O.C(C(=O)N(C(C)=O)C1CC1)SC c1(C(=O)NCCOC2CN(C(C34CSCC3C4)=O)C2)ccnc(CO)c1 C1(CNC(c2cc(Cl)sc2Cl)=O)CC2CCC1N2C(c1ncccn1)=O Cc1ccc(C(C)C)c(NC(C2CCC(C)N(C(=O)CCNC(=O)CO)C2)=O)c1 c1(C(=O)NCC2N(C(C3C(C(=O)OC)CCCC3)=O)CC2)cn2cccnc2n1 CC1(C)CN(C(C2CCCCCC2)=O)CC1CNC(=O)CSc1ccccn1 C1(NC(CC(C)n2ccnc2)=O)CC(NC(=O)CN2CC3C=CC2C3)C1(C)C c1(C(=O)NCCCCN(C)C2CC2)ccc(CNC(c2cccnc2)=O)nc1 C1(N(C)C(c2cc(C(N)=O)[nH]n2)=O)CN(C(c2ccnc(Cl)c2)=O)CC12CC2 N1(C(c2c(C)ocn2)=O)CCN(C(C2(CC(C)C)CCCC2)=O)CC12CCC2 N1(C(C(C)NC(C)(C)C)=O)CCC(NC(c2ccccc2CO)=O)C(C)(C)C1 N1(c2nc(C)nc(C(C)C)c2)CCN(C(=O)C2=CCCCC2)CC(C)(F)C1 C1(NC(CC(C)(F)F)=O)CCN(C(c2c[nH]cc2C(F)(F)F)=O)CC1(C)C c1(OCCC)c(C)cc(-c2cnc(NC(=O)CCN(C)C)c(O)c2)cc1C c1(OC)ncc(C=CC(N2CCC(CNC(=O)CCn3ccnc3)CC2)=O)cn1 C1(C(=O)NC(CC=C)CNC(=O)CCc2cc(C)no2)CC12CCCCC2 C1(C(C)NC(C(C)C2CCOC2)=O)CCCN(C(c2nncs2)=O)C1 C1(C(N(CCOC)CCc2ccncc2)=O)CCCC2CCCN12 c1(C(N2C3CC(NC(=O)CCSC4CCCC4)(C3)C2)=O)occ2c1CCCC2 c1(C(N2CCC(N(CCC)C(c3cncn3C)=O)C2)=O)n[nH]c(CC)c1C CCCCC(C)CCC(=O)NCC1(F)CCCN(C(C2(C#N)CCCC2)=O)CC1 c1(C(=O)NCCC2CCN(C(c3ccn(COC)n3)=O)C2)ccc2nn[nH]c2c1 C(C1=CCN(C(C2CC(OCC)C2)=O)CC1)NC(CC(C=C)C)=O N1(CCc2cn(C(C(=O)OC)C)nn2)CC2CCN(c3ccc(Cl)cc3)C2C1 C1(CC(C(=O)OCC)F)(NC(c2ccc(C)c(Cl)c2)=O)CCCCCC1 N1(C(CNC(CCC)=O)=O)CC2CC1(CNC(c1cccc(CC(C)C)c1)=O)C2 C1(C)(C(N(CCC(C)NC(=O)C(C)(C)CF)C)=O)CNC(=O)C1 c1(C(=O)NCC(C23CCC(CC2)C3)NC(=O)CC2CC2)cc2ccc(F)cc2s1 N1(C(C(C(C(C)C)OC)O)=O)CCC2(C1)CN(C(=O)COC1CCOC1)C2 c12ccc(cc1)NS(=O)(=O)C2.c1(NC2CC3CNC2C3)ccc(Cl)cc1 C1(O)(C(=O)NCc2cn(CCC)nn2)CCN(C(C2CC(OC)C2)=O)CC1 N1(C(c2nccc(C)n2)=O)CC(CNC(c2n[nH]c(C)n2)=O)OC(C)(C)C1 c1(C(=O)NC2CCCC(C(=O)N3CC(O)CO3)C2)ccc2c[nH]nc2c1 C1(C(N(CC(CC)NC(C2(C)CCOCC2)=O)C)=O)CC2(C1)CC(O)C2 CCCCC(CC)C(=O)N1CC2CCC(CNC(C3SCCS3)=O)C2C1 c1(C(N2CC(C(C)NC(=O)C(C)(Cl)Cl)C2)=O)cccc2c1CCC(=O)N2 CC(C)P(=O)(CC(=O)N(CC(O)CN(C)C(c1cnc(S)n1C)=O)C)C(C)C c1(C(N2CC(C)(NC(C(COC)O)=O)C2)=O)c(C)cc(C)nc1S CC(C)(C(=O)NCCC(=O)NC1(C2CCCO2)CC1)C1(O)CCC1 CCCCCCCC(F)C(=O)N1CC(CNC(=O)C(C)=C(C)CC)CC1(C)C C1(NC(CN(C)C2CC2)=O)CN(C(=O)CNC(C2CC(C)(C)C2)=O)CC1(C)C c1(C(=O)NC2CC(CCNC(C3CCC(C)(C)C3)=O)C2)cnn2c1CCC2 N1(C(C2CC(=O)C2)=O)CCC2(CCC2)C(NC(=O)Cc2cnccn2)C1 C1(C(N2C(CNC(=O)C(F)CC3CC3)CCCCC2)=O)C2CCC3C(C2)CC13 N1(C(C2C(C(=O)OC)(CC)C2)=O)CCC(C(C)NC(=O)CC(C)(C)SC)CC1 c1(NC(=O)NC(C(F)(F)F)c2ccccc2)cccc([N+](=O)[O-])c1 c1(C(N2C(C(N3CC(n4cccn4)C3)=O)CC2)=O)ccnnc1O C=CC1(C(=O)NCCC2CC2C2CC2)CCN(C(=O)C(=O)CC(C)C)C1 N1(C(CC2C(C)(C)CC2)=O)CCC2C(C1)CN2C(c1ccc(C(F)F)c(F)c1)=O C(=O)(CC(C(F)(F)F)n1ccnc1)NCCN(C(CC(C)(C)SC)=O)C(C)C c1(C(=O)Nc2cccc(NC(CS(C)(=O)=O)=O)c2)cccc2nccnc12 C(CCCCC(=O)NC1CCN(C(c2cn[nH]c2)=O)CC1CC)OCC N(C1CCCc2cc(CNC(C3(C)CCC3)=O)ccc21)C(CC(C)(C)OC)=O C=CCC(CNC(=O)CC(C)NC(C)=O)NC(=O)C=CSC C1(C(N2C3(C)CC3CC2)=O)CCC2CCC1N2C(=O)CCCc1cnn[nH]1 N1(C(c2cc(C)sc2)=O)CCN(C(=O)CCN2CCC(F)C2)CC12CC2 c1(OCC)ccc(CNC2CCCCCC2c2ccccc2)c(Cl)c1O N1(C(CC(C)C2CCCO2)=O)CCC=C(CNC(C2CC(=O)NC2(C)C)=O)C1 CCC(C(=O)OC)C(=O)NC1CCN(C(=O)CC2CCC(=O)NC2=O)CC1C c1(C(N2CCCC(C)(NC(CC(C)C(C)(C)C)=O)C2)=O)nn(C)c2c1COCC2 N1(C(C2C(CC)CCCC2)=O)CCCC(NCCOC)C1c1ccccc1 C1(C(=O)OC)CC2CCC1N(C(c1c(Br)ncn1C)C(=O)NC1CCCCC1)C2 N#Cc1cncnc1C(=O)NCC1CC(CNC(=O)C=C2CCCC2)CO1 C1(C2CC2)(CNC(C2CC(C)(C)C2)=O)CCN(C(c2cc(Cl)cc(F)c2N)=O)C1 C#CCC(C)(C)C(=O)N(CC(O)CN(C)C(c1cnc[nH]1)=O)C O=C(C#CC1CC1)NCC(O)CNC(=O)CC(c1ccccc1)n1ccnn1.C1(C)CC1 c1(C(N(C2CCN(C(=O)CC3CCC(O)C3O)CC2)CCOC)=O)cc(C)cnn1 c1(C(N2CCC(CNC(COC)=O)CC2)=O)cc(Cl)c(F)cc1O Cc1cc2[nH]c(C(=O)NC3CC(C)N(C(=O)C(C#N)=CC4CC4)C3)cc2s1 Cc1cn2ccnc(C(=O)NCC(O)CCNC(=O)C3=COCCC3)c2n1 C1(NC(c2cccc(F)c2)=O)CC2CC1CN(C(c1coc3ccccc13)=O)C2 CC1CN(C(C2(F)CC=CCC2)=O)CC1c1cn(CCNS(C)(=O)=O)nn1 C(C)(c1ccccc1C)=CC(=O)NCC1N(C(C2CC(CC)C2)=O)C2CCC1C2 CC(CNC(c1ccsc1)=O)(CO)NC(=O)CCCNC(N)=O Cc1c(C(=O)NCCC2CCN(C(=O)CCS(C)(=O)=O)CC2)nn2c1CCCC2 C1(CNC(C(C)CN(C)C(C2(C)COC(=O)N2)=O)=O)CCC2(CC2)CO1 C1(C(=O)NCC(CN(C(C2(CCC)CC2)=O)C)C)CC(C)(C)OC(C)(C)C1 Cc1ncoc1C(=O)NCc1cn(CCCC)nn1.N1(CC2CC2)CC1 N1(C(CCCOC)=O)CCCC(NC(c2oc(SC)cc2C)=O)C1C C1(C(N(CCN2CCN(C(CCC(C)OC)=O)CC2)C)=O)CC2CCCC(C1)C2 c1(CC)ccc(C(=O)NC23CCC2CN(C(=O)COCC2CC2)C3)cc1N Nc1cc(C(=O)N(C2CC(NC(=O)CN3CCOCC3)C2)CCO)cc(O)c1 N1(Cc2c(OC)ccc(C)c2)CCC2(CCN(C(=O)CN3CCCS3(=O)=O)C2)C1 N1(C(N2CC=CC(C(=O)N(C3CCCC3)Cc3ccco3)C2)=O)CCC2CC1CO2 C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1(C)CCCN(C(C(C(=C)Cl)(C)C)=O)C1 N1(C(C(C)OC(C)(C)C)=O)CC=C(C(=O)NCC2(C)CCCC(=O)N2)CC1 Cc1cccc(-c2cccc(C3(NC(c4ncncc4I)=O)CCC3)c2)c1 c1(C(=O)NC(c2ccccc2F)CNC(CC2C(C)OCC2)=O)cc(F)cc(Cl)c1 C(=O)(C1=CC(C)(CC)C1)NC(c1ccccc1)CNC(CN(CC)SCC1CC1)=O c1(CC(=O)NC2CC(C)(NC(=O)CC(F)F)C2)ccc(Br)cc1[N+](=O)[O-] C1(O)(C(N(CCCCN(C(c2nn(CC)c(O)c2)=O)C)C)=O)CCCC(C)(C)C1 C1(Nc2nccc(C)n2)CCN(C(c2c(C)cccc2C)=O)CC1O c1(C(N2CC(COC)N(C(=O)Cc3nnc(C)s3)CC2)=O)c(Cl)ccc(F)c1C C1(NC(C(C(COC)C)C)=O)CC2CCC(C1)N2C(c1csnn1)C CC(CC(=O)N1CCCC1C1(CNC(=O)COCc2ccsn2)CC1)N(C)C O=C(CC(O)C(Cl)(Cl)Cl)NC1(C2CN(C(C3COCCOC3)=O)C2)CC1 C1(C(=O)NCc2ncccc2O)CC=CCN1C(=O)CC1CCC=CCC1 N1(C(c2cn(CC)nn2)=O)CCCC12CCCN(C(=O)CC1C=CCC1)C2 C1(C2CC2)(NC(C2=CCN(C(C3CCCC(C#N)C3)=O)C2)=O)CCCCC1 C1(F)(C(=O)OC)CCN(c2nnc(-c3cc(C)[nH]n3)n2CC2CCCCO2)C1 N1(C(C2C(OCC)CC2)=O)CCC2(CCC2NC(c2nc(=O)n(C)[nH]2)=O)CC1 c1(OC)ccccc1C(N1CCCCC1CCNC(c1ccoc1Br)=O)=O c1(OCC(C)(C)C)ccc(C(=O)NCCC(C)(C)NC(C2CC(O)C2)=O)cc1 c1(C(N2C(CCNC(c3c(C)ccs3)=O)CSCC2)=O)ccc(F)c(C(C)C)c1 CCC(C)(C)C(O)C(=O)N1CC2(CC2)CC1CNC(=O)Cc1ncc(Cl)s1 C(=O)(C(F)CC(C)(C)NC(=O)OC(C)(C)C)Nc1c(C)ccnn1 c1(C(=O)NC2C(NC(C(CCC)NC(C)=O)=O)COCC2)nc2cnccc2s1 CCCCC(C)(F)C(=O)NC1CCCC1C(=O)NCCc1cscn1 c1(C(=O)NC2(CNC(c3ccc(Cl)c(Cl)c3)=O)CC2)ccc2nc(Cl)nn2c1 C(=O)(C(C)(O)C(F)(F)F)NCC1(C)CN(c2nccc(SC)n2)C1 CCCC(F)C(=O)NC(Cn1ccnn1)C(N1CCCC(CN(C)C)C1)=O Cc1cc(Br)cc(C(=O)NCC2(NC(c3cncn3C)=O)CC2)c1C c1(C(C2(C)CC2)OC)nc2ccccc2[nH]1.C123CC(C1)(C2)C(=O)OC3=O c1(OCCOC)ccccc1CNC(C1C=CCN1C(=O)C(CO)OC)=O C1(NC2CC2)CC2CN(C(=O)C3=C(Cl)CC3)CC12.CC1(C)CNC1=O C1(CNC(C=CC(CC)=CC)=O)CC(C)N(C(c2cc[n+]([O-])cc2)=O)C1 N1(c2cc(NCc3c(F)ccc(C)c3)nc(C)n2)C2CCC1CC(F)C2 C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CCCC2CC12)NCC1CC(SC)C1 O=C(N=c1ccc(O)n[nH]1)Nc1snnc1C1CCC1 CC(C(=O)NCCN(C(c1ccsc1)=O)C1CC1)C(C)n1cccn1 N1(C(c2cc(C)sc2)=O)CCC2(CCN(C(c3cc(C#N)cn3C)=O)C2)C1 c1(C(=O)NCCCN(C(=O)Cn2cccn2)C2CC2)cccc2oc(O)nc12 c1(CC)nc(C(=O)NC2CC(C(C)NC(c3cnc(C(N)=O)s3)=O)C2)co1 Cc1nc(C(=O)N(C(C)CNC(C2(c3ccccc3)CC2)=O)C)c2n1CCCC2 N1(C(Cc2ccc(C)o2)=O)CC2(CCCC2)C1C(N1CC(C)(O)C1)=O C1(NC(CCCC#C)=O)CCN(C(=O)C=C(C)c2ccsc2)CC1O C12(C(C)NC(C3C(C(C)NC(C4CC(=C)C4)=O)C3)=O)CCC(CC1)C2 c12cc(ccc1Br)C(=O)N2.C1(COC)(NC(=O)OC(C)(C)C)CC=CC1 c1(CC2CCN(C(C3(OC(CC4CC(OC)C4)=O)CC3)=O)C2)ccc(F)c(Cl)c1 N1(C(c2nnn(CC)c2C)=O)CCN(C(=O)C=CCOCCOC)CC1C Cc1c(CNC(=O)C(C)CNC(=O)CC(C)CN(C)C)cnn1C Cc1cc(F)c(C(=O)NCc2ccc(C(N3CCOC(CO)C3)=O)s2)c(Br)c1 Cc1c(Br)ccc(CNC(=O)C(=O)NCCS(=O)(=O)CCO)c1I c1(C(=O)NC(CC=C)C(=O)NCC2CCOCC2)c[nH]c2ccncc12 C1(C)(NC(C(C(=O)OC)C)=O)CCC(NC(c2ccc(C)o2)=O)CC1 c1(C(N2CC(C(C)NC(C3(CC=C)CCC3)=O)C2)=O)cnn(CCOC)c1C C(=O)(CCS(N)(=O)=O)N(CCCNC(CCCOCCOC)=O)C(C)C C1(C(=O)NC(C(=O)N(CCCC(C)C)C)Cn2cccn2)COCCC1C N1(CC(=O)NC(c2ccsc2)C)CC2CCC1CN2C(=O)C(c1ccccc1)F N1(C(c2nn(CC)c(O)c2)=O)CCN(C(=O)CCCn2ccnn2)C2CCC12 C1(C(=O)NC(C(=O)NCCC)CC)CC2(C1)CC21CCC1 n1(C(C)C)c(SCC(N2C(CNC(C)C(=O)O)CC2)=O)nc2ccccc12 c1(C(N2CCC(NC(c3cc([N+](=O)[O-])cs3)=O)C2)=O)cnc(Cl)c(F)c1 c1(C(N2CC(F)(F)CC2CC(N)=O)C(=O)NC)cn2cc(F)ccc2n1 N1(C(C2C(COC)CC2)=O)C(C(=O)NCCCCC2CCCC2)CC1C N1(C(C)=O)CCCN(S(=O)(=O)c2cccnc2NCc2nocc2Br)CC1(C)C C1(C(=O)NC(C)CN(C(=O)Cc2cnn(C(C)(C)C)c2)C)CCCC12CC2 S(=O)(=O)(c1cccs1)NC1C(C)CN(C(=O)CCC(=O)NC(F)(F)F)C1 c1(C(N2CCC(NC(C=C(COC)C)=O)CC2)=O)cc(Br)ccc1N c1(C(=O)NCc2ccc(C(F)(F)F)o2)cc2n(c1)CCN(CC)C2 c1(C(=O)NC(C(C)NC(c2cc(Cl)ncc2O)=O)C)cccc2nc(O)n(C)c12 C1(O)(C(C)CNC(c2cocn2)=O)CCN(C(=O)CCOc2ccccc2O)C1 C1(NC(c2cccc[n+]2[O-])=O)C2CCC1N(C(=O)C1=CCC1)C2 N1(C(=O)Cc2ncsc2Cl)CC2(CCN(C(c3c(F)cccc3F)=O)CC2)C1 Cc1cc(O)nc(SCC(=O)NC2CCC(N(C(=O)CC(C)F)C)CC2)c1C#N C1(C(N2CCC(C(C)NC(c3c(CC)n(C)nc3)=O)CC2)=O)CC2CCC(C1)O2 c1(N2CC3C(NC(C(CC)(C)C)=O)C3C2)nc(C)c(C#N)cc1Cl c1(C(CNC(c2ccc(C(=O)OCC)cc2)=O)O)c(C)nn(C)c1Cl C1(CC(=O)NC2(CN(C(=O)C(C)(C)C)C)CC2)CCCC(=O)N1 N1(C(C=C(C)Cl)=O)CCN(C(C2CCCN2N=O)=O)C2COCC12 c1(CC)cn2c(C(N3CC=CC(NC(=O)C(COC)N(C)C)C3)=O)cccc2n1 N1(CCNC(c2nccc(=N)[nH]2)C)CCC(c2ncco2)CC1 c1(OC)cnc(F)c(C(=O)NCC(C)(CO)NC(=O)CC2CC3(CC3)CO2)c1 N1(c2nnc(C)s2)CC2C3CCC(C2C1)N(C(=O)CCCC1CCOCC1)C3 c1(SC(C)C)ccc(C(=O)NCCOCCNC(=O)CSS(C)(=O)=O)cc1 N1(C(=O)NCc2nnc(CC)s2)CCC(CC(O)C(F)(F)F)CC1 C12(CNC(C3CCN(C(CCSC)=O)C3)=O)CC(CN1C)C2 c1(C(N2CC(NC(C3CC(OC)C3)=O)C(SC)C2)=O)cc(C)c(C)nc1C C1(NC(C2(C)CCCS2)=O)COC2CN(C(C3(c4cccc(Cl)c4)CC3)=O)CC12 C1(OC(N2CC(C(C)NC(=O)CSCCCc3ccccc3)C2)=O)CCCOC1 CCCCC(C)CCC(=O)NCC1COCCN1C(c1cc2nnn(C)c2s1)=O c1(C(=O)NC(CN(C(CSCCOC)=O)C)C)cnc(OCC(F)(F)F)c(C)c1 C1(C(N2CCC(N(C(=O)CCc3cncs3)CC#C)CC2)=O)CCCCC(=O)C1 C(=O)(C#CC1CCCCO1)N1CCN(C(CNC(c2ccns2)=O)=O)CC1 C1(C(N(C(C2CCCCC2)CO)C)=O)CC(F)(F)CN1C(c1cncn1C)=O CCC(CCOC)C(=O)NC1CC(OCC(=O)NC(C)C(C)F)C1 N12CCOC(C1)CN(C)CC2=O.c1(C(=O)O)ccn(CCN2CCCCC2)n1 N1(C(C2(F)CN(C(C3CC(CC#C)C3)=O)C2)=O)CCCC(C#C)CC1 c1(C(=O)NC2C(CC(=O)N(CCN(CC)CC)C)CCCC2)cc(C)nc(C)c1 CC1(F)CN(C(c2nc(O)[nH]c(=O)n2)=O)CCN(C(=O)CCC2CCOC2)C1 c1(-c2cc(CNC(CC(C)C)CCO)on2)cc(F)c(O)c(F)c1 c1(C(=O)NCC2N(C(C(C=CC)O)=O)CC(F)C2)ccncc1N=[N+]=[N-] C1(C(=O)NCC2(OC)CCCCC2)CCN(C(=O)C2=NOC(C)C2C)C12CCC2 C12(C(=O)NCC3CC(F)(CNC(=O)C=C4CCOCC4)C3)CCCCC1C2(F)F S(=O)(=O)(CCC(=O)NCC1C(C)CCN1C(=O)C(O)COC)NC C1(C(=O)NC2(CNC(=O)CCc3ccccc3Cl)CC2)Cc2cc(Cl)ccc2O1 c1(CC)cc(CC(N2CCCC2CCNC(=O)CC2(OCC)CCC2)=O)n(C)n1 N1(C(c2cc(C(N)=O)[nH]n2)=O)CC(NC(=O)CC2CCOC2)C2(CC2)C1 c1(CNC(c2ncn(CC)c2)=O)cnn(C)c1C(=O)NC(c1ccccc1)CC CC1CCC(C(=O)NCc2cccc(NC(=O)Cc3cncn3C)c2)C(=O)N1 CN1CC(NC(=O)NCC2CN(CC(F)(F)F)C2)CC1=O c1(SCC(NOC)=O)ccc(-c2cn(-c3cnc(OCC)cn3)nn2)cc1 CC(CC(=O)N(CC(F)F)C)C(C)(C)NC(=O)C(c1cnn(C)c1)C c1(C(=O)Nc2ccc(C(=O)NCCC(CSC)OC)cn2)ccc2c(n1)CCC2 C(CCCCC(=O)NCC12CC(CO1)N(C(c1cc3sccc3s1)=O)C2)OC c1(CCC(=O)NC(CNC(COCCOCC#C)=O)(C)CO)cccc(C)c1 c1(C(=O)NC2CC(C(N3CCN(CC(C)C)CC3)=O)C2)cccc2ccccc12 C(=O)(CC1=Cc2ccccc2C1)N1CCN(C(C2N(C)CCC2)=O)C(C2CC2)C1 N1(C(C(C(C)C)O)=O)CC2CC(NC(=O)C(C)(C)n3ccc(C4CC4)n3)C2C1 S(=O)(=O)(c1cc2sc(=NC3COCC3C)[nH]c2cc1Cl)NC(CCCC)(C)C Cc1nccn1CCNC(C1CC(C)N1C(=O)Cn1cc(CO)nn1)=O c1(C(=O)NC2(CNC(c3cc(C(=O)OC)on3)=O)CCC2)cccc(Cl)c1Cl c1(C(=O)NC(C)CC2CN(C(c3cccc(F)c3Cl)=O)C2)cc(Cl)ccc1F C=CCCCC(C(=O)NCC1CC2CCC2C1)NC(=O)C(C)N=[N+]=[N-] c1(NC(C2CC(=C)CN2C(c2nc(C3CC3)cs2)=O)=O)ccc(Br)c(Br)c1 CC(C)(C)C(C#N)C(=O)NC(C(N1CC(O)(C2CC2)C1)=O)C1(O)CCC1 C(c1cccnc1)=C(C(=O)NC(C(C)NC(CNC(=O)OC)=O)CO)C c1(NC)cncc(C(=O)NCCC(O)CNC(=O)CNC(=O)CCC(C)C)c1 C1(NC(c2c(OC)nsc2)=O)C(C)CN(C(c2cc(Br)ccn2)=O)CC1C Cc1cc(C(=O)NCC2CCCCC2NC(C2CC23CCCCC3)=O)nc(C)n1 n1(C(C)C)c(SC(F)(F)F)nc2ccccc12.c12cn(nn1)CC(F)CCNC2 C12(C(N3CC(CC)OCC3)=O)CC(C)(CN1C(c1c(C)ncnc1C)=O)C2 N1(C(C2N(C(CSCC)=O)CCC(F)C2)=O)CCn2cc(C)nc2C1 c1(C(=O)NCC2C(C)(C)C(NC(=O)CCNC(N)=O)C2)cccc(O)c1Cl c1(-c2nc(-c3ccc(OC)cc3)nn2-c2ccc(O)c(F)c2)ccc(Cl)cc1Cl c1(N2CC(CN(C(c3c(C)cns3)=O)C)OCC2)ncnc2onc(C)c12 C(CNC(=O)CCCC1CCC1)(CC(=O)N(c1ccsc1)C)OC C(=O)(C1=C(CCCCl)N(c2cccc(F)c2)C(=S)NC1c1cc(C)[nH]n1)OCC Cc1ccc(C(C)N(C2C(NC(=O)CC#N)CCC2)C)cc1 c1(-c2ccc(C)cc2)csc2ncn(-c3cccc(C(C)C)n3)c(=O)c12 S(=O)(=O)(CCN=C(NC1CCOCC1)NC12CC(C1)C2)N1CC(C)OC(C)C1 c1(C(N(C(CNC(C(COC)O)=O)C)C)=O)cc(S(=O)(=O)N(C)C)oc1C C1(CNC(C2(C(=O)OC)CCCC2)=O)CCCCN1C(=O)Cc1cnsc1 N1(C(C(C)O)=O)CCCC(CCNC(c2ccc(C3CC3)cn2)=O)C1 c1(CNC(C(CCSC)N(C(C)COC)CC(C)C)=O)ccc(Cl)c(Cl)c1 CN1C(=O)CCC1C(=O)NCC=CC(=O)NC1CC(CO)C1(C)C N1(c2nc(C)nc3c2CCC3)CCc2cc(ON3CCC(C#N)C3)ccc2C1.CN(CC#N)CC c12ncccc1C(=O)NC2.CC1CCCC1CC(=O)N(CC)CC1CNC(=O)C1 C1(NC(C=CC)=O)C2CCN(C(c3ccc4cnoc4c3)=O)CCC12 c1(C(N2CC(OCCNC(c3cc(C)[nH]n3)=O)C2)=O)cc2c(C)cccn2n1 c1(C(N(CC(C)CNC(=O)C(C)C2CCCC2)C)=O)cnc2ccnn2c1O c1(OCC(=O)NCC(CN(C)C(c2cccc(Cl)c2N)=O)O)ccc(F)c(Cl)c1 N1(C(C=C(C)C(F)(F)C(F)(F)F)=O)CCC2(CC1)CC(CNC(C1CC1Cl)=O)C2 C1(O)(CNC(C(C=CC)O)=O)CC2CCC(C1)N2C(c1ncccc1C(F)F)=O c1(C(=O)NC2CCCN(C(C(CC=C)C)=O)CCC2)c[nH]c2ccc(OC)cc12 C=CC(C)(O)CC(=O)N1CC2CC2(CNC(=O)Cn2cncc2C(=O)OC)C1 C1(NC(C2CC(C)=C(C)CC2)=O)CN(C(c2coc(Br)c2)=O)CC2(CC2)C1 CC1(C)Cc2ccc(C(=O)NCCNc3ncc4cc(Cl)ccn34)cc2O1 Cc1cc(OC(C)C(N2CCCC(N(C)C(c3ccncc3)=O)C2)=O)cc(C)c1 c1(C(=O)NCC(CC)NC(c2occc2Cl)=O)ccc(N(C)C)c(F)c1 C(=O)(CC(COC)NC(C1(C(C)(C)OCC)CC1)=O)NCCSCC#C C#CC(Cc1ccc(F)cc1)N(C)N(C)C1CCS(=O)(=O)CC1.C(C)(C)C N1(C(C(CSC)OC)=O)CC(CNC(c2ccc(CC(C)C)cc2)=O)CC1C CCC(C)C(=O)NCC(=O)NC1(C(=O)NC(C)C(C)(C)O)CCCC1 C(=O)(C(CCC(C)C)OC)NCC(CCOC)NC(c1cnc(OC)c(C)c1)=O c1(C(N2CC(CNC(CCC(=O)NC)=O)C2)=O)ccc(OC)c(Cl)n1 CC1(C)CC(CC(N2CC(OCCNC(C3CC4(CCCC4)C3)=O)C2)=O)CCO1 c1(C(=O)OC)ccc(-c2nn3cc2COC3)cc1.N1(CC)CCC(C)C1 c1(N(C)CC2(C)CCCC2)nc(N2CCCC(C3CC3)CC2)nc2ccsc12 c1(C(N2C(CNC(C3(C(C)C)COC3)=O)CC3(CC3)C2)=O)cc[nH]c2nccc1-2 c1(C2C(CNC(C(CN(C)C)N)=O)C2)ccc(F)cc1 CN1CCCC1CC(=O)NC1(CCNC(C2(N(C)C)CC2)=O)CC1 O=C(C1CCc2nccn21)NCC1(CNC(C2CC23CCOCC3)=O)CCC1 C1(C(=O)NC2CN(C(CCCOC)=O)C(C)CC2)Cc2cncn2C(=O)N1 C1(C(=O)NCCC2N(C(C(CC(N)=O)O)=O)CCOC2)CCc2nnc(O)n2C1 C(=O)(C#CC1CCCCO1)N1C2C(NC(c3nc(OC)cc(OC)n3)=O)C(C2)C1 CC1COC(CNC(c2ccc(CNC(C3CC(CC4CC4)C3)=O)o2)=O)C1 Cc1c(CN2CC(=O)N(CC3CC3(C)C)C2=O)sc2cncn12 CC1CN(C(=O)Cn2ccnn2)CCN1C(C1CCCCCC1C)=O c1(C(=O)NCCCCC)ccoc1CNC(=O)CCNC(N)=O C1(NC(C2N(C(CC(=O)NCC)=O)CC(F)(F)C2)=O)CN(C)C(=O)C12CC2 C#CCC(CC(F)F)C(=O)N1CCC(C(=O)NCC2CC3CCC3C2)C1C(C)C C1(NC(CC2CC(NC(C(C)c3cccs3)=O)C2)=O)CC(F)(F)C1(C)C C(=O)(C(=O)N=c1cc(-c2cn(C)nc2C)o[nH]1)Nc1cccc(OCOC)c1 C(C1CN(C(C2(C)CC(OC)C2)=O)CC1C(N1CCSC(C)CC1)=O)=CC n1(CC)ncc([N+](=O)[O-])c1C(=O)NCC1(O)CN(C(=O)Cc2cc(OC)cs2)C1 N1(C(C2CCN(C(CC)=O)C2)=O)CCC(CO)(CNC(c2ccc[nH]2)=O)C1 N1(C(c2cc(C(C)=O)oc2C)=O)CCC2CN(C(=O)CC3CC4(CC4)C3)C2C1 N1(C(C(C)Cn2cccn2)=O)CCn2nc(C(=O)O)cc2C1.C12(CC1)C(=O)N2 C1(C2CC2)(NC(CC(CCC)C)=O)CCN(C(=O)CSc2nncn2C(C)C)C1 N1(C(c2n(CC)nc(C)c2)=O)CC=C(CC(=O)NC2CCN(C(C)(C)C)C2)CC1 c1(OC)cc(F)c(-c2cn(C(c3nc(C(C)O)n[nH]3)C)nn2)c(F)c1 c1(C(=O)NCCCCCNC(COCCC=C)=O)cncc(C)c1Cl N1(C(C(CCC)NC(C2CC=CC2)=O)=O)CC2CC(CO)C(C2)C1 CCCCCC(C)(C)CNC(=O)C(C1CCN(C(C2CCC(CC)CC2)=O)C1)C C#CCC(C)(C(=O)N1CCN(C2CC2)C(C)C1)NC(c1cc(C(C)C)no1)=O C1(NC(C(C2CCOCC2)OC)=O)C(CN=c2[nH]ncs2)CCC12CCC2 c1(C(N2C(CNC(C(CC)COC)=O)CC2)=O)c2ccc(Br)cc2nn1C c1(CC(=O)NCCC(C)NC(C(F)OC)=O)cccc([N+](=O)[O-])c1Cl c1(CC(=O)NC(c2cn(CC3CC(=O)N(C)C3)nn2)CCC)cc(F)cc(Br)c1 N#Cc1ccc(C(N2CCC(C(F)C(=O)N(CCO)CC3CC3)C2)=O)nc1 C1(O)(CC(=O)NCC2CC(C)N(C(c3cn(C)[nH]c3=N)=O)C2)CCCCCC1 c1(C(=O)NC(CN(C(C(=O)OCC)=O)C)(C)C)ccc(OC)c(Br)c1N Cc1cccc(C(=O)NC(C(=O)NC2(CCF)CCC2)C(C)C)c1O CCC(CC(=O)NC1CCN(C(=O)Cc2ccns2)C1C(C)C)SC c1(CN(C)CC2CCCCC2O)c(O)ccc(Br)c1Cl C12(C(N(CC(C)O)CCNC(C(CCC)(C)O)=O)=O)CC(C)(C1)OC21CCC1 C(C(CO)N=c1[nH]c(Cl)nc(C2CC2)c1F)NC(c1csc2nnsc12)=O Cc1ccnc2ccc(C(=O)NC3CCC3NC(=O)CCCS(C)(=O)=O)cc12 c1(C(=O)NC2CN(C(C3N(N=O)CCC3)=O)CC2O)csc2c(O)ccnc12 CC(CNC(=O)C(CN(C)C)NC(=O)CCc1nc(O)n[nH]1)N=[N+]=[N-] Cc1nn(CC(N2CCC(O)(CNC(=O)Cc3ccc(Cl)s3)C2)=O)c(=O)o1 C1(C(C)C)CN(C(=O)CCN(C(=O)Cc2cn(C)cn2)C)CC(=O)N1 N1(c2ncc(C(=O)OCC)nc2)CC2CC(NC(c3cnn(C)n3)=O)CC1C2 C1(NC(CCC(=O)NCC)=O)C2CCC1N(C(=O)Cn1nnc(C3CC3)n1)C2 Cc1cnc(C(=O)NCCCN(CCO)C(c2cnc(C(C)C)o2)=O)cn1 C(=O)(C(C(C)C)SC)N(CCn1cc(CSc2ccc(N)cc2)nn1)CC c1(C(=O)NCC2C(NC(c3n(CC=C)ccc3)=O)COC2)cc2[nH]ccc2s1 N1(C(C2(F)CC(C(=O)OCC)C2)=O)CCOC(CCNC(=O)CC2CCOC2)C1 NC(=O)CCCC(=O)N1CC2C(N(C(=O)COC(F)(F)F)C3CCC3)C2C1 N1(CC(=O)NC2(CNC(CCC(C)OC)=O)CC2)CCCNS1(=O)=O C1(C(=O)NC(c2cc(C)cc(C)c2)CO)CCC2C(=O)NCC(=O)N2C1 C1(CC(NOCC(C)(C)O)=O)CN(C(C2C=CCCC2)=O)C(C)(C)C1 N1(C(C2CC(=C)C2)=O)CC(CNC(=O)C=CCN2CCOCC2)C(C)(C)C1 CC(C)C(F)C(=O)NCCCN(C1CC1)CC1CC(C)(C)C1 N1(C(=O)OC(C)(C)C)CCN(CC2CCOC(c3nccn3C)C2)CC1 c1(NC(C2CC3CC3N2Cc2cnc(Cl)cn2)=O)nccc(Cl)c1Cl c1(C(=O)NC(CC(C)NC(C2(C=C)CC2)=O)C)ccc(C)n1C c1(-c2c(C(=O)NCCCCCCN(C(CC)=O)C)c[nH]n2)ccc(F)c(Cl)c1 C1(CN(C(=O)CC2CCC=CCC2)C)C2CN(C(=O)Cn3ccccc3=O)CC12 c1(CC(=O)NC(C(C)C)CCNC(=O)C(C)(O)C2CCC2)cn2ccccc2n1 C1(CNC(COCC=C)=O)CCC(C(=O)Nc2cn(C)nc2Cl)CC1 N1(C(=O)CN2CCCC2)CCC(N=c2[nH]nc(CCO)s2)(CO)CC1 N1(C(C2CCCC(C(=O)OC)C2)=O)CCC2(NC(c3ccn(C)c3)=O)CCCC12 Cc1cc(CNC(=O)CC2(NC(=O)CC(C)F)CCCC2)c(C)cc1O C(CCC(C)C(=O)NCC(C1CCCN1C(=O)Cc1cncn1C)(C)C)OC C1(CCNC(c2csc(Cl)n2)=O)CCCCN1C(=O)C(c1cccnc1)O C(=O)(CC1=Cc2ccccc2C1)NC1(CN(C)C(C2CC23CC3(F)F)=O)CC1 C1(CNC(C2CCN(C)C2)=O)C2CCC(C2)N1C(C1(S(C)(=O)=O)CC1)=O C1(C)(C(=O)NCc2c(C(=O)NC(CC#C)C)con2)CCCCO1 Cc1nn(C)cc1C(=O)NC(C1CCCN1C(=O)C=CBr)(C)C C1(NC(COCC=C)=O)CC(CNC(c2ccc(CC(N)=O)cc2)=O)C1(C)C N1(C(C2C(COC)C2)=O)CC(CNC(c2cc(=O)c(OC)c[nH]2)=O)OC(C)(C)C1 Cn1nc(C(N2CCC(CNC(=O)CC3CC34CC4)C2)=O)cc1OC(F)F Cc1ccc(CCC(=O)N(C)CC2(CNC(=O)CCc3cnccn3)CC2)cc1 C(CCSC)(C(=O)Nc1cn(C2CN(C(C3C=CC(CO)C3)=O)C2)nn1)OC N1(C(c2c(C)csc2Cl)=O)CCN(C(=O)CC2CC(=O)NC(=O)C2)CC(C)(F)C1 C(=O)(C(C(C)(C)C)c1cc(F)cc(F)c1)NCC(CC)NC(=O)C(F)CC N1(C(C=CC)=O)CCC(O)(C(=O)Nc2ccc(C)c(Cl)c2)CC1 C(C(=O)OC)(C(C)C)c1nnc(SCCC)n1C O=C1OCC2CN(c3ccc(S(=O)(=O)NC4CC4C(F)(F)F)cn3)CCN12 C1(NC(=O)Cc2ccon2)CC=C(C(=O)NC2Cc3cscc3C2)C1 c1(C(N(CCCNC(=O)COCC2CCCOC2)C(C)C)=O)ccc(N)cc1Cl C1(C(=O)Nc2cccc(C(=O)OCC)c2)CC12CCN(Cc1c[nH][nH]c1=N)C2 C(=O)(C1=C(F)CN(C(=O)C2=C(Cl)CCOC2)CC1)NC1(CC(=O)OC)CC1 c1(C(CNC(c2csc(C3CCCC3)n2)=O)=O)csc(C(=O)O)n1 C(N=c1[nH]c2ccc(OC)cc2s1)C1(CNC(C(CC)(C)C)=O)CCC1 C1(C(N2CC(C)C(N(C)C)C2)=O)CNC(=O)CN1C(=O)C(O)Cn1cncn1 C1(C(=O)NC(C(COCC)C)OC)CC(OC)CN1C(c1c(OC)noc1C)=O c1(C(=O)NCC=CCNC(=O)Cn2nnnc2C2CC2)nccc2occc12 C(=O)(CCCCCC(=O)OC)N(C1CCN(C(c2cc(C)cs2)=O)CC1)CCC Cn1cc(C(F)(F)F)nc1C(=O)NCCCNC(C1CCCN1C1CC1)=O C1(C(C)C)C(NC(C2CC(C(C)C)C2)=O)CCN1C(=O)CN1CCOCC1 Cn1cc2c(CN3CCCC(CNC(c4cnc(F)c(F)c4)=O)C3)cccc2n1 C12C(C)CCCN1CC2.c1(-c2cn(CCCC(=O)NC)nn2)ncc(F)cc1F S(=O)(=O)(c1ccc(S(=O)(=O)Nc2ccc(COC)cn2)cc1)NCC CC(C)CC(O)C(=O)N(C1CCCN(C(c2ccc(CO)nc2)=O)C1)C CC(C)CC(CC(=O)NC(C)C)NC(C1(C(F)F)CCOC1)=O c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(C2(C)CC2)CO)cn(C2CC2)cn1 N1(C(C2CC(=C)C2)=O)C2CCC1(CNC(c1cnc3n1CCS3)=O)CC2 c1(CCC(=O)NC(C(C)NC(C2CNC(=O)N2)=O)(C)C)cccc(F)c1F n1(CC(=O)NCC2CCN(C(CC(C=C)CC)=O)C23CC3)c(C)cc(O)cc1=O N1(C(C2(C#C)CC2)=O)CC2CCC1CN2C(=O)COc1cc2c(s1)CCC2 n1(CCC(=O)NCC2CCCCN2C(=O)Cc2ccsn2)cccnc1=O CCCS(=O)(=O)C(C)C(=O)NCC(O)CNC(c1c(N)sc2c1CCC2)=O S(=O)(=O)(CC(=O)NCC(F)CNC(=O)C(C)OCOC)NCC CCC(CC(C)C)C(=O)N1CCC12CN(C(c1nonc1N)=O)C2 C(=O)(C(C)CC(F)(F)F)N1C(C(N(C2CC(C)C2)C)=O)C(O)CC1 C12(NC(CCCC=C)=O)CCC1CN(C(c1ccc(OCCOC)cc1)=O)C2 C12(CNC(CCCCSC)=O)CCC1CCN2C(=O)CSCCN1CCCCC1 c1(CN2CCC(C(N3CCC(C(=O)OC)C3)=O)C2)ccncc1O C1(c2cn(CCN(C(C)=O)C)nn2)N(C(=O)CN2C(C)CCC2C)CCCC1(C)C C=C(C)CN=C(NCC(=O)NC(C)C)NCC12CC(C1)C(C(F)(F)F)O2 CC(C)C(O)C(F)(F)C(=O)N1CCC(NC(=O)CN2CCCOC2=O)C1 Cc1nc(C(=O)NC2CC(C(=O)OC(C)(C)C)C2)c(-c2ccc(F)cc2)s1 C1(C)(C(=O)NCC(CNC(CCOCC(C)C)=O)(C)O)CCCNC1=O c1(SC)ncc(C(=O)N(C(C)CN(C)C(C2C=CC=CC=C2)=O)C)n1C C1(C(N(CC(C(=O)NC)C)C)=O)COCCN(C(c2ccccc2N(C)C)=O)C1 N1(C(C(C)(C)CNC(c2cnccn2)=O)=O)CCC2(CCCOC2)C1 N1(CCN(C(C(C)NC(C2CCC2)=O)=O)C)CCN(C(=O)CC(C)(F)F)CC1 C1(COC)(NC(=O)Cc2nccs2)CN(C(=O)C(c2ccc(C)s2)C)C1 c1(C(N2CCC(CCNC(CSCCCC)=O)C2)=O)ncccc1C(F)F N1(C(CCCC2C(C)C2)=O)CC(C)(C)OCC1CNC(c1c[nH]cc(Cl)c1=O)=O c1(C(=O)NC2CN(C(c3cncc(NCC)c3)=O)CC2F)c(F)cc(C)cc1Cl C(=O)(CC(C)C(F)(F)F)N1CC(C(=O)NCCC(C)SC)(CC)C1 CC(C#N)C(=O)NC1(CCNC(=O)CN(CC(C)(C)C)C)CC1 C1(NC(=O)OC(C)(C)C)CCc2nc(C(N3C4CCC3(C(F)F)CC4)=O)cn2C1 N1(C(C2C(=C)C2)=O)CCN(C(C2(c3ccc(Br)s3)CCC2)=O)CC1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(C(=O)NCC(=O)NC(C)C)CC(C)(C)C1 Cc1nc(C(C)C)oc1C(=O)NCC(C)N(C(=O)CCc1cccnc1F)C c1(C(=O)NCC(C)(C)O)nc2ccc(-c3cnn(C(C)(C)CO)c3)cc2s1 C(C(C(=O)N1CC=CC1CF)NC(C1CCOC1C(C)C)=O)OCC C(=O)(CCCC(F)F)NC1CCC(C)(CNC(c2ccc(C(N)=O)o2)=O)C1 c1(C(N(C2CN(C(=O)CCn3cnnn3)CC2F)C)=O)ccc2cccc(F)c2n1 N1(C(C(C)Oc2ccccn2)=O)CCC(F)(CNC(=O)C=CC2CCC2)C1 c1(CC(CNC(C(c2cnn(C)c2)OC)=O)C)nnc(C)n1C C(CC)(CC)(CCNC(=O)C(C)(O)C1CCC1)NC(C(CCC)NC(C)=O)=O Cc1ccc(F)c(NC(C2N(C(COc3ccccc3ON)=O)CCCC2)=O)c1 c1(OC)cc(C(N2CCC(NC(=O)Cc3nnc(O)s3)C2)=O)ccc1OC(C)C C(=O)(N=c1cc[nH]cc1)NCC(=O)N(C1CCN(CC(C)O)CC1)C C(=O)(C1=CC2CCCCCC12)N1CCCC(c2cn(C(C(C)O)C)nn2)C1 C=C(Cl)CC(C(=O)NCCc1ccn(CC)n1)NC(C1CCC2CC12)=O C(=O)(C1=CC(O)C(NC(C2(CF)CC2)=O)C1)NC1C(OC)COCC1 C(=O)(CCC(C)(C)C)N(C)CC1CN(C(=O)CC2CS(=O)(=O)C2)CCO1 CC1(C)CC(NC(c2cc(C3CCC3)n[nH]2)=O)CN1C(C1CC1F)=O N1(C(C2C(CC)C2)=O)CCC(CN(C(=O)COCC(F)(F)F)C)C1 C#Cc1ccc(C(=O)NCC2CN(C(=O)COC)CCO2)c(C(F)(F)F)c1 C(=O)(C#CC1CCOC1)NC(C(=O)NC1(C)CCSC1)CC1CCCC1 N1(C(CC2C(C)(C)C2)=O)CC(NC(=O)CNc2nccs2)CC12CCOCC2 C(=O)(CCC(=O)c1ccc(Cl)cc1)N(CCN(C(C1(CC#C)CCOC1)=O)C)C CC1CCC(CNC(=O)CSCC#N)N(C(c2cc(-c3ccccc3)ns2)=O)C1 C1(NC(C)=O)CCN(C(=NCCC2(F)CCC2)NC(c2ccccc2)C)CC1 C(=O)(C(CCCC(OC)OC)N1CCN(S(C)(=O)=O)CC1)NCC(=C)C N1(C(CC2(CC)CC2)=O)CC(CNC(=O)CC2(C)CC2(F)Cl)C(C)C1 c1(-c2nc(N(C(=O)C(C)SC3CCC(C)CC3)CC)sc2)ccc(F)c(F)c1 C1(NC(CCSCC(N)=O)=O)CC2(C1)CC(CNC(C1CCCCC1F)=O)C2 N1(CC(=O)NCCCCNC(C2(C(C)(C)C)CCCC2)=O)CCCOC1=O C(N=c1[nH]c2c(c(=NCC3CSCCO3)[nH]1)COC2)C1(C)CCN(C)CC1 C1(NC(c2ccon2)=O)CC(F)CN1C(C1(c2cccnc2)CC1)=O c1(NC(=O)NC2CCCC2C(=O)NC(=O)C(F)F)cccc(Br)c1 c1(NC)ccc(C(F)(F)F)cc1C(=O)NCC(C)(CO)NC(=O)C=C1CCCC1 c1(CNC(C2CC2CF)=O)cccc2c1CN(C(c1csc(Br)c1)=O)C2 c1(C(=O)NC2CC(CCNC(C3C(OCC)C3)=O)C2)c(Br)cnn1CC Cc1nccc(CCNC(C23CC2CN(C(=O)C(C)CC2CC2)C3)=O)n1 C1(NC(CC=C)=O)CN(C(c2cc(C)c(F)cc2O)=O)CCC1(C)C N1(CC(=O)NCCCCC#C)CCCN(C(c2ncoc2CC)=O)CC1 c1(OCCCC)c(OC)cc(CN(C)CC2CCCCC2C)cc1Cl C(=O)(N=c1ccc(N2CCCC2)n[nH]1)c1ccn(C(c2ccccc2)C)n1 C1(NC(CCN(CCC)C)=O)C2CC3C(C2)C13C(=O)NC(c1ncc[nH]1)C CC1CC(=O)NCC1C(=O)Nc1cccc(CNC(c2cc(C3CC3)on2)=O)c1 N1(C(C2(COC)CCCO2)=O)CCCC(CC(=O)NC(CC2CC2)C2CC2)CC1 O(NC(=O)C(C1(O)CCCCC1)NC(=O)CCC1CCOC1)CC(C)C C(CCC(=O)N(CC(C)CNC(c1cnn(CCF)c1)=O)C)OCCC CC(C)(O)C(C)(CO)NC(=O)C=CCNC(=O)C(F)C(F)(F)F Cc1csc2c(N3CCC(CCNC(C4CC4(C)C)=O)C3)ncnc12 N1(C(c2n(C(C)(C)C)ncc2)=O)CCN(C(C2CCCC2(C)C)=O)C(C2CC2)C1 CCC(CC(=O)NCCC(=O)NCCCC1C=NNC1=O)C(F)F c1(C(N2CCC(NC(C3(CC)CCNC3=O)=O)C2)=O)csc2cc(OC)ccc12 c1(CNC(C(=O)Nc2n(C(C)C)ccn2)=O)cn(C(F)F)c2ccccc12 N1(C(c2cc(C)c(C)s2)=O)C2CCC1CC(CNC(C1(CF)CCC1)=O)C2 C(=O)(CC(C)(C(F)F)N(C)C)N1CC(CCCCNC(c2c(C)oc(CO)c2)=O)C1 CN1CCCCCC1C(=O)NCC1(CNC(C2(C)CCOC2)=O)CCC1 c1(COC)noc(CNC(=O)C(C2CC2)NC(c2sncc2C)=O)n1 n1(CC(=O)NC(CCCNC(C(C)OCCC(C)C)=O)C)cnccc1=O c1(C(=O)NC(CC=C)CNC(=O)CCCc2ncco2)ccc2ncccc2n1 c1(C(N(CCC(C(C)(C)C)NC(C2C=CCC2)=O)C)=O)ccc2ccoc2c1 CN=c1nc(N2CCC(CCO)C2)[nH]c(=NCc2ccnc(Br)c2)[nH]1 c1(C(=O)NCC(C)(C2CC2)NC(C2CCC(C)CC2)=O)ccc(F)c(C(N)=O)c1 c1(CSCC)cccc(C(=O)NC2C3CCN(C(C4CCC(CC)CC4)=O)C23)c1 c1(C(=O)NC2CN(C(COCC=C)=O)C(C)(C)C2)cnc2n1CC(C)CC2 C(=O)(C1CCc2cc(F)ccc21)NC12C(CN(C(c3cccc(C#C)c3)=O)C1)C2 C12(C(=O)NCC3(F)CCN(C(Cc4c(C)n(C)cn4)=O)C3)CC1COC2(C)C C(C(C(=O)N(CCCNC(=O)C(CO)N(C)C)C(C)C)OC)OC C(CN=c1ccnc(NCCCC2CCCCO2)[nH]1)NC(=O)C1CC1 N1(C(C(C)(C)CNC(=O)CC2CCC(=O)NC2)=O)CCNC(=O)CC1 CN1CC(NC(C2CC=CCN2C(c2nocc2Cl)=O)=O)C(C)(C)C1 c1(CC)ccc(C(=O)NC(C)CCNC(c2cc(C(C)CC)no2)=O)cn1 c1(C(N(CCCNC(C2(OCC)CCC2)=O)C)=O)nc(C(F)(F)F)sc1C N1(C(=O)Cc2cn[nH]c2)CCN(C(c2c(O)cc(F)cc2F)=O)CC2(CC2)C1 C12(CNC(CSc3cn(C)nc3)=O)CCCC1N(C(=O)CCCF)CCC2 Cc1nc(C(=O)NCCn2cc(CNC(C3(C)CCOCC3)=O)nn2)c(C)n1C N1(C(CCC=CCC=C)=O)CCC(C2CC2)C1C(N1CC2CC2C1)=O c1(C2(C(=O)NCC3C(NC(c4cn(C)nc4)=O)CCC3)CC2)c(F)cccc1Br C(=O)(C(C)(F)C(=O)NC1CCCC1CC(=O)NCC(C)C(C)(F)F)OC C(=O)(CCCC(C)CC)N(CCCCNC(c1nc(COCC)sc1)=O)C CC1CC(=O)NC(C(=O)NC2C=CC(CC(=O)NC34CCC(CC3)C4)C2)C1 C1(NC(CCN(C(=O)CN2CCCCC2)CCO)=O)CC2CCC(C1)O2 c1(N2CC(CC)N(Cc3sccc3C(=O)OC)CC2)ncnc2c1CCCC2 c1(C(=O)NCC(C2CCCC2)NC(COC)=O)cc(=O)n(-c2ccccc2)[nH]1 Cc1ccc(=N)[nH]c1C(=O)NC1CCCCC1N(C)C(c1cc(=O)n(C)o1)=O c1(C(N(CC(C)NC(C2(C(F)F)CC(F)(F)C2)=O)C)=O)cc(S(N)(=O)=O)c[nH]1 C(Cc1ccccc1)(CCNC(=O)CCC1(C)CC1)NC(C(C1CC1)OCC)=O c1(C(=O)NC2CC3CN(C(C(C(CC)O)C)=O)CC32)cc(C)c2c(c1)CCCN2 C(C)(CNC(C1COCC1(C)C)=O)(C(C)C)NC(c1n(CCC)ncc1)=O c1(C(=O)NC(CC(C)NC(C2(CCCC)CCCC2)=O)C)cnc(Cl)cn1 c1(CNC2C3CCN(C(COCCCOC)=O)C32)coc2cccc(O)c12 C1(C(=O)NC2CC(O)(CNC(=O)CCc3cncnc3)C2)CCC2(CC2)C1 CCC(F)C(=O)NCCN(C(=O)C(C)(C)N1CCCCC1)CC c1(C(C(=O)NC2C(CNC(C3C4(CC(OCC)C4)C3)=O)C2)O)cc(F)cc(F)c1 c1(C(N(C2CN(C(CC(CC)(F)F)=O)CC2(C)C)C)=O)cc(C)cc(C)c1O N1(C(CCCn2c(C)ncc2)=O)CCC(NC(=O)COC(F)(F)F)C(F)C1 Cc1cc(C(=O)NC(CNC(C2(O)CC(CF)C2)=O)CO)ccn1 c1(C(=O)OC(CCC)C)ccc(NC(C)=O)c(CC)c1 c1(N2CCC(CC=C)(NC(=O)CCN(C)CCC)C2)cc(C)nc(CC(C)C)n1 c1(OCCC(N2CCC(N3CCCOC3=O)C2)=O)ccc(-c2nn[nH]n2)cc1 c1(C(=O)NCCCN(C(CN2CC(C)C2)=O)C2CC2)c[nH]nc1C1CCC1 Cc1nc(C)c(CN2CC(NC(C3(C4CCCO4)CCC3)=O)C2)s1 C1(C)(CC)CN(C(c2coc(CNC(C3CCC(=O)C(C)C3)=O)n2)=O)CCO1 c1(C(N2CCC(F)(CNC(CCC=CC)=O)C2)=O)cc(Br)c(N)cc1C c1(OC)c(C(=O)N(CCC(C(C)C)NC(=O)CN2CC(C)(C)C2)C)occc1=O c1(C(C)C)nc(NC(C2CC(C)(C)C2)=O)cc(=NCCC=C(C)C)[nH]1 c1(C(=O)NC(C(C)NC(c2c(CC)nn(C)c2)=O)C)c(C)cccc1Cl c1(C(=O)NC2(C(=O)NC(CNC)C)CC2)ccc(Cl)cc1Oc1ccccc1 N1(C2(C#C)CC2)CC(C#N)(S(C)(=O)=O)C1 c1(OC)ncc(Br)cc1C(c1nnnn1C1CCCC1)NCCC(C)(C)OC C1(CC(=O)N(CC#C)CCO)CN(C(c2cccc(F)c2)=O)CC12CC2 c1(-c2n(COCC(F)(F)F)nc(CC3CCC3)n2)coc2c1CCCC2 N1(C(C)=O)CCC(C(=O)NCC(C)NC(c2csc(C(=O)OC(C)(C)C)n2)=O)C1 c1(C(N2C(C)C(NC(=O)CCC3CC3)CC2)=O)cncn(C)c1=O C123CCC(CN(C1)C2=O)C3.c1(CNC(C2CC2C(F)F)=O)ccc(F)cc1 C1(C(N2C(CNC(=O)C=CC(F)(F)F)CC2)=O)CC2CCC(C1)C2(F)F N1(C(C=CC=C(C)C2CC2)=O)CC2CCCC(C1)N(C(c1ccc(C)c(C)n1)=O)C2.C(C(=O)O)=CC=C.CCCl C1(C(=O)NCCCCNS(C)(=O)=O)COCC2(CNC2)O1 CN1C(=O)C(F)CC1C(N1CCC(NC(c2ccc(-c3ccncc3)o2)=O)C1)=O C=C=CC(C)C(=O)NCC1(CNC(=O)C(C(C)O)NC)CC1 Cc1cncc(CCC(=O)NC2CN(C(c3c(C)noc3C)=O)CC2C)c1 C1(NC(C2CN(S(N)(=O)=O)C2)=O)CN(C(=O)COC2CCOC2)CC2(CC2)C1 CC1CN(C(=O)CCC(C)(C)F)C(C)CN1C(=O)Cc1ncc(F)cc1F n1(CC(=O)N(CC(CC)NC(=O)C=CSc2ccccc2)CC)cccc(C)c1=O C1(CC)CCCCN1c1nnc(Cc2cccs2)n1CC1CC1 c1(C(=O)NC2CCC(CNC(C3CSC3)=O)C2)cccc2c(O)nncc12 C1(C)(CNC(c2c(CC)scc2)=O)CCN(C(=O)C(C)(C)CF)C1 C12(NC(CC3N(C)CCC3)=O)CCOC(CNC(c3cncc(C#N)c3)=O)(C1)C2 Cc1ccc(F)c(C(=O)NCC2CC(O)CN2C(c2cc3n(n2)CCO3)=O)n1 N1(C(CCCCC#C)=O)C2CCC1CC(NC(c1cc(CC)ccc1O)=O)C2 CC(C)C(O)C(C)C(=O)NCC(C(=O)N1CC2CCC2(C)C1)C(C)C C1(NC(=O)OC)CCN(C(=O)NC2CCN(Cc3ccccc3)C2C)CC1 c1(C(N2C(C)(CNC(C3ON=C(C(C)C)C3)=O)CCC2)=O)ccccc1[N+](=O)[O-] n1(Cc2ccc(C)cc2)c(C)ccc(C(N2Cc3nc(C)sc3C2)=O)c1=O Cc1c(C(=O)NC(C)CNC(=O)C(C)Sc2ccccn2)ccc(F)c1F c1(CNC(=O)NCCCn2ncc(C(=O)OCC)c2)c(C)nn(C)c1OC N1(C(COc2c(C)ccc(Cl)c2)=O)CCCCC2(CCN(C(=O)C(C)C#N)C2)C1 C=CCC(CNC(=O)C(F)=CC1CC1)NC(c1ncoc1CCCC)=O c1(C(=O)NC(C2CCCC2)CNC(c2n(CC)nnc2)=O)cc(Cl)ncc1NC C1(CCC)CN(C(=O)CC2CC(=O)NC2=O)CCN1C(=O)Cn1cc(CC)cn1 N1(C(c2c(OC)ccnc2)=O)CCC=C(C(=O)N2CCNC(=O)CC2C)C1 c1(OC)ccc(S(=O)(=O)N2CCCC2C(=O)Nc2ccc(=O)n(C)n2)cc1 c1(C(=O)NC(CN(C(=O)Cc2cccc(F)c2)CC)C)n[nH]c(C)c1Cl C1(CCC)CCC(C(=O)NC2CCC(NC(C3(O)CCC3)=O)CC2)CC1 c1(CC)ccc(C(=O)NC2CN(C(=O)CC3(O)CCC3)CC2(C)C)cc1Br CC1CC(C(=O)N(CC(C)N(C)C)C)N1C(=O)COC1CCCOC1 c1(C(N(CCNC(CC(C)C(C)(C)C)=O)C2CC2)=O)cnc2c(cnn2C)c1N c1(C(=O)NC2(C)CCCN(C(CCC(C)C#N)=O)C2)n[nH]c2c1CCSC2 C=CC(C)(CC)C(=O)NCC1(CO)CCCN(C(=O)CCOCCCOC)C1 c1(CC)ocnc1C(=O)NC1CC1CNC(=O)C(F)=CC1CC1 C1(CNC(=O)Nc2c(OC)csc2)COCCN1C(=O)C(C)c1cccs1 C(=O)(C(C(C(C)CC)OC)N1CCCCCCC1C)NCCC C(C)(CCC(=O)NCC(C)(C(C)C)NC(=O)COCC=Cc1ccccc1)SC C1(NC(C2(OCC)CCOC2)=O)C=CCCC1C(=O)NCCCCC1CC1C C(=O)(C1=CC2(CCOC2)C1)NC(CNC(CCC1CC(OC)C1)=O)C(C)C C1(C(=O)NCCc2ccc(C)nc2)CC12CCN(C(c1cc(C)nc(O)c1)=O)C2 C1(CNC(CCCCC)=O)C(C2CC2)CCN1C(=O)Cn1cnc(C(N)=O)n1 c1(OC)ccc2onc(C(N)=O)c2c1.C12CCCN(C1)S(=O)(=O)CC2 C1(SC)CN(C(=O)C2CC2)CC1C1CC1.c1(-c2ccccc2)cc(C)c(CC=O)o1 Fc1cc(Br)ccc1C1CCN(CN2CC=C(Br)CC2)C1 CC1CC(C)(C(N2CCC(CNC(=O)C(O)C3CCCC3)C(C)C2)=O)CC(C)O1 C(=O)(C1CCCc2ncnn21)NCC1CC(NC(c2cnn3ccccc23)=O)C1 c1(COCCCNC(N(CCC(c2ccccc2)O)C)=O)ccc(Cl)cc1 C(=O)(C(CC(N)=O)NC(C1CCCSC1C)=O)NCC(C(C)O)O c1(NC(CNC(c2cccc(C)c2)=O)C(F)(F)F)scc2c1CCCC2 CCC(CC(=O)NCC1(C)CCCN(C(=O)COCCCOC)C1)C(F)F N1(C(CC(CCC)CC)=O)CC2(C)CN(C(=O)C(C3CCC(=O)N3)C)CC2(C)C1 C12(CNC(c3cc(C(N)=O)[nH]n3)=O)CC1CN(C(C1CC(F)C(=O)N1)=O)C2 c1(-c2cc(C(=O)NCc3cccnc3Br)c(Cl)nc2)cnc2c(F)cccc2c1 [N-]=[N+]=NC1CCC(C2CC2)CN1C(c1ccc(OCC2CC2)cn1)=O c1(C(=O)NCCC(CNC(C2(C)CCCO2)=O)O)c(Br)ccc2n[nH]cc12 C(=O)(CC1NC(=O)c2ccccc21)NC1(CC=C)CN(C(c2occc2Br)=O)C1 S(=O)(=O)(c1cccc(Cl)c1F)NC1CN(C(c2ccnc(OC)c2C)=O)CC1O C1(NCc2n(Cc3cccc(OC)c3)ccn2)CCC2CC(F)(F)CCC12 C1(C(=O)NC(C)CNC(c2cn(CCCF)nn2)=O)CCC2C(CC1)C2(F)F N1(C(C(N2CC(CNC(C(CC)=CC)=O)C2)=O)C)CCN(C)CC1 C1(C(N2CCCC(F)(CNC(C=CCCC(C)C)=O)C2)=O)CCc2ccnn2C1 c1(CC)ccc(C(=O)NC2CC(CC(=O)OC)C2)cc1[N+](=O)[O-] CC(C)C(C(=O)N1CC(NC(C2CN(C(N)=O)C2)=O)C(O)C1)c1cccc(Cl)c1 C1(C(=O)NCC2(F)CC(NC(COCCOCC#C)=O)C2)CCCN(CCC)C1 C(C)(C)(CC(=O)NCCc1cnn[nH]1)NC(COCCC=C)=O CC(=O)C(C)CC(C)C(=O)N1CC(O)CCC1C(=O)NCc1noc(C)n1 CCCCC(C)CCC(=O)NCC1CCC(C(=O)NOCC(F)F)C1 C1(NC(CCC=C)=O)CC2CCC(C1)N2C(=O)COc1ccc(Cl)nc1 c1(C(N2CCCC(CN(C(C(COC)C)=O)C)C2)=O)csc2cnccc12 C(=O)(CC(C)(C)C)N1C(CNC(C(C)N(C(=O)CSC2CC2)C)=O)CC1 c1(C(=O)NC2(C)CCN(c3sc(C(=O)OC)c(Cl)n3)C2)noc2cc(Cl)ccc12 CC(C)(C(=O)NCCCCC(N)=O)C1=CCN(C(c2ccc(C3CC3)o2)=O)C1 C(=O)(C1=NOC(C)(C)C1)N(CCOCCC(=O)NC(CCOC)C(C)C)C N1(CCC(N2C(CNC(CN3CC(C)(OC)C3)=O)C=CC2)=O)CCNC(=O)C1 C=Cc1ccc(C(N2CC(NC(c3cc(Br)cnc3O)=O)C(F)(F)C2)=O)cc1 C(N=c1[nH]cnc(Cl)c1F)C1(NC(COC2CCN(C)CC2)=O)COC1.C(COC)S C1(CN(C(=O)C(c2cccnc2)O)C)CCCN1C(c1c[nH][nH]c1=N)=O N1(C(c2nc(CC)sc2N)=O)CC2CC(C1)CN(C(C1C3CS(=O)(=O)CC13)=O)C2 c1(C(=O)NCCN(C(Cc2c(C)nsc2)=O)C2CC2)cn(CC(F)F)nc1C C1(C(N2C(CCNC(c3cc(CC)n(C)n3)=O)CSCC2)=O)CCCCC12CC2 N1(C(C2C(C(N)=O)C2)=O)CC2CC(C1)N(C(=O)CC1(N(C)C)CC1)C2 C1(C(=O)NC2(COC)CC2)CCC=CC1NC(=O)CN(C1CCC1)C C(=O)(CC(C(C)(C)C)NC(=O)Cc1cncs1)NC(C1CCOC1)C C(C(CC(C)C)NC(=O)C(=O)NC1CC1c1nccn1C)NC(C)=O c1(C(=O)NC2CCC3CCN(C(C(CC)CC)=O)C32)ccc2c(c1)C(=O)C(=O)N2 c1(-c2c(C)occ2)nc(C(O)CC(F)F)n(CC2CCSC2)n1 c1(C(N(C(C)CCNC(c2ccc(C3CC3)cc2)=O)C)=O)ccc(S(C)=O)cc1 N1(C(C2C(OCC)C2)=O)CCN(C(=O)Cc2ccsn2)C(c2ccccc2)C1 c1(OC)cc(C)c(CN2CCC(O)(C(=O)Nc3ccc(O)cc3C)C2)cn1 N1(C(CCC)CC(=O)OC)CC(C2=NOC(C)(C)C2)C1 c1(CC(=O)NCCNC(C(CC)(C)F)=O)cc(F)cc2c1OCOC2 C1(CNC(C2CCC(CCNC(CC)=O)C2)=O)CC(C(=O)OC)=NO1 c1(C(N(C(CN(C(C)=O)C)C)C)=O)ccc(C2CC2)o1.C1(=O)C(C2CC2)CN1 C(=O)(C(C)(C)CO)NCC1CCC(C(N2C(C(C)C)C(C(C)C)C2)=O)C1 c1(N(C2CC(=C3CCC3)C2)C(N2CC(N3CC(O)C3)C2)=O)nccc(CO)n1 c1(NC(=O)CN2CC(C(F)(F)F)C(O)C2)ccc(Cl)c([N+](=O)[O-])c1 C1(NC(C2CCCC2)=O)CCN(C(C2CCCCO2)=O)CCC1CO c1(NC23CC(C(=O)NCC4CCCN(C(C)=O)C4)(C2)C3)ccc(C#N)n1C c1(OC)ccc([N+](=O)[O-])cc1.C1(c2cn(C(C)C)nn2)C(C)CCN1CC.C1(=O)CO1 CCCC(CNC(c1cccc(CNC(=O)C(C)CC(C)C)n1)=O)CCC C(=O)(C(N=[N+]=[N-])C(C)C)N(CCC(=O)Nc1cc(C)c(F)nc1)CCO CCC(CC(=O)N1CCC(CCN(C(=O)C(CC)(CC)CC)C)CC1)C(F)F c1(CCC(N2CC(COC)C3(C2)CC3)=O)ccnc2ccccc12 N1(C(C(C(COC)C)C)=O)CCC2(CCOC2)C(CNC(C2(COC)CC2)=O)C1 C12(NC(C(C)CO)C)CCC(C)(CC1)OC2 c1(C(=O)NC(C(C)NC(c2conc2C2CCC2)=O)CO)ccc(O)cn1 c1(CNC(CN2C(C)CCC2C)=O)nnc2n1CCC2 C1(C(=O)NCC2(C)CCN(C(C(F)=CCC)=O)C2)CCC2C(=O)NCC(=O)N2C1 C1(C(C)NC(C2C(COC)C2)=O)CCN(C(=O)CC(=O)Nc2nccs2)CC1 c1(OC)ccc(C(F)(F)C(=O)NC(C)CC(C)NC(=O)CCCCC2CC2)nc1 C1(C(=O)OC)COCC1COC(=O)C(F)C1CC(C(C)(C)C)C1 c1(CC)nn(C)cc1C(N1CCC(C(=O)NOCC(=O)N(C)C)C1C)=O N1(C(C(F)=CC)=O)CC(C)(C)OC2(C1)CN(C(=O)CC(C)SC)C2 N1(CCC=CCCC)CCC(N(C(=O)CC(C)n2ccc(C)n2)C2CC2)CC1 N1(C(=O)Cc2cc[nH]n2)CCC2(CCCC2C(N2CCCOCC2)=O)C1 N1(C(c2cnn(C)c2C#N)=O)CC(C)(C(N2CC(CO)C(O)C2)=O)CC1(C)C n1(CC(=O)N(CC2N(C(CC)=O)CCCC2)CC)ncc2ncccc12 Cc1ccc(C(N2CCCC(C)C2CCNC(C2CNC(=O)O2)=O)=O)c(F)c1F c1(CS(N2CCC(O)C2c2ccccc2Cl)(=O)=O)cc(F)ccc1Cl C1(C(=O)N(C2CCCC2)CCO)CC=CC(N(C(C)=O)C(c2cn(C)cn2)=O)C1 Cc1cc2c[nH]nc2cc1C(=O)NCC(O)CN(C(=O)CCC1CC1(C)C)C n1(CC(N2CCCCC(N(C)C(=O)OC(C)(C)C)C2)=O)cc(F)ccc1=O N1(C(C2=CCN(C(CC(CC)SC)=O)C2)=O)CCCC2(CCC2)C1 c1(C(=O)NC2CCC(C(N(CC#C)Cc3ccco3)=O)C2)cc2ccccc2[nH]1 c1(CCn2cc(CNC(c3c(C)cc[nH]3)=O)nn2)ccc(Br)nc1 c1(C(N2CC(C(=O)O)(C(F)F)OCC2)=O)cc2c(s1)-c1ccccc1OC2 C1(NC(c2ccn(COC)n2)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(C)O N1(C(CC(=O)Nc2ccccc2)=O)CCC2CN(C(C3CC4(CC4)C3)=O)CC2C1 C12(C(N3CC(CNC(C4CCCOC4)=O)OCC3)=O)CC(CO)(C1)OC21CCC1 c1(CC)ncc(C(=O)NC2COCC2NC(=O)COc2ccsc2)[nH]1 Cc1ccc(CN2CCC(C(=O)NCCNC(c3ccccc3)=O)CC2)cc1C C1(C(=O)Nc2cccnc2C(F)(F)F)CC(F)(F)CN1C(=O)CC1CCCC1 c1(C(=O)OC)cncc(C(=O)NC2(CNc3ncncc3Br)CCCC2)c1 c1(OCC)nccc(C)c1NC1(c2nnnn2CCCSC)COCC(C)C1 c1(NC(C2N(C(c3c(CC)nns3)=O)CC(O)C2)=O)ccc2c(c1)COC2 Cc1cc(N(C)Cc2ccc(Cl)cc2)ncc1S(=O)(=O)NC1CCN2CCCCC12 Cc1ccnn1CC(=O)N(CC(=O)N(C(C)CO)C)C(C)C Cc1oc(CO)cc1C(N1CCC(CF)(NC(=O)CSc2ccncc2F)C1)=O N1(C(c2ccc(C(C)=O)[nH]2)=O)CCN(C(c2ncsc2C(F)(F)F)=O)CCC1C N1(C(c2cnc(C)nc2O)=O)CCC2CCC(NC(=O)CC3C=CCCC3)C1C2 C(=O)(CCC(=O)NCCCC(C)C)C1(CN2C(SC)CCC2)CC1 N1(C(C2N(C(c3n(OC)cnc3C)=O)CC2)=O)CCC2(CNC(=O)N2)C1 CC1CN(C(c2cccc(=O)n2C)=O)CC(CCNC(c2sccc2CO)=O)O1 N1(C(c2cccc3c2OCO3)C(=O)NCCC)CCC2OCCCC2C1 c1(CN2C(C)CN(C(=O)C(C)(C)C)CC2)c(O)nc(=O)n(C2CCCCC2)c1N C1(C(N(C2CCN(C(Cc3c(C)noc3)=O)C2)C)=O)CC(C)CCC1C(C)C c1(C(N2CCOCC2Cc2cn(CC(F)(F)F)nn2)=O)ccc2scnc2c1 n1(CC=C)cc(C(=O)N(C(C)CNC(=O)C(O)CN2CCOCC2)CC)cn1 c1(CN(CC(F)(F)F)CC(N2CCCC(CS(C)(=O)=O)C2)=O)ccc(C#N)cc1 CCC(C)(COC)C(=O)NCCCCC(=O)Nc1cc(C)ccc1CO Cc1cc(CNC(=O)COC2CCN(C(c3ncccc3N)=O)C2)sc1C C1(C)(C(N2CCN(c3nsc(C4CC4)n3)CC2)C)CCCOC1 C1(CC(=O)NC)CN(C(C2CCCCC2(F)F)=O)CCN1C(=O)CC1(O)CCC1 C1(C)(C(=O)NC2CCCN(CCC)C2)CCCN(C(=O)C=Cc2ccc[nH]2)C1 c1(NC(CCC)(C)c2nnnn2-c2c(C)cccc2C)cc(F)c(Br)cc1C n1(C(C)C)ncc(C(=O)NC(C)CCNC(c2ccc(C#N)[nH]2)=O)c1C1CC1 C(=O)(C(C)(C)CCC)N(CC(CN(C(c1cnc(CCC)s1)=O)C)O)C c1(OC)c(Cl)cc(C(=O)NCCOCCN(C)C(C2CN(C)CC2C)=O)nc1Cl c1(CC)ncc(C(=O)NC(C)(CNC(c2nocc2C(C)C)=O)C2CC2)s1 N1(C(C(c2c(C)ccc(F)c2)=O)=O)CCC2(CC1)CN(C(c1ncnn1C)=O)C2 C1(C(=O)NCCCCC(C)(C)C)(NC(c2c(CCC)nco2)=O)CCC(C)(C)C1 C=CC1CN(C(=O)CCC2(C)CCC(=O)N2)CC1NC(=O)C=CC(C)(C)SC N1(C(c2ccnc(C)c2O)=O)CC2CC(NC(=O)C(C)SC(F)(F)F)C(C2)C1 c1(C(=O)NC2CN(C(CC3CC(CC)C3)=O)CC2F)c([N+](=O)[O-])cnn1C S(=O)(=O)(c1cccnc1NCC1(CC2CCC2)CC1)N1CCN(CC(C)O)CC1 CC(N=c1nc(N2CCN(C3CCCC3O)CC2)c2cnn(C)c2[nH]1)C(F)F C1(N(C)C(c2ncoc2C(C)(C)C)=O)CCC(NC(=O)CCc2nncn2C)C1 c1(C(N2CC3(OCCN(c4c(C)cncn4)C3)C2)=O)c2n(c(=O)n1C)CCCC2 C(=O)(C1=CNC2=NCCC2=C1)N1C(C2(C(=O)NC(CC)(C)C)CC2)CCCC1 c1(C(=O)NC2C(NC(c3ccc(Cl)s3)=O)C2)sccc1Cl CC(C)C(C(=O)NC1C=CCCCC1)NC(=O)CCN(C)CCO C1(C)(C(=O)NCC23CN(C2)C(=O)CC3)CCN(C)CC1.CCC(C)(C)OCC.OCC C1(C)(C(=O)NC(COC(C)C)(C)C)CCN(C(=O)CC2CCC(=O)C2)CC1 c1(C(C=C)C)nc(C2CCOC2)nn1CCCOC c1(CC(=O)NCC2CC2CO)cc(C(=O)Nc2cccc(SC)n2)cc(N)c1 C(=O)(C(C(C)O)NC(c1cnc(S)[nH]1)=O)NCc1nc(C(C)C)on1 N1(CCCC(=O)NC(C(C)NC(c2c(C(=O)OC)csc2)=O)C)C(=O)CCC1=O c1(C(=O)NCC2(F)CC(NC(CC3CCCC(OC)C3)=O)C2)ncc(C)cc1C C(CN=C(NCc1occc1C)NC(C)C)c1ccc(SC)cc1 C#CC1(NC(C2CCC3(CC3)N2C(C2C3CN(C)CC23)=O)=O)CCCCCC1 O=C(C1=NOC(c2ccccc2)C1)NCC1CCCN1C(C1CCS1(=O)=O)=O CC1(C)Cc2cc(C(=O)NCC3C4CN(C(C5CCC(=O)O5)=O)CC34)ccc2O1 c1(C(C)=O)cc(C(=O)NC(C)CCNC(c2c(OC)cccc2O)=O)ccc1C c1(C(N2C3CN(Cc4nccc(C#N)c4)CC32)=O)cc2n[nH]cc2cc1Cl C=C(C)C(CC(=O)NCC1(OC)CN(C(c2cc(Cl)sc2Cl)=O)C1)OCC C1(O)(C(C)NC(=O)CCN(c2ccc(Cl)cc2)C)CCN(C(C2(Cl)CC2)=O)CC1 C1(C(N(CCCNC(c2ccsc2C(F)F)=O)CC)=O)CN(C)CC1C(F)(F)F N1(C(C(=O)NCCC#N)c2cn[nH]c2)CCC2(CCC2)C1 Cc1cc(=NC(=O)C2C=CC(NC(=O)C(CO)C(C)(C)C)C2)[nH]n1C1CC1 C(=O)(C1=C(C)CC1)NCCn1cc(C(N2CC(C(=O)OC)(OC)C2)=O)nn1 C1(N(C(=O)NC2CC(CC(N)=O)C23CCC3)CC)CC2CCCCC2C1 N1(C(c2cc(C3CC3)[nH]n2)=O)CC2CC(C1)CN(C(c1csc(Cl)n1)=O)C2 Cc1cn2c(n1)CC(C(=O)NCC1CN(C(=O)C(C)OC3CCCC3)CC1O)C2 C(=O)(C1=CC2CCC(C1)C2)N1C(C(=O)NCC(CC)C(C)C)C(O)CC1 O(NC(=O)C1=COCC1)CC(N1C(C)CC(C(c2ccccc2)=O)CC1)=O N1(C(C(CC2CCCC2)OC)=O)CCNC2=C1S(=O)C=CC=C2 c1(NC(N2CCC2C(=O)NC2CC(=C(F)F)C2)=O)ccnc(OC(F)F)c1 C1(C(N2CCCC(NC(CCCNC(C(C)(C)C)=O)=O)C2)=O)CC2CCCC2C1 C1(C(N2C(CSC)CCC2)=O)CN(C(C2CC3(CSC3)C2)=O)CC1(F)F S(=O)(=O)(c1ccccn1)NCC1CCN(CS(C2(CC=C)CC2)(=O)=O)CC1O c1(C(N(C)CC2CN(C(CN(C)C(N)=O)=O)CC2O)=O)cccc2[nH]ncc12 c1(C(=O)NCC(C)(C2CCC2)NC(C(CN(C)C)N(C)C)=O)cc2cccnc2s1 CC1(NC(c2coc(CNC(c3cnns3)=O)n2)=O)CC(O)(CO)C1 N1(C(C(C)(C)CF)=O)CC(NC(=O)COCCF)C2(CC2)C1 C1(N(C(=O)CCOCCCN(C)C)CCC)CCN(C(=O)C(C)SC(F)(F)F)C1 c1(OCC)c(Cl)cc(C)nc1C(N1CCC(F)C(NC(c2cc[nH]c2C)=O)C1)=O CCC(CC)C(=O)N(C)CC1(NC(c2cn(-c3ccccc3F)nc2C)=O)CC1 N1(C(c2cnc(N)c(CO)c2)=O)CCCN(C(C2CCS(=O)CC2)=O)CCC1 C1(C(=O)NCC(C)(C)NC(CC(C(=O)OC)C)=O)CC12CCS(=O)(=O)CC2 C1(NC(C=C(CC)C)=O)CCCN(C(=O)CCC2C(=O)ON=C2C)C1C CCC(C(=O)NC1CCCC1NC(C1CCC(=O)N1)=O)OC C1(CC(C(=O)NC2CC2)N(C2CC(F)(F)C2)C)COC(C)(C)C1 c1(CC(N2CC(C)(NC(c3c(C(C)C)noc3)=O)C2)=O)cnc2n1CCCC2C c1(C(C)NC(=O)NC2C(CC(=O)OC)CCC2)ccc(OCF)cc1 C12(C(=O)NCCN(C)C(c3cc(C4CCCC4)n(C)n3)=O)CCC(CC1O)C2 CC(C)CC(=O)NCC1CC1CNC(=O)COC(F)(F)F c1(C(N2C(C)CCN(C(C(CC)(C)OC)=O)CC2)=O)ccc(C)c(S(N)(=O)=O)c1 N1(C(CC2C(C)C2)=O)CCCCC2(CCN(C(=O)Cc3cc(Cl)ccc3Cl)C2)C1 C(C(O)CC(=O)NCCOC1CCN(C(=O)CC(C)(C)C)C1)N(C)C C(=O)(C1=CC2(CCOC2)C1)NCCC1(NC(C(C2CC2)OC)=O)CC1 c1(C(N2CC3C(NC(c4cc(CC(C)C)[nH]n4)=O)(C3)C2)=O)cnc([N+](=O)[O-])n1C C=CC1OCCC1C(=O)NCC(C)(CNC(=O)Cc1cccnc1O)C1CCC1 c1(C(N2CCC(C(C)NC(C3(CC#C)CCOC3)=O)C2)=O)nc(O)nc(O)c1N C1(CC)C(NC(=O)CC2CCCOC2)CCCN1C(=O)Cc1ccnc(O)c1 c1(C(=O)NC2CC(NC(=O)CC3C=CS(=O)(=O)C3)C2)cc(Cl)cc([N+](=O)[O-])c1O N1(C(C(CCC)OC)=O)CC(NC(c2cn(CC)nn2)=O)C(S(C)(=O)=O)C1 CC(C)CC(O)CC(=O)N1CCC(CCNC(=O)COCC(C)C)C1 N1(C(C(COC)(C)C)=O)CC2(CC(CC(N3CCCNC(=O)C3)=O)C2)C1 CC1CCC(NC(C2CCCC2C2CC2)=O)CN1C(=O)Cn1cccn1 c1(-c2c(C)nc(NCC3CCCCO3)s2)cc(C)c2c(c1)CCC(=O)N2 N#CC1CN(S(=O)(=O)CC2CC2)CC1NC(C1(c2ccc(F)nc2)CC1)=O c1(C(=O)NC2C3CCN(C(CCN(C(C)=O)C)=O)C32)cc2cccc(F)c2o1 c1(NC(N2CCCC(C(=O)Nc3ccccc3)C2)=O)ccc(Br)c2ncccc12 N1(C(=O)Cc2cccnc2)C2CC1CN(C(c1cnc(Cl)c(Cl)c1)=O)C2 Cc1cc(C(=O)NC(CNC(C2(C)CCCO2)=O)C2CC2)c(O)c(C)n1 C1(OC)CCCC(C(=O)NCCCCC2CCN2C(C2CC(N3CCCC3)C2)=O)C1 N1(c2cc(OC)nc(OC)n2)CCC(NC(=O)CC2CCCCN2C)C12CCC2 N1(C(C2C(C=C(C)C)C2(C)C)=O)CC2OCCN(C(=O)Cc3ccsn3)C2C1 CCC(C)(C)CCCC(=O)N1CC(O)(C(F)C(=O)NC2CCC3CC23)C1 CC(C)CC(CNC(C12CC(C)(CO1)C2)=O)NC(=O)C(C)(F)CC1CCCC1 S(=O)(=O)(C1CC1c1ccccc1Br)NCC1(C(=O)OCC)CCC1 N1(C(CCCCC)=O)CCC2CCC(C1)N2C(C1CCS(=O)(=O)N1C)=O c1(OC)ncnc(C(=O)NC2COCC2NC(=O)CC2CC3CC3C2)c1F C#CC1CN(C(=O)CSS(C)(=O)=O)CCN1C(=O)CC=CC(C)(C)C C1(NC(c2cccc(C)c2Cl)=O)CCN(C(=O)Cc2scnc2C)CC12CCC2 C1(OC)(CNC(=O)C(CC)SC)CCN(C(=O)C(F)(F)c2nccn2C)C1 c1(C(=O)NCC=C)ccccc1NCc1ccccc1N1CCCC1 N1(C(c2cc(C#N)oc2)=O)CC2=C(C1)CN(C(c1ncnc(O)c1Br)=O)C2 c1(C(C(=O)NC(CC)CNC(=O)Cn2cnnn2)=O)cc(F)ccc1C C1(CC)C(C(N2CC(O)(CO)C2)=O)CCN1C(=O)CCn1cccc1 c1(N2CC3(C)CN(C(CSCCC)=O)CC3(C)C2)ncnc2c(Cl)cc(Cl)cc12 N1(C(CCSCC(=O)OC)=O)CC2CCN(C(C3OC(C)CC3C)=O)CCC2C1 C12(C(N3CCC(C)(NC(CNC(=O)OC)=O)C3)=O)CCC(CO)(CC1)C2 C1(C(N2CCC(C(=O)NC)CC2)=O)CCc2cnn(C)c2C1 c1(C(N(CCNC(c2noc3ncccc23)=O)CC)=O)cc(C)cc2ccoc12 N1(C(c2c[nH]c(=N)o2)=O)CC2(COC(CNC(C3Cc4nccn4C3)=O)C2)C1 CC1CN(C(=O)C(c2ccccc2)F)CC1(C)C(N1CCC1CC(C)(C)C)=O N1(C(C2C(C3(C)COC3)C2)=O)CCC(C(=O)N2CC3CC2CS3)=C(F)C1 N1(C(CC(C=C)CC)=O)CC2(C1)CN(C(=O)CC1=CCCCC1)CCO2 c1(NC2(CNC(=O)Cn3cnc(-c4ccccc4)n3)CC2)ccc(Cl)cc1Cl C1(C(=O)NC2CC(C)(CNC(COCC#C)=O)C2)CCc2nnc(C)n2C1 c1(C(N2CCC(C(=O)NCc3cnccn3)O2)=O)cccc([N+](=O)[O-])c1 CCC(C)CCCCC(=O)N(C)CC=CC(=O)NCC1CCCCC1C N1(C(C2CC(F)CN(C(=O)CSc3ccncc3)C2)=O)CCC2(CC1)COC2 C1(NC(c2c(CCC)n[nH]c2)=O)CCC(C)N(Cc2cc(-c3cccs3)on2)C1 c1(CC(=O)NCC2C(NC(C3C(C)CCC3)=O)C2)cc2ccccc2cc1O N1(C(CCCC#N)=O)CC(C2CCCN(C(C3CCC(C(F)(F)F)O3)=O)C2)C1 N1(C(C(n2c(C)ccn2)C)=O)CCC(N(CCO)C(C2CC2[N+](=O)[O-])=O)CC1 CCCC(C)C(C)(c1nnnn1CCCSC)NCc1cc(SC)nn1C N1(C(c2ccc(OC)s2)=O)CC2CCC(CNC(c3ccnnc3)=O)C2C1 N1(C(C(C)(C)SC)=O)CC2CCCC(CNC(=O)C=C(C)c3ccco3)C2C1 N1(C(c2c(N)cc(F)c(Cl)c2)=O)CC2CC(C1)CN(C(c1ccnc(S)c1)=O)C2 C(=O)(C(C(C)C)NC(=O)CCSCC(N)=O)NCCC(C)(C)OC C(=O)(C(CC(F)F)c1ccccc1)NC(CCN(C(c1nccc(C)n1)=O)C)C CC(C)(C)C#CC(=O)N1CCN(C(=O)Cn2cc(C3CC3)nn2)C(CC2CC2)C1 C1(N(C(CSc2nc(C)[nH]n2)=O)C)CCCC(N(C)C(c2nc(O)sc2C)=O)C1 C=CCC(CC(C)C)C(=O)NC1C2CCN(C(=O)C(O)CSC)CC12 Cc1nn(C)c(C)c1CC(N1CC2(CC2C(=O)Nc2nnnn2C)C1)=O C=CCCCC(C(=O)NC1COCC1F)NC(C1CC12CCOCC2)=O S(=O)(=O)(c1ccc(F)c(F)c1)NC1CCC(C(N2C(C(N)=O)CCC2)=O)CC1 c1(N2CCN(c3c(OC)nccc3)CC2)c(C)nc(C(=O)O)nc1C C1(C(=O)NC(c2ccoc2)C)CCCN(C(=O)C(O)c2cnc[nH]2)CC1 C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(CO)CCN(C(c2cncc(NC)c2)=O)C1 C1(C)(NC(CNC(CCCC)=O)=O)CCCC1NC(c1ccsc1COC)=O N1(C(CCc2cc(C)on2)=O)CCOC(C(C)NC(c2[nH]ccc2C2CC2)=O)C1 C1(C(=O)NCCc2ccccc2O)CCCCCN1C(=O)CC1CCC1 C1(CC(N2CC(CN(C(CCC(C)C)=O)C)OCC2)=O)CCCCC12CC2 c1(C(O)CNC(=S)Nc2ccccc2F)ccccc1[N+](=O)[O-] c1(C(C(=O)NCC(CCC)C)NC(=O)C=Cc2cncn2C)c(C)cccc1Br C1(C(=O)NC(C(=O)NCC2CN(CC)C(=O)O2)c2ccoc2)CC1C1(C)COC1 c1(C(=O)NC(C(=O)NCC(n2cc(C3CCC3)nn2)C)C)ccc(Br)o1 CCCC(CCC)CC(=O)NC1CCCN(C(c2ccccc2O)=O)CC1 C1(C(N(C2CCCN(C(C3CC3C(C)(C)C)=O)C2)CC)=O)CN2CCC1CC2 c1(CCN(CCCN2CCOC2=O)CCOC)c(F)cccc1F Cc1ccc([N+](=O)[O-])c(N(CCCNC(=O)Cn2cnc([N+](=O)[O-])c2)C)c1 c1(OC(C)C)cnccc1C(=O)NC(C)C(C)(C)NC(=O)Cc1cccnc1 c1(C(=O)NC(CNC(CCCSC)=O)C(C)C(C)C)cc2nc[nH]c2cc1N C(C(C)(C)CNC(c1nnn(C)n1)=O)N(C(=O)CCN1CCC(F)C1)C c1(CC(=O)N(CC(C)NC(CCC=CCC=C)=O)C)ccc(C#N)cc1F C(=O)(C(C)C1=CCCC1)NCC(=C)CCNC(=O)C1=CCCCC1 c1(C(N(CCNC(=O)CC2(C)CCCO2)CC)=O)n[nH]c2c1CN(C)CC2 N1(C(c2ncn(CC)c2)=O)CCN(C(c2ccco2)=O)C(C2CC2)C1 CCCCC(O)C(=O)Nc1ccc(C(=O)NS(=O)(=O)CC2CNC(=O)CO2)cc1 c1(CCCNCCO)c[nH]c2cnccc12 c1(C(N2C(CNC(Cc3scc(CC)n3)=O)CC2)=O)ncccc1C c1(C(=O)NC(CC)CNC(=O)C(C(C)C)N(CC)CC)cc(Cl)ncc1F N1(C(C2(C=C)CC2)=O)CCCC(C(=O)NCCNC(=O)CP(C)(C)=O)C1 CCC(C(=O)NC(C1CCN(C(c2cc(C(C)C)oc2C)=O)CC1)C)C(C)C C(C)(C)(CCCC(=O)NC1CN(CC)CC1C)NC(C(COCC)C)=O c1(NC(C(C(C)NC(C2C(=C)C2)=O)C)=O)ccc2nc[nH]c2c1 C1(C(=O)Nc2nc(O)cs2)CC2CCCCC2N1Cc1cc2cc(Br)ccc2s1 C12(C(N(CCNC(C(CCCC)O)=O)CC)=O)CCCCC1CCCC2 C1(NC(C2N(C(COCCSC)=O)CC=CC2)=O)CC=C(C(C)C)CC1 N1(C(C2C(=O)NCC2)=O)CCCCC1C(N1CCCC1C1CCCC1)=O N1(C(CCOCC)=O)CCC(NC(C2CC2Sc2ccccc2)=O)C1 N1(C(CCN(CCCCC)CC)=O)CCCC(CNC(=O)C(F)CC2CC2)C1 Cc1cn2cc(C(N3CCC(C(C)NC(=O)C4=CCCC4C)CC3)=O)nc2s1 O=C(C1=CC2C=CC(C1)C2)NC1(CNC(c2cncc(O)c2)=O)CCOC1 c1(CCC(=O)NC(CN(C(c2n(CC)ccc2)=O)C)C)c(F)cccc1Cl c1(CN2CCC(NC(C3(N=[N+]=[N-])CC3)=O)C2)nnc2n1CCCCC2 Cc1nc(CC2CC2)sc1C(=O)NC1C2CN(C(=O)CCC3CC(F)(F)C3)CC12 N1(C(C2(COCC)CC2)=O)CC2(CCCCN(C(=O)CCSCC)C2)C1 N1(C(C(C)CC2CC2)=O)CC(NC(c2ccc(-c3nccs3)cc2)=O)C(CO)C1 C1(CC)(NC(=O)CCN(C)CCO)CCN(C(C2(COC)CC2)=O)CC1 C(C)(C)(CCN=c1cc[nH]cc1S(=O)(=O)NC1CCC2CCCC1C2)OC N1(C(CCCC#CC)=O)CC2ON=C(CNC(=O)CCn3ccc(C)n3)C2C1 N1(C(c2c(SC)nccn2)=O)CCCN(CCNC(C2(C(F)F)CC2)=O)CC1 c1(C(C)=O)ncc(C(=O)N(C2CCN(C(=O)CCN(C(=O)CC(C)=O)C)C2)C)s1 c1(CN(C(=O)C(=O)NCCCc2cccnc2)CCN(C)C)ccc(F)cc1 C1(NC(c2ccc(OCCC)cc2)=O)CC(N=c2[nH]cnc3cc(I)sc23)C1 C1(C(=O)NC2CC(CNC(c3ccc(O)cc3Cl)=O)C2)CC2C=CC1CC2 C1(C(C)NC(CN(C)CC)=O)CN(C(=O)C(C)C(C)c2ccc(F)cc2)CCO1 CC1(C)C2CCC(C(=O)NCC3CC3CNC(C3(F)C(C)(C)C3(C)C)=O)C1C2 C1(CC)CC(C)CN(C(C2(C(C)C)CCCN2C(c2ccn(COC)n2)=O)=O)C1 Cc1nc(S)sc1CC(=O)NC(C(=O)NC1(C)CC(NC(=O)CN(C)C)C1)C(C)C Cn1nc2c(c1NC(C13CC1CN(Cc1ncccc1[N+](=O)[O-])C3)=O)CCCC2 C#Cc1cccc(C(=O)NCC2CC(F)(CNC(C3(F)CCOC3C)=O)C2)c1C C#CCC(C)(CNC(=O)CSCCNC(C1CCSCC1)=O)CO Cc1ccc2c(C(=O)NNC(C3(C)CCCS3(=O)=O)=O)[nH]nc2n1 Cc1cc(C(=O)NC2CCC2C(=O)NCCOCCCO)cs1 CC1(C)CC(CN(CCC(=O)NC)C(=O)C(=O)O)CN1C(=O)C1=CCOC1 CCC(C)C(C(=O)N(C1CCN(CCCOC)C1)C)NC(C)=O C(=O)(CC(C)CC(=O)NCc1ccc(C(N(C)Cc2ccccc2)=O)cc1)OC C1(O)(CCNC(=O)CC2(O)CCC2)CCCN(C(=O)CCc2cscn2)C1 N1(C(=O)NC)CCCC(N(C)C(C2CCCN2CCOc2ccccc2C)=O)C1 C(=O)(C(CCS(C)(=O)=O)OC)N(CCC)CCNC(=O)Cn1ncc(Cl)c1C CC1(C)CCCN(C(C2CCCCN2C(c2cncn2-c2ccccc2)=O)=O)C1 c1(CC(N2CCCC(CN(C)C(c3csc(=N)[nH]3)=O)C2)=O)ccc(F)c(F)c1 c1(C(=O)NC(C)C(=O)N(C)CC2CCOC2)cncn1C c1(NCCN(C)C(C2CC2OC(C)(C)C)=O)cc(=O)n(C)c(=O)n1C N1(C(C2=CC(C)(CC)C2)=O)CC2(CCN(C(=O)CC3CC(C(C)(C)C)C3)C2)C1 C1(C(N2CCC(C(C)NC(=O)C(F)CC(C)C)CC2)=O)(OC)CCCCCCC1 C12(C(=O)NC3C(C)(C)CN(c4nc(Cl)c(C#N)s4)C3)CC3CC(C1)CC(O)(C3)C2 C1(CNC(C(C(=O)OC)C)=O)CN(C(c2cc(CC(C)C)on2)=O)C(C)(C)C1 N1(C(C2CN(C)C2)=O)CCOC2(CCN(C(C3CCCCS3(=O)=O)=O)C2)C1 n1(C(C(N2C(C)CC(NC(CCC=CCC=C)=O)C2)=O)C)nc([N+](=O)[O-])cc1C C1(CC)CN(C(=O)Cc2ccc(C(C)OC)cc2)CCN1C(=O)C1=C(C)OCC1 c1(CCC)cc(C(=O)NC2CC(CCNC(c3ccnc(S)c3)=O)C2)n(C)n1 C(C(CC(C)C)C(=O)NC(C)CC1CC1)NC(CCCOCCC)=O N1(C(CCCCC)=O)CC(CNC(C2(C)CC2)=O)OC(C)(C)C1 N1(C(Cc2scc(C)c2)=O)CCCC(F)(C(=O)NCCCN2CCOC2=O)C1 C1(F)(C(=O)NC(CN(C(=O)CNC(c2ccncc2)=O)CC)C)CCC(=O)CC1 CCCC(C)(CC)C(=O)NC1CCCCCC1C(N1CCCC2(CC2)C1)=O Cc1ccc(CC(=O)NCc2nc(C)c(C(=O)NC3CCCCC3C)o2)cc1 C(=O)(CCCCCNC(C1C=C(C)CS1)=O)NCC1CC(OC(C)(C)C)C1 c1(C(N2CC(N(C(c3cc(C)ncc3)=O)C)C(C)(C)C2)=O)cn(C)c(=O)cc1C CC1(C)CN(C(c2nocc2Cl)=O)CC1NC(=O)CC1CC1(Cl)Cl C=CCC(C(=O)NC12CCC(NC(=O)CC(=O)OC(C)(C)C)(CC1)C2)C(C)C CCCC(C)(C)C(=O)OCC(=O)NC(C1CN(C(N)=S)C1)=O CC1(C(N2CC(NC(C3(c4cccs4)CC3)=O)C3(CC3)C2)=O)CCCS1(=O)=O C(=O)(CS(=O)(=O)N(C)C)N1CC(CC(c2ccccc2)NC(CCCC)=O)C1 N1(CCO)CC(S(=O)(=O)N2CCOCC2)C1.Cc1n[nH]cc1Cc1nnnn1C C#CC1C(C(=O)NCC(C)(C)CN(C(=O)CC=C(C)C)C)C1(C)C c1(NC2CC3CN(C(C(CC)OC4CCCC4)=O)CC32)ccc(Br)c(C)c1[N+](=O)[O-] C1(CC(=O)OC)CC2(CCN(C(=O)OCc3ccc(C(C)(C)C)cc3N)C2)CO1 c1(C(=O)NC2CN(C(C3(OC)CCSCC3)=O)CC2C)ccc2c[nH]nc2c1 N1(C(C2(OC)CCOC2)=O)CC(NC(C2CCSCC2)=O)CC(F)C1 C(=O)(CCCCC(c1nnnn1C1CC1)NCCn1ccccc1=O)N(C)C c1(C(=O)NCCC(C)N(C(C#CC(C)C)=O)C)cc2cccnc2nc1N C(=O)(C1=CCCCC1)N1CC(CCC=C)(C(=O)NC(C)CC2(O)CCC2)C1 N1(C(Cc2ccc(C)s2)=O)CCOC2(CCC(NC(=O)CC(C)N(C)C)CC2)C1 C1(O)(CNC(c2ccsc2)=O)CC(NC(c2cn(CC3CCOC3)nn2)=O)C1 N1(C(COCCCOC)=O)CCC(C)(C(=O)NCC(C)(O)CCO)CC1 S(=O)(=O)(c1ccc(Cl)cc1)N1CC2(C1)C(=O)N2.c1(-c2cccs2)cc(Cl)nc(Cl)c1 C1(CC(C)NC(=O)C(O)CC2CCOCC2)CCN(C(=O)CC2CS(=O)(=O)C2)CC1 CC(C)(CCNC(C1C=CCCC1)=O)NC(=O)CCCC1CC1 c1(C(=O)NCC(=O)NCC(CSc2ccc(O)cc2)OC)cncc(C2CC2)c1 C1(C(N2CCOC(C3CC3)C2)=O)C2C3CC4C1C2C34C(=O)NC1CC(O)C1 N1(C(c2c(SCC)cncc2)=O)CCN(C(C2(F)CCCC2)=O)CC(O)C1 S(=O)(=O)(c1cc(C(=O)NC2COc3ccccc3C2)ccc1Cl)N(C)C C1(F)(C(N2CCC(N(C)C(c3cncc(C(F)F)c3)=O)CC2)=O)C2CCCCC12 c1(C(=O)NCC2(F)CN(C(C3CC4CCC3O4)=O)C2)cccc2ccncc12 C1(CC)C(NC(=O)Cc2cc(F)ccc2C)CCCN1C(c1coc(Cl)n1)=O c1(NC(C)=O)cnccc1C(N1CCOC(CC(N2CC(C)(C(N)=O)C2)=O)C1)=O c1(N2CCC(C)(C#N)C2)nc2ccccc2c(=NCc2cc(Br)cc(Br)c2)[nH]1 N1(C(c2ccc(CCC)cc2)=O)C2CCC1CC(NC(C1CSCC(=O)N1)=O)C2 C1(C(N2C(CN(C(=O)CC3CC4(COC4)C3)C)CCC2)=O)CSCC(=O)N1 C#Cc1ccnc(C(=O)NC2(COC)CCN(C(c3ncn(C)n3)=O)C2)c1 CC1CN(C(c2ccc(F)s2)=O)CC1CC(N1CCSC(C)C1)=O c1(NC(C(C)C)C)ccc(C(F)(F)F)cc1S(=O)(=O)N(C1CN2CCC1CC2)C c1(CO)ccc(S(=O)(=O)NCCCCN2CC(Oc3ccc(Br)cc3)C2)cc1Br CN1CCC(C(=O)N(C2CN(C(C34CC(C)(C3)C4)=O)CC2O)C)C1=O CC(CNC(c1cc(CO)ccn1)=O)CC(=O)NCC(C)C#N C(C(=O)NCCN(C(=O)C(F)(F)c1cncs1)C1CCCCC1)(C(C)C)SC c1(NC(c2ccc(NC(C3CC3F)=O)c(F)c2)=O)nccc2ccccc12 C1(NC(c2cc(OCC)no2)=O)CN(C(=O)C(F)C2CCOC2)CCC12CCC2 C12(C(C)C)CCN(C1)CCNC(=O)CCCNC2=O.C1(CC)CCC1 Cc1c(C(=O)NCC(C)CNC(=O)CCc2ncccn2)sc(Cl)c1Cl CC1(C)OCc2c1n[nH]c2C(=O)NC1CCCN(C(c2coc(C3CC3)n2)=O)C1 C=CC(C)(CCOC)C(=O)NCC1(F)CCC(NC(=O)CN2CCCNC2=O)C1 C1(CNC(=O)C=C2CCCCC2)C2CCC2CN1C(=O)CC1CCCO1 c1(CC)[nH]nc(Cl)c1C(N1CCCC(CNC(C2(SC)CC2)=O)C1)=O C(C(=O)NC(C)CC(C)NC(=O)CN1CCCCC1=O)(C(C)C)SC c1(OC)cc(C(=O)N(C(C)CNC(=O)CCc2cnoc2)C)cc(F)n1 c1(SCC)cccc(CC(=O)N(CCN(C)C(C2CC(O)C(F)C2)=O)C(C)C)c1 C(=O)(C1=NN2CC(C)CN=C2N1)N(CCNC(c1ncn(C(C)C)n1)=O)C1CC1 c1(C(=O)NC2CCC(CNC(c3c(C)[nH]cc3)=O)C2)ccc(-c2cnco2)cc1 C(CC(CNC(C1C=CCCC1)=O)NC(c1ccsc1Cl)=O)OC Cc1c(C(N2CCN(C(=O)CC(C)NC(N)=O)C(CO)C2)=O)ccc2c1CCC2 C(=O)(CCC(=O)N1CCC(O)CC1)N(C)CC1CCCN1C(C1(F)CC1(F)F)=O C#CCC(C)C(=O)NC(C1CCCC1)CNC(=O)Cc1csc(C2CCCC2)n1 C12CCN(C1)C(=O)NC2=O.c1(C(C)CN(C)Cc2cocn2)ccccc1.NC N1(C(CC2CC(OC)C2)=O)CCC(CNC(=O)Cc2nn(C)cc2Br)CC1 c1(C(N2CCCC(NC(c3ccc(C)cc3C)=O)C2)=O)ccc2ncc(Br)n2c1 c1(C(=O)NC(C(C)NC(CC=C=C)=O)CO)cn(C)nc1C1CCCC1 C1(NC(C2C(C)CCS2)=O)CCN(C(=O)C=Cc2ccsc2Br)CC1 c1(CCC(=O)NCC(C)CNC(C2(C)CNC(=O)C2)=O)cnc2n1CCOC2 c12ccc(cc1)CC(=O)C2=O.C(=O)(CC(C)CF)NC1CC(C(C)=O)C1.CCCCN c1(C(=O)NCC2CN(C(C3(OCC)CCOCC3)=O)C2)cc(C(C)C)ccc1N C=CC(C)(C)C(=O)N1CCC1CNC(=O)C(Cc1ccc(F)cc1)N(C)C Cc1ccc(CC(=O)NCC2CC2NC(c2nc(=N)cc[nH]2)=O)cc1Br N1(CCc2ccc(C(=O)OC)cc2OC)CC(C)CS(=O)(=O)CC1 N1(C(C2N(CC)CCC2)=O)CC2CC(C1)N(C(=O)Cn1nnc(C(C)(C)C)n1)C2 c12cnc3ccc(nn13)[nH]c2=O.C=CC(C)(O)CC(=O)N1CCN1C=O C1(C(N2CC(OCCNC(=O)C(c3cccc(F)n3)(F)F)C2)=O)CCC(F)(F)C1 Cc1cc(O)c(C(=O)N(C2CN(C(c3ccc(F)c(F)c3)=O)CC2F)C)nn1 c1cc(F)cc(Cl)c1.c1(C=O)cccc(I)c1O c1(C(=O)NCC2(CCNC(C34C=CC(CC3)C4)=O)CC2)c(F)ccc2occc12 c1(C(C)C)cc(C(=O)NC2CC(N(C)C(C3(C4CCC4)CC3)=O)C2)cc(O)n1 C1CN=C2N=C(C=C(C)N2)N1c1ccccc1.N1(C(C)=O)CC(OC)C1 c1(CNC(CC2CCN(C(C3(N(C)C)CCC3)=O)C2)=O)ccc(F)cc1F C1(NC(C2OCCN(CC)C2)=O)CN(C(C2CCC(CC)CC2)=O)CC1C1CC1 c1(C(=O)NCCC(C)(C)NC(C2C(C)(C)C2(F)F)=O)cncc2cnccc12 CC1CCCCC1(CNC(c1ccc(CO)nc1)=O)NC(=O)CCC1CC1(C)C O=C(C#CC1CCCC1)NCc1cc[nH]c1C(=O)NC(C1CCOC1)CO c1(CC)ccc(C(N2CC(N(C(=O)CC3(CO)CC3)C)C2)=O)cc1CC Cc1cc(CC(N2CCC(NC(=O)COCP(C)(C)=O)C(F)C2)=O)cc(C)c1 C(=O)(CC(C(F)(F)F)n1cccn1)NCCC1CC(OC)CN1C(=O)CO C1(C(N(C)CC2CCN(CC)C2)=O)CC(O)CN1C(c1oc(C)cc1C)=O C(CC(C)C)(C(=O)NCC=CCOC)NC(CC1CC(OC)C1)=O c1(C(C)C)ccc(CC(=O)NCC(F)CNC(C23CCC2C3)=O)cc1 N1(C(C2C(=C)CC2)=O)CC(NC(c2c(C)cc(C)oc2=O)=O)CC12CCCCC2 CC1CCC(F)(F)CN1C(=O)C(Cc1cc[nH]n1)NC(=O)C=CC(C)(C)C C(=O)(C1=C(C)N(C)c2ncnn2C1)NC1C(C#C)C1 c1(OC)cccc(C(N2CC(O)(CNC(C3CCCS(=O)(=O)C3)=O)C2)=O)c1OC c1(C(N(c2nnc(-c3ccccc3)s2)C(C)C)=O)cc(Cl)c(Cl)s1 C1(C(=O)NCCNC(CN(CCC(C)(C)C)C)=O)CC2(CCC2)CO1 C1(C(=O)NCC2(OC)CCOC2)CCN(C(=O)C(C)CC2CC2)CCO1 C1(C)(NC(C(C(C)CC)NC(c2cccc(CC)n2)=O)=O)CCCCC1(C)C c1(CC(=O)NCCNC(CCCCC#N)=O)ccc2c(c1)CCC2 C1(NC(CCCC)=O)CCN(C(=O)Cc2cc(C)cc(F)c2)C(C)C1 c1(CC(=O)NCCC2CCN(C(C(CCC)CC)=O)C2)coc2ccc(C)cc12 c1(C(=O)NCC2(CO)COC2)cc2ncc(-c3cccnc3)cc2[nH]1 N1(C(CNC(=O)NC)=O)CC(NC(=O)CC2(CO)CCC2)CC12CCOC2 CC(CC(=O)N1CCC(C(C)(C)C(=O)NCc2cnccc2Cl)C1)C(F)F c1(C(=O)NCC2CN(C(c3c(OC)scc3)=O)C(C)CC2)cc(F)c(C)cc1O c1(C(=O)NC2C(NC(Cn3c(C)ncc3)=O)COCC2)cc(O)nc(O)n1 C1(C(=O)NC(c2cnn(C)c2)C)(CO)CCCN(C(=O)CCc2nncs2)C1 c1(C(=O)NCC2CN(C(c3c(OC)cccc3)=O)CC2C)cc(C)nnc1O c1(OC)ccc(NC(=O)C(N2C(C)CN(C)CC2C)=O)c(C(=O)NC2CC2)c1OC Cc1cc(C)c(C(=O)NC(C2CC2C(=O)NC(C)Cc2ncn(C)n2)C)cn1 c1(CN2CC(NC(C3CCCN(C)C3)=O)C(F)(F)C2)cc(F)c(F)cc1O C1(CC(=O)NCC2(CNC(=O)CC3CCCC34CC4)CC2)CCCC2(CCC2)O1 CC1CC2(C(=O)NCC3CCCN3C(c3cocc3C(N)=O)=O)CC12 C1(CNC(c2c(CC)n(C)cc2)=O)CN(C(=O)C(C(C)C)OC)CC1(C)C CC(O)(CNC(=O)CCC1CCCOC1)CNC(c1ccoc1)=O CC1CN(C(=O)CC2COCCN2C(=O)Cc2ccc(Cl)cc2F)CC(C)O1 CCC(CC)(CN=c1[nH]c2c(c(=NC3CCS(=O)(=O)C3)[nH]1)SCC2)OC c1(C(=O)NC2CCC(NC(C(C)=C3CC3)=O)CC2)ccc(C)c2c1CCC2 N1(C(c2nc(COC)sc2)=O)CC(F)CC1CNC(=O)CC1CCCC(C)C1 C1(CNC(c2c(C)nn(C(C)C)c2)=O)CC2(CC2)CN1C(=O)Cn1ccsc1=N CC1CC2(CCN(C(=O)C3=CCN(C(C4CC5CCC4CC5)=O)C3)C2)C1 Cc1cc(C(N2CCN(C(c3ncsc3C)=O)CC2CCO)=O)c2occc2c1 C1(CNC(c2cnc(C)[nH]2)=O)CCCCN1C(=O)CNC(=O)CN(C)C CN1CCC(C(=O)NCC2(O)CCOC2)(NC(c2cc(C(F)F)[nH]n2)=O)C1 C1(C(=O)NCC2C(CNC(c3cnn(CCC(F)(F)F)c3)=O)C2)(CO)CCCO1 c1(C(=O)OC)ccc(C(N2CC(CC(N)=O)(NC(c3cccnc3)=O)C2)=O)cc1 C#CCCCCCCCC(=O)N1CCN(Cc2ncnn2CC)C(C)C1 c1(C(=O)NCC(C)(O)CNC(c2cnccc2Cl)=O)nc2cccnc2s1 C(=O)(C1c2ccccc2CN1C(c1ccc(C)nc1Cl)=O)N(CC=C)CC=C CCCC(C)(CCC)C(=O)NC1CCN(C(c2csc(-c3ccccn3)n2)=O)C1 N1(C(Cc2cccc(C)n2)=O)CC2CCC(NC(=O)C(c3ccccc3)C)C2C1 c1(C(=O)NCC=CCNC(C2(n3cccc3)CC2)=O)ccc2scnc2c1 c1(C(=O)NC2C(NC(CCC#C)=O)CCCC2)cnn2ccc(Cl)c(F)c12 c1(C(N2CC(NC(c3c(OC)n[nH]c3)=O)C2)=O)c(C)nc(O)nc1C C(=O)(C(F)CC(C)(C)NC(c1ccc(F)s1)=O)Nc1ccc(COC)cc1 C1(CNC(c2c(Cl)cc(C)s2)=O)CC2CCC(C1)N2C(=O)CC1CNC(=O)C1 c1ccccc1.c1(C(C(=O)NC)NC(C2CSC2)C)ccc(I)s1 C1(C(=O)NCC(CC)OCC)CN(C(c2cc(CO)n(C)n2)=O)CC1(C)C C1(N(C(CC2C(C)=NNC2=O)=O)C)CN(C(c2cnsn2)=O)CC12CC2 c1(COC)nc(Cl)cc(=NCCC(C)NC(=O)CS(=O)(=O)N(C)C)[nH]1 CCCC(C(=O)N1CC(C)(C(N2CCC(O)CC(C)C2)=O)C1)C(C)C C(=O)(C1=CCCC1)N1CC(COC)(CNC(=O)CCNC(C)=O)C1 c1(CN(C)CC2CC(OC(C)(C)C)C2)ccc(-c2ccco2)cc1F N1(S(C)(=O)=O)CCN(C(=O)C(F)=CCCF)CC1.C12CC(C1)N2 CN1CCN(C(c2ncccc2N)=O)C(CNC(C2CC3CC2CO3)=O)C1 c1(OC)oc(C)nc1C(N1CCC(C(=O)NCCN2C(=O)CNC2=O)C1)=O C1(NC(C2C(=C)C2)=O)CCC(NC(c2oc(CCC)nc2C)=O)CC1 CC1(CNC(c2ccc3c(c2)CCO3)=O)COCCN(C(C2(C)CC2(Cl)Cl)=O)C1 C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(c2cn(CCF)nn2)=O)C1(C)C c1(-c2ccc(C(N3C(C)(C(=O)Nc4cscn4)CCC3)=O)o2)cccc(F)c1O c1(C(N2C(CNC(c3c(Cl)ccc(NC)c3)=O)CC2)=O)ccnc2cc[nH]c12 Cc1oc(C(F)(F)F)nc1C(=O)NC1CCC(NC(C2CCC2(C)C)=O)C1 C(=O)(C1CCc2cccnc21)N(CC(C)CNC(c1cccc(=O)n1C)=O)C c1(CN(C2CC(C#N)C2)C(C=CC(CC)C)=O)cccc(NC)c1.C12CN(C1)C2 C1(c2nnnn2C2(C)CC3(CCC3)C2)(NCc2c(C)csc2)CCC(=O)NC1 CC12CC3(C(=O)NCCOCCNC(=O)CCC4CC4)CC(C)(C1)CC(C)(C3)C2 N1(C(CC2CCC(C)(C)CC2)=O)CC2(CCCN(C(=O)CN3CCSCC3)C2)C1 c1(C(N2CC(NC(c3cc(Cl)c[nH]3)=O)CC(C)C2)=O)cc([N+](=O)[O-])ccc1Cl CC(O)(CNC(c1cnc(C2CC2)o1)=O)CNC(C1(n2nccn2)CC1)=O C=CCC(C(=O)NCC1CC2CC2N1C(C1CN(C(C)C)C1)=O)c1ccccc1 CC1CN(C(c2c(N)cccc2F)=O)CCC1CNC(=O)CCCC(=O)C1CC1 CCC(CC(=O)NC(C)CCNC(=O)C(C(C)O)N(C)C)C1CC1 n1(CC)cc(C(=O)C(=O)NC2(CN(C(=O)C(C)NC=O)C)CC2)cn1 c1(NC(C(N2CCc3sccc3C2)CCC)=O)cc(C)cc([N+](=O)[O-])c1N CC1CCc2nc(CNC(=O)CCn3ccc4ccccc34)sc2C1 C(C(C(C)C(C)C)NC(=O)CCCCCF)NC(c1ccc(N(CC)CC)nc1)=O Cc1ccc(Br)cc1C(N1CCC(C2CCCN2C(C2CN(S(N)(=O)=O)C2)=O)C1)=O c1(CNC(c2n(C(CC)(C)C)nnn2)c2ncc(CO)s2)ccncc1C C1(C(N(CC(C)(C)NC(c2ccc(C)s2)=O)C)=O)CC2(CC2)CO1 Cc1ccncc1CC(=O)NCC1CCCN(C(c2cnc(N(C)C)cn2)=O)C1 C1(O)(C(=O)NCCC(C)NC(CN(C)CC)=O)CCc2cc(Br)ccc2C1 C(CCCCCNC(=O)C(C)(C)CO)NC(C1C(C)CC1C)=O N1(C(C(C)OCC#C)=O)CC(NC(c2ccc(Cl)cc2CC)=O)C(N=[N+]=[N-])C1 CC(C)(C#N)CCC(=O)N1CC(F)(F)CC1CCNC(=O)C=Cc1ncc[nH]1 c1(OC)ccccc1N1CCN(Cc2nc(C(C)(C)C)co2)CC1 c1(N2CCC(O)C(C3CC3)C2)ncnc2cc(C(F)(F)F)ccc12 c1(OC)[nH]c(=NC(=O)c2csc(C)c2OC)ccc1Br c1(C(=O)NC2CN(C(CC3CCC(C)CC3)=O)CC2O)cnc2[nH]ccc2n1 C1(NC(CC(C=C)C)=O)CN(C(c2cc(C3CC3)ncc2Cl)=O)C2(CCC2)C1 C=Cn1nncc1C(=O)NCC(CC(=O)NCCC1C=CCC1)C1CCC1 C=CCC(CC=C)C(=O)NC1CCC(C)(CNC(=O)CC(C)=C(C)C)C1 c1(NC(CCN(C)C)(C)C)nc2c(c(=NCc3ncc(Cl)cc3F)[nH]1)SCC2 c1(CCNC(C(C2CCCO2)NC(c2ccco2)=O)=O)ccccc1F c1(C(=O)NCCC(CC)(C)NC(=O)C(C)Cc2cnc[nH]2)cccc2ccoc12 c1(C(N2CC(O)(CN(C)C(C3CC4CC3C4)=O)C2)=O)c(C2CC2)cnn1C C(=O)(C1CCCc2sc(=N)[nH]c21)NCC1N(C(C23CCC(C)(C2)CO3)=O)CCC1 C(=O)(C(COC)N(C)C)NCC(CC)NC(=O)Cn1ccsc1=N C1(C2CCCO2)(C(=O)NCC2CN(C(C34C(C)(C)OCC3C4)=O)C2)CCCO1 N1(C(c2cc(C)c(C)o2)=O)CCCCC(NC(=O)C=Cc2cccn2C)C1 c1(CC)cccc(C(=O)NC(c2ccccc2)CNC(=O)CC2CC2(C)C)n1 c1(C(N2CCC(CNC(c3n(CC)ncn3)=O)C23CC3)=O)cc(Cl)c(F)c(Cl)c1 N1(C(CC2(OC)CN(C(C3(C#N)CCCCC3)=O)C2)=O)CC2CCCC(O)C2C1 C1(C(N(CCCCCCNC(C2(CO)CCCCC2)=O)C)=O)CCCCN1N=O C1(NC(C(C(CNC(C2(C=C)CCCCC2)=O)C)F)=O)CCc2n[nH]cc2C1 c1(OC)ccc(CC(C)(O)CNC(C)C(F)F)cc1OC N1(C(C(=O)N2C(C(=O)OCC)CC2)CCC2CCCCC2)CCn2cnnc2C1C C=C(C)C(C)(C)C(=O)N1CCC(CCNC(c2c[nH]ccc2=N)=O)C1 C(CC(C)(C)C(=O)NC(C1CCN(C(=O)Cc2c(F)cccc2F)CC1)C)SC C1(NC(C(C2CC2)OCC)=O)CCCCC1CNC(=O)C(C(C)C)n1cnnn1 c1(C(=O)NCC2(F)CC(NC(c3c(OC)n[nH]c3)=O)C2)csc(C)c1C1CC1 CC(C)C(C#N)C(=O)NCc1cc(C(=O)NCC(c2ccsc2)C)on1 CC(C)C(O)CC(=O)NC1CN(C(=O)CC(C)C2CCCCC2)CCC1C(C)C C1(C(N(CC(CCC=C)O)C)=O)C(C2CC2)CCN1C(C1CCN(CC)C1)=O C1(C(=O)NC(CSCC)C(=O)Nc2ccc(Cl)c(O)c2)CC2(C1)CC(O)C2 CCCC(CCC)CC(=O)NCCCC(CO)NC(=O)CC=C(C)C CC1CCN1C(=O)C(C1CC1)NC(=O)Cc1ccc[nH]1 C(=O)(C1=C(C)OCC1)N1C2CC(NC(C3CC(=C)C3)=O)(C2)C1 CCCCCC(C)CC(=O)NC1CC(NC(c2cc(Cl)nnc2O)=O)C1 C1(CNC(c2cnc(O)s2)=O)(NC(C2CC(CCO)C2)=O)CCOCC1 C1(F)(C(N2CCC(NC(c3c(C)oc(C(F)(F)F)n3)=O)C2)=O)CCC(F)(F)CC1 CCCCC(CC)C(=O)N1CCC(C)(NC(c2ccc(NC(C)C)cc2)=O)CC1 c1(C(=O)NC2(CF)CCN(C(c3c(C)ncn3C)=O)C2)cc2cccn2c(O)n1 CC1CCCc2ncc(C(N3CCN(C(=O)C(F)=C4CCC4)C(C)C3)=O)n21 CCCC(C)(C)C(=O)NCC(F)CNC(=O)Cn1nnc(C(C)(C)C)n1 c1(NC)cnncc1C(N1CCOC(C(C)NC(=O)CN2CCOCC2)C1)=O c1(SCC(=O)NCC2(F)CCN(C(C(C)(C)O)=O)C2)cc(=O)n2ccsc2n1 O=C1CCCC(C(=O)NC2CCOC(C(N3CCC4(CC4)C3)=O)C2)C1 C1(NS(CCOC)(=O)=O)CC2(CC2)CN1CCN1CC2(COC2)C1 CCC#CCCNC(=O)C(CO)N(C)C.C12(CC(COC)C1)C(=O)N2 n1(CC(=O)Nc2c(C)cc(NC(=O)C(C)N(C)C)cc2)c(C)nc2ccccc12 c1(C(=O)NC(CC=C)CNC(c2cnc(O)o2)=O)cccc2c1ccn2C(C)C c1(C(N2CC(CC(=O)Nc3n(C)nnc3)OCC2)=O)ccc(Br)c(Br)c1 c1(N)ccc(C(F)(F)F)cn1.C1(C(=O)NCC(C)NC(C2CCCO2)=O)CC(CF)C1 C1(CC)CN(C(=O)C(C)(C#N)CC)CCN1C(=O)COc1ccc(C)cc1 CC1CCSCCN1C(=O)CCN(C)C(C1CCC(=O)NC1)=O N1(C(c2n(C)cnc2)C(=O)NCC2CCCO2)C2CCCC1CC(=O)NC2 c1(C(N2CCC(OC3CC3)C2)C(=O)NCC(F)F)cccc(-c2ccccc2)c1 C1(C)(C(=O)NC(C(=O)N(CC)CC)C)CCN(C(=O)CCCn2ccnc2)C1 c1(C(=O)NCC2C(NC(COCC(C)C)=O)COC2)cc2c(F)c(F)ccc2[nH]1 C1(C)(CC(=O)N(C(CNC(c2cc(CO)[nH]n2)=O)C2CC2)C)CC1(F)Cl S(=O)(=O)(c1cnc(Cl)nc1)N1CC2C(C(=O)NCc3cccc(Cl)c3F)(C2)C1 CN1C(=O)c2ccccc2C1CC(=O)NC1CCC(NC(=O)Cc2ccsn2)C1 c1(CC(=O)NC2C(NC(C3C(C)CC=CC3)=O)CC2)ccc2nc[nH]c2c1 c1(CC(N2C(CO)CC(NC(C(C)(C)OC)=O)C2)=O)ccc(CO)c(C)c1 N1(C(Cc2c(C)occ2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)C2CCCCC12 C(=O)(C1=NOC(C)C1)N1CCC(CC(=O)NC(c2c(C)cccn2)C)CC1 N1(C(c2cc(SC)oc2)=O)CCC(CCc2ccccc2)CC1.C(=O)(C)NCC1CC1 N1(C(c2c(OC)csc2)=O)CCCC(O)(CNC(c2cccnc2N)=O)C1 c1(C(N(C(C)C(=O)NC2(CCC)CCC2)CCC)=O)cc(C)c(O)nn1 c1(C(c2nnnn2C(C)C)NCCc2onc(OCC)n2)nc(C)[nH]c1Br C12(CNC(C3CCN(CCO)C(=O)C3)=O)CCCC1CN(C(c1cnsn1)=O)C2 N1(C(CC=C=C)=O)CCC(C)(CC(=O)NC(C)Cc2nncn2C)C1 C1(CN(c2cnn(C)c2)C(=O)OC)COC2COCC12.C1CC(=O)N1.C1(=O)CO1 Cc1ccccc1NCC1CCCCN1CCC1C=CCC1 N1(C(c2c(OC)n[nH]c2)=O)CC(CNC(=O)Cc2cncnc2)C(F)(F)C1 N1(C(CCC)=O)CCCOC(CNC(=O)CSc2nccn2C)C1 N1(C(CCNC(C)=O)=O)CCC(C)(CNC(C2CC2c2ccc(F)cc2)=O)CC1 C1(C(N(CC2N(C(C3CCC(CC)O3)=O)CCC2)CC)=O)CCC(C)C(C)C1 C=C(C)CN=C(NCC(c1c(C)noc1C)C)N1CCOCC2(C1)CC2(F)F c1(CCC)cc(C(=O)N(C)CCOCCC(=O)NCCCc2nncn2C)no1 C(=O)(C1Cc2ccccc21)NC1C(CNc2nccc(C(=O)OC)n2)C1 C1(C(=O)NCCCCCCN(C(c2cc(COC)on2)=O)C)CCS(=O)(=O)CC1 c1(C(=O)NCCCN(C(CCN(CCC)C)=O)CCC)ccc2oc(S)nc2c1 C(CCNC(C1(CC(C)=O)CC1)=O)(C(=O)N1CCCC1CCC(C)C)OC C(=O)(C1COc2ccccc21)NC1CCN(C(Cc2c(OC)ccc(Cl)c2)=O)C1 C1(CNC(C=C(C)CNC(=O)COCC2CC2)=O)CC2(CCC2O)C1 C(C)(C(O)C(=O)N1CC(O)(CNC(c2ccnc(C3CC3)c2)=O)C1)SC N1(C2CCN(C(C=CC=CC)=O)CC2)CCN(C(c2scc(C)c2Cl)=O)CC1=O c1(C(N2CCC(CNC(C3CCCC(C)C3)=O)C2)=O)cn2cccnc2n1 c1(N2C(CNC(C(C3CCCCO3)C)=O)CC2)nccc(-c2ccnn2C)n1 N1(C(C2(C(=O)OCC)CC=CC2)=O)CCCC(CNC(c2cc(=O)cc[nH]2)=O)C1 Cc1ccccc1C=CC(=O)NCC1CC1CNC(C1(C(C)(C)C)CCC1)=O N1(CCOCCC)CC(CN=[N+]=[N-])C(C)C1 c1(CC(=O)NC(C2CCOC2)CNC(C)=O)c(C)cc(C)c(C)c1Br C1(NC(c2cccc(OC(F)F)c2F)c2n(CCSC)nnn2)CCCOC1(C)C C1(NC(CCCCC(C)C)=O)CCC2(CCCN(C(c3ccsc3)=O)C2)C1 C1(NC(C(CSC)C)=O)CC2(CCCCN2C(C2(O)CCCC(C)CC2)=O)C1 CC1OCCCC1C(=O)NC1CCCC1NC(C1(c2ccon2)CC1)=O C1(CC)C(NC(=O)Cc2nnc(C)o2)CCN1C(=O)C=CCOC1CCOCC1 C1(C)(C(=O)NC(C)(C)CCNC(c2cnc(-c3ccncc3)s2)=O)CCC(=O)C1 CCC(C)(CNC(=O)CCC1CCOCC1)NC(=O)COC1CCC1 N1(C(Cn2cnc(C#N)n2)=O)CCOCCC1C(=O)NCC1CCC(F)(F)C1 c1(C(N(CCCN(C)C(c2cc(C#N)ccn2)=O)C)=O)cc2cccnc2cn1 N1(C(CCOCC)=O)CC(NC(=O)CCc2cnccn2)CC(F)C1 C1(NC(=O)OC(C)(C)C)CCOCC1C(=O)NCCNC(c1ncccn1)=O C1(C(=O)NC2CCC(C(=O)NCC(=O)OCC)C2)CC2(C1)CC2(F)F c1(C(N(C2CCCN(C(=O)C3=NNC(=O)C3)C2)CC)=O)cc(C)nc(C)c1 C(c1cccc(CO)c1)=CC(=O)NCC(CNC(CC1C(C=C)C1)=O)C N1(C(CCC2CC(CC)C2)=O)CCN(C(=O)CCn2cnnn2)CC1C1CC1 c1(C(=O)NC23CC(CNC(=O)C=C4CCC4)(OCC2)C3)ccc2nnn(O)c2c1 C#CC1CC2(CC(C(=O)NCC3CCCN3C(=O)C(O)Cc3ccccc3)C2)C1 N1(C(=O)C=CI)CCC(C(F)F)(CNC(c2cc(-c3ccccc3)ncn2)=O)C1 N1(C(c2ncn(-c3ccccc3)n2)=O)CCC(O)(C(=O)Nc2cnnc(Cl)c2)C1 Nc1ccc2c(c1)CCC(C(=O)NC(c1c(F)cccc1F)CC1CCCC1)C2 C1(NC(C(N2CCOC3C(N(C)C)C23)c2cnc(CC)s2)=O)CCC(F)(F)CC1 c1(CC(=O)N(C2CCCN(C(=O)CCCNC(C)=O)C2)CC)c[nH]ccc1=O Cn1ncc(C#N)c1C(N1CCC(C)(CC(=O)NC(C(N)=O)C2CCCC2)C1)=O c1(C(=O)NCC2(NC(c3sc(C)c(O)n3)=O)CCCC2)c(F)cccc1Cl C(C(C)(C)C(=O)N1CCC(NC(c2cncc(Br)c2)=O)C1)OCC C(=O)(CCCCCN(C(=O)CNC(=O)CN(C)C)C)NC(COC)CO.C(C)(=O)O c1(C(=O)NCC2(C(=O)NCC3(O)CCCCC3)CCCO2)ncccc1O c1(COCCCC(=O)NC2C3CN(C(COCCOC)=O)CC32)cc(Cl)cc(Cl)c1 N1(C(C2CC(=O)NC2)=O)CCOC2(CCC(NC(c3csc(Cl)n3)=O)CC2)C1 CCCCC(C)CCC(=O)N1CCC(=CC(=O)NCCCCCCN(C)C)CC1 C1(N(c2cc(C)nn2C)C(C2(c3ccccc3)CC2)=O)CCNCC12CC2 C(C)(C(=O)N(C)CC1(CNC(=O)CSC)CCC1)SCC C(=O)(CC(O)CC(C)(C)C)NC1CN(C(C)C)C(CO)C1 c1(NC(c2cccc(F)c2)C)cc(NC(C2(c3cccc(Cl)c3)CC2)C)ncn1 Cn1nc(C(N2CC3CC3(NC(=O)CC3(n4cccn4)CC3)C2)=O)cc1C(F)(F)F CC(C)S(=O)(=O)CC(=O)N1CC(NC(=O)Cc2ccc(Cl)cn2)C(C)C1 N1(C(C23CN(C(C4C=C(C)CS4)=O)CC2(CO)C3)=O)CC2CCOC(=O)C2C1 c1(OC)cccc(Cl)c1CC(=O)N(CC(=O)OC(C)(C)C)CC1CCCO1 CC1CCN(C(C2(F)CCOCC2)=O)CC1CC(=O)NCC1CC(N(C)C)C1 C1(NC(CCC(C)c2ccccc2)=O)CC12CCC(NC(c1cnsc1)=O)CC2 CC(C)C(O)C(C)(C)C(=O)NCC1CCCC(CNC(=O)CC(F)(F)Cl)C1 C1(NC(C2=C(C)OCC2)=O)CCC2CC1CN2C(c1ccc(NC=O)cc1)=O C1(CNC(c2cc(C)no2)=O)CCN(C(=O)CC2(N3CCCC3)CC2)CC1O c1(CN(CC(C)NC(c2nc3cccnc3s2)=O)C)cccc(P(C)(C)=O)c1 C=C1CC2(C1)C(=O)N(CCC)C2.c1(C(=O)Nc2ccccc2)cccn1C(C)C C(=O)(C(C)(C)n1ccc(NC(=O)OC(C)(C)C)n1)N(CCCN(C)C)C1CC1 N1(C(c2ccc(C)c(Cl)c2Cl)=O)CCCC12CCC(NC(=O)C1=CCOC1)CC2 c1(CNC(=NCC)NCC2CC(C)OC(C)C2)c(C)cccc1[N+](=O)[O-] c1(CCC(=O)NC2C3CN(C(=O)C=CCO)CC23)cncc(F)c1 Cc1nc2c([nH]1)CN(C(=O)C(C)(C)C(C)NC(=O)C1Cc3ccccc31)CC2 CCC(O)C(F)(F)C(=O)NC(CNC(c1ccc(OC)nc1OC)=O)C1CCC1 c1(CCC)ccc(CNCc2nc(C(=O)OC)n[nH]2)s1 C1(COC)(CNC(=O)CC2CCCO2)CCCN1C(=O)CN1CCOCC1=O C1(CNC(=O)NCC2CC(C)S(=O)(=O)CC2)CCC2COCCC2O1 N1(C(c2nc(COC)[nH]n2)=O)CC(CNC(=O)C(F)CC2CCCC2)CC1C N1(C(C(C=C)(C)C)=O)CCC2C(CCCN2C(C2OCC3CCCC2C3)=O)C1 N1(C(c2c(C)sc(Br)n2)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CC1C CN1CCN(C(C2CN3CCC2CC3)=O)C(CNC(c2cnc(N)cn2)=O)C1 c1(-c2nc(-c3cn(C(C)C)nn3)n(CCC3CC3)n2)ccc2nc[nH]c2c1 C12(C(CNC(C3CCCC3)=O)N(C(=O)C(c3ccnn3C)O)C)CCC(CC1)C2 C1(C(=O)NC2(C)CN(C(c3cnc(C)o3)=O)C2)CC(O)CN1C N1(C(C2C3CCN(C(C(C)(C)O)=O)CC32)=O)CC2(C)COCC2(C)C1 CC(CS(C)(=O)=O)C(=O)N1CCOCC(NC(=O)Cc2cnn(C(C)(C)C)c2)C1 N1(C(CCCC(C)=O)=O)CC2(CNC(c3[nH]cnc3C)=O)CCC1CC2 C1(C(N(C(CC)CNC(c2cscc2C(=O)OC)=O)C)=O)CCOC(C)(C)C1 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C1CN(C(=O)CCN2CCCCC2)C1)C c1(-c2cc(C)c(C(=O)O)cc2)cc(=NC(=O)C(O)CC2CCCCC2)[nH][nH]1 C(=O)(C1Cc2ccccc21)NCC1OCCCN(C(C2C(C)C2)=O)C1 CC1OCCC1(C)C(=O)NCC1CCC(C(=O)NCCC2(O)CCOC2)CC1 c1(C(N(C2CCN(C(=O)CC(C)CN(C)C)CC2)CC)=O)ccc(C)c(F)c1F.C1(O)CC1 C(C)(N=c1[nH]c(=NCC=CBr)[nH]c2c1CC(C)CC2)c1n(CC)ncc1 Cc1cc(Cl)cc2[nH]c(C(N3CCC(N(C(=O)CC4CCOC4)C)C3)=O)cc12 C1(O)(CNC(CC(C)(C)C)=O)CCCN(C(=O)CN=S(C)(C)=O)CC1 c1(C(N2C(CNC(C3C(=C)CC3)=O)CCCCC2)=O)cccc2sccc12 CC(C)(CC(=O)NCCCCCNC(c1csc(C(F)(F)C(F)(F)F)c1)=O)C(F)F N1(C(COc2c(C)ccnc2)=O)CC(F)(F)CC1CC(=O)O c1(CC(N2CCC(F)(C(N(CCC#N)C3CC3)=O)C2)=O)cc(F)ccc1Br C1(C#N)(OC)CC(C(=O)NC(CC2CCCC2)C(=O)NC2(CO)CC(C)C2)C1 c1(C(=O)NCC(C2CC2)NC(c2cc(C)c(Cl)s2)=O)cc2ccncc2cc1F c1(C(=O)NCC2(CN(C(C(CCC)O)=O)C)CC2)ccc2cccnc2c1 c1(C(=O)NC2CN(C(CC=C=C)=O)C(C)CC2)ccc2ccccc2c1 C(=O)(CCCCCCCS(C)(=O)=O)NCCOC(CNC(CCC=C=C)=O)(C)C C1(C(C(C)C)NC(=O)C(C)(C)C)CCCN(C(C2(CC(F)F)CCC2)=O)C1 Cc1cc(CC(=O)NCCN(CC(=O)O)C(N)=O)on1 S(=O)(=O)(c1ccc(C(=O)NCCNC(=O)C(C)C2CCOC2)cc1)NCC CCC(O)CC(=O)NCC(C)(C1CC1)NC(=O)CC1CN(C(C)=O)C1 N1(CCNC(c2ncc3ccsc3n2)=O)CC=C(c2ccccc2)C1 c1(CCC(=O)NCC2(NC(C3CC3(F)Cl)=O)CCCCC2)ccc(F)cc1 C1(CC(=O)NC2(CCC)CC2)CCCN1.C1(C=O)CCC1(F)F C1(CNC(C(COC)(F)F)=O)CCC2(CCCC2)C1 Cc1ccc(CC(=O)N(C2CCC(NC(c3cc(C)c(C)[nH]3)=O)C2)C)cn1 CS(=O)(=O)C(C(=O)NC1CN(C(=O)CCc2ncc(F)cn2)CC12CC2)C1CC1 CN1CC(C(=O)N(O)Cc2cn(-c3ccc(Br)cc3)nn2)OCCC1=O CC1CC(C(=O)N(CC(C)C(=O)Nc2ccc(O)cc2N(C)C)C)=NO1 c1(-c2cn(CCC(N3CCC(=C)CC3CC(=O)O)=O)nn2)cc(F)c(Cl)c(F)c1 CC1C(C)N(C(c2cc(C3CC3)cs2)=O)CCN1C(=O)Cc1sc(S)nc1C N1(c2n(CC(=C)C)c(Cc3ccccn3)nn2)CCCCC(C)(F)C1 N1(C(c2cn(C)c(=O)cn2)=O)CC2ON=C(CNC(C3(C)CC(F)(F)C3)=O)C2C1 c1(C(=O)OC)ccc(C(F)CNC(C2C(CC3CC3)C2(C)C)=O)cc1 C(C(C)(C1CC1C(=O)O)NC(=O)NCC1(C(F)(F)F)CCC1)OC C1(CC)(NC(=O)C(C)C2CCCC2)CCN(C(=O)C(F)C(F)(F)F)CC1 c1(OC)ccc(Br)c(CN2CCCC(C)(C(=O)NCC(C)O)C2)c1 N1(CCNC(CSCC)=O)CCN(CCNC(=O)Cc2ccccc2)CC1 N1(CC)CCC(C(=O)NCC2CCN(C(=O)CCCc3sccc3C)C2)CC1 c1(C(=O)NCC(C)CNC(c2ccc[nH]2)=O)cc2cc(Br)cc(F)c2o1 N1(C(COCC(=O)OC)=O)CC(OC)C(C(=O)N(C)Cc2cccnn2)C1 c1(SCC(N2CCC(C)(NC(CC)=O)CC2)=O)ncc(C(=O)OC)cc1[N+](=O)[O-] C1(C(=O)NCC2(F)CN(C(C(F)=C(C)C)=O)C2)CCCC2(CCCCC2)C1 c1(C(N2CC(C(C)NC(c3[nH]cc(C)c3)=O)C2)=O)ccc2c(c1O)OC(C)(C)C2 C1(NC(C2C(C)(C)C(NC(C3(O)CCOC3(C)C)=O)C2)=O)CCCCC1(C)C c1(CCC(N2C(C)(CC)CCC2)=O)nc2cccc(Cl)c2[nH]1 Cc1nn(-c2ccc(Cl)cc2)c(C)c1C(N)C(=O)NC(C)CO c1(CCC)cc(C(=O)NCC2CCCCN2C(=O)CSC(C)C)ccn1 C=CCC(CNC(=O)COC)C(=O)NC12CCC(CC1)C2 C(=O)(C(C)CC(C)(F)F)NCCN(C1CCCCCC1)C(c1nc(C)c(C)s1)=O Brc1scnc1-c1noc(-c2ccon2)n1 C=CCC(CC(F)F)C(=O)N(C(C)CCNC(C1CCC2(CCC2)C1)=O)C N1(C(c2cncc(OCC)c2)=O)CCCC(O)(CNC(c2nscc2C)=O)CC1 CC1CCCC(C(=O)NC(C)C(C)(C)NC(=O)CCc2cccnc2)O1 C1(O)(CNC(C=C(C)c2ccsc2)=O)CCN(C(=O)CC2(C)CC2F)CC1 C1(NC(CS(C)(=O)=O)=O)CCN(C(=O)CCc2ccoc2)CC12CCC2 C(=O)(CCCC(C)(C)C#N)NC(CC(=O)Nc1c(C)n[nH]c1C)C(F)F N1(C(c2c(CC)cncc2)=O)CCCC12CCN(C(C1OCC1(C)C)=O)C2 C1(NC(C(CCSC)O)=O)CCN(C(C2(F)CC3(CCC3)C2)=O)CC1(C)C C12(NC(c3cc(Cl)ccc3F)=O)CC3CCC(C1C2)N3C(C12CSC(C1)C2)=O N1(C(c2ccc(C(C)(C)C)o2)=O)C2CCC1CC(CNC(c1ccon1)=O)C2 C#Cc1ccc(C(=O)NCCCC(CCC)NC(=O)C(C)CC(OC)OC)nc1 N1(c2scc(C)n2)CCC(C(=O)NCC(C)NC(C2(C3CC3)CC2)=O)CC1 c1(C(=O)NCC2CCN(C(C(C(CC)C)C)=O)C2)c[nH]c2ncccc12 C1(C(=O)NC(C)CC2CN(C(=O)C(F)CC3CC3)C2)CCC2CC2CC1 C1(NC(c2cnc(O)[nH]2)=O)CC2CC1CN2C(C1CC=CCC1)=O C(CN=c1nc(C(C)(C)C)nc[nH]1)N(C(=O)C(C)(C)F)C N1(C(c2cc(C(C)C)no2)=O)CCC(NC(c2cc(C3(C)CC3)on2)=O)C12CC2 c1(C(N2CC(CNC(c3cnccn3)=O)OCC2)=O)n[nH]c2ccccc12 C=CCCCN=C(NC1CCOCC1)NC1CCOC(CC)C1 Cc1c[nH]cc(C(=O)NC2CC(NC(c3cnn(C4CC4)c3)=O)C(O)C2)c1=O Cc1cccc(CCN2CCN(C3(C)COC3)CC2)c1Cl C(Cn1ccnn1)(C(=O)N1CC(C(=O)OC)(CC)C1)NC(C=CC)=O C1(C(=O)NCC(CC)NC(c2ccc(N)cc2Cl)=O)CC(C)c2nc(C)cn2C1 CC1C(C)N(C(=O)Cc2cccnc2Cl)CCN1C(c1cc(C(C)(C)C)n[nH]1)=O C1(C)(C(=O)NC)CCN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC1 O(P(C)(=O)CCNC(=O)NC(c1cccc(OC)n1)C(C)C)CC C12(CNC(C3C(C)C3(F)F)=O)CC1CN(C(=O)C1=NOCC1)C2 CCS(=O)c1ccccc1C(N1CCC(C)(NC(=O)Cn2cnc(=N)[nH]2)C1)=O c1(C(N2CC(C(F)(F)F)C(C)C2)C(=O)NCC=C)cnc2c(c1)COC2 N1(Cc2cccc(OC)n2)CC2CN(C(C3CCN(C)C3)=O)CC12 c1(C(N2C(CNC(C(CC)C)=O)CC2)=O)cnn(CC)c1Br CCCCCCC(C)CC(=O)N1CC(NC(C23CC(C#N)(C2)C3)=O)C1 CCC(C(=O)NCC=CCNC(=O)C(C)Cc1cnc[nH]1)c1ccccc1 Cc1nc[nH]c1CNC(C1CCOC1CNC(c1ccsn1)=O)=O CCC(F)(F)CC(=O)NC1CN(C(c2ccc(OC)c(C3CC3)c2)=O)CC1C c1(C(=O)NCC(CC)(C)NC(C2CCOC2)=O)cc2cc(Cl)ccn2n1 C1(O)(CNC(C2(NC(C(=O)NCC3CC3)=O)CSC2)=O)CCCOC1 C(=O)(C1=CS(=O)CCC1)NCC(CC)NC(c1ccc2cnnn2c1)=O N1(C(c2ccc3ncnn3c2)=O)CCC2(CCCN2C(C2CC2Br)=O)CC1 Cc1cc(C)c(C(N2CC(CNC(C3CCCN3N=O)=O)CC(C)C2)=O)c(O)n1 N1(C(C2(C=C)CCC2)=O)CC2CCOCC2(NC(c2ccc(CC)c(Cl)c2)=O)C1 c1(C(C(=O)NC(C)C)N(CCC(=O)OCC)CC)ncc(SC(C)C)s1 C(=O)(C(C)(CC)CCC)NC(CCC)CNC(C1(F)CCCCC1)=O C(=O)(C=C(Cl)Cl)NCC1(CNC(COCCCC)=O)CCC1.COC n1(-c2c(C)cccc2)[nH]nnc1=NC(=O)N(C(Cc1ccccc1)C(N)=O)C1CC1 Cc1ncc(Cl)c(C(=O)NN2CC(CC(C(=O)N3CC(CC4CC4)C3)F)C2)n1 c1(CC)cccc(C(=O)NCCC2C(C)CCCN2C(c2occc2Cl)=O)c1F C1(NC(c2ccc(C)c(C)n2)=O)CCC2CN(C(c3cccc(O)c3)=O)CC2C1 N1(C(C(c2cccs2)SC)=O)CCC(O)(C2(NC(=O)CCCN(C)C)CC2)CC1 CN1CC(N=c2nc3sccc3c(N3CCc4nccc(N)c4C3)[nH]2)CC1=O Cc1ccncc1CC(=O)NC1CN(C(c2cccnc2)=O)CC1C N1(C(COc2ccc(C(C)=O)cc2)=O)CCC(C)C2CNC(=O)C12 c1(C(=O)NC)cccc(C(=O)NCC2CC(NC(=O)Cc3csnn3)C2(C)C)c1 C(=O)(C(C)(CO)NC(=O)Cc1cccnc1O)N(C1CC2CC2C1)C C(=O)(CCCCC(C)(C)C)N1CCOCC(CNC(C2ON=C(C)C2)=O)C1 C#CCCCC(C)C(=O)NC1CC(CC(=O)NC(c2ccco2)CO)C1 N1(C(C(C)=C(CC)C)=O)CC2(CCC2)CC1C(=O)Nc1nccc(OC)c1OC c1(OC)ccc(C=CC(N2CCC(C)C(NC(=O)Cc3cc(C)[nH]n3)C2)=O)cc1 C(CC(C)(O)C(=O)NCCc1cc(C(=O)NCCc2ccccc2)no1)N(C)C c1(C(CNC(=O)C(F)(F)CO)NC(C(C)SCCCC)=O)ccc(F)cc1F C1(N(C(CCCC)=O)C)CN(C(c2cc(C)n(-c3ccc(Cl)cc3)n2)=O)CC1O CCC(CC)CC(=O)N(CCCNC(=O)C(C)(C)Nc1ccccn1)CCO C=CCN=C(NCCc1cnn(C)c1C)N(C)Cc1cccn1C N1(C(c2c(CC)ncs2)=O)CCC(C)(C(N2CCC(C)C2C(=O)OC)=O)C1 N1(C(c2cc(CNC(C3C(C)CCOC3)=O)ncc2)=O)CCCC2(C1)N=N2 CC1=NN(c2ccc(Br)cc2)C(=O)C1CC(=O)NCC(CO)C(C)C CCC(CC(=O)N1CC2(CCC2)C12CCC2)C(C)(C)C.N12CCCC(CC1)C2=O C1(NC(CN(C)C2CC2)=O)CCOCC1NC(=O)Cn1ncccc1=O c1(OC)ccnc(C(=O)N(C2CCN(C(=O)C(F)Cc3ccccc3)C2)C)c1 S(=O)(=O)(c1cccnc1NCc1cn(CC)nn1)N(CCCC=C)CCOC N1(C(C(CC)F)=O)CC2CC(CNC(C3(OC)CC3)=O)CC1C2 N1(C(c2n(C)cnc2Cl)C(=O)NC2CCOCC2)CCc2ncncc2C1 C(CCC)(CCCNC(=O)CN1CC(=O)NC1=O)NC(C(c1n(CC)ncc1)=O)=O C1(C(=O)N(C(C)C(N)=O)C)(CC)CCCN(C(=O)CC#N)C1 C(=O)(C1=CC(C)(C)C1)N1CC(CC(C(=O)NCCc2n(CC)cnn2)F)C1 c1(C(=O)NCC(C(C)(C)C)NC(C2CC(N=[N+]=[N-])C2)=O)cc([N+](=O)[O-])ccn1 C1(N(C(c2c(C)cn(C)c2)=O)C)CC2CCC(C1)N2C(=O)CCC(C)CN(C)C C=CCCCCC(=O)N1CCCC(C)(CCCNC(=O)C(CC)C(=O)OC)C1 C1(CNC(CN2CC=CCC(C)(C)C2)=O)CCCC2(CCCCC2)C1 N1(CCC)CCC(CCNC(c2ccccn2)CCc2ccccc2)CC1 c1(C(=O)NC(C2OCCN(C(c3c(C)nccc3)=O)C2)C)ccn2nnnc2c1 c1(C(N2CC(N(C(CC(=O)NCC#C)=O)C)C(F)C2)=O)ccc2nnn(C)c2c1 C1(SC(C)C(=O)N(C(c2ccccc2)CCNC(=O)C(C)O)CCO)CCCCO1 c1(N2CC(C)CS(=O)CC2)ncccc1S(=O)(=O)NCCO.c1(C)ccccc1 C1(CC(N2CCC(C(C)NC(=O)COc3ccon3)C2)=O)CCCCC1C c1(SC(=O)CSC(C(F)(F)F)C2CCOCC2)ccc(O)cc1 c1(NC(C2(NC)CC2)=O)ccc2c(c1)C(O)CC2 C(=O)(C1(O)CCCc2ccccc21)N1CCS(=N)(=O)C2(C1)CCC2 N1(C(C2CN(C(N)=O)C2)=O)CCC2(NC(c3nccc4occc34)=O)CCCC12 c1(CNC(CCSCC)=O)ccnc(N2CCN(C(C3CCOC3=O)=O)CC2)c1 N1(C(CC(CC)N(C(=O)C(C)NC(=O)OC)C)=O)CCc2nnnn2CC1 c1(C(=O)NCC(CC=C)NC(c2ccn3ncccc23)=O)c(F)ccc(N)c1F C(=O)(C(CCC1CC1)NC(=O)CC(C1CC1)C1CC1)N(CC(COC)C)C C(CCNC(c1ncc[nH]1)=O)(C(C)C)NC(Cn1ncc(C)c1)=O CCC(O)C(C)C(=O)N1CCC(NC(c2cn(-c3ccccc3Cl)nn2)=O)CC1 N1(C(C(CC)NC2CCN(Cc3cccnc3)C2)=O)CCCC(CC)C1 N1(C(=O)CC2(O)CCOCC2)CC(NC(C2(F)CCCC2)=O)CC12CCCC2 c1(CC(N2CCN(S(C)(=O)=O)CC2)=O)c(F)cccc1Br c1(C(C)C)nn(C)cc1C(N1CCOC(CCN2CCCC(O)C2)C1)=O C1(CCNC(CC2(OC)CC2)=O)CSCCN1C(=O)CC(C)CF CC1CN(C(c2ccc(C#N)[nH]2)=O)CCN1C(=O)CCOCC1CCCO1 C(CC(C)(C)C)(C(=O)N1CC(O)CC1C(=O)N(C)CC1CCC(=O)N1)OC c1(C(C)C)cccc(OC(C)C(=O)NC(=O)Sc2nncs2)c1 Clc1cccc(Cn2ccnc2-c2ccc(-c3cc[nH]n3)s2)c1CN1CCCCC1 Cn1ncc(C(=O)NC2CCOC(C(=O)NCCC(C)(C)C3CC3)C2)c1Cl c1(C(=O)NC2C(NC(C(C=C)OC)=O)COC2)cncc(C)n1 c1(C(=O)NC(C2CCOC2)CNC(C2(COC)CC2)=O)ccc(OC)cn1 CCCC(C)(C)CNC(=O)NC1CCOCC1O C=C(Cl)CC(C(=O)N(CC)Cc1cncs1)NC(=O)C(C)OCCN(C)C n1(C(CC)(C)C)nnnc1C(c1occc1C)NCC1CCCO1 CC(C)C(C(C)NC(c1cnc[nH]1)=O)NC(c1cc(-c2ccc(Br)s2)on1)=O N1(CCC(=O)NC(CCCNC(C(C)n2ccnn2)=O)C)CCC(O)CC1 N1(C(CC(=C)C)=O)CCCOC(CNC(c2nc(C)sc2C)=O)C1 N1(C(c2cnn(C)n2)=O)CCCN(C(c2cc(C3CC3)ccc2F)=O)CC1CO c1(NC(CC2(N(C(C(C3CC3)OC)=O)C)CC2)=O)csc(CC2CSC2)c1 N1(C(COCCC)=O)CC2C(CN(C)C(c3oc(Br)cc3C)=O)C2C1 N1(C(C(COCC)NC(=O)COC(C)=O)=O)CC2CCCC2(COC)C1 C(C(C)(CC)C(N)=O)NC(CN(C(=O)C(O)CCCC)CC#C)=O c1(CNC(C(COC)(C)C)c2nnnn2-c2ccccc2)cnc(C)c(Cl)c1 c1(C(=O)NC(CNC(c2cc(OCC)n[nH]2)=O)(C)C)ccc2ncc(C)cc2c1 C(CCCCC(=O)NCCCCC(C)NC(C1C2COCC12)=O)NC(C)=O N1(C(Cn2ncc(C)c2)=O)CC=C(C(C)(C)C(=O)N2CCC2CN=[N+]=[N-])C1 N1(C(C23CCC(C(=O)OC)(CC2)C3)=O)CC(CN)C(S(C)(=O)=O)C1 CC(CSC(F)(F)F)C(=O)N(C)CC1CCCN1C(=O)CSc1ccccc1 CC(C)(C(=O)N1CCCC1)N(C(=O)COC1CCC1)CCNC(=O)C1=CCC1 C(=O)(C1=NNC(C(F)(F)F)C1)NC1C=CC(CNC(c2c(C)ccnn2)=O)C1 C1(c2ccccc2)(C(=O)NC2C(NC(C(=O)NCCOC)=O)C2)CCN(C)C1 Cc1nc(N(C)C)sc1NC1CCCCC1SCc1ccccc1 C(=O)(C1Cc2ccccc21)NCC(CNC(c1cc(C)nc(C)c1O)=O)OC c1(CC(=O)N(C(C)CNC(c2c[nH]c(=N)s2)=O)C)cnn2ccccc12 N1(C(CCC2C(C)C2)=O)CCC(CNC(c2c(C(F)F)nn(C)c2C)=O)C(C)C1 c1(NC(C2CCN(C(c3cc(C)oc3C)=O)C2)=O)ccc(Cl)cc1C#N C(=O)(C(O)C(F)(F)F)NCC1C(C)CCN1C(=O)Cc1nc(=N)[nH][nH]1 C#CCCCC(=O)NC(C(C)NC(c1ccc(CSCC)cc1)=O)C(C)C c1(C(C(=O)N(CC2N(C(CCC#C)=O)CCC2)CC)C)ccc(CC)cc1 c1(CC(C)(C)C)nnc(N2CCC(O)(C(Cl)(Cl)Cl)C2)n1CCCN1CCCCC1 N1(C(CCCC)=O)CCC2(CC1)CC(NC(c1ccc(S(C)(=O)=O)cc1)=O)CO2 c1(C(C)NC(C2(c3cc(C)no3)CCCC2)=O)cnc(O)c(C(F)(F)F)c1 C(c1ccnn1C)=CC(=O)N(CC(=O)NC1(C)CC(=C)C1)CCC CCC(C)(O)Cc1cn(C(C)C(=O)NC(c2ccccc2)c2ccccn2)nn1 c1(CC)cc(=NC(=O)CC(CC)N(C(=O)CC2CNC(=O)O2)C)[nH]n1C CC(C(=O)NC1CCCC(NC(C2CCC=CCC2)=O)C1)C(C)O Cc1cc(Cl)ccc1C(N1CCC(C)(CNC(C2C3CCC23)=O)CC1)=O CC1CC2(CCN(C(C3NC(=O)OC3C)=O)CC2)CN1C(=O)C1=CCCSC1 C1(C(N(C2CN(C(c3c(C(C)C)nn(C)c3Cl)=O)C2)C)=O)CC2CCCC(C1)C2 c1(C(=O)NCCCN(C(CCOC(C)=O)=O)C)cc(S(=O)(=O)N(C)C)c[nH]1 C1(N(C(=O)CCC2CC2)C)CCCC(N(C)C(c2nn[nH]c2Cl)=O)C1 N1(CC)CCCC2C1CCCN2C(COC(=N)O)C(=O)Nc1ccccc1 c1(CC(=O)NCC2CCCN(C(C3(C)CC(C#N)C3)=O)C2)ccc2ncsc2c1 c1(C(=O)NC2CN(C(C(C)C(C)(C)C)=O)CC23CC3)ccc2c(c1)NC(=O)C2 c1(C(=O)NCCc2ccc(C)cn2)coc2c1CN(C(=O)C1=CCCC1C)C2 CCC(CC(=O)N(C)CCc1ccncc1)NC(C1CC(C)CCO1)=O c1(C(N2CC3CCC2CN3C(C2(C(F)(F)F)CC2)=O)=O)cc(O)cc([N+](=O)[O-])c1 C=C1CCC(C(=O)NCC=CCNC(c2ccncc2N(C)C)=O)CC1 C(=O)(CC(C)P(C)(C)=O)NC1CC(CCNC(c2[nH]cc(C(=O)OC)c2)=O)C1 Cc1cc(F)ncc1CNC(=O)NC(C)COCc1ccccc1 CCCCC(C)N(C(=O)C(=O)N1CC(OCCOC)C1)C N1(C(C2=CCC(NC(C(CC)=CCCC)=O)C2)=O)CCc2c(cnn2C)C1 n1(CCC)cc(C(=O)N(C2CCN(C(=O)CSCCCC(C)C)C2)CC)nn1 c1(C(=O)NCCN(C(C2CC2c2cccnc2)=O)CC2CC2)cnc(Cl)s1 C1(C(=O)NCc2nccc(C(=O)NC(COC)C(=O)OC)c2)CC2C=CC1CC2 C(c1cccc(F)c1F)=CC(N1CC2CC2(CNC(C2(CO)CC2(F)F)=O)C1)=O N1(C(C2CCCN(C(C(C)NC(CC)(C)C)=O)CC2)=O)CC2(C1)OC(=O)NC2C CC1=NN(C)C(=O)C1CC(=O)N(C1CN(C(=O)C(=O)Nc2ccccc2)C1)C N1(C(CC2ON=C(CC)C2)=O)CC2CCOC2(CNC(=O)C2=C(C)CCCC2)C1 CCCC(CNC(=O)C(N)=O)C(=O)N1CCC(COC(C)=O)C1 C(=O)(CS(=O)(=O)CCOC)N1C2CN(Cc3cccc(CCCCC)c3)CC1C2 c1(C2(CNCC3CCC(C(=O)OC)CC3)CC2)ccc(Cl)c(F)c1 C1(C(=O)NCCC(C)NC(C(C(CC)O)C)=O)C2CC3CC(C2)CC1C3 C1(CNC(C(C=C)CC)=O)CN(C(c2ccnn2CCC)=O)CC12CC2 c1(C(=O)NC2C3(CC(NC(c4occ(C)c4C)=O)C3)C2)ccn2ccnc2c1 C(C)(CCCCNC(c1ccc(Cl)cn1)=O)NC(CCN(C(CCC)C)C)=O C1(N(C(c2c(CCC)nco2)=O)C)CCCN(C(=O)Cc2ccccc2)CC1 CC1(C)C2CCC(C2)C1C(N1CCN(C(c2cnc(N(C)C)o2)=O)CC1CO)=O C1(C(CC)CC)CC(NC(=O)NC2(C(=O)OC)CS(=O)(=O)C2)CCO1 c1(CC(CC)C)nc(C2CCC(O)CN2)n(-c2ccc(F)nc2)n1 Cc1cc(C(=O)N(CCCN(C(=O)COCC(C)C)C)C)nc(O)c1 c1(CCN)ncccc1C.C1(CCCC)CC(c2nnnn2C)(N)C1 c1(OC)ccc(C(CNC(=O)C(F)n2cccn2)NC(c2ccc(F)s2)=O)cc1 C(=O)(CC(C)(C)CC(F)(F)F)NCC1CCN(C(C(c2ccc(F)cc2)C)=O)C1 C1(NC(C2CCC(NC(C(CC3CC3)OC)=O)CC2)=O)CCC2(CCC2)C1 c1(C(=O)NC(C)CC2CN(C(c3cn(C(F)F)cn3)=O)C2)ccc2ncccn12 C1(CNC(c2c(C)nns2)=O)N(C(=O)COc2cccnc2Cl)CCCC1(C)C N1(C(C2CC(C)OCC2)=O)CC(C)(C)OC2(C1)CN(c1ncnc3c1COC3)C2 CCCC(CC(=O)N1CCOCC1CC(N)=O)NC(=O)CC(C)CC C1(CNC(CCc2cc(OC)no2)=O)CN(C(=O)C2=CCC2)CCC1C(F)(F)F CCCCCCC(C)C(=O)N(CCN(C)C(c1c(F)ccnc1F)=O)C(C)C N1(C(CN(CCC)C)=O)CCC(NC(c2ccnc(C(N)=O)c2)=O)C2(CCC2)C1 c1(C(N2CC(NC(C(C)N3CCC3)=O)C(F)CC2)=O)ccc(O)c2ncccc12 c1(C(=O)NC2(C)CCN(C(C3CC(n4cnnc4)C3)=O)C2)cc2c[nH]cnc-2n1 C1(C(N(CC)CC2CCCCN2C(=O)C=C(C)C)=O)CCCCCN1C N1(C(=O)CC2(c3ccccc3)CC2)CC2(CO)CC1(CC1CC1)C2 C(=O)(C1Cc2ccc(Cl)cc21)OCNC(C(CC(C)C)(C)O)=O C1(C(=O)NCCc2c(CNC(c3cc(F)cs3)=O)nco2)CCc2cnnn2C1 c1(C(=O)NCCOCCNC(C(C(CC)CC)C)=O)ccc2c(C)noc2c1 N1(CC(=O)O)CCN(C(c2ccc(CNC(C3CC3(F)F)=O)nc2)=O)CC1=O C1(NC(CC=CCC)=O)CCCC12CCN(C(=O)C(C)(O)CC(C)C)CC2 Cc1cccc(OCC(=O)NC(C)(C)CN(C(=O)CC2CCC(C)(C)O2)C)c1C N1(C(C2CCCN(S(CC=C)(=O)=O)CC2)=O)CCC2(CC1)OCCc1ccsc12 N1(C(C(C)(C)C#N)=O)CCOC(C)(CNC(C23CC=CC(C2)OC3)=O)C1 C1(C)(CNC(C(C2CC2)OC)=O)CN(C(=O)Cc2ncoc2C)CCO1 c1(C(=O)OC)c[nH]c2ncnc(N3CCOC(CNC(=O)C(C)(C)N(C)C)C3)c12 CC(C(=O)NCC(C)NC(c1cnc(Cl)s1)=O)C1CCOCC1 c1(C(=O)NC(C2CCCN2C(C2CCCCO2)=O)C)cnn(C(C)(C)C)c1N c1(CC(=O)N(C2CCN(C(C3CCN(S(C)(=O)=O)C3)=O)C2)CC)ncn(C)c1C N1(C(c2c(C(F)F)ccc(C)c2)=O)CC2(CCC(CNC(=O)C(C)O)O2)C1 N1(C(C(C)=CC2CC2)=O)CC2(NC(c3ccc(C)nc3O)=O)CCC1C2 Cn1cc(CNC(=O)C(N2CCCCCC2)=O)c(C(F)F)n1 C1(NC(CC(C)CN(C)C)=O)CN(C(=O)C(C)n2ccnn2)CCC1O c1(C(=O)NCCCNC(C(CCC)(C)CC)=O)cc2ccccc2[nH]c1=N c1(C(=O)NCC23CC(NC(c4c(CC)cco4)=O)(C2)C(C)O3)cn2ccccc2n1 N1(C(c2cnc(CCC)s2)=O)CCC(CCNC(c2cnn(CCC)c2)=O)CC1 c1(OC(C)C)ccc(C(=O)N(C2CCCCC2NC(c2c[nH]c(=N)o2)=O)C)cn1 c1(C(=O)NCC2C(SCC(=O)Nc3cn[nH]c3)CC2)ccc(Cl)c(Cl)c1O C(=O)(C(C)(C)NC(=O)NC1CC(C(=O)NCCc2ccccc2)C1)NCC CC(C)CC(O)CC(=O)NCc1cccc(C(=O)NCC2CC(CO)CO2)n1 C1(C(=O)NCC2C=CCN2C(c2cnc(C(C)(C)C)o2)=O)(OC)CCSC1 c1(N(C)C)ccccc1C(=O)NCC1CCCC1NC(=O)CC1(C2CC2)CC1 C1(C(=O)NCC(C)C(=O)OC)(OC)CCN(C(=O)C=CCN(C)C)C1 N1(C(CC(=O)OC)=O)CC(NC(C2(F)CCOC2)=O)Cc2ccccc21 C1(=O)C(N(C2(C)CC2)C)CCC2C(C(C(=O)OC)N1)C2.OC CCCCCCCCCCC(=O)NC(CNC(c1ncoc1CC)=O)CO c1(CC(=O)NC2CCC3(C2)CN(C(C2CC=CCC2)=O)C3)cc2ccccc2s1 Cc1cc(C(=O)NC2CC3C(NC(=O)C4=NNC(=O)C4)C3C2)c(F)cc1Cl c1(C(=O)OCCc2cc(C)on2)ccc(Sc2ccc(Br)cc2)cc1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(CC)N(C(C2CCC(C(N)=O)CC2)=O)CC1 C12(CNC(CC(C)(C)OC)=O)CCCC1N(C(=O)C=C(C)C1CC1)CCC2 Cc1ccc(C(=O)N(C23CCC(CC2O)C3)CCCNC(N)=O)c(O)c1.CCCN=[N+]=[N-] C1(NC(=O)CN2CCOCC2=O)(CC2CC2)CC2CCCC12.C12CC(C1)NC2=O C1(CC(=O)N(CCOC)CCNC(C2(CO)CCOCC2)=O)CCCC(C#N)C1 Cc1cccc(CNC(C2CC(C)CN(C(=O)CCNC(=O)CO)C2)=O)c1F N1(C(C2CCCC(C)O2)=O)CC(C2(NC(=O)Cc3ccsc3Cl)CC2)C1 C1(c2nnnn2C2(C)CC2)(NCc2cccc(CC)c2)CCN2CCCCC12 c1(NC(N2CC3C(CC(=O)NC(CCO)C(F)(F)F)C3C2)=O)cc(Cl)ncc1F c1(C(=O)NC2C(CNC(C(=Cc3ccncc3)C)=O)C2)cncc2cnccc12 N1(C(=O)NCC2CCCCC2(F)F)CC=C(c2cccc(Cl)c2F)CC1 Cc1oc(C(=O)NCC2CCN2C(C2(C)CC(C3CC3)=NO2)=O)cc1S(N)(=O)=O c1(C(N2C(CNC(C3C(=C)CC3)=O)CCC2)=O)cc2c(Br)cccc2[nH]1 c1(CN(C(c2c(CC)c[nH]n2)C(=O)NCc2cccs2)C)nc2ccccc2o1 S(=O)(=O)(c1cnc(NC2CCC3(CCCC3)C2)c(Cl)c1)N1CCC(C#N)(F)C1 N#Cc1ccccc1CN1CC(NC(c2ccc(F)cc2Br)=O)C(C#N)C1 C1(C(C(=O)N(CCNC(C(CCC)=CCC)=O)CCC)O)CCS(=O)(=O)CC1 C1(NC(C2C(COC)C2)=O)CCCCN(C(c2ccc(F)cc2N)=O)C1 c1(C(=O)NC2CC(CCNC(C3(CF)CCOCC3)=O)C2)cn2ncccc2n1 c1(NC(CCCCCC)(C)c2nnnn2C2CCC2)ccc2c(c1)CC(C)(C)O2 c1(C(=O)NCC2CC(C(=O)OCC)OC2)occc1C.c1(C)ccc(CC)[nH]1 C1(NC(c2c(C)nc(C)s2)=O)CC(C)CN(C(=O)CNC(=O)C(F)(F)F)C1 C(=O)(C1CCCc2c(O)cccc21)N1CC(CNC(CC=CC=C)=O)C2(C1)CC2 C#CC1CN(C(c2sc(COC)nc2C)=O)CCN1C(C1CCCN1C(C)=O)=O C(C)(C(=O)N(C1(OCCOCC(O)CO)CC1)C)SCC.C1(=O)CN1 N1(C(c2c(C#C)c[nH]n2)=O)CC(O)CC1(C)C(=O)NC1(CSC)CC1 Cc1cc(Cl)cc(C)c1C(=O)NC1CCCC1CNC(=O)CCCc1cc[nH]n1 c1(C(C(=O)NC(CNC(c2ccn(CCC)n2)=O)C)(C)C)ccc(Cl)c(Cl)c1 N1(C(C2N(C(c3c(C)n(C)nn3)=O)CC3CC32)=O)CCCC(C)(O)C1 C1(CNC(C2=NOC(C)C2)=O)CN(C(c2ccc(N)c(O)c2)=O)CCC1(C)C N1(CCNC(c2c(O)cccc2Cl)=O)CCS(=O)(=O)C2(CCCCC2)C1 N#Cc1ccc(O)c(C(N2CCC(NC(=O)Cc3ccsc3)C(O)C2)=O)c1 N1(C(c2ncc(OC(C)C)nc2)=O)CCN(C(C2(C)CC2(F)F)=O)CC(CO)C1 C(C(C(=O)NC1CC(NC(N)=O)C1)NC(=O)C(C)c1cccs1)OC N1(C(C(COC)C)=O)CCN(C(c2cn(-c3ccccc3OC)nn2)=O)C(C)C1 c1(C(=O)NCC#CCNC(c2cocn2)=O)ccc(Cl)cc1C(F)F C1(C(N(C2CCN(C(=O)COC3CCC3)C2)CCC)=O)CCC(=O)N1C N1(C(CNC(c2cccs2)=O)=O)CCOC(NCc2ccnc(C(F)(F)F)c2)C1 C1(N(C(c2cnc(SC)s2)=O)C)CCCC(N(C)C(c2cccnc2)=O)C1 CC(CNC(=O)C(O)CC1CCCCC1)(CO)NC(=O)CCc1csc(=N)[nH]1 C(=O)(C(C)(C)CCC#N)NCCN(C(C1CC(CC(=O)OC)C1)=O)C(C)C CP(C)(=O)C(O)C(=O)N1CC2(CNC(c3cnnc(O)c3)=O)CC2(C(F)(F)F)C1 C1(C(N2CCC(C)(CC(=O)N(CCCCCC)CC(N)=O)C2)=O)CC2(C1)CC(C)C2 CCC(C)C(CC(=O)NCC(O)C(C)(C)O)NC(c1cc(C)sn1)=O CC(C)(C(=O)NC(c1ccccc1)CNC(c1cc(Cl)c[nH]1)=O)C1CCCO1 c1(C(=O)NCC(CNC(c2c(C)csc2)=O)(C)O)cc(S(N)(=O)=O)cn1C c1(NC(C(=O)N(C(C)CS(C)=O)C)=O)ccc(Br)nc1Cl N1(C(c2c(C)c(N)ccc2)=O)CCC(C)N(C(c2cc(Cl)cnn2)=O)CC1 C1(NC(C2(COC)CC=CCC2)=O)CCN(C(=O)C2=COCC2)CC1CO N1(C(CNC(c2c(C)cccc2)=O)=O)CCC2(C1)CN(C(c1cccs1)=O)CCO2 C(=O)(C1COc2cc(C)c(C)cc21)NC1(CCNC(CC=CC=C)=O)CCC1 n1(CC(=O)NC2(CC=C)CN(C(=O)CCC3CCOC3)C2)ncc(Br)c1C C(=O)(CC(=O)NC(CO)C(=O)N1CCC1(C)CCO)N(C)C C(=O)(C1=CCOCC1)N1CCC(C(=O)NC(COC)CO)(OC)C1 C1(F)(C(N(CC(CCC)O)C)=O)CCN(C(=O)COC2CCC2)C1 C1(C(C(=O)N(CC(=O)NCC)C)NC(C2CN(C(C)C)C2)=O)CC=CCC1 C1(NC(C=NOC)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)C12CC2 C(=O)(C(O)CCCc1ccccc1)NC(CNC(c1ncc(C)nc1)=O)CO c1(CN(C(C2CCCOC2)C(=O)NCSc2ccccc2)C)c(Cl)cccc1Cl C1(C(=O)NC(C#C)C)CCN(C2CCN(C(=O)C3CC3)CC2)CC1 c1(C(=O)NC(C2(CNC(CCOC)=O)CC2)C)c[nH]c2nc(Cl)ccc12 c1ccc(F)c(Cl)c1.C(CC(=O)NC)(OCC)OCC.c12cc(n[nH]1)NC2=O C#CCC(C(=O)NC(C)(C)C(C)NC(=O)CN(C1CCCC1)C)C1CC1 c1(C(N2CCC(CC)CC2)C(=O)NCc2cccs2)cnc(OC)c(Br)c1 N1(C(c2c(C)cnn2C(C)C)=O)CCC(C)N(C(C2CN(C)CCO2)=O)CC1 c1(OC)cc(C(O)C(=O)NC2CCCN(C(=O)CCC3(C)CC3)C2)c(F)cc1O C(C(C)(C)CC(C)C)NC(C(CCC1CCC1)NC(CC1C(CC)C1)=O)=O O=C(CC(C(F)(F)F)NC(=O)CSC1CC1)NCC12CC(CO)(CO1)C2 N(C(=NC1CC1)NCC1(N(C)C)CC(C)CC(C)C1)C(C#C)CC C1(NC(c2cnn(-c3ccccc3)c2)=O)CCN(C(C2CC(CF)C2)=O)C1 CCCCC(O)C(C)C(=O)NCC1CCN(C(C)C)CC1 C12(C(=O)NCC(C3CC3)NC(CCSCC(N)=O)=O)CC(F)C1C2 N1(C(CC(C(C)C)O)=O)CCOC2(CCN(C(c3cnn4c3CCC4)=O)C2)C1 c1(C(=O)OC)cccc2nc(COC(=O)C(C3CCCCC3)N(C)C)cn12 C(=O)(C1c2c[nH]nc2CN1C(=O)CC(O)C(C)C)NC(CSC)C C(=O)(C(C)C(O)C(C)C)NC1(CO)CCN(C(CCCc2c(C)cccc2)=O)C1 C1(CC)CCN(C(=O)C(=O)Nc2cc(C)n(CC(=O)OC)n2)C(c2ccco2)C1 N1(C(c2c(N(C(C)C)C)cccc2)=O)CCC(NC(=O)CC(C)(C)O)C(C)C1 Cc1c(C(N2CC(CN=c3[nH]ncs3)(C(F)(F)F)C2)=O)cnn1C(C)C(C)(C)O N1(C(c2nnc(C)s2)=O)CCC2(CCN(C(C3COCCO3)=O)CC2)C1 C1(NC(C(C)OCC#C)=O)CN(C(c2cc(C)c(O)nn2)=O)CC1S(C)(=O)=O c1(CCC(=O)NCC(C)CN(C)C(C2CN(C)C2)=O)ccccn1 c1(OC)cc(C)cc(F)c1CNC(C12CC1CN(C(=O)COC1CCCCC1)C2)=O c1(C(N2CCCC(N(C(=O)C=C3CCCCC3)C)C2)=O)cccc(P(C)(C)=O)n1 c1(C(=O)NC(C(C(C)C)NC(C2(O)CC(F)(F)C2)=O)C)cn(C)c(=O)n(C)c1=O N1(C(c2cnc(C)nc2C)C(=O)NC(C(=O)OC)C)CCC(C)OC(C)C1 c1(COCC)nc(COC)cs1.C12(COC1)CC(=O)N(C)C(C)CN(C)C2=O.N(C)C c1(C(=O)NC(CNC(C2(CF)CC2)=O)CO)cc([N+](=O)[O-])c(Cl)cc1Cl c1(C(=O)NC(CCOC)CNC(=O)C(C)c2cccs2)ccc(S(N)(=O)=O)s1 C1(C(=O)NCC(CCNC(C2(NC(N)=O)CC2)=O)O)OCC2COCCC12 C(=O)(C(C(C)(C)C)C1CCC1)N1C(C(C)NC(c2cccnc2)=O)CCCC1 c1(C(N(CCN(C(CC2C(C)CCC2)=O)C)C)=O)ncccc1S(C)(=O)=O N1(C(c2c(NCc3c(C)cncc3)ccs2)=O)CCN2CCOCC2C1 c1(SC)cc(C)ccc1C(=O)NCC1CC(O)CN1C(=O)CC1(N(C)C)CC1 N1(C(CCSCCCC)=O)CC2CC1CCN2C(=O)Cc1ccc(F)cc1Cl C1(F)(CNC(c2c(C)scc2)=O)CCN(C(c2ccnnc2)=O)CC1 C(CN=C(NCC1CCC1)NCC(c1ccccc1)(C)O)c1ncc(C)cn1 c1(NC(c2c(CCC)n(-c3ccccc3)nn2)=O)cnc2n1CCCC2 CC(C(=O)N1CCOC(C)(CNC(=O)Cc2ccc(F)cc2F)C1)C(C)(C)C CCCN=C(NCCN(C)C)N1CCC(O)(C(F)(F)F)C1 N1(C(C(C(C)(C)C)NC(C(C(CC)C)N(C)C)=O)=O)CCC2(CC=CCO2)C1 C1(OC(N2CCC(c3scc(C)n3)C2)=O)CC2CN(C(=O)OC(C)(C)C)CC2C1 C1(NC(C(C2CCCN(C(CCC#C)=O)C2)C)=O)CCN(C)CC1(C)C Cn1cnc2sc(C(N3CC(NC(c4cc(C#N)c[nH]4)=O)C(C4CC4)C3)=O)cc12 c1(C(N2C(CN(C)C(C3CCN3C)=O)CC(F)C2)=O)cccc2c[nH]nc12 C(=O)(C1=C(CC)N(CC)C(=S)NC1c1cc(C(C)C)c(Br)s1)OCc1cc(C)on1 CC(C(=O)NCCC(C)NC(=O)Cn1ccc(C(F)F)n1)S(C)(=O)=O c1(CC(=O)NC(C)CNC(=O)C=CC(N2CCOCC2)=O)ccc(S(C)=O)cc1 c1(C(=O)NCC2C(NC(C3(COC)CCC3)=O)C2)ncc2ccccc2c1O c1(CC(=O)N(C(C)CNC(c2csc(C(F)F)n2)=O)C)cccc(F)c1Cl c1(C(N(CCCCCNC(=O)C(C)C2CCOC2)CC)=O)cccc2c1OCC2 C1(NC(c2c(C)coc2C)=O)CN(C(=O)Cn2[nH]cnc2=N)Cc2nccn2C1 O=C(N=c1ccn(CCC(=O)OC(F)F)[nH]1)NN1CCCCC1 c1(CNC(=O)NC2C(C)(C)CN(Cc3ccccc3)C2)cc2ccccc2[nH]1 C(C1=NOC2COCC12)NC(CCC1CCCN(C(CCC(C)SC)=O)C1)=O c1(NC(C2CCN(C(c3cnc(C)[nH]3)=O)CC2)=O)cc(F)cc(C)c1Br c1(C(N(C2CCCN(C(=O)C#CC3CC3)C2)C)=O)ccc(CO)cc1F c1(CCOC)n[nH]c(=NCC2CCCN2C(=O)C(C)CF)s1 C(=O)(C1=CC2CCCCCCCC12)N1CC2C(NC(CC(C)F)=O)C2C1 C(=O)(CC(CC(=O)O)C(F)(F)C(F)(F)F)NCC(N1CCCCC1)C C1(C(N2CCC(C(F)CNC(c3ccc(C)o3)=O)CC2)=O)(CC)CC(C)(C)C1 C=CCC(CC=C)C(=O)NC1(C(=O)NCCCC(=O)NO)CC1C O=C(C1=C(Cl)CCOC1)NCC(O)CNC(c1ccc2nc[nH]c2c1)=O C1(C(N2CCN(C(=O)C(C3CC3)OC)C(COC)C2)=O)(OCC)CCCCCC1 C=CCCC(O)CNC(=O)CC1(NC(=O)CC(CC)SC)CCCCC1 C1(CNC(c2n(CC)c(O)nc2)=O)CCN(C(c2cc(=N)[nH]n2C)=O)CC1C c1(C(N2CC(C)N(C(c3cc[nH]c(=N)c3N)=O)CC2)=O)cc2cc(Cl)ccn2n1 c1(C(=O)OCC(C(=O)OCC)CC2CC=CCC2)ccccc1.c1cccnc1 c1(OC)ccc(NC(=O)CCN(C(=O)CC2CCCC(C)O2)C)cc1F CCC(C(=O)NCC1C=CC(CNC(=O)C(F)(F)C2CCOCC2)C1)N(CC)CC C(=O)(C1CCCc2ccnn21)N(C)CC1CCN(C(c2c(OC)cc(C)s2)=O)C1 c1(CN2CC(CS(=O)(=O)N(C)C)NCC2)cc(Cl)cc(Br)c1 c1(C(C)=O)cc(C)[nH]c(=NCCCCCCNC(c2cnoc2C2CC2)=O)n1 c1(C(=O)NC2(C(NOCC(=C)Cl)=O)CC=CC2)cn(C)c(C)n1 S(=O)(=O)(c1cnc(NC(C)(CO)CCF)c(Cl)c1)NC(C)COCC1CC1 N1(C(C(COC)(C)C)=O)CC(C)CN(C(c2cnc3ccncc3c2)=O)C(C)C1 C1(NC(C(C2CCN(CCCOC)CC2)C#N)=O)(CO)CCC(C)(C)C1 CCC(C(=O)N(CCCCO)CC)NC(N)=O N1(C(c2c(CC)nc(C)nc2)=O)CCCC2(C1)CN(C(=O)CNC(N)=O)CCO2 CCC(C)C(O)CC(=O)N1CC2C(c3cn(C(c4c(C)noc4C)C)nn3)C2C1 c1(C(N2CC(OC)(CO)C2)=O)coc2c1CN(C(=O)CC(=O)NC1CCCC1)C2 C(=O)(C(C)(C(C)C)ON)NC(CC=C)CNC(=O)Cc1cncc(C)c1 C1(C)(C(N(CC(C)(C)CNC(C2CC(CC(C)(C)C)C2)=O)C)=O)CCSCC1 Cc1cc(C)n(CCN(C(=O)CN2CCC(N(CCc3ncc[nH]3)C)CC2)C)n1 C1(NC(CCC2C(C)(C)C2)=O)COCCC1C(=O)NCC1CN(C(N)=O)C1 n1(CC)c(N(CCOCc2ccccc2)CCNC(C)=O)nnc1C(C)O c1(CCSCC)nc(-c2cnn(CCO)c2C)n(C(c2ccncc2)C)n1 N1(C(C(C)(CO)NC(c2cc(O)cs2)=O)=O)CCN2C(=O)NCC2C1 CC1CCCC1C(=O)NCCCOCCNC(=O)C(C)n1ccnc1 C1(C(=O)NC(C(C(C)C)O)C)CCCCN(C(=O)Cc2nc(=N)[nH][nH]2)C1 c1(NC(C2CCN(CCC)C2)=O)cccc(-c2cccs2)c1 c1(NC(N2CCC(c3cncc(OC)c3)C2)=O)cn2ccc(OC)cc2n1 c1(C(N(C23CCCC2N(C(C2CC2(C)C)=O)CC3)C)=O)ncnc2c1cnn2C C1(C(=O)OCC)CCCCN1C(C1CC(O)CN1C(C1CC1C)=O)=O CC(C(=O)NCC1CC(NC(c2csc3ccccc23)=O)C1)C1=CCCC1 N1(C(c2cccc(OC)c2)=O)CCC2CN(C(=O)C(CC(C)C)C(N)=O)CC2C1 CCC(O)C(=O)N(C)CCN(C(=O)CC1CCCOC1)C N1(C(CN(S(CC)(=O)=O)C)=O)CCOCC1CNC(=O)C=C1CCN(C)C1 c1(CN2CC(NC(C3CCCN(C)C3)=O)C(F)C2)cc(Cl)ccc1Cl N1(C(COCC)=O)CCCC(C)(C)C1CNC(=O)CC1(C)CCOC1 C1(C(N2CC(C(C)NC(c3cnn(C4CCCC4)c3)=O)C2)=O)CC2CC1C1CC21 c1(OC)ccc(CCC(=O)N(C)CC2CCCN2c2nccnc2F)cc1 C1(CN(C(c2ccncc2)C(=O)NC)CC)CCCN1CC1CCOCC1 C(=O)(C(C)C(O)C(C)CC)N(CC(=O)NC1CC(O)C1OC)CCOC C(=O)(C1=C(Cl)CCCC1)NCC1N(C(C(C(C)C)C#N)=O)CC(C)(C)C1 C(CC(O)C(F)F)NC(c1ccn(CCNC(=O)CC2C=CCC2)c1)=O O=C(CCCCCCNC(C1(n2cccn2)CC1)=O)N1CCC12CCC2 c1(C(N(C)CC2(CNC(C(CC=CC)C)=O)CC2)=O)cc2scc(Cl)c2[nH]1 c1(C(N2CC(CC)C(NC(=O)C(C)(C)C)C2)=O)ccc(C)c(S(N)(=O)=O)c1 c1(C(=O)NCC2N(C(C(C)OCOC)=O)CCN(C)C2)n[nH]c2ccc(C)cc12 C1(C(=O)NC(CCNC(=O)C(=O)Nc2ncc[nH]2)C(C)C)(OC)CCCCCC1 C12CC(C1(C)C)NC(=O)C2.c1(CCC(=O)N(CCOC)CCOC)nc(O)n[nH]1 c1(-c2nc(NC(C=NOC)=O)sc2)ccnc(NC(=O)OC(C)(C)C)c1 c1(OC)cncc(NC(C2COCCN2C(=O)Cn2nccc2C)=O)c1 N1(C(Cn2cc(CNC(COC)=O)nn2)=O)CCC(NC2CCC(O)CC2)CC1 S(=O)(=O)(CC(=O)N1CCC(C)(NC(=O)CC(C)C2CCCCC2)C1)NCC c1(N2CC(NCc3cccc(Br)n3)C3(C2)CC3)ncnc2c1CCCC2 C(CC(=O)N1CC(NC(c2c(C)cnn2C)=O)C(F)C1)(C(F)(F)F)OC CCCC(C#N)C(=O)NCCCCCC(=O)NCC(C)(COC)CC CCCCCCC(C)(C)C(=O)NC(C)CCCNC(=O)C(C)NC(C1CC1)=O N1(C(c2cc(C)c(Br)o2)=O)CCCOC(CNC(C2(C)COC2)=O)C1 c1(C(=O)OCC)cc(F)c(NS(=O)(=O)CCOCC2CCCO2)cc1OC c1(CNC(N2CCOC(CF)C2)=O)cc(F)cc(Br)c1Cl C1(C(N2CC(SCC)C2)=O)CC(C)(C)CCN1C(c1cc(C)co1)=O CCC(C(=O)OC)C(=O)NC(CC)CCC(=O)NC1(COC)CC1 n1(CC)c(N2CCOC(C3CC(F)(F)C3)C2)nnc1-c1nc(-c2ccsc2)no1 c1(CCC(=O)NCC2CCCCN2C(C2CCCC(F)C2)=O)ccc(F)nc1 C(C(C)N=c1cc(NCCCC(C)CO)nc(C2CC2)[nH]1)c1c(C)cccc1 C=CC1CN(C(=O)CCc2nc(C)c(C)[nH]2)CC1NC(c1ccc(F)cc1F)=O Cc1nc(N(CCCCN(C)C(c2cccn3ccnc23)=O)C)c(C)c(Cl)n1 c1(CC)ccc(CNC(=NCC2CCS(=O)(=O)N2)NC(C)C)cc1 C1(CCNC(c2n(CCC)ccc2)=O)CN(C(=O)C(C)=CC(C)(C)C)CCO1 CC(CC(=O)NC(C1CCN(CC(=O)N2CCC2)CC1)NC1CC1)C(F)(F)F C1(NC(c2c(CC)nc[nH]2)=O)CCCCN(C(C2CC2(C)C(C)C)=O)C1 c1(CC)nc(C)[nH]c1C(=O)NCC1(F)CCN(C(=O)C(=Cc2ccccc2)C)C1 N1(C(c2ccn(CCF)c(=O)c2)=O)CCC2(COC(CSc3ccccc3)C2)C1 CN1C2CCC1CC(CNC(=O)CC(C)(C)NC(C1CC3(CCC3)CO1)=O)C2 CS(=O)(=NC(=O)C1CCCC(C(=O)O)C1)c1ccc2ccccc2c1 Cc1cc([N+](=O)[O-])ccc1N1CCC(N2CCCC2c2ccc(O)cc2)CC1 C(CC(F)(F)F)N(C(=O)C(C1CCOC1)NC(c1c[nH][nH]c1=N)=O)C C(=O)(C(CC(C)C)C(N)=O)NC(CCNC(COc1cc(C)on1)=O)C(C)(C)C C1(C(=O)NC2(CNC(c3cc4cnccc4o3)=O)CC2)CNc2ccccc2O1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC(NC(=O)C(C(C)C)C2CCC2)C(C)C1 N1(C(C(C)(C)OCC(F)(F)F)=O)CCC2CN(C(C3CCCSC3)=O)C2C1 N1(C(C(CCC)O)=O)CCCN(C(=O)CCCc2ccc(Cl)cc2)CC1 C(=O)(C1=CC2C=CC(C1)C2)NCC1(O)CN(C(c2n(C)ncc2C(F)F)=O)C1 c1(OCC(=O)NC(CC)CNC(c2ccoc2C)=O)ccc(C#N)cc1Cl N1(C(c2cnc(C)[nH]2)=O)CCC2C(CCN2C(=O)Cn2cc(P(C)(C)=O)cn2)C1 N1(CC(NNC(c2c(OC)cccc2)=O)=O)CCC(F)(C#N)C1 C12(C(N(CC(=O)NCC(N3CCC(CC)C3C)=O)C)=O)C(=O)C3CC1C2C3 C1(n2ncc(C(=O)OC)n2)CCN(N2CC(O)CC2(C)C)CC1 C=CC1CN(C(=O)NCCC(C)(C)COCC)CCO1 C#CCC(C(=O)NC)NC(=O)CCn1cc(CN2CC(O)CCC2=O)nn1 C1(NC(CCCCC)=O)CCN(C(c2cccc(-c3nc[nH]n3)c2)=O)C(C)C1 C(=O)(CCC(=O)NC1(n2cc(Cc3conc3C)nn2)CC1)NC1(COC)CC1 C(=O)(CCC1=CCCCC1)N1CCC(=CCNC(c2csc(CO)n2)=O)CC1 N1(C(c2cn(CC)nn2)=O)CC(CNC(=O)C(c2ccc(OC)cc2)=O)CC1C Cc1cc(C)c(C(=O)NCC2CCC2NC(=O)CC2CCN(C)C2=O)c(O)n1 c1(C(N2C(C3(NC(C4CCCC4CF)=O)CC3)CCC2)=O)cc2ncccn2n1 c1(OC)c(C(N2CC(CC(C)(C)O)C2)C(=O)OC)cccc1C C1(C(=O)N(CCC(N)=O)C)(CC)CCN(C(=O)C(CCC)OC)C1 C1(CC(=O)N(CCC(C)(C)O)C)CN(C(=O)OC(C)(C)C)CC(C)(C)O1.OCC(F)F c1(-c2c(CNC(N3C(C)CC(O)C3)=O)nccc2)cnn2c1C(=O)N(C)CC2 c1(CCCC(=O)NCC2CC(NC(=O)Cc3cnoc3)C2)nc2ccccc2s1 C1(NC(c2c(CC)nn(C)c2)=O)CCN(C(=O)CCCC(C)(F)F)CCC1CO C(c1cccc(CO)c1)=CC(=O)NC1CN(C(C2(CC#C)CCOC2)=O)CC1O C1(C(=O)NC(C#C)(CC)CC)C2CC3C(C2NC(=O)C(C(C)CC)N(C)C)C13 N1(c2ccnc(NCC3(C)CCOCC3)n2)CCC2(CNC(=O)O2)C1 S(=O)(=O)(c1ccc(Br)cc1)N1CCCC(C(N2CC3CCC2CC3)=O)C1 CC(C(=O)NC1C2CC1N(C(=O)C#CC(C)(C)O)C2)C(F)(F)F C1(CCOC)CN(C(c2cccc(C)c2)=O)CCN1C(C1CCCN1C(N)=O)=O c1(CNC(C2CC3(CC3)CN2C(=O)CC2CCOCC2)=O)nc(Cl)ccc1F c1(OC)cc(-c2ccc(C(=O)NCc3cnco3)nc2)c2cn[nH]c2c1 N1(C(c2c(C)nc[nH]2)=O)CCCC(C2CCN(C(c3coc(Cl)n3)=O)CC2)CC1 c1(C2N(C(c3c(C)cns3)C(=O)NCCC3(C)CC3)CCC2)cccc(Br)c1C C1(C(=O)NCCCN(C(c2c(C)nc(C(C)OC)s2)=O)CC)CCC(C)(C)CC1 N1(C(C2(OC(C)=O)CC2)=O)CC2CCCN(C(C3CCCOC3)=O)C2C1 C1(C(N(CCCO)CC#C)=O)CCCN(C(c2cccc(CO)c2)=O)CC1 c1(C(=O)NC(c2ccnn2C)C(=O)NC(c2nn(C)cc2O)C)cnn2c1CCC2 C1(NC(CCOCCOC)=O)CC2CCC1(NC(=O)CN1CCCCC1=O)C2 c1(C(=O)OC)cnc(N(C2CCN(C(=O)CC34CCCC3C4)C2)C)c(C)c1 c1(C(=O)OC)ccc2c(c1)CN(CC1CCN(C(=O)CCCC(C)(C)C)C1)C2C c1(C(=O)NCCO)ccnc(Cl)c1O.C1(OCC=O)CCN(C(C2CCC2)=O)C1 Cc1nn2ncccc2c1C(=O)NCC1C2CN(C(C3CC(F)C(=O)N3)=O)CC12 c1(C(=O)NCC2C(C(=O)NCC(C)(C)NC(C)=O)C2)cccnc1C N1(C(c2c(C)cnnc2)=O)CCC(C(=O)Nc2ncccc2F)C(O)C1 c1(C(=O)OC)cnc(CO)[nH]c1=NC1CC(CNC(c2cnc(S)n2C)=O)C1 Cc1cc(C(=O)NCC2CN(C(=O)C(C)C3CCCC3)CC2C)c(F)cc1N N1(C(c2ncncc2F)=O)CC2CC(C1)N(C(C1CCCCCS1(=O)=O)=O)C2 C=CCC(C)C(=O)NC1(CNC(c2ccc(N(C)C)cn2)=O)CC(OC)C1 S(=O)(=O)(c1cc(C)cc(Br)c1)NC1C(C(=O)Nc2cc(SC)ncc2)C1 C=CC1(NC(=O)CC2(C)CCN2C(=O)Cc2sccc2C)CCOCC1 n1(CC(=O)NC2CCC(CC(=O)NCC(F)(F)CO)C2)cnnc1O N1(C(C2C(C(=O)NCCCC(C)C)CC2)=O)CCC(C2CCOC2)C1 C1(CC(=O)NCCN2CCCC2=O)CC2(C1)CN(C(c1ccccc1)=O)C2 N1(C(C(C)OCC)=O)CC2CC2(C(=O)N(CC(O)CO)C(C)C)C1 C1(C(N(C(CC)CSC)C)=O)CCN(C(=O)C2=COCCC2)CC1(C)C c1(C(=O)NCC2C(C(N(C(CC(C)C)C)C)=O)CCO2)cnccc1C#N C(=O)(C(O)CCC(C)C)NCC1C(NC(CCCCSC)=O)CC1 N1(C(CCC(CC)C)=O)CCS(=O)(=O)C(CCNC(=O)CC(F)(F)C(F)F)C1 C1(NC(c2cnn(CCF)c2)=O)CC2(C1)CN(C(=O)C(C1CCCO1)C1CC1)C2 c1(C=O)c(Cl)cc(F)cc1Cl.N1(NC)CCNC(=O)C1 C=C1CC(CF)(NC(=O)CNC(=O)CNC(C2COCC2C(=O)OCC)=O)C1 C(C1CCCCCC1)=CC(=O)NCC1CC(C(F)(F)F)CN1C(C1C2COCC12)=O Cc1cc(C(=O)NCCC2CN(C(C3CCC(=O)N3C(C)C)=O)C2)cc(C)c1Cl C1(CC)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(=O)Cc1csc(Cl)n1 Cc1ncc(Br)c(C(=O)NCCCNC(=O)C(n2cc(Cl)cn2)C)n1 C1(C(=O)NC2C(C(=O)NC(COCCOC)C)CCCC2)C2CCC(C2)C1C CN1CC(C(=O)NOCC(=O)NCc2cncc(F)c2)CCC1=O N1(C(c2ccc(-c3c(OC)ccc(Cl)c3)cc2)C)c2ccccc2NC(=O)C1C C1(C(=O)NCCOC(C)(C)CNC(C2CC(O)CN2C)=O)(OC)CCCOC1 c12ccccc1C(=O)N2C1CC1.c1(CNC(N)=O)cn(Cc2ccno2)nn1 c1(C(N2CC(CC(C)NC(c3cc(COC)[nH]n3)=O)C2)=O)cccc(C)c1SC N1(C(C2C3CCCCC23)C(=O)NC2(C)CC2)Cc2ccccc2CCC12CCC2 CN1C(=O)CCCc2occ(C(=O)NC3CCN(C(C4(Cl)CC4)=O)C3)c21 C1(C(=O)NC(C(=O)NC(CCC(C)C)C)C2CCCC2)CCCCC(=O)N1 c1(C(N(CC(C)NC(c2cnc3n2CCOC3)=O)C)=O)cc(Cl)c(F)cc1Cl CC(CNC(c1cncc(CO)c1)=O)CC(=O)NC1(CO)CC(F)C1 C1(NC(C2CC3CCC2O3)=O)CCCN(C(C2(CO)CC2)=O)CC1 N1(c2c(N)cccn2)CCC(N=c2nc[nH]c3[nH]c(Br)cc23)C1 c1(C(=O)NCCC(=C)CNC(c2cccc3nn[nH]c23)=O)cccc2c1CCC2 c1(CC(N2CC(C)C(NC(C3CCCN3C3CC3)=O)C2)=O)cccc2c1OCO2 C1(C)(C(N2CCC(O)(C(C)NC(C3CC(OC)C3)=O)C2)=O)COC(C)CO1 C1(CNC(c2cc(C)no2)=O)CCN(C(C2(C)C=CCC2)=O)CCC1(F)F C1(COC)(CNC(C2CCOC2C)=O)CCCN1c1ccc(C(F)(F)F)nn1 C1(NC(C2N(C(CC3(OCC)CCC3)=O)CCC2CC)=O)CCN(C)CC1C c1(OCc2cccc(C(=O)OCC)c2)nc(=O)c2cc(C(=O)OC)ccc2s1 C1(C(=O)NC(c2cccc(C)n2)C)(OC)CCN(Cc2ccc(OC)cc2)CC1 Cc1nonc1C(c1nnnn1CCC1(C)CC1)NCCCCCF N1(C(CCCCCC)=O)CCC2(CC1)C(OC)CC2NC(c1nccn1CC)=O N1(C(CCC=C(C)C)=O)CC2CC(C1)N2C(c1ccc(C(C)(C)C)o1)=O c1(C(c2n(C(C(=O)OC)C)nnn2)NC(C)(C)CF)nc2c(s1)CC(C)(C)CC2 C1(CN(C(=O)CCOC2CCCOC2)C)CCN(C(C2CCOC2(C)C)=O)CC1 C(=O)(C(CC(C)C)ONC(=O)OC(C)(C)C)N(C(C)CNC(c1ccnn1C)=O)C C(=O)(C(F)CCC(C)C)NC(CCC=C)C(=O)NC(CC)CCO c1(C(N2CCC(NC(CC=C(C)C)=O)(CO)CC2)=O)cc2c(N(C)C)cccc2s1 O(NC(=O)C(C)(C)C(C)NC(=O)C(C)S(N)(=O)=O)CCCC CC1(C(=O)NC23CC2CN(C(c2nnn(C(C)(C)C)n2)=O)C3)CC2(CCC2)C1 C(=O)(CCCCCCCC(=O)N1C2CCC1CC(NC(C1CCCO1)=O)C2)OC C#Cc1ccc(C(N2CC(NC(C3CCN(C)CC3)=O)C(C#N)C2)=O)cc1Cl C12CC3CCC(C1)N3C(=O)CCNC2=O.C1(C(=O)NC2CCSC2)CCOCC1 C(=O)(C(C(C)(C)C)OC)N1C(CC)C(NC(=O)CC2(O)CCCCC2)CC1 N1(C(C=CC(C)C)=O)CC2CN(C(c3cc(F)c(Br)cc3Cl)=O)CC2C1 CCCCCCCC(F)C(=O)N(C(C)CNC(=O)COC1CCC1)C Cc1nc(N2CCCCC2CNC(c2cnoc2CC(C)C)=O)c(F)c(C)n1 c1(-c2cc(C(=O)OC)cc(O)c2)ccc(S(=O)(=O)OC)c(Cl)c1 C1(NC(C(CN(C)C(C2CCCCC2(C)C)=O)(C)C)=O)CC12CCCCC2 C1(C(CO)NC(C2C(C)C(=O)C2)=O)CCN(C(C23CCC(C2)C3)=O)CC1 N1(C(=O)C(O)Cn2cncn2)CC(O)CC1C(=O)NC1CCCC1.C1(=O)CN1 CC(C)(CC(=O)NCC(C)(C)C(=O)N1CCC(C)(CO)C1)C(F)F C1(C(=O)NCc2ccc(C)o2)CC(C)CN(C(=O)CC2CN(C)C2)C1 CCCCCCCCC(C)CC(=O)NCCC1OCCCO1 C1(CNC(Cn2c(C)ccc2C)=O)CCC(C)N(C(=O)CCC2CCC(=O)C2)C1 C1(C(N2CC(n3cc(-c4nc(Cl)cs4)nn3)C2)=O)CC(=O)N(O)C1 c1(N2CCOCC(NC(c3nccc(OC)c3F)=O)C2)ncc2ncn(C)c2n1 C1(NC(C2COCCO2)=O)CN(C(c2cn3c(n2)COCC3)=O)C2(CCC2)C1 N1(C(CC=C(C)C)=O)CCC2(C1)CN(C(c1cnn(CCC#N)c1)=O)C2 Cc1ccc(=O)n(CC(N2CCC(NC(C3CC4(CCC4)CO3)=O)C2(C)C)=O)n1 C(C(CCO)CC(C)C)NC(c1nnnn1C1COC1)C1CC(C(C)C)C1 Cc1onc(Cl)c1C(N1CCC(CCN(C(=O)Cc2ccccc2)C)CC1)=O c1(CC(=O)NC(CCCC)CNC(=O)C(C)(C)C2CCCO2)cccc(Cl)c1Cl N1(C(CN2CC(=O)NCC2)=O)CC(CNC(C2(CCO)CC2)=O)N2CCC1C2 N1(C(CC2(C=C)CC2)=O)CCCC(C)(CNC(=O)C=C(C)C(F)F)C1 Cc1ccc(C(=O)NCCC2CN(C(=O)CCCc3ccc(CO)cc3)C2)nc1 C(N=c1[nH]c(C(N2CCC(N3CCCC3)C2)=O)cs1)c1c(C)cco1 C1(C(=O)NC(CNC(C(CC)n2cccn2)=O)(C)C)C2CCCOC12 C(CC(C)(C)CC(=O)N1CCCC(C)(c2cn(-c3ccccc3Br)nn2)C1)OC C(=O)(CC(O)C(C)CC)N(CCOCCC(=O)NC(CC=C)CC(=O)OC)C Cc1cc(O)c(C(N2CCOCC2CNCc2c(F)ccc(Cl)c2Br)=O)cc1Br Nc1cccc(Cl)c1C(N1CC(N2CCCC2)C(F)C1)=O c1(OC)nc(C(=O)NC2CCCC(CNC(=O)C(C)(C)c3cscn3)C2)sc1C n1(CC(=O)NC2(CNC(C(C)O)=O)CCOC2)cnc2sccc2c1=O N1(C(C2CCCN(CC)C2)=O)CCC(NC(=O)CSCCC(C)C)C(F)C1 C12(NC(c3c(C)oc(C(C)C)n3)=O)CCCC1CN(C(=O)C(C)N(C)C)C2 c1(CNC(C2C(C(N)=O)CC2)=O)ncccc1C(N1CCC(c2cc[nH]n2)C1)=O c1(CN(C)CC2(CC)CCCOC2)c(O)ccc2c1CCC2 N1(C(C(F)OC)=O)C2CCC1CN(C(c1ccc(-c3ccccc3)cc1)=O)CC2 c1(C(N2CC3(CCN(C(c4ccns4)=O)C3)C2)=O)nc2n(c1Cl)CCCC2 C1(NC(C2C(C)CN2C(=O)C=Cc2cnccn2)=O)CC2CC1CC2O C1(CC2N(C(CC(c3cc(C)cc(Cl)c3)N)=O)CC2)CCc2cc(F)ccc2O1 C1(NC(C2(C3N(C(CCC#C)=O)CCC3)CC2)=O)CCN(CC=C)C1=O Cc1cc(Br)ccc1C(=O)NC1CC(CNC(=O)CN(C)C(C)C)C12CCC2 C(=O)(CN=S(C)(C)=O)N1C(C2(NC(c3nc(C(C)OC)oc3)=O)CC2)CCC1 N1(C(C(CC)OC)=O)CCCCC(CNC(=O)C(C)(C)COC(C)=O)C1.OCC C1(C)(NC(CNC(CC)=O)=O)CCCCC1C(=O)NCC1(F)CC1 Cc1nc(NCc2csc(C)n2)cc(N(C)Cc2cccc(C)c2F)n1 C(CC(C(C)C)NC(=O)CSc1ccc(F)cc1)N(C(C1C(C)=C1)=O)C C1(C(=O)NC(C2CCCC2)C)CCCN(CC=Cc2ccccc2)C1 C1(NC(Cc2cn(CC)nc2)=O)CN(C(C2CC(=O)C2)=O)C2CCCC12 C1(C(N(C(C)CC(C)C)CCOC)=O)CC(NC(=O)CSC)C(O)C1 C1(NC(CCC(C)SC)=O)COC2(CCN(C(C3CC(F)C3)=O)CC2)C1 C1(NC(CCC)=O)CC2(CCN(C(c3nc(C)ncc3F)=O)CC2)C1 C1(CCNC(C(C(C)C)NC(C)=O)=O)CN(n2cc(CN(C)C)nn2)CCCO1 C=C(C)CCC(=O)NC1C=CCN(C(=O)C(C)(C)c2cnco2)C1 c1(C(N(CC(CN(C(=O)CC2CCC(=O)N2)C)O)C)=O)cnn(C)c1Br C1(NC(c2csc(C)c2N)=O)CCN(C(c2cc(O)nn2C)=O)CC1(C)C c1(C(N2C3C(NC(c4n(CC)ncn4)=O)CC(C3)C2)=O)nc2cc(F)ccc2s1 c1(C(=O)NCC(CNC(C(C)c2ccsc2)=O)F)scnc1C1CC1 c1(C(=O)NC(CCOC)CNC(=O)C(CC(C)C)N(C)C)cnc2c(c1)COCC2 N1(C(c2cc(CC)on2)=O)CC(NC(=O)C(=Cc2ccncc2)C)C2CC12 Cc1cn(C(C)C)cc1C(N1CC(NC(=O)CCOCCN(C)C)C(O)C1)=O c1(OC)ccc(C(N2CC3CC3(NC(c3cnn[nH]3)=O)C2)=O)c(Cl)n1 c1(C(=O)NC2C(CNC(CC(C)C(F)F)=O)C2)cc(=O)c2ccccc2n1C c1(CN2CC(F)CC(C(N(CCC)CCC)=O)C2)ccc(F)c2ccoc12 N1(C(CSCC(N)=O)=O)CC2OCCN(C(=O)CCc3ccc(N)c(F)c3)C2C1 n1(CCNC(C(C)C(=O)NC(N)=O)(C)C)cc2ccccc2n1 c1(C(=O)NCCCN(C(C2CC(F)C2)=O)CC)ccnc(OC(C)C)c1 C1(CCNC(c2cc(COC)no2)=O)CN(C(=O)C2=CCC2)CC1C C1(NC(C(C=C=C)C)=O)(CO)CCCN(C(c2coc(-c3ccccc3)n2)=O)C1 N1(C(C2CC(CC)C2)=O)CCN(C(c2cc(Br)sc2C)=O)CC1C N1(C(c2ccc(C)o2)=O)CCC(CNC(C2(COC(C)C)CC2)=O)CC1 C1(N(C(CSCCC)=O)C)CC2CCC(C1)N2C(C1(C)CCC(C)=C(C)C1)=O CCCC(C(=O)NC(C1CC(NC(c2cnc(C)nc2)=O)C1)C)N(C)C c1(CC2C(=O)O2)cccc(N(CC#N)C(C)C)c1.C1C(=O)N1.C(C)(=O)OC N1(C(=O)NCCc2nnc(S)n2C2CC2)CCC2(CC1)COC(CO)C2 N1(C(Cc2scc(CC)n2)=O)C(=O)NC2(CCS(=O)(=O)CC2)C1=O c1(C(=O)NC(c2nocc2C(=O)NCc2cnn(CCO)c2)C)cc(=O)cc[nH]1 c1(C(N(C2CCCCN(C(C(C)n3cccn3)=O)C2)C)=O)nc2cccnc2s1 CC1(F)COCCN(c2cc(NCc3nc[nH]n3)nc(C(F)(F)F)n2)C1 C1(N(C(c2cnc(C)o2)=O)OCC)CCN(C(=O)C2CC2)CC1 c1(NC(C2CCOC(c3cnn(C)c3)C2)=O)c(O)cc(C(=O)OC)cc1I c1(C(C(=O)OC)N(CC(C)C)Cc2ncc(C(=O)OC)s2)cnccn1 c1(OC)ccc(F)c(C(=O)NCC2C(C)CCN2C(c2cc(C)ccn2)=O)c1 S(=O)(=O)(c1cccs1)NC(C)C(N1CCC(O)(Cn2cc(C3(O)CC3)nn2)C1)=O N1(C(c2c(OC)nn(C)c2)=O)CCN(C(c2cnns2)=O)CC1c1cnn(C)c1 N1(C(C2C(C(C)=O)C2(C)C)=O)CC(C(N2CCC(C#N)CC2)=O)C(C)(C)C1 C#CC1(C)CCCN(C(=O)CC2CCCN(C(=O)CCC(C)(C)OC)C2)C1 Cc1ccc(-c2nc(C3CCOC3)nn2C)c(C(F)(F)F)c1 CCC(C)C(O)CNC(=O)CC(CC)N(C)C(C1(C)CCC1)=O c1(C(C(=O)NCCCCCC)N(C)C(C2(C)CC2)C)nccnc1OC(C)(C)C C1(NC(CN(C(C)=O)Cc2csnc2Br)=O)CCCC(NC(C)=O)C1 C1(C)(CC)CC(NC(=O)CCNC(N)=O)CN1C(=O)C1=C(C)CCC1 Cc1ccc(S(=O)(=O)N2CC(O)CC2C(N2CC(O)C2)=O)cc1C Cc1nccc(Br)c1NC(C1CCC(O)C1O)=O N1(C(C(CC)C)=O)CC2CCC(C1)N2C(c1cnn(-c2cccc(F)c2)c1C)=O C(C)(CC(C)N=c1nc(C2CC2)[nH]s1)NC(C(C)=C1CCC1)=O N1(C(c2cn(CCCF)nn2)=O)CC2CC(C1)CN(C(C1CCS(=O)CC1)=O)C2 N1(C(C(C)Oc2ccccn2)=O)CCC(C)CC1CNC(c1c(Cl)nn(C)c1Cl)=O CCCCC(O)C(C)C(=O)NCC(C)NC(=O)C(C(C)C)N(CC)CC N1(C(C(C=C)(C)C)=O)CCC(C2CC(NC(c3nn(C)cc3Cl)=O)C2)C1 C1(C(CCNC(C(C)N(C(=O)CN(C2CCCC2)C)CCC)=O)O)CCCCC1 N1(c2n(C(C)CN3CCCC3)c(-c3cc[nH]n3)nn2)CCC2C(C1)C2(F)F c1(C(=O)NCC(C(=O)N(CC(=O)NCCC)C)N(C)C)cccc(CC)c1 c1(CC(=O)NC(CN(C(C2CCCC(C)(C)C2)=O)CC)C)cc2ccccc2s1 C1(F)(C(=O)NCC(C)(C)C)CN(C(=O)COCC(=O)OC(C)(C)C)C1 C1(CNC(CN2C(C)CC2)=O)CC12CCN(C(=O)COc1ccsn1)CC2 c1(C(=O)NCC(CC(C)C)NC(=O)C(F)C(F)(F)F)cc2c(cc1Cl)CCCC2 CC(C)CC(C(=O)NC1CCCC1NC(c1ccc(Cl)[nH]1)=O)C(C)C c1(C(=O)NCC(CC=C)NC(=O)CC2CC3CC3C2)c(C)ccc(C)c1N C12(NC(CC=C(C)C)=O)CCCC1N(C(c1cc(C(N)=O)ccc1O)=O)CCC2 CC(CC(=O)N1CC(NC(=O)CCCCN2CCCCC2)CC(O)C1)C(F)F N1(C(CC2C(C)CC2)=O)CCN(C(=O)CCCCC2CC2)C2CC12 C1(CCNC(CCCOCC)=O)CN(C(c2cnc(-c3cccs3)s2)=O)CCO1 N1(C(c2cnn(C)n2)=O)CC(NC(=O)CN2CCCC2=O)C(O)C1 c1(C(N2CC(NC(C3(CF)CC3)=O)C(F)C2)=O)c[nH]c2cccc(Cl)c12 Cc1nc(NC(=O)CC2(CO)CC2)ccc1C(=O)OC(C)(C)C C(CCC(C(=O)NN1CCCCC1=O)OC(=O)Nc1ccccc1)OC Cc1cnc(NC(=O)CC2CCCCN2Cc2ccc(Cl)s2)c(Cl)c1 C(CCN=C(NCC)NC(C)CC1(C)CC1)(C1CCCC1)OCC C(=O)(C(Cc1ccoc1)NC(C1CC1C(N)=O)=O)NCC(C)C#N c12cnc(cc1C)NC(=O)C2N(CCCCC)C.c1(C(=O)OC)ccccc1 c1(C(=O)NCC(CCCC)NC(c2ncnc(C)c2C)=O)ccc2nc[nH]c2n1 c1(C(NOC2CCN(CC(=O)OCC)C2)=O)cc(CC)cc(O)c1 C1(C(=O)NC(C)C(=O)NCCN(C)C(c2ccoc2)=O)CC2CCC2C1 C=C1CCN(C(C2COCOC2)=O)C(C(=O)NCCc2ccc(C)s2)C1 c1(C(N2CCC(CCC(=O)N3CC(c4ccon4)C3)C2)=O)cncc(Cl)c1 C1(NC(C(c2ccc(C)cc2)(C)C)=O)COC2CN(C(=O)C3=CCCOC3)CC12 N1(C(C2N(C(C(CCCC)F)=O)CSC2)=O)CCCC2C(O)CC12 NC(=O)CCC(=O)NC1CCC1CNC(=O)CN1CCCCCC1 C1(c2cn(C)nc2)CCCCN1C(c1c(I)cnn1C)C(=O)NC1CC1 c1(N(C(c2c(C)ccs2)=O)C)cc(CN(C)C)n(C)n1 N1(C(COc2cn(C)nc2)=O)CC2C=CC1C(C(N1CCOC3CC13)=O)C2 c1(C(=O)NCC2CCC(NC(CN(C(=O)OC)C)=O)C2)noc2c1CCCC2 c1(C(N2CCN(C(C(CC=CC)C)=O)CC2CCOC)=O)nccn2ccnc12 C(=O)(CCC(C)(C)C)N1CC(O)(C(C)NC(C2CCC(F)(F)C2)=O)C1 N1(C(C(Cc2ccoc2)NC(CN(C(=O)OCC)C)=O)=O)CCC(F)(F)CC1C c1(CNC(c2ccc(CC(N)=O)cc2)C)cc2ccccc2nc1F C1(CC(=O)NCC2(CN(C)C(c3ccc(Cl)s3)=O)CC2)CC(O)C12CCC2 Cc1ccncc1CC(=O)NCC(C)NC(=O)CO Cc1cc(Cl)cc(C)c1OCCNC(=O)OCC1CCCCC(O)C1 N1(Cc2cc(C)ncc2)CCC(F)(F)C(C(=O)Nc2cnccc2CO)C1 c1(CN2C(C(N(CC(CC)NC(c3ccccc3)=O)C)=O)CC2)ccc(C)nn1 CCCCC(O)CC(=O)N1CCN(C)C(CNC(=O)COC(CC)CC)C1 C(c1cc(Cl)c2c(c1)OCCO2)=CC(=O)NCC1CN(C(CCOCCC)=O)C1 c1(C(=O)NCCCN(C(C2CC(C)OC2)=O)C)cn(C)nc1-c1cccnc1 C1(Cc2coc(C3CCCCN3)n2)CN(CCC)CCO1 N1(C(C=CCN(C)CC)=O)CC2CCC1C1CN(C(=O)C#CC(C)(C)C)CC21 c1(C(=O)OC)c(C(=O)NCCN(C(=O)C(F)(F)CN(C)C)C)[nH]c2ccccc12 c1(C(CC)CC)cn(CC(CNC(C2(Cl)CC2(C)C)=O)OC)nn1 Cc1cccn2ncc(C(=O)NC(C)(CNC(c3cnc(C)n3C)=O)CO)c12 c1(C(=O)NCCC(C)NC(c2cnn[nH]2)=O)cccc(-c2cc[nH]n2)c1 c1(N(C)C)cnc(C(c2nnnn2CCCF)NC2CCCC2F)nc1 N1(C(Cc2nc(C)[nH]n2)=O)CCOC(C2CCOC2)C1 C(=O)(C1=Cc2ccccc2C1)NC(CCOCC)C(=O)NCCCOC(=N)O c1(C(N2C3C(NC(CCN4CCC(C)CC4)=O)C(C3)C2)=O)ccc(C#N)c(F)c1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CC(C(=O)NOCC2CCCO2)C2(CCC2)C1 c1(C(=O)OC)cc(NC(=O)CC2(C)CN(C(C3NC(=O)NC3=O)=O)C2)ccc1Cl C(=O)(CCCCC(=O)NC)NC1C(NC(CC(CC)SC)=O)CCC1 Cc1scnc1C(=O)NCC(O)CNC(=O)CCC1CC1(F)F Cc1noc(C(=O)N(CCCNC(C2CC2F)=O)Cc2ccccc2)c1C C(=O)(CCCCC(C)=O)N(CCC(=O)NCC(CO)CC(C)C)CC=C c1(C(=O)NCCN(C)C(C2(c3cnn(C)c3)CCCO2)=O)cc(Cl)cnc1O CC1CC(N=c2nc(O)c3cnn(C)c3[nH]2)CN1C(=O)CCC(F)(F)CN=[N+]=[N-] c1(C(N2CC(C)C(NC(C3COCCO3)=O)C2)=O)cc(CO)ccc1Cl C1(C(C=CCCC)=O)CN(C(C2C=CC2C(=O)NCC)=O)CC1OCCSC C1(O)(CN(C(=O)C(C)(C)N2CCCCC2)C)CCCN(C(C2(C)COC2)=O)C1 CCC(C)CCCCC(=O)NCC1(C)CC(OC)CN1C(=O)C(O)Cn1cncn1 C=C(F)C1(CC(N2CC(F)(CNC(=O)COC(C)C)C2)=O)CCOCC1 C1(C(N(CC(CC)NC(c2cn(C(C)C)cn2)=O)CC)=O)CCCCC1O c1(CNc2c(C(N3C(C#N)CC(F)C3)=O)nccc2)ccc2nonc2c1 C1(CNC(C=C(C)C(F)F)=O)CN(C(=O)CC2CCCCCCC2)CC(C)(C)O1 c1(C(=O)NCC(CC)NC(c2cc(C(C)C)[nH]n2)=O)[nH]nc(C)c1O c1(CC(=O)NCCNC(C2C(COC)CC2)=O)cc(OC)ccc1OC N1(C(C(C)NS(CC)(=O)=O)=O)CC2CC2(CNC(c2ccc(N(C)C)cc2)=O)C1 c1(C(CC)O)nc(-c2ccnn2C(C)C)n(-c2cccc(Br)c2)n1 c1(OC)cccc(OCC(=O)NC2CN(C(c3ccc[nH]3)=O)C3CC23)c1 N1(C(CC=CC=C)=O)CCC(C2CCC2)(CNC(=O)C(C)O)CC1 C1(NC(C(C)(C)CF)=O)CCN(C(C2CC3(CCC3)C2)=O)CC(O)C1 c1(C(=O)NC2CCN(C(CC3OCC(C)OC3)=O)C2)cc(F)cc2ccncc12 C1(N(C)C(c2cc[nH]n2)=O)C2CN(C(C3(C)CC3Br)=O)CC12 c1(CN(C)C)ccc(C(C)NC2(c3n(CCCCCC)nnn3)CCOC2)cc1 C(=O)(C(F)C(CC)CC)NCC1CCN(C(CCCOCC)=O)CC1O CC1(C)CCN(C(C2CC(=O)C2)=O)CC1C(N1CC2CC=CCC2C1)=O c1(CNC(C2CN(C(c3ncn(C)c3C(F)(F)F)=O)C2)=O)ccc(F)nc1F Cc1cccc(C(C)NC(=O)C(C)NC(c2cccc(F)c2)=O)c1 c1(C2(C(=O)O)CCC2)ccc(C(=O)NCC2(O)CN(C(=O)C(F)C3CC3)C2)cc1 N1(C(c2c(CC)occ2)=O)CC(C(=O)NOCC2(O)CCCCC2)CC(C)C1 C(=O)(CC(C)(F)F)NCC(C)(C(C)C)NC(CCC(C)C)=O N1(C(C(CC(C)C)O)=O)CC2(C1)OC1(C)CC2(NC(=O)CS(=O)(=O)N(C)C)C1 C1(C(=O)NCCn2c(CSC)ncc2)CN(C(C2(O)CCOC2(C)C)=O)CC1(C)C CCC(C)(CNC(C1CCOC(C)(C)C1)=O)C(=O)NCc1ncccn1 CP(C)(=O)C1CCCC=C1C(=O)N1CC(F)(CNC(=O)CN2CCSCC2)C1 C(Cc1ccc(C)cc1)(CC(=O)O)NC(COC(CC)C)=O c1(CCC(=O)N(C2CCN(C(c3csc(COC)n3)=O)C2)CC)nc(C)c(C)o1 N1(C(C2CN(C)C(=O)N2)=O)CCC2CN(C(c3cc(C#N)ccc3O)=O)C2C1 c1(C(=O)NCC(C)NC(=O)CS(=O)(=O)NC(C)(C)C)cccc(O)c1[N+](=O)[O-] N1(C(CCc2cnc(C)o2)=O)CC(NC(=O)CCC(C)C)C(N=[N+]=[N-])C1 C1(CNC(COCc2cccc(OC)c2)=O)CCN(C(=O)C(C)N(C)C)C1(C)C N1(CCNC(c2ccc(COC)cc2)=O)CCC(N=c2[nH]nc(C(N)=O)s2)CC1 N1(C(COC(CC)CC)=O)CCCC(CC)(NC(c2cccc(=O)n2C)=O)C1 C12(COC)CC(CNC(C3CCN(C)C3=O)=O)(CN1C(c1nccnc1N)=O)C2 C1(C(=O)NCc2c(C)scn2)C(C2CC2)CCN1C(=O)C(CN(C)C)N(C)C C1(CNC(c2n(CC)cnn2)=O)C2CCCC1N(C(C1CC=CC1)=O)C2 CC1(CNC(=O)C(Cn2cncn2)NC(=O)COCC2CCCC2)CCCC(=O)N1 c1(C(=O)NCC2C=CC(NC(c3cnc(CC)s3)=O)C2)nc(C)c(C)nc1C C(=O)(CCN1C(=O)CCc2ccccc21)NC(C(C)NC(C1=NOC(C)C1)=O)C c1(C(=O)NC2CCN(C(CC(CC)SC)=O)CC2)cc2ccc(F)cc2s1 c1(NC(Cc2cc(CC)no2)=O)ccc2c(C)cc(C)cc2n1 c1(C(=O)NC(CC)(CNC(=O)CC2CCCC(OC)C2)CC)ccc(N)c(O)c1 Cc1noc(C2CC2NC(=O)CNC(=O)CNC(=O)C(N)=O)n1 c1(C(=O)NCC2(OC)CN(C(c3cncnc3)=O)C2)cnc(O)c(F)c1 C1(CC(=O)NC23CCCCC2C3)CCN(C(=O)C2CC2)CC1C1CC1 c1(C(=O)NC2(C)CCN(C(c3cc(Br)no3)=O)C2)cccc(C#N)c1 c1(C(=O)NCC2(CCNC(=O)COc3cn[nH]c3)CC2)ccnc(F)c1F N1(C(C(c2ccccc2)OCC)=O)C2CCCC1CC(NC(C1CC1CC)=O)C2 N1(C(C2CC(CC)OCC2)=O)CCC2(C1)CN(C(C1CCCC3CC13)=O)CCO2 C(CC(C)(C)C)(C(=O)NC(CCN(C(=O)CCC(F)(F)F)C)C(C)(C)C)OC C1(C(=O)NC2CCC(NC(c3n(C)c(C#N)cc3)=O)C2)CC2CC(O)C(C1)C2 C1(NC(c2nc(CC)sc2N)=O)CC2CCC(C1)N2C(C1CCOCC1)=O Cc1ccc(Br)c(C(=O)NC2CC(NC(c3sccc3-n3ccnn3)=O)C2)c1 C1(CNC(CCC=CCC=C)=O)CCC2CN(C(c3ccon3)=O)CC12 C1(CNC(CSCC#C)=O)Cc2ccccc2CN1C(=O)C(C)(C=C)CC C(CCC[Si](C)(C)C)NC(C#CC(OCC)ON)C.C1CCC1 c1(C(N2CCC(OCCNC(Cn3nnc(=N)[nH]3)=O)C2)=O)cccc2cc[nH]c12 c1(N2CCCC(CSC)C2)nc(C2CC2)nc2c1CCCC2 c1(-c2cn(NCC3N(C(CC(C)(C)C4CC4)=O)CCC3)nn2)cccc(Br)c1F N(C(=NCCCc1cn[nH]c1)N1CCC(c2cc(OC)ccn2)C1)CC(=C)C N1(C(COC(C(C=C)c2ccccc2)=O)=O)CCS(=O)CC1 c1(C(N(c2c(C)cccn2)C)=O)nc2n(c1Cl)CCN(C(c1ccsc1)=O)C2 Cc1ccc(C(N2CC3(CC3)CC2CNC(C2CCCS2)=O)=O)cc1C c1(OC)ccc2c(c1)CC(C(=O)NC1CC1NC(c1csc3nccn13)=O)O2 C1(C(=O)NCCCC(=O)NC(C#C)C(C)OC)CC(=O)NC1(C)C C1(C(=O)NCCCNC(c2n(C)c(=O)ccc2)=O)CCN2CCOCC12 c1(NC(C2CC(=C)CN2C(c2ccc(N(C)C)c(C)c2)=O)=O)cc(F)ncc1C N1(CC(=O)NCC(CO)NC(c2c(C)ncn2C)=O)CCn2ccnc2C1 C1(CNC(Cc2ccc(OC)cc2)=O)CN(C(=O)CC(C)C(F)F)C(C)(C)C1 C(=O)(C1CCc2nccn21)NC1(C)CCN(C(c2c(N)cn(C)n2)=O)C1 N1(C(=O)NC2CCCCC2C(=O)NCC(F)(F)F)CCN(c2cnccn2)CC1 CC1(CNC(=O)CN(C2CCC2)C(c2cc[nH]n2)=O)CCC(=O)N1 C1(OC(=O)CCn2cncn2)CCCC(c2ccccc2)C1 c1(C(N2CC(C(C)(C)O)(CNC(C3(CC#C)CCCO3)=O)C2)=O)cc(C)nn1C O(N1CCC(CC(=O)NC2CCCN(C(c3sccc3OC)=O)C2C)CC1)CC N1(C(C2N(C)CC(C)(C)C2)=O)C2CCC1CN(C(C1CC(C)(C)CN1C)=O)C2 c1(C(=O)NC(CC)(C)CNC(=O)C(C)C(F)F)cc2sc(Br)cc2[nH]1 C1(NC(C(CC(C)=O)C)=O)CN(C(c2ccc(Cl)s2)=O)CC12CCC2 C1(C(=O)NC2(CF)CCN(C(c3scnc3Cl)=O)C2)CC2(CCC2)CO1 CC(C)CCCCC(=O)N1CCCCCC1CNC(c1ccc(CO)s1)=O C1(CC(=O)NCc2c(C)csc2)CCC(NC(=O)CN2CCCCCC2)CC1 C1(C(C2(C3CCCCO3)CC2)=O)(CNC(c2ccc(CSC)s2)=O)CCOCC1 CCC(O)C(F)(F)C(=O)NCC12CCC(CC1)N2C(C1(C)CNC(=O)C1)=O c1(C(=O)NCC2(OC)CCN(C(C3CC(O)CN3C)=O)C2)cccc(F)c1SC C(CCC(C)(C)C(=O)N1CC2(CC(CO)CO2)C1)NC(C(C)S(N)(=O)=O)=O c1(C(=O)NC(C2OCCN(C(c3c(C)[nH]cc3)=O)C2)C)ccnc2c1ncn2C Cc1cc(C(=O)NCC2CN(C)CCN2C(=O)C#CC(C)C)ccc1Cl c1(-c2c(OC)ccc3ncccc32)nc(=NC2CCN(CC)C2)[nH]c2ccccc12 CN1C(=O)OCC12CN(C(C1C=CCN1C(=O)CC1OCCC1(C)C)=O)C2 c1(C(=O)NC(CN(C(C23CCC(OC)C2CC3)=O)C)(C)C)ccc2c(c1)CCN2 c1(C(N2CC(CCC)N(C(=O)C(CO)N(C)C)CC2)=O)cc2c(C)cccc2o1 C1(CNC(C(C)c2cc[nH]n2)=O)CN(C(C2CC(C)(C)C2)=O)C(C)(C)C1 CC1=C(C(=O)N2CC3(C)CC2(C(=O)NC2CCCCC2C#N)C3)COCC1 C1(CNC(c2n(C(C)C)nnc2)=O)CCN(C(c2ncoc2C2CC2)=O)C1(C)C CC(C)CC(CNC(c1cnsc1)=O)NC(C1(c2cccc(Cl)c2)CC1)=O C1(CNC(C(C(C)C)O)=O)CN(C(c2cc(CCCO)on2)=O)CCC1(C)C c1(C(N(CCC(C)NC(=O)CC2CCC=CCC2)C)=O)ccc(=N)[nH]c1 C(c1ccc(C)cc1)=CCC(=O)NC(CC)(C)CCNC(C1OCCC1C)=O N1(C(C2(CC=C)CCCN2C(=O)CCc2ccncn2)=O)CCOCC(CO)C1 c1(C(=O)NCC#CCNC(C2C(C(=O)OC)C2)=O)n[nH]c2nccc(Cl)c12 c1(OCC)cccnc1C(=O)OCCCCOC(C)CC(C)OC C(=O)(N=c1ccn(CC2CCCC2)[nH]1)N1C(C(C)(C)F)CCC1 c1(C(C)C)cc2c(N3CCC(O)C(C(=O)N(C)C)C3)ncnc2s1 c1(OC)ccc(C(=O)NC2CC3COCC2O3)nc1C N1(C(C=C(CC)C)=O)CCN(C(=O)CC2(C)CCOC2)C(C)C1 c1(CCC(=O)NCCC(C)NC(=O)CCNC(C2CCN(C)C2)=O)cccn1C N1(C(COCC#C)=O)CCC(NC(c2ccc(OC(C)C)nc2)=O)C(C)C1 C(=O)(C(C)CC(F)(F)F)NC(C(N1CC(CC)N(C)CC1)=O)Cc1cn[nH]c1 N1(C(c2ncc(C(F)F)s2)=O)CC2C(CNC(C3(CC(F)F)CC3)=O)C2C1 c1(COC)nc(NC(C2CCCCC2)C)cc(=NCc2noc3c2CCCC3)[nH]1 CCCCCCCCNC(=O)CC(CC1CC1)NC(=O)CC1(C)CCOC1 C(CCCC(CO)NC(C1CCCN(CC(F)F)C1)=O)NC(CCCN(C)C)=O c1(OC)ccc(-c2nc(C)c(C(C3CC3)NC34CCCC3C4(F)F)s2)cc1OC C1(CNC(c2n(CC)c(O)nc2)=O)CN(C(=O)C(C)n2ccnc2)CC1(C)C C1(CC=C)(C(N2CC(C)(F)C2)=O)CCN(C(=O)CC(C)CC)C1 C1(C(=O)NCC(CC=C)NC(c2scnc2C(C)C)=O)CCCC(C)O1 Cc1nc(CC(=O)NCC2CCN(C(=O)C(C)CC3CCCC3)CC2)[nH]c1C c1(C(=O)NCCN(C(C2C(C)(CC)C2)=O)CC2CC2)cc(C(F)F)ncn1 C1(NC(c2cnco2)=O)CCCCN(C(=O)CCc2ccc(F)c(F)c2)C1 C1(N(C(C(C=C=C)C)=O)C)CCCN(C(=O)C(F)=CC2CC2)CC1 C1(NC(c2cc(O)ncn2)=O)CCS(=O)(=O)C12CN(C(C1CCCCC1)=O)C2 Cc1sncc1C(=O)NOCC(=O)N(C1CCOCC1)C1CC1 CC1CN(C(=O)C(O)CN(C)C)CC1C(=O)N(C1(C)CCCC1)C c1(C(=O)OCC23CC(C)(OCC2)C3)c(F)ccc2c1OCC2 CCC(C)(C)C(C)CC(=O)N1CC(F)CC1CN(C(=O)COCCOC)C N1(C(C(=O)NCCNC(C)=O)=O)CCC(NC(C2CC3CCN2CC3)=O)C(C)C1 Cc1ccc(C(=O)NCC(CO)NC(C2CC3(C2)CC3(F)F)=O)cc1N C1(NC(C2(CC=C)CC=CC2)=O)CC2CCC(C1)N2C(C1CC12CC2)=O c1(NCCS(CC)(=O)=O)ccc(S(=O)(=O)NCC(=O)OC)cc1[N+](=O)[O-] C(=O)(C(CC)CCc1ccccc1)N(CCOCCCNC(C1C(=C)C1)=O)C c1(C(=O)NCC2N(C(CCC(C)=O)=O)CCN(C)C2)cn(C)c(C)cc1=O C(=O)(CCC(COC(=O)COC(=O)C(F)(F)F)C(F)(F)F)OC N1(C(COC(CC)CC)=O)CC(O)(CNC(c2ncsc2C)=O)C1 c1(CC(=O)NCCCCCN(C(=O)CCC2CCC2)C)ccc2oc(O)nc2c1 N1(Cc2onc(C)n2)CCC2(CC1)CC2C(=O)NCc1nnc(O)o1 c1(C(N2C(C)CCC(NC(c3c(CC)occ3)=O)C2)=O)cc(F)c(F)c(Cl)c1F N1(C(C2N(C(CN(C)C(N)=O)=O)CC2)=O)CC2CCCC(C1)N2C N1(C(C2CCC(=O)NC2)=O)CCC2CCCC12C(=O)NC1CCCOC12CCC2 C(c1nc2ccccc2o1)=CC(N1CC(OCCNC(C=CCCC)=O)C1)=O N1(C(c2n(CC=C)ccc2)=O)CCCC(NC(=O)CCC(C)CC)C1C c1(C2C(C(=O)NCC(C(C)C)Cc3nnc(C(C)C)o3)C2)ccc(F)cc1F C1(NC(=O)CN2CC=CC2)CC2CC(NC(=O)C(F)(F)c3cnccn3)C1C2 N1(C(CS(N)(=O)=O)=O)C2CCCC1CC(NC(=O)C(F)CC1CCOC1)C2 n1(C(C)C)cc(C(=O)NC2CCC(NC(C3(CCO)CC3)=O)C2)ccc1=O C(=O)(C(CC1CCC1)NC(C1(NC(=O)CC(C)SC2CC2)CCCC1)=O)OC c1(C(=O)NCCC2CN(C(C(COC)OC)=O)CC2C)cc(C#N)ccc1F N1(C(Cc2ccc(C)o2)=O)CCCC(C(C)C(=O)NC(C(C)C)C(C)C)C1 N1(C(c2cccc(OCC)c2)C(=O)NC2CCC2)CC(CC)OC(C)(C)C1 C(=O)(CCCCCCCC1CC1)N1CC(O)(C(C)NC(C(C(C)C)OC)=O)C1 C#CC1(C(N2CCC(C(C)CNC(=O)C(CN(C)C)N(C)C)CC2)=O)CCCC1 C#CC1CN(C(=O)C=CC(C)(C)NC(=O)Cc2cccs2)CCO1 C1(NC(C(C=C)(C)C)=O)CN(C(C2CC3CCC3C2)=O)CC1N=[N+]=[N-] C1(C(N2CCCC(OC)C2)=O)CC12CCN(CC(=O)NC1CCCC1)CC2 C1(NC(C(C)OCCC(C)C)=O)CN(C(=O)C=Cc2ccccc2)CC2(CC2)C1 c1(OC)c(Cl)cc(CC(=O)NC2(CNC(=O)C(F)OC)CCCC2)cc1Cl c1(NC(C2CC(NC(C)=O)C2)=O)ncnc2c1ncn2C1CC(O)C1(C)C CCC(CC(=O)N1CC2CC(NC(=O)CN3CC(C)C3)C1C2)C(C)C c1(CC)cnc(C(N2CC(C)CC2c2ccccc2F)C(=O)NCCSC)cn1 N1(C(C=C(C)C(C)C)=O)CCC(C(F)(F)F)C(NC(c2ncnn2C(C)C)=O)C1 c1(C(N2CC(C)C(C)(C(=O)NC(C)CS(C)(=O)=O)C2)=O)cc2cccnc2[nH]1 Cn1oc(C(=O)NCC(CO)NC(c2ccc(CSCC(F)(F)F)o2)=O)cc1=O c1(CCC(=O)NC(CC(C)NC(c2c(C)nn[nH]2)=O)C)c(F)cccc1Cl N1(C(C(CC(F)F)NC(c2cncnc2)=O)=O)CC23CCC2(COC3)C1 c1(C(=O)NC2CCN(C(c3ccc(Br)c(Br)c3)=O)CC2)cnc2ccoc2c1 CC(C)C(C(=O)NC1CCC(NC(=O)CC(C)(F)F)C1)c1ccccc1 c12cc(S(N)(=O)=O)cnc1N2.C1(C(=O)O)COCCOC1 C1(c2n(CC(=C)C)nnn2)(NCC(C(=O)OC(C)(C)C)C2CC2)CCC(=O)NC1 C1(CCC(N2CC(=C)C2)=O)CCN(C(c2ccncc2)=O)CC1 C1(NC(=O)OC(C)(C)C)CCCC(C(=O)N(C2CCCC2(C)C)CCO)CC1 CCC(C)CC(=O)N(CCCn1cc(CCN(C)CCOCCO)nn1)C C=CC(CC)CC(=O)NCC1CN(C(=O)C=C=C(C)C)CC1CCC c1(C(=O)NCC2CCCN(C(C=CSC)=O)C2)cc(OC(F)F)cc(Cl)c1 C(CCCCC(=O)NCCc1ccc(F)nc1)NC(C1(CC)CC(C)(C)C1)=O C1(C)(NC(C2(NC(c3n(COC)ncc3)=O)CC2C)=O)CCCC1C N1(C(C(C)(F)F)=O)CCC(CO)(CNC(=O)CCC2CCCCC2)CC1 c1(C(=O)NCC(CCOC)NC(C2CC(=O)N2)=O)ccc(C2CCC(=O)N2)cc1 CC1(C)C(NC(=O)CC2(NC(c3ccncc3C3CC3)=O)CC2)CC1(F)F c1(OC)c[nH]c(C(=O)NC(CNC(=O)C(=O)NC(C)C)CC(F)(F)F)cc1=O C=CCC(CC=C)C(=O)NCCC1CCN(C(c2cc(Br)co2)=O)C(C)C1 Cc1ccc(=O)n(CC(=O)N(CC(C)NC(c2scc(C)c2Br)=O)C)c1 N1(C(CCCCOC)=O)CC2ON=C(CNC(c3cn4c(n3)CCC4)=O)C2C1 C1(CC(=O)NC(C2CCOC2)C#C)COCCN1C(C1CC(CN(C)C)C1)=O c1(C(N2C(C(=O)NC(CCC)C(=O)NC)C(CC)CC2)=O)cnc(N)c(Cl)c1 C(CC(C)C)(C(=O)N1CCCC1CF)N(C(CN(CC)CC1CC1)=O)C C1(C(N2C(CCCNC(CCn3ccc(C)n3)=O)CCC2)=O)C2CC3C(C2=O)C13 c1(C(N(CCNC(C2(CC#C)CCCCC2)=O)C(C)C)=O)ccc([N+](=O)[O-])s1 C1(C(=O)NCC2(OC)CN(C(c3n(CC)ncc3)=O)C2)OCCC1(C)C C(C(COC)CC(=O)NCC(CO)NC(c1ccc(C(=O)N(C)C)cn1)=O)OC N1(C(CC=CCC)=O)CCN(C(c2cccs2)=O)C2CC12 C(C(CC(=O)NN1CCC1C(C)(C)C)CO)NC(=O)C=Cc1cscn1 C1(CNC(C2(NC(C3CCS(=O)(=O)C3)=O)CCSC2)=O)CCC2(CC2)C1 c1(C(=O)NCCC2(OC)CCN(C(c3ccoc3)=O)C2)cn2c(n1)CCC(C)C2 CS(=O)(=O)CC(F)(F)CC(=O)NCCNC(c1ccc(O)cc1OC(F)(F)F)=O CCC(CC(=O)NCC1CC(C)(O)C1)N(C)C(C1CCN1C(C)(C)C)=O C1(C(N2CC(O)(CCNC(C3(CC)CCNC3=O)=O)C2)=O)CS(=O)(=O)CC(=O)N1 CSC1=C(C(=O)N(C)CCN(C(=O)C(N2C(=O)CCC2=O)C)C)CCCC1 N1(C(Cc2cccc(SCC)c2)=O)CC(NC(c2cocn2)=O)CC12CCOC2 N1(C(C(=O)N(C(C)C)CCN(C)C(c2n[nH]cc2Br)=O)C)CCCC(O)C1 C(=O)(CC1COc2cc(O)ccc21)N1CC(CNC(c2c(OC)cc(C)s2)=O)C1 CCN=c1ccc(C(N2CC(NC(C3CC3CCOC)=O)CC23CCC3)=O)c[nH]1 c1(CC)ccc(C(N2CCC(O)(C(C)NC(=O)Cc3ccccc3)C2)=O)nc1 Cc1cc(C(=O)NCC2CN(C(=O)C=CCN(C)C)C3(CCC3)C2)cc(N)c1Cl C(C(=O)N(C(C)CC(=O)NCCCN(C)C)C)(C(C)C)SC C12(NC(=O)CCOc3cccc(F)c3)CCCC1CN(C(C1(CF)CCC1)=O)C2 c1(CC)c(C(=O)NC2CCC(NC(=O)C=CSC)CC2)nnn1-c1ccccc1 N1(C(C(C)c2cncs2)=O)CC2(CC(NC(=O)CCC(C)(C)C)CO2)C1 C1(C(=O)O)(CN)CCCCC1.C12CCCN1C(=O)C(=O)N(CC#C)C2 C1(C(=O)Nc2c(C)occc2=O)CC2CN(C(=O)OC(C)(C)C)CC2C1 C(C(C)(C)CC(C)O)NC(c1n(CC(=C)C)nnn1)C1(CF)CC1 c1(CC(N2CC3(C2)CN(C(c2ccc(O)nn2)=O)C3)=O)cc(Br)ccc1F c1(C(=O)NC2CN(C(c3ccc4nonc4c3)=O)CC2F)cnc2snnc2c1 C1(NC(NC(CC)C)=NCC=CCl)CCn2c(C)cnc2C1 C1(C(=O)NC(C2CN(C(c3ccc(C4(C#N)CC4)cc3)=O)C2)C)C2CCC(F)(F)C12 c1(OC)cccc2c(-c3cc(C(=O)O)ccc3C)cccc12 C(=O)(C(F)(F)C(F)(F)C(F)F)N(CC(C)CNC(c1nnn(C)n1)=O)C c1(C(=O)NCC2N(C(c3cc(C)on3)=O)CC=C2)ncnc2cc[nH]c12 C1(NC(c2n(CC)c(O)nc2)=O)(CO)CCCN(C(=O)CN2CSCC2=O)C1 N1(C(C(C2CCCO2)NC(Cc2cc(C)n(C)n2)=O)=O)CCC(O)CC(C)(C)C1 c1(OC)ncc(C(=O)NC(C(=O)N(C)CCn2cncn2)c2ccoc2)s1 n1(CCN(C)C(=O)OC(C)(C)C)cc(C(C(=O)Nc2ccsc2)N(C)C)nn1 c1(NC(C2COCCN2Cc2ncc3ccccn23)=O)cc(Br)cnc1[N+](=O)[O-] N1(C(C2N(C(C)=O)CCC2)=O)CCC(CNC(=O)CCc2ccco2)C(C)C1 N1(C(CC2C(C)CC2)=O)CCC2(CCCN2C(c2cc3nc(=O)ccn3[nH]2)=O)C1 C1(CN(C(=O)CCc2ccc(N)nc2)C)CCCN(C(=O)CC2CC(F)C2)C1 CC1CN(C(c2cnn(-c3ccccc3)c2Br)=O)CCN1C(=O)C(C)(C)O c1(-n2ccc(C(=O)Nc3c(C(=O)NC)nc[nH]3)n2)ccc(OCCOC)cc1 c1(C(=O)NC)ccc(C)c(N(C)C(=O)OC(C)(C)C)c1.C1(C)CCN1 C1(NC(c2c(C)cn(C)n2)=O)CCN(C(c2cnc(C)n2C)=O)C1(C)C N1(Cc2c(OC)cc(OC)cc2C(=O)O)CCCC1C1OCCO1 N1(C(C2C(C)(C)CCN2C(C2CCS2(=O)=O)=O)=O)CCc2ccccc2C1 CC(C)(C)C(C(=O)NC1CN(C(c2cc(F)cnc2O)=O)CC1O)C1CCCC1 C1(CC(=O)NC2CC(NC(c3ccc(C)cc3)=O)C2)CC(C)(C)CCO1 CN1CC(NC(=O)NCCOC2CN(C(=O)OC(C)(C)C)C2)C(C)(C)C1 C1(NC(c2c(C)cccc2O)=O)CN(C(=O)CC2=CCOCC2)CC1C1CC1 N1(C(C2N(C(=O)Cc3ccccc3F)C3C(C2)C3)=O)CCC2(CCOC2)C1 C(=O)(CC(C)(C)CC(=O)N1CCC(NC(C2(C)CC(C(F)(F)F)C2)=O)C1)OC C1(CNC(c2[nH]cc(C)c2)=O)CCN(C(=O)C(C)c2ccsn2)C(C)C1 CCCC(CCC)CC(=O)N1CCC(CF)(NC(=O)CC2CCC(=O)NC2=O)C1 C(=O)(CC(C(F)F)NC(=O)C(C)OC(C)=O)N(CC(COC)C)C N1(CC(=O)NC(C)CCCOCC)CCCCC1CCCC c1(C(=O)NCCCN(C(c2ccc(C)c(O)c2)=O)C)ccc(F)c2cccnc12 C1(C(N(C(C)C(C)(C)O)C)=O)(NC(c2cn(C)cn2)=O)CC(F)(F)C1 N1(C(COC)=O)CC2(CCCCN2C(c2ccc3c(C)[nH]nc3c2)=O)C1 c1(C(N(CC(CC)NC(C2(CO)CCCO2)=O)CC)=O)ccncc1NCC c1(CCOC)n[nH]c(=NC(=O)NCC2(CSC)CC2c2ccccc2)s1 N1(C(C2CC(C)(NC(=O)CC3(O)CCOCC3)C2)=O)CC(S(N)(=O)=O)C1 C1(NC(c2cnc(OC)nc2)=O)CS(=O)(=O)CC1NC(C1SCCCS1)=O c1(N2CCN(Cc3cc(SC)c(Br)cc3)CC2)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] C1(C(=O)NC(c2ccc(C)s2)C)CC2CCC1N2C(c1ncsc1C)=O C1(C2(O)CCOCC2)(NC(c2n(C(C(=O)OC)CC(C)C)nnn2)C(C)C)CC1 N1(C(C2(C)CCC(=O)C2)=O)CCCCC(CNC(c2n[nH]c3c2CCC3)=O)C1 c1(OC)ncc(C(=O)NC2CC(CCNC(c3nccc(C(F)F)n3)=O)C2)cn1 CC(=O)CCCC(=O)NC1(CO)CCN(C(C23CC(CF)(CO2)C3)=O)C1 c1(C(=O)OC)c(C)sc(C(N2CC3CC2CN3CCF)C(=O)NC(C)C)c1Cl CCCC(CC)C(=O)NC(CO)CCCNC(C1CCCS1)=O c1(CC)[nH]nc(C(=O)NCC(O)CN(C(=O)C=Cc2cnc[nH]2)C)c1Cl n1(CC(=O)NC(CC)CN(C(=O)C(COC)OC)CC)cccc(C)c1=O N1(C(CCc2n(C)ncc2)=O)CCC2CN(C(=O)CN3CCCC3=O)CCC2C1 CC(C)(CC(=O)NCC(C)(C)CNC(c1cccc(-c2cc[nH]n2)c1)=O)C1CC1 c1(C(N2CCC(CCC(=O)NCCSCCCO)C2)=O)ccc2cc[nH]c2c1 C(N1CCC2(CCCCO2)C1)c1n(CCCCC)nc(-c2cnn(CCO)c2)n1 CC1CCN(C(c2cc(C3CCC3)nn2C)=O)CC1CNC(C1(Cl)CCC1)=O S(=O)(=O)(c1cn(C)nc1C)C(=O)NC1(c2c(OC)cccc2)CCC1 C1(NC(c2cncc(OC)c2)=O)CCCC(NC(c2ccnc(O)c2)=O)CC1 CC1(NC(c2cnc(S)[nH]2)=O)CC(NC(=O)CSCC(N2CCCC2)C)C1 Cc1cn(C)cc1C(=O)N(C)CCN(C)C(C1(CO)CC1(F)F)=O N(C(=NC1CCCC1)NC1CC1C1(Cl)CCCC1)CC(C)C C(C1(C)CCOCC1)=CC(=O)NCC(C)NC(c1ccc(CO)o1)=O C(N=c1cccc(S(=O)(=O)NCCC2CC3CC3C2)[nH]1)C1(CC(C)(C)C)CCC1 CC(C)(C)CCNC(=O)CC1CCC(=O)N1.N1(CCC(=O)NCC#N)CCCCC1 c1(C(C(=O)NCC=CCNC(=O)CCn2cncn2)O)ccccc1Br c1(NC(C2OCCN(C(Cn3ccc(C)cc3=O)=O)C2)=O)ccccc1N=[N+]=[N-] CC#CCCCC(=O)NC(C)C(C)(C)C(=O)NC(c1ncn(C)n1)C c1(C(=O)NC2C3N(C(C(C)(C)N(C)C)=O)CC(CC3)C2)c[nH]c(=O)c2ccnn12 c1(C(=O)NCC(CC=C)NC(=O)CN2CC(C)(OC)C2)c(C)ccnc1O C1(NC(C(C)(C)OC(C)=O)=O)CCCCC1N(C(=O)CNC(=O)C1CC1)C CN1CCC(C)(C(N2CC(NC(=O)Cc3ccon3)C(n3ccnn3)C2)=O)C1 N1(C(C2CC(OC)C2)=O)CCCC2(NC(=O)CCCc3nc(C)no3)CCCC12 c1(CNCC(C(=O)NC)(C)C)ccc2oc(Cl)cc2c1 C=CCC(CC)C(=O)NC(C)CNC(=O)CC1NC(=O)NC1=O C1(NC(c2cnc(OC)nc2)=O)CC2CC(C1)N(C(c1sncc1C)=O)C2 C1(CCN(C(c2nc(COC)oc2)=O)C)CCN(C(C2(SC)CCC2)=O)CC1 c1(CN(C)C(C2COCCN2C(=O)CSC(F)F)=O)ccc(=O)n(C)c1 N1(C(c2c(=NCC=C)[nH]ccn2)=O)CCC2(CCCCN(C(=O)C=CC)C2)C1 c1(C(N2CCC(F)(C(N(CC(CSC)O)C)=O)C2)=O)c[nH]c(C#N)c1C C1(CC)(NC(=O)CCOCCN(C)C)CCN(C(c2cc(Br)c(C)o2)=O)C1 N1(C(C2N(CC)CC2)=O)CC2CCC1CN2C(=O)Cn1cnnc1O CC1CC(C)(C(=O)NC2CC(CNC(=O)Cc3cccc(F)c3Cl)C2)CC(C)O1 CCCCC(=O)NC(C1CCN(C(c2cscc2Cl)=O)C1)C N1(CC(N2CC(C(=O)NCCC3CCC(C)O3)(SC)C2)=O)CCC(O)CC1 C(=O)(C1CCOc2ccc(Cl)cc21)N1CC(C)N(C(c2csnc2Cl)=O)CC1 c1(C(N2CC(OC)(CNC(C3CCCOC3)=O)C2)=O)cc(O)cc(N)c1C N1(C(COCC#C)=O)CCN(C(c2cccnc2)=O)CC(C)(F)C1 Cc1cc(C(=O)N(C)CC2CN(C(=O)C(c3ccnn3C)C)CCO2)ccc1Cl Cc1ncnc(C)c1C(N1CCC(CN(C)C(C2(C)CC=CCO2)=O)C1)=O Cc1cc(C(=O)NCCN(C(=O)C(C)CC2CC2)C2CC2)ccc1-n1cnnn1 N1(C(C2C(CCC#C)C2)=O)CCC2(CCCCN(C(C3CCC3)=O)C2)C1 S(=O)(=O)(c1ccccc1F)NC(C)C(N1CCC(N)C(C)(C)C1)=O c1(C(=O)OC)cc2cc(C(=O)NCCN(C(=O)C(C)CS(C)=O)C)sc2s1 c1(C(=O)NC(C(C)NC(C(F)=CCC)=O)C)cnc(C2CC2)[nH]c1=N C1(CC=C)(NC(=O)CC=CC)CCN(C(c2cc(C(F)(F)F)[nH]c2C)=O)C1 N1(C(C)C)CCCC(NC(=O)CC(C)(C)N(C)C(C2CC2C(C)(F)F)=O)C1 C(Cc1ccccc1)(CC(=O)O)C(=O)NCc1cc(C)on1 c1(C(=O)NC23N(C2)C3)cnn(C(C)CC)c1CC.C(C=O)SCC.C#CCSCC c1(CCOC2CN(C(CCN(C(CC)CC)C)=O)C2)snnc1CCOC c1(C(=O)NCCC2CCC(NC(=O)CCc3ccco3)C2)occ2c1CCCC2 c1(C(C)=O)cc(C(=O)NCc2ccccc2CNC(=O)CNC(N)=O)ccc1F c1(C(N2C(CO)CC(NC(C(CC)(C)O)=O)C2)=O)cc(C#N)cc2ccccc12 N1(C(c2c(NC)cnnc2)=O)CCC=C(C(=O)N2CC(CO)C2)C1 C1(CC)C(NC(c2ocnc2CC)=O)CCCN1C(C1CCCC1OC)=O C(C(=O)NCC1(C2CCCN2C(=O)CCOC2CC2)CC1)(C(C)(C)C)N(C)C N1(C(C(CCC)NC(c2cncc(OC)c2)=O)=O)CCOC2(CC2)C1 N1(C(COC(CC)C)=O)CCC2(CC1)CN(C(c1cncs1)=O)C2C(C)C C1(C(=O)NC2CC(n3cc(Cn4ncc(C#N)c4)nn3)C2)OC2CCC1CC2 CC1(C)CC(CNC(c2ccc[nH]2)=O)CN(C(=O)C(c2ccc(F)c(F)c2)=O)C1 C1(C(N(CCCCC(=O)NCCCN2CCC(O)C2)C)=O)CC2(C1)CC2(F)F C1(CC(=O)NC(CNC(c2c(C)cco2)=O)C)(COC(C)(C)C)CCCCC1 n1(CC(N2CCC(CN(C(C(C3CC3)OC)=O)C)CC2)=O)nnc2c1CCCC2 C1(O)(CC(=O)NC(C(=O)NCc2ccccc2)C2(C)CC2)CCCOC1 N1(C(CC(CCCC)O)=O)CCCC2(CCCN2C(=O)CC(Cl)Cl)C1 n12cc(cn1)C(=O)NCC2.N1(C(CC2CC(=C)C2)=O)CCC(N2CC(O)C2)C1 N1(C(C2(CCC)CC2)=O)CC(NC(c2cnc(C)c(C#N)c2)=O)C(C2CC2)C1 N1(C(CNC(CC)=O)=O)CC2CCCC2(NC(c2cc3cccnn3c2)=O)C1 C(C(C)(C)CN=[N+]=[N-])N(C(CC1CCCN(C(C)=O)C1)=O)C1(C(=O)NC2CCC2)CC1 CC1CCOC(C(N2CCOC(CCNC(=O)C(F)(F)c3ccccn3)C2)=O)C1 CC1CCC(CNC(C2CC=CC2)=O)CN1C(=O)CCc1ccccc1Cl C1(O)(CNC(C(c2ccoc2)NC(c2c(COC)ccs2)=O)=O)CCN(C)CC1 c1(CCC(=O)N(C(C=C)C)CC)ccccc1-n1cc(CCCN)nn1 C(=O)(CN=S(C)(C)=O)NCCCCC1(NC(C(C)C(=O)N2CCOCC2)=O)CC1 c1(CC)cnc(C(=O)NC2CCN(C(=O)CCc3nncs3)C2)nc1 Cc1ccc2c(n1)CN(C(=O)C(O)C1CN(C(c3coc(N(C)C)n3)=O)C1)C2 c1(OCC)ccc(NC(=O)NCc2[nH]c(C)nc2C)cc1OC [N-]=[N+]=NCCNC(=O)C(C1CCCC1)NC(=O)CCc1cnoc1 C1(NC(c2cc(OCC)n[nH]2)=O)CCCC(NC(c2cnn(C(C)C)c2)=O)CC1 c1(C(=O)NC2CC(NC(c3c(C)csc3)=O)CC2O)cn2ccnc2cn1 C12(C3CC3)CCN(C1)C(=O)C(=O)N2.c1(OC)c(OC)cccc1C(N)=O N1(C(C(C)SC)=O)CCN(C(C2(c3cccc(F)c3F)CCCC2)=O)CC1CO C12(C(=O)NC(C)CC3CN(C(c4ccc(N)c(N)n4)=O)C3)C3C4C1C1C2C3C41C N1(C(c2ccc(C)c(C)c2)C(=O)Nc2ccccc2)CCCCC(S(C)(=O)=O)C1 c1(C(N2C(C)(C(=O)NCC3CCN(C)CC3)CCC2)=O)ccc(C#N)nc1 C(C(C)(C)CC(=O)NC1CCN(CCNC(=O)C(CSC)OC)CC1)OC c1(C(N2C(CNC(c3n(C=C)ncc3)=O)CCCC2)=O)c(Cl)cc(Cl)nc1N C(=O)(CC(C)C1CC1)N(CC(C)NC(c1[nH]ccc1-c1ccccc1)=O)C Fc1ccc(Br)c(CNC(c2nnnn2C2CCOCC2)CCc2cccs2)c1 C(=O)(C1CCCc2scnc21)N(CCNC(=O)CN(C)C(N)=O)CC N1(C(C(CC)(C)O)=O)CC2OCCN(C(=O)C(C)Oc3ccc(C)cc3)C2C1 Cc1nc(CN2CCC(NC(=O)Cc3cccnc3)C2)ccc1Br C(=O)(CC(C)CC(=O)N1CCCC(N(C)C(C2CN(C3CCC3)C2)=O)C1)OC N1(C(c2cnn(CC)c2)C(=O)NCC=C)CC(C)c2ccc(OCC)cc21 C(=O)(C1CCc2nccn21)N1CC(C)N(C(C2CCC(=O)NC2)=O)C(C)C1 N1(C(c2n(CC)ccn2)=O)CCCC(C(=O)NCCC(=O)NO)C1C C12(NC(=O)CNC(=O)C3CC3)CCC(CNC(c3cc([N+](=O)[O-])c[nH]3)=O)(C1)OC2 C1(NC(C(CSC)OC)=O)CCN(C(=O)CCCC2CCC2)CC1C(C)C c1(CC(CC)NC(c2ccccc2N(C)C)=O)cccc(Br)c1 c1(CC(N2CCC(NC(CCC(=C)Br)=O)C23CC3)=O)cn(C)c2ccccc12 O=C(N=c1cc(C2CCCC2)[nH][nH]1)C(=O)N1CCN(c2nnc(O)s2)CC1 C(=O)(C1=NOC(C)(C)C1)NC(c1cn(C)nn1)C(N1CC(F)(C(=O)OC)C1)=O C(=O)(C1=CC2(CCOC2)C1)N1C(CC(=O)Nc2c(OC)cc(O)cc2)CCC1 C1(C(=O)NCCOCCC=C)COCCC1NC(=O)Cc1csc(C)c1 N1(C(C2C(=C)CC2)=O)CC2CN(C(c3cc(C)ccc3Br)=O)CC2C1 C1(CC(=O)O)(NC(C2CCN(Cc3cccc(OC)c3)CC2)=O)CCN(C)CC1 c1(C(=O)NCC(CNC(c2n(CC)nnc2)=O)O)coc2c1N(C)C(=O)CCC2 c1(OC)nc(C(=O)NC(C)(CNC(c2ccn(CCF)n2)=O)CO)cc(O)n1 c1(OCCN(C)C)ccc(C(=O)N(CCN(C)C)Cc2ccc(O)cc2)cc1 c1(CN(C(CC(=O)OC)=O)CCCNC(c2n[nH]cc2F)=O)ccc(Cl)cc1 C=C1CC2CC1CN2C(C1CCC(C)N1C(=O)CSC1CC1)=O C1(CCC)CN(C(=O)C(C)Cn2ccnc2)CC1NC(=O)Cc1ccnnc1 C12(CNC(CCOCCC)=O)CCC(C1)N(C(c1cc(=O)n(C)cn1)=O)C2 S(=O)(=O)(c1ccc(N2CC(C)CC(O)C2)nc1)N1CCC(C2C(CCC)C2)CC1 c1(C(=O)NC2CC(C(=O)NC(CC)COC3CC3)C2)ccc(OCC)cn1 c1(C(=O)NCCN(C(=O)CC2CCC(O)C2)C)ccc(NS(C)(=O)=O)cc1O C1(CC)CCCN(C(=O)Cc2ccnn2C)C1CNC(=O)CCNC(N)=O C(CC(O)C(=O)N(CCCNC(c1nocc1C(C)(C)C)=O)C(C)C)SC C1(COC)(NCCNC(C)=O)CCCN(C(C2CCOC2C)=O)C1 C12(CNC(c3c(C(C)C)con3)=O)CCC(CN(C(c3ncncc3N)=O)C1)C2 C#CCC(CC(F)F)C(=O)N1CCC(C)N(C(=O)Cn2ccnc2C)CC1 C1(CCC(=O)N(C)Cc2cccnc2)CCCCN(C(C2(O)CCSCC2)=O)C1 C1(C(N2C(CCNC(C(COC)O)=O)CSCC2)=O)CN2CCCN1CC2 c1(C(CCOC)NC(C2CCOCC2)CC)ccc(OC)cc1C C#Cc1cncc(C(=O)NC2CCN(C(=O)Cc3ccc(F)cn3)C2C(C)C)c1 C(=O)(C1CCCn2ccnc21)NCC(C)(CO)NC(=O)Cc1ccsc1 Cc1cnc(C(=O)N(C(C)CNC(c2ccc(OC(F)F)cc2)=O)C)c(F)c1 C1(C(N(C(C=C)C2CC2)C)=O)CCN(C(=O)C#CC2(C)COC2)C1(C)C CC(C)CC(C)(C)C(=O)NC1CC(NC(=O)CCC(C)N(C)C)C(O)C1 C(C(=O)NCC1CCCN1C(=O)C(C)N(C)C)(C(C)C)n1ncc(C)c1 C1(C(N(CCOCCNC(c2c(OC)cccn2)=O)C)=O)CCn2cnnc2C1 C1(CNC(C(=O)NCC#C)=O)CCN(C(=O)CSC2CC2)CC1 C12CCCCN1C(=O)CCn1cc2nn1.C1(Cc2cc(C)no2)CC(O)(C#N)C1 C1(F)(CNC(C=C(C)Cl)=O)CCCN(C(c2csc(CC(F)F)n2)=O)C1 c1(OC)cc(C=CCN(C)Cc2ccsc2)ccc1O C1(NC(c2c(C)oc(S(=O)(=O)N(C)C)c2)=O)CC12CCc1ccccc12 OCCN(C(CO)c1ccccc1)N1CCCC(O)(CO)C1 C1(C(=O)NC(C#C)CCC)COCCN(C(C2CCN(C)CC2)=O)C1 N1(C(c2c(C)c(F)ccc2)=O)CCCN(C(=O)C(C)P(C)(C)=O)CC1C(C)C C1(C(C)C)(C(N2CCCC2)=O)CCN(C(c2csc(F)c2)=O)C1.C1(C=O)CC(C)(C)C1 N1(C(c2c(CCC)n[nH]c2)=O)CCC(NC(=O)C(O)Cc2cn(C)cn2)C1(C)C C1(CNC(c2cc(C(C)=O)sc2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC1 c1(COC)cc(C(=O)NC(C)(CSC)CO)n[nH]1.C1(C)C=CC(=O)N1 C(C(=O)NCC1(NC(C2CC3(CSC3)C2)=O)CC1)(C(C)C)OCC C(CC(C)C)(C(=O)NCC(CO)NC(c1cnc(C)nc1C1CC1)=O)OC N1(c2ccc(C#N)o2)CCc2nc(C(=O)Nc3ccc(F)c(O)c3)cn2CC1 c1(NC(C(CCC)C)C)ccc2[nH]ccc2n1 Nc1ccc(C(=O)NC2CN(C(C3CC4OC3C3CC43)=O)CC23CC3)cc1F N1(C(C2CCOC3(CCC3)C2)=O)CC2(CCN(C(=O)C(F)n3cccn3)CC2)C1 CC1CCC(N(C(=O)CCc2cccn2C)C(=O)COC(=O)CO)C1 c1(C(=O)NCC(C2CCC2)NC(C2(O)CCCCC2)=O)cccc(F)c1[N+](=O)[O-] c1(CC(N2CCC(C(C(=O)N(CC(C)OC)C(C)C)F)C2)=O)ccc(C#N)cc1 c1(CC)ccc(C(=O)NC2CN(C(C3CC(=O)N(C)C3)=O)C(C)(C)C2)c(N)c1 N1(CC(=O)O)C(=O)CN(CC2CCCC(C3CC3)O2)CC1=O N1(C(C(CO)OC)=O)CC2(CCCC2)C1C(=O)NCCC1CCOC1=O N1(C(c2ccc(COC)o2)=O)CC2CCN(C(=O)CCC3CC3(F)F)C2C1 c1(C(N2CC(CCNC(CC(CC)C)=O)(OC)C2)=O)cn(C)c2c(Cl)cccc12 Cn1nc(C(=O)NC2CC(CCC(=O)NC3CCC3O)C2)cc1C#N c1(C(N(C2CN(C(=O)C#CC(C)(C)C)C2)C)=O)cc(Br)c2occc2c1 N1(C(C(c2nc(C)sc2)=O)=O)CC2=C(C1)CN(C(=O)CC1CCCC(C)O1)C2 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1C(CNC(COCCN(C)C)=O)C1 S(=O)(=O)(c1ccc2[nH]c(=NC3CCC(C4CC4)C3)sc2c1)NCCC(CC)C(C)C CC1CC(C(=O)NCC2(C)NC(=O)NC2=O)CCN1C(c1ccn(C)c1)=O c1(C(N2CCCC2CC(F)(F)F)C(=O)NC(CC)(C)C)ccn(C2CC2)c1 N1(C(c2cc(CNC(C(c3ccn(C)c3)C)=O)no2)=O)CCN2CCC1C2 C1(C(=O)NCCC(CCC)O)CC2(CCC2)CN1C(c1cccn2cncc12)=O c1(SC)cnc(NCc2ncccc2-c2cncc(CN3CCOCC3)c2)nc1 CCCC(O)C(=O)N1CCC(C(N2CCSC(CC)C2)=O)(CO)C1 N1(C(NNC(C2S(=NC)(=O)CCNC2)=O)=O)c2ccccc2Sc2ccccc21 C1(N(C(CSC)=O)CCO)CCCN(C(=O)C(C)=C2CC2)C1 c1(C(N2CCC(CCNC(CNS(NC)(=O)=O)=O)C2)=O)ncnc(O)c1Cl c1(C(N(CCCNC(=O)CC2CCCO2)C(C)C)=O)noc2c1CC(F)(F)CC2 c1(N2CC(CCOC)(OC)C2)nc(C)ccc1C(=O)OC.c1(C(=O)NC)cnsn1 C1(CNC(C(n2ncc(C)c2)C)=O)CN(C(=O)COC2CCCCCC2)CCO1 N1(C(C(c2ccc(F)cc2)(C)C)=O)CCC2OCC(=O)NC2C1 c1(NC(C2(CC)CCN(C(=O)CC3(O)CCC3)CC2)=O)cccc2c1OCO2 C1(N(C(C(c2cccc(F)c2)C)=O)C)CCC2CN(C(C3CC(F)C3)=O)CC12 C1(NC(=O)COCCF)CCC12CCN(C(=O)Cc1ccc3c(c1)COC3)CC2 N1(C(CC(C)N(C)C)=O)CCCC2CN(C(=O)CC3CC4(CC4)CO3)CC12 c1(C(=O)NC(CC)CN(C(=O)C(N2CCOCC2)C)CC)cc(C)n(C)c1 N1(C(C(c2ccccc2Cl)C)=O)CCN(CCOc2ccc(CO)cc2)CC1 C(=O)(CCC(C)(C)C#N)N1CCC(NC(c2ncc(OC)nc2)=O)(CF)C1 N1(C(c2cc(C)oc2C)=O)CCC(NC(c2cc3n(n2)CCCN3)=O)C(C)C1 C1(C(=O)OC)CC2CCC(C1)N2C(c1cc(CO)co1)=O.C12CC(C1)NC(=O)C2 N1(C(c2c(C)nc(C(C)C)o2)=O)CC(C)N(C(=O)CSCC(F)(F)F)CC1C C1(C)(C(C(N2C(C(C)NC(=O)CC3(c4ccccc4)CC3)CCC2)=O)F)CCOCC1 C1(NC(CCCOCCOCC)=O)CCN(CCc2ccc(Cl)c(Cl)c2)CC1C N1(C(C(CC)n2nccc2C)=O)CC(OC)CC1CNC(c1ccc(C#N)o1)=O CN1CCc2[nH]nc(C(=O)NC3CC(NC(c4c(N)cc(Cl)cc4Cl)=O)C3)c2C1 N1(C(C(CC)CC)=O)CCOCCC1C(=O)N(CCCF)C Cc1cc(C(=O)NC(CNC(=O)CC2CCC3CC23)C2CC2)cc(N)c1O c1(OC)c(C(=O)NC)csc1C.C1(CC(C)C2CCC2)CCN(C(=O)COC)CC1 C(=O)(C(C)(C)C(C)(F)F)N1CCCC(F)(CNC(C2CC(C)NC(=O)C2)=O)C1 c1(C(C(=O)NC2C(CC)N(C(=O)CCC(F)F)CC2)C)ccc2c(c1)OCCO2 c1(C(N2C(CN(C(CC3(C=C)CC3)=O)C)COCC2)=O)cncc([N+](=O)[O-])c1 CC1(NC(=O)CC2CC(F)C2)CCC(NC(c2cn(CC3CC3)nn2)=O)CC1 CN=C(NCC1CC1c1ccsc1)NCc1nc(N(S(C)(=O)=O)C)no1 c1(C)cc(C(=O)C(C)=O)cc(Cl)c1OC.N1(C(COC)(C)C)CCN(C=O)CC1 C(=O)(C1c2cc(Br)ccc2CCN1C(=O)COc1ccc(CO)cc1)OC c1(C(=O)NCCOCCNC(C(=O)N(C)C)=O)ccc(S(C)(=O)=O)[nH]1 C(C1OCCc2sc(I)cc21)NC(=O)NC(C(F)(F)CO)C1CC1 N1(C(c2nc(CC)oc2)=O)CC2CCC1C(NC(C1(F)CCC1)=O)C2 C1(CC(=O)NCC(CC)N(C(=O)CCC2CCOCC2)C)CC(C)(C)C(=O)N1 N1(C(CN2CCC(C)CC2)=O)CCC2(CC1)CC2NC(=O)CN1CCC(C)(C)C1 N1(C(C2CC23CCOC3)C(=O)NCC(C)C)CCC(C2CC2)C1 N1(C(CC(n2ccc(C)n2)C)=O)CCN(C(=O)C=Cc2cccc(Cl)c2)CC1C O(N1CCC(CC(=O)N(CCNC(=O)CC(CC)SC)CCOC)CC1)CC c1(N2CCCC(CNC(C)=O)C2)nc(N2CC3CC2C3)c2c(n1)CSC2 C1(NC(C2CCN(Cc3ccncc3)CC2)=O)CCC2C(CC1)C2(F)F c1(C(=O)NCC2(CO)CCCN(c3nccc(SC)n3)C2)cc(C)cn2ccnc12 c1(C(=O)NCC(C2CCN(C(C(CC)(C)O)=O)CC2)(C)O)occ2c1CCC2 CC#CCC(C(=O)NC(c1ncccn1)C)NC(=O)C(CC)=CCCC CC(CCC(=O)N1CCCC1c1ncc[nH]1)NC(C1CC(=C2CC2)C1)=O C=C(C)CC(C(=O)N(CCCCCCNC(c1cccc(Cl)c1)=O)C)OC Cc1c(C(=O)NCC2(OCC(=O)NCc3nc[nH]n3)CC2)sc2cncn12 N1(C(C(CC)n2cncn2)=O)CCC(C)C1CNC(=O)C(F)=C(C)C1CC1 C(c1ccc2c(c1)COCC2)=CC(c1nc2cc(Cl)ccc2o1)=O N1(C(C(C)C2CCC2)=O)CCN(C(c2cc(-n3[nH]nnc3=S)ccc2F)=O)CC1C c1(C(=O)OCc2cc(C(=O)OCC)ncc2)cc(C)c2c(c1)CCC2 CCC1=C(C(=O)N2CCCC2(C)CNC(C2CC3(CCCC3)CO2)=O)CCCO1 N1(C(CCSCCC)=O)CC2CCOC2(CNC(=O)C(C)(C)CCSC)C1 c1(C(=O)NC(C(=O)NCCC(C)N(CCC)CC)CN(C)C)cnn2c1OCC2 c1(CC)[nH]c(=N)sc1C(N1CC(NC(=O)C=CC(c2ccccc2)=O)CC1C)=O c1(C(N2CCN(C(CNC(C=C(C)Cl)=O)=O)CC2)=O)ccc(C)c(Cl)c1 N1(C(CCC)=O)CCN(C(C2CCCO2)=O)CC1c1ccc(OC)cc1 Cc1ncc(C(=O)NC(C)CCN(C(=O)CC(=O)Nc2nccs2)C)n1C(F)F C12(NC(C3OCCN(C)C3)=O)CCCC1N(C(c1scc3c1CCCC3)=O)CC2 c1(C(=O)NCC2CCN2C(C2CN(CC(F)(F)F)C2)=O)cccc(C2CCC2)c1 C1(CNC(c2occ(C)c2)=O)CC(O)C(O)CC1C(N1CCC1(C)CCO)=O C1(n2ncc(C)c2)CCN(C(=NCCCCc2cccs2)NCC(C)(C)C)C1 CC1CCC(NC(=O)Cc2cnc(C3CC3)[nH]2)CN1C(c1csc(S)n1)=O C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(C)CC1(C)C S(=O)(=O)(c1ccc2c(c1)CNC(=O)O2)N(C1(CC)CC1)Cc1nnc2cnccn12 N1(C(CC(C)N(C)C)=O)CCOCC1CNC(=O)CC1(CSC)CCOCC1 C1(CNC(c2cc(SC)oc2)=O)CC2CCC1N2C(=O)C(C)C1CCCO1 c1(C(=O)NC2(C)CN(C(C(C(CC)C)O)=O)C2)cc2n(n1)C(C)CCC2 N1(C(C(C)C2CCC2)=O)CCCCC1CN(C(=O)Cc1ccc(N)cc1)C c1(C(=O)NC23CC(NC(C4CCC(OC)C4)=O)(C2)C3)c(C)nn2cc[nH]c(=O)c12 n1(CC)cnc2nc(=NCc3ccoc3)[nH]c(N3CCC(C(F)(F)F)(CO)C3)c12 C=CC1CN(C(=O)COCC(F)(F)F)CC1NC(=O)CCCCC1CC1 c1(C(N)=O)ccccc1OCC(=O)NCC=CCNC(C1CC2CC2C1)=O c1(CN(C)Cc2cccn2-c2ccc(OC)cc2)cccc(Br)c1F CC1(C)CCCN(C(c2cocn2)=O)C1CNC(c1cc(O)cc(Br)c1)=O C1(C(=O)NCC=CCNC(c2ccc(OCCOC)nc2)=O)CCCNS1(=O)=O C1(N(C(CC=C=C)=O)CC)CCCN(C(c2cc(C)sc2C)=O)C1 c1(-c2nc(NC(c3cnc(N(C)C)s3)=O)sc2)ccc(CN2CCSCC2)cc1 N1(c2nnc(C)s2)CCC2(CC1)C(NC(=O)C=Cc1nc(C)cs1)CS2(=O)=O N1(C(CCNC(=O)OC(C)(C)C)=O)CC(C(N)=O)(CNC(=O)Cn2ccnn2)C1 c1(C(=O)NCC(C)O)cc2ccccc2cc1CC(=O)NCC(c1ccccc1)C Cc1ccc(S(=O)(=O)N2CCN(C(=O)CN3CCCC(C)CC3)CC2)cc1CN N1(C(=O)Cc2cnoc2)CCC(c2cn(CCCF)nn2)C1 c1(CSC)nnc(N2CCN(CCOC3CCOC3(C)C)CC2)n1CC1CC1 c1(C(N2CCC(CC(N3CC(O)C(F)C3)=O)CC2)=O)cnc2cc(Cl)ccc2c1 c1(COC)ccoc1C(=O)NC1(C(=O)NC(c2cnc[nH]2)C)CC1(C)C C1(NC(CC(=O)NCC#C)=O)CCC(NC(c2nc(C3CC3)n[nH]2)=O)CC1 C1(NC(c2cc(COC)c(NC(C)=O)cc2)=O)CCCCC1S(C)(=O)=O N1(C(=O)C=CCN2CCCC2)CCN(C(C2Cc3ccccc3S2)=O)CC(O)C1 c1(CNC(C2CCCOC2)C)ccc(C2CCCCC2)cc1 N1(C(c2cn(C(C)C)nc2)=O)CCC(O)CC1C(=O)Nc1cc(I)ccc1F C1(NC(C(C)(C)SC)=O)CCCCC1NC(C1(CN(C)C)CCOCC1)=O C1(C(=O)NCC2(NC(=O)C=C[N+](=O)[O-])CC2)CCC2C(CC1)C2(F)F CC(C)C(CNC(=O)CCc1cnc2ccccn12)N=c1[nH]nc(CC#N)s1 C(CC(=O)N1CCC2CC12)(C(C)OC)NC(CCN(CC)OC)=O N1(C(C(CC)N(C(=O)Cc2cccnc2)C)=O)CCCC(N(C)C)CC1 C1(CCNC(C2(C)CNC(=O)C2)=O)CCN(C(c2csnc2Cl)=O)CCC1(F)F C12(CN(C(C3(C(C)=O)CC3)=O)C1)CC(=O)N2C.C(CF)(CF)OC C1(CCC(C)C)CCCN(C(=S)Nc2ccnc(F)c2)C1 C1(CNC(C2(CNC(C3CCCN3C3CC3)=O)CC(=C)C2)=O)(CC)CCCCC1 C(C)(CCC(=O)NC(c1ccc(F)cc1)C)NC(C1C(OCC)CCC1)=O N1(C(C(C)C2(O)CCC2)=O)CC(C(=O)NC2CN(C)CC2C)CC1(C)C N1(C(C2SCCS2)=O)CC2CN(C(C3CC34CCC4)=O)CC(C1)O2 C1(C(N2CC(C(C)NC(c3c(CC)nccc3)=O)C2)=O)CC2(CCO1)CC2 Cc1cc(Cl)c(NC(=O)CN2CCC(N(C(=O)CN(C)C)C)C2)c([N+](=O)[O-])c1 c1(C(=O)OC)ccc(C(=O)N(CC(C)CNC(C2(C)CC2(F)F)=O)C)n1C C1(OC)CN(C)C(C)(C(N2CC(CC(C)NC(=O)Cc3cccc(Cl)c3)C2)=O)C1 N1(C(C=CSC)=O)CCC(C)(NC(=O)COCC2CC2)C1 c1(C(=O)NC2CCN(C(c3c(COC)scc3)=O)C2C)cnn2c1CCCC2 C(=O)(CS(=O)(=O)C(C)C)NCC=CCNC(c1ncnc(C)c1C)=O N1(C(c2c(C)n[nH]c2C)=O)CCN(C(c2ccc(CO)s2)=O)CC2(CC2)C1 C(C(C)(C)CCl)(C(F)(F)F)N(CC(C)(C)C)C(CC)C.N(C)CCN(CC)CC C1(NC(C(CC)=O)=O)CN(C(c2c(F)cccc2Cl)=O)CC12COC2 N12CCC3(CC3C1=O)C2.N1(CC(C)C)CC(C(N2CCCC2CCO)=O)CC1=O N1(C(=O)NCCCc2n(C)ncc2)CCc2c(Cl)ccc(Br)c2C1 C1(n2cc(CC(C=C)O)nn2)CC2CCC1(NC(=O)CN(CC(C)(C)C)C)C2 CCC(O)(CCCc1ccccc1)NS(=O)(=O)CC1(Cl)CC1(F)F C(c1cncn1C)=CC(=O)N(C1CCC(NC(=O)Cc2cnnn2C)C1)C C1(OC)CCC(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(C)C#N)C2CC2)C1 N1(CC(=O)NCC2(OC)CN(C(c3ccc(N)cc3C)=O)C2)CCS(=O)(=O)CC1 c1(SC)ccc(-c2cncc(C(N3CCCC(Br)C3)=O)n2)cc1 c1(C(=O)NCCNC(c2ccc(-c3nnc(C)o3)cc2)=O)c(F)cccc1F c1(CC(=O)NCCN(CCC)C(C2CCC(C)S2)=O)cnccc1Cl C1(C(C)(C)C)C(NC(=O)C(=O)NC2CC2)CCN1C(=O)CC1(C(F)(F)F)CC1 C(C1=CCCN(C)C1)NC(C1C(C)CCN1C(C1OCCC1C)=O)=O N1(C(C(C)C(F)(F)F)=O)CCCCC12CN(C(c1cc3occc3s1)=O)C2 c1(C(N2CCC(NC(C3COCCO3)=O)C2C2CC2)=O)cc2cnccc2[nH]1 C(=O)(CCCCC(N)=O)N(CC(CC)NC(c1ccc(C)c(C)c1F)=O)CC Cc1ccc(C(C)(C)CC(=O)NCCOCCNC(=O)C(C)C2CCC2)cc1 C=C(C)C(CC(=O)NC1CCC(F)(CNC(c2cc(O)n(CC)n2)=O)C1)OCC C1(C2(NC(=O)Cn3nccn3)CC2)CCCN1C(=O)Cc1nccs1 N1(C(c2cc(C)cc(C)c2)=O)CC2(CCCC(CNC(C3CS(=O)(=O)C3)=O)O2)C1 CC1(C)CC(=O)NCC1C(=O)NCC1CN(C(C2CCC(=O)O2)=O)CCC1(F)F N1(C(=O)Cn2ccccc2=O)CC(C2CN(C(C3C=CCCC3)=O)C2)C1 c1(C(N(C(CNC(=O)COCP(C)(C)=O)C2CC2)C)=O)c(F)cc(F)cc1Cl C(C(CC)CC(F)F)N(c1ccsc1)CCCOC C(=O)(C1COc2ccccc21)NCCN(CCCN(C)C)C(c1ccn(C)c1)=O c1(CNC(N2CCC(NC3CC3)C2)=O)cnc2sccn12.C12CN(C1)CC(=O)N2 c1(C(N2CC(CC)(NC(c3cc(C(F)F)[nH]n3)=O)C2)=O)onc2cc(C)ccc12 Cc1oc(C)c(C(=O)NCC(C)C(F)C(=O)NC2CCC2)c1C c1(CC)ccoc1C(=O)NCC(CC)NC(=O)C(=O)Cc1cccs1 C(c1ccc[nH]1)=CC(=O)NC1(CC(=O)NC2CN(C3COC3)C2)CC1 c1(CC(N2CCC(c3cn(N(C(C)=O)C)nn3)C2)=O)cccc2c1OC(C)(C)C2 c1(C(N2CCC2Cn2cc(-c3ccnn3C3CC3)nn2)=O)cscc1Br C12(NC(CC(C=C)(C)O)=O)CCC(CC1)N(C(c1cnn(CC(F)(F)F)n1)=O)C2 c1(CNC(C2C(C(=O)NC3(CC)CCOCC3)C2)=O)ncc(Br)cc1C c1(C(=O)NC2(c3cc(OC)c(Br)cc3)CC2)cc2c(o1)CCCNC2=O CCC(O)C(C)C(=O)NC1(C)CCCN(C(c2cc(C(F)F)ccn2)=O)C1 c1(SCC(=O)NC2CCC(C(=O)NCCNC(C)=O)C2)ccc(O)cc1 Cc1ncc(Cl)cc1C(=O)NC1COCCN(C(=O)CC2CN(C)C2)C1 C1(C(N(C2CCN(C(=O)C(O)P(C)(C)=O)CC2)CC)=O)CCC(=O)N(C2CC2)C1 c1(N2CCC(OCC(C)C)CC2)nccc(=NC2CC(C)SC(C)C2)[nH]1 C(=O)(C(C)(C)C(=O)NCC1CCN(C(=O)Cc2cncc(C)c2)C1)NC N1(C(C=C=C(C)C)=O)CCCCC(NC(c2cnc(C)s2)=O)C1 C1(NC(C2(CC)CC2)=O)CC(CCNC(=O)C(C)OC2CCOC2)C1 C1(CC#C)(C(=O)NC(C)CC(C)NC(=O)CCC2CC2(F)F)CCCCC1 Cc1cc(C(=O)NCC(CO)NC(c2nccn2C)=O)c2cccc(O)c2n1 c1(CC(N2CCC(N(C(=O)CC3CC(OC)C3)CC)CC2)=O)c(F)cncc1Cl CC1CN(C(C2(C3CC3)CCCCC2)=O)CCN1C(c1cc(C(F)(F)F)ns1)=O CCC(O)C(C)(C)C(=O)NCC(C1CC1)NC(c1ccc(F)c(CSC)c1)=O C1(O)(C(C)NC(=O)CN2CC3CC3C2)CCN(C(=O)CC2(C)CCCCC2)C1 Cc1cccc(OCC(=O)NCC2CCCC2NC(=O)C(C)(C)N(C)C)c1 N1(C(CCN(C(C)=O)C)=O)CC(C(=O)Nc2nc(Br)ccc2Cl)CC(F)C1 C1(OCC)CCN(C(C2CCOC2CNC(c2c[nH]cc2C)=O)=O)C1 c1(C(=O)NCCN(C(=O)C(Cl)=CCl)CCOC)cc2c(cc1N)CCC2 N1(C(c2ccc(F)c(F)c2F)C(=O)NCC(C)C)CCCC2(CCN(C)C2=O)C1 C(=O)(CCC(C)(C)C#N)NC1C(C)CN(C(C2CCN(CC(F)F)CC2)=O)C1 N1(C(C(CC#C)(C)C)=O)CC2CC(NC(=O)CN3CCCC3C)C(C2)C1 C1(C)(C(=O)NCCOCCN(C)C)C=CCN1C(c1ccnc(CO)c1)=O C(CC(=O)NC1CC(NC(=O)C(c2ccc(N(C)C)cc2)C)C1)(C(C)C)OCC N1(C(C(N2C(=O)CCC2=O)C)=O)CCCCC12CC(NC(C13CCC(C1)C3)=O)C2 C(=O)(CCC(C)(C)CO)Nc1cn(CC(N2CCCC(C)C2)=O)nn1 c1(CC(=O)NC2CCC(CNC(CC3CCC(C)CC3)=O)C2)csc2nccn12 c1(C(N2CCC(N(C)C)(CC)C2)C(=O)NC(C)(C)C)cc(Br)ccc1Cl N1(C(C(CC(CC)C)NC(c2sc(C)cc2C)=O)=O)Cc2nncn2C(C)C1 Cc1cnc(C(=O)NCC2CCCCC2NC(c2[nH]cnc2C)=O)nc1 c1(OC)cc(-c2cn(CCCCCC(=O)NC(C)C=C(C)C)nn2)ccc1C C1(NC(CCCC)=O)CCN(C(=O)CN(C)C(=O)C2CC2)CC1C(N)=O c1(CCNC(C(C2CCCC2)NC(C2CC=CCC2)=O)=O)ccncn1 C1(NC(C(OC)OC)=O)CCN(C(c2[nH]nc(C(F)(F)F)c2C(C)C)=O)C1(C)C C1(C#C)(C(N(CC#C)CCOC)=O)CCN(C(=O)C(C(C)C)C(C)C)CC1 N1(C(c2c[nH]nc2CC(C)(C)C)=O)CCN(C(=O)CC2CSC2)C(OC)C1 C12(CN)CCCC1C2(F)F.n1(CC)cc(C(c2nnnn2CCC2CC2)N)nn1 C12COCCN(C1)C2=O.C1(C(=O)NCCOC2CCCCC2)C2CC3C(C2)C13 C1(NC(CNS(CC)(=O)=O)=O)CN(C(c2ncnc(C)c2C)=O)CCC1(C)C c1(C(=O)NC2CN(C(CC3(CC=C)CCOCC3)=O)C(C)C2)ccnc(C)c1O N1(C(CC2(C)CC2)=O)Cc2n[nH]cc2C1C(=O)N1CC(C)(C)C1C1CC1 N1(C(=O)CSC(F)(F)F)CC(NC(c2csc(S)n2)=O)C(C(F)(F)F)C1 C1(C(=O)NC2(CNC(C3CCCN(CCC)C3)=O)CCOC2)CCS(=O)(=O)CC1 C12(C(=O)NCCC3CCN(C(=O)CSCC4CCCO4)CC3)CCCC1C2(F)F CC1(CNC(=O)C(CC2CC2)NC(=O)CC(C2CC2)C2CC2)CC2CC2C1 N1(Cc2ccc(OCC)cc2F)CCC2C1CCCN2c1ccnc(C(C)C)n1 C1(C(=O)Nc2cc(C)c(NC(C3CC(F)(CO)C3)=O)cc2)CSc2ccccc2O1 c1(C(N(CCNc2nccc(C(=O)OC)c2C)CC)=O)nc(OC)ccc1OC C1(C(=O)NC2CCC(NC(C3C(C)(C)NC(=O)C3)=O)CC2)CC2(CCOCC2)C1 c1(C(=O)NCCN(C(CCCCOC)=O)C)cn(C(C)C)c(=O)nc1O c1(C(=O)NC2C(C)N(C(c3ccccc3F)=O)CC2)[nH]c2ccccc2c1Br c1(C(Cc2ccc(Cl)cc2)NC(N(CCOC)C(C)C)=O)ccc(F)cc1Cl Cc1ccccc1C(=O)NC1CCN(C(c2ccc(NS(C)(=O)=O)cc2)=O)C1 C1(C(N2CCCCC(CNC(C3C(=O)NCC3)=O)C2)=O)CC2(CCCC2)CO1 C1(C(C)NC(=O)Nc2nc(C(=O)OCC)c(C)s2)CC(c2ccccc2)=NO1 C1(COC)(NC(=O)CC(C)(C)O)CCCN(C(=O)CN2CCCOC2=O)C1 Cc1cc(C(=O)NC2CCOCC2C(N2CCC(C(C)O)CC2)=O)cnc1C CCC(C)(C)CC(=O)N1CC(O)(C(C)NC(c2csc(C(C)OC)n2)=O)C1 C1(C(=O)Nc2cncc(C)c2C)CC12CCOc1ccc(Cl)cc12 c1(OC)ccc(OCC(=O)N(CC(O)CNC)CCSC)cc1.C1(C)CS(=O)(=O)C1 C(CC(=O)N1CCC(C)(NC(=O)CC2(CS(C)(=O)=O)CC2)C1)(C(F)(F)F)OC c1(CCC)ccccc1CNC(=O)CC1CCN(C(c2c[nH]c(=NC)s2)=O)C1 C1(CNC(CC2C(C)C2)=O)CN(C(c2cc(O)cc(O)c2)=O)CC2(CCC2)O1 C1(C(N2CCCC(N(C(C(=O)NCCOC)=O)CCO)C2)=O)CCC2(CC1)CC2 c1(C(C(=O)NCC2C(NC(C(C)Cc3cnc[nH]3)=O)CC2)O)ccc(Cl)cc1 CCCC(O)C(C(=O)O)NC(c1cc(-c2ccc(C)cc2)no1)=O N1(C(c2ncn(CC)c2)=O)CC(CNC(=O)CCOC)CC12CCOCC2 c1(OC)ncc(C)c(C(=O)NC(C)C(c2ccccc2)NC(=O)CC#N)c1Cl C1(C(N2CCN(C(CC(C)(C)OC)=O)CC2CO)=O)CC(C(C)(C)C)=NO1 Cc1cccc(C(F)(F)C(=O)N(C)CC2CCN(C(C3CCCC34CC4)=O)C2)c1 C12CC(C13CCC3)C(=O)N2.c1(OC)cc(C=CC(=O)Nc2cc(F)ncn2)sn1 N1(C(C(C)(C)O)=O)CCC2(CCCN(C(=O)C3Cc4c(Cl)cccc43)C2)C1 c1(NC(c2cccc(CN3CCCCCC3)c2)=O)ncnc(O)c1F c1(CC)oc(C)cc1C(N1CC(NC(C2CCC(F)C2)=O)C(F)C1)=O c1(NC(C2CCN(Cc3occc3Br)CC2O)=O)nc(Cl)c(Br)cc1I C(=O)(C(C)C(C)(F)F)NCC(CN(C(Cc1c(C)nc(C)s1)=O)C)(C)C CC1CCN(C(C2(c3ccc(Cl)cc3)CCCC2)=O)CC1NC(C1(O)CCC1)=O C1(C(=O)NCCSCCCO)C=CCCN1C(c1ccc[nH]1)=O C1(C(N(C)Cc2ccn(CC)n2)=O)CCOCCN1C(=O)CCn1ccnc1C c1(OC)ccc2c(c1)OCCC2N(C)C(=O)NCc1ccc(C)cc1OC C(=O)(C#CC1(C)CCCO1)N(C1CN(C(c2ccc(OC)c(I)c2)=O)C1)C c1(C(N2C(CCNC(CNS(N(C)C)(=O)=O)=O)CCC2)=O)n[nH]cc1[N+](=O)[O-] CCC(CC(=O)N(CCCNC(C1CC(C(=O)OC(C)C)C1)=O)C)C(C)C CC1CCN(c2nnc(CCc3ccc(Br)cc3)n2C)CCC1(F)F c1(C(=O)NC(C(=O)NCCc2cn(CC)nc2)C2CCCO2)ccc(O)cc1 C(=O)(C1CCCc2nn[nH]c21)NC(C(C)C)(C)CNC(=O)Cc1nn(C)cc1Cl CCCCC(C(=O)OCC1CCC=CCC1)ON=C(C)C c1(N(C2CN(C(CCc3nnc(C)n3C)=O)C2)C)ccc([N+](=O)[O-])cn1 C(=O)(CC(C)N(C(c1nc(C)ns1)C(=O)NC1CCCC1)C)OC C12(NC(C(C)NC(N)=O)=O)CCC(CN(C(=O)COc3ccccc3O)C1)C2 C(=O)(C(C(C(C)C)OCC(=O)OC(C)(C)C)N(C1CCN(C)CC1C)C)NCC CC(C#N)CN(C(=O)CC1(NC(=O)CCC2OCCO2)CCC1)C c1(C(N2CCN(C(C3C=CCCC3)=O)C3CCC23)=O)ccc2n[nH]cc2c1 C1(CNC(c2c(C(N)=O)scc2)=O)CCCCC1N=c1nc(C2CCCC2)[nH]s1 CP(C)(=O)c1cnc(C(N2CCCC(CNC(c3ccc[nH]3)=O)C2)=O)nc1 C1(CCC(=O)NCCNc2sc(C(=O)OC)c(C)n2)OCCOC1(C)C C1(CCC(=O)NCC2C(NC(Cn3ncc(C)c3)=O)CC2)CCCC(=O)N1 c1(CNC(NC2CC(OCC)C2)=NCCc2ccccn2)ccc(C)c(F)c1F N1(C(c2cccc(OC)c2O)=O)CCN(C(C2CC2C(F)F)=O)CCC1C C12(C(N3C(C)CCC(NC(C(C(C)O)C)=O)C3)=O)CCC(C(F)F)(CC1)CC2 N1(C(=O)OC(C)(C)C)CC2CCCC2(C(N)=O)C1.c12ccc(cc1)NCC2 c1(C(N)=O)cc(F)c(Br)cc1NC(C1CCCC1NC(=O)CCS(C)(=O)=O)=O c1(NC(C2C(NC(c3ccc4ncnn4c3)=O)C2)=O)c(Cl)cc(Cl)cc1[N+](=O)[O-] c1(N2CCC(C(C)NC(c3ccc(CC)cc3)=O)C2)nc2cccc(C)c2o1 C1(NC(C(CC)OCC)=O)CCOC12CCN(C(c1nnsc1C)=O)CC2 Cc1cnc2nc(C(=O)NC(CNC(c3n[nH]c(C(C)(C)C)n3)=O)CO)nn2c1 c1(NC(C(C(C)C)C)CNC(=O)C(n2cc(Cl)cn2)C)ccnc2ncnn12 C=CCCCC(=O)NCC(CCCC)NC(=O)C(C)Oc1ccc(OC)cc1 c1(OC)cc2ncc([N+](=O)[O-])c(N3C4CCC(O)C3CCC4O)c2cc1C(C)C C(C(C)(C(=O)NCC1(F)CC(NC(=O)C(F)=C2CCC2)C1)OC)OC c1(C(=O)NCCC(C)NC(=O)Cn2cnc(=N)[nH]2)ccc(C(F)F)c(F)c1 C1(NC(C2CCC(=O)N2)=O)CN(C(c2nccc(Cl)c2F)=O)CCC12CCC2 c1(C(=O)NCC(CNC(c2c(COC)noc2)=O)C)cn2ccsc2n1 C(=O)(C(CNC(=O)C(C)(C)CF)CCC)NC(CC#C)CC(=O)OC CN1CCC(C(N2CC(NC(=O)C=CCO)C(c3ccc(F)cc3)C2)=O)C1=O C=CC1(NC(C23CCC(NC(=O)CCCC4CCC4)(CC2)C3)=O)CCOCC1 c1(CCC)ccc(C(N2CCC(C(C)NC(C3CCCO3)=O)CC2)=O)cc1 C(CCSC)(C(=O)N1CCC2C(NC(c3ccn(C)n3)=O)C12)OC CCC(C)C(O)C(C)C(=O)N1CCCOC(CNC(=O)CS(=O)C(F)(F)F)C1 C1(NC(c2cnc(C(C)C)s2)=O)CCN(C(=O)CCC(C)CN(C)C)CC1CO c1(OCC(=O)NC(C2CCN(CCCC(=O)O)CC2)C)ccc(F)cc1 c1(C(=O)NCCC2CC(NC(CN(C)C)=O)C2)ccc2nccn2n1 C1(C(=O)NC2(CCC)CC2)CCCCN(C(c2cc[nH]n2)=O)C1 CC1(C)CN(C(=O)CC(F)(F)C(F)F)CCN(C(c2cn[nH]c2)=O)C1 c1(CNC(CCNC(C(C)(C)c2ccno2)=O)=O)ccc(O)c(F)c1 Cc1nc(C=CC(=O)NC2CCN(C(=O)Cn3nccn3)C23CC3)[nH]c1C C(=O)(C1=NOC(C)C1)N1C(Cn2c3c(nn2)C(=O)N(C)C3(C)C)CCC1.CC C1(C(=O)NCCN(C(=O)Cc2cccc(C(F)(F)F)c2Cl)C)CCCC(C#N)C1 C1(C(N2CC(C(CC)C)C2)=O)C=CCN(C(c2cn(C3CC3)nn2)=O)C1 S1(=O)(=O)c2ccccc2CN1C.c1(NCCOC(F)F)ccc(F)cc1 c1(CC(=O)NCC2C(NC(=O)CCN3CCOCC3)CC2O)csc(Cl)n1 N1(C(C(CC)(C)O)=O)CC(NC(=O)COc2cc(Cl)ccc2C)CC2(CC2)C1 C(=O)(C(F)(F)CCCC)N1CCC(N(CC#C)C(C2CCCCCN2C)=O)C1 Cc1nc(NC(C)(C)CCNC(c2cccc([N+](=O)[O-])c2)=O)c2cnn(C)c2n1 c1(C(C)(C)NC(CCCc2nnc(C)n2C)=O)ccc2ncsc2c1 N1(S(c2cnc(CCC)s2)(=O)=O)CCc2ccc(C)cc2C1C [N-]=[N+]=NCCCC(=O)NC1CCN(C(C2CC23CCSCC3)=O)CC1O C(=O)(C(COC)N=[N+]=[N-])N(CC(=O)NCC1CC(C(C)C)C1)CC#C c1(-c2nnc(N3CC(C)(C(=O)OC)OCC3)n2CC(C)C)cn2c(n1)COCC2 C1(CNC(c2c(C)nc(C)o2)=O)CCN(C(C2(C)CC3(CCC3)C2)=O)CC1(F)F CCCC(C)CC(=O)NC1CC(OC)CN(C(=O)CCC(=O)N(CC)CC)C1 c1(N(CC(C)N(C(C)=O)C)C)ccncc1S(=O)(=O)N1CCC(CC(C)C)CC1 C1(NC(CN2CCC(CNC(C#CC(OCC)OCC)=O)C2)=O)CCS(=O)(=O)C1 Cn1cc(NC(=O)C(N2CCC(Oc3cccc(Cl)c3)CC2)=O)c(Br)n1 c1(OCC=C)cccnc1C(=O)NC(CNC(=O)C(Cl)=CCl)C(C)C N1(C(=O)NC(CCc2ccc(OCC)cc2)C)CC(=O)Nc2ccncc21 N1(c2cccc(C)c2)CCN(CC(=O)NC(c2nc(C3CC3)cs2)C)C(C)C1=O c1(N2C(=O)CC(N(C3CCCN(C(C(C(C)C)O)=O)C3)C)C2)ccc(F)c(F)c1 C1(CC=C)(NC(C2C3CCCC23)=O)CCCN(C(C2CCCN2S(C)(=O)=O)=O)C1 C(=O)(C(F)(F)C(C)NC(CCC1OCC(NC(=O)OC(C)(C)C)C1)=O)OC c1(C(N(C(CCNC(CC(CC)OC)=O)C)C)=O)cc(Cl)ccc1O C1(NC(CC(C)SC)=O)CCN(C(c2ccc(N)c(F)c2)=O)CC(C)(C)C1 CCC(C(=O)N1CC(C(n2cc(Br)cn2)c2nn[nH]n2)C1)c1cccnc1 c1(C(=O)NC(CC=CC)C(=O)Nc2cccc(C(C)C)c2)cc2cccnc2[nH]1 C1(C(N2CC(O)(NS(C)(=O)=O)C2)=O)CN(C(=O)CCCn2cccc2)CCS1 C1(C(=O)NCC(C)(O)CNC(C(COCC)N(C)C)=O)CCN(C)C1=O N1(C(C2C(C)=C2)=O)CCCC2(CCN(C(c3cc(F)c(O)c(Cl)c3)=O)CC2)C1 c1(N2C(CNC(C3C(C)CC(=O)N3)=O)CC(F)C2)ncnc2cc(C3CC3)nn12 CC1CC(NC(c2csc(C(C)(C)C)n2)=O)CN(C(c2ccc(Br)o2)=O)C1 N(C(=NCCC1CCCC1)NC(C)Cc1ccccc1)C(C)C c1(CC)nc(C)c(C(=O)N(C)CC2(NC(=O)C(C)Sc3ncccn3)CC2)s1 Cc1cnc(NCC2CSC2)c(S(=O)(=O)NC(c2cnsc2)C)c1 c1(C(=O)NCC(C(C)C)NC(C2CC3CCC(C2)O3)=O)nnc(O)nc1O C1(=O)CC(C)(C)c2cn(nn2)CCCN1.Cc1cnn(CCCN2CCCC2)c1 c1(C(N2CCC3(NC(c4c(CC)cc[nH]4)=O)C(C2)C3)=O)cn2cc[nH]c(=O)c2n1 Cc1cnc(C(=O)N(C2CN(C(c3ccn(CCF)n3)=O)CCC2O)C)cc1C c1(CC(=O)NCCC(C)(C)NC(Cc2ccc(OC)nc2)=O)ccc(Cl)c(F)c1 CCCC(C)(CCC)C(=O)NC1CC(O)C1CC(=O)NCCc1cc[nH]n1 CC(CC(=O)NCC1C=CC(NC(C2CC=CC2)=O)C1)c1cccnc1 c1(C(=O)NC2CN(C(c3cccc(C(C)(C)C)c3)=O)CC2O)nccc(Cl)c1F C1(CC(=O)Nc2c(SC)nn(C)c2)CN(C(=O)CCN2CCC2)CCC1C c1(CC)ccccc1NC(C1CCCN1C(=O)COCc1ccnc(O)c1)=O c1(C(N(C2CCC(NC(C3(CC#C)CC3)=O)C2)C)=O)nccc2[nH]ccc12 CC1NC(=O)C=C1N1C(=O)N(C)C(CSCCS)C1 C1(C(=O)NC2CCCN(C(c3ccn(CCC)n3)=O)CC2)CCn2cncc2C1 C1(C(=O)NCCCCCNC(c2c(C)nc[nH]2)=O)COCC2(CCC2)O1 c1(CC(=O)NCCC(C)NC(C(CSC)O)=O)ccc2oc3ccccc3c2c1 N1(C(CC(C=C)C)=O)CC(C2CCCN(C(c3cc4c(C)n[nH]c4cn3)=O)C2)C1 c1(C(=O)NCC2CCCN(C)C2)ccc(-c2cccc(C(F)(F)F)c2)c(F)c1 c1(NC)cc(C(N2CCC(NC(c3c[nH]nc3C)=O)C(O)C2)=O)cc(Cl)n1 C1(CNC(C(C)CF)=O)CC(C(C)(C)C)CCN1C(c1cnc2sccn12)=O N1(C(CNC(=O)CCCCO)=O)CCC2(C1)CN(C(=O)Cc1ccccc1)C2 C1(NC(c2cn(CCC=C)nn2)=O)CN(C(C2CCCCS2(=O)=O)=O)CCC1F CCC(CC(C)C)C(=O)NCC1CC(O)CN1C(=O)Cc1cnc(C)o1 N1(C(C(COC)N(C)C)=O)CCC2(C1)CN(C(C1CC1C(=O)OCCO)=O)C2 C1(C(C)C)CCC(C(=O)NC(CNC(=O)CN2CCC2C)C(C)C)CC1 C1(C(N2CC(NC(c3cc(Cl)ccc3Cl)=O)CC(C)C2)=O)CNC(=O)C(C)(C)C1 C12(NC(C(CC)N(CC)CC)=O)CCCC1N(C(=O)C(c1ccc(F)cc1)=O)CC2 c1(CC)cc(C(=O)NC2(C)CN(C(c3sc(C4CC4)nc3C)=O)C2)nn1CCO N1(C(CNC(C)=O)=O)CC2CCCC2(CNC(c2cc(C3CC3)[nH]n2)=O)C1 Cc1c(C(=O)NCC(C)(C)NC(=O)CC2CCOC2)sc2cc(F)ccc12 CC1(C)CN(C(C2CN3CCN2CC3)=O)CC1NC(=O)CCc1ccncc1 c1(C(=O)Nc2n(C(C)C)ncc2)ccc(-c2cncc(-c3cccs3)c2)cc1 C1(O)(C(C)NC(C2C(C(C)O)C2)=O)CCN(C(C2CCN(C)C(=O)C2)=O)CC1 CCCCCC(C(=O)Nc1cccc(NC(=O)C(C)OC)c1)C(C)C CC(C)C(C(C)NC(=O)CCc1cocn1)NC(c1nc(Cl)cs1)=O c1(C(N2CCC(C)(CCNC(C3CCCOC3)=O)C2)=O)cc2ccccc2s1 C1(OC)CC(CNC(=O)Cn2cc(Br)cn2)N(C(=O)CC2(C)CCCC2)C1 C1(NC(CCC(C)SC)=O)CCN(C(=O)CCC(C)(F)F)CC1OC C1(C(N2CCC(C(C)NC(=O)C(C)(C)O)C2)=O)CCN(Cc2ccccc2)CC1 C1(C(=O)NC(CC#C)C)CN(C(C2(C)SCCCS2)=O)CC1F C(=O)(C1=CC(O)C(OC)C1)NC1CC(C(NOOCC2CC(=C)C2)=O)C1 c1(C(=O)NCC(CNC(c2ccn(C(CC)CC)n2)=O)C)csc2nccn12 C1(CC)CN(C(=O)CCc2cc(F)ccc2F)CCN1Cc1ccc(C)cn1 Cc1noc(N)c1C(=O)NCC(C)NC(c1cnn(C(C)C)n1)=O C12(CC)CN(C(=O)COc3ccc(Br)cn3)C(CNC(=O)CCF)(C1)C2 C(C(C)C(=O)N1CC(CNC(=O)C=CCN2CCOCC2)(OCC)C1)OC C(CN=c1[nH]c(C(=O)OC)nc(=N)[nH]1)C1CCC(NC(CCC(=C)Cl)=O)C1 N1(C(C(C=C)CC)=O)CC(C)(CNC(=O)C(C(C)C)C(C)C)CC1(C)C CC(C)(CNC(=O)COc1ccccc1F)CCNC(=O)Cc1ccc(F)cc1 C(CC(C(C)(C)C)NC(c1cnc(C)[nH]1)=O)N(C(c1n(C=C)nnc1)=O)C c1(OC)cc(C(N2CCN(C(=O)CN(C3CCC3)C)CC2)=O)nnc1C1CC1 n1(C(C)C)cc(S(=O)(=O)NCC23CCC(CN2)C3)cn1 c1(C(=O)OCC(=O)Nc2c(OC)ccc(NC(C)=O)c2)c(N)cc(F)cc1Br C1(C2CCN(C(=O)CCC3CCOC3)C2)(NC(c2nc(C)c(C)s2)=O)CC1 C1(NC(c2cc(OC)n[nH]2)=O)CCN(C(c2nccc(OC)c2F)=O)CC1CO C1(C(=O)NC(C)(C)CC=CC(=O)NCC(O)C(F)F)Cc2nccn2C1 C12(CNC(c3nc(C)sc3)=O)CCC1CN(C(=O)COc1ccc(F)cc1)C2 Cc1cc(C)c(C(=O)N(CCC(C)NC(=O)CC2CCC(=O)N2)C)[nH]1 CC1CCOCCN1C(c1c[nH]nc1CNC(=O)CCC(C)(C)F)=O N1(CC(C(=O)N(CC=C)Cc2ccco2)N(C)C)CCc2ccccc21 N1(CCC2(C(=O)NC(Cc3cn(C)nc3)=O)CC2)CCN2C(=O)NCC2C1 c1(C(N2CCC(OCCNC(C3CSCC(=O)N3)=O)C2)=O)cnn2ncccc12 c1(C(=O)NCC2CCCN(C(c3n(C)ccn3)=O)C2)cc(Br)ccc1N N1(C(C(CCSC)NC(C)=O)=O)CC2CCC1C2CN(C)S(=O)(=O)N(C)C CC(CCC(C)(C)C)C(=O)N1CCC2(C1)CN(C(C1CC(O)CN1C)=O)C2 C1(NC(c2ccc(C#N)s2)=O)CCN(C(C2(c3cc[nH]n3)CC2)=O)CC1CO C1(NC(c2c(CNC(CCCSC)=O)cnn2C)=O)CC2C(C1)C2(F)F Cc1ccc(S(=O)(=O)N2CCN(C(=O)NC(C)CC(F)F)CC2)cc1 CC1CC(NC(c2ncnc(O)c2Cl)=O)CCN1C(=O)CCCc1ccccn1 C#Cc1cc(C(N2CCN(C(=O)C(C)C3(O)CCC3)CC2)=O)cc(Br)c1 C(C(=O)NCCCN(C(=O)Cc1cc(C(F)(F)F)n(C)n1)C1CC1)(C(C)C)SC Cc1nccnc1C(=O)NC(C1(O)CN(C(c2cncnc2C2CC2)=O)C1)C N1(C(C(CC)C(C)(F)F)=O)CC2CN(C(C3CC(C)(C)C3)=O)CC2(C)C1 N1(C(c2noc(C)c2C)=O)CCN(C(=O)CC(C)(C)C)C2(CCC2)C1 c1(OCCOC)cccc(NC(C2(C3N(C(C(CC)O)=O)CCC3)CC2)=O)c1 c1(C(=O)NC2(CF)CCN(C(CC3OCC(C)(C)C3)=O)C2)coc2c1CCCC2 N1(C(C2C(CC)CCC2)=O)CCCC(C)(CNC(=O)C(C)Cn2ccc(C)n2)C1 C1(C(N2C(C(C)O)CC2)=O)N(C(=O)CC2CCC(=O)C2C)CCC1(C)C c1(N2CC3C(CNC(=O)C(C4CC4)C4CC4)C3C2)nc(Cl)nc2c1S(=O)(=O)CC2 O=C(CCCCc1cnn[nH]1)NC(C1CCOC1)CNC(=O)Cc1nnc(O)s1 Cc1cc(C(=O)NC2(C(=O)NCCC3CCCO3)CC2(C)C)nc(O)c1 c1(C(N(C(c2cc(C)on2)C)C)=O)ccc2c(c1)CCC(C)N2 C#Cc1ccc(C(N2CCC(C)(CNC(=O)C(F)=C(C)C)C2)=O)cc1F C1(NC(C(C(C)C)OCC)=O)(CC)CCCN(C(=O)COCC(C)C)C1 N1(C(CC2CC(OC)C2)=O)CCN(C(=O)C(=Cc2cncn2C)F)C(CCO)C1 C(N=c1[nH]nc(-c2ccon2)s1)C1(CNC(=O)C2CC2)CC1.C1CCCC12CC2 c1(OC)cccc(C(=O)Nc2nccc(F)c2F)c1OC(F)F Cc1cc2[nH]c(=NC(C)CC(C)NC(=O)CN(C)C(N)=O)c3ccccc3n2n1 c1(C(N2CC(CNC(C3=C(C)OCC3)=O)OCC2)=O)cccc2c(Br)ccnc12 c1(C(N2C(CC(=O)OCC)CSCC2)C(=O)NC(C)CC)ccc2c(c1)COC2 C(=O)(C1COc2ccccc21)NCC1(NC(C2C(C)C2(F)F)=O)CCC1 N1(C(c2cc(C(N)=O)oc2)=O)CC2(CCN(Cc3cccc4nonc34)C2)C1 C1(NC(c2c(C)nc(C3CC3)[nH]2)=O)CC(C)CN(C(C2C(C)(C)C2(C)C)=O)C1 c1(CC(=O)NCCNC(CC(c2ccc(Br)cc2)C)=O)cc(O)nnc1O C1(C)(C(=O)NCC2C(CC(=O)NCC(C#C)CC3CC3)C2)COCCO1 C1(OC)CC(F)CN(C(C2CC=CCN2C(c2ncccc2Cl)=O)=O)C1 N1(C(=O)NCC(=O)N(C)C)CCCC(c2cn[nH]c2)C1 c1(C(=O)NCC2CC(NC(CC(CC)SC)=O)C2)cc2cccnc2o1 c1(CC(=O)NCC2CC2Cn2cc(-c3cscn3)nn2)c[nH]c2ccc(Cl)cc12 C(=O)(C1=CCCN(C(c2cc[nH]c2C2CC2)=O)C1)N1C(C)(CCO)CC1 C(C)(CC(=O)N1CCC2(CCN2)CC1)(C(=O)O)N(C)C CC(O)C(C(=O)NCC12CC(CCO1)C2)NC(c1cnc(S)nc1)=O N1(C(c2ccc(CC)o2)=O)CCC(NC(c2c[nH]nc2OC)=O)C(CO)C1 c1(CC(C)C)cc(C(=O)NC2CC(CNC(=O)C=Cc3cc[nH]n3)C2)no1 CON(CCC(=O)NC(C)CCO)C(=O)C12CCC(C)(C1)OC2 N1(C(C2COCCN(C(C(CC)N)=O)C2)=O)CCCC(C2CCCNC2)C1 C1(C(=O)NCCCCC(C)NC(C(n2ccc(C)n2)(C)C)=O)CCCC(C)(C)C1 C1(N(C(C=NOC)=O)C)CCN(C(=O)C=Cc2ccsc2C(F)(F)F)CC1C c1(C(=O)NC(C=C)C)cc2c(-c3cnc(OCC)nc3)cncc2s1 C=CCC(CC)C(=O)NC(C1CN(C(=O)CCc2nc(-c3ccco3)no2)C1)C c1(CC(N2CCC(OC)(CNC(C3(Cl)CC3(C)C)=O)C2)=O)cc2ccccc2o1 CCC(O)C(C)C(=O)NCC1CCCCN1C(C1CCCN1C1CC1)=O C1(F)(CNC(C2CCC(C)(C)C2)=O)CCCN(C(C2(C)CC2(C)C)=O)CC1 O(C1CCC(=O)c2ccccc21)C(Cc1nc(CCCC)sc1)=O C1(NC(C(c2ccc(OC)cc2)O)=O)C2CC1CN(C(c1cnn[nH]1)=O)C2 c1(C(=O)NCCC#CCC)oc(CNC(=O)C=C(C)c2ccco2)nc1C c1(C(N2C(CNC(CC=CC)=O)CCC(C)(C)C2)=O)cnc2nc(C)[nH]n2c1=O O=C(CC(F)(F)c1ccccc1Br)NCCCN1CCCC1=O C1(N(C)C(C2CCNC2=O)=O)CCCN(C(c2cccc(O)c2)=O)CC1 c1(C(C)COCCNC(C(=O)NC(C)Cc2ccccn2)=O)ccccc1F.OC c1(NC(C2C(CNC(C(CC)n3ccnc3)=O)CCO2)=O)ccc(C)nc1 N1(C(c2c(F)ccc(OC)c2)=O)CC2(C1)SCCC2NC(=O)CCC1CCCO1 c1(C(N(CCN(C(C)C)C(c2cnn(C)n2)=O)C)=O)c[nH]c2cc(C#N)ccc12 N1(C(COc2ccc(OCC)cc2)=O)CCN(C(=O)CCCC2CCC2)CC1C C(=O)(C1CCc2cccnc21)NC(C1N(C(CC(C)(C)OC)=O)CCC1)(C)C C1(C)(NC(C(C2CCC2)NC(c2n(C)ccn2)=O)=O)CN2CCC1CC2 N1(C(C2(CC=C)COC2)=O)CC2(CCCC2NC(c2cc(C(C)C)oc2C)=O)C1 N1(CC(=O)NCCCC(=O)NCCc2cn(C)nn2)CCOCC1=O C12(NC(c3occ(C)c3C)=O)CCC1CN(C(C1(F)CCS(=O)(=O)C1)=O)C2 N1(C(c2c(OCC)ccs2)=O)CCC(CO)(CNC(c2conc2CC)=O)CC1 CC1(NC(=O)CC2CCCCO2)CCN(C(=O)CSCc2cccnc2)CC1 N1(C(CCSC)=O)CC2C(NC(=O)CC3CCCSC3)C2C1 c1(C(N(CC(C)NC(=O)C(C)N(C)C(=O)OC(C)(C)C)C)=O)c[nH]c(Br)c1 C(CCCCC(=O)NCC(C)CN(C)C(c1cnc(O)n1C)=O)OCC c1(-n2cc(CC3CC(OCC)C3(C)C)nn2)ccc(Br)cc1C C(=O)(CCCCC(C)=O)NC1CC=C(C(=O)NC(CCCC)C)C1 N1(C(c2[nH]c(=N)sc2)=O)CCc2[nH]nc(CNC(C3CC4C=CC3C4)=O)c2C1 N1(C(CC2(OC)CCC2)=O)CC(N(C(=O)C(C)OCCC(C)C)C)C(C)(C)C1 Cc1nc(N)cnc1C(=O)NCCC1CN(C(C2CCCS2)=O)CCO1 C(N=c1nc(N2CCOC(C)CC2)c2sccc2[nH]1)C1N(C(C)=O)CCC1 C(=O)(C1=CS(=O)CCC1)N(CC(CNC(Cc1ccc(C(C)=O)cc1)=O)C)C N1(C(c2n(C)ncc2)=O)CCC(CF)(NC(C2CC23CC(O)C3)=O)C1 C#CC1(C(=O)NC2COCC2CNC(C2(C)CC(C)(C)C2)=O)CCCC1 N1(C(Cn2c(C)ccn2)=O)CC2CC1CC2NC(=O)Cc1ccccc1Cl N1(C(CC2N(C(C(COC)N(C)C)=O)CC(F)C2)=O)CC2CCCCC2C1 C(=O)(C(C)(C)CC(C)C)NCC1N(C(c2cc(C)n(C3CC3)n2)=O)CCOC1 c1(CC(=O)NC2CCC(NC(C(n3cc(Cl)cn3)C)=O)C2)ccc2c(c1)CCC2 CCC(C)CC(=O)NCC1(CNC(c2csc(C(C)(C)C)c2)=O)CCC1 c1(C(c2ccn(C)n2)NCCOC)nnnn1CC1(OCCO)CCC1 Cc1cccn(CC(N2CCC(NC(C3(n4cccn4)CC3)=O)C2C)=O)c1=O C(CC(O)CC)NC(C(N1C(CC(=O)NC)CC1)=O)=O O=C(NNc1ccc2ccccc2n1)NCC1Cc2ccccc2CN1 C1(CCCC)CCCC1(c1nnnn1CCCSC)NCCS(=O)(=O)CC Cc1csc(C)c1S(=O)(=O)NC(c1nccn1C)C(C)C C1(NC(C=Cc2cccc(C)c2)=O)CC2(CCC(NC(=O)COC(F)F)CC2)C1 N1(C(c2cc(C)[nH]n2)=O)CCCN(Cc2cccc(F)n2)CC1C c1(C(C2CCC2)=O)nncn1C.C(C(C)CN)C=O.C(CO)OC c1(CN2CC(NC(=O)CNC(C3CCCCC3)=O)C(F)C2)cccc(Cl)c1O C(=O)(C(C)CC(F)F)NC1(C(=O)NCCCC)CCC1 C1(C(=O)NCC(C)CNC(=O)C=C2SCC(=O)N2C)CCc2cc(F)ccc2O1 C=Cc1cccc(CNC(=O)CC2CCCN2C(c2cc(O)nc(O)n2)=O)c1 c1(NCC2CCC(NC(C3(C)CC3Br)=O)CC2)ccc([N+](=O)[O-])c2cccnc12 C1(NC(C(C2CN(C(C(C)OC)=O)C2)O)=O)CCCN(C2CC2)C1 c1(SCC(=O)NC2CN(C(c3c(C)nn[nH]3)=O)C(C)(C)C2)cncc([N+](=O)[O-])c1 C1(C(=O)NCCC#C)(CNC(=O)CSCC(F)F)CCCCC1 CCC(CC(=O)NC(C(=O)NC1CN(C(C)C)C1)C1(C)CC1)OC C1(C)(CNC(COCC(=C)C)=O)CN(C(=O)CCSc2nccn2C)CCO1 C1(CNC(=O)C=Cc2cnc[nH]2)CC12CCN(C(c1nnc(O)nc1O)=O)CC2 C(=O)(CC(F)(F)C(F)F)N1CCCC(CCNC(=O)C(O)C(F)(F)F)C1 N1(C(C(C(C)(C)C)(C)C)=O)CCC2(CC1)CC(NC(=O)C#CC1CCCOC1)C2 N1(CC(=O)N(CCCNC(C2CCN(C)CC2)=O)C)CC(C(F)(F)F)CCC1=O c1(CC)cncc(C(=O)NC2CCCC(N(C(=O)Cc3cnc[nH]3)C)C2)c1 C1CC(O)C(=O)N2CCC2C(=O)N1.Cc1nccn1C(C)C(=O)N(C)C c1(-c2cn(CCOC)nc2)nc(-c2ccnn2C)nn1CC(F)F CC(O)CCCC(=O)N(CC(C)CNC(=O)CNc1cccc(Cl)c1)C N1(C(C2C(=C)CC2)=O)CC(C)(C)CC1CNC(c1c(OC)ccnc1OC)=O CCC1=NOC(C(N2CC=CC(C(=O)NCC(=O)NC(C)C)C2)=O)C1 C(=O)(CCP(C)(C)=O)NCC(CCOC)NC(c1cc(C(C)(F)F)ccc1C)=O c1(C(N2C(CNC(CCOCC#C)=O)CC2)=O)cn2cccc(C(F)(F)F)c2n1 N1(C(C2C(C=C)CC2)=O)CCC2(CCC2)C(NC(c2ccc(F)cc2)=O)C1 c1(C(N(c2cccc(C(F)(F)F)c2C)CC)=O)cc(S(C)(=O)=O)c(Cl)cc1Cl C1(C)(NC(CN(C(c2c(C)scc2)=O)CC2CC2)=O)CCCC(C)(C)C1 c1(CC)ccccc1CC(=O)NCC1CCCCN1C(C1CC(=O)C1C)=O CN=S(C)(=O)c1cccc(C(N2CC(CCNC(=O)CCCNC(N)=O)C2)=O)c1 N1(C(CCCCC)=O)CCCC(O)(CNC(c2cn(C3CCC3O)nn2)=O)CC1 n1(CC)nc(C(=O)NC(CCOCCO)C(=O)NC2CN(CC(F)F)C2)cc1C c1(C(=O)OC)ccc(NC(=O)Cc2cnn(C(C)C)c2)c2ncccc12 C(=O)(C(CC)(CC)CC)NCC(C)(C)NC(CC(CC)C1CCC1)=O N1(C(c2n(CC(C)C)ncc2)=O)CC(O)CC1CNC(=O)C(C)C C12(C(N3CC(CNC(C=CC=CCCCCC)=O)OCC3)=O)COCC1C2(F)F Cc1cc(C(=O)NC23CCC2CN(C(C2(F)CCCCC2)=O)C3)c(C)cn1 O=C(N=c1[nH]n(-c2ccc(F)cc2)cc1Br)Nc1c(C(=O)O)nn2c1CCCC2 c1(C2C(=O)N2C2CC2)cn(C)nn1.C1(C(C)C)CC1C(=O)OC(C)(C)C c1(CC)cnccc1C(=O)NCCC(=O)NC1CCSC1 CCC(C)(CCO)NC(C1CN(C(c2cc[nH]n2)=O)CC1OC)=O N1(C(C2C(C)OCCC2)=O)CCCCC(CNC(c2cc(CO)ccc2Cl)=O)C1 N1(C(CCSCCC)=O)CC2CC(NC(=O)COCCCC(C)C)C(C2)C1 Cn1[nH]c(C(N2CCCC2CCNC(c2cccc(O)n2)=O)=O)nc1=O N1(C(C)C)CCC(N(C(=O)C(N)CC2CCNC2=O)C)C1=O c1(CN=C(NCC2CCCC(C)(C)C2)NC2CCCCC2)ccc(C#N)c(Cl)c1 C1(NC(c2c(C(C)C)c[nH]n2)=O)CN(C(c2cc(C3CC3C)on2)=O)C(C)(C)C1 C(C)(C)(C(=O)NC1CC(CCC(=O)NCC2CC2(F)F)C1)OC c1(C(N2CC3C(C(=O)NCCC=C)C3C2)=O)ccc(F)c(S(C)(=O)=O)c1 Cc1ccc(Br)nc1N(C1CCNCC1)C(=O)Cn1cc(C2CC2)nn1 CCC(=O)CCC(=O)NCC(C)(C)OCCNC(c1ccccc1OC)=O Cc1ccoc1CC(=O)Nc1nc(C2CCOC2)cs1 NC(=O)CC(O)C(=O)NC1CCCC(C(=O)Nc2ccc(O)cc2Cl)C1 CCS(=O)CC(=O)N1CCN(CCN(C)C(C2(C3CC3)CCC2)=O)CC1 C(=O)(C(O)CC(F)(F)F)N1CCN(C(CCC=CCC=C)=O)C(C(F)F)C1 c1(C(N2CC(CNC(C(C)N(C)C)=O)C(C)C2)=O)cc(Br)c2n[nH]cc2c1 c1(C(=O)NCC2CC(C)N(C(=O)CCC(N)=O)C2)cnc2c(ccn2C)c1 N1(C(c2c(C)n(C)nn2)=O)C2CCC1C(C)C(NC(=O)Cc1cncs1)C2 C1(OC)CC(C(=O)Nc2cnn(CC(C)C)n2)C12CCOCC2 C=CCCCC(C)NC(=O)COC1CCN(C(c2n[nH]c(C)c2C)=O)C1 C1(OC)CC2CC(C1)N(C(=O)NC1CC3(CCCCC3)C1)C2 c1(C(C)=O)ccc(NC(C2(C)CCN2Cc2c(F)cccc2I)=O)c(C#N)c1 C=CCCCCCC(=O)NCC=C1CCN(C(C2CC2(C(C)C)CC)=O)CC1 Cc1nn(C)cc1C(=O)NC1CCC(NC(c2ccc(CSC(F)F)o2)=O)CC1 Cc1csc(CCC(=O)NCC2(C(C)(C)O)CN(C(c3cncnc3)=O)C2)n1 c1(C(C(=O)NCCN(C(C2COCCO2)=O)CC)C)ccc(C)cc1 C1(C(N2C(C)CC2CO)=O)CCOCCN1C(c1nc(Cl)cs1)=O c1(C(N(CC(CC)NC(C(CC)SC)=O)C)=O)c(C)nn(C)c1F c1(C(=O)NCCOC(CC)C(=O)OC(C)(C)C)cc([N+](=O)[O-])ccc1OC c1(CC(N2CC(NC(C3C(C=C)CC3)=O)C2)=O)c(C)cccc1Cl Cc1ccncc1C(N1CC2CC1(C(N1CCC(F)CC1)=O)C2)=O C=C(C)C(C)(O)C(=O)N1CCCC(CNC(c2sc(-c3ncc[nH]3)nc2C)=O)C1 c1(C(=O)NCC2(O)CC(NC(=O)CC3CCC3)C2)cccc2c1CCO2 CCCC(CC)CCC(=O)NC12CCC(CC1)CC2.C1(=O)NOC(C)C12CC2 C(=O)(CCCC(F)F)N(C1CCCN(C(C2(CC)CCCC2)=O)C1)CCO C1(CCNC(c2cc(C(N)=O)ncc2)=O)CN(CCn2ccnn2)CCCO1 c1(CC)cc(C(=O)NCC2CC2CNC(C2CCC2)=O)c(C)o1 C(c1ccc(C)c(C)c1)=CC(N1CCN(C(C=C(C)C)=O)C(c2cn[nH]c2)C1)=O C12(CNC(c3nc(C#C)sc3)=O)CC(CO1)N(C(=O)C(C)CC(C)C)C2 c1(CN2CC(F)CC(C(N3CCCC(CCO)C3)=O)C2)cc(F)c(F)cc1O N1(C(c2ccc(CC)o2)=O)CCC2(NC(=O)CC(C)(C)SC)CCCCCC12 c1(C(N2C(CNC(C(CC(C)C)OC)=O)CCC2)=O)cc2occ(Br)c2[nH]1 C1(CNC(=O)N(CC(C2CCCO2)O)CCO)CCS(=O)(=O)CC1 c1(C(N2CC3C(CNC(c4cnc(=N)[nH]c4)=O)C3C2)=O)cnc(O)c([N+](=O)[O-])c1 c1(NC(C2C(CNC(C(C(C)C)OC)=O)C2)=O)cccc([N+](=O)[O-])c1C Cc1csc(C(O)CC(=O)NCC(C)N(C(=O)C=Cc2ccsc2)C)c1 N1(C(COCC)=O)CCC2(CCC(NC(=O)CCNC(=O)C=CCl)CC2)CC1 CC1(C)C(CNC(=O)CC2=CCCC2)CCN1C(c1ccc[nH]1)=O Cc1ccnc(CNC(=O)CC(CNC(C2(CO)CC2)=O)C2CCC2)c1F N1(C(CN(C)C)=O)CCN(C(CNC(=O)CCc2cn[nH]c2)C(F)(F)F)CC1 Cn1ncc(Cl)c1C(=O)NC1CC12CC(NC(=O)CCc1ccncn1)C2 C1(NC(C(C)OCCOCC)=O)CC2CCC1N2C(=O)CCC1CCC1 c1(N(CC(=O)NCC)C)nc2cccc(F)c2c(=NCC2(Cl)CC2(F)F)[nH]1 c1(CC(N2CC(O)(CN(C(c3[nH]c(=NC)sc3)=O)C)C2)=O)cccc2c1CCC2 CCCC(C)(CC)C(=O)N(CCCNC(=O)C(C(C)C)n1cnnc1)CC C(c1ccc(F)cc1)=CC(N1C(C2CCN(C(=O)CC(O)C3CC3)C2)CCC1)=O c1(C(=O)NCC(CNC(c2ccc(C)c(N)c2)=O)C)cccc2oncc12 C(=O)(CC(O)C(C)C)NC1CC(CCNC(C(n2c(C)cc(C)n2)C)=O)C1 N1(C(CNC(C)=O)=O)CCC(NC(=O)C(c2ccc(F)cc2)(C)O)C(O)C1 C1(CNC(C2(C=C)CC2)=O)CC(C)N(C(c2ncccc2N(C)C)=O)C1 c1(C2C(NC(=O)NC(CNC(CC#N)=O)C3CCC3)C2)ccccc1 CCCCC(O)C(C)C(=O)NCCCC(CO)NC(=O)CC1(CSC)CC1 Cc1ccc(C(=O)NCC2CC3CC3N2C(=O)CN2CCCCC2=O)cc1 CCC(CC(=O)NC1CCCC1CNC(C1(O)CC(C)(C)C1)=O)C1CCC1 N1(C(C(N2CC(C)C2)C)=O)C(CNC(=O)Cc2ccnn2C)CC2CCCC12 C(=O)(C(C(C)(C)C)c1cc[nH]n1)N1CCC(N(C)C(c2ccnnc2O)=O)C1 C1(C(=O)NCC(CNC(C2(C(=O)OC(C)(C)C)CCC2)=O)F)NC(=O)C2CC12 C1(C(C)NC(c2cnn(CC(F)(F)F)n2)=O)CCCN1C(=O)CC1CCCC1O C1(N(C(c2c(CCC)nco2)=O)C)CCCC(NC(C2(F)CCC2)=O)C1 C(=O)(C(CC(N)=O)NC(c1ccnc(C)n1)=O)N1CCCC(CCC#C)C1 c1(OC)cc(N(C)C)ccc1C(=O)NC(C1(O)CCN(C(=O)C(C)(C)CO)C1)C Cc1c(C(=O)NCC(C)(C)OCCNC(c2nn(C)cc2C)=O)[nH]ccc1=O CCCCCCC(CC)(CC)C(=O)N(CC(C)(C)NC(C1CS(=O)(=O)C1)=O)C C(=O)(C(CC(C)(C)C)OC)NCC=CC(N1CC(CC)N(C)CC1)=O C(=O)(CS(N)(=O)=O)NC1C(CC)CCN1C(C)=O CC(C)C(C#N)C(=O)NCC1CCN1C(c1ccnn1C(C)(C)C)=O C1(NC(C2CCCO2)=O)CN(C(=O)C(F)=CCCF)CC12CCCC2 C1(CC=C)(NC(=O)C(C)(C)F)CCN(C(c2ccc(F)c(C(F)(F)F)c2)=O)CC1 c1(C(=O)NC2C(NC(c3cc(C)n(C)n3)=O)CCC2)ccc2nccn2n1 CC(C)C(C(=O)NC(C(N1CCOC(CCF)C1)=O)C1CC1)C(C)C C1(C)(NC(C2N(CC)CCC2)=O)CCN(C(=O)CCCc2nc(C3CC3)no2)C1 C(=O)(C1CCCc2c(O)cccc21)N1CC(NC(=O)C(C2CCCCCCC2)O)C1 C(=O)(C1=C(CF)N(CCc2ccc(OC)cc2)C(=S)NC1c1cc(Br)co1)OC c1(C(=O)NCC(CNC(=O)CC2CC(n3cccn3)C2)CO)cc(F)cc(Cl)c1 c1(C(=O)NCC2C(NC(c3c(C)cnnc3)=O)C2)c[nH]c(=O)c2ccncc12 C1(NC(c2c(COC)nn(C)c2)=O)CC2CC(C1)CN(C(=O)CC1CCC1)C2 C(=O)(C(C)CC(F)F)N1CCC(NC(Cn2cc(-c3cnc(C)o3)nn2)=O)CC1 Cc1cc(NC(c2occc2F)=O)ccc1NC(=O)CN1CCCS1(=O)=O c1(CNC(NC2C(C)(C(F)F)C2)=NCC2CCOC2)nc2ncccn2n1 N1(C(C(C(C)O)C)=O)CC2CC(C)N(C(c3cccc(OCCF)c3)=O)C2C1 c1(C(N2CCN(C(c3ccc(C)o3)=O)CC2C(F)(F)F)=O)ccc(F)c(C)c1Cl N1(C(COCCC)=O)CCC2(CCC2NC(=O)C(F)C(C)(F)F)CC1 N1(C(c2c(C)cns2)=O)CCC(C)(C)CC1C(N1CC2CC2(CO)C1)=O c1(N2CC(C)SC2)nc2c(c(=NCc3cc4cc(Cl)ccc4o3)[nH]1)CC(C)CC2 CCC(C)CC(=O)N1CCCC1C1CCN(C(C2CCN(CC)C2=O)=O)C1 CC1(C)CC(NC(c2cc(C(N)=O)co2)=O)CCN(C(=O)C=CBr)C1 c1(CCC(=O)NC(CCCC)CNC(c2snnc2C)=O)ccc(OC)cc1F N1(C(C2CCC(CNC(=O)Cc3ccccn3)C2)=O)CCC(CF)CC1 c1(C(=O)NC2C(NC(=O)COC(F)F)CCC2)c(Cl)cc(Cl)cc1Cl C1(NC(c2ccc(N)c(F)n2)=O)CCN(C(c2cccc(Cl)c2)=O)CCC1(F)F c1(OC)ccc(Cl)c(C(=O)NC2CCC(F)(CNC(C3CCCCO3)=O)C2)n1 C1(NC(C(CC(C)C)OC)=O)CCN(c2nc(C)cc(C)n2)CC12CCC2 N1(C(CCC2N(C)CCC2)=O)CCCC(C)(CNC(c2ccccn2)=O)C1 N1(C(C2CCCC(=O)C2)=O)CCCCCC1CNC(=O)CC1CC=CC1 S(=O)(=O)(c1ccc(Br)c2ccccc12)NC(C(=O)OC)C(C)C1CC1 N1(N(C(=O)NCC(C(=O)OC)CC2CCCC2)C)CC(C)(C)Oc2ccccc21 c1(C(=O)NC(C2CCN(C(C3(C#N)CCCC3)=O)C2)C)nncc2c1CCCC2 CCCCCCC(C)C(=O)NCC(C(C)(C)C)NC(c1c(Cl)n[nH]c1C)=O CC1(C)CCC(CS(N2CCCC2c2ccco2)(=O)=O)OC1 C=C(Cl)CCC(=O)NCC(C)=CC(=O)Nc1cnn(CC)c1C C1(NC(CNC(CCC)=O)=O)CCN(C(C2OCCCO2)=O)CC1C C(=O)(CCCCC(N)=O)NC1(CCNC(c2c(C)cccc2F)=O)CC1 C(CN=S(C)(C)=O)NC(C(CO)NC(C(CC)n1ccnc1)=O)=O C1(NC(CCC(C)O)=O)CCC2CN(C(C3(C)CCCS3(=O)=O)=O)CC2C1 c1(C(=O)NCCCN(C(C2(C#N)CCCCC2)=O)CC)ccnc(P(C)(C)=O)c1 N1(CC(=O)NCCS(CC#N)(=O)=O)CC(O)C(O)C1 CC(C1CCCc2ccccc21)NC(=O)NNC(=O)c1nccs1 Cc1nn(CC(N2CCOCC2CNC(C2(CF)CCOCC2)=O)=O)cc1Cl C12(NC(C3CCN(C(C)=O)CC3)=O)CCCC1N(C(=O)CCC1(C)CC1)CCC2 N1(C(C2(C(=O)OC)CCCC2)C(=O)OC)CCc2[nH]c3ccc(F)cc3c2C1 C(C1CCCN1C)=CC(=O)NC1(CC(N2CCC(OCCNC(C)=O)C2)=O)CC1 c1(C(=O)NCCC(C)NC(=O)CCCCC(F)F)cn(C)c(=O)c2c1CCCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C(=O)N(C(C=C)C1CC1)C)C)C N1(C(C=CC=CCC)=O)CC=CC(NC(c2ccc(-c3nnc(S)o3)cc2)=O)C1 Cc1cc(C(=O)NCCCC(C)NC(c2ccnn2C2CCCC2)=O)cc(N)c1 N12CCOC(CC1)C2=O.c1(NC)cnccc1C(N1CC=CC(OC)C1)=O N1(C(C2CN(C(C)=O)C2)=O)CCC(CO)(CNC(=O)CSC2CCOCC2)CC1 c1(C(=O)NC2CCCN(C(C(CC=C)CC)=O)C2)cc(C#N)ccc1C C1(NC(c2c(C)nns2)=O)CC2(C1)CC1(CC(NC(=O)CN3CCCCC3)C1)C2 CCC(C(=O)NCC1CC1NC(c1cc(COC)[nH]n1)=O)OC N1(C(C2CC(C)C2)=O)CCC(C2CN(C(C3CC3c3ccncc3)=O)C2)CC1 c1(C(=O)NCC2CC(NC(CCCC(N)=O)=O)CC2O)ccc2scnc2c1 S(=O)(=O)(c1cnccc1NCCCc1ccsc1)N1CCCC(C)(CO)C1 c1(N(C)Cc2cscc2Br)ccc(S(=O)(=O)N2CC3COCC3C2)cc1F CC1CN(C(=O)CC(CNC(C2(C)CC2(C)C)=O)C2CCC2)CC1O c1(C(=O)NC2C(C)CN(C(=O)C=Cc3ncc[nH]3)C2)cc(O)nc(O)c1 Cc1cc(C(=O)NC2CC2CNC(=O)CCC2CCCOC2)c(C)[nH]1 C(=O)(CC(C)CC(F)(F)F)NC1CC(C)(NC(Cn2c(C)c(Cl)cn2)=O)C1 C(=O)(C1=NOC2(CCN(C(C)C(=O)Nc3cc(C)ccc3C)CC2)C1)OC c1(C(=O)NC2CCCC2C(=O)NCc2ccccc2SCCO)ccc(F)cc1O c1(C(C)C)nn(C)cc1C(N1CC(NC(=O)Cc2cnc[nH]2)C(O)C1)=O C1(CC)(NCCNC(=O)Cn2cnc(Br)n2)CCN(C)CC1 c1(-c2nnn(C(COCCOC)(C)C(=O)O)n2)ccccc1-c1ncn(CCO)n1 c1(C(=O)NCC(CC)NC(=O)C=C(C)C(C)(C)C)cc(C2CC2)oc1C1CC1 CCCC(O)CC(=O)NCC1CC(F)(CNC(c2sccc2SC(F)F)=O)C1 c1(CN2C(C(=O)Nc3c(OC)cc(C)cc3)CC(F)(F)C2)ccc(C#N)cc1Br n1(CC(CCOC)O)c(-c2cc(C)n(C)c2C)csc1=Nc1ccc(OC)cc1 c1(NC(CC(C)C)CNC(C2CCC(C)C2)=O)nc(C2CC2)nc2c1CCC2 CCCCCC(F)C(=O)NCC1CN(C(=O)C(C)(C)C(C)(C)C)CCC12CCC2 N1(C(c2cc(C)sc2C)C(=O)NCC=C)CCCSCC1C c1(OC)cc(C(=O)NC(C)CCCNC(=O)Cc2cn(C)nn2)c(C)cc1O CC1CCOC(C(=O)N(C)CC2CCCN2C(=O)CC2(C)CCN(C)C2)C1 C1(NC(=O)COCc2cncc(F)c2)CC(NC(C2CCCC2)=O)C(O)C1 C1(CNC(CCc2nc(C)sc2)=O)CCN(C(C2CCCC2)=O)C(C)C1 N1(C(c2cscn2)=O)CCC2C(CCN2C(c2c(F)cccc2I)=O)C1 C(CCO)(C(C)(C)C)NC(C(C1CCN(C(=O)C2=CC(C)(C)C2)C1)C)=O CCCCS(=O)(=O)CC(=O)NCC=CCNC(c1cn(CCCC#N)nn1)=O N(C(=NCCc1ccccc1)N1CCCC(O)CC1)Cc1cccc(C#C)c1 C1(NC(C(C)C)=O)CCC2(CCN(C(c3ccc(Cl)c(O)c3)=O)CC2)C1 c1(OC)ccc(C(C)(C)C(=O)NC(c2ccccc2)CNC(=O)CC(C)F)cc1 c1(C2(C)CC2)ccc(CO)cn1.c12ccc(cn1)C(=O)N1CC(n3cc-2nn3)C1 N1(C(c2c(CC)cco2)=O)CCC(NC(C2CC(F)(CSC)C2)=O)C(CC)C1 C=CCCC(CC)(c1nnnn1CC(F)F)Nc1cnc(CSC)nc1 C1(CCC)C(=O)NCCN1C(=O)C(C)(C)C(C)NC(c1nnn(C)c1C)=O c1(OC)cc(C)cc(C(=O)NCC(C2CC2)NC(c2ccnnc2)=O)c1O c1(CNC2CCN(C(c3nc(C)n(C)c3)=O)CC2O)n[nH]c2ccc(Cl)cc12 C(CCC(CCC)NC(c1cnccc1C(F)(F)F)=O)NC(C(C=C)(C)C)=O CCCCC(C)(F)C(=O)N1CCC(O)(CCNC(c2nccnc2CC)=O)CC1 c1(C(N2CC(CC(C)NC(=O)C(C)NS(C)(=O)=O)C2)=O)cnc(C)[nH]1 C1(NC(c2cn[nH]c2)=O)CC2CCC(C1)N2S(=O)(=O)c1ccc(Br)s1 N1(C(C(c2c(C)cncc2)C)=O)CC2(C)CC1C2NC(c1csc(Cl)n1)=O CCCCCCC(C)C(=O)NCC1C(C)CCN1C(C1CCC1)=O c1(C(N2CCC3(NC(Cc4nc(C)[nH]n4)=O)C(C2)C3)=O)cnc2c(c1)CNC2=O Cn1c2c(ccc1=O)C(NC(C1(C)CCC(=O)CC1)=O)CCC2 C1(NC(C2(C)CNC(=O)C2)=O)CC(F)(F)CC1NC(=O)Cn1nccn1 O=C1Cc2ccc(C(N3CC=CC3CNC(=O)C(F)CC3CCC3)=O)cc2N1 c1(NC(c2ccc(C(C)OC(C(C)(C)CO)=O)cc2)=O)cc(Br)ccc1F N1(C(C(COC)C)=O)CC(OC)C(NC(=O)CCSc2cccc(OC)c2)C1 CC12CC3CC(CC(NC(=O)NC4CCOCC4c4ccc(F)cc4)(C3)C1)C2 N1(C(C(CCCC)O)=O)CCC(C(=O)NCc2cc(F)cc(F)c2)=C(F)C1 c1(C(=O)NC(CNC(CN(CCCCCC)C)=O)C)ccc(Br)c(C)n1 N1(C(C2CN(C)C(=O)N2)=O)CC(=O)NCC1C(=O)Nc1cnn(C)c1 Cc1cc(C(=O)NC2CCC(NC(=O)C(C)OC3CCCCC3)C2)sn1 S(=O)(=O)(c1cc(C)cnc1N1CCC(O)C(F)C1)N(CCCC(=C)C)C CC1(C)CN(C(C2(C)CC=CCO2)=O)CC(CNC(=O)CCc2ccsc2)O1 C(=O)(C1=CC(C)CC1)N(CCCNC(C1C(OC)(OC)CC1)=O)C c1(NC(C)=O)ccc(Cl)c(C(N2CC(O)(CCNC(=O)CC(C)C(F)F)C2)=O)c1 c1(C(=O)NC2(CNC(c3cnc(CCCC)s3)=O)CC2)cnn(CCC#N)c1C C12(CNC(c3cnccn3)=O)CCCCC1N(C(c1ncc(F)cc1F)=O)CC2 Cc1cc(C(c2nnnn2C)NCCOCC2CC2)cc(C)n1.C1CCOCC1 N1(C(c2nc(C)sc2Br)=O)CCC2(CCCCC2NC(C2CC23CC3)=O)C1 C1(COC)(CNC(C2(C)CCOC2)=O)CCCN1C(c1cccnc1S)=O C(=O)(CC(O)C(C)C)NCC(C)NC(=O)Cc1ccc(-n2cnnn2)cc1 C1(NC(C2CCN(C)C2)=O)(CF)CCN(C(=O)C=Cc2ncc[nH]2)C1 N1(CC(=C)C)C2CCC(C2)C1CNC(C1CCCC(C)C1)=O c1(C(N(CCCCNC(=O)CC2NC(=O)NC2=O)C)=O)ccn(CCO)c(=O)c1 c1(C(=O)NC2CC(NC(CCCc3scc(C)n3)=O)C2)cccc2nc[nH]c12 Cc1cccc(C(N2CCC(O)(CNC(=O)CCC3CCN(C)CC3)C2)=O)c1O N1(C(c2cc(CC)[nH]n2)=O)CCC2CN(C(c3c(C)nn(C)c3Cl)=O)CCC12 c1(C(=O)NC(C)C(C)NC(=O)CCc2cn[nH]c2)ccnc(N(C)C)c1 N1(C(N2CCC(=C)C2)=O)CCc2c(F)ccc(OC)c2C1 c1(OC)ccc(C(C)CNC(=O)Cc2nc(-c3ccc(C)s3)oc2C)cc1OC C1(C)(C(N2CCC(C(C(=O)NC(C3CCCC3)C#C)C)C2)=O)CNC(=O)C1 c1(NC(c2c(CNC(Cc3ccc(C)s3)=O)cco2)=O)ccc[n+]([O-])c1 c1(-c2ccc(OC)s2)cccc2c(C(N3CCC(OC)CC3)=O)[nH]nc12 c1(C(N2CCCCC(CNC(C3CC(O)C3)=O)C2)=O)ccc2ccc(Cl)cc2n1 c1(NC(c2cnn3c2CCC3)=O)ccc2occc2c1 c1(C(N2CCC(O)(C(C)CNC(C3(F)CC3)=O)C2)=O)cccc(F)c1N n1(CC(=O)NC2CC(NC(C3C(C(=O)OC)C3(C)C)=O)C2)nc(C)ccc1=O c1(CC)ccc(OC)c(CN2CC(C)CC2C(N2CCCC(O)C2C)=O)c1 c1(C(=O)NC2CC(C)(NC(CC(COC)C)=O)C2)ccc2c(c1)COC2 N1(C(CCC=C)=O)CCC(C)N(C(C2CCOC(CC)C2)=O)CC1 C1(C(=O)NCCOCCCNC(=O)OC(C)(C)C)CCCN1c1ccncn1 N1(C(CC=CC=C)=O)CCC(NC(=O)COc2ccon2)C(F)(F)CC1 CC1CC(CC(=O)NCCc2cn(C3CC3)cn2)CN1C(C1CCC1)=O C(=O)(C(C)(C)CS(N)(=O)=O)N(CC(C)N(C(C=Cc1ncc(C)[nH]1)=O)C)C C1(NC(=O)Cc2ccsc2)COC2(C1)CN(C(c1cc(Cl)ns1)=O)C2 C1(CC(=O)Nc2ccccc2SC2CCCCCC2)Oc2ccccc2NC1=O C1(C(=O)NCc2ncn(CC)n2)C2CC2CN1C(c1cc(Cl)no1)=O Cc1c(C(=O)NCCC(O)CNC(c2c[nH]nc2CCC(F)(F)F)=O)cnn1CC C(CN=c1cc(C)c(S(=O)(=O)NC2CN(C)CC2OC)c[nH]1)N(C(C)C)CC C12(CNC(CSCC)=O)CCC(CC1)N2C(C1CCC(F)(F)CC1)=O C1(OCC)CC(C(=O)NCCc2ncccc2Br)CN(C(=O)NC(C)(C)C)C1 c1(NC(C2SCCN(C(CNC(C)=O)=O)C2)=O)cccc(C2CC2)c1Cl c1(C(=O)NC(C(C)(C)C)c2cncs2)ccc(I)cc1F CC(C)CC(CC(=O)N(CC(C)C)C)NC(=O)CC1CCCCCC1 Cc1nn(CC(=O)NCC(CO)NC(=O)CN2CCC(O)CC2)c(C)c1Br c1(C(N2C(C)CN(Cc3nnsc3Cl)CC2)=O)ccc2cc[nH]c2n1 N1(C(c2cc(C)sn2)=O)CC=CCC1C(N1CCN(C(C)C)CC1)=O C12(C(=O)NC(CN(C(c3c(C)n(C)nc3)=O)C)C)CCCN1CCC2 C(=O)(C(C)CCC(C)(C)C)NCC1OCCN(C(c2c(C)cc[nH]c2=N)=O)C1 C1(C(=O)NC(C=C)CO)CCOCCN1C(=O)Cc1nocc1C C(=O)(C1=CC2CC(C1)CC2O)N1CC(COC)C(c2ccccc2)CC1 N1(C(C(C(C)(C)C)O)=O)CCOC2(C1)CN(C(=O)C(C)(C)Cc1cnn[nH]1)C2 C1(CNC(c2ccn(CCC)n2)=O)CN(C(=O)CCC2CCC(=O)NC2)CCO1 C1(NCC2CC(=C)C2)CCC(C)N(C(=O)Cn2nc(C)cc2C(F)F)C1 CC1(CNC(=O)CCN(C(=O)CC2OCCCO2)C2CC2)COCCO1 CCC(C)(C)C(=O)C(=O)N1CCC(C2CC2)C1C(=O)NCC(=O)OC(C)C CN1CCN(C(c2ccccc2Cl)=O)C(CNC(=O)CCCC(N)=O)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CCC(C)(CNC(c2c(CC)cccc2)=O)C1 N1(C(C(CC)n2nccc2C)=O)CCC(NC(=O)Cc2n[nH]c(C)n2)CC1C c1(CCC)cc(C(=O)N(C(C)C(=O)NCC2C=CCOC2)CCC)no1 C1(CNC(=O)C(CC2CC2)NC(=O)CC=C(Cl)Cl)CC12CC2(F)F c1(C(N2C(C(C)NC(CCN(CCCCC)C)=O)CCC2)=O)oc(SC)cc1C N1(C(C2CC(CC)C2)=O)CC2CCN(C(c3cccnc3S)=O)CC12 C1(CNC(CCC2CC(NC(c3c(OC)nccn3)=O)C2)=O)CC(=O)N(C)C1=O N1(C(C(=O)N(CCO)Cc2cc(CC)no2)=O)CCC(C)CC1 CC1(C(=O)NCCCCCCNC(c2cccc(C3CC3)c2)=O)CCCCCC1 N1(C(c2cnn(C(C)C)c2Cl)=O)CCCC(CNC(c2cc(C#N)c[nH]2)=O)CC1 N1(C(CN(C(=O)OC)C)=O)CC2=C(C1)CN(C(=O)CC1CCC(F)(F)CC1)C2 c1(OC)cc(-c2c(C(=O)Nc3c(C)ccnc3Br)cccc2F)c(OC(C)C)nn1 c1(C(N2CCOCC(NC(CCc3ccn(C)c3)=O)C2)=O)cc(S(C)(=O)=O)co1 c1(CC(=O)NC2(CNC(=O)Cn3nccn3)COC2)cccc(Br)c1 C1(F)(CNC(c2cncc(OC)n2)=O)CCN(CC2CCCC2)CC1 Cc1cc(CC(=O)NCCCC2CCCN2C(=O)CCCOCC2CC2)ccn1 N1(CC(=O)NC2C(SC)CN(C(=O)C(c3cccnc3)O)C2)CCCCS1(=O)=O C1(C(N2C(C)CC(F)C2)=O)CN(C(C2CCC(C)(C)OC2)=O)CC1(C)C c1(C(=O)OC(C)(C)C)ccc(F)c(OC(F)F)c1.C1(O)CCN(CC(=O)NC)CC1C C12(C(N3CC(N(C(=O)CCC4CCCC(=O)N4)C)C3)=O)CC=CC(C1)OC2 c1(C(N2CC(NC(C=CC(C)(C)C)=O)C(F)C2)=O)c[nH]c2c(Cl)cccc12 c1(NC(c2n(CC)nnn2)C2CC2C(F)(F)F)ccc(Br)c2c1CCC2 Cn1nc(C2CC2)nc1CC(=O)NCCC1(C)CCN(C(C2CCCCO2)=O)C1 CC1CC(NC(C2CC(N(C)C)C2)=O)CN1C(=O)Cc1cccc(O)c1 CC(N=[N+]=[N-])C(=O)N1C(C(=O)NC2CCC(O)CC2)CCC1C(C)C C(CC(C(C)(C)C)NC(c1c[nH]nc1C(F)F)=O)N(C(COC(C)=O)=O)C CP(C)(=O)C1CCC(NC(C2CCN(c3ccc(F)cc3)C2=O)=O)C1 c1(CCC(=O)NCC2(O)CC(NC(C(C)CO)=O)C2)cccc(C(F)(F)F)c1 c1(C(=O)NCC(C2CCCC2)NC(C2C(C=C)C2)=O)ccnc(COCC)c1 C=CCC(C)(CC)C(=O)N1CC2CC(NC(C3(SC)CCC3)=O)C(C2)C1 c1(C(=O)NC2C(NC(c3cccnn3)=O)C2)ccnc2c1CCC2 c1(C(=O)NCC(=O)NC2CCCC2NC(C2CCCCC2)=O)cc(O)cc(F)c1 c1(C(=O)NC2C3CCN(C(C4(C5CC5)CCCO4)=O)CC23)cc2ncccn2n1 C1(CCC(C2CC23CCC3)=O)CCCCC1NCCn1cc(CNC(N)=O)nn1 Cn1nccc(C(=O)NCC(CO)NC(C2(C)CS(=O)(=O)C2)=O)c1=O c1(NC2CC(=O)NC2)ncnc2c1ncn2C(c1ccc(OCCO)cc1)CO C1(NC(C2(CC)CCOC2)=O)CCN(C(c2cnc(C)nc2)=O)CC1(C)C C1(O)(C(C(=O)NCCOCC(N)=O)NC(C2C(OC)CC2)=O)CCCCC1 n1(CCC)ccc(C(=O)NCC2CCC(NC(=O)COCC(C)C)C2)n1 O=C(CCC1CCc2ccccc21)NCC12CC1CN(C(c1cocn1)=O)C2 N1(C(CN2CCC(C)(O)C2)=O)CCC2(CC(NC(=O)C3=C(Cl)CCCC3)C2)C1 n1(CCC=C(C)C)cc(C2CCCN2C(=O)C(CC)N(c2ccccc2)C)nn1 N1(C(C2(C#C)CCCCC2)=O)CCC(CNC(=O)C=CC(=O)N(C)C)C(F)(F)C1 c1(NC2C(C)(C)C(NC(c3cccc4ccsc34)=O)C2)ncnc(Cl)c1C#N C1(C(N2CC(C)OCC2)=O)C2C3CC4C1C2C34C(N1CCC(C#N)C1)=O c1(OC)cccc(NC(=O)C=CC(=O)NC(CNC(=O)C(O)C(C)C)C(C)C)c1 C(c1ccc(C(F)F)o1)=CC(=O)N(CC(C)NC(C1CCN(C)CC1)=O)C CC(=O)C(C)CC(C)C(=O)N1CCC(CC(=O)NCC(C)N(C)C)CC1 C1(NC(C(C)C)=O)(CNC(c2cnc3ccnn3c2)=O)CCC(C)(C)CC1 c1(OC)nc(N(C)C)ccc1NC(=O)Cc1ccc(Cl)c(F)c1 C(CC(C)(C)C(=O)NCCN(C)CCO)NC(C(C)NC(CC)=O)=O C(=O)(CC(CC)OC)NC(C(=O)NC(CCC=C)C)(C)C CCC(C)CCC(=O)N1CCCC(O)(CCNC(=O)CCc2cnn(C)c2)C1 c1(CNC(C(=O)NCc2onc(CC)c2C)C)c(OC)cc(OC)cc1OC CN1CC(C)(C)CC1C(N1CCC(Cn2cc(CCN3CCCCC3)nn2)C1)=O C=C1CC2CCC(C1)N2C(c1cnc(NC)s1)=O c1(C(N(C(CCNC(CSCC=C)=O)C)C)=O)cc(CC)ccc1Cl c1(CC)cc(C(N2CC(CO)C(C)(C)C2)C(=O)NCC(F)F)ccc1OC CN1CCCC(NC(=O)CC2CCN(C(=O)CC3CC=CCC3)C2(C)C)C1=O N1(C(C2C(CC)C2)=O)CCOC(C2CN(C(=O)Cc3cc(C)[nH]n3)C2)C1 c1(CNC(C(C)n2cccn2)=O)ccccc1CNC(=O)CC1CCC(=O)N1 N1(C(c2c(CC)occ2)=O)CC2CC1C2C(=O)NCCc1cccc(OC)c1 c1(NCC(C)Cc2cccnc2)ncccc1S(=O)(=O)NC1CC(C#N)C1 Cc1cc(C(=O)NC2CCC(N(C(=O)Cn3cccn3)C)C2)c(C)n1CC1CC1 c1(C(=O)Nc2cccnc2Cl)cnn2ccc(-c3cc(F)c(F)c(F)c3F)cc12 C(CCCC(=O)N(C)CCNC(=O)CCCSC(C)(C)C)OCC CN1CCC2(CCN(C(=O)CC3CC(C)(C)CN3C(=O)CCc3nncs3)C2)C1 C1(CC(=O)NC(CC)(C)CNC(=O)CC2CCN(C)C2C)CC(=O)NC(=O)C1 C(C(CC(C)C)NC(C1CCC(=O)NC1)=O)NC(C1(CCCC)CCCC1)=O c1(C(=O)NC2CCN(C(C3CCC4(CC4)C3)=O)C2)ccn2c(O)nnc2c1 C1(C(=O)NC(CC2CCOCC2)C(=O)N2CC(OCC(F)F)C2)CCCC(F)C1 N1(C(CCCOCCC)=O)CC2CC2(CNC(=O)CC2CCNC(=O)C2)C1 c1(C(=O)NC2C(NC(c3cnc(CC)[nH]3)=O)CCC2)ccc2c(c1)CCCO2 c1(C(=O)NCCCC(C)NC(c2nc(C)sc2)=O)cc2ccc(O)nc2s1 Cc1nc(Br)oc1C(=O)N(C1CCCC1)CCCNC(C1CCCCO1)=O C1(CNC(C(C(C)O)C)=O)CC(N=c2cc[nH]c(C#N)n2)C1 c1(C(N2CC(CNC(C(COC)(F)F)=O)C(C)C2)=O)cc(Cl)ccc1O C(=O)(CCS(N)(=O)=O)NCCCCCCN(C(=O)CC1CC1C1CC1)C N1(C(c2coc(C3CC3)c2)C(=O)NCc2cccs2)CCCC2CCC(O)CC12 Cc1c(-n2cc(CC3(F)CCCN(C(=O)OC(C)(C)C)C3)nn2)cccc1Br CCC(C)CCCCC(=O)N(CC(C)CNC(c1nn(C)cc1S(N)(=O)=O)=O)C N1(C(C2(c3cccc(F)c3)CCC2)=O)CCCNC(=O)C12CCC2 N1(C(C2C(C)(C(C)C)C2)=O)C2CCC1C(CNC(=O)C(C)n1cncn1)C2 C1(CNC(c2ccc(F)s2)=O)CN(C(=O)C(F)CC2CCC2)C2(CCC2)C1 Cc1cnc(C(=O)NC2CCCC(CN(C(=O)CCCn3cccc3)C)C2)cn1 C1(CC(=O)N(CCNC(c2cc(COC)sc2)=O)C(C)C)CCCC1(F)F N1(C(C(C(C)(C)C)O)=O)CCC2CN(C(c3cc(Br)ncc3Cl)=O)CC2C1 C1(CC=C)(NC(c2scnc2CC)=O)CN(C(c2n[nH]c(C)n2)=O)C1 N1(C(C(CCC2CC2)NC(C(COCC)C)=O)=O)CCC(F)(F)C(F)C1 C1(CNC(C(CC=C)OC)=O)CC2(C1)CN(C(=O)CCCCCC)C2 CCC(C)C(O)C(=O)N1CC(n2cc(CNC(=O)Cc3cncc(O)c3)nn2)C1 N1(C(c2[nH]c(=N)sc2)=O)CCCN(C(c2cccc3c2OCC3)=O)CCC1 Cc1c(CC(=O)N(CCC(C(C)C)NC(=O)CCC2CCCO2)C)cnn1C CN1CCC(O)(CNC(=O)COCCNC(C2CCOC2)=O)CC1 C12(C(=O)NCC3C(C)OCC3)CCCC1CN(C(=O)CC1CCCO1)C2 c1(C(=O)NCC(CNC(C=CC=CCCCCC)=O)O)cc(F)cc2cnccc12 C1(CNC(C2(CC=C)CCN(C(c3ccncc3F)=O)C2)=O)CC(O)C12CCC2 c1(C(N2CC3C(NC(C(C)n4cccn4)=O)C3C2)=O)ccc(C#N)cc1Br CCC(CNC(=O)CC1CC2(CCC2)C1)(CC)C(=O)N1CCC(F)C1 C(=O)(CC(C)(C)C(=O)N1CCCC(C(C)(O)CNC(c2cnnn2C)=O)C1)OC N1(C(C)=O)CC2C(COC(=O)NC(=O)CCc3ccccn3)C2C1 c1(C(N2CCC(N3CCCC(COC)C3)CC2)=O)cc2c(s1)CN(C)CC2 c1(NC(C(N2CCCCC(C)C2)C=C)=O)c(C)cccc1C C1(C(=O)N(CC(=O)NCC#CCOC)CC2CC2)C2(CC2)C12CC2 N1(C(C2(CC)COC2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1CO N(C(=N)N1CC(O)CC(C)(C)C1)Cc1c(C(F)(F)F)nn(C)c1CC1CC1 C=CCCCCCCC(=O)N(CC(C)(C)CNC(C1(F)CCS(=O)(=O)C1)=O)C C(=O)(C1=CN(C(=O)OC(C)(C)C)CCC1)N1CC2C(NC(CSCC)=O)C(C2)C1 N1(CCCCC)CCN(c2nnc(C(C(C)C)SC)n2CCC2CCOC2)CC1 c1(C(=O)NCC2CCN(C(CCCC(C)=O)=O)C23CC3)ccc(S(C)=O)cc1 N1(C(C2C(C)CC=CC2)=O)C2CCCC1CN(C(C13CCC(C)(CC1)OC3)=O)C2 C1(C(=O)NC(C2CN(c3ccnc(Cl)n3)C2)C)Cc2cc(F)ccc2O1 C(C)(CCC(=O)NCCN1CCC(NC(C2C(C)C2(F)F)=O)CC1)OCC C(=O)(C(F)CC(C)C)N1C(CC)C(NC(=O)COCCF)CC1 c1(NC(CCC=C)c2nnnn2C(C)(C)C)ccc(Cl)c(OC)c1 N(C1CCCc2ccoc21)C(c1n(CCCOC)nnn1)c1cnn(C)c1 CC1(C)CC(C(=O)NCCCCC2CC2)CCN1C(=O)CCCOc1ccccc1 N1(C(CC2CC(C(=O)OC)C2)=O)CCCC1CNC(c1scnc1C)=O CC1CN(C(=O)C=CCF)CC1CNC(=O)CCC1CCC(=O)C1 C1(C(C)(C)O)(CNC(C2CCCN2C)=O)CN(C(=O)C(C2CCCCC2)O)C1 CC(C)C(CCNC(=O)C(C)(C)C1CC1)NC(c1ncoc1-c1ccco1)=O C12(C(N(C)CC3N(C(C=C(C)C4CC4)=O)CCCC3)=O)CCC(C1)C2(C)C C1(NC(C(C)CN(C)C)=O)CCC12CN(C(=O)CSc1cccc(F)c1)C2 Cc1cc(-c2nc(CCN(C)C)no2)ccc1CSc1cccc(I)c1 C(C(=O)NNC(=O)c1ccccc1Cl)Nc1cc(SCC)ncc1 N(C1CN(C(=O)C(F)C2CCC2)CCc2ccccc21)C(C(C(CC)C)O)=O C(=O)(CCCCCCSC)NC1CCN(C(c2ccn(COC)n2)=O)C(C)C1 S(=O)(=O)(c1ccc(NCC2CCC(F)(F)C2)c(Cl)c1)N1CC(CO)CC(C)(C)C1 C1(C(=O)NCC(C2CCC2)NC(C2(CC#C)CCCC2)=O)CCOC1C=C C(C)(C(=O)N(CC1CC1)OC)NC(C(C)NC(CC)=O)=O c1(C(=O)NC(C(=O)NC(C=C)C)CC2CCC2)cnc(O)n1CC C(CC(=O)NC(C)(CNC(=O)CCc1ccc[nH]1)C1CCC1)OC(C)C c1(C(NOCC(=O)NCC2CC(O)C(O)C2)=O)ccc2[nH]nc(Cl)c2c1 c1(C(N(C2CCN(C(C3C(OC)C3)=O)CC2)CCO)=O)cc(Cl)cc(F)c1F c1(OC)cc(F)ccc1OC(=O)CC1CCC(=O)NC1=O C1(C)(COC)CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CN(C)C(C)C)C1 CCC(CC(F)(F)F)C(=O)N1CCN(C(c2cnc(C#N)s2)=O)CC1COC c1(C(N(CCOCCN(C(=O)COCC(C)(C)C)C)C)=O)ccnn1C1CC1 N1(CC(C2CCC2)OC)CCC(NC(=O)Cc2ccccc2F)CC(C)(C)C1 C1(NC(c2nc(C)c(C)s2)=O)CC2CCC(C1C)N2C(=O)CN1CC2CC2C1 CC(C)CC(C)(C)C(=O)NC(C)Cc1ccc(CNC(C2(C)CC2)=O)cc1 C(=O)(CCCCC(F)F)NC1CCCN(C(C2(CC(C)C)CCNC2=O)=O)CC1 c1(C(N2C(CN(C(C(C)OCC#C)=O)CC)CCC2)=O)ccc(O)cc1C Cc1c(C(N2CC(NC(=O)CC3CC4CC4C3)CC2CO)=O)cnn1CCO C=CCC(C)(C)CC(=O)NC1CC2CC1N(C(=O)Cc1cccc(C(C)C)c1)C2 CC1CCN(C(C2CC(C3CC3)C2)=O)C(C(=O)NCCCC2CCOC2)C1 N1(C(C2N(C(=O)OC)CCC2)=O)CC2CC(C1)N(C(=O)CCN(C)CCO)C2 c1(C(N2CCSC(COc3ccccc3)C2)C(=O)NC)ccc2cccnc2c1 C(N=c1[nH]c(=NCCCC(C)C)[nH]c2c1CCC2)c1cccc(OC)c1 C1(C(=O)NC2C(NC(C(C)(C)OC(C)C)=O)CCC2)CCC(C)CC1 N12CCC3CN(CC13)C(=O)COCC2=O.c1(Oc2ccc(C)s2)ccc(Cl)cn1 c1(N(C(c2c(C)c(Cl)c(Cl)cc2)=O)CC2CCCNC2)[nH]cnc2nc(Br)cc1-2 N1(CC(=O)NCc2cccc(OCCC)c2)CCc2c(CC)cccc21 C(C(O)CF)N(C(C(C)N(C(=O)CSCC(F)F)CC)=O)C CC(=Cn1ccnn1)C(=O)N1CC(F)CC1CNC(=O)C(C)n1ccnc1 CC(C)S(=O)(=O)C1CCN(c2ncnc3c2ncn3C(c2n[nH]c(=N)s2)(C)C)C1 c1(CC)cc(NC(=O)C(C2CC=CCC2)NC(=O)C(O)C(F)(F)F)cc(O)c1 c1(C(N2CCC(CN(C(CCc3cc(C)no3)=O)C)C2)=O)ccc(C)c(C)c1F C1(C2CC2)(C(=O)Nc2c(N3CCCC(C)(C)C3)cccc2)CCOCC1 c1(C(=O)NC2CCCN(C(c3ccnnc3)=O)C2)cc(OC(F)(F)F)ccc1O C1(NC(C=CC(CC)=CC)=O)CCN(C(C2CC(=O)N(C(C)CC)C2)=O)CC1O c1(C(=O)NC2C(CC)CN(C(=O)C3CC3)CC2)ccc2n[nH]cc2c1F c1(NC(=O)NC(CCOC)C)c(F)c(Br)c(F)c(Br)c1F C(C(O)C(=O)NC(C)(C)CCNC(C1CCN1S(C)(=O)=O)=O)SC N1(C(c2c(C)csn2)=O)CCN(C(C)CNC(=O)C(c2cncn2C)O)CC1 Cc1ccc(C(=O)NC(C)(C)CCCNC(C2CCCCC2C)=O)c(=O)n1C c1(CC(N2CCC(NC(C(C)SC(C)C)=O)C2C)=O)cc(F)c(F)cc1F C1(OC)CC(NC(=NCc2ccnn2C(F)(F)F)NC2CCC2)C12CCC2 Cc1ccnc2nc(C(=O)NC(C)CCNC(c3cc4ccsc4[nH]3)=O)nn12 N1(C(C=C(C)c2cccs2)=O)CCC2(C1)CN(C(C1CC(S(N)(=O)=O)C1)=O)C2 CCCCC(CCCC)NC(=O)CCCCCNC(C1(CF)CC1)=O C1(C(=O)NC2C3(CN(C(CC(CC)(C)C)=O)C3)CC2)CC2CCCC(C1)C2(F)F c1(C(=O)NC(C2(C(N3CCCCC3C3CC3)=O)CC2)C)cc2cc[nH]c2cn1 C(CC)(C(=O)N1CCC1CC(=O)N(CCCCO)C1CC1)=CC N1(C(c2nc(C)sc2)=O)CCCCC(N(C)C(C2CC(N3CCCC3)C2)=O)C1 CCCCN=C(NCc1c(OC)cccc1C)NC1CC(OC(C)(C)C)C1 N1(C(C(CC(C)C)(C)C)=O)CCC2(COCC(CNC(=O)CCN(C)CCO)O2)C1 C1(CCOC)(NC(=O)CN(C)C(C)C)CCN(C(=O)CC2(OC)CCCC2)C1 c1(C(C)C)nnc(C(=O)NC(C2CCCN2C(C2CC(=O)N2)=O)(C)C)s1.C1CC1 N1(CCCCSCC)CC(C)OC(C)C1.c1(C(C(=O)CN)C)c(Cl)cccc1Cl C1(NC(C2Cc3c(C)ncnc3CC2)=O)CCN(C2CCc3c(F)cc(F)cc32)CC1 C1(CNC(c2ccc(OC)nn2)=O)CN(C)CCN1C(C1CCN1C(C)(C)C)=O c1(OCCCCCC)ccc(CNC(=O)CC2(Cc3ccccc3)COC2)cn1 S(=O)(=O)(c1[nH]c(=NCC2(C(F)(F)F)CC2)ccc1Br)NCCC1(OC)CCC1 CCC(C)C(O)C(C)C(=O)NCCOCCC(=O)NC1COCCC1O C(=O)(C(=O)C(C)(C)C)NCC1(CNC(C(CC)F)=O)CCCCC1 C1(NC(=O)OCC)CCN(C(C2CCN(C(C3CC(C)(CC)C3)=O)C2)=O)C1 C(=O)(C1=CCCN(Cc2c[nH]nc2-c2ccccc2)C1)NCc1nc(C)sc1 Cn1ncc(C(N2CC(NC(C3CCCCC3)=O)C3(CCC3)C2)=O)c1S(N)(=O)=O c1(NC(C(N2CCC(c3nc(C)[nH]n3)C2)=O)=O)ccc(Cl)c(F)c1 CCCCCCCC(=O)NC1CCCC(C(N2CCCC(O)CC2)=O)CC1 C12(C(=O)NC3(CC(=O)OCC)CC3)CCN(C(c3cnncc3C)=O)CCC1C2 C1(C(=O)N(CCCNC(c2ccc(CN3CCCC3)o2)=O)C)(CC)CC(C)(C)C1 N1(C(c2c(Cl)ccc(OCC)n2)=O)CCC2(CCCN(C(c3cocn3)=O)C2)C1 CC(C)(C(=O)N(C1CCN(C(=O)Cn2cc(N)cn2)C1)CCO)c1ccccc1 c1(NC(C2N(Cc3cc(OC)c(Cl)cc3)CCC(F)C2)=O)cccc2c1OCO2 CC1CN(C(C2(O)CCC2)=O)CC1NC(c1ccccc1CC(C)(C)C)=O c1(-c2cn(CC3N(C(C4(C)ON=C(C)C4)=O)CCC3)nn2)cc(F)cc(F)c1 N1(C(CCCC(=O)OCC)=O)CCC(CNC(=O)CCC(C)(C)F)C(F)(F)CC1 N1(C(C=C(C)C2CC2)=O)Cc2n[nH]cc2C1C(=O)N(C)CC1CCCN1C C1(C(N(C2CCCN(C(=O)CCNc3cncnc3)C2)C)=O)CCNC(=O)C1 c1(CC(=O)NCC(CN(C(C(C2CCOCC2)C)=O)C)O)ccc(F)cc1 C1(NC(CCCC=C)=O)CCC2(CC1)CC2NC(c1ccnc(CN(C)C)c1)=O CCC(CC(C)C)C(=O)NCc1ccoc1C(=O)NCCSCC(C)C c1(SC)nc(Cl)cc(=NC2(CNC(=O)CNC(C3CCC3)=O)CCCC2)[nH]1 n1(CC(=O)Nc2cc(Br)nn2C2CCCCO2)c(C2CC2)nc2ccccc12 C1(NC2CC(C)(F)C2)CCN(C(=O)CCP(C)(C)=O)C(C)(C)C1.C1C(=O)N1C c1(C(N2CCC3CN(C(C4(CF)CCC4)=O)CC23)=O)ncc2n1CCCC2 Cc1ncc(C(=O)NCC2(CCNC(c3cc(F)cc(Cl)c3)=O)CC2)cc1N N1(C(c2cnc(C(C)C)s2)=O)CCC(C)(NC(=O)C(C)OC2COC2)C1 C1(NC(C(CSC)O)=O)CN(C(C2(NC(N)=O)CC2)=O)CC2(CCOCC2)C1 C(=O)(CCCC(=O)NC(C(=O)NCC#CCCO)C(C)O)OCC N1(C(c2nc(C)n(C)c2)=O)CCC(C)C(NC(=O)CN2CC(F)(F)C2)C1 c1(N(C(CC)C)C)ccc2c(C)nn(C3CCc4ccccc43)c2n1 CCCCC(CNC(=O)CC1C(=O)NN=C1C)NC(=O)C(C)=CC(C)(C)C N1(CC(n2cc(-c3nccnc3C(=O)N(C)C)nn2)C)CCC(C)C(F)(F)CC1 N1(C(CC2(OC)COC2)=O)CCOCC1CNC(c1cnc(C)[nH]1)=O CC(C(=O)N(C1CCCC1)CCNC(=O)CCCc1ccccc1)C(F)F C1(C(=O)NCC2CC(NC(C3(C)CNC(=O)C3)=O)C2)COCCN1C=O c1(C(=O)NCC2CCC(NC(COCCCC(C)C)=O)C2)ccc2n[nH]cc2c1 c1(NC(CNC(C2CCN(C(c3n[nH]c(C)c3C)=O)C2)C)=O)cc(O)nc(O)n1 c1(CN(C(Cc2c(C)cccc2)C)C)ccc(Cl)nc1C C1(C(N(CCCCNC(CC(C=C)(C)C)=O)C)=O)CCS(=O)(=O)C12CCC2 C12(NC(CC)=O)CCCC1CN(C(c1n[nH]cc1Cl)=O)C2 C=CC1CN(C(=O)CCc2n[nH]c(=N)s2)CC1NC(=O)C(C)CC(N)=O CC1=C(C(=O)NC(C)(CNC(=O)CC2CCOC2(C)C)CO)C(C)(C)CCC1 c1(C(CNC(C=CC(CC)C)=O)NC(=O)CCCN(C)C)ccccc1 c1(OC)ccc(C(N2CCCC(n3ccnn3)CC2)=O)cc1OC(F)F C1(CCC(=O)NCCCNC(C)=O)CCN(C(=O)CCc2ccc(F)cc2)CC1 N1(C(CC(C(C)C)C)=O)CCOC2(CCN(C(=O)CCN3CCOCC3)CC2)C1 c1(C(=O)NCC2(C)CCN(C(c3cc(Cl)no3)=O)C2)cc(CN)nnc1O C1(F)(CNC(=O)Cc2cn[nH]c2)CCN(C(=O)COc2cncc(Cl)n2)CC1 C(=O)(C1=NN(C)C(=O)CC1)NC12C(CN(C(CCc3c(C)noc3)=O)C1)CCC2 c1(C(=O)NCCc2ncc(C)cn2)n[nH]c2c1CN(C(C1(O)CC1)=O)C2 Cc1c(N)ccc(C(=O)NCC2(NC(=O)Cn3ncn(C)c3=O)CCC2)c1C N1(C(C2C(C)(CC)C2)=O)CCC12CN(C(=O)CCc1ccccc1OC)C2 CC(C)(CO)C(=O)NC1CC(NC(C2CCCN2C(=O)C(F)(F)F)=O)C1 C(C)(C(O)C(F)F)NC(CC1N(C(CCSCC)=O)CCC1)=O CON(Cc1ccco1)C(=O)CC1CCCN1C(c1coc(C(C)C)n1)=O C=CCCC(C)C(c1nnnn1C1(C)CC1)NCCCn1ccnn1 C(=O)(C(O)CC(C)(C)C)NCC(C)(C1CCC1)NC(c1c(C)cccn1)=O c1(C(N2CC(O)(CCNC(C(C)n3ccnc3)=O)C2)=O)ccnc2[nH]ncc12 c1(NC(N(C2CCCC(SCC)C2)C)=O)ccc(S(=O)(=O)NC(C)(C)C)nc1 CCCCC(CC)C(=O)NCC1C2CCC(C2)N1C(=O)COC1CCOC1 n1(C(CC)C)nccc1C(c1nnnn1C(C)(C)C)NCCCc1cncnc1 N1(C(c2c3ccc(C)cc3[nH]n2)=O)CCC(NC(C2(F)CCCC2)=O)C(C)(C)C1 CN1CCC(C)(CNC(C2(NC(=O)Cn3cnnc3)CCOCC2)=O)C1 CCCC(C#N)C(=O)NC(C)(C)C(C)NC(c1ccccc1NC)=O CCCC(CC(C)C)C(=O)NC1(CNC(=O)CS(=O)(=O)CCO)CCC1 N1(C(CC=CC=C)=O)CCCC(C(C)NC(=O)CN(C2CCCCC2)C)C1 C(CCC)(C(=O)NC1CN(C(=O)CCN2CCC(C)CC2)C2CC12)=CCC Cn1cnc2c1CCCC2C(=O)NCC1CN(C(C2CCCCO2)=O)C1 C(N=c1nc(-c2ccc(Cl)c(Cl)c2)o[nH]1)c1ccc(=N)[nH]c1 C1(CC(N2CCC(C)(COC)C2)=O)CCCN(C(=O)C(O)CC(N)=O)CC1 c1(CC(=O)NC(CNC(c2c(CC)c[nH]n2)=O)C(C)(C)C)cccc(F)c1F c1(NC(CCc2onc(C(C)OCC)n2)=O)ccc(C)c(CN)c1 C1(NC(CCC=C(C)C)=O)CC(C(=O)Nc2cn(C)nc2O)C12CCC2 c1(C(C)C)ccc(S(=O)(=O)NC2(CO)CCOC2)cc1 C1(C(=O)NC2(C)CCCN(C(COCCCCC)=O)C2)CCC12CCOCC2 C1(NC(C(COC)O)=O)CC2CCC(C1)N2C(c1ccccc1SC(F)(F)F)=O N1(C(C(=O)NCCSC)c2ccon2)CCCC(c2ccnn2C)CC1 c1(C(=O)Nc2nc(-c3ccnnc3)cs2)c(F)cccc1Br c1(C(N(C2CCN(C(C(C)OC3CCCC3)=O)C2)C)=O)cccc(CO)c1 c1(C(N(CCOC)CCNC(C2(SC)CC2)=O)=O)ccc(-n2ccnn2)cc1 Cn1c(=O)c2nc(C3CCN(CCC4(C)CCS(=O)(=O)C4)CC3)[nH]c2n(C)c1=O N1(C(=O)CC2CCCO2)CCC2C(C1)CN2C(=O)CN1CCCCC1=O c1(C(=O)NC2CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)c(F)cc(F)cc1Cl C(=O)(CC(C)(C)N(C)C(c1cccc(Cn2ccnn2)c1)=O)NC N1(C(Cc2cccc(C)c2)=O)CCC2C(CCN2C(c2cnn(C)c2C#N)=O)C1 Cc1nc2ccc(C(=O)NC3CC(F)(CNC(C4(N(C)C)CCC4)=O)C3)cn2n1 C(=O)(C1=CCCSC1)N(C)CC1CCCN(C(c2ccnn2CCC(F)(F)F)=O)C1 c1(C(=O)NCC2(F)CC(NC(C3CC3c3ccsc3)=O)C2)cc(F)cc(Cl)c1O C1(C(N2C(CCNC(CCCSC)=O)CSCC2)=O)CCCC2CCCN12 N1(C(C(F)OC)=O)CCC(CNC(=O)C(F)(F)C2CC2)C(C)C1 C1(c2n(CCOC)nnn2)(NCc2nc(COC)sc2Br)CCCC1OC N1(CCC(=O)NC2CN(C(C(CC)C)=O)C2)CCOCC1=O C1(CNC(C2OCC(C)C2)=O)CN(c2ncc3c(ncn3C)n2)CCC12CCC2 c1(N2CC3C(C)C3C2)ncc(S(=O)(=O)NC2CC2)cc1Cl.CCS(=O)CC(F)(F)F C12(CNC(c3cc(C)c(Cl)s3)=O)CCC1CCN2C(=O)Cc1cn[nH]c1 c1(CC(=O)NCC2(C(N3C(COCC)CCC3)=O)CC2)c(C)noc1Cl Cc1ncccc1C(=O)N(CCNC(=O)CCC1CCCCO1)C1CC1 CC(C)CC(C(=O)NCC1CN(C(c2nnc3ccccn23)=O)C1)C(N)=O c1(CNC(=O)NCCCCSC)ccc(-c2noc(C)n2)cc1 C1(C(N2CC(O)(CNC(C(CC)Nc3ccccc3)=O)C2)=O)CCCC(C)(C)O1 N1(C(C2CC(C(C)C)C2)=O)CCC(C(=O)NCC2(C)CCOC2)=C(F)C1 CC1CCCN1CC(=O)NC12CC(C(=O)NC3CCNC3=O)(C1)C2 N1(C(c2ccc(CCC)[nH]2)=O)CCN(C(C2CCOC2CC)=O)C(C2CC2)C1 C12(NC(C(C)SC(F)(F)F)=O)COC(CNC(C3CC(O)CN3C)=O)(C1)C2 C1(C(=O)NC(CCNC(c2c(C)[nH]nc2Cl)=O)(C)C)CC2(CCC2)CO1 C12(C(N3CC(NC(C(CC)n4ccnc4)=O)C3)=O)CCCC1C2(F)F c1(C(=O)NCC(CNC(c2n(CCC)ccc2)=O)OC)ccc(OC)cc1O C1(C)(CNC(C(CC)Oc2ccccc2)=O)CCN(C(c2csc(O)n2)=O)CC1 C1(C(=O)N(C2CC(C)(C)C2)C)(CC)CCCN1C(C1COC(=O)N1)=O Cc1nc(S(=O)(=O)NC2CNC3(CCC3)C2)nn1-c1ccc(F)cc1 C1(C(N(C2C(C)CC2)C)=O)CCC(C)CN1C(c1cccn1C)=O CN1CCC(CCN2C(=O)CN(CC(=O)N(C(C)(C)C)C3CC3)C2=O)CC1=O N1(C(C(CC)(C)OC)=O)CCC(C2(NC(c3cnc(Cl)c(Cl)c3)=O)CC2)CC1 C1(NC(COC(C)C)=O)CCN(C(c2cccnc2SC(F)F)=O)CC1C(C)C N1(C(C2C(=C)C2)=O)CCC2(CC(NC(c3ccc(F)c(C(F)(F)F)c3)=O)C2)C1 Cc1[nH]c(C)c(C(=O)NCC(C)(CO)NC(=O)C(O)C(C)C)c1C N1(C(C2C(C(=O)OC)C2(F)F)=O)CC(C)(C)CC1CNC(=O)CSC(F)F c1(C2CC(C(=O)NC(CCOC)CNC(=O)C(C)=C(C)C)C2)ccc(Br)cc1 C(=O)(CC1=NN(C)C(=O)C1)NCC1(CC2C(CC(=O)N(CCOC)C)C2)CC1 C(CCC(C)(C)C(=O)NC(CCO)C(F)F)NC(C(C)Cn1ccnc1)=O c1(C(=O)NC2CN(C(C(C)(C)CC3CC3)=O)CC2F)ccc(C2CC2)cc1F CCCCS(=O)(=O)NC(C)C(=O)NCC1CCCN1C(C1(CSC)CC1)=O c1(N(CCC)CCNC(c2cncc(F)c2)=O)ccc([N+](=O)[O-])c(SC)c1 c1(CCN2CCN(CCNC3N(CC)CCC3)CC2)c(C)nc2ncnn2c1C C1(NC(C(C=C)C)=O)CN(C(=O)C(C)(C)COC(C)C)CC1CO CCCCCCC(CC)C(=O)NCCCCCNC(=O)C(O)CN(C)C C12(CC)CCC(C(=O)NC3(C4CCN(C(=O)C5=NOCC5)C4)CC3)(CC1)CO2 CCCCCC(C)CC(=O)N1CCC(CCNC(C)=O)(NC(c2scnc2C)=O)C1 Cc1cc(C#N)cc(C)c1-c1noc(C(C)NCCCCS(C)=O)n1 c1(C(=O)NCCNC(c2ccoc2I)=O)ccc(F)cc1F C1(CC=C)(NC(=O)Cn2cnc(Br)c2)CCCN(C(=O)C(COC)OC)C1 c1(C(C(=O)NCC(F)F)N(CCCC)C)cn2c(F)cccc2n1 c1(C(C)C)ccc(F)c(C(=O)NCC2CC(F)CN2C(c2ccc(N)cc2)=O)c1 c1(C(N2CC3C(CNC(CN(CC)CC)=O)(C3)C2)=O)ccc(C)cc1OC c1(C(CN(CCCC)CCC)O)ccccc1C N(C(=NCC1CC1)NCCc1ccco1)CC1N(CC)CCC1 CCC(C(=O)NCC(CNC(=O)CC1CCN(C)CC1)OC)C(C)(F)F c1(CCC)nccc(N2CCCC2C(=O)NC(CC(C)C)c2ccccc2)n1 c1(C(=O)NCC(CC=C)NC(c2ccc(OC)c(F)c2)=O)cc(C)c(CC)cn1 CCC(CNC(C1CC=CCC1)=O)(CC)N=c1[nH]ncs1 c1(OC)cc(CO)ccc1NC(=O)CC1CCCN1Cc1ccc[nH]1 Cc1nc(S)sc1CC(=O)NC1COCCC1NC(=O)C=CBr O=C(O)CN1C(=O)COc2ccccc21.C(C1OCCc2sc(F)cc21)CC(N)=N N1(C(C2(CC)CC(C)(C)C2)=O)CCN(C(c2coc(CO)c2)=O)C(C(C)(C)C)C1 N1(C2C(NC(CN(CCOC)C)=O)COC2)CCN(C(=O)Cc2cn[nH]c2)CC1 c1(NC)ccc(-c2ccc(CNC(C3CCOC3)=O)c(F)c2)cc1F.c12cn-1nn2 c1(NCC(C2CCCC2)NC(C(C)(C)CF)=O)ncnc2[nH]cnc12 C1(CNN2C(=O)CCC2C(N2CCOCC2)=O)CCC(=O)NC1c1ccnn1C C1(C2N(C(c3c(CC)n[nH]c3)=O)CCC2)CCN(C(=O)C(C(C)C)OC)CC1 C1(C(=O)NC(CCC)C(=O)NCCC2COCC2O)CCn2nccc2C1 C12(CNC(C(CCOC)NC(C3ON=C(CC)C3)=O)=O)CCCC1OCC2 CCC(C(=O)NC(C(=O)NC1(C)CCSC1)C(C)OC)C(C)(C)CC CCC(CC)CCCC(=O)NC(CO)C(=O)NC1(C2CCCO2)CC1 N1(C(CNC(CC)=O)=O)CCC2CCN(C(=O)COc3ccc(F)cn3)C2C1 Cc1cccc(C(=O)NC(Cc2ccco2)C(=O)NCCCCO)c1N Cn1cc(F)c(C2CCN(C34CCC(C3)NC4)CC2)n1 N1(C(CC(C)SC)=O)CCC(C2CCN(C(=O)CC(C)CC(C)C)CC2)C1 Cc1cc(=NC(=O)C2CN(Cc3ccc(Br)s3)CCS2)[nH]c(C)c1C#N C1(C(C(=O)NCCOCC)N(CCC(F)(F)F)Cn2ccnc2)C2COCC12 c1(C(=O)NC(C(C)NC(C2CCC(F)(F)C2)=O)(C)C)cc(Cl)c2c(c1)OCO2 C12(CNC(C(C)CN(C)C(c3cnn(C)n3)=O)=O)CCCC(CO1)C2 c1(C(C)NC(=O)CCC2CCC(NC(=O)C(C)(C)n3cncn3)C2)cccnc1F C(CN=C(NCC(C)(C)SC)N1CCC2OCCCC2C1)OCC Cc1cc(-c2noc(-c3cc(Br)cs3)n2)c(C)o1 C(=O)(CC1=CCN(C(=O)CS(=O)(=O)CC)CC1)NCC1(CC)CCCC1 C1(NC(c2c(CC)scc2)=O)CCCN(C(C2(C)CCCC2)=O)C1 c1(C(=O)NC2(C3CCCN3C(C3CC34CCC4)=O)CC2)cc(C2CC2)ccc1Cl C1(CN(C(C(F)=CCC)=O)C)CCCC(NC(c2cc(C3CCC3)nn2C)=O)C1 c1(C(=O)NC2(CCCC(N3CC(CO)C(O)C3)=O)CCC2)occ2c1CCC2 N1(CN2CCC(N(S(C)(=O)=O)C)C2)C(=O)NC(Cc2ccsc2)C1=O c1(C(=O)NC2C(C)(C)C(CNC(c3csc(Cl)n3)=O)C2)csc(=NC2CC2)[nH]1 CCC(CC)C(CNC(c1cc(C2CC2)[nH]c1C1CC1)=O)CO N1(C(=O)CCC2CCOCC2)CC=C(C(=O)N2CCC(O)CC2C2CC2)CC1 C(=O)(CC1=CCCCC1)N1CCCC(NC(CCC2CCC(C)O2)=O)(CO)C1 c1(C(N(C2CN(C(=O)C=C3CCOCC3)C2)C)=O)c(Br)ccc(F)c1N N1(C(c2c(CC)noc2)=O)CCC(C)(C)C(C(=O)NCCc2c(C)n[nH]c2C)C1 CCC(CC)CC(=O)NCCN(C(=O)CC1(O)CCCOC1)CCOCCO Cc1n[nH]c2cc(C(N3CCC(CNC(C4(F)CC=CCC4)=O)CC3)=O)ncc12 C1(CNC(C2CC(C)(C)O2)=O)CCCCN1C(=O)CSCc1ccccc1 N1(C(CC2(CNC(c3c(C)scn3)=O)CC2)=O)CCC2CN(C)CC2C1 C(CCC(=O)N1CC(N(C(=O)C(C)=CC2CC2)C)C1)OCC=C c1(CCC)nc(C(=O)NCC(C2CCC2)NC(C2C(C(F)F)C2(C)C)=O)co1 c1(C(C)NC(C23CC2CN(Cc2cnn(C)c2Cl)C3)=O)cc(Cl)ccc1O C1(C(=O)OC)(NC(=O)C(C)C2CCCC2)CCN(CC(=O)NCC2CCCC2)CC1 N1(C(CC(C=C)C)=O)CC2CCC(NC(=O)C=C3CCCCC3)(C2)C1 C(=O)(CC(F)(F)C(F)F)NCCC1(C(=O)NCC(CC)OC(C)=O)CCC1 N1(C(C(C(C)O)N(C)C)=O)CC(C)OC2(CCN(C(C3(F)CCCC3)=O)CC2)C1 N1(C(C(NOC)=O)=O)CC2CC(C(N3CC(OCC(C)C)C3)=O)C(C2)C1 c1(C(C(=O)NCCOCCN(C(COC(CC)C)=O)C)C)ccncc1C C1(NC(C(CCC)OC)=O)CN(C(=O)COC(F)F)C2CCCCC12 C1CCCCNCCCN1C.C(=O)(C(C)N1CCC1)N1C(C)C1.C(C)(C)C C(CC(C)C(=O)N1CCOC(C(=O)NCC(O)C(C)(C)O)C1)=CCC CC(C)(C)CC(F)C(=O)NCc1ccc(C(=O)NCCC2CCCC3CC23)cn1 C12(CNC(c3cnn(C4CCCC4)c3)=O)CC1CN(C(=O)Cc1nncs1)C2 N1(c2n(C)ncn2)CCn2ncc(S(C)(=O)=NC(=O)Cc3ccco3)c2C1 c1(C(N2C(C)C(NC(=O)CNC(c3ccco3)=O)CC2)=O)cccc(F)c1F c1(C(=O)NCC(CO)NC(COc2c(CC)cccc2)=O)cc2cscc2s1 C1(COC)CC(O)CN1C(=O)C(N1CCC(O)CC1)C.c1(SC)ccccc1 CCCC(C(=O)NCCN(C(=O)C(C(C)C)n1cccc1)C)c1ccc(Cl)cc1 c1(C(=O)NCC(CC)NC(=O)C(C)(F)CC)cc(OC)cc(C(F)F)c1 c1(SCC(=O)NC2CCC(N(C)C(c3sccc3F)=O)C2)ncnc2[nH]cnc12 C(=O)(C(CNC(C1(NC(C)=O)CCC1)=O)CC(C)C)NC(CC)C1CCC1 C1(NC(CN2CCN(C)CC2)=O)CC2CC(NC(=O)Cc3nn(C)cc3Cl)CC12 n12cnc(c1)NC(=O)C1(CC1)C(=O)NCC2.C12CCCC1C2.CSC N1(CCCC=C)CCC(NC(c2occ3c2CCC3)=O)C(F)C1 N1(C(C=CSC)=O)CCCC2(C1)C(NC(=O)CCc1cnc(C)o1)CCN2C C(=O)(CN=S(C)(C)=O)N(CC1(NC(CNC(=O)OCC=C)=O)CC1)CC C1(CN(C)C(C2CCCC2CNC(C2(n3cccn3)CC2)=O)=O)CCCC2CC12 c1(OC(N(CC(C)C)CC(=O)N(c2ccco2)C)=O)ccc(Br)cc1 CC1CC=C(C(=O)N2CCCCC2CCNC(=O)Cn2cc(F)ccc2=O)CC1 C1(CC(=O)NC(C(=O)NCCn2c(C)cnn2)CC2CCC2)CCCOCC1 C1(CNC(C2(C)CC(F)(F)C2)=O)COCC2(CCN(C(=O)C=CBr)CC2)O1 N1(C(C(C(C)O)NC(C(C(CC)C)N(C)C)=O)=O)CCOCC(C)(C)C1 c1(NC(N2CCN(C(=O)OCC)CC2)=O)ccc2ncc(I)n2c1 C1(C(N(CC(C)NC(c2c(C)nc(-c3ccsc3)s2)=O)C)=O)CC2(C1)CC(O)C2 CCCC(C)CC(=O)N1CC(C)(C)CC1CC(=O)N(C(C)CSC)C Cc1cc(C(N2CCOCC2CNC(C23CC(C)(CO2)C3)=O)=O)nc(C)n1 c1(C(=O)Nc2c(C)cc(C(=O)OCC)s2)cc(C)c(C)cc1N c1(C(N(C(CN(C(Cc2c(C)con2)=O)C)C)C)=O)ncnc2sccc12 C1(C)(C(=O)NCC(c2ccccc2)C)CCCN1C(=O)COCC(F)F CC1CN(C(C2(C)CCC(=O)N2)=O)CCN1C(c1cc(C2CC2)no1)=O c1(CNC(=NCCOC)NCC(c2nccs2)C)cc(C)cc(Cl)c1.C(CO)S N1(C(c2c(CC)csc2)=O)CCC2(CC2)CC1C(N1CCC1CF)=O CCCC(C(=O)OC)C(=O)N1CC2(C(=O)NC(CC(=O)OC)C3CC3)CCC1C2 C1(CNC(c2ccccn2)=O)CC2CCC1N2C(c1ccc([N+](=O)[O-])s1)=O N1(C(C2CCOCC2)C(=O)NC(=O)OC(C)(C)C)CCN(c2cncs2)CC1 CC1COCCC1C(N1CCCC1(C)CNC(=O)Cn1cc(C(F)(F)F)nn1)=O N1(C(CCCCSC)=O)CC(F)(F)CC1(C)CNC(C1CC12CCSCC2)=O C1(NC(c2ccc(=O)oc2)=O)CC2CN(C(=O)CSCC(F)(F)F)CC2C1 c1(C(=O)NCCN(C(C2CN(C(C)C)C(=O)CC2)=O)C)cc(N)c2ncccc2c1 C12(CNC(CC(C)(C)O)=O)CCCC1CN(C(=O)C1=C(Cl)CCCC1)C2 c1(C(c2n(CCCC)nnn2)NCC2CC2(C)C)cccc(N(C)C)c1 N#Cc1cc(C(=O)NC2CCN(C(c3ccc(F)c(O)c3)=O)CC2F)ccc1F c1(C(N2CC3C(NC(C(CC)N(C)C)=O)(CC3)C2)=O)ccc(F)c2[nH]ccc12 N1(C(COCCOC)=O)CCC2CN(C(=O)Cc3ccc(C)cc3)CCC12 C(=O)(CC1=CCN(C(=O)C=CC2CCOC2)CC1)NC(C(CCC)C)CO N1(C(c2nccc(CC)c2)=O)CC(CNC(=O)C(C)(C)CCSC)CC(C)C1 c1(C(=O)NCC2C(C)CN(C(=O)CSCC(N)=O)C2)noc2cc(Cl)ccc12 c1(OC)cc(C(=O)NCC=C2CCN(C(C3CCC(=O)N3C)=O)CC2)cc(C)n1 Cc1cc(C(=O)NC2(CC=CC(N3CCCC(C(N)=O)C3)=O)CCC2)nn1C C1(NC(=O)Cc2nc[nH]n2)COCCN(C(C2CCCNS2(=O)=O)=O)C1 CCC(F)(F)CC(=O)N1CCC(CCCCNC(=O)CC(O)C(C)C)CC1 C#CC1(CO)COCCN1C(C1CN(C(=O)OC(C)(C)C)C1)=O C#CC1(C(=O)NC2(CC=C)CN(C(=O)Cn3cc(C4CCOC4)cn3)C2)CCCC1 C1(c2nc(C(C)OCC)nn2Cc2ccc(Br)cc2)CC2C=CC1C21CC1 C1(C#N)(C(=O)NC(CC=C)CC(F)F)CC2CCC1C2 C1(NC(CCN2CCN(C)CC2)=O)CCN(C(=O)Cc2cnco2)C12CCCC2 CC(C)C(C)(C(N)=O)NC(C1CCCCC1NC(=O)C(F)C1CCCC1)=O CC1CN(C(c2cccc(CC3CCC3)c2)=O)CC1NC(C1NC(=O)OC1C)=O C(=O)(CC(C)CC(C)C)N1CCC(C(=O)NCC)C(O)C1 c1(OC)cc(=NC(=O)C(C2(O)CCCCC2)NC(=O)Cc2cnc(C)s2)[nH]n1C CCS(=O)(=O)CCNC(=O)C(n1cc(C(C)(C)NC(=O)OC(C)(C)C)nn1)C N1(C(c2cc3n(c2)CCCC3)=O)CCOc2ccccc2C1C(F)F C1(CC)CCC(C(=O)NC2CCCC2CNC(c2sccc2C(C)(C)C)=O)CC1 CC(c1cccc(Cl)c1)=CC(N1CCC(N(C(=O)CN2CCCC2)C)C(C)C1)=O Cc1ccc2c(c1)CN(C1CCCC1NC(=O)C(c1ccc(Cl)c(F)c1)O)C2 C(C(CNC(C1(CCCF)CC1)=O)CO)NC(CCOCCC)=O C(C(O)C(F)(F)F)NC(=O)NC(c1csnn1)CC c1(CNC(CCCOCC)=O)ccc(CCNC(=O)C(C)(C)C2CCC2)cc1 N1(C(COCCC)=O)CCN(C(=O)C(C)CSCc2ccccc2)CC1C c1(N2CC(c3c(OC)cccc3)OCC2)nc(C)c2c(n1)CCCC2 C1(NC(c2cc(OCC(F)F)ccn2)=O)C2CN(C(C3CC(O)C3)=O)CC12 C=CC1CC(NC(C2CCCC2CNC(=O)C(=C2CCCCC2)F)=O)C1 C12(C(=O)NCC(CC)N(C)C)CC(C)(CN1C(=O)C(C)SC)C2 C(=O)(C(C)CCC(C)(C)C)NCCN(C(C)C)C(C1CCCN1N=O)=O N1(C(C2(COC)CCCO2)=O)C2CCC(C2)C1CNC(C1C(C)(C)C1(C)C)=O C(=O)(CCCC(=O)NCC1CCN(C(=O)CC(C)O)C12CC2)NC Cc1oc(C#N)cc1C(=O)NCc1nocc1C(=O)NCC12CCCC1C2 C=CC1(C(=O)NC2CC(CCNC(c3cc(CC(C)C)[nH]n3)=O)C2)CCCC1 C1(CNC(C=C(C)C)=O)CCCC1NC(c1ccc(-c2cc[nH]n2)s1)=O C1(NC(c2cc3ncccc3[nH]2)=O)CC12CCC(NC(C1CC1F)=O)CC2 c1(OC)ccc(NC(C)=O)c(CS(=O)Cc2ccccc2Br)c1C#N C1(C(=O)OC)C2CC1N(C(C1CC1C(=O)Nc1nc(Br)cn1C)=O)C2 CCC(C(=O)NCCN(C(=O)Cc1c(C)nc(O)nc1O)C(C)C)C(F)(F)F N1(C(C2C(C)CCO2)=O)CCN(C(=O)Cc2csnn2)C(C2CCC2)C1 CC(C)(C)C(CCc1cccc(F)c1)NCc1ccc([N+](=O)[O-])o1 C(=O)(C(O)C(F)(F)F)N1CCC(C(C)NC(=O)Cc2cnn(C(F)F)c2)CC1 C1(CNC(c2[nH]nc(OC)c2Cl)=O)CC12CCN(C(=O)Cc1cncnc1)CC2 C(=O)(CS(=O)(=O)CCO)NC1CCCC(NC(c2cccc(C)c2)=O)CC1 c1(CNC(CC2CC(NC(c3ncn(CO)n3)=O)C2)=O)cccc(Cl)n1 N1(C(CCCC(C)C)=O)CCN(C2CCCN(C(=O)Cc3cc[nH]n3)C2)C(=O)C1 N1(C(CCCCCC)=O)CCC(C2(O)CN(C(=O)C=C3CCC3)C2)CC1 c1(NC2CN(C(Cc3cccc(COC)c3)=O)C(C)C2)ccc([N+](=O)[O-])c(C#N)c1 N1(C(c2cn(C)nc2)=O)CCN(C(=O)Cn2ccnn2)CC(C)(F)C1 N1(C(CC(CC)C)=O)CCCC2C1CCN2Cc1ccc(C#N)cc1C C=C1Cn2c(C(=O)NC3CC(NC(C4(OC)CCSC4)=O)C3)nnc2S1 C1(NC(C2CC(C)N(C(=O)Cc3sc(SC)nc3C)C2)=O)CC(CC=C)N(CC)C1 C1(C(N(C2CCN(C(c3cc4sccc4[nH]3)=O)C2)C)=O)CCCCN1N=O C1(NC(C2CC(=O)N2)=O)CN(C(c2cc3occc3s2)=O)C2(CCOCC2)C1 C1(C(N)=O)CCCC(C(=O)NCC2(NC(=O)C(CF)=CC3CC3)CCC2)CC1 Cc1cc(Cl)cc(Cl)c1OCC(=O)NCC1CC1NC(=O)CSC(C)C CC(C)C(F)(CNC(C1(CO)CCCO1)=O)C(=O)N1CCCCC(CO)C1 C1(CC=C)(NC(=O)CCOc2cc(F)cc(F)c2)CCCN(C(=O)C(C)SC)C1 S(=O)(=O)(c1ccc(F)cc1)NCCC(=O)NC1C(NC(CNC=O)=O)CCOC1 C1(C(N(CC#N)CC#N)=O)CCCC12CCN(C(C1CCC3(CC1)CC3)=O)C2 c1(CC)cc(C(N2CC(OC)CC2CNC(C2(CC)CC2)=O)=O)ccc1O Cc1ncc(C(N2CC(C(=O)NCc3ccc(Cl)cc3)C(C(C)C)C2)=O)c(C)n1 CC1(C#CC(=O)NC2CC3CC4C(C3)C24C(N2CC(O)(CO)C2)=O)COC1 c1(C(=O)OC)ccccc1C(N)CNCCCC1CCC1 N1(C(C2N(S(CCCC)(=O)=O)CCC2)=O)CCN(C(=O)Cc2cn[nH]c2)C2CC12 c1(CC)ccc(F)cc1NC(=O)C(C(C)C)NC(=O)Cc1sccc1C C(=O)(C(CCC)CC(C)C)NC(C(=O)N1CC(=C)C1)Cn1ccnn1 CN1CCn2ncc(C(=O)NC3CN(C(=O)C=Cc4cccn4C)CC3O)c21 CC1(C(N2CCC2CNC(c2cccc(N)c2O)=O)=O)CCCS1(=O)=O C(=O)(C1=CCOCC1)NCC1OCCN(C(C(C)(O)Cc2cccc(F)c2)=O)C1 c1(C(=O)NCC(C)N(C(Cc2c(C)ncs2)=O)C)cc(OC(F)F)cc(F)c1 N1(C(Cn2cnc(C#N)n2)=O)CCCC2CN(C(C3CCCC3(F)F)=O)CC12 C1(NC(CNC(CN2CC(C)(OC)C2)=O)=O)CC2C(O)C(O)CC12 N1(C(c2cc(C)c(F)cn2)=O)C2CCC1CC(NC(=O)C(C)(C)CN(C)C)C2 C(CCC(=O)N(C)CCNC(C1CC1c1cnn(C(C)C)c1)=O)NC(=O)OC n1(CC)nc(C)c(C(N2CCCC2CN(C)C(c2cc(O)cc(Cl)c2)=O)=O)c1Cl N1CC2CC(C=O)C1C2.O=C1NC(C2(c3ccnn3C3CCC3)CC2)CO1 N1(CCn2cc(CC(=O)OC)nn2)CCN(C(=O)C(C)(C)C)CC1 C1(C(=O)NCCOCCCN(C(=O)CC2CC(n3cnnc3)C2)C)CC1[N+](=O)[O-] C(N=c1nc2scnc2c(N2CCSC(C(C)C)C2)[nH]1)c1nc(C)[nH]n1 N1(C(c2cnc(OC)c(Cl)c2)=O)CCC(C2CC2)C1CNC(=O)OC(C)(C)C CCC(C(=O)N1CCC(CC2CCN(C(C3(O)COC3)=O)CC2)CC1)C(C)C C1(C(=O)NC2CCN(C(c3cnn(CC(F)(F)F)c3)=O)CC2)CCC2(CC1)N=N2 C1(CNC(C2N(C(=O)NC)CCC2)=O)CCCCN1C(c1sc(F)cc1Cl)=O O=S(=O)(c1ccc(Br)cc1NCC1COCO1)NCc1cc(F)c(Cl)cc1Cl C(=O)(C(C)S(C)(=O)=O)N1CCC(O)(CNC(COCC(=O)NC)=O)C1 C12(C(N3CC(F)(CNC(C(C)NC(=O)NCC)=O)C3)=O)CCC(CC1)CO2 N1(C(Cc2c(C)scc2)=O)CCc2sc(CNC(C3(F)CC4(CCC4)C3)=O)nc2C1 C1(CCC)C(=O)NCCN1C(=O)N(CCCNC(c1ccc(C)cc1)=O)C C1(NC(C(CC)(C)F)=O)CCC2(CC1)CCN(C(c1n[nH]c(C)n1)=O)CC2 C(CCCCCC(=O)NCC1CCOCC1C)NC(CCOCCC)=O N1(C(c2n(COC)ncc2)=O)CCC(C(=O)N(C2CCCCC2)C)C1(C)C N1(C(c2cc(C)on2)=O)CC2CCN(C(=O)C3=NOC(c4ccccc4)C3)C2C1 C(C)(C)(CCCNC(=O)Cc1sc(O)nc1O)NC(CCc1cc(OC)no1)=O c1(C(N(CCNC(C=NOC)=O)C2CC2)=O)cc([N+](=O)[O-])ccc1N1CCCC1 C1(CNC(C2CC(=C)C2)=O)CN(C(=O)CCc2ccc(C(F)(F)F)cc2)CCO1 C1(C(N2CC(NC(c3cn(C)c(=O)cn3)=O)C3C(C2)C3)=O)CCn2cnnc2C1 C=CCC(CC)C(=O)NC1CCC(C(=O)NCc2nn(C)cc2C)CC1 C1(C(N2CC(C#C)(F)C2)=O)COCCN(C(c2c[nH]c(=NC)o2)=O)C1 C=C=CCCC(=O)NC(C)(C)CC=CC(=O)NCC1CCCC1CF C12(CCNC(c3c(C)cco3)=O)CCC1CN(C(=O)CC(C1CC1)C1CC1)C2 c1(C(=O)NCC(CNC(C(CCCCC)O)=O)F)[nH]nc2c1CCCC2(C)C N1(C(C2CN(C)C(=O)N2)=O)CCN(C(c2scnc2Cl)=O)C2COCC12 c1(OC)nc(C)ccc1C(=O)N(C1CCN(C(c2cc(Br)cs2)=O)C1)C CN1CCCC(C(C)(C)C(=O)N2CCC2CNC(=O)Cc2cnn(C(F)F)c2)C1 C(=O)(C=C1SCC(=O)N1C)N1C2C(NC(CC(=O)NCC#C)=O)(CCC2)CC1 Cc1nc2cc(NC(=O)C(C)OC(c3cc(Br)c(C#N)s3)=O)ccc2s1 c1(C(=O)NC2(CNC(c3ccc(F)s3)=O)CC2)c[nH]c2ncccc12 CCCCC(C)(F)C(=O)NCC1(CNC(=O)C(=O)NCCOC)CCC1 N1(C(C(CC=C)NC(=O)CC#N)=O)CCN2CC(C)CC2C1 CCC(O)C(C)C(=O)NC(C)(C)C=CC(=O)N(C1CCCC(O)C1)C N1(C(c2c(CC)n[nH]c2)=O)CCC(F)(CNC(C2(C3CCCO3)CCC2)=O)CC1 c1(C2N(C(C3(O)CCCCCC3)=O)CCC2)ccc(NN2C(=O)CCC2=O)cc1 Cc1csc(C(C)C(N2CCC(Cn3cc(CCOCCO)nn3)C2)=O)n1 C1(OC)CN(C(C2CC(C(F)F)C2)=O)C(C)(CNC(c2cc(F)cc(Cl)c2)=O)C1 C1(C(=O)NCc2n(C)c(O)nn2)CCN(C(C2C=CCC2)=O)C1(C)C C(C(N=[N+]=[N-])C(=O)N(CCCCN(C(=O)Cc1cc(F)ccc1O)C)C)OCC N1(C(=O)CC2CC2)CCC2C1CCCN2C(c1cncc(I)c1)=O C1(CNC(c2ccc(SC)o2)=O)CN(C(c2cscc2F)=O)CCC1(C)C c1(C(=O)NC2CN(C(c3c(Cl)ccnc3Cl)=O)CC2O)cc2cccnn2c1 c1(-c2ccc(CCCC)cc2)cc(C(=O)NCc2ccc(Br)s2)c2cn[nH]c2c1 N1(C(CC2CN(C)C2)=O)CCC(NC(=O)CCc2ccsc2)C(CO)C1 C1(CCNC(=O)Cc2cc[nH]n2)CN(C(c2nc(Cl)c(Cl)s2)=O)CCO1 c1(C(N2CC(CNC(C(C)(C)C)=O)C(C)(C)C2)=O)n[nH]c2ccc(Br)cc12 N1(C(c2cncc(NC)c2)=O)CC23CCCC2(C1)CN(C(C1CC1F)=O)C3 Cc1ccc(C)c(CNc2nccc(N3CCCC(F)C3)n2)n1 C1(CCNC(=O)CC2CNC(=O)O2)CN(C(=O)CC2CC=CC2)CCO1 C1(CNC(c2cc(C(=O)OC)n(C)c2)=O)(NC(=O)C(C)CSC)CCCCCC1 N1(C(c2c(C)csn2)=O)CCCC(CNC(C2(CO)CCCC2)=O)CC1 C1(C)(C(=O)NCCCOCC=C)CN(C(=O)CC2CC2C2CC2)CC1C c1(OC)cc(C(N2CC3CC(C2)N3C(c2cn(C)cn2)=O)=O)ccc1I Cc1ccc(F)cc1C(=O)C(=O)NCC1CN(C(=O)Cc2ccoc2)CCC1C N1(C(CCSC)=O)Cc2ccccc2C(NC(C2(F)CCOC2)=O)C1 N1(C(C2C(CCOC)C2)=O)CCCC(O)(CNC(c2cc(N(C)C)ccn2)=O)C1 c1(CC)nc(C(=O)NC2CC2CNC(c2c[nH]nc2-c2ccnn2C)=O)cs1 Cc1cnccc1C(=O)NC(CNC(=O)CC1(C2CC2)CC1)C1CCC1 N1(C(C2C(C)C2c2ccccc2)=O)CC2CC2(CNC(=O)CSC2CC2)C1 c1(CC)n[nH]c(=NC2CC3CC(C2)N(C(=O)CCC(F)(F)F)C3)o1 CN1C(=O)OCC12CN(C(=O)CN(C(C1CC13CCOC3)=O)C1CC1)C2 N1(C(CC(C)C2CC2)=O)CCC(NC(c2nn(C(F)F)cc2Cl)=O)CC(C)(C)C1 Cc1cncc(C(=O)NC(C)CCCNC(c2cc[nH]c2C2CCCC2)=O)n1 C1(NC(Cn2ccc(C)n2)=O)CC2CCC(C1)N2C(=O)CCc1nc(C)cs1 c1(C(N2CCC(N(C(c3csc(SC)n3)=O)CC)C2)=O)ccc(N)c(F)c1 Cc1ccc(NC(c2ccc(F)c3ccccc23)=O)cc1S(N)(=O)=O N1(C(=O)CN2CCSCC2)CCC2CC1CN(C(C13CC(F)(C1)C3)=O)C2 C1(OC)(CNC(c2cnsn2)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C1 C(=O)(CC(C)(C)C(F)F)NCCC1OCCCN(C(C2CCCC(OC)C2)=O)C1 c1(C(N2CC(C(C)NC(C(c3ccccc3)C)=O)C2)=O)cnc(-c2ccco2)s1 N1(C(CN(CCC)C)=O)CC2CC(C)N(C(c3cc(C)ncc3C)=O)C2C1 C1(CNC(COCCC=C)=O)CC2(CCN(C(c3csc(C)c3N)=O)CC2)CO1 C1(C(=O)NCc2ccnc(OC)n2)CN(C(=O)CC2OCCCO2)CCN1C c1(C(CC)NC(=O)C(=O)NCc2ccc(F)cn2)ccc(C)cn1 N1(C(COC(CC)CC)=O)CC(F)(F)CC1CNC(c1cc2[nH]ccc2s1)=O CC1(C)CCC(C(=O)NC(C)(CNC(=O)COc2ccon2)C2CC2)C1 C(=O)(CC(CNC(c1occc1CN(C)C)=O)OC)N1C(C(=O)NC)CC1 c1(C(N(CCOC)CCNC(c2c[nH]nc2F)=O)=O)cc(C)cc(Cl)c1 Cc1cc(C)c(C(=O)NC(C(=O)N(C2CC2(C)C)C)c2cccs2)cn1 C1(C(N(CC(F)Br)C)=O)CC(NC(=O)C=CC2(C)COC2)CCO1 Cc1c(C(=O)NC2(c3ccccc3)CC2)c(C#N)c2n1CCC2 C1(C(=O)NCC(CC=C)NC(C2CCCC2OC)=O)(COC)CC(F)(F)C1 c1(C(=O)OCCCn2cncn2)ncnc2sc(C(F)(F)F)nc12.O=CC=CC CC1(C(=O)NCc2cn(CC(=O)NCc3nnns3)nn2)CCCOC1 n1(CC(=O)NCC2CC(OC)CN2C(c2sccc2SC)=O)ccc([N+](=O)[O-])n1 C(=O)(CCCC1CC1)NCCCCN(C)C(c1nocc1-c1ccccc1)=O C1(C(C)NC(C2CN(C)C2)=O)CCN(C(C2CCCN2C(=O)C2CC2)=O)C1 c1(OC)cc(I)ccc1C(N1C2CC1CN(C(c1cccn3cncc13)=O)C2)=O c1(C(N(C2CCN(C(c3cnn(C)n3)=O)CC2)CCC)=O)ccccc1CC#N Cc1cccc(F)c1-c1nc(-c2cnn3c2CCC3)cs1.N12CCCC1C2=O N1(C(C2C(NC(c3ccsc3Br)=O)C2)=O)CCOC(NCCn2cccn2)C1 Cc1nc(C(F)(F)F)ccc1CNC(N1CCN(CC(O)C(F)(F)F)CC1)=O c1(-c2c(C)c(O)ccc2)ccc2c(c1)CCN(C(c1ccc(Cl)cc1I)=O)C2 c1(C(=O)NC2CC(O)CN(C(=O)C=CC3CC3)C2)cnc2ccoc2c1 CC#CCCCC(=O)N1CCC(C(=O)N(C2CCN(C(C)=O)C2)C)O1 C(=O)(C(N=[N+]=[N-])C(C)C)N(C(C(=O)NC(C(=O)OC)CO)CC(C)C)C CC(CC(=O)NC12CC(CNC(C3(F)CCOC3)=O)(C1)C2)C(F)F C1(N(C)C(C2CSCCS2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C C(=O)(CC(C(C)OC(F)F)N)NCC(C(=O)CN1CCCC1CC1CCC1)=O c1(NC(c2cncc(-c3cc(NC)c(C)cc3)n2)=O)nc2cc(F)ccc2s1 CCC(C)CC(=O)N(n1cc(C2CCC2)nn1)C1CC(C2CCCCC2)C1 CC(C)C(CC1CCCC1)C(=O)N1CC2CC1C2CNC(C1(CO)CC1)=O C1(C(=O)N(CCC(C)N(C(c2ccc(C)cc2)=O)CCO)CC)CC2C(C1)C2(C)C c1(Cn2cc(C3N(C(c4sc(CC)c(Br)c4)=O)CCC3)nn2)cc(Cl)ccc1Cl C=C1CCC(C(=O)NC2CC(NC(c3cc(C)[nH]n3)=O)C2)CC1 Cc1cc(N2CCCC(CNC(c3scc(C)c3Cl)=O)C2)nc(C)n1 c1(OC)ccc(F)c(C(=O)NCC2C3CN(C(=O)CCc4n[nH]c(=N)s4)CC23)n1 N1(C(C2CC(C#C)(O)C2)=O)CC2CC1CN(C(c1sccc1OCC)=O)C2 C1(C(C)NC(=O)Cn2cnc(Br)c2)CCCN(C(=O)CN2CCC(C)(O)C2)C1 N1(C(C(CC)CC2CCCC2)=O)CCN(C(=O)C(C)(C)CF)CC1CC(=O)NC C1(CNC(C(CC)=CC)=O)CCN(C(C2CCC(C(C)(C)O)CC2)=O)CC1 N1(C(COC)=O)CCN(C2CCCN(C(=O)Cc3ccco3)C2)C(=O)C1 c1(C(=O)NCC(CNC(=O)CC(C)F)OC)cc(F)c(F)cc1O C(=O)(C(C(C)(C)C)NC(=O)Cc1ccon1)NC(c1ncn[nH]1)C c1(CCNC(C(C)C)Cc2ccc(F)cc2)cnc2c(C(=O)O)cnn2c1 CC(C)(CCC(=O)NCC1(CCCO)CC1)NC(C1CC2(CC2)CO1)=O C1(C(N2C(C)CC(NC(CC=C)=O)C2)=O)CC2CC1C1CC21 Cc1ccc2ncc(C(=O)NCC3(F)CCC(CNC(C45CC(C4)C5)=O)C3)n2c1 Cc1cc(F)ncc1C(=O)NCCC(C)N(C(=O)C(CO)c1ccccc1)C C1(N(C)C2CC2)CC(C(=O)NCCN(C(CCNC(=O)OCC)=O)C)CO1 C1(OCC)COCCC1NC(Cc1ccccc1C)C1CCC1.C(C(=O)OC)C1CC1 C1(CNC(C2(CC(C)C)CCC2)=O)CCC(NC(=O)Cc2c(Cl)cnn2C)CC1 N1(C(C2(C#N)CC=CC2)=O)CC2(CCC2)CC1CNC(=O)CCc1cnccn1 N1(C(C(CCC)CC)=O)CCN(C(C2(CC(F)F)CCC2)=O)CC(O)C1 C1(NC(CCC=C)=O)CC(N=c2[nH]c(C3CCCC3)nc(Cl)c2C)C1 N1(C(C2CC3CCCC23)=O)CCOC2(CCN(c3ncnc(O)c3Br)CC2)C1 C1(C(N2CCC(N(C(c3ccc(COC)o3)=O)CC)C2)=O)CC(=O)CCO1 C(=O)(C1=NOC2(CCOC2)C1)NC(CCNC(c1cnc(C)o1)=O)C C1(C(N2CCC(F)(F)C2)=O)CC2(C1)CN(Cc1ccc(Cl)cn1)C2 c1(C(=O)NCC2CN(C(C(C)n3cccn3)=O)C(C)(C)C2)ncn2c1COCC2 C1(C(=O)NC(CNC(c2cc(CCOC)on2)=O)(C)CO)CC(C)(C)OC1(C)C C1(CNS(N(C)Cc2ccccc2)(=O)=O)CC2COCC(C1)C2(F)F n1(-c2ccn(CC)n2)nc(COC)nc1C1CC(n2cccn2)(OC)C1 CC1(C)CC(C)(C(=O)NCC2CC(C(=O)NC3CC3CCF)C2)C1 N1(C(CCOC(CC(C)C)C)=O)CCC(O)(CNC(c2cnnn2C(C)C)=O)C1 C1(C2(O)CN(C(=O)C=Cc3cnccn3)C2)(CNC(=O)CCc2ccoc2)CC1 c1(CCCC)nc2ccccc2n1CC(=O)NCC1CN(C(C)=O)CCC1(F)F C1(CC(=O)NCCSCC(F)(F)F)CCCCC1O.C1CC(=O)N1n1cnnn1 c1(OC)cc(C(=O)NC(C)CC2CN(C(c3csc(NC(C)=O)n3)=O)C2)nn1C c1(NC(C2CC(=O)NCC2)c2nnnn2CCCC2CC2)ccc2c(c1)COC2 C12(NC(C(C3CCC3)OC)=O)CCCC1N(C(C1(F)CCC(=O)CC1)=O)CC2 CCCCCC(O)CC(=O)NCc1ocnc1C(N1CC(N2CC(F)C2)C1)=O C1(C(N(CCN(C(C)C)C(c2cnccc2Br)=O)C)=O)CCC12CCC2 CCCCCCC(C)(CCC)C(=O)N(C1CCN(c2ccccc2OC)C1=O)C CC1CCC(NC(C2CC3(CSC3)C2)=O)CN1Cc1ccc(C(F)F)cn1 C1(NC(C(C(CCC)C)C)=O)CCN(C(=O)CN(C)C(=O)OCC)CC12CCC2 N1(C(=O)NC(c2cccc(OC(C)C)c2)CC)CCOCC1C1CCOCC1 CCCC(C)CCCC(=O)N(CCCNC(=O)C(O)C1CCCC1)CCO C1(NC(C2(CC)CCC(O)CC2)=O)CCN(C(=O)CCNC(C)=O)CCC1CO c1(C(N(C2CCN(C(C3CCOCC3)=O)C2)CC)=O)ccc(C)nn1 C1(C(=O)NCC2C(NC(C(CC)N(CC)CC)=O)CCC2)CCC(CSC)CC1 N1(C(C2C(C(N)=O)C2)=O)CC2CCC1CN2C(=O)Cn1ccc(C(F)F)n1 C1(NC(C=NOC)=O)CCN(C(c2cc(C)nc(C)c2)=O)CC(C)(C)C1 C(=O)(CC(CC)C(C)C)N(CCC(C)NC(C1(COC)CCCC1)=O)C N1(C(C2CN(C(C(C(=O)OCC)OC)=O)CC2F)=O)CC2CCC1CC2 C1(C(=O)Nc2ccc(Nc3cc(C)ncn3)c(F)c2)CCCN2CCCC12 c1(N(CCC(O)C(C)(C)C)C)nccc(=NC2CSC2)[nH]1 c1(SCC)cnc(O)c(C(=O)NC2CCCCC2NC(c2snnc2CC)=O)c1 c1(NC)ccc(C(=O)N(C)CCN(C(=O)C=C(C)C(C)(C)C)C(C)C)c(F)c1 NC(=O)C#CC(=O)N1CCC(NC(=O)COc2cccnc2)CC1 C1(C)(CNC(C(CCN(C)C)(C)O)=O)CCCN(C(=O)C(C)S(C)(=O)=O)C1 c1(C2C(COCC(CN(C(C)(C)C)C3CC3)(C)C)C2)ccc(F)cc1Cl c1(C(=O)NCC2COCC2NC(C2(O)CCSC2)=O)cncc(-n2ccnn2)c1 CCC(C)CC(=O)NC1CC(CNC(c2ccnc(N(C)C)c2)=O)CC1O N1(C(c2c(C)cns2)=O)CC(C(N2CCCCC2C2(O)CC2)=O)CCC1(C)C c1(C(=O)NCC(CNC(C2=C(C)CC2)=O)(C)F)cc2n(n1)CCC2 c1(C(=O)NCC2CCC(NC(C(CC=C)CC)=O)C2)cnc2snc(C)c2c1 N1(C(C2(OCC)CCC2)=O)CCC(NC=O)CC1.C1(N)CCN(C(C2(C)CC2)=O)C1 Cc1ccc2[nH]cc(C(=O)CNC(C3CCCCNCC3)=O)c2c1 CC1(C)Cc2c(Br)cccc2C1OC(=O)N1CCC(NCCO)c2ccccc21 C#CCCC(C(=O)NCC1(O)CC2CCC1O2)NC(=O)Cn1ccc(C)c1 C1(CC(=O)N(C(CNC(c2ccc(C)nc2)=O)C)C)CCCCC1(F)F Cc1cc(C(=O)NCc2csc(CNC(=O)C(C)(C)F)n2)ncc1C#N C1(C(=O)Nc2c(C#C)cccc2)CCN(C(=O)CSc2ccncc2)CC1(F)F c1(C(=O)NCC2(O)CCCC2)ncn2cc(-c3cccc(O)n3)sc12 Cc1cc2c(C(=O)NC(C)CC(C)NC(c3c(C)ccn3C)=O)ccc(C)c2[nH]1 C1(C(=O)NC2(CNC(CCn3ccc(C)n3)=O)CCCC2)CC(S(C)(=O)=O)C1 N1(CCCCCNC(CCCC)=O)CCN(C(=O)CN(S(C)(=O)=O)C)CC1 N1(C(=O)COc2ccccc2O)CCC2CCCN(C(C34CCC(C3)C4)=O)C2C1 c1(OC)cc(F)c(C(N2CC3CC2C3C(=O)Nc2cc(O)ccn2)=O)cc1F c1(CC(=O)NC2CC(NC(C34COC(CO)(C3)C4)=O)C2)ccc2c(c1)OCCO2 C1(C2CCCNC2)(C(N2CC3CCCCC23CO)=O)CC1 C(CC(C(C)(C)C)NC(=O)Cc1cnco1)N(C(c1c(C)snc1)=O)C c1(C(=O)NCCNC(=O)CCSC2CCCC2)ccc(Cl)c(F)c1O N1(C(C2CCN(C(C3CC34CCCCC4)=O)CC2F)=O)CCCNC(=O)C12CC2 C1(NC(CC(n2c(CC)ncc2)C)=O)CC12CC(NC(c1ccc(F)cc1)=O)C2 c1(C(CC(=O)OC)NCc2nscc2Br)ccc(SC(F)(F)F)cc1 C1(NC(CC2(NC(Cn3c(C)nc(C)n3)=O)CCCCC2)=O)CN(C)CC1(C)C C(C)(CCC(=O)N1CCC(C)(F)C1)NC(CC(C)=C(C)C)=O Cc1ccnc(C2CCN(C(=O)Nc3sc(Cl)cc3Cl)C2)c1 n1(CC)nc(C)c(C(=O)NCCC2(NC(C3C4CCCC34)=O)CC2)c1Cl C12(NC(CC3CC(=C)C3)=O)CCC(NC(C3(C(N)=O)CCC3)=O)(CC1)CC2 N1(C(c2c(CC)cno2)=O)CCC2(C1)CN(C(c1cccc(C)c1Cl)=O)C2 S(=O)(=O)(c1ccccc1N1CCOCC1)NC(=O)C1CC1.c12ccccc1CNC2 CCCCCC(C)CC(=O)N1CCCC1(C)C(N1CC(C)(O)C1)=O C1(C(=O)NCc2ncc(CC)[nH]2)C2CC2CN1C(c1ncc(F)cn1)=O N1(C(C(C(C)(C)C)SC)=O)CCN(C(=O)CCC(C)(C)C)CC12CC2 C1(NC(CC(C)F)=O)CC12CCN(C(C1(C)CCOC1)=O)CC2 c1(C(=O)NC(C2CCN(C(C3CNC(=O)N3)=O)CC2)C)ccnc2c1ncn2C C#CCC(C)(C(=O)NCCc1nnc(O)o1)NC(=O)C(O)C(C)(C)C O(NC(=O)C(CNC(=O)Cn1cccc1)C(C)C)Cc1cccc(C)n1 C1(C(=O)NCC(CNC(c2cc(CCC)n(C)n2)=O)OC)CS(=O)(=O)CC(=O)N1 C(=O)(C(Cc1cc[nH]n1)NC(c1cnsn1)=O)NCC(C)F N#CC1(C(=O)NCC2CCCN2C(=O)CCC2CCCCCC2)CC2CC2C1 N1(C(C2CCC(C)CC2)=O)CCN(C(C2CCCCCN2C)=O)CC1C c1(NC(=O)N(C2CCO2)CC2CCC2)cccnc1F c1(C(N2C(C(=O)Nc3cc(C)cc(C)n3)CC(C)C2)=O)cc(F)c(Cl)c(C#N)c1Cl c1(N(CC(C)NC(CCc2cc(OC)no2)=O)C)nc(Cl)nc2nc(Cl)n(C)c12 N1(C(c2cc3ncccc3[nH]2)=O)CCC2CCC(NC(C34CCC(C3)C4)=O)C1C2 Cc1ccc(F)c(CC2CCCCC2CCNCC(N)=O)c1 N1(C(C2C(CC)CN(C(=O)CC3CCC3)C2)=O)CCCCCC1C(C)C CCCC(CC(C)C)C(=O)N1CC(C)(C)OCC1CNC(=O)C=C(C)C(C)C C1(C(=O)NCC=CCNC(=O)C(c2ccccn2)O)CC2C=CCC(C1)C2 N1(C(C(C(CCC)NC(COC2(C#C)COC2)=O)O)=O)CCCC(C)(C#N)C1 c1(NC(N(c2ccc(Br)cc2)CCOC)=O)cccc2c(F)ccnc12 CCS(=O)(=O)CC(=O)NCc1cccnc1CNC(=O)CC1CCN(C)C1 c1(C(=O)NC(CNC(C(CCCC)(C)F)=O)CO)[nH]c2c(c1C)CCCC2 c1(C(N2CCCC(NC(C3C(OC)CCCCC3)=O)C2)=O)cc(C#N)cc(C)n1 C(=O)(C#CC(C)(C)CNC(C1CC=C(C)CC1)=O)NCCSCC#C c1(CC(=O)NCC(C)N(C(c2ccnnc2)=O)CC)ccc(S(=O)C2CC2)cc1 c1(OC)ccsc1C(C(=O)NC1CC1)N(C(c1cccnc1)C(C)C)C C12(CC(=O)Nc3c(OC)nsc3)CCC1CN(C(=O)C(C)(O)CCN(C)C)C2 O=S(=O)(c1[nH]c(=NC2CC(CF)C2)ccc1Br)NC1CCOCC1O C1(CC(=O)NCCCNC(C(c2n(C)cnc2)O)=O)CCCC(C)(C)C1 N1(C(CC(C=C)CCC)=O)CCn2nc(CNC(=O)CCN3CCCC3)cc2C1 C1(C(=O)NC2CN(C(=O)NC3CC(C)(C)C3C(F)(F)F)C2)CC12CCOCC2 CC1(C)CCCC(C(=O)NC2CCCC(NC(C3CC3(Cl)Cl)=O)C2)C1 N1(C(C=CCN(C)CC)=O)CCCC(O)(CNC(C2CC2(Cl)Cl)=O)CC1 N1(C(c2ccc(C)cc2C2CC2)=O)CCC2CN(C(=O)C(C)(C)OC(F)F)CC12 C1(S(N)(=O)=O)(C(=O)NC(C2CN(C(=O)CC(C3CC3)C3CC3)CCO2)C)CCC1 n1(CC(N2CC(C(C)NC(C(CCSC)O)=O)C2)=O)ccc([N+](=O)[O-])n1 c1(CSC)ccc(C(=O)NC2CC2NC(=O)COCCCN(C)C)cc1 C1(OC)CN(C(C2CC2(C)C)=O)CC1C(=O)NC1(C(O)CO)CC1 C(=O)(CC(C)(C)C(C)=O)NCC(CCC)C(=O)NCC1(CO)CC12CCC2 N1(CCCCNC(C2(N(C)C)CC2)=O)CCCN(C(=O)CN2CC3CC3C2)CC1 C(=O)(CC(C)C(=O)NC1CCC(NC(=O)C=C(C)C(C)C)CC1)OCC N1(C(c2cccc(SCCC)c2)=O)CC(NC(=O)CCC2OCCO2)CC(O)C1 c1(CC(C(=O)OC)NC(=O)Cc2ccc(Cl)c(C#N)c2)ccc(F)c(Br)c1F C(=O)(CS(=O)(=O)c1ccccc1Cl)N(CCNC(C(COC)C)=O)C1CC1 c1(OC)cc(Cl)ccc1NC(=O)NC(c1ccnn1C)C CCC(C)(C(=O)N1CC2CC1C2NC(=O)CC1(CN(C)C)CCOCC1)C(N)=O c1(CCNC(c2ncn(CCNC(CCOCC(C)C)=O)c2)=O)ccccc1O C1(CNC(c2c(C)cc(F)s2)=O)CC(C)(C)CN1C(c1ccc(Cl)nc1C)=O CCCCCC(C)C(=O)N1CCC2C1CCN2C(=O)CN1CCOC1=O Cc1cnn(C(C)C)c1C(=O)NC1CCCC(N(C(=O)CC=CC(C)(C)C)C)C1 CC1CCC=C1C(=O)N1CCC(N(C(=O)C=Cc2ccoc2)CCO)C1 c1(OC)ccc(CN2CC(C(=O)NC(CCO)C(C)C)CC(F)C2)c(F)c1F C1(CNC(Cc2cc(C)c(F)cc2)=O)C2CCC1CN(C(=O)CCCN(C)C)C2 C1(CC(=O)NCc2ccc(CNC(C3(O)COC3)=O)cc2)CC2(CCC2)CCO1 CCCC(O)C(CO)NC(=O)CN1CCN(C(=O)CC2CCCO2)CC1 C(=O)(CCCC(N)=O)N.C(CC(O)C(=O)NC1(C)CCC1)SC.C12CCCN1C2=O C1(CC)(CC)CN(C(=O)CC(C2CC2)NC(=O)CN(C2CC2)CC)C1 c1(CC(=O)NC2C3CCN(C(C4CC(CC)(CC)C4)=O)C32)ccc(F)c(C#N)c1 n1(CC)cc(C(N2CC(F)CC2C(N2CCC(Br)C2)=O)=O)c2ccccc12 Cc1[nH]c2c(F)cccc2c1CCNC(N1CCC(CC2CC2)CC1C)=O N1(C(C)C(=O)NC23CC(C2)N(C(=O)C(C)(O)c2ccccc2)C3)CCCCCC1 Cc1c(C(N2CC(CC(=O)NC(C3(CO)CC3)C)CC2(C)C)=O)c[nH]c1C#N N1(C(C(n2nnnc2C(C)(C)C)C)=O)CCC(N(C)C(C2(O)CCC2)=O)CC1 CCCC(O)C(=O)NCCC1(NC(c2nccn2C)=O)CCCC1 CCCCC(CCC)N.c1(C2N(C(=O)O)CCC2)cnc(N)cn1 c1(COC)nc(C(=O)NCC(=C2CN(C(=O)CCc3cnc(O)[nH]3)C2)F)cs1 c1(C2C(c3ccc(C)c(C)c3)C2)nc(C)c([N+](=O)[O-])cc1Cl N1(C(C(CCC)C)=O)CC(NC(c2oc(CC3CC3)nc2C)=O)CC(F)(F)C1 CCC(C(=O)N1CCN(C(=O)Cc2cnnn2C)C(CC(=O)NC)C1)C(C)C C#CCCC(O)CCNC(C1C2CCN(C(=O)C=CC3CCC3)CC12)=O c1(C(=O)OCC)nc(C)ccc1.C1(C(=O)OCC)(C(=O)OCC)CCC1 C(C)(C)(CC(=O)N1CCC(NC(=O)CSc2nc[nH]n2)C1C(C)(C)C)SC c1(C(=O)NC2C(CNC(c3n(CCCC)ncc3)=O)C2)cc2ccc(Cl)cn2c1 N1(C(C(C)OC)=O)CC2(CCNC(C3(Sc4ccccc4)CC3)=O)CCC1C2 c1(C(=O)NC(C2CN(C(c3nncn3C)C)C2)C)cc2sccc2s1 C1(NC(c2cc(C)nn2C)=O)C2CC3CN(C(=O)CSCC4CCCO4)C1C3C2 CC(C)CC(O)C(=O)NC1(CNC(c2ccc(Oc3ccccc3)nc2)=O)CC1 n1(CC)nc(C(=O)NCC2(F)CCN(C(C3(CO)CC(C)(C)C3)=O)C2)cc1O Cn1cc(C(=O)NCC(CNC(=O)Cn2cc(CO)nn2)CO)c(C(C)(C)C)n1 C1(CNC(C2(CSC)CC2)=O)(NC(c2ncc(OC)cn2)=O)CCCCC1 C1(OC)CC2(C1)CC(NC(=O)NC1CCN(C(=O)OC(C)(C)C)C1)C2 C1(CC=C)(C(=O)NCCC2CC(C(N3CC(COC)C3)=O)C2)CCOCC1 N12CC3CCC3(C1)C2=O.N1(C(C)(C)C)CCC(NC(c2cncs2)=O)C1=O N1(C(CC2C(C)CCN(C(=O)CC3CCSC3)C2)=O)CC2C(=O)NC(=O)C2C1 C1(CN=[N+]=[N-])CCCN1C(=O)Cn1cc(Cl)cn1 Cc1ncnc(C)c1CC(=O)N(C1CN(C(C2CCCC3(CC3)C2)=O)CC1O)C C(N=c1cc(C)[nH]cc1[N+](=O)[O-])C1CN(C(c2c(SC)ccs2)=O)CC12CCC2 C#CC1(CNC(C2(CNC(=O)CC3CCCCC3)CC2C)=O)CCCC1 C#Cc1cccc(C2CC2C(=O)Nc2ccc(NS(C)(=O)=O)c(F)c2)c1 C(c1ccc(F)c(F)c1)=CC(N1CC(C)(C)C(NC(=O)C=Cc2cnc[nH]2)C1)=O n1(CCCC)ncc(C(N2CCCC(N(C(=O)C(C)SCC)C)C2)=O)c1C C1(NC(CN(C2CC2)CC)=O)C(C)CCN(C(=O)CCOCCN(C)C)C1C.C(C)=O C1(C(=O)NC(C2CCCC2)CO)COCCC1NC(C1(O)CCCC1)=O C1(C)(CNC(C2(COC)CCOC2)=O)CCCNS1(=O)=O C(=O)(C(CC(C)C)NC(C)=O)NCC12CC(NC(CC3(OC)CCC3)=O)(C1)C2 CC(O)C(C)(C)CN=c1[nH]c(N(CC2CCc3ccccc32)C)nc2cc[nH]c12 C1(C(=O)NC2CCCC2NC(=O)CNC=O)(COC)CC=CCC1 c1(C(=O)OC)cc(CC(N2CC(O)(CCNC(c3nccs3)=O)C2)=O)ccc1O N1(C(C(C)SC)=O)CC(CNC(c2cc(Br)no2)=O)C(O)C1 Cc1cnc(C(=O)NC(C)CC2CCN(C(=O)CCCC3CC3)CC2)c(C)c1 c1(NC(C(N2C(C)CC(NC(c3cnc(C)[nH]3)=O)C2)=O)=O)ccc(C#N)c(Cl)c1 CC(C)C(CCN(C)C(c1cnn(C)c1)=O)N=c1cc[nH]c(C#N)n1 C(C(C(=O)NCc1ncc(C)cn1)C(C)C)NC(CC(C=C)C)=O c1(CNC(C)=O)ccc(C(=O)N(C)CC2(O)CCN(C(=O)C=CCF)C2)cc1 c1(C(=O)NC2CCCN(C(C3N(C(C)C)CCC3)=O)C2)cc(Cl)ncc1F c1(OC)cc(CCNC(=O)C(=O)NC(c2ccc(Br)c(Cl)c2)C)cc(OC)c1O C1(O)(C(=O)NCCC(=O)NC(C)Cc2cccs2)CCSCC1 c1(SC)ccc(F)cc1-c1ccnc(CNC(=O)CCc2ccc(C)c(F)c2)c1 C1(CC)(CNC(=O)COC2CCOC2)CCN(C(=O)CCc2c(C)noc2Cl)C1 N1(C(C=COCC)=O)CCCC(C(C)(O)CNC(c2ncccc2N(C)C)=O)C1 c1(-c2cc(C(=O)NC)c(Cl)nc2)ccc(S(=O)(=O)NCc2ncccn2)cc1 CC1CCN(C(=O)C=CC2CCCC2)CCN1C(C1CCCS(=O)(=O)N1)=O N1(C(C(C)(C)C2CCC2)=O)CC2COCCC2(NC(=O)CCn2cnnn2)C1 C1(C(N(CC(C)NC(=O)C(c2nc(C)cs2)C)CC)=O)CC2(C1)CC1(CC1)C2 Cc1cccn2cc(C(N3CCC(N(C(=O)CCC(C)C)CCO)C3)=O)nc12 C1(CNC(C(CC)C(C)C)=O)CN(C(c2nnsc2C(F)F)=O)CC(C)(C)C1 C(CCCC(C)NC(c1cc(C(C)(F)F)n[nH]1)=O)NC(c1cc(CCC)[nH]n1)=O c1(C(N(C)NC(C(=O)NCCOCC)=O)=O)ccccc1OC.C12CC(C1)C2 C1(O)(C(C(=O)NC(C)CN(C(=O)Cn2cc(C3CC3)nn2)C)(F)F)CCCCC1 N1(C(C(C2CC2)SC)=O)CCCC(CC(N2CCOCC2)=O)C1 c1(C(=O)NC(CN(C(=O)CCCC(=O)NC)CC)C)cc(C)nc2[nH]nc(O)c12 CC(C)(F)CCC(=O)NCC1CCCCC1NC(=O)CN(CC(=O)N(C)C)C C(=O)(C(C)C(C)NC(c1cccnc1O)=O)N1CC(CC)(OC)C1 C1(CC)C(NC(C2C3CCCCC23)=O)CCCN1C(=O)CNC(c1ccsc1)=O C1(NC(C2(C)CC=CCC2)=O)CC2CC(NC(=O)CCCCC#N)C2C1 c1(C(N2C(CCNC(C3CC(CCC)C3)=O)CCCC2)=O)cc(C)cnc1N N1(c2n(Cc3cncc(C)c3)c(C3CCCN3C)nn2)CCC2(CC1)CC(Br)C2 CCC(C)(C)CC(=O)N1CCCCC1CCC(=O)Nc1cc(CO)cc(F)c1 N1(C(c2n(C(C)C)ccn2)=O)CCN(C(C2CCC=CO2)=O)CC1C c1(OC)noc(C)c1C(=O)NCC1CCCCC1NC(=O)COC1CCOC1 Cc1cc(C(=O)NC2(C(=O)NC3(C(C)C)CC3)CCCC2C)nc(C)c1 C1(C(C)C)OCCC1C(=O)NCC1CCCC1NC(=O)CNC=O c1(SCC)c(C(=O)Nc2cccc(NC(c3cccc(F)c3)=O)c2)cccc1F c1(CN2CCN(C(C(N)=O)=O)C(CF)C2)ccc(F)cc1[N+](=O)[O-] N1(C(C(C2CCOC2)OC)=O)CCCCC1CNC(c1oc(C2CC2)nc1C)=O c1(C(N(CC(C)NC(=O)Cn2ccnn2)CC)=O)cnc2c(ccn2C)c1 C1(NC(c2ccc(C(C)C)o2)=O)CCN(C(=O)CC(=O)NC2CC2)C(C)C1 C1(C(=O)NC2CN(C(C3(CC#C)CC3)=O)CC23CC3)COc2cc(Cl)ccc2C1 N1(C(C(CCC2CC2)OCC)=O)CCC(CO)C(O)C1.C1(C)CCC(=O)N1 c1(OC)ncccc1S(=O)(=O)Nc1cc(-c2cc(C)ccc2C)cs1 C1(O)(C(=O)NC(C2(O)CN(C(c3c(C)c[nH]n3)=O)C2)C)CCc2ccccc2C1 CCC(C)(C(=O)NC1CCC1NC(c1ccnc(-c2ccco2)c1)=O)C(N)=O c1(OC)ccc(CN2CCOCC2CC(N2CCC(C)C2)=O)cc1I c1(C(N2CCCC(NC(C(CC)CO)=O)CC2)=O)cncc2c(O)nccc12 c1(NC(CCC#C)=O)ccc2c(c1)CN(C(c1ccc3cccc(Br)c3c1)=O)C2 CC1Oc2ccccc2OC1C(N1CCN(C(c2ccco2)=O)CC1)=O C1(CNC(c2ccc(C)cc2F)=O)CN(c2ccnc(N(C)C(C)C)n2)CC(C)(C)O1 C1(COC)CC(CNC(c2c(Cl)cnn2C)=O)N(C(=O)C=C(C)C(F)F)C1 C(C(C(C)(C)C)N)NC(C(C)C#N)=O.N(S(N)(=O)=O)CC(=O)C=O CCC(C)(C(=O)N1CC(CC(C)NC(=O)CN2CCC(C(N)=O)CC2)C1)C(F)F C1(NC(=O)C2=COCCO2)CCC2CN(C(=O)CO)CC2C1 C1(C(N2CCCC2c2nc[nH]n2)=O)CCC(O)CN(C(=O)C#CC2CCOC2)C1 CC1OCCC1(C)SCC(=O)N(C1CN(C(C)C)C1)C(=O)CSC1CCSC1=O c1(N2C3CCN(Cc4ncn(C)c4)C3CCC2)ncnc2c1cnn2C(C)(C)C N1(NC(C2C=CC(Cc3cccc4[nH]ccc34)C2)=O)CCc2ncccc2C1 C12(NC(c3n(C(C)C)ccn3)=O)CCCCCC1N(C(c1n[nH]c(O)n1)=O)CC2 c1(C(=O)NCCC2(CNC(c3c(CC)ccs3)=O)CC2)cccc2ncnn12 C(=O)(CC(C(F)(F)F)c1ccn(C)n1)N1C(CN(C(CC=C)=O)C)COCC1 C(CC(F)F)(C(=O)NC1CC1F)NC(C(C)=NOCC#N)=O c1(SCC(=O)NC2C3(NC(=O)C4=CCCCO4)CCC(C2)C3)nc2ccccc2s1 c1(NC(C2CC(F)CN2Cc2cccnc2F)=O)ccc(Cl)cc1O C1(NC(c2ccc(OC)c(C)c2)=O)CCCCN(C(c2cnco2)=O)CC1 C(C)(CN=c1[nH]nc(CO)s1)(C1CC1)NC(C1(C(N2CCCC2)=O)C(C)C1)=O N1(C(c2cnc3[nH]cnc3c2)=O)CCN(C(=O)C2=CCOCC2)C2(CCC2)C1 c1(C(=O)NCC23CC(CN2C(c2cnc(O)o2)=O)C3)cc2ccccc2o1 c1(C(C(=O)OC)CCC(c2nccn2C)N)ccccc1I.C1CCC1 C1(CNC(C(N)=O)=O)CC(O)CN1C(c1cnn(C2CCCC2)c1)=O c1(C(=O)NCC2CCCN2C(c2cc(CF)on2)=O)cc(OCCSC)ccn1 c1(OC)cc(CN2CC3C(C2)N3C(=O)C(c2ccc(Cl)cc2)=O)cc(SC)c1 c1(C(=O)NCCC2CN(C(C(c3ccccc3Cl)C)=O)C2)nccn2ccnc12 c1(C(=O)NCC2(OC)CN(C(C3CC=CCC3)=O)C2)cc2cnccc2o1 C1(C(N2C3CC(NC(C4(CC)CCC4)=O)C3CC2)=O)CC2(C1)CC(F)C2 C1(NC(C2CCC(C(C)C)N2C(c2ccc(C#N)[nH]2)=O)=O)CCc2c[nH]nc2C1 C(N=c1[nH]c(=NCC2CCC(F)C2)c2cc(OC)ccc2[nH]1)c1nnn(CC)n1 CC(C(=O)NC(CNC(=O)CCOCC(F)F)C1CC1)NS(C)(=O)=O C12(C(=O)NCC#CCNC(C(C=C)c3ccccc3)=O)CC1Cc1c[nH]nc12 C(=O)(C(CC(C)CC(C)(C)C)N1CCCS(=N)(=O)CC1)NCC=C c1(C(=O)NCC23C(CN(C(C(CCC)C)=O)C2)C3)cc(N)cc(S(C)(=O)=O)c1 C1(NC(c2c[nH]c(=NCC)s2)=O)C(C)CN(C(C2CC(N(C)C)C2)=O)CC1C C=CC(C)(CC)C(=O)NCC1CC1.c1(CC2CN(C)CCO2)ccc(C)cc1 Cn1cc(C(N2CC3CC3(CNC(=O)COc3ccccc3F)C2)=O)n(C)c1=O C1(C(CNC(CCC#C)=O)C)CCN(C(c2cnc(Cl)n2C)=O)CC1 C12(C(N3C(C(=O)OCC)CCC3)=O)CCCC1CCN2C(=O)CCC1CCOC1 C1(O)(CNC(C(n2nnnc2C(C)(C)C)C)=O)CN(C(c2n[nH]cc2C2CC2)=O)C1 c1(N(CCCCC=C)C)cccc(S(N)(=O)=O)c1S(C)(=O)=O C1(C(=O)NCC2CC(C(N(CC(C)C)CC3CCCO3)=O)C2)CCC(F)(F)C1 C1(NC(C2CC(OC)C2)=O)CN(C(C2CC(=C3CC3)C2)=O)CC12CC2 Cc1nn(C)c(C)c1CC(=O)NC(C)CNC(=O)C=Cc1cc[nH]n1 C1(NC(CN2CCN(C(c3n(C)nnc3)=O)CC2)=O)CCC2(CC1)N=N2 c1(C(=O)NC(C(=O)NCc2c(CC)n[nH]c2)Cn2cncn2)ncn2ccccc12 C1(CNC(Cc2c(OC)ccnc2)=O)CN(C(C2C(C)C2C)=O)CCN1C c12ccc(cc1)C(=O)NCC2.C(C)(CC(C)(C)C)NC(C=CC=C)=O.CC C12(C(=O)NC3CC(CNC(C4C(OC(C)=O)C4)=O)C3)CCCCC1OCC2 N1(C(c2n(OCC)nnc2)=O)CCC12CCC(OCC)CC2 c1(C(N2C(CNC(=O)C(C)CO)CC(OC)C2)=O)occ2c1CCC2 N1(CC(=O)N(CCC(=O)NCC(=O)NCC#C)C(C)C)CCC(C)CC1 N1(C(C(CC=CC)CC)=O)CC2(CCCC2)C1C(=O)NCc1cccc(O)n1 C1(C(=O)NCc2cc(C)ncc2)N(C(=O)C(C2CCOCC2)F)CC12CCCC2 C1(C(=O)Nc2cnc(O)nc2O)CCC2(CN(Cc3ccc(F)cn3)C2)O1 CC1(C)Cc2ccccc2C1NC(=O)NCc1ccc(C2CCCCC2)cc1 CCC(C)(O)C(=O)N1CC(CO)(NC(c2csc(C)c2OC)=O)C1 C(=O)(C(C(C)C)n1cnc(C)c1)NCC1N(C(CCOCC)=O)CC1 c1(C(=O)OC)cc(OC)ccc1CC(=O)Oc1ccccc1F Cc1cc(C(=O)NC2CC2NC(=O)C(C(C)C)Sc2ccccc2)nn1C C1(C(=O)NCCC2(O)CN(C(C(C)NC(CC)(C)C)=O)C2)CC=C(C)CC1 CCC(CC(=O)NCCc1ccncc1F)NC(C1CCCC1)=O c1(C(=O)NCCNC(C(C)Oc2ccc(OC)cc2)=O)ccc2c(c1)COCO2 CC1CC(C(N2CCC(C(=O)NC(C)(C)CC3CCC3)CC2)=O)CCO1 CN1CCC(=CC(=O)N(C2CCC(NC(c3cc(F)n[nH]3)=O)CC2)C)CC1 C12CCCOC1C1=NC=CNC(CC)SCC(=O)N(C)CC1CCCCNC2=O N1(C(CCCC(=O)OCC)=O)CCC(N(C(=O)COC2CC=CC2)CCO)C1 C1(C(N2C(C#C)CCC2)=O)C(C)OCCN1C(=O)C(C)=C1CCCC1 N1(CC(=O)NC(C2CC(NC(C3CCCCS3)=O)C2)C)CC(C)(C)C1 N1(C(C(=O)NCC)=O)CC(NC(=O)C(F)C2CC2)C(C)C1 c1(C(N2CCC(NC(CC3C(C)CCCC3)=O)C2)=O)c[nH]c2cccnc12 C1(CNC(C2(SC)CC2)=O)CCC2(CCC2)CN1C(C1CCCC(=O)CC1)=O C(CCCCCNC(=O)C(C)(O)C1CCOC1)N(C(=O)CN1CCSCC1)C C(=O)(CCS(=O)(=O)C(F)(F)F)N(CC(CC)NC(C1CCSC1)=O)CC C(CCC)(C(=O)N1CCCCC1C(C)NC(c1nocc1C1CC1)=O)=CCC N1(C(CC2(C)CC2(Cl)Cl)=O)CCC(C2CC2NC(c2cc3n(c2)CCC3)=O)CC1 N1(C(C(C)OCCC=C)=O)CCN(C(c2occc2C2CC2)=O)CC1CC1CC1 C1(C(=O)NCC(C)(C2CC2)NC(COCCC=C)=O)CCCOC1C CCC(C)(CNC(=O)C(CCOC)NC(=O)CC1C(=O)NN=C1C)CC c1(C(N2C(CNC(CSC)=O)C(C3CC3)CC2)=O)cc2ccc(OC)cc2o1 c1(CCNC(N2CCC(O)(c3cccc(F)c3)C2)=O)cccc(F)c1O C1(NC(=O)C(F)=CCCF)CC2CN(C(C34CCCN3CCC4)=O)CC12 C1(CNC(C(CSC)OC)=O)CCCN(C(c2cn(C)nc2C(C)C)=O)CC1 c1(C(=O)NC2(CNC(CC(C)F)=O)CCOC2)cc(Br)cc2c1OCCO2 c1(OC)cncc(C(N2CC(CNC(=O)CCc3ccnc(Br)c3)C2)=O)n1 CC(CC(=O)N(CCCCNC(=O)C(C)(Cl)Cl)C)c1ccccc1 C(N=c1[nH]cnc2cc(Br)ccc12)C1CN(C(c2c(CC)noc2)=O)CC1C c1(CC(=O)NCC(CCNC(C2(SC)CCC2)=O)O)c[nH]c2cc(Cl)ccc12 N1(C(C(CC)OC)=O)CC2CN(C(C3(Cc4cccc(Cl)c4)CC3)=O)CC(C1)O2 Cc1ccncc1CC(=O)NC(C)CCCNC(c1cccc(C(C)C)n1)=O C12(CNC(c3cc(CC)nn3C)=O)CCCC1CCN2C(=O)Cc1nnc(C)o1 c1(C(N2CCN(C(=O)CC3(C(F)(F)F)CC3)C3C2C3)=O)cc2cc(Cl)cnc2[nH]1 c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC2C)ccc2c(c1)C(C)CN2 c1(C(N2CCC(c3ccc(OC)cc3)C2)=O)c(C)n(C)n(-c2ccccc2)c1=O C(=O)(C1=Cc2ccccc2C1)N1CCC(NC(c2c(C)cc(SC)o2)=O)C(F)C1 c1(C(=O)NCC(CN(C(C2CS(=O)C2)=O)CC)(C)C)cccc(C(F)(F)F)c1 C#CCC(C(=O)NCC=CCNC(=O)CN1CCN(C)C(=O)C1)C1CC1 c1(C(c2cccs2)C(=O)N(CCCC(F)(F)F)CC)cccc(Cl)c1 N1(C(C)C(=O)NC2CCCC2)CCC(F)(c2cccc(Cl)c2)C1 c1(CCCC(N2C(CN(C)C(C3(C)CCC(=O)N3)=O)CCC2)=O)cccc(Cl)c1 C1(NC(C=CCOC)=O)C2CC3C1C3C2C(=O)Nc1cnc(F)c(C)c1 N1(Cc2nc(C)sc2)CCc2[nH]nc(C(=O)Nc3c(Cl)cc(Cl)cc3I)c2C1 C=CCC(CNC(=O)CN1CCOCC1)C(=O)NCCc1ccccc1C C1(C(=O)NCCC2CC(C)C2)CCN(C(=O)c2c[nH]ccc2=O)O1 Cc1ccc2nonc2c1C(=O)N(C)CCN(C(=O)C=Cc1ccoc1)C C(C)(C)(CCN=c1cc[nH]cc1S(=O)(=O)NC1(C)CCC(C(C)(C)C)CC1)OC c1(CCC(=O)NCCCCC2CN(C(C3(C(N)=O)CC3)=O)C2)cccc(F)c1F CCCCCCCCC(=O)N1CC=CC(NC(c2ncccc2OCCC)=O)C1 c1(CC(C)NC(c2c(CC)c(C)ccc2)=O)c[nH]c2c(C)cccc12 C1(O)(CC(N2CC3(C2)C(=O)NC3)=O)CCOCC1.C1(C(N)=O)CC(=O)CO1 CCCC(CC)CCC(=O)N1CCC(N=[N+]=[N-])CC1C(=O)N1CC(C)(O)CO1 c1(C(N(C2CCCN(C(CCCOC(C)C)=O)C2)C)=O)cc2scnc2[nH]1 C#Cc1cccc(C(=O)NCC2(C(=O)NCc3coc(C)c3)CCCC2)c1C N1(C(c2cc(C(C)=O)n(C)c2)=O)CCCC(O)(CNC(=O)C2=CCCC2)C1 c1(C(=O)NC23CN(C(C(C(C)C)SCC)=O)C(C2)C3)cc(C(C)(C)C)ccc1N C1(C)(C(N(CCCNC(C(C2(OC)CCCC2)(F)F)=O)C2CC2)=O)CCCC1O c1(C(C)C)nc(C(C)(C)C)cc(=NC(C)CNC(=O)C(c2ccnn2C)O)[nH]1 C1(C(=O)NCCC(C(C)C)NC(c2cn(C(C)(C)C)nn2)=O)CNC(=O)CC1C N1(CC(N2CCC(N(C(=O)C(C)OC)CC)C2)=O)CCOCC1=O C1(=CC(=O)NCCCCN(C(=O)C2=C(Cl)CCOC2)C)CC2CCC(C1)N2C C(=O)(C(C)(F)C(C)(C)F)NC(C1(O)CN(C(c2cnc3ccnn3c2)=O)C1)C CC(C)(C(=O)NCC(CO)NC(=O)C(F)(F)c1ccncc1)C1CCCCO1 c1(C(N(C2CCN(C)C2)CCOC)=O)cccc([N+](=O)[O-])c1C C(C(O)C(=O)NC1(CNC(C2CCC(=O)C2)=O)CCC1)SC C1(C(=O)NC(C=C)C)CC2(CC2)CN1C(c1ccc(OC)nn1)=O CC(C)CCCCC(=O)N(C(C)CN(C(=O)CNC(=O)Nc1ccccc1)C)C c1(C(=O)OC)nc(=NCC(CO)c2ccc(Cl)cc2)cc[nH]1 C1(C(=O)OC)(OC)CN(C(c2ccc(I)cc2C)=O)CC1OC C1(C)C(C(C)C)C(=O)N1.n1(CC#C)cccc1C(=O)NCC(N)=O.C1CS1 N1(C(C2CCCCO2)=O)CCN(C(c2cc(Cl)cnc2O)=O)C(CC2CC2)C1 C=CC(O)(C(=O)NC(CNC(c1ccc(C2CCC2)cc1)=O)CC)C(F)(F)F C1(C(=O)NC2CCN(C(CC)C)C2)CCS(=O)(=O)N1 Cc1cc(CC(N2CCC(NC(C3CCC=CO3)=O)CC2C)=O)cc(C)c1 c1(C(CC)C(=O)NCC(C)N(C(=O)C(=O)NCC)CC)cccc(C(F)(F)F)c1 c1(OC)cccc(C(=O)NCC#CCNC(=O)C(C)C2CCC2)c1 Cc1cn(C)cc1C(=O)NC1CC(O)(CNC(c2cc(C(F)(F)F)ccn2)=O)C1 c1(C(=O)NCCCCN(C(C2(C#C)CCC2)=O)C)csc2c(F)cccc12 c1(C(N2CCC(CN(C(CN(C)C)=O)C3CC3)CC2)=O)ccc2c(c1)C(=O)NC2 CCCC(C)(CCC)C(=O)N1CCCC(CCNC(C2(OC)CC(C)C2)=O)CC1 CC(C)CCCCCCC(=O)N(C1CN(C(C2CCCSC2)=O)C1)C N1(S(CC=C)(=O)=O)CCCC2(CCCN(Cc3c(F)ccc(Br)c3C)C2)C1 c1(C(N2CCCCC(CNC(C3(CC#C)CC3)=O)C2)=O)c(C)ccc(Cl)c1N c1(OC)ccc(O)c(NC(=O)CC23CCC2CN(C(C2(C)COCCO2)=O)C3)c1 n1(CC(=O)NCCN(C(C23CCC(CC2)C3)=O)CC)nc(C2CC2)n(C)c1=O C1(NC(C=CCOC)=O)COC2(CCN(C(=O)Cn3nc(C)c(Cl)c3C)C2)C1 CC1(NC(=O)CC2(c3ccccc3)CC2)CCN(C(C2CC23CC3(F)F)=O)CC1 c1(OC)ccccc1C(=O)C(=O)NCCCN(C)C(C1CC(=C2CC2)C1)=O C12(CNC(=O)CCc3cncs3)COCCN1C(=O)CN(C(c1cnc[nH]1)=O)C2 C1(CC(N2CCC(N(C(=O)CCC3CCCCO3)CC)C2)=O)CC(=O)NC1=O c1(-n2c(C(C(CCC)C)NCC(C)(C)c3ccns3)nnn2)ccc(Cl)cc1F Cc1noc(C)c1C(=O)OC.C12CCN(C1=O)CC(=O)O2.C123CC(C1)(C2)C(=O)N3 C1(C(=O)NCc2nncn2C2CC2)CCN(C(=O)COCC2CC2)O1 Cc1ccc(C)c(C(=O)NCc2ccnc(Br)c2)c1O c1(CCC(=O)N(CCNC2CCCCO2)CC)cc(Cl)no1.C(=O)(COC)NC1CC1 C1(CC=C)(C(=O)NC(c2nccn2C)C)CN(C(c2csc(=N)[nH]2)=O)C1 CC#CCCC(=O)NC(C)(C(=O)NC(C)C(C)CC)C1CCC1 C1(CNC(C2=CC(C)(C)C2)=O)(NC(c2nncs2)=O)Cc2ccccc2C1 Cc1nc(C(N2CC(C(N)=O)(CNC(=O)C(=O)NCCC(N)=O)C2)=O)sc1C CC1(C(=O)NC2CCN(C(=O)Cn3cnc(C(N)=O)n3)CC2F)CCCNC1=O C1(C)(CNC(c2c(CN(C)C)ccs2)=O)CCN(C(c2nn(C)cc2Cl)=O)C1 N1(C(CC2(OC)CN(C(=O)Cn3cnc(C#N)n3)C2)=O)CC(CO)CC(C)(C)C1 c1(N2CCC(=C)C2)nccc(C)c1C(=O)CNC(=O)C(CCC)N(C)C CCCCC(C)CCC(=O)N1CCCC2(NC(c3cccn3C)=O)CCCC12 N(C(=NCCCF)N1CCCC(S(=O)(=O)N(C)C)C1)CC1CC(C)OCC1 C1(NC(C(CCSC)(C)C)=O)CC2CCC(C1)N2C(=O)Cc1ccc(CO)cc1 C(=O)(CC(C)C(F)(F)F)NCC1(C)CCN(C(C2CC(OC)(OC)C2)=O)C1 CCCCC(C)C(=O)NC1(CNC(C2(F)CCOCC2)=O)CCCCCC1 c1(C(=O)NC(C)CCNC(C2CNC(=O)C2)=O)cc2c(cc1N)CCC2 C=C1CCC1(C(=O)NCC(C1CC1)N(C(=O)Cc1cn(C)nn1)C)C(=O)OC CC1(C)CCCC(O)(C(=O)NC2CC3CCCCN3C2=O)CC1 c1(C(=O)NCC2(NC(C(CC(C)C)OC)=O)CCCC2)cc([N+](=O)[O-])cn1C c1(C(=O)NC2C(C(=O)Nc3c(C)cc(Cl)cc3)CC2)cnc2ccccn12 N1(C(C)=O)CCCC2(CCCCCN2C(c2cccn3nncc23)=O)C1 Cc1cc(C(=O)NC2CC2C(=O)NC2CN(C(C)C)C2)cc(C)c1 c1(C(N(C2CCN(C(CC(=O)OCC)=O)C2)CC)=O)cc(C(C)C)nn1C C(=O)(C(C(C)O)N(C)C)NC(CNC(CC=CCC)=O)(C)Cn1cccn1 C1(CC(N2C(CNC(=O)CCn3cccn3)CC2)=O)CC=CCC1 C1(O)(C(=O)NC2CN(C(C(C)C3CC3)=O)C(C)CC2)CCc2ccccc2C1 C12(COC)CCC(C(N3CCOC(C)(CNC(C4(OC)CC4)=O)C3)=O)(CC1)CO2 C1(C(=O)NC(c2ncc[nH]2)CC)C=CCCN1C(C1CCN(C)C1=O)=O C12(CNC(c3c(=N)[nH]cnc3)=O)CCC(CC1)N(C(c1cnc(S)[nH]1)=O)C2 C1(n2c(-c3ccc(OC)cc3)ncc2)NC(=O)N(C2CCCC(C)(C)C2)C1=O Cn1nnc2cc(C(=O)NCCNC(=O)CO)cnc12 N1(C(C23CN(C(C(CC=C)CC)=O)C(C2)CO3)=O)CCC(O)CC(C)(C)C1 N1(C(C(CCCC)O)=O)CCCC12CCCN(C(C1(C#N)CCSCC1)=O)C2 N1(C(Cc2nc(NC(C)=O)sc2)=O)CCN(Cc2nc(C3CC3)no2)CC1 c1(C(N(C(CC)C(N2CC(OC)C(O)C2)=O)C)=O)ccccc1F C1(NC(C(C)(N)Cc2ccccc2F)=O)CC2CCCC(C1)N2 CC1(C)CCCC(CNC2(CC(=O)O)CC2)C1 c1(OC)ccc(N)cc1C(=O)NS(=O)(=O)CCCn1cccn1 C(CCCC(=O)N(C)Cc1ccccc1)N(C(=O)CNC=O)C c1(CC)cccc(C(=O)NC(c2cn(C3CCC3)nn2)c2nncn2C)c1 C1(C(=O)NCCc2n(C)cnn2)CC2CC1CN(C(c1cncnc1)=O)C2 N1(C(c2cnc(C)s2)=O)CCC(C2(NC(=O)CCN(C)CCO)CC2)CC1 C=CC(C)(C)C(=O)NCC(=O)OC.C1C(O)C(=O)N1 C1(C(C(=O)NCCCC(C)NC(Cc2ccc(C)s2)=O)F)CCCCCC1 N1(C(C(C)c2cccs2)=O)CCC(C(=O)N(C)CC2CCCS2)C1 C1(C(=O)NCCN2CCC(F)CC2)C2CN(C(=O)CC3CC3C(F)(F)F)CC12 N1(CC(C)NC(=O)CSc2ccccc2Cl)CCN(C(C2CCNC2=O)=O)CC1 C(=O)(CCCS(C)(=O)=O)NCC(N(C(C(C=C)c1ccccc1)=O)C)C1CC1 c1(C(N2CCC(NC(C(F)=CCC)=O)C2)=O)ccc(C2CC2(C)NCC)cc1 N1(CC#C)CCC(CNc2ccnn2C)C1 C(=O)(C1=NOC2COCC12)NC(CCC#C)C(=O)NC1CN(C)C(=O)C12CC2 c1(C(N(CCOCCNC(C(C)C2CC2)=O)C)=O)sc2ncccc2c1Cl c1(OC)ccccc1.C1(C2CCCC2)C(=O)NCCCSCCCN(C)CC1C N1(C(C(=O)NCCCC(=O)OC)CCc2ccco2)CCCC1P(C)(C)=O N1(c2nc(=N)[nH]c(=N)[nH]2)Cc2cc(F)c(F)cc2C1 C1(C(N(C(C)CNC(=O)COc2cn[nH]c2)C)=O)CC(=O)NC(=O)C1 CCC(CC(=O)NCC(C)C(C)O)NC(=O)CC1(COC)CC1 C(CN=c1[nH]c2cc(F)ccc2o1)C1CC(NC(c2ccn3cc(C)nc3c2)=O)C1 c1(OC)ccc(C(=O)C(N2CCC(O)(CNC(c3cc(C)on3)=O)C2)=O)cc1 CCCCCC(C)(C)C(=O)NCC(C)CN(C)C(c1cnn(C)c1C(F)F)=O C1(NC(C2N(N=O)CCCC2)=O)COC2(C1)CN(C(=O)C(F)(F)C(O)C1CC1)C2 N1(C(C(C)(C)CO)=O)CCN(C(c2cc(O)cc(Br)c2)=O)C(CO)C1 C12(CNC(c3c(C)ncs3)=O)CC(NC(=O)C(F)C(C)C)C(CO1)C2 c1(C(=O)NCC2CCCN2C(c2sccc2C(F)F)=O)cnn2c(=O)cc[nH]c12 CC(C)CC(C(=O)NCCCC(C)(C)C(=O)N(C)Cc1ccn(C)n1)C(N)=O c1(CCC)cc(C(=O)NCc2cc(C(=O)NC3CC3C)no2)no1 CC1(C(=O)O)CN(C(=O)CCn2cc(CCCC(O)C(C)(C)C)nn2)CCO1 c1(CC)ncccc1C(=O)NCc1cc(C)c(C(=O)NCCC2CCCO2)o1 Cc1c(C(=O)NCC(C)NC(C2(C)CCCO2)=O)cccc1S(N)(=O)=O C1(CNC(c2cc(C)ns2)=O)CC2(CCN(C(C3C(C)(C)C3(C)C)=O)C2)CO1 c1(NC(C(c2cccnc2)NC(=O)Cc2ccco2)=O)cccc([N+](=O)[O-])c1 C12(C(=O)NC3CC(F)(CNC(CCCOCCOC)=O)C3)CCC(=O)N1CCS2 C1(NC(C(C)OC2CCOC2)=O)CCC(C)N(C(c2ccc(=O)n(C)n2)=O)C1 CC(CCC(C)(F)F)C(=O)N1CCC(F)(CNC(=O)CCCC(N)=O)C1 CC(C)S(=O)(=O)C(C)C(=O)NC1CC(C)(NC(=O)C=CC2CCCN2C)C1 C(=O)(NN1CCCC1C(N1CC(O)C(O)C1CO)=O)C1CCC(C)(C)O1 C#CCC(O)C(=O)NC1C(C(=O)NCCOc2ccccc2)C1(C)C C1(C2CN(C(C3CC3(F)F)=O)C2)(NC(CC(C)c2ccccc2)=O)CC1 N1(C(C(F)=CC)=O)CC2CCC2(NC(c2ccc(OC3CCOCC3)cc2)=O)C1 c1(OC)ccc(CCNC(=O)C(c2ccc(Br)cc2F)(C)C)c(C)n1 Cc1cnc(Oc2ncnc(O)c2Cl)c(C)c1 C(=O)(CC1OCc2ncccc21)N1CCC(CCNC(c2cc(CC)[nH]n2)=O)C1 C(CCCC(CO)NC(C1CC(=O)N(C(C)C)C1)=O)NC(c1cc(C)ncc1)=O c1(NC(C(CC(=C)Cl)NC(=O)CC(C)n2cccc2)=O)ccc2nncn2c1 N1(C(C(N2CCOCC2)C)=O)CC2CCN(C(C3CNC(=O)N3)=O)CC12 C12(NC(CN(C(=O)CN3CCOCC3)CCOC)=O)CC1COC2(C)C c1(C(=O)NC(CNC(C(=O)Nc2c(C)cccc2C)=O)C)ccc2cnoc2c1 c1(CC(N2CCC(CCNC(C=CC(CC)=CC)=O)C2)=O)cccc2nsnc12 c1(CN2CCC3(C(C(=O)NC(=O)Nc4ccccn4)C3)C2)cccc2c1OCO2 C1(CNC(=O)C(O)C2CC2)(CO)CCN(C(C2CCCCCCC2)=O)CC1 C1(CCNC(CC2CC(=C)C2)=O)CSCCN1C(=O)C(C)CN1CCCCC1=O C(=O)(C(C(C)(C)O)NC(c1cc(C(C)=O)on1)=O)NC(C#C)C(C)(C)C CC1(C)CCC(CC(N2CCC(CNC(c3nnn(C(C)(C)C)n3)=O)C2)=O)CC1 N1(C(Cc2scc(C)n2)=O)CCCC(NC(c2cc(C3(C)CC3)on2)=O)C1C C(=O)(CC(CNC(C1CCCN1C(C)C)=O)C1CCC1)NC(CC)C c1(C(=O)NCCC2(NC(=O)C(O)CC(F)(F)F)CCC2)cc2c(F)cccc2s1 N1(C(C(CSC)O)=O)CC2CC(NC(c3conc3C3CCCC3)=O)CC1C2 CC(Cc1ccccn1)C(=O)N1CCCC1CCNC(c1ccn(C)n1)=O C(=O)(C(CC(C)C)CC(C)C)NCC(CC=C)NC(=O)C(C)(C)NC(=O)NCC N1(C(c2cc(C)sc2)=O)CCC(F)(CNC(C2CCC(CN(C)C)C2)=O)CC1 C1(C(=O)NCC2(CN(C(=O)CN(C)S(N)(=O)=O)C)CC2)CCc2nncn2CC1 c1(OCCCC(N2C(CNC(CC)=O)C(C)CCC2)=O)nc2ccccc2s1 C(=O)(C(C)CCCC(C)=O)NC1(C(=O)NCC(CCOC)(C)C)CCC1 Cn1nc2c(c1C(=O)NCC13CC1CN(C(c1cc(C(F)F)no1)=O)C3)CCC2 C1(OC)CC2CC(NC(=O)C(C)(C)C(C)NC(c3cnccc3C)=O)CC12 S(=O)(=O)(CCCNC(=O)NCC1CCCCN1C)NC.c12cccc(c1)C2 C(=O)(CN=c1ccc(C#N)c[nH]1)N1CC(NC(C(CCC)CC)=O)C(SC)C1 N1(C(CC)=O)CCN2C(=O)C(NC(c3ccc(Cl)c(C)c3OC)=O)CC2C1 N1(Cc2nc(OC)sc2)C(=O)NC(C2CCCO2)C1=O N1(C(CCN(C(C2(C#N)CC3CC3C2)=O)CC)=O)CCc2nn(C)cc2C1 CS(=O)(=O)c1ncc(C(=O)NC2(CO)CCCN(C(=O)CCOC3CC3)C2)s1 C(c1cccnc1)=C(CC)C(N1CC(NC(=O)CC(C)F)C(n2cccn2)C1)=O c1(SC)ccc(C(=O)NCC(=C2CN(C(=O)CCCF)C2)F)cc1 C1(C(=O)NC(CCC)CCC)CC12CCN(C(C1(C)CC(=O)C1)=O)C2 N1(C(C2CCCCC2O)=O)CC(C2CCCCC2)CCC1C(F)(F)F C1(c2n(C(C)C)cnn2)CCN(N(C)CC2CC2c2ccccc2)C1 C1(CNC(CNC(CCC)=O)=O)CC2CCC1N2C(c1cccc(OC)c1N)=O C=CC1CCN1C(c1cc(CNC(c2nsnc2O)=O)no1)=O Cc1cc(C)c(C(=O)NC2CCCC2CN(C(=O)C(F)C(C)(C)O)C)cn1 c1(NC2CN(C(C(CCC)C(C)C)=O)CC2C)ccc([N+](=O)[O-])c(C)n1 Cc1cc(=NCCN2CCC(C)C(CO)C2)[nH]c(=NCCC(C)N2CCCC2)[nH]1 CCCC(C)(O)CC(=O)N(CC(CO)(CO)NC(=O)C(C(C)C)SC)C c1(NC(CCC(C)(C)NC(C2CC2(F)F)=O)=O)cccc(N=[N+]=[N-])c1 C1(OC)(CNC(=O)C(C)(C)n2cccn2)CCN(C(=O)C(C)NS(C)(=O)=O)C1 C1(C(C)C)CN(C(=O)COCCNC(c2c[nH]c(C#N)c2)=O)CCN1C c1(C(C(=O)NCC#CCNC(C2C(C)CCC2)=O)(F)F)ccc(C2CC2)cc1 C=CC1(C(=O)NC(c2nccs2)CC)CCN(C(=O)C(CO)OC)C1 N1(C(CC2C(CNC(C3(C)CCCO3)=O)C2)=O)CC(F)CC1CO c1(CNC(c2cnn(CC3CCC3)c2)C)cccc(Br)c1 c1(NC(CSc2n(-c3ccc(C)cc3)c(C)nn2)=O)nc2c(s1)CCC2 C1(CNC(c2coc(Cl)c2)=O)CC2COCC2N1C(=O)CCc1ccon1 Fc1ccc(CNc2cc(-c3cccc(CC(F)(F)F)c3)ccn2)c2cc[nH]c12 c1(C(N(C)CC2(NC(c3nc(OCC)oc3)=O)CC2)=O)cn2ncccc2n1 C1(N(C(=O)CC2CCCO2)CCC)CCN(C(=O)CNC2CCOC2)C1 N1(C(CCNS(CC)(=O)=O)=O)CCN(C(=O)CN2CCOC2=O)CC1CCO C1(NC(CCOC)=O)CCC2(CC1)CC(NC(=O)CC1(N(C)C)COC1)C2 Cc1nc(C)c(C(=O)NCCCNC(c2ccc(C(C)(C)C#N)cc2)=O)c(C)n1 c1(C(N2C(C)(CNC(C(C3CC3)OCC)=O)CCC2)=O)noc(C)c1[N+](=O)[O-] C1(NC(C=CC(C)NC(c2c(C)[nH]cc2)=O)=O)C=CCCC1CO N1(C(C(CCC)O)=O)CCn2ncc(S(C)(=O)=NC(=O)C=CCC(C)(C)C)c2C1 c1(C(=O)NC(C(=O)OCC)C)nn2c(c1-c1ccc(N3CCC3)c(C)c1)CCCC2 N(C1CCc2cc(CNC(c3n[nH]cc3C(C)C)=O)ccc21)C(C=C(C)C)=O c1(C(=O)NC(CCCC)CNC(c2[nH]nnc2C)=O)cc(C)c(C)c(C)c1 N1(c2nnc(C)o2)CC2CCCC(NC(c3cc(C(F)F)ncn3)=O)C2C1 C1(C)(C(N(CCCCNC(C2CCN(C(CC)=O)C2)=O)C)=O)CCOCC1 c1(CC)nc(C)ncc1C(N1CC(C2(NC(C3CC3CN(C)C)=O)CC2)C1)=O c1(CC(=O)NCC(C(=O)N2CC(CO)(CO)C2)OC)c(C)n[nH]c1C C(=O)(C(F)CCC(C)C)N1CCC2C(C(NOC3CCCN(CC)C3)=O)C2C1 N1(C(C(=O)NC(C)C)=O)CC2CC2(NC(C2(c3ccccc3)CNC(=O)C2)=O)C1 C(=O)(C(CNC(=O)CC(O)C1CCCC1)C(C)(C)C)NCC1(C)CCN(C)CC1 c1(CC(=O)NCC(CO)NC(=O)CCCCn2ccnn2)cc(O)nnc1O C1(C(N2CCC(C)(NC(C)=O)C2)=O)CC1C1CN(C(c2cnn(C)c2N)=O)C1 Cc1cc(N2CCC(F)C(F)C2)c([N+](=O)[O-])cn1 C(=O)(C1=NOCC1)NC1(CCCCNC(c2c(CC)occ2)=O)CC1 N1(C(=O)OC(CC)CC)CCc2c(OC)ccc(C)c2C1 C=CCC(CNC(=O)COC1CCOCC1)C(=O)NCC(=O)OCC C1(NC(c2cnc(C)n2C)=O)CCC12CN(C(=O)CC(O)CN(C)C)C2 CC(CS(C)(=O)=O)C(=O)NCC1CC1CNC(C1(C(F)F)CCCO1)=O c1(C(=O)NC(CNC(COCCCC#C)=O)C2CC2)ccc(OCCCl)cc1 c1(NC(CC2(N(C)C)COC2)=O)cc2c(cc1C(F)F)OCO2 Cc1nn(C)c(C(=O)NCC2(O)CN(C(C3(C#N)CCCC3)=O)C2)c1Br C#CC(CC(C)(C)C)NC(C1(NC(=O)OC(C)(C)C)CC(O)C1)=O N1(C(CC2C(C)CC2)=O)CC2CC(C1)CN(C(C1CC1c1ccncc1)=O)C2 c1(CC(=O)NCCN(C(C2CCC3CC23)=O)CC2CC2)ncn2c1CCCC2 C1(CCNC(c2c(SC)ccs2)=O)CCN(C(C2CC(F)(F)C2)=O)C(C)C1 N1(C(C(C)Oc2ccccn2)=O)CC(NC(c2cncc(Cl)c2)=O)CC(C)(C)C1 c1(OC)ccc(CO)cc1C(N1CC(O)(C(C)NC(c2coc(CO)n2)=O)C1)=O C1(NC(=O)NC2CN(S(C)(=O)=O)C2)CCCCC1F CCC(CCOC)C(=O)NCC1CCC1NC(c1ccc(CN=[N+]=[N-])o1)=O C#Cc1cccc(C(N2CC(C(=O)N(CC(C)COCC)C)C(CCC)C2)=O)c1 c1(OC)ncc(F)cc1C(=O)NC1CCCC(CNC(=O)CCc2cnn[nH]2)C1 C1(C(=O)NCc2cc(C)cc(O)c2)CN(C(=O)CS(C)(=O)=O)CCC1(F)F n1(CCNC(Cc2ccc(C)c(Cl)c2)=O)c(O)nc2cccnc12 C1(NC(C(CC)CC2CCCCC2)=O)CC2CCC(C1)N2c1nnccc1C#N N1(C(C=C(C)Cl)=O)CC2CCC(NC(=O)Cc3cnc(C)nc3O)CC2C1 C1(NC(=O)CC2CCN(C(=O)CCC3CCCC3)C2)C2CN(CCF)CC12 C1(CC)CCCCC1OCCc1cn(C(C)CNC(=O)Cn2cnnc2O)nn1 C(=O)(CCC(=O)NCC1CCCN(C(c2cn(C(F)F)cn2)=O)C1)OC(C)(C)C N1(C(COCC(C)C)=O)CC2(C1)SCCC2NC(=O)CCC1CCCO1 CC(=O)CCCC(C)C(=O)N1CCC(CNC(=O)CC2(C)CC2)C(F)(F)CC1 N1(CCc2nn(CC)nc2C)CCCOC(COC(=O)OC(C)(C)C)C1 C(C)(CCC(=O)NCC1(C)CC1(F)F)NC(CSCC=C)=O N1(C(=O)C(O)C2CC2)CC2CCN(C(=O)Cc3ccoc3)CCC2C1 C(CC(=O)N=c1ccn(C)[nH]1)N(CC(C)C)C(C1CCC(C#N)CC1)=O c1(C(=O)NC2CCN(C(C=Cc3c(C)ccs3)=O)CC2)ccc2nccn2c1 c1(OC(C)C)ncc(Br)c(N2CCC(NC(c3ccc(C)nc3)=O)C2)n1 N1(C(CC2(NC(=O)C(C3CCOCC3)=O)CC2)=O)CC(CO)C(C2CC2)C1 Cc1nc(-c2cc(C)[nH]n2)sc1CCNC(=O)N(C)CCC1CC1 C(=O)(C1=CCCCC1C)NC1C(OC)CN(C(=O)C(O)CCSC)C1 N1(C(C=CC=CCN(C(=O)Cn2cccnc2=O)C)=O)CCCc2occc2C1 Cn1cncc(C(N2CC3(CNC(c4ccc(Br)cc4)=O)CC2CO3)=O)c1=O c1(C2C(NC(NC3CCC(CC)CC3)=S)C2)ccc(Br)c(F)c1 Cc1nc(C(=O)NCC2(F)CCC(NC(C3(F)CC=CC3)=O)C2)c2ccccn12 C(=O)(CCCCC(F)F)N1CCC(CC)C1CNC(c1cnn(C)n1)=O c1(CC2CCN(C(c3cnc(C4CC4)o3)C(=O)NCCC)C2)ccc(F)cc1.OC n1(-c2nccc(C)c2)nc(C2COc3ccccc32)nc1CC12CCCC1C2 C(C)(C(O)C(C)C)NC(c1c(CNC(CCNC(COC)=O)=O)occ1)=O N1(C(CCc2nc(C)sc2)=O)CCCC(CNC(C2C(C)C2C)=O)C1 N1(C(c2c(Cl)ccc(OC)c2)=O)CCC2(CCN(C(c3ccc(C)[nH]3)=O)C2)C1 c1(CC=O)cc(O)nc(O)n1.C1(C=O)(CO)CCCC1.N12CCC(C1)N2C C#CCC(C)(C(=O)N1CCC(C)(COC)C1)NC(c1cccc(C)c1O)=O c1(CCC(N2C(CNC(C(C)=C(CC)C)=O)C=CC2)=O)cccnc1Br c1(CNC2CCC(NC(c3cscn3)=O)C2)ccc(O)nc1 CC(C)(C)C(C(=O)N1CCCC(O)C1)NC(C1CCCC(=O)N1)=O c1(OC)n[nH]cc1C(=O)NCC(O)CNC(=O)CN1CC2CC2C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CN(C(=O)Cn1nccn1)C)(C)C N1(C(c2cc(C)ns2)=O)CCOC(C)(CNC(=O)C(C)(C)C2CCCCO2)C1 O=NN1CCCC1C(=O)NC12CC(NC(C3(F)CCOC3)=O)(C1)C2 N1(C(c2cn(CC)nc2C)=O)CCC(NC(=O)CCC2(C)CC2)C(F)C1 CCCCC(C)C(=O)NC(C)CCN(C)C(c1cc(O)ccc1C(F)(F)F)=O C(=O)(CCC(=O)NC)NCC1C(NC(CC2(OCC=C)CC2)=O)C1 C12(C(=O)NC(C)CCCCNC(C3CCOC3C)=O)C3CC(CC13)C2(F)F c1(C(=O)NCCCN(C(C2C(CC)CCO2)=O)C)ccc(C)c(S(C)(=O)=O)c1 c1(OC)c(F)cc(C(N2CC(CNC(c3ccc(O)nn3)=O)C(C)C2)=O)cc1Cl C(=O)(CCC(C(C)C)NC(C1CC(O)CCO1)=O)Nc1cccc(CC)c1 C1(NC(C(C)N(C)C)=O)CCC2CN(C(c3cnoc3)=O)CC2C1 C#CCCCCCC(=O)N1CCOC(CC(=O)NC2CC3CCCC3C2)C1 c1(C(=O)NCC(C)N(C)C(c2cnsn2)=O)cnc(O)c2cnccc12 C1(Cl)(C(N2CC(CC(CNC(CC(C)C)=O)(C)C)C2)=O)CC12CCOCC2 C1(C(=O)NCC2CN(CCC)C2)CCN(C(=O)CCC(=O)NC)C(CC)C1 N1(C(CC2OCC(C)(C)C2)=O)CC2(CCCC2NC(C23CCC(C)(C2)OC3)=O)C1 N1(C(CN(C)C(N)=O)=O)CC(NC(C2(C#N)CCCO2)=O)CC12CCOCC2 CC1CN(C(=O)COC2CCOC2)CCCN1C(c1ccsc1C(F)(F)F)=O c1(SCCC(=O)NC(CNC(COC(C)(C)C)=O)C2CCC2)nccn1C C#Cc1ccc(C(=O)NC2CCCC(N(C)C(c3coc(C)n3)=O)C2)cc1F Cc1nc2ccc(C(N3CCC4CN(Cc5cccn5C)CC34)=O)cc2[nH]1 N1(C(c2c(CC)n(C)nc2)=O)CCN(c2ccnc(C#N)n2)CC(C)(F)C1 C12(NC(=O)C=CC3CCOCC3)CCOCC1CN(C(C1(Cl)CC1)=O)C2 c1(C(=O)NC2(C)CN(C(CCC(=O)NCC)=O)C2)ccc2ccnc(O)c2n1 C(C)(C)(CC(=O)NCCC1(O)CCN(C(=O)C(F)Cc2ccccc2)C1)SC N1(C(c2c(C)cc(N)cn2)=O)CCCC2(C1)CN(C(=O)Cn1ncc(Cl)c1C)C2 C=C(CNC(=O)CC1(C)OCCO1)CCNC(c1ccnn1CC(C)C)=O CC1=NOC(C)(C(=O)NC2CC(CNC(=O)C(c3cccc(Cl)c3)(C)C)C2)C1 c1(NC(c2scc(C(=O)OC)c2)c2nnnn2C(C)C(=O)OC)cncc(C#N)c1 c1(C(c2nnnn2CC2CCOCC2)NC2(COCC)CC2)cnccn1 C1(C(=O)N(CC(C)(C)CNC(=O)Cc2c[nH]nc2C)C)(COC)CCOC1 C(=O)(C(O)C(F)(F)F)NCC1(OC)CN(C(=O)CC2COC(C)(C)CO2)C1 C1(CS(C)(=O)=O)CCC(C(=O)NCC2CN(C(=O)C(O)Cc3cn(C)cn3)C2)O1 CC1CC=C(C(=O)NC2(CO)CCCN(c3ncnc4[nH]cnc34)C2)CC1 C1(CN(C(C2CCC2F)=O)CC)CCCN(C(c2ccc(F)cn2)=O)C1 C12(C(N3CCCC(C(=O)Nc4scc(OC)c4)C3)=O)CC1CCC2(F)F C(=O)(C(C)C(O)C(C)C)NCCCOCCCNC(CC(CCC)C)=O Nc1ncc([N+](=O)[O-])cc1C(=O)NC1CCC(NC(C2CCC(F)C2)=O)CC1 C1(NC(C(F)=CCC)=O)CC2(CCCCN2C(c2cccc3c[nH]nc23)=O)C1 c1(C(=O)NC2(CNC(CC3(C)CC3F)=O)CCCC2)ccc(N)c(Cl)n1 N1(C(CCc2ccc(C)s2)=O)CC(O)CC1CNC(C1CCCN(C(N)=O)C1)=O C1(CNC(c2cc(CC)on2)=O)CC2(CC2)CN1C(=O)C(COC)N(C)C.C1CC1 c1(C(=O)NC(C)CC(C)NC(C23CCC(CC2)CO3)=O)cc(Cl)c(F)cc1O c1(C(=O)NC(C(=O)NC)C)ccnc(CNC(=O)CCc2nnc(C)o2)c1 C1(CNC(C(N)=O)=O)CC2(CCOCC2)CN1C(=O)CC1CCCOC1 c1(N2CCC(N(CCC)C(c3ncsc3Br)=O)C2)ccc(C#N)nn1 C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCC(CN(C)C(C2(C3CC3)CC2)=O)C1 Cc1ncnc(C)c1C(N1CC(CC(C)NC(C2CCC2c2nncn2C)=O)C1)=O c1(C(N2C(CN(C(C(C)OCCC=C)=O)C)CCC2)=O)cc(Cl)cn1CC n1(CCCC)nnnc1C(C)(CCSC)NCCCn1cnnn1 C1(C(N2C(CNC(C3CCCC4CC34)=O)CCC2)=O)COc2ccc(O)cc2O1 C(=O)(C(C)CC(F)(F)F)NCc1c(C(=O)NC(CC)C2CC2)con1 N1(C(CCCS(CC)(=O)=O)=O)C2CCCC1CC(n1cc(C3CC34CC4)nn1)C2 CC1C(NC(=O)C(C)(C)c2ccno2)CCN1C(=O)Cc1csc(C2CC2)n1 c1(C(=O)NCC(CC)NC(=O)C(C)S(N)(=O)=O)cc2ncccc2[nH]1 c1(CC(=O)NC2C=NN(c3cccc(Br)c3)C2=O)ccc2c(c1)OCO2 Cc1cn2cc(C(N3CC4(CCN(C(C5(C)CCC(=O)N5)=O)C4)C3)=O)ccc2n1 CCCCCCN(CC(=O)NCC1CC1CNC(=O)CN1CCCC1)C N1(C(CCn2cc(CCCCSC)nn2)=O)CCN(CC2CC2(Cl)Cl)CC1 C1(NC(CN(C(=O)CC2CCCSC2)CCOC)=O)CCCC(O)CC1 C1(CC(=O)NCC(C)(C2CCC2)NC(C(CCCC)C)=O)CC2(CCCC2)CO1 C1(CC(N2CCC(CCNC(c3cc(C4C(C)C4)on3)=O)C2)=O)COC(C)(C)C1 C1(NC(C(C)OCCCC)=O)CCN(C(=O)Cc2cnc[nH]2)CC1O C(=O)(CCCCC(F)(F)F)NCC(C)(C1CC1)NC(=O)C=Cc1nccs1 N1(C(C(C)c2ccco2)=O)CCCC(F)(C(=O)NCCN2CCCC(O)C2)C1 N1(C(=O)CCCC2CC2)CC2(CCCCN2C(=O)C2Cc3ccccc32)C1 CC1CN=NC(=O)CN1C(=O)CCCn1cc(-c2cccc3ncnn23)nn1 O(NC(=O)COCCNC(c1ccoc1C1CC1)=O)C(CC)C CC(=O)CCCC(C)C(=O)NC(C)C(C)NC(C12CCC(CC1)CO2)=O C(C(C)(C)C(=O)N1CCN(CCN(C(=O)C(C)n2cccn2)C)CC1)OC(C)C Cc1ccccc1NC(=O)C(CC1CC1)N1CCC(N2CCCC2)C1 C(=O)(C#CC(C)(C)O)NC(C1CN(C(=O)C(O)c2ccsc2)CCO1)C O=S(=O)(c1cnc(NCC2CC3(CCC3O)C2)c(Cl)c1)N1C2CCCC1COC2 c1(CC(=O)NC2C(CNC(c3n(CC(C)C)ncc3)=O)CC2)ccc(Br)cc1 Cc1ccc(CC(=O)NC2(CNC(c3cc(-c4ccncc4)on3)=O)CC2)o1 c1(NCC(N2CC(C(C)NC(CC(=O)NCC)=O)C2)=O)ccc2c(c1)CCCC2 N1(C(c2ccc(C#C)o2)=O)CC=C(CC(=O)N2CCC(SC)C2)CC1 C1(NC(C(CC)O)=O)(CNC(=O)Cc2ccc(C(C)=O)cc2)CCOCC1 N1(C(=O)NCC2(OC)CCCCCC2)CCC(O)CC(C)C1 C(=O)(C(C)(C)Cc1cnn[nH]1)N(CCCNC(C(c1scc(C)n1)(F)F)=O)C C(=O)(C(CC)CC(F)(F)F)N1CC(N(C(COCCC#C)=O)C)C(C)(C)C1 C1(OC)C(C)(C)CN(c2nc(C)ns2)C1(C)C C(C(O)C(=O)NOCCO)NC(c1cccc(F)c1)=O Cc1ncc(CC(=O)NC(CNC(C2(c3cncnc3)CCCC2)=O)C2CC2)s1 C1(NC(C2CSCCS2)=O)CC1C1CCN(C(=O)CCC2CCC2)CC1 C1(N(C(C2(N3CCOCC3)CCSC2)C(=O)NC)C)CCC(C(F)(F)F)CC1 CC1CCC(C(=O)N(C)CC2CCCS2)N(C(=O)COCCCN(C)C)C1 N1(CC(=O)NCC(C)(CO)NC(CC)=O)C(=O)CC(C)(C)C1=O c1(OC)cc(F)c(C(N2CC(C)(NC(=O)CC3C=CCC3)C2)=O)c(Cl)c1 c1(C(c2nnnn2C2CCC2)NC(C)C(C)(C)F)ccccc1C(C)(F)F C#CC1CN(C(C2(C(C)C)CCN(C(=O)CCc3nncs3)C2)=O)CCO1 N1(C(C2CC(O)(CC#C)C2)=O)CCC2C(C1)CN2C(=O)CC(C)c1ccncc1 c1(OC)csc(C(N2CCN(C(=O)Cc3ccccc3Cl)CC2)=O)c1OC C1(SCc2cn(C(COCC)C(=O)N(C)CCC3CCC3)nn2)CCCCCC1 n1(CCC(N2CC(CNC(C3CC(=C)C3)=O)OCCC2)=O)cc(S(N)(=O)=O)cn1 N1(C(C(CC)(C)F)=O)CC(NC(c2cc3c(s2)CCC3)=O)C2CCCC2C1 c1(C(N2CCC(CCC(=O)NC(C3C(C(=O)OC)C3)C)C2)=O)sc(O)nc1C c1(C(=O)NCC(CNC(C(C(=O)OCC)(C)F)=O)C)cccc2c1OCC2 C1(C(=O)NC2(C)CC3(CCC3)C2)CC2CN(C(c3cc(F)cc(F)c3)=O)CC2C1 Cc1nc(CC(=O)NC2CCCC(NC(C3(O)CCSC3)=O)C2)c(C)s1 c1(C(=O)NC(CCNC(CC(CC)OC)=O)C(C)C)cccc2oc(C)cc12 C1(C(=O)NCC2(CC)CCC(=O)N2)CN(C(c2ccsc2C#N)=O)CC1C1CC1 C1(C(=O)NCC2(NC(=O)Cn3cc(Br)cn3)CCOC2)CC2CCC(C1)O2 c1(SCC)nnc(N2CCC(C(F)F)CC2)n1CCCSc1csc(C)c1 C1(NC(c2n[nH]c(C)c2C)=O)CCSC12CN(C(c1cc(C3CC3)n(C)n1)=O)C2 N1(C(c2cnc(CC)s2)=O)CC2CS(=O)(=O)CC2(NC(=O)C2=CCSC2)C1 c1(CC(N2CCCC(NC(C(OC)OC)=O)CC2)=O)cn2cccc(C)c2n1 C1(C(N(CC(C)NC(C2(CO)CCC2)=O)C)=O)CCCC(N(C)C)C1 C1(OC)CCCC(CC(N2CC(CCNC(=O)CCC3CCCC3)C2)=O)C1 c12cc(ccc1F)NC2=O.CC(C)(C(=O)NCC(=O)NOC(C)(C)CO)C1CC1 N1(C(CC2C(C)C2)=O)CC(C2CCCN(C(C3CCC(=O)N3C)=O)C2)C1 C1(CC(=O)NCCCCCN(C)C(c2ccsc2)=O)COc2ccccc2O1 c1(C(=O)NC2CC(N(C)C(C34CCC3C4)=O)C2)cccc(-c2ccc[nH]2)c1 CCC(C)C(=O)C(=O)NCC(CNC(=O)Cn1nc(C)oc1=O)OC C1(COC)CN(C(c2cccc(CO)n2)=O)CCN1C(=O)C(C)CC(=O)OC N1(C(C2(CC)CCOC2)=O)CCC2CN(C(=O)CC34CCC(CC3)C4)C2C1 CCC1c2ccsc2CCN1Cc1c(OC)cccc1C C(=O)(CC(C)P(C)(C)=O)NCC1(C(C)NC(c2c[nH]nc2C(F)(F)F)=O)CC1 Cc1ncc(Cl)cc1CC(=O)NC1CN(C(=O)CCF)C(C)(CO)C1 c1(CC(=O)OCC(c2ccc(F)cc2)C)ccc(C(F)(F)F)cc1 N1(C(c2c(C)cn(C)n2)C(=O)NCCC2(C)CC2)CCC(C)CC(C)C1 c1(C(=O)NC2CC(CCNC(C(C)n3ccnc3)=O)C2)cnc2nccn2c1 c1(C(=O)NCC2CCN2C(c2scnc2C(F)F)=O)ccc2c(c1)NCC2 C(=O)(C1=CCCN(C(=O)Cc2ccn(C)c2)C1)N1CC(C)C(N(C)C)C1 CCC(C(=O)N1CCC(CNC(c2ccc[n+]([O-])c2)=O)CC1)C(C)O C1(=CCNC(c2ccc(C)s2)=O)CCN(C(=O)Cc2cccnc2)CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NC2CCN(C(C3CCC(=O)NC3)=O)C2)c1Cl c1(C(N2C(C)(C(=O)O)C=CC2)=O)ccc2oc(O)nc2n1 Cc1nc(N(C)C)sc1C(N1CCC(CCNC(c2ccc(F)o2)=O)C1)=O c1(C(NC(=NC)NCC(COC)OCC)C#C)ccccc1Br C1(NC(CCCNC(COC)=O)=O)CCC(CNC(=O)C(C)(C)NC(C)=O)CC1 C1(C(=O)NCC(C2CCN(C(CC(C)(F)F)=O)CC2)O)CC2C=CC1CCC2 C1(NC2(C(N)=O)CCCCCC2)CCc2c(cnn2CCC2CCCC2)C1 c1(NC(CC2CCCC(NC(c3c(NC)scn3)=O)C2)=O)cc(O)cc(F)c1 c1(-c2nnc(N3CCC(CCOC)C3)n2C)cc2sccc2s1 C1(COC)(NC(=O)C(F)C(C)C)CCCN(C(=O)CC2(N3CCCC3)CC2)C1 C1(C(=O)NC(C(C)NC(CCNC(C=C(CCC)C)=O)=O)C)CCCCN1CC c1(C(C)C)nnc(CC(N2CCC2CNC(c2ccc(-c3cccs3)o2)=O)=O)o1 N1(C(CCCOC(C)=O)=O)CC(CNC(C2(C3CCCCO3)CC2)=O)C(O)C1 N1(C(CN(C(=O)NCC)C)=O)CC2CC1CCN2C(=O)CC(C)(C)OC N1(C(c2c(C)noc2C)=O)CCOCC(NC(=O)C=Cc2ccn(C)c2)C1 c1(OC)ncc(C(=O)NCC2(C)CCN(C(C3CCC4(CC4)C3)=O)CC2)cc1C C(=O)(CS(=O)CCC(F)(F)F)NC1(C)CCCN(C(c2cc(O)cc(F)c2)=O)C1 C12(CNC(c3c(COC)noc3)=O)CC(NC(C3CC3(C)C)=O)(CCO1)C2 C(C1CCCC1)=CC(N1C(CNC(C(c2cncn2C)N(C)C)=O)CC1)=O C1(NC(C(C)NC(CC)=O)=O)CCC(CCNC(C2(C(=O)N(C)CC)CC2)=O)C1 CCCCS(=O)(=O)CC(=O)N1CC(NC(c2cc(F)ccc2Cl)=O)C(C)C1 N1(C(C(CC)SC)=O)CCCN(C(c2ccc(OC)c(OC)c2C)=O)CC1C C1(CNC(CCC(N)=O)=O)(NC(c2cnn3c2OCC3)=O)CC2CCC1C2 c1(C(N2CC(CN(C(C(F)OC)=O)C)OCC2)=O)ccc(F)c(N(C)C)c1 C1(C(=O)NCC(n2ccnn2)C)CCN(C(=O)CSC2CC2)C12CCC2 c1(NC(=O)CCN(C(C2CC2(F)Cl)=O)C2CC2)cccc(CCO)c1 c1(C(N2C(CNC(C=C(C)C)=O)C=CC2)=O)cncc2nc(C(F)(F)F)n(C)c12 c1(CCC(=O)NCCCOCCN(C(C(C)C)=O)C)cccc(O)n1 C(=O)(CS(=O)(=O)C(C)C)N1C(CNC(CS(CC)=O)=O)C(O)C(O)C1 CCC1=C(C(=O)N2CCCN(C(C3CCCN(C(N)=O)C3)=O)CC2)CCCO1 C1(CC(=O)NCC(C)CNC(C2CC3(CCC3)CO2)=O)CCOC(C)(C)C1 CCC(CC(=O)NCCCC1(NC(c2cc(C#N)c(C)cn2)=O)CC1)C(C)C C1(CNC(C(=C(C)C2CC2)F)=O)CN(C(c2ccc(N)c(N)c2)=O)CCC1(F)F C1(CC(=O)NC(C2CN(C(C3(C)C(C(=O)OC)C3)=O)C2)C)CCCN(C(C)C)C1 N1(C(c2ccc(OC)c(C)c2)=O)CC(NC(=O)C(C)OC2CC2)CC2(CCC2)C1 N(C(=NCCn1ccnc1)N1CCN(S(C)(=O)=O)C(C)C1)C(CC)C N1(C(C2CC(SC)C2)=O)C2CCC1CC(N(C)C(C1(O)COC1)=O)C2 C(=O)(C(C(=O)NC(CCC(F)Cn1cc(Cc2nncs2)nn1)=O)OC)OC c1(C(=O)NCC(CNC(=O)CCn2cccn2)F)ccc(Br)cc1F CN(C)C(=N)N1CCN(C(c2cnc(C3CC3)[nH]2)=O)CC1 c1(NC(C2N(Cc3c(C)nc[nH]3)CCC2O)=O)c(Br)c(CN(C)C)nn1C Cc1c(C(=O)NC2CCCCN(C(C3(CO)CCC3)=O)C2)nn(C)c1N C12(CNC(C(C(C)C)O)=O)CCC1CN(C(=O)CCC(C)(C)F)C2 c1(CC)nn(C)c(CC(=O)NCC2(F)CC(NC(=O)Cn3cccc3)C2)c1Cl CC(CC(=O)NCCC1(O)CCCC1)C(C)(C)NC(c1coc(CO)c1)=O C1(CCC)CN(C(=O)C(c2ccc(C)s2)C)CC1NC(=O)COCC1CC1 N1(C(C(C)C(F)F)=O)CCOCC(NC(=O)C(F)(F)CN(C)C)C1 CC(C)C(C(C)NC(C1(C(F)F)CCC1)=O)NC(=O)CC=C(Cl)Cl C1(C(=O)NC2C3(CN(C(c4c(C)ocn4)=O)C3)CC2)CCc2nnc(O)n2C1 C=C=C(C)CC(=O)NC1CC(CNC(C2CCN2C(C)(C)C)=O)C1 c1(-c2ccc(NCC(N3CCCC4(CCOC4)C3)=O)cn2)ccc2c(c1)CCO2 N1(Cc2cccc(C=O)c2Cl)CCC2CN(S(=O)(=O)N(C)C)CC12.N(C)(CC)CC n1(CCCC(=O)N(CC(CC)(C)O)C)c(C)cc(=O)cc1C c1(COC)ccc(NC(C2CCCN(Cc3cc([N+](=O)[O-])cs3)CC2)=O)c(C)c1 C1(CC(=O)NCCCCN(C(C)C)C)CN(C(C2COC(=O)N2)=O)CCO1 c1(C(=O)NC2C(NC(CSCC=C)=O)CCC2)cc(N2CCC(O)CC2)ccn1 C(=O)(C(F)C(C)(F)F)NC1CC(C(N(c2ccc(O)cc2)CC)=O)C1(C)C O=C(CCC(=O)c1cccc(Cl)c1)NCCCCO.n12cc(nn1)CCOC2=O C1(NC(CC2N(C)CCCC2)=O)COC2CN(C(=O)Cc3sccc3Cl)CC12 c1(C(=O)NCC(C2CCN(C(C(C=C)O)=O)CC2)C)cc2ncccn2n1 C1(NC(C2C(C)C2C)=O)C2CC3CN(C(c4cncc5ccccc45)=O)C1C3C2 c1(OC)cc(OC)c(N(C2CC3(CNC3)C2)C(c2cc(C)c(F)cc2Br)=O)cc1Br Cc1ccc(C(=O)NCC(C)CNC(=O)C(C)N(C)C)c2cccnc12 N1(C(CS(C(C)C)(=O)=O)=O)CC2(C1)CN(C(=O)CN(c1ccncc1)C)CCO2 CCC(C)(F)C(=O)NC1C2CN(C(c3c[nH]nc3-c3ccc(Cl)nc3)=O)CC12 CC(C)(CC(F)C(=O)NCC1CSCCO1)NC(=O)CC1CCCCC1 C1(N(C(CCCC#C)=O)C)CN(C(=O)C(n2nc(C)cc2C)C)CC12CC2 c1(C(C(=O)N(CC(C)Nc2ncc(C(=O)OC)nc2)C)O)ccc(F)c(Cl)c1F CCS(=O)(=O)c1ccccc1Nc1cnn(CC(C)(C)O)c1C c1(C(=O)NCC(C(C)(C)C)NC(C2(C3CCC3)CC2)=O)cccc2ccnn12 c1(CNC(C(=O)NC23C(CN(C)C2)C3)=O)cn2c(n1)CCCC2 C1(O)(C(=O)NCC(CNC(C(C)c2ccco2)=O)F)CC(C)(C)C1 c1(CC(=O)NC2C(F)CCN(C(C3(SC)CCC3)=O)C2)ccc2c(c1)COCC2 C1(CNCCSCC(=O)NC(CC2CC(=C)C2)=O)CC2C=CC1C2 C1(C2(O)CCC2)(C(=O)NC(c2cccnc2)C(=O)NCc2c(CC)nco2)CC1 CC1(C)CC(N)CC(C(N2CCCC(CN3CCCC3)C2)=O)O1 C1(C(=O)NC2CC(C)N(C(=O)Cc3cccc(N)c3N)C2)CCc2c[nH]nc2C1 C1(CC(=O)NCCN(CC(C)O)C(C2C=C(C)CS2)=O)CC(CC)=NO1 c1(C(=O)NC(CC)CN(C(=O)CCOCCCOC)CC)cc[nH]c(=N)n1 N1(C(=O)CO)CC2CCN(C(c3cnc(N4CCS(=O)(=O)CC4)nc3)=O)C2C1 C(=O)(C(C#N)C(C)C)NC(C(=O)NC(c1c(C)nc(C)[nH]1)C)C(C)C c1(C(=O)NCC2N(C(C(CCC)C)=O)C3C(C2)C3)cnc2sccc2c1 C1(CC(=O)NC2(CC=C)CN(C(c3c(C)ncn3OC)=O)C2)CCCNC(=O)C1 C1(C(N2CCC(C(=O)NC3(C=C)CCC3)C2)=O)CC1C1(C)COC1 c1(C(=O)NC2CC(C)(NC(C(C)SC)=O)C2)ccc(N)cn1 C1(C(N(c2ccc(SC)cc2)CC)=O)COC2(C1)CN(C(=O)C(CSC)OC)C2 c1(OC)ccc(Cl)c(C(=O)NC2CN(C(=O)C(C)CC(N)=O)C3(CCC3)C2)c1F CCC(C)(CNC(=O)COC1(C)CCC1)C(=O)N=c1ccn(C(F)F)[nH]1 C1(NC(C2(NC(C3N(C(C)=O)CSC3)=O)CCCC2)=O)CC(=O)N(C(C)C)C1 N1(c2scc(C)n2)CC2C(C3CCCN3C(=O)C(F)(F)F)C2C1.C(=O)C1=NOCC1 C(=O)(CC(C)CC(C)C)N1CCCC(O)(CN(C(c2cnc(C)o2)=O)C)C1 C(=O)(C(O)CC(C)(C)C)N(CCNC(C(c1c(OC(C)C)cccc1)(F)F)=O)C C(C(C)(F)CNC(=O)CNC(c1ccccc1)=O)NC(CN(CC)CC)=O N1(C(c2ccc(=NCC)[nH]c2)=O)CC(C)CN(C(=O)C(C)COC)C(C)C1 C1(C(N2C(C(C)NC(CC=C)=O)CCC2)=O)CN(C)C(=O)N1 C1(C(=O)NC2CCN(C(=O)CCCN3CCCC3)C2)CCCC2(C1)CC2(F)F n1(CC2N(C(CN(C)C(C)=O)=O)CC2)cc(CCN2CCOC2=O)nn1 C1(C(=O)NCC2(NC(C(C)OC)=O)CCC2)CN(S(N)(=O)=O)C1 C1(C(=O)N(C2CCN(C(c3coc(C)c3)=O)CC2)C)(OC)CCS(=O)(=O)C1 CC1CN(C(=O)CCc2ccoc2)CCC1NC(c1nnn(C(C)(C)C)n1)=O c1(CN(C(=O)CCC2CCC(=O)N2)C)cc2nc(Cl)ccc2s1 c1(C(N2CC(NC(C(COCC)C)=O)C2)=O)ccccc1C(c1ccccn1)=O Cc1cc(Br)c(C(N2CC(CNC(=O)CCCn3cccc3)C2)=O)cc1F c1(OC)ccc(CC(N2CCCC(CN(C(=O)Cc3cnccn3)C)C2)=O)nc1 c1(C(N2CCC(N(C(CSc3c(C)n[nH]c3C)=O)C)C2)=O)ccc(S(C)(=O)=O)s1 C12(CNC(CC#N)=O)CCC(CNC(C3CCCC3O)=O)(CC1)CO2 N#Cc1ccncc1C(N1CCC(C(=O)NCCN2C(=O)CSC2=S)C1)=O C(C(O)C(=O)N1CC(C(N)=O)(CNC(=O)C(C)(C)C2CCCCC2)C1)N(C)C N1(CC=C)C2CCC1CC(NC(=O)C(C)c1ccsc1)C2 c1(CCC(=O)NC2CN(C(C(CCC)(C)C)=O)CC2O)nc2cccc(C)c2[nH]1 C(=O)(C(C)(C)C(F)(F)F)NCC1CCN(C(c2c(CC)n(CC)nc2)=O)CC1C O(N(C(=O)c1occc1Cc1cn(-c2cnn(C)c2C)nn1)C(C)C)OCC c1(C(=O)NCC2(C)CCN(Cc3cc(C)cc(F)c3)CC2)cnn2ncccc12 c1(OC)cccc(CNC(C2CC(F)CN(C(C3CCCC3)=O)C2)=O)c1F NC1CCCOc2cc(F)ccc21.c1(NC)cccc(CN(CC(=O)NC)C)c1 N1(C(c2c(CC)c[nH]n2)=O)CCCC(C2CCCN2C(=O)CO)C1 c1(OC)cccc(C(F)(F)C(=O)NCCCC(C)NC(=O)CC2CCCOC2)n1 c1(C(=O)NCCCCC2CN(C(C(C)SCC)=O)C2)cncc2nc(O)[nH]c12 Cc1nc(C)c(CNC(C2CCC(CNC(c3cccnc3C)=O)CC2)=O)[nH]1 CC1CCC(NC(=O)Cc2nccn2C)CN1C(c1ccc(C(F)(F)F)nc1)=O c1(OC)cc(C(=O)NCC2CCCCC2(C)NC(=O)C(C)N(C)C)cnc1OC n1(CCC=C)c(N2CCCC2C2CCC(=O)NC2)nnc1C1(C)CC1 N1(C(c2c(C)nc[nH]2)=O)CC(NC(=O)Cc2cc(C)n(C)n2)C(F)C1 c1(NCC(C)C2CCC2)ccc(S(=O)(=O)NCC#CCCO)c(Cl)c1 C1(C(=O)NC)(Cc2ccccc2)CCN(C(=O)Cc2ccc(O)nc2)C1 c1(C(N2CCCC(F)(CNC(c3cnn[nH]3)=O)C2)=O)cc(F)c(Cl)cc1Cl C1(CN(C)Cc2ncsc2Br)CCN(C(=O)C(=O)N(CC(F)F)C)CC1 N1(C(C(CC)N(C)C)=O)CC2CCN(C(c3cccc(CCO)c3)=O)CC2C1 CCC(O)CC(=O)N=c1ccn(C2CN(C(c3cccc(I)c3O)=O)C2)[nH]1 C1(CC(N2CCC(NC(CC(=O)OC)=O)C2)=O)CCCC(C)(C)O1 N1(C(C(C2CC2)NC(C2(C)CNC(=O)N2)=O)=O)CCC2(CO)CCCC12 C(=O)(CP(=O)(C(C)C)C(C)C)NCC(CNC(=O)Cc1ccc(F)cc1C)OC C(CC(C)C)(C(=O)NC(CCO)C1CCC1)N(C(c1ccn(CC)n1)=O)C c1(NC(CN2CCN(C(CC(CC)C)=O)CC2)=O)c(O)ccc2nc[nH]c12 C1(C(N2CCC(C)(COC)C2)=O)CN(C(=O)CN2CCCCC2C)CCN1C C=CCC(C)(C)C(=O)N1CC(F)(F)CC1C(=O)NCc1c(Cl)cncc1Cl C1(NC(C(C)(C)CO)=O)CN(C(c2ccc(N)c(OCCO)c2)=O)CC1C1CC1 C1(OC)CC2(CCN(C(c3cn(CC(C)C)nn3)C(=O)NC(C)C)CC2)C1 c1(NC(C)C)ncccc1C(=O)NCC1CN(C(c2ccc[nH]2)=O)CCO1 c1(C(N2CCN(C(C3CCCS3)=O)CC2C(F)(F)F)=O)cc2ccc(Cl)cc2s1 C(CC(C)(C)C(=O)NC(C)Cc1cc(C)[nH]n1)NC(CCC=C(C)C)=O c1(CC)nn(C)cc1C(N1CCC(C(=O)NC(C)C2CC2)(CF)C1)=O c1(OC)ccc(C=CC(N2CCC(NC(=O)CC3CC4CC4C3)CC2)=O)cc1Cl c1(OC(C)=O)ccc(F)c(C(N2CC(NC(=O)C(C(C)C)NC(N)=O)C2)=O)c1 S(=O)(=O)(C1CC2(CC2C(=O)O)C1)CN1CCCCC(C)(F)C1 N1(C(c2c(SCC)cccc2)=O)CC(C2CN(C(c3cc(CC)oc3C)=O)C2)C1 c1(C(C(=O)CCc2cscn2)=O)cncc(CO)c1.C1(O)(CCN)CN(C(=O)C2CC2)C1 C1(CNC(C(c2cnccn2)C)=O)CCCC2CN(C(C3(C4CC4)CC3)=O)CC12 CC1CN(C(c2ncnn2C2CCOCC2)=O)CC(C)N(C(C2CCOC2)=O)C1 Cc1cc(N)c(C(N2CCC(CNC(C3(n4ccnn4)CC3)=O)C2)=O)c(F)c1 CC(C)C(F)(CNC(=O)C(C)SC1CC1)C(=O)NOC1CC2CCC1C2 c1(C(=O)NCCN(C(=O)CCC(N)=O)CCOC)cccc2sccc12 c1(C(C(=O)NCC2N(C(c3c(C)nc[nH]3)=O)CC2)(F)F)c(C)noc1C C(=O)(CC(C(F)F)NC(=O)C(F)=CC1CC1)N1CCC(OC)C1C(C)C CCC(C(C)(F)F)NC(=O)CN(C(=O)C=C(C)C1CC1)C Cc1ccc2c(=NCC3OCCOC3(C)C)[nH]c(=NCCC(C)C(C)C)[nH]c2c1 n1(CCCCC(C)NC(=O)NCC(CC(C)=O)(C)C)c(O)nc2ccccc12 c1(CCSc2c(C)oc(C(C)(C)C)c2)cc2c(O)ncnc2cc1F c1(C(=O)NCC2CN(C(CC(C)(C)O)=O)C3C2C3)sccc1S(N)(=O)=O c1(OC)cnc(F)cc1C(N1CC(NC(=O)CCn2cc(C)cn2)CC(C)C1)=O c1(CC)cc(Cl)ccc1C(=O)NC(CNC(c1cnc(C(C)(C)C)[nH]1)=O)C1CC1 c1(C(CCSC)NC(=O)C(C)=CCN)ccccc1[N+](=O)[O-] C1(C(N(CC(CCC=C)O)C)=O)CCN(C(c2ccn(C)c2)=O)C12CC2 N1(C(C2C(C(F)(F)F)CC(=O)N2)=O)CCC12CN(C(=O)C=CC1CCOCC1)C2 Cc1cn2c(=O)c(C(N3CCSCC3C(=O)NCc3ccncn3)=O)cnc2s1 c1(CC(=O)NC2C(NC(CC(C)n3ccnc3)=O)COC2)cnn2c1CCCC2 Cc1cc(CNC(c2nnnn2CCN2CCOCC2)C23CCCC2C3)cc(Br)c1 N1(C(C(C)n2cccn2)=O)CC2(CCCN(C(C3(CF)CCC3)=O)C2)C1 C1(NC(C=CC)=O)CCSC12CN(Cc1cncc(-c3ccc(C)cc3)c1)C2 Cc1cc(C)c(C(=O)NCC2CCCCN2C(c2cnco2)=O)c(O)c1 N1(C(C)COCCO)C(=O)NC(Cc2ccccc2)C1=O C1(CC(=O)N(C(CNC(Cc2cc(C)sc2C)=O)C)C)Cc2cc(F)ccc2O1 C1(N(C(c2ccsc2)=O)CC)CCCN(C(=O)C(C2CCOCC2)F)C1 N1(C(COCc2n(C)ncc2)=O)CCCC(C)(NC(c2ccc(F)o2)=O)C1 C(=O)(C1CCCn2c(Br)cnc21)NC1(CNC(C2CSC2)=O)CC1 C(=O)(CCCCC(F)(F)F)NC1CN(C(CS(CC)=O)=O)CC(C)(C)C1 CCCCC(CNC(C1CC(C)CO1)=O)NC(c1oc(C(=O)OC)cc1C)=O C(=O)(C1=CS(=O)CCC1)N1CC(C)C(NC(c2nccc3ccncc23)=O)C1 C1(C(N(C2CCS(=O)(=O)C2)CC#C)=O)CC2(CCOC2)C1 C1(C2CC2)(C(=O)NC2(c3ccc(C(F)(F)F)cc3)CC2)CCC1 C=CCCCC(C(=O)NCC1(CO)CC(C)(C)C1)NC(c1coc(C)c1)=O c1(NC(=O)NC2C(C)COCC2)cnc(Cl)c(Cl)c1 C1(NC(C2C(C)C2C)=O)Cc2ccccc2N(C(=O)C2=CCCOCC2)C1 N1(C(Cc2onc(C)n2)=O)CCOCC(NC(C2CCN2C)=O)C1 C(CS(=O)(=O)Cc1cn(CCOC(C)(C)C)nn1)C(=O)OCCCCC1C(C)C1 c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)C)nc(=N)cc[nH]1 N1(c2snc(CC)n2)CCCC(NC(c2ccc(-n3cccn3)c(C)c2)=O)C1C CC(C)CC(C)C(=O)NCCSCC(=O)NC(C)C(=O)NCCF Cc1ccc(CNC(C2CCN(C(c3cccc(Cl)c3)=O)CC2)=O)cc1 N1(C(C(N)=O)=O)CCOCC(F)(CNC(c2ccoc2C(F)(F)F)=O)C1 C1(NC(C2C(C)(C)CO2)=O)CCCC2CN(C(=O)C(C)(O)C3CCC3)CC12 c1(C(C(=O)NCC(=C)C)N(C)Cc2snnc2C)cccc(C)n1 CS(=O)(=O)CC(=O)NCC1CCN(C(c2cnc(-c3ccccc3)cn2)=O)C1 N1(C(C(=O)NCc2ccccc2)=O)CC2=C(C1)CN(C(=O)Cc1csc(Cl)c1)C2 Cc1cccc(CN(C)C(C2CC(CN)C2)=O)c1.c1cc(C)c(Br)s1 C1(CNC(c2cc(C)nnc2O)=O)N(C(=O)C(C)NC=O)CCCC1(C)C N1(CCC)C2(CCC(CCO)C(=O)N2C(C)C)C(=O)N(C)CCCC1=O Cc1[nH]nc2ncnc(N3CCCN(CCc4ccccc4)CC3)c12 N1(C(C(CCC)F)=O)CC2(CCCC2NC(c2nc(C)c(C)s2)=O)C1 c1(C(N2CC(NC(C3(OC)CCSC3)=O)C2)=O)ccc2[nH]nc(C(F)(F)F)c2c1 N1(C(C(Cn2ccc(C)n2)F)=O)CCC(c2cn(C3(C(=O)O)CC3)nn2)C12CC2 C1(C(N(C2CCN(C(C3CSC3)=O)CC2)C)=O)CC=CC(O)C1.CCCC c1(C(=O)NCc2c(CNC(=O)COCCF)nccc2)ncc2c(F)cccn12 C1(C(=O)NC(CNC(CC(=O)NCC2CC2)=O)C2CC2)CCC(F)CC1 C1(C)(NC(C(CCOC)NC(=O)CN2CCNC(=O)C2)=O)CCC(=O)NC1=O C(=O)(CC1CCc2cc(Br)ccc21)NCC(CNC(CSCCCC)=O)O Cc1ccc(S(=O)(=O)NC2CCN(C(c3cc4cccn4cn3)=O)C2)c(C)c1 CCC(CC)C(=O)N1CC(NC(c2coc(O)n2)=O)C(C)C1 S(=O)(=O)(c1cnc(C(F)F)s1)NC1(C)CCN(C(=O)OC(C)(C)C)C1 C(C(C)C(=O)N1CCC(C(=O)NCC(C)(C)OCCO)C1)OC c1(C(=O)NCC2(C)C(C)CN(C(CC(CC)OC)=O)C2)cccc2[nH]ccc12 N1(C(C=CS(C)=O)=O)CCCC2(C1)CN(C(c1[nH]nnc1-c1ccccc1)=O)C2 C1(C(=O)NCC(C=C)(C)C)(CNC(C2CC(CC)C2)=O)CC12CCC2 N1(C(CC2(OC)CC2)=O)CCN(C(=O)Cc2c(Cl)cnn2C)C(C2CCC2)C1 C(CCC(C)C(=O)N1CCN(C)CC1CNC(c1ccc(Cl)nc1C)=O)OC N1(C(CSCC=C)=O)CCC(=O)NC2CN(C(=O)CCc3cc(C)no3)CCC12 C1(CNC(C(C)N(C)C(C2(C#N)CCC2)=O)=O)CCCC1(C)C c1(OCCC)ccc(C2(C(=O)N(C3CCCC(N)C3)C)CCCCC2)cc1 N1(C(CC2(NC(C)=O)CC2)=O)CC2CCC1CN2C(=O)CN1CC2C=CC1C2 Cc1cc(C#N)ccc1C(=O)NCC#CC(=O)NC1(c2cccs2)CC1 C1(CNC(COCCCC)=O)CN(C(=O)C(c2ccc(Cl)nc2)(F)F)CC1(C)C C1(=O)C(C(C)(C)C)OCC(=O)NC2CCN1C2.C(=O)(C(C)CN(C)C)NC CCCC(O)CC(=O)NCCCN(C(=O)C(F)(F)C(F)F)CC N1(C(c2cnn(C)n2)=O)CCC(C(=O)NCCC2CCC(C)(C)O2)=C(F)C1 C1(C(N2C(COC)CN(C(=O)CN(C)C(N)=O)CC2)=O)CCc2c(nnn2C)C1 C12(C(=O)NC(CCC=C)CO)CC(C)(CN1C(C1CCCCCC1)=O)C2 N1(C(CCOCCC)=O)CCC(O)(CCNC(c2cccnc2CC)=O)CC1 C(c1ccccc1)=CC(=O)NC(C(=O)N(CCOC)CC1CC1)C Cc1cc(Cl)ccc1C(=O)NCC(CNC(c1cccc(C2CC2)c1)=O)CO c1(C(=O)NCc2ccc(C(N(C)CCc3nnc(O)o3)=O)s2)ccccc1C#N Cc1nc2ncccc2cc1C(=O)NC1CN(C(C2CC2C(N)=O)=O)C1 C(=O)(C#CC1CCCCO1)NC1CCC(C)N(C(=O)CC2CCC(=O)NC2)C1 C(CC(=O)c1ccccc1)(C(F)F)NC(=O)NCCNC1(OC)CCCC1 CCCC(O)CC(=O)N1CC(CCNC(C2CC(n3ccnn3)C2)=O)C(C)C1 C=C1CCN(C(=O)C(C)=C2CCCC2)C(C(=O)NC(C)C(C)(C)O)C1 c1(C(C=CC(=O)N(C2CCC(NC(c3csc(Cl)n3)=O)C2)C)=O)ccc(F)cc1 N1(C(C=C(CNC(CCOCC)=O)C)=O)CCC(CO)C(F)(F)C1 C1(CNC(c2n(C)ncc2)=O)CCCC2(CN(C(=O)CCC3CC3CC3CC3)C2)O1 N1(C(C(c2ccccc2)SC)=O)CCC(C(C)NC(c2cnc(C)[nH]2)=O)CC1 CC(O)C(F)(F)C(=O)N1CCC(NC(=O)C(c2ccc(F)c(F)c2)C)C(C)C1 C(c1cnc(C)nc1O)=CC(=O)NCCCCNC(COC)=O N1(C(C2CCN(CC)C2)=O)CC(C(=O)NCc2cscc2C)CC1(C)C N(C1COc2cc(Br)ccc21)C(=O)Nc1c(C)ccc(CS(N)(=O)=O)c1 C(C(CNC(c1cnnn1CC)=O)S(C)(=O)=O)NC(c1cncc(CC)n1)=O CC(C)CC(C(=O)NC1CCC(NC(=O)CC(O)c2ccccc2)CC1)N(C)C S(=O)(=O)(c1cnccc1NC1CC(C)n2ncnc21)NC(c1ncc(C)s1)(C)C N#Cc1cc(S(=O)(=O)NC2CC(CNC(=O)Cc3cccnc3Cl)C2)ccc1F N1(C(CC(=O)OCC)=O)CCCC2(CCCN2C(=O)C(C)CSC)C1 C(c1ccc(Cl)nc1)=CC(=O)NCC(C)NC(C(C)=CC1CC1)=O C1(CC(=O)NCCC2CCCCC2)CN(C(=O)CC2CC3C=CC2C3)CC12CC2 CC1CC(CO)CN(C(C2CCN(C(c3coc(N(C)C)n3)=O)C2CO)=O)C1 c1(-c2cc(F)c(C)c(F)c2)nc2c(s1)CC(C(=O)NCC13CCN(CC1)C3)CC2 N1(C(c2cc(C)c(F)cn2)=O)C(C(=O)NC2CC3CC3C2)C2CC(O)C1C2 N1(C(C2CN(CCOC)C(=O)C2)=O)CCn2nc(C(=O)Nc3cncs3)cc2C1 c1(C(N(CCC(C)NC(C(C=C)O)=O)C)=O)cccc(F)c1 N1(C(c2c(C)nc(O)cc2)=O)CCC2(CCOC2)C(CNC(=O)C(C)CO)C1 N1(C(C(=O)N(C(C)CO)CC=C)=O)CCOC2(CCOC2C)C1.C(COC)N C#CC#CC(C)(C)NC(=O)CC(CNC(=O)CN1CCNC1=O)C1CCC1 C(N=c1nc(NCc2cc(C(C)(C)C)n[nH]2)c2sccc2[nH]1)c1c(CC)[nH]nn1 C1(C(=O)NCCC)(Cc2ccccc2)CCCN1C(=O)C(F)=C(C)C C(C1=NOC2CN(C(=O)Cc3ccccc3O)CC12)NC(c1cc(CC)no1)=O Cc1ccc(OCCC(=O)NC2CN(C(c3ccncc3Cl)=O)CC2F)cc1C N1(C(C)=O)CCc2cc(C(=O)NC3COC4(C3)CN(C(=O)CNC=O)C4)ccc21 c1(C(=O)NC(C(C)(C)CO)c2n(C)ncc2)cccc2c1NCCC2 C=CC1(C(=O)NCCc2cc[nH]n2)CCN(C(c2ccoc2CC)=O)CC1 c1(OC)ccc(C(N2CCC(OC(=O)N(C)C)CC2)C(=O)NC)c(C)c1 C1(C(=O)NC(CNC(C(C(C)C)OCC)=O)C)Cc2cc(OC)ccc2O1 C(=O)(CCC[N+](=O)[O-])N(C)CC1OCCN(C(C=C(C)I)=O)C1 C(=O)(C(C)(C)CC(C)(C)C)N(CCOCCNC(CC(C)n1cccn1)=O)C N1(C(CCc2n(C)cnn2)=O)CC(CNC(=O)C2=CCC2)C(F)(F)C1 c1(NC(=O)OC(C)(C)C)cc(NC2CCC3CC23)ncn1 c1(OCCOC)ccccc1C(N1CCC(CNC(c2nccnc2N)=O)C1)=O CC(C)(C#N)C(=O)NC1CN(C(c2coc(C(F)F)c2)=O)CC1c1ccccc1 C1(C(N2CCCC(C(N(C3CCCCC3(F)F)C)=O)C2)=O)CCCC2(CC2)C1 C1(OC)CC(CNC(=O)Cc2ccon2)N(C(c2cc(Br)c(C)o2)=O)C1 Cn1nc(C2CC2)cc1C(=O)NCCC1CCCN(C(=O)C(F)(F)CF)C1.CSC C1(F)(CNC(C(=O)NCCOC)=O)CCCN(C(c2ccccc2C(F)F)=O)C1 N1(C(CCc2ccc(C)o2)=O)CCC2(CC1)CC2NC(c1cc(C)nc(C)c1)=O N1(Cc2ccc(O)c(C)c2O)Cc2ccc(NC(c3cc(O)n[nH]3)=O)cc2C1 Cc1cc(C(=O)NC2CC(CC(N3CCNC(=O)CC3)=O)C2)cc2c[nH]nc12 N1(C(CC)=O)CCSCC1CCNC(=O)CC(F)(F)Br C12(C(N)=O)CCC(CNC(C3CCN3C(=O)CC3CC=CC3)=O)(CC1)CO2 c1(C(=O)NCC(C)NC(c2cc(C)sn2)=O)cccc2c1ncn2C N1(C(CC2(CSC)CC2)=O)CCC(C)(c2cn(CCN3CC(C)C3)nn2)CC1 C(=O)(CCCCC(=O)N1CC(C2CN(C(=O)C(F)(F)C3(O)CCC3)CCO2)C1)NC CC(C)(C)C(C)(O)C(=O)N1CCCC(NC(=O)COCCF)CC1 CCCC(C)(C)CC(=O)NC1CCCC(NC(=O)CCC2CCN(C)CC2)CC1 c1(C(=O)NCCOC2CCN(C(C3CC(=C)C3)=O)C2)cc2cnccc2[nH]1 N(C(=NCC1CCOC1)NC(C)CCc1ccccc1)Cc1ccn(CC)n1 C1(C(=O)NC2(CC=C)CN(C(=O)COC(C)(C)C)C2)COCC2(CCC2)O1 Cc1coc(C(C)C)c1C(=O)NCC(C(C)(C)C)NC(=O)CC(C)C1CCCC1 CC1(C)C(CC(=O)NCC2(O)CC(O)C2)CCN1C(C12CSCC1C2)=O C(=O)(C1=NOC(C)C1C)N1CCC(N(C(=O)Cc2cn(C3CC3)cn2)CC)C1 C1(C(=O)NCCCCC2CN(C(c3n(C)ccn3)=O)C2)(N(C)C)CCCCC1 c1(NC(C(N2C(CC(C)C)(CCO)CCC2)=O)=O)cnc2ccc(Br)cn12 C1(F)(C(=O)NC2CCCN(C(CN(c3cnccn3)C)=O)C2)CC12CCCCC2 C1(C(=O)N(C)CC2(C#N)CCC2)(CC)CCCN1C(C1CCCOCC1)=O CC(O)C(C)(C)C(=O)NCCN(C(c1cn(C)c(=O)cn1)=O)C1CC1 C=CC(C)(CCOC)C(=O)NCCC1(C(=O)NC2COC(C)(C)C2)CCC1 C1(NC(C2(COC)CCCCC2)=O)CCC2CC1CN2C(C1CCCOC1)=O C1(C)(NC(COCCSC)=O)CCC(NC(=O)C(O)C(C)C)CC1 c1(C(N2CCC(C)(C)C2CNC(=O)CS(N)(=O)=O)=O)c[nH]c2cnccc12 C1(C)(OCC(=O)NC2(CCOC)CCC2)CN(C(C2CCCOC2)=O)C1 C1(CNC(c2cc(COC)on2)=O)CC2(CO1)CN(C(=O)CC1(C)CCCC1)C2 Cc1nnc2ccc(NC(=O)COC3CCCOC3)cn12 C(C)(N=c1[nH]c(=NC(C)c2ccco2)[nH]c2c1COC2)c1ncc(C)o1 C(CN=c1cc[nH]c(C(F)(F)F)c1)C(=O)C1CC1.O C(C(N=c1nc[nH]s1)C(C)C(C)C)NC(c1cc(C)c2c(n1)cccc2)=O C12(OC)CCC(C(N3CCN(C(C4CC4(F)F)=O)CC3C)=O)(CC1)C(=O)C2 c1(OC)ccc(Br)c(CN2CC(c3ncccc3Br)(O)C2)c1F c1(N(CCC)C(C2CCN(C(=O)CC#N)C2)=O)ccc(Cl)nc1OC c1(C(=O)NCC2CC(NC(C3(COC)CCC3)=O)C2)ncccc1Cl Cc1ccc(C(=O)NC2CCC2NC(=O)Cc2cccc(C)c2Cl)c(C(C)C)n1 S(=O)(=O)(CC(CC(C)(C)C)OC)N1C(C(=O)NCC)C=CC1 CC12CC(C(=O)NC3CC4CN(C(=O)CN5CCOC5=O)CC34)(CCO1)C2 c1(OC)cc2nn[nH]c2cc1C(=O)N(C(C)CNC(c1cnco1)=O)C C1(NC(C(C)O)=O)CC2CC(NC(=O)Cc3cc(C4CC4)no3)CC2C1 C1(C(C(=O)N(C)Cc2cn(-c3ccccc3)nn2)F)CCCNCC1 C(CCC(C)C)(C(=O)N(CC(C1CCC1)OC)C)NC(c1ccnc(OC)n1)=O CC(C(=O)N1OC2C=CC1CC2)C1CCN(C(=O)C2=NOC3COCC23)C1 CC1Oc2ccccc2OC1C(N1CCOC(CN(C)C(C2CC2F)=O)C1)=O N1(C(c2ccc(C(C)C)cc2)=O)CCCC(O)(CCNC(=O)Cn2cnnn2)C1 C1(NC(=O)Cn2cc(Br)cn2)CCC2(CCN(C(=O)CCF)CC2)C1 c1(C(N2CCCC(F)(CNC(CCOCCOC)=O)C2)=O)c([N+](=O)[O-])cnn1C c1(C(=O)NCCN(C(CCC(=C)Cl)=O)C2CCCC2)c(C)nc(C(C)C)nc1O c1(NC(C2C(C(=O)OC)(C(C)C)C2)=O)c(C#N)cnn1-c1ccccc1Cl C(=O)(CCC(C)C)NCCCC(C)N(C(CSCC(=O)OC)=O)C1CC1 C1(C(=O)NCC(CC)NC(=O)CC2COC(=O)C2)CCn2nnnc2C1 S(=O)(=O)(C1CCN(C(=O)C(c2ccccc2)Sc2ccc(Br)cc2)CC1)NC N1(C(C(C)=C2CCC2)=O)CCOCC1CCNC(=O)C(C)n1ccnn1 C(=O)(C1=COCCO1)NC1CCCN(C(C(C)(C)C2CCOC2)=O)C1 CCC(CC)(CC)C(=O)NCCCCNC(=O)CC1CC(OC)C1 Cc1c(-c2nc(C3CC3)nn2CCCO)cnn1CCO C1(NC(CC(COC)(C)C)=O)CN(C(=O)CCc2cc(C)n(C)n2)CCC1(C)C C1(NC(C2(C(N)=O)CC2)=O)CC(NC(=O)C=CI)C1 c1(C(N(C2CC3CNC2C3)C(C)C(C)(C)C)=O)ccc2cncn2c1 C(=O)(N=S(C)(=O)CC1(C)COC1)c1c(C(=O)OCC)scn1 N1(C(CCN(C)CC)=O)C2CCC1CC(CO)C2.C12CC(C1)OC(=O)CNC2=O C1(CNC(CCNC(N)=O)=O)CN(C(=O)CC2CCCCC23CC3)C2(CCC2)C1 c1(C(N(c2cc(Cl)ccc2F)CC)=O)ccc(C#N)c2[nH]ccc12 C1(C(=O)NC(C2CCN(C(C3(C)CCC(=O)N3)=O)CC2)C)CCc2ccnn2C1 C12(CNC(c3ccc(CC)s3)=O)COCCN1C(=O)CN(C(=O)CCS(C)=O)C2 Cc1cc(C)n(C(C)C(=O)N(C)CCN(C(=O)C(C)C(=O)N(C)C)C)n1 C1(C(CO)NC(c2nc(C)sc2)=O)CCN(C(C2CCC2C)=O)CC1 N1(CCCCCOC)CCC(NC(=O)CC2(C)CC2(Cl)Cl)C(O)C1 CC(C)C(C(=O)N(CC(C)NC(C1(CCO)CC1)=O)C)Oc1ccc(Cl)cc1 c1(N2CCC(NC(C3C(C)CCC3)=O)C(C)(C)C2)ncnc2c1ccn2C N1(C(Cc2ccc(C(N)=O)cc2)=O)CC(NC(C2(F)CCC2)=O)CC12CCC2 c1(C(N2CCC(COC)(NC(=O)CN(C3CCCC3)C)C2)=O)cc2n(n1)CCC2 C1(NC(c2c(CC)scc2)=O)CN(c2cc(COC)nc(SC)n2)CC(C)(C)C1 C1(C(=O)NCC2C(NC(COCC(=O)NC)=O)COC2)CC(=O)NC(C)C1 CC1CC(C(=O)N2CCCC(C(C)(C)C(=O)N(C)Cc3ccoc3)C2)=NO1 c1(SCC(=O)NC2CC(NC(c3ncn(CC)c3)=O)C2)ccsc1[N+](=O)[O-] c1(SC(C(=O)NC2(CC=C)CN(C(=O)CCC=C(C)C)C2)C)ccc(C#N)cc1 C1(C2(O)CCN(C)CC2)(C(=O)NCC2C(CNC(c3c(C)cn(C)c3)=O)C2)CC1 N1(C(CCC)=O)CCC(CNC(c2ccnc(N3CCCC3)n2)=O)C(O)C1 CC(CN(C)C(C1CCCN1C1CC1)=O)N=c1[nH]c(C(F)F)nc(=N)[nH]1 c1(C(=O)NCC2(CNC(C(CC)C(C)O)=O)CC2)ccc2nccnc2c1 C=CCC(F)(F)CN(C)C(C1(CNC(c2ccns2)=O)CCCO1)=O CC(F)(F)C(F)C(=O)OC1CCCOC1 N1(C(C(COC)C)=O)CC2CC(NC(=O)C(C)CN3CCOCC3)C1C2 C1(CNC(C2CCC2(F)F)=O)CCCC12CCN(C(C1SCCS1)=O)CC2 C(=O)(C(C)(C)C(N)c1ccccc1)NCCC(=O)N(C(c1ccccc1)C)C CCC(C)CN=c1[nH]c(N2CC3CC=CCC3C2)nc2c1CC(C)CC2 N1(C(C(C)CNS(=O)(=O)c2ccccc2)=O)CC2CCCC(C1)C2O C(=O)(C(O)CC(N)=O)NC1CCCC(NC(CCCn2ncc(C)c2)=O)C1 N1(C(C2(C)N(C)CCC2)=O)CCC2C(C1)CN2C(=O)CNC(c1ccoc1)=O n1(CCC=C)cc(C(=O)NC(C)CN(C(=O)CC(C)N(C)C)C)nn1 CC(c1cccnc1)=CC(=O)NCC1CCCC1NC(=O)CCc1n[nH]c(=N)s1 C1(CCC=C)CCCN(C(=O)NC(c2ccc(Cl)cc2)C(C)(C)C)C1 C1(CC)C(=O)N(C)CCN1C(C1CC(C)N1C(=O)C(CC)(CC)CO)=O N1(C(c2nc(CC)oc2)=O)CCSCC1C(=O)NC(C1CCOCC1)CC C1(C(=O)NCC(CN(C(C2CCOC2C)=O)CC)(C)C)CC(=C(F)F)C1 C1(CC(=O)NCC2CN(C(c3ccc(O)nc3)=O)CCO2)CC2(CCCC2)CO1 C(C(C(=O)NC1CCCC1NC(=O)CCCCOCC)C(C)(C)C)OCC=C CC(C)CC(C(=O)N1CCCC1C=CC(=O)NCC1(CO)CCCO1)C(N)=O c1(C(=O)NCC(CNC(C(CC)C)=O)F)ccc(CO)cc1OC c1(C(=O)NCC(CC=C)NC(=O)C(CC)NC(N)=O)cccc(C(F)F)c1OC c1(CNC(CCSCCC)=O)ocnc1C(=O)NCC C1(NC(c2ccc(=N)[nH]n2)=O)CCCCCN(C(c2ccnc(O)c2)=O)C1 Brc1ccc(-n2nccc2-n2nnnc2N2CCCCC2c2ccon2)cc1 C1(NC(C(C=C)O)=O)CC2CCC1N(C(c1ccc(C(F)(F)F)cn1)=O)C2 N1(C(c2c(C)nn(CCO)c2)=O)CCCC2(NC(C3CCC(F)C3)=O)CC2C1 c1(OCC=C)cc(OC)ccc1C(N1CC(NC(=O)CC)CC1C)=O c1(COC)nc(C(=O)NC2CC(NC(c3cc(C(N)=O)c[nH]3)=O)C2)cs1 Cn1nc(Br)cc1S(=O)(=O)N1CCC(c2ccc(F)cc2F)C1 C1(C(C)NC(c2cc(CC)no2)=O)CCN(C(C2(C(F)(F)F)CC(O)C2)=O)CC1 CCCCCCCC(=O)N1CCC(C)(C)C1C(N1CC(=O)N(C)C(C)C1)=O CC(C(=O)NCCCNC(=O)CCCOCCOC1CCC1)SC(F)(F)F N1(C(CN(C)C2CC2)=O)C(CNC(c2cc(-c3ccccc3)co2)=O)CC2CC12 C(CNC(C1(C(N)=O)CC1)=O)(C(C)C(C)C)NC(Cc1c(C)noc1C)=O c1(C(N2C3C(NC(c4ccc(CC)cc4)=O)CC(C3)C2)=O)cc(C)[nH]c(=NC)n1 CC(C)(C)CCC(F)C(=O)NCC1(C)CCCC1NC(=O)COC1CCC1 CC1CN(C(=O)CN(c2cnccn2)C)CCCN1C(=O)C1=CCCOCC1 c1(C(N2CCC(C)C2CNC(=O)CC2(O)CCCOC2)=O)cc2cnccc2o1 c1(CC(N2C(C(C)NC(c3cn(CC)nc3)=O)CCC2)=O)c(C)cc(C)cc1C N1(CCNC(C2C(C)OCC2)=O)CCC(NC(=O)CN2C(=O)CCC2=O)CC1 c1(C(C2CC2)NC(C(C)OC(=O)C(C)(C)NC(C)C)=O)nnc(O)n1C C1(NC(=O)C(F)(F)c2cncs2)CN(C(C2(CC3CC3)CCC2)=O)CC1F N(C1CCCn2ccnc21)C(C1OCCC(NC(CSC)=O)C1)=O C1(C(N2CCCC(N(C(=O)CCOC(C)C)CC)C2)=O)CC2(C1)CS(=O)(=O)C2 CCC(C#N)C(=O)NC1(CN(C)C(C2COCCN2C)=O)CC1 CC1(NC(C2CCN2S(C)(=O)=O)=O)CN(C(=O)C(C#N)C2CC2)C1 c1(C(N2CCN(C(=O)CC(F)(F)F)CC2C2CC2)=O)cc2ccoc2cc1F CCCCN=C(NCc1ccc(Br)cc1Cl)N1CCC(C(=O)OC)CC1 c1(C(=O)NCC2C(C)CCCN2C(=O)C=C2CCC2)ccc(P(C)(C)=O)cn1 c1(OC)ccnc(C(N2CC(CNC(=O)CC3CCCN(C)C3)C2)=O)c1O C1(C(=O)OC)CN(C(c2ccc(Cl)s2)C(=O)NCc2cccs2)CCC1C C#Cc1cccc(OCC(=O)NCC(C)(O)CNC(C2CCN(OC)CC2)=O)c1 c1(C(C)(C)C)cccc(CC(N2CC(O)(CCNC(=O)C(F)(F)CO)C2)=O)n1 c1(C(C(=O)NC(C(=O)OC)Cc2ccccc2C)OC)ccccc1O c1(NC(C(C2CC2)NC(C(N2CCOCC2)C)=O)=O)ccc2c(c1)CCO2 C(=O)(N=S(C)(=O)C1CC(CN)C1)C1(N(C)C(c2ccc3nnc(C)n3c2)=O)CC1 c1(C(N2CCCC(N(C(C(CC)F)=O)C)C2)=O)ccc(F)c2c1OCC2 N1(C(C(CC)(F)F)=O)CCCCC(CCC(=O)NCCn2ncnn2)C1 N1(C(Cn2cnc(=N)[nH]2)=O)CCN(C(c2cncc(F)c2Cl)=O)C2CC12 CC(CC(=O)NC1(C(=O)N(C(C)C(N)=O)C)CCN(C)C1)C(C)(C)C C1(O)(CNC(CCN(C(C(C)n2cccn2)=O)C)=O)CCCC1(C)C C1(C(C)(C)C)CC(N=c2[nH]c3c(c(=NCC4CC(C(N)=O)C4)[nH]2)CCC3)CCO1 N1(C(C2CC(=O)NCC2)=O)CCC(C(=O)NC(c2ccc(Cl)cc2)CO)C(O)C1 Cc1cc2[nH]c(C(=O)NCCC(C)N(C)C(C3(C)CC4CC4C3)=O)cc2o1 C(=O)(CCC(=O)NCCOC(C(=O)OC(C)(C)C)C1CN(CC)C1)OCCCC c1(C(=O)NCC(CNC(c2ccn3nccc3n2)=O)F)ccc2ccncc2n1 Cc1cc(NC(c2conc2CNC(c2cnc(C)s2)=O)=O)cc(Cl)c1 N1(C(C(C)OCCN(C)C)=O)CCN(C(CCc2c[nH]c(=N)s2)=O)CCC1C S(=O)(=O)(c1cccs1)NC(C)CC(=O)N(C)CCN(C)C(C1(C)CCCN1C)=O N1(C(C(C)OC)=O)CCOC2(CCCN(C(c3ccccc3I)=O)C2)C1 CC1(CNC(C2C=CCCN2C(C2CCC(=O)O2)=O)=O)CCC(=O)N1 Cc1ccccc1OCCCC(=O)NCCCC(C)NC(C1C2(CC2)C12CC2)=O c1(CC)ncc(C(=O)NC2CC(C(N3CC(C)(O)C3)=O)C2)s1 C#CCCCCCCN=c1nc(N(CCCO)C)c2sccc2[nH]1 Cc1cc(C)c2[nH]c(=NC3CCCCC3NC(C3(O)CCCC3)=O)sc2c1 C1(CNC(CCCCC)=O)CC2(CCN(C(C3COC3)=O)CC2)CO1 CN1CC(C(=O)NC2CN(C(C3C4CCCCCC34)=O)C2)OCCC1=O c1(N2CCN(C(CN3C(C)CCC3C)=O)CC2)ncnc(Cl)c1[N+](=O)[O-] c1(C(N2CCC(C)(CNC(c3cc(C)c(Br)o3)=O)C2)=O)cc(N)cc(F)c1 c1(C(N2C(C(=O)Nc3cc(C)cc(O)c3)CC3CC32)=O)cccc2ncccc12 N1(C(C(C)c2ccsn2)=O)CCC2(CC(NC(c3cnc4cc[nH]c4c3)=O)C2)C1 n1(CC)cc(S(=O)(=O)N2CCC(C(=O)NCCN(C)C)C(O)C2)cn1 C1(C)(C(N(CCC(=O)NC(C2CCC2)C)CC2CC2)=O)CCCO1 c1(NC(C)=O)ccc(NC(c2ccc(-c3c[nH]nc3C)cc2)=O)cc1Cl N1(C(C2CCC(=C)CC2)=O)CCCC(O)(CN(C)C(c2conc2C(C)C)=O)C1 C1(C(N(C)Cc2cnco2)=O)CCOC1CNC(=O)CCc1cccs1 CC(C)(C)C(Br)C(=O)N1CC2CC1(C(=O)O)C2 C1(CC(=O)N(CCC)CCNC(CC2CCOC2)=O)C=CS(=O)(=O)C1 C1(NC(=O)NC(CC)CS(C)(=O)=O)COc2ccc(F)cc2C1 c1(C(N)=O)ccnc(C(=O)NC2CC(NC(C3CCCN3C=O)=O)C(O)C2)c1 C1(NC(C(=O)NCC)=O)CC2C1CCN2C(=O)CCC(CC)OC C1(C(=O)NC2C(C)CN(C(c3cnn(CCF)c3)=O)C2)CCC(=O)N(C2CC2)C1 c1(OC)cc(C=CC(=O)NC(C(C)NC(=O)C(=O)NC(C)C)C(C)C)ccc1F C(CC)(CC(=O)N(CCC(=O)O)OC)CC.CCO c1(NC(C(=O)NCCN(OC)C)=O)cccc(S(=O)(=O)C(F)F)c1 C#CCCC(O)C(=O)N1CCCC(CCNC(=O)Cc2csc(COC)n2)CC1 C(=O)(CC(CNC(c1nc(Br)c(C)cc1F)=O)C(F)(F)F)OC N1(C(C2CN(C(c3c(C)c(F)ccc3)=O)CC23CC3)=O)CCCC2OCCC2C1 c1(C(N(CCOC)CCNC(C2(C)CC(=O)N(C)C2)=O)=O)[nH]nc([N+](=O)[O-])c1Cl S(=O)(=O)(c1c(C2OCCO2)cnn1C)N1CCCC(c2onc(C)n2)CC1 c1(NC(C(C)OC(=O)Cn2nnc(=N)[nH]2)=O)ccnc2c1cnn2C c1(OC)cc(Br)ccc1CNC(C1CCCN(c2cncc(CO)n2)CC1)=O c1(C(N2C(CN(C(C(CC)F)=O)C)COCC2)=O)cc(Cl)cc(C(F)(F)F)n1 c1(OC)ccc2cc1-2.c1(C(=O)Nc2cncs2)ccc(-c2cncn2C)cc1 c1(NC(C)C)cnccc1CNC(=O)Cn1cc(CCS(=O)(=O)N(C)C)nn1 C12(NC(c3c(OC)cccc3)=O)CCCC1(F)CN(C(=O)C(C)NC=O)C2 N1(C(c2cc(C)c(C)o2)=O)CCCC(C)C1CNc1ncc(F)cn1 n1(CC)nc(C2CC2)cc1C(N1CC2CC2(CNC(=O)CCS(C)=O)C1)=O N1(C(C(C)OCC=C)=O)CCCC(C)(C)C1CNC(c1ccc(=O)oc1)=O C(=O)(CC1NC(=O)c2ccccc21)NCCCCNC(=O)CC1CCS(=O)(=O)C1 C#CC(CC)(CC)NC(=O)C(C1CN(C(C2CC=C(C)CC2)=O)C1)OC c1(C(=O)NC2C(SC)CN(C(=O)C=CC3CC3)C2)ccn2cccnc12 n1(CCC(=O)N(C)CC2(NC(C(F)=C(C)C)=O)CC2)cnc(C)cc1=O Cc1cccc(C)c1C(=O)N(C)CCN(C(=O)Cc1cncs1)C(C)C C1(NC(Cc2cc(C)no2)=O)CN(C(c2ccc(C(C)C)cc2)C)CC1F S(=O)(=O)(c1ccccc1)C(N1CC(C2CCNCC2)OC(C)C1)C(C)C C1(C)(CNC(c2c(OC)c[nH]n2)=O)CCN(C(C2CCC(N(C)C)CC2)=O)CC1 C(=O)(CC(C)(C)CCOC)NC1C(C(=O)NC(CCC)C(C)(C)C)CCC1 c1(C(C(=O)NC2CCCC2)N(CC(C)C)C2CC2)ccc(F)c(Cl)c1F C(=O)(C1CCCc2c[nH]nc21)NC1(C2CCCN(C(CC(CC)O)=O)C2)CC1 c1(OCC#C)ccc(Br)c(CNCc2cnc(CC)s2)c1 C1(C(=O)N(C2CC(=O)N(C)C2)C)(OC)CCN(C(=O)Cc2ccsc2)CC1 c1(CCC(C)C)cc(C(=O)NC(C)CNC(c2cnc(C(C)O)s2)=O)no1 C1(C2CCN(c3ncnc4onc(C)c34)CC2)(NC(C2N(CC)CC2)=O)CC1 N1(C(C(c2ccc(OC)nc2)(F)F)=O)CC2(CCN2C(c2nnsc2C)=O)C1 C=CCCC(C)C(C(=O)NCc1ccc(F)cc1)N1CC(C(=O)OC)C(CCO)C1 c1(C(N(CCNC(C2CC2CC(C)(C)C)=O)CC)=O)[nH]c2c(C)cccc2c1C C(=O)(C1=C(C)OCC1)NCC1C=CC(NC(C2C(OC)CCCC2)=O)C1 C#Cc1cc(C(=O)NCC2CN(C(C3(C#N)CCC3)=O)CCO2)ccc1Cl O=C(O)C(O)C(F)(F)N1CCCC(CNC(C2CCC(F)(F)CC2)=O)C1 c1(SC)ccnc(O)c1-c1nccn1C1CN(Cc2ccon2)C1 C1(N(c2ccc(O)c(F)c2F)C(c2ccc(C)[nH]2)=O)COC2(CCNCC2)C1 c1(N2CCC(N(C(C3CCC4C(C3)C4(F)F)=O)CC)C2)ncc2ccccc2n1 C(=O)(CCCCCNC(=O)C(CC)N(C)C)N1CCC(CCCC)C1 c1(CCCNC(=O)NCC2(c3cccc(F)c3)CCC2)cccc(Cl)c1 C1(C(CNC(c2c(C)occ2)=O)C)CCN(C(=O)C(C)(C)c2cccs2)CC1 c1(OC)ccc(CCC(=O)NC2C3CN(C(c4c[nH]c(Br)c4)=O)CC23)c(OC)c1 N1(CC)CC(NC(=O)C(C2(O)CN(C(=O)Cc3cc(C)n(C)n3)C2)F)CC1=O CC1(CCNC(=O)CCCNC=O)CCN(C(=O)CCC(N)=O)C1 Cn1nnc2cc(NC3C(C)CCN3C(=O)OC(C)(C)C)ccc12 c1(CC(N2CCCC(N(C(C=CC(C)C)=O)C)CC2)=O)ccccc1[N+](=O)[O-] N1(C(CCCCN(C(=O)CSC(F)(F)F)C)=O)CCCC2CCCC12 N1(C(C(c2cscn2)N(C)C)=O)CCC2(CCC2NC(=O)CCCC(N)=O)CC1 n1(C(C)C)cncc1C(=O)NCC1(O)CN(C(=O)Cn2nccn2)C1 c1(C(=O)OC)nc(N2CCCCC2C2CCN(C(C3CCOC3)=O)C2)ncc1Cl c1(NC(CNC(c2nnnn2C)C(C2CC2)OC)=O)ccc(F)c(Cl)c1 N1(C(C2CN(CC(C)C)C2)=O)CCC2C(C1)CN2C(c1oc(C(C)C)nc1C)=O Cc1ccc(CC(=O)N(C2CN(C(=O)C(O)C(F)F)C2)C)cc1C c1(C(=O)NCC2(C(C)NC(CCCOCCC)=O)CC2)ccc(F)c(F)c1 c1(C(N(C2CCN(C(=O)CCCCc3cnc[nH]3)C2)CC#C)=O)ncc[nH]c1=O Cc1cc(C(=O)NC2CN(C(c3cc(F)ccc3O)=O)CC2C)cc(Br)c1 C12(C(N3CCC(C(C)(C)C)CC3)=O)CC(CCO1)N(C(=O)Cc1ccccc1)C2 c1(N2CC(C(C)NC(C(COC)C)=O)C2)nc(C#N)c(Cl)s1 C1(CNC(CC(C)(C)C)=O)N(C(C2CCCN(S(C)(=O)=O)C2)=O)CCC1(C)C C1(C(=O)NC(C)C=CC(N2CCC(C(C)(C)C)C2)=O)(SC)CC(=O)C1 N1(C(CCN(C(C(COCC)(C)C)=O)C)=O)CCC12CCC(C)CC2 C1(CNC(c2c(C)cnn2C)=O)C2CCCC1N(C(C1CCCN1C)=O)C2 c1(C(N2CC3C(CNC(C4CCCS(=O)(=O)C4)=O)C3C2)=O)cn2cnnc2cn1 C1(n2cc(C(CC)CC)nn2)CON(C(=O)C2CC(=O)N(CCC(C)C)C2)C1 N1(C(C(C(=O)OC)C)=O)CCC2(CC1)CN(C(C1(C(=O)NC(C)(C)C)CC1)=O)C2 c1(C(=O)NC2CCC2CNC(c2coc(C3CCC3)n2)=O)ccc2snnc2c1 N12CCOCCC1CN(C)CC2=O.c1(SCC(=O)NCC2CC2)ncc[nH]1 C(=O)(CC(C)(C)C(F)F)N1CCC(CN(C)C)C1CNC(=O)C1=CC2C=CC1C2 Cc1cc(C(N2CCC(F)(CNC(C3CN(C)C3)=O)C2)=O)c(N)s1 c1(OC)cc(C(=O)NCC(C)(C(C)C)NC(=O)C(F)=C(C)C)cc(OC)c1C c1(NC(C)=O)cccc(C(=O)NC2(CNC(=O)C(C3(O)CCCC3)F)CC2)c1 c1(OC)cc(C(=O)Nc2ncc(-c3ccc(CO)c(F)c3)s2)c(F)cn1 c1(CC(=O)NC2CN(C(CNC(CC(C)C)=O)=O)C2)ccc(Br)cc1F C1(NC(CCCC)=O)Cc2ccccc2C1NC(=O)CCCn1ccnn1 C(C)(CCC(=O)N(C(CNC(=O)C(C)N1CCCC1)C1CC1)C)SC C1(CNC(c2scc(C)c2)=O)CCC(N(C(=O)CNC(c2ccoc2)=O)C)CC1 c1(C(C(N2CC(C(C)NC(c3csnn3)=O)OCC2)=O)O)cc(F)c(F)c(F)c1 N1(C(CCN(C(C2CC(C(=O)OC)C2)=O)CCO)=O)CCN(C)C(C(C)C)C1 C1(C(N2CC(C#C)(C(=O)NC(C)CSC)C2)=O)CCC=CCCC1 C1(C(=O)NC(C)CNC(c2cc(-c3csc(=N)[nH]3)c[nH]2)=O)COCC(C)(C)O1 c1(C(N(C2CCC(NC(c3ccc(F)o3)=O)C2)C)=O)cccc2c1CCC2=O CCCCCC(O)C(C)C(=O)NCC(C)NC(c1cc(C)sc1Br)=O C(=O)(C1=COCCO1)NC(CCCNC(CC1C(C(=O)OC)CCC1)=O)(C)C C1(NC(C2(CN(C)C)CC2)=O)C2CC1N(C(=O)CCCn1ccnn1)C2 C1(C(N(CCCCCC=C)C)=O)CCN(C(=O)C(CC=C)CC(C)C)O1 N1(C(COC(CC)C)=O)CCN(C(c2sc(C)nc2C)=O)CC(O)C1 c1(C(N2CCC(NC(C(CC(C)C)OC)=O)C2(C)C)=O)cc2ccccc2n1C C(=O)(CC(C(F)F)NC(=O)C(F)OC)NC1(CCOC)CCN(C(C)=O)C1 C(=O)(C(C)(C)C(C)(F)F)NC1C=CC(CNC(Cc2cc(C)[nH]n2)=O)C1 c1(CC)[nH]c(=NC(C2=CCCCC2)c2nnnn2CCCC2CC2)[nH]c1C1CC1 CCC#CCN=c1[nH]c2c(c(=NC(C)Cc3cccs3)[nH]1)SCC2 N1(C(C2CN(C(C)=O)C2)=O)CCC2(CO)CN(C(c3ccn(C)c3)=O)CC2C1 C12(C(N3CC4C(CNC(c5ccno5)=O)(C4)C3)=O)CC3CC(CC(C3)C1)C2 C1(C(N2CC(CC)C2)=O)CC2C=CC1N(C(=O)CCc1nc(=N)[nH][nH]1)C2 C1(C(N2CCC(OCCNC(=O)C=C(Cl)Cl)C2)=O)CC2(C1)CC(F)C2 [N-]=[N+]=NC1CCN(C(C2(F)CCCN(C(C3CC4(CC4)CO3)=O)C2)=O)C1 N1(C(C=CCC2(NC(C(C)=CC(C)(C)C)=O)CCC2)=O)CCN(C)CC1CO N1(C(C(C)CCO)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)Cc1ccco1 C(C(=O)NCc1cn(C2CN(C(c3cccc(F)n3)=O)C2)nn1)(C(C)C)OCC C(CC(=O)N(C1CCC1O)C)N(C(=O)CC1CC(SC)C1)CC c1(C(N2CCC(O)(C(C)NC(=O)C(Cl)=CCl)C2)=O)c[nH]cc(Cl)c1=O c1(CNCC2(O)CCC(C)C2)cc2c(cc1Br)OCO2 C=C1CC2CCC(C1)N2C(=O)C(C)(C)CNC(=O)C(C)O c1(C(c2nnnn2CCNC(C)=O)NC(CCC(=C)C)C)cc(C)cc(C)c1 N1(C(C2OCCN(C)C2)=O)CC(C)(C)OCC1CNC(c1ncccn1)=O CC(C)C(CC(=O)NCCOCCN(C)C(C1CCC(=O)C1)=O)c1ccccc1 c1(C(N(C(C)=O)C)C)ncc(-c2ccco2)n1C(c1ccccc1)C c1(-n2ncc(C(=O)NCC(C(C)(C)C)NC(C=C(C)Cl)=O)c2)cccc(Cl)c1 Cc1cc(OC(CNCCCOc2ccccc2Cl)C(=O)O)nc2ccnn12 c1(C(N2CC(C)(NC(C3CCCC(O)C3)=O)C2)=O)cc2nccnc2cc1F c1(CCC(=O)NC2CC(N(C)C(c3ccc(Cl)o3)=O)C2)cnc2n1CCCC2 c1(C(N(C2(C(=O)OC)CCCC2)C2CC2)=O)cnncc1O c1(C(=O)NCC2(F)CC(NC(C3(O)CCC(CC)C3)=O)C2)nccc(C)c1N CCC(C(=O)N1CCC(C(=O)N(CC(C)(C)OC)C)C12CC2)C(C)C N1(C(CCCCSC)=O)C2CCC1C(C)C(NC(C1CC3CCCCN3C1)=O)C2 CC1CN(C(=O)CC2CCC(=O)NC2)CC1NC(=O)CCCn1cccc1 C1(CC(=O)OC)CC(NC(C2(O)CN(C(=O)C=CC(=O)N(C)C)C2)C)C1(C)C c1(CN(CC(O)CN2CCOC3(CCCCC3)C2)C)nc2ccc([N+](=O)[O-])cc2s1 CC(C)CC(C(=O)NC1CC1NC(=O)CCc1ccn(C)n1)N(C)C C1(C(N2CCN(C(c3c(CC)n(C)nn3)=O)C3C2C3)=O)CC2CC(O)CC(C1)C2 c1(C(N2C(CCC)CN(C(=O)CCS(C)(=O)=O)CC2)=O)cnc2nncn2c1C N1(C(CC=CC=C)=O)CCCC2CN(C(C3CCCCNC3=O)=O)CCC12 C(CCCCCn1ncc(NC(C)=O)c1)N(C(=O)C(C)OC1CCOC1)C(C)C N1(C(C2CC(SC)C2)=O)CC2C(CNC(c3ccc(CS(C)(=O)=O)cc3)=O)C2C1 Cc1ccnc(C(=O)NCCC(O)CNC(=O)Cn2ccccc2=O)n1 C#Cc1cccc(C(N2CCN(C3CN(C(=O)C(C)c4ccsc4)C3)CC2)=O)c1 N1(C(CC2(OC)CN(C(=O)Cc3cccc(Br)c3)C2)=O)CCCC2CCCCC12 Cc1cc(C)cc(C=CC(N2CC3CCC2CN3c2ncncc2C#N)=O)c1 C=CCCCCCC(=O)N1CC(N(C(=O)C(O)CF)C)C(C)(C)C1 c1(C(=O)OC)sccc1SC(C)C(=O)N1CC(Cc2ccco2)C1 CCN=c1ccc(C(=O)NCC2(O)CN(C(=O)C(c3ccc(Cl)s3)C)C2)c[nH]1 C(CCCCC)N(CC(=O)NCc1conc1C(C)(C)C)CCN(C(=O)CC#N)C C1C(F)C(=O)N1.C1(CN(CCOCCN(CC)CC)C)CCN(C)C1 C1(N(C(C)(C)C)OC(CC(=C)C)=O)(CF)CCN(C(=O)C=CC(C)C)C1 c1(OC)cccc(Cn2nnnc2C(c2ncco2)NC2COCCOC2)c1 C1(CC(=O)NCC2CC(C(N3C(C)(CC)CC3)=O)C2)CCCC(C)O1 N1(C(C=C2CCC(C)CC2)=O)CC(C(N2CC(C(C)O)C2)=O)C(F)(F)C1 c1(NC(c2n(Cc3nnn(C)n3)nnn2)C2C3CCCC23)cccc([N+](=O)[O-])c1 c1(CN(C(=O)C(=O)NCCc2cccc(OC(F)F)n2)C)cccc(F)c1 C1(NC(CCC=C)=O)CCN(C(=O)C(C)(C)c2sccc2Cl)CC1C C1(C(=O)NCc2c(C(=O)NC(C3CCCCO3)C)nco2)CC2(CCC2)C1 C1(C(C)NC(C2(CF)CCC2)=O)CN(C(c2ccnn2C2CCCC2)=O)CCO1 c1(CC)nc2c(C(=O)N(C3CCC(NC(=O)CCS(C)(=O)=O)C3)C)ccnc2[nH]1 O=C1OCc2cc(COC(C3CC4CC3C3CCCC43)=O)ccc21 c1(OC)ccc(C(N2CC(NC(=O)C(O)Cc3ccccn3)C(O)C2)=O)cc1N CC(CC(=O)N=c1ccnc(C2CN(c3cnccc3F)C2)[nH]1)C1CCCCC1 N1(C(CCCCOC)=O)CCC(NC(=O)CCC(F)(F)F)C(F)C1 N1(C(c2cncc(C)c2)=O)CCC(CNC(C2COCCC2C)=O)C(O)C1 C1(C(=O)NC)(C(=O)ONC(C(CO)NC(c2ncoc2COC)=O)C)CCCCO1 c1(CC(=O)NCCCN(C(C2CC(C)CC(C)C2)=O)CC)nc([N+](=O)[O-])n[nH]1 C1(C(=O)NCCC2CC(C(=O)NCC3(C(C)C)CCC3)C2)CCCN1C=O N1(C(Cc2cnc(C)[nH]2)=O)CCC(N(C(=O)CCC2CCC2)C)C2(CC2)C1 c1(C(C(N2CCOC(CNC(c3cnn(C4CC4)c3)=O)C2)=O)O)cccc(F)c1 c1(C(=O)NC2C(NC(C(CC#C)C)=O)CCOC2)ccc(Br)c(O)n1 N1(C(C2(CO)CN(C(C3C(C)CCC3)=O)C2)=O)CC(CO)C1(C)C C(=O)(CCCCCSC)NC(C1(O)CN(C(C23CCC(OC)C2C3)=O)C1)C N1(C(Cc2c(C)ocn2)=O)CC2CN(C(c3cccc[n+]3[O-])=O)CCC2(CO)C1 N1(C(CCC(C)OC)=O)CCN(C(=O)CC(C)(C)c2ccccc2)CC(C)(F)C1 C1(C(=O)NCCC(CC)(C)C)CC2(CC(NC(C3COCCO3)=O)C2)C1 c1(C(N2CCC(NC(C(F)=CCC)=O)C2)=O)oc(SC)cc1C c1(C(=O)NC2CN(C(CCCC(C)C)=O)CC23CC3)cn2ccc(Cl)c(F)c2n1 N1(C(CCCSC)=O)CC(NC(C2CC(=O)NC2(C)C)=O)CC(C)(C)C1 CCCC(C)CC(=O)NC(CCOCC)C(=O)NCC1(CO)CC1 N1(C(CC2(C=C)CN(C(C34CCCN(CC3)C4)=O)C2)=O)CCC(N=[N+]=[N-])CC1 CC1(C)CC(CNC(C2CCCCC2n2cccc2)=O)CN(C(=O)C(N)=O)C1 c1(NC)ccccc1C(N1CCCCC1CCC(=O)N1CCC1CF)=O C(C(F)(C(=O)NCC(C)CC1CC1)C(C)C)NC(C(n1ncc(C)c1)C)=O c1(CNC(CC(CC)(C)C(=O)OC(C)(C)C)=O)c(C)oc2ncn(C)c(=O)c12 c1(C(N2CCC(C)C(NC(=O)CCC3CCCCO3)C2)=O)n[nH]c2c1CCOC2 c1(NC(C2CCCN2Cc2cccc(OC(F)F)c2Br)=O)cc(Cl)c(Cl)cc1F C1(OC)CN(C(c2cc(C(N)=O)c[nH]2)=O)CC1NC(=O)CNC=O C1(NCC2(C)N(C(=O)OC(C)(C)C)CCC2)COCC(C)(C)C1 c1(CC2(CO)N(C(C(CCN)F)=O)CCC2)ccc(Cl)c(F)c1 C(=O)(C(C)CC(C)(C)C)NC(C(=O)NCCC(CC)CC)CSCC c1(CNC(C(CN(C(C(CC=C)NC(C)=O)=O)C)C)=O)ccc(C)cc1O c1(C(C(N2CCCC(NC)C2)=O)(F)F)cccc(F)c1F C12(c3nc(CCP(C)(C)=O)on3)CCOC1CN(C(=O)OC(C)(C)C)C2 CC1(CO)CCN(C(C2CCC(NCc3c(O)ccc(F)c3F)CC2)=O)CC1O c1(C(=O)NCC(c2ccc(OCC)cc2)O)cccc2oc(=N)[nH]c12 c1(CC)ccc(C(C)C(=O)NC2CC(NC(=O)CCn3cccn3)C2)cc1 c1(CC(=O)NCC(CNC(Cn2c(C)ccn2)=O)(C)C)cccc(C(F)F)c1 N1(C(CC2CC(CC)C2)=O)C(C(=O)OC)CC1C.C12C(C1(C)C)NC2=O N1(C(c2scc(C)c2)=O)CCCC2(CCN(c3nc(C(F)(F)F)cc(C)n3)C2)C1 Cc1cc(C(N2CCC(N(C)C(C3CCC(=O)N(C4CC4)C3)=O)C2)=O)cc(C)c1 CCC(C)(C)C(C)NC(=O)COCCNC(C1CN(C(C)=O)C1)=O C1(NC(C2CC(=C)C2)=O)CCOCC1NC(=O)CCn1cncn1 C1(C)(C(=O)NCCC2N(C(C(CC)=CC)=O)CC(F)(F)C2)CCCCNC1=O C1(CN(C(c2c(C)ocn2)=O)C)CCCCN1C(=O)Cn1cccc1 N1(C(C(C)OCCOCC)=O)CC2CCCC(NC(=O)C(C)(C)CO)C2C1 C1(CC#N)CN(C(c2c(O)cccc2Br)=O)CCN1C(c1ccc(Br)cc1F)=O c1(OC)ccc(OCC(=O)N(CC(C)CNC23CCC(C)(CC2)C3)C)cc1C C(C)(C)(CCCNC(c1c(Cl)cnn1C)=O)NC(C1C(OCC)C1)=O c1(NC(C(=O)NCC(CC)NC(c2cc(CO)ccn2)=O)=O)ccc(C)c(F)c1 CCCC(CCCNC(=O)CNS(=O)(=O)NC(C)C)N=c1cc(C)nc(CO)[nH]1 C1(NC(C2CC(C#N)(OC)C2)=O)CN(C(C2CN(C)CCO2)=O)CCC1CO CCCC(C)(O)C(=O)NCC1CCCN(C(c2occc2Br)=O)C1 c1(C(n2cc(CC3N(C(C(C)CF)=O)CCOC3)nn2)C)ccc(Cl)c(F)c1 c1(OC)ccc(CNc2ccc(C(=O)NCC=C(C)C)nc2)c([N+](=O)[O-])c1 c1(NCC(=O)NC2C3CN(C(c4c(C)occ4)=O)CC32)ccc(C#N)cc1 N1(C(c2c(CC)ocn2)=O)CC2CCC2(CNC(=O)Cc2nccn2C)C1 C=C(Br)CC(C)(C)C(=O)NCC1(NC(C2C(F)(F)C23CC3)=O)CC1 c1(N2CC(CC)C(O)CC2)nc(N2CCC(C(N)=O)C2)c2sccc2n1 N1(C(CCN(CC)CC)=O)CC2=C(C1)CN(C(=O)CC1OCCC1C)C2 C1(C(N(CC(C)O)CCNC(c2c(OC)ccc(F)c2)=O)=O)CC(C)(C)OC1(C)C C(CC(CNC(=O)COCc1nc[nH]n1)NC(=O)C(CO)NC(C)=O)OC C1(NC(CC2C(C)CN(C(=O)CC3(C)OCCO3)C2)=O)C2CCCC1CC2 C(C1CCOC1)=CC(=O)NC1CCN(C(=O)CCCC2CCC2)C1 c1(OC)cc(C(N2CCN(C)C(CNC(c3cccs3)=O)C2)=O)cc(F)n1 c1(C(=O)NCC2(F)CCN(C(CC(C)CN(C)C)=O)C2)cc(F)ccc1F Cc1oc([N+](=O)[O-])cc1C(=O)NC1CCN(C(=O)CC2CCC(=O)N2)C1C N1(Cc2cccc(OCC)c2)CCC(N2CCOCC2C(=O)NC)C(C)CC1 CC1CN(C(c2ccc(Br)nc2O)=O)CCN1C(=O)C(F)CC1CCC1 S(=O)(=O)(c1ccc(N(C)CC2CCSCC2)c(Br)c1)N1CC(C)S(=O)C(C)C1 C1(CCC(=O)NC(c2cccnc2F)C)CCCN(C(=O)CC(C)(C)O)C1 C(=O)(CCCC(=O)N(C1CCCN(C(c2cc(C)nc(CO)n2)=O)C1)C)OCC Cc1[nH]c(=N)sc1C(=O)NC(C)(CNC(=O)C(C)(C)n1ccnn1)CO c1(OC)cnc(C(N2CCOCC2CCNC(=O)COC2CCOC2)=O)cn1 CC(C)CC(O)C(C)C(=O)N1CC(O)CC1CC(N1CCC12CCCC2)=O c1(C(N2C(CN(C(=O)C(C)C)CC)CCC2)=O)cnn(C2CCCC2)c1C C12(CC(=O)NCC=CCO)CC1CN(OC(C)(C)C)C2.C1(C(=O)OC)CCC1C=O N1(CCC)CCCC(C(=O)NC2CC(CCNC(c3csc(=N)[nH]3)=O)C2)C1 c1(C(=O)NC2CC(CNC(C(C=C)O)=O)C2)ccc2oc(C)nc2c1 C12(CNC(CC3CN(C(C)=O)C3)=O)CCN(CC1)CC2 CCC(CC(F)F)C(=O)NCC(C1CCCC1)NC(c1ncn(C)c1C)=O n1(CC(=O)NC2CC(NC(c3ccc(C)nn3)=O)C(O)C2)nc(C)c(C)c1C c1(C(=O)NCCCC(C)NC(CC(C)SC)=O)cc(O)ccc1N N1(C(C(CC=CC)NC(=O)CCOCC(C)(C)C)=O)CCC2CCN(C)CC12 C1(C)(CC)C=C(C(=O)NCC(C2CC2)NC(c2ccc(C(C)(C)C)s2)=O)C1 c1(C(=O)NC2C3(CC(NC(C(C4CCC4)OC)=O)C3)C2)cc(C#N)c(F)cc1F S(=O)(=O)(c1ccc(F)c(NC(=O)C(N)CC2CC2(F)F)c1)NC C1(C)(C(=O)NC(C)COCC(F)(F)F)CNCCO1 n1(C(C)C)ccc(=NC(=O)CC2CCN2C(=O)Cc2cnsc2)[nH]1 C(=O)(N=c1cc(C)n(CC(=O)N(C)C)[nH]1)c1nc(NC(C(C(C=C)C)C)=O)sc1 N1(C(C(C)OCC)=O)CCN(C(c2c[nH]c(=N)c(C)c2)=O)CC1C1CCCC1 [N-]=[N+]=NC1CCC2(C(=O)OCC3CCc4c[nH]nc4C3)CC12 N1(C(C2(c3ccc(Cl)cc3)CCC2)=O)CC(O)CC1Cn1cc(CO)nn1 c1(C(c2n(C)nnn2)NC(C)(C)CSC(C)(C)C)ccc(S(C)=O)cc1 C=CC1COCC1NC(=O)CN(CC(C)C)C(c1nccnc1OC)=O Cc1sc(C)c2sc(C(N3CCC(CN(C)C(C4CCNC(=O)C4)=O)C3)=O)cc12 C(=O)(C(C)CCCOC)N1CCC(C2N(C(CCC(=O)NC)=O)CCC2)C1 Cc1nc2c(o1)CCN(C(=O)C(C(C)O)NC(=O)C(C)CO)C2 c1(C(N2CCC(N(C(=O)Cn3cnccc3=O)CC)C2)=O)ccc(C)c(F)c1N C(=O)(C(O)CC(C)C)NC1C2CC(NC(CS(CC)=O)=O)CC21 c1(CC(=O)NC2CC(C)N(C(=O)CC3CN4CCC3CC4)C2)ccc(F)c(Cl)c1 C1(C(=O)NC2(CC=C)CN(C(=O)CCCN3CCCC3)C2)CCOC2(CCC2)C1 N1(C(C=CC=CC)=O)CCN(C)C(CNC(C2CCN(C)C2C)=O)C1 c1(COC)nc(NCC2COCC(C)O2)cc(=NCCOC(=O)N(C)C)[nH]1 c1(CC(CC(=O)NC2CC2O)NC(=O)CCc2cn[nH]c2)ccc([N+](=O)[O-])cc1 C1(NC(=O)NC2CCC(c3ccc(OC)cc3)(O)C2)CNCCC1C#N CC(C)(CCNC(=O)CCN1CCOC1=O)NC(=O)Cc1cncnc1 C(C(C(C)C(C)C)NC(c1ccc(C(C)C)c(O)c1)=O)NC(c1cc(C)[nH]n1)=O c1(C(N(CCCNC(=O)CCC2CC2(Cl)Cl)C)=O)sc([N+](=O)[O-])cc1Cl c1(C(=O)NC(CC)CN(C(=O)CCc2nc[nH]n2)C)ccc(Br)c(C)c1 c1(NC(C(C(=O)OCC)(C)F)=O)nccc2[nH]ccc12 c1(C(N2C(CC(=O)Nc3c(OC)ccnc3Br)CC2)=O)cnn2cccc(C)c12 c1(C2(NCc3ccn(C)c3)CC2C)ccc(F)cc1 c1(C(N2CC(NC(CC(CC)OC)=O)C2)=O)cc2cccc(Cl)c2cn1 c1(CNC(C2(CCC=C)CN(C(C3CCC(=O)O3)=O)C2)=O)ccncc1F c1(C(N2CCC(N(C(C3CCC(C)CC3)=O)C)C2)=O)cnc2c(Cl)cccn12 c1(OC)ccc(Cl)cc1N(Cc1ccc(C(F)(F)F)nn1)CC1CC1 N1(C(C2CCC(C)CN2C(=O)C(C)Cn2ccnc2)=O)CC2C3C=CC(C3)C2C1 CC1C(C(=O)NCC(F)Br)CCCN1C(=O)C(C)c1cc[nH]n1 C(CCCC(C)NC(c1cncnc1C1CC1)=O)NC(CSCCC)=O N1(C(C2(CC=C)CC=CC2)=O)CC2=C(C1)CN(C(C1CC(O)C(F)C1)=O)C2 C(C)(N=c1[nH]c(=NCCCS(C)=O)c2c(F)cccc2[nH]1)c1nnc(OCC)s1 O=CN1CCC(c2nnnn2CN2CCCC2=O)(NC2CN3CCC2CC3)CC1 c1(CN(C(C)C(=O)NCCC(O)CNC(=O)C(F)(F)C2CC2)C)ccc(F)cc1 C(=O)(C1=CCCC(C)(C)C1)NC(C)CCCCNC(=O)Cc1ccn(C(F)F)n1 N1(C(CC(C)SC)=O)CCC(CO)(NC(c2oc(SC)cc2C)=O)CC1 c1(C(=O)NCC(CO)NC(C2CC2c2ccc(F)nc2)=O)csc(=NC2CC2)[nH]1 c1(C(=O)NCC(C)N(C(c2cnnc(O)c2)=O)CC)cnc(O)cc1C C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NC(C)CNC(C1CCC(C2CC2)C1)=O C(=O)(C(C)CC(C)(C)C)N1CCC2C(NC(c3c(NCC)cccc3)=O)C2C1 C1(O)(CC)CCC(C(=O)NC(C)CNC(=O)CN2CCCCC2)CC1 C#CCCCC(C)C(=O)NC1(CNC(C2(C3CCCO3)CCC2)=O)CCCCC1 CCCC(C(=O)Nc1cccc(NC(c2cc(Br)oc2C)=O)c1)OCC Cc1c(Br)cnn1CC(=O)NCC(C)(C)CNC(c1c[nH]c(=N)o1)=O N1(C(C)=O)CCCC1(C)C(=O)NCCC1(C)CCN(C(c2ncc(F)cn2)=O)C1 C(=O)(C(CCC)=Cc1cccs1)N(C)CC1N(C(COCC(=C)C)=O)CCC1 N1(C(C2(NC(=O)COc3ccccc3)C(C)CCC2)=O)CC(C)C12CCOCC2 CC1CCC(NC(=O)CC(C)(C)C#N)CN1C(C1CCCS(=O)(=O)C1)=O C#Cc1cc(NC(C23CC(NCc4ccc(Cl)c(O)c4)(C2)C3)=O)ccc1C Cc1ncc([N+](=O)[O-])cc1C(N1CCC(CNC(c2nccc(Cl)c2O)=O)C1)=O Nc1cccc(C(=O)NNC(=O)C2CC3C=CC2C3)c1F.C12CN(CC1CO)C2=O N1(C(CN(CC(C)(C)C)C)=O)CC(NC(c2cccnc2O)=O)C(F)C1 C(=O)(C1=CCCSC1)NC(=O)OC(C)(C)C.C1CC(=O)NC(C2CCC2)CN1C Cc1cccc(F)c1CC(N1CCC=CC1c1ccccc1)=O C(=O)(C(C)(C)CC(=O)NCCC1CCCCN1C(=O)CCCCSC)OC N1(C(C2CC(SC)C2)=O)CCc2c(c(CNC(C3(O)CCSC3)=O)nn2C)C1 N1(C(c2c(C)nc(Br)s2)C(=O)NC2CCOC2)CC(C)OC(C)(C(F)F)C1 c1(OC)ccccc1-c1nc(COC(=O)COc2ccccc2C)no1 Cc1[nH]nc2cc(C(=O)N(C3CCN(C(C4CC5CC4CC5O)=O)C3)C)ccc12 C1(CC(=O)NCC2CCC3(CN(C(C4(O)CCC4)=O)C3)C2)SC2=NCCN2C1=O N1(CCC)CCCC(C(=O)NC2CCCC(NC(=O)Cn3nnnc3C)C2)C1 c1(C(C(N2CCC(CNC(C3(C)C(C)C3)=O)C2)=O)(F)F)ccc(F)cc1 Cc1ccc(C(N2CC3(CC3)CC2CNC(C2CC2(C)C)=O)=O)cc1[N+](=O)[O-] N1(C(CCCC(C)=O)=O)CCCN(C(=O)CCn2cnc([N+](=O)[O-])c2)CC1CO C1(C(=O)NC(CCCNC(c2c(C)nc(CC3CC3)o2)=O)C)CCCCNC1=O C1(C(c2ncc(C3CC3)cn2)N2CCCC2)COC2(CCNC2)C1 c1(C(N2CCC(NC(C(C)(C)C(N)=O)=O)C(O)C2)=O)n[nH]c2ccccc12 N1(C(C2C(CC)C2)=O)CCCC(C2CC2NC(C2(C)CC2C(F)(F)F)=O)C1 C1(CNC(c2c(CC)non2)=O)CC2(CCN(C(=O)CCC(F)F)C2)CO1 CCC(C)(C)CS(=O)(=O)N(C1CC1)C(c1ccc(Br)c(F)c1)C N1(C(COCCOCC#C)=O)CCN(C(=O)CC2C=CCC2)C2COCC12 CC(C)(C(=O)NCC=CCNC(C1(c2cc[nH]n2)CCC1)=O)n1ccnn1 Cc1ncnc(N2CCC(C)(CNC(c3cccnc3)=O)CC2)c1Br Cn1ncc(CCC(=O)NC2CN(C(C3CC3(C)C(F)F)=O)C2)n1 c1(C(=O)NC(C)CNC(c2cc[nH]n2)=O)cccc2ncnc(O)c12 C1(C(C)(C)C)(CNC(C(C)=C(CC)C)=O)CCN(C(C2CCN2C)=O)C1 Cc1cc(Cl)c(C(=O)NC2CC(CCNC(c3cccc(F)c3)=O)C2)cn1 c1(NC(=O)NC(c2cc(F)cc(Cl)c2)CC2CCCC(C)C2)ccnc(F)c1Br C1(NC(=O)CCC2CCOC2)CC(N=c2[nH]nco2)C12CCC2 CN1CCCC1C=CC(N1CCC(CCNC(C2(C#N)CC=CC2)=O)C1)=O C(C(=O)N1CC(O)CCO1)N(CCC)C(c1cnc(C)[nH]c1=N)=O CC(C)(C)C1=NOC(C(=O)NCC2CC2CNC(=O)CCc2ccc(Cl)s2)C1 S(=O)(=O)(c1cn(C)c2c(Br)cccc12)NC(c1ccc(C)c(C)c1)C(=O)O N1(C(C(C)=C2CC2)=O)CCCCC2(CCN(c3ncc(S(C)(=O)=O)cc3Cl)C2)C1 Cc1cnn(C)c1C(=O)NC1CC(CNC(=O)C=C(C2CC2)C2CC2)C1 c1(OC)ccc(N(C(C(=O)N)c2cnsc2)C)cc1.N(CCSC)(CC)CC C1(CC)CC(C(N2CCCC2(CNC(=O)C=CC(=O)NC)COC)=O)CC(=O)N1 N1(C(=O)CCC2CCCO2)CC2CC(C1)N2C(=O)C=Cc1ccccc1F N1(C(C(C)Cc2ccncc2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 CCC(CC)(CO)C(=O)NCC(C)(C)CN(C(=O)CC1CN2CCC1CC2)C CCC(CC)CCCC(=O)NC1COC2(C1)CN(C(c1cc(CO)c(C)o1)=O)C2 N1(C(C2N(C(c3coc(C)n3)=O)CCC(=C)C2)=O)CCC(O)CC(C)(C)C1 c1(NC(C(c2ccccc2)OC)=O)oc(=NC2CCC(=O)CC2)[nH]c1C N1(C(C2ON=C(CC)C2)=O)CC=C(C(C)(C)C(=O)NC(CC)C(N)=O)C1 c1(CNC(C2(N(C(C(CO)OC)=O)C3CC3)CCC2)=O)ccc(O)nn1 C(=O)(C1=CSCCO1)N(C1CCN(C(=O)C2=NOCC2)C1)CC Cc1ccc(CNC(C2(CNC(c3ncsn3)=O)CC2)=O)cn1 C1(CCNC(C=CC(=O)N(C)C)=O)(NC(=O)CC2NC(=O)NC2=O)CCOCC1 C=CC(C)(C)CC(=O)NC1C2CC1N(C(c1c(F)cncc1Br)=O)C2C Cc1ncc(CCC(N2CC3CC2CN3C(C2CC(=O)NC(=O)N2)=O)=O)c(O)n1 C(=O)(C1CCN(C)c2ccccc21)N(CC(CC)NC(c1cccc(O)n1)=O)C Cc1ccn2cc(C(=O)NC3CC4(C3)CN(C(=O)CC(C)C(F)F)C4)nc2c1 c1(CN2CCCN(C(c3c(C#C)cccc3)=O)CC2)c[nH]c2ccncc12 N1(C(c2cc(C)nc(O)n2)=O)CCN2C(=O)C(NC(=O)CC3CCCC3)CC2C1 C1(CNC(C=C(COC)C)=O)COC(CNC(c2nccn2C)=O)C1 c1(N2CCC(NC(C(C)S(C)(=O)=O)=O)C(C)C2)cc(C#N)ccc1[N+](=O)[O-] Cn1ncc(CNC(C2(F)CCN(C(=O)CCC3CC3(C)C)C2)=O)c1O C1(CN(C(CN(C(COC)=O)C)=O)C)CN(C(=O)C(C2CCCC2)OC)CC1O C#CCC(CC#C)C(=O)NC1CC1NC(=O)CCCN(C)C(C)=O c1(C(N2CCC(C(C#C)C)CC2)C(=O)NCCSC)ccc(Cl)c(Cl)c1Cl C1(C(=O)NC2C(C)CN(C(=O)C3=CCCS3)CC2)C2CCCCCCC12 C(=O)(C(O)C(C)(C)SCC#N)NCCN(C1CCCC1)C(CNC(CN(C)C)=O)=O n1(C(C2(C)CC2)C)nc(-c2cccnc2)nc1CCS(C)(=O)=O O=C(CCCC#Cc1ccccc1)OCC(Cl)=CCl Cc1noc(C(=O)O)c1C(N1CCCCC1c1nnc(CC(F)(F)F)o1)=O N1(C(C(C(CC)C)OC)C(=O)NCCC2CC2)CC2CCC(C1)C2(F)F C1(C(=O)NCC2(C)CCN(C(=O)C(O)CC3CCCC3)C2)CCC2(CCC2)CO1 c1(OCC)ccc(CNC(c2nnnn2C2CCOC2)CCOC)c(Cl)c1 c1(CC)cccc(C(N2CC3CC2CN3OC(=O)Cc2nonc2C)=O)c1C c1(N(C)C)cccnc1C(=O)NC1CCCCC1NC(=O)CCNS(C)(=O)=O c1(C(N(CCNC(C(CC#C)(C)C)=O)C2CC2)=O)c(C)cc(OC)cc1F N1(C(c2c(C)nns2)=O)CCC(CNC(c2cn(CCO)nn2)=O)C(O)C1 C1(N(C(CN(C(=O)C(C)C(C)O)CC)=O)C)CN(C(=O)OC(C)(C)C)CCO1 Cc1csc2cc(C(N3C4CCC3CC(NC(=O)CC(C)C(F)F)C4)=O)[nH]c12 N1(C(c2c(C)cc(N)cc2)=O)CCC2(CCC(NC(c3cncs3)=O)C2)CC1 c1(OC2CC3(C(=O)OCC)C2C3)ccc(Cl)c(C)c1 Cc1cc(C(=O)NCCC2(O)CCN(C(=O)COCCF)CC2)ccc1C(F)(F)F N1(CC(=O)NC(C2CC(NC(Cc3nc(C)sc3)=O)C2)C)CCC(O)CC1 C1(S(N)(=O)=O)(C(N(CCCCNC(c2cnc(C(C)OC)s2)=O)C)=O)CCCC1 C1(C(N2CC(=C(CNC(C(CO)N(C)C)=O)F)C2)=O)COc2ccccc2O1 N1(C(c2nc(-c3ccc(C)c(C)c3)on2)=O)CC(C)C(O)C(C)C1 c1(C(=O)NCCNC(C=C)=O)nc2ccc(-c3cnc(C)c(C)c3)cc2cc1C C1(N(C(C2CC2c2ccc(Br)o2)=O)CC)CCN(C(=O)C(F)F)C1 Cc1c(Br)ccc(C(=O)NC2CC(NC(c3c(F)ccc(O)c3F)=O)C2)c1C CC1C(NC(=O)CC2CCCC(=O)C2)CCN1C(c1cncc(C(N)=O)c1)=O Cc1ccc(C(CNC(c2c(C)n[nH]c2C)=O)NC(=O)CS(C)(=O)=O)cc1 C1(NC(C(CC)C)=O)CC2CC(C1)N(C(=O)CCCN1CCCCC1)C2 CC1CCC(C(=O)NCC(C)(CO)NC(=O)Cc2cc(C3CC3)on2)CC1 c1(C(=O)NC(CC)CNC(c2cc(C3(C)COC3)no2)=O)cc(Cl)cn1C Cc1cnc(C(=O)NCCC2CCN(C(=O)CCCC3CCCCC3)C2)nc1 N1(C(C(C(=O)OCC)C2CC2)=O)CCCCC(CNC(=O)Cc2nccn2C)C1 C(C(CC(C)C)C(=O)NCCC1COCCO1)NC(c1nc(C)n(C)c1)=O c1(OC)cc(C(N2CC(NC(=O)CC3(O)CCCCC3)CC2C)=O)c(N)c(C)c1 N1(C(=O)CN2CCCCC2)CC2CCCN(C(C3CN4CCCN3CC4)=O)C2C1 C1(NC(c2cc(C)sn2)=O)CCC2CCN(C(C3CCC4CC3C4(C)C)=O)C1C2 N1(C(C2=C(C)OCC2)=O)CC2(CCCC2NC(c2cc(N)c(F)cn2)=O)C1 c1(OCC)cc(C(=O)NCC2(NC(C3CC4CC4C3)=O)CCOC2)oc(=O)c1 CC(C(C)(C)C(=O)N1CC2(CC2)C1)NC(=O)CSC1CC1 Cc1nc2c(s1)CC(C(=O)N(CCNC(=O)COCC1CCOC1)C(C)C)CC2 n1(CC(=O)NCC2CCN(C(C(CCC)CC)=O)C(C)C2)cc([N+](=O)[O-])c(C)n1 c1(SC(C)C)ccc(NCC2C=CCOC2)cn1 C1(N)(C(=O)NCC2(CC)CCCCC2)CCC2CCCC12 c1(NC2C(OC)CCCC2)ccc(Br)c(C)n1 N1(C(COCCOCCOC)=O)CCC(C)(C)C1CC(=O)NC1C=C(C)CCC1 C(=O)(C(C)C(=O)NCCCOCCNC(=O)CNC(=O)C(F)(F)F)OC Cc1cc(Br)c(N)cc1C(=O)NC1CN(C(=O)Cc2c(C)cccc2C)C1 CC(C)C(CN(C)C)C(=O)N(C1CCCN(C(=O)C(C)(C)OCC(F)(F)F)C1)C C1(NC(CSc2nc(C)[nH]n2)=O)CN(C(=O)C(C)C)CC1CC(C)(C)C N(C)(C(=NCCC1(C)CC1(F)Cl)NCCc1cccs1)CCNC(C)=O N1(C(C(CCOC)(C)C)=O)CCCN(C(C2CC(N(C)C)C2)=O)C(CO)C1 C1(N(C(=O)COC2CC=CC2)CCC)CCN(C(=O)C=CC(=O)N(C)C)C1 CC(C)(C)CC(O)C(=O)N1CC(O)(C2(CNC(C3(C(F)F)CCCC3)=O)CC2)C1 Cc1cncc2cc(C(N3CCC(CC(C)NC(=O)CCC#N)CC3)=O)sc12 c1(C(N2C(C)(CNC(=O)C(O)C3CC3)CCC2)=O)nc(Br)n2ccccc12 C(=O)(C1CCCc2n[nH]cc21)N(C)CC1CCCN1C(c1cc(I)c[nH]1)=O c1(C(=O)NC(CCN(C(C(CC)OCC)=O)C)C(C)C)ccn2cccc2c1 N1(C(C(CC)(C)CO)=O)CCCC(C2(NC(C3CCCCC3)=O)CC2)C1 C#CC(C(C)OC)N(C(c1cn(C)nn1)C(=O)NCCCOC)C CCCCCCC(F)C(=O)N1CC2CC1CN2C(=O)C(=C1CCCCC1)F C1(NC(C(C)=CC2CC2)=O)CCCN(C(=O)C(C)Cc2ccccc2C)C1 c1(C(C)C)cncc(C(N2CCOC(C(C)NC(c3cccnc3S)=O)C2)=O)c1 c1(C(N2CC(C)C(CNC(c3ccoc3)=O)C2)=O)sccc1S(=O)(=O)C(F)F N1(C(C2(CF)CCN(C(c3c(C)cnnc3)=O)C2)=O)CC(F)(F)CCC1C c1(CC)ccc(CCC(=O)NC2(C)CCCC2NC(=O)C=C2CCC2)cc1 c1(OC)ncc(F)cc1C(=O)NC1CC(NC(c2cc(F)ccc2O)=O)C1 C1(NC(C2(C#C)CCC2)=O)CN(C(C2(N(C)C)CCCOC2)=O)CC1OC Cc1nnc(O)c(C(=O)N(C)CC2CCN(C(c3ccc(F)cc3Cl)=O)C2)c1C c1(C(N2CC(CC=C)(NC(C3CN(C(N)=O)C3)=O)C2)=O)csc2nccn12 N1(C(C2C(C)(C)C2)=O)CCC(CCC(=O)NOCCCCF)CC1 c1(C(N2CCCC(n3cc(-c4cnccn4)nn3)C2)=O)coc(=O)c(Cl)c1 C=C(C)CC(C(=O)NCCOC)NC(=O)CN1C(=O)CCCC1=O N1(C(C2OCCC(C)C2)=O)CC(C2CCN(C(=O)Cc3cccc(O)c3)CC2)C1 C1(NC(C(C)(C)OC)=O)CCCC(NC(=O)COc2ccsn2)C1 c1(C(=O)NC(c2cnc(C)s2)C)c(CNC(=O)CNC(=O)C(C)(C)C)cnn1C c1(C(=O)NCC2N(C(CCc3cnc(C)o3)=O)CC2)cccn2nccc12 c1(OCC(C)C)ccc(C(N2CC(O)(C(=O)Nc3nc(=O)o[nH]3)C2)=O)cc1 c1(C(=O)NCCC(C)N(C(CCCOCCC)=O)C)ccc(C(C)C)c(C)c1 N1(c2ccc(S(=O)(=O)N(C(C)C)C)cc2)Cc2ccccc2OC2(CCOC2)C1 O=S(=O)(c1cc(F)c(F)c(Cl)c1)NC(C1CCCCC1)CNC1C2COCC12 C1(NC(CCc2onc(CN)n2)=O)COc2ccc(F)cc2C1 C1(C(C)C)CCC(C(=O)NC(C)Cc2cccnc2)N1C(c1cnc[nH]c1=N)=O N1(C(C(C)=C(C)C)=O)CCC(CF)(NC(=O)CCC(=O)c2cccc(Cl)c2)C1 CC(CC(=O)N1CCCN(C(c2ccc(F)c(C3(C)CC3)c2)=O)CC1)C(F)(F)F c1(C(N2CC(NC(C(C(C)SC)O)=O)C2)=O)cc(C)cc2c1CCC2 c1(C(=O)NCCCC(C)NC(C(CC(C)C)OC)=O)cc2c(cc1F)NCCC2 n1(CC)cc([N+](=O)[O-])c(=NCC(=O)N(C)CCN(C(=O)CSC(C)C)C(C)C)[nH]1 C1(CNC(c2occ(C(=O)OC)c2)=O)CN(C(=O)C(=O)CC(C)C)CCCO1 c1(C(=O)NC2CC(F)(CNC(C3(C)CC3F)=O)C2)cc(N)c(F)cn1 C(CC(=O)Nc1ccc(O)cc1C)(C(F)F)NC(C(COC)COC)=O N1(C(Cc2ccn(C)n2)=O)CC(NC(=O)C(F)(F)CO)C(F)C1 Cc1cc(C#N)ccc1C(N1CC(NC(=O)CC2(O)CCC2)CC(C)C1)=O C1(NC(C(=O)NCC2CC2)=O)C2CC3CN(C(c4c[nH]nc4Cl)=O)C1C3C2 Cc1sc(C)c(C(N2CCC(NC(c3cccnc3)=O)CC2)=O)c1C c1(C(=O)NCCN(C(C(CC)C(=O)OC)=O)C)cc2cc(F)cc(F)c2[nH]1 CN1CCC(CC(=O)NC2CC23CC(NC(=O)CCC2CC2(C)C)C3)CC1 CCC(C)CCC(O)CC(=O)N1CC(F)(CNC(=O)CC2CCC=CCC2)C1 N1(C(CC2CN(C)C2)=O)CCOC2(CCC(N=c3ccnc(S(C)(=O)=O)[nH]3)CC2)C1 c1(C(=O)NCC2CC(NC(CCC)=O)C(O)C2)nc2ccccc2[nH]1 C(=O)(CCCCCN(C(=O)C(=O)N(C)C)C)NCC1NCCN(C)C1 c1(N2CC(C)=C(C)C2)[nH]c(=NCCC2CCC2)nc2c1cnn2C Cc1cc(C(C)(C)C(=O)N2CC(NC(c3cnc(C4CCOC4)s3)=O)C2)cs1 C1(n2cc(-c3cnc(OC)s3)nn2)CN(C(c2sccc2OC)=O)CC1O c1(OC)ncc(C(=O)NC(C2CCCN2C(=O)CN(C(=O)C(C)C)C)C)nc1C c1(C(N(CC(C)O)CCNC(=O)C2=C(Cl)CC2)=O)cccc2sncc12 N1(C(c2c(C)cncc2)=O)CC(NC(C2CNC(=O)N2)=O)CC(C)C1 c1(C(=O)OC)ccc(C)nc1N1CCOC(CNC(C2(C)CCCOC2)=O)C1 CC1CN(C(=O)C(=O)Nc2ncc(-c3ccccc3)s2)CC(C)(C)O1 C=CCC(CC(=O)N1CCOCC1C(C)(C)C)NC(=O)C=CC(C)(C)C C1(C(=O)NC2C(NC(C3(C=C)CC3)=O)C2)CC2(C1)C(C(=O)OCC)C2(F)F N1(C(c2cn(CC(=O)OC)nn2)=O)CCC(N(C(=O)C(COC)N(C)C)C)CC1 c1(NCC2C(NC(c3nc(OC)cc(OC)n3)=O)CCC2)ncc(C)cc1[N+](=O)[O-] c1(C(=O)NCC2(F)CC(NC(C(CC)n3cccn3)=O)C2)ccc(Cl)c(C)c1N C1(C(N(c2cccc(C)c2)C2CC2)=O)CCC2C(OCCN2C(=O)OC(C)(C)C)C1 C1(C(=O)NCc2cc(C)c(C(N3CCCC(C(C)C)C3)=O)o2)(OC)CCCCC1 CCCCC(C(=O)N1CC(C2(OC)CC2)C1)NC(=O)CNCC(N1CCCC1)=O C1(C(N(C2CCN(C(C=C(CC)CC)=O)C2)C)=O)CCCN(S(N)(=O)=O)C1 c1(Cc2scc(C)n2)nc(COc2ccccc2)nn1-c1ccnc(Br)c1 N1(C(Cn2ncc(C#C)c2)=O)CCCC(O)(CCNC(=O)C(C)NS(C)(=O)=O)C1 N1(C(C2C(CNC(C3(COC)COC3)=O)C2(C)C)=O)Cc2cccnc2C1 Cc1ccccc1OCCC(=O)NCC1CCCN1C(C1CCSC1)=O c1(C(=O)NCC2N(C(C(CCCC)O)=O)CCN(C)C2)c(OC)ccc(F)c1N c1(C(=O)NC(CNC(c2c(C)[nH]nc2CO)=O)C(C)(C)C)cc(Cl)cc(Cl)c1 c1(OCC)ccccc1C1CCN(Cc2nccn2C)CC1 c1(NC(c2ccn(C)c(=O)c2)c2n(CCCCCC)nnn2)c(C)cccc1C C1(C)(CC)C=C(C(=O)N(C2(CC(=O)NCCC#CC(C)(C)C)CC2)C)C1 N1(CCCc2cccc(C)c2)CC2CCC(NC(=O)COC3CCCC3)CC2C1 C1(NC(C(=O)NC(C2CCCOC2)C)=O)CCC2(C1)CC2(F)F C=CC(C)(O)C(=O)N1CCCC(C(C)NC(c2nncn2CC)=O)C1 Cc1ccc2c(c1)C(N(S(=O)(=O)CC1(c3ccccc3)CC1Br)C1CC1)CCCO2 N1(C(c2c(C)ccc(O)c2)=O)CCC2CN(C(c3ccc(Br)cc3Br)=O)CC12 c1(-c2nc(C(C)OCC)nn2CC2CCCOC2)cc2ccccc2cn1 c1(C(C(=O)OC)N(C)C(=O)NC(C)C)ccc(OC)c(Cl)c1 N1(C(C(CC#C)CC#C)=O)CCC2(CCN(C(=O)C=C(C)C(F)F)C2)C1 C1(NC(C2(C)CCOC2)=O)CCOCC1NC(c1ccnn1CC(F)(F)F)=O O=S(=O)(c1c[nH]ccc1=NCC1(COC)CC1)N(CC(F)F)CC(C1CCC1)O C1(CC(N2CC(CC(C)NC(c3ncoc3Br)=O)C2)=O)CCCCC1 C1(NC(C(CC=C)CC(C)C)=O)CN(C(=O)COCC(F)F)C2(CCOCC2)C1 C1(NC(c2ccc(C(CC)=O)cc2)=O)(CC)CCCN(C(c2sncc2C)=O)C1 C=CCC(C)(CC)C(=O)NCC1CC1C(=O)NC1(c2ccc(O)cc2)CC1 C1(NC(C=CCN(C(=O)CCNC(N)=O)C)=O)CN(C)CC12CC2 c1(C(=O)NCC(CC)(CCO)NC)ccc(F)c2occc12 c1(CC(=O)N(C2CCN(C(C(C)(C)SC)=O)C2)C)oc2ccccc2c1C C1(CNC(c2nc(C)oc2)=O)CC2(CCN(C(=O)CCC=CBr)C2)CO1 N1(C(Cc2c(CC)noc2CC)=O)CC2CC1CN(C(=O)C(C)(C)CF)C2 N1(C(C2(c3cccnc3Cl)CC2)=O)CCCC(C(=O)N(CC(C)OCC)C)C1 c1(C(=O)NC(C2CCN(C(c3cnn(C)n3)=O)C2)C)c(F)ccc(Cl)c1N C(=O)(CC(C)(C)CC)N(CCCC(=O)NCCCCOCC)C C(=O)(C1=CCCN(C(=O)CC2CCC(C#N)C2)C1)NCCOCC=C C1(N(C(C(=O)NC(CN(C)C)CCO)=O)C)COC(C)(C)C1 c1(COC)nc(C(=O)NCC(C(C)C)NC(c2conc2C2CCC2)=O)co1 n12cnc3c(ncn3c1=S)CC2.Cc1ccc(C(F)(F)F)cc1N1C(=O)CNC1=O C1(C(N2CCC(NC(C3(c4ccccc4)CCCO3)=O)CC2)=O)CC2CCC1O2 Cc1nc(CO)ncc1C(N1CC=CC1CNC(=O)CC(C)n1cccn1)=O N1(C(C)=O)CC(O)CC1C(=O)N(C)CCN(C(=O)C=Cc1ccn(C)c1)C N1(C(CCN(C(C(c2ccn(C)n2)C)=O)C2CC2)=O)CCC(C2CCCC2)C1 N1(C(CC(CNC(C2(COC)CCOC2)=O)C)=O)CC2(CCNC2=O)C1 C#CCCCC(C)(N)C(=O)NC(CN1CCC1)CC CCCC(C(F)(F)F)NC(C1(CCNC(=O)CN2CC(C)(C)C2)CC1)=O CS(=O)(=NC(=O)C1(N)C2CCCCC2C1)c1ccccc1Cl C1(C(=O)NCCOCCCNC(C2CCOCC2)=O)CC(=O)N(C2CCCC2)C1 N1(C(CN(C)C(=O)C2CC2)=O)CC2C=CCC(C2)C1.c1ncn2c1CCC2 N1(C(CCNC(COC)=O)C)CCN(C(=O)CC23COC(CF)(C2)C3)CC1 c1(C(N2C(C)(CNC(C3C(Cl)(Cl)C34CC4)=O)CCC2)=O)ccc(O)nc1Cl c1(-c2cnc(NC)nc2)cc(C(=O)Nc2nc(OC)ccc2Br)c2[nH]ccc2c1 c1(NC(C)=O)ccc(C(=O)NC2CN(C(=O)COCCO)CCC2C)cc1F c1(OC)ccc(C(=O)N(C)CC2CCCN2C(c2nn(C)cc2N)=O)cc1O C1(NC(C(C)Cc2ccccc2)=O)COCCN(C(c2cc(F)cs2)=O)C1 Cc1ccc2c(c1)c(CCOC(c1ccc(OC3COC3)cc1)=O)cn2CC(N)=O N1(C(C(c2ccc(C)s2)C)=O)CC2(CC2)CC1CNC(=O)CC1CCSCC1 C1(NC(C2C=CCCC2)=O)CC(=O)N(C2CN(C(c3cn(CCO)nn3)=O)C2)C1 c1(NCC2CCC(NC(CC(C)(C)c3ccccc3)=O)CC2)cc(Cl)cc(I)c1 c1(C(=O)NC(C)(C)CNC(c2cccc(Br)c2)=O)ccc(N)c(Cl)n1 c1(NC(C)=O)cnccc1C(=O)NCCCN(C)C(c1cc(C)sn1)=O n1(-c2cccc(C(C)=O)c2)[nH]c(=NCc2ccsc2)cc1C N1(C(CC2C(C)C(=O)CC2)=O)CCC2CCC(NC(=O)C=CC3CCOC3)C1C2 C=CCCC(C(=O)NCc1nn[nH]n1)NC(=O)CC1CC(=O)NC1=O Cc1cc(NC(=O)COc2ccsn2)ccc1NC(C1CCC(=O)N(C)C1)=O c1(CC)nc(Cl)c(C)c(=NC2CN(C(c3ccnn3C(C)CC)=O)CC2(C)C)[nH]1 N1(C(CNS(CC)(=O)=O)=O)CC(F)(F)CC1CNC(=O)C=C(C)C(F)F Cc1ccc(Cl)cc1OCC(N1CCC1CNC(=O)CC1CCNC1=O)=O CN1CCC(C(=O)NCC23CCCC2C3)(NC(=O)CC2CCCCO2)C1 c1(C(=O)NC2C(CNC(=O)CC3(CO)CCC3)C2)cnn(-c2ccccc2)c1F C(c1ccc(F)c(F)c1)=C(C)C(=O)N(C)CC1(O)CN(C(c2cnnn2C)=O)C1 c1(C(=O)NCC2(C(C)(C)O)CN(C(CCCOCC)=O)C2)ccccc1CC#N CC(CC(C)(C)C)C(=O)NCC1(C(C)(C)O)CN(C(=O)CCCNC(=O)C2CC2)C1 C1(C(N2C(C)CC2C(=O)NCC2CC(CN=[N+]=[N-])C2)=O)CC(F)CN1C c1(CCC(N2CC(NC(CCOCCC)=O)(CF)C2)=O)ccc(F)cc1 N1(C(C2CN(C(N)=O)C2)=O)CC(NC(=O)Cc2ccncc2Cl)CC12CCOC2 Cc1c(C(=O)NC2CC(NCc3cc(F)cc(F)c3)C2)ccc2c1OCCO2 C1(C(=O)NCCOCCNC(=O)CC2CCC3CC23)CC(=O)N(O)C1 N1(C(N(c2c(C)cccc2)C)=O)CCCN(C2COC2)CC1 c1(OCC)ccc(F)c(C(=O)NCC(O)CNC(C2(C)CCCC2)=O)c1N c1(SCC(N2C3(CNC(CN(C)C(N)=O)=O)CC(C2)C3)=O)nc2ccccc2[nH]1 C#CCC(C)(CC)C(=O)NCCC(Cc1ccccc1)NC(=O)C(C)CCC C(=O)(C1=NOC2(CCN(C(=O)C(c3ccccc3Br)O)C2)C1)NCC(=O)NC CCC(CC(=O)NCC1CCCN(C(=O)C(=Cc2cccnc2)F)C1)C(C)C Cc1nn(C)cc1CC(N1CCN(CC(N2CC(C)(F)C2)=O)CC1)=O c1(CNC(CCN(C)CC)=O)ncc(F)cc1F.c12ncoc1CCNC2=O c1(CN2C(C(N3CCCC(O)C3)=O)CC(C)C2)cccc2cn[nH]c12 c12ccc(c(F)c1)-c1cc(ccc1OC(C)C)COC2=O.CCC(C)N(C)C CC1CN2CC1N=C1C3=C(NC(SC(F)F)=NC(Cl)=C2C#N)CCC13 N=c1c(C(N2CCCCC2CCNC(C2(F)CCCC2)=O)=O)c[nH]cc1Br C12(CNC(=O)C(c3ccccc3)N3CCCC3)CC(CO1)N(C(c1ccco1)=O)C2 N1(C(c2nnn(C)n2)=O)CC2(C)CN(C(c3ccc(=N)[nH]c3)=O)CC2(C)C1 c1(CNC(=NCCC#C)NC2CC2CF)c(C)[nH]c2ccccc12 C1CC(NC(C)=O)C(=O)N1.C(C)(C(N)=O)N(C(C=CC)=O)CC CC1CN(C(C23CC(F)(C2)C3)=O)CCCN1C(=O)C(Cc1ccccc1)C1CC1 N1(C(c2c(CC)cncc2)C(=O)NCCOC)CC(C)(C)OCC1C N1(C(c2cccc(OC)n2)=O)CCC2CCCN(C(=O)CCCS(N)(=O)=O)C2C1 c1(CCC(=O)NC(c2cccc(Cl)c2)CNC(CC=CCC)=O)cccc(F)c1 c1(NC(N2CCC(c3ccc(Cl)nc3)CC2)=O)cnc(Cl)c(Cl)c1 C1(OC)CN(CCOC2CCN2C(=O)C(C)=CC(C)(C)C)C1 c1(CCC(=O)NCC(CNC(C=CC)=O)O)ccc(Br)cc1 C(=O)(C1=CCC(F)(F)CC1)N1CC(SC)C(CNC(c2cc(C)cc(O)n2)=O)C1 c1(C(C)NC(=O)NC2CCCN(C(CC)C)C2)cc(OC)cc(OC)c1 Cc1nn(C)c(Cl)c1C(=O)N(C1CCC(NC(C2CCCCCC2)=O)CC1)C N1(C(c2cc(C)nnc2O)=O)CC2CCC1CN2C(C1CC(=O)N(C)C(=O)N1)=O c1(Oc2cc(C(N3CCC(OC(C)=O)C3)=O)ncc2)ccc(S(C)(=O)=O)cn1 C1(NC(c2c(C)nn[nH]2)=O)CCC2CN(C3CCC=CCC3)CC2C1 Cn1ccc(C=CC(=O)NC2COCC2n2cc(CCC3CCCOC3)nn2)c1 Cc1ccc(Cl)c(NC(=O)NC2CC2C(=O)NCc2cccc(F)c2C)c1 c1(OC)cc(C)c(C(=O)N(C2CN(C(C3CCCC(C)(C)O3)=O)C2)C)cc1Br C12(NC(CCN(CC)CC)=O)CCOCC1CN(C(=O)C(C)SC(C)C)C2 Cc1c[nH]cc(C(=O)NC2COCC2NC(c2ccc(Cl)c(F)c2)=O)c1=O c1(N(CCOC)C)ccnc(C(=O)NC2CCN(C(=O)C(O)CC3CCCC3)C2)c1 c1(C(=O)NC(CCCNC(c2c(CC)n[nH]c2)=O)(C)C)cnc2n1CCOC2 c1(C(=O)OC(c2c(Cl)cccc2Cl)C)cc2c(s1)CCCCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NCC1C2CCCCC12)C1(C)CC1 N1(C(C(CC)(F)F)=O)CCN(C(=O)CC2CCCNC(=O)C2)C2CCCC12 c1(C(=O)OC)ccc(Cl)c(CN2CCC(CC(=O)Nc3nccs3)CC2)c1 C1(CN(C)C)CCCCN1C(C1C=CCN(C(C2CNC(=O)O2)=O)C1)=O C1(NC(c2cc(OC)ns2)=O)CC2CCCC(C1)N2C(C1(F)CCN(C)CC1)=O C1(C(=O)NC2CCN(C(C(C(C)(C)C)NC(C)=O)=O)C2C)CCn2nccc2C1 c1(C(=O)NCC=CCNC(C2(C)CCC(C)C2)=O)csc(=NC2CCCCC2)[nH]1 c1(NC(=O)NC2CC(NC(Cc3cccc(OC)c3)=O)C2)ccc(C#N)cc1I C(CC(C(C)(C)C)NC(C1(F)CC=CCC1)=O)N(C)C(C1(C)COC1)=O C(CN(C(C1CCN1C(C)(C)C)=O)CC)(C(C)C)NC(CN(CC)CC)=O C1(OC)CC(C(=O)NC2(CCOC)CC2)N(C(C2C3CC(=O)CC23)=O)C1 C1(C(=O)NCC2(CNC(c3c(CC)[nH]cc3)=O)CC2(F)F)CC2CCC(C1)N2C Cc1cncc(C(N2CC(F)(CNC(C3CCN(C)C3C)=O)C2)=O)c1 CC1(C)CCC(CC(N2CCC2C(=O)NCCN=S(C)(C)=O)=O)O1 C1(NC(C(CCN(C)C)NC(=O)CCCn2cccn2)=O)CC2CC3C(C2)C13 Cc1noc(CNC(=O)NC(COC(C)(C)C)C(F)(F)F)c1C CC1(C)CCCCC1CN(C(=O)C(=O)NCC1CC(C(N)=O)=NO1)CC1CC1 C12(C(=O)NC3CN(C(c4n(C(C)C)ncc4Cl)=O)C(C)C3)CC(C)(C1)OC2C C(=O)(C1=CCCOCC1)NCCOCCCN(C)C(c1[nH]cc2c1CCCC2)=O C1(CNC(CNC(C)=O)=O)CCCC1C(=O)NCCN(C)C(C)=O CCCC(C(=O)N1CCC1CC(C)C)NC(=O)C(C1CC1)OCC n1(CC(=O)NC2CCCN(C(CCC(=C)Br)=O)C2)cc(F)ccc1=O C(C(CNC(C12CCCC1(C(N)=O)C2)=O)C(F)(F)F)NC(Cn1c(C)ccn1)=O c1(C(=O)NC(Cc2cnn(C)c2O)C(=O)NCC(C)(C)O)cnn2cccc2c1 c1(CC)ccc(C(=O)NC(CO)CCCNC(=O)C2CC2)cn1 c1(NCCC(C)(C)NC(C(C(CC)(C)C)O)=O)ncc(C)c(S(C)(=O)=O)n1 c1(CC)cnsc1C(=O)NC1(C)CC(NC(C2CC2(C)C(F)F)=O)C1 C1(OC)CN(C(c2cc(C)c(O)nn2)=O)C(C)(CNC(=O)CC2CC(=O)C2)C1 C1(C(=O)NC(CNC(C2(C)CCCCO2)=O)C(C)C)(COC)CCCCO1 c1(C(N2CCC(C(=O)NC)C2)=O)cc(OCC(O)CF)ccn1 c1(NC(C(=O)NC(C2(c3ccccc3)CC2(F)F)C)=O)cnn(-c2ccccc2)c1 c1(C(N2C(C(=O)NCC3CC(COC)C3)CCC(O)C2)=O)cccn2ccnc12 Cc1cc(CCC(N2CC(C)(NC(=O)CC3(C)CCOC3)C2)=O)on1 c1(C(N2C(CNS(CC)(=O)=O)CC2)=O)cnoc1-c1ccc(Cl)s1 c1(C(=O)NCCCNC(C=CCN(C)CC)=O)c(OC)ccc(OC)c1[N+](=O)[O-] N1(C(C2C(C)(C)OCC2)=O)CCN(C(c2csc3nnsc23)=O)CC1CF c1(OC(C)C)ccc(C(=O)NCC(C)(O)CNC(C2CCC(CO)O2)=O)cc1 C1(C(N(C)CCn2cccn2)=O)C(C2CC2)CCN1C(=O)C=Cc1ccc[nH]1 c1(CC)c(C(c2nnnn2CCCF)NCCOC)ccn1C.OC(F)F N1(C(CC(C=C)C)=O)CC2(C=C(C(=O)N3CCC(O)C34CCC4)CO2)C1 CCCCC(O)C(=O)N(CCCCNC(c1oc(C(F)(F)F)nc1C)=O)C c1(C(=O)NC2CCCN(C(C3OCCN(C)C3=O)=O)C2)cnn2c(=O)cc[nH]c12 CCC(C(=O)N1CC(C(F)(F)F)CC1CNC(c1cc(F)n[nH]1)=O)C(C)C CC1(NC(=O)C2=CSCCO2)CCC(NC(=O)CNc2nccs2)CC1 C1(NC(C=C(C)C(C)C)=O)CC(N=c2ccnc(C(F)(F)F)[nH]2)C12CCC2 C1(NC(C(CC)CC)=O)CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC(F)(F)C1 c1(CC(C(=O)NCC(CNC(C=CC=CC)=O)(C)C)C)ccc(F)cc1F C1(C)(C(=O)NC(C2(O)CN(C(C3N(CC)CCOC3)=O)C2)C)CCN(C)C1=O N1(C(CCN(C(CCC)C)C)=O)CC(F)CC1CNC(=O)CS(=O)(=O)N(CC)CC C1(CNC(C(C=C=C)C)=O)CN(C(c2sccc2Cl)=O)CCC1(F)F c1(C(C)=O)cc(NC(N2CCC(CO)CC2C)=O)ccc1C CC12CC(NC(C3CCOC3)=O)(C1)N(C(c1ccncc1O)=O)C2 c1(C(C)C)nc(C(N2CCC(O)CC2)C(=O)C(=O)N)n(C)n1.C1CCOC1 C(C(O)CCNC(=O)Cc1ccn(CC(F)(F)F)n1)NC(C1(OC)CC1)=O c1(C(=O)NC2C3CN(C(c4c(CC)ccs4)=O)CC32)cccc2c1C(=O)CCN2 c1(SCC(=O)NC(C)CCNC(c2ccon2)=O)ccccc1F C(C(O)CC(C)(C)C)NC(C1(CCNC(C2C(OCC)CC2)=O)CCCC1)=O c1(C(N2CC(C(C(=O)OC)OC)C2)=O)sc(OC2CC2)nc1-c1ccccc1 c1(NC(c2ccc(F)cc2)C(=O)OC)ccc(Br)c(C)c1I c1(OC)ncc(F)cc1C(=O)NC1C2CN(C(=O)Cc3ccccc3C#N)CC12 Cc1ncccc1C(N1C(C(=O)NC(c2cscn2)CO)CC1C)=O N1(C(c2c(C)ccnn2)=O)CC(O)CCC1C(=O)NC1CCOCC1F C1(C)(CC)CC(NC(=O)C(F)=C(C)C)CN1Cc1ccc(F)cc1F c1(NC(C2CC(O)CN2C(=O)C=CCF)=O)ccc(N2CCOCC2)c(Cl)c1 c1(CC(=O)NC2C(C)N(C(C3CCC(F)C3)=O)CCC2)cn2c(n1)CCCC2 N1(C(CC(=O)NC)=O)CC(CNC(=O)C=Cc2ccc(C)o2)CCC1C c1(CC)cc(C(N2CCCC(N(C)C(c3nccnc3N)=O)CC2)=O)cc(O)n1 c1(C(=O)NCCN(C(c2sccc2C(C)(C)C)=O)CC)ncccc1Br C1(CCNC(c2nnnn2C2CC2)(COC)C2CC2)CCC2(CC1)CC2 c1(OC)ccc(C(=O)OC2(OC)CCO2)c(O)c1 C1(CC)(NC(=O)COCC2(F)CC2)CCCN(C(=O)C=Cc2cnn(C)c2C)C1 c1(CC)ccc(C)c(C(=O)N(CC)CC2CCN(C(=O)CS(=O)CC)C2)c1 c1(OC)cncc(C(=O)NCCC2CN(C(C3(F)CC3C)=O)C2)n1 N1(C(CC(C)c2cccnc2)=O)CCCC(C(=O)NC(C)(C)C)C1 C1(CNC(C(=O)NCC(CO)OCC(=O)NCC(F)(F)F)=O)CCCCO1 c1(N2CC(CNC(COC(CC)(C)C)=O)OCC2)c(C#N)nnc2ccccc12 C(=O)(C1=CSCCO1)N(C1CCN(C(=O)CC2CCC(C)(C)CO2)C1)C Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)CCC2CCCC2)nn1C(C)C c1(C(C(=O)NCCN(C(C2(COC)CCC(=O)N2)=O)CC)SC)cccc(Cl)c1 N12CCOC(C)C1C2=O.N1(C(C=C(CCC)C)=O)CCC(OC2CCC2)C1 C1(NC(=NCC=C)NCC(c2cccnc2)CO)CCc2cnn(CC(C)C)c2C1 n1(CC(=O)N(C(CNC(C2CC2C(C)(C)C)=O)C2CC2)C)cccc([N+](=O)[O-])c1=O N1(C(c2ncc(C)cn2)=O)CCC2(CCCC2NC(C2CCSCC2)=O)C1 Cc1cc(Br)ccc1C(=O)NCCC1(NC(C2CC23CCCC3)=O)CC1 C1(CNC(CC2CCC(C)CO2)=O)CCn2nnnc2C1.C1=CC(=O)N2C1CC2 N1(C(C(c2ccccc2)OC)=O)CCCC(NC(=O)C(=O)NC2CCCC2)C1C O=C(CC=C(Cl)Cl)NC1CCC(CC(=O)NC2CCCC2F)CC1 C1(C(N2CC(O)CC2c2ccc(F)cc2)=O)CC2(CC(N3CCOCC3)C2)C1 Cc1cc2c(C(=O)NCC3CCCN3C(=O)CCN3CCOCC3)cccc2o1 C1(c2cn(Cc3c(C)c[nH]n3)nn2)CCCN(C(C2CCCN2C)=O)C1 c1(C(N2CC3C(NC(=O)CC4CC4)C3C2)=O)cc(Br)cc2[nH]ccc12 c1(OC)nn(CC(=O)NC(=O)Cc2ccc(C)s2)cc1I N1(C(CCN(CCCCC)C)=O)CCOC(CNC(=O)CC2CC2(Cl)Cl)C1 c1(OC)cc(CCNC(C2C3CN(CC(N)=O)CC23)=O)ccn1 N1(C(C2C(C3C(C)C3)C2)=O)CC(C2CCCN(C(c3ncccc3F)=O)C2)C1 C(=O)(CC(C)(C)CN(C)C)NC1C(C(=O)NCC(C(CC)C)O)CCCC1 C1(NC(C2(OC)CCSC2)=O)CN(C(c2cccc(COC)c2)=O)CC1C C1(NC(CCCNC(C)=O)=O)CCN(C(=O)CCCc2cncs2)CC1(C)C c1(C(C)NC2CCOCC2N2CCOCC2)nc2ccccc2s1 N1(C(C2(CC#C)CCC2)=O)CC(CO)C2(CCN(C(=O)C=CSC)CC2)C1 N1(C(c2cnc(OC)s2)=O)C2CCC1CN(C(=O)CC1CCOC1)CC2 CC1(CNC(c2ccc(C3CC3(F)F)cc2)=O)CCCN1C(=O)CCC(F)F C1(N(C(c2nc(=N)[nH][nH]2)=O)CC)CCCN(C(=O)Cc2cnn(CC)c2)C1 c1(N2CC(C(N=c3ccc(OC)n[nH]3)=O)SCC2)ncc2ccc(F)cc2n1 N1(C=O)c2ccncc2CC1C.C#CCCCCCCN(C)N(C(C)(C)C)C(=O)CC c1(C(=O)NC(C2CCN(C(c3c(C)ncn3C)=O)C2)C)cc(N)nc(Cl)c1 CCCCC(C)(CO)NC(=O)C(C)N(C(=O)Cn1ncccc1=O)CC C(=O)(CN=c1cc[nH]cc1)N1CC(NC(CC(C(C)C)OCC)=O)C(O)CC1 c1(OC)cc(CNC2CCCCC2n2cccn2)c(OC)c2c1CCCC2 C(C(C)(O)CC(=O)N1CCCC1CNC(c1ccc(N2CCCC2)nn1)=O)OC c1(C(=O)NC2CC(C)(NC(CC(CC)C)=O)C2)cn2cccc(F)c2n1 C(CCCCC1OCCO1)(c1n(CCOCC)nnn1)NCC1CCC1 C#CCC(CC(F)F)C(=O)N1CC(C)CN(C(=O)C(CO)C(F)(F)F)C(C)C1 C1(C(N2CSCC2C(=O)NC(C2(O)CCC2)C)=O)(OC)CCC(C)C1 C12(CNC(C(CC)(C)C)=O)CC(NC(=O)CSCC(C)C)(C1)C(C)O2 C1(CC)C(C(=O)NC(CC(=O)NC2(CCF)CC2)C2CC2)CCN1C N1(C(CC(C)OC)=O)CCCCC(NC(c2cc(F)ccc2Cl)=O)C1 C1(C(=O)NCC(CO)N(C)C)CCC2(CC2)N1C(c1ncc[nH]1)=O c1(C(N2CC(O)(CNC(C3(C)CC=CCC3)=O)C2)=O)ccc2c(c1)NCCC2 c1(NC(=O)NCCCC)ccc(C(=O)NCCN(C2CCN(C)CC2)C)c(Cl)c1 c1(C(=O)NC2C(n3cc(CC(C)O)nn3)CCC2)ccc2nncn2c1 C(=O)(CC(COC)CN(C)C)NCc1nccc(C(N2CC(C(CC)C)C2)=O)c1 C1(OC)CC2CC(C(=O)N(CCNC(c3ccccc3Cl)=O)C(C)C)CC12 c1(C(N2C(C)CN(C(=O)Cc3cncs3)CC2)=O)c(F)cc(F)c(O)c1F Cc1ccccc1SCC(=O)NC1CCCC1CNC(=O)CNC=O C1(C(=O)NCCN(C(=O)C(c2ccc(F)cc2)=O)C)CCC(=O)NC1 C1(NC(COCCCC#C)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CC1(C)C Cc1cn(C(C)C(=O)NCc2cn(C3CCN(C(=O)CC4CC4)C3)nn2)cn1 N1(C(c2cc(C)c(Cl)c(C)c2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)C2CCCC12 CC(C)(CCCNC(c1ccsc1)=O)C(=O)NC1CCC2CCCC1O2 N1(C(=O)CC2CC3(CC3)C2)CCN(C(C2C3CCCCCC23)=O)CC(O)C1 N1(C(c2cc(OC(C)(C)C)ncc2)=O)CC2CCCC2(NC(c2cncs2)=O)C1 C1(C)(C(N(CC(=O)N(C)Cc2cc(C)n(C)n2)C)=O)CCC(=O)NC1 c1(C(N(C2CC(NC(=O)C(F)(F)C3CC3)C2)C)=O)cc(Br)c2[nH]nnc2c1 OC1(C2CC2)CCCN(N2CCOC(c3ccc(F)c(Cl)c3)C2)C1 c1(C(=O)NC(CCCC)CNC(=O)CCNC(=O)CCC)cc(F)cc(Cl)c1 CCC(C)(Br)C(=O)N1CCOCC1c1nc(C(F)(F)F)n[nH]1 CCCC(C)(CCC)C(=O)N1C2CCC1CN(C(C1C(C)C1C)=O)CC2 c1(CC(=O)NCC(CC)NC(C2(OC)CC3CCC2C3)=O)c(C)ncnc1C c1(C(N(C(C(=O)NC(CCOC)CO)C2CC2)C)=O)cnnc(C)c1 c12ncnc3c1nnn3N2C1COC1.Cc1ccnc(C)c1CC1CCCCC1 N1(C(COCCCC)=O)CCCC2(C1)CN(C(c1cccnc1N)=O)C2 N1(C(c2n(CC)ccc2)=O)CCC=CC1C(N1CCCCCC1)=O C1(CNC(C(C2CC(F)(F)C2)OCC)=O)CCCCN1C(=O)CCCOC(C)=O N1(C(C(F)=C(C)C)=O)CCC2(CC1)COC(CNC(=O)C(C(C)C)NC(C)C)C2 Cc1cc(C)n2ncc(C(=O)NCC3CCCN3CCC3CCCC3)c2n1 C1(NC(c2cccc(Br)c2)=O)CCN(Cc2ncccc2F)CC1F c1(C(=O)NCC(CNC(C2(C(CC)=O)CC2)=O)C)cn2cccnc2n1 c1(-n2c(-c3[nH]c4c(c3C)CCCC4)nc(C)n2)cc(Cl)cc2ccccc12 c1(C(N2CCC(CC=C)C2)C(=O)NCC)cncc(C(C)(C)C)c1 c1(OC)cc(N)c(C(=O)NC2(CCNC(c3cncnc3C)=O)CC2)cc1OC N1(C(c2ccc(Cl)cc2Cl)C(=O)NCCC)CC(C(=O)OC)C(C2CC2)C1 N1(C(c2c(C)nc(C)s2)=O)CCC(CNC(=O)CSC(F)(F)F)C(C)C1 c1(OC)ccc(Br)cc1C(=O)NCC1CCN(C(=O)CC2CCCC2)C1 C1(C(=O)NCCC(C)(C)NC(C=C(CC)CC)=O)CCN(C)S1(=O)=O c1(OC)cc(C(N2CC(C(=O)Nc3cc(F)c(Cl)nc3Cl)C2)=O)cc2n[nH]cc12 C1(C(=O)OCC)CCCN1NC(=O)C(C1CC1)Nc1ccccc1CC Cc1noc2ncc(S(=O)(=O)NCC3CCCC3N3CCCC3)cc12 Cc1cc(=NC(=O)Nc2ccc(-c3csc(=N)[nH]3)cc2)cc[nH]1 C=CCCC(C(=O)NCC(=O)OCC)NC(=O)C(C1CCC1)OCC Nc1ncc(Cl)cc1C(=O)NC1CC1CNC(C1(n2cccn2)CCC1)=O N#CC1CN(Cc2nccs2)CCN1C(c1ncc(Cl)nc1Cl)=O Cc1cnc(C(=O)NCC2(C)CCCN2C(=O)CN2CCC(C)(C)C2)c(F)c1 C1(CCC=C)(C(N2CCCC2CNC(C)=O)=O)CN(C(=O)C(C)N2CCC2)C1 c1(C(N2CC3CC4C(NC(C=C(C)Cl)=O)C2C3C4)=O)ccc2c(c1)NCCC2=O C(=O)(CCC(=O)c1cccc(F)c1)NC(CN(C(CC1(OCC)CC1)=O)C)C c1(C(N(C2CN(C(=O)Cc3cc[nH]n3)C2)C)=O)cc(F)c(O)c(Br)c1 Cc1ccc2nc(C(C)NC(=O)COC3CN(C(c4ccccn4)=O)C3)[nH]c2c1 c1(C(N2C(C(N(CCCCC(C)C)C)=O)CC2C)=O)cccc2[nH]ccc12 C1(CC)(NC(=O)C(C(C)O)N(C)C)CCCN(C(c2ccc(F)c(OC)c2)=O)C1 C1(NC(C(CCC)NC(=O)Cc2cccnc2F)=O)CCCCCC1CO N1(C(c2cc(C)oc2C)=O)CCN(C(C2CC3C(C2)C3(C)C)=O)CC1C(C)(C)C C1(C(=O)NC(C)C(C)C)C2CCC(C2)C1NC(=O)CCC(=O)N(C)C C1(CNC(C(CC)F)=O)CN(C(=O)COC2CCC(F)(F)CC2)CC2(CCC2)O1 C1(N(C(COc2c(C)cccc2)=O)C)CCN(C(=O)CCn2cccn2)CC1C N1(C(C)=O)CS(=O)(=O)CC1C(N1CC2(CCN2C(c2cc3c(s2)CCC3)=O)C1)=O N1(C(C(CC(C)C)(C)C)=O)CCCC(C2CN(c3nc(C(F)F)nc(=N)[nH]3)C2)C1 C(=O)(CCCCC(F)F)N1C(CNC(C2N(S(C)(=O)=O)CCC2)=O)CCCC1 c1(C(N2CCN(C(C(C(C)(C)C)NC(C)=O)=O)CC2C)=O)ccc([N+](=O)[O-])c(C)c1 C1(C(N2CCC(CNC(c3cncn3C3CC3)=O)C2)=O)CCc2ncsc2C1 CC(C)C(F)C(=O)NC1CCCCC1CNC(c1ncoc1C(C)(C)C)=O c1(C(=O)NCc2ccc(C(=O)NC3C(CC)CCC3)o2)c(SC)cnn1C CCC(CNC(c1coc(C(C)(C)C)n1)=O)(CC)NC(=O)COC1CC=CC1 CCN=C(NCC(CC)CCO)NCC1CCCC1c1cccc(F)c1 Cc1cc(C=CC(=O)NCC(CNC(C2C=CCS2)=O)CO)ccc1F C1(CN(C(C(C2CN(C(c3n(CC)ccn3)=O)C2)OC)=O)C)OCCC1(C)C O=C(C(F)(F)c1cnccn1)NCc1ncc(Br)s1 N1(Cc2cc(C(=O)OC)sc2Cl)CCCC12CCC2 N1(C(CCN(C(C(C)OC2CCCC2)=O)C)=O)CC(N(C)C)C(C)(C)C1 N1(C(CC(COC)C)=O)CCN(C(=O)C(=Cc2cccnc2)C)C(CF)C1 Cc1cc(SC2CCCC2(C)O)c(F)cc1[N+](=O)[O-] N1(C(CC=C)=O)CCC2CN(C(=O)Cc3ccc(F)cc3Br)CCC2C1 N1(C(c2ccc(OC)nc2)=O)CC(C)(C)CCC1CNC(c1cc(F)n(C)n1)=O c1(C(=O)NC(COC)CNC(=O)CSS(C)(=O)=O)cc(C)sc1C C1(C(=O)NC(CC)CNC(=O)CCc2cc(C)on2)C2Cc3c(Cl)cccc3C12 n1(CCSC)nnnc1C(C1CCOCC1)N(CC(C)OC(F)F)C1CC1 C1(O)(CC(=O)NCC(CC)Nc2cncc(C#N)n2)CCN(C)CC1 C1(C(N2CC(NC(C3CSCC(=O)N3)=O)(CO)C2)=O)CCc2nc[nH]c2C1 c1(NC2CCN(C(C(=O)NC(N3CCOCC3)=O)=O)C2)ccc2c(c1)OCO2 C(=O)(CC(O)CNC(C1CC(CC2CC2)C1)=O)NCC1(CCOC)CC1 N1(C2CN(N3CCC(C)C3)C2)CC(NCC=O)CC1=O.n1(CC(=O)N)cncn1 c1(CCC)cnnc(C(=O)NCCCNC(=O)C(C)Cc2c(C)n[nH]c2C)c1 c1(C(N2C(C(=O)NCC(=C)CC)CC2C)=O)cc[nH]c(=NC)c1 c1(C(N2CCC(C)(CNC(C3(F)CCC3)=O)C2)=O)cc2n(n1)CC(F)C2 C1(CNC(=O)C2=NOCC2)CN(C(C2CC(OC(F)(F)F)C2)=O)CCCO1 C1(C(N2CC(COC)(NC(=O)C(C)CC3CC3)C2)=O)CCCCC(F)(F)C1 C(C(C)(C)C(=O)NC1CCC(NC(=O)CCc2nnc(C)n2C)C1)OCC C1(CCC)CCC(O)(C(=O)NC(CNC(=O)CC(F)(F)F)C(C)(C)C)CC1 N1(C(C(C)(C)n2ccc(C3CC3)n2)=O)CCC2(CCC2(C)C)C1 C#CC1CN(C(=O)C(CCN(C)C)NC(=O)C(C)OCC(C)C)CC1O c1(N2CC(CO)(NC(=O)C(F)Cc3ccccc3)C2)nc(Cl)nc2sccc12 C(=O)(C(C)CCC(C)(C)C)N1C(C(=O)NCC(CCC)C)CCCC1 c1(C(=O)NCCC2(C)CCN(C(C3C=CCC3)=O)C2)cc2cnc(Cl)cc2s1 CN1CCCC1C=CC(=O)NCC1CC(O)(CNC(=O)CCC2CCOCC2)C1 N1(C(c2cnc(OC)c(F)c2)C(=O)NC2CC2)CCOC2(CCN(C)C2)C1 C12(NC(C=C3CCC(C)C3)=O)CC1CN(C(c1cc(-n3cnnc3)ccn1)=O)C2 N1(C(C(C2CCN(C(=O)NC3OCCC3(C)C)C2)C)=O)CCCC(CCF)C1 O=C(C1=CC2CCCCC12)NCC1CCCCC1NC(c1ncc(F)cc1F)=O c1(C(N(CC(C)(C)CNC(=O)CC23CCCC2C3)C)=O)cc2ncccc2[nH]1 C(C)(C(C(C)C)NC(c1cnn(C2CC2)c1Cl)=O)NC(C=COCC)=O c1(C(=O)NCC(C)CN(C)C(c2cc(Cl)ncc2N)=O)cccc2nccn12 C1(C)(CC(N2CCN(C(CCCSC)=O)CC2)=O)CCC(C(F)(F)F)CC1 N1(C(c2c(NC)cccc2)=O)C(C(=O)NC(C2CCCCC2)C)CC2CCCC12 C1(N(C(C2CCC(OC)CC2)=O)C)CCCN(C(C2(F)CCOC2)=O)CC1 C1(CC#C)(C(=O)NCCCCNC(C2CCOC2c2ccncc2)=O)CCOC1 C1(C(=O)NC2CCC(CNC(=O)C=Cc3ccsc3)C2)COC2COCC12 C1(C(=O)NCC2(CO)CCCN(C(CC(C=C)C)=O)C2)CCn2c(C)nnc2C1 N1(C(C2(C(F)(F)F)CCN(C)CC2)=O)CC2CN(C(c3csc(CO)n3)=O)CC12 c1(C(=O)NCC2CN(C(C3(N(C)C)CCC3)=O)C2)csc(Cl)c1 c1(OC)nc(C(=O)NCC(C)(C2CC2)NC(=O)CC(=O)N(C)C)co1 n1(C(C(=O)NCC(C)(C)OC)C)cc(CC2CCCOC2)nn1 c1(CN2CCC(C(C(=O)NC(C)C#N)C)CC2)ccc(C2CC2)cc1Cl CC1=C(C(=O)NCC(C)(C)CNC(C2SCCC2C)=O)CCC1 c1(-n2c(C(COC)NC(C3CCCCC3)CCO)nnn2)ccc(F)cc1 C(O)(CN=c1cc(C(F)(F)F)nc[nH]1)C1CN(C(c2nc(C)oc2)=O)C1 N1(C(=O)OC(C)(C)C)CCC(OC(CC(F)C2CC2)=O)C1 N1(CC)CC(C(=O)NC2CCC(N(C)C(C3CC3C(C)(C)OC)=O)CC2)CC1=O N12CC(CC(C)C1)NC(=O)CCc1nc(no1)CC2=O.c1(CCC)nnc(C)o1 C1(N(C)C)C=CCN(C(=O)C(Cn2cncn2)NC(c2cscc2C2CC2)=O)C1 C#CC1(C(=O)NCCOC(C)=O)CCN(C(=O)CN(C)C(C)=O)C1 c1(C(N(C)CC2N(C(C=CC(C)(C)SC)=O)CCC2)=O)cccc2c1CC(=O)N2 C1(CNC(COCC#C)=O)CCN(C(C2CCOC2C)=O)C1(C)C c1(C(N2C(CNC(=O)CCCC3CCCO3)CC(F)C2)=O)cnc2n1CCC2 CCCCCC(C)CC(=O)N(C1CCCN(C(c2cnn(C)c2Cl)=O)C1)CCF c1(OC)ccc(-n2cc(C3CN(C(=O)CC4CCCC4OC)C3)nn2)cc1 c1(C(CN(C(CC2(CO)CNC2)=O)CC)O)ccc(F)cc1Cl C1(C(=O)NC2CCOC(CO)C2)(NC(CC(=O)NCC(F)(F)F)=O)CC(F)(F)C1 c1(CN2CC3C(C(N4CC(F)(F)C(F)(F)C4)=O)(C3)C2)c(Cl)cc(F)cc1Cl C1(NC(=O)CN2C(=O)CCCC2=O)CN(C(c2ccoc2)=O)CC2CCCC12 [N-]=[N+]=NCCCC(=O)N1CCC(NC(c2ccc(-n3cncn3)cn2)=O)C1 n1(CC(=O)NC2(CF)CCN(c3nnc(C(C)C)o3)C2)c(=O)oc2ccccc12 Cn1cnc(CC(O)C(=O)NCCCCCNC(=O)C=CSCc2ccco2)c1 CC(c1ccsc1)=CC(N1CCOC(CCCNC(c2cc(C)cs2)=O)C1)=O N1(c2nnc(CC)s2)CCC(C2CCCN(C(=O)CN(C)C(N)=O)C2)C1 N1(CC)CCCC(CC(N2CCC(NC(=O)CCc3ccc(C4CC4)[nH]3)C2)=O)C1 N1(C(C2CC(C)(O)C2)=O)CCCCCCC1C(=O)Nc1cccc(O)c1 C1(F)(C(=O)NCC2CCC(=O)N2)CCCN(C(c2cccc(F)c2O)=O)C1 C1(C2CC2)(C(N(C)CCNC(=O)CN(c2cnccn2)C)=O)CCOCC1 C(=O)(CCC(O)C(C)(C)C)NC(C)CC1CN(C(=O)Cc2nncn2C)C1 Cc1cc(C)c(CC(N2CCC(CN(C)C(C3CCSC3)=O)CC2)=O)c(O)n1 N1(C(C2CC=CCO2)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc(O)cc1 c1(C(=O)NC2C(C)CCN(C(=O)C(F)(F)C(F)F)C2)cccc2ccnn12 C1(C(N2C(C(C)NC(=O)C(C#N)=CC3CC3)CCC2)=O)COC(=O)N1C Cc1cc(I)ccc1C(N1CCN(Cc2cnn(C(C)C)c2)C2CC12)=O c1(C(Cc2ccccc2OC)N(CCCCCC)C)cc(Cl)cnc1OC CCCCC(CC)C(=O)NCC(CC1CCCC1)C(=O)NC1CCN(CC)CC1 c1(OC)ccc2c(c1)nc(CNC1CC3CCC1C3)n2C c1(NCC2(CNC(=O)CC(O)C3CC3)CC2)cc2nn[nH]c2cc1[N+](=O)[O-] C1(C(=O)NC(CNC(c2cnc(S)[nH]2)=O)C2CC2)CCS(=O)(=O)C12CCC2 c1(OC)ccc2c(c1)C(C(=O)NCCC1CC(NC(C3(OC)CC3)=O)C1)CC2 C(=O)(CC1CS(=O)(=O)c2ccccc21)NC(CC(C)NC(CCSC)=O)C c1(C(=O)NCC2C(NC(C(C)OCC#C)=O)CCC2)cccc2sncc12 n1(CCC)cc(C(=O)N(CC(C)CNC(C2CCN2C(C)(C)C)=O)C)cn1 c1(C(=O)NCCC2CCCN(C(C3CNC(=O)N3)=O)C2)nccc2c[nH]nc12 c1(N2CCC(C)C(NC(=O)CCc3nccn3C)C2)ccnc2ncnn12 N1(C(c2cnc(-c3ccco3)s2)C(=O)NCCCOC)CCCCC(C)C1 N1(C(C2(CC)CCCCC2)=O)CC2CCC(C1CO)N2C(c1cccnc1)=O CCCCC(C(=O)NCC1(F)CCOC1)NC(c1scnc1Cl)=O C1(NC(CC(C=C)C)=O)C2CC(CN(C(=O)CCOC3CCCC3)C2)C1CO N1(c2c(C)ccnc2)CCN(N(C)Cc2cccc(C#N)c2)CC1 C(CCC(N1CC2CC1CO2)=O)(C(F)F)NC(=O)OC(C)(C)C C(=O)(CC(C(C)(C)C)NC(C1CC(C)C1)=O)NCC(CC)(C)Cl C1(C(N2C(CNC(C3(C)CSC3)=O)CCC2)=O)CCC2(CCC2)C1 C1(CNC(C2(CC=C)CC2)=O)CCCCN(C(=O)COCCF)C1 c1(CC(=O)NC2(COCC)CCCC2)ccc(OC)nc1.C12CCCC1C(=O)N2 c1(C(N2CCCN(C(c3cnc(Cl)s3)=O)CC2)=O)nccc2c1NCCC2 c1(C(=O)OC)ccccc1C(=O)NC(C)CCNC(c1ccc(CCF)cc1)=O c1(C(N(C(CN(C(C2CCC(C)O2)=O)C)C)C)=O)ccn2ncnc2c1 Cc1cc(O)ncc1C(=O)NC12CCN(C(c3ccoc3Br)=O)CC1C2 N1(C(c2c(CNC(C(C)(O)C3CC3)=O)n[nH]c2)=O)CCCC(C#N)C1 Cc1cc(Br)ccc1C(=O)NC(C1CCN(C(C2(C#N)CCCC2)=O)C1)C C1(CNC(Cc2cc(C)sc2)=O)CCCN(C(c2c(Cl)nn(C)c2C)=O)CC1 N1(C(Cc2c(C)ccs2)=O)CCCCC(NC(=O)C(C)NS(C)(=O)=O)CC1 C(=O)(C(COC)CC(C)C)NCC(CCSC)O.C12(CCC1)C(=O)N2 N1(C(Cc2cnc(C)[nH]2)=O)CCC2(CCCN2C(c2n[nH]c3ccccc23)=O)C1 CC1CCCC(C(=O)NC(C)CN2CCN(C(=O)CC3CCSCC3)CC2)CC1 C12(NC=O)CCC(C(=O)NCCOC)(CC1)C2.Cc1sncc1C(C1CC1)=O C1(C(N(C(C)CNC(=O)C(C)COc2ccccc2)CC)=O)CC12CCOCC2 C1(NC(CCOCCN(C)C)=O)CC2CC(NC(c3cc(Br)cn3C)=O)C2C1 C(=O)(C(CC1CCOC1)N(C(=O)OC(C)(C)C)Cc1ccccc1)NCCCC CC(CCC(=O)NCC1(O)CN(C(=O)CC2CC3CC3C2)C1)N(C)C c1(OCC(=O)NC2(C)CN(C(=O)Cc3ccc(Cl)s3)C2)ccc(Br)cn1 CCCC(CCCO)C(=O)N1CC(NC(=O)C(C)=C2CC2)C(C)C1 c1(C2(C(N3CC(NC(CC4C(C)C4)=O)C3)=O)CC2)ccc2ccncc2c1 N1(C(C(C(C)(C)C)O)=O)CCC2(CC1)CC(NC(c1cc[nH]n1)=O)CCO2 CC1(NC(=O)CC2CCCCN(C(c3cc(C4CC4)on3)=O)C2)CCCCCC1 c1(NC(C2CCCC(NC(CCNC(C)=O)=O)C2)=O)cccc(F)c1Br Cc1c(F)c(F)c(CNC(C2CNCC3(CCC3)C2)=O)c(F)c1F CCC(C)(C)C(O)C(=O)NCC(c1ccc(C)cc1)NC(C1CC1(Cl)Cl)=O CC1(C)CCC(CC(=O)NCC(C2CCN(C(=O)CCC3CC3)CC2)O)O1 c1(NCCCC)nc(N(C)CC2(CO)CC2)nc2ncn(C)c12 CC1(C)CN(C(c2ccncc2Cl)=O)C(CNC(C2CC2(C)C(F)F)=O)CO1 C(=O)(C1CCCc2scnc21)NCC1(C)CCCN(C(=O)CCOCC(F)F)C1 C(=O)(C(O)CC(F)(F)F)N1CC2(CC(NC(c3cc(Cl)ccc3F)=O)C2)C1 CCC1=NOC(C(N2CCC(C)C2CNC(c2ccc(C)cc2)=O)=O)C1 C1(CNC(CN(C(c2n(CCC)ccc2)=O)C2CC2)=O)(CO)CC2CCCC12 C1(NC(C2(NC(C)=O)CCCCC2)=O)CC2CN(C(=O)C(C)CC(F)(F)F)CC2C1 c1(NC(C)=O)ccc(C)c(C(=O)NC2CN(C(=O)C=CC3CC3)CC2C(F)F)c1 CON1CCC(C(=O)NC(CCN(C(=O)CC2=CCCC2)C)C(C)C)CC1 CC1CCN(C(C2CC(=O)C23CCC3)=O)CC1CC(=O)NC1CC2C=CC1C2 C1(C(=O)NC2C(NC(C(CC(C)C)(F)F)=O)CCC2)CCc2cc(F)ccc2O1 N1(C(C(C)SCC)=O)CCN(C(=O)C=CSCc2ccco2)CC1C1CC1 Cc1nc(C(=O)NCC2CC2CNC(c2cccn2C(C)C)=O)ccc1[N+](=O)[O-] CC1=C(C(=O)NC23CC2CS(=O)(=O)C3)CCS1(=O)=O N1(C(C(C#C)(C)C)=O)CCC2(CCCN(C(=O)C(C)Sc3ncccn3)C2)CC1 C1(CCC)(NC(=O)C(C)COC)CCCN(C(=O)CCCc2n[nH]c(=N)s2)C1 c1(OC)cc(C(=O)NC2CN(C(=O)CN3CCC3C)CC2(F)F)cc(F)c1 CC(C)CC(C)C(=O)NCCCCC1CCN(C(=O)CCCC#N)CC1 c1(OC)cnccc1C(N1CCSCC1C(=O)NC(C)C(C)(C)O)=O CC1=CCC(C(=O)NCC2(CCNC(=O)Cc3ccc(C)s3)CC2)CC1 C1(CN(C)C(c2cc(C(C)(C)C)ccn2)=O)COCCN1C(=O)C=CC=C(Cl)Cl Nc1ccc(F)c(C(=O)NC2CCC2NC(=O)C=CC2CCCO2)c1 C1(C(=O)NC2CC(C)(NC(c3cccc(Cl)c3)=O)C2)CCc2ccccc2C1 N1(C(COCC(C)C)=O)CCC(NC(c2cc(Cl)cc(Cl)n2)=O)C(O)C1 C1(C#CC(=O)N2CC(NC(=O)C(C)COC)C2)(CC)CC1 n1(CCOCC)nnc2c1CCN(Cc1nc[nH]n1)C2 CC1C(=O)NCCCN1C(=O)NCCN1CCN(c2ccccc2)CC1 c1(CN(C(=O)C(O)COC2CCOCC2)CCOC)ccncc1Cl c1ncnc(C)c1C.C1(c2cn(CCOCCO)nn2)CCCN(CC)C1 c1(C(C)NC(CCOC2CN(C(CC3(OC)CC3)=O)C2)=O)nnc(C)o1 N1(C(C(CC)C#N)=O)CC(CNC(c2sccc2SC)=O)CC12CCC2 NC(Cc1ncccn1)C(=O)Nc1cnoc1CC(=O)O C1(CNC(C)=O)CCCN(C(C)C(=O)NCC(c2ccc(Cl)cc2)C)C1 CC(CC(C)NC(c1ncnn1C1CCOCC1)=O)NC(=O)C=Cc1ccoc1 Cc1scnc1C(=O)NC1(C(=O)NCCN(C)CCOCF)CCC1 C1(CNC(CC)=O)CN(C)CCN1C(c1cc(OC(F)F)cc(Br)c1)=O N#Cc1cnccc1CNC12CC(C(=O)Nc3c(Br)ccnc3Br)(C1)C2 N1(C(C(CC)NC(C)=O)=O)CCOC(C2(NC(=O)C(CCOC)OC)CC2)C1 Cc1cc(Cl)cc(C(=O)NCC2CCN(C(=O)COc3ccccc3Cl)C2)c1O C(=O)(N=c1[nH]nc(Cl)cc1Br)C1(C)CN(C(c2cc(C)oc2C)=O)C1 S(=O)(=O)(c1ccc(C#N)cc1Cl)Nc1cccc(-c2nc(C)c(Br)s2)c1 C12(C(=O)NC(c3cn(-c4c(F)cccc4Cl)nn3)CCC)CCCCN1CCC2 c1(C(=O)NCC(c2cccc(F)c2)(C)C)ccccc1C1CC1(F)F c1(CNC(C2(C)CCC2)=O)ccccc1-n1cc(C2COC(C)(C)C2)nn1 C1(NC(Cn2c(=O)ccc(C)c2)=O)CC2(CCN(C(C3CCOC3(C)C)=O)C2)C1 c1(CC(N2CC(NC(C3CC(C)(O)C3)=O)CC(C)C2)=O)ccc(F)cc1[N+](=O)[O-] C(=O)(C(C)CCO)NC(CCNC(COCC)=O)Cc1ccccc1 Cn1cc(C(N2CC(Nc3cc(F)ncn3)C(O)C2)=O)c(C2CC2)n1 C(=O)(CCC(C)(F)F)NCC1CCC(NC(CCc2nnc(C(C)C)o2)=O)C1 CCC(C)(COC)C(=O)NC1CCC(C(=O)N(CC(C)(C)CN(C)C)C)C1 N1(C(C#C)C)CCCN(C(=O)NCC2(CCOC)CCCC2)CC1 c1(C(=O)NCCCC(C)NC(c2cnc(C)o2)=O)cc(C)c2nc(C)cn2c1 C1(C(=O)NCC2(O)CN(C(CCc3nc(C)sc3)=O)C2)CCC(O)CC1 c1(C(=O)NCC=CCNC(c2cncc3nc[nH]c23)=O)occ2c1CCCC2 c1(C(N2CCC(C)C2Cc2ccccc2)=O)ccc2nc(S)[nH]c2c1 c1(NC(C2N(CC)CCC2)=O)cnc(F)cc1C(N1CCN(C)CC1CCO)=O C(CNC(=O)C(c1ccccc1Cl)O)(CC(F)(F)F)NC(=O)Cc1ccsc1 CCC(C)(C(=O)NCCCN(C(=O)C(C)(C)CF)CCO)C(N)=O C=CC1(CC(=O)N(CC(C)COC)C)CN(C(c2n[nH]c(C)c2Cl)=O)C1 Cc1ccc(C(N2CCN(CC(C)NC(C3CCCO3)=O)CC2)=O)c(C2CC2)c1 C(CC)(CC(=O)NCc1cc(C(=O)OC)co1)N(C(CSCC#C)=O)C N1(C(CC)=O)CC(C(F)(F)F)CC1CNC(=O)CC(O)c1ccccc1 c1(NCCN(CCOC)C)[nH]c(=NCc2scnc2C)nc2c1cnn2C(C)C C1(CC(N2C(CC)(CC)CC2)=O)CN(C(C2CCCOC2)=O)CC12CC2 N1(C(C(C2CCN(C(c3c(C)ccnc3)=O)CC2)C)=O)CC2CCC1(CO)C2 C1(CNC(c2c(CNC(=O)CC3CC=CCC3)cco2)=O)CC1C1CCC1 N1(C(C(CC)NC(C)=O)=O)CCC(N(C(c2ccccc2F)=O)CC2CC2)CC1 c1(CNC(C(N2C(C(N)=O)CC(O)C2)=O)=O)cc(F)ccc1F Cc1c(Br)ccc2c1CCC2NCCc1ccc(F)c(C(F)(F)F)c1 N1(C(CCC(C)OC)=O)CC(C2CCCCN(C(C3(C)CCCC3C)=O)C2)C1 N1(C(C(C)n2ccnn2)=O)CCN(C(=O)CC2(CO)CC2)C2CCCCC2C1 c1(C(=O)NC2CN(C(Cc3ccc(C)nc3)=O)CC2C)cnc2c[nH]nc2c1 c1(CC)ncnc(CC)c1C(=O)NCCC1(NC(=O)CC2COC(C)(C)C2)CC1 C1(C(F)F)(OC)CCCN(C(=O)CCc2ccc(Br)c(F)c2)C1 C(CN=c1ccc(C#N)c(C)[nH]1)C1C(NC(Cc2scc(C)c2)=O)CCCC1 c12ccccc1[nH]c(=O)[nH]2.N1(CC)C(C(=O)NC2CCS(=O)(=O)C2)CC2CC12 C1(NC(C(Cc2ccsc2)NC=O)=O)CC2(CCN(C(C3(F)CC3)=O)CC2)C1 C#CC(C)(C)C(=O)NC1CCC(C)(CNC(=O)C=CBr)C1 c1(NC(C2(CNC(c3cccc(C(F)(F)F)c3)=O)CC2)=O)nc(F)ccc1Br NS(=O)(=O)c1ccc(C(=O)NC2CC2CNC(C2CC2C(F)(F)F)=O)c(F)c1 c1(C(N2C3C(c4cn(CCOCC)nn4)C(C3)C2)=O)c(O)ccc(OC)c1F.C=O Cc1nc2c(C(=O)NC3C4CC3N(C(c3cc(C)sn3)=O)C4)ccnc2[nH]1 Cc1ccc(SCC(N2CCCCC2CNC(=O)CC2CCC23CCC3)=O)cc1 N1(C(C2OCCC(C)C2)=O)CC(NC(=O)C(C)n2cccn2)CC2(CCC2)C1 c1(C(=O)NCC(CC)(C)NC(=O)C(C)C(F)F)c(C)noc1C Cc1ccc(OCCN(C)CC2CCN(C(c3nc(C)c(Br)s3)=O)C2)cc1 CCCCCC(C)(C)C(=O)NC1CC2CC(C1)N(C(=O)CCSCC(N)=O)C2 C12(C(N3CCCC(COC)C3)=O)CCCC1CCN2C(C1SCCCS1)=O CC(CNC(C1CCN(C)CC1)=O)CC(=O)NCC1CC[Si](C)(C)C1 Cc1coc(C)c1C=CC(N1CC2CC(NC(C3CCC34CCC4)=O)C1C2)=O N1(C(C2C(CC(C)(C)C)C2)=O)CCC(NC(=O)CCC2CCOCC2)C12CC2 c1(C(=O)NC2(C(C)C)CCC2)cccnc1CNC(=O)C(F)CC1CCOC1 C(CCCCCNC(=O)Cc1nccnc1C)n1cc(-c2cnc(NC)s2)nn1 Cc1nc2ncc(C(=O)N(C3CN(C(=O)CCC=CC(C)C)C3)C)c(=O)n2[nH]1 N1(C(c2ccc(OC)nc2Br)=O)CCCC2C1CCN2C(c1ccnc(O)c1)=O C(CCCCC(=O)N1CCCC(F)(C(=O)Nc2ccccc2)C1)NC(N)=O Cn1c(C(=O)N(C2CC(C#N)C2)CC(=O)N)cccc1=O.N1(CCF)CC(C#N)C1 C(CCCCC(=O)N1CCC(F)(F)CC1)NC(c1c(CCC)[nH]cc1)=O C=C(Cl)CC(C(=O)NCC(C)C1CCC1)NC(=O)C(F)OC(F)(F)F Cc1c(NC(C)C)cccc1C(N1CCOC(CNC(c2cncs2)=O)C1)=O c1(CN=c2cc(-c3c(OC)cccc3)[nH]cc2)cc(O)n2nccc2n1 c1(Cc2cn(CC(CNC(COCC)=O)(C)C)nn2)ccc(C(=O)NC)cn1 N1(C(c2ncc[nH]c2=O)=O)CCC(N=c2[nH]c3ncc(Cl)cc3s2)C1 C1(C(=O)OCC)CN(C(C2CC3CCC2C3)C(=O)NC(C)C(=O)OCC)CCO1 N1(C(C(CC#C)(C)C)=O)CCC2(CC1)CN(C(c1cc(S(N)(=O)=O)cs1)=O)C2 c1(C(=O)NC2C(C)CN(C(c3cccnc3C3CC3)=O)C2)cnn2ccncc12 CS(=O)(=O)c1ccc(OCC(=O)NCCNC(=O)C=CCF)cc1 N1(C(c2cc(C)c(Br)s2)=O)CCC(F)(CNC(C2CCOC2)=O)CC1 C1(C(=O)NCC2(C(=O)NCC3(C(=O)OC)CC3)CC2)C(C(F)F)C1(C)C.COC Cc1ccc(CNC(=O)CC2CN(C(c3cn(CCO)nn3)=O)CCO2)nc1 C1(CNC(c2c(OC)cccn2)=O)(NC(=O)CSCC(C)C)CC2CCC1C2 N1(C(C2CCC3CCCCN23)=O)CCCC2(CCN(C(=O)C(O)C3CC3)CC2)C1 N1(Cc2ccc(CNC(C)=O)cc2)CCC2OC(=O)OC2C1 C(CC(CC)C(=O)Nc1cccc(CCF)c1)=CC.N12CCCCC1CCC2=O N1(C(C(CCCC)NC(c2ccnn2COC)=O)=O)CCn2nc(C)cc2C1 N1(C(C2CCC(CC)O2)=O)CCC(C)(C)C(C(=O)NC2CC(C)(O)C2)C1 N#Cc1ccnc(N2CC=C(CCNC(=O)CCn3cccn3)CC2)c1[N+](=O)[O-] N1(C(C(CSC)O)=O)CCc2nc(CNC(C3CC4CCC(C3)S4)=O)sc2C1 c1(C(N2CCCC(NC(C(C(C)C)SCC)=O)C2)=O)ccc2sccc2c1O C(=O)(CCCCN=[N+]=[N-])NCC1CCC(C(=O)NC2CCN(C)C2)O1 c1(C(=O)NC2COC3(C2)CN(C(C2CC(F)C2)=O)C3)ccc2ccc(O)nc2n1 C1(NC(C(C)(F)F)=O)CN(C(=O)Cc2cccc3nsnc23)CC2(CC2)C1 c1(OC)cc(OC)c(OC)cc1C(=O)NCC1CCN1Cc1ncn(C)n1 c1(OC)cc(C)cc(C(N2CC3(CCCC3NC(=O)C3=COCC3)C2)=O)c1O S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NC(c1cc(Cl)cc(Br)c1)CC(=O)O O(C1CCc2c(Cl)ccnc21)C(C1(Cl)C(C(=O)O)C1)=O C12(NC(c3cnc(CN(C(C4CC=CCC4)=O)C4CC4)nc3)=O)CCN(CC1)CC2 C(CCCCCC1CC1)NC(=O)CCCn1cc(C2CC=CCC2)nn1 C(=O)(C(C)(C(F)F)N)NCc1ccccc1.Cc1n[nH]c(C)c1NN1CCC(C)C1C N1(C(c2ncc(N)nc2)=O)CC(NC(=O)CC2(O)CCC2)CC12CCC2 Cc1cc(=NCCP(C)(C)=O)[nH]c(N2CC3CC(C)(C)C3C2)n1 c1(NC(N2CCC(CCC)C2)=O)ccc(F)cc1OCc1cccc(C)c1 CCCC(O)C(=O)N1CCOCC1CC(=O)NCc1ccoc1C(N)=O c1(C(=O)NC2CCC(NC(c3ccc(Cl)nc3O)=O)C2)cnc2c(c1)CCCO2 Cc1ccc2c(C(=O)NC3CN(C(C4CCOCC4)=O)CC(F)(F)C3)csc2c1 N#Cc1ccc(-c2cn(CCC3CCN(C(=O)CCCCCF)CC3)nn2)cn1 Cc1ccc(C(=O)NC(C)CCNC(=O)Cc2ccccc2CC(N)=O)c(O)n1 N1(CC)CC(NC(C2(CNC(C3C=CCC3)=O)CC=CC2)=O)CCC1=O C(=O)(C(F)(F)C(F)(F)F)NC1C(SC)CN(C(=O)COc2ccc(C)cc2)C1 C(CC(C(=O)NC1CC(C(F)F)(OC)C1)NC(c1cccc(O)n1)=O)OCC Cc1cccc2c1CN(C(=O)CC(CNC(=O)C=Cc1ccc[nH]1)C1CCC1)C2 C1(NC(C(c2cccs2)NC(CCNC(COC)=O)=O)=O)CCOC2(CCC2)C1 c1(C(N2CC(C(C)NC(C3(C(=O)OC)CCC3)=O)C2)=O)cc(CC2CC2)c(C)s1 c1(C(C)NC2CN(CC(F)(F)F)C2)nc2c(s1)CN(C)CC2 c1(CCC)nnc(S)n1CC(=O)NCC(C)NC(C12CCC(CO1)C2)=O c1(C(N(C(C)CN(C(=O)CSC(F)(F)F)C)C)=O)cc(F)cc2nc[nH]c12 C1(C(N2CC(C)(C)C2)=O)COC2CN(C(c3cc4ncsc4[nH]3)=O)CC12 CC1(CCC(=O)NCc2ccncn2)CN(C(c2ccsn2)=O)C1 C1(CNC(C(C)(C)OCC)=O)CC2(CC(NC(=O)CN3CC4CC4C3)C2)C1 Cc1cccc2nc(C(=O)NCCC(C)N(C)C(c3cc([N+](=O)[O-])c[nH]3)=O)cn12 c1(C2(O)CC(C(=O)NC(C)CNC(C3COC(=O)O3)=O)C2)ccccc1Cl c1(C(=O)NC2CC3C(NC(Cn4ncc(CC)c4)=O)C3C2)cc(C)c(O)nn1 c1(C(=O)O)cc(OC(F)(F)F)cc(NC(C2CCCC2c2ccc(F)cc2)=O)c1 Cc1c(C(=O)NC(C)CCCCNC(=O)CN(C)C2CC2)nnn1C1CCOC1 C1(C(=O)NCC(C)NC(C2(SC)CCC2)=O)Cc2nnsc2S1 C(C)(C)(CC(=O)NC1CC(N2CCCC2)C1)N(C(C(=O)OC)=O)C Cc1cncc(C(=O)NC2CCC(N(C)C(c3cc(Br)co3)=O)CC2)n1 N1(C(c2c(OC)n(C)nc2)=O)CCC2CC(C1)CN(C(=O)CC1CCCC1)C2 c1(C(N2CCCC(N(C(=O)Cc3cnccc3Cl)C)C2)=O)cnc2scnc2c1 C1(NC(C2CC(NC(c3c(OCC)nccc3)=O)C2)=O)CC2CCCCCC12 CC1(C(N2CCCC2CNC(c2c(Cl)ccc(F)c2F)=O)=O)CCC(F)(F)CC1 N1(C(c2c(C)sc(C)c2C#N)=O)CCCC12CCN(C(c1cscc1Cl)=O)CC2 C(CN=c1[nH]cnc(C)c1Br)NC(C1(CCC)CC1)=O C1(C(=O)NCCC(=O)NC(C)COC(F)(F)F)CCCCCCC1 N1(C(CCCC(N)=O)=O)CC2CS(=O)(=O)CC2(NC(c2[nH]ncc2C#N)=O)C1 C=CC1(CC(=O)NC2CCN(C(c3nccn3C)=O)CC2F)CCOCC1 Cc1cc(C(N2CC(C)CN(C(c3cccs3)=O)CC2C)=O)cc2nc[nH]c12 N(C(=NCCF)NCC(=C)C)C1C(C=C)OCC1 C(=O)(C(C)CC(F)(F)F)N1CC(C(=O)NCCCc2ncn(C)n2)(SC)C1 O=NN1CCCCC1C(=O)NCCN(C1CCCC1)C(=O)CC1C=CCCC1 C1(CCNC(CCC=C)=O)CN(C(=O)Cc2ccc(OC)cc2)CC(C)O1 N1(C(c2c(C)cns2)=O)CCC(C2CCN(C(=O)CC3CCC(=O)N3)CC2)CC1 C1(NC(=O)NCn2ccc(C)n2)CC2CN(c3nc(C4CCC4)cn3C)CC2C1 C12(NC(C3(C(C)C)CCC3)=O)CCC(NCc3sc(Br)nc3Br)(CC1)C2 C(=O)(C(C)(F)CC1CC1)NC(C)CNC(=O)COc1ccc(F)cn1 c1(C(N2CCC(NC(C3(CC)CC3)=O)CC2C)=O)cc2ccc(Br)cn2n1 N1(C(c2cc(C(C)C)no2)=O)CC(F)(F)CC1CNC(=O)CNC(=O)CN(C)C C1(OCc2cc(C(N3CCCC3CO)=O)n[nH]2)CCS(=O)(=O)NC1 C1(CC)(Nc2cc(C3CC3)nc(Cl)n2)CCN(C(=O)CC2C=CCC2)CC1 Cc1ccc2c(O)c(C(N3CC4CC(C)N(C(=O)C(C)(F)F)C4C3)=O)cnc2n1 C1(C(N(CCN(C(=O)C2=CCCOC2)CC)CC)=O)C(C)(C)CCCC1(C)C C12(NC(C(CC3CCC3)NC(c3ccnnc3O)=O)=O)CCC(O)(CC1)CC2 Cc1ccc(C(N2CCCCC2CNC(c2nc(Br)c(C)s2)=O)=O)c(O)c1 N1(C(COCC#C)=O)CCOC2(CCN(C(=O)CNC(=O)OC)CC2)C1 C1(NC(C(=O)NC(c2ccc(N3CCCC3)cc2)C)=O)CC2(C1)OCCO2 C1(C(=O)OC)CC2CC1CC2NC(C(=O)O)C1(C)CC1 c1(C(N2CC(=O)NCC2C(N2CCSC3(CCC3)C2)=O)=O)ccc2n[nH]cc2c1 N1(C(C(C)(C)C2CCOC2)=O)CC(C(=O)NCc2ccon2)C(C2CC2)C1 C1(CCNC(C2CCCCO2)=O)(NC(C(C=C)O)=O)CCOCC1 N1(C(CC2CCCC(OC)C2)=O)C2CCC1CN(C(C1CC3(CC3)C1)=O)C2 C1(NC(CCc2cccc(OC)n2)=O)CC2CCCC(C1)N2C C1(O)(C(C)NC(C2(c3ccncc3)CC2)=O)CCN(C(=O)CC(C)F)C1 c1(OC)ccc(Cl)c(C(=O)NCC(c2cccc(C)c2)NC(=O)C2=CCC2)n1 CCC(C)CC(=O)C(=O)NCC(C)(CC)C(=O)N1CCC(C(F)(F)F)C1 C1(CN(C(C(CN(CC)CC)F)=O)C)CN(C(=O)CCSC)CCO1 CC1CCN(c2nnc(-c3ccccc3)o2)CC12CCC2 N1(C(C)=O)CCCCC1C(=O)NCCC(O)CNC(c1n[nH]cc1C1CCC1)=O C12(C(=O)NCCn3cc(CNC(c4nc(O)n[nH]4)=O)nn3)CC=CCN1CCC2 Cc1cc(C)cc(C=CC(N2CCN(C(=O)CCc3ccccc3)CC2C)=O)c1 CC1CCC(NC(C2CC(=O)C23CCC3)=O)CN1.C1(CCN)CCCCCC1 N1(C(c2cncc(C(C)=O)c2)=O)CCCC(NC(C2(N(C)C)CCC2)=O)CC1 C(=O)(C(C(C)C)C1CCC1)N1C(C(=O)NC(C2CCCCC2)CC)(CC)CCC1 c1(C(=O)NC2CN(C(c3cc(Br)c[nH]3)=O)CC2F)cc(Br)ccc1I C1(C(=O)NC23CC(NC(C(C)c4ccsn4)=O)(C2)C3)CC2(CCCCC2)S1(=O)=O n1(CC(=O)NC(C2CCO2)C)ccc(C2CC2)n1 CCCC(CC)CC(=O)NC1CC2CCC(C1)N2C(C1(O)CC(C)(C)C1)=O c1(CC(=O)NCC(CC)NC(C2CCCN(CC(F)F)C2)=O)ccc(OC)cc1 C1(C(=O)N)CC(F)(F)CN1C(c1cc[nH]n1)=O.C(CCCCN(C)C)OC c1(C(=O)NC2CC(C)N(C(=O)C3=CCCCO3)C2)cccc2occ(Br)c12 c1(C(N(C)CC2N(C(CCOC)=O)CCCC2)=O)c(O)cnc2cc(F)ccc12 c1(OC)cc(C(=O)NCC=CCNC(c2cc(Cl)c(F)cc2N)=O)cc(F)c1F c1(C(c2n(CC)nnn2)NC2CCOC2)ccc2c(c1)C(=O)OC2 CC1OC2(CNC(=O)C=CBr)CC1(NC(C1OCCC1C(F)(F)F)=O)C2 C1(CC=C)CCCN(C(=O)C(CN(C)C)NC(=O)CC(CC)OC)C1 N1(C(C(=O)N(C)C)=O)CCC(CCNC(C2CCC(O)CN2C)=O)C(F)(F)C1 c1(C(=O)NCC2C(NC(c3cc4c[nH]nc4s3)=O)CCC2)cccc2sccc12 C12(C(=O)NC3C(CNC(c4c(OC)c(Cl)sc4)=O)CCCC3)CCC(C)(C1)OC2 C1(CC(=O)NC(CC)C(C)O)Cc2ccccc2CN1Cc1ncc(Br)cc1Br Cc1ncc(Br)c(C(=O)NCC2CCN(C(=O)CCP(C)(C)=O)C2)n1 c1(C(N(C2CCN(C(=O)COC3CCSC3)C2)C)=O)cnn(C2CCOCC2)c1 N1(C(c2cc(C)c(F)cc2)=O)CCC(F)(F)C(C(=O)NC2CCCN(C)C2)C1 C(=O)(C1=CC2CCCCC12)NC(C1CCCC1)CNC(c1c(C)nc(CC)o1)=O S(=O)(=O)(c1ccc(C(=O)NC(C)(C)CCNC(=O)CSc2nncs2)cn1)NC c1(C(=O)NC2C(CNC(Cc3nc(COC)sc3)=O)CC2)ccn2nnnc2c1 CN1c2ccccc2CC1C(=O)NCC12CC(CN1C(C1CCN1C(C)(C)C)=O)C2 c1(C(N(C2CCN(C(C3CCCC(=O)N3C)=O)C2)CC)=O)ccc(F)c(C)c1 c1(C(=O)NCC2N(C(c3cc(OCC)no3)=O)CC2)ccc2c(c1)OCC2 Cc1ccnn1CC(=O)NC(Cn1ccnn1)C(=O)NCCNC(N)=O C(c1ccccc1C)=CC(N1C(CNCc2c(N(C)C)cccc2)CCCC1)=O N1(C(C2C(CC)CCO2)=O)C2CCCC1CN(C(c1csc3cncn13)=O)C2 C(=O)(C1=CC(O)CCC1)N1C(CCCNC(C=C(C)c2cccs2)=O)CCCC1 CC(C)(F)CCC(=O)N1CC(CNC(=O)Cc2cccc(C#N)c2)C2(CC2)C1 N1(C(CN(C(C(=O)N(C(CC(C)C)C)C)=O)C)(C)C)CCC(N(C)C)CC1 CCCC(C)N=c1[nH]c(=NCCCN2CCCC(CO)C2)[nH]c2cccnc12 C1(C(N(C2C(N(C(CNC(=O)NC)=O)C)CCCC2)C)=O)CCC2(CCC2)C1 N1(C(CC(C(C)C)O)=O)CC2CCC1CN2C(c1cc(C(F)(F)F)cc(O)n1)=O N1(C(Cc2scc(C)n2)=O)CCCCC1C(C)NC(=O)CCSc1nnnn1C c1(C(=O)NCC2(NC(c3nc(OC)oc3)=O)CCCC2)cc(F)cc(Cl)c1O C1(CNC(c2cc(CCC)nn2C)=O)CN(C(=O)C#CC(C)(C)C)CCCO1 c1(N(C)C)ccc(CN2CCCC(CNC(=O)C(c3ccccc3)O)C2)cc1 c1(CC(=O)NCCC(C)NC(C(COCC)C)=O)cccc(C)c1Br C1(NC(CCSC)=O)C=CCN(C(=O)CCCN2C(=O)CCC2=O)C1 n1(CC)nc(C(N2CCC(C3CCCN3C(=O)Cc3csnn3)C2)=O)cc1O N1(CC(N2C(C)(CNC(c3csc(Cl)c3Cl)=O)CCC2)=O)CCS(=O)(=O)CC1 c1(CC(N2CC3C(NC(CCC)=O)(C3)C2)=O)ccc(S(=O)(=O)NS(C)(=O)=O)s1 C1(NC(=O)Nc2ccc(-n3cccn3)cc2)CS(=O)(=O)C12CCCC2 CCC(O)C(C)C(=O)N1CCC(C)(CNC(=O)C(C)Cc2ccc(F)c(F)c2)C1 C1(CNC(c2cc(Cl)c(F)c(Cl)c2)=O)CN(C(c2cccnc2)=O)C2(CCC2)C1 C12(CNC(c3c(CC)onc3C)=O)CCC1CCN2C(c1cc(C)ncn1)=O Cc1ccc(C2(NC(=O)NC(C(=O)OC(C)(C)C)Cn3cccn3)CC2)cc1C C12(C(=O)NC3CN(C(c4nc(C)oc4C)=O)CC3O)CC(CC(C)O1)C2 c1(C(N(CC(C)NC(C(COC)OC)=O)C)=O)cnc(-c2nn[nH]n2)c(C)c1 C(=O)(C(C)(F)C(=O)NCc1cc(C)c(C(=O)NCC2CCCCO2)o1)OC c1(C(N2CC(CCn3cc(C(CC)(C)O)nn3)C2)=O)nnn2c1COCC2 C(=O)(CCCCC(=O)NC)NCCC(C)NC(c1c(SCC)cccc1)=O N1(C(C(CC2CC2)OC)=O)CCC(C(=O)NC2(C(N)=O)CCCCC2)CC1(C)C C1(C2CCCN(C(c3cc(C)nc(C)n3)=O)C2)(NC(C(CC)(CC)CO)=O)CC1 C1(NC(C2C(OC)CC2)=O)CCC2CCN(C(c3ncoc3C3CCC3)=O)C1C2 N1(C(C(C2CCCC2)OC)=O)CCCN(C(c2cccc3c2NCC3)=O)C(C)C1 C(c1cnccn1)=CC(=O)NC1(CC=C)CN(C(C2CC(=O)C2(C)C)=O)C1 Cc1cc(C(=O)NCC(C)CNC(=O)C(C)NC(C2CCC2)=O)c2occc2c1 c1(NC)ccc(C(N2CC(NC(=O)C=C(C)c3ccsc3)C3CC23)=O)nc1 CCCC(C)CC(=O)NC1COCCC1NC(c1cccc(OC)c1C)=O c1(C(N2CC(COC)(NC(c3ccc(OC)cn3)=O)C2)=O)cccc(C)c1O Cc1ccc(-c2noc(C(C)Oc3ccc(Cl)cc3)n2)c2ncccc12 N1(C(C2(C(=O)OC)COC2)=O)CC2CC(C1)N(c1ncnc(=N)[nH]1)C2 C(=O)(C1=CCCCO1)N1CC(C(C(=O)NC(C=C)C(F)(F)F)OC)C1 c1(CC)ncc(Cl)c(C(=O)NC2CCN(C(c3cc(=N)[nH]c(=N)[nH]3)=O)CC2C)n1 N1(C(C=COCC)=O)CCCC2(C1)CN(C(=O)Nc1cc(C)ccc1C)CCO2 C1(NC(CC)CCc2ccccc2)CN(C)CCN(C)C1 C(C)(C)(C(C)CC(=O)NC1(C)CCCCC1)NC(COC)=O Cc1c(C(=O)NCC2COCC2NC(=O)C=Cc2cnc[nH]2)oc2ccccc12 C1(C(=O)NC23CC(NC(C(C)Oc4ccccc4)=O)(C2)C3)CCC12CCCO2 C12(C(=O)NCCCCN(C(c3ccc(CCC)s3)=O)C)CC1COC2(C)C C1(c2n(CCCCC)c(N(C)CC3CCCCC3)nn2)COc2ccccc2C1 N1(C(c2scc(C(C)=O)c2)=O)CC2CCC1CN2C(C12CCCC1C2(F)F)=O C=CCN=C(NCc1ccc(OCC(=O)NC)c(OC)c1)N1CCCC(C)(C)C1 C(C(=O)N1CC(CNC(c2cnn(C(C)C)c2Cl)=O)C(C)C1)(C(C)C)NC(C)=O C1(C(C)C)CCC(C(=O)N(C)CCN2CCCC2)C(=O)N1 Cn1cc(C(=O)NC2C3CC2N(C(=O)CC2CCCCC2)C3)cc1Br c1(C(C(=O)N(CC(C)NC(C2CC(C(F)(F)F)C2)=O)CC)O)cccnc1 N1(C(c2cncc(CNC(CN(CC)CC)=O)c2)=O)CC(N(C)OC)C1 C(=O)(CCS(=O)(=O)CC(C)C)NCC1(C)CCN(C(C(C)OCCCC)=O)C1 C(C(=O)Nn1nnc2c1CCCC2)N1CC(OC(C(NOC)=O)=O)C1.C(C)C N1(C(c2c(CC)n(C)cc2)=O)CC(N=[N+]=[N-])CC1C(N1CC(O)C(C)(C)C1)=O c1(OC)ccc(C(N2CCN(Cc3ccc(OC)nc3)C(C(C)C)C2)=O)c(Br)n1 c1(C(=O)NCC2C(C)(C)CN(C(=O)CCC3CC3)C2)cnc2c(F)cccn12 C(=O)(C(C(C)(C)C)NC(N)=O)NC(CC(C)NC(CSc1ccc(OC)cc1)=O)C Cn1cnc2nc(N3CCC(C4CCC4)CC3)[nH]c(=NC3C=CCC3)c12 CCCCCC(C)(C)C(=O)NC1CCC1C(=O)NCCC(=O)N(C)CC C(CCCCCCO)N(C(c1ccccc1F)CC)C(=O)COCC(F)F Cc1c(C(c2nnnn2C(C)C)Nc2ccnn2C)cccc1C(F)(F)F C(=O)(C(C)(C)CO)NCc1c(C(=O)NC(CC)Cn2cncn2)occ1 c1(NC(=O)NC2(CNc3ccnc(F)c3)COC2)cccc(I)c1 c1(CC(=O)NC(C2CC=CCC2)C(=O)NC2(CC)CC2)cnc(O)cc1C CC1CCC(C(=O)NCC23CC2CN(C(C2CCN(CC4CC4)CC2)=O)C3)CC1 N1(C(c2nc(C)on2)C)CCc2ccccc2C1CNC(c1ccsc1)=O c1(N(C)Cc2ccc(C(C)C)cc2)nc2ccccc2c(=NC(C)c2cnsc2)[nH]1 c1(N2CCN(C(Cn3c(C)cc(C)n3)=O)C3(C2)CC3)ncnc2ccc(F)cc12 c1(OC)c(Cl)cc(CNC2CC(NC(c3nc(Cl)cs3)=O)C2)cc1Cl CCC1=C(C(=O)NC2(C3CCN(C(=O)C(CO)OC)CC3)CC2)CCCO1 C1(S(N)(=O)=O)(C(N2CC(C)C(CNC(=O)C3=NNC(C(F)(F)F)C3)C2)=O)CCC1 c1(C(N2CC(C)CC(NC(C3=C(C)CCC3)=O)C2)=O)cn2nc(C)sc2n1 c1(CC)ccc(-c2nc(CCc3nc(C)no3)n(C(C)C(C)(C)C)n2)cc1 Cc1csc(CCCC(=O)NC(CNC(=O)Cc2cnccn2)C2CCC2)n1 N1(C(C(N2CCC(C)CC2)=O)=O)CCC=C(CNC(C2CC(O)C2)=O)C1 c1(C(=O)NCC(CNC(c2n(C=C)nnc2)=O)F)ccc(C)c(C)c1N N1(CCCC)CCCCC1NC(C1CC(F)(CNC(=O)C=C2CCC2)C1)=O c1(CC(=O)OC)cccc(C(=O)N(C)CC2CN(C(=O)CC3CSC3)CCO2)c1 c1(OC)cccc2c1CCC2(CO)NC(=O)NC1CCC(O)CC1 N1(C(C(C)SCCOC)=O)CC(NC(=O)C=Cc2ccc(OC)cn2)C(C)(C)C1 C(=O)(CC1OCc2cc(Cl)ccc21)N(CCN(C(C1(CC=C)CCOC1)=O)C)C n1(CCCC)nnnc1C(c1[nH]nnc1C)NCc1nncn1CC c1(OC)ccc2c(c1)OCC2CC(=O)NCCCNC(c1cc(C)ccc1N)=O C(C(C(=O)NCc1ccccc1)N(CCOC)C1CC1)(C1CCCCC1)OCC N1(C(CNC(C)=O)=O)CC2CC1CN(C(c1cn(C)cc1C)=O)C2 c1(NC(CSC)C)[nH]c(=NC2CC3C(C2)C3(F)F)nc2c1cnn2C c1(C(N2CCN(C(c3ccc(CC)[nH]3)=O)C(C)C2C)=O)nc2ncc(C)cn2n1 C(=O)(CCC(=O)NC(C)CCN(C)C(c1sccc1OC)=O)NC N1(C(CN(CC)CC)=O)C2CCC1C(CNC(=O)Cc1cnc(C)[nH]1)C2 Cc1nn(C(C)C)c(C)c1C(=O)NCC1CCCN1C(C1CCCNS1(=O)=O)=O c1(C(=O)NCC(C2CC2)NC(c2c(CCC)[nH]cc2)=O)c(C2CC2)noc1C c1(Sc2c(C(=O)NCCNC(CN(C)S(N)(=O)=O)=O)cccc2)ccc[n+]([O-])c1 c1(C(=O)NCC2(F)CC(NC(c3ccc(N)cc3O)=O)C2)ccn2ncccc12 c1(CNC(C2CC3CCCC3C2)=O)c(F)ccc2nc[nH]c12.C12(CC1)C(=O)NC2 c1(OC)ccc(CC(c2cc(C)ccn2)NC(=S)NC(C2CCC2)C)cc1 C1(N)CC12CCCCCC2.C1(c2n(C)nnn2)CCC2(CCC2)OC1 Cc1cc2cccnc2nc1C(=O)N(CCNC(=O)CN1CC2CC2C1)C1CC1 CCC(C)C(O)CC(=O)NC1CCOC(C(=O)NCC2(C)CCCC2O)C1 C1(CC)CN(C)CCN1C(C1CC(O)CN1C(=O)Cc1c(C)cccc1C)=O C1(NC(Cc2ccc(CC)cc2)=O)CCN(C(c2csnn2)=O)CC1(C)C Cc1c(C(=O)NC2(c3cn(CC(C)(C)C)nn3)CC(C#N)C2)cnn1C C1(C(=O)NCC2(F)CN(C)C2)CCCCCCN1C(C1CCC1(F)F)=O C12(NC(c3c(C)cccc3)=O)CCC(CNC(=O)Cc3ccsn3)(CC1)OC2 C#CCC(CC#C)C(=O)N1CCOCC(NC(=O)C(F)(F)CN2CCCC2)C1 C1(NC(c2ccc(OC)c(Cl)n2)=O)CN(C(=O)C#CC(C)C)CCC12CCC2 N1(C(c2c(F)ccc(C)n2)=O)CCC2(CCC(NC(=O)C(C)C3CCCO3)C2)C1 c1(NC(C(CN(C(c2ccccc2F)C)CC)O)=O)cc(S(C)(=O)=O)co1 c1(C(CCC(=O)NCCCNC(C2C(OCC)C2)=O)=O)ccc(F)c(F)c1 n1(CC)nccc1C(=O)NCC1(F)CC(NC(c2cc(CO)[nH]n2)=O)C1 N(C1CCc2cccnc21)C(C(N(C(c1ccc(C)cc1)=O)C)C1CC1)=O c1(OC)ccc(Br)c(F)c1CNC(=O)NC1CC(C(C)(C)C)C1 C1(C#N)(OC)CC(C(=O)NC(c2nocc2C(=O)NCC2CN(C)CCO2)C)C1 Cc1ccc(I)cc1CCNC1CCN(C(=O)CC(C)O)CC1 c1(C(N2C(C(=O)Nc3cncc(C)c3)C(C)CC2)=O)cc(C)ccc1C C1(CNC(C2C(C)(C)C(F)(F)C2)=O)CC2CCCC2N1C(=O)CC1CCCCO1 C1(NC(CC(CC)SC)=O)COC2(C1)CN(C(=O)C(C)(C)c1ccno1)C2 C(=O)(C(O)CCC(C)C)NC1CC(NC(C(CCC)OC)=O)C(O)C1 CC(O)(CC(=O)NC1CN(C(C2CCC3(CC2)CC3)=O)CC12CCC2)C(F)(F)F N(C1CCCn2ncnc21)C(C(=O)NCCCC1CCOCC1)=O CCCC(C(=O)NCC1CCCN1C(=O)Cc1sc(C2CCC2)nc1C)OC N(C(=NCCN1CCOCC1)NCC(C)(C)CC1CC1)C1CC(C)OC1 c1(C(=O)NC(C)C(C)NC(c2cnc3c(c2)COC3)=O)nnn2c1CSCC2 N1(C(c2c(C)ocn2)=O)CCN(Cc2nnc(C)n2N)CC1 c1(CC(N2CC(COC)(NC(=O)CC(O)C3CC3)C2)=O)sc(S)nc1C C=C(Cl)CC(C(=O)N(C1CC2CC2C1)C)NC(=O)C1=CCCCO1 N1(C(C(C)OCC(C)C)=O)CC2CC1CCC2NC(C1CCC(C)(C)CC1)=O Cc1cc(C(=O)NC(C(=O)N(C)Cc2ccco2)C2CCCO2)cc(O)n1 c1(C(=O)NC(CN(C(=O)COc2cccc(C#C)c2)CC)C)cccn2nnnc12 N1(C(CC2C(C)C2)=O)CCCC(N(C(=O)COc2cn[nH]c2)C)C1 C1(NC(c2c(OC)cncc2)=O)CCc2onc(C(=O)N3CC(O)CO3)c2C1 C1(C(N(C2CCS(=O)(=O)C2)CCC)=O)CCN(CC(N2CCCCC2C)=O)CC1 c1(CC)ccc(Br)cc1C(=O)NCCCNC(C1(CSC)CC(F)(F)C1)=O C(=O)(C(F)(F)CC1CC1)NC(CC(C)NC(c1cnc(C#N)s1)=O)C c1(C(N(CCCN(C(C2C(C)(C(=O)OCC)C2)=O)C)C)=O)cnc(C(C)(C)C)s1 c1(C(N2CC3C(C2)N3C(c2ccc(F)c(O)c2)=O)=O)ccc(O)nc1Cl c1(C(=O)NCC2CC(F)(F)CN2C(C23CC2C3)=O)c[nH]c2cccnc12 C(=O)(C1CCOc2ccccc21)c1[nH]c(=NCC2CCC(C)(C)CO2)[nH]c(=N)n1 c1(C(=O)NC(C)CC2CN(C(=O)C=Cc3ccccc3)C2)cc([N+](=O)[O-])c[nH]1 C1(OC)CC(CN(C)C)N(C(c2csc(-c3csc(C)n3)c2)=O)C1.C(C)(C)(C)O C(=O)(CCC(C)CC(=O)NOC(C)(C)C)NC(CC(C)CN(C)C)=O c1(NC(C2C(C(N3CCCCC(C)C3)=O)C2)=O)ccc2scnc2c1Br N1(C(CC2C(C)C2)=O)CC2(CNC(C3CC3(F)F)=O)CC1CO2 c1(C(N2CCC(C3(NC(c4c(C)ocn4)=O)CC3)C2)=O)cnc2n1CCCC2C Cn1cccc1CC(=O)NCC(C)(C1CC1)NC(=O)C(O)CN1CCCC1 c1(C(=O)NC2(C)CCN(C(=O)C(F)(F)C3(O)CCC3)C2)ccc2ccsc2c1 C1(NC(c2n(C)ncc2)=O)CN(C(=O)Cn2cnc(Br)c2)C2CC12 CC1CN(C(C2(O)CCOC2)=O)CCCN1C(=O)CCN(c1cnccn1)C C1(O)(CC)CCC(NC(=O)C=C=C(C)C)CC1.C1(=O)C(COC)N1C c1(N2CCN(C3(OC)CC3)CC2)ncnc2ccsc12 c1(CCCC(=O)NC2(CNC(c3coc(O)n3)=O)CCCC2)ccc(F)cc1 N1(C(=O)Nc2c(C)cc3cccc(C)c3n2)CCC2(CC1)NCCC2C(N)=O c1(OCC(=O)NC2C(C(C)C)N(C(C3CC(C)(C)O3)=O)CC2)ccc(F)cc1Cl N(C1CCc2cc(F)cc(Br)c21)C(N1CC(CC)N(C(=O)C2CC2)CC1)=O C(=O)(CC(C(C)C)OCC)NCC1(F)CCN(C(C=CCC)=O)C1 c1(CC)ccc(C(N)C(N2CCC(C3CC3)C2)=O)cc1 Nc1cc(F)cnc1C(N1CCC(C(=O)NCc2ccccc2F)C1)=O Cn1ncc(C(=O)NCC(C)(C)CNC(C2(C)CCCC2O)=O)c1Cl N1(C(C2CC(=C)CN2C(c2ccnc(OC)c2)=O)=O)CCN2CCOCC2C1 c1(CC(=O)NC2CC(C)N(C(C3COCCO3)=O)CC2)nc2ncccn2n1 CCCC(CC(=O)N(CC(N)=O)CC(N)=O)NC(c1cnn(C(F)F)c1)=O c1(OC)cccc(Cl)c1C(=O)NCCCN(C(=O)COc1ccc(F)c(F)c1)C N1(C(CCC)=O)CC(C(=O)NC2(c3csc(C)n3)CC2)OC(C)C1 c1(C(=O)OC)cccc(C(N2CC(O)(CNC(=O)CSc3nc[nH]n3)C2)=O)c1C C1(C)(C(=O)NCCC(C)NC(c2ccc(OC)o2)=O)CCC(=O)NC1 N1(C(CCC2(C)CN(C(C3CCC4(CC4)C3)=O)C2)=O)CC2CC2C2CC12 c1(C(N2CCC(N(C)C(c3cnc(O)[nH]3)=O)C2)=O)cccc(OC(F)F)c1 C1(C(=O)NCCN(C(c2conc2-c2ccc(Cl)cc2)=O)CC)CCCN1N=O c1(C(=O)NC23CCCC2OCC3)cccc2c1OCC2 c1(C(=O)NCC(C)N(C)C(c2cccc(CN=[N+]=[N-])c2)=O)ccc(N)c(Cl)c1 N1(C(CSC(C)(C)C)=O)CCN(C(=O)CC2CC3CCC2C3)C(C2CCCC2)C1 c1(OC)ccc2ccccc2c1C(C(=O)O)CN1CCC(C(F)(F)F)C(N)C1 C1(C(=O)OC)CC(n2cc(-c3cccnc3C)nn2)CN1C(C1CCC1C#N)=O N1(C(=O)NC(C)CCC2CCCCC2)CCCCC12CCC2 C1(NC(C2(COC)CN(C(C3CCC3)=O)C2)=O)CC2(C1)CC(O)C2 C12(NC(CCCOCC)=O)CCCCCC1N(C(c1cnc(O)c(F)c1)=O)CC2 c1(C(=O)NCC(CNC(c2cc(C)n(CCO)n2)=O)(C)O)cccn2cnnc12 CCCCC(CC)CC(=O)NC1CCCC2CN(C(C3(C)CC(C#N)C3)=O)CC12 Cc1nn(C)c(N)c1C(=O)NC1(C(N2CCC(C)C(CO)C2)=O)CSC1 N(C1CCc2ccccc21)C(c1ccnc2c1CCC2)c1ccccc1 c1(OC)cc(-c2cnc(NC(c3cnc(NC(C)=O)o3)=O)c(O)c2)ccc1OC C(=O)(C#CC1(C)CCCO1)NC1CCC(C)(C)CC1CNC(=O)Cc1cccs1 Cc1nc(C)c(CC(=O)NCC(C)CNC(=O)C=C2CCC(C)CC2)c(O)n1 N1(C(=O)CC2CC3(CC3)CO2)CC2CCC1CN2C(=O)CNC(c1ccsc1)=O C1(C(=O)NC(C)C(C)(C)NC(=O)CCSC(F)(F)F)CN2CCN1CC2 N#Cc1cn[nH]c1C(=O)NCC1CN(C(C2CCCC3CC23)=O)C1 c1(C(=O)NCC(CNC(=O)C2=CSCS2)F)cc(O)nc2ccccc12 CCC(C(=O)N(CCNC(=O)CSc1cc(F)ccc1F)C1CC1)C(C)O CC(C)CC(C(=O)N1CCC(CC(C)C)(CC(=O)O)C1)N(C)C C1(NC(c2cnc(Cn3cccnc3=O)o2)=O)CCc2ccccc2OC1 C(=O)(CCCCCSC1(O)CC(NC(C2(CNC(C)=O)CC2)=O)C1)NCC(=C)C C1(N(CCC#N)C(C)C)CCN(C(=O)C(C)Oc2ccccc2C)CC1 N1(C(c2nc(C)nc(O)c2)=O)CCCC(C)(C)C1CNC(C1CC=CCC1)=O c1(C(N2C3CCN(C(=O)NC(C(=O)OC)C)C3CC2)=O)c(O)ccc2nc[nH]c12 c1(CN(C(C(C)OC(c2nn(C)cc2Br)=O)=O)C)ccc(F)cc1Br c1(C(N2CCCC2CNC(C2CC2c2ccsc2)=O)=O)cccc(NC2CC2)c1 C1(N(C)C)CN(C(=O)C(C)(C2CC2)N(C(=O)Cc2cccnc2O)C)CC1O c1(C(=O)OC(C(C)C)C(=O)N2CCC(O)CC2)nnc2c(C(F)(F)F)cccn12 c1(C(N2CC(NC(C(F)=C(C)C)=O)CC3(C2)CC3)=O)ccc2oc(=O)oc2c1 CCCC(CNC(=O)Cc1ccn(C)n1)C(=O)NOC1CCOC1 Cc1n[nH]c(C)c1C(C)NC(=O)CC1CCCC1NC(C1C=CC=CC=C1)=O C(=O)(C(O)C(CCC)NC(c1ccnc(O)c1)=O)NCCCCC#CC N1(C(C2(C)CCCN2C(c2sc(Br)cc2Br)=O)=O)CCOC(C#N)C1 c1(C(C)NC2CN(CCC)C(=O)C2)cc(F)c(Cl)cc1Cl CC#CCC(C(=O)N1CCCC(CCC)C1)NC(=O)CSC C(=O)(C1=C2CCCN=C2NN1)NC(C1CCN(C(C(C)(C)CF)=O)C1)C1CCCC1 C1(N(C(C(C(C)C)NC(c2cc(C)n(C)c2)=O)=O)C)CC(C)CC(C)C1 C1(NC(C(COCC)NC(=O)CN2CC=CC2)=O)CC(=O)N(C)C1 c1(C(=O)NC2CCC(CCCC)C2)cc(NC)nc(Cl)c1 C1(O)(CCNC(C2C(C)CCCC2)=O)CCN(C(=O)CC2CCNC2=O)CC1 CC(C(=O)N(C(C)CNC(=O)CCc1ccc([N+](=O)[O-])cc1)C)C(C)S(C)(=O)=O CC(CF)C(=O)NCC(CO)NC(=O)CNC(C1CCC1)=O C=Cc1cncc(C(N2CCCCC2CCN(C)C(c2cc[nH]n2)=O)=O)c1 CC1CCCN(C(=O)CC(C)(C)CN(C)C)C1CNC(=O)C(=O)NCCC(N)=O C1(C(=O)NC(CCC(C)C)=O)CCN(C(=O)CO)CC1O C1(NC(c2n[nH]cc2CNC(C23CC2CNC3=O)=O)=O)CCC12CCCC2 c1(C(N2C(C(=O)NCc3cc(Cl)nc(Cl)c3)C=CC2)=O)cc2cc(F)ccc2o1 C(CC(CC)C(=O)NCC(C)NC(=O)C=Cc1ncccc1C)=CC C1(C(=O)NC2(CC=C)CN(C(=O)CC3CCCCCC3)C2)CCS(=O)(=O)N1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CC(C)CN(C(=O)C(C)(C)N(C)C)CC1C S(=O)(=O)(c1cnccc1N(C)Cc1cncn1C)NCCc1nccc(C)n1 C1(CC)OC2(CCN(CC(N3CC4(CC(CN)C4)C3)=O)CC2)NC1=O Cc1ccc(C(=O)N(CCCC(=O)N(CCCC(C)(F)F)C)C)c(O)c1 N1(C(c2scc(C)c2)=O)CCCCC1CCNC(=O)C(C)c1cc[nH]n1 C12(C(N3C(C(C)(C)C)CCCC3)=O)CCC(CC1)CO2 c1(N2CC3CC(NC(C4=C(C)CCCC4)=O)CC3C2)nc(Cl)nc2c1CCOC2 N1(C(COCCOCC)=O)CC(NC(=O)C(O)COC)CC1(C)C C1(C(N2CC(=C)C2)=O)CC(NC(=O)CN2CCCNC2=O)CCO1 N1(C(C(CC)O)=O)CC(CNC(C2(c3cc(C)no3)CCOCC2)=O)C(O)C1 N1(C(C(C)N(C(c2c(CC)c[nH]c2)=O)C2CC2)=O)CCOCC1COC C=CCCCCCC(=O)N1CCC1(C)CC(=O)NC1(C)CCC(=O)N(C)C1 N1(C(c2c(CCC)nco2)=O)CCCC(C2CN(C(c3cnnn3C=C)=O)C2)C1 N1(C(c2cnccc2Br)CC)CCC(C)C1c1cccc(C)c1 c1(C(=O)NCC(C)C(=O)NC2CCn3cnnc3C2)ccc2cc[nH]c2n1 Cc1cc(C(=O)NCCCN(CCO)C(c2cnc(N(C)C)nc2)=O)c(C)s1 C1(NC(c2c(C)cc(CC)o2)=O)CC12CCN(C(=O)Cc1coc(C)n1)C2 Cc1c(C(N2CC(O)(CNC(c3nnn(C(C)(C)C)n3)=O)C2)=O)nnn1C c1(NCC)ccc(C(N2CCCC(CO)(CNC(C3(N(C)C)CC3)=O)C2)=O)cn1 C(CCCCC(=O)N1CCC1NC(C1(C(F)(F)F)CC=CCO1)=O)c1n(C)ccn1 C1(NC(C(C)OCCCCCC)=O)CCC12CCN(C(=O)CNC(C)=O)CC2 c1(NC(C)CNC(C2(O)CCSCC2)=O)ncnc2c1COC2 C1(CNC(C(CSC)O)=O)CN(C(C2(C)CCCC2)=O)CC(C)(C)C1 C(=O)(C1CCC(=O)c2ccccc21)N1C(CNC(c2[nH]cc(C)c2)=O)CCC1 C1(NC(c2c(CC)c[nH]n2)=O)CN(C(=O)C=Cc2cc(C)no2)CC1C CN1c2ccccc2N(CCNC(=O)NC2CCCC3(C2)N=N3)S1(=O)=O CC1CC(CNC(C2CC2C)=O)CCN1C(c1ccoc1)=O c1(OC)n[nH]c(C(N2CC(CCNC(C3(CF)CC3)=O)(OC)C2)=O)c1Cl C1(C)(NC(C2C(NC(C3C(OC)CC3)=O)CCO2)=O)CCCC1(F)F C1(C(=O)NC(CC#C)C(=O)OCC)(CC)CCN(C(c2cc(CC)on2)=O)CC1 S(=O)(=O)(c1c(C(F)(F)F)cccc1Cl)NCC(=O)NC1CCN(C)CC1 C1(CNC(c2cn(CCO)c(=O)nc2O)=O)CC2(CO1)CN(C(=O)C=CBr)C2 C1(CCC)CN(C(=O)CCn2ccnc2C)CC1NC(c1c(C)csc1OC)=O C1(CNC(CCC(=C)C)=O)CC(C)(C)CCC1NC(=O)C=CC1CCCCC1 C1(C(=O)NCC2(F)CC(NC(=O)CCCc3ccc(F)cc3)C2)CC2C=CC1C2 C(=O)(C1=NNC(=O)C1)NCC(CC(=O)NC(C(C)C)C1CC1)C1CCC1 C(c1cnccc1C)=CC(N1C(CNC2OCCN(C(C)=O)C2)CCC1)=O C(CN=c1nc(C(F)(F)F)[nH]s1)(C1(C(=O)O)CC1)NC(=O)CCc1ncccn1 C12(C(=O)NCC(CNC(=O)Cn3ncnn3)F)CC(C1)C(C(F)(F)F)O2 N1(C(CCC(=O)OC)=O)CCCC(NC(c2nccnc2C(F)(F)F)=O)C(F)C1 N1(c2ncc(C)c(O)n2)CCC2(NC(=O)CCN3CCCS3(=O)=O)CCCC12 N1(C(C2(C=C)CCN(C(c3cc(C)nc(O)n3)=O)C2)=O)CC2(CCC2)CC1CO N1(C(C(C)OCCCC)=O)CCCC(N(C(=O)Cc2ccns2)CC2CC2)C1 c1(OC)c(C(N2CCN(C(c3cncnc3C)=O)CC2C(C)C)=O)ncnc1C N1(C(CCN(C)CCO)=O)CCCCC(C2CN(C(=O)C(C)(O)C3CCC3)C2)C1 C1(CNC(c2ccc(C(N)=O)o2)=O)CC(C(=O)NC2CC=CCC2)=NO1 CON(CCC(=O)O)C(=O)N1CCCC(c2nnc(O)n2C)C1C c1(C(=O)NCC2OCC(C(=O)NCCC=CC)C2)ccc(F)c(O)c1 C12CCN(CC1O)C2.c1(CNC(=O)CCC2CC2)ccnc(N2CCCC2)c1 C1(CNC(c2c(CC)nccn2)=O)CN(C(=O)CNS(N)(=O)=O)CC(C)(C)O1 c1(C(N(CCCNC(CSCCCC)=O)CCO)=O)cn(CCOC)nn1 N1(C(C(C)OCC=C)=O)CC(C2CCN(C(c3scc4c3OCCO4)=O)CC2)C1 N(C(=NCC1CCS(=O)(=O)C1)NCC(F)F)C(C)C(c1ccccc1)C S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(=O)C(C3CC3)SC)C2)c1)NCC C1(NC(c2ccc(C(N)=O)o2)=O)CS(=O)(=O)CC1NC(c1cccc(CO)n1)=O CN1CCN(C(=O)C(C)(C2CCC2)NC(=O)CN2CCNC2=O)CC1C1CC1 C(C(O)C(=O)NCC1CCCC1NC(=O)CCc1cnoc1)N(C)C c1(C(=O)OC(c2ccc(Cl)cc2F)C)cc([N+](=O)[O-])ccc1C=O C1(C)(C(=O)NS(C(C)CCN)(=O)=O)C2CC3CC(C2)CC1C3 N1(C(CC2ON=C(C)C2)=O)CC2CCCC1C2CNC(=O)COc1ccn(C)n1 c1(CC)cc(CNC(=NC)NCC(C2CCCCN2C)(C)O)ccc1C c1(C(N2C(CN(C(=O)C(O)C(F)(F)F)C)CCCC2)=O)cc(F)ccc1Cl CCCCCCCC(=O)NCC1CCCN(C(=O)CCNC(C2CCC2)=O)CC1 C(C(=O)n1c2ccccc2c(=NC2CCCC2CCO)[nH]1)OC(C)C C(=O)(C(C)(C)C(F)(F)F)N(C1CCN(C(c2cn(CCO)nc2C)=O)CC1)CC Cc1noc2nc(C(N3CCCC(NC(C4(C)CCOC4)=O)C3)=O)ccc12 c12sc(nc1C)CN(C)C2C.C1(C(=O)Nc2ccncc2)CCC(COC)C1 N1(C(=O)COc2ccccc2F)CC2CC1CN2C(C1CC2(CC2)CO1)=O CC1(C)CN(C(c2ccoc2CNC(=O)C(C2CCOCC2)O)=O)CC1CO CCCCC(CNC(=O)Cc1c(C)noc1C)NC(=O)CC1CCOC(CC)C1 C1(NC(CCNC(C(C)(C)C)=O)=O)CC2CCC(C1)N2C(C1CCCOCC1)=O CC(CNC(=O)CCCC1CCCC1)C(F)C(=O)NCC(C)(C)N(C)C N1(C(CCN(C)CC)=O)CCCC2CN(C(C3CCCC3C(F)(F)F)=O)CCC12 c1(C(N(C2CCN(CC(=O)N(CC=C)CC=C)C2)CC)=O)ccnc(F)c1OC C1(F)(C(=O)NC(C(C)F)C)CCCN(C(c2csc(C#N)c2)=O)C1 C(=O)(CCP(C)(C)=O)NCC1CC(C)N(C(c2cc(C(C)(C)C)n(C)n2)=O)C1 N1(C(C(C)(CO)OC)=O)CCC(CNC(=O)C#CC2CCC2)C(F)(F)C1 CC(C)(C)C1=NOC(C(=O)OCc2cc3cnccc3o2)C1 Cc1cc(=O)c(C(=O)NC(C)C=CC(=O)NCC(C)CN2CCCC2)c[nH]1 n1(CC)ccc(C(=O)NC(C)C(=O)NCCC(N)=O)n1 c1(C(=O)NCC2(C)CC(NC(C34CCC(C3)C4)=O)C2)cc2cnccc2o1 C1(C(N2CCC(C(C)NC(=O)COCP(C)(C)=O)C2)=O)(CC)CCC(O)CC1 c1(C(N2CC(NC(CC(=O)OC)=O)(CO)C2)=O)c(C)cnn1C(C)C c1(NC(=O)CC2CCC23CC3)cccc(Cl)c1N1CCCCC1 c1(CCCNCc2n(CCCF)nnn2)cccnc1Cl.C1(C)CCCCO1 c1(C(N(C(C)CN(C(=O)CCCc2nc(C3CC3)no2)C)C)=O)ncc[nH]c1=O C1(C(=O)NCC(C)(F)CNC(=O)C(O)C2CCC2)CCn2nnnc2C1 CCCC(C(=O)NCC1(OC)CN(C(=O)C(O)C2CC2)C1)OCC C1(NC(C(C)OCC(C)C)=O)CCCCCC1C(N1CCC(n2cncn2)C1)=O c1(C(C)C)cc(C(=O)NCCCOCCCNC(=O)CC2CN(C)C2)on1 c1(C(=O)NCC2(C(=O)NOCCC(C)O)CC(=C)C2)cc(CO)c(C)o1 C1(C(=O)OC)(NS(=O)(=O)c2cccs2)COC(C)(C)C1 N1(C(c2n(C)ccc2)=O)CCCC2CN(C(C3(c4cccs4)CC3)=O)CCCC12 CC(C)C(F)(F)CC(=O)N1CC(NC(c2c(O)cccc2Cl)=O)C(C)C1 C#CC1CN(C(=O)CC2CCC(C)C2)CCN1C(c1cc(F)c(F)cc1N)=O c1(OCC=C)ccccc1C(N1CCCC(NC(=O)C(C)CO)C1)=O C1(OC)CN(C(=O)CC2CC3(CC3)CO2)CC1NC(=O)OC(C)(C)C C(=O)(C1=COCCC1)NC1CC2C(NC(C(C)(N(C)C)C3CC3)=O)C2C1 CCC(C)CCCCC(=O)N1CC=CCC1C(=O)N(C1(COC)CC1)C C1(C(N2C(CN(C(c3cc(C(C)C)no3)=O)C)CCC2)=O)C2(CCC2)C12CCC2 C1(N(CCCCCc2ccccc2)C(C2C3C(=O)OCC23Br)=O)CCS(=O)(=O)C1 CC(C)C(CNC(c1ccnnc1O)=O)C(=O)NC(C(F)F)C(C)(C)C c1(CN2CC(CC)N(C(c3ccnc(OC)c3)=O)CC2)cc(Cl)c(Cl)cc1F CC(C)CCCC(=O)NCC(F)CNC(C1CC2C(C1)C2(C)C)=O C=CCC(C)C(=O)NC(C(=O)NC1CCOCC1C)C(C)OC c1(C(=O)NC2CC(C)(NC(c3ccc(SC)o3)=O)C2)cc(C2(Cl)CC2)n(C)n1 C1(C(=O)OC(C)(C)C)(SC)CCCN(C(c2c(N)cncc2Br)=O)C1 C1(NC(Cc2c(F)ccc(C)c2)=O)CC2CN(C(=O)C(=O)CCC(C)C)CC2C1 C1(C)(CC)CCN(C(C2CN(C(=O)C(CCN(C)C)OC)CCO2)=O)C1 N1(C(C(COCC)C)=O)CCC2(CC1)CC(NC(=O)CC(C)CC(C)(C)C)C2 CC(C)C(C(=O)N1CCC(=CCNC(=O)CC2CCCCC2O)CC1)NC(N)=O C#CC1(C(N2CC3C(NC(=O)CCc4nc(C(C)OC)no4)C3C2)=O)CCCC1 Cc1cc2[nH]c(C(N3CC(NC(C4CC5CCCC(C4)C5)=O)C(O)C3)=O)cc2o1 C1(NC(CCCC=C)=O)CN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC12CC2 c1(C(N2CCN(C(c3ccc(C)cc3)=O)CC2C)=O)cc(F)c(C)c(N)c1F C1(OC)C(NC(C2CCC2CNC(C2(C)CC=CC2)=O)=O)CC1O C=CCCCCCCC(=O)NC1C=CCCC1C(N1C(CO)CC1C)=O O(N(Cc1ccc(C)o1)C(=O)C1(C(C)(C)C)CCCO1)CC c1(C(=O)NCC(C(=O)NC2C(O)CCC(C)C2)(C)C)cc2cc[nH]c2cn1 C1(C(=O)NCCCN(C(C2C(CCOC)C2)=O)C)CCC(F)(F)CC1(C)C N1(C(C(CCSC)NC(N)=O)=O)CCCC(C)(CNC(c2ccc(F)cc2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(C(COC)(C)O)=O)C2)cnc2cc(C)[nH]c2c1 C(CC(C)C(=O)N1CCC(NC(c2c[nH]nc2C2CCCCC2)=O)CC1)OC CC(C)CC(C)C(=O)NCC1CC(F)(F)CN1C(c1ccoc1C1CC1)=O C1(NC(c2cc(CC)[nH]n2)=O)C=CCC(C(N2CCC2C(N)=O)=O)C1 C12(CNC(C(CC)SC)=O)CCCC(CN1C(=O)CCC=CBr)C2 c1(C(CC)C(=O)N(C)CCNC(=O)CC2(C)CC2(Cl)Cl)ccc(OC)cc1 C(C(C(C)C(C)C)NC(C1(C(=O)NC2CC2)CCC1)=O)N(C(CC)=O)C Cc1[nH]nc(C(N2CCC(C)N(C(=O)Cc3ncn(C)c3C)CC2)=O)c1[N+](=O)[O-] N1(C(CSCC=C)=O)CCCC(CC(=O)NCC(=O)NOC)C1 Cc1ccc(C(=O)NCCCN(C(=O)Cc2nc(=N)[nH][nH]2)C2CC2)c(=O)n1C C1(C(=O)NC(C#C)C)CCCN1C(=O)C=CC1CCCC1 C1(CNC(Cc2ccc(C)s2)=O)C2CN(C(=O)Cc3ccccc3)CC12 c1(C(=O)NC(CC)CNC(=O)C(F)(CC)C(=O)OC)ccc2c(c1)OCCC2 c1(NC(C2(CCC)CC2)=O)cc(Cl)c(C(F)F)cc1F N1(C(C2CSCC(C)N2)=O)CC2Oc3c(F)ccc(F)c3OC2C1 C(=O)(C1=COCCC1)N(C(CNC(C1CCC(NC(C)=O)CC1)=O)C)C1CC1 C1(CCNC(C(CC)O)=O)CCN(C(=O)Cn2cnc(C3CC3)n2)CCC1(F)F N1(C(c2cnc(C)[nH]2)=O)CN(C)C(=O)N(C)C1 c1(OCC)nc(N(C2CCNCC2O)Cc2ccc(Cl)c(F)c2)ncc1OCC Cc1ccc(OCCC(=O)NCC2(NC(C3CCC(=O)CC3C)=O)CC2)cc1C c1(NC(CC(Cc2cccc(Br)c2)NC)=O)cc(Br)cnc1Br c1(CC)cc(C(=O)NC2CCN(C(c3cn[nH]c3)=O)CC2C)c(C)nn1 N1(C(C2CC(C)OC2C)=O)CCCCC(CNC(c2ccc(C(N)=O)[nH]2)=O)C1 C1(C(=O)NCC2(O)CC(CNC(CNC(C)=O)=O)C2)CC(=O)N(OC)C1 C=CC1(C(N2CCSC(CC)C2)=O)CCN(C(=O)CCCC(C)(C)C)CC1 CCC(CCOC)N=c1[nH]c(=N)[nH]c(=NC(C)c2cncc(F)c2)[nH]1 c1(CC)cc(F)ccc1CN1N(CCN(C)C(=O)C)C(=O)C(C)C1 c1(C(N(C)CC2CCN(C(C3(C)CCN(C)CC3)=O)C2)=O)cc(S(C)(=O)=O)cs1 C1(C(=O)NC(c2cncnc2)C)C=CCCN1C(=O)CN1CCOCC1 N1(C(C2(C)CC(F)C2)=O)CCC2(CC(NC(c3c[nH]nc3C3CCCO3)=O)C2)C1 C=C=C(C)CC(=O)NC(C1(O)CCN(C(=O)CN2CSCCSC2)C1)C C(=O)(C(O)C(F)(F)F)N1CCC(CC(=O)N(C)CC2CC2C2CC2)C1 c1(-n2cc(CN3C(COCC)CCC3)nn2)cnc(C(F)(F)F)cc1C Cc1c(Cl)c(C(N2CCN(C(C3CCCC3C(F)F)=O)C(C)C2)=O)nn1C c1(CNC(C=CC(C)NC(=O)Cc2cccnc2)=O)cccc(C#N)n1 CC(CC(=O)NC1(CO)CCCN(C(=O)CCC(F)(F)F)C1)CC(C)(C)C C1(NC(=O)Cc2ncc(C(F)(F)F)[nH]2)CCCN(C(C2CCCO2)=O)CCC1 c1(C(c2n(CCC)nnn2)NCC(C)C2CCC2)c[nH]ccc1=O C1(NC(c2ccc(OCC)nc2)=O)CCC2CN(c3ccc(C#N)nn3)CC2C1 Brc1ccc2nnc(CNCC34CCCNC3COC4)n2c1 CCCC(C)CC(=O)NCC(C1CC1)NC(=O)CSCc1nnc(C)n1C c1(C(=O)OCCF)ccc2ccc(C3=CCOCC3)cc2n1 C1(F)(C(=O)NCC2CC(NC(=O)CCCC3CC3)C2)CS(=O)(=O)CC12COC2 CC(=O)CCN=C(NCC(C)C)NC1CCC(C(N)=O)C1 C(CC(C)C)(C(=O)NCC1CCCN(C(c2cnc(SC)o2)=O)C1)N(CC)CC C1(CNC(c2c(F)cccc2F)=O)CN(C(c2ccccn2)=O)CC12CCC2 CC1(C)COC(CC(N2CC3C(CC(=O)NCC(F)Cl)C3C2)=O)C1 c1(CC(=O)NCC2CCCN(CC(=O)NC(=O)OC)C2)cccc(Cl)c1Cl C1(NC(CS(CC)=O)=O)CN(C(c2cccc(C)c2Cl)=O)CC1C1CC1 C1(CNC(C2(CC=C)CCOC2)=O)CC2(CO1)CN(C(C1(CO)CCCC1)=O)C2 N1(C(C(Cc2c(C)n[nH]c2C)C)=O)C2CCC1CC(N(C(=O)C(O)C1CC1)C)C2 C(=O)(CCCCN=[N+]=[N-])NCC(C)(CNC(=O)C(=Cc1cscn1)F)OC c1(C(=O)NCCc2nc(C)c(C)s2)cc2ccccn2n1 N1(C(=O)OC)CCC(c2nnnn2CC(F)F)(NCC2CCCSCC2)C1 C=C(CNC(=O)NC(c1ccccc1F)CF)C(F)(F)F N1(CC(N2C(C(=O)NC(COC)(C)C)CCC2)=O)CCC(F)CC1 C12(NC(CC(CC)O)=O)CCC(n3cc(CN4CCCC4CO)nn3)(CC1)C2 C1(CC)C(C(N2CCC(O)CC2)=O)CCN1C(C1CCSCC1)=O N1(C(C(CC)CC)=O)CCN(C(=O)CN2CCC2)CC1c1ccccc1Cl N1(C(CO)=O)CCOC2(C1)CN(C(C1CC1C)=O)C2.C#Cc1cc(C=O)cc(Br)c1 N(C1c2ccccc2CC1NC(=O)C(C)(F)C(F)(F)F)C(C(C(C)C)(C)C)=O C(c1ccc(C2OCCO2)o1)=CC(=O)NC1CC(NC(=O)CC2CCCCO2)C1 N1(C(COCP(C)(C)=O)=O)CC(CNC(=O)CC2CC(=O)C2)CC12CCC2 C1(NC(c2nc(C)n(C)n2)=O)CCCCC12CCCN(C(=O)CC(C)F)C2 CC(CN(C)C)CC(=O)NCCC1CCN(C(=O)CCC2CCC2)C1 CCCCCC(C)CC(=O)NC(C1CCN(C(=O)CCS(C)=O)C1)C CC(=NOOC#N)C(=O)NCCCOCCC(=O)NCc1cnn[nH]1 c1(C(C)O)ccccc1Oc1ccccc1.c12cn(nn1)CC(=O)N1CCC21 c1(N2CCC(c3ccccc3)(NC(CC)=O)C2)cc(C)nc2ccnn12 CC1(CNC(=O)CCNC2COC2)CCN(C(=O)CCc2cnoc2)CC1 C(CCN(C(=O)C=CC1CCCC1)C)(C(C)C)NC(C(COCC)C)=O c1(C(=O)Nc2cc(C(=O)OC)ncc2Br)cnc2onc(C)c2c1 c1(C(N2CC3C(CNC(c4c(C)noc4)=O)C3C2)=O)c2n(c(=O)n1C)CCCC2 N1(c2cc(OC)ncn2)CCCCC(NC(c2ccc(F)c(F)c2)=O)C1 C1(NC(C2CC(=O)N2)=O)CC2CCC1CN(C(c1cc(C(C)(C)C)sc1)=O)C2 N1(CC(CC)CC)CCC(CC(C)N(C(=O)CCCF)OC(C)=O)CC1 C=CCC(CNC(=O)CCC=C(C)C)C(=O)NC(C(O)CO)C1CC1 CN1CC(NC(N2CCCC2CNC)=O)CC12CCC2.c1(O)ccc(C#N)cc1 N1(C(c2cccc(OC)c2)=O)CC2(CCCC2NC(=O)C(C)CC2CCC2)C1 N1(C(C(c2ccc(C)cc2)C)=O)CC2(NC(=O)OC(C)(C)C)CCC1C2 c1(C(=O)NC(c2ccccc2F)C(=O)O)cc2c(Br)cccc2c(=O)o1 C(CCCC(=O)NCC=CC(=O)NCc1occc1C)OC C1(CNC(C(C(=O)OCC)F)=O)CC2CCC(C1)N2C(=O)C(C1CCOCC1)O C1(C(=O)NCC2CCN(C(c3c(C)noc3N)=O)C2)OCC2CCCC12 n1(CC(=O)NC2CC(CNC(C3OCC(C)(C)C3)=O)C2)cc(S(C)(=O)=O)cn1 C(=O)(C(C)N=[N+]=[N-])N(CC(=O)NCC=C=C)CCOC c1(CN(CC)CC)cc(C)cc(Br)c1.c12ccc(o1)CN2CC Cc1ccc(C(N)CC(=O)NC2(CO)CCOC2)cc1 CCC(C)(C)C(C(=O)N1CCN(C(=O)C(=Cc2ccncc2)C)CC1)OC c1(C(=O)NC(C)CCCNC(=O)C(=Cc2cccnc2)F)cccn(C)c1=O c1(CC)nnsc1C(N1CCC1CNC(=O)CC1CCNC1=O)=O c1(C(C)C)ccc(N)c(C(N2CCC(NC(C3(F)CC4(CCC4)C3)=O)C2)=O)c1 CCC(C)C(C)NCCCl.S(=O)(=O)(CCn1cnnn1)NCC N1(C(=O)OC)CCC(C(=O)NC(C(=O)C(=O)C(C)SC2CC2)C(C)C)CC1 c1(N2CC3CN(C(c4ccc(Br)c(C)c4C)=O)C3C2)ncc2[nH]cc(I)c2n1 c1(C(N2CC(CC)C(C(=O)NC3CCN(CC)C3)C2)=O)nc(C)ccc1C C=CC1(NC(C2(N(C)C(C3(C)CC4CC4C3)=O)CC2)=O)CCCC1 CC(C)C(C(C)NC(C1(F)CCCCC1)=O)NC(c1coc(CO)c1)=O c1(CC(N2CC(O)(CNC(c3c(C)noc3)=O)C2)=O)cc(Cl)ccc1Br CC(N=[N+]=[N-])C(=O)N1CC2CC1(C(=O)NCCCCN=[N+]=[N-])C2 C(=O)(CCCCC(N)=O)N1CCC=C(CNC(c2c(C)ccnn2)=O)C1 C1(CNC(c2c(C)cc(SC)o2)=O)COCCN(C(=O)C(C)OC2CCOC2)C1 CC1=CCCN(C(=NCc2ccc(OC)cc2)NC(c2cccs2)C)C1 N1(C(CC(CCC)NC(C(CC=C)C)=O)=O)CCCC(C)(C#N)C1 N1(C(CCCCCC#N)=O)CCC2CCN(C(c3ccnc4[nH]nnc34)=O)C2C1 N1(C(c2c(C)nc(C)s2)=O)CCCC2(CCC2NC(c2csc(O)n2)=O)C1 Cc1ccncc1CC(N1CCC(O)(CNC(c2coc(C(F)(F)F)n2)=O)C1)=O C(CC(=O)NC1CN(C(C)C)C1)(C(F)(F)F)NC(CCC)=O CCC(C(=O)N1CC(O)(CCNC(C2CC2Cl)=O)C1)NC(C)=O C1(CN2CCOCC2)C2CN(C(c3ncccc3F)=O)CC12.C12(CC1)N(C)C2=O C1(NC(C(C)SCCCC)=O)CCCCC1CNC(=O)C(C)C1CCC1 C1(CC)(NC(=O)Cc2ccccc2O)CCCN(C(C2(C(=O)OC)CCC2)=O)C1 O=C1CCN(CC2CCC3(COC3)O2)C(=O)N1CCCOc1ccccc1F CC(O)CCCCCC(=O)NC(C)CNC(=O)CCC1CC1 C1(C(N2CCN(CCNC(=O)CC3(C)CC3)CC2)=O)(CC)CC(F)(F)C1 CC1CCN(C(c2cc(CO)on2)=O)C1C(=O)NC1CCOCC1F Cc1[nH]c2ccc(Br)cc2c1CC(N1CCCCC(c2ccc(F)cc2)C1)=O Cc1cc(F)ccc1C(O)C(=O)NCCN(C)C(C1CC1c1ccco1)=O n1(CC(=O)N(C2CCCN(C(=O)C(O)CF)CC2)C)ccc([N+](=O)[O-])n1 C1(C(=O)NCc2ccc(CC)o2)CC(O)CN1C(c1ccn(C)n1)=O CC(=O)CC(C)(C)C(=O)N1CC(=C(F)CNC(=O)Cc2cnn(C(C)(C)C)c2)C1 CC(C(=O)NOCC(N1CCC(c2ccco2)C1)=O)N1CCC1 N1(C(COC2CC(NC(C(C(C)C)F)=O)C2)=O)CCn2ccnc21 CC1CCNCCC1N(C(c1cc(O)ccc1O)=O)C(c1cccc(Cl)c1)C C(=O)(C(C(C)(C)C)n1ccnn1)NCCC(C)N(C(C=CC(C)(C)SC)=O)C Cc1cn(C)nc1C(=O)N(CC(=O)NC1CC(C(N)=O)C1)C1CCC1 c1(C(N(CC(CNC(CCCOCC)=O)(C)C)C)=O)cccc2c1C(C#N)C2 C1(NC(COCC(=O)NCC)=O)CN(C(C23CC4CC2C3C4O)=O)CC12CCC2 CC(C)C(CCN(C)C(C1CCC(F)C1)=O)NC(=O)CSC1CC1 N1(CC(CC)C)CC2CCC(NC(c3cc4n(n3)CCCC4)=O)CC2C1 CC1=C(C(=O)N2CC3CC2CN(C(c2ccc4cccnn24)=O)C3)CCCO1 CCCC(C)(CCC)C(=O)NC1C=CCC(C(=O)NOCCCC2CC2)C1 c1(C(=O)NCC(C)(C)OCCNC(C2(F)CCOC2)=O)cnc(Cl)[nH]1 N1(C(C2(C)CNC(=O)C2)=O)Cc2nccn2CC(NC(c2cscc2Cl)=O)C1 C1(C(C)NC(N)=O)CCCN1C(=O)C(C1CCCCC1)C CC1(C)CCC(C)(C(N2CC3CCC3(CCNC(=O)CSC3CC3)C2)=O)CC1 N1(C(C=CC=CC)=O)CCOC(C)(CNC(=O)C(C)Oc2ccc(Cl)cc2C)C1 Cc1cc(-c2ccnc(NCc3cccc(O)n3)c2)cc2c[nH]nc12 c1(OC)cc(C2(C(=O)N(C3CC(O)C3)C)CC2)nc2ccccc12 C1(NC(c2csc(Br)n2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CCC1CO Cc1ccc(C(=O)N(C2CCC(C(=O)NCC(N)=O)C2)C)o1 c12cccc(c1F)NC(=O)C(=O)N2.C1(C(C)C)CC(C(=O)N(C)C)CCO1 C(c1cc2ccccc2o1)=NC(=O)CCCn1cc(C2(CN(CC)CC)CC2)nn1 c1(C(N2C(CNc3cc(OC)nc(C)n3)COCC2)=O)cc2nc(C)ccc2o1 c1(CNC(C2N(C(C3N(C)CCOC3)=O)CCC2)=O)ccc(F)cc1F c1(CC)cccc(F)c1C(=O)N(C1CCN(C(=O)C(=O)C(C)(C)C)C1)C Cn1nc(CNC(=O)C(C)(C)F)c2c1CCN(C(c1ccccc1C#N)=O)C2 C1(CC)CC2CN(C(=O)CCOC(C3OCCN(C(C)(C)C)C3)=O)CC12 c1(C(=O)NCCCC(C)NC(c2cccc(C(F)(F)F)n2)=O)csc2cncn12 c1(C(N2C(C)CN(C(=O)CN(C)C)CCC2)=O)cc2ccc(Cl)nc2s1 c1(C(=O)NCCC2N(C(C(CC)CC)=O)CCC2)cccc2cncn12 O=C1CC(CCN2CCCC(C3CCCCN3C(C3CCSC3)=O)C2)C(=O)N1 N1(C(c2c(CC)ncs2)=O)CCCCC(CNC(=O)Cc2conc2C)C1 C1(C(=O)NC(C)C(C)(C)NC(c2cc(C3CCC3)[nH]n2)=O)CC2COCC2C1 C=C(CNC(=O)C(O)C1CCCC1)CCNC(c1csc(C(C)C)n1)=O N1(C(c2cc(SC)c(F)cc2)=O)CCC2CCC(C1)N2C(=O)Cc1ccoc1 CC1(C)CC(NC(C2C3CCCCC23)=O)CN1C(=O)Cc1ccoc1 c1(N2CC(NC(CCC(=O)N(C)C)=O)CC(C)(C)C2)nccc(S(C)(=O)=O)n1 Cc1c(NCc2cn(C(c3cc(C(F)F)on3)C)nn2)cc(F)cc1Br c1(C(N2CC3(C2)NC3)=O)cc([N+](=O)[O-])ccc1NC.c1cncc(C)c1C.OC N1(C(C23CC(OC)C2C3)=O)CCN(C(c2cnc(N)c(N)c2)=O)CC1CO N1(C(C(COC)OC)=O)CC2CCC1C1CN(C(c3cc(C(C)=O)c[nH]3)=O)CC21 C1(C(=O)NC2C(CNC(c3noc(CC)c3C)=O)C2)CC(=O)NC(=O)N1 n1(CC)nc(C)c(CC(=O)NCCC2CCCCN2C(c2c[nH]c(=N)s2)=O)c1C N1(C(c2c(Cl)cn(C)n2)=O)CCC2CN(C(=O)CCc3cc(Cl)no3)CCC12 c1(OC)ccc2c(c1)CCC2C=O.C1(NC(C23CC4CC2C3C4)=O)C2CCN(C)C12 C1(CC)CN(C(=O)C(c2c(F)cccc2F)C)CCC1NC(c1[nH]cnc1C)=O CC1CC(NC(c2cc(C3CC3)nc(O)c2)=O)CN(C(=O)CC2CCC(=O)O2)C1 N1(C(C(N2CCOCC2)C)=O)CCC(NC(=O)CCc2cc(Cl)no2)CC1C C(=O)(C(F)(F)C(C)O)NC1CCC(CC(=O)NCc2n(CC)nnc2C)C1 C(=O)(C(C)(C)CC(=O)NC1C2CC1CN(C(C1CC(n3cnnc3)C1)=O)C2)OC C(=O)(C(O)Cc1ccccc1)N.c1(C(N2CCC2CC2CC2)C)nnc(C(C)(C)C)o1 C1(C)(CC(N2CC(O)(CN(C(=O)CCC3CCCO3)C)C2)=O)CC(F)(F)C1 C1(C(N2CCC(C(CO)NC(C3(CF)CC3)=O)CC2)=O)CN2CCN1CC2 N1(Cc2c(C)noc2C)CCCCC(NC(c2c(Cl)cncc2Cl)=O)C1 n1(CC(=O)N(C2CCN(C(CC(CCC)CC)=O)C2)C)cc(C#N)c(O)nc1=O C12(NC(c3cc([N+](=O)[O-])ccc3O)=O)CCOCC1CN(C(C1CCSC1)=O)C2 N1(C(c2cn(C)nn2)=O)CCC(C2CC2NC(=O)CSc2nncs2)CC1 C(=O)(CCCCC#N)N1CCC(C(C)(C)NC(=O)CC2CC3(CCC3)C2)C1 S(=O)(=O)(c1ccc2nc(NCC(C)CC(C)C)sc2c1)NCCOCC=C C1(C)(CC)CCCC1NC(C1CC1CNC(c1cc(COC)cs1)=O)=O c1(C(=O)NCC(CC)(C)NC(=O)CN2CSCC2=O)cnn2ncccc12 C(N=c1nc(O)c2ccccc2[nH]1)C1CN(C(CCOCC#C)=O)CC1C N(C(=NCC1CC(=O)N(C(C)C)C1)NCC1CC(Cl)(Cl)C1)C(CC)CO N1(CC)CCc2cc(Br)c(S(=O)(=O)N3CCCC(O)(CCN(C)C)C3)cc21 C(=O)(C(C)(O)C(C)c1ccccc1)NCCOCCNC(Cc1c(C)scc1)=O N1(C(c2cc(CC)nn2C)=O)CCC(C2CC2)(CNC(C2CCCOC2C)=O)C1 c1(C(=O)NC(C2(O)CN(c3ccnc(C(F)(F)F)n3)C2)C)ncccc1Cl N1(C(C2CC(=O)NC2)=O)CCC2C(C1)OCCN2C(c1cnc2[nH]ccc2c1)=O C(=O)(C1CCCc2ncnn21)NC(C)(CNC(c1ccco1)=O)CO c1(C(N2CC3(C2)CN(C(=O)C(F)n2cccn2)C3)=O)ccc2c(c1)CCNC2=O c1(C(C)C)ncc2c(n1)CCN(N1CCC(Cc3cccc(F)c3)C1)C2 c1(CC)c(C(N2CC=CC2CNC(C2CCOC2C)=O)=O)cccc1C C1(F)(CNC(C(N2CC(C)C2)C)=O)CCN(C(=O)CCc2cocn2)C1 C1(CC(=O)N(C)CC2CCN(C(c3cncc(N)c3)=O)CC2)CCCC2(CC2)C1 c1(SC)ccc(C=CC(=O)NCC2(F)CN(C(C3CC4CCC(C3)O4)=O)C2)cc1 S(=O)(=O)(c1ccc(CC(N2CC(NC(=O)CC3CCC3(C)C)C(O)C2)=O)s1)NC C(CC(C)(CC)NC(C12CCCCC1C2)=O)NC(CC(=O)OCC)=O c1(C(N2CC=CC(NC(C3(CO)CC3)=O)C2)=O)cc2c(=O)cc[nH]c2s1 n1(CC)cc(C(=O)NCC2CC(NC(=O)OC(C)(C)C)C(OC)C2)c(C)n1 C(C1(C)CCOCC1)=CC(N1CCCC(CN(C(=O)C=CS(C)(=O)=O)C)C1)=O c1(CC(=O)NC2CN(C(=O)CCC(F)(F)F)CC2O)ccc(Br)c(F)c1 CCC(C)CCC(=O)N1CC(C)C(C)(CNC(c2c[nH]c(=N)nc2O)=O)C1 c1(C(=O)NCC2CCCCN2C(C2CC3CC3C2)=O)cnc2c(c1)COCC2 C1C(C)(CC(C)C)C(=O)OCCN(CCC#N)C(=O)N1.C(C(C)(C)C)OC C1(C(=O)OCC)CCC(C(C)C)N1C(=O)C(C)CN(c1ccccc1)C c1(C(N2CCC(N(C(c3n[nH]cc3F)=O)CC)C2)=O)oc2ccc(C)cc2c1C S(=O)(=O)(c1ccc(Cl)s1)Nc1cc(C(=O)OCC(=O)NCC(=O)OC)c(C)o1 c1(C(N2CCCC(CCNC(c3cc(Br)ncc3Br)=O)C2)=O)cc(Cl)ncc1Cl CC1CCN(C(C2CCC3(CC3)N2C(=O)C(O)CN2CCCC2)=O)CC1(C)C C(=O)(C(C(C)(C)C)OC)N(CC(C)NC(c1cnc(C(=O)OC)s1)=O)C C(CC(=O)NCC(O)CO)=CC=C.C1CC(=O)N1 N1(C(CC2(C)N(C(CCC#CC)=O)CC2)=O)CCc2ccc(O)cc21 C1(NC(c2cnn(C)c2Cl)=O)CN(C(C2COC3COCC23)=O)CC(C)(C)C1 c1(-n2c(C(CCCC)[SH2]CC=CC3CC3)nnn2)ccccc1Cl c1(C(=O)NC2C3CN(C(c4c(SC)ccs4)=O)C(C3)C2)c(C)cc(C)nc1C CCC(CC)CCC(=O)N1CC(C(=O)NCC2(CN(C)C)CC2)(COC)C1 c1(C(=O)NCCC(C)NC(C=Cc2nc(C)sc2)=O)ccc2ccn(C)c2c1 CCC(C)C(C)CNC(=O)C(C)(C1CC1)N(C)C(c1ncccc1Cl)=O C1(C(=O)NCCCC(=O)Nc2cnn(C)c2)(CC)CCCCO1 CC1(C)CC(CNC(C2CCCO2)=O)CN1C(c1cc(C(F)(F)F)on1)=O C1(C(=O)NCC(C)C)CCC(NC(c2n[nH]c(=N)[nH]2)=O)C1.C(C)(C)(C)O C1(N(C)C)(C(=O)NC2CCCC2NC(=O)COCc2nc[nH]n2)CCCSC1 C(C)(C)(C(=O)N1CCC(OCC(=O)N(C2CC2)Cc2cnn(C)c2)C1)N(C)C c1(-c2cn(C)nc2)ccc2nccc(C(=O)N=c3[nH][nH]cc3-c3ccccc3)c2c1 c1(-n2ncc(C)c2)cccc(C(=O)NC(C)CC2CN(C(=O)CSC(F)F)C2)c1 C1(C(=O)O)CC1C1CC1.N1(C(CSCCN(CC)CC)=O)CC(O)C1 C1(CNC(C2CN(C)C(=O)C2)=O)CC12CCN(C(c1scnc1C(F)F)=O)CC2 C(CCCCC(=O)OC)N(C(Cc1c(CC)ccs1)=O)C N1(C(=O)CC2OCCCO2)CCCC(F)(C(N2CCC2C2CCCCC2)=O)C1 C#CC(CC)(CC)NC(C12CC(CN1C(=O)Cc1ccccc1F)C2)=O c1(C(=O)NC2(C)CCCN(C(CC3(C)CCOCC3)=O)C2)cnc2c(c1)COC2 c1(C(=O)NC2C(CNC(c3c(C)cc(C)nc3O)=O)C2)ccc2ccccc2n1 N1(C(C=CCCC)=O)CCC2(CCCN2C(c2cnccc2Br)=O)C1 Cc1cnc(NC2CCN(CC)C2)c(S(=O)(=O)NC2CN(S(=O)(=O)N(C)C)C2)c1 c1(C(=O)NC2CN(C(COCCOC)=O)C2)ccc(SC(F)(F)F)[nH]1 Cc1cc(C(=O)NC2CC(F)(CNC(c3ccc(C#N)n3C)=O)C2)ccc1Br CC(C)(O)C(F)(F)C(=O)NCCCNC(c1ccccc1-n1ccnn1)=O CC1CC=CCC1C(N1CCCCC1C1CC1)C(=O)NCc1cc(Cl)cs1 c1(CC)cc(C(=O)NCC2COC(CNC(=O)CCc3nccn3C)C2)c(C)o1 C1(C(=O)NCCC)CC2(CN2C(=O)Nc2ccc(-c3ccccc3)cc2)C1 CCCS(=O)(=O)C(C)C(=O)N1CC(NC(c2ccsc2COC)=O)C2(CCC2)C1 c1(C(N2C(C(C)(C)C(=O)NCCCCF)CCC2)=O)c[nH]c2ncccc12 C1(CC(=O)NCC2CC(NC(C3N(C)CCC3)=O)C2)OCCCC1(C)C N1(C(C2C(C)C2)=O)CC2(CCN2C(=O)Cc2cccc(OC(F)(F)F)c2)C1 CN(C)NC(=O)CCC(=O)N(C1CCCC(NC(C2CN(C(=O)N(C)C)C2)=O)C1)C c1(C(=O)NC(CCCC)CC)cccc(S(=O)(=O)NCc2ccc(OC)cc2)c1 c1(C(=O)NC(CNC(CCOCCC)=O)C(C)(C)C)ncc(C2CC2)cc1C N1(C(C(CCCC)=O)=O)C2CCC1CC(NC(c1ncc[nH]c1=O)=O)C2 Cc1cc(C(=O)NCCN(C(=O)C(C)CC2CCC2)CC(C)O)c(C)n1C C(C(C)(C)CC(=O)NOCC1(F)CCC1)NC(c1nc(C)sc1C)=O c1(CC(=O)NCC2C3CN(C(=O)C=C4CCCCC4)CC23)ccccc1F c1(C(=O)NC2CC(CNC(CCNC(C)=O)=O)C2)cccc(C)c1O N1(C(C(CC)O)=O)CCCC(O)(CN(C)C(c2cn(C)nc2C(C)(F)F)=O)C1 CN1CCCCC(C(=O)NCC(C)(C)CNC(=O)CCCc2cccnc2)C1=O C(=O)(C#CC1(C)COC1)NCCC1N(C(Cc2c(C)cccn2)=O)CCCC1C CC1CCCn2c(C(=O)NC3CN(C(c4c(N)cccc4Cl)=O)CC3C)cnc21 N1(CC(N2C3CC(NC(C4CC(SC)C4)=O)CC2CC3)=O)Cc2ccccc2C1 C=CCC(C(=O)NCCC1CCN(C(=O)Cc2csnc2C)C1)NC(C)=O C12(NC(c3c(N)cn(C)n3)=O)CCCCC1CN(C(C1CC1C1CCCC1)=O)C2 C1(C(N2C(C(N(C)C)=O)CC2)=O)CC2(CCN1C(C1CC3CCC1CC3)=O)CC2 N1(C(=O)OCC)CCC(ON2CCC(N(C(C34CC(CO)(C3)C4)=O)C)CC2)CC1 CC(C)(C)C(O)CNC(c1ccoc1CNC(C1CCNC1=O)=O)=O N1(C(C2N(C(c3sc(C)c(Br)c3)=O)CC2)=O)CCCCC(F)(F)C1 c1(CS(=O)(=O)N(CCC)Cc2cnn(C)c2C#N)ccc(Cl)cc1F C(=O)(C#CC1CCCCO1)NCCC(=C)CNC(c1ccc(C(=O)NC)cc1)=O c1(C(N2CC(C(C)NC(C3(CO)CCC3)=O)OCC2)=O)ccc(F)c(F)c1F C1(C(C)C)N(C(=O)C(C)C(C)O)CC12CCN(C(C1CC(C)CO1)=O)CC2 C1(C(N2C(CC(=O)NCC=CCOC)COCC2)=O)CC(=O)NC(C)C1 CN1CC(N2CCC(c3nncn3C)CC2)C(C)(C)CC1=O C1(CNC(c2n(CC)ccc2)=O)CCN(C(=O)Cc2nnc(S)n2C)CC1O C(=O)(C1CCc2cc(F)ccc21)NCC1CC(C)N(C(c2ccnn2C)=O)CC1 C1(NCC#C)CCN(CC(=O)NCc2ccc(-c3ccc(F)cc3)o2)CC1 C1(C(=O)NCC(C)CC(=O)N2CCC2C(C)(C)O)CC2CCC1CC2 C1(NC(C(C(C)O)NC(=O)CC2CCN(C)C2=O)=O)CC2C=CCC(C1)C2 N1(C(c2cc(C)c(Cl)cc2)=O)CCC2CN(C(=O)C(C)(C)F)CC12 CC1(C(=O)NC2CCC2NC(c2ccc[n+]([O-])c2)=O)CC=CCO1 Cc1cc(=NCC(O)c2ccc(Cl)c(F)c2)[nH]c(N(CC(C)CO)C)n1 CC1(C)CCC(CCN2CC(CNC(C3CCCCC3n3cccn3)=O)C2)C1 Cc1sc(=O)n(C(=O)N(C2CN(c3ncnc(C(C)(C)C)n3)C2)C)c1C c1(C(C)C)ccccc1OCC(N1CCC(C)C1CNC(c1ccsc1)=O)=O n1(CC)cc(C(=O)NC(C)(CO)C(=O)NCCSC)c(C)n1 C1(NC(CNC(CN(C)C)=O)=O)(CNC(=O)CC2CCSC2)CC2CCC1C2 c1(C(N2CCN(CC3CN(C(=O)NCC)C3)CC2)=O)nccc(OC)c1OC c1(C(=O)NC(C)CC2CN(C(C3CCCC34CC4)=O)C2)cccc2c1OCCO2 CCC(C)(C#N)C(=O)NOCC(=O)NCCN(C)C(C)C C(C)(C(C(=O)OC(C)(C)C)NC1CC1)C(=O)SCC(N1CC(OC)C(SC)C1)=O C(=O)(C(F)C(=O)NC(c1ccccc1)CNC(=O)COC1CCN(C)CC1)OC C1(C(=O)NC(C2N(C(C(C)Cc3ccncc3)=O)CCC2)(C)C)CCCN1C=O N1(C(C)C)CCCCC1C(N1CCCC1C1(NC(=O)C2=CCCO2)CC1)=O c1(CC)cnc(C(N2C3CN(C(c4cccnc4N(C)C)=O)CC23)=O)nc1 C(CO)(C(C)N=c1[nH]c(=NC2CC(C(F)(F)F)C2)[nH]c2c1CCCCC2)SC S(=O)(=O)(c1cc(C)cnc1NCCCCCCSNCCC)N1CCCC(C=C)C1 C(N=c1cc(Cl)nc(C2CCC2)[nH]1)C1CN(C(c2cc3n(n2)CCCO3)=O)C1 Cc1cccnc1C(F)(F)C(N1CC(NC(C2CC2C(C)(F)F)=O)C(O)C1)=O c1(CC(=O)NC2CC(F)(CNC(C(Cn3ccc(C)n3)C)=O)C2)cccc(F)c1 CC1C(=O)N(CC(=O)NCc2cccc(CNC(=O)C=CC(N)=O)c2)C(=O)C1C C12(C(=O)OC)CCC(C(=O)NC3CCC3NC(=O)C=Cc3scnc3C)(C1)C2 C(CC(O)CC(=O)NC1CCCCC1CNC(=O)CCc1ccncn1)SC c1(CSCC(=O)NC2C(CNC(C=C)=O)C2)cccc(O)c1 C(=O)(CCCCSC)NC1CC(CNC(COC)=O)C1 C=CC1(CC(=O)NCC(C)(C)OCCNC(=O)C(O)C2=CCC2)CCOCC1 c1(-c2nc(C(C)OCC)nn2-c2cnc3ccsc3c2)nccc2[nH]ccc12 CC1CC(C(=O)NC2CCC(NC(=O)CN(c3ccnc(Cl)n3)C)CC2)CCO1 Cn1nccc1NC(C1CCCN1c1nnc(-c2ccccc2)o1)=O N1(C(c2cc3ccc(Br)cc3o2)=O)CCCC(S(=O)(=O)N2CCCC2)C1 C1(OCC(=O)NCC(CC)N(C)C(c2nc(Cl)oc2C)=O)CCCCCC1 N1(C(C2(C)N(C)CC(OC)C2)=O)CC2CCC(C1)N2C(c1ccoc1C)=O C1(CNC(CC=C(C)C)=O)CCN(C(=O)CCCCOc2ccccc2)C12CC2 Cc1cc(NC(=O)CCC2CCC(O)CC2)ccc1NC(=O)C(C)O C1(C(N(C2CCN(C(c3n(CC#C)ccc3)=O)C2)CC)=O)CC2(C1)CC2F c1(CNC(C2N(C(c3n[nH]c(C)c3C)=O)CCCC2)=O)ccc2c(c1)CCO2 C(=O)(CCCN(C)N=O)NC(CN(C(c1ccc(=O)n(C2CC2)c1)=O)CC)C C1(C(N(C)CC2CCN(C(c3snc(O)c3Cl)=O)C2)=O)CC2CCCC(C1)C2 C1(NC(CCOC)=O)C2CC3CN(C(=O)C(c4ccccc4F)C)C1C3C2 c1(C(NOC(C(=O)OC)C)=O)cncc(CNC(=O)C=CCF)c1 Cc1coc(C(=O)NC2(CO)CCN(C(c3coc(Cl)n3)=O)C2)c1C C1(NC(c2c(Cl)cc(C)s2)=O)CCN(C(=O)CCc2ccc[nH]2)C(C)C1 C1(C(=O)O)CN(C(c2ccc(F)c(Br)c2)=O)CC12CN(C(=O)CCCCCl)C2 C1(C(=O)NC2CC3C2CCN3C(c2ccccc2C(F)F)=O)Cc2nncn2C1 Cc1nc(SC(F)(F)F)sc1CC(=O)NCCNC(=O)CN(C)C c1(Cc2ncc(C(=O)NC3CC(N(C(CC=C)=O)C)C3)o2)ccc(Cl)cc1 C12(CNC(=O)C=Cc3cnc[nH]3)CC1CN(C(=O)CC1CSCCS1)C2 C1(C(=O)NCC(CC)C)CC2CCC(C1)N2C(=O)CCCC#N c1(CNc2c(C(=O)OCC)[nH]c3ccccc32)c(C)cc(C)c(C(C)=O)c1C c1(CNC(=O)NC2CN(c3n(C)nnn3)C2)cc2ncccc2s1 c1(NCC(C)Cc2cccc(O)c2)ccc(Br)cc1Cl c1(C(C)N(C(CC2(C)CCOC2)C(=O)NC2CC2)C)ccc2c(c1)OCO2 C1(C(N2CCC(CCN)C2)=O)Nc2ccccc2S(=O)(=O)N1 C12(CNC(c3cc(SC)oc3)=O)CC1CN(C(=O)C(C)Cn1ccnc1)C2 C1(C(CCC)NC(=O)CC(C)C)CCN(C(c2ccc(CO)o2)=O)CC1 C1(C(N(CC(C)NC(=O)C(C)(C)C2CCCO2)CC)=O)CCS(=O)CC1 Cc1nc(C2CC2)[nH]c1C(=O)NC(CNC(=O)Cc1cccnc1Cl)C1CCC1 N1(C(CC(COC)C)=O)CCOCC(C)(CNC(C2(CO)CCCCC2)=O)C1 c1(-c2nn(CC=CC)c(CCS(N)(=O)=O)n2)ccc(N2CCN(C)CC2)c(F)c1 n1(CC(=O)N(C2CCN(C(=O)CCCn3ccnc3C)C2)CCC)nnc(=O)[nH]1 N1(C(CC(C)NC(=O)C2CC2)=O)CCCC(C)(C)C1C(=O)OC(C)(C)C c1(C(CN(CCC(C(=O)OC)N)C)=O)ccc(C#N)cn1 c1(OC)cc(F)c2c(C(=O)N(CC(C)NC(=O)Cc3ccsc3C)C)n[nH]c2c1 C(=O)(CCC1=NNC(=O)CC1)NCCNC(CSc1n(C)cnn1)=O C(CCSC)(C(=O)N(CC(C)N(C)C(c1ccc(C(C)(F)F)cc1)=O)C)OC n1(C(C)C)ncc(C(=O)N(C)CC2CCCCN2C(=O)C(C)C2CCCC2)c1Cl c1(N2CCC(CNC(C(C)(C)c3ccccc3)=O)C23CC3)ncc2c(n1)COC2 c1(NC(COC)C)[nH]c(=NCC(C(C)C)N2CCN(C)CC2)nc2scnc12 c1(C(=O)NCC(CNC(CCCC#CC)=O)F)cc(C)c(C)cc1Cl N1(C(=O)CCCc2cc[nH]n2)CC2(CCN2C(c2ncccc2Cl)=O)C1 C1(C(C)C)CC(O)CN1C(=O)CC1CCC(NC(C2COCC2(C)C)=O)CC1 N1(C(COCCC=C)=O)CCC(CCCCNC(C2(C)CC2Br)=O)CC1 Cn1nnc2c1C(C(=O)NC(CNC(C13CCC(CC1)CO3)=O)C1CC1)CCC2 C1(N(C(CN(C2CCCCCC2)C)=O)C)CN(C(=O)C(O)C2CCC2)CC1(C)C c1(C(N2CCC(CNC(CCSCC(N)=O)=O)C2)=O)c(Cl)n[nH]c1C1CC1 C(N=c1nc2c(ncn2C(C)C)c(N2CCC(C3CC3)C2)[nH]1)c1cnc(C)o1 N1(CC2CC(CC)C2)CCOCCC1c1ccccc1 C1(C(N2C(CC)C(O)CC2)=O)N(C(C2CC(C)(O)C2)=O)CCCC1(C)C C1(C(N(CCCCCC)CCNC(=O)C(=O)NC(C)C)=O)CC(=O)N(C(C)C)C1 C1(CNC(C(CN(C)C)(C)C)=O)CN(C(c2nnsc2N)=O)CC12CC2 C(CCSC)(C(=O)NC(CNC(c1cc(C(C)(F)F)ccn1)=O)C1CCC1)OC C(=O)(C1=C(c2ccccc2)CCCC1)NC1C(C)CN(C(=O)CC2CC(F)C2)C1 CCC(CC(=O)N(CC(O)CN(C(=O)CCC1(C)CC1(F)F)C)C)C(F)F N1(C(C(CC)=CCCC)=O)CC(NC(C2CCCOC2)=O)CC(F)C1 Cc1ccc(CC(=O)NCCC(C)N(C)C(c2nnn(C)n2)=O)c(F)c1F CCC(C)C(O)C(=O)NC1CC(CO)N(C(C2CCCCN2C(=O)CC)=O)C1 C1(NC(C2COCCO2)=O)CCC12CN(C(=O)Cc1cccc(C(F)(F)F)c1)C2 c1(OC)ccc(C(O)C(=O)NCCCNC(=O)C(=O)N(C)C)cc1 c1(C(=O)NCC2(F)CC(NC(C(C)C#N)=O)C2)cc(C(F)(F)F)ncc1[N+](=O)[O-] N1(C(C(OCC)OCC)=O)CC=CC1(C)C(=O)NCCC(C)(C)CC N1(CCCOC(COC2(C#C)COC2)=O)C(=O)CNC1=O C1(NC(c2cc(F)cc(Cl)c2)=O)CC2CN(C(=O)CC3CCCCC3)CC12 c1(C(N2C(CNC(C3N(C(C)C)CCC3)=O)CC2)=O)ccc2cc(O)ccc2n1 N1(C(C(C)OCCCC)=O)CCC(CN(CCC=O)C)CC1.C(CCO)S(C)(=O)=O C1(C(=O)NC2(CNC(Cc3cnc(C)[nH]3)=O)CCC2)CC2CC1C1C2C1(F)F C1(C(=O)OC)N(C(c2cccc(OC(F)F)c2)=O)CC12CCC(F)(F)CC2 CC1CN2CCN1C(C(=O)NC1C=CCN(C(=O)Cc3ccccc3CO)C1)C2 C1(CC(C)NC(CCC=CC)=O)CCN(C(c2ccccc2SCC#N)=O)CC1 c1(C(N2CC(n3cc(CC(C(C)C)O)nn3)C2)=O)ccc(Cl)c(C2CC2)c1 CC(=O)CCCC(C)C(=O)NC1CC(CNC(C23CCC(CC2F)C3)=O)C1 Cc1cc(O)nc(C)c1C(=O)NCCCOCCNC(=O)C(C)(C)C Cc1cccc(CC(N2CCC(CNC(C3CN(C)C(=O)N3)=O)C2)=O)c1C C1(NC(c2cc(F)cc(F)c2)=O)C2CCC(C2)C1C(=O)NCCCC(O)CO c1(OC)cc(NC(N2CC(OC)C(C(=O)OC)C2)=O)c2c(c1)COC2 N1(C(C(N2CCC(C)CC2)=O)=O)CCC2C(CCCN2C(=O)CC23CC(C2)C3)C1 C(C(CC(=O)NCC(C)(Cn1cccn1)NC(c1cnc(Cl)s1)=O)C(F)F)OC C1(C2N(C(c3cc(CCC)[nH]n3)=O)CCC2)CCN(C(C2CNC(=O)N2)=O)CC1 C1(CC)CCN(C(c2nccnc2N)=O)C1CNC(C1CCC(C)(CC)O1)=O C=CCC(CC=NOCC(=O)NCCNC(=O)N(C)C)C(=O)OCC CCC(CC(=O)NCCOC1CCN(C(c2nn(C)cc2C(C)=O)=O)CC1)OC CCC(O)C(F)(F)C(=O)NCC(C)(C1CC1)NC(=O)CCC1CCCO1 C1(N(C)C(c2ccc(-c3ccco3)s2)=O)CCC(NC(C2COC2)=O)C1 c1(CC)cccc(C(N2CC=CC2(C)C(=O)NCCCN2CCCC2C)=O)c1 C1(NC(c2ccc(C(C)C)o2)=O)CN(C(c2cccc(O)c2Cl)=O)C(C)(C)C1 c1(OC)ccc(-c2nc(C3CC34CC4)nn2Cc2cccnc2)cc1OC N1(c2n(CCC3(OC)CC3)nnn2)CC2CCCC(C1)C2(F)F CCCC(C)(CCC)C(=O)N1CC(CNC(C2(CC#N)CCOC2)=O)CC(C)C1 C1(C)(C(=O)NCC2CN(C(c3n(CCOC)ncc3)=O)C(C)C2)COC(=O)OC1 c1(C(=O)NC(C2(O)CCN(C(=O)CC3CC(=O)C3)C2)C)cc2n(c1)CCC2 C(=O)(C(COC)CC(C)C)N(C(C)C(=O)NCc1csc(C)c1)CCC Cc1cc(CNC(C2CCCSC2)=O)oc1C(N1CC(N2CCCC2)C1)=O C1(CC)CCCCC1C(=O)NCCC1CCCN(C(C2CCCC2OC)=O)C1 c1(C(=O)NCCc2cnc(NC(c3ncn(CC)n3)=O)s2)cc(C)c(C)cc1Cl C1(C)(NC(c2cnc(CC)o2)=O)CCCCC1C(=O)NCc1conc1C1CC1 C1(CNC(CC)=O)CCCCCCN1C(=O)CC1CCSC1 C(=O)(C1(C)COc2ccccc21)NCC1CC(NC(CCC(C)OC)=O)C1 N1(C(CCC=C(C)C)C(=O)Nc2c(C)cccc2C)Cc2ccccc2CC1C N1(C(c2cc(F)c[nH]2)=O)CCN(C2CCN(C(C3CC34CC(O)C4)=O)CC2)CC1 C1(CNC(=O)OC(C)(C)C)CCC(C(=O)O)N(C(=O)CCSc2nnnn2C)C1 C1(OCC2CCCN2C(=O)OC(C)(C)C)COCC1CN(C)Cc1cnn(C)c1 C1(NC(C(CC)C#N)=O)CN(C(c2nccn3nccc23)=O)C2(CCOCC2)C1 Cc1cccc2c(C(=O)NC(C)(CNC(C3CC(C)N(C)C3)=O)CO)csc12 c1(C(=O)NCCN(C(=O)CSCc2cncn2C)CC)c[nH]c2c(Cl)cccc12 C1(OC)CC2CC(C(N3CCCC3CCNC(=O)C(C(C)C)C3CCC3)=O)CC12 C1(CC)(CO)CCN(C(=O)Cn2ccnc2C)C1.c12cncc(c1)CNC2=O CC1CCCC=C1C(=O)NCc1ccsc1C(=O)NCC1CC(=C2CC2)C1 c1(C(N2CC(CNC(C(COC)(C)OC)=O)OCC2)=O)cc2sc(C)cc2[nH]1 N1(C(C(C)N(C)C)=O)CCN(C(=O)C(C)(C)N2CCOCC2)CCC1C C1(F)(CNC(c2cccnc2-n2ccnn2)=O)CCCN(C(c2cnsc2)=O)C1 O=C1NC2C(=O)N1C2.c1(SCC(F)Cl)ccccc1-c1cccnc1 C(=O)(CC(F)(F)Cl)NCCN(CCC)C(c1csc(COC)n1)=O c1(CN2CC(S(C)(=O)=O)C2)nc2c(F)cccc2o1 N1(C(CC(C)N(C)C)=O)CCC(NC(=O)CCc2cncnc2)C(O)C1 c1(C(=O)NC2(CNC(=O)C(O)C(F)F)CCCCC2)cc2cccnn2c1 S(=O)(=O)(c1ccccc1NC(C1CC(OC)C12CCC2)=O)N(CC)CC CCCC(C(F)(F)F)NC(=O)CC1CCC(NC(=O)CCCCOC)CC1 N1(C(C(COCC)C)=O)CCOCC(NC(c2csc(S)n2)=O)C1 C(=O)(C(N)C(F)(F)C(F)(F)F)NC(C(=O)OC)(C)Cc1ccc(Cl)cc1 N1(C(C2CC(C)CC(C)C2)=O)CCN(C(C2(Cl)CC2)=O)CC2(CC2)C1 CC1OC(=O)NC1C(=O)NCCCCCCN(C(=O)CNS(N)(=O)=O)C N1(C(C(CC)OCC)=O)CCOC2(CCCN(C(=O)Cc3n[nH]c(=NC)s3)C2)C1 c1(CCCC)ccc(C(=O)NC2COC(C(C)C)C2)c(C)n1 C#CCCCCCCC(=O)N1CCCC1(C)C(N1CCC(O)(CO)C1)=O C1(CCC(c2ccc(C(=O)OC)o2)(C)CO)CC(C)(C)NC1=O C(C(CNC(=O)C(C)Sc1ccccn1)S(C)(=O)=O)NC(c1c(CC)nn[nH]1)=O c1(CC)ccc(Cl)c(C(N2CCOCC(NC(C3CCS(=O)(=O)N3)=O)C2)=O)c1 C1(NC(c2cc(CCC)[nH]n2)=O)CCCN(c2cc(C(F)(F)F)ncn2)C1 N1(C(c2c(C)nns2)=O)CCC(C(=O)NCc2nc(N(C)C)n[nH]2)(C(C)C)C1 c1(CC(=O)N(C2CCC(NC(=O)C(c3cccnc3)=O)C2)C)ccn(C(F)F)n1 C1(C(=O)Nc2cccnc2-c2ccccc2)COCCN(C(=O)C(F)(F)CO)C1 c1(CC(=O)NCCCN(C(c2c(C#N)cnn2C)=O)CC)ccc(F)c(F)c1 C1(C(=O)NC(C(=O)NCCOCCCC)CCC2CC2)CC(=O)NC(C)C1 C(=O)(C(C)P(C)(C)=O)NCCCN(C(C(c1ccc(C)o1)C)=O)CC1CCCC1 CON(CCC(=O)N1CCn2c(C)nnc2C1)C(=O)C1CC(=O)C12CCC2 c1(OCCCC(N2CC(NC(c3cscn3)=O)(CO)C2)=O)ccccc1Cl c1(C(=O)NCCC2CCCN2C(C2CC2C2CCC2)=O)ccc2cnccc2n1 N1(C(c2csnn2)=O)CCN(C(c2cnc(-c3ccccc3)s2)=O)CC(CO)C1 CCC(CC(C)C)C(=O)NC(C1CCCC1)CNC(c1cccc(Cl)c1F)=O C1(CN2C(c3cc(C(=O)OC)no3)CCCC2)CCCC2(CCC2)O1 n1(CC(=O)NCC(C(C)C)NC(=O)C(C2CCOCC2)F)cnc([N+](=O)[O-])n1 c1(C(N2CCC(N(C(c3c(C)cnn3C)=O)C)C2)=O)cc(N)nc(Br)c1 c1(C(=O)NCC2N(C)CCN(C(C34CCC3C4)=O)C2)cccc(C#CCO)c1 N(C(=NCCC(=O)N(C)C)NC1CC1c1c(F)cccc1F)CC1C(C)CCO1 C(=O)(C1=CS(=O)CCC1)NCC12C(CN(C(CNC(CNC(C)=O)=O)=O)C1)CC2 c1(NCCCNC(C(N=c2cc(C)o[nH]2)=O)=O)ccc(N=S(C)(C)=O)cc1 N1(C(CC2(CSC)CC2)=O)CCC(NC(=O)Cc2cocn2)CC1C1CC1 C(=O)(C(CC(=C)C)NC(C1CC1C(F)F)=O)NC(C1CCOC1)C#C CC1(C)CC(NC(=O)CCP(C)(C)=O)CN1C(c1cnc(C2CC2)nc1)=O CCC(F)C(=O)N1CCC(CCNC(=O)CCSC(F)(F)F)C1 N1(C(C(C)OC)=O)CCC2(CCC2)C(Nc2cc3nnc(C)n3cn2)C1 C1(C(N2CCC2c2cn(CCOC3CC3)nn2)=O)CC12CCOc1ccc(Cl)cc12.O=CO.N C1(C(=O)NC(Cn2cc(-c3c(OC)nccc3)nn2)C)CCCC12OCCO2 c1(CNC(c2nc(C3CCN(C(C)C)CC3)nn2C)C)ccc2c(c1)CC(C)O2 C1(CCC)CN(C(C2CCOCC2NC(c2cc(Cl)no2)=O)=O)CCO1 N1(C(c2scc(COC)c2)=O)CCC2CCN(C(=O)C3=CCS(=O)(=O)C3)CC12 C#CCCCCCCCCC(=O)NC1CC12CN(C(=O)CC(O)CCCCC)CC2 c1(C(N2CC3C(NC(C(C)N(C(C)=O)C)=O)(C3)C2)=O)cc(C#N)c(F)cc1F c1(OC)ncccc1C(=O)NC(CNC(=O)C(C)Oc1ccc(F)cc1)C(C)C C1(OC)CC(CCNC(=O)Cc2scnc2C)N(C(=O)CCSC)C1 C1(NC(C2CCC(NC(C)=O)CC2)=O)CN(C(c2ccoc2)=O)C2(CCOC2)C1 C1(C(=O)NCC(C)C(C)(C)C)(NC(C(COC)C)=O)CCc2cc(Br)ccc2C1 N1(C(C(CCCC)O)=O)CCC2C(C1)CN2C(C1CN(S(N)(=O)=O)C1)=O Cc1nn(C2CC2)cc1C(=O)NC1(C)CCN(C(c2coc(Cl)n2)=O)C1 C1(NC(C(c2cc(C)oc2C)C)=O)CCN(C(=O)C=Cc2cnc(C)s2)C(C)C1 C(=O)(CN=c1ccc(Cl)n[nH]1)N1CCN(C(CC(COC)C)=O)C(C(C)C)C1 c1(C(N(C(CNC(=O)CSCCC#N)C2CC2)C)=O)cnoc1-c1cccs1 C1(CCNC(CCN(CCC)C)=O)CCCCN1C(=O)C(C)OC1CCOC1 c1(OC)cc(C(=O)NC2CCN(C(=O)COC3CC3)CC2CO)cc(F)c1F.C(C)=O N1(C(C(OC)OC)=O)CC(CNC(=O)C2=COCC2)C(c2ccccc2)C1 c1(C(N(C(C)CNC(C2CN(C)C(=O)N2)=O)C)=O)cc2ccc(Cl)nc2s1 CC1CN(C(=O)CC2CCN(C(=O)CCc3nccs3)CC2)CC(=O)N1C CCC(CC(=O)N1CCC(C)(CNC(C2CC(=O)OC2(C)C)=O)C1)C(C)C c1(CC)ncc(C(=O)N(CCC(=O)NCCCC(=C)C)C2CC2)cn1 n1(CCC(=O)NC2CC(NC(C3CC4CCCC4C3)=O)C2)ccc2ccccc12 N1(C(C)C)C(=O)COCC1C(N1CCCC1CNC(c1cc(N)ccc1F)=O)=O c1(C(N2CCC3CN(C(=O)C(F)(F)C4CC4)CC23)=O)cncc2cc(Cl)ccc12 C(CN(C)C(C1COC(C(=O)OC(C)(C)C)C1)=O)(C(=O)OC)OC1CN(C(C)=O)C1 CCC(CO)C(=O)N(C(=O)C(N1CCCC(C)C1)=O)C(C)COc1ccccc1 c1(C(N2C(CCNC(C3C(=C)C3)=O)CC(F)(F)C2)=O)cc2cc(Cl)ncc2[nH]1 C(=O)(C(C)CC(F)F)N1CC(CCC(=O)NC2(C(=O)OC)CCCC2)OCC1 N1(CC(=O)NC(C2N(C(CN(C3CCC3)C)=O)CCC2)(C)C)CCS(=O)CC1 N1(C(C(C(C)C)(C)C)=O)CCC2CC(NC(=O)CSc3ccccc3)CCC2C1 N1(C(C2(O)CCN(c3ccnc4ccnn34)C2)=O)CCN2CCCC2C1 C#CCCC(O)C(=O)NCc1nc(CNC(C2CC3CC2CC3O)=O)cc(O)n1 N1(C(CSCCCC)=O)CCN(C(=O)Cc2cc[nH]c2)C(C2CCC2)C1 C1(C(N2CC(C3CC3)(C(=O)NCCCCCCF)C2)=O)CCC(C2CC2)C1 Cc1cc(=O)n(C)cc1C(=O)NC1CCN(C(=O)CC2CCCC2)C1C c1(OC)cnncc1C(=O)NC1CC(CNC(c2ccc(C(F)F)cc2)=O)C1 N1(C(=O)OC(C)(C)C)CCC1C=CC(=O)NC1CC(CCC(=O)O)C1 CC1CCOCC1C(=O)NCCCCN(C(=O)CN1CCC(C(F)(F)F)CC1)C c1(C(=O)NC(CC(C)C)CNC(=O)Cn2cccc2)cccc2cc(O)ncc12 C1(NC(=O)NC(c2ccc(C)cn2)CC)CN(Cc2ccccc2)CC1O c1(CCC)ccc(CCCC(=O)NCC2CC2CNC(=O)CCSC2CC2)cc1 C1(C(=O)NC2CC(NC(CC(=C=C)C)=O)C2)CC12CCC1(CC1)CC2 c1(CC)ccc(C(N2CCC(CO)(NC(C3CC4OC3C3CC43)=O)C2)=O)c(Cl)c1 C1(CC(C)C)C(=O)N1.C1(O)(CC#C)CC(C(N2CC(O)(C(F)(F)F)C2)=O)C1 C12(C(N(CC(C)NC(C3ON=C(C)C3)=O)C)=O)CCCC1CCC2 c1(C(=O)NC2CCN(C(Cn3c(C)cc(C)n3)=O)C2C)cc(S(N)(=O)=O)c(C)o1 N#Cc1cc(CNc2ccccc2C(N2CC(O)CC2C(N)=O)=O)cc(F)c1 c1(C(=O)NCC2OCCN(C(C(CC)F)=O)C2)cc(OC)cc(OC)n1 N1(C(c2nn(C)c(C(N)=O)c2)=O)CCC2(CO)CN(C(=O)C=CCF)CC2C1 CCC(C(=O)NC(C)CC1CN(C(c2ccc(C(=O)CF)cc2)=O)C1)C(C)(F)F c1(-c2ccc(C(N3CCC(NC(=O)Cc4ccncc4)C3)=O)o2)ccccc1F c1(C(N(C2CCN(C(CCC#C)=O)CC2)CCO)=O)cccc2nccnc12 c1(C(N(C2CCN(C(=O)CC3OCCO3)C2)CC)=O)c(F)cccc1F c1(CC)cc(OC)ccc1C(N1CCN(C(=O)C(C)SC)C(CC)C1)=O n1(CC)cc(CC(N2CCC2CC(=O)NC2(C(C)C)CCC2)=O)cn1 N1(C(C(COC)O)=O)CC2(Cn3cc(CSc4nccn4CC)nn3)CC1CCO2 C(CCN(C(=O)CC1CCCCCC1)C)(C(C)(C)C)NC(c1c(C)cncc1)=O C(CCC(O)C(=O)N1CCOC(C#N)C1)NC(c1nc(C)oc1C)=O C1(NC(C(C)(C)NC(=O)CC2CC(=O)C2)=O)CCC(=O)NC1(C)C C1(NC(CCC(=C)Cl)=O)CN(C(c2ccccc2C(F)(F)F)=O)CC(C)(C)C1 C12(CNC(=O)CCc3ncc(F)cn3)CCCCC1C2(F)F CCC(CN(C)C)CC(=O)N1CCC1CNC(C1(CCOC)CCC1)=O C1(CC(=O)NC2CC(O)(CNC(C3CCCC(C)C3)=O)C2)CCS(=O)(=O)CC1 N1(C(C(CCC)C(=O)O)=O)CCOC2(CCN(C(=O)CSCCC#N)CC2)C1 Cc1cccnc1C(N1CCC1(C)CC(=O)NCC(O)CCC1CC1)=O C1(NC(CCc2cncc(OC)c2)=O)CN(C(=O)CC(C)(C)F)CC12CCC2 c1(N(CC(=O)NCC2N(C(C(C=C=C)C)=O)CCCC2)C)nc2ccccc2s1 c1(C(=O)NCC23N(C(CC(CC)C)=O)CC(CCC2)C3)noc2c(F)cccc12 C1(NC(CC=CC)=O)CC2CC(C1)N(C(=O)COc1ccc(C(=O)NC)cc1)C2 c1(-n2c(CC3CCC(=O)NC3)nc(-c3ccccn3)n2)ccc(F)cc1F CC1CCN(C(c2csc(Cl)c2)=O)C(C(=O)N(C)CCN2CCCCC2)C1 C1(NC(CCOC(C)C)=O)CCN(C(c2ccc(CO)nc2)=O)CC(O)C1 c1(C(=O)NCCOCCN(C(C2CCC(C)O2)=O)C)cccc(CN(C)C)c1 CC(CC(C)(C)C)C(=O)NC1CN(C(c2cnc3ccccn23)=O)CC1C(F)F c1(Oc2c(I)cccc2)ncnc2n[nH]cc12 CCC(CNC(=O)C(C1CCN(C(=O)CC2CC=CCC2)C1)C)(CC)C N1(C(C(C)=C2CC2)=O)CCC2CN(C(=O)CSc3ccc(Cl)c(Cl)c3)CC2C1 CCCCCCCCOCC(=O)NC(CNC(C1CCCC1)=O)C1CCC1 C(CCC)(C(O)C(=O)NCc1cccnc1C)NC(C(C)OCCC=C)=O Cc1occc(=O)c1OCC(=O)NCC1(F)CCN(C(c2cnsn2)=O)C1 C1(N(C(CCC=C)=O)C)CN(C(c2nn(C)cc2C(C)=O)=O)CCC1O c1(C(N2CCC(O)(C(C)NC(C3CN(C)C3)=O)C2)=O)c[nH]c2cnccc12 c1(C(N(C(CCNC(C(C)NC(COC)=O)=O)C)C)=O)cc2cc(F)ccc2o1 c1(CC)nc(C(=O)NCCCNC(=O)COCC2CCCO2)cs1 Cc1nnccc1C(N1CCCC1(C)CNC(c1sccc1SC(F)F)=O)=O C(CC(C)C(=O)NCC(C)C(=O)N(CC)Cc1ncnn1C1CC1)=CCC c1(C(=O)NCC(C(=O)NCC2(CO)CCC2)OCC)ccc(Cl)c(O)c1 C1(C(=O)NC2CN(CCC)C2)C2CC3C(C2NC(=O)C(C)(CC)OCC)C13 c1(C(N(CC(O)CN(C)C(C2CCC(F)(F)C2)=O)C)=O)cc2n(n1)CCO2 C1(C(=O)NC(C2CCCC2)CNC(c2ccnnc2)=O)(OC)CCC(C)(C)C1 C1(CCC)CC(NCCc2cccc(F)c2)CCO1 C(=O)(CCCCCCCC1CC1)NCC1C(C)CCCN1C(=O)CC1=CCCC1 c1(C(N2CC3C(NC(c4ccc(C=C)cc4)=O)(C3)C2)=O)cc2cc(Cl)sc2[nH]1 C1(NC(c2n(CCN(C)C)ncc2)=O)CN(C(c2cc[nH]c2)=O)CCC12CCC2 c1(SC)ncc(C(=O)NC2CC2NC(c2nnn(C)n2)=O)n1-c1ccc(F)cc1 c1(OC)cc(C(CC(=O)O)N(C)CCC2CC2)ccc1NC(=O)NOCCO c1(OC)cccc(CC(=O)NCCC2CSCCN2C(=O)C(C#N)CC)c1 c1(COC(c2c(C(C)C)cccc2)=O)ccc2c(c1)CCCN2C C1(C(=O)NC2CCN(C(c3c(C)cc(C)[nH]3)=O)CC2C)CCc2nccn2C1 N1(C(C2(CCC)CC2)=O)CCOC(CNC(=O)C(c2cccnc2)O)C1 c1(OC)cc(C(O)C(=O)N2CC(NC(=O)CC(C)F)C2)c(F)cc1O c1(C(=O)NC(CNC(CCC=CCC=C)=O)C2CC2)nc(C(F)(F)F)ccc1F C(CC(=O)O)(CC(C)C)N(C(c1ccccn1)CC)CC C(CC(C(C)C)NC(=O)CN1CCCCC1=O)NC(C(CC)c1cccnc1)=O N1(c2nnc(CCC(C(C)C)NC(=O)CCC(F)(F)F)s2)CCc2ccccc21 c1(C(N(CCNC(c2scc(C(C)=O)n2)=O)C)=O)nc2c(s1)CCCC2 c1(CN2CCCC(C(N(C(C)C)C)=O)C2)cccc2ccncc12 c1(CC(N2CC(F)(CNC(CC3C(CC)C3)=O)C2)=O)c[nH]c2c(F)cccc12 C1(CCNC(C2(CC)CC2(F)F)=O)CCCN(C(=O)C(C)(C)c2ccsc2)C1 CC(CC(N)=O)C(=O)NCCCN(C(=O)CSc1nc[nH]n1)C C(=O)(C1CCCn2cnnc21)N1CC2(CCN(CCCCCOC)CC2)C1 C1(NC(c2c(C)sc(Br)c2)=O)CC(C)CN(C(c2nonc2N)=O)C1 C#CC(C)(C)C(=O)NC1CCOC(CNC(=O)CC2C(C)(C)C2(C)C)C1 c1(C(=O)NC2CN(C(Cc3ccc(C)cc3)=O)CC2C#N)cccc2ccnn12 C1(CCN)(NC(=O)NCC2(CCO)CCOC2)CCOC1 C1(C(=O)OC)C(Nc2nc3ccc(OC(C)C)nc3s2)C2CCCCCCC12 c1(C(=O)OC)cc(F)c(C)cc1NC(N1CCOC2CC12)=O N1(C(C(C(C)C)N(C)CC)=O)CC2CCCC(C1)N2C(=O)C(C(C)C)NC(N)=O C1(CC(N2CC(C(N)=O)(OC)C2)=O)CCN(C(=O)Cc2cc[nH]c2)C1(C)C C(=O)(C(C(C)C)c1ccc(C)cc1)N(CCN(C(CNC(=O)NC)=O)C)C1CC1 Cc1cccc(C(N2CCN(C(C3CC3(F)F)=O)C(C3CC3)C2)=O)c1C(F)(F)F c1(OC)ccc(Cl)c(C(N2CCCC2CNC(=O)CCSc2nccn2C)=O)n1 C1(NC(C(c2ccn(C)n2)C)=O)CCCCCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 C1(NC(=O)CCc2cnc[nH]2)CCC2(CCN(C(=O)C(C3CCCCC3)F)C2)C1 n1(C(CC)C)ccc(=NC(=O)CCNC(=O)C(CCSC)OC)[nH]1 c1(C(N(CC(C2CCCCC2)OC)C)=O)ccc2c(n1)CCC(C)(C)C2 c1(CC(C(=O)NCC(C)NC(C2(CC)CC(C)(C)C2)=O)C#N)ccc(C#N)cc1 C12(NC(c3n(C)ccn3)=O)CC(C1)N(C(=O)C(C)(C)c1ccno1)C2 C1(=O)C(CC(C)C)ONC(=O)C(C)(C)N1.C(=O)(CCCc1cncs1)NC c1(CC)cc(F)c(C(N2CC3C(CNC(=O)C(C)C(O)CC)C3C2)=O)cc1F C1(CNC(C2N(C)C(=O)OC2)=O)CCCCN(C(=O)C(F)(F)c2csc(=N)[nH]2)C1 CC1CCN(C(c2scnc2C(F)(F)F)=O)CC1NC(c1cc(C(N)=O)[nH]n1)=O N1(C(c2nc(C)[nH]n2)=O)CC2(CNC(=O)Cc3csc(C4CC4)n3)CC1CO2 N1(C(CCCCSC)=O)CCC(CNC(c2cnc(C(C)C)s2)=O)C(C)C1 c1(CN2CC(C(=O)Nc3c(C(=O)OCC)n[nH]c3)C2)cc2ccoc2cn1 C(=O)(C(O)C(C)(C)C)N1CC(O)(C(CNC(C(C)C(F)F)=O)(C)C)C1 c1(C(CC)C(=O)N(CCCNC(=O)Cn2nccn2)C)c(C)noc1C c1(C(N(C2CC(C(N(C)CC3(O)CCC3)=O)C2)C)=O)cnn2ccccc12 Cn1cc2ccc(CN3CCC(C(=O)Nc4ccc(C#N)s4)C(O)C3)cc2n1 Cc1cccc(O)c1C(=O)NC(C)CCCCNC(C1CC(=O)N(C)C1)=O c1(C(=O)NC2CCC(NC(c3n[nH]cc3Cl)=O)CC2)cc2n(n1)CCCCC2=O N1(C(c2cn(CC)nc2)=O)CCC(C)(C)C1C(=O)NC(CO)C1(C)CC1 N1(C(n2nccc2C2CC2)=O)CC2CC2(C(=O)NCC(c2ccc(O)nc2)O)C1 C1(N(C(C(CC)F)=O)CC)CCN(C(C2(CC)CCOCC2)=O)CC1 CC(C(=O)NC1CCN(C(C2CC(OC(C)(C)C)C2)=O)CC1)C(C)(F)F C1(NC(C2(NC(c3c(C)cc[nH]3)=O)CC2)=O)CC1C1CCCC1 c1(OC)ccc(Cl)c(-c2ccc(C(=O)N(Cc3ccccc3Cl)OC)o2)c1 C(=O)(CCCC(C)(C)C(=O)OC)NC(CC=C)CNC(c1ccc(SC)cc1)=O S(=O)(=O)(c1cnc(Nc2ccccc2OC2CCNCC2)s1)N(C)C N1(C(C(C=C)O)=O)CCC(n2cc(NCc3cn(C)nc3C)cn2)CC1 N1(C(C=CC(=O)N(C)C)=O)CCC(C(=O)NC2(C(N)=O)CCC2)C1 CCCCCCC(=O)NC1CN(C(=O)CCCN(C)C(=O)OC)CC1OC N1(C(CC2CC(N(C)C)C2)=O)CC2(C1)CN(C(C1(C(N)=O)CCC1)=O)CC2CO c1(NC(CNC(c2c(C)cc(CC)o2)=O)C2CC2)cnc(C#N)cn1 c1(OC)ncc(C(=O)NC2CC(NC(C3C(C(F)F)C3(C)C)=O)C2)nc1C c1(C(=O)NC2(C)CCN(C(C(CCCC)=O)=O)C2)cnn2cc(OC)ccc12 N1(C(Cn2ccc(C(=O)OC)n2)=O)CC2(CCN(C(C3(C)CCOC3)=O)C2)C1 N1(CC)CCCCC1C(N1CC(OC)C(C(=O)NC(C)(C)CO)C1)=O S(=O)(=O)(c1cc(C)sc1C)N1C(CSc2n(-c3cccc(CC)c3)nnn2)CC1 C#CCCCC(C(=O)Nc1ccccc1Br)N1CC=C(CO)CC1 Cc1cc2[nH]c(C(=O)NC(CNC(c3coc(C#N)c3)=O)C(C)(C)C)cc2o1 C1(C(=O)NCCOCCNC(COCC)=O)Cc2ccc(F)cc2C(=O)O1 c1(C(=O)NC2CCN(C(c3c(C)ncc(Br)c3)=O)C2)cc(F)cc(Cl)c1N CC1(C)CCN(C(=O)C(c2cccnc2)N2CCCC2)c2ccccc21 C(=O)(C(C)C(F)(F)F)N1CCC(C)(NC(c2ccc(OC)s2)=O)C1 C1(C(N(CCNC(=O)C(CSC)OC)CC)=O)CCCCC(F)(F)C1 CC(C)CC(F)C(=O)NCC(C(C)C)NC(c1[nH]nnc1C1CC1)=O C(CCCC(=O)N1CCC(C2CCCN2C(c2coc(C(F)F)n2)=O)CC1)SC N1(C(Cc2cc(OC)no2)=O)CCC2C(CCN2C(C2CCCN(C)C2)=O)C1 C(C(C)(C(=O)NCc1ccc(C)o1)NC(=O)CCN(C)C)SC c1(C(=O)NCC2CN(C(=O)C(F)=CCCF)CCCO2)ccc2occc2c1 N1(CC(c2ccccn2)N)CCOC(C(N2CCNCC2)=O)C1 C1(CNC(C(C)CF)=O)CC2(CC2)CN1C(=O)CC1(O)CCCCC1 C(=O)(CCCOC(C)C)N(CC(=O)NCC(C)OCC)C1CC1 CC1CCNCCC1N(CCCCCN1CCOCC1)C(c1ccc(I)cc1Cl)=O c1(OCC(=O)NCC(CC)NC(=O)CSc2cncn2C)ccncc1 C1(CNC(C(CC)N(CC)CC)=O)CN(C(=O)C=Cc2scnc2C)CC1C C(=O)(C(F)C1=CCCCC1)OCC1C(C)CCCN1C(=O)OC(C)(C)C N1(C(c2ccc(N)cc2Cl)=O)CC(NC(=O)CC(=O)NCC(F)F)CCC(O)C1 C1(C(=O)NCC(CN(C(=O)CC2(O)CCC2)C)(C)C)CC(=O)C1C(C)(C)C CC(C)CC(F)(F)C(=O)N1CCC2(CC1)CC2Nc1nccc(OC(C)C)n1 CC1CCN(C(c2cccc(N)c2)=O)CC1NC(c1ccc(C(C)(C)C)s1)=O Cc1cc2[nH]c(C(N3CC(C)N(C(=O)C=Cc4ccccn4)CC3C)=O)cc2o1 S(=O)(=O)(c1ccc(C)cc1Cl)N(S(CC(=O)OCC)(=O)=O)CCC1CCCNC1 N1(C(c2cnc(C(C)(C)C)nc2)C(=O)NCCC#N)CCc2nc(=N)[nH]cc2C1 c1(NCC2(CNC(C(CC)(C)OC)=O)CCC2)ncnc2sc(C)nc12 c1(C(=O)NC2(CN(C(c3c(C)nccc3)=O)C)CC2)cc2c(F)ccc(F)c2[nH]1 c1(C(N(CCCNC(=O)CCOc2cccnc2)CC)=O)ncncc1C c1(C(=O)NC2CCC(F)(CNC(CCC(C)OC)=O)C2)[nH]c(C)c([N+](=O)[O-])c1C c1(C(=O)NC2CC(NC(C(C)(C)F)=O)C23CCC3)cncc(S(C)(=O)=O)c1 Cc1ccccc1CC(N1CCC(C)(C(=O)NCCn2cccc2C=O)C1)C CC1CN(C(C2CN(C(c3cnccn3)=O)CC2(C)C)=O)C(C)C1C c1(C(=O)NCC2N(C(CNC(CC)=O)=O)CCCC2)c(C)ccc2ncccc12 CC(c1cccc(Cl)c1)=CC(=O)NCCNC(C1CNC(=O)CC1C(F)(F)F)=O c1(C(N(CCNC(C2CCC(C)S2)=O)C)=O)cnc2c(N)cccc2c1 c1(C(N2CCC(c3nncs3)C2)C(=O)NCCSC)nc(C)c(Br)s1 CC1CN(C(=O)CC2COCC(C)(C)O2)CCCN1C(=O)CC1(O)CCCCC1 Cc1cnc2cccc(C(=O)NC3CCCC3CNC(=O)C=CBr)n12 C(C(=O)N1CCC(NC(c2ccc(C)cn2)=O)C1C)(C(C)C)NC(C)=O C(=O)(C(C)CC(F)(F)F)N(CCCNC(C(C=C)(F)F)=O)CC1CCCC1 c1(C(N2CCCCCC2CNC(C2(C3CC3)CC=CC2)=O)=O)cn2cnnc2cn1 C1(CNC(CCNS(CC)(=O)=O)=O)CN(C(c2ccsn2)=O)CC(C)(C)C1 N1(C(C(C(CC)CC)C)=O)CCC2(CCN(C(c3ccccc3C(C)C)=O)C2)C1 n1(CC(=O)NCCC2(O)CCN(C(CC3C(C)C3)=O)CC2)cc2ncccc2n1 Cc1ccc(CNC2(c3ncccc3C)CC2)c([N+](=O)[O-])c1.N12CCCC1C2=O c1(C(N2C(C)CC(NC(c3c(CC)nco3)=O)C2)=O)cc(N)ccc1O Cc1c(C(N2CCOCC(C(=O)Nc3ccccc3O)C2)=O)cccc1Br c1(NCCNS(CC)(=O)=O)[nH]c(=NCC#Cc2cnn(C)c2)nc2ncn(C)c12 c1(N(C)C)cccc(CNC(=O)NCC(c2ccc(Br)c(F)c2)(C)O)c1F c1(OC)cc(N)c(Cl)cc1C(=O)NCC1CCN(C(C2CNC(=O)N2)=O)C1(C)C c1(C(=O)NCC2(COC)CN(C(C3CCCOCC3)=O)C2)ccc2nn[nH]c2c1 N1(C(C2C(C(C)C)C2)=O)CCC(CCO)C1.c1(N2CC2=O)sccc1C(N)=O c1(C(N2C(CNC(c3snc(C(C)(C)C)n3)=O)CC2)=O)ccc2oc(O)nc2c1 N1(C(CCCCC#N)=O)CC(NC(=O)Cc2cnccc2Cl)CC2(CC2)C1 C1(CN(C(=O)CN2CC3CC3C2)C)CCCN(C(c2ccnn2C2CCC2)=O)C1 c1(C(=O)Nc2ccc(C)o2)nn2ccccc2c1C(=O)NCCN(CCO)CCO CC1C(NC(=O)C(c2cccc(F)c2)O)CCCN1C(c1cnc(O)nc1O)=O N(C(=NCCCOC)N1CCN(CC2CCOC2)CC1)CCC(=C)C c1(C(=O)NCC2CN(C(c3cc(SC)c(C)o3)=O)C2)c(C)nn(C)c1N Cc1sc2ccccc2c1C(=O)NC1CN(C(=O)CC2CCOC2(C)C)CC1C c1(CC)ccc(C)cc1C(=O)N(CC(O)CNC(c1cc(N)cc(F)c1)=O)C N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CCC2CCN(C(=O)CC(O)C(C)C)C2C1 Cc1nccnc1C(=O)NOC1CN(C(C2CC3CCC3C2)=O)CC1C c1(OCC(=O)NC2CCCN(C(CCC)=O)C2)ccc([N+](=O)[O-])cc1 C1(C(F)(F)F)(C(=O)NC(C(C)NC(c2cc(C3CCC3)[nH]n2)=O)C)CCN(C)C1 c1(NC)ccc(F)cc1C(=O)NCC(C1CCCC1)NC(=O)CN1CCC1C c1(COCC)nccc(N2CCN(C3CCN(C(=O)CC4(CO)CC4)C3)CC2)n1 C(=O)(C1CCCn2ccnc21)C1CN(C(=O)C(O)CCCc2ccccc2)C1 CCCC(C(=O)NCCCCC(C)NC(=O)CCc1ccc(O)cc1)N(C)C n1(CC(=O)NC2CCC(NC(c3ccccc3)=O)CC2)cccnc1=O C1(C(=O)NCC2CN(C(C3(CO)COC3)=O)C2)CC(=O)N(O)C1 C1(C(=O)NC2(CNC(c3c(C)ncs3)=O)CCOC2)CCCN(C(C)C)C1 C1(NC(C2(N(C)C)CCC2)=O)CCCCN(C(=O)C(c2ccc(N)cc2)(C)C)C1 N1(C(c2ccc(NC(C)=O)s2)=O)CCOC2CN(C(=O)C(O)CC(C)(C)C)CC12 N1(CC)CCN(C(C2CCC3CCC2N3C(C23CCC(C2)C3)=O)=O)CC1(C)C Brc1c(SCCC2CCCO2)n[nH]c1-c1ccccc1 c1(C(N2CCCC2Cn2cc(COC3COC3)nn2)=O)cc(Br)n2ccccc12 N1(C(CN(C(=O)CCn2cccn2)C2CCC2)=O)CCC2CCCCC12 C=CCC(CC(=O)N1CCCN(C(C)C)CC1)NC(=O)C(C)CC c1(OC)cccc2c1CCC(NC(c1nnnn1-c1ccc(F)cc1)C(C)C)C2 CC1(C)CCCc2ccccc21.c1(N)nc(C2CCCNC2)cs1 c1(NC(C2CN(CCSCc3cccnc3)CCN2)=O)nc(C(F)(F)F)ccc1Cl C(=O)(C(CC(C)C)N(C)C)NC(CN(C(C12CC(CO1)C2)=O)CC)C C(CC(C)(C)C)(C(=O)N1CCN(CC(C)O)CC1)NC(c1c(C)cn(C)n1)=O C1(F)(CNC(C=CC=CCC)=O)CCN(C(=O)CC(=O)NCC)CC1 C1(NC(C2CCC(CC)O2)=O)CCN(C(C2(CN(C)C)CC2)=O)CC1C c1(NC(N2CCC(NC(=O)CCCC3CC3)C2)=O)cccc(Cl)c1F C(=O)(CCC1CC(OC(N2C(CN(C)C)CC2)=O)C1)OC(C)(C)C c1(C(=O)NCC23N(C(COCC)=O)CCC2CC3)ccc(S(=O)(=O)NC)c(F)c1 c1(CC)nn(C)cc1CNC(=O)NCC(C)(C)C(C)O C(N=c1[nH]c(=NCc2ccc3c[nH]nc3c2)[nH]c2ccsc12)C1C(C)CCCC1 N1(C(C2(C(=O)OC)CC2)=O)CCC(C2CC2)(NC(=O)COc2ccccc2Cl)C1 C1(NC(=O)CCc2cncs2)CN(C(c2conc2C2CCCC2)=O)CCC1F C(=O)(CCC(=O)NCC1CC(CNC(=O)C(C)(C)CO)C1)N(CCC)CCC c1(OC)cccc(C(N2CC(O)(C(F)C(=O)NC(C)(CO)C3CC3)C2)=O)c1 c1(C(=O)NCC(CC)(O)CC)c(C)c(C)nn1C c1(CC)c(C(=O)NC(C2CCCC2)CNC(=O)C(Cl)=CCl)cnn1C(CC)CC N1(c2n(CC)c(Cc3csc(C)n3)nn2)CC(=O)NCC2(COC2)C1 c1(C(N2CC(F)CC(C(=O)Nc3cnsc3)C2)=O)cc(O)cc([N+](=O)[O-])c1 C(=O)(C(C)(C)CC(=O)NC(C)(CNC(C12CC(CO1)C2)=O)CC(C)C)OCC c1(C(N2C3(CNC(=O)CCC4CCCO4)CC(C2)C3)=O)cc(O)c(O)c(O)c1 CC1C(C)N(C(=O)COc2cccc(C#N)c2)CCN1C(c1cnccn1)=O C=CCC(CCCCC)C(=O)NCCC(C)CCNC(c1[nH]c(C)nc1C)=O c1(CC(N2CCC(NC(CCSC)=O)C2c2ccccc2)=O)ccc(C#N)cc1 C=CCC(C(=O)N1CCC(CO)(CNC(=O)C=CCCC=C(C)C)C1)C(C)C CC(C)C(C)C(CNC(=O)C(F)C(C)(C)O)NC(=O)CN1CCC(CO)CC1 c1(OC)cc(SC)ccc1C(=O)NC(C1COCCN1C(=O)CC1CC=CC1)C C1(C(C)NC(=O)C2CC2)CC(O)C(O)CC1CCCOc1c(C)cc(OC(F)F)cc1 O=C(CCC(F)(F)Cn1cc(CCCO)nn1)NCCc1cc(Br)no1 c1(C(C2CCCC(O)C2)NC(c2snc(C)n2)=O)ccc(F)cc1F C1(C(=O)NCC(C)(C)SC)CC(NC(c2c[nH]c(C)c2)=O)C1(C)C c1(C(N2C(CNC(C3N(S(CC)(=O)=O)CCC3)=O)CCC2)=O)c(C)nsc1C C1(NC(c2cc(CCC)c(C)s2)=O)COCCN(C(c2ocnc2C(F)F)=O)C1 N1(C(C(C)OC)=O)CC(C(=O)N(C)CCn2cc(C)cn2)C(F)(F)C1 c1(C(N(CCNC(CC2(C)CC2(F)Cl)=O)C2CC2)=O)ccc(F)c(OC(F)(F)F)c1 c1(C(=O)NC2CCN(C(C(C)Oc3ccccc3F)=O)C2)cc(O)cc(=O)o1 C(=O)(C#CC1(C)COC1)NC1CCCN(C(c2c(C)con2)=O)C1 C(=O)(CC(C)(C)c1ccccc1)NC(CNC(c1c(C)con1)=O)(C)C1CCC1 N1(C(C(CC)C(C)C)=O)CCN(C(=O)C(c2cccc(OC)c2)C)CC2(CC2)C1 C12(C(=O)NC(C(=O)OC)CO)CC(CN(C(C3CCCS3)=O)C1)C2 c1(NC(C2CCCN2C(=O)CNCc2cc(B(O)O)co2)=O)cc(Cl)c(Cl)cc1Br C(=O)(C1=C(C)OCCS1)NC1CC(NC(C(C)OC)=O)C1 C(=O)(C(CO)C(F)(F)F)NCC(CC)N(C)C(C1CCC2(CCC2)CO1)=O C1(CC(=O)NCC(C(C)C)NC(c2ccsc2-n2cnnn2)=O)CCC(C)CO1 N1(C(CC(C)(C)N(C)C)=O)CC(CNC(C2CC3CC(=O)C2C3)=O)C(F)(F)C1 c1(C(N2CC(NC(COCC(=O)OC)=O)C(C)C2)=O)ccc2nc(C)nc(O)c2c1 c1(CC(N2C(CN(C(CCCOC)=O)C)CCC2)=O)ccc2nonc2c1 c1(SC)cc(C)c(C(=O)NCC2(F)CCN(C(c3c[nH]nc3C3CC3)=O)C2)o1 N1(C(C=CC(CC)C)=O)CC(=O)CC1C(=O)NCC(C)(O)CCOC c1(Cc2onc(-c3cc(C)sn3)n2)cc(Cl)c(Cl)nc1C CCCC(C)(CC)C(=O)NC1(CCNC(c2cnnc(O)c2)=O)CCC1 c1(CC)c(C(N2CCC(C)(CNC(C3CC4(CC4)CO3)=O)C2)=O)nnn1C N1(C(c2ccc(OCC)nc2)=O)CC(NC(C2CCOC(=O)CC2)=O)CC(F)C1 C(C(C(C)(C)C)NC(=O)C(c1ccc(Cl)cc1)N(C)C)NC(c1c(C)ocn1)=O CC(C)C(CNC(=O)CNS(C)(=O)=O)NC(c1ncc(C(F)F)s1)=O c1(OC)cc(=O)n(C)cc1C(=O)NCC1=CCN(C(C2(C)CCC(=O)C2)=O)CC1 C(CC(=O)NC1CCS(=O)CC1)(C(F)F)NC(c1cn(C2CC2)nn1)=O C12(NC(c3cc(C)ncc3)=O)CCCN(c3cc(C(C)C)nc(C(C)C)n3)CC1C2 C(=O)(CC(C)CC(C)(C)C)N(CCNC(=O)CC1CC=CCN1C)CC c1(NC(CCc2c(N=[N+]=[N-])cccc2)=O)ccc(O)c2ncccc12 c1(C(=O)NCCCN(C(CS(CC)(=O)=O)=O)C)ccn(C(=O)OC(C)(C)C)n1 CC(CC(=O)N1CCCC(N(C(=O)CSc2cccs2)CCF)C1)CC(F)(F)F C1(O)(CC(N2C(C)CC(CNC(Cc3scc(C)c3)=O)C2)=O)CCCCCC1 C(CC(C)(C)C)(C(=O)NCC(O)C(F)F)NC(CCCOCC)=O c1(C(CNC(c2occ(C)c2C)=O)NC(=O)C(Cl)=CCl)ccc2ccccc2c1 c1(C(C)C)ccc(C(=O)NC2C(CNC(=O)C=CCF)CCC23CCC3)c(F)c1 c1(C(=O)NC(CNC(c2cc(C)nnc2)=O)CC(C)C)cccc2c1ccn2C c1(C(=O)NC2CN(C(c3c(Cl)cn(CCC)n3)=O)CC2O)ccn2nncc2c1 C1(C(N2CC(CCCC)N(C(C34CC(C3)C4)=O)CC2)=O)CC2CSCC(C1)C2 C1(c2c(OC)cccc2)CC2(CCCC2)CN1Cc1cc(F)c(F)c(F)c1 CCC(CNC(=O)C(C)=CCNC(=O)CC1CCOC1C)(CC)CO c1(CN(C(C(C(=O)OC)CC)=O)C)cc(OC)cc(O)c1.C1(=O)C(C)N1 N1(C(C2C(C)CN(C(=O)C(C)c3cccs3)CC2)=O)CCc2cccnc2C1 C(C(C)C(C)C(=O)N(CCCCN(C(=O)C=Cc1cncc(O)c1)C)C)OC N1(C(c2ccc(CC)cc2F)=O)CCC(NC(=O)CC2CCCO2)C2(CCC2)C1 C(=O)(CC(C)(C)CC(=O)NCCc1ocnc1CNC(=O)C(CC)CC)OC C1(C(=O)NC2C3(CCN(C(CS(CC)(=O)=O)=O)CC3)C2)COc2ccccc2O1 CC(=NOCC#N)C(=O)NC(CO)C(=O)NCCCc1ccco1 c1(C(N2CC3CN(C(c4c(OC)csc4)=O)CC3C2)=O)ccc2nc(Br)sc2c1 N1(C(c2n(CCC)ncc2)=O)CCC(C(N2CCC(NC(C)=O)C2)=O)C1(C)C C1(CC(=O)NCC2N(C(C3OCCC(C)C3)=O)CC2)CCCC2(CCC2)O1 c1(C(N2CC(NC(c3n(CC)ccc3)=O)C(F)C2)=O)sc(Cl)c(Cl)c1N C(C(C)(CC(=O)N(CCCNC(C1CC(N(C)C)C1)=O)CCO)C(F)(F)F)N(C)C Cn1nc(C(N2CCN(C(=O)CC(F)(F)F)CC2)=O)c2c1CCOC2 C1(CC(=O)OCC)CC12CCN(C(=O)Cc1ccco1)CC2 c1(C(=O)NC2CN(C(CC3C(C)(C)CCO3)=O)C2)nc2ccc(Br)cn2c1F C(CS(=O)(=O)c1ccccc1F)NC(=O)NC1C2(CC(OC)C2)C1 C(=O)(C1=CCCC(C)(C)C1)NC1C(CNC(Cc2cccc(OC(C)C)c2)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)NC(C)(C)CCNC(=O)C(O)CC1CCOCC1 C=CC(C)(C)C(=O)NC1(C(=O)NC(c2csc(C)n2)C)CC1 CC1(NC(c2cc(F)cs2)=O)CC(NC(c2cncn2C2CC2)=O)C1 C(=O)(CC(F)(F)CC(=O)OC)NCC1N(C(Cc2cccc(OCC)n2)=O)CC1 c1(C(=O)NC2C(CNC(C3(OC)CCOCC3)=O)COC2)ccc(O)cc1Cl C1(C2CC2)(NC(C2=CC(C)(CC)C2)=O)CCN(C(=O)C(C)(C)C(C)(C)C)C1 CCCC(CC)C(=O)N(C1CC(NC(c2ccc(-n3cncc3)cc2)=O)C1)C c1(OC)c(C(N2CC=CC2CNC(C2CC2(F)F)=O)=O)csc1Cl c1(-c2onc(-c3c(C)cc(F)s3)n2)cc2occc2s1 c1(C(=O)NC(Cc2cn[nH]c2)C(=O)N2CC(OCCO)C2)ccccc1F C(C(C)(C)CNC(=O)CCCc1cccs1)N(C(=O)CCn1ccnc1)C C(=O)(C1=CCC(NC(c2ncnc(O)c2F)=O)C1)NC1CCC(C(C)(C)C)C1 c1(C(C)C)ncc(C(=O)NCC2CCC(NC(C3CC(C(F)(F)F)C3)=O)C2)[nH]1 N1(C(c2nc(OC)c(F)cn2)=O)CC2COCCC2(NC(=O)Cc2ccsn2)C1 C(CN=c1[nH]c(N2CCN(C3CC3)C(C)C2)nc2c1CCCCCC2)SCC=C C1(NC(Cc2ccn(C)n2)=O)CC2CC(NC(=O)C=Cc3ccc(Cl)cc3)CC12 c1(C(N(CCN(C(=O)CC2C=CCC2)C(C)C)C)=O)ccc(C(F)(F)F)nc1 CC12CN(C(=O)Cn3nnc(=O)[nH]3)CC1CN(C(c1cc3c(s1)CCOC3)=O)C2 Cc1ccc2n[nH]cc2c1C(N1CCN(C(C2CN(C3CCC3)C2)=O)C(C)C1)=O C1(NC(c2cnc(C(C)=O)s2)=O)CN(Cc2cc(C)sc2C)CC1(C)C N1(C(C(CC)OC)=O)CC2(NC(C3(CN4CCCC4)CCCC3)=O)CCC1C2 c1(C(N2C(C)(CC(C)C)CCC2)C(=O)NC(C)(C)C)ccc2cc(Cl)ccc2c1 C1(NC(c2cc(C3CC3)cs2)=O)CN(C(c2ncoc2Br)=O)CC1O C1(C)(CC2CCC2)CCN(C(C(=O)NCCOC(C)(C)C)C2C(CC)C2)C1 C(CC(C(=O)Nc1cnn(CC(C)C)c1)NC(c1cccnc1C)=O)SC c1(SCC(=O)NC2CCC(NC(=O)Cc3csnn3)CC2)ccccc1[N+](=O)[O-] N1(C(c2c(C)snc2)=O)CCN(C(c2cnnn2C)=O)CC(O)C1 C1(C(N2CCC(OCC=C)C2)=O)CCN(C(=O)C(C(C)C)SCC)C(C)(C)C1 n1(CC)ncc(CNC(C2CCC2NC(c2cc(C)n(C)n2)=O)=O)c1C N1(C(C2CC2C2CCC2)=O)CCC2CCN(C(c3ccns3)=O)C2C1 N1(C(C2(OC)CCSC2)=O)CCC2CCC(C1)N2C(C1COC1)=O Cc1cc(C(=O)NCC2CN(C)CCN2C(C2COCCO2)=O)cc(F)c1 C1(NC(c2ncn(C)n2)=O)CCCC12CCN(C(=O)CS(=O)(=O)NC1CC1)C2 c1(C(C2CC2)NC(CC)CNC(c2cn(C)nc2C(C)C)=O)cnc(N)c(CO)c1 C1(CNC(=O)OC(C)(C)C)CC2(C1)CN(C(=O)Cn1ncc(Br)n1)C2 c1(CNC(c2ccns2)=O)cn(C2CCCC2)nn1 CCC(C#N)C(=O)NC1CC(N(C(=O)CCN2C(=O)CCC2=O)C)C1 N1(C(C2(CC#C)CCOC2)=O)CC(NC(C2(NC(N)=O)CC2)=O)C(C)C1 C1(CC)(NC(=O)CCc2nnc(C(F)F)o2)CCN(C(=O)CNC(C)=O)CC1 C1(CNC(C2CCN(C)C2=O)=O)CCCC2CN(C(=O)Cc3cc[nH]c3)CC12 Cn1cc(S(N)(=O)=O)cc1C(=O)NC1CC(NC(=O)C#CC(C)(C)C)C12CCC2 C1(C(=O)Nc2nc(OCC)oc2)CCN(C(=O)CCOC)C(C)(C)C1 N1(C(c2c(C)cc(F)nc2)=O)CC2(CCN(c3ncnc(=N)[nH]3)C2)C1 S(=O)(=O)(c1cc(Cl)c(OC)cc1Br)NC(C1(c2ccc(OC)c(OC)c2)CC1)=O CC1(C)COC(CC(N2CC(NC(C3(F)CCCCC3)=O)CC2CO)=O)CO1 C(CCC1CC1)(C(=O)NCCN1CCC(C)C1)NC(c1c(CCC)n[nH]c1)=O C1(C(=O)NCC2N(C(C(C)C(F)F)=O)CCC2)CN2CC3CC2(CO1)C3 C1(NC(CCCN(C)C)=O)CCC12CN(C(c1ccc(C(F)(F)F)o1)=O)C2 C1(CN(C(=O)CCc2cn[nH]c2)CC)CCCN(C(=O)C(C)CO)C1 c1(C(N2C(C)CC(CNC(c3ncc(Cl)n3C)=O)C2)=O)cc(S(C)(=O)=O)co1 C1(CNC(CC(C)CF)=O)CCCCCN1C(=O)CSc1nc[nH]n1 N1(C(C(=O)NCc2cc(CC)sc2)=O)CCC(S(=O)(=O)CC)C1 c1(COC)ncc(C(N2CC(NC(=O)Cc3cnn(C)c3)CC2(C)C)=O)c(O)n1 c1(C(CC)C)ccc(OC)c(O)c1.C12(CC1)CCC2 Cc1c(C(N2CCSCC2CCNC(C2CC(C3CC3)=NO2)=O)=O)nn(C)c1N c1(C(=O)NCC(CC=C)NC(C2(CC#C)CCOC2)=O)nnn(C)c1CC N1(C(c2cn(CCC)nn2)=O)CC(O)CC1C(=O)NC(C)CCN(C)C1CC1 C(=O)(C(C)(C)CC#N)NC(C)CNC(=O)CN(C)CCO c1(OC)cc(C(=O)NCC=CCNC(=O)CN(S(C)(=O)=O)C)c2c(c1)CCO2 C1(C(=O)NC(C)(C)CNC(=O)CCC2CNC(=O)N2)CCCC2(CCOCC2)O1 N1(CC(COC)O)CC2CC1CN2C(=O)C(c1ccc(F)cc1)N1CCSCC1 C1(C(=O)NC2CCC(F)(CNC(=O)C=CC3CC3)C2)CCc2c[nH]nc2C1 N1(C(C2(SC)CC2)=O)CCCC2(CCC(NC(=O)C3=CCCCO3)C2)C1 c1(C(N2CCC(c3ccccc3)C2)=O)cc(N2CCC(O)C2)ccc1[N+](=O)[O-] C1(CC(=O)NC(CNC(c2nc(C)oc2)=O)CO)Sc2ccccc2NC1=O c1(CCCCC)cc(C(=O)NC2COCC2CNC(c2cnc(C)s2)=O)n[nH]1 C(C(O)CC(=O)NC(c1ccns1)C)NC(C1(C(C)C)COC1)=O c1(C(N2CCCC(C(C)NC(c3cc(C)no3)=O)C2)=O)cn(C)c(=O)cc1C Cc1nc(C)c(C(C)NC(C2(C(C)C)CCCN2C(=O)C(CO)N(C)C)=O)[nH]1 C(C(O)C(=O)N1CCC(C(C)(C)NC(C2CC2C(F)F)=O)C1)SC N1(C(C(CC)OC)=O)CCCC(N2CCN(C(C3CC=C(C)CC3)=O)CC2)C1 c1(C(=O)NC(C2OCCN(C(C3(CC(C)C)CCC3)=O)C2)C)cc(N)c(F)cn1 C1(C#CC(=O)NC2CN(C(=O)C(F)(F)c3cnn(C)c3)CC2(C)C)(CC)COC1 c1(C(=O)NCC2CCN(C(C3(C)CSC3)=O)C2)nc(S(N)(=O)=O)c2ccccn12 N1(C(CC2(CC(=O)OC)CC2)=O)C2CCC1CN(C(=O)NC1CC(CC)=NO1)C2 N1(C(CCC(C)NC(=O)C(F)CC(C)(C)C)=O)CCC2(CC1)CSC2 N1(C(C(F)=CC)=O)CCC(NC(=O)COc2ccc(Br)cc2F)CC1C c1(NC(C2CN(C(c3cnc(O)nc3O)=O)CCO2)=O)ccnc2c1CCO2 C=CCC(C(=O)N1CCCCC1CCC(=O)NC(C)(CO)CCC)OC C12(CNC(CC3(C=C)CC3)=O)CCC(CNC(c3nn(C)cc3Cl)=O)(CC1)CO2 c1(C(C)(F)F)cc(C(=O)NCC2(NC(C3CCCC3O)=O)CCOC2)no1 C12(C(N3CC4(N(C)CC4)C3)=O)CCCC1CCN2C(=O)CC1CC(=O)C1 N1(C(c2cc(C(C)C)c(O)cc2)=O)CCN(C(=O)C2=CCCS2)C2CCCCC12 C1(C(=O)NC(CC=C)CNC(c2[nH]c(C)c(C(C)=O)c2C)=O)CCCS(=O)(=O)N1 N1(C(CC(C)=C(C)C)=O)CC(NC(=O)C=Cc2ccncn2)CC1C CC(C)CC(CNC(=O)CSCc1ccccn1)NC(=O)CCn1ccnn1 N1(C(c2cc(Cl)cc(C)c2C)=O)CC(C2CCN(C(C3(CO)COC3)=O)CC2)C1 Cc1cn2cc(C(N3CCN(C)CC3CNC(C3C(Cl)(Cl)C34CC4)=O)=O)nc2s1 c1(C(C)C)cn(CC2CCN2C(=O)CC2CCCC2)nn1 c1(CC(=O)NC2CN(C(C(CC)(C)O)=O)CC2(C)C)c(C)nc2nc[nH]n2c1=O c1(C(=O)NC2C(CNC(c3ccc(C)c(C4CC4)c3)=O)C2)cccc2c1CCN2 C(=O)(C(O)CC(C)(C)C)N(C)CC1CCCCN1C(c1ccnc(Cl)c1N)=O c1(OC)cc(=NC(=O)C2CCC3(CC3)N2C(C23CSCC2C3)=O)[nH]n1C C(=O)(C(C(C)(C)C)NC(C1C=CC=CC=C1)=O)NCCc1cc(C)ns1 N1(C(CC)=O)CCC(CNC(=O)CCCC2CCCC(=O)N2)C12CC2 C1(C(=O)NCC2C(CC(=O)N(CC(C(C)C)C)C)C2)CCC2(CCC2)O1 C1(CNC(C(C2CC2)SC)=O)CC(C)N(C(=O)CCc2ccc(C)cc2)C1 c1(OC(C)=O)cc(C)c(Br)cc1CN1CC(O)CC1C(N1CC(F)(F)CC1C)=O c1(CCN(CCN(C)C)Cc2ccccc2)cc2ccccc2n1C c1(C(=O)NCCCN(C(=O)COC2(C)CCCC2)CC)ccc(SCCC)o1 C=CCCC(C)(C)C(=O)N(C)CCOCCCN(C(=O)CCN(C1CCC1)C)C CCC(C)CC(C)NC(=O)NCC(C)CC1NC(=O)NC1=O n1(CC)[nH]c(C)nc1=NC(=O)NCC(C1CCCOC1)O c1(C(=O)NCC2C(C)CCN2C(=O)C(C2CC2)C2CC2)cnc(O)c([N+](=O)[O-])c1 CC(C)(C)CC(F)C(=O)NC(C)(C)CCCC(=O)NC1(C)CC(C)(C)OC1=O N1(Cc2cccc(OC)c2)CC2CN(C(c3cnc(N(C)C)o3)=O)CC12 C(=O)(C1=CSCS1)N1CC(CCNC(C(C)(C)c2cncnc2)=O)C1 CN1CCC(C2CCN(Cc3ccc(-c4nn[nH]n4)o3)C2)C1 C(=O)(CCC(=O)NN(C)C)N(CCC(=O)NCCC1CCN(C)C1=O)CC#C C(CC1CCc2ccccc21)n1c(CCC#C)nnc1N(C)CCOCCOC C#CCC(C)(C(=O)NCC(n1cccn1)C)NC(=O)C(C)CCCC N1(C(c2oc(C)c(CO)c2)=O)CC2N(C(=O)C(O)CN(C)C)CCC2(C)C1 Cc1ccc(Br)c(CCC(=O)N2CCC2Cc2cn(C(C3CCOC3)C)nn2)c1 C(=O)(C(O)CCCNC(=O)CC1CC2(CCC2)C1)N(CC(CC)C)C c1(C(=O)NC2(C)CCN(C(C3C(=C)C3)=O)C2)ccnc2cc(Cl)ccc12 O=C(C(C1=NOC2CC12)N1CCc2c(Cl)cccc21)NCCC1CC1 CCCCCCCC(=O)NC1CN(C(c2ccc(Cl)c(C)c2Cl)=O)CC1C(F)F CCS(=O)(=O)CC(=O)N(C)CC1CCCC(NC(=O)COC(=O)CO)C1 C=CC(C)(C)CCNC(C1(CNC(=O)CCc2ccncn2)CC12CCC2)=O Cc1nc(C2CC2)[nH]c1C(=O)NCC1CC(NC(c2c(Cl)cnn2C)=O)C1 c1(C(N2C(C(N(CC=C)CCOC)=O)CC(O)C2)=O)cccc(C)c1C Cc1ccc2[nH]nc(C(=O)Nc3cc(C)c4nccn4c3)c2c1 C(C)(C)(CC(=O)NCC12CCCCC1C2)C1(CNC)CCC1 C1(C(=O)NCC2CC(Cn3cc(C(C(C)C)(F)F)nn3)C2)CCCC(F)(F)CC1 n1(CCOC)ccc(=NC(=O)C(C(C)O)NC(=O)CC(C)CC(C)C)[nH]1 CC(C)CC(CNC(c1ccc(CO)o1)=O)C(=O)NC(C1CCCC1O)C O=C1CCCC(C(=O)NCCC2(C(=O)NC3CC4(CCC4)C3)CC2)N1 C(=O)(CC(C)CN(C)C)NCCC1(NC(c2scc(C)c2)=O)CCC1 c1(C(=O)NC2(CNC(C34C(C(N)=O)(CCC3)C4)=O)CC2)cc(O)cc(Cl)c1Cl C1(C(=O)NC(c2nc(C)sc2)C)C2CC3C(C2NC(=O)Cc2ccc(F)cc2)C13 Cc1cc(C(N2CCCCC(NC(=O)C=CC3(C)CCOCC3)C2)=O)ncc1F N1(C(c2c(CC)onc2C)=O)CCCC(CC(=O)NC(CC)CCO)CC1 C1(NC(c2c[nH]c(Br)c2)=O)CCCN(C(c2coc(O)n2)=O)CC1 c1(C(=O)NCCN(CCC)C(C2(OC)CCSC2)=O)ccc2c(c1)C(=O)NC2 c1(C(=O)NCC23CN(C(CC#C)=O)C(C2)CO3)cc(SC)ccc1[N+](=O)[O-] N1(C(C(CC=CCC)C)=O)C2CCC1CN(C(C13CC(C(=O)OC)(C1)C3)=O)C2 C1(C(N2CCN(C(CC(CC)C)=O)C(C)C2)=O)Cc2cccc(OC)c2O1 C1(NC(CSCC=C)=O)CCCN(C(=O)Cn2ccnn2)C1CC C1(CCNC(=O)NC(C)CCN2CCCC2)CCCN1C(=O)OC(C)(C)C N1(C(CCC#C)=O)CCCC(O)(CCNC(=O)C=CI)C1 c1(COC)nocc1NC(=O)C(Cc1cn[nH]c1)NC(=O)C=CC(C)(C)C S(=O)(=O)(C1CCOc2ccccc21)NC(CCN1C(c2ccc(C)o2)CCC1)=O c1(CC(=O)N(C2CN(C(=O)CNS(C)(=O)=O)C2)C)cc[nH]c(=N)c1 C1(C(=O)Nc2nc(C(F)(F)F)cc(Cl)n2)CCCC12CCN(C(c1ccns1)=O)C2 N1(C(C(C)n2ccnc2)=O)CCSCC1CCNC(=O)C(=O)N(C)C N1(C(CC(C)SC)=O)CC2CC(C(=O)NC3(CN(C)C)CCCCC3)CC2C1 C1(CNC(c2c(C)sc(Cl)n2)=O)CC2(C1)CN(C(=O)CC1CCCC(=O)N1)C2 Cc1ccccc1C(=O)NCc1nc(-c2cc[nH]n2)nn1C1CCSCC1 C1(C(=O)OC2CN(C(C(C)=O)=O)C(=O)C2)CCC(C)(C)CN1 C1(CNC(c2n(C)c(S)nn2)=O)CC2CCC1N(C(=O)Cn1cc(CO)nn1)C2 CC1CC(O)CCN(CC2(C)CC(O)CN2C)C1.C1(NC=O)C2CCCC2C1 c1(CC(=O)N(CC(CNC(C(C(C)C)F)=O)O)C)csc2ccc(Cl)cc12 C12(C(=O)NCCC(=O)NC)CC(CN(C(=O)CC3OCCO3)C1)C2 c1(OC)ccc2c(c1C(=O)NC1(C(CC(=O)N3C(CCC)CC3)C)CC1)CCC2 C(=O)(C(C)(C)CC1CC1)N1CCC(CNC(c2ccc(C(C)C)s2)=O)CC1(F)F Cc1nn(C)c(C)c1C1CC(n2cc(-c3cc(N)n(C)n3)nn2)C(O)C1 CC(C)(C)CCC(N)C(=O)N1CCC(C2NCC2(C)C)CC1 N1(C(c2c(C)nc(O)cc2)=O)CCC2(CC(NC(C3(C)CCC3)=O)CO2)C1 C1(C(N2CCCC(Cn3cc(CN(C)C)nn3)C2)=O)CCc2nnnn2CC1 c1(CC(=O)NC(C)(C)CCCNC(C2(O)CC(F)(F)C2)=O)ncc(F)cc1F N1(C(C2(COC)COC2)=O)CCC(CCNC(=O)Cn2ncn(C)c2=O)CC1 Cc1nc(O)c(Br)cc1C(N1CC2C(NC(=O)C(C3CC3)N(C)C)C2C1)=O C1(C(=O)NCC2(C(N)=O)CN(C(C(C)(C)OCC)=O)C2)CCC12CCCO2 C1(c2cn(C)nc2)CN(Cc2ncc(-c3ccccc3)s2)CCO1 C12(CC(O)C1)C(=O)N2CC(=C)C.C1(N(CC(=C)C)CCC)CCOCC1 c12c[nH]nc1S(=O)(=O)N1CC3COCC3(C1)C(=O)NC2C.C1(CSC)CNC(=O)C1 N1(C(C(C)(C)n2cccn2)=O)C2CCC1CC(NC(C1Cc3nncn3C1)=O)C2 C(C)(C(=O)NCCC1(C(=O)N(C)CCC2CCCO2)CCC1)=C(C)C C(C(CC)(CC)N=c1[nH]nc(C(F)(F)F)n1C)N(C(CC)Cc1ccccc1)C CS(=O)c1cccc(C(=O)NC2(CNC(c3cn[nH]c3)=O)CC3CCC2CC3)c1 c1(CC)nn(C)cc1C(=O)NCc1ncoc1C1CN(C(=O)C(C)C(C)O)C1 c1(C(=O)OC)ccc(N(C(=O)C(=O)N2CC(OC(C)(C)C)C2)C)c(Br)c1 c1(C(N2C3CCN(C(c4ccccc4)=O)CC3CC2)=O)cc2c(cn1)OCCC2 N1(C(CCC2N(C(c3cncc(C)n3)=O)CCC2)=O)CC2(CCOC2)C1 c1(C(N2CC(OC)C(NC(=O)C(C)NC(C)=O)C2)=O)ccc(S(C)(=O)=O)c(C)c1 N#CC1(C(=O)NC2CCC2CNC(c2cnn(C3CC3(F)F)c2)=O)CCSCC1 Cc1nc(C(=O)NC2CC2NC(C2CCC(=O)N2C)=O)c(C)n1C C(=O)(C(O)C(F)(F)F)N(CC(C)N(C)C(c1cccc(CO)c1)=O)C Cc1nc(=N)[nH]cc1C(=O)NC(C)CN(C)C(c1cnc(O)nc1O)=O Cc1cccc(CN(C(=O)C(=O)N(C)Cc2ccc(CN3CCC3)cc2)C)c1 CC1CN(C(C2CCC(NC(c3cc(O)ccc3Cl)=O)C2)=O)CC(C)O1 Cn1cncc(C(=O)NCCCCCCNC(c2cccc(OC(F)F)c2)=O)c1=O C1(CC(=O)N(C(CNC(=O)CC2SC(=N)NC2=O)C2CC2)C)COC(C)(C)C1 c1(OC)c(C(=O)N(C)CC2CCCN2C(C2CC2c2ccsc2)=O)c(C)nn1C C(=O)(CCS(=O)(=O)N(C)C)N1CC(CC(C)NC(c2ccnc(CO)c2)=O)C1 C(=O)(C1CCc2cccc(O)c21)N1CCC(CC)(NC(c2csnn2)=O)CC1 c1(C(N2CC(OCC(=O)NC3CC(C)(C(=O)NC)C3)C2)=O)cnc2n1CCC2 C1(C(=O)NC2CCCC(NC(CCC=C(C)C)=O)C2)Cc2ccccc2C(=O)O1 C1(C(=O)NCC(CC)(O)CC)C2CCCC2CN1C(c1csnc1OC)=O Cc1ccc(C(N2CCCC(C)C2CNC(c2cnoc2C)=O)=O)c2c1CCC2 CN1CCc2cc(C(=O)NCC34COC(CNC(c5ccsc5)=O)(C3)C4)ccc21 c1(OC)cc(CNC(=O)C(C2(O)CCCOC2)(C)C)cc([N+](=O)[O-])c1 N1(C(C(CC)CC2CC2)=O)CCN(C(=O)CCc2c(C)noc2C)CCC1C CC1CCC(CNC(=O)Cc2cc[nH]n2)CN1C(=O)CCNS(C)(=O)=O C1(C(N2CC(N(C(=O)CC3CCC(=O)N3)C)C2)=O)CC12CC(O)C2 c1(OC)ccc(C(=O)NCC2CN(C(=O)CCC(N)=O)CC2(F)F)c(C)c1 c1(C(C)C)ccc(C(=O)NCC=CCNC(=O)C(C)Oc2ccccc2Cl)nc1 CC1C(NC(C2CCC(F)(F)C2)=O)CCN1C(=O)CCCC1CCCC1 N1(C(=O)NCCn2cnc(C(=O)OC)n2)CCC(C(=O)OC(C)(C)C)CC1C CC(C)C(CNC(C1CCC(=O)N(C)C1)=O)N=c1ccc2c([nH]1)CCCC2=O C1(C)(C(N(CCNC(CNS(CCOCC)(=O)=O)=O)C)=O)CCC(C)C1 N1(C(c2ccc(C)o2)=O)CC(NC(C2C3COCC23)=O)C(C2CC2)C1 N1(C(C=Cc2cn(C)nn2)=O)CCC2(CC1)CC2NC(C1(Br)CC1(F)F)=O N1(C(c2c(=N)cc[nH]c2)=O)CCN(C(=O)COCc2ccccc2)C2CCC12 N1(C(C(CC)C2CCOCC2)=O)CCC(CO)(NC(C2CCCSC2)=O)CC1 c1(C(=O)NCC2(C)NC(=O)NC2=O)n[nH]c2cc(N)ccc12 C1(OC)CCCN(C(c2ccnc(Br)c2)C(=O)Nc2ccc(F)cc2)CC1 c1(C(N(C(CC(=O)NC2(CC=C)CCOC2)C)C)=O)c(Cl)cnn1CC C(=O)(N=c1cc(-c2ccc(Cl)cc2)o[nH]1)NCC1CCN(S(C)(=O)=O)C1 C(CCCCCC(=O)N1CCN(C2(C)CC2)CC1)NC(C(CC=CC)C)=O Cc1ccc(C(CNC(=O)CC2CCOCC2)NC(c2n[nH]cc2Cl)=O)cc1 CC(C(C)(C)C(=O)N(C1CC2CC2C1)C)NC(=O)C(O)C(F)(F)F C(N=c1[nH]c(Cl)c(C#N)s1)C1N(C(C2N(CC)C(=O)CC2)=O)CCCC1.C1CC1C C(C1=NOC2CCCC12)NC(=O)Nc1cn(C)nc1C1CCC1 Cc1ccc(C#N)c(N2CCN(C(=O)OC(C)(C)C)CC2)n1.C12(C)CCC(O1)S2 c1(C(=O)NC2CCC(CNC(C3CC4CCC3O4)=O)C2)cccc2cnnn12 N1(C(=O)C(F)C2CCOC2)CC2C3CCC(C2C1)N(C(C12CC(F)(C1)C2)=O)C3 CCC(C)(C(=O)NC1C2CC1N(C(c1nnc(O)cc1O)=O)C2)C(N)=O C1(CNC(=O)NC(CCC)C2CCCC2)CCC2(C1)CC2(F)F CCC#CCCNC(=O)C=CC(C)NC(=O)CCc1conc1C C1(CNC(c2c(C)cns2)=O)CN(C(C2CCOC(C)C2)=O)CCC1(F)F C(=O)(CCCCC(C)C)N(C1CCCCC1)CCNC(c1c(OC)n[nH]c1)=O c1(C(=O)NC2(CC(=O)NC(c3cccc(F)c3)C)CC2)ccc(N)c(F)n1 c1(-c2cncc(OC)n2)n[nH]c2ncc(C(N3CCC4(C3)CC4(F)F)=O)cc12 N(C(=NCCCCl)NC1CCCCC1)CC1(C)CCCCC1O.c1(N)ccccc1 C1(CNC(C)=O)CC(O)CN1C(=O)C(O)CC1CCS(=O)(=O)C1 C=CCCCCCC(=O)N(CC(C)O)CCNC(c1cnc(NC(C)=O)o1)=O C1(CC(=O)NC2CCC(NC(c3cc(C)ncn3)=O)C2)OCCOC1(C)C c1(C(C(=O)NCC(c2c(C(C)C)cccc2)N)O)ccc(Cl)cc1Br Cc1cnc(CNC(=O)Cc2ccc(Br)s2)s1.C1(C)CCCCO1 C(=O)(C(CCC1CC1)NC(=O)C=Cc1nccs1)N1CCC(C2C(C(C)(C)C)C2)C1 C(C(CC(F)(F)F)NC(=O)C(C)COc1ccccc1)Nc1cnc(OC)s1 Cc1cc(C(=O)NC(CC2CCOCC2)C(=O)Nc2cccc(O)c2)nn1C C1(NC(c2nc(CCCC)sc2)=O)CS(=O)(=O)CC1NC(=O)C1CC1 N1(C(c2n(C)cnn2)C(=O)NC2CCOC2)CCOC2(CCC2)C1 c1(C(=O)NC2C(NC(C(C(C)C)SCC)=O)C2)cc(F)cc(Cl)c1N c1(C(=O)NCC2(OC)CC2)c(C)[nH]c2ccnn2c1=O.C(=O)(C1C(=O)N1)OCC c1(C(C)=O)ccc(NC(=O)CC2CN(C(=O)C(C)(C)C)CCO2)c(C)c1 c1(C(N2CCCC(CNC(CCNC(N)=O)=O)C2)=O)ccnc(F)c1O C1(C(=O)NC(CC)CNC(C2(C)CCCC2CC)=O)CC2CCCCCCC12 c12ccc(cc1)C(=O)NC2.c1(CC2C(NC(=O)C=C3CCC3)C2)ccc(F)cn1 N1(C(Cc2c(C)ccc(C)c2)=O)CC2CCC1C(C(=O)NCCC(C)O)C2 Cn1cc(Cl)cc1C(=O)NCC(=C1CN(C(c2cnnc(C3CC3)c2)=O)C1)F C1(NC(CNS(CC)(=O)=O)=O)CCN(C(c2ccoc2Br)=O)C(C)C1 C12(CC(N3C(C)CC(NC(CCCC(C)=O)=O)C3)=O)CCC(CC1)C2(C)C N1(C(C(CNC(Cc2n(C)cnc2)=O)CC2CC2)=O)CC(O)CC12CCCC2 C1(O)(C(N2CCC(n3cc(CCCSCC)nn3)C2)=O)CCCC(C)CC1 C(=O)(C(O)Cc1cnc[nH]1)NCC(CC)N(C(=O)CC(C)n1ccnc1)C Cc1ccc(OCCNC(=O)CS(=O)Cc2noc(CCN)n2)c(C)c1 CCC(CC(=O)N(CCCCNC(c1ccc(OC)cc1OC)=O)C)C(C)C C12(C(N3CC(C)SCC3)=O)COCC1CN(C(c1ccc(O)c(I)c1)=O)C2 O=C(CC1=CCCC1)NCC1CCCN(C(c2ccc(O)c(F)c2)=O)C1 CC(F)C(C)N=c1[nH]c(=NCc2cccc3c2OC(F)(F)O3)[nH]c2ccsc12 CC(C)(CNC(=O)COc1ccccn1)CC1CN(C(c2nsnc2O)=O)C1 N1(C(=O)Cn2cccc2)CCN(C(c2cnns2)=O)C2CCCCC2C1 c1(C(=O)NCC(CN(C(C2(C(=O)NC)CCC2)=O)C)C)ccc(C)o1 N1(C(c2cc(C(=O)N(C)C)on2)=O)CC(C(N2CC=CC2COC)=O)C2(CC2)C1 C1(CNC(c2snc(O)c2Cl)=O)C2CN(C(C3(CO)CC3)=O)CC12 C=CC(C)(CCOC)C(=O)N1CCC(O)(CCNC(C2CC2CN(C)C)=O)CC1 N1(C(C(CC)(C)O)=O)CCOC2(CCN(C(=O)C(C)(C)S(C)(=O)=O)CC2)C1 N1(C(c2c(CC)ncnc2)=O)CCC=C(C(=O)NCC(O)CN(C)C)C1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(NC(c2cn(C(C)(C)C)cn2)=O)CC1C N1(C(C(c2cccc(C)c2)(C)C)=O)CCC(CO)(NC(=O)CC(C)C(C)C)CC1 c1(C(=O)NC(CNC(C(C(C)O)NC(C)=O)=O)(C)C2CC2)cc2c([nH]1)CCCC2 Cc1nnc(C(C)NC(c2conc2C(C)NC(c2ccoc2Cl)=O)=O)s1 CN1CCCC1C1CCCN1c1nnc(-c2c(F)cc(Br)cc2F)o1 S(=O)(=O)(c1ccc(N2CC3CC2C3)cc1Br)N(C)C1CC1.C12CC(O)CN1C2 C(=O)(C(CCC(N)=O)n1cc(-c2cccc(C(F)(F)F)c2)nn1)NC1(C)CSC1 CCCC(C(O)C(=O)NCC(F)F)NC(=O)Cc1cccnc1 N1(C(C=C(C)C)=O)CCC2(CCOCC2C(N2CCCC2CN(C)C)=O)CC1 C1(NC(CCC2(C)CN(C(C3CC3[N+](=O)[O-])=O)C2)=O)CCC=CCCC1 C1(C(=O)NCC(C)OC(C)(C)C)CCCCN1N=O.c12ncc(cc1Cl)[nH]2 CCC(CC)C(C)C(=O)N(CCNC(C1CC1C1CCC1)=O)Cc1ccccc1 CC(C)CC(C)CC(=O)NC(CNC(C)=O)C(=O)NCCOCCN=[N+]=[N-] Cc1ncnc(C)c1C(=O)NC12CC(CNC(=O)Cc3ccc(C(N)=O)cc3)(C1)C2 C1(C(=O)NC(C(N2CC(O)(CC(C)C)C2)=O)C2(C)CC2)CC12CCCC2 Cc1cc(F)c2cc(CC(N3CC(NC(=O)CC(=O)N(C)C)C(O)C3)=O)[nH]c2c1 n1(CCOCCOC)ccc(C(=O)N(C)CCNC(=O)CC2CCCCC2)n1 N1(C(CCC2C(NC(C3C(C(C)C)C3)=O)CCC2)=O)CCC2CCCC12 Cn1ccc2ccc(C(N3CCC(NC(C4CC(C#N)C4)=O)C3)=O)cc12 N1(C(C(C)C2CCC2)=O)CCC(N(C(=O)C(O)c2ccsc2)C)C1 C#CC1(C)CCCN(C(C2CC(C)(C)CCN2C(c2ncn(C)c2C)=O)=O)C1 C1(C(C)C)CN(C(=O)CC2CCCN2C(C23CCC(C2)C3)=O)CCO1 C1(F)(CNC(CC(C=C)(C)C)=O)CCCN(C(C2CC=CCO2)=O)CC1 N1(C(CCOCC)=O)CCCC(C(C)C(=O)N2CC(CC(F)F)C2)C1 c1(OC)cc(Br)cc2c1C(NCC1C3(CC3)C13CC3)CC2 N1(C(C(C=C)O)=O)CCC(NC(C2CC(N(C)C)C2)=O)CC1 N#Cc1cc(CNC(=O)Nc2ccc3c(c2)C2CCC32)cc(F)c1 N1(C(c2c(CSC)cccn2)=O)CC2CCCC2(CNC(=O)C(Cl)=CCl)C1 C1(C(=O)OCC)CCN(C(=O)CCN(C(=O)CCOC2CCC2)C(C)C)C1C C1(CN(C(=O)CC2(C)CCCO2)C)CCCCN1C(c1cscc1Br)=O c1(OC(C(=O)N(CC(C)NC(C2SCCS2)=O)C)(C)C)ccc(Cl)cc1 C1(C(=O)NC2CCC(NC(c3coc(O)n3)=O)CC2)CC2CCCCCCC12 c1(OCC)cc(C(=O)NC(C2CCOC2)CNC(c2cnn(C3CC3)n2)=O)[nH]n1 N1(C(C(c2cccc(C)c2)F)=O)CC2(CCN(C(=O)CC3CCCO3)C2)C1 Cn1nc2c(c1C(=O)NC1CCCC1C(N1CCC(CC#N)CC1)=O)CCC2 C1(CCC)CN(C(C2CN(S(=O)(=O)CC)C2)=O)CCN1C(c1ccc(OC)s1)=O C(CN=c1ncc(F)c[nH]1)OC(C1CC(=O)N(Cc2ccccc2)CC1)=O N1(C(C(N2CCOCC2)C)=O)CCC(N(C(=O)CCC2CCCC(=O)N2)C)CC1 C1(C#N)(C(N(CC)CC2CCN(C(C3(C)CCCO3)=O)CC2)=O)CCCOC1 C(=O)(C1=NOC2(CCCN(C(c3cc4ccccc4[nH]3)=O)C2)C1)NC(C#C)C N1(c2cc(C)[nH]n2)CCN(C(C(=O)NCC2CC2(F)F)C2CC2)CC1 C1(CNC(=O)COCCC(=O)c2cccs2)CCCCC1.C12(CC1)C(=O)NC2 CCC(C)C(O)CC(=O)N1CC=C(C(=O)N(C)CCN2CCCC2)CC1 C1(NC(CCC)=O)CCN(C(=O)CC(C)(C)C#N)CC1CO c1(CN2C(=O)CN(CC(CCCC)CC)C2=O)ccc2c(c1)C(=O)NCCC2 C(c1ccccc1)=CCOCCSCC(=O)OC1CC(C(=O)NC2C(=O)OCC2)C1 C#Cc1cccc(C(N2CCN(C(C3CC(C)=NO3)=O)CC2C2CC2)=O)c1F c1(CSCC=C)cccc(C(=O)N(C)CC2C3CN(C(=O)CNC(C)=O)CC23)c1 C1(CC(N)=O)(NC(C(CCSC)O)=O)CCN(C(c2cccc(Cl)c2Cl)=O)CC1 c1(COC)cnccc1C1C(C(=O)NCCC(=O)NCCO)(C(C)C)C1 C1(C(=O)NCCC2CCCN2C(=O)C=C2CCC2)C2CCN(CC2)S1(=O)=O CCCC(CCC)CC(=O)N1CC(CNC(c2oc(C3CC3)nc2C)=O)C(C)C1 C#CCCCC(C)C(=O)N1CC(CNC(C2CCSCC2)=O)OC(C)(C)C1 c1(C(=O)NC2CCN(C(C3C(C(C)C)CCC3)=O)C23CC3)cc(Cl)c(F)cc1F N1(C(C(CC)C(C)O)=O)CCC2(CCCN(C(c3nnc(Cl)cc3N)=O)C2)C1 C1(NC(CC)=O)CCCN(c2nnc(CC(C)C)n2CCOC)C1 c1(OC)ccc(CC(=O)NC2C=CCN(C(=O)C(F)n3ccnc3)C2)cn1 c1(CC(=O)NCC(C)NC(COc2ccc(C)cc2F)=O)c(C)cc(C)cc1C CC(C)C(O)C(C)C(=O)NC(C(N1CCCC(F)(F)C1)=O)c1ccco1 CC(C)C(F)(CNC(=O)C(C)Cn1cccn1)C(=O)NCCc1cncs1 c1(CC(C(=O)NCC(C(=O)OC(C)(C)C)F)(C)C)cc(Cl)ccc1Cl c1(C(N(C2CCC(C)(C)C2)CC)=O)cc2nc(-c3ccco3)cc(C(F)(F)F)n2n1 CC1(C)C(NC(C2(F)CCCN(C(C3CCCSC3)=O)C2)=O)CC1(F)F C1(C(=O)NCC2CC(C)(C)CN2C(=O)C2=COCCO2)CCCC2CCCN12 C1(NC(c2ccc(COC)cc2)=O)CCN(C(c2ccnc(F)c2N)=O)C(C)C1 c1(CC(=O)NC(CNC(CCOCC)=O)C2CC2)cc2ccccc2c(=O)o1 C1(NC(Cc2cc(C)[nH]n2)=O)CN(C(C2CCN(C)CC2)=O)CC1C#N c1(C(=O)NC2CC(C)N(C(C3COCCOC3)=O)CC2)cncc2ccccc12 c1(N2CCCC(CCCC)C2)ccc(S(=O)(=O)NC2CCSC2)cc1C#N C1(NC(C=CC)=O)CN(C(=O)Cn2cc(C3CC3)cn2)CC(C)(C)C1 O=C1CC(CNC(=O)CC2(CNC(=O)COCC3CCC3)CC2)CCN1 c1(CC)ccc(Cl)c(NC(=O)C(N2CCCC(O)(c3nn[nH]n3)C2)=O)c1 N1(C(Cn2ncc(C(=O)OC)c2)=O)CCC(N(C)C(C2CC2C(N)=O)=O)CC1 c1(C(=O)NCCCCCCNC(C2C3C4CCC(C4)C23)=O)cc2c(o1)CCCC2 C1(C(N2CCC(CN=c3[nH]nc(CC)s3)C(C)C2)=O)C(O)C(=O)N(C)C1C N1(CC)CCCC(C(N(CC)Cc2nccn2-c2ccc(OC)cn2)=O)C1 C(CF)(C(F)(F)F)NC(C1C=CCN1C(C1CC1(F)Cl)=O)=O C=C=CCCC(=O)NCc1cc(C(=O)NCCC(C2CC2)C2CC2)co1.C C1(NC(CC2C(C)(C)COCC2)=O)CCC2(CC1)CC(NC(C1CCSC1)=O)C2 C12CCCC(CC1)NC2=O.N1(CC(C)=C)CCCC(O)C1.C1(C=O)C=C(C)CS1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC(NC(CN(C)CCO)=O)CC12CCCC2 N1(C(Cc2cn(C(c3nccs3)C)nn2)=O)C(C(=O)OC(C)(C)C)CC2CCCC12 N1(C(C(C)OCC(F)(F)F)=O)CCC(C)(C)C(CNC(C2C3CNC(=O)C23)=O)C1 C1(NC(C2C(C(N)=O)C2)=O)CC12CC(NC(c1ccncc1)=O)C2 CC(CC(F)(F)F)CS(=O)(=O)NCc1cn(CCN2CCOCC2)nc1C1CC1 C(=O)(C(O)CCC)NCC(CC)NC(c1cn(-c2ccccc2)nn1)=O.n1(CC)cccn1 C1(CCCCC)CCC(C(=O)NC2CC(C)(NC(C3CCS3(=O)=O)=O)C2)O1 c1(C(N2C3C(C(=O)OC)C(CC3F)C2)=O)c2n(c(C)cc1=O)CCC2 C(N=c1[nH]c(=N)[nH]c(=NCCn2cnc3c(cnn3C)c2=O)[nH]1)C1N(C)CCC1 CC(C)CC(C(=O)NCCCCNC(c1cccnc1F)=O)C(N)=O N1(C(=O)NCCCC2CC2(F)F)CCCCCCCCCC1 c1(COC)nccc(=NCCC2CCCC(NC(=O)CCc3cnc(C)s3)C2)[nH]1 c1(C(=O)N(c2ncc3[nH]ccc3n2)CC2CCNC2)cc(Br)ccc1[N+](=O)[O-] C1(NC(c2cc(C)no2)=O)CC2(CCC(CNC(C3C=CCC3)=O)OC2)C1 C(CCN=c1[nH]c(=NCC(CC)(CC)C(N)=O)[nH]c2cc(OC)ccc12)OC N1(C(CCCOCCC)=O)CCCC(C(=O)N(CC)CC2(C)CCCCO2)C1 CC(CCCC(=O)NCc1nccn1C)NC(C1CC(=O)NC(=O)N1)=O c1(-c2ccc(NC(c3cc(Br)ccc3F)=O)cn2)ccc(F)c(O)c1F C(C1CCC(C)CC1)=C(C)C(N1CCC(N(C)C(c2cccc(Br)c2)=O)C1)=O C1(C)(NC(C2N(C(c3c(OC)n(C)nc3)=O)CCN(C)C2)=O)CCC2(CC1)CC2 C1(C(=O)NCC(C(C)C)C(C)C)CC2C=CC1N(C(=O)C1CC1)C2 C#CCCCCCCNC(=O)C(CNC(=O)C=CC(C)(C)SC)CC1CCCC1 c1(CSC)ccc(C(=O)NCCOCCNC(=O)C=Cc2ncco2)cc1 CC(CCl)(CCl)CN(C)Cc1cc(C(F)(F)F)on1 C(CC(=O)NCC(C)N(C(=O)C(C)c1cc[nH]n1)C)SC N1(C(c2ccn(C3CCCC3)n2)C(=O)NCCOCC)CCOC(C)C1C c1(CSC)c(C)nc2ncnn2c1N1CCC(OC2CCOC2)CC1 c1(OCC)cccc(C(=O)NCC(F)CNC(=O)CCOC(C)C)c1 c1(NC(N(Cc2c(CC)cccc2)CC)=O)cc(-c2ncco2)ccc1C C(=O)(C1CCCc2nn(C)cc21)NCC(CC)NC(c1cc(C#N)cn1C)=O N1(C(=O)Cc2cc(F)cs2)CC2(C1)CN(C(c1ncccc1Br)=O)C2 c1(CC)cc(CC2CC2)nc(N2CCCC(C)(NC(=O)C#CC3CC3)C2)n1 N1(C(=O)CN2CCOCC2)CC2CCN(C(=O)CCc3ccc(Br)cc3)C2C1 C1(NC(C2OCCN(C(C)C)C2)=O)(CO)CCCN(C(c2cnn(C)c2N)=O)C1 c1(C(=O)NCC23N(C(C4(CSCC)CC4)=O)C(CC2)CC3)ccc2oncc2c1 c1(C(=O)NC2CN(C(C3(C)CS(=O)(=O)C3)=O)CC23CC3)cc2ccccc2s1 n1(CC)nc(COC(=O)C(C2CCC(F)(F)C2)O)c(Br)n1 C1(C(=O)NCCCn2cc(CCSCC)nn2)CCc2ccccc2OC1 CC(C)CCCCCC(=O)NCC(C1CC1)N(C)C(c1ccoc1)=O c1(CCC)[nH]ccc1C(N1CC(NC(C2(COC)CC(=O)C2)=O)C1)=O C1(CC(=O)NC(C(C)C)C2CC2)(OC)CN(C(C2CC2c2ccco2)=O)C1 c1(OC)ccc(C(=O)NC(C)CNC(C2(c3ccno3)CC2)=O)c(N)c1 C1(CNC(CCCC)=O)CN(C(=O)CC(CC)SC)CCC12CCOCC2 Cc1ccc(F)c(C(=O)NCC2C(C)CCCN2C(=O)CC2COCCO2)c1 c1(CCCC(=O)N(C2CCC(N)C2)C)nnc(C2CC2)n1-c1cccc(O)c1 c1(NC(c2n(C)cc(NC(c3cc(C#N)c[nH]3)=O)c2)=O)ccc(Cl)c([N+](=O)[O-])c1 N1(C(C2C(C)C(=O)C2)=O)CCOC(CNC(=O)CC2CC3CC3C2)C1 N1(C(C2(CCC=C)CC2)=O)CCCC(F)(C(=O)NCCC2CCCC2)C1 Cc1c(C(=O)NCCNC(=O)Cc2cn(C)nn2)oc2c1ccc1ccccc21 C(C1=NOCC1)(NC(=NC)NCC(C)C#N)C1CCCCC1 C(=O)(C(CC(C)C)C(C)C)N1CC(CC)N(C(c2sccc2OC)=O)CC1 CC1(C)CC(NC(=O)CC(CNC(=O)CCc2ccccc2)C2CCC2)C(=O)O1 Cc1ccnc(O)c1C(=O)NC1CCC(NC(C2CC3(CCC3)C2)=O)C1 O=C1OCC(COC(c2cn(-c3ccccc3)nn2)=O)O1 c1(C(=O)Nc2nnc(CN(C)C)s2)coc2c1C(O)CCC2 N(C(=NCCF)NCC1CC1)C(c1cn(-c2ccccc2OC(C)(C)C)nn1)C N(C(=NCCS(=O)(=O)C1CC1)NCCC(C)(C)C#N)C(COC)C.OC C(c1cn(C)nn1)=CC(=O)NC(C(=O)NCCCCN(CC)CC)CC1CC1 N1(C(C2CCC(C)(C)C2)C(=O)NCCCC)CCC(C)C2(CCC2)C1 C=CC(C)(CCOC)C(=O)N1CC(N(C)C(c2csc(C#N)c2)=O)C1 c1(C(N(C)CCN2CCN(CC(=O)O)CC2)=O)ncnc2c1c(Br)nn2C c1(NC(=O)Cn2nnc(-c3ccc(Cl)cc3)n2)cc(F)cc(Br)c1Br C1(NC(=O)Cn2cnnc2)CCN(c2nnc(C(F)F)o2)CC12CCC2 N1(C(C(C=C)O)=O)CCn2ncc(CNC(=O)C(n3cc(Cl)cn3)C)c2C1 CC1(C)CCC(C(N2CC3(CC3)CC2C(=O)NCC(CC2CC2)CO)=O)CO1 C#CC1CCN(C(C2CCCCC2CNC(C2CC(n3cnnc3)C2)=O)=O)CC1 C12(NC(c3cn(CC(=O)NC4C(CNC(C)=O)C4)nn3)=O)CC(CO)(C1)C(C)O2 c1(C(=O)NCC2(C(N)=O)CN(C(C3CCC4(C3)N=N4)=O)C2)n[nH]c2ccccc12 C1(C(N(CCCN(C)C(C2CC2(Cl)Cl)=O)C)=O)OCC1(C)C C1(C(N(CC(=O)NCC(F)Cl)CC)=O)COCCN1CC N1(C(c2cccc(OCC)c2Cl)=O)CCC2(CCCC2C(=O)Nc2cnc[nH]2)C1 CC(O)CCCCCC(=O)N1CCC(CC(N)=O)(NC(=O)CNC=O)CC1 C1(NC(=O)C(F)CC2CC2)CC(F)CN(C(c2ccsn2)=O)C1 c1(C(CNC(=O)CCC2CC2)NC(CNC(C)=O)=O)cccnc1 CCCC(C)(O)CC(=O)NCC1(CNC(c2cc(Br)cn2CC)=O)CC1 N1(C(CN(C)CC)=O)CCC(c2n[nH]cc2CNC(C2(C(=O)OC)COC2)=O)C1 Cc1n[nH]c2cc(C(=O)NC(CNC(=O)C3=CCCS3)C(C)C(C)C)ncc12 C1(NC(c2cc(F)n[nH]2)=O)COC2(CCN(C(c3cccc4nsnc34)=O)C2)C1 C1(C(=O)NC(CCNC(c2cc(C)c(F)cc2Cl)=O)C)CC2COCC(C1)C2=O CC1CCN(C(C23CC(C2)CN(C2CC2)CC(=O)N3)=O)CC1O.C1CC1 N1(C(CCc2scc(C)n2)=O)CCC(C2CCN(C(C3CCCSC3)=O)CC2)C1 c1(NC(C2CC(=C)CN2Cc2c(F)cccc2Cl)=O)c(C)cc([N+](=O)[O-])cc1Br C=CC(CCC)CC(=O)NC1CC(CC(=O)NC(c2nncn2C)CO)C1 Cc1scc(C(N2CCCC(C(C)NC(=O)CC3(C)OCCO3)C2)=O)c1C1CC1 CN1CCCC(C(=O)NC2CN(C(C3(C#N)CCCO3)=O)CC2F)C1 c1(CC)nc(CCNC(=O)C(C2(C)CC2)NC(c2cocn2)=O)n[nH]1 C1(CCNC(c2scc(C)c2C)=O)CCCN(C(C2CC3(CCCO3)C2)=O)CC1 C1(CC=C)(C(=O)N(C)CCO)CCN(C(=O)CC2(O)CCOCC2)CC1 c1(CCC(=O)NCC2C(NC(c3c(CC)noc3)=O)CCC2)ccccc1CC Cc1cnnc(O)c1C(=O)N(C)CCOCCNC(=O)CC1CCCN(C)C1 Nc1c(C(N2CCC(F)(c3cn(-c4cccc(F)c4Br)nn3)C2)=O)ccc(Cl)c1F Cc1cc(=O)n(C)cc1C(=O)N(CC(C)(C)C(N1CCCC2(C1)N=N2)=O)C Cc1cc(CC(N2CC(NC(c3cc(C(F)F)ncn3)=O)C2)=O)c(C)s1 C1(NC(C2(CCN=[N+]=[N-])CC2)=O)CCCCC1C(=O)NC1C=CCCCC1 C1(NC(c2ccc(OC)s2)=O)CCC2(C1)CN(C(c1ccc(F)c(F)c1C)=O)C2 C1(CC(=O)N(CCC#C)C2CC2)CCCN(C(=O)C(C)CC=CCC)C1.C1CO1 C1(CC(=O)NC(CC)CCOC)CC(C)(C)CN1C(c1cnn2c1OCC2)=O C1(CNC(C=CC)=O)CC2(CO1)CN(C(=O)C(O)c1ccco1)C2 C(C(C(C)C(C)C)NC(c1ccoc1C1CC1)=O)NC(C1(CCCC)CCC1)=O c1(NC)ccc(F)cc1C(=O)NCCC(C)(C)NC(=O)CC(C)n1ccnc1 C1(C(N(C)CC2CCC(CNC(CCCOC)=O)CC2)=O)OC2CCC1CC2 C#CC1(C(=O)NC(c2cccc(C)n2)C)CCN(C(c2cc(C3CC3)no2)=O)C1 c1(CC)ccc(C(=O)NC2CCN(C(=O)CCn3cncn3)CC2CO)cc1Cl C1(NC(C(C)NC(c2cc(OCC)c(F)cc2)C)=O)CCc2ccsc2C1 c1(C(C(C)C)NC(C(=O)NCC(c2ccc(C)o2)(C)O)=O)ccc(Br)cn1 C1(C)(CNC(C(N2CCCOCC2)C)=O)CN(C(=O)C(F)C(F)(F)F)C(C)(C)C1 C(=O)(C1=CC2(CCOC2)C1)NCC(C)NC(c1cccc2cccn12)=O c1(C(N(CC(CC)NC(=O)COc2ccc(CC#N)cc2)C)=O)cnccc1C c1(C(N2CCC(CNC(Cc3cc(C)on3)=O)C2)=O)cnn(C)c1C N1(CC(C)NC(C(C)C)=O)CCN(C(C2CC2C2CC2)=O)CC1 C(=O)(C(O)C1=CCCCC1)N1C(CCC(=O)NC2CCSCC2)CCC1 C(=O)(C1=NOC(C(C)(C)C)C1)NC1(COC)CN(C(C2ON=C(CC)C2)=O)C1 c1(CN2CC(NC(c3cccc4ccoc34)=O)C(F)C2)cc(Cl)c(O)cc1F CCCC(O)CCNC(=O)CN(C(=O)Cn1ccnc1)C1CC1 c1(C(N2CC(N(C(c3[nH]cc(C)c3)=O)C)C(O)CC2)=O)ccc2[nH]nc(O)c2c1 c1(C(=O)OC)cc(C)nc(N2CCCC2CNC(c2[nH]c(C)nc2C)=O)n1 C(C(C)(O)C(F)F)NC(C(C)NC(COCCC)=O)=O C(=O)(CCCCCS(N)(=O)=O)N1CC2C(CNC(C(CCC#C)O)=O)C2C1 C1(C)(CC(=O)N(CCC(C)(C)O)C)CCN(C(c2ccccc2)=O)C1 C1(NC(C=CCCC)=O)C2CC3CN(C(c4nccn5nccc45)=O)C1C3C2 N1(C(C(CC)NC(C)=O)=O)CCCC(C(=O)NCc2ccc(Br)s2)CC1 C1(C(C)(C)NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2cccnc2O)CC1 C(C(CC(=O)N(CCCNC(c1ccc(Cl)c(F)c1O)=O)C)C(F)F)N(C)C c1(C(N(C)CC2CCN(C(=O)CCc3cn[nH]c3)C2)=O)cncc(F)c1Cl c1(COC)ccc(C(=O)NCC2CN(C(=O)C(c3nc(F)ccc3Cl)C)C2)cc1 CC(N=c1[nH]c(N2CCCC(N3CCC3)CC2)nc2c1COC2)C1CC1 N1(C(C2(SC)CN(C(=O)CC3(C)CC3)C2)=O)CCCC(CCO)CC1 c1(C23C(=O)NCC(C2)OC3)ccc(OC(F)(F)F)c2ccc(O)cc12 c12nc(C3OCCc4ccccc43)nn1C2.Cn1cc(-c2cnn[nH]2)cn1 C#CCCCC(C)C(=O)N1CC2CC1(c1cn(-c3ccc(F)c(F)c3)nn1)CO2 Cc1ccn2ncc(C(=O)N(C(C)CCNC(c3cc(O)ccc3N)=O)C)c2n1 C1(NC(C=C(C)C)=O)C2CCC1CN(C(=O)C(C)C1CCCC1)C2 c1(C(N2CC(C)(C)C2C(=O)OC)C(=O)NCCCCCC)ccnc(Cl)c1Br N1(C(c2cc(C)oc2C)=O)CCCC(C)(CNC(=O)CCc2cccc(F)c2)C1 C1(NC(c2ccc(C)nn2)=O)CN(C(=O)C(C2CCCCCC2)C)CC1C1CC1 Cc1ccccc1C(=O)NC1CC(F)(CNC(C2(C)CCOC2)=O)C1 c1(C(=O)NC2CCN(Cc3c(C)noc3)CC(C)C2)ccc2cccnc2n1 c1(C(=O)NCC(CN(C(C(CCC)(C)CC)=O)C)O)cc2cc(F)cc(F)c2[nH]1 C1(C(=O)NC(CC(C)NC(c2cccc(OC)c2N)=O)C)CS(=O)(=O)CC(=O)N1 c1(C(N2C(c3cn(C)nn3)CCC2)=O)cccc(C(F)(F)F)c1Cl N1(C(C(C(=O)OC)NC(C)(C)C(C)SC)=O)CCN(C2CC2)C(=O)C1 C1(CNC(C(C=CC)O)=O)CC(F)(F)CN1C(c1ccc(CCC)c(Cl)c1)=O C=CC1CN(C(=O)C(CC)C(C)C)CC1NC(c1ccc(OC)s1)=O CCCC(C(F)(F)F)NC(=O)C1=CCN(C(C2(OC)CCCOC2)=O)C1 C1(C(=O)OC)CC(CSCCC(=O)NC2CCOC2)N(C(=O)CO)C1.C(C)(C)C C(=O)(CCC(=O)N(CCCOCCNC(C1CCCSC1)=O)C)OC N1(C(CS(N)(=O)=O)=O)CC2(C1)OC1(CO)CC2(NC(=O)CN2CCOCC2)C1 c1(C(N2CC(C(=O)Nc3c(C)cccc3Cl)SCC2)=O)c(F)ccc(O)c1F c1(C(N(CCCNC(c2cccc(F)c2Cl)=O)C2CC2)=O)ccc2snnc2c1 N1(Cc2cnn(CC)c2C)CCCC(F)(F)C1C(=O)OC(C)(C)C.C(=O)(NC)O O(NC(=O)C#CC1CCC1)CC(N1CCC(c2ccc3cc[nH]c3c2)CC1)=O C1(NC(c2c(C)scn2)=O)CCN(C(c2[nH]ccc2-c2ccccc2)=O)C(C)C1 C1(C(=O)NCCC(=C)CNC(c2ccc3c(c2)COC3)=O)CCCC2(CCC2)O1 C(N=c1[nH]c(C)cc(=NCC(C)N2CCc3ccccc32)[nH]1)c1c(C)nccc1 CC(CC(C)N=c1[nH]c(=NCC23CCC(CC2)OC3)[nH]c2cc[nH]c12)C(F)F c1(C(=O)NCC2(NC(c3csnn3)=O)CCCCC2)ccc2sncc2c1 Cc1cc(C=CC(N2CC(NC(C3(C)CC3(Cl)Cl)=O)CC23CCC3)=O)c[nH]c1=N N1(C(=O)CCF)CCC(NC(C2(C3CC3)CC2)=O)C1 C1(NC(CCCN(C(C)=O)C)=O)CCN(C(=O)CNC2CN(C(C)=O)C2)C1(C)C CC1(C)C(CNC(C2CCCCC2O)=O)CCN1C(C1CCN(C2CC2)CC1)=O Cc1nnc(N2CCC3(NC(=O)COC(F)F)CCCCCC23)c(C#N)c1C C(=O)(CC(C)(C)C)NCCC(CNC(=O)C(C)n1ccnn1)OC N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(=O)C(C)C(O)CC(C)C)C2(CCC2)C1 CC(C)C(C(=O)NC1C2CC1N(C(c1ccn(C)n1)=O)C2)N1CCCCC1 N1(C(C2CCCC(OC)C2)=O)CC2(CCCC2N=c2nc(C#N)[nH]cc2Cl)C1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CCCC(CNC(=O)C=CC(C)CC)C1 Cc1c(C(=O)NCC2(CCNC(C3C4CC5C(C4)C35)=O)CC2)cnn1C c1(C(C)C)ccc(C(=O)NCCNC(=O)C(=O)NCC(F)F)o1 C1(C(=O)NC(C2(O)CN(C(COCCOCC#C)=O)C2)C)CC12CCCCCC2 C1(C(=O)NCCC2N(C(C(CC)CO)=O)CCSC2)CC12CCCCC2 CCCCC(C)(C)NC(=O)C(C1CCCN(C(=O)C(C(C)C)SCC)C1)C N1(CC)CCC(C(N2CCC(C(=O)N(c3ccccc3Br)CCO)C2)=O)CC1 C(N=c1[nH]cnc2c1CCC2)C1N(C(c2ccccc2OC(F)(F)F)=O)CCC1 c1(C(=O)NC2C(NC(C(CCC)OC)=O)CCOC2)nn2c(c1Br)CCC2 C1(CC(=O)NCC2CCCCN2CC2CCC(O)C2)CCC=CCC1 C(=O)(N1OC2CCC1C2)C1(CNC(=O)Cc2ccco2)CCCO1 c1(OC)cccc(CCC(=O)NCC=CCNC(c2ccc(COC)cn2)=O)n1 N(C1CN(C(C(C)(C)C)=O)CCc2ccccc21)C(C1=C(C)OCCS1(=O)=O)=O N1(C(C(C)OC)=O)CC2(C1)CN(C(C1(C(F)(F)F)CCCCO1)=O)C2 C1(CNC(C2(COC)CC2)=O)(NC(C2C(C)(C)C2(C)C)=O)CCOCC1 c1(OC)ncc(CNC(c2cncc(C)n2)c2nnnn2C2CC2)cc1Br Cc1ccc(C(C)(F)F)cc1NC(=O)C(C1CCC2CC12)N c1(SC)nn(C)cc1C(=O)NCC(O)CNC(=O)C(C)Oc1ccc(SC)cc1 c1(C(N2CC(NC(C(C)C(C)(C)C)=O)(CO)C2)=O)cc(F)c(F)cc1NC(N)=O C1(C(=O)NC(COC)C)COC2(CCN(C(c3cc(Br)c(C)cc3F)=O)CC2)C1 c1(C(N(C2CCN(C(c3cc(Br)c[nH]3)=O)C2)C)=O)ccc2nc(O)n(C)c2c1 c1(N(CC=C)C)cc(Br)ccc1S(=O)(=O)NCCC(C)(C)F C1(NC(CC2CC(C)(C)C2)=O)CC2CN(C(c3cc4nc[nH]c4cn3)=O)CC2C1 Cc1cc(C(=O)N(CCCNC(=O)C(N2CCC(O)CC2)C)C)c(Cl)cc1F Cc1cc(Br)cc(C)c1CC(=O)NCCCCN(C(=O)CC(C)C(F)F)C C(C(CO)(CO)NC(C1CC1C1CCCO1)=O)N(C(C(F)=C(C)C)=O)C N1(C(c2c(C)nc(CCC)s2)=O)CCN(C(=O)C(F)=C2CCCC2)C(CF)C1 C(=O)(CC(C)C(=O)N(C(C)(C)CC(=O)Nc1cn(C)nc1C#N)C)OC C(CCCCC(=O)NOC1CCOCC1)NC(C(N1CC(C)C1)C)=O N1(C(C(CC(C)C)(C)C)=O)CCC2CCC(NC(=O)Cc3c(Cl)cnn3C)C1C2 N(C(=NCCc1cncs1)NCC(=O)NC(C(C)(C)C)=O)C(C1CCCO1)C C(=O)(C(CC(C)C)OC)NCC1(CNC(c2c(OC)oc(C)n2)=O)CC(F)(F)C1 c1(OCC)ncc(C(=O)NC(C)CCCNC(c2c[nH]nc2C)=O)cc1Cl C1(N(C(CCSC)=O)C)CCCC2CN(C(C3Cc4ccccc4C3)=O)CC12 Nc1cc(Cl)cc(F)c1C(=O)NCCC(O)CNC(c1cnccn1)=O C1(CNC(C(C(C)(C)O)F)=O)CCC2CN(C(=O)CC3CSCCS3)CCC2C1 Cc1ccncc1C(N1CCOC(CNC(=O)Cc2ccc(Br)nc2)C1)=O C(CC(F)CN=[N+]=[N-])NC(C(CC1CCC1)NC(c1ccc(C(C)C)o1)=O)=O c1(OC)cnc(Br)cc1C(=O)NCC1CCCCN1C(c1n[nH]c(C)n1)=O C(=O)(CN=c1[nH]c(=NCC2(CCO)CCCC2)c2ncccc2[nH]1)NCC c1(N2CCC(C)C(NC(c3c(CC)ncs3)=O)C2C)cc2nnc(C)n2cn1 C1(C(N(CCN(C(c2nc(CCOCC)oc2)=O)C)C)=O)CCn2cnnc2C1 C1(C(=O)NCc2ccc(C(=O)NC(C(C)C)(C)C)cn2)CC1C1CCCC1 c1(C(=O)NCC2(C(N)=O)CN(C(CC3(COC)CC3)=O)C2)cccc(F)c1N C(=O)(C(C)(F)C(=O)NCC1(CNC(c2c(C)csc2C)=O)CC12CCC2)OC C12(C(N)=O)CCCC1(C(=O)NC1CCN(C(c3cnsc3)=O)C1C1CC1)C2 c1(Oc2nc(C)c3c(n2)cccc3)ccc2c(c1)nc(C)c(=O)n2C CC1C(C(=O)NC2CC=CCC2C(=O)Nc2cccc3occc23)=NOC1C c1(NC(C2CCN(C(C(C)NC(=O)C(C)(C)C)=O)C2)C)nc(Cl)nc2c1SCC2 c1(OC)cc(NC(C2CCN(C(c3cn[nH]c3)=O)CC2O)=O)c(Br)cc1C C1(NC(C2(NC(=O)CC3CCCO3)C(C)(C)C2)=O)CCC2(CCC2)CC1 N1(C(CC2(C=C)CC2)=O)CCCC(N(C(=O)CCc2cnn(C)n2)C)C1 C#CCC(C)(C(=O)N1CCC(OCC2CC2)C1)NC(=O)CN(CC)CC C1(C(N(C2CCNCC2)CC)=O)COCCN1Cc1ncccc1C(F)(F)F C1(NC(C(CC)C)=O)CS(=O)(=O)N(C)C12CCN(c1nnc(C3CC3)o1)CC2 C12(NC(CCN(S(C)(=O)=O)C)=O)CC1CN(C(c1nnn(C)c1C(F)F)=O)C2 C12CC(CCC1O)C(=O)OC2=O.C1(N(CC)CC)CCC(C)(C)CC1 C1(CC(=O)NCC2(OC)CN(C(CCS(C)=O)=O)C2)CCC(F)(F)CC1 N1(C(C2(CCC)CC2)=O)CCC(NC(=O)CSC2CCCCO2)C(C)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CC2CC1(CNC(=O)CCc1cccs1)C2 C(CC(C)NC(=O)Cn1cc(-c2ccc(Cl)cc2C)nn1)(C(=O)O)SC C1(Nc2c(OC)cc3c(c2)OCCO3)C2CC3CN(C(=O)OC(C)(C)C)C1C3C2 C=C=CCCC(=O)NC1CCCC1CNC(=O)COc1ccc(F)nc1 C1(O)(C(c2cccc(Cl)c2)NC(C2CC(N(C)C)C2)=O)CCN(C(=O)CC2CC2)CC1 C(CCN=C(NCC12CCC(CC1)OC2)N1CCC(c2cscc2C)C1)OC CC1CN(C(C2(N3CCCC3)CC2)=O)CC(C)N(C(=O)C2=CCCCC2C)C1 c1(CC(N2CCC(O)(CNC(CN(C)C3CC3)=O)C2)=O)nc([N+](=O)[O-])n[nH]1 C1(C(=O)NCC#CCNC(c2ccc(C(C)=O)o2)=O)(OC)CC2CCC1C2 c1(C(=O)NC2C(CNC(=O)Cn3nnc(C4CC4)n3)C2)c(N)cc(Cl)cc1Cl Cc1cccc(C(=O)NC2COCCC2C(N2CCC(F)(C#N)C2)=O)c1O Cc1cc(F)ccc1C1CC1C(=O)NC(C)CC(C)NC(=O)CCCC(C)O C1(CCC)CN(C(=O)CN2CCN(C(c3cc(C)nn3C)=O)CC2)CCO1 C(=O)(NNC(=O)Cn1cnc(C(F)(F)F)n1)C1(C)CCCC1 c1(C(=O)Nc2cc(CO)ccn2)ccc(-c2c(F)ccc(O)c2F)c2cc[nH]c12 C(=O)(C(O)CC(F)(F)F)NCc1ccc(C(=O)NCC2(CO)CC3C=CC2C3)cc1 CC1OC2(C(=O)NCC3C(C)CCCN3C(=O)CC3CCC3)CCC1CC2 N1(C(c2cncc(F)c2)=O)CCN(C(C2CC2c2ccsc2)=O)C2CCC12 c1(-c2c(C)c(C#N)ccc2)ccc2cc(C(=O)NCC3CCO3)[nH]c2c1 C1(C(=O)NCCc2n(CC)cnn2)N(C(c2cncnc2)=O)CCC1(C)C c1(C(=O)NCC(CC=C)NC(=O)CC2(CO)CC2)cnc(C)c(N)c1 c1(C(N2CC(CCNC(C3(C)CC3(F)F)=O)OCC2)=O)[nH]cc2c1CCC2 C1(NC(c2n(C(C)C)ncc2)=O)CC12CCN(C(C1CCCCC1(C)C)=O)CC2 N1(C(CC2CC(=O)OC2)=O)CC=C(CNC(=O)CSc2cn[nH]c2)CC1 N1(C(=O)C=Cc2cnccn2)CCC2CCN(C(=O)CC3CCCS3(=O)=O)C2C1 C(=O)(CC(C)(C)CCC)NC(c1ccccc1F)CNC(C(C=C)C)=O Cc1cc(C(=O)N(C(C)CN(C)C(C2CCCN2N=O)=O)C)ncc1S(N)(=O)=O C(=O)(C(C)C(C)CC)NC1CCC(NC(C(Br)=CC)=O)CC1 CCC1=NOC(C(=O)N(CCC(=O)NC(c2ccncc2)C)CCO)C1 CCS(=O)(=O)CC(=O)NC(C)(CNC(c1ccnn(C)c1=O)=O)C1CC1 c1(C(N2CCC(NC(C3C(CC)OCC3)=O)C2)=O)ccc(Cl)c(Cl)c1O C(=O)(C#CC1CCCO1)NCCC1OCCN(C(c2c(C)[nH]c(=N)s2)=O)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC(C2(NC(c3coc(Cl)n3)=O)CC2)C1 c1(C(=O)NCC2OCCC(NC(c3c(C)nc[nH]3)=O)C2)ncnc2c1CCC2 c12ccc(cc1)C(=O)NC1CN(CC1C)C(=O)c1cc-2on1.C=CCCC1CC1 C(C)(C)(C(C)CC(=O)NC(c1cncs1)C)NC(c1c(C)nccn1)=O CC1CN(C(=O)CCCCCC#N)CC(C)C1NC(=O)CCCCc1cnc[nH]1 C(=O)(C1=COCC1)NC(CC(C)NC(C(CC)F)=O)C C(=O)(N1Cc2ccccc2CO1)C1CC(C)(NC(C(C(C)C)CN(C)C)=O)C1 c1(C(N(CCN(C(CCCOCCC)=O)C)C)=O)ccc(N)c2ncccc12 C1(NCCNC(C(C)NCC)=O)CC2(CO1)CN(C(=O)CNS(C)(=O)=O)C2 N1(C(CSCCC(C)C)=O)CC2ON=C(CNC(c3cc([N+](=O)[O-])n[nH]3)=O)C2C1 C=C(Cl)CC(C(=O)N1CC(=O)NC(=O)C1)NC(c1cn(CC)nn1)=O C1(N(c2nc(SC)nc(O)c2)C(=O)C(C)CN)CCC2(CCNC2)CC1 c1(NC(C2CCN(C(c3cnc(OCF)o3)=O)C2)=O)ncc(Br)cc1Cl N1(C(c2nccc(OC)c2OC)=O)CC(C)N(C(=O)CSCC(N)=O)CC1C C(=O)(C1=CC2CCC1C2)NC1(CNC(c2cnccc2Br)=O)CCOC1 C(=O)(CC(F)(F)C(F)F)NCC1(CNC(C2(C(=O)OCC)CCCC2)=O)CC1 c1(C(N2CC3CN(Cc4ccccc4)CC3C2)=O)ccc2oc(=O)oc2c1 C(C1=CCN(C(=O)CC(C)CF)CC1)NC(c1cn(CC(CC)O)nn1)=O c1(OC)ccc(Cl)cc1C(N1CCCC(O)(CCNC(C2(F)CCC2)=O)C1)=O CCC(C)C(C(=O)N(C1CCNCC1)CCN(C)C)OC N1(C(C(C)OCCC=C)=O)CC(CNC(C2(N(C)C)CC2)=O)CC1C N1(C(CCCCCC#N)=O)CCC(CNC(C2CC3(C2)CC3F)=O)C(F)(F)CC1 c1(C(=O)NCC(CN(C)C(c2ccc3c(c2)NCC3)=O)O)ccnc2ncnn12 c1(C(=O)NCCCNC(c2c(C)nn(C3CC3)c2Cl)=O)cnc2ncccn12 C(=O)(C1=CCCCO1)N1CCC(N(C(=O)CC2CCCCN2C)CC)CC1 C1(NC(CC2CN(C(CC(C)C3CC3)=O)C(C)(C)C2)=O)CN(C)C(=O)C12CC2 C(=O)(C(C)(CO)NC(=O)C(C)n1cncn1)NCC(CC)N(C)C N1(C(c2cccc(SC)c2)C(=O)NC2COC2)CCOCC2(CCOCC2)C1 C1(c2n(C)c(N3CCC(c4ccc([N+](=O)[O-])cc4)C3)nn2)CCC2(CCCCC2)C1 c1(C(N2CCC(CN(C(C(CC)NC)=O)C)CC2)=O)ccc(F)c([N+](=O)[O-])c1C C(c1cc(C)nn1C(C)C)=CC=CC.c12cccc(c1)C2 c1(NC(C)=O)ccc(C(N2CCC(N(C(=O)C(C)SC3CCCCC3)C)C2)=O)s1 C(F)(C(=O)N(C)CC=CC(=O)NCC1(CC2CCC2)CC1)=CCC C1(C(=O)NCCC(=O)NC(C)(C)C)CC(F)CN1C(c1csc(C(F)(F)F)n1)=O Cc1cc(C)c(NC(=O)CSCc2nnc(CCO)s2)c(Br)n1 N1(C(c2ccccc2N2CCC(CO)C2=O)=O)CC2COCC2(CO)C1.CO N1(c2cc(C)nc(N3CCC(C)(CO)C3)n2)CCC2(CCC2)CC1 N1(C(c2ccc(C(C)=O)cc2F)=O)CCC2(CO)CCCC12 c1(CC(=O)N(CC(C)NC(=O)C(c2ccc(Cl)s2)C)CC)cccc2nonc12 C1(C(=O)NCC2N(C(CCCC(=O)NCC)=O)CCC2)CC2CC1CC2(F)F C1(C(=O)NC(C)CCNC(C2(F)CCCOC2)=O)(OCC)CCCCCC1 c1(C(N2CCN(C(CSC)=O)CC2CC(F)(F)F)=O)nc2nc(C)ccn2n1 C(C#Cc1cccc(F)c1F)NC(c1nc(-c2cccs2)no1)C(C)C C(CC(O)C(=O)N1CCCC1CC1CC1)SC.C1(C)(C)C(=O)N1 c1(C(=O)NC(CN(C(=O)CC2CCCN2CCC(C)C)CC)C)cccc(F)c1F c1(C(=O)NCc2scc(C(N(C3CC(C#N)C3)CC#C)=O)c2)ccc(CF)cc1 C(=O)(C#CC1CCCCO1)NC1(C)CN(C(c2cc(Cl)ncc2O)=O)C1 N1(C(=O)NCC(C)(C)N(C)C)CCC(F)(F)C(C(=O)O)C1 C1(C(=O)NCC(C(C)C)NC(C(C(C)C)SCC)=O)CCCCCN1C c1(C(CCO)N(C(CC=C)C)C(=O)NCCCN2CCC(F)C2)ccc(Cl)c(F)c1 N1(C(C(C)OCC)=O)CCCC12CCN(C(=O)Cc1ccc3nonc3c1)C2 c1(C(=O)OC)cc(CCO)cc(NC(OC(=N)O)=O)c1.n1(CCl)cc(CC)nn1 c1(C(N2C(C(=O)O)C3C=CC2C3)=O)ccc2cc(C)ccc2c1 c1(OC)cccc(C(c2ccc(Cl)nc2)NC(c2nc(CCSC)no2)=O)c1 Cc1cc(C)c(C(=O)NCC2CC3(CC(NC(=O)Cc4cc[nH]c4)C3)C2)c(O)n1 c1(COCc2sccn2)n[nH]c(=NC2=NCCCC2)s1 C#CCC(C)(C)C(=O)NCC1CC2(CC2)CN1C(=O)Cc1n[nH]c(=NC)s1 c1(C(C(N2CCN(C(c3cccc(CSC)c3)=O)CC2)=O)C)cccc(C#N)c1 c1(C(=O)NCCCN(CCO)C(C2CC3CCC(C2)O3)=O)cc2ncccc2s1 C=C(CS(=O)(=O)CC)CC[N+](C(=O)C(c1cnccn1)C)([O-])NC.C12CC(C1)NC2=O c1(C(=O)Nc2nc3cnccc3s2)cc2cn[nH]c2cn1 Cc1sc(C(=O)NCC2CCN2C(=O)C(C)(C)C#N)cc1[N+](=O)[O-] N1(C(C2(CC)CCC2)=O)CC2C(CN(C(=O)Cc3cccnc3C)C)C2C1 C1(N(C(C23CC(OC)C2C3)=O)C)CCN(C(C2CCCCN2C(C)C)=O)CC1 c1(C(=O)NC2C(NC(C(CSC)O)=O)CCCC2)nnc(C)c2ccccc12 c1(OCC)nc(C)ccc1C(=O)NC1CCC(CCNC(c2cc(C)c[nH]2)=O)C1 c1(C(=O)NCCN(C(c2ccc(C(C)C)s2)=O)CC)cnc2[nH]c(C)nc2c1 Cn1cccc1C(=O)C(=O)NCC1CCCN1C(=O)CCCc1nc(C(F)F)no1 N1(C(c2[nH]cc(C(N)=O)c2)=O)CC(F)CC1CNC(=O)CCc1cncs1 C(=O)(C(CC(F)F)NC(c1c[nH][nH]c1=N)=O)NCCCCS(C)=O c1(C(N2C(CN(C(C(=O)NCCOC)=O)C)CCC2)=O)cc(OC)ccc1OC C1(C(N(C)Cc2cnn(C)n2)=O)CCN(C(=O)OC(C)(C)C)C1(C)C N1(C(COCC(C)C)=O)CCCOC(C(=O)NC2CC2CCN(C)C)C1 CC1CCN(CC(N2CCC(CC(N3CCCC3CC(N)=O)=O)C2)=O)C1 C1(C(N2CC(c3onc(C)n3)C2)=O)CNC(=O)CN1C(c1ccncc1N)=O [N-]=[N+]=NC1CNC(C(=O)NCC2(Cl)CC2)C1 c1(OCC#C)ccc(C(N2CCSCC2CCNC(=O)CCNC(C)=O)=O)cc1 C1(C(=O)OC)CC2(CCN(C(=O)Cc3csc(C(F)(F)F)n3)CC2)C1 C1(CC)C(NC(c2ccncn2)=O)CCCN1C(C1CC(C)=NO1)=O C(CCCC(=O)NCCN(C(=O)C(C(C)C)c1cnc(C)s1)C(C)C)OC C1(C(=O)NCCN(C(c2c(C)ccnc2C)=O)C2CC2)CCc2n[nH]c(C)c2C1 c1(N(CC(F)(F)Cl)CCOc2c(CC)cccc2)ncnc(C)c1Br c1(CC(=O)OCC(=O)NCc2nn(C)c(=O)o2)nccc2occc12 c1(N(C2CN(C(Cc3c(C)nc(Cl)cc3)=O)C2)C)nc(Cl)nc2c1CC(C)CC2 CC1(C)COC(CC(N2CCC(CNC(=O)CCC3CC3)C2)=O)CO1 CC(C)N=C(NC1CCC1)NCC(c1cc(F)cc(F)c1)O C(CCN=C(NCCc1ccc(C2CC2)cc1)NCC1(Br)CC1)SC C1(C(N(CCC(=O)OC)CC=C)=O)CC(O)CN1C(=O)CC1(C)OCCO1 C1(NC(C(CC)OCC)=O)CC12CC(NC(=O)CCOc1ccccc1)C2 n1(CC(=O)NC2CN(C(c3cnn[nH]3)=O)CC3(CC3)C2)cc([N+](=O)[O-])ccc1=O C1(C(=O)NCCC2CC(NC(c3c(CC)c[nH]n3)=O)C2)CCCCC1(F)F C1(C(=O)NCCNC(CC(N2CCCC2C2CCC2)=O)=O)CCCC1C(N)=O C=C(Cl)C(C)(C)C(=O)N(CCCN(C(=O)CC1CC(O)C1(C)C)C)C C(=O)(C(C)(F)C(=O)NC1CCC(NC(c2ccncc2)=O)CC1)OCC c1(C(=O)NC(CC(=O)OCCC)C(C)C)cc(C)nc2c1nc(C)n2C c1(C(=O)NCc2cc(C)[nH]n2)cc2ncc(-c3ccnn3C3COC3)cc2[nH]1 N1(C(C2CCC(C)C2)=O)CCN(C(c2ccc(CO)nc2)=O)C(C)C1 CC(c1ccsc1)=CC(=O)NCC(C)CN(C(=O)C(CO)N(C)C)C c1(CNCc2ccc(CCCCC)cc2)cc(C)cc(Cl)c1 C(=O)(C1CCCn2ncnc21)NC(C1CCCC1)CNC(c1cncc(OC)n1)=O C(=O)(CCCC(C)(C)C#N)N1CCCC(N(C(=O)CSc2nnnn2C)C)CC1 C1(C)(C(N2CCCC(N(C(CN(C)CC)=O)CCO)C2)=O)CC(C2CC2)=NO1 c1(CC)cc(C(=O)N(CC(C)NC(=O)C(CCSC)OC)CC)ccc1OC c1(NC(C)CCNC(c2conc2-c2ccccc2)=O)ncnc(=N)[nH]1 c1(C(=O)NCC2CCCN(C(c3ccsc3C(F)F)=O)C2)ccc2ccoc2c1 c1(C(=O)NC2C(F)CCN(C(CNS(C)(=O)=O)=O)C2)cccc2nsnc12 N1(C(C2(CC=C)CCOC2)=O)CC=C(C(=O)NCC(c2ccccc2)O)CC1 C1(CC#C)(C(=O)NC2CCCC(NC(C3(C)CSC3)=O)C2)CC=CCC1 Cc1c(NC(C2CCN(C(=O)CC3CC3)C2)=O)ccc(Br)c1Cl c1(CC)cc(C(=O)NCC=CCNC(c2ccc(C(C)F)cc2)=O)cc(Cl)c1 c1(CNC(c2cncc(Br)c2)c2n(C(CC)C)nnn2)n[nH]c(C)c1Cl C1(C(N(CCC)CCNC(c2nnsc2SC)=O)=O)CC2C(C1)C2(F)F n1(C(CC)C)nc(C(=O)N(CC(C)CNC(=O)CC(O)CC2CC2)C)cc1C c1(C(=O)NCC(c2ccccc2)C2CCCC2)ccc2ccccc2c1[N+](=O)[O-] n1(CC(=O)NCC#CCNC(=O)C(F)C(F)(F)F)ncc2ncccc12 C(=O)(C1=CCCC1C)N(CCC(C)NC(c1coc(C2CCC2)n1)=O)C c1(C(=O)NC(C2CCN(C(CSCCCC)=O)CC2)(C)C)cc(C#N)n(C)n1 c1(OC)cc(CN2CCCC(CN(C(=O)CNS(C)(=O)=O)C)C2)c(O)c(Br)c1 c1(C(=O)NCC2C3CN(C(CCCCC=C)=O)CC32)c(F)cc(OC)c(F)c1F n1(C(C(=O)NCC2OCCN(C(CC(C)SC)=O)C2)(C)C)cc([N+](=O)[O-])cn1 N=c1nnn(CC(=O)NCCN(CCOCCO)C(c2ccoc2C2CC2)=O)[nH]1 CC(C)(Cc1ccc(Cl)cc1)CC(=O)NCC1(NC(c2occc2F)=O)CCC1 N1(C(C(CC)n2cncn2)=O)CCCC(NC(c2c[nH]cc2Br)=O)C1 CC1=CCC(C(=O)NC(CN(C)C)C(=O)NCC(=O)NC(C)(C)C)CC1 C1(CC(=O)NCC(C(C)C)(C)NC(c2cncc(F)c2)=O)CCCCC(=O)N1 c1(COC(c2c(COC)ccc(Br)c2)=O)nc2cc(Br)cc(F)c2[nH]1 C1(NC(N2C(c3cc(CC)no3)CCCC2)=O)CCCCC1S(C)(=O)=O CC(C)C(O)C(C)C(=O)NCCCCC(C)NC(c1ccn(C)c1)=O c1(C(=O)NC(C(=O)NC(C=C)(C)C)(C)CO)ccc(F)cc1C CC(CN=c1c(C#N)c[nH]c2c(F)ccc(Cl)c12)N(C)CC1CCC1 c1(OC)cc(C(=O)NCC(O)CNC(=O)C(C)=C(C)C)cc(Br)c1 C1(C(=O)NC2(C)CCN(C(C(C)(CO)OC)=O)C2)CC2(C1)CC(O)C2 c1(N(C)Cc2ccc(OC)nc2)nc(N2CCC(F)C2)nc2cccc(F)c12 Cc1ccc(O)c(CC(N2CCC(C)C2c2cn(CC(F)(F)CO)nn2)=O)c1 N1(C(C)=O)CCC(C(=O)Nc2cccc(NC(C3(N(C)C)CCC3)=O)c2)CC1 C1(C(=O)N)CC2(CCCC2)CO1.C(CC(=O)N(CCCCC)CC)N(CC)CC C1(OCC)(OC)CC(C)(C(=O)NCCN(C)C(c2ccc(C(C)(C)C)nc2)=O)C1 CCC(CC(F)F)C(=O)N1CCC(N2CCN(C(=O)CC(C)CC(C)C)CC2)C1 C1(C(=O)OCc2onc(Cc3c(C)occ3)n2)Cc2nn(C)cc2C(=O)N1 N1(C(CNC(CSCCC(C)C)=O)=O)CCC2CC2C1 c1(C(=O)NC2CC3CCC2N3C(C23CCC(CC2)C3)=O)cc(Cl)c(F)cc1F C(Cc1ccccc1Br)(C(=O)N(O)CC1CCCCC1)NC(C)(C)C.C(N)(=O)O C12(C(N3CCC(C(CNC(Cc4ncc(C)[nH]4)=O)C)CC3)=O)CCC(CC1)CC2 C1(F)(CNC(c2cc(C)on2)=O)COCCN(C(c2ncn3c2CCCC3)=O)C1 Cc1cnc(C(=O)NCC2CN(C(=O)C(C)NC(C3CCC3)=O)CCO2)cc1C N1(C(C2(C(=O)OC)CC2)=O)CC2(CC2C(=O)Nc2ccc(C(C)O)cc2)C1 c1(C(=O)NCCCNC(=O)C=C(Cl)Cl)cc2ccc(Br)cc2o1 c1(OCC=C)ccc(CC(=O)NC2COCC2NC(=O)C(F)OC(F)(F)F)cc1 c1(OCCC)cccc(CNC(=O)C(N2CCCOCC2)=O)c1C CCC(CC)CC(F)C(=O)NCC1CC12CCN(C(=O)C1=CC(C)C1)CC2 c1(OC)c(F)cc(C(N2CCN(C(c3cc(O)ncc3Br)C#N)CC2)=O)cc1F Cc1coc(-c2nc(Cc3cccc(F)c3)nn2C2CCCC2)c1C c1(C(N(CCCNC(C2C(CC)CCC2)=O)Cc2cccnc2)=O)cn(C)cc1C C1(NC(C(c2c(C)cncc2)C)=O)CC1C1CCN(C(c2cocn2)=O)CC1 c1(C(=O)NCC2(NC(CSC)=O)CCOC2)cnn(CCC(C)C)c1C c1(C(C)C)nc(N2CCc3nocc3C2)cc(NCc2cn3ccccc3n2)n1 Cc1cc(OCC(N2CCC2CNC(C2CCCCN2C)=O)=O)cc(C)c1 CN1NC2=NC(=O)C3CC3C(=O)NC1=C2.c1(C(F)(F)F)cc(F)c(F)cc1Br N1(C(c2c(C)sc(O)n2)=O)CCCC(C)(CNC(c2cnn(C(C)C)c2C)=O)C1 Cc1ccc(Br)c(F)c1C(N1CCN(Cc2c(F)cccc2Br)CC1C(C)C)=O C(=O)(C(O)CCNC(=O)CC1CCCCC1)N(CC(=O)N(C)C)CC CC(=O)CC(C)(C)C(=O)N1CCC(C(=O)NCCC2CC3C=CC2C3)(CF)C1 C(c1cccc(CO)c1)=CC(=O)NCC(C)(CO)NC(=O)C(Cl)=CCl Cn1ncc(Br)c1CN1CCCC(CNC(C2CCC(C(F)F)CC2)=O)C1 C(N=c1[nH]c(=NCC(C)C2CCC2)[nH]c2c1CCCC2)c1c(C(C)C)n[nH]c1 CC1CN(C(c2ccc(CC#N)cc2)=O)CC(C)N(C(=O)CO)C1 c1(NC(C2CCCC(NC(Cc3ccc(C)nc3)=O)C2)=O)cc(F)c(F)cc1Br C1(NC(CCCCSC)=O)CC(NC(c2c[nH]ccc2=N)=O)C12CCC2 C1(NC(c2n(C)ncn2)=O)CN(C(C2CCCCNS2(=O)=O)=O)CC2(CC2)C1 N1(C(=O)COc2ccon2)CCC2CCCN(C(=O)CCC(F)(F)F)C2C1 N1(C(CNC(CNC(C)=O)=O)=O)CC2(NC(C3(C4CCCCO4)CC3)=O)CC1C2 c1(NC(C2CC3CC3N2Cc2ccn(CCF)n2)=O)ccc(C2CCOCC2)cc1 C1(C=O)CCCC12CCN(S(=O)(=O)c1ccccn1)C2.N#Cc1ccc(I)cc1 C(C(O)CNC(C1CCOC1)=O)N(C)C(C1CC(CC(C)(C)C)C1)=O C1(CCC)(NC(=O)C2=CSCCO2)CCN(C(=O)CCNc2ccccn2)CC1 c1(OC)cc(CNC(=O)CC2CCCN2Cc2cnn(C3CC3)c2)cc(Br)c1 c1(C(N2CC(C(C)NC(=O)CC#N)OCC2)=O)ccc2cccc(F)c2n1 N1(C(CCC#N)=O)CCC2(NC(=O)CCc3c(F)cccc3F)CCCCCC12 N1(C(c2c(N)c(O)nc(O)n2)=O)CCC2(C1)CN(C(C1CCCCS1(=O)=O)=O)C2 N1(C(c2cc(C)ncc2)=O)CCCC(C)(C)C1CNC(=O)CC(C)C1CCCC1 C1(CN(C(c2c(CC)occ2)=O)C)CCCCN1C(=O)CCCF C1(C(F)(F)F)(C(=O)NCC=CCNC(C=C(C)C(C)(C)C)=O)CC2CCC1C2 C1(C(N2CCCC(C(=O)NCC(=O)OCC)C2)=O)CCC2(CC1)OCCO2 C(C(=O)NC(C)COC(F)F)(C(C)CC1CCC1)N1CC(n2ncc(C)c2)C1 CC1=C(C(=O)N2CCCC2(C)CNC(=O)C(C)(F)F)Cc2ccccc2O1 C1(C(=O)Nc2cn(CCSCC)nn2)N(C(=O)OC(C)(C)C)CC1(C)C N1(C(CC=C)=O)CCC(C2CCN(C(c3cc(CC)ccc3OC)=O)CC2)CC1 c1(C2(C)C(C(=O)NC3(COC)CCNCC3)C2)ccc(F)c(F)c1 n1(C(CC)C)nccc1C(N1CCC1CNC(c1sccc1CSC)=O)=O C1(COc2cccc(OC)c2)CC12CCN(C(=O)OC(C)(C)C)C2 c1(C(N2C(CNC(c3ccc(C)[nH]3)=O)CCCC2)=O)cnc2c(Cl)cccn12 c1(NC(N(OC)Cc2ccccc2)=O)cccc(Br)c1OC(F)F N1(C(c2nn(C)c(C(F)(F)F)c2Br)=O)CC(N)CC2(CCC2)C1 C1(CNC(=O)Cn2ccc(Br)n2)CC2(CCC2)CN1C(C1CC1(F)F)=O N(C(=NCCc1cccc(C)n1)Nc1ccc(OCC)c(OCC)c1)C(C=C)C C(=O)(CC(CC)C(C)C)NCCOCCCNC(C1N(C(C)=O)CSC1)=O C1(NC(C(CN(C)C)NC(C2CC(=O)CS2)=O)=O)CCCC(C2CC2)C1 N1(C(CSC)=O)CCOCC1C(=O)Nc1ccc(-c2ccccc2)nc1 c1(CN2CC(F)CC(C(=O)Nc3c(OC)cc(I)cc3)C2)cc(C)cc(Br)c1O CCN=c1[nH]cc(C(N2CCCC(C(C)NC(=O)C(C)=C(C)C)C2)=O)s1 N1(C(CC2N(C(C(C)=C3CC3)=O)C3C2CCC3)=O)CC2CCC(C1)C(=O)N2 C1(C(N(C(CCNC(C(C)NC(CC)=O)=O)C)C)=O)C2COCC12 c1(C(N2CCC(NC(C(c3c(C)cncc3)C)=O)C2C)=O)cc(Br)cnc1O C1(CNC(C2N(CCS(C)(=O)=O)CCC2)=O)CCC2(CC2)CN1 N1(C(C)(C)C)CC(C(=O)NC2CC(CCNC(c3cnn(C)c3F)=O)C2)CC1=O c1(OC)cc(CC(=O)NCC(C)CN(C)C(C2OCC2(C)C)=O)cc(Br)c1 C1(NC(c2cn(C)nc2)=O)CC2CC1CN(C(c1cc(Cl)ccc1Cl)=O)C2 Cc1cc(C)c(OCCNC(c2ccc(NS(=O)(=O)CC#N)cn2)=O)c(C)c1 C(CCN=c1[nH]c(Cl)ncc1[N+](=O)[O-])N(C(CCCC1C(C)C1)=O)C1CCCC1 C1(c2nnnn2Cc2nnn(C)n2)(NC(CCCC)C)CC2(CCC2)C1 C#Cc1ccc(CC(=O)NC2(CCNC(c3coc(N(C)C)n3)=O)CCC2)cc1 c1(OC(C)C)cccc(CN(C(=O)C(=O)N(C)CCN2CCCC2)C2CC2)c1 c1(OC)ccccc1CC(=O)N(CCCCNC(=O)CC1CCC(C)(C)C1)C N1(C(C2C(CC)CCO2)=O)CC2CC2(CNC(c2nn(C)cc2C)=O)C1 C1(NC(C2=CC(C)CC2)=O)COC2(CCN(C(=O)CCC(C)(C)F)C2)C1 c1(OC)ccc(F)cc1-c1cc(C(=O)NC2CCC(F)(F)C2)ccn1 N1(C(c2c(C)onc2O)=O)CCN(C(=O)CN(C2CCSC2)C)C2(CC2)C1 CC(C)CC(C)C(=O)NCC1(C(C)(C)O)CN(C(c2ncn(C(C)(C)C)n2)=O)C1 CS(C)(=O)=NCCNC(c1cn(C2CCCC2)nn1)=O CCS(=O)(=O)NCC(=O)NCCCN(C(=O)CC1CCCC1)C(C)C n1(CCNC2CCN(c3ncccc3CC)CC2C)cnc2ccccc12 c1(CC(=O)NC(C2OCCN(C(C(C(C)C)(C)O)=O)C2)C)ccc(S(C)=O)cc1 Cc1c(C(=O)NC2(C)CN(C(c3cn(C)c(=O)n3C)=O)C2)[nH]c2c(C)cccc12 CCCC(C)CC(=O)N1CC(C(C)NC(=O)CC(C(F)F)c2ccco2)C1 N1(C(C(n2c(C)ncc2)C)=O)CCC(C)(CNC(=O)C(c2cccnc2)C)CC1 C1(NC(c2n[nH]cc2Br)=O)CCCCC12CCCN(C(c1cnnc(Cl)c1)=O)C2 N1(C(c2c(C)ccs2)=O)CC(NC(c2[nH]cc3c2CCC3)=O)C(C#N)C1 C(C)(C)(CCCC(=O)NCC1CCC1C)NC(C(CC=CCC)C)=O c1(-c2n(C(C=C)C)nc(CC(C)CC)n2)cnn2cc[nH]c12 C1(NC(C2N(C(CC#N)=O)CCCC2)=O)CCCCCCC1CO C(CNC(c1c(C)cnn1C)=O)(CC(=O)NCC=CCSC)OC Cc1n[nH]c(C)c1C(C)C(=O)N(C(C)CNC(c1ccc(F)cc1)=O)C N1(CC(=O)NCC2CC(NC(c3conc3C3CCCO3)=O)C2)CCSCC1 c1(C(=O)NC2C(NC(CCCCOC)=O)CCC2)sc2cccc(F)c2c1CO N1(C(C(CC#C)O)=O)CC(C)(C)CC1CNC(c1[nH]c(O)nc1C)=O N1(C(C2(C)N(C(CCC(C)SC)=O)CCC2)=O)CCOC2(CCC2)C1 c1(NS(c2ccc(OCC#C)cc2)(=O)=O)cc(OC)c(OCC)cc1[N+](=O)[O-] C1(C(=O)NC2C(C)CN(C(=O)Cn3cccn3)C2)CC(S(C)(=O)=O)C1 Cc1cc(C(=O)NCC(CC(C)C)NC(C2CC(C)N(C)C2)=O)ncc1C(N)=O c1(CC(N2CCN(C(c3cnns3)=O)CC(O)C2)=O)coc2c(Cl)c(Cl)ccc12 C(=O)(C1Cc2ccc(F)cc21)NC1C(NC(=O)COCc2nc[nH]n2)CS(=O)(=O)C1 N1(CC)CCC(NC(C2OCCC2CNC(c2cc(C)n(C)c2)=O)=O)C1=O c1(C(=O)OCC)nc(C(C)OCC(F)(F)F)n(-c2nc(C)nn2C)n1 CC1(c2cn(Cc3ccno3)nn2)CCN(C(C2(S(N)(=O)=O)CCC2)=O)CC1 C1(CNc2cc(C(C)=O)ncn2)CN(C(c2nnc(C)cc2O)=O)CC1(C)C C=CC(C)(C)CCCNC(=O)C(C(C)OC)NC(c1cc(CC)ccn1)=O Cn1cc(C(F)=CC(=O)NCC23CC2CN(C(=O)CN2CCCOC2=O)C3)cn1 C=C1CCN(C(c2sccc2OC)=O)C(C(=O)NCC23CC(CN2C)C3)C1 C1(N2CCN(c3nccc(OCC)n3)CC2)CCCCN(C(=O)CNC(N)=O)C1 N1(C(C(C)OCCN(C)C)=O)CCC(F)(CNC(c2csc(Cl)c2)=O)CC1 c1(OC(C)C)cc(NCCC2CCC(NC(=O)C(C)(O)C3CC3)C2)ncn1 C1(C(=O)NCCN(C(=O)CCc2nnc(C(F)F)o2)CCOC)CCS1(=O)=O N1(C(C(F)=CCC)=O)CC2(CNC(=O)C(CCSC)N(C)C)CC1CCO2 CC1C(=O)CC2CCC1N2C(c1ccc2c(c1)CCN2)=O C1(NC(=O)CCC2CCCCO2)CCCOC12CCN(C(=O)COCCF)CC2 c1(CCNC(C(=O)NCCCS(=O)(=O)Nc2ccccc2)=O)c(Cl)ccnc1Cl N1(C(Cn2ncc(CC)c2)=O)C2CCC1C(CNC(C1CC1(C)C)=O)C2 C(=O)(C(O)CC(C)C)NC1(CCOC)CCN(C(C2(CC#C)CC=CCC2)=O)C1 C(=O)(C(CP(C)(C)=O)C(F)(F)F)Oc1c(C)oc(C(N2CC3(CCOC3)C2)=O)n1 c1(C(N(C(C)C)CCNC(c2cnc(Cl)s2)=O)=O)ccc2c(c1)C(=O)NC2=O C1(NC(=O)CCc2nccs2)CC2CCC1N(C(=O)CC1CCCC1)C2 c1(OC)ccc(C(=O)OCC(=O)NCC(c2ccccc2)C)cc1 c1(NC(C23C(CN(C(C4CCC(=C)CC4)=O)C2)C3)=O)cc(Cl)cc(Cl)c1Br c1(C(CNC(=O)C(C)=C2CCC2)NC(CC(=C=C)C)=O)ccc(F)cc1F C1(C(N(C2(COC)CC2)C)=O)CN(C(C2(F)CCCCC2)=O)CC(C)O1 N1(C(C)=O)CCOCC1C(=O)NC1CCC(CNC(=O)CCCn2ccnn2)C1 c1(OC)ccccc1C(N1CCC(F)(C(=O)NCCCP(C)(C)=O)C1)=O c1(C(=O)NCCN(CCC)C(c2cnc(C3CC3)o2)=O)cc(Cl)cc(Cl)c1 CC1(C)C2CC1CN(C(C1CNC(=O)CN1C(=O)CC(F)(F)F)=O)C2 C12CN(C(C3CCCO3)=O)CC1C(C)C2.N1(CCC)CCCC1CC(N)=O N1(C(c2ccc(SC)o2)=O)CCC2CC12C(=O)NCCCC1CCOC1=O c1(C(N2CCC(N3CCCCC3C)CC2)=O)ccc(Sc2cc(C)[nH]n2)cc1Br CC1(C)OCCN(C(=O)OC(C)(C)C)C1C(=O)NCc1cc(Br)ccn1 C=CCC(C)(CC)C(=O)NCc1csc(C(=O)NC(C)C(O)C(F)F)c1 C12(C(=O)NCCC(C)N(C)C(c3ccc(CO)cn3)=O)CC(CO)(C1)OC2C C1(C(=O)NC2(CO)CCN(C(C(CC(=C)C)C)=O)CC2)CC2OC(=O)OC2C1 N1(C(c2nnn(C)n2)C(=O)NC2CC(F)(F)C2)CCN(Cc2nc[nH]n2)CC1 c1(C(C(=O)NCc2cc(N3CC(C)OCC3)ncc2)=O)ccc(F)cc1F c1(OC)cc(CCC(=O)NCCC(C)N(C(=O)C=C(C)C(C)C)C)ccc1F c1(C(=O)NC2C3CN(C(C(C(C)O)C)=O)CC2C3)ccc2nccnc2c1 Cc1cc(=NCc2cccnc2Br)[nH]c(=NCc2cccc(N)c2)[nH]1 C1(C(N(CCNC(C2C(=C)C2C=O)=O)CCC)=O)COCC2(CCC2)O1.CC C1(NC(CSCCC)=O)CCCC12CN(C(C1C3C4CCC(C4)C13)=O)C2 C1(CNC(c2cc(SC)oc2)=O)CN(C(C2CC3(CC(OC)C3)C2)=O)C(C)(C)C1 c1(C(=O)NC2C=CCN(C(=O)C(O)C3CCCC3)C2)cncc2nc[nH]c12 c1(C(=O)NCC2(O)CN(Cc3cccc(OCCC)c3)C2)nccc2[nH]ccc12 C=CC1(CC(=O)NCCCOC(=N)O)CN(C(C2CCC(CO)CC2)=O)C1 C1(C(N(CC(C)NC(C(CCSC)O)=O)C)=O)CCC2C(C1)C2(F)F c1(C(=O)NC2(C3CN(C(=O)C4CC4)C3)CC2)cc2c(Br)cccc2o1 N1(CC2CCC(COC)CC2)CCC(NS(C)(=O)=O)CC1.C=C1CC12C(=O)NC2 N1(C(C2CCC(=O)C2)=O)CC(F)CC1C(=O)NCc1cnco1 c1(C(C)C)nc(NCC(C)CCO)cc(N2CCC(CCCO)C2)n1 C(=O)(C1OCCn2ccnc21)NC1C(CC)N(C(c2ccc(F)cn2)=O)CC1 N1(C(CCCC(CC)C)=O)CCN(C(=O)CC2CCCS2(=O)=O)C2(CCC2)C1 Cc1n[nH]c(C)c1CC(C)C(=O)NCC=CCNC(=O)CCC1CCCCN1C c1(N(C)C)ccc(C(=O)NCC2CCCC=C2Br)c(F)c1 C(=O)(C(C)CNC(=O)C(O)CNC(c1cnc(S)[nH]1)=O)OC(C)C C1(NC(Cc2c(C)ocn2)=O)CCN(C(=O)CC23COCC(C2)C3)CC1 CC1CCN(C(=O)C=CCN2CCC2)C(NC(c2cc(=O)n(C)cn2)=O)C1 N1(C(CNC(C2C(C)C2)=O)=O)CCC2(CCN(C(C3C4CC(=O)CC34)=O)C2)C1 C(=O)(CCCCCC#N)N1CC(CC(=O)NCC(C)C(C)(C)C)OCC1 N1(C(C(C)(C)N2CCCC2)=O)CCOCC(F)(Cn2cc(CNC(N)=O)nn2)C1 C1(COC)CN(C(C2CC(=O)N(C)C2)=O)CCN1C(c1ccc(C(C)=O)cc1)=O C1(C(=O)N(CC(C)(C)NC(=O)C(C)NC(N)=O)C)(COC)CCOC1 c1(OC)coc(C(=O)N(C2CCC(NC(=O)CC(=O)N(C)C)C2)C)cc1=O CCC(C)(CCNC(=O)Cc1cc(C)nn1C)NC(=O)Cc1cncc(F)c1 C=CCCCCCCCC(=O)NCC1CC1CNC(c1cncc(Cl)c1C)=O N1(C(C2CC23CC3)=O)CC2CCN(C(C3C4CCC5C(C4)CC35)=O)C2C1 N#CC1(NC(C2CCN(C(c3c(I)ccnc3F)=O)CC2O)=O)CCOCC1 C(CC1=CCOCC1)NC(CN(C(=O)C(CC(C)C)OC)CCC)=O c1(C(N2CC(NC(CC=C=C)=O)C(F)C2)=O)cc(Cl)c(C)cc1OC N#Cc1cccc(CCC(=O)NC(CNC(=O)Cc2cnn(C(F)F)c2)C2CC2)c1 C1(CN(C)C(c2ncc[nH]2)=O)CC(F)CN1C(=O)CC1CCC(C2CC2)O1 N1(C(C2(CCNC(C3(CC(C)=O)CC3)=O)CC2)=O)CCSCC(C)C1 C1(NC(C2(C)CCC3CC3C2)=O)CC2CCC1CN2C(C1(C(N)=O)CC1)=O Cc1c(NC(C2CC(C)CN2C(=O)C(C)NC=O)=O)cccc1CO C1(C(=O)NCC2N(C(C=CCCC)=O)C3C(C2)C3)CC2(CCCCC2)S1(=O)=O C1(CC)(NC(C2CC(F)C(=O)N2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1 N1(c2ccc(OC)cc2OC)C(=S)NC(c2ccco2)C2=C1CCCNC2=O C1(C#N)(C(=O)NC(CC#C)C(=O)NC2CC(C)(CC)C2)CCCOC1 C1(NC(C(=O)NCCC2CC(C)(C)OCC2)=O)C2(CCC2)C12CCC2 Cc1cc(CCC(=O)N(CC(c2cccc(C(=O)O)c2)=O)C)cc(C)c1 N1(C(C2CC=C(C)CC2)=O)CCN(C(c2cccc(F)c2)=O)CC(O)C1 C(=O)(C(C)(C)CC(F)(F)F)N1CCC(CN=c2nc(CCOC)[nH]s2)(C)CC1 CC1CC(C)(C(N2CC(NC(C3CC(N4CCOCC4)C3)=O)C(O)C2)=O)CCO1 N1(C2CN(C(c3cc(C(C)=O)sc3)=O)C2)CC(NC(c2nsnc2O)=O)CC1=O c1(CNC(c2ccc(COC)o2)=O)ccc(SC)cc1.C12(CCOC1)C(=O)N2 N1(C(=O)CCOC2CCOC2)CCC2(CC1)CN(C(C1CCC1(F)F)=O)C2 N1(C(C=CCCC=C(C)C)=O)CC2CC1CC2NC(=O)C=Cc1ccc(C(F)F)o1 C1(NC(=O)CN2CC3CC3C2)CCN(C(c2ccc(C3CC3)cn2)=O)CC1F C(CCC(C)C)(C(=O)NCC1(C(C)(F)F)CC1)NC(C(C(=O)OC)OC)=O CC1COC(CO)CN1C(C1CC(C)(NC(=O)CCOC(=O)CO)C1)=O C1(CNC(C(C)(C)C)=O)CCCC2(CCN(C(c3c[nH]nc3F)=O)CC2)O1 C(=O)(C(O)C1=CCCCC1)N1CCCCC(NC(C(=O)N(C)C)=O)C1 Cc1cc(=NC(C)COC(C)(C)C)[nH]c(=NCC2CC(C)CO2)[nH]1 C(=O)(C1CCc2nccn21)N1CC(CNC(c2c(CC(C)C)onc2)=O)C(O)C1 C12(NC(=O)COCC3CCCC3)CCCN(C(c3cccc(Cl)c3)=O)CC1C2 CCC(C(=O)NC(C)(C)CNC(c1cnc(OCC)s1)=O)n1ccc(C2CC2)n1 C#Cc1ccc(OC)c(C(=O)NCC=CCNC(=O)CC2OCCC2C)c1 N1(C(C=Cc2ncc(C)[nH]2)=O)C2CCC1CN(C(=O)C(C)S(=O)(=O)C(C)C)CC2 Cn1cnc2nc(=NC(C)CCO)[nH]c(CCNCCCC(F)(F)F)c12 c1(C(=O)OC(C)(C)C)ccc(N2CCOC(CCC(F)(F)F)C2)nc1 C(=O)(CCCCCF)NC(C)(CNC(=O)CC1CC2C=CC1C2)C1CC1 CC1CSCCN(CC(=O)N(C)C(c2n[nH]cn2)c2ccco2)C1 N1(C(C2(C)CCN(C)C2)=O)CCC(N=[N+]=[N-])(C(N2CC(N3CCCC3=O)C2)=O)C1 N#Cc1c[nH]cnc1=NCC1CCC2(CCC2)C1NC(c1cncnc1)=O C(=O)(C(O)C(F)(F)F)Nc1cccc(CNC(CC2C(CC)C2(F)F)=O)c1 N(C1CCCc2sc(Cl)cc21)C(Cc1c(C)oc(-c2ccco2)n1)=O N1(C(c2ccc(C)cc2O)=O)CCC(C)N(C(=O)CC2CC(O)C23CCC3)CC1 n1(CC)cc(CNC(C2CCC(CNC(=O)C(C)SC)C2)=O)cn1 C1(CN(C(C2NCCOC23CCC3)=O)C2CC2)CCCC2(C1)OCCO2 c1(-n2c(C(c3c(C)scn3)NC(C)CCF)nnn2)ccc(Cl)cc1F C(CCC(C)CC(C(=O)NCC1CCOC1)N1C2CCC1CN(C)C2)=C(C)C C1(C(C)C)CCC(C(N2CCOCC2CNN(C)C(C2CC2(C)C(F)F)=O)=O)CC1 c1(C(C(=O)NC(CC)C)N(CCCC(C)(F)F)C)cc(C)ccc1Cl N(C1CN(C(c2cnoc2)=O)CCc2ccccc21)C(CCC(C)(C)C)=O C(C)(C(C)(C)C(=O)N(C)CC1(C)CCCC1)NC(COCCSC)=O C(=O)(CC1C(=O)Nc2cc(OCC)ccc21)NCCCNC(CCCC(=C)C)=O c1(NC(c2nccn2C)CC)ncc(C)cc1S(=O)(=O)N(C1CCN(OC)C1)C C(CN=C(NCc1ccc(F)cc1O)N1CCC(OC)C(OC)C1)OC N1(C(CSCC)=O)CCCC(C2CC2NC(=O)C(F)OC)C1 C12CCCN(C1)C(=O)C1CCCC21.c1(S)ccc(C(F)(F)F)cn1.CO C1(CNC(C2(COC)CCOC2)=O)CCCCN(C(c2cc(O)ncc2F)=O)C1 N1(C(CCCC=C)=O)C2COCC1CC(NC(=O)CC1CCCO1)C2 Cc1ccc(C(C)(C)C(=O)NC2CCC(N(C(=O)CCC3(C)CC3)C)C2)cc1 Cc1cccc(C=CC(N2CC3CC2C3NC(=O)C(C)Oc2ccccc2)=O)c1 N1(C(C2C(NC(Cc3cnc(C)s3)=O)COC2)=O)C(C)CCC1(C)C c1(-c2c(OCC)ccc(F)c2)cnc2c(C(=O)NC(CO)CC(C)C)cccn12 c1(C(=O)NCCN(CCCCCC)C(=O)C(C)C#N)c(Cl)nsc1Cl C1(C)(C(=O)NCC2C=CC(NC(COCCC#C)=O)C2)CCCN1C c1(OC(C(N2C(C)(c3nn[nH]n3)CC2)=O)CO)ccc(Cl)cc1[N+](=O)[O-] C12CN(CC1CC1CCCCC1)NC(=O)N2.c1(OC(C2(C)CC2)=O)ccccc1 N1(C(c2ccoc2Cl)=O)CC(C2CCCN(C(C3CCC4CCC3O4)=O)C2)C1 C(=O)(CC(=O)NC(c1ccccc1)C(C)NC(C1(C(=O)OC)CC1)=O)NC C1(NC(C2N(C(C3CC(OCC)C3)=O)CC(O)C2)=O)=CC=C2C=C2SC(Cl)=NC=C1 c1(C(N2C(CNC(C(=O)NCC)=O)COCC2)=O)cc(F)c(F)cc1I C1(CN(C(C2(SC)CN(C(C34CCCC3C4)=O)C2)=O)C)CCCC1(C)C c1(N2c3cncc(c3)C2=O)ncc2c(ccn2C)n1.C1CCNC1.CCO c1(C(=O)NC(C#C)CO)nnn2c1CSCC2 c1(C(=O)NC2(CO)CCN(C(Cc3c(C)ccs3)=O)C2)ccc2nn[nH]c2c1 c1(C(N(C2CCCC(NC(c3c(C)ocn3)=O)C2)C)=O)ccc2nnn(O)c2c1 N1(C(C(CC=CC)CC)=O)CC2(CCN(C(c3c(C)nsc3N)=O)CC2)C1 N1(C(C(COC)OC)=O)CCC2CN(C(c3ccnc(OC(C)C)c3)=O)CC12 C1(NC(COCC(=C)C)=O)CC(C(=O)NC2CCSC2)C1 c1(CNC(NC2C(C)C2)=NCCc2ccc(F)cc2)ccc2c(c1)CCC2=O CCCCC(C)CCC(=O)N1CC2CC(C1)CN(C(C1(C#N)CCOC1)=O)C2 C(=O)(C(F)C(F)(F)C(F)(F)F)NC1CCN(C(CNC(=O)OCC=C)=O)CC1O c1(NC(C2(O)CCN(C(c3nc(CC)sc3)=O)CC2)=O)cc(F)c(O)cc1C C1(CCC)CN(C(c2cc(C3(C)CC3)on2)=O)CCN1C(=O)COC1CCC1 N1(C(C(C)C2CCC2)=O)CCCCC2(C1)CN(C(C1(CO)CCCC1)=O)C2 Cc1cc(C(=O)N(C2CN(C(=O)Cc3sccc3Br)CC2O)C)oc1C c1(OC)cc(Cl)sc1C(N1CCC1(C)C(=O)Nc1ccccc1SC)=O C(=O)(C(F)(F)C(F)(F)F)Nc1cc(C(=O)NC)cc(C)c1 Cc1cc(C(=O)N(CCCCNC(=O)CC(C)C)C)c2c(C)n[nH]c2n1 c12cc(ccc1C)CNC(=O)CCO2.C(C)(C)(C)CCNC(C)=O N1(CC(=O)NCC2C(NC(C(C)OCC(C)C)=O)CCCC2)CCC(=O)NC1=O N#Cc1csc(C(=O)NCC2(NC(=O)CC3CCCS3(=O)=O)CCOCC2)c1 N1(C(C2CC(=O)C2)=O)Cc2n[nH]cc2C1C(=O)NCc1cccs1 Cc1sc(C)c(C(=O)NC2CCCC2CNC(=O)C2=CCSC2)c1C#N N1(C(C=Cc2ccc(C)cc2)=O)C2CCC1CN(C(=O)CC1CC1C(F)(F)F)C2 n1(CC)cc(C(N2CCCC2CN(C(=O)C(F)(F)c2csc(C)c2)C)=O)cn1 CCC(C)(CC)C(=O)N(CC(C)NC(c1cc(C)ccc1Cl)=O)C C1(NC(c2n(C)nnc2)=O)CCN(C(=O)CSc2cccc[n+]2[O-])CC(O)C1 N1(C(CN(C(C)=O)CC)C)CCC(n2cc(CNC3CCOCC3)nn2)C1 O=C(C1COc2ccc([N+](=O)[O-])cc21)N1CC2CC2(NC(C2(CF)CCC2)=O)C1 Cc1ccc(C)n1CC(N1CC2CC1C2CNC(=O)C(c1cncn1C)O)=O C(CCCC(F)(F)F)NC(C(C(C)NC(=O)CN(C1CCC1)C)C)=O CCC(C)(CNC(C1CC1c1ccco1)=O)NC(=O)CCc1cnccn1 CC1(CNC(C2C=CC=CC=C2)=O)CCCN(C(C2(CO)CCCO2)=O)C1 c12nc(ncc1Br)C(=O)N2.c1(SC)ccc(OCCO)nc1 N1(C(CC(C)(C)C)=O)CC2CC(NC(c3cnn(CC(F)F)c3C3CC3)=O)CC1C2 C(=O)(C1Cc2ccc(F)cc21)N1CCC(NC(CCc2ccc(C)s2)=O)C1(C)C CCCCCCC(C)(CCC)C(=O)NCC(C)NC(c1c(C)cc(C)oc1=O)=O O=C(C(CCc1cn[nH]c1)NC1(c2ccc(Cl)cc2)CC1)NCC1CC(F)(F)CO1 c1(C(N(C(C)C)CCN(C(=O)CCNC(=O)C=CCl)C)=O)ncccc1F c1(CC)cc(N2CCOC(CNC(=O)C(C)n3cccn3)C2)nc(C)n1 Cc1ccc2[nH]cc(CC(=O)NCCCCCCNC(C3(C#N)CC3C)=O)c2c1 N1(C(CSSC)=O)CCC2(COC(CNC(=O)Cc3cn[nH]c3)C2)C1 C1(NC(c2cscn2)=O)COC2(CCN(C(=O)CCCCC(F)(F)F)C2)C1 CC(C)CC(C(N)=O)NC(=O)Cc1cnc(C(F)(F)F)s1 C1(CC)CCCC(C(N2CC3CC2(c2nc(N4CCCCC4)no2)C3)=O)C1 CC(C)(CS(N)(=O)=O)C(=O)NC1CN(C(c2ccc(=N)[nH]c2Cl)=O)CC1O c1(NC(C2(CNC(c3c(C)nc(Br)cc3)=O)CC2)=O)ccc(S(C)(=O)=O)c(Br)c1 C(CC)(C(=O)N1CC(C(=O)NC(c2csnn2)C)(COC)C1)OCC c1(C(=O)NCC(C)(C2CCC2)NC(C(CCC)O)=O)ccc2c(c1)N(C)CC2 C(c1ccc(C)cc1)=CC(=O)NCC1(CNC(CC(CC)OC)=O)CCC1 C#Cc1cccc(C(=O)N(C2CCCN(C(=O)C(CC)C(=O)OC)C2)C)c1C N1(C(CC#N)=O)CC2(CO)CC1(CNC(=O)CS(N)(=O)=O)C2 C1(NC(C2CCCC3(CC3)C2)=O)CCCCCC1NC(C12CCN(CC1)C2)=O Cc1nccc(CCC(=O)NCC2CC2CNC(=O)C(C)OC2CCCCC2)n1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)C=Cc2ccc(Cl)cc2)CC1C C1(CNC(c2cc3sccc3s2)=O)C2CCC(C2)N1C(=O)CC1CC=CCC1 c1(C(N2C(C)CC(CNC(CN(C(C(C)C)=O)C)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(CC(COC)NC(C2CCCCC2O)=O)=O)CCCNC(=O)C1 C1(C(C)NC(CSCC=C)=O)CCN(C(c2ccc(N(C)C(C)=O)cc2)=O)CC1 C1(N)CCCN(C(=O)Cc2cnn(CC)c2)C1COC.C(CC=O)=CCC N1(C(c2c(C)snn2)=O)CC2CCC1CN2C(c1ccccc1C(C)(C)C)=O C1(C(C)NC2(C(=O)OC)C=CCC2)CC2(CCCC2)CO1 C1(C(c2n(C3(C)CC3)nnn2)NCc2ccnnc2)CCCC(C)(C)C1 CCCC(C)(C)C(=O)N(CCNC(C1(F)CCOC1)=O)C1CC1 C1(COC)CN(C(C2OCCOC2(C)C)=O)CCN1C(=O)CCCCCF c1(CC(=O)NC2CC(F)(CNC(c3cc(CC)ncc3)=O)C2)c[nH]c(=N)nc1O c1(C(=O)NCC(CNC(C2(COC)CCCC2)=O)CO)cccc(Cl)c1 N1(C(CC=C(C)C)=O)CCCC2(CNC(c3cnc(C4CC4)s3)=O)CCCC12 Cc1c(C)c(C)c(C(N2CCCCCC(NC(C3CCCO3)=O)C2)=O)c(C)c1C Cc1cnc(C(N2CC=CC(NC(C3CNC(=O)N3C)=O)C2)=O)c(C)c1 C(C(C)(C)C(=O)NCC1CN(C(=O)C=C(C)c2ccco2)CC1O)SC N1(C(C(C)Cc2ccco2)=O)CCC2(CC(C(=O)N3C4CCC3COC4)=NO2)C1 CCC(C(=O)Nc1nc(C)c(C(N2CCOC(CO)C2)=O)s1)C(C)C N1(C(CC)=O)CCCN(C(C2CN=C3N=CNN3C2)=O)CC1C C1(CNC(CSCC=C)=O)C2CC1N(C(c1scnc1CC)=O)C2 c1(-c2cc(CS(N3CCC(OC(C)=O)C3C)(=O)=O)no2)ccc(Cl)cc1 c1(C(C(=O)OCC(C)CN(C)C)Sc2ccccc2)cnn(C)c1 N1(C(C2C(CC)CCCC2)=O)CC2CN(C(=O)C(F)=C3CCCC3)CC12 c1(OC)cccc(C(=O)O)c1OCC(C)C.n12ncc(c1C)NC(=O)CC2 C1(C(=O)NC)CS(=O)(=O)CCN1C(c1ccc2c(c1)CCC2)C(=O)NCC(C)C C=CC(C)(CCOC)C(=O)N1CCC(CNC(=O)Cc2ccoc2)C(F)(F)C1 N1(C(C(C)(C)C#N)=O)CCCC2(NC(C3CCC=CO3)=O)CC2C1 C1(C(N2CC(O)(CCNC(CCOCC#C)=O)C2)=O)CCN(CC(F)F)CC1 C1(COC)(NC(=O)C(C)C2CCCC2)CCN(C(c2cnccc2Br)=O)C1 N1(C(c2c(C(C)(C)C)c[nH]c2)=O)CC(NC(c2ccsc2Cl)=O)C2(CCC2)C1 C(CCC(C)C(=O)N(CCCN(C(=O)C(c1ccc(F)cc1)CO)C)C)OC CCC(C)C(C(=O)N1CCC(C(=O)NCCCOC(F)(F)F)C1(C)C)N(C)C c1(CCC(=O)NCCCOCCNC(=O)C=CC=C(Cl)Cl)cc(Cl)no1 CC(C)CCCOCC(N1CCC(N(C(=O)CC2CCC2(C)C)C2CC2)C1)=O c1(OC)cc(C(N2CCCCC(C(=O)Nc3ncc(C)nc3C)C2)=O)cnc1Cl N1(C(C(C2CC2)OCC)C(=O)NC(c2ccccc2)C)CCC2(CC1)OCCO2 CCCCC(C)C(=O)NCC1COCC1NC(c1nc(Cl)ccc1OCC)=O c1(C(=O)NCC2N(C(COC(CC)C)=O)CCCC2)cc2cc(N)ccc2[nH]1 C(CC(C)C)(C(C(=O)NCSc1ccccc1)N1CCC(F)(CF)C1)OC C#CCC(C)(CC)C(=O)N1CCN(C(C2CCN(c3ccccn3)CC2)=O)CC1 C(C)(C)(CC(=O)NC(=O)NC1(C)CCCCC1)N(C)C(=O)C1CC1 c1(C(=O)NCC(C)NC(c2nocc2C2CC2)=O)c(O)nnc2c1CCCC2 c1(CC)nn(C)c(CC)c1C(N1CCCC(CC)(NC(c2sccc2Cl)=O)C1)=O c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CCC2)c(C)cc(Cl)cc1C C(=O)(C1CNc2ccccc21)N1CCCC(C(C)NC(c2ccc(O)nn2)=O)C1 C(=O)(C(=O)N1CC(O)CCO1)NCc1cnc(CC)s1 C(c1c(F)ccc(Cl)c1F)=CC(=O)NC1C(C)(C)CN(C(C2CCC2(C)C)=O)C1 c1(SCCCC)cccc(C(=O)NC2CN(C(C3COC(=O)C3)=O)CC2C)c1 S(=O)(=O)(c1cc(C=CC(=O)N(C)C(C)C2CC2)ccc1OC)NC C=CC1CN(C(C2(c3cccc(C)c3)CC2)=O)CC1NC(=O)CN(C)C C1(NC(C2(CC#C)CCCO2)=O)CCC2CN(c3ncnc(C)c3Br)CCC2C1 Cn1cnc2nc(=NCCc3cc(Br)ccc3Cl)[nH]c(NCCc3cc[nH]n3)c12 C1(OC)CCC(C(N2CCC3(C2)C(=O)N3)=O)CC1.O(C(=N)O)CCO CCCCCCCCCC(=O)NC(CNC(C1CC(C)(C)CN1C)=O)CC C(CC(C(=O)NCCc1[nH]nnc1CN)c1ccccc1)=C(C)C c1(C(=O)NC(C(C)NC(c2c(SCC)nccn2)=O)C)cc(C)c(Cl)c(C)c1 C1(CCCC)CN(C(c2cnoc2C)=O)CCN1C(=O)COCC(C)(C)C C1(C(=O)NCCC2CCCN2C(C2CCOCC2)=O)CC2CCC1O2 N1(C(C(=O)N(C)C)=O)CCC(C(F)(F)F)C(CNC(=O)C(O)c2ccco2)C1 N1(C(c2c(C)nccn2)=O)CCC2CC2(C(=O)Nc2ccc(CCO)cc2)CC1 c1(CC)nc[nH]c1C(=O)NC1CC1NC(=O)Cc1ccccn1 Cc1ccc2c(n1)CN(C(=O)C(C)CN(C)C(C1CCC1C)=O)C2 C1(CNC(=O)Cn2ncnn2)COCCN(C(C2(C(F)F)CC2(F)F)=O)C1 c1(CNC(C2(NC(=O)CC3(C)CC3)C(C)CCC2)=O)cc2n(n1)CCC2 N1(C(c2cc(C)c(Br)cn2)=O)CC2(COC(CNC(c3ccncn3)=O)C2)C1 c1(CC)cc(O)ccc1NC(=O)CCN(C(=O)C(C)C1CCC1)CCCO C1(NC(c2cc(F)cc(Cl)c2)=O)CC2CCC1CN2C(=O)CC1CCCC1O C12(C(=O)NCC3CCC(NC(C(C(C)SC)O)=O)CC3)CC3CC(CC(C3)C1)C2 c1(C(N2CCC(C(=O)NC(CCC(C)C)C)(C(C)C)C2)=O)cccn2ccnc12 c1(OC)nc(C)ccc1C(=O)NC1CC(CNC(C2C(C)CC2C)=O)C1 C(=O)(CC(C)(C)F)NCC(CCOC)NC(=O)CCCN(C)C(C)=O C(C(CC)(CC)C(=O)N1CCC(OC(C)C)C1)NC(C(C=C)CC)=O c1(N(C2CCCN(C(C(NOC)=O)=O)C2)CCO)ccc([N+](=O)[O-])cn1 c1(C2(C(=O)NCC3C4CN(C(C5C(C(C)C)C5)=O)CC43)CC2)cccc(Cl)c1F C1(NC(C2C(C(C)O)C2)=O)CCSC12CN(C(c1cc3n(n1)CCC3)=O)C2 c1(C(N2CC(O)(CCNC(C3CCC34CCCO4)=O)C2)=O)ccnc2c1CCO2 N1(C(CC2(OC)CCC2)=O)CCC(COC)(NC(C2CC=CCC2)=O)C1 c1(CC)cc(=NCC(C2CC2)NC(C2(C)CCC(C)C2(C)C)=O)[nH]c(CC)n1 C1(CNC(=O)NCC2CC(SC)C2)CCCOCC1 C(CSC)(C(=O)N(CCC(=O)NC1CCSC(C)C1)OC)OC N1(CCCC(=O)NC(CC=C)CNC(C2CCC2OCC)=O)C(=O)CNC1=O CC1CC=CCC1C(=O)NCC(CO)NC(c1cc(CO)[nH]n1)=O C(CCC(C)(C)NC(=O)CNC(C1CCOCC1)=O)NC(c1ccc(SC)s1)=O C1(C(=O)NC(C2CN(C(C3(CC#C)CC3)=O)C2)C)CC(C)(C)C1 C=CC(C(=O)N(CCCOCCNC(C1CCS1(=O)=O)=O)C)OC N1(C(c2nn(CC)c(O)c2)=O)CCCC(CC)(NC(C2CC(N(C)C)C2)=O)C1 O=C1CC(C2CC2)(C(=O)NC2CCN(C(=O)C=Cc3cncs3)CC2CO)C1 N1(C(CC(=O)OC)=O)CCc2c(CNC(=O)C(=CC3CCCC3)C)cccc2C1 c1(C2C(C)CC2)nc(-c2ccncc2)nn1Cc1cccnc1 c1(C(=O)NCC2(C(N)=O)CN(C(C3COCCC3(F)F)=O)C2)ccnc(Cl)c1O C1(O)(CN(C(CC2CC(=C)C2)=O)C)CCN(C(=O)C(C)CC2CCC2)C1 C=C=CC(C)C(=O)N1CCC(OCCNC(C2(C(F)(F)F)CC=CCO2)=O)CC1 C(=O)(CC(C)(C)C(=O)N1CCCC(NC(c2cc(C)c(C)[nH]2)=O)C(F)C1)OCC C1(CC)CC(C(=O)NC2CCC(C)CC2)CCN1C(=O)C#CC(C)C N1(C(C(C)OC2CCCC2)=O)CC2(CCNC(=O)C=CC(C)(C)C)CCC1C2 Cc1cc(C(N2CCN(C(=O)C3CC3)C(C(C)C)C2)=O)c(C)n1-c1ccncc1 C1(C(=O)O)CCN(C(C2CC2C(F)(F)F)=O)CC1C(c1ccccc1)C1CC1 Cc1scc(C(=O)NCC2(C)CC(NC(=O)CC3SC(=N)NC3=O)C2)c1C Cc1nc(C(=O)NCC2CN(C(C34CC5CC3C4C5)=O)CC2O)ccc1Br c1(CC)nc(NC(=O)C(=O)Nc2ccc(OC)nn2)sc1C c1(C(CC(=O)OC)NC(=O)NC(C)CCOC(C)(C)C)ccc(Cl)cc1 C1(NC(C(C)=CC)=O)COC2C(NC(C3(C)CCC34CCC4)=O)COC12 c1(C(C)C(N2CCC(CNC(c3ccc(N)cn3)=O)C2)=O)c[nH]c2ncccc12 N1(C(c2nccc(C)n2)=O)C2CCCC1CC(NC(=O)Cc1cncc(F)c1)C2 C1(CCC)CC(C(=O)N(CC(=O)NCCC2CC2CCF)CC)C1 C=CC(C)(CCOC)C(=O)NC1CC1CNC(=O)Cn1nc(C)cc1C CC(C)C(C)N(C)C(C1(N(C(=O)C=CCN2CCC2)C)CC1)=O C(=O)(CCCC(C)(C)C)NCCC(CCNC(CC1ON=C(CC)C1)=O)C C(C1=CCN(C(=O)CC2(CO)CCC2)CC1)NC(C1CC(C)OC1)=O N1(S(CCOC)(=O)=O)C(C(=O)Nc2cnc(Br)nc2)CC2CCCCC12 C1(COC)CN(C(=O)CC#N)CCN1C(c1cnn(CCC(F)(F)F)c1)=O c12ccc(cc1)S(=O)(=O)NC2=O.c1(CN(C)C(=O)C2CC2)nc(O)n[nH]1 C1(OC(c2ccccc2)C)CCN(S(=O)(=O)NCC2CCCC3CCCCC23)C1 CCC(C)C(CC(=O)NCC1(CC2CC2)CC1)NC(=O)CCC(C)N(C)C N1(C(CC(CCC)O)=O)CC2CC1CCN2C(=O)CNc1ccc(C(N)=O)cc1 N1(C(c2c(CC)nco2)=O)C(C(=O)N(C)Cc2cn(C)nc2C)CC2CCCC12 N1(C(c2ccc(CC)c(N)c2)=O)CC(C)N(C(=O)C(=O)N(C)C)CC1C C(=O)(CCC(=O)OC(C)(C)C)NCCN(C(=O)Cc1ccsc1Br)C(C)C C=C(CNCCC(C)(C)C(=O)OC)c1cccc(F)c1 c1(C(C(=O)NCCC(=C)CNC(C2CCN2CC)=O)N(C)C)ccc(F)cc1 C1(N(C(c2c(C)cc[nH]2)=O)C)CCC2CN(C(=O)Cn3ncnn3)CC12 c1(C(=O)NCC2N(C(C=C(COC)C)=O)CCCC2C)[nH]nc2c1CCC2(C)C C(=O)(C(=O)CC(C)C)N1C(C(CNC(CCNS(CC)(=O)=O)=O)(C)C)CCC1 CC1=CCSC1C(=O)NCC(c1ccccc1)CNC(=O)CCOC1COC1 CC1=C(C(=O)NC2(C(=O)NCc3nc(N(C)C)no3)CC2(C)C)COCC1 C1(NC(C2C(=C)C2)=O)CCCN(C(=O)C(C(C)CC)NS(C)(=O)=O)C1C C1(CNC(C(C)C2CC2)=O)CC2CCC(C1)N2C(c1ncccc1C1CC1)=O C(=O)(C#CC1CCOC1)N(C(C)CNC(c1sccc1Cl)=O)C C1(C(=O)NC2C(C)OCCC2)CCN(C(C2CS(=O)C2)=O)C1(C)C C1(C(N(CCCNC(C2CCCO2)=O)C)=O)CCS1(=O)=O c1(C(=O)NC(C)CNC(C2CC3(CCCO3)C2)=O)cc2ccc(Cl)cc2c(=O)o1 N1(C(C2CCN(C(c3c(CC)cno3)=O)C2C(C)C)=O)CCC12CCOCC2 c1(N2CCN(C(C)=O)C(C)C2)ccncc1S(=O)(=O)NC(c1nc(C)oc1C)C CN1C(=O)N(C)C2(CCN(C(C3CCCN3C(c3cccs3)=O)=O)C2)C1=O c1(CC(=O)NC2CC2CNC(C2CCC(=O)NC2)=O)c[nH]c2cc(F)ccc12 N(C1c2ccccc2CC1NC(C1CCC1C)=O)C(c1cc(C)c(O)c(N)c1)=O c1(C(C(=O)NCC(F)F)N(C(C)C2CC2)CC)cc2cc(Cl)ccc2s1 C(=O)(C1CCCc2cccnc21)N1CCC(O)(CNC(CCCCC)=O)C1 N1(CC)CCN(C(c2ncc(C)s2)C(=O)NC(C)C(=O)OC)CC1C CC1CN(CCC(=O)Nc2cccc(F)c2)CCC1NC(c1cc(CF)no1)=O CC1(C)CC(C(N2CCSC(C)(C)C2)=O)CN(C(=O)COCCCF)C1 C1(C(=O)NC(CC)CN(C(=O)C=CCOC)C)CN2CCCN1CC2 N1(C(c2cnn(CCC)c2C)=O)CCN(C(c2ccoc2CC(N)=O)=O)C2CC12 c1(C(N2CC(CCNC(C(CCC)O)=O)C(C)C2)=O)cc(C)c(C)nn1 N1(C(C(C)NC(C)(C)C)=O)CC2CCN(C(=O)CNS(=O)(=O)N(C)C)C2C1 c1(C(=O)NC23CC(C(=O)NC4CC(C(=O)O)C4)(C2)C3)ccc2ccccc2n1 CC(CCNC(=O)CC1CCOC1)N(C(=O)CCc1cn[nH]c1)C Cn1ncc(C(=O)NCC2C=CCN2C(c2cnc(=N)[nH]c2)=O)cc1=O c1(C(c2nnnn2CC)NCCC(C=C)C)c(C)nc2sc(C)nn12 CC(C)(C(=O)NCC1CC1NC(=O)CCCOc1cccnc1)c1ccccn1 c1(OC)c(Cl)cc(C(=O)NCC2CCC(CO)CC2)c2ncccc12 c1(C(=O)OC)cnccc1N1CC(O)(CCNC(c2cnoc2C2CC2)=O)C1 c1(C(N(CCC(C)NC(=O)CCCCC2CC2)C)=O)c(Cl)ccc2c[nH]nc12 c1(CC(=O)NCC2CC(NC(C(C=C)O)=O)C2)cccnc1Br C1(NC(C2CN(C)C2)=O)CCOC12CCN(C(=O)C1CNc3ccccc31)CC2 c1(CC)cn2c(n1)CC(C(N1CCCC(F)(CNC(=O)CCCC#N)C1)=O)CC2 C1(CNC(COCC(=O)NC)=O)COCCN1C(=O)C(CCSC)NC(N)=O c1(CC(=O)NCC(C)CNC(=O)CC2CCCCCC2)ccc([N+](=O)[O-])c(N)c1 c1(N2CC3C(COC)(C3)C2)nc(C)nc2c1CCC2 C(CN=C(NCC1(OC(C)C)CCOC1)N1CCCC2(CC1)CC2(F)F)OCC CCCCC(CN(C(=O)C(CC(F)F)NC(=O)CN(C)C(C)=O)C)CCC Cn1cnc2ccc(C(N3CCC(C(F)CNC(C4CCCO4)=O)CC3)=O)cc12 Cc1cccc(C(=O)NCCC(C(C)C)NC(=O)CCC2CCCC(=O)N2)c1C Cc1c(C(=O)NCCC2=CCN(C(=O)CCOC3CC3)CC2)[nH]c2c1CCCC2 N1(C(CC(=C)C)=O)CCC(NC(=O)C(C)(C)C2CC2)CC1C Cc1c(C(=O)NC(C(N)=O)C(C)(C)C)[nH]c2ccccc12 c1(OC)ccncc1C(=O)NCCCN(C(=O)CCc1nc(C)cs1)C c1(C(N(C(CCNC(C(C=CCCC)O)=O)C)C)=O)ccn2ccccc12 C(=O)(C#CC1CCCC1)NC1CC(OC)CN(C(=O)C=Cc2nc(C)co2)C1 Cc1cc(C(=O)NC2(CNC(=O)COc3cnn(C)c3)CCC2)c2nccn2c1 C1(NC(c2c(CC)onc2)=O)CCCC12CCN(c1ncn(C)c(=O)c1Br)CC2 CCC(C)(CCC(C)C)C(=O)NC(c1ccc(-c2ccc(O)c(F)c2)cc1)C N1(C(C(C(=O)OCC)C2CC2)=O)CC2CCC(C1)N2C(=O)CS(=O)CC c1(C(=O)NCC(=C2CN(C(CSSC)=O)C2)F)ccc(=O)n(O)c1 CS(=O)CCC(=O)NCC1(O)CC(CNC(C2CC(F)(CO)C2)=O)C1 N1(CC)CCC(c2nnnn2CC(F)F)(NCCCc2ccccc2F)C(C)C1 C1(NC(c2cncc(OC(C)C)c2)c2nnnn2C2(C)CC2)CCCCC1(C)C C12CC(C1(C)C)OC(=O)C(=O)C2.c1(C(C)=O)cc(OC(C)(C)C)cs1.NCS C(N=c1[nH]n(CCOC)cc1[N+](=O)[O-])C1CCC(NC(CCC=C)=O)C1 Cc1nnc(O)c2c(NC(=O)Nc3ccc(SC(F)(F)F)cc3)cccc12 C1(CNC(CC2(OC)CC2)=O)CCC(C)(C)CN1c1ncncc1I C1(C)(CCNC(C2C(CCOC)C2)=O)CCN(C(c2ccsc2NC(C)=O)=O)C1 C(C(C(C)C(C)C)NC(c1coc(CCC)n1)=O)NC(CC(=C)Br)=O c1(CNC(C(N2CC(C#N)CC(C)C2)=O)=O)cc(O)c2ccccc2c1 C(=O)(C1CCCc2ccccc21)N1C(CNC(CSCC)=O)CC(OC)C1 c1(C(=O)NC2C(C)N(C(=O)CCC3CC(C)(C)CO3)CC2)ccc2c(c1)CC2 N1(C(c2ccc(COC)o2)=O)CCOC(C(=O)NCC#CC2CC2)C1 S(=O)(=O)(c1cnn2ccc(N(C)CCOC)nc12)NCC1CC(=C)C1 C1(OC)CN(C(C2(SC)CC2)=O)CC1NC(C1(C(C)C)CNC(=O)C1)=O C(=O)(C(C)CC(=O)c1cccc(F)c1)NCC1(CNC(C(CC)CO)=O)CC1 c1(C(=O)NC2CN(C(C3(CC)CC3(F)F)=O)CC2F)c(F)cc(F)cc1F c1(NCCC2N(C(C3C(C)=C3)=O)CCCC2)cncc(C#N)n1 C1(CC(=O)NC(c2ncc[nH]2)C)CCCC(NC(c2ccncn2)=O)C1 CC(C)C(F)(F)CC(=O)N(C(c1ccccc1)CNC(C1CC(CCO)C1)=O)C C(CS(=O)(=O)CC(=O)NCC(C)CN(C(=O)C(=O)N=S(C)(C)=O)C)OC Cc1cc(C(N2CCCN(C(C3OC4CCC3C4)=O)CC2)=O)ccc1Br Cn1cc([N+](=O)[O-])cc1C(N1CCC(NC(=O)NCCc2ccccc2)CC1)=O C(=O)(CCCC(=O)c1ccc(Br)cc1)N(C)Cc1cn(CCC=C=C)nn1 C(=O)(C1=CCN(C(C2CCSC(C)C2)=O)CC1)N(C)Cc1cc(C)n(C)n1 C1(O)(CNC(c2cc(C(N)=O)ncc2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC1 c1(C(C)=O)cc(C)nc(N2CC3CN(Cc4ccc(N5CCCCC5)s4)CC23)n1 N1(C(CCCCC#C)=O)CC(CO)C2(C1)CN(C(=O)C(CCC)N(C)C)C2 C1(C(=O)NCc2occ(C)c2)CCC(C(C)C)N1C(C1CC1C(F)F)=O N1(C(C2(NC(C)=O)CC2(C)C)=O)CCCC(CC(=O)NCC(=O)NC(C)C)C1 CC1(F)CN(C(c2cc3ccncc3s2)=O)CCN(C(C2CC23CCCC3)=O)C1 c1(C(=O)NCCC2(C)CN(Cc3ccc(Cl)cc3)C2)cnc2c(F)cccc2c1 c1(OC)cc2ccc(NC(=O)C(C)C3CCC3)cc2cc1OC C(=O)(C(C(C)(C)C)C1CCC1)NC1CC(NC(c2ccc(CSCC)cc2)=O)C1 C1(NC(Cc2c(C#C)cccc2)=O)CC2(CCN(C(=O)CO)CC2)C1 N1(C(C)C(=O)N2CCC2)CCC(N(C)N2CCN3C(=O)NCC3C2)CC1 C1(C(=O)OC)CCN(C(=O)CC2CC2CNC(C23C=CC(CC2)C3)=O)O1 c1(C(=O)NC2C(NC(C3CCC(=O)C3)=O)CCCC2)cc(F)cc(F)c1 c1(N2CC(OC)C(O)C2)ccc(Cl)cc1[N+](=O)[O-].c12ccc(cc1)C(=O)NC2 CCCCC(=O)C(=O)N1CC(CC(=O)NC2CCCCC2(C)C)(OCC)C1 Cc1sc(C(=O)NC2CC2CNC(C2CCN(C)C2=O)=O)cc1[N+](=O)[O-] C1(N(C(c2c(OC)csc2)=O)C)CC2CC1N(C(c1occc1C)=O)C2 N1(C(c2c(CCC)[nH]cc2)=O)CC(C)(C)CC1C(=O)N(C)CC1(C)CCC1 c1(SC(C)C(=O)NC2COCC2NC(=O)C(C)(C)n2ccnn2)nncn1C Cc1nc2ccnn2cc1C(N1CCC1CNC(c1sc(F)cc1C)=O)=O c1(C(=O)NCC(CCNC(CSCCN(C)C)=O)O)ccnc(F)c1 c1(C(=O)NCC(CN(C(C(C)NC(CC)=O)=O)C)O)ncc([N+](=O)[O-])cc1C Cc1cc(C(=O)NCCOCCNC(=O)C(C2CCC(=O)N2)C)nc(O)n1 N1(C(CC2(CC)CCCC2)=O)CCCC(O)(CNC(C2CCC2C)=O)C1 N1(C(C(C)OCCC(C)C)=O)CCOC(C(=O)NC2CCOCC2F)C1 c1(C(=O)OC)ncc(NC(=O)C=Cc2ccc(C(F)F)o2)cc1F Cc1oc(-c2ccccc2)cc1C(=O)NC(C1CCCN1C(=O)C=C(Cl)Cl)C c1(CC(=O)NC(C)CC2CCN(C(c3cn(C)cn3)=O)CC2)c(Cl)cccc1Cl N1(C(C(C)OC)=O)CCC(NC(c2c(C)nc(Cl)nc2Cl)=O)C(C)(C)C1 C1(NC(c2cncc(C)c2)c2n(CCCC)nnn2)CC2(C1)CC2(F)F c1(C(=O)Nc2cccc(NC(C(CC#C)(C)C)=O)c2)[nH]nc2cnccc12 c1(CCC)n[nH]c(=NC2CCN(C(c3cc(C)cnc3F)=O)C2)s1 C1CC(O)C(=O)N1SC.c1(C(N2CCC(C)C2)=O)ccnc(OC2CCCC2)c1 Cc1[nH]c2ccccc2c1CC(=O)NC1CC1NC(=O)Cc1cncnc1O C(CS(=O)(=O)CC(=O)N(C1CCC(=O)NC1)C)OC N1(C(C(C)(CC2CCC2)OC)=O)CC2(CC(NC(=O)Cc3conc3C)CO2)C1 CC1C(NC(=O)CN2CCC(NCC(C)(C)C)C2)CCN1C(=O)C=CCF Cc1c(N(C(=O)CCc2cc(Br)c(Br)s2)C)cccc1F N1(C(C(C(C)C)OC)=O)CCOC2(CCN(C(C3CC(=O)NC3(C)C)=O)C2)C1 N1(C(CC(C)O)=O)CCCC(F)(C(=O)NCC2CC3CCC2CC3)C1 C1(C(C(C)C)NC(C2(NC(C)=O)CC2)=O)CCN(C(=O)Cc2ncoc2C)CC1 N1(C(C(CCNC(=O)CC2(O)CCC2)OC)=O)CCC2(CCOC2=O)C1 C(CC(=O)Nc1ccccc1OCF)(C(F)F)NC(c1cnn(C(C)C)n1)=O C1(C(=O)OCCCC)CC(NC(=O)CNC(=O)CCCN(C)C(C)=O)CCO1 N1(C(c2cc(OC)c(OCC(F)(F)F)cc2)=O)CCC2(CCC2(C)C)C1 C1(C(=O)NCC2C(C)CCN2C(C2CCCSC2)=O)CCCCN(C)C1=O CC(CCCNC(c1ccccc1)(CCC1N(CC)CC1)CC)NC(=O)C(=O)N(C)C Nc1c(C(N2CCCCC(CNC(=O)CC3=NNC(=O)C3)C2)=O)cc(Cl)cc1F C(=O)(C1=C(C)CCCC1)NCC(C)N(C(c1nc(COC)[nH]n1)=O)C c1(OCC)cc(CO)ccc1C(N1C2CC1CN(c1cc(NC)ncn1)C2)=O S(=O)(=O)(c1nc(N2CC3COCC3C2)ccc1Br)N1CCCS(=O)(=O)CC1 c1(C(C)=O)ccc(F)c(C(=O)NC(C)(C)C(C)NC(=O)C2=C(Cl)CC2)c1 C1(C)(NC(CNC(=O)OCC)=O)CCN(C(c2sc(Cl)cc2Cl)=O)C1 c1(-n2cc(CC(C(=O)O)NC(c3cn(CC)nn3)=O)nn2)ccc(Cl)cc1 c1(CC)nc(C)c(C(=O)NCC2(C)CCCN2C(=O)C(O)C(F)F)o1 c1(N2CCC(S(C)(=O)=O)CC2)nc2c(c(=NCc3csc(Cl)n3)[nH]1)CCCCC2 N1(C(c2c(C(C)NC(=O)CN3CCCNC3=O)cco2)=O)CCCN(C)C(=O)C1 N(C(=NCCCCl)N1CCC(c2ccccc2)C1)CC1(CC)COC1 c1(NC(C(C)N(C(c2c(COC)cc[nH]2)=O)C)=O)cc(C)c(F)cc1O c1(NC(C2CCCN(C(CC(CC)OC)=O)C2CC)=O)cnc2c(c1)CCC2 CC(CCO)C(=O)N1CCCCC1C1CCCN(C(c2cccc(CO)c2)=O)C1 c1(C(=O)OCC)cc(CC(=O)N(C2CCOC2)C2CC2)c2cccnn12 C(=O)(CCCCC(N)=O)N1CC(CNC(=O)CCCN2CCCC2)CC(C)C1 c1(CNS(C)(=O)=O)cn(C2CCC(NCc3csc(CC4CCC4)n3)C2)nn1 c1(C(N2CC3(CN(C(C4N(C)C(=O)CC4)=O)C3)C2)=O)ccc2c(=N)[nH]cnc2c1 C(=O)(C(C)(C)C(C)(F)F)N1CCC(N(C(CC2CN(C)C2)=O)C)C1 c1(COC)c(C(N2CC(NC(=O)CC(C)(C)C)C3CC3C2)=O)sc2ccccc12 C12(NC(C(=O)NCC)=O)CCC(CN(C(=O)CC(O)C(Cl)(Cl)Cl)C1)C2 c1(CC(=O)NC(CNC(CC2(C)CCOC2)=O)(C)CO)cnn2ccccc12 N1(C(c2cccc(C)c2)=O)CCN(C(c2nc(C)ccc2Br)=O)C2CC12 C(CC(C)C)(C(=O)O)N(C=O)Cc1c(C)oc(-c2ccc(F)cc2)n1 N1(C(C2N(C(Cc3nc(C)[nH]n3)=O)CC(F)C2)=O)CC(C(N)=O)CC(C)C1 c1(C(N(C2CCCCN(C(C(C)OC)=O)C2)C)=O)oc2ccccc2c1C N1(C(CC(C)F)=O)CCC(C)(C)CC1C(=O)N1CC(O)C(O)CO1 C(=O)(CCCCC1CCN1C1CC1)OC(C)C(=O)NC1CCCCCC1 Cc1nn(C)cc1CC(N1CCCCC1CN(C)C(C1CCC(F)(F)C1)=O)=O N1(C(C(CC#C)(C)NC(=O)CCCCC)=O)CC2CC(CO)C(C2)C1 CC1CN2CCN1C(C(N1CC(NC(=O)C(C)c3cc[nH]n3)C(C)(C)C1)=O)C2 Cn1cc(Br)cc1CNS(=O)(=O)Cc1cscc1Br N1(C(c2ncc(C)nc2)=O)CCC2(C=C(C(=O)N3CC4CC5CC4C3C5O)C2)C1 N1(C(C(CN(C)C)NC(c2ncc(OC)nc2)=O)=O)CCCC(F)(CO)C1 C1(C)(CNC(C(C)C#N)=O)CCCN(C(c2ccc(Cn3cc(F)cn3)o2)=O)C1 N1(C(C(COC)C)=O)CCCCC1C1(CNC(=O)C(C(C)O)NC(C)=O)CC1 Cc1n[nH]c(C)c1SCC(=O)NC(C)C(C(C)C)NC(=O)CCc1ncco1 c1(C(C)C)ccc(C(=O)NCC2CCC2NC(C2COC(=O)N2)=O)s1 N1(C(c2cc(C)n(C)c2)=O)CCCC2(NC(=O)CC(O)CC(C)(C)C)CCCC12 C1(C(N)=O)CCC2(CC1)CN(S(=O)(=O)Cc1ccc(Br)cc1)C2 c1(OC)c(F)cc(CCNC(=O)N(C2CC2)CC2CCCOC2)cc1F c1(C(=O)NCC(CC)NC(c2cccc(F)c2NC)=O)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)OC)cc(Br)c(NC(N2CCC(O)CC23CC3)=O)nc1C C(=O)(C1CCCc2ncccc21)NC1CCC(NC(C2C(C(C)O)C2)=O)CC1 C(C(COC)CC(=O)NC1CN(C(c2ccon2)=O)CC1OC)OC c1(OC)ccnc(NCC(N2CCC(NC(=O)C(F)(F)c3cccnc3)C2)=O)n1 c1(C(C(=O)NC(C)CCNC(c2cccc(=O)o2)=O)O)ccc(O)c([N+](=O)[O-])c1 C12CCCCN1C(=O)c1cnn(c1)C2.O=C1CCCN1CCC1CCN(CCl)C1 Cc1[nH]nc2cc(COc3ccccc3C(=O)NC(c3cscn3)C)ccc12 c1(C(=O)Nc2ccc(OC)c(Cl)c2)csc2cnccc12 c1(N2CCC(C(C)NC(C(CC(C)C)C)=O)CC2)cc(C#N)c(F)cc1[N+](=O)[O-] CCCC(CCC)C(=O)N1CCC(C(=O)N(CC(N)=O)CC(C)C)CC1 C(=O)(C(C)(C)CC(F)(F)F)NC1C(CNC(c2cc(C)nc(O)n2)=O)CCC1 N1(C(C2C(CC)CN(C(C3C4COCC34)=O)C2)=O)CCCC12CCOCC2 N1(C(c2cc(C)c(Cl)cc2)=O)CCC(C2CCCN(C(=O)C(C)NC=O)C2)C1 C(=O)(C(C)CC(C)(C)C)N1CCC(CC=C)(NC(=O)CCC2CCCO2)C1 N1(C(CNC(C2CCN(CC)C2)=O)C)CCN(C(C2CCCS2(=O)=O)=O)CC1 C1(CNC(CCOCC)=O)(NC(=O)CCC=Cc2ccccc2)CCCCC1C C(=O)(C1=COCC1)NC(C)CNC(=O)C(C)CNC(=O)CSCc1ccccc1 c1(C(=O)NCC(CN(C(C2C(C=C)C2)=O)C)C)nccc2ncccc12 C(CN=c1nc(C(F)F)nc[nH]1)C1(O)CCN(C(=O)C=Cc2ccncc2)CC1 C1(NC(CN2CCC(C)(O)C2)=O)(CO)CCCN(C(c2cc(C(F)F)[nH]n2)=O)C1 N1(C(CN(C)C(N)=O)=O)CCCC(CNC(=O)C(=Cc2c[nH]cn2)F)CC1 C12(C(=O)NCC3C(C(=O)NC(c4ccncc4)CO)C3)CCN(CC1)CC2 C(CC(C)(C)N(C(=O)CSCC(C)C)C)NC(CNC(=O)OCC=C)=O C1(NC(=O)CCN2CCOC2=O)CN(C(C2CCCCO2)=O)C2(CCCCC2)C1 c1(C(N(CC(C)O)CCNC(C2CCCO2)=O)=O)cc(Br)cc(F)c1F C(=O)(C1=COCCC1)NC1(C)CC(NC(C2C3CNC(=O)C23)=O)C1 c1(NCC2C(NC(c3ccc(C(=O)OC)o3)=O)C2)cc(OC(F)(F)F)cc(Br)c1 N1(C(=O)CSCc2ncc[nH]2)CCCC(CO)(NC(C2CCCOC2)=O)C1 CC(C)CC(C(=O)NC1C2CCC1N(C(=O)CCOCCN(C)C)C2)C(C)C c1(CC)ccccc1C(=O)N(CCCNC(C1(C(F)F)CC(F)(F)C1)=O)C1CC1 c1(C2C(OCC)C2)nc(-c2cccc(Br)n2)nn1CC(F)F c1(C2(C(=O)NCCOC(C3(C(N)=O)CCC3)=O)CC2)ccc(Cl)c(Cl)c1 CC1CCC(Cl)=C(C(=O)NCC2(O)CCCN(C(c3cc(Cl)cn3C)=O)C2)C1 c1(C(C)C)c(C(N2CC(F)(CNC(=O)C=C3CCN(C)C3)C2)=O)cnn1C N1(C(CCCC=C)=O)C(CNC(c2n[nH]cc2C2CCC2)=O)CC2CCCCC12 c1(C(N2CCC3(NC(c4cnc(O)o4)=O)C(C2)C3)=O)cc(F)c(F)c(F)c1F c1(C(=O)NCC(C)(Cn2cccn2)NC(=O)C2CC2)cc2ccncc2[nH]1 C1(NC(CCc2ncc(C)[nH]2)=O)C2CCC1N(C(=O)C=Cc1cnc[nH]1)C2 Cc1oc(CNC(C2CCCC(C)C2)=O)nc1C(=O)NC1CSCC1C C1(CC)CN(C(=O)CC2CN(C(C)=O)C2)CCC1NC(c1cnc(S)n1C)=O C(=O)(C1CCCc2sc(C)nc21)Nc1c(C(=O)OCC)c(C)nn1C c1c(COCCOCC2CCCO2)nn2c1CNCC2 Cc1cccc(C(N2CC=C(CNC(=O)C(F)C3CCOC3)CC2)=O)c1C C1(N(C)C(c2cccc(N(C)C)n2)=O)CS(=O)(=O)CC1O C1(C(NOCCC(=C)C)=O)(CC(=O)OC)CN(C(=O)Cc2ccnn2C)C1 N1(C(c2cccc(CC=C)c2)=O)CCC(C)C(NC(C2(C(C)(F)F)CC2)=O)C1 CCC(C)CC(=O)NC1CC1CNC(=O)COc1cccc(OC)c1 C(=O)(C1CCCc2cncn21)N1CC2CC(NC(c3nc(OCC)oc3)=O)C2C1 C1(COC)(NC(c2nc(O)sc2C)=O)CCN(C(=O)Cc2c(F)cccc2Cl)CC1 N1(C(C(CCC)CC)=O)CC2(CC(C(N3CC(C(C)(C)O)C3)=O)CO2)C1 c1(OC)cccc(NC(C2CCC2C(=O)O)=O)c1Br C(CCCSC)(C(=O)NC1CC(F)(F)C1)N(C1CCOC(C)C1)CC(=O)OCC c1(C(=O)NCC2CCN(C(CCCC(CC)C)=O)CC2)cc2cccn2c(O)n1 CC1CCC=C1C(=O)N1CCN(C)CC1CNC(c1ccn(C)c1)=O C=CC(C)(CCOC)C(=O)NCC1COCC1NC(=O)CCc1cc(C)no1 c1(N2CCC(NC(CN3CC(=O)NCC3)=O)C(F)C2)ccnc2ncnn12 CC1(C)OCCOC1CS(N1CC2(CC(c3ccccc3)C2)C1)(=O)=O Cc1c(NC(=O)CC(C)(C)CNC(c2c[nH]cc2C(C)C)=O)cccc1Cl CC(C)CCC(=O)NCC1CCCCC1NC(C1CCC(C)(C)O1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C1(O)CN(C(C2(C)CCC2)=O)C1)C C(CCCCC(=O)N1CCC(C(=O)N(C(COC)CC)C)(OC)C1)=CC N1(C(C(CC)NC(N)=O)=O)CCC(F)(F)C(CNC(c2ccc(C)nn2)=O)C1 CC1(C(=O)NCC2(C(C)(C)C)CCN(C(=O)CC3C=CCC3)C2)CCNC(=O)C1 C1(NC(C2C(=C)C2)=O)CC12CCN(C(=O)CC1C=CCCC1)C2 Cc1ccc(F)c(N)c1C(N1CC(NC(=O)COCCCF)CC(F)C1)=O C1(C(=O)NC2CN(C(COCC#C)=O)C(CC)(CC)C2)CCS(=O)(=O)C12CCC2 c1(C(=O)NC2CN(C(CC(C)(C)O)=O)CC2C(F)F)cnc(O)c2c1NCCC2 CCC(F)(F)CC(=O)NCC1CCCCC1NC(c1nc(C)ccc1F)=O C12(O)CCN(C1)C2.c1(CC(=O)Sc2ccccc2)ccnc(C(F)(F)F)c1 N1(C(CC(C)F)=O)CCCC2CN(C(=O)C(=Cc3ccccc3)C#N)CCC12 N1(C(CCC(=C)Cl)=O)CCC2CCN(C(=O)CC(C(F)F)C(C)(C)C)CC2C1 N1(CC(=O)N(CCN(C(c2c(CC)cco2)=O)CC)C2CC2)CCC(C)(O)C1 C1(CNC(C=CCCC)=O)CCN(C(c2ccc(Cl)c(C(F)F)c2)=O)C12CCC2 C(=O)(C(C)S(N)(=O)=O)NC1C2CN(C(C(C3CCC(=O)N3)C)=O)C1C2 C(c1ccccc1F)=CCC(=O)NC(CNC(c1[nH]cc2c1CCC2)=O)C1CC1 C(C)(CNC(C12CC(C)(C1)C2)=O)(CC(C)C)NC(C(CC)SC)=O c1(C(N2CC(NC(=O)C(F)F)C3C(C2)C3)=O)cnc2cccnc2c1 c1(C(=O)NC2C(C(=O)NC(C#C)C3CCC3)CCCCC2)cc(C)cc(C#N)c1 Cc1cc2c(cc1C(=O)NC(C)CNC(c1cc(CC(C)C)nn1C)=O)OCO2 N1(C(C(C(CNC(C2(C=C)CCCC2)=O)C)F)=O)CCCOC(C)(C)C1 CC12CC1CCN2C(=O)CC1C=CC(NC(C2CCCC2)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CC)(NC(=O)Cc2ccoc2)CC1 C1(NC(C=CC(C)(C)SC)=O)CC2CC1N(C(=O)Cn1ccc(C)cc1=O)C2 N1(C(c2c(C)cc(C3CC3)cn2)=O)CC2(CCCCN2C(=O)C2=CC(C)(C)C2)C1 N1(C(C(C2CCC2)OC)=O)CCN(C(=O)C(c2ccn(C)n2)C)CC1CCO CN1CCOC(C(N2CC3CC2C3C(=O)NCC2COC(C)(C)C2)=O)C1 c1(NC(CNC(CNC(C2CCC(OC)C2)=O)=O)=O)cc(CO)cc(F)c1 CC1(C)CCCN(C(=O)CCC=CBr)C1CNC(c1cncc(N)n1)=O CC(C)CCC(F)C(=O)NC(CCC1CCC1)C(N1CCC(F)(F)C(O)C1)=O C=CC1(CC(=O)NC2CCCC(NC(C3CCC=CCCC3)=O)C2)CCCCC1 N1(C(C2(CCNC(=O)C(F)CC3CCOC3)CC2)=O)CCCC(F)C1 c1(C(=O)NC2CCCC(N(C(CNS(CC)(=O)=O)=O)C)C2)c(C)cc(=O)oc1C C1(C(=O)N(C2CCOC(C)C2)C)(COC)CCN(C(c2c[nH][nH]c2=N)=O)C1 CCCCC(C(=O)N1CCC(OCC(=O)NC2CCCC(N(C)C)C2)C1)C(C)C N1(C(c2nccc(C(C)(C)C)c2)=O)CCC2(CC1)CC2NC(=O)CCC(N)=O c1(C(N2CC(O)(CNC(C(C)OCCC=C)=O)C2)=O)cnn2c(C)cc(C)nc12 N1(C(C(C)OCC)=O)CCC(NC(c2cccn(C)c2=O)=O)C(OC)C1 C1(NC(C(C)C)=O)CN(C(C2CCc3cncn3C2)=O)C2CCCCC12 C1(Nc2nc(C)nc(N3CC4CCC4C3)c2)CCOC2(CCSC2)C1 Cc1cccn2nc(C(N3CCCCC3CNC(C3CCS(=O)CC3)=O)=O)cc12 C(N=c1[nH]c(Cl)nc2c1SCC2)C1(CNC(C2=CC(C)(CC)C2)=O)CCC1 c1(SCC=C)ccccc1C(N1CC2C(CNC(=O)CC3OCCCO3)C2C1)=O C(=O)(C1=CS(=O)CCC1)NCC1CCC(NC(c2cnc(OC)c(Cl)c2)=O)CC1 c1(C(N(C2CC(NC(C3(F)CC3C)=O)C2)C)=O)cccc(C(F)(F)F)c1 N1(C(Cc2nc(COC)sc2)=O)CCN(C(c2c[nH]c(C#N)c2)=O)CC(C)C1 c1(C(N(CC(CNC(C=C(C)Cl)=O)O)C)=O)nc(C)n(C)n1 C1(OC)COCCC1CC(=O)NC1C2CN(Cc3nccs3)CC12 C1(NC(CC(C)n2ccnc2)=O)CC(O)CN(C(=O)COC2CCOCC2)C1 Cc1nc(CC(=O)N(CCC(C)NC(c2ccn(CC(C)C)n2)=O)C)c(C)s1 CC(C)(C#N)CCCC(=O)NCC1CC(F)(F)CN1C(=O)CCS(C)(=O)=O C1(CNC(C2C(C)CC=CC2)=O)CN(C(=O)CCSC(F)(F)F)CC2(CCC2)O1 C1(NC(c2ccc(Cl)[nH]2)=O)CC(c2ccccc2)(NC(c2ccncn2)=O)C1 c1(C(=O)NC(CCNC(C(CCCC)CC)=O)C)n[nH]c2c1CC(C)(C)CC2 CC1C(CC(N2CC(C(C)(C)O)C2)=O)CCN1C(=O)C=Cc1cccnc1 c1(C(C)(C)C)nnc(C(=O)NCCC2(CNC(C3SCCS3)=O)CC2)s1 C1(N(c2nccn2CCl)C(C2CN(C(=O)OC)C2)C)CCNCCC1C CC1(C)COC(CC(=O)NC(CC2CC2)C(=O)NCC2(C)CCC(=O)N2)C1 N1(c2c(C)ccc(S(=O)(=O)N3CCCC3)c2)CCN(S(=O)(=O)N(C)C)CC1 C(c1cnn(C)c1C)=CC(N1CC(O)(C(CNC(COCC#C)=O)(C)C)C1)=O CCCC(C(=O)NCc1cn(C(C)CNC(=O)CC(Cl)Cl)nn1)OC CCCCCC(F)C(=O)N(CCCNC(=O)CCC=Cc1ccccc1)CCC CCC(O)C(=O)NC1CC(F)(CNC(=O)CCN2CCOCC2)C1 c1(SC)nccc(=NCC2CC(C)(C)CCC2NC(=O)C(c2cccnc2)O)[nH]1 C(=O)(C1=CCCN(C(=O)C(O)C(C)(C)C)C1)N(C)CCC1CCCO1 C1(C(=O)NC2(C(=O)NCC(CC)N(C)C)CC2)CC(F)(F)C1 C1(C(=O)NCc2cn(CCC)nn2)CN(C)CCN1C(=O)CCc1nncn1C C1(NC(C(CC#C)NC(c2cccc(C)c2O)=O)=O)CCc2nn[nH]c2C1 c1(C(=O)NC2CN(C(=O)Cn3cnnc3)CCC2O)cnc2ccccc2n1 N1(S(C2C(C)OCC2)(=O)=O)CCC(N)c2cc(Cl)ccc21 C1(CCCCCOC)CN(C(=O)C(C2CC2)SC)CC(C)O1.C1C(=O)N1 Cc1ccc2[nH]c(C(=O)N(CCN(C(=O)C(F)C(F)(F)F)C)C(C)C)cc2c1 N1(C(CCN(C(C)=O)C)=O)CCN(C(=O)C(C)(C)CO)CC1CCO C1(CC(=O)NCC(C)CN(C(=O)C(F)(F)c2ccnn2C)C)CCCS1(=O)=O N1(C(Cc2ccc(OC)c(O)c2)=O)CCC2(C1)CN(C(C1(O)CCOCC1)=O)C2 C1(C(=O)NCCOCCOCCNC(CC(C)C)=O)CN(C)CC1C(F)(F)F CC(C)C(O)C(F)(F)C(=O)NC(C)CC(C)NC(c1csc(Cl)c1Cl)=O n1(CC)nc(C(=O)NC2(CO)CN(C(C3(OC)CCC3)=O)C2)cc1C1CC1 C1(C(=O)OC)C=CCN(C(C)=O)C1.C(c1cccs1)=CC(=O)N.C1CC(=O)N1 N1(C(C2CN(C)C2)=O)CCN(CC2CN(C(=O)C(C)(C)c3csc(Cl)c3)C2)CC1 C12(c3cn(Cc4c(C)c[nH]n4)nn3)COC(CN1C(=O)Cc1cnn(C)c1)C2 c1(NC)ncccc1C(=O)NCCN(Cc1cncc(SC)c1)CC1CC1 N1(C(C=C=C(C)C)=O)C2CC1CN(C(c1coc(C(N)=O)c1)=O)C2 N1(C(C=COCC)=O)CCC2CCN(C(c3c(O)ccc(Cl)c3F)=O)CC12 N1(CC(=O)NC2C3CN(C(CC(CC)O)=O)CC32)C(=O)N(C)C2(CCCCC2)C1=O c1(OC)cccc(C(C)C(N2CCN(CC(=O)NC(c3nccs3)C)CC2)=O)c1 CCC(C)(C)CCCC(=O)N1CC(C(=O)NCC(C)C2CCC2)OC(C)C1 c1(C(=O)NC2CN(C(c3c(O)ccc(C)c3)=O)CC2F)c(C)[nH]c2ccccc12 C(N=c1[nH]c(=NC(C)c2ccc(C#N)cc2F)[nH]c2cc[nH]c12)C1(CCC)CC1 C12(CNC(C(C)(C)NC)=O)CC(C)(CCO1)C2 C1(COC)(NC(C2CCSC2)=O)CCN(C(=O)C(C)Sc2ccccc2)CC1 C(C)(CCC#N)(c1n(CCCC)nnn1)NC(c1ccc(F)cc1)C(N)=O C(=O)(C(C)(CF)c1ccccc1)N1CC(N(C(=O)Cn2ccc(C3CC3)n2)C)C1 C12(CNC(CN(C)Cc3cccc(Cl)c3)=O)CC1CN(C(=O)CC1CC=CC1)C2 C1(CN(C(=O)CC2CCCOCC2)C)COCCN1C(=O)CCc1cn(C)cn1 C12(NC(C3CCC(C)C3)=O)CC(C1)N(C(c1ccn(C)n1)=O)C2 c1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CCN(C)C2)ccc(P(C)(C)=O)cc1 CC(C(=O)N1CCC(O)C1C(=O)N(C(CCO)C(F)F)C)C(F)F C(=O)(C1=CC2CCCC12)NCc1ccc(CN(C(C(CSC)(C)C)=O)C)cc1 c1(C(=O)O)nccc(N(CCc2nn[nH]n2)C2CC2)n1.CCSCC1CC1 N1(C(CCN(CC)CC)=O)CCC(F)(CNC(=O)CC(C)SC)CC1 C1(CNC(c2cc(C3CC3)ccn2)=O)CN(C(=O)CCCn2ccnc2)C2CC12 c1(C(C(=O)NC(c2ccccc2Br)(C)C)N)ccccc1F N1(C(C2C(CC)CCCC2)=O)CCC2(C1)CN(C(c1c(OC)cccc1C)=O)C2 N1(C(=O)COc2csc(Cl)c2)CCOC2(CCN(C(C3(CO)CCCC3)=O)C2)C1 c1(CNC(C2(CSC)CCC2)=O)csc(C(=O)N(CC(F)(F)CO)C)c1 CC1CCCCC1(CNC(=O)CCNS(C)(=O)=O)NC(C1(C#N)CC1)=O C1(NC(CC(C)(C)OC)=O)CCCCN(C(=O)C(C)(C)F)C1 c1(CCNC(=O)NCC(n2ccnn2)C)nn(C)cc1C(F)(F)F CC#CCN=c1nc(N(CC2OCc3cc(Cl)ccc32)C)c2c(ncn2CC)[nH]1 c1(C(=O)NC(C2CN(C(c3cc4c(ncn4C)[nH]3)=O)C2)C)ccnc2c1CCC2 CCCCS(=O)(=O)CC(=O)Nc1cccc(CNC(=O)C(C)(CC)OC)c1 CC(O)C(C(=O)N1CC(NC(=O)C2=COCC2)C1)C.C(C)(C)(C)OC(=O)NC(C)C N1(C(C(C)(C)C2CC2)=O)CCC2(COC(CNC(c3cccc(=S)n3O)=O)C2)C1 CC(C)C(C)(CNC(=O)C(=C1CCCCC1)F)NC(C1CCC(=O)NC1)=O C#Cc1ccc(Cl)c(C(=O)NCC2(CN(C)C(C3CC3(C)C(F)(F)F)=O)CC2)c1 C1(OCCCNC(C(C)=O)=O)CCN(C(=O)CC2OCCC2C)CC1 C1(C(N2CC3(CCCC3)C2)=O)CN(C(=O)C2=NOCC2)C2(CCC2)C1 NC(=O)CCCCC(=O)NC1CCCCN(C(c2cc(Cl)n[nH]2)=O)C1 c1(C(N2CCC(NC(c3c(C)cco3)=O)CC2C)=O)cnc(C)c(C#N)c1 CC(O)C(C(=O)NCC(N1C(CNc2cccnn2)CC(C(F)(F)F)C1)=O)N(C)C C=CC(C)C(C)C(=O)N1CCC(N(C(=O)CCC(C)(C)OC)CC)CC1 C(C1=CCCCCC1)NC(C(=O)OCCC(C(=C)C)OC)C C1(C(C)C(=O)NCCOC(F)F)CN(C)CCN1C(c1cnn(CCO)c1)=O CC(C)CCCC(=O)NCC1(C)CCN(C(c2ccccc2F)=O)C1 C1(NC(C2CCC23CCC3)=O)CCCN(C(c2ccc(SCCO)cc2)=O)CC1 Cc1ccc(C)c(C(=O)NCCN(C(=O)CO)CCN(C)C)n1.C1C(=O)N1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NC1CCN(C(CCCOCCC)=O)C1 CC1(C)OCc2c1n[nH]c2C(=O)NC1CCC(NC(C2CCOC2(C)C)=O)CC1 c1(C(N)=O)ccccc1CNC(C1CCCN(C(=O)CSC2CCCO2)C1)=O N1(C(C2(COC)CC(=O)C2)=O)C(C(=O)NCC(C)(C)CO)C2CC(O)C1C2 C1(C(=O)NCCSCCC=C)COC2(C1)CN(C(C1(C)CCC3CC3C1)=O)C2 O=C(CCCCN1CCCCC1)NCCC1CCCN1C(c1cccs1)=O C1(NC(CC=CC=C)=O)CC2CC(NC(c3cc[n+]([O-])cc3)=O)C2C1 N1(CC)CC(C(=O)NCC2CC3(C2)CN(C(=O)C=C(C)Cl)C3)CCC1=O C1(NC(COc2cc(C)on2)=O)C2CCC(C2)C1C(=O)NCCC(O)C(F)(F)F N1(C(CCNC)=O)CC(C)CCC1CNC(=O)CCCNC(=O)OC CCC(F)(F)C(=O)NCC(=O)NCC1(CC)CC(C)(C)C1 C(C1CCCN1C(=O)Cn1ccccc1=O)=CC(=O)NC(CC=C)C1CC1 CCC(C)C(C(=O)OCC1CC1)Nc1nnccc1C(F)(F)F C(=O)(CCC(C(=O)NCCNC(c1cc(OC)cc(Br)c1)=O)N(C)C)OC c1(C(=O)NC2CC(CCNC(CSCCCC)=O)C2)ccnc(F)c1O c1(NC(C2C(OC)(OC)CC2)=O)ccc(CNC(C2CC2C(F)(F)F)=O)cc1C Cc1ccc2cc(C(=O)NCC3CCN(C(=O)CC(C)CF)C(C)C3)[nH]c2c1 N1(C(CN(CC)CC)=O)C2CCC1CC(O)(CNC(c1csnn1)=O)C2 N(C(=NCCC1(O)CCCOC1)NCC1CCCCO1)CC1CCN(C(C)C)C1 N1(C(C(C)OCCN(C)C)=O)CC(NC(=O)C2=CCCOCC2)OC2(CCC2)C1 N1(C(c2c(C)c(Cl)ccc2)=O)CCC2(CC1)CC2NC(=O)C=Cc1ccnn1C C(=O)(C1CCc2nccn21)N1CCC(CCCNC(=O)CC2CCC(=O)N2)CC1 C(=O)(C1CCOc2ccccc21)N1CCC(NC(Cc2c(C)nc[nH]2)=O)C(F)C1 CC(CC(=O)N1CCN(Cc2c[nH]c3cccnc23)C2CC12)CC(C)(C)C c1(CC)ocnc1C(=O)N(C1CCCC1)CCNC(C1CCOC1C(F)(F)F)=O C(=O)(C1CCCc2cncn21)N1CCC(NC(Cc2c(C)noc2C)=O)C1 C=CCC(C)(C)C(=O)NCC1CN(C)CCN1C(C1CCC2CC2C1)=O C(=O)(C1=NOC2(CCOC2)C1)N1C(C(C)(C)CNC(=O)C(C)(C)CO)CCCC1 CON(CCCO)C(=O)C1(C=C)CCN(C(=O)CC2CC=CCN2C)C1 c1(C(=O)NC(CNC(c2c(CCC)nns2)=O)(C)CC)ccc(N)c([N+](=O)[O-])c1 C1(C(C)NC(=O)Cc2nnc(O)s2)CN(C(c2ccc(Cl)o2)=O)CCO1 CCCCCCC(C)(CC)C(=O)N(C)CCNC(=O)CC(c1ccc(F)cc1)C N1(C(C(C)CCO)=O)CCCC(C2CCN(C(=O)CCn3cccn3)C2)C1 Cc1nc(N2CCCC2C2CCN(C(c3cnc[nH]3)=O)C2)c(C)c(Cl)n1 N(C(=NCCC1(O)CCOC1)N1CCc2nnc(O)cc2C1)C1CCS(=O)(=O)C1 C(=O)(CC(C)CC(C)(C)C)N1CCOCC(CNC(Cc2scc(C)c2)=O)C1 N1(C(C2C(CC(C)(C)C)C2)=O)CCC2C(C1)CN2C(C1CNC(=O)C1)=O C(=O)(C1CCc2ccccc21)N1C2CC(NC(c3cccs3)=O)C(C2)C1 c1(OC)ccccc1CC(N1CCC(C2(NC(=O)C(=O)NC)CC2)C1)=O C1(CNC(C2COCCO2)=O)CN(C(c2cn3ccsc3n2)=O)C2CCN1C2 C(=O)(CCC(CF)CF)NCC1(C)CCCN1C(C1CN(C2CCC2)C1)=O Cc1nn(C)c(C(=O)NCCC2CCCN(C(C3CC3CF)=O)CC2)c1Cl Cc1cncc(C(N2CC(CNC(c3cc(CCO)on3)=O)CC(C)C2)=O)c1C c1(OC)ccc(C)c(CNC2CC3CCC23)c1Br N1(C(C(CC)ONC(=O)C2CC(O)C2)=O)CC(C(C2CCCC2)=O)CC(F)C1.NC CCC1=NOC(C(=O)NCC(C(=O)N(c2cscc2C)CC)OC)C1 C(=O)(C1=CCN(C(=O)C(C)n2ccnc2)CC1)NCCN(C)CC Cc1cc(C(=O)NC2(C3CN(C(=O)C=C4CCC(C)CC4)C3)CC2)ncc1C#N C(C1C(C(=O)NC2(CCCNC(=O)C=C(C)c3cccs3)CC2)C1(C)C)=C(C)C C1(NC(C2=CC(C)(CC)C2)=O)CC2CCC1CN(C(=O)C(C)COC)C2 c1(CC(=O)NCC(CNC(c2ccc(C#N)cc2)=O)O)cccc2cnccc12 c1(C(=O)NC2CC(CNC(=O)C=C3CCCCC3)C2)cc(F)cc(F)c1 N1(C(CCCSC)=O)CCOC2(CCN(C(=O)Cn3nccc3C)C2)C1 CC(C)CC(C(=O)NCCCCN(C(=O)Cc1csc(=N)[nH]1)C)C(C)C c1(CNC(c2cc(OC)ncc2)(C)C)ccc(Br)cc1F c1(C(=O)NCC(C)NC(c2cc(OC)no2)=O)cc(C)cc(F)c1N C1(NC(CCCNC(=O)OC)=O)CCN(C(=O)C(C)(C)CS(C)(=O)=O)CC1(C)C Cc1cnccc1CCNC(=O)CC(O)CNC(=O)CC1OCCCO1 c1(C(=O)NC(CC(=O)NC(CC=C)C2CC2)C2CC2)cnn2c1OCC2 c1(CN(CC(=O)NC2(C)CC(C(=O)O)C2)C(C2C(C)C2)=O)ccccc1Cl C1(C(F)(F)C(=O)NCC2CCC2NC(c2cc[nH]c2)=O)(OC)CCOCC1 CCN=c1[nH]cc(C(=O)NCC2(CNC(C3CCCN3C)=O)CCC2)s1 C1(C(=O)NC2C(NC(c3c(COC(C)(C)C)ccs3)=O)CC2)CCCNC1=O N1(C(CC2(OC)CCCC2)=O)CC2CCC1CN2C(c1csc(C(C)OC)n1)=O N1(C(Cn2nnc(=N)[nH]2)=O)CC(NC(=O)C=CC2CCC2)CC2(CC2)C1 c1(C(=O)NCCC2N(C(CC(C)(C)F)=O)CCCC2)cc(C(F)(F)F)cnc1O C1(NC(c2ccc(C(C)C)o2)=O)CC(NC(c2cnns2)=O)C12CCC2 N1(C(C2(C)CC(OC)(OC)C2)=O)CCN(C(c2cn(C)cn2)=O)C(CC(F)F)C1 CC1c2ccccc2OC1CC(N1CCC(NC(=O)C(C)(C)CO)C1)=O C1(c2cc(OC)c(F)c(F)c2)CCCN(N2CCCC(O)(C(C)(C)C)CC2)C1 N1(C(C(CC=C)NC(C2CC(=O)C23CCC3)=O)=O)CCSCCC1C CC(C)CCCCCNC(=O)CC1CN(C(C2(C(=O)OC)CC2)=O)CCC1C C1(COC)CN(C(=O)Cc2ccco2)CCN1C(=O)CC1CCCC(C)(C)O1 c1(C(c2nnnn2CC2CC2)NCC2C(C)(C)C2)ccoc1C(F)(F)F C1(C(N(CCNC(c2nc(C)nn2C)=O)CC)=O)CC(=O)NC1(C)C N1(CC(CC(C)C)C)CCCOC(CNC(c2c(Cl)cncc2Cl)=O)C1 C1(NC(COC(C)(C)C(F)(F)F)=O)CCCCCC1NC(C1(C)CC1(F)F)=O C1(CNC(c2c[nH]cc2Br)=O)CN(C(=O)C=CC(=O)N(C)C)CC1O CC1CC(NC(=O)CC2CSC2)CCN1C(C1(C)CCN(C)C1=O)=O N1(C(C(c2ccccc2)OCC)=O)CC2C(NC(=O)C(CC)n3cncn3)C2C1 c1(C(=O)NC2CCCN(C(C(C3CCC3)OC)=O)C2)ccc2nc(O)oc2c1 c1(NC(C23C(CN(C(c4ccc(C)cc4F)=O)C2)C3)=O)cc(Cl)c(Cl)cc1C#N N1(C(COC)=O)CC2(NCCOCCNC)CCC2(CCC(=O)COCC)C1 c1(C(N2CCC(C(C(=O)N(CC(CC)CC)CCC)F)C2)=O)cnccc1C C1(C(N2CC(c3onc(C)n3)C2)=O)CCOCC1NC(=O)COCC1CCOC1 C1(NC(CN2C(C)CCC2)=O)CC2CC(NC(=O)Cn3cnnc3)C1C2 C1(CCC)(CNC(c2cc(OC)cs2)=O)CCN(C(=O)C(O)CCSC)C1 Cc1[nH]c(C#N)cc1C(=O)NC1CC(NC(=O)CC2CC(C(F)F)C2)C1 c1(C(N2CCCCC(N(C(CC)=O)C)C2)=O)nn2c(c1C)CCCC2 C(C)(C)(CCC(=O)N1CCCC1CC(N1CCC(CCO)C1)=O)OC N1(C(c2c(C)nco2)=O)CCC(C)C1C(=O)NCCN1CCCOCC1 N1(C(CC=CC)=O)CC2CCCN(C(=O)CC3CCCC3O)C2C1 Cc1cc(F)ncc1C(=O)NCC1CCCN1C(=O)CN(c1ccccc1)C c1(CC)cc(C(=O)NC(C)CCN(C)C(c2ccc(C3CC3)s2)=O)ccc1Cl c1(CCC(=O)NC(CNC(C(CC=C)C)=O)(C)CO)ccc(S(N)(=O)=O)cc1 C1(NC(C2C(=C)CC2)=O)CC2(CCN(C(c3nc(C)n(C)n3)=O)C2)C1 c1(C(C(=O)NCCCSCC)N(CCC(C)C)C)ccc(OC(F)F)cc1OC CC1(C)CC(NC(=O)CC2(O)CCOCC2)CN(C(=O)CC2(CO)CCC2)C1 C(=O)(CC(O)CNC(C1CCCOCC1)=O)NC(C(=O)N(CC)CC)C C12(CNC(CN3CC(CC)C3)=O)CCCC1CCN2C(=O)CC1CCOCC1 C1(C(=O)NCC(C)N(C(c2nc(Cl)sc2C)=O)CC)CCN(C)S1(=O)=O c1(C(N(C2CCN(C(C3CC3CCC)=O)CC2)CC#C)=O)cccc(F)c1CC C12(C(N3C(CC#C)CCCC3)=O)CC(CO)(CN1C(=O)COc1cccnc1)C2 N1(C(COCC(=C)C)=O)CCC(C2CC2)C1CNC(=O)C=CCN(C)CC C1(C(N2CC(NC(C=Cc3nc(C)sc3)=O)C(C)C2)=O)CCc2nn[nH]c2C1 N1(C(C(CCC)OC)=O)CC(NC(c2ncc(Cl)s2)=O)C2CCCCC12 Cc1cc(C(N2CCOC(CCCNC(C34CC(C3)C(C)O4)=O)C2)=O)nc(O)n1 CC(CC1CCC1)C(=O)NC1(C(=O)N(C2CCC2)C2CC2)CCCC1 N1(C(CCNC(CC(C)C)=O)=O)CCC(NC(c2ccc[n+]([O-])c2)=O)CC1C C#CC1(C(=O)NCCN2CCCC(C)C2)CCN(C(c2ccc(C)n2C)=O)C1 C(=O)(CCC(C)CN(C)C)N1CC(CC=C)(NC(=O)C(C)CC2CC2)C1 CCC(CC)(CCNC(c1nnn(C)c1C)=O)NC(=O)C=Cc1nccs1 Cc1noc2nc(C(=O)NC34CC(C3)N(C(C3(C(=O)NC5CC5)CC3)=O)C4)ccc12 N1(C(C(n2cnc(C#N)n2)CC)=O)CCCC(CNC(=O)CC2CSC2)CC1 N1(C(C2(OC)CCC2)=O)CCC(NC(=O)C=Cc2cncc(C)c2)C2(CCC2)C1 c1(C(N2CCC(N(C)C(C34CCC3CC4)=O)C2)=O)cnc2ccoc2c1 N1(C(C=CCCC)=O)CC(CCNC(c2ccc(C(N)=O)nc2)=O)OC(C)C1 C(=O)(C(CNC(c1cccc(F)c1F)=O)CC(C)C)NCc1ccc(C)c(F)c1 Cc1oc(C)c(C(=O)NCC(CC(C)C)NC(=O)C(F)C(F)(F)F)c1Br N1(c2nnc(Cc3c(OC)cccc3OC)n2C2CC2)CCC(S(N)(=O)=O)C1 CC1OC2(C)CC1(C(N1CC(F)(CNC(c3ccc(-c4ccco4)s3)=O)C1)=O)C2 C1(CC(=O)NC(C(=O)N(CC)CC(C)(C)CC)C)CC(F)(F)C1 C1(C(=O)NCCCOCCNC(Cn2ccc(C)c2)=O)COCC(C)O1 C(=O)(CC1c2ccccc2C(=O)N1C)N(C1CCN(C(=O)CNC=O)C1)CC Cc1cc(OC)c(C(=O)NCCN(CCc2ccccc2)C(C2CC2Cl)=O)s1 C1(C(=O)NCCN(C(c2nnn(C)c2C)=O)CC)CC(c2cccc(F)c2)=NO1 C1(NC(C2C(NC(C(CC)C3CCC(=O)N3)=O)CCO2)=O)CCN(C)CC1C c1(C(=O)NC2(CC(=O)OC)CCC2)ccc(Cl)c(Cl)c1N c1(COCC(=O)NCCN(CCOC)C(C2CC(C)(O)C2)=O)ccnn1C N1(C(c2c(C)cc(CNC(CC(CC)O)=O)o2)=O)CCC2(CCCCO2)C1 CCCCCCCCC(=O)N1Cc2[nH]nc(C(N3CCOC(CC)C3)=O)c2C1 C#Cc1ccc(C(N2CC3CCCCC23)C(=O)NCCC)cn1 C1(NC(CC)=O)CN(C(=O)COc2ccc(OC)cc2)CCC1C(F)(F)F CCCCS(=O)(=O)CC(=O)N1CCC(NC(=O)C(C)CC=CCC)CC(O)C1 c1(C(N2CC(OC)(CNC(=O)Cn3ccsc3=N)C2)=O)cnc(C)[nH]c1=N c1(CC(=O)NCCCCN(C(=O)CCCc2ccncc2)C)ccsc1Cl C1(NC(=NC)NCc2ccc3c(c2)COCC3)CCc2[nH]c(=N)sc2C1 N1(C(c2ncc(C)nc2)=O)CCC(C(=O)NCC2CCC2C)C(C)C1 C(=O)(C(C)(O)C(C)C)NCC(CCNC(CC1(CC)CCC1)=O)(C)C c1(N(C)CC2CCCN2C(c2cc(Cl)nc(Cl)c2)=O)nc(O)c2c[nH]nc2n1 CC1(C#CC(=O)NC(CNC(c2cc(F)c(F)cc2F)=O)C2CCC2)CCCO1 C123COC(C1)(C2)C3.C1(C(=O)NCCCN(C(CC)=O)CCC)C(C)CC1C C=CC1(CC(=O)NC2CN(C(c3cocc3C)=O)C(C)(CC)C2)CCOCC1 CCCC(CC)CC(=O)NC(CCN(C)C(c1ccc(N(C)C)nc1)=O)C(C)C CC1(C)c2ccccc2CN1CCN=c1cc[nH]cc1C(F)(F)F CC(C)S(=O)(=O)CC(=O)NC1(C2CCCN2C(=O)Cc2ccnc(Cl)c2F)CC1 n1(CCCOC)nnnc1C(C)(CCCl)NCCOC(C)C C1(CC)CCN(C(=O)CN2CCCCC2C)C1CNC(c1cocc1C)=O N1(C(C2(C(C)(C)O)CC2)=O)CCC(NC(c2sccc2Cl)=O)C(CO)CC1 C(=O)(C1CCOc2ccccc21)NCCC1N(C(Cc2nnc(C)s2)=O)CCC1 C1(CN(C)C(C2(C)CC=CCO2)=O)CCCCN1C(=O)C1=CCC1 c1(C(=O)NCC2CCCCN2C(=O)CN2CCC2)ncc2ccnc-2[nH]1 CCC(CN(C)C)CC(=O)NC(c1ccccc1)C(C)NC(C12CC(F)(C1)C2)=O c1(-c2n(CCSC)ccn2)cc(-c2ccc(CN(C)C)cc2)ccn1 C1(CC)(NC(c2nocc2Cl)=O)CCCN(C(=O)Cc2ccnc(O)c2)C1 C(=O)(CC(=O)NC1CC(O)C1CC(=O)N1CC(C(F)(F)F)C1)NCC#C c1(C(N2CC(C)(NC(C(c3ccccc3)OC)=O)C2)=O)cnnc(C2CC2)c1 N1(C(C2(C)CC2(Cl)Cl)=O)C2CCC1CN(C(C1C3(CC3)C13CC3)=O)C2 N1(C(c2cccc(C(C)C)n2)=O)CCCCC(C2CN(C(=O)C(C)C(C)O)C2)C1 C1(C(N2CC(CC)C(C(=O)NC(C)C(C)(C)C)C2)=O)CC2(CC2)CN1C N1(C(CCC2OCC(C)(C)C2)=O)CC2(CCC(CNC(=O)CC3(CO)CC3)O2)C1 C1(OC(C2CC2)=O)CCS(=O)(=O)C1.C(C1CCCC1)=C(C(=O)NC(CN(CC)C)C)C C1(N(C(CC2N(C)CCC2)=O)CCc2ccco2)C2CCC1CNC2 C(=O)(C1=CCN(C(=O)COC2(C)CCCC2)CC1)NCC1N(C)C(=O)COC1 C1(NC(C2(C)CCCS2)=O)CCN(C(c2ccsn2)=O)CC1CO C1(C(=O)NCc2c(C)n(C)nn2)CCCCN(C(=O)C(C)S(C)(=O)=O)C1 C12(C(=O)OCC)CCC(NC(C(=O)NCCCC3CCOC3)C(C)C)(CC1)C2 C#CCCCC(=O)NC1CC2(C1)CC2NC(c1c[nH]cc1Br)=O CC1=NOC(=O)CN1C(=O)C(c1ccc(-c2cc(Br)cn2C)nc1)N1CCSCC1 N1(C(C2(NC(C=CCC)=O)CC2C)=O)CCC(CC)CC1 C(CN=c1ncc(O)c[nH]1)C1CCCN(C(C=CCC)=O)C1 C1(CNC(C(C)C=Cc2ccccc2)=O)CC(F)(F)CN1C(=O)Cc1cocn1 O=S(=O)(c1ccc(OC)c(Cl)c1Cl)N(CCCO)Cc1nccs1 C1(NC(C(C)OCC#C)=O)CC12CCN(C(=O)Cc1cccs1)CC2 C1(NC(C=C(CNC(CC=C)=O)C)=O)CCCCC12CC2 C(=O)(C(C)(C)CCN(C)C)NCC1N(C(c2c(C)c(Br)no2)=O)CCC1 C1(NC(CC(CC#C)NC(=O)CC2CC2CC)=O)CN(C)CCN(C)C1 C12(NC(c3ccncc3F)=O)CCC(NC(C3(O)CCSCC3)=O)(CC1)C2 c1(CC(=O)NC2C(NC(c3cccc(C)c3)=O)CC2)c(F)cncc1Cl C1(N(C(C(C)CO)=O)C)CCN(C(=O)CCc2ccccc2)CC1 Cc1sc(O)nc1C(=O)N(CC(C)C(=O)N(C)CCn1ccnc1C)C c1(NC(C)=O)cc(CC(=O)NCC(O)CN(C)C(C2CC2(C)C)=O)ccc1F N1(C(CNC(CC)=O)=O)CC2CN(C(C3CC34CCCCCC4)=O)CC2C1 c1(OCC)cccc(C(=O)NC2CCCC2CNC(c2cnc(C)o2)=O)c1N N1(C(c2ccc(CC)o2)=O)CCN(C)CC1CNC(c1ncsc1C(C)C)=O Cc1c(CN(C2(C(=O)OCC)CCOCC2)C2CC2)cccc1F C(=O)(CCCCCCNC(C12COCC1C2)=O)N(CC(CC)OC)C C1(C2CN(C(c3nnc(O)nc3O)=O)C2)(NC(=O)CN2CCNC2=O)CC1 Cn1cc(C(N)=O)cc1C(=O)NCC1COCC1NC(C1CC1(C)C)=O C1(NC(C(COCC)(C)C)=O)CC2CCC(C1)N2C(C1CC(CC(=O)OC)C1)=O Cc1ccc([N+](=O)[O-])cc1C(N1CCN(C(=O)Cc2conc2C)CC(O)C1)=O c1(C(C)(C)C)nnc(C(N2CCC(Oc3ccccn3)C2)=O)s1 c1(C(=O)NC2(c3cccc(OC(C)C)c3O)CCOCC2)cc(Cl)cc(F)c1F C1(C2CC2)(NC(CS(CC)=O)=O)CCN(C(C2CCCN(C(N)=O)C2)=O)C1 c1(C(N(CCCNC(=O)Cc2ccoc2)C)=O)cccc(N2C(=O)CCC2=O)c1 N1(C(C)=O)CCCC1C(=O)NC1(CC(N2CCC(O)C2)=O)CCC1 C1(OCC)COCCC1CC(=O)N(C)CCNC(=O)C=C1CCCCC1 c1(OC(C)C)ccc2[nH]c(C(=O)NNC(=O)c3cncnc3)cc2c1 N1(C(CC(C)c2ccco2)=O)CCN(C(=O)C2=CCCCC2)CC12CCC2 C1(C(N2C3C(CNC(C(C)C(C)O)=O)C(C3)C2)=O)CCc2n[nH]cc2C1 c1(C(=O)NCCOCCCOCC(=O)NCc2cccs2)cc2ccccc2o1 N1(C(Cc2c(C)nccc2)=O)CCC(C2CC2)C1Cn1cc(CCCCCO)nn1 CC1CC(NC(=O)C(C)(C)c2cnsc2)CCN1C(c1cc(Cl)c(Cl)[nH]1)=O c1(CN=C(NC(COC)C)NCC2(C)CCCS2)cc(OC)cc(OC)c1 C1(C)(OCC)CCN(Cc2nc(CCO)c(C)s2)CC1 Cc1cc(C)c(C)c(C(N2CCN(C(=O)CCCN=[N+]=[N-])CC2)=O)c1C CCC(C)(CCC(C)C)C(=O)NCC1CN(C(=O)CC2CCOCC2)CCCO1 C(=O)(CC(C)C1CC1)OC(=O)CC.C1(=O)CC(c2ccccc2)CCN1CCC c1(C(=O)NC(C2CCCCC2)CC)cc(C)[nH]c1C.c12n[nH]cc1NC2 c1(C(=O)NCC2(NC(=O)CSC(F)(F)F)CCCCC2)cc2cccnc2[nH]1 N1(CC(=O)NCC2CC(F)CN2C(C2CCOC2)=O)CCC(F)CC1 c1(CC(=O)N(C2CCN(C(C3CCC(C)(C)O3)=O)C2)CC)ncn2c1COCC2 Nc1ccnc2c(C(N3CCCC3CNC(c3ccnnc3O)=O)=O)cnn12 C1(C(=O)NC(CNC(CN(C)C(c2ccccc2)=O)=O)(C)C)CCC(N(C)C)C1 c1(C(=O)NCC(CCNC(CC(CN(C)C)O)=O)O)cnc2n1CCS2 CON(CCCO)C(=O)c1cc(CNC(=O)CCOC2CCC2)no1 C1(NC(c2nc(OCC)oc2)=O)CCN(C(c2ccoc2CC)=O)CC1CO C1(CNC(C(C(C)(C)O)F)=O)CC12CCN(C(=O)C=Cc1cnccn1)CC2 N1(C(c2cc(C)nnc2)=O)CC(C)C(C)(CNC(=O)CCn2cnc(=N)[nH]2)C1 c1(C(=O)NC(C(C)NC(Cc2c(C)n(C)nc2)=O)C)cc2ccc(O)cc2[nH]1 c1(CC(N2CCC(Cn3cc(C(C)(C)OC)nn3)C2)=O)csc2ccccc12 C(CC(F)F)(C(=O)N1CC(C)C1(C)C)NC(c1n(CC)ccc1)=O c1(C(N(C2CCC(NC(c3ccncc3O)=O)C2)C)=O)cc(Cl)cnc1O CN1N=C(C(=O)NCC2CCN2C(C2CCC=CO2)=O)CCC1=O c1(C(=O)NCCCOCCNC(C(C)CC2CCC2)=O)cn(C)c(=O)n1C c1(C(N2C(CN(C(C(F)=CCC)=O)C3CC3)CCC2)=O)cc(N)c(Cl)cn1 C1(C2CCCC2)(C(=O)NC(CCNC(CN(CC)CC)=O)C)CCNC1=O Cc1coc(C=CC(=O)NC(C)CCCNC(=O)CCC2CCN(C)CC2)n1 C1(NC(C(CCC)NC(=O)COCCSC)=O)CCC(=O)NC1(C)C c1(CN(C(CC2C(C)C2)=O)C)cccc(CNC(=O)COC2CCOCC2)c1 c1(C(C)(C)C)ncccc1C(=O)NCCC1(NC(C2CC3CCC2O3)=O)CCC1 CCC(C)C(O)C(=O)NC1CCC(NC(c2coc(Cl)n2)=O)CC1 C1(C(=O)NCCC2(OC)CN(C(=O)CN3CC4CC4C3)C2)CCCCN1N=O c1(OCC(=O)N(CC(CC)NC(c2ccc(O)c(F)c2)=O)C)nc(O)nc(O)n1 N1(C(c2cnn(C)c2Cl)=O)CCC(C)(C)C(NC(=O)Cc2ccns2)C1 c1(OCC(=O)NCC(CN(C(c2c(C)cns2)=O)C)C)cc(F)cc(F)c1 c1(CC)c(C(=O)NCC(CCNC(c2ccon2)=O)OC)cccc1C C12(C(=O)NC(CNC(COCCOC)=O)CC)CCCN(CC1)S2(=O)=O C#CC1CC2(CC(C(=O)N(C)CCNC(=O)C(C)CSC)C2)C1 CC1(C(=O)NCC2CCOCC2)CC(O)CN1C(C1C2CCC(F)C12)=O C(c1cccnc1)=CC(=O)NCC1CCC(NC(C2CCC(O)N2)=O)C1 N1(C(=O)OC(CC2N(c3cccc(C(=O)OC)n3)CCC2)=O)CC(C)CC(C)C1 Cc1cccc2c(C(=O)N(C3CCN(C(C4COC4)=O)CC3C)C)csc12 c1(OC)ccnc(OC)c1C(=O)NC1CCCC1NC(=O)CC1CCOC1=O C(=O)(C(CCNC(=O)CCCOC)OC1CCCC1)NCCC(CC)O n1(CC(=O)OC)cnc(C)c1C(=O)NC1COCC1NC(C1CNC(=O)C1)=O CCCCCC(=O)NCC(=O)NC1C=CCN(C(=O)Cc2ccc(C)s2)C1 N1(Cc2ncc(C)nc2)CCC2C(CCCN2C(c2cccn2C(C)C)=O)C1 N1(C(C(CCOCC)NC(c2cnc(C)cn2)=O)=O)CC(=O)NC(C)C1 C1(CNC(CSCC#C)=O)CN(C(=O)CC(c2ccccc2C)C)CCC1C C1(C(N2C(CNC(C34CCC(C(=O)OC)(C3)C4)=O)CCC2)=O)CC12CCOCC2 Cc1ccc(C(N2CCCC2C(C)NC(C2CCC(C)(C)O2)=O)=O)cc1F c1(C(=O)NC(C=C)C2CC2)ccc(C)cc1-n1cc(-c2ccncc2C(=O)O)nn1 CCCC(C(O)C(=O)N1CCC(CC(N)=O)CC1)NC(=O)CC(C)(C)CCC c1(CC)cc(=NCCC(C)NC(c2c[nH]c(Br)c2)=O)[nH]c(CC)n1 C1(C(=O)Nc2c(CC)cc(C)cc2)(CNC(=O)OC(C)(C)C)CCCC(F)(F)C1 n1(CC(=O)N(C)Cc2ccc(Cl)c(Cl)c2)cc(Cl)c2cccnc12 c1(C(=O)NC2(CNC(C(CC#C)C)=O)CC2)ccc2cccnc2c1N N1(C(C(CC)OC)=O)CCC2CCCC(C1)N2C(=O)C(F)(F)CC(C)C C(C(C)(C)CC(=O)NC(C)CNC(=O)C(c1cccc(C)c1)F)OC N1(C(C(CC)n2ccnc2)=O)CCCC(NC(=O)CCC(=O)C2CCCCC2)C1 CCCCCOCC(=O)NC1CC1C(=O)NCCOCC(F)F N1(C(c2scc(OC)c2)=O)CCC=CC1C(=O)NCC(c1ccncc1)C C(=O)(C(O)CCCc1ccccc1)NC1CCN(C(C2CCC(=O)NC2)=O)CC1 c1(C(CNC(=O)C(O)c2cncs2)NC(C(C)=CC2CC2)=O)cc(F)cc(Cl)c1 C1(C)(C(=O)NC2C(CNC(c3c(COC)scc3)=O)C2)CCCNS1(=O)=O C(=O)(C(CC)CC(C)C)N1CC(C)(CNC(CC(C=C)(C)C)=O)OCC1 c1(C(=O)NCC2(CNC(CC3CCC(=O)CC3)=O)CC2(F)F)ncc(F)cc1F C1(CNC(C23CCCCC2OCC3)=O)CC2CCCC2N1C(=O)CCOC1CC1 CC1(C(=O)NCC(C2CCOC2)NC(c2ncsc2Br)=O)CCCC1 c1(C(N2CC(C)CC(NC(C(Br)=C(C)C)=O)C2)=O)c[nH]c2c(F)cccc12 N1(CC)CCCCCC1c1ccc(NCCN(CCOC)C2CC2)o1 N1(C(c2coc(C)n2)C(=O)NC(CC)C)CCOC2(CC1)CCS(=O)(=O)C2 CC1CC=C(C(=O)NC(C(=O)NCc2ccccn2)C2CCCC2)CC1 Cc1nc2n(c1C(=O)NCC1(C)CCOC1C1CC1)CC(C)CC2 n1(CC)ncc(C(N2CC(CNC(=O)CCCC3CCCO3)C2)=O)c1C N1(C(c2cnc(CC)nc2)=O)CCN(C(=O)CNC(C2CCOCC2)=O)C(C)C1 c1(C(N(C2CCC(NC(c3occc3Br)=O)CC2)C)=O)ccc(P(C)(C)=O)cc1 C1(N(C)C(c2cc(Br)ncc2Cl)=O)CCc2ncccc2C1 C1(CC)CN(C(C2CC(=O)N(CC)C2)=O)CCN1C(c1c[nH]nc1F)=O c1(OC)ccc(C(N2CCCCC2CNC(=O)C(C)SC)=O)c(OC)c1 Cc1nsc(Br)c1C(=O)N(CCCCCNC(c1coc(CO)c1)=O)C C1(C(=O)NC(COC)CC(=O)NCC23CCCCC2C3)CC2(CCO1)CC2 Cc1cc(C(=O)O)c(C)cc1-c1ccnn1CCC(C)C C=CCCCCC(=O)NCC1(CNC(C2CC2Cl)=O)CCC1 CC1CC(C(=O)O)N(C(=O)COC2CCCCCC2)CC1C C1(CC(=O)N(C2(CNC(C3CCC(=O)N3C3CC3)=O)CC2)C)CCCOCC1 N1(C(C2(F)CN(C(C3CCC(CCCC)CC3)=O)C2)=O)CCCCC(C)(F)C1 C(=O)(N=S(C)(=O)c1ccc(Br)cn1)c1c(CCC)n(-c2ccc(Cl)cc2)nc1 c1(C(N2CCC(OCC(=O)NC3(CCN(C)C)CC3)C2)=O)cc(COC)no1 C1(C(N2CCC(C)(CNC(=O)C(O)C3CC3)C2)=O)CCCC(F)(F)CC1 N1(C(Cc2c(OC)c(Cl)ccc2)=O)CC2C(NC(=O)CO)CS(=O)(=O)C2C1 N1(C(CC(C(C)C)O)=O)CCC2CCC(C1)N2C(C1C2CCC(C2)C1(C)C)=O C1(n2cnnn2)(C(=O)NC(C)CCNC(=O)CCC2CC2(F)F)CCOCC1 C1(NC(=O)NC(C(C)(C)CO)c2ccco2)COCCC1(F)F N1(C(C(C)C(F)F)=O)CC2CCCC2(NC(=O)Cc2cncnc2)C1 Cc1nsc(C(=O)NCC2CC(O)CN2C(=O)CCNC(N2CCCC2)=O)c1N Cc1cc(=NCC2CC3CC2CN3C(c2cnc(C(C)(C)C)nc2)=O)[nH]cn1 c1(CNC(C(=O)NC(CSCC)CO)=O)ccc(Nn2cc(C)cn2)cc1 C1(NC(N2CCS(=O)CC2c2cccc(F)c2)=O)CC2CC1CC21CC1 C1(C(=O)NCC2(COC)CCN(C(C=CC=CC)=O)C2)CC2CCCC(C1)C2 c1(C(=O)NC(CCN(C(CCOCC#C)=O)C)C)ccc(S(N)(=O)=O)nc1 c1(C(=O)NCC(CNC(c2c(SC)cccn2)=O)O)cccc2ncnc(O)c12 CC1=NC(C(=O)NCC2CCN2CC(=O)NCC(C)(C)C)CS1 C=C(Br)CC(C)(C)C(=O)OCc1cc(Cl)ccc1F c1(C(=O)NC(CC)(CNC(C2(F)CCOC2)=O)CC)c[nH]c2cc(Cl)ccc12 CC(=O)CCCC(C)C(=O)N1CCSCC1C(N1CCC(C)(N(C)C)C1)=O N1(C(c2cc(OC)no2)=O)CC(CNC(=O)COCCF)C2(CC2)C1 C1(C(=O)NC(c2ccccc2)C(=O)OC)CCC(NC(=O)C#CC(=O)O)CC1 CON1CCC(NC(=O)C(C2CC=CCC2)N(CC(=O)OC)C)CC1 C(=O)(C(N)C1(CC)CCC1)NCC=CC=C c1(OC)ccccc1OCC(=O)NCCC1CC(NC(C23COCC2C3)=O)C1 c1(C(N2CC(NC(=O)CNc3cccnc3)CC(C)C2)=O)cccc2[nH]ncc12 N1(C(C2CN(C(C)=O)C2)=O)CC2(CC(C(=O)NCCCN3CCCCC3)CO2)C1 C(=O)(CC(C(C)C)C(C)C)N1CC(SC)C(NC(C2OC3CCC2CC3)=O)C1 c1(C(=O)NC(c2cn(C(C)C(C)O)nn2)CCC)conc1C(F)(F)F C(CN=c1[nH]c2c(c(=NC3CCC(C4CC4)C3)[nH]1)SCC2)(C(C)C)OCC=C C12(CO)CCCN1C2=O.c1(C(=O)NCCN(C)CC)cc[nH]n1 N1(C(C2C3(CC(OCC)C3)C2)=O)CCOC2(CCN(c3ncncc3C)C2)C1 C(CCCCC(=O)N1CCN(C(C2CCC(=O)O2)=O)CC1C1CCCC1)OCC C(=O)(C(C)(C)CC(=O)N(C1CCCC(C)C1)CC1C(NCC(=O)NCC)C1)OC c1(C(C)NC(C23CC(CCC(F)(F)F)(C2)C3)=O)ccnc(Cl)c1F N1(C(C2(c3c(-c4c(OC)nccc4)cccc3)CC2)=O)CC(F)(F)C(F)(F)C1 Cc1nc(C2CCCOC2)sc1C(N1CCC(CSCc2cn(CC)nn2)C1)=O N1(C(C=CC(=O)OC)=O)CCCC1C1CCCCN1C(c1ccc(C)cn1)=O C(=O)(C(O)CCNC(=O)Cn1cc(C)cn1)NCC(C)SC Cn1cnc2sc(C(=O)NCCOCCNC(=O)CC3CCOCC3(C)C)cc12 C(CC(C(=O)NC1CCCCC1OC)NC(c1cc(O)cs1)=O)OCC c1(OC)cc(C(=O)NC2(C(=O)NCC3CC3c3ccoc3)CC(O)C2)on1 C1(C(=O)NCC(C(C)C)C)CCC2(CC2)N1C(C1CC2(CCC2=O)C1)=O C1(C(=O)NCCC2CC(C(=O)NCC(N3CCOCC3)=O)C2)CCCCNC1=O C1(C(=O)NC2CCC(CNC(CC3CC(=O)C3)=O)C2)CC2CCCC(C1)C2 n1(CC)c(C(N2CC(N(C(=O)COCC(C)C)C)C(F)C2)=O)cc2ccccc12 c1(-c2cc(C(=O)NCC3CN(C(C4N=C(C)SC4)=O)C3)on2)cccc(C)c1 C1(C(=O)NCCCCCN(C(=O)CN2CCOCC2)C)CSCCS1 CC(C)CC(F)C(=O)N1CCC(O)(CN(C(=O)CCc2cnn(C)c2)C)C1 C=C(C)CCCC(=O)NCCC(O)C(=O)NCc1nncn1C1CC1 N1(C(CCOCC(C)C)=O)CC2(COC(CNC(=O)C(=O)Nc3ncc[nH]3)C2)C1 C1(C(c2n(C)nnn2)Nc2ccc(-c3nc(C4CC4)no3)nc2)CCOC(C)(C)C1 c1(C(N2C(CNC(=O)Cc3conc3C)CC(OC)C2)=O)ccc(O)c(CO)c1 c1(C(N2C(C(C)NC(c3nc(COC)oc3)=O)CCC2)=O)oc(C(N)=O)cc1C c1(-c2n(C(C3(C)CC3)C)nc(C3CCOC3)n2)csc2cc(C)ccc12 c1(CC)nonc1C(=O)NCCCC(=O)NCC(C1CC1)OC Cc1cn2c(C(=O)NCC3(F)CC(NC(=O)COCC(C)C)C3)c(C)nc2s1 O=C(N=c1cc[nH]cc1-c1nn[nH]n1)C12CCC1CN(C(c1cnnc(Cl)c1)=O)C2 c1(CN(C)C(C2CCCN(c3ncc(I)cn3)C2)=O)ccc(Cl)cc1Cl N1(C(CC=CC=C)=O)CCC(CF)(NC(=O)C2CC2)C1 C(=O)(C1c2c[nH]nc2CN1C(C1CC2(CC2)CN1C)=O)N1CCCC(CC=C)C1 C1(NC(C2CC3(CSC3)C2)=O)CC(=O)N(C2CN(C(C3C4CCC(=O)C34)=O)C2)C1 C1(NC(C(C=C)O)=O)COC2C(NC(c3csc(C(C)OC)n3)=O)COC12 C12(NC(CS(C)(=O)=O)=O)CCC(CC1)N(C(c1csc3ccccc13)=O)C2 CC1(C(=O)NC23CC(F)(C2)C3)CCN(C(=O)CC23CCC(CC2)C3)C1 c1(C(N(CCC(C)NC(C2(C)CCCCO2)=O)C)=O)ccc(N=[N+]=[N-])cc1 C1(CCNC(C2C(C(C)C)CCC2)=O)CCN(C(=O)CCN2CCCC2)CC1 c1(C(=O)NC(C2COC(C)(C)O2)CO)cc2n(c1)CCCC2 c1(C(C(=O)NCCOC)N(C)CC2CC=CC2)cc(OC)c(Br)c(OC)c1 S1(=O)(=O)c2cnc(c(Cl)c2)NCC2C(CC)CCN12.C1(=CCC)CCNC1 C(=O)(CC(COC)NC(c1nnn(C)c1N)=O)NC(c1n(CC)ccn1)C c1(CCC)c(C(=O)Nc2ccc(C3(OC)COC3)cc2)cnn1C1CC1 c1(C(=O)NCC2OCC(CNC(C(=O)N(C)C)=O)C2)ncccc1Br C1(C(c2n(CCOC)nnn2)NCCCCc2nccs2)CCSC1(C)C c1(CCCC)nc(C)c(CC(=O)NC2CN(C(=O)CCC3CCCC(=O)N3)C2)s1 CC(C)(C)CC(=O)N1CC(NC(C2(C(C)(C)C)CCCCC2)=O)C(O)C1 CCCCC(C)CCC(=O)NC1CCCCC1NC(c1ccc(C#N)cc1Cl)=O C(CCC(C)C(=O)N1CCC(CNC(=O)Cc2ccco2)C1)OC N1(CCC(N2CCC(CNC(C3(C=C)CCC3)=O)C2)=O)CCN(CC)CC1 C1(C(=O)NCCC(N2CCCCC2)=O)CC12CCN(C(c1ccoc1)=O)CC2 N(C(=NC1CCS(=O)(=O)C1)NC1CCC1(C)C)Cc1ccc2c(c1)N(C)CC2 c1(C(N2CCC(C3N(C(CCCCSC)=O)CCC3)C2)=O)ccc2c(c1F)CCC2 N1(C(C2(C)CC2(F)F)=O)CCN(S(=O)(=O)c2cn[nH]c2)C2(CC2)C1 C1(CCC)CCCC1C(N1CC(CCCCNC(c2nocc2C)=O)C1)=O Nc1cc(Cl)ccc1C(=O)NCC1(NC(C2CSCCS2)=O)CCCCC1 c1(C(N2CC(O)(CNC(c3c(C)nc(Br)cc3)=O)C2)=O)cccc2c1CCC2 CC(C)C(C(=O)NCC(C(C)(C)C)NC(=O)Cc1ccno1)n1ccnc1 c1(CNC(c2cccc(-c3ccccc3)c2)C)cc(Cl)ncc1Br C(=O)(C(C)(C)CC(C)(C)C)N(C)CC1CCN(C(Cc2c(C)occ2)=O)C1 c1(C(=O)NC(C2CCN(C(CCCSC)=O)C2)(C)C)[nH]c2c(c1C)CCCC2 CC(C)CCC(C(=O)OC(C)(C)C)OC(=O)NCC1CC(C)(C)C(=O)N1 C#CCC(O)C(=O)N1CCC(OCCNC(C2CC(CC)C2)=O)C1 C(C)(C(=O)NC(CO)C(C)NC(=O)CCN1CCCCC1)(C(C)C)NC(C)=O c1(NCc2cn(C(CSC)C(=O)NCC(O)(COC)CO)nn2)cc(=O)cc[nH]1 CC12CCCC1N(C(C1CCCOCC1)=O)CCN(C(C1SCCS1)=O)C2 c1(C(=O)NCCN(CCCCCC)C(=O)C(O)CC2CC2)cc(C(F)F)n(C)n1 C(=O)(CCN1C(=O)COc2ccccc21)N(C(C)CN(C)C(c1cnn[nH]1)=O)C c1(C(=O)NC2(CCNC(=O)CC=C(C)C)CCC2)ccn(COC)n1.C1CC1 c1(NC(N2C(Sc3cccc(C)c3)CCCCC2)=O)cc(Cl)c(Cl)cc1N C1(C(N2CCCC(CCNC(C(C(=O)OC)F)=O)CC2)=O)CN2CCCN1CC2 c1(-n2cc(CNC(CNC(C3C(C)N(C)CC3)=O)=O)nn2)cccc(F)c1F C1(N(C(CCC2(C)CC2)=O)CCCO)CCSC12CN(c1nc3ccccc3s1)C2 C(=O)(C1=CC(O)C(O)C(O)C1)N1CC(C#N)N(C(c2ccc(Cl)c(Br)c2)=O)CC1 c1(C(=O)NCC2CN(C(c3scc(CC)n3)=O)C2)c(C(F)(F)F)ccc(F)c1F C1(NC(c2ccc(C(C)(C)C)s2)=O)CCC(NC(C2(CC(F)F)CC2)=O)CC1 c1(-c2cccc(C(C)C)n2)cc(O)cc2ccccc12 Cc1cnc2cccc(C(=O)NCCN(C(=O)CCC3CC3C)CC(C)O)c2c1 C1(C(N(CC#C)CC=C)=O)CN(C(=O)C(c2ccccc2)F)CC1C n1(CC(=O)N(C2CCN(C(=O)CC(C)F)CC2)CCC)nc(C)c2cccnc12 C(=O)(CC(C)(C)CCC)NC(CC#C)C(=O)OC c1(C(N2CC(CNC(Cc3cn(C)nn3)=O)C3(C2)CC3)=O)cc2ccccc2[nH]1 CN1C(=O)C(NC(c2ccc(Cl)nc2O)=O)c2c(F)cccc21 Cn1cnc(S(N)(=O)=O)c1C(=O)NC1CCN(C(c2cn[nH]c2)=O)C1C1CC1 O=C1CC(COCC(F)(F)F)NC(=O)N1Cc1nc(C2CC2)sc1Br N1(C(Cc2cn(CC)nc2)=O)CCc2c(C(=O)NCCc3ccsc3)n[nH]c2C1 c1(NCC)cccnc1C(N1CCC(NC(c2c(C3CC3)noc2C)=O)C1)=O CCC(CC)C(C)C(=O)NCC(C(=O)NCCC(C)(C)N(C)C)C(C)(C)C N1(C(CSc2ccc(N)c(Cl)c2O)=O)CCC2(CCN(C(C34CC(C3)C4)=O)C2)C1 C(=O)(C(CC(C)C)n1ccnc1)N(C1CCN(C(CCCCOCC)=O)C1)CC C1(CC(=O)NC(C2CCCCC2)C(C)NC(c2csnn2)=O)CC2(CCC2)CO1 Cc1c(CC(N2CC(N)CC2C(=O)NCC(C)C)=O)cccc1[N+](=O)[O-] n1(C(C)C)nccc1CC(=O)NCC(C)NC(c1csc(-c2ccccn2)n1)=O C1(NC(c2c(C)cccc2F)=O)CCN(C(=O)CC2NC(=O)NC2=O)CC1(C)C N1(C(C2N(C)CC(F)C2)=O)CC2=C(C1)CN(C(C1CCNC(=O)C1)=O)C2 Cc1csc(=NCC(=O)N(C(C)CCNC(c2nnn(C)c2C)=O)C)[nH]1 C(C)(CC(C)(C)OC)NC(CCOC)=O.C12CCOC1C(=O)NC2 C1(NC(C(Cc2ccoc2)NC(=O)CCOC2CC2)=O)CCCCCC1F CC(C)C(O)(C(=O)NC(C)CCNC(C1CCOCC1)=O)C(F)(F)F CC(C)C(F)C(=O)NCC1CC(F)CN1C(=O)CNC(=O)CCCc1ccsc1 C1(F)(CNC(C2(C#C)CCC2)=O)CCN(C(C2CC(CC)=NO2)=O)CC1 Cc1cc(C)c(C(=O)NC2COCCN(C(=O)CNC(=O)CC(C)C)C2)c(Cl)n1 c1(OC)cc(C(C)NC(=O)NCCCOc2ccsc2)on1 C#CCCCC(C(=O)Nc1cccc(OC)c1)N(CC=C)Cc1ccccc1Cl C1(C(C)C)CN(C(=O)CCCCCF)CCN1C(c1cccc(C(C)(C)C)c1)=O c1(CNC(N2CCOC(c3nccs3)C2)=O)ccc(CO)cc1 Cc1cccc(C(N2CC(CNC(c3cc(C)c(C)o3)=O)C(O)C2)=O)c1[N+](=O)[O-] C(=O)(CCCCn1ccnn1)NCCN(C(=O)C(C)(CO)OC)CCC N1(C(COCCC)=O)CCCC2(NC(c3cncc4sccc34)=O)CC2C1 CCC(C)C(O)C(=O)NCCOC1(CNC(c2cc(C)no2)=O)CCOCC1 C1(C(=O)NCC2(C#C)CCCC2)C2CCC(C2)C1NC(=O)C(C)N=[N+]=[N-] C(=O)(CC1OCCc2ccsc21)NC1CN(C(C(CC#C)O)=O)CC1C(F)(F)F c1(C(C)C)ccc(C(=O)N(CCCN(C(=O)C(O)CN2CCCC2)C)C)s1 c1(C(=O)NCc2ncc(-c3ccnn3-c3ccccc3)cn2)ncc(Br)cc1O N1(C(=O)Nc2n(C(C)CC3CCCC3)ccn2)CC2COCC2(C(=O)O)C1 Cc1cc(S(=O)(=O)NC(c2cc3ccc(F)cc3s2)=O)c(C)o1 Cc1ccnc(C)c1C(=O)NCC=CCNC(=O)CC1CCC(F)(F)CC1 Cc1ccc(Br)c(C)c1C(=O)NC1CCN(C(C2CCCS2)=O)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CCN(C(c2ncc(N)cc2C)=O)C(C)C1C N1(C(CCN2CCN(CC)CC2)=O)CCCC(NC(C2(N(C)C)CCC2)=O)CC1 c1(C2C(N(C(C3CC4(CC(OC)C4)C3)C(=O)NC)C)C2)ccc(S(C)(=O)=O)cc1 CC1CCC(C)N(C(C2CCCN(C(c3cnn4c3OCC4)=O)CC2)=O)C1 N1(C(C#CC2(C)COC2)=O)CCN(C(C2(CF)CCC2)=O)CC2CCCCC12 Cc1nc2c(C)cc(C(=O)NCC3CCN3C(C3(C)C=CCC3)=O)cn2n1 C1(C(=O)NCc2coc(C3CC3)n2)(CC)CCCN(C(C2CCC3CC2CO3)=O)C1 c1(C(=O)NCCc2cc(O)no2)scc(Br)c1Br C12CCCCC1NC(=O)C2.C1(CNC(COC)=O)CCC1C(=O)OC(C)(C)C C#Cc1cc(F)c(C(N2CC(NC(=O)C(C)(C)c3cscn3)C(O)C2)=O)cc1F C(=O)(C(C)(C)CC(C)C)N1CC(SC)C(NC(=O)Cc2cscn2)C1 c1(CC(=O)N(C2CCN(C(C3OCCO3)=O)C2)CC)ccc(F)cc1C c1(C(N(CC(CC)NC(C2(n3cccn3)CC2)=O)C)=O)nn(C)c(C2CC2)c1C Cc1cccc(Cl)c1OCC(N1CCC(NC(=O)CC2(C)CCC2)C(CO)C1)=O N1(C(CC(CC)OC)=O)CCC(CNC(C2CC(C)(C)C(C)(C)C2)=O)C(F)(F)C1 c1(-c2nc(CC)[nH]n2)ccc(C(=O)N(C)CCNC(C2CC2(C)C)=O)cc1 C(C(C(=O)NCc1cn(C)cn1)NC(=O)CCC=CC(C)C)OC C12(C(=O)NC3C(=O)NCC3)CC(CN1C(c1ocnc1C1CC1)=O)C2 C(=O)(C(F)CCC(C)(C)C)N1CC(CNC(=O)CCC2(C)CC2)CC(C)C1 N1(C(c2c(CC)nn(C)c2)=O)CCC(N=c2nc(C(F)(F)F)[nH]s2)C(C)C1 C(=O)(C1=CCCC1C)N1CCCC(CCNC(CCc2ccc(C)o2)=O)C1 C1(NC(C2(OC)CC2)=O)CCC(C)(C)CC1CNC(=O)Cn1cnc(C(N)=O)n1 N1(C(c2nc(COC)sc2)=O)CC2(C)CN(C(c3cnn(C)c3N)=O)CC2(C)C1 C1(NC(CCC#C)=O)CCCCC12CCN(C(c1cccc3nn[nH]c13)=O)CC2 C(CC(=O)N1CCCCC1C1CC1)(CC(C)C)NC(Cc1cccc(C#C)c1)=O c1(C(=O)NCC=CCNC(c2c(N)nccn2)=O)ncc(C(N)=O)cc1Cl c1(C(N2CC3CCN(C(C(C)OCC=C)=O)C3C2)=O)c(C)nn2c(C)cccc12 C1(CNC(CN(S(CC)(=O)=O)C)=O)CCCCN(C(C2(C)COC2)=O)CC1 C(=O)(C(C)(C)c1cnn(C)c1)N1CC(N(C(C2C(OCC)C2)=O)CC)C1 C(CN=c1ccc2c(I)cccc2[nH]1)N1C(=O)CCNCC1 C(=O)(C1=COCCC1)NC1CC(C)(NC(=O)CN2C(=O)CCCC2=O)C1 CCC(N=c1[nH]c(=NCCCCS(C)=O)[nH]c2ccsc12)c1ncccn1 C(=O)(C(C)C(O)C(C)C)N1CC(OC)C1(C)C.C12CCN(CC1)c1ccc(s1)CO2 C1(NC(C2(F)CN(C(CN(C(C)C)C)=O)C2)=O)CC(C)OC1=O c1(CN(CCC(C(C)C)NC(=O)CSCC(F)(F)F)C)cnn2c1CC(C)CC2 CC1(C(N2CCC(n3ccnn3)C2)=O)CCN(C(=O)Cn2cccnc2=O)C1 c1(CNC(C(C2CN(C(C3(COC(C)C)CC3)=O)C2)O)=O)nccn1C c1(C(=O)NC2C(NC(C3N(CC)CCCC3)=O)C2)ccc2cc(F)c(F)cc2n1 c1(C(=O)NC(C(C(C)C)NC(=O)CCC(C)(C)F)C)nc2cc(O)ccc2[nH]1 CN1CCC2(CCN2C(=O)C(CNC(C2CC(=O)CC(=O)N2)=O)N(C)C)C1 c1(-c2ccc(C)cc2O)cnc2c(C(=O)Nc3nc(Br)cn3C)c[nH]c2c1 c1(CC)ccccc1C(=O)N(C)CCNC(=O)C(c1cnn(C)c1)OC CCC(CC)C(C(=O)N1CCCCC1CNC(c1ccc(Br)o1)=O)OC c1(NC(C(C)NCCc2conc2Br)=O)ccc2c(c1)CCC2 C(C(C)CC(=O)N1CC(C)(C)C1)NC(C(OC)OC)=O c1(OC)ccc(NC(=O)C(C2CCCO2)NC(=O)C(C#N)C(C)C)nc1C Cc1nc(C(N2CC3(C2)CN(C(=O)CC2CC4CCC2C4)C3)=O)cc(O)n1 C1(CC)C(NC(=O)CS(=O)(=O)NC)CCN1C(C1CC(F)C(=O)N1)=O N1(C(C2CN(C(C(CNC(=O)NC)O)=O)C2)=O)CCC(CF)C1 C12(NC(C(C)OCCOC)=O)CC(CNC(c3cc(Cl)c[nH]3)=O)(C1)OC2C Cc1cccn2c(CC(=O)N(C3CCN(C(C4CC4C)=O)CC3)CCC#N)cnc12 n1(CC(=O)NC2CCN(C(CCCC#C)=O)C23CC3)cnc2ccccc12 Cc1cc(NC(C2CCN(C(c3ncc(Cl)cc3Br)=O)C2)=O)ccc1F C(C#Cc1cccnc1)NC(C1(C#C)CCN(C(=O)C(F)CCC)C1)=O c1(C(=O)NCC(C)(C2CC2)NC(C2CC3(CCO3)C2)=O)cc(F)ccc1Cl N1(CC)CCN(CC(=O)NCC2(F)CCN(C(C3CC(C)=NO3)=O)C2)C(=O)C1=O c1(C(C)C)nnc2cc(N(CC(O)CN(C(=O)C(C)C3CCC3)C)C)ncn12 CC1CN(C(C2CCCC23CCCC3)=O)c2ccc(F)cc2O1 Cn1c(=O)oc2ccc(CNC(=O)NCc3noc4c3CC(F)(F)CC4)cc12 C(C(=O)N(CC(C)C(=O)NCc1cncc(OC)n1)C)(C(C)C)SCC Cc1nc(C=CC(=O)NCCNC2CCN(C3CCC(C)CC3O)C2)[nH]c1C C(CCC1CC1)(C(=O)N1CCC2CC12)NC(C=CC=CC)=O C(=O)(CCCC(C)(C)C(=O)N1CCN(C(C2CCN(C)C(=O)O2)=O)CC1)OC c1(N2CCC(N(C)C(C3(Cl)CC3)=O)C2)ccc(C#N)cn1 c1(CCNC(c2ncc(-c3ccccc3)o2)C)cccc(Br)c1 C1(C(=O)NCCC(C)O)OCCC1NC(=O)C(C)C1CCCO1 C1(NC(C2C(OCC)COCC2)=O)CCN(C(C2CCC3(CCC3)O2)=O)CC1O c1(CN(S(=O)(=O)CC)CC)cn(C)nc1C1CCCO1.C12CCN(C1)C2=O CC(C)CCCC(=O)N1CCC(O)C(N(C(=O)CCS(C)=O)C)C1 Cc1cn2ccnc(C(=O)NC3CCCC3NC(c3ccnn3CC#N)=O)c2n1 c1(NCc2ccc(OCC)c(-c3cc(O)ccc3F)c2)cc(Br)ccc1[N+](=O)[O-] CCC(CC(=O)NC1CC=CCC1C(=O)N(c1ccccc1)CC)SC CC1=C(C(=O)N2CC(C)N(C(c3ccncc3Br)=O)CC2C)CCCO1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(C2CC(NC(=O)C(CN(C)C)C(C)C)C2)C1 c1(NC(C(=O)Nc2c(C)n(C(C)C)nc2)=O)ccc(I)c(Cl)c1 Cc1cc([N+](=O)[O-])ncc1C(=O)NC(C)C(C)NC(C1Cc2ccccc2C1)=O CC(CCC(C)(C)C)C(=O)NC1CC1NC(c1ccc(Cl)c([N+](=O)[O-])c1)=O Cc1cccc(C(=O)NCC2(O)CCN(C(C3(O)CC3)=O)C2)c1O C=CC1(C(=O)NC(CC)C(=O)N(C)C)CCN(C(c2coc(CC)n2)=O)C1 C1(C(=O)OC)CNC(=O)CN1C(=O)CCC(C)NC(=O)CNC(=O)C1CC1 CC1(C)CCc2c(C(=O)Nc3ccccc3C(=O)NCC(N)=O)csc2C1 C12(NC(c3ccn(CC)n3)=O)CC1CN(C(=O)CCc1cnc(C3CCC3)o1)C2 N1(C(c2n(C(CC)CC)ncc2)=O)CCCN(C(c2cnn(C)c2OC)=O)CC1 C1(CC(=O)NC(COC(C)C)(C)C)N(C(C2CS(=O)(=O)C2)=O)CCC1(C)C Cc1ccc(Br)c(C(N2CCCCC2C2CCCN(C(=O)CC#N)C2)=O)c1 c1(C(=O)NCC2C(NC(c3cnn(CC)c3Cl)=O)CCCC2)ccnc(O)c1F C1(CC)(CNC(=O)C=CCC(C)(C)NC(C2CC(=O)C2(C)C)=O)CCC(=O)N1 N1(C(CNC(CCOC)=O)=O)CCN(C(c2cccc(-c3nccs3)c2)=O)CC1 c1(CC(=O)NC(CN(C(c2cnoc2C)=O)CC)C)ccc(OC)cn1 c1(C(=O)NC2(c3ccccc3)CC(NC(C(CC)=CC)=O)C2)nnn(C)c1C C(=O)(CCCC#N)N(C1CCCN(C(=O)C(N2CCOCC2)C2CC2)C1)C N1(C(C(CC)=CC)=O)CCC2(CC1)CN(C(C1CCCN(C(=O)OCC)C1)=O)C2 CCCC(C(=O)NC1CC(C(F)C(=O)NCCC2CCC(C)(C)C2)C1)OC Cc1cc(C)c(C(=O)NC2CC(C)N(C(c3ccncc3F)=O)C2)[nH]1 c1(SC)ccccc1OCC(=O)NC1(CCNC(=O)C(C)C2CC2)CCC1 c1(NCC2N(c3ccc(C#N)c(C4CC4)n3)CCC2)ncc2ccc(Br)cc2n1 CCC(CNC(c1cn[nH]c1)=O)(CC)NC(c1cnn(CC(F)(F)F)c1)=O c1(-c2ccn(C)n2)nc(-c2cc(O)ncn2)n(CCOCC2CCCCC2)n1 c1(OC)c(C(=O)NCC2(O)CCN(C(C3CC34CC4(F)F)=O)CC2)c(C)nn1C c1(CC)cc(C(N2CCOCC2CNC(c2cncc(Br)c2)=O)=O)nn1C c1(NCC(CC)CC)ncc(C)cc1S(=O)(=O)N1CCC(P(C)(C)=O)CC1 C1(C(=O)NC(C)C(N2CC(F)(CF)C2)=O)C2CCCCCC12 c1(OC(C)C)ccc(C(=O)NC2(C)CCN(C(C3CN(C)CCO3)=O)C2)cn1 C1(C(N(CCCO)CCC)=O)N(C(c2cc(C)cc(C)c2)=O)CCC1(C)C c1(OC)cncc(C(=O)NCC(C(C)(C)C)NC(=O)C=CCF)c1 C(=O)(C1=NNC(C(F)(F)F)C1)NCCC1(OC)CN(C(CCC(=C)C)=O)C1 CCC(C)CCCCCC(=O)N(CCNC(=O)CC1NC(=O)CNC1=O)CC CC1(C)CCC(NC(=O)CCNC(=O)CCCC2CCCO2)CC1 CCC(CC(C)C)C(=O)NCc1cc(C(N2C(CO)CCC23CCC3)=O)ccn1 c1(CC)cccc(CC)c1C(=O)NC1CCCCC1CNC(c1cnsc1C)=O N1(C(c2c(C)nn(C3CC3)c2)=O)CC2CC1CN2C(=O)CCOCC(C)C(C)C c1(SC)ccc(C(C)NC(=O)Nc2ccc(Cc3ccc(C)nc3)cc2)cc1 C(CC(=O)N1CC2CC(CO)C(C2)C1)(C(F)(F)F)NC(C1C2CCCC12)=O c1(C(=O)NC(C2CCCN2C(=O)C(C#N)=CC2CC2)C)ccc(C(F)F)cc1 c1(C(C)C)ccc(C(=O)NCCC2(O)CCN(C(=O)CC3CCOC3)C2)c(O)n1 C1(C(=O)NCC2CCC(NC(CC(=O)OCC)=O)C2)CC12CCOC2 N1(C(c2c(O)ncc(CC)c2)=O)CCC2(CCCN(c3cc(Cl)c(O)nn3)C2)C1 c1(C(N2CCN(C(C3CCC3)=O)CC(O)C2)=O)c(F)ccc2c1OCC2 c1(C(N2C(CNC(c3n(C)nnc3)=O)CCC2)=O)c(C(F)(F)F)ncn1O C(=O)(C(O)CC(F)(F)F)N1CC(C(C)(C)O)(CNC(C(CO)N(C)C)=O)C1 C1(NC(C=CC)=O)CN(C(c2ccc(-n3cnnn3)cn2)=O)CC1OC Cn1nnc2c1CCC(C(=O)NCCCCNC(=O)Cc1cncnc1)C2 C1(C)(CNCC2OCCN(C(c3c(C)ccnn3)=O)C2)CCCC1(F)F C1(COC(c2n(CCC)nc(C)c2)=O)CCN(C2CCc3c(F)cccc32)CC1 C12(CCNC(CNC(C)=O)=O)CCC(C1)N(C(=O)CCC1CCC(=O)C1)C2 C1(CN(C(=O)CCN2N=N2)C)CCN(C(C2CC2(c2ccccc2)C)=O)C1 N1(C(C(C)=CC2CC2)=O)CCCC1C(C)NC(=O)C=CC1CCC1 N1(C(CCCC#N)=O)CCN(C(=O)Cc2cccs2)CC12CC2 N1(C(C(COC)(F)F)=O)CCC(C)(NC(C23CC(F)(C2)C3)=O)CC1 N1(C(c2cc(C(C)C)no2)=O)CCC2CN(C(=O)CCc3ccc[nH]3)CC12 c1(NC(N(CCC(C)C)C)=O)scc(C(F)(F)F)c1C#N c1(N2CC(C)C(O)C(C)C2)nc(N2CC(Cc3ccoc3)C2)c2c(n1)CCCC2 C(=O)(C(C)(C)C(C)(F)F)N1CC(NC(C(c2cscc2)N(C2COC2)C)=O)C(C)C1 C(=O)(C1=NOC(CNC(=O)Cc2cscn2)C1)NCC(C#C)C(C)C N1(C(COC(CC)CC)=O)CC2CC(C)N(C(c3cnn(C(F)F)c3)=O)C2C1 c1(CC)cc(C(=O)NCC#CCNC(=O)CCc2cncc(C)c2)c(C)nn1 c1(C(=O)OCC)sc(CCC(=O)NC2C=CCN(C(=O)OC(C)(C)C)C2)nc1C N1(C(c2ccc(N(C)C)c(F)c2)=O)CC(NC(c2coc(Cl)c2)=O)CC12CCC2 C1(C(N2CCC(N(C(=O)CCSc3ccccc3Cl)C)C2)=O)CCCCC(=O)N1 C1(C)(CNC(c2c(C)cnnc2O)=O)CN(C(=O)C(C)SC(C)C)C(C)(C)C1 Cc1cc(C(F)(F)F)nc(C(=O)NC2CCCN(C(=O)C(F)(F)CO)C2)n1 N1(C(CN(C(C)=O)C)=O)CC(NC(C2(C#N)CCOC2)=O)CC2(CCC2)C1 c1(C(N(CCNC(c2cccnc2Cl)=O)CC2CC2)=O)ccccc1C1CCC1 n1(CC(CC)NC(=O)NC2(C)CC(=C)C2)ncc2ccccc12 Cc1cc(C(=O)N(C(C)C(=O)NCC2(CO)CCCO2)C2CC2)cnn1 C1(=O)C(CC(C)C)N1.c1(C(C(=O)OCC)N(C(CC)CC)CC)nc(Cl)sc1Cl CC(C)C(C)C(C)CC(=O)NCc1ccc(CN(C(=O)CC=C(Cl)Cl)C)cc1 C(=O)(C(C)CN(C)C(C1CCC(=O)C1)=O)NCC(c1ccncc1)C N1(C(C2=C(C)OCCC2)=O)CCCC(C2CC2NC(=O)COC2CCOC2)C1 C1(NC(c2ccn3cncc3c2)=O)CCN(C(=O)Cc2cc[nH]n2)C12CCCC2 N1(C(C=C(C)c2ccco2)=O)CC2(CCCC2NC(C2CC3CCC2C3)=O)C1 C1(C(=O)NC(C(C)NC(c2ccc(OC)c(O)c2)=O)(C)C)C2CCC3C(C2)CC13 CC1CC1C1CC1NC(=O)CCN(C(=O)COC1CC1)CCO C1(CC2C(NC(C)=O)C2)CCCCN(C(N2CC(C)C2)=O)C1 C(=O)(C(C)(C)CNC(=O)CC(C)CN(C)C)NCc1c(C)n[nH]c1 c1(C(N2C(Cn3cc(CCCSC)nn3)CCC2)=O)cncc(Br)c1C C=CCC(C)(CC)C(=O)NCC1CN(C(=O)C=CC)C(C)(C)C1 c1(CC(N2CC(NC(CCC)=O)C3(C2)CC3)=O)ccc(OC)c(OC)c1Cl C(=O)(CC(F)(F)Cl)NCC(CC=C)NC(c1cccn1C)=O C=CC1CCCCN1C(=O)C(O)CCCNC(=O)C1CC1 c1(OC)cc(C(=O)NC2CCN(C(c3cc(F)n[nH]3)=O)CC2O)nc(C)c1 C1(C(C)O)CCCCN1C(c1cc(CNC(c2ccc(C(F)F)o2)=O)cs1)=O C1(NC(c2cnn(C3CCCC3)c2Cl)=O)CCC2CC1CN2C(=O)CCF Cc1c(C(=O)NC2CC2NC(c2cc(C(F)(F)F)nn2CC)=O)noc1C1CC1 c1(NC2(CNC(c3cccc(CC)n3)=O)CCCC2)cccc(OC)c1[N+](=O)[O-] Cc1cc(C(=O)NCCSc2ccncc2)ccc1[N+](=O)[O-] C#Cc1ccc(C(=O)NC2CC3CC(C2)N(C(C24CC(C)C2C4)=O)C3)c(OC)c1 C1(C(N2CC(CC(C)NC(CN(CCCCCC)C)=O)C2)=O)CCCC(C)(C)O1 C1(C(=O)NC2CCC(OC)C2)CC(N=[N+]=[N-])CN1C(=O)C=CC(=O)N(C)C c1(C(N2CC(CC(=O)OC)C(C)C2)=O)cc2ncc(Br)cc2o1 C1(C(=O)N)CCC2CN(CC3C4CCCC34)CC2CC1.C1(NC=O)CCOCC1 Cc1cc(NC(=O)COC2(C)CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)cc(F)c1 C(C(=O)NCc1occc1C(=O)NCC(C)(C)CC1CC1)(C(C)C)SC C1(NC(C2(O)CCN(C(CSCCC(C)C)=O)C2)=O)CC1C1CCCCC1 CCCCC(CNC(=O)C(F)CC)NC(c1ncccc1C(F)(F)F)=O C(CCCC(=O)NCC1CC1NC(=O)Cc1ccc(C(C)C)cc1)OCCC=C N1(C(CNC(CC)=O)=O)CC2CN(C(=O)CCC(N)=O)CCC2(CO)C1 C1(CNC(CC(C)O)=O)CC2CCC(C1)N2C(c1ccc(F)cc1N)=O CC1CC(CC(=O)NOCC(C)(C)O)CN1C(c1ccncc1N(C)C)=O Cc1cc(NC(C2CCC(NC(=O)C3=NNC(=O)CC3)C2)=O)cc(C)c1Cl Cc1ccc(C=CCC(N2CC(NC(=O)Cc3c[nH]nc3C)CC(F)C2)=O)cc1 C(=O)(C(CCCC(C)C)N1CC2COC(=O)C2C1)NCCOC C12(C(=O)OC)COC(C(=O)NCCCCN(C)C(C3CNC(=O)C3)=O)(C1)C2 C1(NC(=O)CCC(F)F)CCN(C(c2cc(Cl)c(Cl)s2)=O)CC1O N(C1c2ccccc2CC1NC(C1(F)CCS(=O)(=O)C1)=O)C(CCC=C(C)C)=O CCCC(C(=O)NC1C=CCN(C(c2cnn[nH]2)=O)C1)c1ccccc1 N1(C(c2c(CCC)[nH]cc2)=O)CCN(C)C(CNC(c2snnc2C(C)C)=O)C1 C1(C(=O)NCC2(F)CC(NC(C(C)(Cl)Cl)=O)C2)CC(C2CCC2)C1 c1(CNC(=O)CC2COCCN2C(c2cnn(CCO)c2)=O)ccc(F)cc1O C(N=c1[nH]c(N2Cc3cccnc3C2)nc2c1CSC2)C1(C)CCOC1 c1(C(N2C(C)CCN(C(=O)CC3(C)CCOC3)CC2)=O)ccnc2c1nnn2C c1(CC#N)cc(-c2cc(N)ccc2Cl)cc([N+](=O)[O-])c1 C1(CNC(C=CCOC)=O)CCN(C(=O)CCOCC2CCCO2)CC1C C(Cc1cc[nH]n1)(C(=O)N1CCC(F)C1)NC(CCN(C)CCO)=O C1(C(N(C)Cc2c(C)n[nH]c2)=O)CCN(C(C2CC2(C)C)=O)C12CCC2 c1(C(=O)NCCn2c(=O)cc(C)nc2O)cc2c(o1)C(C)(C)CCNC2=O C12(C(=O)NC3CCC(=O)NC3)CC(CO)(CN1C(c1cnn[nH]1)=O)C2 C(C)(C(C(=O)NCCC1CCOCC1)C(C)C)N(C(C(C)N(C(C)=O)C)=O)C CCC(C(=O)N(C)CC1C2CN(C(c3cnns3)=O)CC12)C(C)(F)F CC1C(C=CC(N2CCC2CNC(=O)CC2(N(C)C)CCCC2)=O)C1(Cl)Cl c1(N(CCCOCCNC(=O)CN2CCOCC2)C)ccnc(CC2CC2)n1 C1(NC(=O)OC)CCCN(C(C2(F)CC(NC3CC3)C2)=O)C1 C1(CNC(c2cc(O)nc(Cl)c2)=O)CCCCCN1C(C1CCOCC1)=O c1(CC(N2CC(CNC(C3CC(O)C3)=O)C(O)C2)=O)ccc(Cl)cn1 C(C(C)(C)C(C)(C)O)NC(C1CCN(C(CC2(OCC)CC2)=O)C1C1CC1)=O C1(CNC(=O)C=CC2CCOCC2)CN(C(c2snnc2C2CC2)=O)CC12CC2 N1(C(C(n2cc(CC3CCCCN3)nn2)C)=O)CCC(O)CC2(CCOCC2)C1 c1(CN(C)C(=O)NCc2cnn(CC(F)(F)F)n2)nc2c(s1)CCCC2 CC(C(F)C(=O)N1CCC(=O)N(CC(F)(F)F)C1)C(F)(F)F C(C1CCCn2c(C)cnc21)Nc1nc(C)nc(N2CCC3CC3C2)c1 C(=O)(CC(O)C(C)C)NCCN(C(c1nc(Br)[nH]c1C(F)(F)F)=O)CC C1(NC(c2cn(CCC)nc2)=O)CN(C(C2CCN(C(C)=O)CC2)=O)CC12CC2 c1(CC)ccc(O)c(C(N2CC(CNC(c3nnsc3C)=O)C2)=O)c1 N1(C(c2c(OC)cccc2F)=O)CC(NC(C2CCOC2)=O)CC12CCCC2 C1(NCC(F)=CCC)CCCC12CCCC2 CC(O)C(C)CNC(c1ccoc1CNC(C1CCN1C(C)(C)C)=O)=O C1(CC)CCC(C)CN1C(=O)CC1CC(OC)CN1C(=O)C(C)N1CC(C)C1 N1(C(c2cccc(C(C)(C)C)c2)=O)CC2CCC(C1)N2C(C1(C)CCOC1)=O c1(C(N(CCCNC(c2ccncc2)=O)CC)=O)cnn2c1S(=O)(=O)NCC2 C(N=c1nc(C2CC2)[nH]s1)C1OCC(CNC(c2cc(-c3ccco3)[nH]n2)=O)C1 CCC(C)CC(=O)NC(C)CNC(=O)CCNC(=O)CCC1CCCCCC1 N1(C(CCc2ccc(C)s2)=O)CCC(C)C(NC(=O)CC2CCCNC2=O)C1 C1(C(=O)N(C)CC2(O)CCN(C(c3nnnn3C)=O)C2)(SC)CCC(F)(F)CC1 C(C)(C)(CCCNC(c1ccc(CNC(c2cccnc2)=O)o1)=O)N(C)C N1(c2c(Br)cnc(OC)n2)CCC(C)(C)C(CNC(=O)CSc2nncn2C)C1 C(=O)(C1=COCCO1)NC(CC1CN(C(C2CCCC(C(=O)OCC)C2)=O)C1)C C(=O)(C1CCc2cc(F)ccc21)N1C(C(=O)NCC2CC(C#N)C2)CC(O)C1 CCC1=C(C(=O)NCC2CCCN2C(=O)C(C)OCC2CC2)SCCO1 CCC(C(=O)N(C)C)C(=O)N=c1[nH][nH]cc1-c1ccc(F)c(F)c1 C(C(N=[N+]=[N-])C(=O)NC1CCCCN(C(=O)C(C)CC(N)=O)C1)OCC C1(S(C)(=O)=O)(C(N2CC(NC(c3ccc(CC)nc3C)=O)C(C)C2)=O)CCCC1 C1(=CC(=O)NCC2N(C(C3C(C(=O)OC)C3(F)F)=O)CCC2)CCC(C)CC1 c1(NCc2c(C)nc(CCC)o2)ccc(S(=O)(=O)N2CCC(CC(C)C)C2)cn1 C=C1CC(C(=O)OC)(C(=O)NC2CC2(C)CC(C)C)C1.C12(CC1)C(=O)NC2 CN1C(=O)CSC1=CC(=O)NC(c1ccccc1)CNC(=O)Cc1ccn(C)c1 Cc1ccc(C(N2CC3CC(CNC(=O)C=C4CCSCC4)C3C2)=O)cc1C N1(C(=O)COc2cccnc2Cl)CC2CN(C(C3(CF)CCC3)=O)CC2C1 c1(NC(C2CC(=C)CN2C(c2c(C)cccc2Cl)=O)=O)cnc2ccc(Cl)nn12 C1(NC(c2c(C)onc2Cl)=O)CCN(C(c2cnc(=N)[nH]c2)=O)C(C2CC2)C1 N1(C(c2ccncc2)=O)CCC(C2CCCN(C(C3CC3F)=O)C2)C1 C1(C(=O)NCCCOCCNC(CC2(C)CC(F)(F)C2)=O)CCc2n[nH]cc2C1 c1(OC)ccc(NC(c2ccc(Cl)o2)=O)c(C)c1.N12CC(C3CC13)C2=O N1(c2nnn(C)n2)CCC2(COC(CNC(C3CCn4c(cnc4C)C3)=O)C2)C1 C1(C(=O)NCC(C#C)CC)CCN(C(C2CCCCC2(C)C)=O)CCO1 c1(C(=O)NC(CNC(C2C(C(=O)OC)C2)=O)C(C)(C)C)ccnc(F)c1OC c1(C(=O)NC(CCC)CNC(=O)C(F)(F)C2CCC2)cc(=O)c(OC)c[nH]1 C1(CCNC(c2cnc(C(C)C)s2)=O)CN(C(=O)C2=NOCC2)CC(C)O1 N1(C(c2n3c(nn2)SC(=C)C3)=O)C2CCC1CN(C(C1CCCCS1)=O)CC2 c1(OCC)ccc(NC(C2CSCN2C(c2ccc(O)cc2)=O)=O)cc1 Cc1c(C#N)c(O)nc(=N)[nH]1.C(=O)(C(C(C)C)C(C)C)NCC(=O)CNC c1(C(N2CCC(C(C)NC(=O)CN3CCOCC3)C2)=O)cncc(F)n1 c1(C(=O)NCCCNC(c2cncc(N(C)C)n2)=O)c(N)cc(Cl)cc1F c1(NCCCCCCN(C(=O)CC2(n3cccn3)CC2)C)cc(O)nc(Cl)c1 c1(C(=O)NCC2CCC(NC(C(C3CC3)OC)=O)CC2)ccc(F)c(C(F)F)n1 c1(C(=O)OC)ccc(C(=O)NC2CC2CNC(=O)C(c2ccccc2)C)cn1 c1(OC)cc(C(=O)NC2CC(NC(c3cc(C)cc(Cl)n3)=O)CC2O)cc(F)n1 c1(C(=O)NC2CCN(C(c3c(CC)cco3)=O)CC2C)cnc2[nH]cncc1-2 c1(C(=O)NCC2N(CC)CCC2)ccc(C)c(CO)c1.C12CN(CC1OC)C2=O c1(C(N2CCC(c3nn[nH]n3)(C(=O)OCC)C2)=O)ccc(C)c(Cl)c1 Cn1cncc(C(=O)NCCCC(N2CCOC3CC23)=O)c1=O c1(CC)sc(C(=O)NCCOCCNC(c2coc(C)c2)=O)cc1C C1(NC(c2cc(CNC(C3C(C(N)=O)COC3)=O)on2)=O)CCC(C#N)CC1 C(=O)(C1CCCc2ccnn21)NCC1CCN(C(C(C)=CC2CC2)=O)C12CCC2 Cc1cc(NC(c2c(Br)n[nH]c2C)=O)ccc1NC(c1cc[nH]c(=N)n1)=O N1(C(C2(C)CNC(=O)C2)=O)CCc2[nH]nc(CNC(C3CC=CC3)=O)c2C1 CC1(C)NC(=O)CCC1NC(=O)CCOCCNC(=O)COC1CCOC1 N1(C(C(CC)C)=O)CCC(NC(=O)CCc2nncs2)C1C(C)(C)C c1(C(=O)NCC2C(NC(C=CCCC)=O)C2)cnc2snc(C)c2c1 NC(=O)CCCC(=O)N1CCCCCC1CNC(C1(CC2CCC2)CC1)=O c1(C(=O)NC2(COC)CCCOC2)n[nH]c2c(C(=O)O)cccc12 C1(C(C)NC(COCC(C)C)=O)CCN(C(c2cnn(-c3cccnc3)c2)=O)C1 c1(CC)cc(C(=O)NCC(C)(CO)NC(=O)C(O)Cc2ccccn2)c(C)nn1 c1(C(N2CC(N(C(C(CC(C)C)NC(C)=O)=O)C)C2)=O)ccc2ccccc2n1 c1(C(=O)NCC2CN(C(C3(SC)CC(O)C3)=O)C2)cccc(C#N)c1 CC1(C(=O)NC2CCC2CNC(=O)Cn2nnc(C(C)(C)C)n2)CCCCC1(F)F c1(C(=O)NCCCC(C)NC(C2C(C)C2)=O)ccccc1CS(C)(=O)=O Cc1ccc(F)cc1CCNC(=O)NCC1CCN(S(=O)(=O)c2cccs2)CC1 C12(N(C(C(C)NC(CC)(C)C)=O)C)CCCC1OCC2.C12CCN(C1)C2 C(CC(CC)C(=O)NCCCC(C)(C)NC(c1ccc(N)c(SC)c1)=O)=CC CCC(C)C(=O)NC(Cn1cccn1)C(=O)N(C)CCn1cnnc1 O=C1CC(NC(C2CN(Cc3cccc4cccnc34)C2)=O)C2CCCCC2N1 Cc1ccc2ncc(C(=O)N(C)CCN(C)C(C3COC(C)(C)O3)=O)cc2c1 c1(NCC2CCN(C(=O)OC)CC2)nccc(=NCC2=COCCO2)[nH]1 CC(C)CS(=O)(=O)N1CCC(N(C)CC2CCN(S(=O)(=O)C(F)(F)F)CC2)CC1 C(=O)(C(C)CC(N)=O)NCC1(OC)CN(C(=O)CCc2cccnc2C)C1 C(=O)(CCCC(=O)C1CC1)N1CCCC(C(=O)NCC2C(C)CCC2)C1 N1(C(c2cnc(OC)s2)=O)CCCC(C(N2CCC(C#N)C2)=O)C1 CC(C)CCC(=O)C(=O)NC1(CC(=O)NCc2nnc(O)n2C(C)C)CCC1 c1(N(C)CC)ccc(C(=O)NCCCCC(C)NC(=O)CN(C)C2CC2)cc1 c1(C(=O)NC(C)C(C)NC(C2(F)CCCCCC2)=O)ccc(S(N)(=O)=O)cc1 c1(C(N2C(CCNC(CC(C)C3CCCO3)=O)CCC2)=O)cc2sccc2s1 c1(C(N2CCC(C(=O)NC3CCCC3(C)OC)(CC)C2)=O)cc2cc[nH]c2cn1 N1(C(C)=O)CCCN(C(c2cnn(C)c2)=O)CC1 N1(C(CC)=O)CCCC(NC(C2CCCN2C(c2cc(C)oc2CC)=O)=O)C1 C1(OC)(OC)CCCN(C(=NCc2cc(C3CCCC3)n[nH]2)NC2CCC2)C1 C(=O)(CC(C(F)F)c1cccc(F)c1)NC(C1(CNC(CC(C)OC)=O)CC1)C C1(CNC(c2cnc(OC)s2)=O)C(C)CCCN1C(=O)C(O)CC1CCCC1 C1(C(=O)NCCCCCNC(CC2CC(=O)C2)=O)CC12CCOc1ccccc12 N1(C(CCC#CC)=O)CC(N=[N+]=[N-])CC1C(=O)NC1C(C)CCC1C C1(C(=O)NCC(C)(C)NC(=O)CNC(c2ccoc2)=O)CCN(C2CC2)C1=O c1(CC(=O)NC2CC3(C(Nc4nc(CC)nc(C)c4)C3)C2)ccc2nonc2c1 C(=O)(C(C)(F)C(=O)N1CCC(c2cn(C3CC(F)(F)C3)nn2)C1)OC C(=O)(C1=CCN(C(c2n[nH]cc2-c2cccc(C)c2OC)=O)C1)OC C(=O)(CC(C)C(C)(C)C)NC(CC1CN(C(CCCCN(C(C)C)C)=O)C1)C C1(N(C)C)COCC1C(=O)NCc1cncnc1.C1C(=O)NCCO1 C#Cc1ccc(C(=O)NCC2(O)CCCN(C(=O)COCC(=O)NC)C2)c(F)c1 N1(C(C(C=C)CC)=O)CC(C)CN(C(c2cccc3c2CCO3)=O)CC1C C=CCC(CNC(=O)CC1CC2CC2C1)C(=O)NCCC1(C)CCCC1 c1(C2(CNC(=O)NC3(CF)CC3)CCC2)conc1C(F)(F)F N1(C(C2(OC)CC2)=O)CCCOC(CCNC(C2(C)CCNC2=O)=O)C1 Cc1nc2[nH]c(C(N3CCC(NC(c4c[nH]cc4C)=O)CC3)=O)cc2s1 C1(C(N(C(C)C(=O)N(c2ccccc2)C)CC=C)=O)CCCC1NC(C)(C)C C1(CNC(c2cn(C)nc2)=O)CN(C(=O)C(C)(C)F)CCC1c1ccccc1 N1(C(CNC(CN(CC(=O)NC(C)(C)C)C)=O)=O)CCCC(F)C1O N1(c2nc(OC)c(F)c(C)n2)CCC2(CN(C(C3(C(N)=O)CC3)=O)CCO2)C1 c1(CC)nc(C(=O)N(C2CCCCC2)CCNC(c2c[nH]nc2OC)=O)n[nH]1 N1(C(C(C)(C)OC)=O)CC2CC1(CNC(C1(C)CCOCC1)=O)C2 N1(C(c2occ(C)c2)=O)CCC(NC(C2NC(=O)C3CC23)=O)CC(C)(C)C1 Cc1cc(C(=O)NCC(C)(C)NC(=O)Cc2cscn2)cnn1 N1(C(CN(C(Cn2c(C)ccn2)=O)C(C)C)=O)CCC(C2=NOCC2)C1 c1(CCOCCOC)n[nH]cc1NC(=O)NC1(C(F)(F)F)CCC1 C1(NC(C(COCC)C)=O)(CC)CCN(C(=O)CC2CCOC2(C)C)CC1 C(=O)(C(C)CC(F)F)NC1C(CNC(Cn2nc(C)c(Cl)c2)=O)COC1 CC1(NC(C2SC3C=CC2CC3)=O)CCC(NC(=O)CN2C(=O)CNC2=O)CC1 C(=O)(C1CCCc2ncnn21)NC1COCCN(C(CCC(=O)OC)=O)C1 O=C(C1CCCc2scnc21)NC1CCC2CN(c3ncc(F)cn3)CC2C1 c1(NCC(c2ncc(C)nc2)=O)nc(N(CCC(C)C)C)nc2ncn(C)c12 c1(C(N(C)CCN(C)C(C23CCCC2C3)=O)=O)c(-n2cccc2)sc2c1CCC2 C1(NC(=O)Cc2cscn2)CCCCN(C(c2cc(F)cc(F)c2)=O)CC1 N1(C(c2c(C)c[nH]n2)=O)CCCC2(C1)CN(C(=O)C(C)CN(C)C)CCO2 c1(CN=C(NC(C2(CO)CCCC2)C)NCC2CC2)ccc2c(c1)NC(=O)CO2 Cc1ccc(O)c(NC(C2CC2C(=O)NCCOc2c(C)cccc2Cl)=O)n1 N1(C(c2n(C)ncc2C2CC2)=O)CC2(CC(NC(C3CC3C(C)(F)F)=O)C2)C1 N(C)(C[Si](C)(C)C)C(C1(NC(C(=O)NC(C)C)=O)CCSC1)=O C1(CC(=O)NC2CC(O)(CNC(c3csnn3)=O)C2)CCC12CCC2 c1(C(=O)NC2(C3CN(C(C4C(OCC)C4)=O)C3)CC2)cc2c(O)cccc2[nH]1 Cc1coc(C(=O)NCCC2CCCCN2C(C2CCSC2)=O)c1C C(=O)(C(O)CC(C)(C)C)N(C)CC1CN(C(c2nncs2)=O)CC12CC2 c1(OC)cncc(C(=O)N(C(C)CN(C(=O)CCCc2ccccc2Cl)C)C)c1 N1(C(CS(=O)(=O)NC)=O)CC2CCC1C(NC(=O)CCCCC1CC1)C2 N1(C(C2C=C(C)CS2)=O)CCC(C2CCN(C(=O)C(C)(C)n3cnnn3)CC2)C1 C(CCCCCNC(c1csc(C(C)OCC)n1)=O)NC(C1(COC)COC1)=O C1(F)(CNC(C2CCN(C(CC)=O)C2)=O)CCN(C(=O)Cn2[nH]cnc2=N)C1 C1(C(N(C2CCN(C(=O)CCc3nccs3)CC2)CC)=O)CCC(C)(C)C1 C1(N(C)C(C2CCCC2c2nc[nH]n2)=O)CCCC2(C1)N=N2 CC1(NC(=O)CC2CCC(=O)O2)CCCN(C(C2CN3CCN2CC3)=O)C1 c1(CN(C)C)ccc(NC2CN(CCOc3ccccc3F)C2(C)C)cc1 CCCCS(=O)(=O)N1CC(C(=O)NC2C=CCN(C(=O)C=CS(C)=O)C2)C1 c1(C(=O)NCC23C(CN(C(C(=O)C=Cc4cccs4)=O)C2)C3)ccc([N+](=O)[O-])cc1 c1(OC)cc(C#N)ccc1C(N1CCC(C(=O)Nc2cc(F)c(C)cc2F)C1)=O CCC(C#N)C(=O)N1CCC(CC(C)NC(=O)C[SH2](CC(=O)N(C)C)=O)CC1.OC c1(C(N(C2CCN(C(=O)C(C(C)C)SC)C2)CC)=O)cnn2cccc(Cl)c12 N1(C(CCC(C)OC)=O)CC2(C=C(C(=O)N(CCCC(F)(F)F)C)CO2)C1 C1(CC(=O)NC2C(NC(c3n(C)nnc3)=O)CCCC2)CCc2ccccc2C1 CC(C)C(C(=O)N1CC(O)CCC1C(=O)Nc1cccc(N(C)C)c1)C(C)C c1(CC)cccc2c(C(=O)NCC3(F)CN(C(c4cc(O)nn4C)=O)C3)c[nH]c12 C1(NC(C2(S(N)(=O)=O)CC=CC2)=O)CCCC2CN(C(=O)C=CI)CC12 C(C1CCc2ccc(Br)cc21)NC(c1ccc(-c2ccncc2)cn1)=O c12ccnc(c1)C(=O)N1CC(C1)O2.C1(C(=O)OC)CC1C(=O)N(CCF)C1CC1 CCN=C(NCCOC(c1cccc(NC)c1)=O)NN(C1CN(C)CCO1)C N1(C(C(CC)=CC)=O)CCC(NC(c2cc(F)c(F)cc2Cl)=O)CC(O)C1 N1(Cc2cccc(OC)c2O)CCC2(CCN(C(c3ncn(C)n3)=O)CC2)CC1 N1(C(c2c(N)cn(C)n2)=O)CC(NC(c2cc(C3CC3)cs2)=O)CC(F)C1 Cc1cc(C(=O)NC2(CF)CCN(C(C3CCC(=O)N(C)C3)=O)C2)ncc1CO CC(CC(N)=O)C(=O)N1CCOCC1C(=O)N(C)Cc1cnnn1C c1(C(N2CC3(C2)CN(C(C2CCCCC2(F)F)=O)C3)=O)nccc2cccnc12 c1(CC)nocc1C(=O)NCCC(=O)NC(c1cnccn1)C C1(C)(COC)CN(C(=O)C(Cn2ccnn2)NC(=O)CC2CCCC2)C1 C1(CNC(C2C(C)CN(S(=O)(=O)C(C)C)CC2)=O)CC(C)(C)OC1(C)C C(C)(CO)(C(=O)NCC(O)CC(=O)NCC(O)CC1CC1)OC C1(C(=O)NCCC(C)NC(=O)Cn2nc(C3CC3)cc2C(F)F)CCS(=O)(=O)C1 c1(COC)cc(-c2ccc(NC(c3ccns3)=O)nc2)ccc1F C1(O)(C(C)NC(C(C)OC2CCCC2)=O)CN(C(=O)C(F)(F)C2(O)CCCC2)C1 CCCC(C)(C)C(=O)NC(C1CCCN1C(=O)CSc1ccc(C)cc1)C c1(C(=O)NCCC2N(C(C(CCCOC)C)=O)CCCC2)cc2ccccn2c1 Cc1cc(Br)c(CC(=O)NC(c2cn(CCCN3CCCC3)nn2)C)s1 C1(C(=O)NCC2CCN(C(C(c3cncnc3)C)=O)C2)CCC2CC1CO2 N1(C(CN(S(CC)(=O)=O)C)=O)CCC(COC)(NC(=O)CCc2cccn2C)C1 CC1CC(CNC(c2ccc(CN=[N+]=[N-])cc2)=O)CN1C(=O)Cn1ncnn1 N1(C(C2(OC(C)=O)CC2)=O)CC(NC(=O)CCC(F)(F)F)CC(C)(C)C1 CC(c1ccccc1)=CC(=O)O.N12CCCC1SCCC2=O CC(C)(CCCCNC(=O)CS(=O)(=O)C1CC1)C(=O)NNC(=O)CCC(F)F C(=O)(C(C)CS(C)(=O)=O)NC1C(NC(Cc2c(C)ncs2)=O)CC1 C1(N(C(CCNC(C)=O)=O)C)CN(C(=O)C=Cc2ccnn2C(C)(C)C)CC1O C(=O)(C(C)C(C)S(C)(=O)=O)NC(CN(C(C=Cc1c(C)cccc1)=O)C)C Cn1ncc(C(=O)NC2CC=CCC2C(N2CCOCC2C(F)F)=O)c1N N1(C(CCC(CC)OC)=O)CCC2C(CCCN2C(c2cc[nH]c(=NC)c2)=O)C1 C1(C(=O)NCC2C3CN(C(c4cc(CO)c(C)o4)=O)CC23)(COC)CCOCC1 N1(C(C(c2ccccc2)OC(C)=O)=O)CCCC(N(C(=O)CS(C)(=O)=O)C)CC1 N(C1COCc2ccccc21)C(C)=O.c12ccc(c(F)c1)c(=O)o2 C(C(C)(C(=O)NCCC(C)c1cn[nH]c1)NC(c1c[nH]c(C(N)=O)c1)=O)SC C1(C(=O)NCCCOCCCNC(C=C(C)C(F)F)=O)CCOC1C(F)(F)F c1(C(=O)NCC2N(C(C(C)C3CC3)=O)CCC2)cc2n(n1)CC(F)C2 N1(C(C2C(C)(C)C2)=O)CC(CNC(c2cc(Cl)c(F)cc2O)=O)C2(CCC2)C1 c1(C(=O)NC(COCC)C(=O)NC(CO)CCSC)cc(C)nc(C)c1 CC1CN2CCN1C(C(N1CC(C(C)NC(c3ccc(C(C)(C)C)s3)=O)C1)=O)C2 CN1CCC(C(=O)NC2CCC(F)(CNC(c3nnn(C)c3N)=O)C2)CC1 n1(CC(=O)N(CC(CN(C(C(COCC)C)=O)C)O)C)ccc(C)cc1=O c1(C(=O)NCCN(C(CN(CC)CC)=O)C2CC2)ccc(F)cc1C#N N1(C(=O)Cc2ccc(Br)cc2Cl)CC2CCN(C(C3CCCCO3)=O)C2C1 CC1(NC(=O)CC2(CO)CCOCC2)CCCN(C(=O)C2CC2)C1 c1(C(N2C(C#N)CC2)C(=O)NC2CCCC2)ccc(Cl)cc1 C1(CNC(C2C3CC2(c2ccccc2)CO3)=O)CC2(CCCC2)CO1 c1(CCC(=O)N(CC(C)NC(C2(C)CC(=C)C2)=O)C)cc(F)ccc1Br C#CCCCCC(c1nnnn1CC1CCCO1)NS(=O)(=O)C(F)(F)F C(C(C(C)C)NC(=O)Cc1ccsc1Cl)(c1ccccc1)NC(C1CC(=C)C1)=O CN(C)NC(=O)CCC(=O)NC1CC1C1CCCN(C(=O)CC2CCCOC2)C1 C(=O)(N=c1c(C)c[nH]cc1Br)C1C(NC(c2cc(OC)c(I)cc2)=O)C1 N1(C(CNS(N)(=O)=O)=O)CCC2C(C1)CN2C(c1cnc(Cl)cc1C(F)F)=O C(CC(C(C)C)NC(c1c[nH]nc1F)=O)NC(C(CC)OCC)=O N1(C(C(C)NC(=O)C(C)(C)C2(O)CCC2)=O)CC(F)CC1C CCC(CC)(CCNC(c1ccn(C2CC2)n1)=O)NC(c1nc(C)sc1C)=O c1(C(=O)NC2CC3CC(NC(C(C)(C)SC)=O)CC32)cc(C)cc2nc[nH]c12 C=CCCCCCC(=O)N(CC(C)O)CCNC(c1cnn(C)c1)=O CCC(F)(F)C(=O)NC1CCC1NC(c1cnn(CCO)c1C(C)C)=O C(=O)(C#CC1(C)CC1)NCC1CN(C(CCCCOC)=O)C1 c1(C(=O)NC(CC)CC(=O)N2CCOCC2C2(C)CC2)cc2occc2[nH]1 C(=O)(C(C)(C)c1cc[nH]n1)NCC1(CC(=O)NC2(CC#C)CC2)CC1 c1(C(N2CC(C(N)=O)(CNC(c3cn(C)c(=O)n3C)=O)C2)=O)c(F)ccc(F)c1F C1(CN=C(NCCOC(C)C)NC2CN(S(C)(=O)=O)C2)CCCS(=O)(=O)C1 N1(C(CN(C(C)=O)C)=O)CCCC2CN(C(c3cnc(N)c(O)c3)=O)CC12 C#CCC(C)(CC)C(=O)NCC(C)(C)CC1CN(C(c2ccncc2Cl)=O)C1 C#CC(C)NC(=O)C=CCN(C(=O)CN(C1CC1)CC)C C1(COC)CN(C(C2(CCC(F)(F)F)CCC2)=O)CCN1C(C1(C)CC=CC1)=O c1(SC)ccc(SC)cc1.C12CCCC(C1)NC(=O)C1CC(O)(C1)c1cn2nn1 c1(CCN(CCOCC)C)cn(CC(C)NC(=O)Cc2cscn2)nn1 C1(NC(C=C(CC)CC)=O)CCC2(CC1)CCN(C(C1CCC(O)C1)=O)CC2 N1(C(c2nccc(C)c2)=O)CC2CCC1CN2C(c1cc(Cl)c(F)cc1F)=O C1(CC)CC(C)CN(C(c2nc(NC(=O)CC3(C)CCC3)cn2C)=O)C1 N1(C(c2nc(CC)oc2)=O)CCC(C2CCCN(C(=O)CCC3CC3)C2)CC1 c1(C(=O)NCc2ccnc(N3CCOCC3)n2)sc2ccccc2c1Br c1(CC(=O)N(CC(C)NC(=O)C(C2CC2)N(C)C)CC)csc2nc(C)cn12 N1(C(C(C)(C)OC(C)=O)=O)CC2(CCN(C(=O)C(C3CC(F)(F)C3)N(C)C)C2)C1 c1(C(N2C(CN(C(=O)Cc3cn(CC)nn3)CC)CCC2)=O)cc([N+](=O)[O-])n[nH]1 C1(N(C(=O)C(=O)Nc2ncc[nH]2)C(Cc2c(C)ocn2)=O)CCCN(C(C)C)C1 c1(C(=O)OC)no[nH]c1=NC(=O)Cc1ccc(CC(=O)NC(C)(CO)CO)cc1 C=CC1(CC(N2CC(N3CCCC3)C2)=O)CN(C(C2(C(C)=O)CC2)=O)C1 N1(C(c2c(OC)scc2)=O)CC2CCC2(CC(=O)NCC2CC(F)(F)C2)C1 c1(N2CC(C)(COC)OCC2)nc(=NCC2CC3CC3C2)[nH]c2c1CCC2 C(CNC(c1ccc(C(=O)N(C)CC)cc1)=O)(CC(C)C)CCNC(CC=C)=O C=CCC(CC(C)C)C(=O)NC(CNC(c1ccc(F)c(F)c1C)=O)C1CC1 C12CC(O)CN1C(=O)C2.C(C(O)CO)(C1CC1)NC(C1CC1C(F)(F)F)=O C1(CC(C)NC(C(C)=C2CC2)=O)CC2CCC(C1)N2C(=O)C(C)(C)C(C)C CC1CCCC=C1C(=O)NC1(C2CN(C(C3(C)CCC3)=O)C2)CC1 C1(NC(C(C)C2CCC2)=O)CCN(C(c2cc(C(F)F)ncn2)=O)C12CCC2 C1(NC(C2CCC(=O)NC2)=O)CC2CC(C1)N(C(=O)Cc1cc[nH]c1)C2 CN=c1[nH]c(C(N2CC(CNC(C3(F)CCOC3)=O)(COC)C2)=O)cs1 CC(CN=c1[nH]c(C#N)c(Cl)s1)(C1CC1)NC(c1ccc2c(c1)CCOC2)=O C12(C(=O)NCC(C(C)(C)C)NC(C3CCC(N(C)C)CC3)=O)CC3CC1C2C3O C=CCC(CC=C)C(=O)NC(C)(C(=O)NC1CC2CCC(C1)O2)C1CCC1 CC1CCCC(C(=O)NC(C)(C)CN2CCN(C(=O)C=CC(N)=O)CC2)CC1 C#CCC(CC#C)C(=O)NCC1CCN1Cc1ccc(F)c(F)c1 C1(C(C)C)CC1C(=O)NCC(C1CC1)NC(C1CC1C(C)(F)F)=O N1(C(C2C(C=C)C2)=O)CCN(C(=O)C=C2CCCCC2)C(CC(F)(F)F)C1 C1(NC(C(C)NC(CC)=O)=O)CCC(N(C)C(c2cc(C(C)=O)on2)=O)CC1 C1(Cc2ccc(OC)cc2)CCN(C(=O)NCc2ncc[nH]2)CC1(F)F N1(C(C2CCCN(CC)C2)=O)CCC(C(=O)NCC2(CF)CC(F)(F)C2)=C(F)C1 C1(CC(=O)NC2(CC(=O)NC3(C(O)CO)CC3)CCC2)CCOC1=O C1(NC(c2ccncc2F)=O)CCC2CC1CN2C(c1cccc2cncn12)=O C12(OC)CCC(C(=O)NCC3N(C(CCCC=C)=O)CCC3C)(CC1)C2 N1(C(c2cc(C(C)C)on2)=O)CCCCCC(NC(C2(F)CCS(=O)(=O)C2)=O)C1 CCC(C)(C(=O)N1CC(NC(=O)OC(C)(C)C)C(c2ccccc2)C1)OC CCCCCCCC(=O)N(C(c1csc(C)c1C)C(=O)Nc1ccccc1)C c1(C(N2CC(NC(CC=CC=C)=O)C(F)CC2)=O)cc(Br)cc2c1OCC2 C1(CNC(C(C)n2ccnc2)=O)CCCCCN1C(c1cn2c(n1)SCC2)=O c1(C(=O)NCCC2CC(NC(C(N3CCNC3=O)C)=O)C2)cn2cccnc2n1 N1(C(c2c(CC(=O)OCC)scc2)=O)CCC(CNC(=O)C=CBr)C(C)C1 N12CCC(CC1)C(C)C(=O)NCC(C)SCC2=O.C1(SCC#C)CCCC1 C12(CNC(c3cc(CC)no3)=O)CCCCC1N(C(=O)CC(F)(F)C(F)F)CC2 C1(NC(c2c(CC=C)cccc2)=O)CC12CCN(C(c1ccc(F)s1)=O)C2 C1(N(C)C(C2CSCCS2)=O)CC2CC1N(C(c1cc(C(F)F)ccn1)=O)C2 c1(C(=O)NCC(C)CN(C)C(C2(C)CC(C)(C)C2)=O)cc2ccccc2s1 c1(C(N(C)CCNC(C23COC(CF)(C2)C3)=O)=O)c(Cl)cccc1Cl N(C(=NCCOCC(C)(C)C)N1CCCC(S(C)(=O)=O)C1)CCSC Cc1c(C)c(C)c(C(=O)OCc2nc3ccc(Cl)cc3s2)c(C)c1C c1(C(=O)Nc2ccc(-c3c(CCC)onc3C)cc2)ccnc(O)c1F Cn1nccc(C(N2CC(O)(CNC(C3CCCCS3(=O)=O)=O)C2)=O)c1=O C1(N)CCCN(C(=O)CCC(C(C)NS(CC)(=O)=O)=O)CC1.c1ccc(F)nc1 C(=O)(C(=O)CCC(C)C)N1CC(n2cc(CNC(c3c(SC)cn(C)n3)=O)nn2)C1 N1(C(Cc2ccc(OC)cc2)=O)CCCCCC(NC(c2c(C)ncn2C)=O)C1 C1(NC(c2c(C)nc[nH]2)=O)C2CC1N(C(c1ccc(OCC3CC3)cc1)=O)C2C c1(C(=O)NCCN(CCCCCC)C(c2nnsc2C)=O)c(C)ccc(C)c1N c1(C(=O)NC(CCCNC(Cc2cn(CC)nn2)=O)C)cc(F)c(C)cc1N N1(C(CSCCC)=O)CCC(NC(=O)C=Cc2ccc(Cl)cc2)C12CC2 C1(NC(C(CC)COC)=O)C2CCCN(C(C3CC(=C4CCC4)C3)=O)C2C1(C)C C1(CC(=O)NC(c2cccnc2)C(=O)NCc2ncc(CC)o2)CC(O)C1(C)C c1(C(=O)NCC2(F)CC(CNC(C=C(C)C(F)F)=O)C2)cnc2nccn2c1 c1(CCC(=O)NC2CC(C)N(C(C3CCCCO3)=O)C2)ccc2c(c1)OCCO2 Cc1ccccc1CC(=O)NC(C)(C)CNC(C1CCC(=O)C1)=O N1(C(C(COC(C)=O)C)=O)C2CCC1CN(C(=O)C(O)c1ccco1)CC2 c1(C(N2CCCC(CN(C(c3ccc(C)o3)=O)C)C2)=O)ccc(S(C)(=O)=O)[nH]1 N1(C(CN)=O)CCCC(CC(=O)C(=O)CC2(C)CS(=O)(=O)C2)C1.CC(=O)NC C1(NC(CC=C=C)=O)CN(C(=O)C(CC=C)OC)C(C)(C)C1 C1(CNC(CCN(C(CCC)C)C)=O)CC2COCC2N1C(=O)CCC(C)SC c1(C(=O)NC2CCC(CNC(C3(OCC)CCC3)=O)C2)cc(F)cc(F)c1N n1(CC(N2CCC(C)(NC(CCSc3nc(C)[nH]n3)=O)C2)=O)nc(C)n(C)c1=O CC(C)(C(=O)NCC1CCC(NC(c2ocnc2C2CC2)=O)C1)C(F)(F)F c1(C(N2CC(C(=O)NC(c3ccno3)C)OCC2)=O)cc2cnccc2[nH]1 N1(C(C2C(CC)C2)=O)Cc2ccccc2C(NC(c2ccoc2Cl)=O)C1 c1(CNC(c2cncc(OC)n2)=O)nc2c(s1)CCN(C(C1CC(C)C1)=O)C2 Cc1cccc(OCCC(=O)NC(C)CC(C)NC(c2cc(F)cs2)=O)c1C c1(NC(C2C(NC(C3CCC(O)C3)=O)CC2)=O)ccc2cccnc2c1 c1(C(=O)NC(C(=O)NCCC(=O)NCC)CCOC)cnc(O)c(C)c1 c1(NC(C2N(Cc3ccc(C)c(C)c3)CCSC2)=O)cc2c[nH]nc2cc1Br N1(C(CC=C(C)C)=O)CCCC1C1CCN(C(C2CCN(CC(C)C)C2)=O)C1 Cn1cc(C=CC(=O)NCCCNC(C2(C)CCC(=O)C2)=O)c(=O)n(C)c1=O N1(C(C(C)(C)CO)=O)CC2(C)CN(C(c3nc(Br)cnc3N)=O)CC2(C)C1 CC1(C)C(C(=O)NCCOC2CCN(C(=O)CSC(F)F)C2)C1C#N C1(CNC(N2C(C=C)CCCC2)=O)CCCc2ccccc2C1 C1(CC(=O)NC(C=C)C2CCC2)CCCN1C(=O)C(C)CC c1(OC)nc(OC)nc(N2CCCC(CO)(NC(C3CNC(=O)N3)=O)C2)n1 N1(C(C(CC=C)(C)OC)=O)CCC2(CC(C(=O)NC3CC=C(C(C)C)CC3)C2)C1 N1(C(c2cc(F)cs2)=O)CC(F)(F)CC1CO N1(C(C)C)N=C(C(=O)NCCN(C)C(C2OC3CCC2CC3)=O)CCC1=O N1(C(c2ncn(CC)n2)=O)CC2CCN(C(C3CC(C)(O)C3)=O)CC(C2)C1 C(C(N=[N+]=[N-])C(=O)N(C)CC1CCN(C(c2ncc(C(N)=O)cc2Cl)=O)C1)OCC c1(CC)oc(C(=O)NCC(C)N(C(=O)C(c2cccc(OC)c2)=O)C)cc1C Cc1nc2c(o1)CCN(C(=NCc1ccc(F)cc1)NCC(F)C(F)(F)F)C2 C1(CNC)CCC2(CCCC2)C1.c12nc(cc(O)n1)CNC(=O)CCC(=O)NC2 c1(OC)ccc(CNC(=O)CC2CN(Cc3c(O)cccc3Cl)C2)c(C)c1OC c1(C(=O)OC)ccc2cc(NC(=O)NCC(=O)OC(C3CCCO3)C)ccc2c1 C1(NC(Cc2c(C)n[nH]c2)=O)CC2CCC1C(NC(=O)Cc1cccnc1O)C2 Cc1nc(O)nc(C)c1C(N1CC(OCCNC(c2ocnc2C(F)F)=O)C1)=O C1(C(=O)NCc2ccc(C#N)cn2)C2CC(O)C(C2)N1C(=O)C(F)(F)CO CC(O)C(C(=O)N1CCC(CCNC(=O)CCSc2nccn2C)C1)N(C)C C1(C(C)C)C(NC(=O)C(F)=CC2CC2)CCN1C(C1C2CN(C)CC12)=O N1(C(C(C2CCC2)OC)=O)C2CCCC1CN(C(=O)COC1CCCC1)CC2 Cc1cc(C(=O)NCc2cccc(NC(=O)CC(C)C(F)F)c2)c2c(c1)CCO2 C1(NC(COCCOC)=O)CC2CC1CN(C(=O)CCCn1ccnn1)C2 c1(OC)ccccc1CCC(=O)NC1CCN(C(c2nn(C)cc2Cl)=O)C1 CC(CC(=O)NC1CC(CN=c2cc[nH]c(-c3nccs3)n2)C1)P(C)(C)=O c1(C(=O)NC2CCC(CCNC(c3c(CC)cco3)=O)C2)cc(F)cc(N)c1F c1(NC(CC2CC(C)N(C(=O)Cn3[nH]cnc3=N)C2)=O)ccc2nncn2c1 N1(C(c2c(C)n[nH]c2)=O)CC2C(CN(C)C(c3cc(N)ccn3)=O)C2C1 c1(C(=O)NC2C(NC(c3nc(N(C)C)oc3)=O)COC2)ccc([N+](=O)[O-])c(Cl)c1 C1(C#N)(C(=O)NCC(CNC(C(CC)c2cccnc2)=O)F)CCOCC1 c1(C(=O)NCCC(C)Nc2nnc(C(=O)OCC)s2)ccc(C)c2[nH]c(C)cc12 c1(C(N2CC3CC(CNC(C4(CC)CC4)=O)C3C2)=O)c(O)nnc2c1COCC2 C=CC(C)(CC)C(=O)NC1C2CCC(C2)C1C(=O)N(C)CCc1cccs1 N1(C(C2C(C(C)C)C2)=O)CC2CCC(C1)N2C(=O)CSc1cccc(Cl)c1 CN1CCC(N2CCC(NC(=O)NC3(CO)CCCC3)C2)C1=O C1(=O)C(C)(CC)CO1.C1(c2nnc(C(C)C)o2)(CC#C)CC=CCC1 N1(C(CCC)=O)CC(NC(c2cc(-c3ccns3)on2)=O)C(C2CC2)C1 C1(C2CCN(C(c3ccc4nsnc4c3)=O)C2)(NC(C(CCCC)O)=O)CC1 C(=O)(CC1=CCCC1)OC.C12CC(n3cc(CCS(C)(=O)=O)nn3)CN1C2=O c1(C(=O)NC(C2CCN(C(c3ccncc3F)=O)CC2)C)ccn(C)c(=O)c1 N1(C(C(CCOCC)NC(=O)CC=CC(C)(C)C)=O)CCOCC(OC)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCCCC1CCC(=O)NCC(F)(F)Cl C(c1ccc(C)cc1)=CC(=O)NCc1c(C(N(CC(CC)(O)CC)C)=O)con1 N#CC1CCC(NC(C2CN(C(=O)COCC3CCOC3)C2)=O)CC1 C1(C(=O)NC2CN(C(c3ccc(F)cc3F)=O)C2)CCc2cnnn2C1 C1(CNC(Cc2cc(C(C)C)no2)=O)CN(C(=O)C#CC2CC2)CC(C)(C)O1 c1(C(N(CCNC(C2CCC2C2CCCO2)=O)CC)=O)ccc(C)c(C)c1 C12(NC(c3c(C)nc(C4CC4)[nH]3)=O)CCCC1N(C(=O)CCCC1CC1)CC2 Cc1nc2ccc(C(=O)NC(CNC(=O)C(C)S(C)(=O)=O)CO)cc2o1 Nc1cccc(F)c1NC(C1CC(Cn2cc(COC(=N)O)nn2)C1)=O c1(NCCN(C(=O)CC2CCCCO2)C)ncccc1C#N c1(C(=O)NCC2CN(C(c3ccc(NC=O)cn3)=O)C2)coc2c1C(O)CCC2 N1(C(CC(C=C)C)=O)CCCCC(NC(c2cc[nH]n2)=O)CC1 c1(OC)cc(OC)c(NC(C23CC2CN(c2cc(C#N)ncn2)C3)=O)cn1 C1(NC(C(CC)N(C)C)=O)(CNC(=O)CCC2CC2(C)C)CC(F)(F)C1 C(=O)(CCCCC(F)(F)F)NCC12CN(C(C(C)=C3CCCC3)=O)C(C1)CCO2 c1(C(N2CCCC(C)(C(=O)NCCCCC3C(C)C3)C2)=O)ccc(Cl)c(Cl)c1OC Cc1ccc(NC(=O)COCCNC(C2CC(=O)C23CCC3)=O)cc1C#N Cc1cc(C(=O)NCCCNC(=O)C(=O)NCC(C)C)c(O)c(Br)c1 N1(C(c2nccc(CC)c2)=O)CCCC(CC)(NC(=O)C2=NOCC2)C1 C(c1ccc(C)nc1)=CC(=O)NC(CNC(c1cncc(COC)c1)=O)(C)C N1(c2nccc(OCCC)n2)CCC2C(CCCN2C(C2COCCO2)=O)C1 C1(CC(=O)N(C2CCN(C(=O)CC3(O)CCOC3)C2)CC)CC=CCC1 N1(C(C(C(=O)OC)C)=O)CC2(CCCC2)C1C(=O)NOCCC#N S(=O)(=O)(c1ccc(=NCc2cc(Cl)cc(Cl)c2F)[nH]c1)N1CC(C)CS(=O)C1 N1(C(Cn2ccc(C)cc2=O)=O)CCCN(C(C2C=CCCC2)=O)C(C)C1 c1(CC)oc2ccccc2c1C(=O)NC1CC1CNC(=O)C(C1CCOCC1)F CC1C=C(C(=O)NCC2CN(C(=O)C(c3c(F)cccc3F)N(C)C)C2)CC1 C(=O)(C1=COCCC1)N1CCCC(C(N2C(C)(C(C)C)CC2)=O)C1 C(CC(C)(C)C(=O)NC(CC1CC1)CC(N1CCC12CN(C)C2)=O)SC NC(CC(F)F)C(=O)NCc1sccc1I N1(C(c2c(C)nsc2C)=O)CC2OCCN(C(=O)CN3CCNC(=O)C3)C2C1 c1(NC(C2=CCC(NC(c3c(C)cncn3)=O)C2)=O)cc(C)c(O)c(C)c1 C(=O)(CC(O)CNC(C1(C(F)F)CCCC1)=O)Nc1cn(CC)nc1 c1(NC)cccc(CNC(=O)NC(=O)CCc2ccc(Br)cc2)c1 c1(C(=O)NCC(CC)NC(=O)CN2CCCC2CO)nc(C)ccc1O CC1CC(CO)N1C(=O)CN(C(=O)CCc1nncn1C)C1CC1 C1(CNC(c2cc(OC)n[nH]2)=O)CCC(NC(C2(C)CC=CCO2)=O)CC1 CCC(C)(CO)C(=O)N1CCN(C2CCC(NC(C34CCC(CC3)C4)=O)C2)CC1 c1(C(=O)NCCCOCCNC(CC(CC)(F)F)=O)ccc(P(C)(C)=O)s1 C(C1CCCN1C(=O)CCc1ccncc1)=CC(=O)NC1C(C)(C)CC1 N1(C(CCCSC)=O)CC(CNC(c2cccnc2C2CC2)=O)C(C(F)(F)F)C1 CC(C)(C)CC(O)CC(=O)N1CC(O)(CCNC(c2cn[nH]c2)=O)C1 Cc1cc(C(N2CC(C(=O)NC3CCNC(=O)CC3)CC2(C)C)=O)cc(F)c1 c1(CNC(NOCCC(C)C)=O)cccc(-c2cncc(F)c2)c1 CC1(C)CC(C(=O)NCC2C=CCN2C(=O)CNC(c2ccccc2)=O)CCO1 N1(C(CC(=O)NCC)=O)CC2(CC(NC(=O)C(c3ccc(C(C)C)cc3)F)C2)C1 Cc1cc(C(=O)C2CC2)c2[nH]cnc2c1.C1(C(=O)NCC=CCN)(CS)CCC1 c1(C(=O)NC)ccc(CNC2CCCC2CO)cc1OC(F)F c1(C(C)C)nc(=NCC(C)(C2CC2)NC(=O)C(C)n2cncn2)s[nH]1 N1(C(c2n(CC)ncc2C)C(=O)NC2CCCO2)CC2CC(C1)N2CC c1(C(=O)NC2(CNC(C(C)(Cl)Cl)=O)CC2)cccnc1N1CCOCC1 C#CCCCCC(=O)N(CCCCN(C)C(C1CC(=O)N(C(C)C)C1)=O)C C1(C(N(CCC(N)=O)C)=O)CC2C=CC1N(C(C1(N(C)C)CCC1)=O)C2 O=C(N1CCC(O)CO1)Nc1cc(Br)sc1-n1cccc1 CCCC(C)(C)CNC(=O)C(C)(CO)NC(=O)CCc1cncnc1 O=S(=O)(c1ccc2c(c1)OCCO2)NCC1CCN(Cc2ncc(Br)cc2Br)C1 N1(C(CCCOC(C)C)=O)CC2(C1)CN(C(c1c(N)cc(Cl)cc1F)=O)CCO2 CC(CC(=O)N(CCCCCCNC(c1ccnn1CC(F)(F)F)=O)C)C(F)F N1(C(C(C)C)=O)CC2CN(C(c3ccccc3CC#N)=O)CC2C1 N1(C(=O)Cc2cccc(N(C)C)c2)CCC2CN(C(=O)CC3(C)CC3(F)F)C2C1 C1(C)(OC)CCCN(C(=O)CC2CCN(C(=O)CCNc3cccnc3)C2)CC1 C(C(C)(COC)C(=O)N1CCC(COC)(NC(C2CC(C)(C)O2)=O)C1)OC c1(NCC2(OC(C)C)CCOC2)[nH]c(=NCc2cnn(C)c2)nc2ncn(C)c12 c1(CCC)ncoc1C(=O)NCC(C)NC(=O)Cn1nnc(=O)[nH]1 C1(F)(CNC(C(COC)NC(C)=O)=O)CCCN(C(c2cncc(OC)n2)=O)C1 C1(NC(CC2(C=C)CC2)=O)CCC2(CCCN(C(=O)C(C)(F)F)C2)C1 C1(C(N2CCOC(CN(C(=O)CN(C)C3CC3)C)C2)=O)(CC)CCC(F)(F)CC1 C(=O)(CCCC(=O)NC)NC1C(CC)CN(C(=O)CSC(C)C)C1 C(CC(=O)NC(CC)CCCO)(C(F)F)NC(CC=C)=O c1(CCNC(C(C)Oc2ncccc2C(F)(F)F)=O)ccc2occc2c1 C(C)(C)(CC(=O)NCC(c1ccccc1)N(C)C(c1csc(CO)n1)=O)OC CC1=NNC(=O)C1CCC(=O)NCC1CCC1NC(=O)Cc1nn(C)cc1Cl C1(NC(c2cnn(C3CCC3)c2)=O)CCN(C(=O)C#CC2CC2)C(C2CC2)C1 c1(NC(=O)NCC(C(=O)OC)(C)O)nc(C)cc(C)c1Br N1(C(C(CC)CC)=O)CC2CCN(C(c3cc(Cl)cc(C)c3N)=O)CC12 Cc1nc(Br)sc1C(=O)NCCC1CC(NC(c2cncc(O)c2)=O)C1 C(=O)(CCCCCS(=O)(=O)Nc1cccn2cc(C(=O)OC)nc12)OC C(=O)(C(C(C)(C)C)OC(c1ccc(-c2ccc(Cl)cc2Br)cc1)=O)OC CCCC(CCCNC(C12CC(C#N)(C1)C2)=O)NC(=O)COc1cccc(F)c1 c1(OC)cc(OC)cc(CNC(c2c(Cn3ccccc3=O)nnn2C)=O)c1 C1(NC(C2CC2c2ccc(F)cc2F)=O)CCCN(C(C2CCOC2)=O)CC1 C(=O)(C(C1CCC1C(F)(F)F)N(C(C)CC1CCCC1)C)NCC(=C)C C(=O)(C(C)(O)C1CCOCC1)NC(C1CCN(C(c2cnsn2)=O)C1)(C)C N1(C(C=NOC)=O)CCC2C(CCCN2C(c2ccc(F)c3[nH]ccc23)=O)C1 C1(NC(C(=O)NCC2CC2)=O)CCCCCN(C(c2ccc(F)c(Cl)c2)=O)C1 C1(NC(C2C3CNC(=O)C32)=O)CN(C(=O)Cc2ccccc2Cl)CC12CCC2 S(=O)(=O)(c1ccc(S(=O)(=O)NC2CCNC2(C)C)c([N+](=O)[O-])c1)N(C)C C1(NC(CN(C(C)=O)C)=O)CCN(C(=O)CNC(=O)OC(C)(C)C)CC1 C(=O)(C(C)(C)C(N)=O)NCC(CC=C)NC(CCOCC#C)=O C1(CNC(=O)CN2CCCC2)CCCC(CNC(c2csnn2)=O)C1 C#CCC(C)(C(=O)N1CC(OCC(C)C)C1)NC(C1CC2C(C1)C2(F)F)=O N1(C(Cc2ccc(C)nc2)=O)CCN(C(=O)CCC(=O)C2CC2)C2(CCC2)C1 N1(C(C2(C(N)=O)CCC2)=O)CC2CCCC2(NC(=O)CCc2n[nH]c(=N)s2)C1 C(CC(=O)NC1CC(C(=O)NC(CCN(C)C)C(C)C)=CC1O)(C(F)(F)F)OC C1(NC(C2CC(C(C)C)C2)=O)COC2(CCN(C(c3c[nH]ccc3=O)=O)CC2)C1 N1(C(c2cc(OC)n[nH]2)=O)CCN(C(c2ccc(CN(C)C)nc2)=O)C(CO)C1 c1(C(N2CCC(NC(COCCCOC)=O)C2)=O)cc2c(Cl)nccc2o1 c1(C(=O)NC2C=CCC(C(=O)NCC(=O)OCCCC)C2)nccc(C)c1F C1(N(CCc2ccc(C)cc2)C)CCCN(C(c2ccc(Cl)cc2)=O)C1=O CCC(CC(=O)NCC(C)(C)CN(C)C(C1CCN1S(C)(=O)=O)=O)SC C1(N(CCN(C)CCO)C)CCc2ccccc2NC1=O C(=O)(C1=C(Cl)CCCC1)N1CC(CCCCNC(C(C)NS(C)(=O)=O)=O)C1 CN1CC(O)CCC1C(N1CCC(C(C)(C)NC(=O)Cc2ccc(F)cc2)C1)=O C1(C(=O)NCCN(C(CCC#C)=O)CC2CC2)CCN(C)C(=O)C1 C1(NC(c2n(C3(C)CC3)nnn2)c2cnn(CCF)c2)CCc2n[nH]cc2C1 n1(C(COC)C)nc(-c2ccccc2Br)nc1-c1ccc(Cl)cn1 C1(C(N(c2ccc(OC)cc2)c2ccc(Br)cc2)=O)CC12CCCNC2 c1(NC(N2CCCN(C(c3c(C)nn(C)c3F)=O)CC2)=O)ccc(Cl)c(Cl)c1O c1(SC)ccc(Cl)c(C(=O)NCCCC(C)NC(C2(C)CNC(=O)C2)=O)c1 C(CCCCCC(=O)N1CCC(OCCOC)C1)NC(C(CCC)NC(N)=O)=O N1(C(CN(C(=O)CC(O)CC(C)(C)C)CC(C)C)=O)CC2C3C=CC(C3)C2C1 C(C(=O)NC(C)CN(C(=O)C(C)n1cnnn1)C)(C(C)C)n1ncc(C)c1 C1(NC(CC(=O)N(C)C)=O)CN(C(c2cnn(C)c2C(F)F)=O)CC2CC12 S(=O)(=O)(c1ccc(C#N)cc1Cl)N.c1(CC(=O)Cc2ncc(C)[nH]2)ccccc1N c1(OC)ccc(C(N2CC3CC3(CNCc3ccc(OC)cc3)C2)=O)c(Cl)n1 CC(C)C(CNC(c1nc(C(C)(F)F)cs1)=O)NC(=O)CCc1cccs1 c1(OC)cc(C(=O)NCC2(O)CC2)c(NCc2cc(C#N)ccn2)cn1 c1(C(N2CC(F)(C(=O)Nc3nccc(C(N)=O)c3)C2)=O)ccc2c(c1)CNC2=O N1(C(C(C)=CC)=O)CCCN(C(=O)C(CC)C(C)(F)F)C(c2ccccc2)C1 C1(C(C)C)CC(NC(c2cnc(-c3cn(CC=O)nn3)o2)=O)CCS1.C1CC1 N1(C(C2CCCC(C)C2)=O)CC2(C1)CN(C(c1cccc(-c3ccco3)n1)=O)C2 N1(C(CC)=O)CCN(C(c2cc(C(=O)OC)no2)=O)C(CCO)C1 C1(C(N(CCN(C)Cc2onc(CC)n2)C(C)C)=O)CCC2(CCC2)O1 N1(C(c2c(C)non2)=O)CCC(C)(C)C(C(N2CCC(C)C2)=O)C1 Cc1nc(NC(c2cn(C)nn2)C)cc(N2CCN(Cc3cn[nH]c3)CC2)n1 CC1=C(C(=O)NC(C)CCNC(=O)C(O)CC(N)=O)Cn2nnnc2N1C c1(C(=O)NC2CC(C)(NC(c3cnc(CCC)s3)=O)C2)cncc(C)n1 N1(C(C(C=C)OC)=O)CCN(C(=O)Cn2nnc(C)n2)C(c2ncc[nH]2)C1 N1(C(C(CCSC)O)=O)CCC(NC(=O)C2=C(Cl)CCC2)C(O)C1 CCC(C)C(C(=O)N1CC2CC1C2C(=O)OC)NC(c1cc(F)cnc1O)=O c1(C(N2CC(CNC(C=CCC)=O)C(O)C2)=O)cc2cnccc2[nH]1 C1(C#CC(=O)NC(C)CCCNC(c2cnc(C3CCC3)nc2O)=O)(CC)CC1 CN1C2CCC1CC(C(=O)NCC1(F)CCCN(C(C3CC4(C3)OCCO4)=O)C1)C2 N1(C(C2C(=O)NCC2)=O)CCN(C(c2cnnc(O)c2)=O)CC1 c1(CC)cc(C(=O)N(CC(C)C(=O)NCCC2CCSC2)C)nn1C O=C(NNc1cccc(C2CCC2)n1)c1cc(I)c(C(F)(F)F)cn1 CC1(C)CN(C(=O)CC2CCOC(C)(C)C2)C(CNC(=O)C2=COCC2)CO1 c1(-c2c(C(=O)NCC(CC=C)O)cccn2)nn(-c2ccc(Cl)cc2)c(=S)n1C Cc1sccc1CN(C)CC1CCCN1C(c1ccccc1)C c1(CN(CC(=O)NCC2(NC(c3cc(Br)co3)=O)COC2)C)ccccc1 CC1CN(C(c2ccncn2)=O)CC1NC(c1nn(C(C)(C)C)cc1Br)=O C1(C(N(CC(=O)N(CC(F)F)C)CC#C)=O)CCCC1C C1(C(N2CC3C(NC(CCCc4[nH]c(=N)sc4)=O)C3C2)=O)CCn2cnnc2C1 c1(OC)ccc(F)c(C(=O)N(CCCNC(C2CCC3CC23)=O)CCO)c1 C(=O)(CCC(=O)c1cccc(N)c1)N(C)Cc1onc(CC)n1 Cc1c(F)cc(C(=O)NNC(=O)Cc2n[nH]c(=N)o2)cc1F c1(CCC)nccn1CC(=O)NC1CCOC1c1cnn(C)c1 C1(CNC(c2c(C(C)C)ccs2)=O)CCN(C(C2Cc3nncn3C2)=O)C1(C)C C1(F)(CNC(C2(C)CCC2)=O)CCN(C(=O)C(c2ccc(Cl)cn2)(F)F)C1 c1(NC(C2CCC3(CN(C(=O)CC(F)(F)F)C3)O2)=O)cc(Br)ccc1[N+](=O)[O-] c1(OC)ccccc1CN(C(=O)C(=O)C(C)C)C1CC1.c12nc(cn1C)NC2=O NC1CC2CN(S(=O)(=O)Cc3cccc(Cl)c3)CCN2C1=O CC(C)(C)C(C(=O)NC1C2CCC1N(C(c1cccnc1O)=O)C2)C1CCC1 c1(-c2n(CCC=C)c(N3CC(C)SC(C)C3)nn2)cnc2[nH]ncc2c1 C1(NC(c2cnn(C)n2)=O)CCN(C(=O)CCC2CCCO2)C12CCC2 N1(C(C23CC2CN(Cc2c(F)ccc(O)c2F)C3)=O)CCC(O)C(F)(F)C1 N1(Cc2c(CC)cccc2)CCC(NC(c2ccc(Br)nc2)=O)C(C)(C)C1 C1(C(=O)NCc2oc(C(=O)NCCOCC(=O)OC)c(C)n2)CCC(O)CN1C c1(C(=O)NCCCCC(C)NC(=O)C(C)(Cl)Cl)cc2ncccc2cc1Cl C12(C(=O)NCC3(CNC(CC4CC(C)(C)OCC4)=O)CC3)CCC(C1)C(C)(C)O2 N#CC1CN(C(C2(CNC(c3ccc(CC#N)cc3)=O)CC2)=O)CCO1 C1(CC)CN(C(=O)C(CN=[N+]=[N-])NC(c2ccoc2)=O)CCCO1 CCCC(CCC)C(=O)NCCNC(c1ccc(Br)nc1OC)=O C1(CC(=O)NC2C(OC)CN(C(C3(O)CCCCC3)=O)C2)OCCCC1(C)C N1(C(c2c(C)con2)=O)CC2CCC(C1)N2C(c1ccn2c1CCCC2)=O n1(CCC)cc(NC(C2CC(n3cc(C4(COC)CC4)nn3)C2)=O)cn1 C=CCC(C(=O)N(C(C(=O)NC(c1nccs1)C)C1CC1)C)C(C)C CC1C2CN(C(=NCc3cc(C(F)(F)F)ccc3F)NC3CCC3)CC12 N1(C(CCC(=C)C)=O)CC(C)CN(C(=O)CN(C)C(c2ccccc2)=O)CC1C N1(C(c2nccc(C)c2)=O)CCN(C(=O)CN2CCCC2=O)CC(C)(F)C1 c1(NCC(C2CCN(C(CC(CC)OC)=O)CC2)C)cc(C)nc(C(C)(C)C)n1 N1(C(C=CCOC)=O)CC(NC(c2ccccc2C)=O)C(c2cncn2C)C1 CC1CCC(NC(=O)Cn2cccnc2=O)CN1C(=O)CCC(=O)c1cccs1 c1(C(N(CC(CO)(CO)NC(c2c(CC)noc2)=O)C)=O)ccc(Cl)nc1N c1(SC2CC2)cc(C(N2CCC(NC(CCC3CCN(C)C3)=O)C2)=O)ccn1 C(=O)(CC(C)(F)F)N(C1CCN(C(C2COCCN2C)=O)CC1)CC c1(N2CCC(OCCNC(c3n(C(CC)C)ncc3)=O)C2)ccc(C#N)nn1 N=C1NC(=O)C(CC(=O)NC2CCCCC2NC(=O)COc2ccncc2)S1 C=Cc1ccc(C(C)NCc2ccc(OCC(F)(F)F)cc2)cc1 C1(OCC)CN(C(C2CC(=O)C2C(C)(C)C)=O)CC1CNC(=O)CSCCOC c1(C(N(CCN(C(=O)CC=C(Cl)Cl)C)C)=O)cccc(S(C)=O)c1 C(CCOCCO)(C(=O)N(C)Cc1cncnc1)NC(C(C1CCC(=O)N1)C)=O N1(C(CC2N(C(C(COC)(C)O)=O)C3CCC2C3)=O)CCC(C2CCOC2)C1 Cc1cc(C)c2c(C)c(C(=O)NCC3CCC3NC(C3CCCOC3)=O)sc2n1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(CCCNC(C(C(C)C)F)=O)CC1 N1(C(C(C)OC)=O)CC(NC(=O)Cc2cnn(C(C)(C)C)c2)CC1COC n1(C(C(=O)NCCNC(CN(CC)CC)=O)C)cc2ccccc2n1 C1(C)(CNC(C2(C)CCC2)=O)COCCN(C(=O)CNS(=O)(=O)C2CC2)C1 c1(C(C)=O)ccc2c(c1)OC2C(=O)N(C)CCN1CCN(C(C)C)CC1 C(c1ccsc1)=CC(=O)NC(CC1CC1)C(=O)NCc1ncsn1 C(=O)(CS(=O)(=O)N(C)C)NC(CC)CN(C)C(c1ocnc1C(F)(F)F)=O C1(CNC(Cn2cc(C(C)=O)nn2)=O)(OC)CCN(C(=O)C(C)(C)CN(C)C)C1 C1(NC(c2c(C)nc(C)s2)=O)CCN(C(c2cccc(N(C)C)n2)=O)C12CC2 Cc1ncc(C(=O)NCC2CCN(C(c3cc(Cl)sc3Cl)=O)CC2C)cc1N C1(NC(=O)CNC(=O)CC2CCCC2)CCCN(C(C23CC4CC2C3C4)=O)CC1 Cc1c(C(=O)NCC(O)CCNC(=O)C2=C(Cl)CC2)c[nH]c2nccc1-2 N1(C(CC(C=C)(C)C)=O)CCCN(C(c2cccc(OC)c2C)=O)CC1C C1(CC)(NC(c2ccc(C3CCOC3)cc2)=O)CCCN(C(=O)CCC2CC2)C1 c1(C(N2CCC(CCNC(CCC(C)SC)=O)C2)=O)cc(N)c(F)c(F)c1F C=CCC(CO)NC(c1occc1CNC(=O)C(n1nccc1C)C)=O C1(NC(c2cc(CC(=O)OC)on2)=O)CCCC12CN(C(C1CCCCC1)=O)C2 Cn1ncc2cc(C(=O)NCC3CCCC3NC(=O)Cc3ccsc3)cnc12 CCCC(CC)CCC(=O)NC(C(=O)NCC(C(C)C)C(C)C)c1cccs1 c1(C(N2CCC=C(C(=O)NC(C)CO)C2)=O)ccnc2c(O)cccc12 Cc1[nH]nc(C(=O)NCc2cccc(NC(C3CCC=CCC3)=O)c2)c1C N1(C(c2ccc3c(c2)OCC3)C(=O)NC)CCN(C(=O)C(C)C)CC1C#N C1(C(N2CCCN(C(C3C(C(=O)O)OCC3)=O)CCC2)=O)CC12CCC(F)(F)CC2 C(=O)(C(CNC(c1coc(C(F)F)c1)=O)CC(C)C)NC1(CSC)CC1 Cc1cn2cc(N(C3CCNCC34CC4)CCO)ccc2n1.C(=O)(CCC(C)C)NCN c1(CNC(C2N(C(CSCC)=O)CC=C2)=O)ccnc(O)c1 c1(C(N2C(CCNC(c3n(C)nnc3)=O)CSCC2)=O)cccc2[nH]ccc12 C1(CNC(C2N(CC(=O)N(C)C)CCCC2)=O)C(F)(F)C12CCC2 c1(C(=O)NCCC(C)N(C(c2ncn(CC)n2)=O)C)nc(C)ccc1O N12CCN(C(C)C1=O)C2=O.C1(NC(=O)OC)CCN(Cc2ccccc2)CC1C N1(C(COCCCCC)=O)CCCC(C(=O)NCCNC(=O)C(CC)C2CC2)C1 c1(Sc2c(C(=O)NCC(C)NC(=O)OC(C)(C)C)cccc2)ccc(Cl)c(Cl)c1 Cn1cnc2c1C(C(=O)NC1CC3C1CCN3C(=O)Cn1ccnn1)CC(=O)N2 C1(NC(CC(c2cccc(OC)c2)C)=O)CC2CN(C(=O)CCOC3CC3)CC12 c1(C)ccccc1.N1(C(C2(CC3(C)CC3)CC2)=O)CC(NC(=O)C=NO)C(O)C1 CCC(CC(=O)NCC(Cc1ccccc1)NC(=O)C=C(C)C(C)C)OC CC(C)C(CC(=O)NCC(C)C1CC1)NC(c1cnn(C2CC2)c1)=O c1(C(N(CC(CNC(C(C(C)OC)O)=O)(C)C)C)=O)nc(C)ccc1O c1(CC)cc(C(=O)NC2CC23CC(NC(=O)CCCC2CC2)C3)cn(C)c1=O C1(NC(C)=O)CCC(C(N2CC(NC(c3nnc(C(C)(C)C)s3)=O)C(C)C2)=O)CC1 CC(C)CCC(F)C(=O)N1CCC(CF)(NC(=O)CC(C)n2ccnc2)C1 N1(C(C(=O)NC2CCN(c3cc(C)nn3C)C2)=O)CCC(C#N)CC12CC2 C1(NC(C2CCCC(OC)C2)=O)CC(F)CN(C(=O)C(C)(CO)NC(C)=O)C1 c1(OC)cccc(NC(=O)NC2CCN(C(c3ccnc(F)c3)=O)C2)c1 N1(C(c2cc(COC)[nH]n2)=O)CCC(N2CCCNC2=O)CC1 CC1CN(C(=O)CSCC(N)=O)CC2(CCN(C(=O)CCc3nccs3)C2)O1 N1(C(c2cnc(NC(C)=O)o2)=O)CC(C2CCN(C(=O)C(C#N)C(C)C)CC2)C1 C1(C(N2CC3(C2)C(=O)OC3)=O)CC(C)CN1C(C1CCC(CC)CC1)=O.CC c1(OC)cc(Cl)ccc1C(N1CCN(C(C2(F)CC2)=O)CC1CS(C)(=O)=O)=O C12(NC(C(C)c3ccsc3)=O)CC(CNC(=O)CCNc3ccccn3)(C1)C2 N1(S(=O)(=O)CCc2cc(Cl)cc(Cl)c2)CCNc2ccc(F)cc2C1 C1(C)(CC)C=C(C(=O)N2CC=CC2(C)C(=O)NCC(C)(C)CC(C)C)C1 C1(CNC(CSCCC(C)C)=O)CCCCN(C(=O)CC2(O)CCOC2)C1 CCCCC(CC)CC(=O)N1CCCC(CC(=O)N(C2CCCC(C)(C)C2)C)C1 c1(CC)cc(C(=O)NC(c2cccc(C)c2)CNC(=O)CC(O)CN(C)C)c(C)o1 C1(C(N2C(C)CC(NC(C3CCCCN3C)=O)CC2)=O)CCc2ncccc2C1 c1(C(=O)OC)cc(C(=O)NC(C)CNC(c2cccc(-c3ncc[nH]3)c2)=O)ccn1 C(CCCCC(=O)N(C1CCCN(C)C1)C)N(C(c1cnc(C)o1)=O)C C1(C(=O)NC(C2CCCN2C(c2ccnc(O)c2)=O)(C)C)CC2CCC1CC2 C12(NC(N(C)Cc3c(C)noc3C)=O)CC3CC(C1)CC(F)(C3)C2 N1(C(=O)C(c2cccc(F)c2Cl)(F)F)CC2(C1)CN(C(C13CCC1C3)=O)CCO2 N1(C(C2C(C)C2)=O)CCC(N2CCC(NC(C3CC4CC4C3)=O)C2)CC1 C1(CNC(=O)Cn2nnc(=O)[nH]2)CCCCCN1C(C1CCS(=O)(=O)CC1)=O c1(C(N2CCC(C(=O)Nc3ccc(C)nc3Br)CC2)=O)cc(F)c(CO)cc1F C(=O)(C(CC(F)F)NC(=O)CCN(CC)CC)NC(CCCC)C C1(CNC(C(C)C(F)(F)F)=O)CN(C(=O)C=CC=C(Cl)Cl)CC(C)(C)C1 c1(NC(=O)C=CCCC=CC(=O)NCCC(=C)C[SH]=C(C)C)cc(C)cc(Cl)c1 N1(C(CC2(C)CC2)=O)CCN(C(C2COC3(CCC3)CO2)=O)C2CCCCC12 N1(C(CCC)=O)CCC2(CC2)CC1C(N1CCCOCC1C)=O C1(C(=O)NCc2ccc(CNC(c3cn(CC)nn3)=O)cc2)CCC2CC1CO2 N1(C(C2CC(OC)C2)=O)CCC2CCC(NC(=O)C(F)C(C)(F)F)C1C2 c1(CC(=O)N(C(C)C(=O)NC(C)Cc2ccccn2)CC#C)ccccc1C#C c1(C(=O)NC2C(C)CN(C(C3CCC(C)C3)=O)C2)cc2c(s1)CCOC2 c1(C(N2CCN(C(C=C(C)Cl)=O)C(C)C2C)=O)nc2cc(O)ccc2[nH]1 n1(CCC)ncc(C(=O)NCC2(F)CC(NC(=O)CCC3CCC(C)O3)C2)c1C N1(C(c2cnc(C)o2)=O)CC23CCCC2(C1)CN(C(=O)CC(C)C(F)(F)F)C3 n1(CCOCC)ccc(=NC(=O)C2CCC(CC)O2)[nH]1.c12coc(n1)CCNC2=O C1(C(=O)N(C(C)CC(N)=O)C)(CC)CCN(C(c2ccoc2C)=O)C1 C#CCCCC(=O)NCC1CC(COC)CN1C(=O)CC1CNC(=O)C1 c1(C(=O)NCCC(C)NC(C2(C#N)CCCOC2)=O)cc2cc(Cl)ccn2n1 C1(N(C(CCC)=O)C)CCCN(C(c2ccc(C(C)(F)F)nc2O)=O)CC1 C(=O)(C(C)CS(C)(=O)=O)NCC(CNC(C(C1C(C)C1)NC(=O)C1CC1)=O)(C)C N1(C(C(CC)CC)=O)CC(NC(c2cnc(C3CCC3)o2)=O)CC(O)C1 C(=O)(CC(O)(CCC)CCC)NC1C(CNC(C(CCC=C)(F)F)=O)CC1 C1(CN(C)C(c2cncn2C)=O)CCCCN1C(c1ccnn1CC(F)(F)F)=O c1(NCCC(N2CC(NC(CC3N(CC)CCC3)=O)C2)=O)oc(C)nc1C#N c1(C(N2CCC(C)(NC(C3N(CCC)CCC3)=O)C2)=O)cnn2c1CCC2 c1(C(=O)NC(CC)CNC(C2CCCCC(=O)N2)=O)cc(C)ccc1S(N)(=O)=O N1(C(C2CC(C)OCC2)=O)CC2(C1)CN(C(c1coc(C3CC3)n1)=O)CC2CO C1(N(C(=O)CSc2nncn2C2CC2)C)CCN(C(c2coc(Cl)n2)=O)C1 N1(C(C(N2CCNC2=O)C)=O)CC2CCCC2(NC(=O)COCC2(F)CC2)C1 C1(C(=O)NCCOC(CNC(c2c(C)onc2)=O)(C)C)NC(=O)CC1C c1(C(=O)NCCOC2CN(C(C3(C)C(C)C3)=O)C2)ccnn1C1CCCC1 N1(C(CCC=CC(C)C)=O)CCC(C)C(NC(c2ncsc2C(C)C)=O)C1 CCC(C(=O)NCC1CC(F)(CNC(=O)CC2(OC)CCCC2)C1)C(C)C C(C(=O)NC1C2CCN(C(=O)CSc3ccc(Cl)cc3)C12)(C(C)C)OC n1(CC(=O)NCCCNC(COCCOCCOCC#C)=O)ccccc1=O C(=O)(CCCC(O)c1ccccc1)NC(C1CCN(C(C2(N(C)C)CC2)=O)C1)C N1(C(c2ncncc2Cl)=O)CC2CCCC2(C(=O)NCCCCCC2CC2)C1 c1(OCC)cccc(Cc2cc(C(=O)OC)no2)c1.C123COC(C1)(C2)C(=O)NC3 c1(C(N2C(C)C(c3ccccc3)CC2)C(=O)NCC2CC2)cc2scc(Cl)c2[nH]1 c1(C(=O)NCC(CNC(c2ccc(CC)s2)=O)(C)O)c[nH]nc1S(N)(=O)=O N1(C(C(CC#C)O)=O)CC23CCCC2(C1)CN(C(c1ccnn1CCCC)=O)C3 CC1CCN(C(=O)CC2CCOCC2)C1CNC(C12CC(C1)C2)=O c1(OCC)cc(C(N2CC3CC2CC3NC(=O)C=Cc2ncc[nH]2)=O)ccc1C CCC1=NOC(CC(=O)N(CC(CC)NC(c2cc(COC)cs2)=O)C)C1 C(=O)(C1=C(C#N)CCC1)N1CCC(C#C)(C(=O)NCc2cc(C)cc(C)c2)C1 CC(CCC(=O)N1CCC(NC(=O)CNC(=O)CC(F)(F)F)CC1)N(C)C c1(C(=O)NCC2(F)CN(C(c3c(C)ncs3)=O)C2)cc2cc(Br)ccc2o1 C1(NC(=O)CN2C(=O)CCC2=O)CC2CN(C(c3cccs3)=O)CC12 C1(C(=O)NCc2cn(C3CN(C(C4CC4N(C)C)=O)C3)nn2)(OC)CCCC1 Cn1cnnc1CNC(C1CC(NC(C2CC2C(F)(F)F)=O)C1)=O c1(CC(=O)NC2CCC2NC(C2CC(C(F)(F)F)C2)=O)c(Cl)cccc1Cl C1(NC(c2c(CC)nn[nH]2)=O)COC2CN(C(=O)C(C)COC)CC12 N1(C(=O)COC2CC(C(=O)Nc3ccccc3F)C2)CCC(F)(F)CC1 CC1(C)OCCC1C(N1CCCCC1CC(=O)N(C1CC1)CC1CCC1)=O n1(CCC)ccc(C(N2CC(C(C(=O)NC(COC)CC)OC)C2)=O)n1 c1(SC)sccc1C(=O)NC1CC(CNC(=O)CCOC2CCOC2)C1 c1(C(N2CC(NC(c3ccc(F)cc3)=O)C3C2C3)=O)cc2cccc(F)c2o1 c1(C(=O)OC)cc(Br)c(C(=O)NCC2OC3(C)CC2(CO)C3)cc1N C12(NC(C(c3cccc(Cl)c3)C)=O)CC1CN(C(=O)C=Cc1ccn(C)c1)C2 C1(C(=O)N(CCCNC(=O)C#CC2(C)CC2)C)(OC)CCCC(C)(C)C1 N1(C(CC(=O)N(C)C)=O)CCCCC(CNC(=O)CCc2cnn[nH]2)C1 C1(C(C2CC(F)(F)C2)C(=O)OC)CN(C(=O)Nc2cncc(O)c2)CCO1 c1(N(CC(CCCC)CC)C)ccc(S(=O)(=O)NCC2(C)CCN(C)C2)cc1Br CC1CC(N(C)C)CN1C(=O)CC1CC(NC(=O)OC(C)(C)C)C1 c1(CC(N2CC(C)CC2(C)C)=O)cccc(F)c1[N+](=O)[O-] C(=O)(C1CCCc2nn[nH]c21)NCC(CNC(C1=NOC(C)C1C)=O)(C)C CC(C)CCC(=O)C(=O)NC(C)(CN(C)C)C(N1CCC([N+](=O)[O-])CC1)=O N1(C(c2c(C#N)ccs2)=O)CCC(C2CCN(C(C3(n4nccn4)CC3)=O)C2)C1 N1(C(CNC(C2C(C)C2)=O)=O)CSCC1C(=O)NCC1COC(=O)O1 C=CCC(C)(C)C(=O)N1CCC(C)(NC(=O)C(Br)=C(C)C)C1 C1(c2cc(-c3c(C)n(C)nc3)[nH]n2)CC2CCC(C1)N2C(C(=O)NC1CC1)C1CC1 C=CC(CC)CC(=O)NCC(=C)CCNC(=O)CCc1cccc(C#N)c1 N1(C(C(c2cccnc2)NC(C2C(C(=O)OC)C=C2)=O)=O)CCC(O)C12CCCC2 C1(NC(N2C(c3ccc(N)cc3)CCC2)=O)CCc2ccccc2C1O C(=O)(CC(C)(C)C#N)N(CCOCCC(=O)NC(c1ncc[nH]1)CC)C c1(NC(c2ccns2)C)ccc(S(=O)(=O)NC2CC(F)C2)cc1C#N c1(CC(=O)N(C2CCN(C(=O)C=CC3CCOC3)C2)C)cccc2nonc12 N1(C(C2OCC(C)(C)OC2)=O)CC2(CCCC2NC(=O)CC2=NNC(=O)C2)C1 C=C=C(C)CC(=O)NCC1CCCC1NC(c1cccc(C(C)=O)c1)=O C1(CC)C(NC(c2ccsc2Sc2ccccc2)=O)CCN1C(=O)C(C)CSC CCCC(CCNC(C1CCOC(CNC(c2cnc(S)nc2)=O)C1)=O)C1CC1 c1(OC)ccccc1S(=O)(=O)N1CCN(CC2(C)CCOC2)CC1 c1(C(N(CCCN(C(=O)CN=S(C)(C)=O)C)C)=O)ccc(C(F)(F)F)c(O)c1 CN1CCC(C2CCN(C(=O)CSc3ccc(N4CCC(O)C4)cc3)CC2)C1 c1(OC)cc(CN2CC(C)CC2C(=O)Nc2ccc(Br)cc2C)cc2c1OCO2 C1(NC(c2nnnn2CC2CCOC2)(COCC)C)CC2(CCC2)C1 C1(CC(C)NC(CCC=C=C)=O)CC2CCC(C1)N2C(c1cnsn1)=O CC1C(NC(C2CCC(F)(F)C2)=O)CCN1C(c1cc(=O)n(C)o1)=O c1(C(N(CC(CN(C(C=CC(=O)OCCCC)=O)C)O)C)=O)nccc(N)c1Cl N1(C(C(C)(C)SC)=O)CC2CC2(NC(=O)CC2CCCOCC2)C1 C#CCCCCCC(=O)N1CC(NC(c2cc(C)c(Cl)c(N)c2)=O)CC(C)(C)C1 c1(C(=O)NC2CC3(CN(C(C(CC)O)=O)C3)C2)cc([N+](=O)[O-])cc(C)n1 C1(N(C)C)(CC)CCN(C(C2C=CC(NC(=O)Cc3ncn(C)c3C)C2)=O)C1 N1(C(C(C)OCCOC)=O)CC2(CCN(C(=O)CCCc3ccncc3)CC2)C1 C1(NC(C2C(C(C)(F)F)C2)=O)CC2COCC(C1)C2NC(C1CS(=O)(=O)C1)=O N1(C(C(CCCC)O)=O)CCCC2(CCN(c3ncc4cccnc4n3)C2)C1 N(C(=NCCCCl)NCc1cc(C(=O)OC)ccn1)C1CCC(CC)CC1 Cc1cc(C)c(C(=O)NC(C2(O)CCCCC2)C(=O)N(C2CCOC(C)C2)C)o1 c1(C(=O)NCCN(C(=O)CC2NC(=O)NC2=O)C(C)C)cn2cc[nH]c(=O)c2n1 C1(S(C)(=O)=O)(C(=O)NC2C(C)CCN(C(C34C(C)OC(C)(C3)C4)=O)C2)CCCC1 N1(C(C(C)SCCCC)=O)CCC(NC(c2cn(C)nc2O)=O)CC1 N1(C(c2ncn(CC)n2)=O)CCC(C)(C)C(C(=O)NC2CCC2(C)C)C1 c1(C(c2n(CC(=C)C)nnn2)NCc2ccn(C3CC3(F)F)n2)nc(C)sc1C N1(C(c2c(CCC)n[nH]c2)=O)C2CCC1C(C(=O)NCCCC(C)(C)C)C2 C(CO)(CO)(CO)NC(C1C(CNC(Cc2cc(C)on2)=O)C1(C)C)=O C1(CNC(CCCC#N)=O)(NC(=O)COCCOCCO)CC2CCCC2C1 c1(C(C(=O)N(CC(F)(F)F)CC(=O)OCC)O)cnn(C)c1O C1(c2c(OC)cncc2C)NC(=S)N(Cc2cccs2)C2=C1C(=O)NC(C)C2 C(=O)(C(CC(C)C)C(C)C)NCC1CCN(C(CC2CC(=C)C2)=O)C12CCC2 c1(C(N2C(CNC(CC(=O)NCC#C)=O)CCC2)=O)cccc(F)c1O CC1CN(Cc2cn(-c3c(F)cc(Br)cc3Cl)nn2)CC(C)(C)C1 c1(CC(=O)NC(CCOC)C(N2CCN(C)CC(O)C2)=O)csc2nc(C)cn12 C1(CC(=O)NCCN2CCC(NC(c3[nH]c(=N)sc3)=O)CC2)CCCCC1(F)F C1(N(CCC)CC)CCCN(C(c2cc(C)n(CC)n2)=O)CC1 N1(C(=O)COC2CC(CF)C2)CCCC1C1CCCN1C(=O)C(O)CC1CC1 C(=O)(CCC(C)(C)C)NC(C(C)C)C(C)NC(=O)C=C1CCCCC1 C(CO)(C(=O)NC(C(F)(F)F)c1cnn(C)c1)NC(C)=O.C1CC(=O)N1 C1(C(N2CCC(Nc3cc(C)no3)CC2)C(=O)NC)C2CCCCCC12 C(CC(C(=O)NC1CCCC1C(C)O)NC(=O)C(CO)OC)SC C12(C(=O)NC3CN(C(=O)CCOC4CCCCC4)C3)CCCC(CCC1)C2 c1(C(N2CC(OCCNC(C3(SC)CC3)=O)C2)=O)ccc(C(N)=O)nc1 N1(C(C2COCC(C)O2)=O)C2CCC(C2)C1c1ccccc1 C1(CNC(C(CC2CCCC2)NC(C(C)c2cncs2)=O)=O)CCC2CC1CO2 c1(C(C2CCC2)NC(CNC(CC(COC)C)=O)=O)c(C)cccc1Br C(=O)(C(O)CCC(C)C)N(CC)CC1CCCN1C(=O)CCc1cncnc1O C1(C2(O)CN(C(c3ccnnc3)=O)C2)(CNC(C2CCN(CC)C2)=O)CC1 Cn1cc(C(N2CCOCC(NC(=O)C(C)(C)N3CCCCC3)C2)=O)ncc1=O S(=O)(=O)(c1cnc(N(C(CF)CF)C)c(Cl)c1)NCCN1CCN(C(C)=O)CC1 C(CCCC(C)NC(=O)CNc1ccccn1)NC(C1(COCC)CCCC1)=O c1(C(N2CC(CNC(C(C)=CC)=O)C(O)C2)=O)nccc(Br)c1C Cn1cc(S(=O)(=O)NCC2CCN(CCCF)C2)cn1 CC1(C(=O)NCC2C=CC(NC(c3ccnn3CC#N)=O)C2)CC2CCC1O2 c1(NC(C2N(C(c3n(C(C)C)ncc3)=O)CCC2)=O)ccc(Cl)cc1[N+](=O)[O-] c1(N2CCN(C)CC2CO)ccc(S(=O)(=O)NC2CC3(C2)CC(F)(F)C3)c(Cl)c1 CCCCCS(=O)(=O)CC(=O)NCCCNC(c1nnc(S)n1C)=O C1(N(C(C2(C(N(C(C)C)C)=O)CC2)=O)C)CN(C(=O)C#CC2(C)CC2)CC1(C)C C1(C(N(C)CCNC(=O)CCC2CCOCC2)=O)CCC2(C1)CC2(F)F N1(C(COC2(C)CCCC2)=O)CCCC(NC(c2coc(C#N)c2)=O)C1 N(C1CN(C(=O)COCCCF)Cc2ccccc21)C(=O)CCC(F)F C1(CC(=O)NC(c2ccsc2)C)CC(C)(C)CN1C(c1cncc2[nH]ccc12)=O C#CCCCCNC(=O)C(c1ccco1)NC(=O)C(C)C=C c1(C(C(=O)NCC2CC2)N(CC#CC)CC#C)nc(C(F)(F)F)n2c1CCCC2 c1(C(N2CCC(C3CC3)C2CNC(C2(O)CCOC2)=O)=O)nccc2occc12 C1(CNC(c2scnc2C(F)(F)F)=O)CN(C(=O)CC2CCCO2)CC1C(F)F C1(C(=O)NC2C(NC(CCCC(OC)OC)=O)C2)CNC(=O)C(C)(C)C1 c1(C(C(=O)NCc2ncc(C(F)(F)F)cn2)F)ccc(F)cc1Cl C(=O)(CC(C)C(C)(C)C)NCC1(F)CC(NC(c2nc(C(=O)OC)sc2)=O)C1 C1(C(N2CCC(NC(=O)C=C(Cl)Cl)C23CC3)=O)CC2(CCCCC2)S1(=O)=O N1(C(C2CN(CCOC)C(=O)C2)=O)CCC2(C1)CN(C(=O)CC1C(C)C1(F)F)C2 C1(NC(c2n(CC)ccn2)=O)CCC2(CCCN(C(c3cccnn3)=O)C2)C1 C(C(C)(O)CC(=O)N1CC(NC(c2c[nH]ccc2=O)=O)CCC1C)OC C1(NC(c2cn(C3CCOCC3)nn2)C)CCC(O)C(C)(C)C1 C12(C(N3CC4C(N(C)C(C5CC56CCCC6)=O)C4C3)=O)CCC(N=[N+]=[N-])C1C2 C1(C(N(CCCF)CC)=O)CCCC(NC(=O)C(F)C2CCCC2)CC1 CCCC1c2ccccc2CCN1C(c1ccc(OC)nn1)CN(C)C C1(NC(C(c2ccc(F)cc2F)C)=O)CCCC2CN(C(C3C=C3C)=O)CC12 c1(C(=O)OC2CC(NC(c3cncc(Cl)c3)=O)(CF)C2)cc2c(s1)CCC2 c1(CN(C(C2C(C)C2)=O)C)cnn2c1CN(C(C13CCC(=O)N1CCS3)=O)CC2 c1(N2CCC(CCC)(CO)C2)nc(=NCCCC(F)F)[nH]c2cc(OC)ccc12 C(=O)(CC(O)(C(F)(F)F)c1ncc[nH]1)NCCCCCCNC(C(CCCC)O)=O c1(C(=O)OC)ccc(N2CCN(C(=O)CCC(F)Br)CC2)c(F)c1 CC1CCC(NC(=O)C(C)(C)c2ccsc2)CN1C(=O)C=CCN1CCOCC1 C(=O)(CC(C)(C)C(F)F)N1C(CN(C)C(c2cnc(F)c(F)c2)=O)COCC1 C1(NC(C(C2CCOCC2)C)=O)CC2(C(N3CC4CC3CN4C)=O)COC1C2 N1(C(CN2C(C)CCC2)=O)CCN(C2CN(C(C34CCC(C3)C4)=O)C2)CC1 Cc1nncn1NC(=O)C12CCC1CN(C(c1cc3ccccc3[nH]1)=O)C2 C1(NC(C(n2cc(C3CCCC(O)C3)nn2)C)=O)COC2(CCCC2)O1 CCC(O)(C(=O)NC(CNC(c1ccccc1)=O)CO)c1ccccc1 Cc1nnc(O)c(C(N2CC(CC(C)NC(C3CC(C(F)(F)F)CO3)=O)C2)=O)c1C CC1CN(C(c2cc(CNC(c3ccoc3C3CC3)=O)on2)=O)CC(CO)O1 C1(OC)CCCCC1C(=O)NCC(C)CN(C(=O)C(C1CCC1)OC)C c1(C(=O)NC(C)C(C)(C)NC(C2CCCCN2C)=O)cccc2c1ncn2C CC1Cc2cc(C(=O)N(C)CC3CN(C(C4CCOC4)=O)CCO3)ccc2O1 c1(N2C(CNC(=O)CCC3CC3(Cl)Cl)CCC2)ccc2c(n1)CCC2=O N1(C(CC(=O)OC)=O)CCCCC1C1(NC(c2c[nH]nc2C(F)F)=O)CC1 c1(OC)ccc2c(c1)CCC(C)N2C(=O)C(=O)Nc1nn(C)c(C)c1Cl N1(C(C(C2CC2)OC)=O)CCN(CC(C)NC(c2cc[nH]c2C(C)C)=O)CC1 O(N(CC)C(=O)CCC1CCCN1C(C1(O)CCOC1(C)C)=O)CC c1(C(=O)NCCCCN(C(=O)C(O)C2CC2)C)c[nH]c2cccc(Br)c12 c1(-c2cccc(-c3nc(C)[nH]n3)c2)cc(C)cnc1F c1(OC)nccc(C(N2CCC(C(F)C(=O)N(C)CCc3cccs3)C2)=O)n1 CC1CC2(CCN(C(=O)CCC3CCN(C(C4(C)CCCN4C)=O)C3)C2)CO1 c1(C(=O)OC)cc(C(=O)NC(C)CN(C(=O)C=CCOCC(F)(F)F)C)on1 C(CCCNC(=O)COC1CCC1)NC(C1(C)CC1)=O C1(OC)CCCC1c1cn(CC(=O)NCCc2nncs2)nn1 C=CCCC(C)(C)C(=O)NCC(F)(C(=O)NCCCN1CCOCC1)C(C)C N1(C(c2cc(C(C)(C)C)on2)=O)CCC(O)(CC(=O)N(CCO)C2CC2)CC1 c1(C(=O)NC(C(C)(C)NC(C(C2CC2)SC)=O)C)ccc(O)nn1 N1(C(C2CCC(C(C)C)CC2)=O)CCOC2CN(C(=O)CNC=O)CC12 c1(C(N2CCN(CCNC(C(CCOC)OC)=O)CC2)=O)c(F)ccc(OC)c1F c1(N(C(C)=O)C)nn(C)c(Cl)c1NCC(C)(CC(C)C)NC(=O)C(F)C(C)(C)O CC(CC=Cc1ccccc1)C(=O)NCCCCCN(C)C(C12CC(C)C1C2)=O C1(C(C)C)(NCc2cc(O)ncn2)CCCN(C(=O)OC(C)(C)C)C1 C1(NC(C(C#C)(C)C)=O)CN(C(c2nc(C)oc2OCC)=O)CC1N=[N+]=[N-] C1(N(C(=O)C2=NOCC2)C2CCN(C(C)=O)C2)CC(C#N)(c2ccccc2)C1 c1(OC)ccc2[nH]cc([N+](=O)[O-])c(=NCCN(C(c3csc(S)n3)=O)C(C)C)c2c1 N1(CC(=O)C2CCC2)CCN(C(=O)NCC(c2ccccc2)N(Cl)Cl)CC1 C1(C(N2CC3CC3(NC(c3cnn[nH]3)=O)C2)=O)(COC)CC=CCC1 C1(C(N2CCCC(O)(CNC(C3CSC3)=O)C2)=O)(COC)CCCNS1(=O)=O c1(OC)cc(C=CC(N2CC3(CC3)CC2CO)=O)cc(OC)c1O c1(OC)ccc2[nH]c(C(N3CCC3CNC(=O)C=CC=C(Cl)Cl)=O)cc2n1 N1(Cc2onc(C)n2)CCN(C(=O)CSCC(=O)OC)CC1 C(=O)(CC(CN(C)C)C(F)F)N(CCCNC(c1c(CC)non1)=O)C1CC1 C(=O)(NNc1cccc(Cl)c1Br)Nc1c(C)c(N2CCCCCC2C)ncc1 Cc1nc(C(N2CCC(C(C)(C)NC(=O)C(F)CC3CCCCC3)C2)=O)cs1 C#CC1(C(=O)NC2CCCN(C(=O)Cn3cccc3)CC2)CCCCC1 c1(C(=O)NC2CCN(C(c3cn[nH]c3)=O)C2)cc(Cl)cnc1Br c1(OC)cc[nH]c(=NCCNC(=O)C(C)CN(C)C(C2CCCCO2)=O)n1 C(=O)(C(O)CC(C)C)N(CC(CC)NC(c1cnn(CCC)c1C)=O)CC c1(C(=O)NCC2C(NC(c3ccc4cnsc4c3)=O)C2)cncc2ccccc12 C1(CC)(NC(=O)CCc2cncn2C)CCN(C(C2CCC(=O)N2C)=O)CC1 C=CC(CC)CC(=O)N(C1CCC(NC(=O)Cc2n[nH]c(=N)s2)CC1)C Cc1cc(=O)n(CCC(=O)NCC(CO)NC(=O)C2=CCOC2)cn1 C1(C(=O)NCC2CCN(C(c3cncc(C)c3)=O)CC2O)CCCCC(F)(F)C1 N1(C(=O)CCF)CCC2C(CCCN2C(c2ccccc2-n2cccc2)=O)C1 C1(C(=O)NC2(CCO)CN(C(COC)=O)C2)CC12CCC2(F)F Cc1[nH]nc(C(=O)NCCC2CCCN2C(c2cccc(N)c2)=O)c1C c12ccc(cc1)NC(=O)Nc1ccnc(c1)CO2.c1(C(C)(C)C)cccnc1 c1(-n2c(C)cc(C(C)NC3CCNCC3)c2C)ccccc1[N+](=O)[O-] C12(CCNC(=O)COCc3nc[nH]n3)CCC(C1)N(C(C1CCOC1)=O)C2 C(=O)(NNC(=O)CCc1ccc(C(=O)O)cc1)NCC c1(OCC=C)ccc(CC(=O)NCCC2CC(NC(=O)CCNC(N)=O)C2)cc1 c1(C(=O)NC(C2(O)CN(C(c3ccc(C(F)F)cn3)=O)C2)C)cc[n+]([O-])cc1 Cc1cn2c(CC(=O)NCc3ccccc3OC(C)C)cnc2s1 CC(C)CCC(=O)NC1CCC(Cn2cc(CCC3CCCO3)nn2)CC1 c1(CNC(CCCC#N)=O)ccc2c(c1)CCCC2NC(C1CCCCO1)=O N1(C(C(C(C)C)NS(C)(=O)=O)=O)C2CCC1CC(NC(=O)CCc1nc(=N)[nH][nH]1)C2 C1(CNC(CC(=O)N(C)C)=O)CN(C(C2CC23CCOCC3)=O)CCC1(F)F c1(OCC)ccccc1OCC(=O)NC1CCCCC1NC(=O)CC(C)(F)F Cc1cccnc1C=CC(=O)N(C(C)CCNC(=O)CCc1nncn1C)C c1(C(=O)NCC2CC(NC(CCC(=O)OCC)=O)C2)ccc2nc(C)ccc2c1 C1(F)(C(=O)NC2CCC(C)(CNC(c3c(C)nsc3)=O)C2)CCCCCC1 C(=O)(CCC(=O)NCC(C)NC(c1sccc1CC#N)=O)Nc1nnc(C)s1 S(=O)(=O)(c1ccc(N2CCOC(CCC)C2)cc1Cl)NCCN(CCC)CCC N1(C(c2c(SC)scc2)=O)CCOC(C(C)NC(=O)CC2CC(C)(C)C2)C1 N1(C(c2c[nH]c(=N)o2)=O)CCCN(C(=O)CC2CC=CC2)CC1c1ccccc1 C1(C)CN(C(C2CN(NC(CSC)=O)CC2C)=O)CCN1CC.c1(CO)ccccc1 C(=O)(C1=Cc2ccccc2C1)N1C(CN(C(C(C)N2CCCC2)=O)C)CCCC1 C1(C)(NC(C=CC2N(C)CCC2)=O)CCCN(C(C2CCN2C)=O)C1 c1(SCCN2CCN(C(=O)CC3CC3(C)C)CC2)cncc(NC(C)=O)n1 c1(C(=O)NC2CN(C(c3c(C)n(C)nc3)=O)C(C)CC2)cccc2ccnn12 CC1CN(C(=O)CC2CCS(=O)(=O)C2)CC1NC(C1(C)CCOCC1)=O Cn1nnc(CNC(=O)CC2(C)CC2F)c1C(=O)NCC=CCO c1(NC(C2C3CN(Cc4cncc(Br)c4)CC23)=O)c(Cl)cc(Cl)cc1Br C=CCC(C)(CC)C(=O)NC1CCN(C(=O)COCc2ncc(C)o2)CC1CO C1(CNC(COC(CC)C)=O)CC(C)CN(C(=O)C(C)SCC)C1 c1(C(N2CC(NC(c3cnn(C)c3F)=O)C2)=O)cc2c(nc1O)C(C)CCC2 CCC(C#N)(CC)C(=O)NCC1(NC(=O)CC(n2nc(C)cc2C)C)CCCC1 Cc1ncc(C(=O)NC2(C(=O)NCC(c3cn(C)cn3)O)CC(O)C2)cn1 C1(CC)(NC(c2scnc2C)=O)CN(C(=O)COC2CC=CC2)C1 c1(CCCC)ccc(C(=O)NCCC(C)(C)NC(=O)C(CC)SCC)cc1 C(=O)(C(N)CCC(=O)O)N1CCC(NCc2cc(C)n(C)n2)C1 C=C(Cl)CC(C(=O)N1CC(F)(CC)C1)NC(=O)C(CC1CCC1)OC CC(C)(C)C(CO)C(=O)NC1CN(C(c2ccnn2C2CCC2)=O)CC1N=[N+]=[N-] c1(CNC(c2n(CCSC)nnn2)c2cn(C)nn2)cc(F)c(F)cc1F N1(C(C(C=C)(C)O)=O)CCC(C)(NC(=O)C(C)Oc2ccccc2)CC1 C1(NC(CC(C)OC)=O)CCN(C(c2cncn2-c2cnn(C)c2)=O)CC1CO C(=O)(C1CN(C)C(=O)c2ccccc21)OC(C(C)C)C(=O)Nc1ccc(Cl)cc1 C1(C(N2C(Cn3cc(C(N4CCCC4)C)nn3)CC2)=O)CC(=O)NC1(C)C C1(NC(CSC)=O)CN(C(c2cc3cc(F)cc(F)c3o2)=O)C2(CCCOC2)C1 N1(C(C2N(CC)CC2)=O)CC(NC(=O)CSc2cccc(Cl)c2)CC(F)C1 C1(COC)CN(C(c2c(Cl)cnn2C)=O)CCN1C(c1ccsc1)=O C1(CC(=O)NCC(NOCC)=O)N(C(C2CC23CCC3)=O)CCC1(C)C N1(C(C(C)NC(c2ccc(C(C)=O)o2)=O)=O)CC(N(C)C)CC1C N1(C(C2(F)C(C)C2)=O)CCC(CNC(c2ncccc2CO)=O)C(F)(F)C1 C(=O)(CC1NC(=O)c2ccccc21)N1CCC(NC(c2cncc(C)c2)=O)C1C C1(CNC(c2cc(C)oc2C)=O)CC(C)CN(C(C2CC(F)C2)=O)C1 C1(C(=O)NC2CC(c3ccccc3)(NC(c3n(CC)nnc3)=O)C2)CC=CCC1C N1(C(CCCOC)=O)CCN(C(c2cnc3c(ccn3C)c2)=O)C2COCC12 c1(SCc2cn(C(C)CNC(C3CC34CCOCC4)=O)nn2)ccc([N+](=O)[O-])nc1 C(CN=C(NCC(C)F)N1CCN(C(=O)N(C)C)CC1)c1ccc(C)cc1C Cc1ncc(C=CC(=O)NCCC(C)(C)CNC(c2ncn(C)c2C)=O)s1 C#CC1(C(=O)NCC(CNC(C2(C)CCCCC2)=O)CO)CCCC1 N1(C(C2(C)C(C)(C)C2)=O)CCOC(C)(CNC(c2ccnc(OC(F)F)c2)=O)C1 C1(C(CNC(C2(CC=C)CCC2)=O)(C)O)CCN(C(c2csc(CC)n2)=O)CC1 C1(CC)CCCC(NC(C2(NC(=O)CCn3ccnc3C)CSC2)=O)C1 Cc1ccc(CCCCC(=O)N(CC(C)CNC(=O)C(C(C)C)N(C)C)C)cc1 C(CCC(=O)NC(C)(C)CN(C)C(C1CCOC1C)=O)=C(C)C c1(CNC(C2CC=CCC2)CCc2n(C)nnn2)c2ccccc2nn1C c1(C(C)=O)cc([N+](=O)[O-])ccc1NC1CCCC1NC(C1CC2CC2C1)=O c1(NC(=O)NCCN2CCC(N3CCCC3)CC2)cc(-c2ccncc2)ccn1 Cc1csc2ncc(C(=O)NCCC3(O)CCN(C(C4CC4(C)C)=O)C3)c(=O)n12 C1(C(=O)NC(CCCNC(c2cnc(C)o2)=O)C)CCCN1S(=N)(=O)N(C)C c1(C(c2cc(C(N(C3CCCC3)CCC#C)=O)sc2)=O)ccc(F)cc1 C1(CNC(CCOCCOC)=O)CCCC1C(=O)NC1(C(O)CO)CC1 C(C1CN(C(c2cc(F)cc(N)c2N)=O)Cc2ccccc21)NC(COCC)=O Cc1cccnc1C(=O)NC1(C)CCN(C(=O)CC(C)n2cc(Br)cn2)C1 CC1(C)CC(C(=O)NCCc2ncc[nH]2)CN1C(C1CCSC1)=O C1(NC(C(c2cccnc2)NC(C(C=C=C)C)=O)=O)CC=C(C(C)C)CC1 C(=O)(CS(=O)(=O)CC1CCCO1)N(CC(C)SC)CCNC(C=CCC)=O C(=O)(C(CO)C(C)(C)C)N1CC(CNC(c2c(CC)ccs2)=O)C(C)C1 CC1CCC(C(=O)NCC#CCNC(c2ncoc2C2CC2)=O)S1 C1(C(=O)NCC(C)CN(C)C(c2c[nH]nc2C2CCC2)=O)CCn2cnnc2C1 Cc1cc(CNC(C2COCC2NC(C2OC3CCC2C3)=O)=O)ccc1F c1(C(=O)NC2CN(C(C(CCC)C)=O)CC2SC)ccc2nc(C(F)F)[nH]c2c1 c1(C(=O)NC2CCN(C(c3cc(C4CC4)on3)=O)CC2)cccn(CCF)c1=O c1(C(=O)OCC(C2(C(=O)OC)CC3(CCC3)C2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 C1(NC(CSCC(C)C)=O)COC2(CCN(C(=O)CC3CC4CCC3CC4)C2)C1 c1(C(=O)NC2CN(C(C(C)n3cccn3)=O)C2)cncc2nnn(C)c12 c1(C(=O)NCC2(CNC(CC=C)=O)CCC2)cc2cc(Br)cn2c(O)n1 CC1CN(C(=O)CCn2cccnc2=O)CCCN1C(c1c[nH]cc(F)c1=O)=O CC1C(NC(c2cnc(C3CC3)o2)=O)CC2CCC1N2C(=O)C1=NNC(=O)CC1 CCC(C)(C)CC(=O)NC1CC(C)(NC(c2ncc(N)cc2Cl)=O)C1 C1(N)CCCN(C(=O)C=CC(=O)N(C2CC2(C)C)C(C)=O)C1C.N(C)C Cc1cc(N2CCC(C(C)NC(c3cn(CCO)nn3)=O)C2)n2nc(C)nc2n1 c1(C2C(NC(Cn3cc(CNC(=O)OC(C)(C)C)nn3)=O)C2)cccc(C#N)c1 C(c1ccc(Br)s1)=CC(=O)N(CCCNC(=O)C(CO)OC)CC N1(C(CN(c2ccccc2)CC)=O)CCC(C(C)NC(=O)CC2(C#N)CC2)C1 Cc1ccc(NC(C2(C)CN(C(C3CC(N(C)C)C3)=O)C2)=O)cc1C#N c1(CCN2C(=O)NCC(CCN3CCOCC3)C2=O)cccc2ccccc12 c1(COCC)c(C(=O)NC2CC2CNC(=O)CC2(C)CC2(F)F)cnn1C C1(CC)CN(C(C23CC(C(C)(F)F)(C2)C3)=O)CCN1C(=O)CC1CC12CC2 c1(N(C2CCC(CO)CC2)C)cc(S(=O)(=O)N2CCCN(C)CC2)ccc1C#N c1(C(N(C)CC2CCCN(C(c3n[nH]cc3I)=O)C2)=O)ccc(F)nc1F c1(CNC(=O)NCC2CC3CCCC3C2)cccc2nccnc12 c1(CC(=O)NC2CN(C(C3(C)C(C)(C)C3)=O)CC2O)nc2ncccn2n1 c1(NC(C2CCN(C(=O)Cc3c(F)cccc3F)C2)=O)nnc2ccc(Cl)nn12 Cc1c(CC(=O)NCCOCCNC(C23CCC(CC2)C3)=O)ncn1C c1(CNC(C(C)c2ccsc2)=O)nn(C)c2c1CN(C(c1csc(O)n1)=O)CC2 CC1CCN(C(c2ccc(N(C)C)nn2)=O)CC1NC(c1cncn1C)=O C1(CNC(C(C=C)(F)F)=O)CN(C(=O)C=Cc2ccsc2)C2CCCC2O1 C(=O)(C(C)(O)CC(F)F)NC(CNC(c1ccc(COC)c(F)c1)=O)C(C)(C)C C12(CCOC1)C(=O)N2.c1(C(N2CCCC2)=O)cnn(C2CCC2)n1.C1CC(=O)N1 CCC(O)C(C)C(=O)NCCN(CCCN(C)C)C(=O)Cc1ccc(Br)cc1 c1(NC(C2N(Cc3c(C)nc[nH]3)CC(O)C2)=O)c(Br)cc(Cl)cc1C#N C(=O)(CC(C)CC(C)C)NCC1(O)CCN(C(CCC(C)OCC)=O)C1 C12(C(=O)NCCC(=C)CNC(c3ccc(CC)[nH]3)=O)CCC(CC1)C2(C)C C1(CNC(c2ccc(C)cn2)=O)CC(C(C)(C)C)CCN1C(=O)C(O)C(C)C N1(C(c2cc(C3(C)CC3)on2)C(=O)NC2CC(F)(F)C2)CC(C)C(C)C1 c1(C(C)OC)cc(C2CCOCC2)nn1C(C)C C1(CNC(C(C)=C(C)C)=O)CN(c2ncc([N+](=O)[O-])cn2)CCC12CCOCC2 C1(CNC(C(C2CCOCC2)C)=O)C2CCC(C2)N1C(=O)C(N)=O c1(C(=O)NC2(CC=C)CCN(C(C3CCCN3C=O)=O)C2)ccc(F)c(OC)c1 c1(OC)c(C(N2CCC3CN(C(=O)C=CC(F)(F)F)CC23)=O)cc(F)cc1F C#CCCCCC(=O)NCC1CCN(C(=O)C(C)NC(=O)OC)C1 N1(C(c2c(C)c(F)cnc2)=O)CCC2CCN(C(c3cn(C)c(O)n3)=O)CC12 N1(CCC)CCCN(C(C2CCCC2CNC(=O)Cn2cnnc2)=O)CC1 C1(C(N(CC(C)NC(=O)CC=CCc2ccccc2)C)=O)(CO)CC1(F)F C12(NC(C(C)SC)=O)COC(C1)C(NC(=O)Cn1nnnc1-c1ccsc1)C2 c1(-c2ccc(C3(CNS(=O)(=O)C4CC4)CC3)c(F)c2)ccc2c(c1)NCCO2 C12(C(N3CCC(N(C)C(C4CCCC4C)=O)C3)=O)CCC(CC1=O)C2 c1(C(=O)NC2CC3CCC2N(C(C2CCCSC2)=O)C3)coc2cc(F)ccc12 c1(C(N2CCC(CNC(C3CCCCO3)=O)C(O)C2)=O)c(F)ccc(F)c1Cl C(=O)(C(C)N(OC)C(=O)CC1CCCN(C(=O)CCCOC)C1)NCC N(C(=NCC1CCCC1(F)F)NC1CCS(=O)(=O)C1)CC1(OC)CCC1 Cc1ccc(CCC(C)NC(=O)C(CCN(C)C)N(C)C)cc1 CC(Cn1ccnc1)C(=O)NCC(F)CNC(c1ccn(CC(F)F)n1)=O CC(CCOC(F)(F)F)C(=O)NC(c1cnn(C)c1)c1ccccc1 N1(C(CC(C)OC)=O)CCC(NC(=O)Cn2cnccc2=O)CC1C C1(N(C(C2C(C=C)C2)=O)C)CCCN(C(c2cc(C)c(Cl)cn2)=O)CC1 C1(C(=O)NCC2N(C(CC(C)C)=O)CCC2)COc2ccc(Cl)cc2C1 c1(C(N2CCC(CNC(C3CCC3)=O)C2)=O)c(Cl)ccnc1Cl C(CCSC)(C(=O)NCCSC)N(c1cccc(C)c1)C(COC)C C(=O)(CC(C)CCc1ccccc1)NCCC(CNC(C(C=C)(C)C)=O)O CC1C(NC(=O)C2=CC(C)(C)C2)CC2CCC1N2C(=O)CCNC(=O)CO N(C1CN(C(=O)C(N2C(=O)CCC2=O)C)CCc2ccccc21)C(C(F)=CC)=O c1(C(=O)NC(CN(C(=O)C(C)Cc2cccc(Cl)c2)CC)C)nc(C)c(C)s1 Cc1cc(Cl)ccc1OCC(=O)NCC1CN(C)CCN1C(C1CC1(C)C)=O C1(C(=O)NC(CCCC)CNC(c2cccc(C)c2)=O)CCc2nc(C)cn2C1 CC1(C)CCC(CNC(=O)CC2CC2C2CC2)CN1C(=O)CCc1cncs1 Cc1c(Br)ccc(C(=O)NC(C(C)NC(=O)CCC(C)C)C(C)C)c1N C(C(=O)N1CC(CC(C)NC(C2C=CCC2)=O)C1)(C1CC1)SC c1(C(=O)NC2(C)CN(C(CC3COCC(C)O3)=O)C2)ccc2c(c1)CCC=C2 C#Cc1ccc(F)c(C(=O)NCC2CC2NC(c2cnoc2CCC)=O)c1 C=CCCC(C(=O)NOCC(O)CO)N(C(=O)CCCC)CC C(C)(CCC(=O)N1CCC(NC(=O)Cn2nnc(-c3ccco3)n2)C1C)OC C(N=c1[nH]cnc(Cl)c1F)C1(C)CCCCN(C(=O)C2=CCSC2)C1 N1(C(C(c2cncc(F)c2)C)=O)CCC(CF)(NC(c2cc[nH]c2)=O)C1 c1(CC(=O)OCc2cccc3[nH]ccc23)ccc2cc(Br)ccc2c1 c1(C(C(=O)OC(C)(C)C)NC(N(C2C=CC(=O)N=N2)C)=O)cc(Br)ccc1F c1(CCC(=O)NCCN(C)C(C2CCO2)=O)ccc2c(c1)CCO2 C1(C(=O)NCC(C(C)C)NC(=O)CN2CCCCC2=O)CN(C)CCN1C CCC(C)C(O)C(=O)NCC(C)(CNC(=O)COCCCC(C)C)OC N1(C(C(S(CCC)(=O)=O)C)=O)CCc2sccc2C1CNC(C12CC(F)(C1)C2)=O C12(C(=O)NCC3CC(NC(C4CN(C(C)(C)C)C(=O)C4)=O)C3)CCCC(C1)OC2 c1(C(=O)NC2C(C)(C)N(c3ncnc(O)c3Br)CC2)cc2n(n1)CC(F)C2 C(=O)(C(CC)C(=O)N1CCC2C(NC(C3CCC3)=O)CC12)OCC CCCC(O)CC(=O)NCC1CCCC(CNC(=O)CNc2ccc(Cl)cn2)C1 C1(N(C(=O)CCc2ccccn2)C)CCN(C(c2cc(O)nn2C)=O)CC12CC2 C1(NC(c2ccco2)=O)CCC2CN(C(=O)CC3CC4(CC4)C3)CCC2C1 N1(C(c2c(COC)cco2)=O)CCC2CCC(C1)N2c1ncncc1Br c1(COC)sccc1C(=O)N(CCNC(C1(C)CCOC1)=O)C(C)C c1(CN=c2[nH]c(=N)nc(N3C(CC=C)CCCC3)[nH]2)ccc2c(c1)CCCC2 c1(C(N2CCC(NC(CC=C=C)=O)C(F)C2)=O)cc2c(C)c(F)ccc2[nH]1 N1(C(C(CCCC)C)=O)CCC2(CC1)CC(NC(=O)CCn1nc(C)nc1C)C2 C(=O)(CCC(C)(C)C)N(C(C(=O)NCC(CC)(C)O)C1CC1)C c1(C(N2CC3CC(NC(c4cc(Cl)on4)=O)C3C2)=O)ccc(OC(F)F)c(F)c1 N1(C(C(=O)NC(C2CN(C(=O)CCCN3CCCC3)C2)C)C)CCOCC1 C1(N(C)C(C2CCCN2C(=O)CN2CSCC2=O)=O)CCCC1(F)F C1(CC)CN(C)CCN1C(=O)Nc1ccccc1CCN1CCOCC1=O C(=O)(CC1=CCOCC1)N1CC(CCNC(c2ccc(C(C)F)cc2)=O)(OC)C1 C=CCC(C)(C)C(=O)NCCCCN(C(=O)C(F)CC)C C(CCC(=O)N1CCC(CCCO)C1)N(C)C(C1(CSC2CC2)CCC1)=O c1(CCC(=O)NCC(CNC(c2c(C(C)C)nns2)=O)F)nc2ccccc2[nH]1 C(=O)(C(C)C(O)C(C)C)NCC(CNC(c1nc(OC)c(C)s1)=O)OC C1(NC(C(C)CCOCc2ccccc2)=O)CC2CN(C(=O)CCC(F)F)CC12 C12(NC(C=CC=CC)=O)CCC(CN(C(=O)C(C)(C)c3ccn(C)n3)C1)C2 C1(C)(C(=O)NCCSCC(=O)N(C)CC2(C)CCC2)CNC(=O)C1 C1(C(=O)NC(C)CC2CN(C(c3cncc(Cl)n3)=O)C2)CCCCC1(F)F CCC(O)C(C)(C)C(=O)NCCCCC(CO)NC(=O)C=Cc1ccco1 CC1CCN(C(c2cnc(Cl)n2C)=O)CCN1C(C1CCCC1(F)F)=O C1(C)(CNC(COCCCC)=O)CCC(NC(c2cc(SCC)cnc2O)=O)CC1 CC1CC(C)CN(C(=O)CCNC(=O)CCC2CC2CN=c2[nH]nc(CO)s2)C1 Cc1nn(CC(=O)NCC(O)CN(C)C(C2C(Cl)(Cl)C23CC3)=O)c(C)c1C N1(C(C#CC(=O)N(C)C)=O)CC2CC1CC2NC(=O)C=Cc1ccncc1 c1(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)CCOC)cc2cncn2c(O)n1 N(C)(C1CCc2c(C)cccc21)C(c1cc(CC)on1)=O c1(CCNC(C(C)OC)=O)ncc([N+](=O)[O-])cc1C N1(C(C=CC(=O)OCC)=O)CCCC1CN(C)CCO.C12CC1C(=O)NC2 CN1CC(=O)N(CC(N2CCOC(CNC(C3CCCCC3O)=O)C2)=O)C1=O N1(CC)CC(C(=O)NC2CC(N(C(=O)C(=Cc3c[nH]cn3)F)C)C2)NC1=O c1(C(=O)OC)cc(C)[nH]c(=NCCCN(C)C(C2CNC(=O)N2)=O)n1 c1(C(N2CCCC(NC(=O)CC3=CCCC3)C2)=O)cc(F)cc2nc[nH]c12 Cn1ccc2cccc(C(=O)NC3CN(C(=O)CC4CC4(C)C)CCC3(C)C)c12 C1(OC)CC(CN(C2CNC(c3ccc(C)cc3)C2)C)C(OC)O1 c1(OC)ncc(Br)c(=NC(=O)c2ccc3[nH]cc(C(=O)NCCF)c3c2)[nH]1 CC1CCN(CCC(=O)NC(=S)N)C1c1ccccc1 C1(NC(C(c2n(C)ncc2)O)=O)CCCC(Nc2ccc(C(C)=O)cn2)C1 c1(C(=O)NCC(CCNC(C(C(C)C)O)=O)O)ccc2cnoc2c1 CC(C)C(Cc1ccccc1)C(=O)NCCCC1CCCN1CC(Cl)=CCl C1(OCCC)CCCN(c2nnc(C(O)C3CC3)n2CC2CCCO2)C1 C(=O)(C#CC1CCOCC1)N1C(C(=O)Nc2c(CC)nc(C)cc2)CC1C Cc1cnn(C2CN(C(=O)CCN(C(=O)C(F)OC(F)(F)F)C3CC3)C2)c1 C(CC(=O)NCCCCC1CC1C)(C1CC1)NC(CC)=O c1(CC)cc(C(N2CC(CNC(c3cscc3CC)=O)C3(CC3)C2)=O)c(C)nn1 c1(C(N2CC(NC(C(C)OC(C)(C)C)=O)C(C(F)F)C2)=O)cccc2ccsc12 C1(CNC(CCCC)=O)COC(C(F)(F)F)CN1C(=O)Cn1nnc(=O)[nH]1 N1(C(C(CC(C)C)C)=O)CCC2(CNC(C3(C(=O)N(C)C)CC3)=O)CCCC12 C#CCC(CC(F)F)C(=O)N(CCCNC(=O)Cc1cc(C)ns1)CCO c1(C(=O)OC)c(C)[nH]c(C(N2CC(O)(C(C)NC(=O)CN3CCC3C)C2)=O)c1C c1(C(=O)NC2CC3N(C(CSCCC)=O)C(CC3)C2)ccc(=O)n2c1CCC2 c1(N(C2CN(C(CCc3c(C(=O)OC)c(C)[nH]c3)=O)C2)C)ncc(Br)c(O)n1 C#CCC(CC(F)F)C(=O)N1CC(OCCNC(=O)Cc2sccc2Cl)C1 C1(CNC(C(CCSC)O)=O)CN(C(=O)COc2ccc(F)cn2)C(C)(C)C1 C1(O)(CNC(c2c(C(=O)OC)coc2)=O)CCCN(C(=O)CC(C)(C)O)C1 C1(N(C)C)CC2CC1CN2C(C1CCCCC(=O)N1)=O C1(C(=O)N(C(C)C(C)SC)C)(N(C(c2ccc(C)nc2)=O)C)CCC(C)(C)C1 C12(C(=O)NCc3c(C(=O)NCC(=O)NCCC)con3)CC(C#N)(C1)C2 c1(C(=O)NCC2(OC)CN(C(=O)CS(N)(=O)=O)C2)cc(F)c(F)c(F)c1F C(C(C(=O)N(C1CCOC1)C)NC(C1CCC1CO)=O)OCC Cc1nc(C)n(CC(=O)N(CC#CCC2C(c3nc(S)n[nH]3)C2)CCO)n1 C1(N(C(=O)C(C)n2cncn2)CC)CCCN(C(c2scnc2C(C)C)=O)CC1 CC(C)(CS(C)(=O)=O)C(=O)NC1CC(F)(F)CC1NC(=O)CC1CCCOC1 c1(C(N2CC3(CCCC3NC(C3CC(O)C3)=O)C2)=O)cc2n(n1)CCCC2 Cc1c(CC(N2CCC(C)(CNC(C3CSCCS3)=O)C2)=O)oc2ccccc12 C1(NC(c2cc(OC)c(Br)nc2)=O)CC2CC1CN(C(=O)C(C)C(C)C)C2 C1(NC(COCCCOCC#C)=O)CC(C)CN(C(=O)C(CC)C(C)C)C1 c1(-c2ccc(OC)nc2)n[nH]c2ccc(C(=O)NCc3cncc(C)c3)cc12 c1(CC)cc(C)c(C(=O)NC2(C)CC(N)C2)o1.C1(=O)C(C)CC1=O.C1CC1 c1(C(N2CCOCC(F)(CNC(C(C)=C(C)C)=O)C2)=O)cccn2c(C)nnc12 c1(C(N2CCC(NC(CC3CCC(C)(C)C3)=O)C2(C)C)=O)nsc2ccccc12 CCCC(CCNC(C1(SC)CN(C(=O)C(C)OCCC(C)C)C1)=O)C1CC1 c1(CN(C)C(C2CCC3(C2)N=N3)=O)cccc(CNC(C2CCN2C)=O)c1 N1(C(C2(OC)CCC2)=O)CCC(CC(=O)NCC2(OCC)CCC2)C(C)(C)C1 Cc1ccc(Br)c(C(N2CCOCC2CNC(c2cc(Br)cc(F)c2F)=O)=O)c1F c1(NC(C(=O)NCc2ccc(CC)cc2)=O)cc(C)nc(C#N)c1 N1(CCCn2c(C)nnc2)CC(NC(=O)CCCN(C)C)CCC1C c1(N(C)CC2CC2(F)F)nc(=NCC2(C(N)=O)CC2)[nH]c2ncn(C)c12 N1(c2n(Cc3ccc(Cl)cc3I)c(C3CCC3)nn2)CCCC12CCNC2 c1(C(=O)NC(C(C)C)CCN(C)C(c2ccns2)=O)ccc(F)c(S(C)(=O)=O)c1 Nc1cncc(C(=O)NCCC2CCN(C(c3cccc(OC(F)F)n3)=O)C2)c1 c1(OC)cc(C)c(C(C)NCc2cc(C(=O)O)on2)cc1OC c1(C(=O)NC2CCN(C(=O)CC3CCCCCC3)CC2)cncc([N+](=O)[O-])c1 c1(OC)ncc(C(N2CCC(CC(=O)N(C3CNC3)C3CCC3)CC2)=O)cn1 C1(C)(C(C(=O)CN)=O)CCC(=O)C1.CCCC(C)CNC(=O)CN C1(C(=O)NCCC=CCC(N2CC(N(C)C)OCC2)=O)C2CC3C(C2=O)C13 C12CCC(CC1)C(=O)N(C)CCOC2.S(=O)(=O)(CC1CCOC1)N(CCOCC)C C#CCCN=C(NCC(=O)OC(C)(C)C)NC(c1ccco1)CN(C)C CC(C)C(CC(=O)Nc1cnn(CCF)c1)NC(C1(CCN(C)C)CC1)=O c1(OC(N2CCOC(c3ccccc3)CC2)C)ccc(N2CCCC(C)C2)c(F)c1 C1(CNC(C(C)N(C)C)=O)CCC12CCN(C(=O)Cn1cnc([N+](=O)[O-])n1)CC2 Cc1noc(C)c1C(=O)NC1CN(C(=O)Cn2nnc(-c3ccsc3)n2)CC1F C(C(C)NC(=O)CCNC(c1ccncc1)=O)(C(C)C)NC(CC=CCC)=O c1(OC)ccc2c(C(=O)NC3CC(CNC(c4c(C)[nH][nH]c4=N)=O)C3)csc2c1 C1(CC(=O)N(CC(CC)(C)COC)CC)CN(C(=O)C=Cc2ccc[nH]2)CC12CC2 Cc1nc2nc(=S)[nH]n2c(C)c1CCC(=O)NC1CC1CNC(=O)C(F)C(C)C C1(C(=O)NCC2CCCN2C(=O)Cc2sccc2Cl)C(C(F)(F)F)C1[N+](=O)[O-] c1(C(N2C(C)CC(CNC(=O)COC3COC3)C2)=O)cc2nn[nH]c2cc1F C(=O)(CCCCCCC(=O)N1CCOCC1)OC.C1(C(C)(C)C)C(=O)N1 C1(NC(c2cccc(C)c2)=O)CCN(C(=O)CC(C)N(C)C)CC1C CC(C)C(C(=O)C(=O)C(C)C)N1CCCC1=O.C(COCCON)N C(=O)(C1Cc2ccccc21)NCC(C)NC(C=Cc1c(C)n(C)nc1)=O C1(CN(C)C(c2cc(C(C)(C)C)nn2C)=O)CCCC(NC(C2CCC3CC23)=O)C1 C(C1CN(C(=O)C=C(C)C(C)C)CC1C(=O)NCc1cccc(COC)c1)=CC C1(CC(=O)OC)C(=O)NCCN1CCc1nc(-c2cccs2)no1 CCC(CC)C(=O)NCCCCNC(=O)C(c1cnn(-c2ccccc2)c1)=O C1(C(=O)OC)CC(F)(F)CN1Cc1cc(C(F)(F)F)cnc1Br Cc1n[nH]c(C)c1C(C1CCCN(C(c2ccc(Cc3ccccc3)[nH]2)=O)C1)=O O=C(C1=CCCN(C(=O)CC2CC2)C1)NCCCc1ccc(Br)cc1 N1(C(C(c2ccc(Br)s2)OC)=O)CCC(c2cn(C(C)C)nn2)C12CC2 C(=O)(C(CC(C)C)NC(=O)CC1CCC12CNC2)NCC(=O)OC C1(NC(c2ccc[n+]([O-])c2)=O)CCC2CC1CN2c1nnc(-c2ccccc2)o1 c1(C(=O)NC2CCC(NC(CC3(OC)CCC3)=O)C2)cc2c([nH]1)CCC(C)C2 NC(=O)CC(O)C(=O)NC12CC(NC(=O)CCCC(=O)NCC(F)(F)F)(C1)C2 CC(CCCNC(=O)CSC(F)F)NC(C1CCCSC1)=O C(CCCCCC(c1nnnn1C)Nc1nc(C(=O)N(C)C)cc(Cl)n1)OC C1(NC(Cc2cccc(C(=O)OC)c2F)=O)CN(C[Si](C)(C)C)C1 N1(C(CN(C(CO)C2CCC2)CC)=O)CCCC1(C)c1cccc(F)c1 c1(C(=O)NCC(C)(CO)NC(C2CC2C#N)=O)cc(F)cc2nc[nH]c12 CCC(C)C(C)CNC(C1COCC1NC(C1CN(C(N)=O)C1)=O)=O C1(C(=O)NCCCN(C(C(C)SC)=O)C)C2CCC1(C)C2(C)C C(=O)(C1=C(C)CCOC1)N1CC(C=C)(CC(N2CCC(N3CCC3)CC2)=O)C1 n1(CC)ncc(C(=O)NCC(C)C(N2CCCCC2c2nc[nH]n2)=O)c1C CCC(CC)CC(F)C(=O)N1CCCC1CCC(=O)NC1(CO)CC(O)C1 CC(C)CC(C)(O)C(=O)NCC1CC(C(N2CCC(O)(CCO)C2)=O)C1 N1(C(C2N(C(=O)OC)CCC2)=O)CC2CC(NC(=O)Cn3cnnn3)C1C2 C1(CC)CCN(C(c2cnc(O)o2)=O)C(C(=O)NCC(O)CF)C1 N1(C(C(C(C)C)NC(C2CCCN2C)=O)=O)CCOCC(C)(F)C1 c1(C(N(CC(C)NC(c2cnnn2C)=O)CC)=O)cccc(OCCF)c1 c1(C(C)C)ncc(C(=O)NCCCC2CN(C(=O)COCC3CCC3)C2)n1C N1(C(C2(C)ON=C(C)C2)=O)CCC(C)(CNC(c2ccc(C)nc2N)=O)CC1 Cc1c(C(=O)NC2CCN(C(=O)CC3OCCCC3(C)C)C2)cncc1N CCCCC(C)C(=O)N1CCCC(CN(C(=O)CN(CC(=O)NC(C)C)C)C)C1 C1(CC)(NC(=O)C(CC)n2ccnc2)CCN(C(C2CN3CCN2CC3)=O)CC1 N1(C(CCC#C)=O)CCCCC2(CCN(C(=O)CC3(N(C)C)CC3)C2)C1 C(C)(CN=c1cc(C)nc(OC)[nH]1)NC(CCCC#CC)=O N1(C(c2ccn(C)n2)=O)CC2CN(C(=O)CCc3ncnn3C)CC2(C)C1 C1(C)(OC)CC(N2CC(O)(C3CCC(=O)N3)C2)C1(C)C C1(CNC(Cc2ccc(CC)c(F)c2)=O)COC(C)(C)CN1C(c1cn[nH]c1)=O C#CC1(C(N2CCCCCC2)=O)CCN(C(c2cc(OC)cnn2)=O)C1 c1(CN2CCCC(O)(CNC(C(CC)C)=O)C2)ccc(O)c(C)c1O C1(CNC(C(CN(C)C)O)=O)CN(C(=O)C#CC2(C)COC2)C2(CCC2)C1 c1(C(N2CC(O)(CNC(C3C(C(=O)OCC)C3)=O)C2)=O)cc(F)cc2ccoc12 C(c1ccccc1Cl)=CC(N1C(CN(C(c2cc(CF)on2)=O)CC)CCC1)=O N1(C(c2csc(CO)n2)=O)CC2CCN(C(c3cc4n(n3)CC(F)C4)=O)C2C1 C(c1cncnc1O)=CC(=O)NCC1(F)CCN(C(C2ON=C(C)C2)=O)C1 C1(C)(C(=O)NCC)CC=C(C)CC1.C(CCNS(C)(=O)=O)NC(=O)CNC n1(CC)cc(Cl)c(C(=O)NCCCN(CCCNC(C2(O)CCOC2)=O)C)n1 CCC(C)(C(=O)NC1CCN(C(=O)COCc2nc[nH]n2)CCC1CO)C(F)F C1(C(=O)NCC(CCNC(=O)C=Cc2ccco2)O)CCOC(=O)CC1 N1(C(C(CCOC)(C)C)=O)CC2CC(NC(C3(C)CCC(OC)CC3)=O)C(C2)C1 c1(C(=O)NC(CCNC(CCN(C)CC)=O)(C)C)ccc2c(c1O)CCCC2 Cc1cc(CNC(C2CCCN(C3CCCC3C(=O)O)C2)=O)ccn1 C1(C(=O)NCC(CC)C#N)CN(C(C2(C3(C)CC3)CC2)=O)CC1(C)C C1(NC(N(C)C)=O)CN(N2CCC(NS(C)(=O)=O)C(C)(C)C2)CC12CC2 CCCC(C)(CC)C(=O)NC1CC(NC(=O)C(CO)C(C)(C)C)C1 N1(C(CCC#CC)=O)CCCC2(C1)CN(C(=O)CSC1CCS(=O)(=O)C1)C2 C1(CNC(C2(CC)CCC2)=O)CC(C)CN(C(c2ncoc2C(C)C)=O)C1 C=CCCCCC(=O)N1CCC(C(C)NC(=O)C(CCOC)OC)CC1 C1(CN2CC(=O)NCC2)CCC2(CCC2)C1.C12(CC(F)(F)C1)C(=O)NC2 C1(NC(c2oc(CC)c(C)c2)=O)CCN(C(c2cnn(C)c2Br)=O)CC1C C(CCC(CO)NC(c1cnn(CCO)c1)=O)NC(C=CSC)=O N12CCC(CC1)NC(=O)C1(CC1)C2=O.C1(CN(C)C(=O)NC2CC2)CC2CC2C1 c1(C(=O)NCCOCCOCCNC(c2c(SC)snn2)=O)nc(C)c(C)[nH]1 c1(C(N2CCC(C(C)NC(c3n(C(C)C)cnc3)=O)CC2)=O)cnccc1C#N c1(C(=O)NC(C2(O)CCCCC2)C(=O)NCCn2c(C)ncc2)cc(CO)n(C)n1 Cc1cc(C(=O)NC(C(C)NC(=O)CCc2ccn(C)n2)C(C)C)oc1C C(CC(C(C)(C)C)NC(c1cc(Cl)ccc1N)=O)N(C)C(c1cscc1F)=O C1(C)(CNC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)CCc2cc(Cl)no2)CC1 c1(OC)c[nH]c(C(=O)NCC2CC2NC(c2cc(C)n(C)n2)=O)cc1=O Cc1nc(CC(N2CCC(C)(NC(C3CCCN3C(C)C)=O)C2)=O)[nH]c1C C1(C(=O)OC(c2ccncc2)C)COC2CCCCC12.C1C(=O)N1 C(=O)(C(C)(C)C(F)(F)F)N1CCC(C)(CN(C)C(c2ncoc2C2CC2)=O)C1 CC1(c2cccc(Cl)c2)CN(N2CCC(CC=O)C2)C1.CCOCS c1(OC)ccccc1NC(=O)CN(S(C)(=O)=O)C.N12CCC(C1)N(C)C(=O)C2 CCCCC(C)C(=O)NC1(C)CC(NC(C2OCCC2C)=O)C1 Cc1ccc(C(C)N(C)C(=O)NC(c2nccnc2C)C2(O)CCCC2)c(C)c1 N1(C(C(n2cc(CC(C)(C)C)nn2)C)=O)CCC12CC(CF)C2 O=[N+]([O-])c1cc(Br)c(F)cc1CN1CCCC(OCC2CC2)C1 c1(NC(=O)NCC(F)CO)cnc2ccc(Br)cc2c1 N1(C(C2CC(C#C)(O)C2)=O)CCN(C(c2ccnc(COC)c2)=O)C(C)C1C c1(C(C(=O)NCC23CC(NC(C4CC(C)(C)C4)=O)(C2)C3)(F)F)ccc(Cl)cc1Cl C1(N(C(c2cc(CC)no2)=O)C)CC2CC1N(C(=O)Cc1cccc(OC)c1)C2 c1(OCC(=O)Nc2cnccn2)ccc(C(=O)NCc2ccccc2)cc1 c1(C(=O)NCC(CCNC(CCCCC)=O)(C)C)c[nH]c2nccc-2c1 C1(C(=O)NCc2scc(CNC(CN3CC(C)(C)C3)=O)n2)OCCC1(C)C c1(C(=O)NC(CNC(C(C)N(C(C)=O)C)=O)C(C)C)ccc2nnn(C)c2n1 c1(C(=O)NCCC2CN(C(C3C(C#C)C3)=O)C2)cc2sc(C)cc2o1 C(=O)(C1CCCc2cccnc21)NC1CC2CN(C(COCC#C)=O)C(C1)C2 c1(COCC)nc(C)cc(=NC2CC(CNC(=O)CC3(O)CCCC3)C2)[nH]1 c1(OCC(=O)NCC#CCNC(C2CC2C2CCOC2)=O)ccc2c(c1)CCC2 c1(C(=O)NCC2CCCN2CCF)coc(-c2ccsc2)n1 CCCCC(O)C(=O)c1ccc(-n2cc(C3CCCCC3)nn2)cc1 C(CC(C)(C)C)(C(=O)NCC(c1ccc(C)cc1)NC(=O)C(C)(C)N(C)C)OC c1(NC(C2(C)CCN(C(CCC(C)=O)=O)CC2)=O)ccc2c(c1)C(=O)NC2 CC1CCOCC1C(N1CSCC1C(=O)NCCC1CC(=O)N(C)C1)=O N1(C(c2c(C)cncc2)=O)CCC2CN(C(c3cnc(S)[nH]3)=O)CCC2C1 S(=O)(=O)(C1CCCCC1)NC12CC(NC(c3cc(F)c(Br)c(F)c3)=O)(C1)C2 N1(C(c2cc(COC)no2)=O)CC2CC1CN(C(c1cncc(C)n1)=O)C2 CN1CCN(C(=O)CN2CCSCC2)CC1CNC(=O)CC1OCCCO1 Cc1ccccc1C(C)C(N1CCCC1CNC(=O)CC1OCCCO1)=O CC(F)(F)C(C)(C)C(=O)NC1CCOC1C(N1CCCC(O)CC1)=O S(=O)(=O)(c1ccc(NCC(C)(C)C2CCCC2)c(C#N)c1)NC1C(C)COC1 CC(C)C(O)CC(=O)N1CC(OCCNC(c2ncsc2C(F)(F)F)=O)C1 N1(Cc2c(C)c(O)ccc2)CCc2[nH]nc(C(=O)Nc3cccc(I)c3)c2C1 C1(C(=O)NCC2N(C(c3c(OC)cnnc3)=O)CC2)CCCC12CCC2 C1(NC(=O)C(F)Cl)CCCCC12CN(C(C1CCCCO1)=O)CCO2 C1(CNC(C2C(C)C2)=O)CC2(CCN(C(=O)C(=Cc3cccnc3)F)CC2)C1 CC(C)C(O)CCNC(=O)C(CN(C)C)NC(=O)CC(C1CC1)C1CC1 Cc1cc(C(=O)NCC2CCN2C(=O)C(C)Cc2cnn(C)c2)oc1C c1(NC(C2C(O)CCN2C(c2cscn2)=O)=O)cc([N+](=O)[O-])ccn1 c1(CCNC(=O)NCc2c(F)cccc2Br)cc(C(F)(F)F)cc(C(F)(F)F)c1 c1(OCCOC)nccc(C(N2CC=CC2CNC(=O)CC2CCC2)=O)c1F N1(C(c2c(C)ccc(O)c2)=O)CC2(CCN(C(=O)CCC3CCCN(C)C3)C2)C1 Cn1nc2c(c1NC(=O)Cc1cccc(Br)c1F)CN(S(=O)(=O)C(Cl)(Cl)Cl)CC2 C1(NC(=NCCOC)NCC23CC(CO2)C3)CC(=O)N2CCCCC12 N1(CCC)CCC2(CC1)CC2NC(=O)CCC(C)(F)F C1(C(=O)NC(CSCC)CO)CC=CC(NC(c2ccc(OC)nc2)=O)C1 C1(c2n(C)cnn2)CCN(C(=O)C(N2CC3CCC2C3)=O)C(Cc2ccccc2)C1 C1(CC)CCCC(c2nnnn2Cc2ccco2)(Nc2cnc(Cl)c(SC)c2)C1 N1(C(C(=O)N(CC(C)NC(C(CC2CC2)OC)=O)C)C)CCCCCC1 c1(C(N2C(CN(C(=O)C=C=NOC)CC)CCC2)=O)ncccc1OC C(CCCC(=O)N(C1CCN(C)CC1)C)NC(C(CC1CC1)OC)=O N1(C(C(C2CCC2)NC(c2cccnc2)=O)=O)CCCC1Cn1ccnn1 c1(C(=O)NC2CCC(NC(C(C(C=C)C)C)=O)CC2)c(C)ccc2nsnc12 C1(c2nnnn2CC2CCOCC2)(NC(C=C)C)CCC(C)(C)CC1C C1(C(=O)NCCc2onc(C)n2)CCN(C(c2ncncc2N)=O)C1C(C)C Cc1cc(Cl)c(C(=O)NC2CC3(C2)CC3NC(C2CCC(=O)O2)=O)cn1 C(C(C)(C)S(C)(=O)=O)c1nnc(C(=O)NC(C)CN(C)Cc2ccccc2)o1 O(N(C)C(=O)CCC1CCCCN1C(=O)Cc1cnccn1)CC(=O)OC C(C(=O)N(CCNC(C1CCC(C)CC1)=O)C1CC1)(C(C)(C)C)OC N1(C(CCCC2C(C)C2)=O)CCC2CC12C(=O)NCCn1cnnn1 N1(C(C(C(=C)Cl)(C)C)=O)CCC2(CCC(NC(c3ccoc3Cl)=O)CC2)C1 C1(NC(CCC2CC(NC(CC=CCC)=O)C2)=O)CCCC1(C)O N1(N(CC2(CC3CC(COCCOC)C3)CC2)OC)CCC2(CCOC2=O)C1 C(C(N=[N+]=[N-])C(=O)N1C(C(=O)N(C)CCOCCO)CCC12CC2)OCC C1(CNC(CCC(C)NC(CN2CCC(C)CC2)=O)=O)CCC(C)(C)CO1 Cn1nc(C(=O)NCC2CCC2NC(=O)CCC2=CCCCC2)c2c1CCCC2 CC(C)CC(C)(C)C(=O)N(CCCNC(c1ccn(-c2cnccn2)n1)=O)C c1(C(=O)NC2CCC(NC(CCSC)=O)CC2)ccnc(C)c1C Cc1nc(C(N2CCC(NC(=O)Cn3ccccc3=O)CC2C)=O)c(C)n1C C1(NC(c2nc(C(=O)OC)sc2)=O)CCCC(NC(C23CC(C2)C3)=O)C1 N1(C(C(c2ccc(C)cc2)(C)C)=O)CC2CCCC(NC(C3CSC3)=O)C2C1 CC(C)CCC(O)C(=O)NC(C(=O)NCC1OCCC1(C)C)C(C)O N1(C(C(C(C)C)N(CC)CC)=O)CCCN(C(=O)CC2COCC(C)(C)O2)CC1 N1(C(CCOCC)=O)CCC(C)(C)C1C(N1CCCC(CF)C1)=O C#CCC(C)(C(=O)NC(c1ncc(C)[nH]1)CC)NC(=O)CCc1cc(C)[nH]n1 c1(C(=O)NCCCN(C)C(C2NC(=O)CC2C(F)(F)F)=O)cn(C)nc1O c1(C(=O)NCC2CN(C(C(C3CC3)OC)=O)CC2SC)n[nH]c2cc(C)ccc12 C1(NC(c2c(C)nc(O)[nH]2)=O)(CO)CCN(C(C2CCC(C)O2)=O)CC1 C1(NC(C2(CC)CC2(F)F)=O)CC2CN(C(=O)CCCCC#N)CC2C1 c1(C(=O)NCC(CNC(C2C(OCC)C2)=O)(C)C)ccc(NC)cc1O c1(CC(=O)NCC2C(NC(c3cc(CC)ncc3)=O)C2)c(C)ncnc1C C1(C)(NC(C(C2CCC2)OCC)=O)CCN(C(=O)COCc2ccccn2)C1 N1(C(=O)CN(C(C2CC2)=O)C)CCOCC(CC2CC2)C1.C1CCC1 C1(CCOC)(C(=O)NC(C)CC(C)NC(c2cc(CF)on2)=O)CCN(C)CC1 C1(NC(=O)CCc2cnc[nH]2)CC2CC1N(C(c1cn(CC(F)(F)F)cn1)=O)C2 C1(O)(CNC(CC2OCC(C)(C)C2)=O)CCN(C(=O)CN2CCNC(=O)C2)CC1 c1(C(N2CCC(O)(CCNC(=O)C3=COCCC3)C2)=O)ccc2c(c1)CCCO2 C(=O)(CC(CNC(=O)CC1CCSC1)OC)NC1(CCOC)CC1 C(=O)(C(C)(C)CCC#N)N1CCC(C(n2cc(C3(S(=O)(=O)N(C)C)CC3)nn2)C)C1 CCC(C)(C(=O)NCCCCC(C)NC(=O)CCCc1nnc(C)n1C)C(N)=O N1(C(c2ncn(C)n2)=O)CC(NC(c2cc(O)n(C)n2)=O)C2CCCC12 c1(C(=O)NCC2CC(C)(C)N(C(=O)Cc3cn[nH]c3)C2)nnc2ccccc2n1 S(=O)(=O)(c1ccc(NC2CCC3CC23)c(F)c1)NC(c1nc(CC)sc1)C c1(C(N2CCC3(NC(CN(CCC)C)=O)C(CC2)C3)=O)cc(O)cc([N+](=O)[O-])c1 CCCCCCCC(=O)N1CC2CN(Cc3cnn(CC(C)C)c3)C2C1 CC(C)(C)CC(O)CC(=O)NCCC1(C(=O)NC2CSC2)CCCC1 c1(C(C)C)[nH]nc(C(N2CC3CCN(C(C4CCC5CC45)=O)C3C2)=O)c1[N+](=O)[O-] C1(C(=O)NCCC2CCN(C(c3n(CC)ccn3)=O)C2)CC2OC(C)(C)OC2C1 O(N1CCC(CC(=O)NCC2CCN(C(=O)Cc3cc[nH]n3)C2(C)C)CC1)CC CC1CC(N(C)C(c2n[nH]cc2CNC(C2CCCC2C2CC2)=O)=O)CC(C)O1 C(=O)(C1CCCc2ccccc21)N1CCC(CNC(C(CC(N)=O)O)=O)(CO)C1 C1(CNC(C2CC(F)(F)C2)=O)CCC2(CN(C(C3COC4CC3C4)=O)C2)O1 C1(C(=O)NCC(C)N(C(=O)CN=S(C)(C)=O)C)CCn2cc(C(F)(F)F)nc2C1 C1(OC)CC(CCNC(=O)CCSC)N(C(=O)CCCOc2ccc(C)cc2)C1 C(=O)(N=c1ccn(CCc2ccccc2)[nH]1)NC(c1cc2c(s1)CCCC2)C c1(C(=O)NC(CNC(C(c2ccccc2)OC)=O)C)c(C)[nH]cc([N+](=O)[O-])c1=O c1(C(=O)NC2(C3N(C(CC4CC(SC)C4)=O)CCCC3)CC2)cncc(Cl)c1Cl c1(OC)ccc(F)c(C(N2CCC(NC(C3(C)CC4CCC3C4)=O)C(C)C2)=O)c1 C=C(C)CCC(=O)NC1COCCC1NC(=O)C(O)c1ccco1 c1(C(=O)NCCC(C)N(C)C(c2ccc(OCCO)cc2)=O)ccc(C#N)[nH]1 Cc1ccc(OCC(=O)NC2CC(NC(C3CC3c3nncn3C)=O)C2)c(F)c1 C1(C(=O)NC(C)Cc2ccncc2)C2CCCC2CN1C(C1OC2CCC1C2)=O N1(C(C2(COC)CCCO2)=O)CC(NC(=O)CSC2CCOCC2)CC(F)C1 N#Cc1cnc2c(F)cc(F)cc2c1C(=O)NCC1(Sc2ncccc2F)CC1 C1(CNC(c2cn(C)nn2)=O)CN(C(=O)C(C)(C)C2CCCO2)CCC1(F)F c1(OC)cc(O)ncc1C(N1CC2CCC1(CNC(=O)C(C)(C)F)C2)=O C1(C(=O)NCC(C2CC2)NC(c2ncccc2C(F)F)=O)CCC2CC1CO2 N1(C(=O)OCCC)CCCC1(CCC)CC S(=O)(=O)(c1cccc2cccnc12)NC1CN(C(CN(C(C)C)C)=O)CC12CC2 C1(NC(C2(CNC(=O)Cc3nonc3C)CC(=C)C2)=O)CCC(F)(F)C1 C1(C(=O)NC(C)Cc2cnccn2)CCN(C(c2ccncc2F)=O)CC1O C1(NC(=O)Cn2nnc3c2CCCC3)CN(C(C2CCC2)=O)C2(CCCC2)C1 N1(CC(N2CC(O)(CNC(CN(C)C3CC3)=O)C2)=O)CCC(C)(O)C1 c1(C(=O)NC2CC(=O)NC2)cnc2c(c1)CCN(Cc1ccc(Br)cn1)C2 N1(C(c2ccc(C)nn2)=O)CCCC2C1CCN2C(c1cc(C)c(C)o1)=O CN(C)S(=O)(=O)NCC(=O)NC1(CO)CN(C(c2ncc[nH]c2=O)=O)C1 S(=O)(=O)(c1ccc(NCc2ncc(C(N)=O)s2)c(Cl)c1)N(CCC#N)CC C1(CNC(CNS(NC)(=O)=O)=O)CN(C(c2cc(N)ccn2)=O)CC(C)(C)C1 c1(N2CCC(N(C)CC)C2)nc2ccsc2c(=NCc2ccc(SC)o2)[nH]1 C1(C(N(CCCOCCNC(C(CC)c2cccnc2)=O)C)=O)CC2CCC1O2 C1(C(N(CCOCCNC(C(C(CC)C)=O)=O)C)=O)Cc2ccccc2C1 C1(C(N2CCC(C(=O)NCCc3cn(C)cn3)(CC)C2)=O)CCCC(=O)CC1 CCC(CC(=O)N1CCOCC1CCNC(=O)CCCCc1ccccc1)OC c1(C(N2CC(NC(COCCCC)=O)CC3(C2)CC3)=O)nc2ccccc2[nH]1 c1(SCC)cccnc1C(=O)N(CC(O)CN(C)C(N)=O)C.c12cccc(c1)OC2 C(C(=O)N1CC(O)C(O)CO1)(C1N(C(C(CC)SCC)=O)CCC1)N Cc1c(C(=O)NC2CCC2NC(c2ccc(Br)cn2)=O)oc2ccccc12 N1(C(CCSC)=O)CC2CC(NC(=O)C=CCn3cncn3)C(C2)C1 CC(C(C)(C)C)N(C)C(c1c[nH]nc1CCNC(=O)CCc1cnco1)=O C1(C(=O)NCCN(C(c2n(CC)ncc2C)=O)C2CC2)CCC2CC1CO2 N1(C(C=CCOC)=O)CCC(C2CCCCN2C(=O)C(C)C(=O)OC(C)C)CC1 c1(CNC(COC)(C)C)ccc(-n2nc(C)cc2C)nc1 C1(C(=O)Nc2c(OC)nc(Br)cc2)CN(Cc2cc(Cl)ccc2Br)CC(F)(F)C1 c1(SC)cccc(NC(N2CCC2(C)CNC(=O)CN2CC3CC3C2)=O)c1 C#CCCC(O)C(=O)NCC1CC(F)CN1C(C1(C2(O)CCC2)CC1)=O O=C(C#CC1CCOCC1)NC1C2CC1N(C(=O)CCc1cnc(C3CC3)o1)C2 n1(CCOCC)nc(C(c2nn[nH]n2)OC(C)(C)C)nc1-c1ccc(C(C)C)o1 C(C(O)C(F)(F)F)SCCN(C(=O)CCSCC(N)=O)C.C1C(=O)N1 N1(C(C2CN(C)C2)=O)CC2CC(NC(C3(C)CCOCC3)=O)C(C2)C1 N1(C(C=Cc2c(C)ncs2)=O)CCCC2(C1)CN(C(c1ccc(CO)cn1)=O)C2 Cc1cc(C)n2nc(C)c(C(N3CCC(CN(C(=O)CC#N)C)C3)=O)c2n1 Cc1cc2sc(C(=O)NC3CC(NC(=O)CCc4ccoc4)C3)c(C)c2cc1C C12CN(CC1NC(C1(Cc3ccccc3F)CC1)=O)C2=O.c1(S)ccc(Cl)cc1.CO C1(C(=O)Nc2cn(CCC)nc2)CN(C(=O)CCC2CCOCC2)CC1C N1(C(=O)C(F)(F)F)C2CCC1CN(C(c1nc(SC)sc1C(=O)O)=O)C2 N1(C(C2CCCO2)=O)CCC2(CC1)CC2CNC(C1(F)CCCC1)=O C1(NC(C2(C)C(C)(C)C2)=O)CCCCC1C(=O)NC(C1CC1)C1CC1 N1(CCC(N2CCC(CN(C(C(C)N(C)C)=O)C)C2)=O)CCP(C)(=O)CC1 c1(OC)cc(NC(C23CC(NC(c4ccc(N(C)C)cn4)=O)(C2)C3)=O)ccc1Cl c1(CNC(=O)CSCCNC(C2C=CCCC2)=O)cnnc(O)c1 C(=O)(CC(CC1CC1)NC(c1ccc(CO)cc1)=O)NCC(CC=C)OC C#Cc1cc(F)ccc1CNC1CC(C(=O)Nc2ccc(Br)c(C)c2C)C1 CC1(C(N2CC(CO)(NC(=O)C(=O)NCC(F)F)C2)=O)CC2(CC2)C1 C1(C(N2CC3C(N(C(c4cc(C)sc4C)=O)C)C3C2)=O)CC(=O)NC(C)C1 C1(NC(C2(NC(C(CC)(CC)OC)=O)CC2)=O)CCCC(C2CC2)C1 Cc1ccc2cc(C(N3CCN(C(=O)CC(C)CN(C)C)C(C)C3)=O)[nH]c2c1 Cc1cc(Cl)n[nH]c1=NC(=O)c1ccccc1NCc1cnc(O)nc1O C1(NC(CC2CCN(C)C2)=O)CC2(CCN(C(c3nc(Cl)cs3)=O)CC2)C1 C1(OC)CC(C(=O)NCc2nc(CNC(=O)C(O)C(C)C)cs2)CC1OC C(CC(C)C)(C(=O)NC(C)C(C)NC(=O)Cc1cc(C)cc(F)c1)NC(C)=O C(=O)(CCCN=[N+]=[N-])NC(C(C)O)C(=O)NCCCC(C)(C)CO c1(CN2C(CC(=O)OCC)CCC2)cc2c(nn1)CCOC2.C1(=O)CS(=O)(=O)N1 CC1(C)CCC(C(=O)NCc2nc(CNC(C3CC=CC3)=O)cs2)C1 C1(C(=O)NC2CCCC(NC(CN(S(C)(=O)=O)C)=O)C2)CSC2(C)CCC(=O)N12 C1(C)(NC(c2ncn(CCNC(C(CN(C)C)O)=O)c2)=O)CCOC1=O CC1(C(=O)NC2(C(O)CO)CC2)CC(O)CN1C(=O)CS(C)(=O)=O N1(C(CCOC)=O)CCC(NC(=O)CC2CCC3(CCC3)O2)C12CCCC2 c1(C(=O)NC(CCNC(C2CC(CC)(CC)C2)=O)C)ccnc(CO)c1 N1(C(c2ocnc2C(F)F)=O)CC2CN(C(C3CC4(CCC4)CO3)=O)CC2C1 N1(C(CC2N(C)CCOC2)=O)CC(NC(c2cccnc2O)=O)C2CCCC2C1 N1(C(C23N(C(c4nccc(CC)c4)=O)CCC2C3)=O)CC(O)(C2CC2)C1.C1CC1 N1(C(CN(CC(C)(C)C)C)=O)CCC2(C1)CN(C(=O)CCc1ncc[nH]1)CCO2 N1(C(C2CC(SC)C2)=O)CCCC2CN(C(c3ccc4c(c3)CNC4=O)=O)CC12 N1(C(C2C(CC)CCO2)=O)CCN(C(=O)C(C2CCOC2)OC)CC1CCOC c1(C(N2C(CC(=O)NC3CN(C)C(CO)C3)CC2)=O)c[nH]c2ccncc12 C1(O)(C(C)CCNC(=O)CCF)CCN(C(c2ccc(-c3cnco3)cc2)=O)C1 N1(C(C=CC(N)=O)=O)CC2(CC(CNC(c3cccc(Cl)c3)=O)C2)C1 c1(NC(C(CCNC(C(c2ccccc2)C)=O)O)=O)ccc2cnccc2c1 N1(C(C(CC)OCC)=O)CCC(OC)CC1.c12ocnc1C(=O)N1CC2C1 N1(C(c2c(C)nns2)=O)CC2CCC1CC2NC(c1cnn2cccc(Cl)c12)=O C1(O)(C(CNC(CCC=CC(C)C)=O)C)CCN(C(C2(Cl)CC2)=O)C1 c1(N2CC(COC)N(Cc3cnc4ccccn34)CC2)ncnc2scc(C)c12 N1(C(c2ccccc2)=O)CCCN(C(=O)CNC2(C(N)=O)CC2)CCC1 c1(C(c2n(CCC(=O)OC)nnn2)NCC2(CC3CC3)CCC2)cc(C)c(Br)s1 n1(CC)cc(C(N2CCCC2CC(C)(C)C)C(=O)NCCC#N)cn1 C1(CNc2cncc(C#N)n2)CCC2(CCOCC2)CO1 CC(C)CC(O)C(=O)N1C(C(=O)NC2(c3nn[nH]n3)CC2)CCC1C c1(CC(=O)NCCNC(C2CCC(F)C2)=O)ccc(F)cn1 C1(F)(CNC(C(C)c2ccsc2)=O)CC(NC(=O)C(F)=C2CCCC2)C1 C=Cc1cccc(SOc2c(NC3CC3C(N)=O)nccc2)c1 C1(C(N(C)Cc2cnn(C)c2)=O)COC2(CCCC2)C1 C(=O)(C1=CCCN(C(=O)CCCC(=O)C2CC2)C1)NC(c1c(C)ncs1)C C12(CNC(=O)NC(CC)C(=O)NC)COC(C)(OC1)OC2 C1(C(N2CC(NC(c3[nH]cc(CC)c3)=O)C2)=O)CCCN(C(C)=O)C1 CC(=O)CCCCC(=O)NC1CCCCCN(C(c2ocnc2C)=O)C1 C1(NC(=O)CCCCCF)C2CC3CN(C(C4CN5CCCN4CC5)=O)C1C3C2 N1(C(C=CCCC(C)C)=O)CCC(C)N(C(=O)CC2CCCC23CC3)CC1 C=CCCCC(=O)NC(C)(CSC)C(=O)N1CCC(CN=[N+]=[N-])C1 Cc1cc(Br)cc(F)c1C(N1CC(N(C(=O)Cn2cncc2C)C)C1)=O C=CCCCC(C(=O)NCC(N1CCCCC1)=O)NC(=O)CCCC(C)C CCCC(CNC(=O)C(CC1CCC1)NC(C1CCC2(CC1)CC2)=O)CCC c1(OCCN(C(C(=O)NCC(c2cccnc2)C)=O)C)ccccc1Br C1(CC(=O)NC2CCN(CCC)C2)CCCN(C(=O)C=Cc2cscn2)C1 C1(C(=O)NCC(C)(C)NC(C2CC23CC3)=O)CCc2nnc(-c3ccon3)n2C1 N1(C(CC2(CSC)CC2)=O)CC(NC(=O)CSCCC(C)C)CC12CCCCC2 c1(C(=O)NCC2(O)CCN(C(c3c(C)nc[nH]3)=O)C2)cnn2c1OCC(F)C2 CCC(CC(C)C)C(=O)NCC1(C)CCCN(C(c2cccn3cnnc23)=O)C1 Cc1ccc(C(N2CCC(NC(c3ccnc(C(F)F)c3)=O)C(C)C2)=O)nc1C CC(C)(C)C(C(=O)NCC1CCCCCC1)NC(c1cc(O)cc(F)c1)=O c1(CC)cc(C)c(C(=O)NC2CCC(NC(=O)C(C)(C)c3cscn3)C2)o1 c1(-n2cc(C3C(C)CCN3C(=O)CC3CN(C)CC3O)nn2)cccn(C)c1=O CC(C(=O)N1CCC(CNC(c2ccnc(OC(F)F)c2)=O)C1(C)C)S(N)(=O)=O CC(C)(C)C#CC(=O)N1CCN(C(c2ccncc2F)=O)C(CF)C1 Cc1cc(C)c(C(=O)NCC(C)(C2CCC2)NC(=O)CCC2CCCCO2)o1 CC1(C(N2CCC(C(F)Cn3cc(CCCO)nn3)CC2)=O)CCCS1(=O)=O Cc1ccc(NC(C2CCN2Cc2csc3ccccc23)=O)c(C)c1Cl N1(C(c2nc(NC)oc2)=O)CCCC(CCNC(=O)Cn2cc(Cl)c(C)n2)CC1 c1(C(=O)NC(C(C)NC(C2(OC(C)=O)CC2)=O)C)cccc2c1oc(=O)n2C c1(-c2ccc(CN3CC(C)NC(=O)C3)c(F)c2)c[nH]c2ccccc12 C1(CNC(c2n[nH]c(C)c2F)=O)(NC(=O)CCn2cncn2)CCCCC1C C=CC(C)N=c1[nH]c(=NCCn2ccc(=O)cc2)[nH]c2c1CCCC2 N1(C(c2c(N(C)C)cncc2)=O)CCC(NC(c2ncccc2Cl)=O)C(F)C1 N1(CCN(C(c2cccc(OCCC)c2)=O)C)c2ccccc2CC1C c1(CC(C)C)cccc(C(N2CC(NC(=O)C(F)CC3CC3)C(C)C2)=O)c1 c1(-c2n(C(c3ccc4c(c3)OCCO4)C(=O)NC)ccn2)cccc2c1CCCC2 N1(C(c2nc(COCC)sc2)=O)CC(NC(c2ccc(C(N)=O)[nH]2)=O)C2CC12 CCC(CN(C)C)CC(=O)NC(C1(C(=O)NCCC(C)C(F)(F)F)CC1)C N1(C(CNC(C2(NC(N)=O)CC2)=O)=O)CCCC2CCCCC12.C1C(=O)N1 C12(C(=O)NC3C(NC(C4CCOCC45CCC5)=O)CC3)CCCN(CCC1)C2 C1(C(C)C)CCC(C(=O)NCC2(NC(=O)C(c3ccccn3)C)CC2)CC1 CC#CCCC(=O)NCC1C2CN(C(=O)C(N)=O)CC12 N1(C(C2CCN(c3nc(=N)[nH][nH]3)C2)=O)CCc2nc[nH]c2C1 N1(C(c2ncc(C)cn2)=O)CCC2C(C1)CN2C(c1cc(-c2ccco2)no1)=O c1(C(=O)NCC2C(NC(C(CC)=CCCC)=O)CC2)ccc(OC)c(Cl)c1OC N1(C(CSCC#C)=O)CCCN(C(=O)C(C(C)C)N2CCC(C)CC2)CCC1 Cc1ccc(C(N2CCC(NC(=O)CC34CCCC3C4)C(C(N)=O)C2)=O)nc1C C(N=c1[nH]c2c(c(=NC(C)C)[nH]1)CCCC2)c1n(CCC)nnn1 c1(N2CC(C(C)C)N(C)CC2)nc(NCC(c2ccccc2)F)c2ncsc2n1 CN1CCN(N2CCCC2(C)C2CCC(F)(F)CC2)CC12CCOC2 C1(NC(c2ccc(CC(C)C)cc2)=O)CCN(C(C2CCCN2C=O)=O)CC1F C1(N(C(CCCOc2ccc(C)cc2)=O)C)CC2CCC(C1)N2C(=O)CC(C)C N1(C(c2c(C)onc2)=O)CCOCC1CN(C(=O)CC1CC2(CC2)C1)C CCC(C)(C)CC(=O)NCC(C1CCCN1C(C1C=CC=CC=C1)=O)(C)C C(=O)(CN=S(C)(C)=O)NCC(c1ccc(N(C)C)cc1)NC(Cc1c(C)n[nH]c1)=O c1(N2CCCC(C)(C)C2)ncccc1S(=O)(=O)NC1CCC(F)(F)CC1 N1(C(C2N(C(CCCCCSC)=O)CCC=C2)=O)CCC(C2CCC2)CC1 Cc1c(Br)c(C(N2CCC(O)C(C(=O)NC(C3CCC3)C)C2)=O)nn1C c1(C(=O)NCc2cccc(CC)c2)cc(OC)ncc1-c1ccc(OC)nc1 Cn1nc(C2CCN(C(=O)NCC3CCCOC3c3cc[nH]n3)CC2)cc1N C(=O)(CC(C)CC)N1CC(OCCNC(CCSCC)=O)C1 c1(CC(=O)N(CCCCNC(=O)COC2CC2)C)c(F)cccc1Br C1(O)(CNC(=O)CC2CC(O)C23CCC3)CCCN(C(C2(O)CCCC2)=O)C1 N1(C(c2n(CCOC)ncc2)=O)CCC2CN(C(=O)CS(=O)(=O)CC)CCC2C1 N1(C(c2nc(CCC)oc2)=O)CCC(C(F)(F)F)C(CNC(=O)C(C)(F)F)C1 c1(C(C(N2CCC(C(C)C)C2)=O)N)cccc(I)c1 C1CCC(C2CCN(Cc3cc(C4CC4)no3)C2)CC1 C=CCC(CNC(C1(CNC(=O)COC2CCOC2)CCCC1)=O)CC(C)C C1(CN(C)C(=O)NC(C2CC2)C2CC2)CC(C(F)(F)F)CO1 c1(NC(c2c(OC)c3c(cc2)CCC3)=O)ccc2c(c1)C(=O)c1ccccc1-2 C1(N(C(C(CCC)NC(=O)NC)=O)c2c(C)noc2C)CCC12CCNCC2 C(C(CC(C)C)C(=O)NCC(C)(F)CNC(c1ccc(N)c(F)n1)=O)OC C=Cn1nccc1C(N1CC(CNC(c2ccnc(OCC)c2)=O)C1)=O c1(N(C(c2csc(Br)n2)C(=O)NCc2c(SC)cccc2)C)ccc(C#N)cc1 n1(CC(=O)NCCNC(c2coc(Cl)c2)=O)cc(I)cn1 CCCCC(C)CCC(=O)NC12CCC(CNC(=O)CC3=CCCC3)(C1)OC2 Cc1cc(NC23CCCN(CC2)C3)ncc1S(=O)(=O)NC(CC(N)=O)C1CC1 c1(OCCC)ccc(C(=O)NC2(CNC(c3cn(C(F)F)c(C)n3)=O)CC2)cc1 CCC(C(=O)NCCCCC(C)NC(c1cnoc1C1CCC1)=O)C(C)C c1(-c2ccc(C)s2)ccc(CCn2c(-c3c(S)cncn3)ncc2)cc1F.C1CC1 C1(CCCC)CN(C(=O)C(CC)CCC)CCN1C(c1cc(C)c(C)[nH]1)=O O=C(NNC(=O)C(=O)Nc1ncc[nH]1)NC1CN2CCCC1C2 C(=O)(C(=O)C(C)(C)C)N1C(CC(=O)NCC(CCC)(C)O)COCC1 c1(C(N2C(C3(C)CC3)CCC2)=O)cc(C=O)ccc1F c1(C(N2CC(CC)C(NC(c3ccc(OC)s3)=O)CC2)=O)c(C)cc(C)cc1N c1(C(=O)Nc2c(C)cc(N3CCCC3)cc2)cccc(Cl)c1N=[N+]=[N-] C1(C(N(CCCCC)C)=O)C=CCN(C(=O)C(F)C(=O)OCC)C1 C(C(CC1CC1)C(=O)NOCC(O)C(C)C)NC(c1c(C)ccc(F)c1)=O CCC(C)CC(CO)NC(=O)CC1(NC(=O)Cc2cnsc2)CC1 C12(NC(c3ccc(OC)cc3)=O)CCC1CN(C(=O)Cc1ccc(SC)cc1)C2 c1(C(NNC(=O)Cc2cc[nH]n2)=O)cc2ccc(F)cc2nc1O N1(C(c2c(SC)csc2)=O)CC(CNC(c2coc(C(F)F)n2)=O)CC1(C)C C1(CCNC(CCc2c(C)ncs2)=O)CN(C(=O)CC23CCC(CC2)C3)CCO1 N1(C(C(CCOC)C)=O)CCN(C(c2cnn(CC(F)(F)F)c2N)=O)C(CF)C1 C(=O)(CCCCC(C)(C)C)NC1(CCNC(c2cc(C(CC)C)c(C)o2)=O)CC1 c1(N2C(CNC(c3c(C)coc3)=O)C(C)CC2)nc2ccccc2s1 N1(C(CCSCC(C)C)=O)CCC2(CC1)COCC(CNC(=O)C(O)CN(C)C)O2 Cc1cc(Br)cnc1C(=O)NC(CO)C(C)NC(=O)C(=O)NC1CC1 C12(C(N(CC(C)O)C(C)C)=O)CC(NC(c3cn(CCO)nn3)=O)(C1)C2 C(c1ccc([N+](=O)[O-])s1)=CC(N1C(CCNC(CSCC#C)=O)CCCC1)=O CC1CN(C(=O)CSc2cnn(C)c2)CC(C)C1NC(C1(O)CCC1)=O N1(C(C(N2CCC(OC)CC2)=O)=O)CC(=O)NC2CCCC2(C)C1 c1(C(N2C(CNC(CC(=C=C)C)=O)C(C)CC2)=O)ccnc2cc(OC)ccc12 C=C1CCN(C(=O)CCCOCC)C(C(=O)N)C1.C(CO)(C(=O)OC)NC(N)=O c1(OC(C(=O)NCC2N(C(C(Br)=C(C)C)=O)CC2)C)ccc(Cl)c(Cl)c1 C1(C(=O)NCC2CN(C(C)C)C2)CC(F)CCN1C(=O)CC(O)CN(C)C C(=O)(CCCC(F)(F)F)N1C2C(NC(C(C3CC3)OCC)=O)C(C2)C1 C1(CC(=O)NCCCN(C(=O)Cc2nc[nH]n2)C)CCCS(=O)(=O)C1 N1(C(Cc2ccc(C)c(O)c2)=O)CC2C=CC1C(C(=O)NCc1nc(=O)o[nH]1)C2 c1(C(=O)NC2(CC)CN(C(c3cc(Cl)no3)=O)C2)cc(C)cc(C#N)c1 CC1Oc2ccc(CNC(=O)C(n3cc(CCC4CCCC4)nn3)C)cc2C1C N1(C(=O)C=Cc2ccoc2)CC2(CCC2)CC1CNC(C12C=CC(CC1)C2)=O c1(NCC2C(NC(C(C=C)OC)=O)CCCC2)ccc(C#N)c(C)n1 C1(CNC(=O)COCC(F)(F)F)CC2CCC1N2C(C1CC2CCC1CC2)=O C1(NC(c2cnc(-c3ccccc3)s2)=O)CCCC(N=c2[nH]nc(C3CC3)s2)C1 Cc1oc(C2CC2)nc1C(N1CC(CCNC(C2(C)CSC2)=O)C(C)C1)=O CN1CCCC(CCNC(=O)C(=O)NCc2cccc(N3CCSCC3)n2)C1 N1(C(c2ccc(Br)cc2OC(F)F)=O)CCCCC12CCCNC2 c1(CC)nn(C)c(NCC(C2CC2)N(C)C(c2ccc(Br)o2)=O)c1[N+](=O)[O-] C(=O)(CCC#Cc1ccccc1)OC(C)(C)C.N12CCC3(CCCC13)NC2=O Cc1nnc2c(C(=O)NC3CCCN(C(=O)COC4CC=CC4)CC3)nccn12 c1(NC(=O)C=CCNC(C2CC23CCC3)=O)ccc2c(c1)CCO2 C1(NC(C2CNC(=O)N2)=O)(CO)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1 c1(C(N2CCCC(O)(CNC(C(C)C(F)F)=O)C2)=O)nc2ccccc2nc1O C(=O)(C1=CC2C=CC1C2)NC(C(CC)C)C(=O)N1CC2CC1CN2CC N#Cc1ccc(CCC(=O)NC2CCOCC2NC(=O)CC2CC=CC2)c(F)c1 CC1(C)CCN(C(=O)C=Cc2ccco2)C1CNC(=O)CCc1ccncn1 c1(C(=O)NCC2(C)OCCN(CC(=O)NC)C2)cc(C)c(Cl)cc1OC c1(C(N2CCC(CNC(C(CC)SC)=O)CC2)=O)nnc2c(F)cccc2c1O Cc1nc(C)c(C(=O)NC2(CC(=O)NCC3CCC(C)C3)CCCCC2)[nH]1 N=c1ccc(C(N2CC(O)(CNC(=O)CCF)C2)=O)n[nH]1 C#CCCCCC(=O)N1CCOC(C(C)NC(c2cc(CC)c(CC)o2)=O)C1 CC(CC(=O)NCC(C1CCC1)NC(=O)CCc1cc[nH]n1)C(F)F Cc1nc(C(=O)NCCC2CCN(C(C3CCN3C3CCCC3)=O)C2)c(C)n1C N1(C(C=CC(C)(C)C)=O)CCC(C(=O)Nc2cnccn2)C1 c1(C(=O)NCC2(NC(c3cc(C)no3)=O)CCCCC2C)ccc2c(c1)NCC2 C1(C(=O)NCC2OCCN(CC)C2)CCCCC1N=c1nc(OC)[nH]c(OC)n1 C1(NC(C=COCC)=O)CC(NC(=O)C(Cl)=CCl)C12CCOCC2 c1(C2C(C(=O)OCC(=O)NCC(C)C)C2)cncs1 N1(C(CC(COC(C)=O)(C)C)=O)CC2(CCCC(CNC(=O)C3CC3)O2)C1 n1(C(COC)C)nc(CO)nc1-c1cccc(-c2ccco2)c1 c1(C(N2C3C(NC(C4CC=CCO4)=O)CC(C3)C2)=O)cn2cccc(F)c2n1 C1(NC(C2(CC=C)CC2)=O)CC1C1CCN(C(c2c(SC)cnn2C)=O)CC1 C=CC(C)(CC)C(=O)N(CC(C)NC(c1cc(-c2ccncc2)[nH]n1)=O)C c1(NCCCOCC=C)[nH]c(=NCC(C2CC2)C2CC2)nc2c1cnn2C CCCS(=O)(=O)CC(=O)NC1CCN(C(C2CCN2CC)=O)CC(O)C1 CC1CN(C(c2csnc2Cl)=O)CC1C(=O)NCc1nc(C#N)cs1 C1(C(=O)NC2CC(C(F)C(=O)NCC(C)CSC)C2)(OCC)CCCOC1 c1(C(N2CCN3CCC2C3)C(=O)NCCCSCC)nn(C)c2ccccc12 c1(C(N(C(CC)CNC(c2ccc(COC)o2)=O)C)=O)ccn2ccsc12 c1(C(CC(=O)OCC)C)c[nH]c2ccccc12.C1(C)(N(C)C(NO)CC)CC1(F)F c1(CNC(C(F)F)CCc2ccccc2)ncc(Cl)cc1Cl C1(C(=O)NC2CC(CCNC(=O)C=C3CCCCC3)C2)Cc2ccncc2N1 O(NC(=O)C(O)C1CCC1)C(C1CCC(Cc2ccccc2)O1)=O N1(C(C=CC(N)=O)=O)CCC(C2CCCCN2C(C2CC=CCO2)=O)CC1 CCC(CCOC)C(=O)OCCO.C12(CCC1)C(=O)N1CC(C1)N(C)C2=O S(=O)(=O)(c1c[nH]c(C(=O)NC(C)CN(C)C(C2(CC(C)C)CCC2)=O)c1)NC CC(C)C(N=[N+]=[N-])C(=O)NCC1CC(C)(C)CCC1NC(=O)C(F)C(F)(F)F N1(C(c2c(CC)nn[nH]2)=O)CCCN(C(=O)CC(C)O)C(CO)C1 N1(C(C#CC2(CC)COC2)=O)CCCC2(C1)CN(C(=O)C=CS(C)(=O)=O)CCO2 c1(OC)cnc(Br)cc1C(c1nnnn1C1CCC1)Nc1cncc(C)c1 c1(OC)ccc(C(=O)NC2CN(C(C3(N(C)C)CCCOC3)=O)CC2F)cc1 C1(NC(C2C(CC)C2)=O)CC2CN(C(c3c(O)cccc3O)=O)CC12 CN1CC(C(=O)NC2CCCC2CC(=O)NC2CC3C=CC2C3)CCC1=O C1(C(N(C)Cc2cccc(C3(N)CC3)c2)=O)CCCC12OCCO2 C(c1cncnc1O)=CC(N1CCC(NC(C(=Cc2ccccc2)OC)=O)C1)=O N1(C(c2c(C)con2)=O)CCN(C)CC1CNC(c1cccc(N)c1O)=O N1(C(CCc2cnc(C)o2)=O)CCC=CC1C(=O)NCC(O)CF c1(C(N2CC(C(=O)NCCCC(C)O)CC2(C)C)=O)c[nH]c2ccncc12 c1(OC)cnnc(C(N2CC3CC2C3C(=O)NCc2csc(C)c2C)=O)c1 C1(NC(C(C)CN(C)C)=O)CN(C(C2(c3cccnc3)CC2)=O)CC(C)(C)C1 C1(NC(C(C)SCCCC)=O)CCN(C(c2ccnc(C(C)(F)F)c2)=O)C(C)C1 c1(C(=O)NCC(C2CC2)NC(c2nc(C)oc2)=O)cc2n(n1)CCCC2O c1(-n2cc(CC=C)nn2)cccc(CNC(=O)CCN2CCC(C)C2=O)c1 C=C(C)CC(C(=O)NC(CNC(c1cc(N)ccc1F)=O)CCCC)OC c1(CC(=O)NC2CCCN(C(C3CCC(F)C3)=O)CC2)ccc(O)c(O)c1 C(C1(C)OCCc2sccc21)NC(c1cc(C)cc(OC)c1O)=O CCCC(CC)CCC(=O)NCC1CCN(C(c2cn(C3CC3)nn2)=O)C1 Cc1nc2nccc(N3CCCC3CNC(=O)CC3(O)CCOC3)n2n1 c1(C(N2CC3C(CNC(=O)CC4OCCO4)(C3)C2)=O)ccc(O)c2ccccc12 C1(NC(c2cc(CCO)on2)=O)CCCC(NC(c2scnc2C(F)(F)F)=O)C1 Cc1cc(CN2CCCC2CNC(=O)C=Cc2ccccc2)cnc1F N1(C(CC(C=C)CC)=O)CC2CCC(C1)N2C(=O)CCCCCF C1(CC#C)CCCN(C(C2CCN(C(C3(N(C)C)CC3)=O)CC2)=O)C1 c1(C(=O)NC2CC(NC(C3CCC4CC34)=O)CC2O)cc2n(n1)CCCC2 C1(CC)CN(C(=O)C=CC2CC2)CCC1NC(C1(CN(C)C)CCCC1)=O C#CCC(CC#C)C(=O)N1CCC(NC(C2(C#N)CCC2)=O)C(c2ccccc2)C1 Cc1ccc(O)c(NC(C2CC3CC3N2Cc2ccc(Cl)nc2Cl)=O)n1 Cc1ocnc1C(=O)N(c1nc(C(=O)O)cs1)CCc1cn(CC(C)(C)C)nn1 Cc1ccc(C=CC(N2CC(O)CC2CCc2cccs2)=O)cc1 c1(NC(CCOc2cccc(C(C)C)c2)=O)cc(F)c(O)c(Cl)c1 CC1(CNC(=O)CC=C(Cl)Cl)CCCN1C(=O)COC1CC1 c1(OC)cc(C)cc(C(=O)NCCC2CN(C(=O)C(C)NC(C)=O)C2)c1O C(=O)(C1=CCCC1(C)C)N1CC(CCC)N(C(=O)C(F)C2CCC2)CC1 C12(CNC(CCCOCCC)=O)CCC(CC1)N2C(c1ocnc1C)=O C12(NC(Cc3ccc(OC)c(O)c3)=O)CCCC1CN(C(=O)CN1CC(C)C1)C2 C1(NC(CN(C(COC)=O)C)=O)CC(F)CN(C(C2(C)CCC(=O)NC2)=O)C1 C(=O)(C(C)(C)CC(C)C)NC1C(CNC(c2c(C)nc(C3CCOC3)s2)=O)C1 C(CCCC(=O)NC1CCCCN1C(=O)CCCN(C)C(C)=O)N(C)CC Cc1nc(-c2ccco2)ccc1C(N1CC(NC(=O)CC2CC2)CC(O)C1)=O N1(CNC(C(CNC(C)=O)(C)C)=O)CCCN(C(C2CC2C2(C)COC2)=O)CC1 N1(C(CC2CC(C)C2)=O)CCC=CC1NC(c1ccc(N2CCCC2)cc1)=O c1(OC)ccc(CCC(N2CCN(C(=O)C(N3CCOC3=O)C)CC2)=O)cc1Br Cc1c(C(=O)N(C(C)CCNC(C2CC2c2cccnc2)=O)C)cnn1C1CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(CNC(C(C(C)C)NC(N)=O)=O)N(C)CC1 N1(C(c2ccc(CO)cc2)=O)CC(CO)C2(C1)CN(C(C1CC3(CC3)C1)=O)C2 C(C(Cc1ccccc1)N=c1[nH]c2c(c(=NCC3CC(F)C3)[nH]1)CCCC2)OC C1(NC(c2coc(-c3ccccc3Cl)n2)=O)CC2CC1N(C(c1csnn1)=O)C2 c1(CC)nc(C)cc(=NC2CC3CN(C(=O)C(C)CSC(F)(F)F)CC23)[nH]1 c1(C(N2C(C)C(NC(=O)C=Cc3cccs3)CCC2)=O)cc(F)cc(N)c1N c1(CC)ccc(C)c(NC(=O)C(CN=[N+]=[N-])NC(c2n[nH]c(C)c2O)=O)c1 CCC(C)(COC)C(=O)NC1CN(C(=O)C=Cc2cncs2)CC1c1nccn1C N1(C(C(CC)SC)=O)CC(CNC(=O)C(=O)NCC2CC2)C2(CCC2)C1 C1(NC(c2[nH]cc(C)c2)=O)CC(NC(c2occc2C2CC2)=O)C(O)C1 c1(CNC(C2(NC(COCCCCC)=O)CC2(C)C)=O)cccc(CO)n1 N1(C(Cc2c(C)con2)=O)CCN2CCN(C(=O)C=Cc3cn(C)nn3)CC2C1 C1(NC(C(c2cccc(F)c2)(C)C)=O)CCCC12CN(C(=O)CC1C=CCC1)C2 c1(C(=O)NC(CC=C)C)cc(CNC(C2CC(C(C)C)C2)=O)ccn1 c1(C(CNC(C(C2CC2)SC)=O)NC(c2coc(Cl)n2)=O)ccc(F)cc1 C1(C(N2C(COC)CCCCCC2)=O)CN(C(=O)CC(C)(C)C(C)=O)CC1C1CC1 C#CCN(OC)C(=O)CCNC(c1cnc(N)cn1)=O C(CCC(O)C(=O)N(C1CC2CCC1O2)C)NC(c1n[nH]c(C)c1Cl)=O C(=O)(CC(C)C(F)(F)F)N1CCC(C(N(C(C)CC2CC2)C)=O)(CF)C1 C1(CC=C)(C(=O)NCC23CC2CN(C(=O)Cc2ccn(C)n2)C3)CCOCC1 N1(C(C(CCSC)O)=O)CCN(C(=O)C(C)(C)CO)CC1CF CC1C(NC(C2(C3CCOCC3)CC2)=O)CC2CCC1N2C(=O)CC1CC(=O)C1 C1(NC(c2ccc(CC)s2)=O)CN(C(c2cc3sccc3s2)=O)CCC1F Cc1cc(C(=O)NCC(C)CC(=O)NCCC2COCC2O)n(C)n1 CC1C(CC(F)(F)F)CC(C)N1Cc1ccccc1C(=O)N(C)Cc1cccs1 CCC(C)CCCCC(=O)N1CC2CC1CN(C(=O)CC1CC=CC1)C2 N1(C(CCCC)=O)CC(NC(=O)C(c2ccc(OC)cn2)(F)F)CC12CCOC2 CC1CN(C(C2CCSC2)=O)CC1(C)CNC(=O)CCOc1ccc(Cl)cc1 C1(NC(c2cnc(SC)[nH]2)=O)CC(NC(c2ccnc(O)c2)=O)C12CCC2 C1(NC(CCC(C)SC)=O)CN(C(c2cccc(Cl)c2F)=O)CC2CCCC12 Cc1cnc(C(=O)O)cc1Cl.C(=O)(CC(C(F)F)C(F)(F)F)NCCC1CC1 c1(COC)cccc(-c2cnc(NC(c3c(C)ccnc3Cl)=O)s2)c1F c1(N(CC(=C)C)C)nc2cc(Cl)c(S(=O)(=O)N3CCCC(C#N)C3)cc2s1 Cc1cccc(C2CC2C(=O)NC2C3CC2N(C(=O)CC2CCCC2(F)F)C3)c1 C1(C(N(C2CCN(C(c3cn(CC)cn3)=O)C2)CCC)=O)CC(=O)N(C(C)C)C1 c1(C(=O)NCCC2(NC(CCc3cnc(C)s3)=O)CCC2)ccc2nncn2c1 C1(C#N)(C(N(C)CCOCCNC(=O)C(C)(C)c2ccccn2)=O)CC1(C)C C1(C(N(CCC)CCN(C)C)=O)C2CCC(C2)N1C(=O)C(C)SC N1(C(CN(C)Cc2cccn2C)=O)CCCC1CN(C)C N1(C(C(C)OCC)=O)CCN(C(c2csc(C(F)F)n2)=O)CC1CS(C)(=O)=O C1(NC(COCCCCCC)=O)CCCC(CNC(=O)CSCCCC)C1 c1(C(N2CCC(NC(C(C)(C3CCOCC3)OC)=O)C2)=O)c(C)cc(=O)oc1C Cc1nc(O)nc(O)c1CCC(N1CC(NC(c2cnco2)=O)C(O)C1)=O N1(C(=O)CCC2OCCO2)CCCCC1C1(NC(=O)CC2(O)CCOC2)CC1 c1(C(=O)NC23CCC(CNC(c4c(C)csc4)=O)(OC2)C3)ccc(S(C)(=O)=O)s1 C1(C(=O)NCCN(C)C(c2cncn2C2CC2)=O)OC(C)(C)OC1(C)C CC(C)CC(C)CC(=O)N1CCC=C(C(=O)N2CCOCC(C)(C)C2)C1 C(=O)(CCCC(=O)N(CC(C)CNC(=O)CCc1ccncc1)C)N(CC)CC C(=O)(C(C(C)CC(C)C)N1CC2CCOC2C1)NC c1(C(=O)NC2CCC(C(=O)NC3CCNC3=O)OC2)cccc([N+](=O)[O-])c1Br N1(C(Cn2c(C)ncc2)=O)CCCC(CNC(c2cc(F)nc(F)c2)=O)CC1 C12(CNC(c3ccncc3)C3CCCCC3)COCC(C1)C2 c1(C(N2CCOCC(NC(C(CC=CCC)C)=O)C2)=O)ccc(OC)c(Cl)c1F N1(C(CSC)=O)CC2CCCCC2(CNC(c2cc(Cl)ccc2O)=O)C1 N1(C(C2(NC(c3c(C)occ3)=O)CCSC2)=O)CCc2nnnn2CC1 Cc1nc(=NC(=O)C2CC2NC(c2c(Cl)cnc(Cl)c2Cl)=O)s[nH]1 c1(NC(C(C)n2cccn2)=O)ccc(NC(C2CNC(=O)C2)=O)cc1F C1(NC(CC=C(C)C)=O)CCC(NC(c2ccnn2C(F)F)=O)CC1 N1(C(CN(C(=O)OCC)C)=O)CCC2(CCCC2NC(=O)CCC(C)(C)C)C1 C12(CNC(C(N3C(C)CCC3C)C)=O)CCC(CN(C(=O)CCC(N)=O)C1)C2 N1(C(c2c(C)ccc(C)c2O)=O)CC(C)CN(C(=O)C(C)O)C(C)C1 C(=O)(C(F)(CNC(c1cnn[nH]1)=O)C(C)C)N(CCC)CCO C1(C(=O)NCCC(=C)CNC(=O)CCC)CCc2cnn(C)c2C1 c1(C(N2C3C(C(N4C(C#N)CCCC4)=O)C(C3)C2)=O)ccc2sncc2c1 C(=O)(C(C)(C)CO)N1CCC(NC(C=C(C)C(C)(C)C)=O)C1 C1(C(=O)NCC(C)CC2CCCC2)(CC)CN(C(=O)Cc2nocc2C)C1 N1(C(c2c(CC)ncs2)=O)CCC2(CC2)CC1C(=O)NC(C)CCCO Cc1nc2c(o1)CCN(C(C1CCN(C(=O)COC3CCC3)CC1)=O)C2 C1(C(=O)NC(C)Cn2cnnc2)CC(N=[N+]=[N-])CN1C(=O)CCn1cncn1 C(C(C)(C)C(=O)NC1CN(C(C2CC23CCC3)=O)CC1c1cnn(C)c1)N(C)C c1(C(N2C(CN(C)C(C3CCCC3)=O)CCCC2)=O)cnn2c1CCCC2 C(c1cccc(F)c1)=CC(=O)NCC1CCC(NC(Cc2n(C)ncc2N)=O)C1 Cc1cc(C(N2CCC(CF)(NC(=O)CCC3CCC(=O)N3)C2)=O)nnc1C C1(C(=O)NC2CCN(C(CCCC)=O)C23CC3)OC2CCCCC2C1C c1(C(N(CC(CNC(CCN(CCC)C)=O)O)C)=O)nc(Cl)c(Cl)s1 O=C1CCC(C(=O)NCC(CNC(C2CCCCC23CCC3)=O)C(F)(F)F)=NN1 c1(OC)cccc(NC(=O)C(c2occc2C)N2CCC(C)C2)c1 c1(NC(C2(C3N(C(C(F)=C(C)C)=O)CCC3)CC2)=O)cccc(C#N)c1 c1(OC)cccc(CC(N2CCC(C)(CCNC(=O)C=CSC)C2)=O)c1F c1(N(C)CCO)ccc(S(=O)(=O)NCc2ccc(C(C)(C)O)cc2)cc1F C(CC(=O)C(C)(C)C)c1cn(C(C(=O)N(C(CCCC)C)CCO)C)nn1 C1(C(N(C(C=C)C)C)=O)CC(NC(=O)Cn2ccnc2C)C1(C)C c1(CN(CC(=O)N(CCOC)C(C)=O)C)ccnn1CC1CCOC1 c1(C(N2CCCN(C(c3cc(C)ncc3)=O)CC2C)=O)ccc2c(c1)nnn2C S(=O)(=O)(c1ccc(NCC2CCCCCC2)c(Br)c1)NC(CC(=C)C)CO N1(C(C(C(C)C)SCC)=O)CCC2CN(C(c3cc(C)c(N)cn3)=O)C2C1 C(=O)(C1=NOC(c2ccccc2)C1)N(CC(C)NC(c1ccc(COC)o1)=O)C C(CCCCC(=O)NC1CC2CC1N(C(=O)C(C)N=[N+]=[N-])C2)OC CCCC(C(=O)NCc1ccnn1CC)NC(C)=O.C1(CCOCCO)C(=O)N1 c1(CC)c(C(=O)NCC(C(C)C)NC(C2CC(=C(F)F)C2)=O)cccc1F C12(CCC(=O)N(CC(C)C)C(C3CCCC3O)=O)COC(C(F)(F)F)(C1)C2 O=C1COC(CNC(C2(CNC(=O)CC3CCCCO3)CC2)=O)CN1 c1(C(N2CC(C(C(=O)N(CCCCCO)C)OC)C2)=O)cccc(C)c1F Cc1c(NCC(c2nccs2)C)ncnc1N1CCC(OCC(F)(F)F)CC1 c1(N2CC=C(CCNC(C3(C)CC3(F)Cl)=O)CC2)ncc(Br)cc1[N+](=O)[O-] C(=O)(CC(C)(C)CC(F)(F)F)N1CC(CC(C)NC(=O)Cn2ccc(O)nc2=O)C1 C1(C(N(CCCC)CCO)=O)(NC(=O)Cc2cn[nH]c2)CCSC1 C1(C(=O)NCC(C)NC(C2(CC=C)CC2)=O)CCC2C(C1)C2(F)F C12(NC(C(=O)NC(C)C)=O)COC(C1)C(NC(C1CC1(Cl)Cl)=O)C2 N1(C(=O)CCc2ccncn2)CCCC2(CNC(=O)C(F)(F)C(F)F)CCCC12 N1(C(c2c(C)c(N)cnc2)=O)CCC2CCN(C(=O)C(O)C(C)C)C2C1 Cc1[nH]c(C#N)cc1C(=O)NCC(CC(N1CCOCC(O)C1)=O)C1CCC1 N1(C(C(CCC)C(C)C)=O)CCC2(CCCN2C(c2cc(C)c(C)nn2)=O)C1 Cc1c(C(=O)NCC2CN(C(=O)C(F)C(C)C)CC2(C)C)sc2cncn12 N1(C(c2c(C)cnnc2)=O)CCC(NC(C2CC(N(C)C)C2)=O)C(O)C1 c1(C(N(CCCCNC(c2c(COC)ccs2)=O)C)=O)nc(O)nc(O)c1F c12cccc(c1)C(CO)N(C)CC(=O)C2.c1(CC)n[nH]c(C)n1 N1(C(CCSC)=O)CC2CCCC2(CNC(=O)CCc2ccccc2C#N)C1 CC1(CNC(C2CCC3(CC2)CC3)=O)CCCN(C(=O)COC(F)(F)F)C1 c1(C(=O)NCCC(C)NC(=O)C=Cc2ccc(Cl)s2)ccn2ccnc2n1 c1(C(=O)NCC(C(C)C)NC(C2(CCOC)CC2)=O)ccc(N)c(C(F)(F)F)c1 C1(C(=O)OC)C(O)CCN1C(=O)CC1(NC(=O)CC2CCCC3CC23)CC1 C(CC(C)C)(C(=O)NC1CC(=O)NC1=O)NC(c1c(C)cccn1)=O C(CO)(C(=O)N(CC(C)(C)C)C)OC.C12CCCN1C(=O)CCOC21CC1 C1(CNC(C2CCC(CC)CC2)=O)CC2(CC2)CN1C(=O)Cc1cnoc1 C(C(C(=O)NNC(=O)c1ccccc1)N(C)C)NC(=O)OC N1(C(CN(C(=O)C(CC)C(=O)OCC)CC#C)=O)CC(O)(C2CC2)C1 c1(SC)c(C(=O)NC2CN(C(=O)CCCc3nncn3C)CC2C)cccc1F C1(N(C)C)(CNC(C2CC2CN(C(C2CCC2C)=O)C2CC2)=O)CCCC1 CC12CN(C(=O)CCN3CCOCC3)CC1CN(C(C1CC13CCSCC3)=O)C2 C(CCC(=O)NCC(C)NC(c1[nH]ccc1-c1ccccc1)=O)OC(C)C CCC(CC)(CO)C(=O)N(C1CCN(C(c2cn(CCO)nn2)=O)CC1)C C(=O)(CS(=O)(=O)C(C)C)NC(C1CCN(C(c2c(C#N)cnn2C)=O)CC1)C c1(C(=O)NCC2CN(C(c3[nH]n(C)c(=O)n3)=O)C3C2C3)ccc(F)c(CO)c1 C(C)(C(=O)N(CC1CC1)OC)N(C(c1n[nH]c(CC)c1C)=O)C c1(OC)ccc2ncccc2c1C(=O)NCC1CC1CNC(c1csc(O)n1)=O C1(C(N(CC(C)NC(=O)C(N2CCCC2)C2CC2)C)=O)CCN(CCF)CC1 C(CCC(N)=O)(C(=O)NC1CN(C(C2CC23CC(O)C3)=O)CC1OC)NC(C)=O C(=O)(C(CC)CC)NC(CNC(CC=CCC)=O)C(C)C c1(C(=O)NC2(CCNC(CNS(CC)(=O)=O)=O)CC2)ccc2c(c1)nc(C)n2C c1(C(=O)NC2C(NC(C3C(C=C)OCC3)=O)C2)cc(C(F)F)ccc1OC C(c1ccc(F)cc1)=CC(N1C(C(=O)NCCc2cccc(C)c2)CCC1)=O C(=O)(C1=CCCOC1)NCC(C)(CNC(C1CC(C)(C)CO1)=O)OC CCC1=C(C(=O)OC)C(c2ccnn2CC(F)F)NC(=O)N1CC1CCC1 C(C)(CC(=O)N1CCC(CCNC(C2CC(C)(C)C2)=O)C1)(C1CCC1)N(C)C C1(CC(=O)O)COCCN(C(C2(CSc3ccccc3)CCCN2)=O)C1 CP(C)(=O)C(O)C(=O)NCCc1ocnc1CNC(C1C=CCC1)=O c1(C(N2CCC(C(C(=O)Nc3cccc(COC)c3)F)C2)=O)cc(C)cc(O)c1 C1(N2CCC(OCCOCC)C2)CCNC1=O.c1(N(CC(C)C)C)ccccc1 N1(C(C=CC(C)NC(=O)NC2C=CCS2)=O)CC(N(C)C)C1 c1(C(=O)NCCCCNC(C(C)OCC)=O)cccc(C)c1O C1(NC(CN2CC(C)C2)=O)C=CC(CNC(C2CC2c2cnn(C)c2)=O)C1 c1(OC)cccc(CC(N2CC(NC(=O)CC3CCC(=O)C3)CC2C)=O)c1 C1(CN)CCCC2(CC(C(=O)N(c3c(O)cc(F)cc3F)CCN)C2)O1 C1(CCNC(CCn2c(C)ncc2)=O)C(C)CCCN1C(=O)CC(C)(C)F N1(C(C2C(CCC)C2)=O)CC(CNC(C2(c3cncnc3)CCCC2)=O)C(C)C1 CC1(C)CCC=C(C(=O)NCC2(F)CCN(C(c3ccc(O)c(F)c3)=O)C2)C1 c1(NC(C2CCCN2C(c2cc(I)ccc2F)=O)=O)cc(Cl)ccc1O c1(C(=O)NCC)cccc(NC(=O)NCCc2nnc(S)n2C)c1 C1(CNC(c2cccn(O)c2=O)=O)CC2(CC2)CN1C(C1CC1CO)=O c1(CN(C(c2n(C)ncc2I)=O)Cc2ccccc2)c(F)cncc1Cl CC(C)(CN=c1[nH]c(=NCC2CCCC(F)(F)C2)[nH]c2c1CCC2)CC(F)(F)F c1(CC(=O)NCCC(C)NC(C(c2cc(C)sc2)(F)F)=O)nc(F)c(F)cc1F c1(OC)cccc(C(=O)NC(CNC(C2CC2c2cnc[nH]2)=O)C2CCC2)c1 C1(C(=O)N(c2cccc(OC(F)(F)F)c2)Cc2cscn2)CC(=O)C1C1CCC1 C(c1cc(Cl)ccc1Br)=CC(=O)Nc1ccc(OC)c(-n2cccc2)c1 CN1CC2CC1(CN(C(=O)C(Cl)Cl)C1CCCC1)C2 CC1(NC(C2C3COCC23)=O)CN(C(=O)C(Cl)=CCl)C1 c1(C(=O)NCCN(C(=O)CS(N)(=O)=O)CCOC)ccc(-n2cnnc2)cc1 C1(NC(CCC(C)OC)=O)CC2CCC1C(NC(=O)C1=CCSC1)C2 c1(C(=O)NCC(C2CCOC2)NC(C2(COC)CC2)=O)cnc2snc(C)c2c1 C1(C(=O)NCCCCNC(C2CN(C(=O)OC)C2)=O)(COC)CCCCO1 N1(C(c2ccc([N+](=O)[O-])cc2Cl)C(=O)NCCSC)CCCC2(CCCO2)CC1 c1(COC)ccc(C(=O)NC2CCC(CNC(=O)Cc3nocc3C)CC2)cc1 N1(C(CSCC)=O)CCN2C(=O)C(NC(=O)CCc3ccc(F)c(F)c3)CC2C1 N1(C(C=C(CC)C)=O)CC2OCCN(C(c3oc(CO)cc3C)=O)C2C1 c1(C(N2CCCN(C(c3c(C)cno3)=O)CC2)=O)ccc(F)c2cccnc12 C1(C(=O)NC2CN(C(CC3CCC(C)CO3)=O)C2)CCc2ncccc2C1 Nc1cc(C(N2CC3CC2CN3C(C2CCc3c[nH]nc3C2)=O)=O)cc(F)c1O c1(C(=O)NC(CCNC(c2cc(OC)nc(F)c2)=O)C)ccc2nc(O)sc2c1 C=CCCCC(C(=O)N(C)C(c1cnn(C)c1)C)NC(=O)CCC(=C)Cl c1(C(=O)NCC2(COC)CCCN2C(c2csc(Cl)c2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(c2c(NS(C)(=O)=O)csc2)=O)CCC2CC(C(=O)NCCOCCO)C2C1 C12C3CC1CN(C3)C2=O.Cc1csc(=O)n1CCC(=O)N.C(=O)C=CC(C)C N1(C(C2CC=C(C)CC2)=O)CCCC(CC(N2CC(F)(F)CC2C)=O)CC1 C(=O)(C1CCc2cccnc21)N1C(CN(C(C(CCCCC)CC)=O)C)CCC1 Cc1ccc(Cl)c(C(N2CC(CNC(c3onc(Br)c3C)=O)C2)=O)c1O c1(CC(=O)NC(C2CCCN2C(c2ccc(F)o2)=O)C)ccnc(F)c1 c1(C(=O)NC(CNC(c2c(CC)c(F)ccc2)=O)C2CC2)cc(S(N)(=O)=O)cs1 C(=O)(CCS(=O)(=O)CC(C)C)NC(CC(=O)Nc1ccc(C)cc1)C(F)F C1(CNC(C2CCN(C)CC2)=O)N(C(c2n[nH]c3c2CCC3)=O)CCC1(C)C C(=O)(C#CC1CCCC1)NC1CC2CC(NC(c3occ(C)c3)=O)C1C2 N1(C(c2ccc(C(=O)OC)n2C)=O)CCCCCC1CNC(=O)C=CC1CCC1 O=C(N=c1cc[nH]c2ccccc12)NCC1CCC2(CCOCC2)O1 C1(CCNC(=O)COC2CC(F)(F)C2)CCCN(C(=O)CSc2nncs2)C1 C1(CC=C)(C(=O)NCCC2CC2C2CC2)CCN(C(=O)CC=CC)C1 c1(OC)ccccc1C(C)CN(C(=O)CCC(=O)Sc1ccccc1)C [N-]=[N+]=NC1CN(C(c2cccc3ccnn23)=O)CC1NC(C1CC1F)=O c1(C(=O)NCC(C)(C)OCCNC(C2C(C)C2C)=O)csc(-c2cn[nH]c2)n1 c1(CC(=O)NCC2CCCCC2NC(=O)CCc2cnco2)cc(F)ccc1O c1(COC)ccc(N)c(C(=O)NCCN(C(=O)C(C)CSC2CC2)C(C)C)c1 C1(CNC(c2c(C)c(CO)ccc2)=O)CC2(CCC2)CN1C(C1CCC(=O)C1)=O C(=O)(CC(O)C(Cl)(Cl)Cl)NC1(CN(C(=O)CCc2cn[nH]c2)C)CC1 N1(CC(=O)N(CCCOCCNC(C2C(COC)C2)=O)C)C(=O)NC(C)(C)C1=O N1(C(CC2(C=C)CC2)=O)CCN(C(=O)CCCC(C)=O)C(CCO)C1 c1(C(=O)NC(C)CCNC(c2cc3c(s2)CCCC3)=O)cccn2[nH]c(=N)nc12 c1(C(=O)NC(CC=C)CNC(c2ccc(C#N)cc2)=O)nc2cnccc2s1 C1(C(=O)NCC(COC)C(C)C)C2CCCC2CN1C(=O)C=C(C)C(F)F C=C=CC(C)C(=O)NC(C1(C)CCCN1CC)=O C1(N(C(CCC=C)=O)C)CCC(NC(c2cn(C)c(C(F)F)n2)=O)CC1 C1(CNC(c2c(C)noc2)=O)(CO)CCN(C(c2cc(C3CC3)cs2)=O)CC1 c1(C(=O)NCC)nc(=N)[nH]cc1NC(=O)COc1ccccc1 CC(C)C(C(=O)NCC1CCC(NC(C2CCOC(=O)N2)=O)CC1)n1cncn1 C12(CCOC)CN(C(=O)CCc3ccc(Br)c(F)c3F)CC(CO)(C1)C2 C1(C(=O)NOCCN(C23CC(F)(C2)C3)C)(CC=C)CCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC(CN(C(C2CCCN2C2CC2)=O)CC)C)ccc(C#N)o1 C(C1=CCCN(C)C1)NC(C1C(CC)CCN1C(c1nonc1CC)=O)=O c1(C(N2CC3CN(S(Cc4cccc(C)c4)(=O)=O)C3C2)=O)cnc2[nH]ncc2c1 N1(C(Cc2cc(C)[nH]n2)=O)CC2(C1)SCCC2NC(C1CCn2nnnc2C1)=O c1(NC(C2C=CCN2)=O)cccc2c1C1CN(C(=O)CC3CCC3)CC1O2 c1(C(=O)NC2CN(C(C3CC(C(=O)OC)C3)=O)CC(C)C2)cnc(O)n(C)c1=O c1(C(N(C)CC2CCN(C(C3CCCCO3)=O)CC2)=O)ccnc2c1cnn2C N1(C(c2cc(C(N)=O)c(F)cc2)=O)CC2CC1CCC2NC(=O)CN1CCC1 C1(NC(C2CN(CC)C(=O)C2)=O)CC2CC(C1)N(C(c1cc(O)cs1)=O)C2 C1(C(=O)NCC=CCNC(c2c(C)cc(OC)nc2)=O)CN2CCN1CC2C C1(C(=O)NC23CC(NC(c4cn(C)[nH]c4=N)=O)(C2)C3)CC1C1CC(F)(F)C1 CN1CCn2nc(C(N3CCC(C(F)CNC(=O)CC4CC4)CC3)=O)cc2C1 C12(C(N3CC(O)(CCNC(CC4CC(CC)C4)=O)C3)=O)CC1Cc1c[nH]nc12 C1(c2n(C3C(C)CCO3)nc(C3CCCC3)n2)C2Cc3ccccc3C12 C1(CNC(C(=O)N(C)Cc2c(C)noc2C)=O)CCCC12NC(=O)NC2=O c1(NC(C)(CO)CO)cccc(C=C2CC3CCC2C3)c1 C1(CNC(c2cnc(C(C)C)[nH]2)=O)CC2(CO1)CN(C(=O)Cn1ccnn1)C2 C1(C(=O)NCCC#C)C=CCN(C(C2CCN2CC)=O)C1 N1(C(c2ccc(CN(C)C)o2)=O)CCC(NC(c2cn(C)c(O)n2)=O)C(C)(C)C1 N1(C(C(C=C)(F)F)=O)CCCC(N(C)C(c2ccn(C)c2C2CCC2)=O)CC1 CCCCCCC(C)C(=O)N1CCCC(NC(=O)COC2CCN(C)CC2)C1C c1(NC(CC2CN(C(c3scc(C)c3C)=O)C2)=O)cc(C#N)cn1C(C)(C)C C1(CN(C(CCN(C)CC)=O)C)CCN(C(=O)CC2CN(C(C)=O)C2)C1 c1(C(N2C(CN(C(Cc3ccc(C)s3)=O)C)COCC2)=O)cc(N)ccc1O C(=O)(C(O)(C(F)(F)F)C1CC1)N(C(C)CNC(c1cccnc1S)=O)C C(C(C)C(C)C(=O)NC1CC(C)(NC(=O)CC2(CN(C)C)CCCC2)C1)OC N1(C(CC=C)=O)CC(CNC(c2ccc(Cl)nc2Cl)=O)C2(CCOCC2)C1 C1(NC(c2nc(NC(C)=O)sc2)=O)C2CCN(C(=O)C=CSC)C12 c1(C(N2C(C(C)NC(CSCC#C)=O)CCC2)=O)ccc(C(F)(F)F)c(F)c1 c1(SCC)ncccc1C(=O)NCC1C(C)CCN1C(=O)Cc1nn(C)cc1Cl C12(CNC(=O)Cc3ccc(C(N)=O)cc3)CCC1CCN2C(c1csc(Cl)c1)=O c1(C(=O)NC2C(NC(=O)CCN3C(=O)CCC3=O)CC2)cc2c([nH]1)CCOC2 Cc1noc(C)c1CC(=O)NC(C1CN(C(=O)C(C(C)C)SCS(C)(=O)=O)C1)C C(=O)(C(C)CCCC)N1CCC(N(C(=O)C(C)c2ccsn2)CCCC)CC1 c1(C(=O)NCC2(F)CN(C(C=CC)=O)C2)cnc(O)c2cnccc12 C(=O)(C(C)(C)c1cnn(C)c1)N(CC(C)NC(C1C(C(=O)OC)CC1)=O)C N1(C(C2CC(C)(C(=O)OC)C2)=O)CCCC(NC(C2(N(C)C)CCCC2)=O)CC1 N1(C(COC(CC)C)=O)CCC(CCNC(C2CC(N3CCCC3)C2)=O)CC1 Cc1c[nH]nc1C(N1CC(C)(NC(=O)C(C)NS(C)(=O)=O)C1)=O Cc1c(C(=O)NCC2CCN2C(C2CCCCC(=O)C2)=O)cnc2nncn12 CC1CC=C(C(=O)NCC2(NC(=O)C(CO)N(C)C)CCCCC2)CC1 C1(C2CCN(C(=O)CCC(C)(C)O)C2)(NC(c2ccnc(CC(C)C)n2)=O)CC1 C1(NC(C=CC(=O)OC)=O)CCN(C(=O)CCC2(C)CC2)CC1C C(CC)(C(=O)NC1(C(=O)NCCSCC(C)C)CSC1)=CCCC C1(CNC(C2CC(C)OC(C)C2)=O)CCN(C(c2n[nH]cc2Cl)=O)CC1(F)F C1(CCNC(C2CN(C(C)C)C2)=O)CCCN(C(=O)CC2CSC2)CC1 c1(C(=O)NCC2(F)CCN(C(Cc3nnc(C)s3)=O)C2)cc2cccc(C)c2s1 C1(NC(C2C(NC(C3(CC=C)CCOC3)=O)CCC2)=O)CC2CCC(C1)O2 CC1CN(C(=O)CSCc2cccnc2)CCC1NC(=O)Cn1cnc(C#N)n1 N1(C(c2cc(C)nnc2O)=O)CCC2CN(C(=O)CSCCC#N)C2C1 C(C(CC1CCCC1)C(=O)NCC(CO)N(C)C)NC(C1(CCC)CC(=O)C1)=O C1(C(=O)NC2CC(NC(=O)C(c3ccc(Cl)c(Cl)c3)O)C2)CCN2CCOCC12 CCCC(C(=O)OC)C(=O)NC1CN(C(=O)C(C)(F)F)CC12CCC2 c1(C(N(CC(C)C)Cc2ncn(CC(C)C)n2)=O)cnn2c1CC(C(C)C)CC2 CC(C)CC(O)C(=O)N(CC(N1CCN(C(c2cncc(N(C)C)c2)=O)CC1)=O)C CN=c1cc(C(=O)NCC2(F)CC(NC(=O)Cc3ccc(Cl)c(F)c3)C2)cc[nH]1 c1(C(N2C(C(=O)NCC(CCCC)O)C=CCC2)=O)cnc(C)c(C)c1 N1(C(C(C)(CO)NC(=O)CN2CCOCC2=O)=O)CC(O)CC(O)C1 O=C(CCCn1cncn1)NN1CCCC1C(=O)NC1CCCCC1 Cc1cc(C(=O)NC2CN(C(C3(C(C)(C)O)CC3)=O)CC2C)n(C)n1 C12(CNC(C3CCC(CC)O3)=O)CC1CN(C(=O)C(C)NS(=O)(=O)CC)C2 N1(C(c2cc(C(N)=O)no2)=O)CC2CC(NC(=O)C3=CCCCC3)C1C2 CCCCCC(O)CC(=O)NCCOCCOC1(CF)CCC(C(F)(F)F)C1 C1(NC(C2(CC(C)C)CCOCC2)=O)COCC1S(C)(=O)=O Cc1ccc(C(=O)NC(C2CCOC2)CNC(c2c[nH]cc2Br)=O)s1 C1(C(N2C(CNC(CC3CC(OCC)C3)=O)CC2)=O)CCCN1C(=O)C(F)(F)F c1(C(=O)NC2(C#N)CCN(S(C(C)C)(=O)=O)C2)cccc2cnccc12 C1(CC=C)NC(=O)N(CCc2cc(O)cc(O)c2)C1=O c1(C(=O)NCC2C(NC(C(CC)n3cccn3)=O)C2)nn(C)c(Cl)c1Cl N1(C(C(=O)NCC2(C)CCC2)=O)CCCC#CCC1 c1(C(=O)NC(CNC(C(CN(C)C)O)=O)(C)CO)cc(=O)cc(Cl)[nH]1 Cc1cccc(CC(=O)NC2CCC(CNC(C34CC(C)(CCO3)C4)=O)C2)c1Cl C1(F)(C(=O)NC2CCC(NC(CC(CC)(F)F)=O)CC2)CS(=O)(=O)CC12COC2 c1(CN2CC3N(C(C4CC(O)C4)=O)C3C2)ccc2ncoc2c1 c1(C(=O)NCCC2CCCN(C(C3C(C=C)CC3)=O)C2)ccc2c(c1O)CCC2 C1(CC)CCCCC1C(=O)NCC1(CNC(=O)CNc2cnn(C)c2)CCC1 C1(NC(C=CC)=O)CN(C(=O)NC(Cc2nn[nH]n2)C2CC2)C1 c1(CC)[nH]nc(Cl)c1C(=O)NCC1CN(C(=O)CCn2c(C)csc2=O)C1 c1(CC(=O)O)ccc2c(c1)N(C(C1SC3C=CC1CC3)=O)CCC2 C1(NC(CN(C2CC2)CC)=O)CCN(C(=O)CCS(N)(=O)=O)CC1O C(CN=C(NCC1CCCSC1)NCC(C)(O)c1ccco1)OC Cc1nc2ccc(F)c(CN3CCC(CC(=O)N(C)CCO)C3)c2[nH]1 CC1CCCC(C)CN1C(=O)CCC1CCC(NC(=O)C2=CCCCCC2)C1 C(=O)(C(C)(C)CCNC(=O)C1=CCCC1)N(CC)Cc1cccs1 Fc1ccc(CNCc2ccccc2)cn1.OCC c1(N2CCC(N(CCC)C(C3(C)CCC3)=O)C2)nc2cccnc2s1 C(C(CCNC(c1cnc(C)[nH]1)=O)OC)NC(C1(CSC)CC1)=O C(C)(CO)(C(=O)NCCCN(C(=O)CCCc1cc(C)no1)CCO)NC(C)=O C1(C)(C(N2CC(NC(=O)OC)C2)=O)CCN(C(c2c(C)ncn2O)=O)C1 CCC(F)(F)C(C)(C)C(=O)NC1CN(C(c2cc(CF)on2)=O)CC1F C(C)(C)(CCC(=O)N(C(C)CNC(c1cn(C2CCOC2)nn1)=O)C)OC CCC(C(=O)N1CCCCC1CCNC(C1CCCC1OC)=O)C(C)O C1(NC(C(C)P(C)(C)=O)=O)CN(C(=O)COc2ccc(F)cc2Cl)CC1C1CC1 C#CCC(C)C(=O)N(CCCNC(=O)C(C)NC(C1CCOCC1)=O)C(C)C C(=O)(C1=C(C)OCC1)NCC1CC(CNC(CC=C)=O)OC1 C(=O)(CC1=CCCCC1)NC1CC(C(C(=O)N(CC(CC)CC)CC)F)C1 C(=O)(C(C)(C)CNC(N)=O)NC(C1CCN(C(c2ccnc(O)c2)=O)C1)C N1(NC(=O)NC(C(=C)C)C(N2CCc3sccc3C2)=O)CC(=O)N(C)C(=O)C1 C=CCCC(C)(C)C(=O)NCC1CCC1NC(=O)C(c1ccccc1)SC c1(CCNC(C2C(C(C)NC(C(C)=CC(C)(C)C)=O)C2)=O)ncccn1 Cc1nn(C)c(Cl)c1CC(=O)N(CC(O)CN(C)C(C1OCC1(C)C)=O)C C(=O)(C1=C(C)C(C)(C)OC1=O)NCC(CC)NC(COC1(C#C)COC1)=O C(=O)(C1CCCn2ncnc21)NCCN1CCN(c2ncc(C#C)cn2)CC1 N1(C(C=CC=CCC)=O)CCCC(C2(NC(c3nc(CC)ncc3Cl)=O)CC2)C1 NC(=O)C(CCC(F)F)NC(=O)Cn1c(=O)oc2ccccc12 C(N=c1[nH]cnc2c1COC2)C1CN(C(CC2CCC(C)C2)=O)CC1C CC(C)(CCC(=O)N1CC(NC(C2(C)CCCCO2)=O)C(C2CC2)C1)[N+](=O)[O-] C#CC1(C)CCCN(C(=O)CCN(C(c2cc(Cl)ns2)=O)C2CC2)C1 N1(C(C(C)=C2CC2)=O)CCC(C2CC2)(CNC(c2ccnc(Cl)c2)=O)C1 c1(C(=O)NCCN(CCC)C(C2CCCC2C)=O)n[nH]c2c1COC2 CC1CCN(C(c2cccc(Cl)c2)C(=O)NCc2ccccc2)CC1O c1(C(N2CC(CNC(c3c(C)snn3)=O)C2)=O)coc2cc(F)ccc12 CC1CCC(C(=O)NCC2CN(C(C)C)C2)CN1C(=O)CCc1ccc(F)nc1 C#Cc1ccc(C(N2CCC(C)CC2C(=O)NC(C)COCC)=O)cc1 C1(NC(C(CO)N(C)C)=O)CCCN(C(c2cnc(-c3ccccc3)nc2)=O)C1 c1(C(=O)NCCC(CNC(CC2C(CC)C2)=O)O)cc(C#N)c[nH]1 C#CC1(C(=O)Nc2cnc(O)c(C)c2)CCN(C(c2ccn(C)c2)=O)C1 C1(C(=O)NCCCN(C(C2(CSC)CC(F)(F)C2)=O)C)CC2(COCCO2)C1 N1(C(C(=O)OCC2CC=CC(C)=NC2)=O)CCC2(NC(=O)OCC)CCCC12 Cc1c(C(=O)N(C(C)CCNC(=O)CNC(C2CCC2)=O)C)ccn1CC1CC1 O(N=C1CCCCCC1)CC(=O)NCCC1CC(NC(=O)COC2CC=CC2)C1 C1(C(N(CCCNC(=O)CCC2CCCCO2)C)=O)CCCC1(F)F N1(C(CCOCC)=O)CCC2CN(C(c3cnn(C)c3C#N)=O)C2C1 c1(C(N2CC(OC)C(NC(=O)C(C)C(F)(F)F)C2)=O)ccc2oc(=O)oc2c1 c1(OC)cc(CN2CCN(C(=O)Cc3nc(C)sc3C)CC2)ccc1C(F)(F)F c1(C(=O)NCC2C(NC(c3ccc(C)cc3)=O)CCC2)ccc2c(n1)NCC2 C(=O)(C1=C(C)OCC1)N(C1C2CN(C(C3C(CC)OCC3)=O)CC21)C S(=O)(=O)(c1cc(C)cnc1NCc1csc(COC2(CF)CCC2)n1)N(C)CC C1(C2CC2)(CNC(c2cc(C)n(C)c2)=O)CCN(C(=O)CC2(O)CCC2)C1 C1(C(=O)NCc2cc(CC)on2)N(C(=O)CN2CCSCC2)CCCC1(C)C Cc1c(NC(c2ccnc(-c3ncc[nH]3)c2)=O)ncc2c1CCOC2 CCC(CC(=O)NCC1CN(C(=O)CCOC2CCOCC2)CCCO1)C(C)C N=c1[nH]c2c(s1)CC(NC(=O)Cc1cc(C(F)(F)F)cc(Cl)c1)CC2 c1(C(=O)NC(CC(C)NC(c2c(C)ccn2C)=O)C)cc2c(nc1O)CCSC2 N(C(=NCCC(C)(F)F)NCc1ccc(C(C)C)cc1)C(COC)C C(C)(C)(CCCNC(C1CCS(=O)(=O)C1)=O)NC(C=C(C)C(C)(C)C)=O C(=O)(C1=CCCC1)N(CCCOCCN(C)C(c1cnn(C)n1)=O)C N1(C(C2CC(=C)C2)=O)CC2CCCC2(NC(c2csc(CO)n2)=O)C1 CC(C)(F)CCC(=O)N1CC(NC(=O)Cc2cc(Cl)cs2)C2(CC2)C1 C(=O)(N=c1cc(-c2cccc(F)c2)[nH][nH]1)C1SCCN(C(CC)=O)CC1 N1(C(c2cnc(OC)s2)=O)CC2CCOC2(CNC(c2cc(Cl)nnc2O)=O)C1 CC#CCCC(=O)N1CCC(N(CC(C)C)C(C2COCCO2)=O)CC1 c1(C(N(C)C)=O)cc(NC(=O)NCCC(C(F)F)c2ccccc2)ccn1 c1(C(=O)NC(CNC(C2C(CC)C2)=O)(C)C2CCC2)c(C)nn(CCOC)c1Cl C#CCC(CC#C)C(=O)N1CCOCC1(C)c1cn(CCOC2CCOC2)nn1 c1(C(=O)NC2CC(c3ccccc3)(CNC(C3C(C)C3)=O)C2)cc(F)c(F)cc1N C12(CN3C(CCC)CN(C(c4cc(C)oc4C)=O)CC3)CC1COC21CCC1 C1(C(=O)NC2CC3(C(NC(=O)OC(C)(C)C)C3)C2)(CC2CC2)CCS(=O)(=O)CC1 c1(C(C)C)cc2c(NC3CCCC3NC(c3c(Cl)nsc3Cl)=O)ncnc2s1 c1(C(=O)NCCC2CCN(C(=O)CCCC3CC3)C2)cnc2scnc2c1 C1(CC)CC(C(=O)NC(C)CCCNC(=O)CSS(C)(=O)=O)CCO1 N1(C(c2cc(CCC)c(C)s2)=O)CC2CCCC2(NC(c2ccncn2)=O)C1 c1(CN(C(=O)CN(CCc2ccc(F)cc2)C(C)C)CC#C)cc(C)ccc1C N1(C(c2ccc(CC)s2)=O)CCN(C(=O)CNC(=O)C(C)c2ccsc2)CC1.C1CC1 N1(C(C2(C)CCC2)=O)CCCC(CO)(NC(=O)Cn2cnnc2O)C1 C1(NC(C(C)Sc2ccccn2)=O)CN(c2cc(Cl)nc(C3CC3)n2)CC1(C)C Cc1ccc(N)c(C(=O)NCC=CCNC(c2csc(-c3ncccn3)n2)=O)c1 CC1CN(C(=O)CCF)CC1NC(c1ccccc1NCc1ccsc1)=O C(=O)(C1=CCC(C)(C)CC1)NC(CCOC)C(=O)NCC1(OC)CCC(C)C1 CC1CCN(CC(=O)N(C)CCNC(C2C(c3ccccc3)C2(C)C)=O)C1 c1(OC)cc(CO)ccc1Cl.C12CCN(C1)C(=O)C1CC1CNC(=O)CN(C)C2 C1(C(=O)NC2CC(=O)N(C3CN(CCO)C3)C2)CCCC12OCCO2 N1(C(c2ccc(OCCC)cc2)C(=O)NCC)Cc2ccccc2C(CO)C1 N1(CCCC)CCC(C(=O)NCC(C)N(C(=O)CC2COCC(C)O2)C)CC1 Cc1ccc(C)c(OCC(=O)NC2CN(C(=O)CC3OCCCC3(C)C)C2)c1 c1(C(N(c2nc(OC)c(C)cn2)C2CNCC2(F)F)=O)cnc2cccnn12 CC1CC(CNC(=O)CC2OCCO2)CN1C(c1ccc(C(F)F)s1)=O C1(CN(C)C(C2CC2(C)C)=O)CN(C(C2CC2(C)C)=O)CCO1 Cc1nc2ncc(C(=O)NCC3(F)CCN(C(C4CC(C)(O)C4)=O)C3)c(=O)n2[nH]1 c1(C(N2C(C)CN(C(=O)Cc3ccn(C(F)F)n3)CC2)=O)cc2ncccc2s1 c1(OC)cc([N+](=O)[O-])c(NC(C2CC(NC(c3nc(C)cs3)=O)C2)=O)cc1C C1(C(=O)NC(C)(C)CCNC(=O)Cc2cccnc2NC)(CC)CCCCO1 c1(C(N2CC(NC(c3c(C)cco3)=O)C(F)C2)=O)cnc2ccnn2c1 N1(C(CCNC(C)C)=O)CCC2C(CCN2C(c2ccccc2Br)=O)C1 CC1(C)CC(C(=O)NC2(C3CC3)CCN(C(c3cnn4ccncc34)=O)C2)=NO1 CCCC(C(=O)N1CCC(CC(=O)NOCCN2CCOCC2)CC1)NC(C)=O n1(CCC)ccc(C(=O)NCC(O)CN(C(=O)C=CC2CCCC2)C)n1 c1(C(=O)NCC2(F)CC(NC(C(C=C=C)C)=O)C2)cccc(O)c1Br Cc1ccc(F)c(C(=O)NCC23CC(NC(=O)Cc4cncn4C)(C2)C3)c1Cl C1(NC(c2cnc(CC)[nH]2)=O)CCC(C)N(C(=O)CN(C)C(C)C)C1 c1(CC(N2CCC(N(C(=O)Cc3nnc(O)s3)CCO)C2)=O)ncccc1O C(C)(CC(=O)N(CC(C)NC(c1ccon1)=O)C)OC c1(OC)nccnc1C(=O)NCC1(O)CC(CNC(C2CCCN(C)C2)=O)C1 Cc1ncncc1C(=O)NCCCC(C)(C)NC(c1cnc(CC2CC2)s1)=O Cc1cc(C(N2CCOC(C(N3CCC(CO)C(O)C3)=O)C2)=O)c2cc[nH]c2c1 c1(C(N2C(C)CC(NC(C(C(C)C)N(C)C)=O)C2)=O)cc(S(N)(=O)=O)co1 C1(F)(CNC(c2c(CC)nc[nH]2)=O)CCCN(C(C2CC2(C)C)=O)C1 Cc1ncccc1-c1cn(Cc2noc(CCCl)n2)nn1.c1[nH]c(C)c(C)c1C N=S1(=O)CCN(C(C2Cc3cccc(F)c3O2)=O)CC12CCC2 CC1CCC(=CC(=O)NCC2(NC(=O)C=C3CCSCC3)CC2)C1 c1(C(=O)NCC(CC=C)NC(=O)Cc2[nH]cnc2C)cc2cc(C)ccc2o1 c1(C2CN(C(C(N3CCC(c4ccc(C)nc4)(O)C3)=O)=O)C2)cccc(Cl)c1F C1(c2nc(-c3scc(C)n3)nn2CC2CCOC2)Cc2ccc(C)cc2S1 C1(CNC(C2N(CC)CCCC2)=O)CC2CCCC2C1.C1(=O)N(CC)C1 N1(C(C(=O)NCCCC2N(C(c3c(C)cco3)=O)CCC2)C)C(C)CCC1C Cc1c(C(N2CCCC(N(C(=O)CC3CC(C)C3)C)C2)=O)cnn1CC(C)(C)O c1(C(=O)NCC23CC2CN(C(C2CCCSC2)=O)C3)cc2ncccc2[nH]1 c1(C(=O)NCCOC2CCN(C(Cc3c(C)noc3)=O)CC2)cc2occc2[nH]1 c1(C(=O)NCC(CNC(c2cccc(C)n2)=O)(C)C)cc(S(N)(=O)=O)cs1 CC1(C)CCC=C1C(=O)NC12CCCC1CN(C(=O)Cn1nnnc1C1CC1)C2 c1(C(=O)NC2C(NC(C(c3scc(C)n3)C)=O)C2)cnc2ncnn2c1C Cc1cc(C(N2CC(NC(c3cscc3F)=O)C(C)C2)=O)c2cc(F)ccc2n1 C1(CNC(C2C(OC)CCCC2)=O)CCN(C(=O)C(c2csc(C)n2)=O)CC1O CC1CC(CNC(=O)CNC(c2ccccc2F)=O)CN1C(=O)C(F)C1CCC1 C1(C(=O)NCCCN(C(c2ccc(C=C)cc2)=O)C)CCC2CCC(=O)N12 c1(C(N)=O)nc(-c2ccccc2)n2c1COCC2.c12ccc(cc1)NC(=O)C2 n1(CC)ncc(CNC(=O)C=CC(C)NC(=O)CC(C)F)c1C c1(C(=O)NCC(CNC(C2NC(=O)OC2C)=O)OC)[nH]nc([N+](=O)[O-])c1Cl C1(OC)CCCCC1C(N1CC(CNC(=O)C(=O)N(C)C)CC1C)=O C12(C(N(CC(=O)NOCC(=O)N(C)C)C(C)C)=O)CC(C)(CCO1)C2 c1(C(N(CC(C)N(C(C2C(C=C)CC2)=O)C)C)=O)cc(C#N)cn1C C(=O)(C1=CCN(C(=O)CSC2CC2)CC1)NCCn1c(C)nnc1 c1(C(=O)NCC23COC(C(F)(F)F)(C2)C3)cccc2cc[nH]c12.C12CC(C1)CN2 c1(CC)ccc(C(=O)NCC2CCN2C(C2CCSCC2)=O)c(C)c1 N(C)(S(=O)(=O)N(C)C)CC(N1CCC(N(CCOC)C(c2ccoc2Cl)=O)CC1)=O c1(C(N2CC(O)(C(C(=O)NC(CCO)C3CC3)F)C2)=O)ncc2ccccn12 C1(C(=O)NC(C(C)NC(COCC)=O)(C)C)CCc2ccc(Br)cc2O1 C12CCCC13CCCN(C3)C2.c1(COC)cccc(NC(=O)C2CC2)c1 c1(SCC)cccnc1C(=O)NCC1(NC(=O)CCC2CCCN(C)C2)CC1 N1(C(c2c(CC)nc[nH]2)=O)CCOCC(CNC(C2CCSC2)=O)C1 CCCC(O)C(=O)NCC1C(C)CCN1C(C1CCCCS1)=O CC1CC(NC(c2cc(-c3ccn(C)c3)[nH]n2)=O)CN(C(c2cc[nH]n2)=O)C1 C1(C(=O)NOC2C(CNC(CSCC=C)=O)C2)(CC=C)CCCC1 N1(C(Cn2cccc(N)c2=O)=O)CC2(CCN(C(C3CC3C3CCCC3)=O)C2)C1 CCCC(CC(=O)NCc1cccnc1)NC(=O)COC(C)CC O=[N+]([O-])c1cc[nH]c(=NCCc2cccs2)c1.C1(N)CCC(c2cncs2)C1 C(Cc1ccccc1)(C(=O)NCCC(O)CNC(C1(CCF)CC1)=O)NC(N)=O C(=O)(CCC(=O)C(C)(C)C)N1C(CNC(C(CC)F)=O)CC(C(F)(F)F)C1 c1(CNC(=O)COc2cccc(F)c2)c(F)cncc1F.CC12CCN(C1)C2 N1(C(CNC(C2CCC(F)(F)CC2)=O)=O)CC2CN(CC3CCC(C)CC3)C2C1 c1(C(=O)NC2CCN(C(C3CC(C)OCC3)=O)C2C)ccnc2[nH]nnc12 N12CCC(CC1)CC2=O.c1(CNC(C2(OCC)CCC2)=O)nocc1C(=O)OC C1(CC(=O)NCCC2N(C(CCCOC)=O)CCOC2)CCCCC12CC2 c1(C(C(=O)NC2(CC(=O)NC3CCN(C(C)=O)C3)CCC2)(F)F)cccc(C)n1 C(CSS(C)(=O)=O)(C(=O)NCC(C1CCC1)NC(=O)Cc1csc(C)n1)OC N1(C(CNC(C)=O)=O)CC2C(CC(=O)Nc3cncc(C(F)F)c3)C2C1 O=C1Nc2cc(Cl)ccc2C1CNC(C1CNCC12CCC2)=O C(=O)(CCCC(C)(C)C)NC(CCN(C(C=C(C)Cl)=O)C)C C=C(C)CCCC(=O)NCC1CN(C(=O)CCOc2cccnc2)C(C)(C)C1 N1(C(C=CCC)=O)CCc2ccccc2C1CCNC(c1ccncn1)=O C1(C(N(CCCNC(C2(CC=C)CC2)=O)C(C)C)=O)Cc2nccnc2C1 Cn1nc(Br)cc1Cn1cc(CCC2CCCNC2)nn1 C1(NC(=O)Cc2nncs2)CCCN(C(C2(C(F)(F)F)CC=CCO2)=O)CC1 N1(N(C)C)CSCCSC1.C12CCC1(c1nnnn1CCC1(C)CC1)N2.C(CC1CC1)O C1(NC(CCc2ccn(C)n2)=O)CCN(C(c2ccc(=O)oc2)=O)C12CCCC2 c1(C(=O)NC2CN(C(CC3CCC(C)O3)=O)C2)cc(F)c(Cl)cc1F N1(C(CCN(C)CC)=O)CCC(C)C(NC(C2CSC(C)=N2)=O)C1C N1(C(c2cc(CSC)c(C)s2)=O)CC(NC(c2cc(CO)oc2C)=O)CC(O)C1 Cc1cccn2cc(CCNC3CC4CCC3C4)nc12 c1(OC)cc(CNC2CCC(C(=O)Nc3cscn3)C2)c(Cl)cn1 c1(C(=O)Nc2ccc(C(=O)Nc3ccc(C)c(Br)c3)nc2)c(Cl)cnc(Cl)c1Cl c1(C(C(=O)NCCN(C)C(C2NC(=O)C3CC23)=O)=O)c[nH]c2ccc(F)cc12 C(=O)(C1=CC2C=CC(C1)C2)N1C(C(C)C)(C(=O)NCc2cnns2)CCC1 C(c1c(C)coc1C)=CC(N1CC2C(NC(Cn3c(C)cc(C)n3)=O)C2C1)=O C1(CCCNC(c2ccoc2Cl)=O)CCCN1C(=O)CC1COC(=O)C1 c1(C(CNC(C2CC(NC(C3(CC(C)C)CCC3)=O)C2)=O)O)cnn(C)c1 O=C(C#CC1CCOCC1)NC1CCCC1NC(c1cc(F)cc(F)c1O)=O CCCC(CC(C)C)C(=O)N(C)CC1(NC(=O)C(c2ccc(F)cc2F)C)CC1 c1(OC)cc(F)ccc1C(=O)Nc1nc(C(=O)NCC(N)=O)cs1 c1(-c2c(C(=O)Nc3cc(C(F)(F)F)[nH]n3)cccc2)cc(F)ccc1[N+](=O)[O-] C12(C(N(CC#C)CC3CCCO3)=O)CCCC1N(C(=O)CCC(C)(F)F)CC2 Cc1ccc(C(=O)N(CC(C)CNC(=O)C2=CC(C)CC2)C)c(C)n1 c1(C(C)C(=O)NCC(F)CNC(=O)Cc2nccn2C)ccc(F)cc1 CS(=O)(=O)c1ccc(C=CC(=O)NC2CN(C(C3CC34CC4(F)F)=O)C2)o1 C1(CC)CCCC(NC(N2CCN(C)C(C(C)C)C2)=O)CC1.c12ccc(cc1)s2 N1(C(c2nc(OCC)oc2)=O)CC(NC(C2CC3CC2CO3)=O)C(CC(C)(C)C)C1 CC1CCOC(C(N2CC(CNC(C3(O)CCC3)=O)C(C)C2)=O)C1 N12CCCCC1CNC(=O)C2.C1(COCCCC)CCCC1 C12(COC(C3C(OC)CCO3)=O)CC(C1)C(C)O2 N1(C(c2c(C)snc2)=O)CCC(C2CC2)C1C(=O)NC1CC2CC1CC21CC1 N1(CCNC(C2CC(NC(C3(CO)CCOCC3)=O)C2)=O)CCNC(=O)C1 [N-]=[N+]=NCCCC(=O)N1CCC2(NC(=O)CCc3ccc(Cl)c(F)c3)CC2C1 N1(C(CSC)=O)CCC(C(=O)NOCC2CC(=C3CCC3)C2)=C(F)C1 C(=O)(CCC(=O)NC(C)(C)C(C)NC(c1ccc(O)nc1)=O)N(C(C)C)C C1(C(=O)NCCCCCCNC(C(C)C(F)F)=O)Cc2nccnc2C1 c1(C(N2CCC(N(C(=O)CCCc3nccs3)C)C2)=O)nnc(O)nc1O n1(CC(c2nnnn2C)NCc2c(C)con2)cc(C(F)(F)F)ccc1=O C1(c2nccc(CC)c2)(CC)NC(=O)N(C(C)CN(C)C(C)C)C1=O C1(C)(C(N2CCC(NC(c3c(CC)n(C)nc3)=O)C(O)C2)=O)CC(C(C)C)=NO1 C1(NC(C2(C=C)CC2)=O)CCN(C(=O)CCc2c(Cl)cccc2Cl)C(C)C1 Cc1cc(C(=O)NC2CCN(Cc3ccc(F)nc3C)C2)cc(C)c1O C1(CCN(C(C(=O)N(CC(=C)C)CC)c2cn[nH]c2)C)NC(=O)NC1=O c1(C(N2CCC(CN(C)C(C3CCC(O)CC3)=O)C2)=O)ccc2nonc2c1 C(CC(=O)NNC(=O)NC1CC2(CC2)C1)c1ccc(C)s1 C(C(CC(=O)N1CC=C(CNC(=O)Cc2cc[nH]n2)CC1)C(F)(F)F)N(C)C c1(SC)ccsc1C(=O)NCCC1CCC(NC(c2ncc(C(F)F)s2)=O)C1 C#CC1CC2CCC1N(C(C1CC(C)CN1C(=O)CC1COCC1O)=O)C2 Cc1c(C(=O)NCC2CC2NC(C2(C(F)(F)F)CCC2)=O)cnc2[nH]ccc12 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)OCC(OCOC)C C(C(=O)NCC1(O)CCN(C(=O)CC2CC=CC2)C1)(C(C)C)OCC c1(C(=O)NC2CN(C(CCCCC)=O)CC2(C)C)cccc2c1C1CCC2CC1 C(C)(CC(C)(C)C)NC(C(c1cnn(C)c1)NC(Cc1cc(C)sc1)=O)=O C1(C(N(CC)CC2CC2)=O)CN(C(=O)CCc2ncc(C)[nH]2)C(C)(C)C1 C=CCC(C(=O)NC1CCCC1NC(c1[nH]c(O)nc1C)=O)OC c1(NC(C2(O)CCN(C(CC)=O)C2)=O)c(C(C)=O)cc(Cl)nc1Cl C1(C(=O)NC(C(N2C(C)(CCO)CC2)=O)(C)C2CC2)CC2(CCO1)CC2 c1(OC)ccc(C(=O)NC(C)CCCNC(=O)C(C)(C)OC)nc1 C1(CNC(C2CC(C)(C(F)F)C2)=O)CCCCCN1C(c1csc(C2CC2)n1)=O c1(CC)sc(=N)[nH]c1C(=O)N(C)CC1CCCN1C(c1ccc(CN(C)C)o1)=O c1(C(N(CCCNC(CCN(CCC)C)=O)C2CC2)=O)cnc2occc2c1 C1(CNC(c2cc(F)c(Br)cc2OC(F)F)=O)CCCC2(CCC2)C1O c1(C(CNC(c2ccccc2)=O)OCCOCCNC(C)=O)ccc(Br)cc1 c1(C(C)C)ncc(C(=O)NCC2CCCC2NC(c2coc(Cl)c2)=O)s1 c1(C(=O)NCC(CNC(c2cnc(OC)nc2C)=O)F)cccc2cnsc12 C(=O)(C(O)CC(N)=O)N1C(CN(C(c2c(C)cc(C)s2)=O)C)CCC1 c1(C(=O)NCCOCCN(C(C(C)OCCC(C)C)=O)C)cccc2ccoc12 C1(O)(C(=O)NC2CCCC2CNC(CN(C)C)=O)CCOC1(C)C.C(=O)(C1CC1)N CC(CC(=O)NCCNC1(Cc2nnn(-c3ccccc3)n2)CC1)C1CCCO1 c1(CC#N)cccc(C(=O)NCC2COCC2NC(c2ccoc2Br)=O)n1 N1(C(CC=CC(C)(C)C)=O)CCC(C)(NC(=O)Cc2ccc(O)cc2)C1 C1(c2c(C(=O)OCC)nco2)CCN(C(C2C(c3ccccc3)C2(C)C)=O)CC1 c12nccnc1C(=O)N2.C(CC(O)CO)NC(CCC1CC(OC)C1)=O C(CCC(C)(C)C(=O)N1CCc2nn[nH]c2C1)N(C(=O)CSC(F)(F)F)C C1(N(CC#C)C(C)=O)CCN(C(=O)C(C)Nn2ncnn2)CC1 C(=O)(C1=CC2(CCOC2)C1)N1CC(NC(c2ncc(C)c(C)c2)=O)C(C)C1 c1(N2CC3C(CCC)(C3)C2)ccnc2cc(Br)nn12 c1(C(=O)O)cc(S(=O)(=O)N2CCN(Cc3nccn3C)CC2)oc1Cl c1(CC(=O)NC(C(C)NC(c2c(C)nsc2)=O)C)ccc2c(c1)CCCS2(=O)=O c1(N(C2CN(C(c3cc([N+](=O)[O-])cs3)=O)C2)C)ncnc2c(Br)csc12 Cn1cnc2cc(C(N3CC(NC(=O)CC4Cc5cccnc5C4)C3)=O)cnc12 CCC(CC(F)(F)F)C(=O)NC1CC(NC(=O)C(C)(O)C(C)(C)C)C1 NS(=O)(=O)c1ccc(C(=O)NC2CCCC(NC(C34CC(CCO3)C4)=O)C2)s1 Cn1ncc(C(=O)NCC2CCCCN2C(C2CN3CCC2C3)=O)c1Cl c1(C(N(CCNC(=O)C(C)Cc2cccc(F)c2)CC)=O)ccc2n[nH]cc2c1 c1(C(=O)NCC2C(NC(c3cnc(C4CC4)nc3)=O)CC2)cc2cn[nH]c2cn1 c1(C(N(CC(CC)NC(c2ccnc(SC)c2)=O)C)=O)nc2ccccc2[nH]1 c1(C(=O)NC(CCN(C(C2C(OCC)C2)=O)C)C(C)C)cc(OC)nc(Cl)c1 c1(CNC2C=CC(C(N3CCN4CCC3CC4)=O)C2)cccc2occc12 CC1(C)C(C(N2C3CCC2CN(C(=O)C=CCF)C3)=O)CCS1(=O)=O Cc1ccc([N+](=O)[O-])cc1CN1C(=O)CCC1c1nc(C(N)=O)no1 c1(C(=O)OC)ccc(CCC(N2CC(O)(C(C)NC(=O)CCF)C2)=O)cc1 c1(OC(C)C)ccc(N)c(C(=O)NC23CC(NC(=O)Cc4csc(Cl)c4)(C2)C3)c1 C1(C(=O)NC2CC(C)(CC3CC3)C2)CN(C(=O)C(=O)NC2CC2)CC1(F)F c1(CC)ccc(F)c(C(N2CCOC(CNC(=O)CC3SC(=N)NC3=O)C2)=O)c1 C(=O)(CS(=O)(=O)c1ccccc1F)NC1CC(C)(NC(c2cccnc2O)=O)C1 c1(C(N2CCCN(C(CC(C=C)CC)=O)C(CO)C2)=O)nc2nccc(C)n2n1 c1(C(=O)NCC2(C)CC(NC(C(C#C)(C)C)=O)C2)ccc2c(c1)COC2 C1(CN(C(C(N2CCCCC2)C)=O)C)CCCCN1C(=O)CNC1CCOC1C S(=O)(=O)(c1cc(F)ccc1Cl)NC(c1cn(CCCF)nn1)C Cc1cccc(CCN(C(Cc2ccoc2)C(=O)NC(C)CCC(C)C)C)c1 N1(C(CCC)=O)CCCC(C)C1CNC(c1cc(O)ccc1OC(F)F)=O C12(CNC(C3(CC#C)CCCCC3)=O)CCC(CC1)N(C(=O)C(CCC)SC)C2 n1(C(CC(N(CC#C)CCOC)=O)OC(CC)C(=O)O)cnc2ccccc12 CC(C)S(=O)(=O)CCN=C(NCc1ccc2cc[nH]c2n1)NCCN1CCCC1 Cn1nc(C(=O)NCCC2CCCCN2C(c2c[nH]c(=N)o2)=O)cc1O c1(C(N(C(CNC(c2cc(C(C)=O)sc2)=O)C2CC2)C)=O)ncn2ccccc12 C#CCCC1=C(C(=O)OCC)C(c2c(CC)nn(C)c2OCC)NC(=S)N1CC N(C(=NCCC1CC(=O)N(C)C1)NCc1cccc(C(N)=O)c1)CC(C)C c1(OC)cc(C(=O)NC2(CO)CN(Cc3ccc(F)cc3Br)C2)ccc1I C1(C(C#C)C)CCN(C(=O)CCC2(C)CCCN2C(=O)C=CC2CCCC2)CC1 C1(C(=O)Nc2c(C)ccnc2)CN(C(c2ncccc2Cl)=O)CCN1C N(C(=NCC1(C=O)CC1)NC1CCN(CC2CCCCC2)C1)NC(C)=O.C1CC1 C1(C(=O)NCC2CCN(C(c3n[nH]c4c3CCC4)=O)C2)CCc2ncnn2C1 CC1CCC(CNC(c2cccc(C3CC3)c2)=O)CN1C(C1CC=CCC1C)=O CCCC(CCC)C(=O)N1CCCC(COC)(NC(c2cscc2CC)=O)C1 C1(N(C)C(c2cc(C3CC3)n(C)n2)=O)CCCCN(C(C2CCC(O)CC2)=O)C1 C1(NC(C2CCC(NC(CC(C)O)=O)C2)=O)(CO)CC(C)(C)C1 N1(C(CCOCC)=O)C2CCC1CC(C(=O)NCC1CCCO1)C2 Cn1cc(C(=O)NCC(F)CNC(C2CCCC(F)(F)CC2)=O)c2ccccc12 C1(CN=[N+]=[N-])CCN(C(c2cc(CNC(=O)CNc3ccccn3)[nH]n2)=O)C1 N1(C(c2c(C)ncs2)=O)CCC(NC(c2n[nH]c(=N)s2)=O)C2(CCC2)C1 CCC(CC)C(F)C(=O)NC1CC12CCN(C(=O)C(C)c1ccco1)C2 C(=O)(C1=C(C#N)CCC1)NCC1C(C)CCCN1C(=O)CN1CC(=O)N(C)C1=O C(=O)(CCCCC(=O)N1CC(CC(=O)NOCCC(F)(F)F)(OC)C1)OC CC1=CCC(C(=O)N(C2CCCCC2N(C)C(c2sccc2F)=O)C)CC1 CC1CCCCC1(CNC(=O)Cc1ccccc1)NC(=O)COC1CCCOC1 Cc1cc(Cl)ccc1OCC(=O)NCCC(C)NC(=O)C(C1CCCCC1)C C1(NC(C2(OCC)CC2)=O)CCCN(C(c2cc(Cl)n[nH]2)=O)CC1 N1(C)CC(N(C2CCCC(O)C2)C(c2c(C)[nH]c(C(=O)NC)c2C)=O)CCC1=O CC(C)CC(C(=O)NC1COCC1C(N)=O)ONC(c1cccnc1S)=O N1(C(C(C)OCc2ccc(C)cc2)=O)CCN(C(c2ocnc2C)=O)C(CF)C1 CC1(C)CC(C)(CNC(C2(CO)CCOCC2)=O)CN1C(C1CC12CC2)=O c1(C(C)C(=O)NCCCOCCNC(=O)C=Cc2cc[nH]c2)nc(F)ccc1Cl Cc1nncc(CNCC2C=CCC2)c1C C1(C(N(C)Cc2c(C)ncs2)=O)(NC(=O)C(C)c2ccco2)CCCCC1 c1(CCCC)nc(C(=O)NC(=O)CC2(O)CN(C(=O)CSC)C2)cs1 Cc1cc(C(=O)NC2(C)CCCN(C(=O)C(F)(F)c3cscn3)C2)cc(C)c1 c1(C(C(C)O)NC(=O)N(C)CCS(=O)(=O)c2ccccc2)nnc2ccccn12 C=CC(CCC)CC(=O)N1CC(CNC(c2cscc2C)=O)C(F)(F)C1 CC1CCN(C(=O)COCCN(C)C)CC1NC(c1ccnnc1O)=O C(=O)(CCC(C)(C)NC(c1csnn1)=O)NC(C1CCCC1)C C1(NC(CC2(C)CCCO2)=O)CC12CCN(C(=O)COCCCF)C2 C1(NC(c2nc(CC)sc2)=O)(CNC(C2CCC(OC)C2)=O)CCC(F)(F)CC1 c1(NC(C)=O)ccc(CNN2CCN(Cc3cnc(O)o3)CC2)cc1 O=C(C#CC1CCCO1)NCCC1CCCCN1C(C1CSCCS1)=O CC1CN(C(C2CC(F)(CO)C2)=O)CC(CCNC(c2cccc[n+]2[O-])=O)O1 c1(C(C(=O)NC(C)(C)CC)N(C(C#C)COC)C)cn2cc(Br)ccc2n1 c1(OCc2oc3ccc(C)cc3c2)cc(C(F)(F)F)cc2cccnc12 C1(CCOC)CN(C(=O)CC2=CCCC2)CCN1C(c1ncn(C)c1C)=O C(CC(CO)NC(=O)CCn1ccnc1C(C)C)OCC c1(C(C(=O)NC(C)C)N(C2CC2)CC2CCOC2)ncc(Cl)cc1Br CCC(F)(F)CC(=O)NCC1(C)CCC(NC(=O)C(c2ccncc2C)C)CC1 N1(C(c2nc(C(C)C)oc2)=O)CCC(CF)(NC(=O)CC2(O)CCCC2)C1 C1(NC(C2(COC)CC2(F)F)=O)CCCC(CNC(=O)CNC=O)C1 C1(C2CCN(C(c3cncs3)=O)C2)(NC(=O)CCSc2ccccc2F)CC1 N1(C(C2(NC(C(C)c3ccsc3)=O)CCC2)=O)CCC12CC(O)C2 O=C1CCCN(Cc2ccccc2)CC1.C12OCCC1NC2=O N1(CCC)CCC(NC(=O)Cn2ccnc2CCCOC)C(C)(C)C1 Cc1cc(NC(c2cc(C)n(C)c2C)=O)ccc1NC(=O)C(C)SCCN(C)C C1(C(N(C(C)CO)CC)=O)CC2C=CC1N(C(c1ccn(C)c1C)=O)C2 C1(NC(CC(=O)NC)=O)CC2CCC(C1C)N2C(C1(C)CCC(=O)NC1)=O Cc1ccc(Br)c(F)c1C(N1CCC(F)(F)C(NCc2ccc(F)c(F)c2)C1)=O n1(CCSC)nnnc1C(c1csnn1)NC(c1nccn1C(C)C)C CC#Cc1ccc(C(C(=O)NCCCF)N(C2CC2)C(C)C)cc1 N1(C(CCC(=O)NCCC)=O)CCC(NC(c2ncc(C)cc2F)=O)C(O)C1 c1(OC)ccc(CC(C2CC2)OC(c2[nH]ncc2C#N)=O)cc1.N12CCC1C2 CC#CCCC(CO)NC(=O)C(C)CSC1CCCCC1 CC1(C)C=C(C(=O)NC2(NC(=O)Cc3ccc(O)nc3)CC(CO)C2)C1 CC(C)C(=O)C(=O)N(C)CC1CCCN1C(C1CC2CCC2C1)=O N1(C(C(CC)=O)=O)CC2CN(Cc3cc(Cl)cc(Cl)c3O)CC2C1 CC1(C)C(=O)NC(=O)N1CCC(=O)Nc1ccc2c[nH]nc2c1 C1(CNC(CCC(=O)NCC)=O)CCC12CN(C(C1CNC(=O)C1)=O)C2 c1(C(=O)NCC(C)(C)NC(c2ccc(CC)[nH]2)=O)ccc(S(=O)(=O)NOC)cc1 c1(CC(N2C(CN(CCC=C=C)C)CCCC2)=O)ccc2nc(O)[nH]c2c1 N1(C(CN(C)C(=O)C2CC2)=O)CCN(C(c2cc(Cl)sc2Cl)=O)CC12CCC2 Cc1ccc(F)c(CC(=O)NC(C)CCNC(C2CC(F)C(=O)N2C)=O)c1 C1(c2cn(CCN(C)C)nn2)CCCN(C(c2conc2C(C)(C)C)=O)C1 c1(CC)cc(N2CCC(NC(C3CC3[N+](=O)[O-])=O)C2C)ncn1 c1(CN2CCC(N(C(=O)CN3C(=O)CNC3=O)C)CC2)cc(Br)ncc1F CC1CCCN(C(=O)C(C)n2ccnc2)C1CNC(c1cc(O)ccc1Cl)=O C1(CNC(CCC=C)=O)CN(C(=O)Cc2cnoc2)CCC1(C)C C(=O)(C(C)C1=CCCC1)NCC(C(C)C)NC(c1c(OC)cnc(Cl)c1)=O C1(CNC(CN(CC(C)(C)C)C)=O)CC(NC(=O)CCC2CCC2)CO1 C1(CN(C(=O)CCCN(C)C)C)CN(C(C2C(C)(C)C2(F)F)=O)CCO1 CC(CC(C)(C)C)C(=O)NC1(CO)CCCN(C(=O)CC2CCCSC2)C1 c1(C(C(=O)NCCC(=C)CNC(c2[nH]c(O)nc2C)=O)OC)ccc(OC)cc1 C1(C2(O)CN(C(c3cc(C(N)=O)no3)=O)C2)(CNC(C2C(COC)C2)=O)CC1 CC1(C)CN(C(c2cc(C#N)ccc2O)=O)CC(CNC(C2(Br)CC2)=O)O1 c1(N2CCC(=CC(N3CCOC4CC34)=O)CC2)ccnc2cc(Br)nn12 CC(C(=O)N1CCN(C(c2sccc2C(F)F)=O)CC1CC(F)(F)F)C(C)(F)F Cc1cc(=NCC(C2CCCC2)NC(C2(O)CC3CCC2C3)=O)[nH]c(CO)n1 CC1(C)CN(C(=O)CC2(O)CCCOC2)CC1CN c1(CC)cc(Br)ccc1C(N1CC(NC(C2(O)CCC2)=O)CC(C)C1)=O c1(C(=O)NCCC2(C)CCN(C(C(CC)(C)O)=O)C2)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)NCC(CC)NC(c2cc(C)c(C)nc2O)=O)c2c(nn1C)CCSC2 N1(C(CCC)=O)CCC(C(=O)N(CC(C)N(C(=O)CC(O)CC)C)C)CC1 C1(NC(C(C)NC(=O)OCC)=O)CCCCC1NC(c1cnc[nH]1)=O C(=O)(CCCC(C)(C)N(C)C)NCC(n1cc(-c2ccc(Cl)nc2)nn1)C C1(C(C)NC(c2csc(S)n2)=O)CN(C(C2CC3(CCC3)C2)=O)CCO1 C(N=c1[nH]c(=NC(C)c2nc[nH]n2)[nH]c2c(F)cccc12)c1c(C)ccc(Br)n1 c1(C(N2C(C(C)NC(=O)CNC=O)CCC2)=O)cccc2c1ccn2C N1(C(C(n2ncc(C)c2)C)=O)CCC2(CC(C(=O)N(CC(C3CC3)N(C)C)C)C2)C1 CN1CC(NC(=O)C(C)(C)CN(C)C(c2ccc3c(c2)CC3)=O)CCC1=O C1(C(=O)NCC2(C(C)(C)O)CN(C(c3ccc(C#N)o3)=O)C2)CCCCN1N=O c1(OC)ccc(C(=O)NC2(CO)CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)c(F)n1 CCC(O)C(C)C(=O)NCCC1CCCN1C(=O)CCNc1ccccn1 c12cccc(c1)SC2.N(S(=O)(=O)N(C)C)CC(=O)NC1(CC)CC(C(=O)O)C1 C1(NC(=O)Nc2sccc2C#N)CCCC(C(N2CC(C(C)(F)F)C2)=O)C1 N1(C(c2ccnc(OC)n2)=O)CCCC(F)(CNC(C2CC2C(=O)NC)=O)CC1 C1(C(N2CCC(NC(C3C(C)=C3)=O)C(C)C2)=O)CCC2CCCCC2C1 c1(C(C(=O)NCC(=O)N(C(=O)CSCCC(C)C)CC)C)ccc(F)cc1 C1(NC(C2C(C=C)OCC2)=O)CC2CCC(C1)N2C(=O)C(N1CCN(C)CC1)C c1(CC(=O)NC(C2OCCN(C(COCCC#C)=O)C2)C)cc(OC)cc(Cl)c1 CC1CCCc2c(C(=O)NC(C)CCN(C)C(c3sc(F)cc3Cl)=O)cnn21 C(=O)(CS(F)(F)(F)(F)F)NCC(CO)NC(COC(CC)C)=O O=C1NCCC2(CN(C(=O)C3=CCN(C(c4ncccc4Cl)=O)CC3)C2)O1 C1(C(=O)NCCN(C(=O)C2=CCC(C(F)(F)F)OC2)C)CC2COCC(C1)C2 c1(OC)cc(F)ccc1C(=O)NCC1(CNC(=O)Cn2nc(C)nc2C)CC1 CCCC(CC(C)C)C(=O)NCCOC1CCN(C(C2(CO)CCCCC2)=O)C1 Cc1c[nH]c2ncc(C(=O)N(C(C)CNC(=O)C=Cc3ccco3)C)cc12 C1(F)(CNC(=O)COc2ccccc2O)CCCN(C(=O)CCc2cnc(O)[nH]2)C1 c1(C(N2CC(O)(CCNC(CSC)=O)C2)=O)cc2ccsc2c(O)n1 c1(C(=O)NC(CN(C(c2c(OC)nsc2OC)=O)C)C)cccc(N)c1N C12(C(=O)NCC3(C)CCCOC3)CC(CO1)N(C(=O)CN1CCCNC1=O)C2 N1(C(Cc2ncc(C)[nH]2)=O)CCC(N(C(=O)Cc2cnccn2)C)C(C)C1 C1(NC(c2nc(COC)oc2)=O)CCN(C(C2(C(F)F)CCC2)=O)CC1 CCC(C)(C)C(=O)NCCN(CC(C)O)C(c1oc(Br)nc1C)=O CC1CCCN(C(=O)CCC2CC(NC(=O)C=CCn3cncn3)C2)C1CO c1(C(N2CCN(CC3(NC(C(CC=C)C)=O)CC3)CC2)=O)cnc2scc(C)n12 c1(OC(C(N2CC(CNC(c3cc(C)no3)=O)C2)=O)C)ccc(Cl)cc1C C1(CC)CCCN(CC(=O)NC2CCN(C(=O)C=C3CCCC3)C2)C1 C1(N(C)C(C2(C)CNC(=O)N2)=O)CC12CCN(C(=O)COc1ccsc1)CC2 c1(C(N(CCCNC(=O)CN2CCCCC2=O)CC)=O)cccc(C#N)c1 CC(C)CCCCC(=O)NCC(C(C)(C)C)NC(C1(O)CC(C)(C)C1)=O C(CC(O)C(=O)NCCC(C)NC(=O)C(=O)NCCCc1ccccc1)SC CCC1CNC(=O)C1.n1(C2(C(=O)NCCN(S(C)(=O)=O)C)CC2)cc(CN)nn1 c1(C(C)C)ccc(F)c(C(N2CCC(C)(NC(=O)C(C)OC(C)(C)C)CC2)=O)c1 N1(C(C(CCSC)(C)C)=O)CC2(CCCCN2C(c2nccn3ccnc23)=O)C1 Cc1sc(C(=O)NC(C)C(C)NC(=O)Cc2ccc(F)cn2)cc1S(N)(=O)=O N1(C(C(CNC(c2cnn(C)n2)=O)N(C)C)=O)CCCC(O)C1 c1(NC(C)=O)cccc(C(N2CC3CC3(CNC(=O)CC3CCCO3)C2)=O)c1C CC(C(=O)NC(C1CC1C(=O)NC1CCCCCC1C)C)S(C)(=O)=O C1(CNC(CC2C(=O)NC(=O)N2)=O)C2CCC(C2)N1C(c1ccc2c(c1)CC2)=O CC(CCCCO)NC(C1CCC1NC(c1coc(C2CC2)n1)=O)=O c1(C(=O)NC2C(NC(C3C(OC)CC3)=O)CCC2)cc2cc(Cl)c(Cl)cc2[nH]1 C(C(COC)CC(=O)NCC1CC1CNC(c1ncc(OC)cn1)=O)OC N1(C(C(C(=O)OCC)C(C)C)=O)CCC2(CC1)CCN(C(=O)CC(C)=C(C)C)C2 C1(C)(C(N2CCCC(NC(C)C)C2)=O)CC12CCN(C(C1C3COCC13)C)CC2 N1(C(c2c(OC)c(F)ccc2)=O)CCC2(CCCN2C(c2cccc(=O)o2)=O)C1 c12cc(no1)CC(C)C1CN(C1)C2=O.C(=O)(C(CN(C)C)N(C)C)N.CSC CCCCC(O)CC(=O)N1CC2(CC(CC(=O)NC3CCOCC34CCC4)C2)C1 N1(C(C2CN(C(=O)Nc3c(C)ccc(C)c3)C(CO)C2)=O)CC2CCCCC2C1 c1(C(=O)NCC2C3CC2N(C(=O)C#CC2CC2)C3)cnc2ccccc2c1 c1(CC(=O)NC(CN(C(c2cc(C(F)F)[nH]n2)=O)CC)C)cn(C)nn1 CCC(CO)(C(=O)NC1CCC(NC(=O)C(O)C(C)(C)C)CC1)OC Cc1cnc(C(N2CCC23CN(C(c2cn[nH]c2)=O)C3)=O)c[n+]1[O-] CC1(F)CCCN(C(=O)C(CCOCCO)NC(=O)C=Cc2ccoc2)C1 C12(C(=O)OCC)CCC(C(N3CC(c4cccc(C)c4)(O)C3)=O)(CC1)O2 C1(NC(C2CCC2)=O)CCCCC12CN(S(=O)(=O)c1ccc(F)c(F)c1)CCO2 CC(C)CC(O)C(=O)N(CC(C)C(N1CCn2ccnc21)=O)C c1(C(=O)Nc2cnc(NCC3CCCO3)nc2)cnc(Cl)cc1Cl Cc1[nH]nc2cc(C(=O)N(C3CCC(NC(=O)CC4CC4)C3)C)ccc12 N1(C(c2cc(C(C)C)on2)=O)CCCCC(C(N2CCCCC(N(C)C)C2)=O)C1 C(=O)(CCC(C)(C)O)N(C(CNC(C1N(CC)CCCC1)=O)C)C c1(C(=O)NC(c2nnc(C3CCC3)o2)C)ccc(N)c(OC(F)(F)F)c1 N1(C(C(CC)(C)O)=O)CCC2(CCN(C(c3cc(C)no3)=O)CC2)C(C)C1 N1(C(c2c(OCCC)cccn2)=O)CC(C2(NC(c3nc(C)sc3C)=O)CC2)C1 c1(C(N2C(C(=O)NCC(C(=O)OC)C)C(C)C2)=O)ccc([N+](=O)[O-])[nH]1 c1(OCC(=O)NCC(CN(C(=O)CN2C(=O)CNC2=O)C)O)cccc(O)c1 N1(C(C2C(CC(C)(C)C)C2)=O)Cc2n[nH]cc2C1C(=O)N1CCCC12CCCC2 C1(NC(c2nc(C(N)=O)sc2)=O)CCN(C(=O)CCn2cccn2)CCC1(F)F C(=O)(C(F)C(F)(F)C(F)(F)F)NCCN(C(C1(F)CCCCCC1)=O)CC1CC1 Cc1cc(C(=O)NCC(C)CNC(C2CC(N(C)C)C2)=O)nc2ccccc12 CN=c1cc(C(N2CC(CNC(=O)CCc3ccsc3)C(C)(C)C2)=O)cc[nH]1 CN1CCN(c2ncccc2OC(C2CCC(C)O2)=O)CC1 O(NC(=O)CCC1(NC(=O)C(O)c2ccsc2)CCC1)CC1(C)CC1 N1(CC(=O)N(C(C)C(=O)N(C)Cc2ncco2)CCC)C(=O)CCC1=O c1(OC)cccc(I)c1NC(C12CC(Nc3ncc(C(F)(F)F)cn3)(C1)C2)=O c1(C(=O)NCCC2CCN(C(=O)C=C3CCCC3)CC2)cccn2c(O)nnc12 C1(CC(=O)NC(Cc2cn(CC=CC)nn2)C(=O)O)CCCCN1C CC1c2ccccc2OC1C(=O)NCC1CN(C(C2CC(n3ccnn3)C2)=O)C1 C(CN=c1ccnc(CO)[nH]1)(c1ccc(OC)c(F)c1)NC(C1CCCOC1)=O N#Cc1cc(Cl)c(C(=O)NCC2(NC(=O)Cc3nc[nH]n3)CCOCC2)s1 c1(CNC2C(C(=O)NC)C3CCC2C3)ccc(F)c(O)c1F c1(C(N2CC(F)(CNC(C(CC)NC(C)=O)=O)C2)=O)c(C)nn2c1CCCC2C c1(OC(C)C(=O)N(CCCN(C(=O)C(C)(C)C(N)=O)C)C)ccc2c(c1)CCC2 N1(c2cc(N3CCCC(C(=O)OC)C3)ncn2)CCCc2[nH]ccc2C1 Cc1cccc(C(N2CC3C(C(=O)Nc4ccc(F)nc4F)C3C2)=O)c1[N+](=O)[O-] C1(N(CCNC(C=CC)=O)C(c2ccc(C(C)C)o2)=O)CCS(=O)(=O)C1 C1(C(N2CCC(CNC(C3CCC(C(=O)OC)CC3)=O)C2)=O)CCCCN1N=O N1(C(C(F)=CC)=O)CC2CCCCC2(NC(c2ccc(C#N)cc2Cl)=O)C1 C1(C(=O)NCCCC(C)(C)NC(=O)CSCC(F)(F)F)CCCC(C#N)C1 N1(C(C(C)C2CCC2)=O)CC(CNC(C2CC3CCC(C2)O3)=O)C(F)(CO)C1 C12(CNC(C(CC)Br)=O)CCCOC1CCN(C(=O)CCNC(=O)NC)C2 CC1(C)CCC(CNC(=O)C(C)(C)CF)N(C(C2CC3OC2C2CC32)=O)C1 C1(C(N2CCCC2CNC(c2cccc(COC)n2)=O)=O)C2CC3C(C2=O)C13 N1(C(=O)NC(C)(C)C(=O)N2CCC2)CCC(c2cccs2)CC1 c1(C(=O)NCCCCC2CN(C(C3CC(SC)C3)=O)C2)cc(Cl)c(F)cc1Cl N1(C(c2c(C)cccn2)=O)CC(NC(=O)C(C)(C)c2cc[nH]n2)CC(C)C1 CC1(NC(C23CC(CO)(C2)C3)=O)CCN(C(c2cocn2)=O)CC1 Cc1c(Cl)ccc(C(=O)NC2(C3CN(C(=O)Cc4c[nH]ccc4=O)C3)CC2)c1O C1(OC)CC(NC(=O)CCCN2C(=O)CCC2=O)CN(C(C2CNC(=O)C2)=O)C1 CCCCCC(C)(CC)C(=O)N1CCC(=O)N(C)CC1.C12CCCN1CC(=O)N2 c1(C(N2CC(c3cn(-c4cn(C)nc4)nn3)OCC2)=O)ccc(F)c2occc12 C1(C(=O)NCCC(C)(C)NC(=O)CNC(C2CCCC2)=O)CCS(=O)CC1 c1(C(N(C(C(C)C)C)C2CC2)=O)c[nH]nc1CCNC(=O)CC1CCC(C)O1 N1(C(c2ccon2)=O)CCN(C(=O)CCc2nncs2)C(C2CC2)C1 C1(NC(C(=O)OC(C)(C)C)Cn2cccn2)C=CC2(CCCC2)CC1 C1(N(C(=O)CC2CC(=C)C2)CC#C)CCN(C(C)C)C1 CCC(CN(C)C)C(=O)NC1(C)CCN(C(=O)C=CC(F)(F)F)C1 C(=O)(C(C)(C)c1cnco1)N(CC(C)O)CC(F)F n1(CC=C)cc(C(=O)N(C2CCC(NC(=O)C=CBr)C2)C)nn1 Cn1ncc(Cl)c1CNCCC1CCCN(C(=O)OC(C)(C)C)C1 c1(C(N2C(C(=O)Nc3c(C)ccnc3F)CCC2)=O)cc2cccnn2n1 N1(C(C(C)CC2CCCC2)=O)CC(NC(=O)CC2(CO)CCOCC2)CC1(C)C c1(OC)nc(C)ncc1C(N1CCCC1CNC(c1cc(C)[nH]c1C)=O)=O CCC(C)(C)C(O)C(=O)N1CCC(C)N(C(C23CCC(C2)OC3)=O)CC1 N1(C(C(=O)NCC(c2ccc(Cl)cc2)C)=O)CC(C)C(N)C1 CC1COCCCN1C(=O)CC(CC1CC1)NC(C1CC(=O)CC(=O)C1)=O CCC1=C(C(=O)NC2CC3CC2CN(C(=O)C(C2CCCCC2)C)C3)CCCO1 C1(O)(C(=O)NC(c2ccccc2F)C)CCN(C(C2CCCCC2N)=O)CC1 C1(C(=O)NCCN2CCC(OC)C2)CC2(CCN(C(=O)C(C)(C)C(C)(C)C)C2)C1 N1(c2cc(NCc3cc4cn[nH]c4cn3)ncn2)CCC2(CCCc3ccccc32)C1 C1(OC)CC(C(=O)NCC(CO)NC(=O)CCc2nc(C)cs2)CC1OC N1(CC)CC(NC(=O)CC=CCNC(C2COCCN2C)=O)CC1=O C1(C(=O)NC(c2cn(C)nn2)C(=O)NC(c2nnc(C)o2)C)COCCC1C C1(C(=O)NC2C(NC(c3c[nH]nc3C(F)(F)F)=O)C2)C2CCC(F)C12 N1(C(=O)Cc2ccnc(C(F)(F)F)c2)CCC2C(CCN2C(=O)Cc2ccsc2)C1 Cc1ccc(C(=O)NCC2(F)CCCN(C(c3cnsc3)=O)C2)c(C)c1 C(C(=O)NC1CN(C(=O)CCF)C1)(C(C)C)SCC c1(N(C)C)ccnc(NC(=O)CNC2CN(C3CCC3)C2)n1 Oc1ccc(CNC(=NCC2CCC2)NCC2CC3CCC3C2)c(F)c1 c1(C(=O)NCC2N(C(C(CC)OC)=O)CCCC2)ccc2c(n1)CCCC2 N(C(=NCc1ccc(F)c(Br)c1)N(C)CC1CCCN1S(C)(=O)=O)C(C)C Cc1cnc(C(N2CC(C)(C)C2Cn2cc(C3(C4CC4)CC3)nn2)=O)cn1 C(C(C)C(=O)N1CCCC1CCC(=O)N(C)CC1CC1(F)F)OCC CCCCS(=O)(=O)CC(=O)NC1CCN(C(=O)C(F)(F)CCn2cccn2)C(C)C1 C(=O)(C(C)(C)CC(=O)N1CC(NC(=O)CCc2cccn2C)CC(O)C1)OCC N1(C(C(CC)F)=O)CCCC(CCNC(c2ccc(N)c(F)n2)=O)CC1 C1(C)(NC(CCc2nc(C)c(C)[nH]2)=O)CCN(CC(c2cncn2C)=O)CC1 c1(C(=O)NC2CCN(C(C3N(S(C)(=O)=O)CCC3)=O)C2)ccc2nn[nH]c2c1O c1(CNC(C2CCCC(NC(C3CC(F)(F)C3)=O)C2)=O)cc(O)ccc1F n1(CC(=O)N(C)CC2(O)CCN(C(CC3(C=C)CC3)=O)C2)c(C)cc(C)nc1=O N1(CCC)CCCCC1C(=O)NC1CCCCC1CNC(=O)CCc1cnn[nH]1 c1(SCC(=O)NC(C(C)NC(c2c(CC)cno2)=O)C)ccc(Cl)cc1 c1(C(N2CCC(NC(c3nc(OC)oc3)=O)C2)=O)sc(C)nc1C CCC(CC)C(=O)NCC(C)(C)OCCNC(=O)C(C)(C)C1CCOC1 c1(C(N2CC(CC=C)(OC(C(=O)NCC)F)C2)=O)ccc2cnoc2c1 C1(NC(CCNC(=O)C=CCl)=O)CC(NC(c2cc(Cl)ns2)=O)C12CCC2 CC1(C)CCCC1(C)NC(C1C2CC3C(C2NC(C2CCCN2C=O)=O)C13)=O CCCC(C)C(C(=O)NCC)N(C1CCN(C2CC2)C1)CC(C)(C)C c1(CC)ccc(OC)cc1C(=O)NCC=C.C(=O)(C(C)CC1CC1)N=CCSC C1(CC(N2C(C(=O)NCCC3(OC)CCC3)CC2)=O)CCC(=O)C1 C(=O)(C1CCCc2sccc21)N1C(CC)(CC)CC(NC(C2CS(=O)(=O)C2)=O)C1 C1(C2(O)CCN(C(c3cc(C)cc(C)c3)=O)CC2)(NC(C(COCC)C)=O)CC1 c1(C(=O)NC2C(NC(c3ccc(C(C)=O)cc3)=O)CC2)cnc2n1CCCC2C c1(CC(C(=O)OCc2cnoc2C2CC2)O)cc(Cl)ccc1Cl CCCCCC(CC)C(=O)NCC(C)NC(c1cc(C)nc(C(F)(F)F)n1)=O c1(C(=O)NCC2N(C(CC(CCC)(C)O)=O)CCCC2)nc2nc(C)ccn2n1 c1(-c2cnc(CSC)s2)cccc(C#N)c1.C1(N2CC2=O)CCOCC1 N1(C(COCC)=O)CCOCC(NC(c2cnoc2C2CC2)=O)C1 c1(N2CCC(C)S(=O)CC2)nc(=N)[nH]c(=NCc2nnc(C(F)F)s2)[nH]1 N1(C(Cc2c(C)con2)=O)CCC(NC(c2ccc(F)c(N)c2)=O)C(CO)C1 N#Cc1ccc(CNC23CC(NC(=O)C(=O)C4CCC4)(C2)C3)cn1 CC1(C)CN(C(c2coc(O)n2)=O)C(CNC(c2nccnc2C(N)=O)=O)CO1 C(C)(CCC(=O)NCC(=C1CN(C(=O)C(C)CN(C)C)C1)F)OC C=CC1(C(=O)NCCCn2nccn2)CCN(C(C)=O)C1 c1(NC(=S)NCC(F)(F)F)ccc2c(c1)CCN(C(C1CCCOC1)=O)C2 c1(NC(C)=O)cnc(-c2nc(-c3ccccc3)co2)cn1 N1(C(C2C(C)(C)C2C#N)=O)CC2CCC1C2NC(c1cc[nH]n1)=O CCC(CC(=O)NCc1c[nH]nc1C(=O)NCc1ncn(C2CC2)n1)C(F)F N1(C(CCC(C)=O)=O)CC2CCC(C1)N2Cc1c(F)cc(Br)cc1Br N1(C(C2(C=C)CCC2)=O)CC(NC(=O)CCc2ncc(F)cn2)C(O)C1 C1(CC(=O)NCCSCCO)CN(C(=O)CCCC)CCO1 c1(C(N2CC3CC3C2)=O)cnc2c(-c3cccc4ncccc34)cnn2c1 N1(C(c2n[nH]c(C)c2O)=O)CC(Nc2ncc3c(n2)CCOC3)CC2(CCC2)C1 C(=O)(C1=C(Cl)CCOC1)NCCC1N(C(C2(C)C(C)(C)C2)=O)CCCC1 c1(CC)c(Cl)nc(C(C)(C)C)[nH]c1=NCC1CCCN1C(c1cncs1)=O O=S(=O)(c1cccnc1NCCCn1cnnn1)N1CCCC2(CCC2)C1 N1(C(=O)COCC(F)F)CCCC2C1CCN2C(C1CCC1)=O n1(CC(=O)NC(CCNC(CCC(C)OC)=O)C)c(C)cc2ccccc12 c1(-n2cc(C(n3cc(CCN(C)C)nn3)C)nn2)cccc(Cl)n1 C(=O)(C(F)C(C)(C)O)NCCC1CC(C(=O)NC(c2ccc(C)s2)C)C1 CCCC(C(=O)NCCSCC(=O)NCC1CC2CCC1O2)N(C)C CCC(C)C(C(=O)NC1(CCF)CCOCC1)N(C(=O)CSC(F)(F)F)C C1(NC(c2c(OC)cccc2)=O)CCN(C(C2(c3occc3C)CC2)=O)CC1O C1(C(C(=O)NC2C(C(C)(C)C)NCCC2)=O)CCC(c2ccccc2)CC1 Cc1cc(C(=O)NCCN2CCN(C(c3nc(=N)cc[nH]3)=O)CC2)nn1C(C)C C(CC(C)C(=O)NCC1(OC)CCN(C(C2C=CCC2)=O)C1)=CCC C(C(C(C)C(C)C)NC(=O)Cn1cncn1)NC(c1cccc(CC)c1)=O c1(C(=O)NC(CNC(C(C)=C2CN(C(=O)OC(C)(C)C)C2)=O)C)c[nH]ccc1=N N1(C(C2CC(N=[N+]=[N-])C2)=O)CCC(NC(=O)CN2CCOCC2)C(O)C1 N1(C(C(C)C)=O)CC(CNC(=O)CC(C)c2cccnc2)CC1(C)C N1(C(c2c(C)cns2)=O)C2CCC1CN(C(C1C3CCC1(c1cnco1)C3)=O)C2 CC(C)C(O)CC(=O)N1CCOC(CNC(=O)C(c2cccc(O)c2)C)C1 Cc1n[nH]c(C)c1C(C)C(=O)NCC(C)(C)NC(=O)Cc1ccoc1 c1(OCC)ccccc1-c1nc(CC2CC2C)n(-c2ccnc(Br)c2)n1 N1(C(c2occ3c2CCOC3)=O)CCC(O)C2(CCOCC2)C1 C(=O)(C1=CCC(C)CC1)N(CCC(C(C)C)NC(=O)Cc1ccoc1)C N1(C(C(c2ccc(C#N)cc2)C)=O)Cc2cccn2CC(C(=O)NCC(C)O)C1 CC(CNC(=O)CCn1cnnn1)C(=O)NC1CCCC1 CCC(C)C(C(=O)NCc1ncc(CO)[nH]1)N(C(=O)C=Cc1cc(C)no1)C Cc1cccc(CC(=O)Nc2ccc(-c3nn[nH]n3)cc2C)c1C Cc1ccnc(O)c1C(N1CCC=C(CNC(C2CS(=O)(=O)C2)=O)C1)=O CC1CC2CN(C(c3cn(CCNC(c4cccnc4)=O)cn3)=O)CC12 c1(C(N2CCNCC2c2ccc(Br)cc2)=O)cccc(O)c1O c1(CNC(c2ccc(N3CCCC3)cc2)C)cccc(C(C)(F)F)n1 N1(CCCNC(c2c(C)cc[nH]2)=O)CCN(c2nncs2)CC1 c1(CC)cccc(C(=O)NC2(C)CC(NC(C3C(C#N)C3(C)C)=O)C2)c1C CC(F)(F)CC(=O)N1CCCCC1CNC(c1cnccc1C(F)F)=O c1(CCC(=O)N(CCCN(C=O)C)C)csc(C)n1.C=C1CC1C=C c1(NC(CN(C2CCC2O)C(=O)OC(C)(C)C)=O)cccc2c1C(=O)CC2 N1(C(C2(CC#C)CCCC2)=O)CCCCC(NC(c2cnoc2COC)=O)C1 c1(OC)cnc(F)cc1C(=O)NC1CCCCC1NC(=O)C(C)=C1CCC1 C1(O)(CNC(C(CO)NC(COCCCC)=O)=O)CC(C)(C)C1 C1(C(=O)NCc2cnccc2Cl)CCC2CCC1N2C(=O)C1=C(Cl)CCC1 N1(C(C2CC(SC)C2)=O)CC2(CCN(C(c3cc(C)n(C(C)C)n3)=O)CC2)C1 C(=O)(CCC(=O)NCC)NC1C(CNC(C=CC(=O)OCC)=O)C1 C(=O)(CCC(C)CN1CCC(CCc2ccc(O)cc2)CC1)OCC S(=O)(=O)(C1CCOCC1)N1CC2C(CNC(c3ccoc3C(F)(F)F)=O)(C2)C1 c1(C(=O)NCC(CNC(CNC(N)=O)=O)CO)cc2cc(Cl)ccc2[nH]1 c1(OC)ncccc1NC(=O)CC1(OC)CN(C(C2CC(C)CO2)=O)C1 C(=O)(C1CCCn2ncnc21)NC1(COC)CCN(C(C2CCOC2C)=O)CC1 CCC1(C)CNC(=O)c2cncc(c2)CNC1=O.c1(CCC(=O)NC)ncnn1C C1(CNC(CCc2cc(C)no2)=O)CC(NC(=O)C=Cc2cocn2)CCO1 Fc1ccc(OCCN=C(NCC(F)(F)C2CC2)NCC2CCCCC2)cc1Cl C(=O)(C1(C)CCn2c(C)nnc21)NCC1(F)CC(CNC(CCCOCC)=O)C1 Cc1ccc(O)c(CNC(C2CCCCN2C(=O)C(=O)C(C)C)=O)n1 C(=O)(C1=NOC2(CCOC2)C1)NC1CC2(CC(NC(CCCC#CC)=O)C2)C1 CCC(CC)C(=O)NCC1CN(C(=O)Cc2ccnn2C)CC1C(F)(F)F CC1(C(=O)NCC2CCCN2C(=O)C(=O)NCC2CC2)CCC(=O)NC1 N1(C(C(CC(N)=O)NC(C(C(C)C)N=[N+]=[N-])=O)=O)CCC2=C(CCCC2)C1 C1(C)(C(=O)NCC2CCCN2)CCCN(C(=O)CNC2OCCN(C)C2)C1 C1(NC(=S)NCC2CCCNCC2)CC2CC1C1CCCC21 N#Cc1ccnnc1N(C(=O)CC1CC(=O)C12CCC2)Cc1ccco1 c1(C(=O)NCC2(O)CN(C(c3cccc(NC)n3)=O)C2)cnc2ccccc2n1 N1(CC(=O)N(CCNC(C(c2ccccc2F)(C)OC)=O)C)CCCCCC1 CCC(N=c1[nH]c(=NCC2C3CCC(F)(F)C23)[nH]c2c1CSC2)c1ccc(C)o1 C1(CN2C3CN(C(c4c(C)nn[nH]4)=O)C(C3)C2)CCC2(CCOCC2)O1 c1(C(=O)NC(CN(C(=O)Cc2cnc(C)[nH]2)CC)C)onc2c1CCCC2 C1(CNC(c2c(CC)c[nH]c2)=O)CC2CCC(C1)N2C(c1ccc(CO)o1)=O N1(C(C=CCC)=O)CCC(C(N2CCC(CCN(C)C)C2)=O)(CF)C1 C#CCC(O)C(=O)N1C(C(=O)Nc2cscc2CC)CCC1C c1(OC)ccc(S(=O)(=O)Nc2snnc2-c2ccc(Br)cc2)c(C(F)(F)F)c1 Cc1cc(S(C)(=O)=O)ccc1CNC1CCC2(C1)CN(C(c1ncsc1C)=O)C2 N1(C(CCCCCC=C)=O)CCN(C(=O)CCCCC(C)=O)C2COCC12 c1(C(=O)NCC(CNC(C(C)OC)=O)O)csc(C)c1C C1(CN(c2cccc(OC)c2)CC)CCN(C(=O)Cc2nnc(C)o2)CC1 c1(C(=O)NCC(CNC(c2c(CC)con2)=O)OC)ccc(-n2ccnn2)cc1 c1(NC(C)=O)ccc(N)c(C(=O)N(C2CCN(C(=O)Cc3cn[nH]c3)CC2)C)c1 C(C)(CCCC(=O)NCC(C)(C)c1cccs1)NC(C)=O C(=O)(CC(C)(C)CN(C)C(C1CCOC(C)C1)=O)NCc1n(CC)cnn1 c1(C(=O)NCC(CC)(C)NC(=O)CCCCSC)ncncc1Br C1(C(=O)NCCC(=C)CNC(c2nnc(O)nc2O)=O)CCS(=O)(=O)C12CCC2 N1(C(CSC)=O)CC(NC(c2ccc(-c3ccccc3)n2C)=O)C(O)C1 C(CC(C)(C)CC(=O)NC1CCCCC1CNC(c1cc(C)n(C)c1)=O)OC CC(C)=C=CC(=O)N(C)CCC1CCN(C(=O)C=CC2CC2)CC1 N1(C(CC=CCC)=O)CCC(NC(=O)Cc2ccsn2)C2(CCC2)C1 Cc1cc(F)c(C(=O)NCC(C2CC2)N(C)C(C2(C)CCCC2C)=O)cc1F CC1CC(NC(=O)CC2CCCCC2O)CN(C(=O)CCc2cnccn2)C1 Cc1ccc(NC(C2CC3CC2N(C(=O)C(C2CCCCC2)O)C3)=O)c(C)c1 C(C(CO)C(F)(F)F)NC(CCC1(C)CN(C(c2cn(C)nc2)=O)C1)=O c1(CC(=O)NC2CC(NC(C(C)C(F)F)=O)CC2O)cc2ccccc2c(=O)o1 N1(C(C(Cc2cn(C)nc2)O)=O)CCCOC(CNC(=O)COC2CCC2)C1 c1(C(N2CCC(N(C(C(C)Cc3ccncc3)=O)C)C2)=O)cc2n(n1)CCCO2 C(=O)(C(C(F)(F)F)C(F)(F)F)NC(CNC(CCc1onc(CC)n1)=O)C c1(N2CCC(OCCC)CC2)nc2c(c(=NCc3cccc(C)c3F)[nH]1)SCC2 C(CC(C(=O)N1CCCC(CSC)C1)NC(=O)C(C)OCC1CC1)SC N1(C(c2[nH]cc(CC)c2)=O)CC2(CCCC2NC(c2cn(C)nc2C)=O)C1 C=Cn1nncc1C(=O)NC(C1(O)CCN(C(=O)CCC(=O)c2cccs2)C1)C C1(CC)CCc2sc(C(N3CC(CNC(=O)C(C(C)(C)C)OC)C3)=O)cc2C1 C(=O)(CCC(=O)NC(C)(C)CNC(c1cnc(C2(C)OCCO2)s1)=O)NCCC C(=O)(C(C)(C1CC1)N(C(=O)CC1C=CCCC1)C)NCCN(CC)CC C1(O)(CC(=O)NCC2CCC2CO)CN(C(c2cc(CO)on2)=O)C1 Cc1cc(Cl)ccc1C(=O)NCC(c1ccccc1)NC(=O)C=Cc1cocn1 N1(C(C(CC)SC)=O)CCCC(CC)(NC(=O)CC(C)SC)C1 N1(C(CC(C)OC)=O)CCCC(CN(C)C(c2cn(CCN(C)C)nn2)=O)C1 CON1CC(C(N2CCC(C(=O)NCC(=O)NC3CCC3)C2)=O)CC1=O c1(C(=O)NCC(Cn2cc(C(C(OC)OC)C)nn2)(F)F)ccccc1C(C)(F)F C(=O)(C#CC1CC(F)(F)C1)NC1CCN(C(CS(N)(=O)=O)=O)C1C1CC1 CN1CC(C)(NC(c2cnn3ccccc23)=O)CCC1=O N1(C(c2ccc(C)o2)=O)CCN(C(=O)CCC2CC2CC2CC2)CC1CF C1(CNC(C(C)c2ccsn2)=O)CC2CCC1N(C(N)=O)C2.C1(=O)CN1 c1(CCC)occc1C=O.N12CCC(C1)OCCNC(=O)CC1CC2C1.SCC c1(C(=O)NC(CNC(C2CC(c3ccccc3)C2)=O)CO)ccnc2ncnn12 CC1CCn2cc(C(=O)NC3CC(CCNC(=O)CNS(N)(=O)=O)C3)nc2C1 N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CC2CC(NC(c3csc(Cl)c3Cl)=O)C2C1 C1(CCC)CC(C(N2CC(CNC(c3c[nH]nc3C3CCCO3)=O)C2)=O)CCO1 c1(OC)ccc(NC(c2cc(Br)no2)c2nnnn2CCCC2CC2)cc1C c1(CN2C(C(N(C)C)=O)CC3CC32)ccc(F)c(C#N)c1 C=CCCC(C)(C)C(=O)NC1C2CN(C(=O)C(C)Cc3ccccc3)CC12 N1(C(c2c(C)cc(C)o2)=O)CCC(NC(c2ccc(CO)c(F)c2)=O)C(F)C1 c1(C(N2CCCC(N(C)C(C3CC4(C3)CC43CC3)=O)C2)=O)c(F)cc(F)cc1Cl Cc1sc(=O)n(CC(N2CCC(O)(C(C)CNC(=O)C(C)(C)C#N)C2)=O)c1C CC1CN2CCN1CC2C(N1CCN(C(c2cc(O)ncn2)=O)CC12CC2)=O C(C(C)(C)CC(=O)N1CCOC(CNC(=O)CC2CSCCS2)C1)OC c1(C(N2C(C3CCN(C(=O)C=CC=C(Cl)Cl)C3)CCCC2)=O)nnc(O)nc1O C1(C(=O)NCC(CN(C(CCN(CC)CC)=O)C)C)CC12CCC2 Cc1cc(C)n2c(CCCC3CC3)nnc2n1.C1(CNC(=O)C(=O)N)CCOC(C)(C)C1 C=C(Cl)CC(C(=O)NCC(C)C(=O)OC)NC(c1cccc(C)c1)=O CN1CCCCC1CNC(C1CNCCN1Cc1nccn1CC(F)(F)F)=O C=CC(C)(CC)C(=O)N1CCN(C(C)CCc2cc(C(F)(F)F)[nH]c(=N)n2)CC1 N1(C(c2nc(C(C)C)oc2)=O)CCN(C(C2SCCS2)=O)C(C)CC1C C(=O)(C(C)(C)C(O)CC)NC(C1CC=CCC1)C(=O)NCc1cnc(CC)[nH]1 c1(C(=O)NCCN(C(=O)C(Cl)=CCl)CCC)cccc(-n2cccn2)c1 C(C(CC(C)C)C(=O)N1CC(CC(=O)NCC(O)C2(Cl)CC2)(OC)C1)OC CCCCC(O)C(=O)NC1CCCCC1CNC(=O)CC1(C(=O)OC)CC1 N1(C(c2nc(CCC)sc2)=O)CC2CC(CNC(c3ccc(N)cn3)=O)C2C1 N1(C(CCc2n(C)cnn2)=O)CCC2(CCN(C(C3CCCC(C)(C)C3)=O)C2)C1 C1(NC(c2c(OC)noc2C)=O)CCCC(NC(=O)CC2(C)OCCO2)CC1 c1(C(N2C(C(=O)NCCCCCC)(CC)CCC2)=O)ccc2cncn2c1 C1(C(N2C(C)C(NC(=O)CC3CCS(=O)(=O)CC3)CC2)=O)CCCCS1(=O)=O N1(C(C(C(C)(C)C)OC)=O)CCC2(CC1)C(NC(=O)CN1CC=CC1)CS2(=O)=O C1(CNC(C(CC)(F)F)=O)CC2COCC2N1C(=O)C(CC)CCOC c1(C(=O)NCCCCNC(c2c(C)[nH]c(C)c2C)=O)coc2c(F)cc(F)cc12 c1(CC(=O)NC)ccc(C(N2CCN(C(=O)C(C)O)CC2)=O)cc1 C1(CCNC(CCCC(N)=O)=O)CC2CCC(C1)N2C(c1cnn[nH]1)=O c1(C(N2C(C(=O)Nc3ccccc3)CCC2C2CC2)=O)cc2ncccc2[nH]1 C(CSCc1ccccc1)(C(=O)N1CCC1c1cn(C(C)(C)C(=O)O)nn1)OC c1(C(N2CC(NC(c3n(CC)ccc3)=O)C2)=O)ccc(-c2csnn2)cc1 C#CCCC(=O)NCC(CC)NC(c1ccc(C2CCOC2)s1)=O c1(C(N(CCCNC(=O)Cn2cncn2)CCC)=O)cc[n+]([O-])cc1 C1(NC(C(C)=CC)=O)CCCC(CNC(=O)CSC)C1 C1(CCO)(CNC(CCOCCC)=O)CN(C(=O)C(C)CC2CC2)C1 C12(NC(c3nccn3C)C(C)C)CC(CN(C(=O)OC(C)(C)C)C1)C2 c1(C(=O)NCC2(C)CC(NC(c3ccsn3)=O)C2)ccc2ccccc2c1F N1(C(c2cc(C(=O)OC)c(C)c(C)c2)=O)Cc2cc(Br)ccc2C(C)C1 C12(C(=O)NC(C3N(C(c4ccc(COC)s4)=O)CCC3)C)CCC(C1)C(C)(C)O2 C(C)(CCC(=O)N(C1CC2(CC2)C1)C)NC(C(C)OCOC)=O C(=O)(N=c1[nH][nH]c2ncccc12)c1c(C)nccc1.N12CC(CC(F)C1)C2=O CCC(CC)CC(=O)NCC1(CNC(=O)C(c2cc(F)cc(F)c2)C)CC1(F)F N1(C(C(C)CO)=O)C2CCCC1CC(NC(c1coc(C(N)=O)c1)=O)C2 Cc1cccc(F)c1C(N1CCC(CNC(=O)CCCC(C)C)C1)=O CC(O)(CC(F)F)C(=O)NC1CC1NC(=O)CCN1CCOCC1 N1(C(CCCC)=O)CCOCC(F)(CNC(c2ccncc2NC(C)=O)=O)C1 c1(NC(C2CCCN(CCCC=C)C2)=O)ccc(C(F)(F)F)cc1[N+](=O)[O-] N1(C(c2cc(CC)[nH]n2)=O)CC(CO)C2(C1)CN(C(=O)C(C)C1=CCCC1)C2 c1(C(=O)NC2CC(C)(NC(C(CC=C)C)=O)C2)cc(=O)c(OC)cn1C C1(CNC(CN(C)C2CC2)=O)(NC(C2CCCC2N(C)C)=O)CCCCC1 CCCS(=O)(=O)CC(=O)NCC1(C2CC2)CCN(C(c2nc(C)sc2C)=O)C1 N1(C(c2cc(SC)c(C)o2)=O)CCCC12CCN(C(C1CCC(C)(C)O1)=O)C2 c1(C(=O)NCC2N(C(C=C(C)C3CC3)=O)CCC2C)cccc2cncn12 C1(C(=O)NC(C=C)C(F)(F)F)CN(C(=O)C(C)(C)CO)CC(C)O1 N#Cc1cccc(NC(=O)CN2CC3CC2CN3C(C2(F)CCCCC2)=O)c1 c1(C(=O)NCC2C(CNC(C(COC)COC)=O)C2)c(O)nnc2c1CCCC2 c1(NC(CC2CC(C)(C)N(C(c3ccon3)=O)C2)=O)ccc2c(c1)OCO2 C1(NC(C2CC(CCC)OCC2)=O)CCN(C(C2CC2CC)=O)C(C)C1 O=C(CS(=O)(=O)CC(F)(F)F)NCC1CCCN(C(c2cnnn2C2CC2)=O)C1 N1(C(C2(Cc3ccccc3)CC2)=O)CCCC2CN(c3ncnc(Cl)c3F)CCC12 c1(C(=O)NC2CCOCC2NC(C2(F)CC2)=O)cccc(C#CC2CC2)c1 CC(C)CC(O)C(C)C(=O)NCC#CCNC(c1cccnc1N(C)C)=O c1(OC)ccncc1CC(=O)NC1(C)CCN(C(=O)CC2C=CCC2)C1 CC1(CNC(C2(n3cncn3)CC2)=O)CCN(C(c2n[nH]c(C3CC3)n2)=O)C1 CC1(C)CCN(C(C2(F)CCOCC2)=O)CC1CNC(c1nc(Cl)cs1)=O C1(C(=O)NC(C2(O)CN(C(c3ccc(F)c(F)c3)=O)C2)C)CC2CCCC(C1)C2 N1(C(CSC)=O)CCCC(C)(C)C1CNC(C1CC(Cc2ccc(F)cc2)C1)=O C#CCC(CC(F)F)C(=O)NC(COC)CNC(c1c(Cl)cnn1C)=O c1(OC)ccc(CC(N2CC3CC2(C(=O)O)CO3)=O)c2ccccc12 c1(C(N2C(C(N(C(C3CCOCC3)C)C)=O)C(C)C2)=O)ccc(O)c(F)c1 C1(CNC(c2cccc(COC)c2)=O)CN(C(=O)CC2COCCO2)CCCO1 N1(Cc2cc(OC)ns2)CCCOC(CNC(=O)CC23CCC(CC2)C3)C1 c1(OCC(=O)NCC(C2CC2)NC(C2CCCCO2)=O)ccc(F)cc1 N1(C(c2c(C)nns2)=O)CCC(NC(C2(Cl)CC2C(C)=O)=O)CC1 CC1(C)OCC2CC12C(=O)NC1CC(CNC(c2ccc(F)cc2Cl)=O)C(O)C1 C(=O)(CS(=O)(=O)C(C)C)NCCCN(C(C1Cc2nncn2C1)=O)CC c1(C(N(CC(C)NC(C2(n3cccn3)CCC2)=O)CC)=O)cnn(C2CC2)c1 c1(OCCC(=O)NCCOC2CCN(C(=O)CN3CSCC3=O)C2)ccccn1 c1(C(=O)NCCC2(O)CN(C(CNC(N)=O)=O)C2)c[nH]c2ccc(F)cc2c1=O C1(C(=O)NCCC2CCN(C(C(CCCC)C)=O)CC2)C2CCC3C(C2)CC13 C#Cc1ccc(N)c(C(=O)NCC2(C)CCCN(C(C3CCC3(F)F)=O)C2)c1 C1(NC(c2c(COC)ncs2)=O)CN(C(=O)CC2OCCCO2)CC2(CC2)C1 C12(C(=O)NCCN(C(=O)C(F)(F)c3nc(C)cs3)CCC)CCC(OC)C1C2 CC(CC1CCC1)C(=O)NCC1CCN1C(c1csc(-c2ccccn2)n1)=O C1(CC(N2CCC(CF)(NC(C34COCC3C4)=O)C2)=O)(CN(C)C)CCCCC1 N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(c2ccc(C)s2)=O)CC1C1CCC1 c1(OCC)cncc(C(=O)NCCC(F)Cn2cc(-c3cccc(F)c3)nn2)c1 CCCCS(=O)(=O)NC(C)C(N1CCOCC1CN(C)C(c1scnc1Cl)=O)=O C1(C(=O)NCCC2CCC(=O)N2)(CNC(C2CCC(=O)C2)=O)CC12CCC2 C(=O)(CCCC(=O)N1CC(N(C)C(c2nc(CC)oc2C)=O)C(C)(C)C1)OCC S(=O)(=O)(c1ccc(NCC2CCCO2)cc1Cl)NC1C(C)(C)S(=O)(=O)CC1 n1(CC)ncc(C(N2CCCC(NC(c3ccc(CCO)cc3)=O)C2)=O)c1Cl N1(CC(=O)NCCCC)CCC(OCCCNc2cnn(C)c2)C1 CC(CC(=O)NC(C(=O)NCC1CC1CO)C1CC1)n1cccc1 N1(C(c2cc(O)cc(F)c2)=O)CCCC2(C1)CN(C(C1(CF)CC(F)(F)C1)=O)C2 C(=O)(CCC[N+](=O)[O-])N1CCC(N(C)C(C2CCCS2)=O)C1 c1(CC)ccc(NC)cc1[N+](=O)[O-].N12CCC(C1)CNC(=O)CC1(CCC1)C2=O c1(C(=O)NC(C2(O)CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)C)cccn2ccnc12 C(=O)(CS(=O)(=O)CC(F)(F)F)NCC(CC(C)C)NC(c1cc(CC)ncn1)=O c1(CC(C)C)ccc(C(N2CCC2c2cn(-c3cnn(C)c3)nn2)=O)s1 Cc1cc(C(=O)NC2(C)CCN(C(C3CCC(F)(F)C3)=O)C2)cc(C)c1N n1(CCC)cc(C(C(=O)Nc2ccccc2)N(C2C3CCCC23)C)cn1 N1(C(C(C)OCC=C)=O)CC2CC(C1)C2NC(=O)C(F)C1CC1 Cn1nnc2cc(C(N3CCC(NC(C4CC4(C)Br)=O)C4(CCC4)C3)=O)ccc12 C1(C(C(=O)NCC2CC2)N(C)CC2CCN(C)C2)CC12CCOCC2 c1(CNC(C2CCN(C(C3(C)C(C)CCC3)=O)CC2)=O)c[nH]c2ccccc12 CC(CNC(=O)C(C1CC1)C1CC1)C(=O)N1CC(O)(c2cc[nH]n2)C1 Cc1cnn(CC(=O)NCC2(O)CC(C(=O)NCc3ncc(C)o3)C2)c1 N1(Cc2nc(C)c(C)s2)CCC2(CN(C(C3CC4CCC3C4)=O)CC(C)O2)C1 c1(OC)cccc(CNC(=O)C(=O)Nc2ccc(Oc3ccncn3)cc2)c1Cl c1(C(=O)NCC(C)NC(c2c(CC)occ2)=O)nc(Br)cn1C(F)(F)F N1(C(C(CC=C)OC)=O)CCC(C2CC2)C1C(=O)NCC(C)C1CCC1 N1(C(c2nccc(C#C)c2)=O)CCC(NC(C2CC(C)(C)CN2C)=O)C12CCC2 C(CCC(=O)NC1CCCCC1)N(C)C(C1CCCCS1)=O C(CCC(C)C)(C(=O)NC(C)CO)NC(c1c(C)cccc1)=O CC1CCC(=CC(N2CCC2NCCN(C(=O)C(N2CCC(C)C2)=O)C)=O)C1 c1(COCC)nc(C(=O)NC2(C)CCCC2)cs1.C1(C(=O)N)CCSC1.C1(=O)CN1 CN(C(=NCCCc1cccs1)NCC1CCOC1)CCC1CCCCC1 C#CCC(CC(F)F)C(=O)N1CCOCC1CC(=O)NCC(C)C(C)(F)F C(c1cnc(C)nc1O)=CC(=O)OOC(C(C(C)C)Oc1cc(C)[nH]n1)=O C=C(Cl)C(C)(C)C(=O)N1CCC(C)C(NC(=O)Cc2ccoc2)C1 CC1CCc2[nH]c(C(=O)NCC3CC3NC(c3cc(Cl)ccc3O)=O)cc2C1 N1(C(CCC(=C)Cl)=O)CCN(C(=O)C(F)(F)c2cncs2)CC1CCO N1(C(C(F)=CC)=O)CC2CCOC2(CNC(c2cn3ccccc3n2)=O)C1 c1(CC(=O)NCC2CC(NC(c3cc(C)c(C)nn3)=O)C2)ccc2sccc2c1 c1(C(=O)NCCN(C)C(c2ccc(Br)cc2Cl)=O)ccc(O)c(N)n1 O=C(Cc1cccc(NCc2cc(Br)cc(Br)c2O)c1)N=c1ccnc(Br)[nH]1 N1(C(CCNS(CC)(=O)=O)=O)CCC(O)(CN(C(=O)C=CC(F)(F)F)C)C1 C1(O)(CCNC(C2C(=C)C2)=O)CCCN(C(=O)Cc2ccccc2C#N)C1 C12(NC(C=CCOC)=O)CCCCC1CN(C(c1cccn3nnnc13)=O)C2 Cc1oncc1C(=O)NCC(=O)NC(C)CCCNC(c1ccc(F)o1)=O N#Cc1cnn(CC(=O)NCc2cccc(NC(C3CC(F)C(=O)N3)=O)c2)c1N C(=O)(C(O)CNC(c1occc1C1CC1)=O)NC(COC)C1CC1 c1(CC(=O)OCCCSCC=C)cccc(F)c1F C#Cc1ccc(C(N2CC(CNC(c3cncc(Cl)c3)=O)C(O)C2)=O)c(C)c1 C1(NC(Cc2c(C)n[nH]c2)=O)CC2C(NC(=O)C(C(C)C)n3ccnc3)C2C1 Cc1ccc(C#N)cc1C(=O)NC(C)(C)CCNC(=O)CN1CCCC1=O CCCCC(=O)NC1CCC(C(=O)NC(C)C(F)F)C1 CCC(C(=O)NCCCSCCO)NC(c1cc(CO)on1)=O c1(OC)ccc(NC(C2CCCC2C2CCCC2)=O)c(P(C)(C)=O)c1 C1(NC(CC2(CC)CCC2)=O)CCC(CNC(C2(C(=O)N(C)C)CC2)=O)C1 c1(C(=O)NCCCCCNC(c2c(C)onc2Cl)=O)cc2c(Cl)nccc2o1 C12(C(=O)NCC3CCCN(C(C(CC)C4CCOCC4)=O)C3)CCOC(C)(C1)C2 N1(C(c2c(C)nc(CO)o2)=O)CCC2CC2(NC(=O)COC(F)F)CC1 Cn1cnc(C(=O)NC2CCCN(C(=O)OC(C)(C)C)CC2)cc1=O c1(-c2n(CCC)nc(CCCO)n2)ccc(OC)c(-c2ccccn2)c1 c1(CC#N)cccc(C(=O)NC2CCOC2C(=O)NC(CO)CCO)c1 Fc1cc(-c2ocnc2Cc2cccnc2)ccc1Cl c1(C(N2C(CNC(CC(C)(C)O)=O)COCC2)=O)ccc(Cl)cc1[N+](=O)[O-] Cc1noc(C)c1C(=O)NCCC1CC(NC(=O)CC2(N(C)C)CCC2)C1 c1(OC)cc(F)ccc1C(=O)NC(C)CCCNC(=O)Cc1cccc(SC)c1 CCCC(C(=O)NCC1(C)CCCN1C(c1cc(CCC(=O)OC)on1)=O)OC C1(CCOC)(NC(c2nc(C)cs2)=O)CCN(C(C2COC(=O)C2)=O)CC1 C(=O)(C(F)(F)C(O)CC)NCC1(CNC(CC(CC)c2ccccc2)=O)CCC1 c1(SCN2CC(=O)NC2=O)cc(C(=O)O)c2n1CCOC2 CC(C)(CCNC(=O)C=CI)NC(c1ccccn1)=O c1(C(N2CC(C3CN(C(CC4CC(=O)C4)=O)C3)C2)=O)cc(F)c(F)c(F)c1F CCCS(=O)(=O)C(C)C(=O)NCC(C)NC(=O)C=Cc1ccc(OC(C)C)cc1 c1(C(N2C(C)C(NC(=O)C=C(C3CC3)C3CC3)CCC2)=O)ccc2c(c1)CCO2 N1(C(CN(CC)CC)=O)CCCC1C(C)NC(=O)CCn1cc(Br)cn1 C(C(N=[N+]=[N-])C(=O)N1CCC(NC(C2CCCO2)=O)C1(C)C)OCC C(C(=O)NC1CCC(F)(F)CC1)(C(C)CCC=C(C)C)N(C(C)COC)CC=C c1(C(=O)NC(CN(C(C(=C(C)C2CC2)F)=O)C)(C)C)ccccc1F CC1C(NC(c2n[nH]c(O)n2)=O)CC2CCC1N2C(c1ccc2c(c1)CC2)=O c1(C(=O)NCCOCCNC(C2N(C(C)=O)CCOC2)=O)cc(C)ccc1Cl C1(NC(c2cscn2)=O)Cc2ccccc2C1NC(c1cccc(F)c1O)=O C1(NC(C=CCOC)=O)CCN(C(=O)C(C2CCCN(C)C2)(C)C)CCC1CO N1(Cc2[nH]nc(C(=O)OCC)n2)CCc2nc(Cl)cc(Cl)c2C1 C1(CNC(CS(CC)=O)=O)CN(C(c2cnn(CC(F)F)c2)=O)CC1(C)C N1(C(C(C)N(C)C(c2ncccc2Cl)=O)=O)CCN(C)CC(O)C1 N1(C(c2cc(SC)oc2C)=O)CC2CC1CC2NC(c1sccc1Cl)=O CCCC(CCC)CCCC(=O)N1CCOCC1CNC(C1CC(CC(F)F)C1)=O C12(C(=O)NC(C)(C)CNC(=O)C(C3CCOCC3)O)CCCC1OCC2 c1(C(N2CC(CNC(C(CC)C)=O)C(C)(C)CC2)=O)cc(F)c2ncccc2c1 CC(C)CC(C(=O)N1CCC(NC(C2CC3CCC2O3)=O)C1)c1ccc(Cl)cc1 O=C(C1=NN(C2CC2)C(=O)CC1)NC1C2CCC(C2)C1Cc1ccccc1 c1(CN(C(=O)NCCCCN2CC(C)OC(C)C2)C)ccc2c(c1)OC(F)(F)O2 C1(C(=O)N(C(CF)CF)C)(OC)CCN(C(C2CC(O)C(F)C2)=O)C1 C1(CNC(CCSCCC)=O)N(C(=O)CN2CCC(C)C2)CCC1(C)C C1(C(N(C2CCCN(C(=O)CCCCNC(N)=O)C2)CC)=O)CCC2(CCC2)O1 c1(C(=O)NC(CCCNC(C(=O)NCCOC)=O)C)c(F)ccc(F)c1O N1(C(CC(CC)C2CC2)=O)CC2(CO)CC1(C(N1CCC1(C)COC)=O)C2 c1(C(=O)OC)ccc(C(N2CCC(C(=O)Nc3ccc(Cl)o3)C(O)C2)=O)cc1O C(=O)(CCC(=O)NCC(C)(C1CC1)NC(=O)CCc1nc(C)cs1)N(CC)CC Cc1nccc(C(=O)NC(C)(C)C(C)NC(=O)CCc2cc(F)cc(F)c2)c1C c1(C(=O)Nc2cncc(C(=O)Nc3ncc[nH]3)c2)ccc2c(c1)CCO2 Cc1cc(NC(=O)NC2CC3CCC2C(N)C3)cc2ccoc12 c1(SC)ccc(N)cc1C(=O)NC(CNC(c1occc1F)=O)C1CC1 CC1CCCC(CC(=O)NCC(O)CNC(=O)C(O)C2CCCC2)O1 C#Cc1cc(F)c(C(=O)NCC2CN(C(c3onc4c3CCCC4)=O)C2)cc1F CCCC(C(=O)N1CC2(C)CC1(C(=O)NCC1(C)CCOC1C1CC1)C2)C(C)C C1(N(C(c2c(CC)cco2)=O)CC)CCN(c2ccccc2Cl)C1=O C1(NC(c2cc(CCC)on2)=O)CN(C(c2c(C)ccn2C)=O)CC1N=[N+]=[N-] CC(C)(C)C(C#N)C(=O)N1CC2(C(N3CC4(CC(F)(F)C4)C3)=O)CC1CCO2 C1(NC(C(CC)OC)=O)CCC2(CC1)CC2NC(c1c(C)nn(C)c1C)=O C1(NC(=O)CC2CCCC2)CCC2CCN(C(C3CCCCO3)=O)C12 n1(CCC)cc(-c2nc(CN3CCC(C)(O)CC3)nn2C2CC2)c2ccccc12 C(=O)(CCCC(=O)NCC1C(C)CCN1C(=O)CN(c1ncccn1)C)NCC C1(O)(CNC(CC=CC)=O)CC(NC(=O)C(C)(C)OC(C)=O)C1 c1(OCC)ccc(OC)c(C=CC(=O)NC2CN(C(=O)C3CC3)CC3(CC3)C2)c1 c1(-c2cn(N)nc2)c[nH]c2nc[nH]c(=NCC(CO)c3cccc(F)c3)c12 N1(C(C(C)OCC(C)C)=O)CCC(OCCNC(C2(S(N)(=O)=O)CC2)=O)CC1 Cc1ccc(F)c(C(N2CCCC2CNC(C2(CO)CCCCO2)=O)=O)c1 C1(C(C)NC(c2cnn(CC)n2)=O)CCCCN1C(c1occc1C)=O c1ccc2c(c1)OC1(CCOC1)CC2NS(=O)(=O)c1cccnc1NCCCF Nc1cc(F)c(Cl)cc1C(=O)NC1CCCC(NC(=O)CC2CC2)CC1 C1(C(=O)NCCCNC(=O)C(F)F)(OC)CC(C)CC(C)C1 N1(C(C(C#C)(C)C)=O)CCC(C2CCN(C(C34CC(O)C3C4)=O)C2)CC1 CCC(Cc1ccccc1)C(=O)N1CC2CC2(NC(c2ccn(C)c2C)=O)C1 c1(C(N2CCN(C(CNC(C(CC)C(C)O)=O)C)CC2)=O)nc2ncccn2n1 Cc1cc(C(=O)NC(CC2CC2)C(=O)NCCOCCN=[N+]=[N-])nc(O)n1 N1(C(CC(COC)C)=O)CC(CC(N2CCC23CC(C(N)=O)C3)=O)CC1(C)C CN1CC2(CC2)CC1C(N1CCCC1C(C)(C)C(=O)N1CCC(C(C)(C)C)C1)=O CC1CN(c2nnc(CC(F)(F)F)s2)CCC1NC(=O)Cc1c(O)ncnc1O N1(C(C(C)O)=O)CC(NC(=O)C(C)(C)O)Cc2ccccc21 C=CCC(CC=C)C(=O)N1CC(CNC(c2ncc(C3CC3)cc2F)=O)C(C)C1 C(=O)(C#CC1(C)COC1)N1C(CC(=O)NC2(C(N)=O)CCCCC2)CCCC1 CN1CC(NC(C2COCCC2NC(=O)C(O)C(F)(F)F)=O)CCC1=O N1(C(c2c(C)cc(F)c(N)c2)=O)CCC2(CCC2NC(=O)C(C)C2CC2)CC1 c1(C(=O)NCC2(C(C)CCO)CCC2)ccc(CN(C)C)cc1 N1(C(c2cc(F)ccc2F)=O)CCC(S(=O)(=O)NCC2CCCO2)CC1 N1(C(C(CC(=C)C)C)=O)CCCN(C(c2ccc(F)cc2NC(C)=O)=O)CC1C c1(CN(C)CC2CCCN(C(c3c(C(C)C)cccc3)=O)C2)c(F)cccc1Cl N1(C(C2CCOC2)=O)CCC(O)(Cn2cc(COc3ncccn3)nn2)C1 N1(C(CC=CCC)=O)CCC2CCN(C(=O)C(C)N(C)C)CC2C1 c1(OCCNCC(C)(O)C(=O)OCc2ccccc2)cccc([N+](=O)[O-])c1 N1(C(C(C(C)C)(C)O)=O)CC(NC(c2cccnc2OC(F)F)=O)CCC(O)C1 Cc1scc(C(=O)NC2(CNC(=O)CO)CC2)c1N c1(OC)cnc(F)c(C(N2CCC(NC(=O)CSc3ccc(F)c(F)c3)C2)=O)c1 N1(C(CCCCNC(=O)Cn2cnnn2)=O)CCN2CC(O)CC2C1 c1(C(C(=O)NCC2CN(C(CCCC)=O)CC2C)O)ccc2ccccc2c1 c1(CC)oc(C)cc1C(=O)N(CC(C)CNC(c1cn(C)nc1Br)=O)C C1(CC(=O)NCC(C)(C)N(C)C)CC2(C1)CN(C(C1CC3CCC1C3)=O)C2 c1(C(=O)NC2CCC(CNC(CN(C)S(N)(=O)=O)=O)C2)cc(-n2ccnc2)ccn1 N1(C(c2ncc(CC)s2)=O)CCC2(CC1)CN(C(=O)CC1CCCCO1)C2 Cc1ccc2c(C(N3CCC(CNC(C4(F)CC4C)=O)C34CCC4)=O)csc2c1 C1(C(N(C)CC2CCCN2C(C2(C#N)CC2(C)C)=O)=O)CC2(CCCC2)CO1 c1(CC(=O)NCCCCCNC(CN(CCC#C)C)=O)cccc(Br)c1F CCC(C(=O)NCCC1(NC(=O)CCOC)CC1)OC1CCCCC1 N1(C(c2ccc(OC)nn2)=O)CC(C2CCCN(C(c3n[nH]cc3C)=O)C2)C1 Cc1cc(C(=O)NCC2CN(C(C3CSCN3C)=O)CCO2)c(C)n1NC(N)=O C1(CC=CCNC(c2n(CC(=O)OC(C)(C)C)ncc2)=O)CCCC2C1C2(F)F N1(C(COCC(=O)NC)=O)CCC2(CCC2CNC(C2CC(OC)C2)=O)CC1 C1(NC2CC3(CCC3)C2)CCCCCC1F.C1(C)C(=O)N1CCC c1(-n2c(Cc3ccccc3)nc(C(C)C3CC3)n2)ccc(Cl)cc1Br Cc1sc(C)c(C(=O)NCCC2(O)CN(C(C3CC(C)(C)CN3C)=O)C2)c1C#N C1(NC(C(C)NC(CC)=O)=O)CCN(c2nc(OC)nc(OC)n2)C12CCCC2 c1(C(N2CCC(C)(CNC(CC3C(C)(C)C3)=O)C2)=O)cccc2ccc(O)nc12 c1(OCC)ncc(-c2cnc(C(N3CCC(C#N)C3)=O)c(C(F)(F)F)c2)cc1F C12(C(=O)NC(CC=CC(=O)NCc3nc(C)ncc3)(C)C)CCC(CC1)CC2 C(N=c1cc(NCCCCCN(C)C)nc[nH]1)c1cc(OC)ncn1 CCC(CC(C)C)C(=O)NC(C)(CO)C(=O)N1CCN(C(C)(C)C)CC1 N#Cc1ccc(C(=O)NC2C3CC2CN(C(=O)CN2C(=O)CNC2=O)C3)c(F)c1 c1(C(=O)NC2(CNC(CCc3cc(C)on3)=O)CCOCC2)ncc(Cl)nc1Cl c1(C(N(CCOC)CCNC(C2(C)CC=C(C)CC2)=O)=O)cc(F)cc2nn[nH]c12 C(C(C)(C)C(=O)NCc1ncc[nH]c1=O)N(C)C(C12CCC(C1)C2)=O N1(C(C23CC(C)(C2)C(C(F)(F)F)O3)=O)CCC2(CCOCC2)CC1 c1(NCC)cccc(C(=O)NCCNC(c2cc(CCOC)on2)=O)c1 c1(NC(C(CCCOC)NC(=O)C(C)O)=O)cccc2cnc(Cl)cc12 C(=O)(C(C)(C)CC(=O)OC)NCC(CC)NC(=O)C(C(C)(C)C)NC(N)=O C1(NC(C(CCC)NC(C)=O)=O)CC2CCCC(C1)N2C(=O)C(Cl)=CCl C1(NC(CCOC(C)C)=O)CN(C(c2cncc(Cl)c2)=O)CC1c1ccccc1 C1(NC(CCN(CCCCCC)CCC)=O)COCCN(C(=O)C(C)(C)O)C1 C1(C(=O)NC2CCN(C(c3ccon3)=O)C2C)(OC)CCCOC1 N1(C(c2c(C(C)(C)C)n[nH]c2)=O)CCC2(CC1)CC2NC(=O)CCc1cncs1 N1(C(c2c(C)nc(COC)s2)=O)CC=C(C(=O)O)CC1 CN1CC(O)CC1C(=O)N(C(C)(C)CC(=O)NCc1ncc[nH]c1=O)C c1(C(N(C(C)CNC(c2cnnn2C)=O)C)=O)cnn2c1CC(C)CC2 Cc1cccc(N(C)Cc2ccc(NC3CC4CCC3N4)cc2)n1 Cc1cn2c(n1)CN(C(=O)CCC(C)(C)NC(=O)CS(C)(=O)=O)CC2 N1(C(Cn2c(C)cnc2)=O)CCOC(CNC(=O)CCS(C)=O)C1 CCCCC(C(=O)N1CCC(NC(C2CC3(C2)CC3(F)F)=O)C1)N(C)C CC(C)CC(C(=O)NC1CC(NC(=O)COCc2nccn2C)C1)C(N)=O CC1CN(C(=NCC2CC2)NCC2CC3(CC3)C2)CC1C c1(C(=O)NC2C(C)CN(c3ncncc3I)C2)c(N)cccc1Cl C1(N(C(c2ccsc2C)C(=O)NCCC)CCOC)CCN(C(=O)NC)CC1 Cc1nc(Cl)cc(=NCC2CCCC(NC(c3ccc(-c4ccco4)s3)=O)C2)[nH]1 N1(C(c2c(C(C)C)nns2)=O)CCC(O)(CNC(=O)Cc2ccno2)C1 C(c1cn(C2CC(NC(c3ccc(C4CCC4)cc3)=O)C2)nn1)=C(C)C C1(C2CC2)(NC(C2CC=CCC2)=O)CCN(C(C2(c3cccnc3)CC2)=O)C1 c1(C(=O)OC)cc(F)cc(C)c1NC(N1CCCCC1CSC1CCCO1)=O N1(C(C2(SC)CC(O)C2(C)C)=O)CCC(C)N(C(=O)OC(C)(C)C)CC1 CN1C(=O)CCCC1C(=O)NCC1(C(=O)NC2(CN(C)C)CC3CCCC23)CCC1 C1(CNC(C2C(C)CCCC2)=O)CC(C(=O)NC2CC2C(C)C)=NO1 N1(C(C2OCCN(C(CN3CC(C)(OC)C3)=O)CC2)=O)CC2CCOC(=O)C2C1 Cc1cc(C(=O)NCCNC(C2CCN(S(N)(=O)=O)CC2)=O)c2cnn(C)c2n1 C=C1CC(C)(C(=O)NC(C2CCCCC2)C(C)NC(=O)CC2CCCC2)C1 c1(C(=O)NCC(CNC(c2c(CC)con2)=O)C)c[nH]c2ncc(Br)cc12 C12(CNC(CCC=C)=O)CCC(CC1)N2C(=O)Cc1c(C)nn(C(F)F)c1C C1(C(=O)NCCCCCNC(C2CCC(C)(C)C2)=O)CCC(F)(F)CO1 C(=O)(CCCC(N)=O)NC1(NC(C2C(C(=O)OC)C2)=O)CC1 C1(NC(C2N(C(CCOCCC)=O)CCC2)=O)CC12CCOCC2 C(=O)(CCC(F)(F)Cn1cc(CN2CC3CC3C2)nn1)Nc1cc(=N)[nH]c(Cl)n1 N1(C(C(CCC)C)=O)CC2(C1)SCCC2NC(c1cc(CC)on1)=O C=CCCCC(=O)NC(C1(O)CCCCC1)C(=O)N1CC(OCC(F)F)C1 CN1CCC(C)(C(=O)NCC2CCN(C(=O)CCC3CCC(C(F)(F)F)O3)C2)C1=O Cc1sc(C(=O)NC(C)CCNC(c2nocc2Br)=O)nc1Br N1(CC(=O)N(CC(C(=O)N(C(C)C(C)C)CC)C)C)CCC(=O)CC1 C(CC(C)(C)C(=O)NC1COCC1NC(c1ccsc1COC)=O)OC N1(C(c2c(C)cncc2C)=O)CCC(C(=O)NC2CCCCCC2CO)C(C)(C)C1 c1(C(n2nnnc2C(CCc2ccccc2)NC2CC(C(N)=O)C2)C)ccccc1 c1(CC)cc(C(N2CCC(C(C)NC(=O)C3CC3)C2)=O)on1 c1(OC)ccc(F)cc1C(=O)NC(C)C(C1CCCCC1)NC(=O)CCF C1(C)(CC)CCN(C(=NCC(O)c2cccc(OC(F)F)c2)NC(CC)CC)C1 c1(C(=O)NC(CN(C(c2c(COC)nn(C)c2Cl)=O)C)C)cc(C#N)ccc1F c1(OC)cc2c(cc1C(N1CCCCC1C(C)NC(C1(CO)CC1)=O)=O)OCO2 C1(CC)CCCC(c2nnnn2CCN2C(=O)CNC2=O)(NC)C1.C1(C)(CC)CC1 c1(SC)cccc(C(=O)NCC2CCN2C(c2cc(C(N)=O)co2)=O)c1 C(CCCO)N(C(=O)C(C)N(C(C1CC(CC2CC2)C1)=O)C1CC1)CC C(=O)(CC(CC)C(C)C)NCC(CC)NC(=O)CCN(S(C)(=O)=O)C c1(C(N(CC(CN(C(=O)CC2CCCCC2)C)O)C)=O)cc([N+](=O)[O-])n[nH]1 C1(SCC(=O)NCC=CCNC(=O)CCc2cocn2)CCOC1=O C1(NC(CCC=C(C)C)=O)CN(C(=O)CC2CN(C)C2)CC1c1ccccc1F N1(C(C=CC(CC)C)=O)CCOCC1CN(C(=O)CCc1cccnc1)CC C1(C(=O)NC(C(=O)OC)C2CC2)CC2CN(C(=O)COCc3nc[nH]n3)CC2C1 C(=O)(C1=C(C)OCC1)NCC(CCOC)NC(C1CCCN(S(C)(=O)=O)C1)=O c1(CS(OC2C(CCC3N(CC)CCCC3)C=CC2)(=O)=O)nn(C)c(Br)c1C CC(C)(C)CCCCC(=O)NCC1CCN1C(C1(C)COCc2sccc21)=O c1(NC(CC(=C)C)CO)ncc(S(=O)(=O)NCCCN=c2nccc[nH]2)cc1Cl CCC(C)C(C(=O)NC(C)CCCCNC(=O)CCC(=O)c1ccc[nH]1)NC(C)=O CC1(C)CCCCC1C(=O)NCCNC(c1cc(Cl)no1)=O c1(C(=O)NCCC(C)O)cc(CNC(=O)C=CCN2CCC2)[nH]n1 N1(C(c2nc(C)nn2C)=O)CC=C(c2c(C)[nH]c3ccccc23)CC1 C=CCC(CNC(=O)CCc1cnc(C)o1)NC(c1cc(C2CCOC2)[nH]n1)=O N1(C(c2nc(OC)c(F)cn2)=O)CC2CC(NC(C3CCCN3C)=O)CC1C2 N1(C(c2n(C)ncc2)=O)CCCC2CN(C(=O)CC3(C)CC(F)(F)C3)CCC12 C(=O)(C(CO)C(C)(C)C)NCc1cc(C(N2CCCC(=C)C2)=O)on1 c1(C(=O)NCC2C(CNC(CSCC)=O)C2)ccc2cccc(F)c2n1 CCC(CC(=O)N1CC2C(N(C)C)C2C1)N(C(=O)CCC(C)SC)C c1(C(=O)NC2CC(NC(Cc3c(C)con3)=O)C23CCC3)cncc([N+](=O)[O-])c1 c1(CNC(CCCOCC)=O)cnn(C)c1C(=O)NCC1CC(CO)CO1 N1(C(Cc2c(C)nn(C)c2C)=O)CC(C)CN(C(=O)CC2(C)CC2)C(C)C1 c1(NCCc2c(OC)cccc2)cc(=NC2C=CCCC2)[nH]c(CC(C)C)n1.C1(N)CC1 C1(C)(CCNC(C(CC)F)=O)CCN(C(c2ccc(C(C)C)cn2)=O)CC1 c1(C(=O)NC(C2(CC(=O)OC)CCCC2)=O)ccc(SC)cc1OC C1(C(=O)NCC(O)CCNC(=O)CCCN2CCCC2)(NC(C)=O)CCCC1 CC1(C)CC1(C(=O)NCC(O)C(N)=O)NC(C1CC(O)C1)=O C1(CNC(c2ccc(N)cc2)=O)CC2CCC1N2C(=O)C=Cc1ccccc1 C#CC1(C(=O)NCCc2nccn2C)CCN(C(=O)C(C)N(C)C)C1 N1(C(c2cc(C)cc(O)c2)=O)CCC(C)N(C(=O)CC(=O)N(C)C)CC1 S(=O)(=O)(c1c(OC)cc(C(=O)O)cc1OC)N1CC2N(C(COC)=O)C2C1 CC1CN(C(=O)CCNS(C)(=O)=O)CC(C)C1NC(c1snc2ccccc12)=O N1(C(c2nscc2Br)C(=O)NCCC#N)CCCC(N2CCCC2)C1 CC1(O)CCN(C(C2(C)CN(C(C3C4CC5C(C4)C35)=O)C2)=O)CC1 c1(OCC(N2CC(F)(CNC(C3CC(C)C3)=O)C2)=O)cccc(O)c1 CCCC(CCC)C(=O)NCc1ccc(C(N2CC(CO)C(O)C2)=O)cc1 C#CC1(C(=O)NCC(=O)NCCO)CCN(C(=O)C=C2CCC(C)CC2)C1 c1(C(=O)NC2C(NC(C(C3CCCCC3)OC)=O)C2)cc(F)c(Cl)c([N+](=O)[O-])c1 C1(C(N2CCC(C)(CCNC(C3(C(N(C)C)=O)CC3)=O)C2)=O)CCCCN1N=O O=C(CCCn1cccn1)Nc1ccsc1C(F)(F)F c1(C(=O)NC2CC(NC(C=CC(CC)C)=O)C(O)C2)ccc2ccncc2n1 c1(C(N2C(C)CC(NC(CC=CC=C)=O)C2)=O)cccc2c1COC2 C1(NC(C2(COC)CCCCCC2)c2n(C)nnn2)CCOC2(CCOCC2)C1 C1(CC)(NC(C2CCSC2)=O)CCCN(C(c2ccc(C(=O)OC)nc2)=O)C1 C(=O)(CCCC(=O)N(C)C)N1CCC(NC(COCc2c(C)ncs2)=O)C1C c1(C(N(C)C)=O)ccc(NC(C2CCC3CC23)=O)cn1 N1(C(C(C)n2ccnc2)=O)CC(O)CC1C(=O)NOCCCN(C)C Cc1c[nH]c2ncnc(N3CCCC(CNC(=O)Cc4ccc(Br)cc4Cl)C3)c12 c1(C(=O)NCC(C)NC(CCOCCCOC)=O)ccc2c(c1)OCCNC2=O N1(C(CN(C(=O)OC)C)=O)CC2CC1(CNC(=O)CC1CCCN(C)C1)C2 Cc1nc2c(o1)CCN(N1CC(C)S(=O)N(C)C1)C2c1ccccc1 C(=O)(C(C)(C)F)N1CC(NC(COCC(=O)NC(c2nccn2C)C)=O)C1 C(=O)(CC(C(C)C)c1ccon1)NCC1(CCNC(CCCC=C)=O)CC1 CCCCC(CCCC)C(=O)NCC1C(CC)CCN1C(C1CC1C1CC1)=O Cc1cc(C(N2CCCCC2CCNC(C2CC2(C)C)=O)=O)cc2c[nH]nc12 c1(C(C2CC3(CSC3)C2)=O)cccc(Cl)c1C.C12(C)CCCN1ONCc1cn2nn1 C(=O)(C1(C)CCCc2ccccc21)N(CC(CN(C(CCCCOC)=O)C)O)C C(CCCCC(=O)N1CCC(c2nn[nH]n2)C1)NC(c1cc(C)ncc1)=O C1(F)(CNC(C(CC)(C)O)=O)CCCN(C(=O)COc2ccc(C)c(C)c2)C1 Cc1ccc2oc(C(N3CCCC3CN(C(=O)CC3CCC3)C3CC3)=O)cc2c1 c1(CN2CC2)nc2c(s1)CC(C(C)(C)O)CC2.Cc1cc(-n2cncn2)cc(C)c1 c1(CC(=O)NC23C(CN(C(C4(N(C)C)CC4)=O)C2)C3)ccc(F)cc1[N+](=O)[O-] C(=O)(C(C)(C)CC(=O)N(CC(C)CNC(=O)CC(C(F)F)n1cccn1)C)OC C12CCCCN1C(=O)C(CC)N(CC)CCC2.C(C(=O)NCC)OCC#C C1(N(C(=O)CCCCCF)C)CCC2CN(C(c3csc(F)c3)=O)CC12 C(F)(c1ccccc1)=CC(=O)N(CCCNC(CCSCC(C)C)=O)CCO c1(-c2cn(CCCCC(=O)NCC(C(=O)OC)OC)nn2)cc(CO)ccc1C O=C(N=c1nc2cc(Br)ccn2[nH]1)N1CCN2C(=O)CCC2C1 C1(CC)C(NC(C23CSCC2C3)=O)CCCN1C(c1ccn(CCF)n1)=O N(C1c2ccccc2CC1NC(=O)C=CC1CCCO1)C(CC1(CSC)CC1)=O C1(C(=O)NC2(CCNC(C(OC)OC)=O)CCCC2)CN2CCN1CC2 c1(CC)nc(Cl)[nH]c(=NCCOCCN(C(=O)CC2CC3CC3C2)C)c1Cl N1(C(C2C(C)(CC)C2)=O)CCC2CCN(C(=O)COC3CCCC3)C2C1 c1(C(C)C)ccc(C(C)C(=O)NCc2csc(-c3ccccc3)n2)cc1 N1(C(CN(C)C(N)=O)=O)CCCC1CCCNC(C1CCC1(C)C)=O C1(N(C(=O)C(C)(C)C)C)CCC2(CC1)CC2NC(=O)CSC(C)(C)C c1(C(=O)NC2CCC(NCc3cc(C)c(F)nc3)C2)cc2[nH]ccc2cc1Cl c1(C(c2n(C)nnn2)NCC2=CCCC2)ccc(S(N)(=O)=O)o1 c1(CNC(C2CC2Cl)=O)n[nH]c2c1CN(C(c1c[nH]c3cccnc13)=O)CC2 N1(c2cccc(CC)c2)C(=S)NC(c2c(Br)cnc(Cl)c2F)C(C(C)C)=C1C N1(CCC(=O)NC(C)CC2CN(C(=O)C=CC3CCC3)C2)CCCCC1 C(CCC(CCC)NC(c1ccc(N(C)C(C)=O)cc1)=O)NC(CCCC#C)=O N1(C(C2(CC(C)C)CC2)=O)CC(CNC(=O)CC2CN(C(C)C)C2)C1 Cc1ccc(Cl)c(C(=O)NCC2(C)CCN(C(=O)C(C)NS(C)(=O)=O)C2)c1N C(CC(C(=O)NCC(=O)NCC(C)C)NC(=O)C(n1ccc(C)n1)C)=CC N1(C(C2C(C(=O)OC)C2)=O)CCOCC(NC(=O)C(C)(C)C(C)C)C1 N1(C(Cc2c(C)ccs2)=O)CCC2C1CCN2C(C1CC1c1ccccc1)=O O=C(CC(F)(F)C(F)(F)F)N1CCCC(n2cc(CO)nn2)C1 c1(NC(C2CC2NCc2ccc([N+](=O)[O-])cn2)=O)ccc(I)cc1[N+](=O)[O-] c1(-n2c(COCCCC)nc(CO)n2)cc(F)cc(F)c1 c1(C(CNC(N(C(c2ccccn2)CCC)C)=O)(F)F)c(C)noc1C c1(C(=O)NC2CCCN(C(c3ccc(C(N)=O)s3)=O)C2)ccc2nc(O)oc2c1 N1(C(C2CCN(CC)C2)=O)CCC2(CCN(C(=O)CCCC(F)(F)F)C2)C1 C(CC(=O)NCC1(NC(C2CC(C)(C)CN2C)=O)CC1)(C(N)=O)NC(C)=O c1(CC(=O)NCC(CC)(C)NC(C2NC(=O)OC2C)=O)ccc(Cl)nc1 C1(C(=O)NC(c2cccnc2)C)(NC(C2C(C)=CCS2)=O)CCCC1C c1(C(=O)NCC2C(NC(c3c(C)nc(C)[nH]3)=O)COC2)cncc([N+](=O)[O-])c1 C1(CNC(C(C)(C)NC(N)=O)=O)CC2(CC2)CN1C(=O)C(C1CCCCC1)O C1(NC(CSCC=C)=O)CCCN(C(=O)CCN(CCCCC)C)CCC1 C(=O)(CC(C)(C)CC(F)(F)F)NC1(C)CCC(NC(C(C(C)C)C)=O)CC1 C1(C(=O)NC(c2c[nH]ccc2=O)C)CCN(C(=O)Cn2cncn2)C12CCC2 C1(NC(c2c(CC)ccs2)=O)CCN(C(=O)C(C)(C)C(=O)N(C)C)CC1C c1(CC)ncc(Cl)c(C(=O)NC(C)CC(C)NC(c2nnsc2C)=O)n1 C1(C(=O)NC2CCCCN(C(CCC(=O)NC)=O)C2)CCc2c(n[nH]c2C)C1 c1(C(N2CCC(CCNC(C=CCC)=O)C2)=O)cc2cccnc2s1 C=CCCC(F)(F)C(=O)NC(CNC(c1ccccc1NC)=O)CO C1(CNC(=O)CC2(C(F)F)CC2)C2CN(C(c3cscn3)=O)CC12 N1(C(C2(OC)CCOC2)=O)CCC(CNC(c2cnc(C#N)s2)=O)CC1 Cc1csc(C(c2nnnn2C2CC2)NCCc2ncccn2)n1 N1(C(=O)CCn2cc(Cc3ccnc(CO)c3)nn2)CCC2(CCCC2)CC1 C1(CC=C)(C(N2CCOC(C(C)C)C2)=O)CCCN1C(=O)C(C)NC(N)=O c1(C(N2CCCC(CCC)C2)=O)ccc2c(n1)CN(C(C1(CO)CC1)=O)CC2 N1(C(CCC(C)C)=O)CCC2COC(CNC(c3ccc(C4CC4)cc3)=O)C2C1 Cc1ccc(C)c(C(C)NC(=O)Cc2ccccc2OCC(C)C)c1 c1(C(N(C2CC(NC(c3c(C)ncnc3)=O)C2)C)=O)cc2cccnn2n1 C1(C(N(CCCNC(=O)C(CCSC)NC=O)CC)=O)CC2(C1)NC(=O)NC2=O Cc1c(NC(=O)CC2CCN(c3ncc(C(F)(F)F)cn3)CC2)ccnc1Br c1(C(=O)NCC2N(C(C(C)C#N)=O)CCC2)cccn2ccnc12 N1(C(C(CC)n2cccn2)=O)CCN(C(=O)CC2CCCS2(=O)=O)CC1C c1(C(N(C2CCN(C(C3CC4(CC4)C3)=O)C2)C)=O)cc(O)ncc1Br CCC(C)(CNC(=O)C(Cc1ccccc1)OC)NC(C1(N(C)C)CC1)=O c1(C(=O)Nc2cc(Br)cc(OC)n2)n[nH]c2c1CN(Cc1ccc(Br)cn1)CC2 C(C(O)CC(F)(F)F)N(C1CCCN(C(N2C(c3nc(C)sc3)CCC2)=O)C1)C N1(C(CC(CC)(F)F)=O)CC2CC(NC(=O)CSc3ccncc3)CC(C2)C1 CC(CC(=O)NCCC1CCCN1C(=O)CCOCC1CC1)C(F)(F)F C1(C(C)O)CCC(NC(=O)C(c2ccccc2)NC(c2cnn(C)n2)=O)CC1 C1(C(=O)NCCCC(=C)Cl)CCN(C(C2CC(F)CN2C)=O)C(C)(C)C1 Cc1cccn2c(C(N3CCC(C)(CCNC(=O)C(C)O)C3)=O)cnc12 C1(NC(c2cnco2)=O)CN(C(=O)Cn2ncc(O)nc2=O)C2(CCC2)C1 c1(C(=O)NCC)ccc[n+]([O-])c1.C12CCCC1C(=O)NCCN(C)CC(=O)N2C CCC(CC)C(=O)N(CCNC(=O)CC1CC1(Cl)Cl)CC1CC1 N1(C(C2CC(OC)C2)=O)CCC2CN(C(c3sccc3-n3cccc3)=O)CC2C1 N1(C(c2nnn(CC)c2C)=O)CC2CC(NC(c3ccc(C(C)C)o3)=O)C(C2)C1 C1(N(C(c2ccc(SC)s2)=O)C)CCC(NC(=O)C(F)(F)c2nccs2)CC1 C12(C(=O)NCCCCCOC(=N)O)CCC(n3cc(C4CCC4)nn3)C1C2 CCCCS(=O)(=O)CC(=O)N1CCOC(CNC(=O)C(C)CSC)C1 N1(C(Cn2cc(C(C)O)nn2)=O)C(CNC(=O)Cc2nccn2C)CC2COCC12 C(CC(C)C(=O)NCC(CC(C)C)NC(c1cscc1Cl)=O)=CC C(O)(CCN=c1c(F)c[nH]cc1F)(C(=O)N(C)C)c1n(C)ccn1 C(N=C(NCc1cccs1)NCC1CCCOC1)c1nnn(C)n1 c1(SCC(=O)N(CCC)CCNC(C23CC(OC)C2C3)=O)c(F)cccc1Cl N1(C(C(n2c(C)ccn2)C)=O)CC2CC1CN2C(=O)CCc1cnn[nH]1 n1(C(C)C)cccc1C(=O)N(CC(C)N(C(=O)C=CC1CCOC1)C)C CC(C)(C)C(CC(=O)NCC1CCCCN1S(C)(=O)=O)C(F)F N1(C(CCc2cccc(OCC)c2)=O)CC2CCC(N)CC2C1 N1(C(COC(CC)(C)C)=O)CC(C2CC2C(=O)N(C2CCN(C)C(C)C2)C)C1 c1(C(CC(N2CCC(N(C(CCC)=O)CCO)C2)=O)C)ccccc1OC N1(C(C(C)C2CCCC2)=O)CC(CNC(=O)CC(=O)NC2CC2)CC1(C)C CCCC(C)(CCC)C(=O)NCC1CN(C(=O)C2=C(Cl)CCC2)CCC1(C)C N1(CC)C(=O)COC(C(=O)OC)C1c1ccncc1.N12CC(F)(C1)COCC2=O C1(CC)CCCCC1NC(C1(CC)CN(C(=O)COC(C)=O)C1)=O.C(C(C)(C)C)N CC1CN(CCCS(=O)(=O)N2CCOCC2)Cc2c[nH]nc21 O(NC(=O)C(C1(C)CC1)NC(C1CC1C(C)C)=O)CC(=O)OCC Cc1cccc(F)c1CC(=O)NC1CC(CNC(C2CCC(C)CC2)=O)C1(C)C N1(C(C(CCCOC)C)=O)CC2CCC(C1)N2C(C1CCC1C(C)(C)C)=O C1(=O)C(C(C)(C)C)CN1.CC(CCNC(N)=O)N(C(=O)C(=O)C1CCCC1)C C12(NC(c3c(C)cco3)=O)CCCCC1N(C(c1nc(O)nc(O)c1N)=O)CC2 C1(CNC(C(CC)C2CCC(=O)N2)=O)CCCN(CC2CCN(CC)C2)C1 c1(N2CC(C)C(NC(c3cc(C(F)(F)F)n[nH]3)=O)C2)ncccc1S(C)(=O)=O CC(C)CCCCCC(=O)NC(C)(C)C(N1CCC(N=[N+]=[N-])C1)=O CC1(C)CC1(C(=O)NCC1CC1[N+](=O)[O-])NC(=O)CCCC1CC1 C1(NC(c2c(CC)scc2)=O)C(CNC(=O)C=NOC)CCC12CCC2 CCC(CC)C(C)(c1nnnn1C(C)(C)C)NCC1CC(=O)NC(=O)C1 C1(C(=O)NCC(O)CC2CCC2)(CNC(C(OC)OC)=O)CC12CCC2 c1(NCCC(N2CC3(OCC(C)C3)C2)=O)cccc2c(=O)c3ccccc3[nH]c12 N1(C(c2nn(CC)c(O)c2)=O)CC(CO)C2(C1)CN(C(c1cc(Cl)cnn1)=O)C2 c1(C(N2CCCC(CN(C(=O)C3=CCC3)C)C2)=O)ccc(N)c(F)c1 N1(C(CCCCC=C)=O)CCCCCCC1C(N1CC(F)(F)CC1C)=O C1(NC(c2nncc(CCC)c2)=O)CC(CNC(=O)Cc2cnoc2)C12CCC2 c1(C(=O)NCC2(C)CCN(C(C(C)=C(CC)C)=O)CC2)ccc2nnn(O)c2c1 c1(NC2CCCN(C(COC)=O)C2)ccc([N+](=O)[O-])cc1Br Cc1ccccc1OCC(N1CCC(O)(CNC(c2c(C3CC3)nnn2C)=O)C1)=O c1(C(=O)NC2CCC(CCNC(C3C(C)(C)C3)=O)C2)nnc(Cl)cc1N C1(NC(=O)Cn2cccnc2=O)CC12CCN(C(=O)C(F)C1CCC1)CC2 C12(C(N3CCC(CNC(C(C4CCC4)OC)=O)CC3)=O)CC1COC2(C)C Cc1cc(C(=O)NCC(F)CNC(=O)C(C)C(F)F)n(C)n1 N#Cc1cc(Cl)c(C(N2CCC(SC(F)(F)CF)CC2)=O)s1 c1(NC(C=CC(=O)NCC)=O)cc(C)cc(C)c1.c12ccc(o1)C(=O)NOC2 C1(OC2CN(C(C(CC)n3cncn3)=O)C2)CCN(C(C2CC2C(N)=O)=O)CC1 CCCC(C)CC(C(=O)NCCCF)N1CC(C(=O)OC(C)(C)C)C2(CC2)C1 C12(NC(=O)OC)CCCC1CN(C(=O)NCC13CCC(OC)(CC1)C3)C2 C=CC(CCC)CC(=O)N1CC=CC1CNC(c1ccc(CC(C)(C)O)s1)=O c1(-n2c(SC)ncc2)ccc(OCC(=O)N(CCc2nn[nH]n2)CC)cc1C c1(C(=O)NC(CNC(C(Br)=C(C)C)=O)C(C)C)cn(CC(=O)N(C)C)nc1C(F)F c1(C(N2CCC(C(C(N3CCC(OC)CC3)=O)(C)C)C2)=O)[nH]ccc(=O)c1C Cn1cc(C=CC(=O)NC(C)(C)CC(=O)NCCCCN(C)C2CC2)nn1 C(CCCC(CO)NC(C12CC(F)(C1)C2)=O)NC(c1c(Br)cn(CC)n1)=O C(CN=C(NCC1CC1)N1CCN2C(=O)OCC2C1)c1ccn(CC)n1 N1(C(C(c2cc(Br)co2)=O)=O)CC2OCC(NC(c3cnco3)=O)C2C1 C1(NC(c2c(C)oc(Cl)n2)=O)CC2CC(NC(C3CCCCC(=O)N3)=O)C1C2 c1(C(=O)OC)ccc2ccccc2c1N(C(=O)Cc1csc(SC)n1)C c1(OC)cc(C(N2CC3C(NC(=O)CCc4ccc(O)nc4)C3C2)=O)n(C)n1 N1(C(c2csc(C(F)F)n2)=O)CCN(C(c2coc(CC3CC3)n2)=O)C(CO)C1 C(=O)(C1=NOC(c2ccccc2)C1)N1CCCC(NC(C2C(CC(C)C)C2)=O)C1 C(=O)(CCCCC(C)C)N1CC(CNC(c2cnc(OC)nc2C)=O)(OC)C1 C=C1CC2CCC(C1)N2C(C1CC1CCOC)=O.C12(C)CC(C1)C(=O)N2 c1(N2C3C(NC(c4c(CC)nccn4)=O)(CCC3)CC2)ncc2ncn(C)c2n1 C12(CC(=O)N(C)CCNC(=O)Cn3cnc(-c4ccccc4)n3)COCC(C1)C2 C1(C2CCN(C(=O)CNC(=O)NC3CC3)CC2)(NC(CC2C(C)C2)=O)CC1 N1(C(c2c(C)cccc2Cl)=O)CCC2(CCCC2NC(=O)C(C)C2CC2)CC1 N1(C2CN(CC)C2)CCN(C(=O)C(c2ccnn2C)OC)CC1.C1(N)CCCC1CC C(c1cccc(C#N)c1)=CC(=O)NCC(C(C)C)(C)NC(=O)CC(C)F Cc1cc(C(N2CCN(C(=O)CN(C)C(N)=O)C(C3CC3)C2)=O)cc(O)c1 C(=O)(C(F)C(F)(F)C(F)(F)F)N(CCN(C(C(CC(C)C)C)=O)C)C(C)C O=C(C1CCCc2sccc21)NCC1(NC(C2CCCC23OCCO3)=O)CCC1 C(=O)(CC(C)C(F)(F)F)NC1N(C(C2(CNC(N)=O)CC2)=O)CCC(C)C1 CN1CC(=O)N(CC(N2CC(NC(c3cc(Cl)sc3Cl)=O)CC(O)C2)=O)C1=O c1(NC(C(N2CCC(C(=O)OCC)C2)c2cnc(Br)s2)=O)ccc(F)cc1 C12(CC)CN(C(c3cc(C)c[nH]3)=O)C(CNC(c3ccnc(OC(C)=O)c3)=O)(C1)C2 CCC(CC(=O)NCC1(O)CN(Cc2ccccc2)C1)C1CCCC1 C(CC)(C(O)C(F)F)NCC(CC1CCCO1)OC CC(C)CCC(O)C(=O)OCCSc1cc(NC(=O)OC(C)(C)C)cn1C CC1CC(C(=O)NCC(O)CSCC(F)(F)F)CCC1=O c1(C(=O)NC2CCN(C(c3[nH]cc(C)c3)=O)C2C)cc(=O)n(C)cn1 N1(C(c2n(C)nc(O)c2)=O)CCCN(C(=O)C=Cc2ccc(F)cc2)CCC1 C(=O)(CC(C(F)F)n1ccnc1)NC1C(NC(CN2CC(C)C2)=O)COC1 C1(NC(CCCC(C)O)=O)CCCCC12CCN(C(=O)CCc1cccnc1)C2 C=CC(C)(C)C(=O)N1CCC(C(N2CCS(=O)CC2C)=O)O1 N#Cc1ccc(CN2CCNCC2C(=O)N(C2CC2)Cc2ccco2)c(Cl)c1 c1(C(=O)OC)cc(OC)cc(OC)c1CN1CC(C(C)C)CCC1C C(CC(=O)NCC1CCCCC1NC(c1ccccc1C)=O)(C(N)=O)NC(C)=O c1(C(=O)NC2CCC(NC(=O)Cc3nc(F)ccc3Cl)C2)coc2ccccc12 c1(N(C(CCCC=C)=O)C2CCNC2)ncnc2ccc(OC)cc12 CC(CNC(C1CC(C)(C)CO1)=O)CC(=O)NCC(C)CC1CC1 C1(C(=O)NCCC2(NC(=O)CSC3CC3)CCCC2)CCc2ccc(F)cc2O1 C(c1ccc(F)c(F)c1)=CC(N1C(CC)C(NC(C2CC(OC)C2)=O)CC1)=O CCC(C)C(O)C(C)C(=O)NC(C)(CNC(=O)CC(C)C)CC(C)C c1(COCC(=O)NC2CCC(NC(c3cnc[nH]3)=O)C2)ccccc1Cl N1(C(C2N(C(C)C)CCC2)=O)Cc2occ(C(=O)NC(C)(C)CC3CCC3)c2C1 C1(NC(c2c(CC)c[nH]c2)=O)COC2(C1)CN(C(=O)CCCCN=[N+]=[N-])C2 C(=O)(CC(CNC(=O)C1=CCSC1)C1CCC1)NCCNC(CC)=O Cc1ccc(Br)cc1CCC(=O)NC(C)(CNC(C1C(C)C1C)=O)CO c1(C(N2C(C(=O)NCCC(C)(O)C3CC3)CC(F)C2)=O)cc(F)cnc1O C1(NC(c2[nH]nc3ncccc23)=O)CN(C(C2CCCS2(=O)=O)=O)CC2(CC2)C1 C1(C(N(C)CC2OCCN(C(c3ccnc(C)n3)=O)C2)=O)Cc2nnc(C)n2C1 C(=O)(C1=C(Cl)CCOC1)NC(C(N1CCCC(CC=C)C1)=O)CCN(C)C c1(C(N2CC(C)CC(OC)C2)=O)cc2c(cc1N)OCCO2 Cc1c(C(N2CC3CC2CN(C(c2ccc(=O)oc2)=O)C3)=O)cnc2ncnn12 C1(NC(c2n[nH]cc2I)=O)CC2CCC(C1)N2CC1CC1 Cc1cc2c(cnn2C)c(NCCc2ccc(F)cc2Br)c1C Cc1cc(Cl)ccc1CC(=O)NC(C)Cn1cc(-c2cn(C)nc2C(F)F)nn1 N1(C(C2CCC(C)(CC)O2)=O)CCC(C2CC2)C1CNC(=O)C=C(C)C(F)F c1(COC)nc(C)c(C(=O)NC2C=CC(CNC(C3(C(N)=O)CC3)=O)C2)s1 c1(C(=O)NC2C(NC(c3ccc(CC)nc3)=O)CCC2)nn(C)c2c1COCC2 CC(CCNC(=O)C(F)=CCNC(=O)OC(C)(C)C)NC(C1(C(F)F)CC1C)=O c1(CN(C(C)CCO)Cc2ccc(Br)cc2)cc2cc(Br)ccc2o1 N1(C(c2cc(Cl)cs2)=O)CC(C2(NC(C34CCCC3CC4)=O)CC2)C1 N#Cc1ccc(CN2CCC(O)(C(=O)Nc3c(F)ccc(F)c3F)CC2)cc1Br C=C(C)CCCC(=O)N1CC2CC(CNC(c3ccc(O)c(Cl)n3)=O)C2C1 N1(C(c2cnc(C)s2)C(=O)N2CCCC2)CCN(C(c2ccc(F)cc2)C)CC1 C1(NC(c2ccco2)=O)CCN(C(C2CCCC3CC23)=O)C12CCC2 c1(OCC)nc(C)cc(=NC(=O)C2CC(F)CN2Cc2cnn(C3CC3)c2)[nH]1 c1(OCC)sccc1C(=O)NC1CC(NC(=O)C(=O)NCC(F)(F)F)C1 C1(C(=O)NCCC(CNC(CCC=CC)=O)(C)C)CCCC(F)(F)C1 C1(CCNC(c2cn(CCC)nc2)=O)CN(C(=O)CCC2CCCOC2)CCO1 C1(N(C(=O)C=Cc2ccsc2)C)CCCN(C(c2cnn(C3CCC3)c2)=O)CC1 C(=O)(C(=O)C(C)(C)C)N1CC2C(CNC(C3C(C=C)C3)=O)C2C1 c1(C(=O)NCC2CCN(C(=O)CC3CC4(CCC4)C3)C2)cc(Cl)c(F)cc1F C1(C(=O)NCc2csnn2)CCN(C(=O)c2cccs2)O1 c1(NC(C)=O)cnc(C)c(C(=O)NC2C=CCN(C(c3ccc(F)o3)=O)C2)c1 N1(C(C(C)OCCCCCC)=O)CCCC2CN(C(c3csc(O)n3)=O)CCC12 C1(NC(CN(CC)CC)=O)CC(C)N(C(=O)CCC2CCC(O)CC2)C1 CCC(CC)C(C)C(=O)NC.C1(C(C)C)C(=O)N(C(C)C)CCN1C n1(CCC(=O)OCC)ncnc1C(C)NCC1CC1F c1(NC(=O)OCC)ccc(C(N2CCCC2c2ccc(-c3cc[nH]n3)o2)=O)cc1 c1(C(=O)Nc2cccc(N3CCN(C)CC3)c2)ccc(NC(N)=O)cc1OC c1(C(=O)NCC(C)CNC(=O)C=C2CCC(C)C2)cccc(O)c1F Cc1nn(CC(F)(F)F)c(C)c1C(C)NCc1nc(C(C)O)nn1C C1(CC)(NC(c2cc(N(C)C)ccn2)=O)CCCN(C(c2cccn2C)=O)C1 C(=O)(CCC(C)(C)C)N1C(C)C(NC(=O)C(C)(C)c2ccno2)CC1 C(CC(O)C(=O)N1CCSCC1CO)NC(c1ccnc(O)c1)=O c1(C(=O)NCC2(O)CN(C(CCSCCC)=O)C2)cc2c(ccn2C)[nH]1 c1(N2CCC(Oc3ccccc3)CC2)nc(N2CCOC(CF)C2)nc2c1CCC2 C1(C2CC2)(CNC(CCC2CCCN(C)C2)=O)CCN(C(=O)CC2CCCC2)C1 Cn1nccc1C(F)=CC(N1CCCC(CNC(C2(C3CCCO3)CC2)=O)C1)=O C(=O)(CC(F)(F)Cl)NCC1CCC(NC(C2(CC=C)COC2)=O)C1 C1(C(C)NC(CC=CC=C)=O)CCCCN1C(=O)CC1(C(=C)F)CCC1 c1(CCCC(=O)NCCCC(C)NC(C2(F)CCC2)=O)ccc(F)cc1 C1(NC(C2CC3(CCC3)C2)=O)CCCC12CN(C(c1ccco1)=O)C2 C1(NCC(N2C(C(=O)NC3CN(C(N)=O)C3)CCC2)=O)CC12CCCCC2 N1(C(COCC#C)=O)CCC(C)(NC(c2cnn(C(C)(C)C)c2N)=O)C1 N1(c2n(C3C(CC)CCCC3)c(C(=O)C3=C(C)OCC3)nn2)CCC2(CCC2)C(CO)C1 c1(OCC=C)cccnc1C(=O)N(CC(C)NC(c1cnc(C)[nH]1)=O)C c1(OC)cc(OC)c(C(=O)N(C2CCCN(C(=O)CCCC(C)C)C2)C)c(N)c1 c1(OC)cccc(-c2cc(COC(=O)C(C)(C)c3cc[nH]n3)n[nH]2)c1 CCCC(O)CC(=O)N1CCN(C(c2ncc(Br)cc2C)=O)C(C)C1 c1(C(=O)NCC(=O)NCC(N2CCC(c3cc[nH]n3)C2)=O)cncc(O)c1 N1(C(c2c(C)ccc(C)c2)=O)CCN(C(=O)CN=S(C)(C)=O)CC(O)C1 c1(C(N2CCOC(CCC(F)(F)F)C2)=O)cccc2[nH]ccc12 C(=O)(CCCS(N)(=O)=O)NCCC1CN(C(C2(C)CC(=C)C2)=O)C1 C1(C(N(C(CC(CC)C)C)C)=O)CCN(C(=O)C#CC(C)(C)C)CC1(C)C N1(C(CCC(C)C)=O)CC2CCCN(C(C3CCN(C4CC4)C3=O)=O)C2C1 N1(C(CC)=O)CC2(C(=O)OC)CC1(C(N1CC(CO)CC(C)C1)=O)C2 C#Cc1ccc(C(=O)N(CCC(C(C)(C)C)NC(C2CCC3(CC3)C2)=O)C)cc1 c1(C(C(N2C(C)(C)CC(C(=O)O)C2)=O)=O)cc(F)c(F)cc1F C1(NC(c2ccc(CCC)[nH]2)=O)CCCCC1NC(c1ccccc1C(C)=O)=O Cc1c(F)ccc(C(=O)NC(CNC(=O)C(F)(F)C2(O)CCC2)CC(C)C)c1N C(N=c1ncc(Cl)c[nH]1)c1ccc(NCCCNC(C(C(C)(C)O)F)=O)cc1 N1(C(C(C=CC)O)=O)CCN(C(c2ncccc2N)=O)CC1CC(F)F C(CS(=O)c1ccccc1F)N1C(=O)NC(C)(C)C1=O.C1CC(=O)N1 C1(NC(C=C(C)Cl)=O)CCN(C(=O)CSCC2CCCCO2)C1C N1(C(C2(OC)CCOC2)=O)CCC(C2(O)CN(C(c3cncs3)=O)C2)CC1 C1(NC(C2C(Cc3c(OCC)cccc3)C2)=O)CC2(NC3CCN3C)COC1C2 C(C)(C(=O)N1CC2(CCC2CNC(=O)COc2cccnc2)C1)(C(C)C)NC(C)=O C=CC(O)C(=O)N(C(C)CN(C)C(c1cscc1Br)=O)C C12(C(N(C)CC3N(C(COCC(=O)NC)=O)CCC3)=O)CCCN(CC1)S2(=O)=O C1(NC(c2cc(C)nn2C)=O)COC2(CCN(Cc3c(F)cccc3Br)CC2)C1 C1(C(N(CC(C)NC(C(CC)NC(N)=O)=O)C)=O)CC(F)(F)CCC1(C)C N1(C(Cc2scc(C)c2)=O)CCC2CCN(C(C3CC3C(N)=O)=O)CC12 c1(C(=O)NC(CNC(C2CCC(c3ccccc3)O2)=O)CO)ncccc1F N12CCCC3CN(CC13)CC2=O.C12(CC3CCN(C(C)=O)C3)CC(C)(C1)OC2C N1(C(c2c(C)ccc(C)n2)=O)CCC2CC2(NC(C2CC3C=CC2CC3)=O)CC1 N1(C(C(C)SC)=O)CCN(C(C2CCc3c(cnn3C)C2)=O)C2(CCC2)C1 C(=O)(C1=CCCCCC1)N1CCC(CCCNC(c2cc(C)nc(C)n2)=O)CC1 c1(Cc2cc(C)sc2)nnc(N2CCC(Cc3ccc(C)s3)C2)n1C C(=O)(C(CC(C)CCC)N1CCOC(CF)C1)NC(CC)C C1(C(N2C(CNC(C(C)SCCCC)=O)C=CC2)=O)CCCCCC1 Cn1ccc(C(=O)NC(c2cccnc2)C(=O)NCC(O)C2(Cl)CC2)n1 c1(OCC(=O)NCC2(CNC(=O)CCC3CCOC3)CCC2)ccccc1F C1(CC#N)CN(Cc2cc[nH]n2)CCN1C(c1cc(C(F)(F)F)cc(Cl)c1)=O C1(C(=O)NC2(CN(C(C=CC(CC)C)=O)C)CC2)CCc2ccccc2C1 C1(C(=O)NCC=CCC(=O)NC2COC(=O)C2)COCCO1 C(CC(=O)Nc1csc(Cl)c1)(C(F)(F)F)NC(Cc1cn(CC)nn1)=O Cc1noc(C(C)(C)NC(=O)CC2C(NC(C3CCOC3C)=O)CC2O)n1 c1(OC(C)C)ccc(NC(C2CCC(NC(=O)C(C)NS(C)(=O)=O)C2)=O)cc1 c1(C(=O)NCC2CC(C)N(C(=O)Cc3sc(O)nc3O)C2)cncc2[nH]ccc12 N1(C(c2nc(CNC(c3ccc(C)nc3)=O)oc2)=O)CCC2(CNC(=O)C2)C1 C1(C(=O)NCC(N(C(CSC(C)C)=O)C)C2CC2)CCCN1C1CCCC1 N1(C(CC(C)C2CC2)=O)CC2CC(NC(=O)CSCc3cccs3)CC1C2 c1(C2C(C(=O)NC3CC3C(=O)NCc3ccoc3)C2)ccc2ccccc2c1 c1(N2C3CC(CN(C(C4CCC(C)C4)=O)C3)C2)ccc([N+](=O)[O-])cc1C(F)(F)F C(=O)(C(CC(C)C)N(C)C)OCCCN(CCCCNc1nc(C)n(C)n1)C c1(C(=O)NC(C(C)(C)NC(CCN(CCCCC)C)=O)C)oc(C2CC2)nc1C C(=O)(C(O)CCSC)N(C(C)CNC(c1cc(Cl)n[nH]1)=O)CC C=CC(C)(C)C(=O)NCCC1CN(C(C2CCCN(S(=O)(=O)CC)C2)=O)C1 O=C(CCCCCO)N1CCCC1C1CCN(C(C23CCCC2C3(F)F)=O)C1 c1(C(=O)NCC(CNC(c2nccc(C)c2)=O)C)cc(C)ccc1OC(F)(F)F c1(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCSC)cccc(C(C)(F)F)n1 C1(C(=O)NC2CC(F)(CNC(=O)Cc3cnn(C)c3)C2)(CC)CCOCC1 N1(C(c2cccc(C)n2)=O)CCC(NC(=O)CC2OCCC2(C)C)C(O)C1 c1(NC(C(C(C)=O)(C)C)=O)ncc(C2=CCSCC2)cn1 C1(COC)(CC2CC2)CCCN1C(=O)CCn1cc(-c2nccs2)nn1 C1(C)(C(N2C(C#C)CCC2)=O)CC(O)CN1C(C1CC1OC(C)=O)=O N1(C(CCOCCOC(C)(C)C)=O)CC2CCC2(CNC(c2sccc2Cl)=O)C1 Cc1cccc(Cl)c1CC(=O)N(CCCNC(c1cnn(CC(F)F)c1C)=O)C S(=O)(=O)(c1cccs1)NCC(N1CC(C2N(C(C(CC=C)C)=O)CCC2)(O)C1)=O CCC(C)(C#N)C(=O)NCC(C)NC(=O)C(C)(CO)NC(=O)OC(C)(C)C CC1(C)CCC(NC(=O)COc2ccsc2)CN1C(C1CC1C(F)(F)F)=O C1(C(C)C)(C(=O)NC(C)Cn2cncn2)CCCN1C(C12CSCC1C2)=O CCC(C)C(CC(=O)NC(COC)C(=O)OC)NC(=O)Cc1ccc(F)cc1 C(C(CC(C)C)NC(=O)Cc1csc(C)c1)NC(C(CN(CC)CC)F)=O CC1(NC(=O)CC2CC(=O)NC(=O)C2)CCCN(C(=O)CC2CCCCC2O)C1 Cc1nccc(C(=O)NCC2CCCC(NC(=O)CS(=O)(=O)N(C)C)C2)c1N c1(C(=O)NC(CC=C)CNC(=O)CCn2cnnn2)ccc(N(C)C(C)=O)cc1 C1(NC(C2(OC)CC2)=O)CCC2CC1CN2C(=O)CC1(CO)CCCC1 N1(C(C=C(C)Cl)=O)CCN(C2CCN(C(=O)C(O)CN(C)C)C2)CC1 c1(C(=O)NC2(CNC(c3c(C)ncs3)=O)CCC2)cnn2c1OCCCC2 C1(NC(CC(=C)C)=O)CN(C(C2CCC(Cn3ccnc3)O2)=O)C(C)(C)C1 CC(C)C1=NOC(C(=O)NC(C2CN(C(=O)C(C)(C)OC(C)C)C2)C)C1 N1(C(CC2(C#N)CC2)=O)CC2(CCN(C(C3CCCC3F)=O)CC2)C1 CCCCC(C(=O)NCc1ccon1)NC(=O)CCN1CCCCC1 c1(C(N(CCC)CCNC(=O)CCC2CCC(C)O2)=O)cc(O)cc([N+](=O)[O-])c1 N1(C(CC2CC(=C)C2)=O)CCC(CNC(c2csc(C(N)=O)n2)=O)(OC)C1 N1(C(c2cccnc2C)C(=O)NCCC)CCN(C)C2(CCN(C)CC2)C1 N1(C(c2ccc(C)cc2N)=O)CC=C(C(C)(C)C(=O)N2Cc3cccnc3C2)C1 C=C(C)CC(C(=O)N1CCC(O)(CC)C1)NC(C1CC(O)C(F)C1)=O c1(C(=O)NC2CCC(CCNC(CC(C)(F)F)=O)C2)noc2c1CCCCC2 c1(NC(C(C2(O)CN(C(Cc3c(C)cnn3C)=O)C2)F)=O)cc(Cl)cnc1O CCC(C)CC(=O)C(=O)N(CCC(N1CC(N(C)OC)C1)=O)CCO N1(C(C(C)OCCC=C)=O)CC(CO)(NC(=O)C(C)NC(N)=O)C1 c1(C(=O)OCC)cc(C(C(=O)NCC(=O)OC)NC(CC)C2CC2)ccc1O c1(C(N2CCCC(OC(C3(CSC)CC3)=O)C2)=O)c2ccc-2c1F.C(C)(C)O C(=O)(N=c1cc(-c2cccc(F)c2)[nH][nH]1)c1ccc(-n2c(C)cc(C)n2)cc1 c1(C(=O)NCC(CCCC)NC(c2oncc2C)=O)cc2c(C)cccc2o1 C1(NC(C2(C#N)CC=CC2)=O)CC12CCN(C(=O)COc1ccc(Cl)cc1)CC2 c1(CC(N2CC(CCN(C)C)C2)=O)ccnn1C.C(CC=O)NCC=C C1(C2(O)CCN(C(C3CC3F)=O)CC2)(NC(C(C(C)C)N(C)C)=O)CC1 N1(C(C2C=CCC2)=O)CCN(C(=O)C=Cc2cn[nH]c2)C(c2ccccc2Cl)C1 c1(C(N2CCN(C(CS(=O)(=O)NC)=O)C(C)C2)=O)cc(F)c(F)c(O)c1F C(=O)(C(C)(C)CC(=O)N1CCC(C(=O)Nc2cnn(C(F)F)c2)C1)OC C1(C)(C(=O)NCC2(C)CCN(C(CCCC=C)=O)C2)CC(C(F)(F)F)=NO1 c1(C(C(C)CCCC)=O)ccc(C(C)C(N2CCCC(OC)C2)=O)cc1 c1(OC)cc(C(=O)N(C2CN(C(C3CC(C)C3)=O)CCC2C)C)ccc1F c1(CC(=O)NCCC2CC(NC(C3CC4CC4C3)=O)C2)ccc(Cl)cn1 c1(CNC(c2coc3c2COC3)=O)c(F)cc(F)c(F)c1F C1(NC(C(C)CN(C)C(c2ocnc2C2CC2)=O)=O)CC2C(C1)C2(F)F N1(CCC)CCCCC1C(N1CCCC(CNC(=O)CC2CCN(C)CC2)C1)=O C(=O)(C1COc2ccccc21)N1CC(NC(C2C(C)(C)CCC2)=O)C(F)CC1 C1(C(=O)NCC2(NC(c3cc(C)nnc3O)=O)CCOC2)CN2CCN1C(C)C2 N1(C(C(=O)NCc2noc(CC(N3CC(SC)(CO)C3)=O)n2)C)CCC(O)CC1 C1(NC(c2c(C)onc2)=O)CCCN(C(C2CC(F)(F)CS2)=O)C1C N1(C(CSc2c(C)n[nH]c2C)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C(C)C1C C1(C(N(C2CN(C(c3nnc(O)nc3O)=O)C2)C)=O)COC2(CCC2)C1 C(=O)(CC(CC(C)C)NC(C1CC(C)CC(=O)N1)=O)NCC(CCOC)O N1(C(C=Cc2c(C)ccnc2)=O)C2CC1CN(C(=O)C(CCO)N(C)C)C2 CN1C(=O)CCCC1NC(C1CC1CC(=O)NCC(Cl)=CCl)=O c1(C(=O)NCC(=C2CN(C(C3CC=CCO3)=O)C2)F)c(Cl)nc2ccccn12 C(=O)(CCCN=[N+]=[N-])NCC1N(C(C2CCCC(C)O2)=O)CC(O)C1 CCCC(C(=O)NC(C)CC(N1CCOC(CO)C1)=O)NC(=O)OC(C)(C)C C=CCC(CC(C)C)C(=O)NCC1CN(C(=O)CC2CC(=O)C2)CC1O c1(C(=O)NC2CN(C(C(CC)(C)C(N)=O)=O)CC23CC3)cc2cnc(Cl)cc2s1 c1(C(=O)NC2(CNC(=O)CCN3CCC(F)C3)CCOC2)ccc([N+](=O)[O-])cc1 N1(C(C2CCC(C)(F)CC2)=O)CC(NC(C2(C(N)=O)CC2)=O)C(S(C)(=O)=O)C1 C#Cc1ccc(C2CC2C(=O)NC2(CNC(=O)C(C)(C)C(=C)C)CCOC2)cc1 C1(NC(c2cn(CCSC)nn2)=O)CCC(F)(F)CC1.C1C(C)C(=O)N1 Cc1ccc(OCC(=O)NC(C)(CNC(=O)Cn2cc(CO)nn2)CO)c(F)c1 C(CCCCCNC(C1CCC1c1nc(S)n[nH]1)=O)NC(=O)C(Cl)=CCl C1(CC)CN(C(=O)C(C)(C)N2CCCCC2)CCN1C(c1cc(F)ccc1O)=O CS(=O)(=O)c1sccc1CNC(C1CC2CC12)=O C(=O)(CC(C)(C)C)NC(C(=O)NCCCC1N(C(c2c(C)con2)=O)CCC1)C Cc1nc(C)c(CNC(=O)C(C2CCCC2)NC(c2cnn(C)c2N)=O)[nH]1 C1(C)(CNC(C2C(CC)C2)=O)CCCN1C(c1cc(C)c[nH]1)=O C1(CNC(C(CC)(F)F)=O)CCCC2(CN(C(C3(CCOC)CCCC3)=O)C2)O1 C1(C(=O)NC(CCOC)CNC(=O)C(C)=CC2CC2)CCS(=O)(=O)C1 c1(CCNC(N2CC(c3ccccc3)CC(C)C2)=O)cc(Cl)c2c(c1)OCCO2 c1(CN(C(c2cc(N3CCCC3)ccc2O)=O)CC2C(C)C2)cccc(C#N)c1 c1(N2CC(CCC)N(C(=O)OC(C)(C)C)CC2)cncc2nnnn12 C1(C(N2C3(CN(C(CNC(C)=O)=O)C3)CC2)=O)C(C)OCC(=O)N1Cc1ccco1 C1(C(=O)NC2(C)CCCC2)CC(F)(F)CC1CNC(=O)Cc1cnc(C2CC2)[nH]1 C12(C(NOCCOCC)=O)CCC(NC(=O)CCN(C)CCO)(CC1)C2 CCC(C)(C)CCCC(=O)N1CCCC1CN(C(=O)CCc1ccncc1)C c1(C(N2CCN(C(c3cc(C4CCC4)no3)=O)C3CC23)=O)nc2ncccn2n1 c1(C(=O)NOCC(=O)C2CC2)ccnc(F)c1Br C(CN=c1[nH]cncc1I)C1CCC(NC(c2cncc(OC)c2C)=O)C1 c1(CC(=O)NC(C)CCCCNC(=O)CCc2nnnn2C)ccc(F)c(F)c1 c1(OC)cccnc1C(=O)NC(CCN(C(=O)C(C)CO)C)c1cccs1 CCC(O)(CC)CCNC(=O)C(C(C)(C)O)NC(=O)Cn1cc(Cl)cn1 C#CCCC(C)(c1nnnn1C1CCOCC1)NCC1CCS(=O)CC1 N1(C(C2CCCCC2CC(F)(F)F)=O)CCn2ncc(O)c2C1 C(=O)(C1=CC(C)(C)C1)NCCC1CCN(C(C2C(C(C)C)CCO2)=O)C1 CC(C)C(F)(CNC(=O)C=Cc1ccc[nH]1)C(=O)NCC12CC(CO)(CO1)C2 CCCS(=O)(=O)NC(c1cn(-c2ccncc2)nn1)=O.n12cc(nn1)CCOCC2 CCC(C)(CNC(=O)Cn1ccnc1)C(=O)NCC(O)CC1CCC1 c1(OCC)ccccc1C=CC(=O)NC(C)C(C)Oc1ccc(F)cc1 Cc1cc(C(=O)NC2CCC(NC(c3oncc3C)=O)C2)c2cc(F)ccc2n1 C=CC(C)(C)CC(=O)NC1CC(CNC(c2ccnc(C)c2)=O)C1(C)C Cc1noc(C)c1C=CC(N1CC(NC(=O)C=C2CCC(C)(C)CC2)C(O)C1)=O C(=O)(C(CC(C)(C)C)OC)NC1CCN(C(CC=CC=C)=O)CC1O c1(N(C)CC2N(C(C(C)=C(CC)C)=O)CC=C2)ccc(C)c(C(=O)OC)c1 c1(C(=O)NCC2(C)CCC(NC(CN(CC)CC)=O)CC2)cc2n(c1)CCOC2 N1(C(C(C)(C)OCCC)=O)CC2C3CCC(C3)C12 CC(C)C(C(=O)NCC(C)(C)NC(=O)CCn1ccnn1)N(C)C C#Cc1cc(C(N2CC(NC(c3ccnnc3C)=O)CC2C)=O)cc(F)c1 C=CCC(C)(C)CC(=O)N1CCC(O)C(NC(C2CC3(CSC3)C2)=O)C1 Cc1cc(Cl)ccc1C(=O)NC1CCN(C(c2coc(C#N)c2)=O)CC1C c1(CCC(=O)N(C2CCC(NC(C=C(CC)CC)=O)CC2)C)ccc(C)c(C)c1 C1(SCCCCCC(=O)OC)CCC2(CCOCC2)CC1 C=CCCC(C)(C)C(=O)NCC(c1ccccc1)N(C)C(c1ncsc1C)=O c1(CNC2C(N(C(Cc3c(CC)ccs3)=O)C(C)=O)C2)c(OC)cccc1C Cn1ccc(-c2cn(Cc3ccc(C(N4CCC(O)C4)=O)o3)nn2)n1 C(C(C)C)(C(O)C(=O)NCC12CC(CO1)N(C(C1C3CC(=O)CC13)=O)C2)OC CCCCCCC(CC)C(=O)N1CCCCC1CNC(C1CC(=O)C1)=O CS(=O)(=O)CCC(=O)NCC1CN(C(=O)C=C(C2CC2)C2CC2)C2CC12 c1(C(N2CCC3(CC(NC(CC(C)O)=O)C3)C2)=O)ccc2[nH]c(=N)n(C)c2c1 C#CCCC(=O)NCCCOCCCNC(=O)C(c1ccn(C)c1)C c1(C(N(CCCCNC(c2c(CC)occ2C)=O)C)=O)cc(C#N)oc1C C#Cc1cnn(C)c1C(=O)NCc1cc(C(=O)NCC2CC[Si](C)(C)C2)no1 CC(CO)(C(=O)NC1CC(NC(=O)Cn2cncn2)C1)c1ccccc1 C(=O)(C(CCSC)NC(=O)CCCNC(c1cncc(Br)c1)=O)NC C1(CN(C)C(C2(F)CCCC2)=O)CCCC(NC(=O)CN2CCCC2=O)C1 N1(C(=O)Cc2cnc[nH]2)CCN(C2CCCN(C(c3ccco3)=O)C2)C(=O)C1 C(=O)(C1CCCc2c[nH]nc21)NC1CC(CNC(CNC(CC)=O)=O)C(O)C1 C=Cc1ccc(C(=O)N(CC(C)N(C)C(c2cc(CC(C)C)[nH]n2)=O)C)cc1 C(=O)(C(C)(C)CC(=O)N(CCCNC(C1CC(COC)C1)=O)C)OCC C(c1c(F)cccc1F)=CC(N1CCC(CNC(c2c(C)cc(C)o2)=O)C1)=O N1(C(CC(CC)C2CC2)=O)C(CNC(=O)C(F)(F)C(O)C2CC2)CC2COCC12 Cc1ccc(C(=O)NCC=CC(=O)NCCNC(=O)C=CC(C)C)c(F)c1 c1(C(N2CCC(NC(c3cc(CC)nn3C)=O)C2)=O)cc(C)n(C)c1C C12(NC(CN(C)C(N)=O)=O)CCCC(NC(=O)C(F)=C3CCCC3)(C1)C2 Cc1ccc(C(=O)NCC23CC(NC(=O)CCc4cnco4)(C2)C3)cn1 Nc1cccc(C(N2CC=CC2CNC(C2CCC3(CCC3)O2)=O)=O)c1Br c1(CC(=O)N(CC(C)NC(=O)CSCCC#N)C)ccc(-c2nc[nH]n2)cc1 Cc1c(N)ccc(C(N2CCC2CNC(C2CCCCC2(F)F)=O)=O)c1Cl C12(CCN(C(=O)CC=C(Cl)Cl)CC1)CCNC2=O.c1(C(COC)C)nccs1 N1(C(C(=O)OC)CC(C)C)CCC2(CCCN2S(=O)(=O)C2CC(SC)C2)CC1 C1(C(=O)NCC2C(CNC(c3cnc(O)s3)=O)C2)CCc2nc[nH]c2C1 C1(CC(=O)NCC(C)N(C)C(c2n[nH]cc2-c2ccncc2)=O)CCS(=O)(=O)C1 CC1(CO)CCN(C(=O)NN2CCCC2)C1 Cc1cc(Br)ncc1-c1ccc(NC(=O)CCC(=O)c2ccccn2)s1 C(CCC(F)(F)F)N(C(CCC1N(C(CCC=C)=O)CCC1)=O)C N1(C(CC(COC)C)=O)CC(NC(c2ccc(SCCCO)cc2)=O)CC(C)C1 C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)NCC1CCC1NC(c1cc(Cl)no1)=O c1(NC(CNC(c2ccccc2F)CCOC)=O)cccc2nnn(C)c12 c1(-c2c(C(=O)NC(c3nn[nH]n3)C3CC3)c[nH]n2)ccc(Br)cc1 C1(C(C)NC(=O)CSc2cn[nH]c2)CN(C(=O)C=CCF)CCO1 c1(CNCCN2CCN(C(C=CC=CC)=O)CC2)c(F)ccc2occc12 Cc1c(C(N2CC(O)C2)=O)[nH]c2ccc(C(=O)NN3CCCC(O)C3)cc12 C#Cc1ccnc(C(N2CCC(NC(c3cccc(Cl)c3OC)=O)C(F)C2)=O)c1 N1(C(CSCC#C)=O)CC2CC(NC(=O)COc3ccc(F)c(Cl)c3)CC1C2 c1(CN2CCC(CC(=O)OC)C2)ccc(-n2ncnc2C)cc1 c1(C(=O)NC2CCC(CNC(Cc3cccc(C)c3)=O)C2)sc2nccn2c1C c1(C(=O)NC2(CNC(C3(CC=C)CC3)=O)CCOC2)cc(C(=O)OC)[nH]c1C O(NC(=O)C(c1ccco1)NC(=O)C(CSC)OC)CC(=O)OCC N1(C(c2nc(CCC)oc2)=O)CCC(CNC(=O)Cc2cc(C)cs2)C12CCC2 C1(NC(c2c(C(C)(C)C)ccs2)=O)CCCC(NC(C2(C#N)CCOC2)=O)C1 C1(CCNC(CN(CCC)C(c2sccc2C)=O)=O)OCCC1C N1(C(c2ncn(C(C)C)n2)=O)CCCC(CO)(NC(C2CCOC2)=O)C1 C=C(C)COCC(=O)NCC=CC(=O)NC1(C(C)C)CC1 N1(C(CCOC)=O)CCC2CCN(C(=O)C(c3cc(C)cc(F)c3)C)CC2C1 C1(NC(C=C(C)C)=O)CCN(C(=O)Cc2cc(C)cs2)CC1C(C)C C1(CC)CCC(C(=O)NC(=O)NC)CC1.c1(N2c3nnc(s3)C2)ccccc1C c1(COC)nn[nH]c1C(=O)NC(C)CCCNC(c1cc[nH]c1)=O c1(C(=O)NC(C2(CNC(C(C)c3cccs3)=O)CC2)C)ccnc(S(N)(=O)=O)c1 CC1CC2CN(C(C3CCN(C(c4cccs4)=O)CC3)=O)CC2N1CC1CCC1 C1(NC2(CC)c3nnnn32)C(CO)C2CCCC12.C1(CO)CCC1 C1(C2CC2)(CC(=O)NCc2ccn(C)n2)CC1.C12CC(C1)C(=O)NC2C n1(CCSCC(=O)NCCOCCOCCNC(CC)=O)cncn1 C#Cc1ccc(C(=O)N(CCN(C)C(C2(F)C3CCCCC23)=O)C(C)C)cc1C C(=O)(CCC(=O)c1cccs1)NC1C(NC(C=CCCC)=O)CCC1 c1(SCC(=O)NCC(C)N(C(=O)CS(=O)(=O)N(C)C)C)ccsc1[N+](=O)[O-] c1(C2N(C(=O)NC3CCOCC3O)CCC2)ncc(NC(N)=O)cn1 c1(C(=O)NCCC2N(C(c3c(C)n[nH]c3)=O)CC(F)(F)C2)ccc2sccc2c1 C(=O)(C(O)C(F)(F)F)NCC=CCNC(c1nnc(C)o1)=O N1(C(c2ccc(OC)s2)=O)CCC2(NC(C3CN(C(C)=O)C3)=O)CC2C1 c1(OCC)ccc(CN2CCN(C(=O)NCC(C)C(C)(C)C)CC2)cc1 c1(SC)cccc(CCNC(=O)CC2CNCC23CC3)c1 C1(NC(C2(OCC)CC2)=O)CC(C(=O)N(C)Cc2ccoc2)CC1O c1(NC(C)=O)ccc(C(=O)N(C2CC3CCC23)C)cc1Cl.C1CN1 CC(C)C(C(=O)N(C)C)NC(=O)CCCCN(C)C(c1cn(C)cn1)=O n1(CC(=O)NCC=CCNC(C2CCC3CCC23)=O)nc(O)ccc1=O n1(C(C)C(=O)NCC2CCCCN(C(=O)CCCO)C2)cnc2ccccc12 CC1CC(NC(=O)Cc2nc(-c3ccsc3)no2)CN1C(=O)CC1(C)CC1(F)Cl c1(-c2c(F)ccc(C(C)=O)c2)cc(C(=O)NCCC(C)(C)O)c2cc[nH]c2c1 CC1CN(C(c2ccc(Cl)o2)=O)CC(C)C1NC(=O)CCNC(=O)CO N1(C(c2cnn3c2OCC3)=O)CC2CCC1CN2C(c1cc(O)cc(F)c1)=O C1(NC(C2CCC23CCC3)=O)(CNC(C2(CO)CCCO2)=O)CCCCCC1 C1(C(=O)NC2C(NC(CC3(OC)CCC3)=O)CCC2)CCC2(CCCCC2)C1 N1(C(C(CCCC)(F)F)=O)CC2CCCC(C1)N2C(C1CC1(C)C(F)F)=O C1(C(=O)NC(CCC=C)C2CC2)CCCCCC1NC(c1cc(O)nn1C)=O C(=O)(C1=CC(O)C(O)C(O)C1)N1C2CC(CN(C(C(CCC)NC(C)=O)=O)C2)C1 CCC(C(=O)NC(C(=O)N1CC(C2CCCOC2)C1)C1(O)CCC1)OC C1(CNC(c2c(CC)c[nH]c2)=O)C2CN(C(=O)C=CS(C)=O)CC12 c1(NC(C2(SC)CCNC2)=O)ccc(OCCCF)cc1 C1(NC(C2(CC)CCCN2C(C2COCC(C)O2)=O)=O)CC2COCC(C1)C2 C(c1ccc(Cl)cc1F)=CC(=O)NC(C1CCCN(Cc2cnn(C)c2Cl)C1)C C12(CN(CC(C)C)C(c3c(C)cc(CC)o3)=O)CC(C)(CCO1)C2.C1C(=O)N1 N1(C(CCNC(COC)=O)=O)CCC2(CCCCC2NC(C2CS(=O)(=O)C2)=O)C1 Cc1cc(C(=O)CSC2(C)CCC(NC(=O)C(F)=CCCF)C2)cc(C)c1 c1(C(=O)NCC2CCCC(CNC(C3C(C=C)C3)=O)C2)cncc(C#N)c1 n1(CC(C)NCc2ncc(F)cc2F)cnc2c(cnn2C)c1=O C1(C)(CNC(c2[nH]cc(C)c2)=O)CN(C(=O)CN2CC(=O)N(C)C2=O)CCO1 c1(C(=O)NCCCc2ccccc2Cl)cccc2c1[nH]c1ccccc21 N1(C(c2nc(C)oc2)=O)CC2CCC1CN2C(=O)C(C)Cc1cccnc1 c1(C(N2C(C(=O)NC)CC(O)C2)C(=O)NCCCF)cc(C)cc(Br)c1 c1(C(N2CC(O)CC(NC(=O)Cc3ccon3)C2)=O)cc2cnccc2[nH]1 N1(C(c2cn(C)cc2C(F)(F)F)=O)CC(NC(=O)C(=O)C2CC2)CC2(CC2)C1 c1(COCCCN2CCC(NC(=O)CCCc3ccsc3)C2)cccc(Cl)c1 C1(C(N(C)CCc2cnc[nH]2)=O)C2CC2CN1C(c1nccs1)=O N1(C(c2ccc(C(=O)OC)o2)=O)CCC(NC(=O)C(F)(F)CF)CC1C1CC1 c1(CC(=O)NCCOC(CNC(CC2CCN(C)C2)=O)(C)C)ncc(F)cc1F C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NCc1cc(OC)c(OC(F)F)cc1 c1(C(=O)NCC(C)N(C(c2c(C)nc(C)[nH]2)=O)C)ccnc2ccc(O)cc12 C1(CNC(Cc2c(C)n[nH]c2C)=O)CCN(C(=O)CC(O)C2CC2)C1(C)C c1(-n2cc(C(N(C(C(C3CCC3)OC)=O)C)C)nn2)cccnc1C(=O)O c1(OCC(=O)NC2CCN(C(COCC#C)=O)C2)cccc(C(N)=O)c1 C1(C(N(CCCNC(=O)Cc2cscn2)CC)=O)CCCSC1 c1(C(=O)NC2CCCN(C(C=C3CCN(C)C3)=O)CC2)ccc(F)c2ccsc12 c1(C(=O)NCC2CC2NC(=O)COC2CC=CC2)c(C(F)(F)F)cncc1F N1(C(C)C)CCC(NC(C2CC3CC3N2C(=O)C(C)(C)C2CCCC2)=O)CC1 CCC(C)CC(C)CC(C)C(=O)OCCCCCCN1CCCCC1 c1(C(=O)NC2(CNC(c3c(C)ccs3)=O)COC2)cc(Br)c(Cl)cc1F C1(CN(C(CCSC)=O)C)COCCN1C(=O)C(C)=CC(C)(C)C C(C)(CC(C)NC(=O)CSc1cn[nH]c1)NC(C(C)NC(CC)=O)=O N1(C(CCC(=C)Br)=O)CCC2CCC12C(=O)NCC1(NC(C)C)CC1 C1(CNC(=NCC2(CO)CC23CCOCC3)NC2CC2)C(F)(F)C12CCOCC2 C1(NC(CCC)=O)C2CN(C(c3ccnc(C)c3)c3ccccc3)CC12 C1(NC(CCCOCCC)=O)CCC(N(C(=O)CN2CCCC2CO)C)CC1 C12(C(=O)NC(C(=O)NC3(COC)CCC3)Cc3cc[nH]n3)CCCC1C2(F)F C1(c2cc(C)no2)CN(C(=O)CCn2cc(C(C3CC3)N(C)C)nn2)CCO1 C1(C(=O)NCC2CCC(CNC(c3ccc(C(C)C)o3)=O)C2)CC2CCC(C1)O2 N1(C(C2(F)CCN(C(c3cc(SC)oc3)=O)C2)=O)CC(C#N)C2(CCC2)C1 c1(-n2c(-c3ncn(CCS(CC)(=O)=O)c3)nc(C(O)CC)n2)cccc(C)c1C c1(CC)cccnc1C(=O)NC1CC(NC(=O)CC2CCSC2)C1 c1(CC)nc(C)c(C(N2CC3CC2C3CNC(=O)CCc2ccc(F)nc2)=O)s1 C1(NC)CCCN(c2ncc(C=CC(N3CCC(C(=O)OC)CC3)=O)cn2)CC1 C1(C(=O)NCCCCN(C(C2(CCC)CCC2)=O)C)COc2ccc(F)cc2C1 C1(C)(C(N(CC(C)O)C)=O)CCN(C(C2CC2Cl)=O)CC1 c1(CC)[nH]c(C(N2CCC(CNC(=O)CCc3cccc(OC)n3)C2)=O)nc1Cl c1(C(=O)NCCC2N(C(C3CC(=O)OC3)=O)CCC2)nnc(O)c2ccccc12 CCC(C)CC(C(=O)NC1CC(C(C)O)C1)NC(c1cncn1C)=O C(=O)(C(=O)CCC(C)C)N1C(CC(=O)NCc2c(C)nn(C)c2)CC(C)(C)C1 c1(C(=O)NC(CNC(Cc2c(C)nc(S)s2)=O)C)nccc2c(Br)cccc12 Cc1nnn(CC(=O)NCc2nc(-c3ccccc3)no2)n1 c1(OCC(N2C(CN(C(=O)Cc3ccon3)C)CCC2)=O)ccccc1F N1(C(C(CC=C)(C)C)=O)CCOC2CCN(C(=O)CSC)CC12 C1(COC)CN(C(c2ncncc2Br)=O)CCN1C(C1CC(F)C1)=O C(=O)(CCC(=O)NCC(O)CCNC(=O)C(C)NC(=O)COC)NCC C(c1ccc(Br)s1)=CC(=O)NCCN(C(=O)C(O)c1cnc[nH]1)CC1CC1 c1(CC)ccc(C(=O)NCC(C)NC(=O)CCN2CCCC2=O)cc1C(F)(F)F Cc1sc(C(=O)NC2CC2CNC(c2ccc(N)c(Cl)n2)=O)cc1[N+](=O)[O-] c1(C2(OC(=O)C=O)C(C)CCC2)ccc(F)cc1F.c1(C(F)(F)F)cccc(Br)c1 N1(c2c(C)c(N3CCN(C)C(c4ncc[nH]4)C3)ncn2)CCC2OC(=O)NC2C1 C12(NC(C(CCC)CC)=O)CCC(CNC(C3CCCC(C)C3)=O)(CC1)OC2 c1(C(C)NCC2CCN(C(=O)OC(c3cncc(Cl)c3)C)C2)cccc(S(N)(=O)=O)c1 C1(C2(O)CN(C(=O)CCC3CC3)C2)(CNC(c2c(C)[nH]nc2C(C)C)=O)CC1 C1(CNC(=O)NCC2C(C)C2)CCN(CCC(F)(F)F)CC1 c1(C(=O)NC2CC3CN(C(C(C)C(F)(F)F)=O)C2C3)n[nH]c2c1CSCC2 N1(C(CCC(CC)OC)=O)C(C)CC2CN(C(=O)CCCC(N)=O)CC12 c1(OC)cccc(CNC2CCCC(NC(=O)CC(O)C3CC3)C2)c1Cl N#Cc1ccc(O)c(NC(C2CC(NC(c3csnc3Cl)=O)CCO2)=O)c1 CCCC(C(C(=O)NCc1ccccc1Br)N1CCCC12CCC2)OC C(=O)(C(C#N)(CC)CC)N1CCC(CCOC)(NC(C(C)SCCCC)=O)C1 c1(OC)cccc(C(N2CC(CN3CCN(C(=O)CC(F)F)CC3)C2)=O)c1 C1(CC(=O)NC2CCC2NC(c2csc(C(F)F)n2)=O)C=CCCC1 C(CC(=O)N(C)CC1(CNC(=O)CCC2CCCCO2)CC1)(C(C)C)OCC c1(C(N(CCN(C)C(C2(O)CCCOC2)=O)C)=O)cnc(Cl)n1C c1(CC)c(C(N2CC(NC(c3[nH]nnc3C3CC3)=O)C(C(F)F)C2)=O)cnn1C C1(C(=O)NCCCN(C(C2CC(OC)C(OC)C2)=O)CC)CCn2nccc2C1 C1(C(=O)NC2CCC(NC(CCc3cc(C)on3)=O)CC2)CCc2nn[nH]c2C1 c1(CN2CC(C(=O)Nc3cc(C)cc(Cl)n3)C2)c(Cl)cc(Cl)cc1Cl N1(C(C(C=C=C)C)=O)CC(NC(c2c(C)nsc2Br)=O)CC2(CCC2)C1 c1(CC)ncc(C(N2CC(CO)(NC(c3cnc(CC4CC4)[nH]3)=O)C2)=O)s1 N(C1CCOc2c(C)cc(C)cc21)(C(CCCC#N)c1nnnn1C1CC1)CC Nc1c(C(N2CCCCC2CCNC(C2CCCC2(F)F)=O)=O)nc(O)nc1O c1(CC)cnc(C(=O)NCc2cccc(NC(=O)Cc3ccon3)c2)nc1 C1(NC(=O)COc2ccsc2Cl)CN(C(=O)CC2(CO)CC2)C2(CCC2)C1 C1(NC(c2c(C)con2)=O)C2CC(NC(c3c(C)ccn3C)=O)CC12 CCCCCC(c1nnnn1C1CC1CC)Nc1cn[nH]c1 CCS(=O)CC(=O)NC1C2CC1N(C(c1cc(C)n(-c3ccc(C)cc3)n1)=O)C2 C(CN=c1[nH]c2c(c(=NCc3c(F)cccc3Cl)[nH]1)COC2)c1c(O)cccc1 N1(C(CCc2ccn(C)c2)=O)CCOCC(NC(=O)COC2CCCCCC2)C1 c1(CC)ccnc(C(=O)NC2CCOC2C(=O)NOCc2ccc(F)nc2)c1 C1(NC(C#CC(C)C)=O)CC(F)(F)CC1NC(C1(C(F)(F)C2CC2)CCOCC1)=O CC(CNC(c1ccsc1C#N)=O)C(F)C(=O)N(CCCc1ccco1)C N1(C(c2c(=N)cc[nH]c2)=O)CC2CC1CC2NC(c1cc2n(c1)CCC2)=O N1(C(c2cc(CC)on2)=O)CCCC(C)(C(N2CCC3C(C(N)=O)C3C2)=O)C1 C1(CNC(C2(C)CC2)=O)(NC(c2ccc(Br)o2)=O)CCCCCC1 c1(C(N2C(CNC(CCC#N)=O)CC(O)C2)=O)cn2cccc(Cl)c2n1 C12(CNC(c3c(CC)nn[nH]3)=O)CCCC1CCN2C(=O)CC1CC=CCC1 c1(CCC)n[nH]c(=NC(C)CC(C)NC(c2cc(OC)ns2)=O)s1 C1(CN(C)Cc2cccc(F)c2OCCO)CCCCC1C1CCCCC1 c1(C(N(C2CC2)CC2(O)CN(C(C3(SC)CCC3)=O)C2)=O)ccc(C)nc1 C1(CNC(C(c2cnn(C)c2)OC)=O)CCN(C(=O)CC2(C#N)CCC2)C12CC2 C(=O)(C(C)(O)C(C)(C)C)NC(CC)CNC(=O)CC1CCN(CC(F)(F)F)CC1 C(=O)(C(C)CC(F)(F)F)N1C(C(C)NC(CCNC(COC)=O)=O)CCC1 CCCCC(C(=O)N1CCCC(O)(CNC(=O)C(=Cc2c[nH]cn2)F)C1)N(C)C C=CCC(CNC(=O)C(F)C(C)(F)F)C(=O)NCCN1CCCOCC1 C1(C(=O)NC(CCNC(c2n[nH]c(C)c2C)=O)(C)C)OCCN(C)C1=O C(N=c1[nH]c2ccc(Br)cc2o1)C1(O)CCN(C(CC(COC)(C)C)=O)CC1 C1(NC(C(C)Sc2ccccn2)=O)CC2CCC1(C(N1CCCC(C)(O)C1)=O)C2 N1(C(CC(=O)OC)=O)CCC2(CNC(c3cn4ccnc4cn3)=O)CCCCC12 Cc1ccc(C(=O)NC(CN2CCCC2)CO)cc1F.c12csc(c1)NC2=O C(=O)(CCCCCNC(N)=O)N1C(CN(C(C(CCC)C)=O)C)COCC1 C=C(Cl)CCC(=O)NC(CCC1CCC1)C(=O)NCC1(CO)CCCO1 N1(C(c2cc(C(C)C)n(C)n2)=O)CC2(CCCC2NC(=O)C2=CCOC2)C1 N1(C(C(C)NS(C)(=O)=O)=O)CCN(C(=O)C=Cc2ncco2)CC1C1CC1 N1(CC(C)C)CCCC1C(=O)NC1CC(CNC(=O)C(F)(F)c2ccnn2C)C1 c1(OC)ccc(C)c(C(N2CCC(NC(=O)C3=CCS(=O)(=O)C3)C2)=O)c1N C1(NC(c2ccsc2Cl)=O)C2CC3CN(C(=O)C4CCc5c[nH]nc54)C1C3C2 C1(C(=O)NC(CC=C)CNC(=O)CC2(CO)CC2)CC2(CCC2)CCO1 c1(C(=O)NCC=CCNC(C2CC23CC(O)C3)=O)cccc(C2CCOC2)c1 C(=O)(N1OC2CCC1C2)C1C(NC(C2(CC=C)CCC2)=O)CCOC1 C1(NC(c2c(C)oc(C#N)c2)=O)CN(C(=O)CC(C)C(C)C)CCC12CCC2 CCC(C)CC(=O)C(=O)NC1CC2(C1)CC(C(N1CC(C)=CC(C)C1)=O)C2 C1(CC(=O)N(CCC(=O)NCc2cscn2)CC#C)CCC2CC12 n1(CC(N2C(CCNC(=O)C(F)OC)CC(OC)C2)=O)[nH]cc2c(=O)ncnc1-2 c1(CCC(=O)N(C2CCC(NC(=O)CNC=O)C2)C)ccc(SC(F)(F)F)cc1 N1(C(c2cccc(CC)c2)=O)CC(OC)CC(NC(C2CC(F)(CO)C2)=O)C1 c1(CC)cccc(C(N2CCCC(C(=O)N(CC)Cc3noc(C)n3)C2)=O)n1 N1(C(c2c(N)non2)=O)CCN(C(=O)COCC(F)F)CC1 c1(C(=O)NCCN(C(CC2C(OC)CC2)=O)CC2CC2)cnc2cc(C)ccn12 O=C(CN=c1cc[nH]cc1)NC1CC(CCC(N2CCCC(O)(C(N)=O)C2)=O)C1 CC1(C)CCC(C(=O)O)N(C(=O)NCc2ccccc2Br)C1 C(C)(C)(CC(=O)N(C(C)C(F)F)C)N(C(CC(C)C)=O)C C(=O)(C1CCCc2c[nH]nc21)NC(C)CCNC(=O)C=Cc1ccccc1F c1(C(C)NC(c2n[nH]cc2CNC(C2CC(C)(C)C2)=O)=O)nccc(O)n1 Cc1ccc2ncc(CN3CCN(C(c4[nH]nnc4C)=O)CC3)n2c1 N1(C(C(CNC(C(C2CCOCC2)C)=O)(C)C)=O)CC2CC1CC2CF c1(OC)cc(Br)c(Cl)cc1NC(=O)C(=O)NC(c1cccc(C)c1C)C Cc1cc(C(N2CCOC(CN3CCN(CC(F)F)C(C)C3)C2)=O)c(C)cc1O C(CCC(O)C(=O)N1CCC(N2CCC2)CC1)NC(C1(C)CCC(=O)N1)=O O=C1NC(Cc2ccc(Cl)cc2Cl)C(=O)N1CCSC1CCCC1 CC(C)(C)C(C(=O)N=c1[nH]oc2cccc(Cl)c12)n1ccnc1 Cc1cc(C(=O)NCCC(O)CNC(=O)CCN2CCCC2=O)cc2nc[nH]c12 C(=O)(C(F)(F)CC1CCCO1)N(C1CCN(C(=O)CSC2CC2)C1)C C(=O)(CCP(C)(C)=O)NCC(C)(O)CNC(C1C2CC1NC2=O)=O Cc1c(C(N2CC3(CCCC3NC(=O)C(C)CO)C2)=O)sc2cncn12 N1(C(C=CSC)=O)CCC2C(NC(=O)C(C)(O)C3CCC3)CC12 C1(CC)(NC(c2ncccc2O)=O)CCCN(C(=O)C(C)NC(=O)NC)C1 C(CC(=O)N(C1CCCCCC1O)C)(C(C)CC)NC(CC(C(=C)C)OCC)=O c1(OC)ccc(F)c(C(=O)NCC2CC(O)CN2C(C2CCN(C)C2C)=O)c1F C(=O)(C1=CCC(C)CC1)NCC1C2CN(C(c3c(Cl)ncc(C)c3)=O)CC21 c1(C(=O)NCC2(NC(C=C(C)C3CC3)=O)CC2)cnn(CC2CC2)c1 c1(C(=O)NCC(CO)NC(C(F)=CCC)=O)cc2cc(OC)c(F)cc2[nH]1 C1(NC(C(C)=C(C)C)=O)C2COCC1CC(NC(=O)CC1CCC1(C)C)C2 C1(C(N2C(CNC(C(CC)CC)=O)CC(C)CC2)=O)COc2cc(F)ccc2O1 C12CCCN(C1)C2=O.c1(C(C)NC(=O)OC(C)(C)C)ccc(SCC(F)(F)F)o1 c1(C(=O)NCC2CN(C(C3N(C)CCOC3)=O)CC2(C)C)ccc2sccc2c1 C(=O)(C(C)CC)N(C1(C(=O)OC)CCC1)C(=O)C1CC1 C1(C(=O)NCCCCC2CN(C(c3cc(C)sc3)=O)C2)CC(C)OC1C C(=O)(CC1=CCN(C)CC1)N1C(C(=O)NC2(C)CCSCC2)(COC)CCC1 N1(C(C(C)NC(c2ccn3ccccc23)=O)=O)CCc2c[nH]nc2C1 C1(C(=O)NC2CCC2C(=O)OC)CCN(C(=O)CC(=O)N(C)C)CC1(C)C C=C(C)c1ccccc1NC(=O)CC1CN(C(c2nc(C)cnc2C)=O)CCO1 Cc1cc(C(=O)N(C2CN(C(C3CCOCC3(C)C)=O)CC2(C)C)C)cc(Cl)c1 N(C1c2ccccc2CC1NC(=O)CC1COCC1O)C(CC1(C)CC1)=O c1(N2CC(COC)(N(C(c3cnn(C)c3CC(C)C)=O)CC)C2)snc(C)c1C#N C(=O)(CC(C)(C)C)N(C1CCN(C(=O)C(=O)NC2CCN(CC(C)(C)C)C2)C1)C Cc1cc(=O)oc(C)c1C(=O)N(C)CC1CC(F)CN1C(=O)CSc1cccs1 c1(C(N2CCC(CC=C)(NC(CSCCOC)=O)CC2)=O)ccncc1N=[N+]=[N-] N1(C(C2C(C)CCC2)=O)CC2CCC1CN2Cc1csc(C2CC2)n1 CC(=O)CCCC(=O)N1CCN(C(=O)Cc2ccnc(F)c2F)C2CC12 C1(NC(C(C)OC)=O)CC2CCC(C1)N2C(C1CC(N(C)C)C1)=O N1(C(c2cccc(Nc3cnc[nH]3)c2)=O)CCCCCC1c1ccon1 c1(C(N2C(Cn3cc(CCSC)nn3)C(C)(C)C2)=O)ccnc2c1ccn2C N1(C(CCOCC)=O)CCCC1C=CCNC(c1conc1CC)=O N1(C(Cc2cn(C)nc2)=O)CCN(C(C2COC3(C)CCOC23)=O)C2(CC2)C1 C1(NC(CSCCC)=O)CCN(C(=O)C(C(C)C)C2CCC2)C1C(C)(C)C c1(C(=O)NC(C2N(C(C(C)OC)=O)CCC2)(C)C)ccnc(OCCO)c1 c1(CCC)cc(=NC(=O)c2cc(Br)no2)[nH]o1 C1(CNC(C2(OC)CS(=O)(=O)C2)=O)(NC(=O)Cc2ccsc2)CCCCC1C C1(C2CCCN(C(c3nn[nH]c3Cl)=O)C2)(NC(c2ccc(C)s2)=O)CC1 c1(-c2ccc(C(=O)OC)s2)[nH]nc2ccc(CN(C3CCS(=O)(=O)C3)CC)cc12 C(=O)(C(CC(F)F)N(C)C(c1cc(CO)n(C)n1)=O)NC(CC)CO c1(C(N(c2nccc(Br)n2)C2CC(N)C2)=O)cnc2ccccc2n1 C12(C(N3CC(NC(COCC)=O)C(F)(CO)C3)=O)CC(COC)(C1)OC2(C)C c1(OC)cc(C(=O)NC2CCC2NC(c2ccc(CS(C)(=O)=O)o2)=O)cc(C)n1 C1(C(=O)NC2(c3nncs3)CC2)CN(C(C2CC(O)C2)=O)CC12CC2 C(C)(C)(CC(F)C(=O)NC1(C)CC(O)C1)NC(c1ccc(C)c(C)n1)=O C=CC(C)C(C(=O)NCc1ccc(F)c(F)c1)c1ccccc1 C1(NC(CCN(C(C(C)C)C)C)=O)CCN(Cc2ccncc2)CC1 N1(C(CCc2ccc(C)s2)=O)CC(NC(=O)CC2(N(C)C)COC2)CC1(C)C N1(c2ncc(C#N)nc2)CCC2(CC(NC(C3(C4CC4)CCC3)=O)C2)C1 c1(C(=O)NC2C(C)CC2)ccoc1CNC(C1CC(=O)C1)=O c1(OC)ncc(C(C)=CC(=O)NC2CCN(C(C3C(C)CC3C)=O)CC2)cn1 N1(CC)CC(C(=O)NC2CC(NC(c3ccncc3Br)=O)CC2O)CC1=O c1(C(=O)NC2CC(NC(CSc3n(C)ccn3)=O)C2)ccc2[nH]ccc2n1 Cc1[nH]c(=N)ccc1C=CC(N1CCCCC1C(C)NC(=O)C1=CCC1)=O c1(C(N2CC3C(NC(C(CC(C)C)C)=O)(C3)C2)=O)cnn2c1OCCCC2 c1(C(N2CCC(N(C)Cc3coc(C4CC4)n3)C2)C)cccc(Cl)c1 C1(C(N2CCC(NC(c3c(C)cns3)=O)C2C)=O)CCC(C#N)CC1 N1(c2n(CCC(C)(C)C)ccn2)C(=O)CC2(SC(F)(F)F)CC2C1=O C(CC(F)(F)CO)N(CC(=O)OC)CC1CC2(CC2)C1 c1(CC)ccc(NC2CN(CC(F)(F)F)C2)nc1.c12ccc(nc1)[nH]2 C1(CC)CCC(C)CN1C(=O)CCNC(=O)CC=CC(C)(C)C N1(C(c2ccnc3ccnn23)=O)CCCC2(CCCN2C(C2C3CCCC23)=O)C1 c1(C(N2C(CC)CC(C)C2)C(=O)NC)ccc(C(F)(F)F)cc1Cl C(=O)(C(C)CC(=O)OC)NCC1CCCN(C(Cc2ccc(OCC)cc2)=O)C1 c1(CC(=O)NCC(C(C)C)NC(C2(CC3CC3)CC2)=O)c(F)cccc1F c1(C(=O)NCCC(C)(C)NC(C2CC3C=CC2O3)=O)nccc2c1CNC2=O C1(C(N(C2(CC)CC2)C)=O)CN(C(c2cc(C#N)n(C)n2)=O)CC1(C)C C1(NC(c2cc(Cl)ns2)=O)CC2CC1CN(C(=O)CC1CCCC1)C2 Cn1c(O)nc2cccc(C(=O)NC3CC(NC(=O)C(C)(C)C(F)(F)F)C3)c12 n1(CCCCNC(CC2(CSC)CC2)=O)cc(Cc2nc(C)no2)nn1 Cc1nc2sccn2c1C(=O)NCCC1(NC(C2CC3(C2)CC(O)C3)=O)CCC1 Cc1cc(=O)c(C(=O)NCCCOCCNC(=O)Cc2cccs2)cn1C Cc1cnc(C(C)NC(c2coc(CNC(=O)CC(C)CN(C)C)n2)=O)nc1 C(=O)(C#CC1CCCOC1)N1C(CN(C(=O)COc2cccnc2)C)CCCC1 c1(OC)cc(CN2CCSCC2C(N2CC3CC3C2C#N)=O)cc(Br)c1OC c1(C(=O)NCC2CCC(NC(c3cccnc3)C)C2)ccc(C(C)C)c(Br)c1 Cc1cnc(C=CC(N2CC=CC2CNC(=O)CC2CCC(F)(F)C2)=O)[nH]1 c1(N2CCCC(CC=C)(NC(=O)C(C)(C)C)C2)nc2ccc(C)nc2s1 CC1CC(NC(=O)CC2CCCC(C)C2)CCN1CCCC1CCS(=O)(=O)CC1 OC1CCCCC1CNC(c1nnnn1CCC1CC1)c1ccno1 C1(CC)CCCCC1C(=O)NCC(N1CCOCC1)C1CC(Cl)C1 C1(CC=CC(=O)NC(C)CO)(NC(C2C(C)C2C)=O)CCC1 c1(C(C(=O)NC2(C)CC2)N(C)CC2CCCN(C)C2)cnc(C(C)(C)C)nc1 c1(C(N2CC3(C2)CN(C(C2C4C=CSC24)=O)C3)=O)ccc(F)cc1Cl c1(C(=O)OC(C(N2CCN(c3cc(C)[nH]n3)CC2)=O)=O)ccc2c(c1)C=CCC2 C(=O)(C(C)(F)C(C)(C)F)N(Cc1cn(CCNC(C(C)=CC)=O)nn1)CC CC1CCCc2nc(C(N3CCC(C)(CNC(C4(CO)CC4)=O)C3)=O)cn21 c1(CC)c(NC(=O)C=CCN(C)C(C2COCCC2C)=O)cnn1CC N1(C(C(C)C)=O)CC2CCC1C(NC(=O)CCc1ccc(C(C)(C)C)cc1)C2 C1(C(=O)NC(C2CCOC2)C#C)CCCCN(C(c2c[nH]cc2CC)=O)C1 C1(C(=O)OCC)CC1(C)C(=O)NCC(C1CC1)NC(c1cnsc1)=O.COC c1(NC(CC)=O)ccc(CNC(=O)C(C)(COC)OCc2ccccc2)cc1F Cn1cc(C(N2CCC(CCNC(=O)CCc3cnn[nH]3)CC2)=O)c(C2CC2)n1 c1(CC(=O)NC(C(C)C)(C)CNC(=O)Cc2ccc(O)nc2)cccc(Cl)c1F C1(C(N(C2CC2)CC2N(C(C3CN(C(C)=O)C3)=O)CCC2)=O)CCCC2(CC2)C1 N1(C(c2ncc(C(C)C)s2)C(=O)Nc2ccccc2)CCSC(C)CC1 Cc1cc(NC2CC(NC(c3cc(O)nn3C)=O)C23CCC3)ccc1[N+](=O)[O-] c1(N(C2CN(C(c3ccc(C)c(C)c3)=O)C2)C)ncnc2sccc12 CC1C(C)N(C(=O)CCN2CCCC2)CCN1C(=O)CCCF C1(C(=O)NCCCOC(C)C)CN(C)CCN1C(=O)Cn1cccn1 c1(N2CCN(CCOC)CC2)cc(N2CCC(C)(CO)CC2)nc(CSC)n1 C1(O)(CC(=O)NC2(N(C(C(C)Cc3cnn(C)c3)=O)C)CC2)CCCCCC1 CCC(C)(C(=O)O)N(C)C(c1ccc(-n2cncn2)cc1)=O C1(C(=O)NC(C)CCNC(C2(c3ccc(O)nc3)CC2)=O)(OC)CCCCCC1 c1(C(N(C)CC2CCCN(C(C3CC3C(C)(F)F)=O)C2)=O)cc2c[nH]cnc-2n1 C1(C(C)NC(C(CC)N(C)C)=O)CN(C(C2CN(CC)CCO2)=O)CCO1 c1(C(N2CCC(CCNC(=O)C(F)OC(F)(F)F)C2)=O)cc2ccccc2cn1 C1(NC(c2ncn(C)c2)=O)CCOCC1NC(=O)CSCc1csc(=N)[nH]1 CC1(C(=O)NCC2CC(F)(CNC(c3csc(CO)n3)=O)C2)CC(F)(F)C1 c1(C(c2n(C(C)C)nnn2)NCc2nocc2C(C)C)cc(Br)ccc1F c1(CNC(c2cc(-c3cncnc3)ccc2CO)=O)ccc(Br)c2ccccc12 C(C)(C(=O)N(C(C)C(=O)NC(COC)C(C)C)CC)OCC#C c1(C(=O)Nc2nc(C(=O)Nc3cc(Cl)ccc3Cl)cs2)cccc([N+](=O)[O-])c1 C(=O)(CCCC(=O)N1CCCC(NC(=O)Cc2[nH]cnc2C)C1C)NCCC Cc1cc(CN(C)C(c2cn(CCNC(=O)Cn3ccnc3)nn2)=O)no1 C(=O)(C(CCF)NC(c1n[nH]c(O)n1)=O)NCC(=O)NC(C)(C)C C1(O)(C(C(=O)NC(C)C(C)n2cccn2)NC(c2nc(C)sc2)=O)CCCCC1 N1(C(C(C=C)O)=O)CCOC2CN(C(c3ccn4cncc4c3)=O)CC12 C1(OC)C(NC(=O)NCc2cc(Br)no2)C2CCCC12 C(C(O)CCCS(N)(=O)=O)NC(CS(N1CCN(C)CC1)(=O)=O)=O Cc1ncnc(C(=O)NCc2cncc(C(=O)NCC3(CC(C)C)CC3)c2)c1C C(C)(CCCN=c1nc(Cl)[nH]c(C)c1C#N)NC(CNS(CC)(=O)=O)=O C(=O)(CC(O)(C(F)(F)F)c1ncc[nH]1)NCC(CC(C)C)NC(=O)C=C1CCC1 C1(NC(CCCCSC)=O)CC2CN(C(C3CC3c3ccco3)=O)CC2C1 c1(N(C)CC2CC2CO)nc(Cc2ccccc2F)c2c(F)cccc2n1 C1(C2CN(C(=O)C#CC(=O)N(C)C)C2)(NC(C2CC(C)CC(C)O2)=O)CC1 c1(C(N2CC3C(CN(C(=O)CCC4CC4)C)C3C2)=O)ccsc1S(C)(=O)=O c1(OCC(=O)N(C(C23CC(C(F)(F)F)(C2)C3)=O)CC2CCCO2)ccc(F)cc1F NS(=O)(=O)c1ccc(C(=O)NCCC2CCCN2C(=O)CC2C=CS(=O)(=O)C2)o1 c1(CS(=O)(=O)NC2CCCN(C(C3(F)CC3)=O)C2)ccc(Cl)cc1 N1(C(C2(C)CCCCC2)=O)CC2CC(NC(C3CCCC3C3CC3)=O)CC1C2 C#CCC(C)(CNC(c1cc(CNC(=O)CC(C=C)CC)nn1C)=O)CO CC1CN(C(c2sccc2F)=O)CCC1NC(c1cc(O)cs1)=O CC(c1cccs1)=CC(=O)NC1CCCC1CNC(c1ccc(C(F)F)s1)=O C12(c3cn(C(C(=O)NC4(COCC)COC4)C)nn3)CCC(C(=O)OC)(CC1)C2 Cc1nn(C2CC2)c(Cl)c1CN1CCC(C)(C(=O)NC2COC(=O)C2)C1 n1(C(CC)C)ncc(C(=O)NCC(CO)NC(C23CCN(CC2)C3)=O)c1C c1(C(N(C2CCC(NC(CC3CC(=C)C3)=O)CC2)C)=O)cccn2c(C)cnc12 C1(NC(C(C=C)O)=O)CC2(C1)CC2NC(=O)COC1CCCCCC1 C=CCC(C(=O)NC1(COC)CN(C(=O)C(=O)NCCO)C1)C(C)C C1(NC(c2cn(CC)nc2)=O)CC(NC(c2ccc(C(C)(C)C)cn2)=O)CC1O N1(C(c2ccc(C)c(Cl)c2)=O)CC(NC(=O)C(C)C2CCC2)CCC(O)C1 c1(C(=O)OCC)cc(C(=O)OC)ccc1C.c12cc(OC)cc(c1)NS(=O)(=O)C2 N1(CC)CC(C(N2CCC(OCCNC(=O)C=CCO)C2)=O)CCC1=O N1(C(C(C2CC2)OC)=O)CCC2CC(C1)CN(C(C1CN3CCN1C(C)C3)=O)C2 C1(C)(OCC)CCN(C(=O)C(CC)N(C(=O)C(F)F)C)CC1 CC(C)C1=CCC(C(N2CCCC(N(C)C(C3CC(F)(F)C3)=O)CC2)=O)CC1 CCC(CNC(=O)C(F)CC1CN(C(=O)CNC(=O)CC(C)C)C1)C(C)C c1(OC)cccc(C(CNC(CC(O)COC2CC2)=O)SC)c1 CC(C)C(C)(O)C(=O)N(CC(C)NC(C1CC1C(N)=O)=O)C c1(OCCC)ccc(Cl)cc1C(=O)NCC1(C)CCC(NC(c2cn[nH]c2)=O)C1 C1(C(=O)NCC2CN(C(c3n(C)ncc3C3CC3)=O)C2)CS(=O)(=O)CC12CCC2 C(C)(CCC(=O)C(=O)CCC(C)OC)SC.C1(N)C2CC(NC(=O)CCC3CC3)CC12 N1(C(C(C)N(C(C)C(C)(C)C)C)=O)CCC(CCc2nn[nH]n2)CC1 CC1CC(C)(C)CC1NCc1ncnn1C1CC1 C(=O)(C(CO)NC(=O)OC(C)(C)C)N(CC(C)N(C(C=C(C)C(C)C)=O)C)C C1(NC(c2cnco2)=O)CC2(CCC(NC(c3cnc(N(C)C)s3)=O)CC2)C1 C1(C2CC2)(NC(CCC(=C)Cl)=O)CCN(C(c2cnc(OCC(F)F)cn2)=O)C1 N1(CC(C)Cc2ccc(C(F)(F)F)cc2C(F)(F)F)CCNC(C)C1C CN1CC2(CN(CC3CCOC3(C)C)C2)OC1=O C(=O)(C(F)(CC)C(=O)OC)NC(CCNC(c1cc(CCCC)oc1C)=O)C C(CC(C(N)=O)NC(=O)C(F)C1CC(NC(=O)CC(=O)OC)C1)OC C(CCCCC(=O)N1CCC(C)(CNC(c2[nH]cnc2C#N)=O)C1)=CC CCC(C)C(C(=O)NC)NC(=O)CCCNC(=O)CC(C)COC N1(CCC(=O)NCC)CCCC(C(=O)N(C)CCc2ccc(Cl)cc2)CC1 C1(C2CC2)(C(=O)NC(C(C)NC(=O)C(O)Cn2cncn2)CO)CCOCC1 CC1(C)CCC(=CC(=O)NCC2CN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)CC1 c1(-c2nnn(C3(CO)CCCS(=O)(=O)C3)n2)cccc2c1sc1ccccc21 C1(C(=O)NCCC(C)(C)NC(c2cc(O)ccc2F)=O)CCn2cnnc2C1 c1(NC(C2CCN(C(C(C)OC)=O)CC2)(C)C)cccc(C)c1C C1(CC(=O)NC(CC)CNC(c2ccc(C(C)C)o2)=O)CCCC2(CCC2)O1 Cc1cc(=O)ccn1CC(=O)NC1C2CN(C(=O)CSc3ccccc3Cl)CC12 c1(C(N2CCC(C(C)(C)NC(C(F)=CCC)=O)C2)=O)ccc(Cl)c(C)c1 N1(C(c2c(CC)noc2)C(=O)NCC2(CC)CC2)CCn2ncc(SC)c2C1 c1(C(C)OC)cn(C2COCC2NC(c2sccc2C(C)=O)=O)nn1 C1(C)(C(=O)NCC2C(NC(C(c3c(C)noc3C)(C)C)=O)CC2)CCCS1(=O)=O c1(C(N2CC(C(C(=O)NCCCC(=O)OCC)O)C2)=O)ccccc1F C1(C(=O)NC2CCC2)C2CCC(C2)N1C(C1CSC1)=O C1(C(=O)N(CC(F)(F)F)C)(COC)CCCN(C(C2CC3(CSC3)C2)=O)C1 C1(CC(=O)NCC2CCN(C(C3CC(C)SCC3)=O)CC2)CS(=O)(=O)CCN1C C(=O)(C(F)(F)CCn1cccn1)NC1CCC(NC(C2CCC(C)C2)=O)CC1 Cn1nc(O)cc1C(=O)NCc1ncoc1C1CN(C(C2CCCC(O)C2)=O)C1 Cc1nc2cc(NC(C3CCN3CC3(c4ccncc4C#N)CC3)=O)ccc2o1 N1(CCC2CCC(C(=O)NC(C=CC3(C)COC3)=O)C2)C2CCCCC1CCC2 c1(COC)nc(=NCC2(NC(c3cc(C(F)F)[nH]n3)=O)CCOCC2)s[nH]1 c1(-c2n(CCC=C)c(N3CCS(=O)(=O)CC3)nn2)sc2ccccc2c1Br Cn1nc(-c2nc[nH]n2)nc1-c1cccc(C(=O)Nc2ccnnc2)c1 c1(C(N2C(CNC(c3c(C)cco3)=O)COCC2)=O)[nH]c(=N)ccc1C C1(C(=O)NC(C)CNC(=O)CCc2nc(-c3nc[nH]n3)no2)CCC2(CCC2)O1 C1(CC)CC(C(=O)O)CN(C(=O)NCc2nn(C)cc2C#N)C1 C(=O)(CCCC(C)(C)NC(C1CCC(C2CC2)C1)=O)N1CC(C)(C(N)=O)C1 C1(NC(c2c(NC(C)=O)cncc2)=O)CN(C(=O)CCC(N)=O)C2(CCOC2)C1 c1(C(N(CC(C)NC(=O)C(O)CC2CCCC2)C)=O)coc(C(C)(C)C)n1 N1(C(C(CC)Cc2ccccc2)=O)CCN(C(c2cc(OC)no2)=O)C2(CC2)C1 c1(C(N(C2CN(C(=O)C3CC3)CC2(C)C)C)=O)cc(Cl)ccc1Br N1(C(CC(CNC(C(CCC=C)(C)C)=O)OC)=O)C2CCCC1CC(=C)C2 Cc1ncccc1-n1cc(CN2CCN(C(=O)CCc3cccnc3)CC2)nn1 C1(NC(C2CC(=C)C2)=O)CCN(C(C2CN(c3ncc(F)cn3)C2)=O)C1C1CC1 c1(C(=O)NC2CCN(C(c3cnc(C(C)=O)s3)=O)C2)cccc2c1SCCC2 C1(C(=O)NCC(C)(C)n2ccnc2)CN(C(c2cc[nH]c2)=O)CC1C1CC1 c1(C(N(CC(=O)Nc2c(CC)noc2)CC2CC2)=O)nn(C)cc1C N#CC1CN(C(c2cnc3n2CCOC3)=O)CCN1c1ccnc(C2CC2)n1 c1(C(=O)NCCC2CCN(C(C(CC)N(C)C)=O)C2)c(C)c2cnccn2c1C N1(C(C(=O)N(C)C)=O)CCCC(F)(CNC(=O)Cc2ccc3occc3c2)CC1 C1(C)(CNC(C2CC(C)OC2)=O)CCCN(C(C2CCCN2C(C)C)=O)C1 S(=O)(=O)(c1cnc(NCC(c2nncn2C)C)c(Cl)c1)NC(CCSC)COC Cc1c(CNC(=O)C(C2CCC2)NC(=O)C=C(C2CC2)C2CC2)cnn1C C1(C(N(CCNC(CC(=O)NCC)=O)C2CC2)=O)CCOC(=O)CC1 c1(CCC)nnc(S)n1CC(N1CCCC(c2ccc(OC(C)C)cc2)C1)=O S(=O)(=O)(c1ccc(Cl)c(C(=O)OCCC2(C)CC2(Cl)Cl)c1)N(C)C CC1CC(NC(=O)C#CC2CC2)CN(C(c2nc(C3CC3)ncc2Br)=O)C1 S(=O)(=O)(c1ccc(Cl)cc1F)N(C(C(CCC)C)C)CC c1(CC)ccccc1C(CNC(=O)C=CCOC)N(CCC(C)(C)C)C.C(C)=O C(=O)(CCCCCNC(=O)CC1CCOCC1)N1C(CC(N)=O)CCC1 C(c1ccc(CC(N)=O)cc1)=CC(=O)NCC1(CNC(C2N(C)CCC2)=O)CC1 C1(NC(C(c2cccc(C)c2)F)=O)CC2CCCC(C1)N2C(C1CC1Cl)=O c1(NC(C2C3CN(C(C4N(C)CCCC4)=O)CC32)=O)cc(Br)cc([N+](=O)[O-])c1 c1(C(=O)NC(C)CN(C)C)n[nH]c2c1CCN(Cc1cc(F)c(F)cc1O)C2 C(CN=C(NCc1cnnn1C)NC1CC1)N1C(CC)CCCC1 c1(C(=O)OC)cc(C(=O)NC(C)(CNC(c2ncc[nH]c2=O)=O)CO)ccc1C c1(-c2cn(C3CC(NC(c4n(CC=C)ccc4)=O)C3)nn2)cccc(N)n1 N1(C(c2cc(CC)nn2C)=O)CCC12CN(C(C1(C)CCCC1)=O)C2 c1(C(=O)NCCC2(CNC(c3cscc3C3CC3)=O)CC2)nnc(O)cc1O CN1CC(C)(C(=O)NCC2(F)CCN(C(C3CC3C(F)F)=O)CC2)CCC1=O c1(CNc2cc(C(=O)OC)no2)ccc(Oc2cccc(F)c2)c(Cl)c1 C1(C(=O)NC2C(CNC(C=CC=CCCCCC)=O)C2)CC2(C1)CC(C)(C)C2 c1(C(N2CC3C(CNC(C(CN(C)C)O)=O)(C3)C2)=O)cccc(F)c1N N1(CC#CCC)CCCC(COC(=O)CC2CCCCC2)C1 CC1OCCOC1C(=O)N(CCCCNC(C1(n2cccn2)CCOCC1)=O)C Cc1nc(CC(=O)N(C)CCNC(c2coc(Cl)c2)=O)co1 c1(OC)c(C#N)ccnc1NC(C1(C)CCCN1C(c1cc(C)nc(O)c1)=O)=O c1(C(=O)NCC(C)(C(C)C)NC(COCCCC)=O)cccc(C)c1Br C(CC(C(=O)N(C1CCCC1)C)NC(=O)CCc1nc[nH]n1)=CC c1(C(=O)NC2CN(C(C=COCC)=O)CC2C)ncc(Br)cc1OC C1(C(=O)NCCC(Cc2ccccc2)NC(c2cccs2)=O)(OC)CCCC1 c1(C(C)(C)C)ccc2[nH]nc(C3(CSC4C(Cl)(Cl)C45CC5)CC3)c2c1 C(=O)(C(C)C(O)C(C)C)N1CC(n2cc(-c3cc(OC)cc(N)c3)nn2)C1 N1(C(C2CC(C)(C)N(C(=O)CCCC#N)C2)=O)CCOC2COCC2C1 c1(N2C3CC(CNC(C4C(CC)OCC4)=O)(OC3)C2)nc(C)nc(C)c1F c1(SC)cncc(C(N2CC(CNC(c3ocnc3C(F)(F)F)=O)C(C)C2)=O)c1 CC(C)CC(F)(F)C(=O)NCCN(C(=O)CN1CCCOC1=O)C1CC1 C1(COC(C)(C)C)CC(C(=O)NC2CCCN(C(c3ccnnc3)=O)C2)=NO1 N1(C(CCCCOCCC=C)=O)CC(CNC(c2ccc(SC)o2)=O)C2(CC2)C1 C1(CN(C)C(c2cccnc2S)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC1 C#Cc1ccc(C(N2CC(OC)C(C(=O)NC3CC(CC(N)=O)C3)C2)=O)cn1 C1(OC)CN(C(=O)CN2CCCCC2C)CC1NC(c1cnn(C2CC2)c1)=O C(C(=O)NCC(O)CCNC(C1CCCOC1)=O)(C(C)C)SCC C1(CNC(C(CCC)C)=O)CC2(CCN(Cc3cccc(OC)c3Cl)CC2)C1 c1(CC)ccc(C)c(C(N2CCCC2C(C)NC(C2CCCN2CC)=O)=O)c1 N1(C(C2C(CN(C)C)C2)=O)CCC(NC(=O)C(C)(C)c2cnco2)C(CO)CC1 C(=O)(CC(C)(C)C(=O)NC(C)CCCNC(C12CCCC1C2(F)F)=O)OC N1(C(Cn2c(C)csc2=O)=O)CCN(C(=O)COc2ccsn2)C(C)C1 C1(CNC(C(COC)(C)C)=O)CCN(C(c2n[nH]cc2C(C)(C)C)=O)CC1C c1(C(N(CCOC)CCNC(C2CNC(=O)C2)=O)=O)cc(F)cc([N+](=O)[O-])c1N Cc1ccc2nc(CNc3cncc(-n4ccnc4)n3)ccc2c1 CC1CN(C(=O)C=CCF)CCC1NC(=O)CCc1ccc(C(N)=O)cc1 c1(NC(CC2C(C(=O)NCCCOCCSC)C2)=O)ccc2ncnn2c1 C(CN=C(NCc1cccnc1Br)N1CCC2(C)C(C1)C2(Cl)Cl)N(CC)CC CC(C)CCCCCCC(=O)NCC1(C)CCC(NC(=O)CCc2nc[nH]n2)C1 C(=O)(CCCN=c1nccc[nH]1)NCC1(F)CC(CNC(C2(CCC)CC2)=O)C1 c1(C(=O)NCCC2(O)CCN(C(c3cc(O)cs3)=O)C2)cc2c[nH]nc2s1 C1(C(=O)NC(c2ccccc2)C#C)C2CC1N(C(C1CCCSC1)=O)C2 N1(C(Cc2cc(C)c(F)cc2)=O)CCC(NC(=O)CCNS(C)(=O)=O)C12CCC2 C1(C(=O)NCC2C(CC(=O)NCCC(C(C)C)O)C2)CCC(O)CN1C CC(C)CC(C(=O)NCC1CC(CF)C1)NC(c1cccn(C)c1=O)=O C1(C(=O)NC2C=CCN(C(c3cc[nH]c3)=O)C2)CCCCCS1(=O)=O c1(C(=O)NCCC2CCN(C(C3CCCN3C3CC3)=O)C2)cc2cccn2cn1 C(CC(C)C(=O)NCCOC1CN(C(C2CC23CC(O)C3)=O)C1)=CCC C(C(=O)N1CCC(OCC(=O)N(CC2CCCC2)CC2CC2)C1)(C(C)C)OC c1(CCC(=O)NCC2(CNC(c3sccc3Br)=O)CC2)cccc(F)c1 N1(C(C(C2CN(C(=O)C(O)Cn3cncn3)C2)OC)=O)CCCOCC1C c1(C(N(C2CCCCC2)CCNC(C(C)NC=O)=O)=O)nn[nH]c1Cl C1(NC(C2=C(C)CC2)=O)CC12CCN(C(C1CCCC(C)(C)C1)=O)CC2 C1(C(N(CCC(C)(C)O)C)=O)CCOCCN1C(C1CCC2CC12)=O O=C1COC(CNC(C2CCC2NC(c2cn(C3CC3)nn2)=O)=O)CN1 C(CC(C)CN=C(NC1CCC1)N1CCC(OCC2CCCCC2)CC1)OC Cn1cnc(C(=O)NCCCNC(C2CC(O)(CCC(C)(C)C)C2)=O)c1 C1(C(C)C(=O)N(CCCNC(=O)Cn2cccn2)C)CCOCC1 C#Cc1ccc(C(=O)NCC2CN(C(c3oc(CC)nc3C)=O)CCO2)c(C)c1 N1(C(c2cc(CC)[nH]n2)=O)CCC(C(N2CCC3(CC3)C2)=O)(CF)C1 C1(C(CNC(C2C(C)C2C)=O)(C)C)CCN(C(C2CCCC2)=O)CC1 C(C(C)C)(C(O)C(=O)NC1(CN(C)C(C2CC(F)C(=O)N2)=O)CC1)OC CCC(CCC(=O)NCC1CC(F)C1)NC(=O)C(O)C1CC1 CC1C(NC(c2noc(C(C)(C)C)n2)=O)CCCN1C(C1CC12CCOC2)=O c1(OC)cc(C(=O)NC(C)(C)CCN(C)C(C2OCCN(C)C2=O)=O)cnc1O C=CC(CC)C(=O)N1CCCC(CCC(=O)N(C)Cc2cnco2)C1 c1(C(N(C(CNC(C2CCC(=O)N2C)=O)C2CC2)C)=O)cncc([N+](=O)[O-])c1 C(C)(CC(C)C)(C(=O)NC(C)C(=O)NO)NC(CC=C=C)=O CCCN=C(NCc1ccc(N2CC=CC2)cc1)NC1CC(OC)C1 CC(O)C(C(=O)N1CC(CO)(NC(=O)C=CC2CCC2)C1)NC(=O)C1CC1 C1(OC)CCCN(C(c2cccc(-c3cc(C(=O)N(C)C)ccn3)c2)C(=O)O)CC1 C1(CC)CN(C(=O)CC2CC3(CC3)CO2)CCN1C(c1cc(C2CCC2)[nH]n1)=O c1(CNC2CN(C(C3N(C(=O)OCC)CCCC3)=O)C2)cnc2ccnn2c1 C(C)(CCC(=O)NCC(C)NC(=O)C(C1CCCCCC1)F)OC c1(C(=O)NC(C2N(C(C(=O)NCCOC)=O)CCC2)C)nc2c(s1)CCCC2 Cc1cc(C(=O)N(C2CCN(C(C3CCCN3C)=O)C2)CC2CC2)cc(F)c1 Cc1ncnc(C)c1C(N1CCN(CC2(O)CN(C(c3cnco3)=O)C2)CC1)=O C(=O)(C1OCCn2ccnc21)N1CC(C)CN(CC(F)(F)F)CC1 C=C(C)C(C)(C)C(=O)NCC1CCN1C(=O)C=Cc1cncc(F)c1 c1(CC(=O)NCC(CC)NC(C(CC=C)(F)F)=O)cn(CC)c2ncccc12 c1(C(=O)NCC2CN(C(CCCOCCOCCOC)=O)C2)cc(N)cc(O)n1 N1(C(c2c(CC)ccc(N)c2)=O)CCC(C2CC2)(NC(C2(CN(C)C)CC2)=O)C1 C1(C(=O)NCC2CCC(NC(COCCOCCOC)=O)C2)CCC(O)CN1C C1(SC)CN(C(=O)C(F)=C(C)C)CCC1C(F)(F)F.C(C(=O)N)(C1CCOC1)SC(F)F n1(C(C)C)ncc(C(=O)NCC2(O)CCN(C(c3ccnc(O)c3)=O)C2)c1Cl C(C1c2ccccc2CN1C(=O)COC1CCOC1)NC(C1C(C)(C)C1)=O CC1(C(=O)N(CCNC(=O)C(N)=O)CCO)CCNC1=O c1(C(=O)NC(C2N(C(C(C(=O)OC)C)=O)CCC2)C)cc2n(n1)CCNS2(=O)=O C=CCC(C(=O)NOCCCOCC)NC(=O)C(C)CC1CCCC1 N1(C(c2cn(C)nc2)=O)CCC(C2(NC(c3nc(O)[nH]c(=O)n3)=O)CC2)C1 C1(Cl)(C(=O)NCC2N(C(c3nc(C)oc3)=O)CC=C2)CC12CCC2 C1(C)(NC(C=CCC)=O)CCCN(C(=O)C(c2ccc(C#N)cc2)O)C1 C(CC1(CO)CCC1)(C(=O)N(C(C)CC)CO)NC(CC)=O.ON N#Cc1sccc1NC(C1CC(F)CN1C(c1cc(Cl)c(Br)s1)=O)=O O=C(C#CC1CCCOC1)NC1CCN(C(c2cnc3n2CCOC3)=O)CC1F C1(NC(C(C2CC2)OC)=O)CC2(C1)CC(NC(=O)CC1COC(=O)C1)C2 Nc1c(C(=O)NC2CCN(C(C3(CC(F)F)CCNC3=O)=O)C2)ccnc1Cl N1(C(C(C)(C)NC(=O)OC)=O)CCN(C(C2CCCN2N=O)=O)C2(CCC2)C1 c1(C(N(C2CCCN(C(CNC(C)=O)=O)C2)C)=O)ccc(Br)c(Cl)c1 C1(C(N2CC(OCCNC(c3nccnc3N)=O)C2)=O)CCC2C(C1)C2(F)F S(=O)(=O)(C1(c2cn(C(c3cccc(F)c3)C)nn2)CC1)NC.C12CCN(C1)C2 c1(N2C(C(=O)NC(CC)C3CCC3)CCC2)ncccc1Cl C(CCC(O)C(=O)N1CCC(CC2CCC2)C1)NC(CCC(C)OCC)=O CCC(CC(=O)N(CC(C)CNC(c1cc(C)n(CCO)n1)=O)C)C(F)F N1(C(C=NOC)=O)CC(C)OC2(CCN(C(=O)C(C)CS(C)(=O)=O)C2)C1 C1(C(C(=O)OC)NC(=O)C(CNC(=O)OC(C)(C)C)CO)CCCN(C)C1=O C1(C(NOCC(=O)N(C)C)=O)CC(NC(C23CC(F)(C2)C3)=O)C12CCC2 N1(C(COc2cccc(NC(=O)NC)c2)=O)CCN(C(=O)C=C2CC2)CC(O)C1 C12(CN(CC)C1)C(=O)OC2.C(=O)(CCCC)OC(C)(C)C.C(=O)(NCO)OCC n1(C(C)C)ccc(=NCc2cc(C3CCCC3)n(-c3ccccc3)n2)[nH]1 CCCCCC(C)(C)C(=O)NC1CC1CNC(c1cnn2ccc(C)cc12)=O Cc1cc(-c2cn(C3CC4(NC(=O)C5=CC(C)CC5)CC34)nn2)ccc1Cl n1(-c2c(CNC(N3CCCN4CCCC34)=O)cccc2)cnc2ccccc12 N1(C(C(C)=C2CCCC2)=O)CCN(C(=O)CC2CCCCC2)CC1CC(F)F C(=O)(C#CC(=O)O)N(CCC(=O)NC)CCCCC(N)=O c1(C(=O)NCCNC(=O)C(c2ccc(F)cc2)(F)F)cc2ccc(O)cc2[nH]1 c1(C(=O)NCCN(C(Cc2cccc(C)c2Cl)=O)C)cc2cccnc2[nH]1 C(=O)(C(C)C(O)CC)N1C(c2nc(SC(c3ccc(Cl)cc3O)C)on2)COCC1 C1(C)(CC)CCC(NC(=O)CC2CC2CNC(=O)CC(C)c2ccco2)CC1 c1(-n2c(C)nnn2)ccc(O)c(C(=O)NC2CC(NC(=O)C(C)P(C)(C)=O)C2)c1 c1(C(=O)NC2(C)CC(NC(c3ccsc3Cl)=O)C2)coc2c1C(O)CCC2 N1(C(c2c(OC)scc2)=O)CC2(CNC(=O)CCCC3CCC3)CCC1CC2 C1(CNC(C(C2CCC2)OC)=O)CCN(C(=O)C(=Cc2cccnc2)F)CC1C C(C(N=c1[nH]c(Cl)ncc1C(N)=O)C(C)C)NC(COCc1cc(C)on1)=O N1(C(c2cc(C)c(C)s2)=O)CCC(C)CC1C(=O)NC1CN(C(=O)C2CC2)C1 C1(C(=O)NC2C3CN(C(CC(COC)(C)C)=O)C2CC3)CSc2ccccc2O1 CC(CC(=O)Nc1cnn(CC2CC2)c1)C(F)(F)C(F)(F)F Cn1cnc2nc(=NCCN3CCNC(=O)C3)[nH]c(NCC3=CCCOC3)c12 C1(CNC(c2cnc(OC)nc2)=O)CCC12CN(C(c1ccnc(Cl)c1O)=O)C2 Cc1cccnc1C(O)C(=O)NCC1COCCO1 C(=O)(CC(C(C)C)NC(c1coc(C)n1)=O)NC(C(CC)C)C N1(C(C(CC)SC)=O)CCCC(CO)(NC(=O)COc2cccc(Cl)c2)C1 Cn1cnc2nc(N3CCCCC(CNC(C4CC(N(C)C)C4)=O)C3)ncc12 C1(C2CCC2)(C(=O)NC(CC(C)NC(c2n(COC)ncc2)=O)C)CCC1 CC1(C)CCc2[nH]nc(C(=O)NCC3CN(C(C45CC(CO4)C5)=O)CCO3)c2C1 Cc1cn2c(n1)CCC(C(=O)NCC1CC(NC(c3cn4c(n3)CCC4)=O)C1)C2 C(N=c1ncc(O)c[nH]1)C1N(C(C23CCCC(C)(C2)OC3)=O)CC1.Cn1nccc1C=C N1(C(CSCCOC)=O)Cc2ccc(C(C)NC(=O)C(C)C3CCC3)cc2C1 C1(C2CCOCC2)(CNC(C(CSC)C)=O)CCN(C(=O)CCCN(C)C)C1 C(=O)(C1CCc2cccnc21)NCC1(C)C(C)CN(C(c2c(C)c[nH]n2)=O)C1 CN1CCC(NC(c2coc(Cl)c2)=O)C12CCCN(C(c1n[nH]c(CO)n1)=O)C2 N1(C(C2CCC(O)C2)=O)CCN(C(C2CC(C3CC3)=NO2)=O)C2(CC2)C1 c1(C(=O)NCCN(C(c2ccc(C#C)cc2)=O)C)cc2cc(OC)c(F)cc2[nH]1 c1(C(C)C)ncsc1C(=O)NCCC1CC(NC(C2CCC2c2nc[nH]n2)=O)C1 c1(CC(N2CCC(OCCNC(CC(CNC)O)=O)C2)=O)cc(C)nc(O)c1 C1(CC(N2CC(CNC(C(C3CC3)OC)=O)C2)=O)CCC(=O)N1C N#Cc1cnc(NC2CCC3CN(C(c4ncccn4)=O)CC23)c(Br)c1 C1(C(=O)NC2(C3N(C(C4(C)CC(=C)C4)=O)CCC3)CC2)CCCN(C(C)=O)C1 Cc1ccc(C)c(C(=O)NCC2(NC(C3CC(C)OC3=O)=O)CC2)c1C CON(C)CC(O)Cn1cc(C(=O)Nc2nnc(-c3ccccc3)o2)nn1 C(=O)(C1=C(C)N(C)c2nnnn2C1)NC1C(NC(C(C(C)C)NC(C)=O)=O)C1 c1ccccc1F.C(=O)(CCOC1CCC1)N(CC(C)NC(=O)CSN)C C(=O)(CCCCC(N)=O)NCCC1N(C(CC2(C#N)CCOCC2)=O)CCOC1 C(=O)(CC(C)C(F)(F)F)N1CC(COC)(CNC(=O)C2=CC(C)(C)C2)C1 c1(C(N2CCC(N(C(=O)CC3COCCO3)CCC)C2)=O)cnnc(C)c1 Cc1ccc(C(=O)NCC(=O)NC2CC2NC(=O)CSc2cn[nH]c2)cc1C c1(C(=O)NC(c2cccnc2)C(C)(C)C)ccsc1C(=O)Nc1ncccn1 C1(NC(c2c(CC)cco2)=O)CCC2CC1CN2C(c1oc(C)cc1C)=O C1(NC(C2N(C(C3N(CCC)CCC3)=O)CC3CC32)=O)CC2COCC(C1)C2 N1(C(C(CSC)OC)=O)CC(C(=O)NC(c2csc(C)n2)C)C2(CC2)C1 C(CCCC(C)(C)C(=O)NNC(=O)CCCC(C)(C)C)NC(C1C(C)CCC1)=O c1(OC)cc(-c2cn(C3CN(C(c4nocc4C(C)C)=O)C3)nn2)ccc1Br C1(C(=O)NC2CC(=C)C2)CC2(CC2)CN1C(=O)Nc1cccc(C(C)(C)C#N)c1 N1(C(C(C)=C2CC2)=O)CC(C)CN(C(=O)CSc2cccc(C)c2)C(C)C1 C1(NC(C2(CF)CCN(C(C3CC3(F)Cl)=O)C2)=O)CCC(F)(F)CC1 c1(NC(C2C3CN(C(C(C)OCC=C)=O)CC32)=O)cc(F)ccc1-n1cccn1 N1(C(CCc2ccn(C)n2)=O)CCCCCC1C(=O)Nc1cccc(C#N)c1 O=C(C1=CC2(CCOC2)C1)N1CCCC(CNC(C2(CC(F)F)CC(F)(F)C2)=O)C1 c1(C(=O)NCC2C(C)CCN(C(=O)CCS(N)(=O)=O)C2)csc(=NC2CC2)[nH]1 c1(N2CCCC(N(C(CCCC#C)=O)C)CC2)nc2c(F)cccc2o1 C1(C(C)NC(=O)CCN2CCC2)CN(C(=O)CC2CCCN(C)C2)CCO1 Clc1cccc2nc(CN3C(c4nc(SCC(F)(F)F)sc4)CCC3)sc12 C(CCC1CCC1)(C(=O)NCc1ncccn1)NC(c1c(CC)occ1)=O Cc1cc(C(=O)NCC2CCCN2C(=O)C(c2ccn(C)n2)C)ncc1F c1(C(C(=O)NCC2N(C(C3C(C)(C)CCC3)=O)CCC2)(F)F)c(F)cccc1F c1(N(CC(CCC)C)C)nc2ccsc2c(=NC2CC3CCCC(C3)C2)[nH]1 c1(C(=O)NC2C3CN(C(c4c(C)con4)=O)C(C3)C2)cscc1S(C)(=O)=O C1(O)(CCNC(c2conc2C2CCC2)=O)CCCN(C(=O)COC2CC2)C1 C(=O)(C1=CCN(C)C1)N1CC=CC(NC(C(C)(C)SC)=O)C1 C1(CC(N2CCC(OC(C)C)C2)=O)COCCN1C(c1cnsc1)=O C(CC(C(=O)N(CC(O)CC)C)NC(=O)Cc1cnccc1C)=CC C12(CNC(=O)Cc3ccccn3)CCC1CN(C(=O)CCCCc1cnn[nH]1)C2 C1(C(=O)NCCC(C)NC(C=C(CCC)C)=O)C(C(=O)OC)CC(=O)N1C c1(C(=O)NCCCNC(C2CC3COCC3C2)=O)cc2cc(F)ccc2[nH]c1=O c1(CN(CC(C)NC(C2(C)CCNC2=O)=O)C)ccc2ccccc2c1 c1(CN2C(CC)COCC2)c(C)nn(CC(=O)NC(=O)C(F)(F)Cl)c1C C(c1cn(C)c2ccccc12)=CC(=O)NC1CC(NC(C(CO)N(C)C)=O)C1 c1(C(C(=O)NC2CCC2)N(C2CCCC2)CC)ccc(OC(C)=O)c(F)c1 CCCC(C#N)C(=O)N1CC(NC(=O)CC2CC(F)(F)C2)C(CC(C)(C)C)C1 C12(NC(C3CCN(C(C)=O)CC3)=O)CCCC1(F)CN(C(=O)CCF)C2 N1(C(CCc2ccc(C)c(C)c2)=O)CC(NC(C2CC=CCO2)=O)CC12CCC2 C1(CCCCC)CCC(C(=O)N(CCCNC(=O)C(C2CC2)SC)C)O1 n1(CC(=O)N(CC(C)NC(c2ccc(OC)nc2)=O)CC)ccc(=O)c(O)c1C c1(C(N2CCCC(CNC(c3cncc(C)c3Cl)=O)C2)=O)cc2n(c1)CCSC2 Cc1cc(C(=O)Nc2nn[nH]n2)co1 C(=O)(C(C)CCCC(C)C)NCC(CC)N(C(c1c(CC)occ1)=O)C C1(C(N(C)Cc2csnn2)=O)CCCCN(C(C2(C3CC3)CC2)=O)C1 C1(CCC=C)(C(=O)NC2CCSC2C)CN(C(c2ccn(C(C)C)n2)=O)C1 C(CN=C(NCCNC(c1ccco1)=O)NC1CCCCC1F)=CCCC C1(C(N2CCC(O)(C(C)CNC(c3ccc(O)nn3)=O)C2)=O)(CC)CCCCC1 CN(CC(F)(F)F)NC(=O)C1(c2ccc(F)cc2)CC1(Cl)Cl c1(C(N2CC3C(CNC(c4c(F)ccnc4F)=O)C3C2)=O)ccc(Cl)cc1Cl C12(C(N(CCOCCN(C(=O)C=C3CCCC3)C)C)=O)CCCC1OCC2 C1(NC(C(F)OC)=O)CN(C(=O)CC(C)c2ccncc2)CC(C)(C)C1 C(=O)(C(O)CC[S+](C)C)N1CCCC(O)(CNC(CCCOCC=C)=O)C1 c1(OC)cnc(F)c(C(=O)N(CCCCNC(=O)C(F)C(C)(C)O)C)c1 c1(C(N(CCC(C)NC(C(CC)C)=O)C)=O)ccc2c(c1)C(C)(C)CCC2(C)C N1(C(C2N(C(c3cc(C)oc3C)=O)CC(C)(C)C2)=O)C2CCC1CC(C)C2 C1(C(=O)NC2(C)CC(NC(=O)CCc3ccsc3)C2)CC2(CCC2=O)C1 C1(CC(N2CCC(N(C(=O)C(C)N(CCOC)C)CCC)C2)=O)COC(C)(C)C1 N#CC1(C(N2CCC2CNC(=O)CCNC(=O)C=CCl)=O)CC1C(F)(F)F CC1(C)C(NC(=O)CC2CC(F)(F)C2)C2CCCN(C(=O)CCC(CF)CF)C12 N1(C(c2c(-c3cnc(COC)c(C)c3)cncn2)=O)CCCC2(CCCC2O)C1 C12CCN(CC1)C(=O)CNC(=O)NC1CC1CNC2=O.N(S(N)(=O)=O)C(C)(C)C c1(C(N2CCC(CNC(C(C=CC)O)=O)C23CC3)=O)cc(F)cc(OC)c1N C(CC(C)(C)C(c1nnnn1CC(F)F)SC(C)(C)C)NC1CC(OC)C1 Cc1cnc(C(N2CC(F)CC2C(=O)NCC2CN(C(N)=O)C2)=O)cn1 C1(CC(=O)N(CCC#C)C)CCN(C(c2ccsc2)=O)C1 C1(CNC(C=CCCC=C(C)C)=O)CN(C(=O)Cc2ccns2)CCC1(F)F N1(C(CC=CC=C)=O)CCCC(N2CCN(C(=O)C(C3CC3)OCC)CC2)C1 C1(C(N2CCC(C)(CNC(c3c(C)onc3)=O)C2)=O)CN2CCCC2CO1 Cc1ccc(C(N2CC(CC(=O)NCCc3cc(C)n(C)n3)CC2C)=O)cc1O C1(C(=O)NC2CCC(C)C2)CCC(CNC(=O)CCCc2cncs2)CC1 C1(NC(c2cc(C)no2)=O)C2CCCN(C(=O)C(F)CC3CCOC3)C2C1(C)C c1(CC(=O)NC2(NC(=O)COC3CCC3)CC2)cccc2ccccc12 C(=O)(C(C)(C)C(C)NC(=O)CCCC(C)=O)NC(CCC=C)CC CCC(CC)CCC(=O)N1CCN(C(c2cnc(N3CCCC3)nc2)=O)CC1C N1(c2cccc(OC)c2)N=C(C(=O)NC2CCC3C(CC2)C3(F)F)CCC1=O c1(OC)ccc(C(=O)NCC2CC(NC(=O)COc3ccccc3O)C2)cc1F C(=O)(CCCC(=O)N(C(C)(C(=O)N1CC(C(C)(C)C#N)C1)C1CC1)C)N(C)C C1(C(=O)NCC2CCN2C(c2ccncn2)=O)CC2CCC(C1)C2 S(=O)(=O)(c1cnc(N2CCOCC3(CC3)C2)c(Cl)c1)NC(CCC)c1ccco1 N1(C(C)=O)CCC(CC(=O)NCCN(CC(C)O)C(=O)CC2OCCC2C)CC1 c1(OCC#C)ccc(CN2CCOCC2CC(=O)Nc2c(Br)cnn2C)cc1 N1(C(CCCC#CC)=O)C2CCC1CN(C(=O)C1=CS(=O)CCC1)C2 CC1(C(=O)NCC(CNC(=O)Cc2cccc(O)c2)CO)CCCNC1=O C1(C(C(=O)NCC=C=C)C)CCN(C(c2cc(CCC)[nH]n2)=O)CC1 c1(OC)ccc(C)c(C(c2nnnn2C2COC2)NC2CCCCCC2)n1 n1(CC(=O)OC)ncc(C)cc1=O.C=C1CC2(C1)C(=O)NCCNC2 C1(C(N(C2CN(C(=O)Cc3ccon3)CC23CC3)C)=O)CCCCC12OCCO2 C1(NC(C2CCCN(C(c3cc(C)oc3C)=O)C2)=O)CC12CCOCC2 O=C(C(CO)C(F)(F)F)NCC1CCN1C(c1cnccc1C(F)F)=O C1(CCNC(CSC(C)C)=O)CN(C(C2CC2(Cl)Cl)=O)CC1C C1(CC(=O)NC2CC(CCNC(c3[nH]cc(C(=O)OC)c3)=O)C2)CCC(=O)N1C C12(NC(=O)C3CC3)CCN(C(=O)CCc3cc(Br)cs3)CC1C2 Cc1ncc(Cl)cc1C(N1CCN(Cc2cnc(Cl)cc2F)C2CC12)=O c1(C(N(CCCCN(C(C2C(C3C(C)C3)C2)=O)C)C)=O)ccnc2cc[nH]c12 CN1CC(O)CC1(C)C(=O)NCC1(CNC(C2(C)CC(C#N)C2)=O)CCCC1 C1(C#N)(C(N2CC3(CN(C(c4c(C)[nH]cc4)=O)C3)C2)=O)C(C#N)C1(C)C c1(C(=O)OC)ccccc1CCC(=O)NCC(C)NC(C1CN(C)C1)=O C(CCCC(=O)N(CC(=O)NC(c1nn[nH]n1)C1CC1)CO)(OC)OC C=CC1(C(=O)NC2CC(C)(C)C23CC3)CCN(C(=O)Cc2ccc(O)cc2)C1 C1(NC(c2csc(Br)n2)=O)CCCCN(C(=O)C(c2ccccn2)O)C1 N12CCN3C(=O)C(CC3C1)N(C)CCC2=O.c1(OC)c(O)ccc(Br)c1C CON1CCC(CC(=O)NCCOCCN(C(=O)CC2CCOC2=O)C)CC1 C1(C(=O)NC)(N(C(=O)C=Cc2ccncn2)C)CCCCC1.C12(CC1)C(=O)N2 c1(C(N2CC(OC)C(NC(c3cnc(C4CC4)s3)=O)C2)=O)ccc(F)c(C)c1 N1(C(CC(CC)SC)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC1C CCC(C)C(O)C(=O)NC1(CNC(C2CCCN(C)C2)=O)CC(F)(F)C1 CC1=NNC(=O)C1CC(=O)NC(C1CN(C(=O)C(F)=CC2CC2)C1)C C1(CNC(C2C(C)C2)=O)CCN(C(=O)CN2CCS(=O)CC2)CC1 c1(C(=O)NCC2N(C(C3CC4(CC(=C)C4)C3)=O)CC2)ccc(Br)c([N+](=O)[O-])c1 N1(C(c2c(COC)cco2)=O)CCCCCCC1C(=O)Nc1ccc(C)cc1C c1(C(C)=O)cnc(C)c(NC(c2nnnn2CC2CC2)(CC)C2CCCC2)c1 N1(C(c2c(C)ocn2)=O)CCC(c2nnc(CNC(c3cnc(O)o3)=O)s2)CC1 c1(C(=O)NC2(C)CCN(C(C3(F)CCCN(C)C3)=O)CC2)cccc2nn[nH]c12 Cc1ccc(=O)n(CC(=O)C(=O)N)n1.C(=O)(C(O)CC1N=N1)N1CC(=C(CN)F)C1 C1(NC(c2c(CNC(c3ocnc3C3CC3)=O)n[nH]c2)=O)CCOCC1F c1(C(=O)NC2(CN(C)C(c3cnn4ccsc34)=O)CC2)ccc(Cl)c(O)c1 C(=O)(C(C)(C)CC(C)C)N(CCNC(c1ccc(-c2nncn2C)cc1)=O)CC C12(C(N3CCCC(NC(c4ccnc(C)c4N)=O)C3)=O)CCCCN1CCC2 C1(CNC(c2ccc(Cl)c(Cl)c2)C(F)(F)F)CCNCC1C1CCCC1 CC(CCC(C)(C)C)C(=O)N(C1CCCCN(C(=O)COC(F)F)C1)C C1(CN(C(=O)CSCC(F)F)C)CCCCN1C(=O)CCCn1cccn1 C(CCC(C(=O)NCCn1cnccc1=O)NC(=O)Cc1cnsc1)OC CCC(CNC(=O)CC1CCCC(NC(=O)CCC(C)OC)C1)(CC)CC c1(N2C(c3ccc(OC)cc3)CCC2)ccc2c(c1)CCC2=O c1(C(N2CCN(C(c3nc(Cl)sc3Cl)=O)C(C(F)F)C2)=O)cnc(O)cc1O C1(CCN2CC(CNC(C3(C#C)CC3)=O)OCC2)Cc2cc(C)c(C)cc2O1 c1(N2CC3(CN(C(=O)CSCC4CCCO4)C3)C2)ncc2c(n1)CCCCC2 c1(C(=O)NC2CC(CNC(C(Br)=C(C)C)=O)C2)ccc2nn(C)cc2c1 n1(CC(=O)NC2C(NC(c3c(CC)nc[nH]3)=O)CC2)ncc(C#N)c1N c1(C(=O)NC2CCN(C(CSC(C)C)=O)C2C)cnn2c1OCC1(CC1)C2 Cc1cc(CC(=O)NCC2CC(F)(CNC(C3(C)CC3(F)F)=O)C2)c(C)s1 C1(OC)CC(CNC(=O)CC2CCC(=O)NC2)N(C(=O)CSc2cn[nH]c2)C1 N1(C(c2oc(CC)c(C)c2)=O)C(C(=O)N(C2CCOC2=O)C)CCC12CC2 c1(-n2cc(C(=O)NC(c3cccc(OC)c3)C)nn2)ccc(F)cc1C(F)(F)F N1(C(COC(CC)C)=O)CCCC(n2cc(CSCC)nn2)C1 C1(C(N(C(C)C)CCNC(C2CC2C(C)C2CC2)=O)=O)Cc2c[nH]cc2S1(=O)=O Cc1cccc(CC(N2CCOCC2CC(=O)Nc2cc(C(N)=O)ncn2)=O)n1 C1(N(C)C)CCCCC1NC(c1cnnn1C)=O.C1(C)(C)CNC(=O)CO1 C1(C#N)(C(=O)NC(C)CCC(=O)NCCS(C)(=N)=O)CC12CCC2 C=CCCCCCC(=O)N1CCC(OCC(=O)NCC(C)(O)CC(C)C)C1 C1(NC(C(C)(C)NC(=O)OC)=O)CN(C(=O)CN(C2CCCC2)C)CC1C C1(C(=O)NCC=CCNC(CC=C(C)C)=O)C2CCC1(c1cccs1)C2 C1(C(N2CCOCC(NC(CC(C)OC)=O)C2)=O)CC2(C1)OC(=O)NC2C c1(CC)ccccc1C(=O)NCC(N1CCN(C(=O)C2=CCCS2)CC1)C CS(=O)(=O)c1ccc(OC(F)F)c(C(=O)Nc2ccc(N3CCCCC3)cn2)c1 c1(N(CC(Cc2cccc(F)c2)OC)C(C)=O)nc2c(C)cccc2s1 O(N=Cc1ccc2c(c1)CCO2)CCOC(C1CC(=O)N(c2ccccc2Cl)C1)=O N1(CC(=O)NCc2cn(C3(C)CC(F)(F)C3)nn2)CCS(=O)(=O)CC1 CN=c1[nH]c(C(=O)NC(c2ccc(C)cc2)CNC(=O)C(C)(C)CC2CC2)cs1 N1(C(CCCC#N)=O)CCCCC(NC(c2cccc(C3CC3)c2)=O)C1 C#CCCCCC(=O)NCC1(F)CC(NC(C2COC(C)C2)=O)C1 N1(C(C=CSC)=O)CCN(C(=O)CN(CC(F)(F)F)C)C(Cc2ccccc2)C1 CC(C(=O)N(CCCCN(C(=O)CSCC(F)(F)F)C)C)NC(N)=O CC1C2C(CCN2C(C2(C3CCCO3)CCC2)=O)CN1C(=O)CCCC(=O)N(C)C C1(C(=O)NC(CNC(c2cn(CC(=O)OCC)nn2)=O)C)COC2COCC12 c1(NC(C(C2CCN(C(CCCCN(C)C)=O)C2)F)=O)cc(O)cc(F)c1 C1(C(N2CC3C(CNC(c4c(C)cncc4C)=O)C3C2)=O)CCCCC12CCC2 N1(C(CNC(Cn2ncc(C(C)=O)c2)=O)=O)CCN(C(=O)C(O)C(F)F)CC1C C1(NC(c2n(CC)nc(C)c2)=O)CN(C(=O)CC2(CO)CC2)C2CCCC12 c1(C(=O)NCC(CCNC(CN(C2CCSC2)C)=O)O)ccc2cccnc2n1 C1(CNC(C2CCCC2)=O)C=CCN1C(=O)C=Cc1cnc[nH]1 c1(COC2(NCCCCSC)CCCC2)ccc(Cl)c(F)c1 C(=O)(C=CS(C)=O)N(C(C)CNC(=O)CNC(c1ccccn1)=O)CC N1(C(CCCC(=O)N(CC)CC)=O)CCC2CCCN(C(=O)C(=O)N(C)C)C2C1 CC(C)(C)CC(C(=O)NCC1(CO)CCOC1)NC(c1cnns1)=O C(=O)(CCCC(=O)N(C(C1CCN(C(=O)C(F)(F)CO)C1)C)C(C)C)OC N1(C(C2(CC(C)=O)CCC2)=O)C2CCC1CC(NC(=O)C(C)N(C)C)C2 C(C(C)(O)C(=O)N1CCC(C(C)CNC(c2ccoc2C2CC2)=O)CC1)OC c1(N2C3CC(CNC(=O)CN4CC5CC5C4)CC2CC3)ncnc2scc(Br)c12 C1(CCOCCN(CCNC(C(c2ccccn2)C)=O)C)CCC(O)CC1 N1(C(C2(C(=O)OC)CC2)=O)CCCC(CCNc2cnn3ccsc23)CC1 C=CCC(CC)C(=O)NC(CNC(=O)Cc1ccc(Br)c(F)c1)CO CC1(C)CCCC(C(N2CCN(CC(=O)NCC(C)(F)C(C)(C)F)CC2)=O)C1 N1(C(c2c(CC)noc2C)=O)CC2(C)CC1(C(N1CCCC1CC(=O)OC)=O)C2 N1(C(c2c(C)c[nH]c2)=O)CCC(C(F)(F)F)C(NC(c2nc(C)c(C)s2)=O)C1 C1(F)(C(=O)NC)CCN(CCn2cc(-c3ccc(SC)cc3)nn2)C1 C1(C(N2CCC(C(=O)Nc3ccc(C)cc3OC)CC2)=O)(CC)CCCCCC1 CC1C(NC(c2cc(CCN(C)C3CC3)on2)=O)CCCN1C(c1cc[nH]c1)=O N1(C(c2c(NC)c(F)ccc2)=O)CCc2cccc(C)c21 CCCCC(C(=O)NC(CNC(=O)CCn1cc(C)cn1)CO)NC(N)=O.C(C)(=O)O C1(C(C)C(=O)N(C)CCC2CC2)CCN(C(=O)CN2CC3CC3C2)C1 C1(C)(CC(=O)NCCC(C)N(C(=O)C(Cl)=CCl)C)CC(F)(F)C1 n1(C(C)C)ncc(F)c1C(=O)NCC(C)CNC(=O)C(C(C)C)N1CCCCC1 c1(C(N2C(C)(CNC(c3cnc(O)o3)=O)CCC2)=O)cc(F)c(Cl)cc1Cl C1(NC(c2[nH]c(=NCC)sc2)=O)CCN(C(=O)C(C)OC2CCCC2)CC1(C)C c1(NCCS(CC)(=O)=O)nc(C)cc(=NCc2ccnc(-c3cncnc3)c2)[nH]1 N1(C(C2OCC(C)C2)=O)CCC(C)(CNC(=O)Cc2ccc(C#N)cc2)CC1 Cn1nc2c(c1N)CN(C(CC1CCC3CC13)C(=O)NC1CCC1)CC2 C1(CNC(CC(=C=C)C)=O)CCN(C(c2ccncc2Cl)=O)C12CC2 C(CCC(=O)N(CC(O)CN(c1cc(C)[nH]n1)C)C)OC CC(O)CC(=O)NCC(c1ccccc1)NC(=O)C(C)(C)c1nncn1C c1(C(N(C2CCN(C(=O)C(C)C3=CCCC3)C2)CC)=O)cc2c(s1)CC(C)(C)C2 C1(N(C(C2CCCOC2)C(=O)NCCC#N)C)C2CCCCC12 Cc1cccc(NC(=O)CCC2CCCN2c2cc(C#N)ncn2)c1F C12(NC(=O)CNC(=O)CC)CC1CC1CN(C2)C(=O)C1(C1CC1)CC N1(C(C=CC(=O)NC)=O)CCC(C)C(NC(=O)CC2C=CCCC2)C1C N1(C(C(C)(C)OC(C)=O)=O)C2CCC(C(N3CCC(O)(C(N)=O)C3)=O)C1CC2 C12(NC(Cc3c(C)ocn3)=O)CCN(C(=O)C=Cc3ccccc3Br)CC1C2 c1(C(=O)NCC2N(S(CC(C)C)(=O)=O)CCC2)c[nH]c2ccc(C#N)cc12 c1(C(N2CCOCC(NC(C3CCCCC3(F)F)=O)C2)=O)ccc2ccsc2c1 c1(N(CC=C)C)ccc(C(F)(F)F)cc1S(=O)(=O)NCC1COc2cscc2O1 n1(CC(=O)NC(C2CC2N(C(=O)C(F)=CC2CC2)C(C)C)C)c(O)nnc1O CC1=NOC(C)(CNC(C2CCC(NC(=O)CC3CCCC3)CC2)=O)C1 Cc1ccc(NC(=O)C(C2CCN(C(c3cncn3C(C)C)=O)CC2)C)c(C)n1 C1(C(=O)NCC2CC(NC(c3cnn(CCO)c3N)=O)C2)(OC)CS(=O)(=O)C1 c1(OC(C(=O)NCC(CC=C)NC(=O)CCC(=C)Cl)C)ccc(Cl)cc1C c1(CC(=O)NCC2C(NC(c3cn(CC)nc3)=O)C2)c(C)nn(C)c1Cl c1(CC(=O)NCC2CC2NC(C2CCc3nc[nH]c3C2)=O)ccc2c(c1)CCC2 C1(C(=O)NC2CCCCN(C(C3(F)CC3)=O)C2)CCn2c(C(F)(F)F)nnc2C1 c1(NCC2C(C)C2(F)F)cc(N2CCOC(CC(F)(F)F)C2)ncn1 N1(C(C(C)NC(CC)=O)=O)CCC2C(CCCN2C(C2SCC=C2C)=O)C1 C1(CNC(CCSCCC)=O)(NC(=O)CC2CCCC23CC3)CC2CCC1CC2 c1(C(N2CCC(N(C(COCCOC)=O)C)CC2)=O)cc(F)cc2ccncc12 N1(C(=O)COCCc2ncon2)CCN(C(=O)CCn2cc(Cl)cn2)CC1 c1(N(C)CC2(O)CN(C(=O)CCCN3CCCC3)C2)ncccc1Cl C(C(N=[N+]=[N-])C(=O)NC1CCN(C(=O)CCCCCSC)CC1)OCC N1(C(C(C)S(N)(=O)=O)=O)CCC2CCN(C(c3ccnc(OC(F)F)c3)=O)CC12 CC1CC=C(C(=O)NCCC2CCN(C(c3cnc(O)n3C)=O)CC2(F)F)CC1 C(=O)(C(CC(F)F)NC(c1csc(O)n1)=O)NC(c1cncs1)C C1(C(C)C)CN(C(=O)C=Cc2cccs2)CCN1C(=O)CSCC1CCCCO1 N1(C(c2cccc(C(=O)OC)n2)=O)CCN(Cc2ccc(I)c(F)c2)CC1C#N N1(C(C23CC(CCC)(C2)C3)=O)CCCN(C(c2nc(Cl)sc2Cl)=O)CC1 c1(N2CC(NC(c3cc(OC)c(Br)cc3)=O)(CO)C2)ncnc2c1CCCC2 Fc1ccc(OC(F)F)c(Oc2ccc(-c3nc[nH]n3)cc2)c1 N1(C(c2cnc(C)[nH]2)=O)CC(NC(C2CC2c2ccccc2F)=O)C(C)C1 c1(C(N(C2CCN(C(c3cnc(Cl)s3)=O)C2)CC)=O)cc(F)c2cn[nH]c2c1 c1(C(N2CCC(CO)C(NC(=O)C(F)(F)CC3CC3)C2)=O)[nH]cc2c1CCCC2 N1(C(C2N(C(CCC(=O)NC)=O)CC(O)CC2)=O)CCOC2C(O)CC12 C1(N(C(CC(OCC)OCC)=O)C)C2CN(C(c3cncc(OC)c3)=O)CC12 C1(NC(c2ccsn2)=O)C2CCCCN(C(=O)CCC34CCC(CC3)C4)C12 n1(CCC(N2CC3CC2CS3=O)=O)sc2ccccc2c1=O CN1CC2CCCC(NC(=O)N=c3[nH][nH]cc3Br)C2C1 c1(NC(c2ccc(-c3cc(C)nnc3)cn2)=O)cc(N(C)C(C)C)ccc1Cl C1(CC)(NC(C2CC2C)=O)CCCN(C(c2sc(C)c(C)c2Br)=O)C1 N1(C(=O)CC2CCOC2)CCC2CCN(C(c3[nH]cc4c3CCS4(=O)=O)=O)C2C1 C1(NC(c2n(C3(C)CC3)nnn2)c2cnn[nH]2)CCN(c2cc(O)ncn2)CC1 C1(C(=O)NCC(C)CNC(c2conc2C(F)(F)F)=O)CCCCC1O C(=O)(CCC(=O)NCC)N1C(CNN(C(CSCC)=O)C(C)C)CCC1 C12(NC(c3[nH]cc(C(=O)OC(C)(C)C)c3)=O)CCC(CC1NC(C1CC1(C)C)=O)C2 CC1CCC(C)(C(N2CC(C(C)NC(=O)Cc3cccnc3O)C2)=O)C1 Cn1nnc2c(C(=O)NC3CN(C(=O)C4=C(C#N)CCC4)CC3(C)C)cccc12 C1(C(C)C)(C(=O)NCC(O)C(C)(C)C)CCN(C(=O)CCc2ccccn2)C1 C12(NC(C(C(C)(C)O)F)=O)CCCC1N(C(c1cc3c(s1)CCC3)=O)CCC2 c1(CCC(N2CC(CNC(C(C)N(S(CC)(=O)=O)CC)=O)C2)=O)ccc(O)nc1 C=CCN=C(NCCCC1CCCCO1)NC1CCOC(C)(C)C1 N1(C(CCCC#C)=O)C(CNC(c2ccc(F)cn2)=O)CC2CCCC12 c1(COC)cc(C(=O)NCC2(NC(=O)C(c3ccccc3)F)CC2)c(C)o1 c1(OCCOCCOC)ccnc(COc2ccccc2OC)c1 c1(C(=O)NC(CCNC(C(C)Oc2cccnc2)=O)C)cnn(C(C)C)c1F C#CC1(NC(C2C3CN(C(=O)C(C)OCOC)CC23)=O)CC2CCCC12 C(CNC(c1ccoc1)=O)(CC(F)(F)F)NC(C(CC)Oc1cccc(C)c1)=O N1(C(=O)COCC(F)F)CC2(C1)CN(C(c1ccno1)=O)CCO2 N1(C(C2COCC(C)O2)=O)CCC2CCCC12C(=O)Nc1cn(C)nc1O c1(NC(C(C2CCN(C(C3CC3(C)C)=O)CC2)C)=O)cc([N+](=O)[O-])ccc1Cl C(=O)(NNC(=O)C(=O)N1CCCC1)C1SCC(C(=O)OC)C1 CCCC(C)C(c1nnnn1C(C)(C)C)NCc1ccc(Cl)o1 c1(C(N(CCOC)CCNC(=O)CSCCC(C)C)=O)c[nH]nc1Cl c1(CN(C(C(n2c(C)ccn2)C)=O)C)ccccc1CNC(=O)CC1CC(C)C1 c1(C(N2C(CNC(c3ccc(C(N)=O)s3)=O)CCC2)=O)cccc(CC2CC2)c1 S1(=O)(=O)c2ccc(s2)C1=O.N1(C(=O)Nc2cccc(C)c2)CCS(=N)(=O)CC1 C(c1ccc(Br)cc1)=CC(=O)NCCCN(C(=O)CC1(O)CCC1)CC c1(NC(C2N(C(CCN(C)C)=O)C3C(C2)C3)=O)ccc2c(c1)CCOC2 CC1CCCC=C1C(=O)Nc1c(Sc2ccc(Cl)cc2)cccc1F C1(O)(C(=O)NCC2N(C(CCCCN(C)C)=O)CCC2)CCc2ccccc2C1 C(C)(c1cccs1)=CC(=O)NC1CC(CNC(CC2C(COC)C2)=O)C1 c1(C(N(CCOC)CCNC(=O)C=Cc2cccs2)=O)ccncc1O C1(NCCC)C2CC3CC(C2)CC13CO.c1(N(C=O)C2CC2)cccs1 N1(C(C(CCOC)OC)=O)C2CCC1CN(C(=O)CC(O)CCSC)C2 CCCC(C)C(=O)N1CCCCC1CCCNC(c1ccccc1Br)=O CONC(=O)C(=O)NCCC(O)C(F)F.C12C(C1(C)C)NC2=O C1(CC(=O)OCCN(C(C2(CN3CCCC3)CC2)=O)CC)C=CS(=O)(=O)C1 S(=O)(=O)(c1ccc(Br)cc1NC1CC(C)C1)NC(c1c(Br)ccc(OC)c1)CO N1(C(C(C)OCCOC)=O)CCN(C(=O)CC2(C)CCCCC2)C2(CC2)C1 C1(C(=O)NC2CC(C(F)F)C2)CC(C)(CC(C)NC(=O)Cn2cccn2)C1 CC1(C)CC(C(=O)NCc2conc2C(=O)O)CN(C(=O)C(O)C(F)(F)F)C1 Cc1cccc2c(C(=O)NC3(C)CCCN(C(=O)C(O)C4CCC4)C3)csc12 c1(N2C(CNC(C(c3ccc(C)cc3)(F)F)=O)C(C)CC2)cc(O)nc(C)n1 C12(OC)CC3CC(C1)CC(NC(=O)C1CC1)(C3)C2.C12CCCN(C1)C(=O)N2 CC1CN(C(=O)CCCC2CC2C)CC(C(=O)NCCN2CCNC2=O)O1 c1(C(=O)NCC(C)C(=O)NCC2CC2[N+](=O)[O-])cccc2occc12 c1(C(=O)Nc2ccnnc2)ccc(Br)c(C(F)(F)F)c1.C12(CCC1)C(=O)N2 N1(C(c2c(OC)ccs2)=O)CC(C(=O)OCC(C)CCCO)C(F)(F)C1 c1(C(=O)NCC2CN(C(c3c(CC)ocn3)=O)C3C2C3)ccc(C(F)F)c(F)c1 c1(CCC(=O)NC2C(NC(C=Cc3ccc(C)o3)=O)CC2)c[nH]c2ccccc12 C1(C(=O)NC(CCOCC)C(=O)NCC2CCSC2)CC2CCCC2C1 C1(OC)CC(NC(c2nc(-c3ccccc3)oc2C)=O)CC(O)C1O CS(=O)(=O)c1cc(CN2CCC(CC(=O)Nc3ccc(O)cn3)C2)ccc1F c1(OC)ccnc(C(N2CCCC(CCNC(C3C(C)C3C)=O)C2)=O)c1F c1(C(=O)NC(CNC(C2(C)C(C)CCC2)=O)(C)C)cccc(S(F)(F)(F)(F)F)c1 c1(C(N2C(C(=O)NCCC(C(C)C)OC)C(C)(C)C2)=O)ccnc2cc[nH]c12 CC1C(C(=O)N2CCC(NC(C3(S(N)(=O)=O)CC3)=O)C(F)C2)=Cc2ccccc21 c1(C(N2CC3(CN(C(C(CC)(CC)CO)=O)C3)C2)=O)cc(N)c2ccccc2n1 C(=O)(CCN=c1[nH]ccs1)NCCC(C)NC(c1cccc2c1OCCCO2)=O C1(CNC(C2CC(CN(C)C)C2)=O)COC(CNC(c2csc(O)n2)=O)C1 C1(C(=O)NCC(CC)NC(c2cn(CC)nn2)=O)CC2CC(OC)C2C1 N1(C(C(=O)NC(c2ncccc2Cl)C)=O)CC2COCCC2(N)C1 N1(C(=O)NC2CC(SCC)C2)CCC(F)(c2ccc(OC)cc2)CC1 c1(C(=O)NC(C2(O)CN(C(C=CC)=O)C2)C)cccc2c(O)ncnc12 C1(CC)CN(C(=O)C(C(C)O)OC)CCC1NC(c1cc(-c2cccs2)on1)=O N1(C(C2OCCN(C)C2)=O)CCCN(CCNC(=O)C(=O)NCCC(N)=O)CC1 C1(NC(c2ccc(CC)[nH]2)=O)CN(C(=O)Cc2sc(SCC)nc2C)CC1OC C(=O)(C1=CC2(CCOCC2)C1)N1CCN(C(CC2CC(OC)C2)=O)C(C)CC1 Cc1ncc(C(=O)NCC=CC(=O)NCCCC2CC2C)s1 N1(C(C=NOC)=O)CCC(NC(C2CC(C)=NO2)=O)C2CC12 C1(CC=C)(NC(CCCC#C)=O)CCCN(C(c2cc3c([nH]2)CCC3)=O)C1 C1(C(=O)NC(C)CCCCNC(c2sccc2C#N)=O)CCC2CCCCN12 CC1CN(C)CC(C(=O)NCc2ccc(CNC(=O)CSCC(F)F)c(F)c2)O1 CCCC(CNC(=O)C(C)NC=O)C(=O)NCc1ccnc(F)c1 c1(CC)cnccc1C(=O)N(C(CC)C(=O)NC1CC12CCC2)C C1(NC(c2ccc(C(C)C)o2)=O)CN(C(C2CCCC(F)(F)C2)=O)CCC1F C=CCC(C(=O)NCC(F)(C(=O)N1CC(C)OCC1CC)C(C)C)C(C)C C(C(CO)C(C)C)NC(C(c1cn(C)nn1)NC(CCC=CC)=O)=O C(CC(CNC(c1ccnn1CCF)=O)NC(C1OCC1(C)C)=O)OC Cc1cc(C(=O)NC2CC(C)(CNC(=O)CCC3CC(C)(C)CO3)C2)ccc1F c1(NCc2n(CCC)cnc2)nc(N2CC3C(C)C3C2)nc2scnc12 c1(C(=O)NC2CC(C)(NC(Cc3ncc(CC)[nH]3)=O)C2)cn(C)nc1C(C)C c1(CCOC)nc(=NCCCCNC(C2CCN(c3ccccc3)C2)=O)s[nH]1 C1(NC(C=CC)=O)CC2(CCC(CNC(c3cnn4c3OCC(C)C4)=O)CC2)C1 C#CC1(C(N2CC(NC(C3(CC)CC(C)(C)C3)=O)C2)=O)CCCC1 c1(CC)ccccc1Nc1ccc(CC(=O)N(C2CCCC2C)C)s1 CCC(CC)C(C(=O)NC1CCC(C(N2CCCCC2CN(C)C)=O)C1)OC Cc1cnc(C(=O)NCC2CCN(C(=O)CC3COC(C)CO3)C2)c(C)c1 n1(CCOC)cc(C(=O)NC2(C)CCC(NC(=O)C3=CCCS3)CC2)ccc1=O C1(C(N(C(C(=O)NCCc2ccc(C)s2)C2CC2)C)=O)CCCC(=O)C1 C(=O)(CCS(N)(=O)=O)N1CC(C)C(CNC(=O)CN2CCN(C)C(=O)C2)C1 Cc1cccc(C2(CNCC3CCCO3)CCCCC2)c1 C1(C(=O)NC(CNC(c2nc(C)n(C)c2)=O)(C)C)CCCC2(CCOC2)O1 C1(CNC(C2(SC)CN(C(c3cncn3C)=O)C2)=O)CC(O)C(F)C1 c1(OC)cc(C(N2CC(NC(c3cc(C)ncc3Cl)=O)C2)=O)nc(C)c1 N=S1(=O)CCN(C(=O)Nc2ccc(-c3nnnn3-c3ccccc3)cc2)CC1 c1(C(N2CC(N(C(C(c3ccc(C)s3)C)=O)C)C2)=O)ccc(F)c(C)c1 C1(CNC(CCNC(=O)CO)=O)CC(F)CN1C(C1CC(CF)C1)=O C(CC(C(=O)NC(c1ccncc1)C)NC(=O)C(n1cc(C)cn1)C)OC N1(C(CCC(=O)N(CC)CC)=O)CCC2CCN(C(=O)CCC3CCCC3)C2C1 N1(C(C(COC)COC)=O)CCCC(N(C)C(c2cccn2C)=O)CC1 N1(C(c2cc(C(C)C)on2)=O)CCC(F)(F)C(NCc2cc(Cl)ccn2)C1 N1(C(C(C(C)C)F)=O)CCC2CCCC(C1)N2C(=O)Cn1ncc(O)nc1=O N1(C(c2cncc(CNC(C3(F)CCC3)=O)c2)=O)Cc2ccccc2C1 C(C1=CCN(C(=O)Cc2ccc(Br)s2)CC1)NC(c1cc(C)c(C)[nH]1)=O O=C(C1=CC2CCCCCC12)N1CCC(Nc2ncnc3c2CCC3)C1 Cc1nc(C(=O)NCCCC(C)NC(=O)CCc2ccoc2)cn1C(F)F c1(C(=O)NC2CCN(C(=O)C(O)c3cnc[nH]3)C2)ccc2c(O)nc(S)nc2c1 Cc1nccc(CNC(=O)Cn2cc(C(=O)O)nn2)c1C c1(-c2ccc(C(NOC)=O)cc2)cnc(C(=O)NCc2nccn2C)cc1C C(=O)(C1=COCCO1)N(CCC(C(C)C)NC(c1ccc(OC)o1)=O)C C1(C(=O)NCc2[nH]n(C)c(=O)n2)CCN(C(=O)C=CCN2CCCC2)C1(C)C N1(CC(c2ccc(CC)s2)=O)CCN(C)C(C2CCOCC2)C1 N1(C(c2cnc(C(C)OC)s2)=O)CCN(C(c2cc(C)cc(O)n2)=O)C2CCC12 Cc1ccc(N(C)C(C2CCCN2C(C2CC(F)C2)=O)=O)c(C)c1 c1(CNC(=O)NC(c2nccc(C)n2)C)ccc2c(c1)CCO2 c1(C(=O)NC(C(=O)N(C)Cc2cc(OC)no2)C2(C)CC2)scc(C)c1C N1(C(Cc2c(C)nccc2)=O)CCN(C(C2(C)CCCCCC2)=O)CC1CCO N1(C(CN(CCC)C)=O)CCCC(C)C1CCNC(=O)CC1CCN(C)CC1 N1(C(C(CCSC)NC(c2cc(CC)[nH]n2)=O)=O)CCCC(C)C1CO N1(C(c2cc(C)[nH]c2)=O)CCCC(C(=O)NCC(C)(C)C(C)O)C1 CN1CCCC(C(=O)N(CCCNC(=O)CCn2cccc2)C)C1 CC1CN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC1NC(c1coc(Br)n1)=O C1(NC(=O)C2CC2)CN(C(c2cnc(C3CCC3)s2)=O)CC2(CCOCC2)C1 N1(C(CC)C(=O)NCC2CCC(=O)NC2)CCc2ccccc21 C1(C(=O)NC(C(C(=O)OC)C)C)CN(C)CCN1C(=O)CCC1CC1(F)F C1(CNC(c2ccc(C(C)=O)cc2)=O)CN(C(=O)Cc2ccccn2)CCCO1 c1(C(N2CCN(C(CCCOCCC)=O)CC2C)=O)ccc2c(c1)C(C)CN2 C1(C2CCCN(C(c3ccnc(C#N)c3)=O)C2)(NC(C(C(C)C)O)=O)CC1 c1(C(N2CCC(N(C)C(c3ncccc3N)=O)C2)=O)coc2ccccc12 Cc1cccc(NCS(=O)(=O)CCOC(C)(C)C)c1.C12CCCN1CC(=O)OC2 c1(C(=O)NC2CN(C(c3c(C)nns3)=O)CC3C2C3)c(N)cccc1[N+](=O)[O-] CSC=CC(=O)NC(C)(CNC(=O)C=Cc1ccoc1)CC N1(C(C(C)C2(O)CCC2)=O)CCC2CCN(C(=O)CC3(O)CCC3)C2C1 C1(CN(C(C(C)OCC2CC2)=O)C)CCCN(C(=O)CN2CCC(C)(C)C2)C1 N1(C(Cc2c(SCC)cccc2)=O)CCC(NC(=O)CC#N)C(C)C1 c1(NC(=O)NCC2(CCOC)CC2)ncc(Br)cc1Br c1(OC(C)C2CC2)cccc(NC(=O)NCc2ccccc2-c2cccnc2)c1 N(C(=NCC(C)C)NCc1cnsc1)C1CC(CC)(CC)C1 c1(CC(=O)NC(C)CCc2cn[nH]c2)csc(-c2ccccc2)n1 c1(C(=O)NC2CC(C(=O)NCC(N)=O)C2)ccc(Br)cc1 c1(C(=O)NCC(=O)N(CC(=O)OC)C)oc2ccc(F)cc2c1-c1ccccc1 C#CC1(O)CC(C(=O)NC(c2cccc(C)c2)CNC(=O)C=CC(C)C)C1 Cc1ncc(C=CC(=O)NC(C2CCCN2C(=O)C(O)CF)(C)C)c(O)n1 C(=O)(C(C)CCCOC)NCC1(C)CCN(C(CN(CCC)C)=O)C1 c1(C(=O)NC2C3CN(C(c4ccc(C)o4)=O)C(C3)CC2)cn2ncnc2nc1C N1(CCOCC(C)C)CCC(C)C(NC(c2cc(F)ccc2F)=O)C1 CC1=C(C)CC(C(=O)NCC2(C(N3CCC(C(N)=O)C3)=O)CC3(CC3)C2)CC1 CN1CC(C(=O)N(C(CNC(C2COC(=O)N2)=O)C2CC2)C)CCC1=O C1(NC(C2CCC(C(=O)OC)CC2)=O)CC(F)(F)CC1NC(C1(C(N)=O)CC1)=O Cc1nc2cc(C(N3CCCC(C)C3CCN=c3cc(F)nc[nH]3)=O)ccc2o1 C1(C)(CNC(C(C)c2ccsn2)=O)CCCN(C(=O)C=Cc2ccsc2)C1 C12(C(=O)NCC(COCC)C)CC(CN(C(c3c[nH]nc3CC)=O)C1)C2 C1(F)(CNC(C(C)(C)c2ccccc2)=O)CCN(C(c2ccc(=O)oc2)=O)C1 CCC1=NOC(CNC(c2c[nH]nc2CCNC(C2CCC2C)=O)=O)C1 CCC(CCC(=O)NCc1nc(=O)o[nH]1)NC(=O)C(C)(O)C(C)C c1(OC)ccc(F)c2[nH]c(C(=O)NCC(C)NC(=O)C=CBr)cc12 c1(C(=O)NCC(=C)CCNC(=O)CCNC(=O)CO)cc(CCCC)n(C)c1C CC(C)C(C(=O)NCC1CCC(C(=O)NOCCCCC2CC2)C1)C(C)C Cc1nc(C)n(O)c1NC(C1CCC(CN(C2CCN(S(C)(=O)=O)C2)C)CC1)=O C1(NC(C23C(NC(C=CC=CC)=O)C4CC2C3C4)=O)CCn2nccc2C1 c1(C(N2CCCC(N(C)C(c3cc(F)ccc3N)=O)C2)=O)cnc2[nH]nnc2c1 n1(CC(N2CC(C)C(NC(=O)CC3(C)CCCC3)CC2)=O)cc2ncccc2n1 c1(C(N2CC(NC(C3OCCN(CC)C3)=O)C(F)CC2)=O)ccc2ncnn2n1 C1(C(N2CCC(OC)(CNC(=O)CCCC(C)=O)C2)=O)CCC(C)=C(C)C1 c1(CN2C(C(=O)NC(c3ccsc3)C)CC2)c(O)cccc1F c1(C(=O)OCC)cccc2cc(SCC3(C(F)(F)F)N=N3)c(=O)oc12 C1(NC(C2CCOCCN2C(=O)C=Cc2ccncn2)=O)CC2CCCCCC12 C1(C(N(CC(C)CNC(C2CC2(F)F)=O)C)=O)CS(=O)(=O)CC(=O)N1 N1(C(C2CC(OCC)C2)=O)CC=CC1C(=O)N(CC(C)(C)CO)C CC(CC(F)F)C(=O)NCC1CCN(C(=O)C=CC2CCCCCC2)CC1O c1(C(=O)NC2CC3CC(NC(C(F)=CC)=O)CC32)cc(Br)c(F)cc1F N1(N2CCC2)CCOC(Cc2nc(=N)[nH][nH]2)C1.Cn1ccc(C=O)n1 c1(NS(CCC)(=O)=O)cccc(C(C)(C)C)c1C.C12CC(OC)CN(C1)C(=O)N2 Cc1ccnc(CNC(=O)C(O)CNC(=O)C=Cc2ccco2)n1 C1(CC(=O)NCCOC)CC(NC(c2cc(C3CC3)[nH]n2)=O)CCO1 c1(C(N(CC(O)CNC(=O)CCS(N)(=O)=O)C)=O)ccc2c(c1)CC(=O)N2 N1(C(c2c(COC)cccc2)C(=O)NCC(C)C)CCC(C2CC2(F)F)C1 C#CCCC(N)=O.C1(=O)CN1.C(CSC(C)C)S N12C3CCC1C(C3)C2=O.C1(NC(C(=O)NC2CC(OC)C2)=O)CC(C)CC(C)C1 c1(ONC(C2N(C(C(COC(C)=O)C)=O)CC=C2)=O)cccc2[nH]ccc12 C1(C(=O)NCCCCN(C)C(c2ccncn2)=O)CCC(C(F)(F)F)O1 CCCCCCC(=O)NCC(O)CN(C)C(c1cc(F)c[nH]1)=O CC1CN(C(=O)Cc2cccc(F)c2O)CC(CCNC(C2(C)CC2C)=O)O1 CCC(CN(C)C)CC(=O)N1CC(CNC(c2csc(C)c2OC)=O)C(C)(C)C1 CN1N=CC(CC(=O)NC(CNC(=O)C(c2cccc(Cl)c2)(F)F)C2CC2)C1=O N1(C(=O)OC(C)(C)C)CCCC2(CCN(CCN3CCOC4CC34)C2)C1 C1(NC(C(OCC)OC2CC(F)(F)C2)=O)(COC)CCN(C(=O)CCOC)C1 C(=O)(CCC(C(=O)NOCc1ccc(Cl)cc1Cl)NC(=O)OC(C)(C)C)OC N1(CC)CC(C(N2CCC(C)(CNC(=O)C(O)C(C)C)C2)=O)CCC1=O C1(C(N2CCC(c3ccon3)C2)=O)CCN(C(=O)CCCC2CCC2)C12CC2 c1(C(C)C(N2CCC(OCCNC(c3coc(CO)c3)=O)C2)=O)cncc(F)c1 C12(NC(c3ccc(F)s3)=O)COC(C1)C(NC(C1CCC3(CCC3)O1)=O)C2 C1(C(=O)NCCOCCO)(COC)C=CCN1C(=O)C(C)Nc1ccccn1 C(CC(O)C(=O)NCC(C(F)(F)F)N1CCN(C(=O)COC(F)F)CC1)SC CC(C)CCCC(C(=O)NCCc1cccc(F)c1)N1CCc2ccc(F)cc21 Cc1cc(C(=O)NC2CC2CNC(c2ccnc(C)c2C)=O)nc(C)n1 C1(NC(c2cc(COC)[nH]n2)=O)CC2CC(NC(c3cnn(C)c3N)=O)C2C1 N1(C(C(CC)=CC)=O)CCC2(CCN(C(=O)CN3CCn4ccnc4C3)C2)C1 c1(N(C)CC2CCN(C(=O)CCc3cccnc3)C2)cccnc1C1CC1 Cc1c(NC(=O)CC2CC(NC(=O)CNC3CCCCC3C)C2)cccc1Cl C1(C(=O)N(CC(=O)NCC(C)(C)N2CCCC2)C(C)C)(OCC)CCOC1 CCCC(CNC(=O)C(C)=NOCC#N)C(=O)N(CCCC(F)(F)F)C C=C1CCC(C(=O)NCCC2CC(OC)CN2C(=O)COCC2CCCC2)CC1 c1(OC)ccc(F)c2[nH]c(C(=O)NCCNC(=O)CC3(C)CCS(=O)(=O)N3)cc12 c1(C(=O)NC2COCCN(Cc3cnc(CCC)s3)C2)cc(O)c(O)c(O)c1 c1(C(=O)NC2CN(C(C(COC)O)=O)CC2O)c(C)nc(C2CC2)nc1O Cc1ccc(C(=O)NC2CC(CNC(c3scnc3C)=O)C2)c(Cl)c1 C#CCC(C)(C(=O)NCC(CO)C1CCC1)NC(=O)CC=CC=C C12(CC(=O)NCCCCO)CCC1CN(C(c1nccs1)=O)C2 N#CCCCCCC(=O)NC1C=CCCC1C(N1CCC2(CC(CO)C2)C1)=O N1(C(CC)C(=O)NC2CC(F)(CNC(=O)C(F)=C3CCCC3)C2)C(=O)CCC1=O CCCC(CCNC(C1(COC)CN(C(c2sccc2C)=O)C1)=O)CCC c1(C(=O)OC)n[nH]c(=NC(CNC(C2CCN(C3CC3)CC2)=O)CO)s1 c1(C(=O)OC)cnn(CC(=O)NCC2CC2NC(C2CC(F)C2)=O)c1 C1(C(=O)NCC(C(C)C)O)CCN(C(=O)C(C)C#N)O1 N1(C(Cc2cc(C)[nH]n2)=O)CCC2CCCC12CNC(c1cc(N)ccc1F)=O c1(C(=O)NC2C(OC)CN(C(=O)CCC(=O)c3ccc[nH]3)C2)cc(C)nc(C)c1 C1(NC(c2nc(Cl)c(Cl)s2)=O)COC2(C1)CN(C(C1CC(CF)C1)=O)C2 C1(NC(C(CN(C)C)N(C)C)=O)CCCC(CNC(=O)CCc2cscn2)C1 Cc1csc2ncnc(N3CC(NCc4c(O)cccc4O)CC(F)C3)c12 c1(C(N2C(C(=O)O)(COC)CCC2)=O)ccc2c(c1)CCCO2 Cc1cnc(CCCC(=O)OCC(=O)CCC2CC2(C)C)[nH]1 C1(CC(=O)NCCCCC=C)CN(Cc2cc(C)cs2)CCO1 S(=O)(=O)(CCC(=O)NCCC(F)Cn1cc(C(N2CCCC2)C2CC2)nn1)N(C)C C1(S(C)(=O)=O)(C(N2CC(CCNC(C(C(C)C)NC(C)=O)=O)OCC2)=O)CCC1 N1(C(C2CC(SC)C2)=O)CCC(CCCNC(c2nc(C)c(C)s2)=O)CC1 C(C(=O)NC(C)(C)C(=O)NCC(F)Cl)(C(C)C)SC Cc1cccc2nc(C(=O)NC3CCCN(C(C4(F)CC4C)=O)C3)cn12 c1(C(c2ccccc2)NCC(C2(O)CN(C(CC)=O)C2)(C)C)cccc(F)c1N C1(NC(C(N2CCOC2=O)C)=O)CC(NC(=O)C(C)(C)c2cnn(C)c2)CC1O c1(CC)ccc(C(=O)NC2(C3CCCN3C(c3cnc[nH]3)=O)CC2)c(C)n1 N1(C(C=CC=CCC)=O)CCC(CN(c2ncncc2C)C)CC1 c1(C(=O)OC)cc(S(=O)(=O)NCc2ccc(F)c(C#N)c2)c(C)cc1C C(=O)(C(CC(F)F)NC(C1CC(C)C1)=O)NCCC(C(=O)OC)O c1(C(=O)NC2CCC(CNC(C3C(C)=C3)=O)C2)cccc2nc(C)sc12 C1(CC=C)(C(=O)NC(C)CCNC(c2noc(C)c2C(=O)OC)=O)CCOCC1 S(=O)(=O)(c1ccccc1)NC(C(=O)N(CC(C)N)Cc1ccc(N(C)C)cc1)=O N#CC1(C(=O)NCC2CCN(C(c3cn(C4CCOCC4)nn3)=O)C2)CCCO1 S(=O)(=O)(c1ccc2c(c1)CCC2)N1CCC2(CN(C(C3C(C)C3)=O)C2)C1 N1(C(c2cn(-c3ccccc3)cn2)=O)CCC12CN(C(C1(F)CCCC1)=O)C2 Cc1ncc(CCC(N2CCSCC2CCNC(c2conc2C)=O)=O)c(O)n1 c1(C(N2CCCC(CNC(c3ccn(CC)n3)=O)CC2)=O)nn(C)c2c1CCC2 CCCC(C(=O)NC1COCC1NC(c1cc(C(N)=O)cc(F)c1)=O)S(N)(=O)=O c1(OC)c(CNC23CC(NC(=O)Cc4ccc(F)cc4)(C2)C3)cc(Cl)cc1Cl N1(C(C(CC)(C)COC)=O)CCN2CCN(C(=O)CCc3csnn3)CC2C1 c1(CCC(=O)NC2CCCC(NC(CC(CC)C)=O)C2)ccc2cnn(C)c2c1 c1(C(=O)NCCN(CC(C)O)C(C2CC2CF)=O)cnc(Cl)cc1N C=CC1CN(C(=O)C(O)C2CCCC2)CC1NC(=O)CC1CC2(CC2)C1 c1(C(=O)NCC2C(NC(c3c(C)nn(C)c3C)=O)CCCC2)cc(Cl)c(F)cc1O N1(C(C(C)OC)=O)CC(CNC(c2ccc(Br)c(F)c2)=O)C(C)(C)C1 n1(CC(=C)C)nnnc1C(c1cc(C)ns1)NCc1nocc1C(C)C c1(C(=O)NC2CCC(N(C(=O)C(=O)NC3CC3)C)CC2)cccc2c1CCC2=O c1(SCC(=O)NC2(C)CC(NC(C3(COC)CC=CC3)=O)C2)c(Cl)cccc1Cl CCC(O)C(C)(C)C(=O)NC1C2CC1N(C(=O)C(C)C(F)(F)F)C2 N1(C(COCCCC)=O)CCC2CCN(C(c3coc4cc(O)ccc34)=O)C2C1 Cc1cccn2cc(CC(=O)N(CCCNC(=O)Cc3ccsc3Cl)C)nc12 O=C1OC2CC(C(=O)NC3(CF)CN(C(C4CCCC(F)C4)=O)C3)CC2O1 N1(C(c2cn(CC)nn2)C(=O)NC)CCC2(CC1)OCC(C)(C)CO2 N1(C(C(C(=O)OCC)CC)=O)CCCN(C(c2cn(C(C)(C)C)nn2)=O)CCC1 C=CCC(CNC(=O)C(C)NC(c1cccs1)=O)NC(c1ccco1)=O CCCC(CNC(C1(C#N)CCOCC1)=O)C(=O)NC1(C(O)COC)CC1 N1(C(=O)OC(C)(C)C)CC2C(CSC3CC(F)(C4CCCN4)C3)C2C1 N1(C(C(C2CCN(C(c3n[nH]c(C)c3C)=O)C2)F)=O)CC(F)(C2CC2)C1 c1(COC)nn(C)cc1NC(C1CN(C(c2cncc(C)n2)=O)CC1C)=O C(CC(C(C)C)NC(c1ccccc1C(C)C)=O)N(C(C1(CC)CC1(F)F)=O)C c1(C(=O)NC(C(C)(C)NC(c2c(COC)nn[nH]2)=O)C)nn(C(F)F)cc1Cl C1(F)(CNC(c2ccccn2)=O)CCCN(C(c2ccc(C(F)F)o2)=O)C1 N1(C(CCC2CCC(C)NC2=O)=O)CC2CN(C(=O)C3=CCCC3)CC2C1 C(=O)(CCCC(=O)N1CCOCC(CNC(=O)CC(O)C2CC2)C1)N(CC)CC Cc1nc(N(C)Cc2cnn(-c3ccccc3)c2)n[nH]1 CC1CN2CCN1CC2C(=O)NCCCN(C)C(c1ccoc1)=O C1(NC(C2N(C(CN(CC)CC)=O)CCCCC2)=O)CCn2ccnc2C1 c1(C(=O)NCC2OCCN(C(C(C(COC)C)C)=O)C2)ccnc2c1CCC2 c1(C(=O)NC(C2CCN(C(c3scc(C)c3)=O)C2)C)sc2nccnc2c1N C1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)c2ccco2)COCCC1(F)F N1(C(C(OCC)OCC(=O)NCC2CC(Cl)(Cl)C2)=O)CCC(OC)C1 C1(C(=O)NC(c2ccc(Br)s2)C)C2CC(CC2F)N1C(C1CCC=CO1)=O C(CN=C(NCCF)NCC1CCCC12CC2)c1cccc(C)n1 N1(C(CC)C)CCC(CN2CCC(CC(C)C(=O)OC)CC2)CC1 c1(OC)cnccc1C(N1CC(CC(=O)NC2CC=CCC2)CC1C)=O Cc1cc(C)c(C(=O)NC(C2CCCCC2)CNC(=O)CC2CC(C(F)F)C2)s1 N1(C(C(=O)N(C(Cc2c(OC)cccc2)C)C)=O)CCCCC(S(C)(=O)=O)C1 C(=O)(C(CC)CC)N1C(CCCSCCNC(C(C)OCC#C)=O)CCC1 c1(CN2CC(CC(=O)Nc3nnc(C4CC4)o3)OCC2)cc(Br)c(Cl)cc1[N+](=O)[O-] c1(C2N(C(=O)NCc3cc(Br)c(Cl)s3)CCC2)ccc(F)cc1 c1(C(=O)NCC2N(C(=O)C=C3CCC3)CCN(C)C2)ccc(=O)n2c1CCCC2 N1(C(c2cc(CSC)cs2)C(=O)NCC)CCN(Cc2cccc(Cl)c2)C(=O)C1 c1(C(N(C(CNC(Cc2cccc(OC)c2)=O)C)C)=O)ccc(NC(C)C)nc1 C1(SC)COCC1N=c1nc2sccc2c(N(CCCNCC(C)(C)C)C)[nH]1 CC1CCCN(C(=O)CC2CCC2)C1CC(=O)N1CCCO1 C1(NC(C2C(c3n(C)cnc3)C2)=O)CC(NC(=O)Cc2cccc(O)c2)CC1O C1(CNC(=O)C(F)CC2CC2)CC12CCN(C(c1ccccc1O)=O)CC2 c1(C(=O)NCC(C)N(C)Cc2ccccc2C(C)(C)C)cn2c(n1)COCC2 N1(CC)CC(C(N2CCC(O)(C(C)NC(=O)CCOC)CC2)=O)CCC1=O C1(CC=C)(NC(C2CC(C)C2)=O)CCN(C(C2COC3(CCC3)C2)=O)CC1 c1(CCC)noc2nc(C)cc(C(=O)NCC3CC(O)CN3C(=O)C=C(Cl)Cl)c12 c1(C(N(C)CC2CCN(C(C=C(CC)CC)=O)C2)=O)c(C)nc(C)n1O c1(C(=O)NCC2C(NC(CC(C)C)=O)CCC2)ccc(OC(F)(F)F)cc1 CC(C)C#CC(=O)NCCS.n1(CCN(C(C)C)CC)cc(C(C)O)nn1 c1(C(N2CCN(C(C(CC=CCC)C)=O)C(CCO)C2)=O)cc([N+](=O)[O-])c(C)s1 C(CC(C)(C)CO)NC(C(C)CN(C)C(c1ccc(Cl)s1)=O)=O C1(NC(COCC#C)=O)CCN(C(c2cc(C)ccc2C)=O)C12CCC2 C(=O)(C(C)S(C)(=O)=O)N(CC(C)CNC(=O)COCCOCCO)C c1(CC(=O)N(C2CCC(NC(c3n(CC)ncn3)=O)C2)C)cc(OC)ccc1Cl CC1CCN(C(c2cc[nH]n2)=O)CCN1C(c1ccnc2ccsc12)=O c1(OC)noc(C)c1C(=O)NC(C)CCCNC(=O)CCCCc1cnn[nH]1 c1(C(=O)NC2C(C(=O)NCCOCC(C)C)CCC2)cc2cnccc2[nH]1 c1(C(N(CC(=O)OCC#C)C)=O)ccc(NC(=O)OC(C)(C)C)cc1 c1(C(=O)NC2C(CNC(C3CCCN(CC(=O)O)C3)=O)C2)cc(F)ccc1Cl c1ccc2c(c1)CC2CCN(C1(C2CCCO2)CC1)C1CC1 c1(C(C(N2CC(NC(c3cc(CCC)[nH]n3)=O)C3C2C3)=O)=O)c(C)nn(C)c1C CC#CCC(C(=O)Nc1cccc(N(C)C)c1)NC(c1cccc(Cl)c1)=O CC1(C)CCN(CCC(N2CCOC(Cc3cn(-c4ccccc4)nn3)C2)=O)C1 c1(C(N(OC)C)=O)c(ONC(=O)NC2C3CCC23)cnn1C Cc1nn(CCNC(=O)C(=O)NC(COCC2CCCO2)C(C)(C)C)c(C)c1C C(CCCCN=c1nc(N2CCC2)cc(Cl)[nH]1)NC(=O)OC(C)(C)C Cc1cc(C(N2CCCC2C(C)NC(=O)C(=O)NC(C)C)=O)ncc1C(F)F C1(C(N2C(CNC(=O)C=Cc3cccc(CO)c3)CC2)=O)CCC2CCCCN12 C1(O)(C(C)NC(=O)CC(C)C2CCCO2)CCN(C(C2(O)CCSC2)=O)CC1 N1(C(c2cn(C)nn2)=O)CCC(C)(CC(=O)NCC2C=CCS2)C1 C1(C2CN(C(C3CC3[N+](=O)[O-])=O)C2)(NC(Cc2cccc(C(N)=O)c2)=O)CC1 C1(C(N(CCC)CCNC(=O)CC2COC3CC2C3)=O)CSc2ccccc2O1 C(=O)(CCC(=O)NCC1COCCN1C(c1ccoc1Br)=O)NC C1(C(=O)NC(C2N(C(C(C)c3cccs3)=O)CCC2)(C)C)CC2CC(=O)C1C2 c1(CC(=O)NCC(C2CCOC2)NC(CC=C)=O)cnc(C)nc1O CC(O)CCCCCC(=O)N(CCO)CCOCCNC(=O)CCNS(C)(=O)=O c1(OC)cc(OC)c(Cl)c(C(=O)NCC(C)CN(C(=O)CC(C)SC)C)c1 C1(C(CC)(C)C)CCC(CNC(c2nnnn2CCCF)(C2CC=CC2)C)CC1 CC1OCCCC1COC(c1cnn(C)c1F)=O CC(N=c1nc(C2CCCC2)[nH]s1)C1CCN(C(=O)CNS(C)(=O)=O)C1 C(CC(O)C(=O)N(C1CC(C(=O)NCC(C)(O)CO)C1)C)N(C)C C1(OC)CC(NC(C23COCC2C3)=O)CN(C(=O)Cc2c[nH]nc2O)C1 c1(C(=O)NCC(C2CCOC2)NC(C(CCOC)(C)C)=O)ccc([N+](=O)[O-])n1C Cc1cc(F)c2cc(C(N3CCC(C)C(CNC(=O)C=CC(C)C)C3)=O)[nH]c2c1 c1(C(=O)NCc2c(C(=O)NC(C)C(C)n3cccn3)occ2)ccc([N+](=O)[O-])o1 C(=O)(C(CC(C)C)C(C)C)NCCC(=C)CNC(c1cc2c(cn1)OCCC2)=O c1(-c2nc(C(CCC)C3CC3)n(-c3ccccc3N(C)C)n2)ccc(C)c(F)c1 c1(CC(=O)N(CCNC(CC=C=C)=O)CCCCCCC)ccc(C(C)C)cc1 Cc1cc(=O)c(C(=O)NC2CN(C(=O)C(C)n3cccn3)CCC2C)cn1C C1(CNC(C(C)C)C(O)c2ccc(Cl)cc2)CCC(C)(C)N(C(=O)OC(C)(C)C)C1 N1(C(c2ccc(CSC)o2)=O)CCOCC1CCNC(=O)COC(=O)CO CCCCC(C(=O)NCC1CC2CCC(C1)N2C(=O)C1=C(C)CCC1)C(C)C Cc1ncc2ccccc2c1C(=O)NCC1CN(C(C)C)C1 CCCS(=O)(=O)C(C)C(=O)N1CC(C)(NC(=O)C=C2CCN(C)CC2)C1 C=CC(C(=O)NCC(C)(CO)NC(c1coc(N(C)C)n1)=O)OC c1(N2CC(NC(C(C)=CC)=O)C2)cc(C)nc(C)n1 CCC(F)(F)C(C)(C)C(=O)NCCNC(c1cnc(N(C)C)s1)=O c1(C(c2nnnn2-c2ccccc2OC)NCC(=C)Br)sc(Br)c2c1OCCO2 N1(C(CC2(C)CCCC2)=O)CCC(NC(=O)Cc2ccc(O)nc2)C(F)(F)CC1 c1(C(CC)=O)ccc(OCC(=O)NCc2csc(-c3cnn(C)c3)n2)cc1 Cc1cc(C(=O)N(CC(C)O)CCNC(=O)Cn2cc(Cl)cn2)cc(C)c1Cl N1(C(C=CC(C)C)=O)C2CCC1CC(NC(=O)CCCn1ccnc1)C2 C(=O)(C1CCc2nccn21)N(C1CC(C)(C)C1)C1CC1.C1(=O)CN(C)N1 N12CC3(CN(CCO3)C(=O)C1)C2.c1(C(=O)NCCC)scnc1C.OC C1(C)(C(N2CC(C)C2C(=O)NCc2ncsn2)=O)CC(=O)N(C)C1 C=CC(O)C(=O)NCC(C1CC1)N(C(=O)C(CC)=CC)C CC1CN(C(=O)CC2CCSCC2)CC1NC(C1OCCC1C(F)(F)F)=O c1(OC)cnc(F)c(C(=O)NCC(C)CNC(C23CC2C3)=O)c1 CCCCC(O)CC(=O)NCC1(O)CCN(C(c2nn(C)cc2SC)=O)C1 Cc1cnc(N2CCC=C(Cl)C2)c(S(=O)(=O)NC(C(C)C)c2cccs2)c1 C1(NC(C(C)NC(=O)NC)=O)CCN(C(=O)CC2CCCCC2C)CC(C)(C)C1 C(=O)(C(F)CC(C)(C)NC(C1CN(C)CCN1C)=O)N1C(C(C)O)CC1 C12CCN(CC1)C(=O)NC(=O)C2SC.C(C)(C(=O)NCCNC1CC1)N(C)OC.CO.N C12(C(=O)NC3CC(NC(C4(CC)CCOCC4)=O)C3)C3C4C1C1C2C3C41CO N1(C(C=NOC)=O)CCCC2(CC(NC(c3ccc(OC)c(C)c3)=O)C2)C1 C(=O)(CCC1=CCCCC1)N1C(CCNC(C2(C(=O)OC)CC2)=O)CCC1 N1(C(c2cc(C(C)C)on2)=O)CC(NC(C2SCCS2)=O)CC12CCCOC2 c1(C(=O)NCC(N2CCC(C(=O)OC)C2)=O)ccnc2ncccc12 C=CCC(CC)C(=O)NCCN(C(=O)CC(O)Cc1ccccc1)C C1(O)(C(=O)NCCCN(C(c2c(CCC)n(C)nc2)=O)C)CCCC(C)CC1 c1(C(C(=O)O)NC(C2C(C)C2)=O)ccccc1-c1ccccc1 c1(C(=O)NC2CCC(NC(Cc3c(C)noc3Cl)=O)CC2)cc(N)c(O)c(F)c1 N1(C(CCC2CC(CNC(C(C)C)=O)C2)=O)CCCCCC1CCO C(CN=c1cc(C2CC2)nc[nH]1)C1CCN(C(=O)Cc2cnoc2)CC1 C1(CC)CC(N=c2nc(NC3CCc4sc(Cl)cc43)c3ncn(C)c3[nH]2)C1 C1(C(=O)NCC(=O)NCC(=O)NCCO)(CC)CCCO1 CCC(C)C(C)C(=O)N(CCC(=O)Nc1cncc(C#N)c1)CC1CC1 C(=O)(CCCCC(N)=O)NC(C(=O)Nc1ccc(C)c(C)c1)(C)CO c1(CNC2CC(CCC)OCC2)ccc(S(=O)(=O)N(C)C)cc1C C(=O)(C(C)(O)C(C)C)NCc1c(C2CN(C(CCc3c(C)ncs3)=O)C2)ocn1 C1(NC(c2n(C(C)C)ncc2)=O)C2CCC1N(C(C1CC(=O)N(O)C1)=O)C2 N1(C(C(C(C)C)=O)=O)CCC(NC(C2CCC(=O)NC2)=O)C(F)C1 C(=O)(CC1OB(O)c2ccccc21)NCC1CN(C(=O)COC2CCCC2)C1 C(C)(CC1=CCCCC1)NC(C1(CO)CCN(C(C(C)SC)=O)CC1)=O c1(C(N2CC(C#C)N(C(=O)Cc3nc[nH]n3)CC2)=O)cn(C)c2ccccc12 Cn1ncc(C#N)c1C(N1CC(CCCCNC(C2CCNC2=O)=O)C1)=O C1(OC)CCCCC1C(=O)NCCNC(c1ccc(C(C)=O)[nH]1)=O c1(C(=O)NC2C(NC(C3(CCCC)CCC3)=O)CCC2)ccc(O)c(CO)c1 CC1(C)Cc2cccc(CC(N3CC(NC(=O)C(F)C4CCOC4)C3)=O)c2O1 C#Cc1cccc(C(=O)N(C2CN(C(=O)CCC=CC(C)C)CC2O)C)c1Cl N1(C(C=CC(CC)C)=O)CC(C(=O)NCc2conc2C2CC2)C2(CC2)C1 Cc1cc(NC(=O)C(c2cn(CC3CCCO3)nn2)N(C)C(C2CC2)C)ccn1 C(=O)(C(CCC)C(C)C)NC(C(=O)N(C)CC1CC(=C)C1)CC1CCOCC1 CCC(C)(F)C(=O)NCC12CC(NC(=O)C(c3cccc(Br)c3)C)(C1)C2 C1(C(=O)NCCC2(NC(C3CCC(CSC)C3)=O)CCC2)CC2CC(=O)C1O2 N1(C(CCSCCC)=O)CCCC(COC)(NC(C2CC(=O)NC(C)C2)=O)C1 C1(C(N(CCCC)CCOC)=O)(CO)CCN(C(c2cc(C)cs2)=O)C1 C1(C(=O)OC)(N(CCCC2CCC2)C)CC(C(c2ccccc2)C)C1 S(=O)(=O)(c1cccc(Cl)c1F)NC1CCC(NC(=O)Cc2ccc(Br)cc2Cl)C1 N1(C(CC2(C)CCN(C(CC(C)C(F)F)=O)C2)=O)CCC2(C1)CC2(F)F c1(CN(CCCCCCCCC)C)cc(=NCC(C)CN(C)C)[nH]cn1 c1(C(N(C2CCN(C(c3noc4ncccc34)=O)C2)C)=O)cnc([N+](=O)[O-])n1C S(=O)(=O)(c1cccc(-c2ccsc2)c1)N.c1(C2C3(CC3)N2C)ccccc1F C(=O)(CC(C)(C)C(=O)N1CCCC2(NC(c3cc(C)no3)=O)CC2C1)OC c1(C(N(CC(C)O)CCNC(CC(C=C)C)=O)=O)cc(S(N)(=O)=O)cc(Cl)c1F Cc1noc(C)c1CC(C)C(=O)NC(C)CN(C(=O)COC1CCCCC1C)C O=C(CCC=CBr)NC1CC(NC(C2CC2c2ccccn2)=O)CC1O O(n1nnc2c1CCCC2)Cc1cccc(NC(CC2CN(C(C)=O)C2)=O)c1 N1(C(CCN(C)CC)=O)CCN(C(=O)CC2OCCC2(C)C)CC1c1ncc[nH]1 c1(NC(C(C)CNC(c2nc[nH]n2)=O)=O)ccc[n+]([O-])c1 N1(C(C(c2scc(CC)n2)(F)F)=O)CCOC2(C1)CN(C(=O)C(F)(F)CO)C2 c1(NC(c2n(C3(C)CC3)nnn2)(C)CCCl)cccc(-c2ncon2)c1 C(=O)(C(C)(CC)CCC(C)C)N1CCC(O)(CNC(C(C(CC)(C)C)O)=O)CC1 C1(NC(CC=CC=C)=O)CCN(C(c2csc(C(=O)OCC)c2)=O)CC1F C1(=O)CCCCCN2CCOC(C2)CCN1.c1(CCC#N)cn(CCF)nn1 c1(NC(N2CCCC2CC#N)=O)ccc(O)c(CCNC(C)=O)c1 C1(C(NOCc2cn(C3CCC(C(=O)O)C3)nn2)=O)CCCCC1O c1(CC)nc(=NC(CNC(c2ccc(F)cc2C(F)F)=O)C2CC2)s[nH]1 O=C(C(O)CC(O)CO)N1CC(O)(c2cn(Cc3nc(C(=O)O)cs3)nn2)C1 C1(COC)CN(C(=O)C(Cn2ccnn2)NC(=O)C(C)CSC)C1(C)C C1(N(C(=O)NC(CCCSC)C)C)CC2CCC(C1)N2C c1(C(=O)Nc2cccc(CNC(CC3(COC)CC3)=O)c2)ccc(S(N)(=O)=O)o1 CC1(C)CC(CNC2CCSCC2)CCN1C(C1C2COCC12)=O C1(CC(=O)NCC(COC)NC(c2nc(Cl)oc2C)=O)C(=O)NN=C1C Cc1cc(=O)n(C)cc1C(=O)NC(C)CC(C)NC(=O)CCCCNC(N)=O CC1(C)C2C1NC2=O.C(=O)(C(O)CC1CCCC1)N(C1CCCC1)CCO C(C(O)C(=O)N1CCCC1c1ncc[nH]1)NC.CC(C(=O)C(C=C)=O)c1ccsc1 C1(NC(C(C)NC(c2nc[nH]c2C(C)C)=O)=O)CCCCN(Cc2cccs2)C1 c1(OCC)cc(C(=O)NCCN(C(=O)C(C)CCOC)C(C)C)cc(F)c1 N1(C(C(C)n2cccn2)=O)CC2COCC2(C(=O)N(C)CC2COCCO2)C1 C(c1ccc(C)cn1)=CC(=O)NC1C(NC(CC(=O)OC)=O)COC1 c1(OCC(=O)NC(CN(C(=O)CC2(C)CCOC2)C)(C)C)ccc(F)cn1 c1(C(=O)NCC(C2CC2)NC(=O)C=CC=C(Cl)Cl)cnc(O)o1 c1(OCCOC(c2ccc(C(F)(F)F)cc2)CS(C)=O)ccc(S(N)(=O)=O)cc1 N1(C(C(CCC)NC(=O)CCCN(C)C(C)C)=O)CCNC(=O)C1CCO C(CC(C(C)(C)C)NC(c1cnc(S)[nH]1)=O)N(C(=O)CC1CCC(=O)NC1=O)C c1(C(N2C(CNC(CCc3scc(C)c3)=O)CCC2)=O)cn(C)c(=O)nc1O c1(CC(N2CCN(C(COCC#C)=O)CC2COC)=O)sc2ccccc2c1C c1(C(N2C(C)CC(NC(c3nonc3N)=O)CC2)=O)cc2ccccc2cc1F CCC(C(=O)NC1CC(CNC(=O)C(C)(C)Oc2ccccc2)C1)C(C)O CC1(C)CCCC(CNC(C2CCCC2CNC(=O)Cc2cc(Cl)cs2)=O)C1 C12(NC(c3cc(=N)[nH]cc3)=O)CCCC1CN(C(C1CCC(=O)N1)=O)C2 C1(CC(=O)NCC(C)(C2CC2)NC(CCCNC(C)=O)=O)CCC(F)(F)CC1 C1(CNC(c2ccc(Br)s2)=O)COCCN1C(c1ccc(OC(F)F)cn1)=O C#CCCN=C(NCC1CCCN1c1nccs1)NC1CCOc2ccccc21 c1(CC)c(Cl)nc(C)[nH]c1=NCC=CCNC(C1CC2CCCC(C1)C2(C)C)=O C1(NC(C2C(OCC)CC2)=O)(COC)CCN(C(c2nnc(S)n2C)=O)CC1 N1(C(c2ccc(CC)o2)=O)CCC(C)(C)C1C(=O)NCc1ncnn1C C1(C)(NC(c2ccc(C(C)=O)[nH]2)=O)CCN(C(=O)CCC(C)N(C)C)C1 C1(NC(c2cn(CCC)nc2)=O)CN(C(=O)C=C2CCCC2)CC1S(C)(=O)=O c1(CCC)cc(C(N2CC(NC(=O)C(C)=C3CC3)C2)=O)cc(O)n1 C1(COC(=O)CCCc2ccccn2)CCCC1C(=O)NC(=O)OC(C)(C)C N1(C(CCc2cc(C)sc2C)=O)CC(C(=O)O)CC(C(=O)O)C1 C1(NC(c2nc(SC)sc2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC1C C1(C(=O)NCC(CC=C)NC(=O)C=Cc2cn[nH]c2)CCC(=O)N1CCC n1(CC(=O)NC(CC=C)CNC(C23CC(C)(C2)C3)=O)ccc2c(C)cccc12 C1(CC(N2C(NC(C(CC)N(C)C)=O)CC2)=O)CCC(C(C)C)CC1 c1(C(=O)NC2CC(C(N3CCn4cc(Br)nc4C3)=O)C2)nccc2ccccc12 C=CCC(C)(C)CNC(=O)C(Cc1cc[nH]n1)NC(c1cn(COC)nn1)=O N1(C(C(=O)NCC2C(c3onc(C)n3)OCC2)=O)CCc2ccccc21 N1(C(CN(CCC)C(c2n[nH]cc2C)=O)=O)CCC(F)(CC)C1 C1(C)(C(=O)NC(C(C)C)Cc2ccc(I)cc2)COC(C)CO1 C1(NC(=O)Cc2ccon2)CCCC1NC(C1(c2ccccc2)CC(O)C1)=O CCCC(C(=O)NC1CCCC1NC(=O)CCc1cccnc1Cl)NC(N)=O c1(OCC)ncnc(OCC)c1C(=O)NCC1CC2CN(C(=O)CCC)CC12 N1(C(COCC(C)C)=O)CC2=C(C1)CN(C(C1CN(CP(C)(C)=O)C1)=O)C2 N1(C(C2=CC(O)C(C(C)(C)C)C2)=O)CCc2cc(Br)c(Br)cc2C1 N1(C(c2nc(OC)oc2)=O)CCN(C(C2CCCNC2=O)=O)C(C2CCCC2)C1 CCC(C)C(C)(O)CNC(C1CN(C(=O)CCC2OCCO2)CC1(C)C)=O C1(OC)CN(C(c2cc(C)sn2)=O)CC1NC(c1ccon1)=O C1(CS(=O)(=O)NC(C(n2cc(-c3ccc(C(=O)O)cc3)nn2)C)=O)CCC(C)(C)C1 n1(C(CC)CC)nccc1C(=O)NC1CC(NC(=O)Cc2occc2C)C1 C1(NC(C(=O)NC(CCCC=C)C2CC2)=O)(CF)CC12CCOCC2 c1(C(=O)NCC2CC3CN(C(CC=CC=C)=O)CC32)c(Cl)nc2sc(C)cn12 C1(NC(C2(C)C(C)C2)=O)CC2CN(C(=O)CCC(=O)N(C)C)CC12 C1(CC)(NC(c2ccc(OC)cn2)=O)CCCN(C(C2CCCC23CCC3)=O)C1 C(=O)(CCC(F)(F)C(F)F)NCCN(C(CCC1C(C)(C)C1)=O)C1CCCC1 C1(C(=O)NCC(C)(C)CNC(=O)Cc2cncnc2O)CC2(C1)CC1(CCC1)C2 C1(CCC)CN(C(=O)Cc2cncn2C)CC1C(=O)N(c1ccc(C)cc1)C Cc1cc(C(N2CC3CC3(CNC(=O)C(C)(C)C)C2)=O)c(Br)s1 C1(NC(CCC(=O)N(C(C)C)C)=O)CCCN(C(=O)CC(F)(F)F)CCC1 N1(C(C2CC3CCC3C2)=O)CCC2C1CCCN2C(c1cccnc1S)=O C1(C(=O)NCCCCOCC)(CNC(C2CCC(C)C2)=O)CC=CC1 C=CCC(C)C(=O)N1CCC(N2CCC(NC(c3snnc3CC)=O)C2)CC1 CCC(C)CCC(=O)NCC(O)CNC(c1csc(Br)c1)=O C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CCCN(C(C(CC)OC)=O)C(CO)C1 C(=O)(C1c2ccccc2C(=O)N1C1CC1)OCCSCC(=O)OCC c1(CC(=O)NCC2(NC(C3CC(Cc4ccccc4)C3)=O)CC2)nccnc1O CC(C)(C(=O)N1CCCC(C(C)(O)CNC(=O)Cn2ncnn2)C1)S(C)(=O)=O C(=O)(C(N=[N+]=[N-])C(C)C)NC(CN(C(C1CC2OC1C1CC21)=O)CC)C c1(C(N2CCC(n3ccnc3)C2)C(=O)NC(C)(C)C)ccc(Cl)c(Br)c1F CC(C)CC(C)(O)C(=O)NC1CCCC1NC(=O)CCc1cnn(C)c1 C1(NCC(=O)OCCCC)CCOC(C(=O)OC)C1 N1(C(C2CN(CC)C(=O)C2)=O)CC(NC(=O)CSCC(F)F)C(C2CC2)C1 c1(CC)nc(C(=O)NCC2(C)Oc3ccccc3O2)c2ccccn12 C1(c2cn(C3CCC3)nn2)(N(C)C)CCN(C(=O)CCc2ccccn2)C1 c1(OC)cc(CCC(=O)NCC(C)(C)NS(C)(=O)=O)ccc1Br c1(C(N2CC(NC(C(C=C)CC)=O)C(SC)C2)=O)nc(C)ncc1Cl C(C1CCCCCC1)=CC(=O)NCC(CNC(C(c1c(C)noc1C)C)=O)F N1(c2[nH]c(=NCc3cn(C)[nH]c3=N)[nH]c(=N)n2)CCc2[nH]c(=N)nc(O)c2C1 C1(C(N(C)CCF)=O)CCCC(NC(=O)CN=[N+]=[N-])CC1 Cc1ccc(C(N2CCCCC(NC(=O)Cc3cc[nH]n3)C2)=O)cc1C c1(COC)sccc1C(=O)NC(C)CNC(=O)CC1(C)CC1(Cl)Cl c1(NC(=O)C(=O)OC)ccc(Cl)cc1OC.c1(OC)ccc(C2CC(=O)O2)cc1 CC1=C(C(=O)NC2CN(C(c3ccc(C(N)=O)[nH]3)=O)CC2(C)C)CCC1 c1(C(=O)NCC2C(C)CN(C(=O)CCCF)C2)ccnc2[nH]cnc12 N1(C(CC2N(C(C)C)CCC2)=O)CCOCC1CNC(=O)CNS(C)(=O)=O c1(C(=O)NCC(C)(CNC(=O)C(=O)N(C)C)OC)cncc(SC)n1 c1(NC(C2(F)CCN(C(C(NC(C)=O)=Cc3cccs3)=O)C2)=O)cn2ccsc2n1 Cc1c(C(N2CC3CN(C(c4cc(C)n(C(F)F)n4)=O)CC23)=O)cc(F)cc1Br c1(C(N2CCC(C)C2CNC(c2cncnc2)=O)=O)cnc2c(F)cccc2c1 Cc1cc(NC(C2CCC2NC(C2CC(=O)C2(C)C)=O)=O)ccc1F C1(NC(C2(C=C)CC2)=O)CCCC(NC(=O)C(c2cccc(C)c2)C)C1 c1(CC(=O)NC2CCN(C(C(CCC)O)=O)C2C(C)C)c(OC)cccc1OC N1(C(C(=O)NCCOCC)C2CC2Cl)CCC(NC(c2oncc2C)=O)C1 CC(C)CC(O)CC(=O)N1CCC(O)(CNC(=O)C(F)=CCCF)C1 c1(NC(C2CCC(NCc3c(Cl)ccc(C)c3F)C2)=O)c(Cl)cc(Br)c(Cl)c1Br Cc1c(C(=O)NCC2CN(C(=O)C3=CC(C)CC3)C2)[nH]c2ccccc12 c1(C(=O)NC2CN(C(CC(C)(C)OC)=O)C(C)C2)c(N)c(F)cc(F)c1F C1(CC(=O)NC(C(C)C)C2CC2)CCN(C(=O)CC2=CCCC2)CC1O C1(NC(=NC)NCc2ccccc2)CCC(C(F)F)CC1 c1(C(N2CCN(C(COCC)=O)C(CC)C2)=O)c([N+](=O)[O-])ccc(C)c1C N1(C(COCC(=O)OC)=O)CCCC1CNC(=O)CNC(c1cnoc1C)=O c1(CC(=O)NC2C3CC2N(C(C24CCCC2C4)=O)C3)ccc(Cl)cc1F C(CC(C)C(=O)N1CCC(C(=O)NC2(C(F)F)CCC2)C1)=CCC CC(C)CC(C(=O)N1CCN(C(=O)CCC(C)N(C)C)CC1C1CC1)N(C)C C(=O)(C(C)(C)C(C)(F)F)N(CCNC(c1snc(-c2ccccc2)c1N)=O)CC Cc1c(C(=O)N(C2CCC(NC(=O)C3=NOCC3)C2)C)sc2[nH]cnc(=S)c12 c1(CC(C(=O)C(C)C)O)cccc(Cl)c1.C1(C(=O)NCCN)(C2CC2)CC1 N1(C(CCCCC)=O)CC2(CCCC2NC(c2ccc(OC)cc2N)=O)C1 N1(C(CC(CC)SC)=O)CC(NC(c2cnc(O)cc2C)=O)CC1(CC)CC C(CC(C(C)C)NC(C1(CF)CC(F)(F)C1)=O)NC(C(C=CCCC)O)=O C1(CNC(CC=CC=C)=O)C(C)CCN1C(=O)CCCNC(N)=O Cc1[nH]c2cccnc2c1C(c1nnnn1C(C)(C)C)NC1CCC1 C1(NC(C2(OC)CCC2)=O)CCCCCN(C(=O)Cc2cnns2)C1 N1(C(=O)C(O)CCCNC(=O)C(F)(F)CO)CCCC2(CCCO2)C1 C(=O)(CC(C(C)C)C(C)C)NC1COCCN(C(CCCC(=O)NC)=O)C1 CCCCCC(CC)C(=O)NCC1CN(CCCC2CCC2)CCO1 C1(O)(CNC(CCCOC)=O)CCCN(C(=O)Cc2ccn(CC(F)(F)F)n2)C1 N1(C(c2cc(CC)cc(F)c2)=O)CCCC2CN(C(C3CC(C(=O)OC)C3)=O)CC12 C1(C(N(C2CCN(C(c3cc(C#N)c[nH]3)=O)C2)CC#C)=O)OCCN(C)C1=O c1(SC)cc(C)c(C(=O)NCC2CC2NC(=O)CSc2ccccc2F)o1 Cc1sc2ncc(C(=O)NC3CC(F)CN(C(C4CCOC4=O)=O)C3)n2c1C N1(C(C(C)C(F)F)=O)CC(C)(C)CC1CNC(=O)C(F)C(C)(C)O N1(C(c2c(C)con2)=O)CCCCC1C1CCN(C(=O)CCn2cnnn2)C1 N1(C(CCCOCC)=O)CC2(CCCC2NC(C2CCC(N(C)C)CC2)=O)C1 C1(N(C(=O)C=Cc2cn[nH]c2)CC)CCC(NC(=O)C(F)OC(F)(F)F)CC1 C1(C(N2CCOCC(CO)C2)=O)CN(C(c2csc(Cl)c2)=O)C2(CCC2)C1 c1(C(N2C(C)(CNC(C3(O)CCOCC3)=O)CCC2)=O)cc(F)cc(F)c1O N1(C(CSCC=C)=O)CC(NC(c2ccc(F)cn2)=O)C(C)C1 N1(C(c2n(C)ncc2)=O)CCC(CO)(NC(=O)Cc2cnoc2)C1 C1(C2CN(C(C3CCNC(=O)C3)=O)C2)(NC(C(c2c(C)n[nH]c2C)C)=O)CC1 CCC(CC(=O)N(C)CC1COCCN1C(=O)Cc1cc(SC2CC2)on1)SC Cc1cn(CC(=O)NC(C)(C)C(C)NC(=O)C=CS(C)=O)nc1C(F)(F)F C(=O)(CS(N)(=O)=O)NCC1(COC)CCCN1C(=O)C(CO)OC N1(C(c2c(CNC(c3nccc(C)c3N)=O)ocn2)=O)CCC12CCN(C)C2 c1(C(=O)NCCOCC(=O)N(CCCC)CC)oncc1C c1(C(=O)Nc2nc(C)c(C(N3C4CCC3CC4)=O)s2)cc(C(F)(F)F)ccc1O S(=O)(=O)(CC(=O)NC1CCC1C(=O)NC1CCN(c2ccccc2F)C1)N(C)C c1(C(N(CCCNC(=O)C(O)CC(F)(F)F)C)=O)ccc2nc(S)oc2c1 CC#CCCC(=O)NC(COCC)C(=O)NCC1(CC)CCOC1 c1(C(N(C(C)C)CCN(C(=O)CC2(C)CC2F)C)=O)cnc(O)c(C(F)(F)F)c1 C1(C(=O)NCC(C)N(C)C(c2ccnc(Cl)c2O)=O)CCc2nncn2CC1 CC(C)C#CC(=O)N1CC(O)CC1CNC(=O)C(C)(C)n1cc(Cl)cn1 CCC(C)CCCC(=O)NCC(=O)NCC(=O)N(C)Cc1csc(C)n1 c1(N(CCOCCN(C(CC(C)OC)=O)C)C)cc(C)ncc1C#N N1(c2n(CCC=C)c(Cc3cccs3)nn2)CCC2(CCC(=O)N2)C1 N1(C(c2c(NC(c3cc(C)no3)=O)cn(C)n2)=O)CCCC(O)(C(C)C)C1 c1(C(=O)NCC2CC(NC(C3(CCC)CC3)=O)C2)cnn2c1OCC(O)C2 Cc1ncc(Cl)cc1NC(C1CC(O)CN1C(c1cnon1)=O)=O c1(C(=O)NCC2CC(CNC(CC=C)=O)OC2)ccc(CCC)nc1 C=CCC(C)(O)C(=O)N1CCC(C(=O)NCCC2(OCC)CCC2)C1 c1(C(=O)NC)ccc(-n2nc(CS(C)(=O)=O)nc2CCOC(C)C(=O)O)cc1 C1(CNC(c2c(C)c[nH]n2)=O)COC(C)(C)CN1C(C12CCCC1C2(F)F)=O CC1(C)CC(CNC(C2(C)COCCO2)=O)N(C(=O)CNC=O)C1 C(=O)(C(C)CC(=O)NC1CCCC1C(=O)NC1(C)CCC(C)(C)C1)OC C(=O)(C1=CC2C=CC1C2)N(C1CCCN(C(Cc2ccn(C)n2)=O)C1)CCO N1(c2nnc(C(C)C)n2C2CC2C)CCC=C(c2ccccc2)C1 c1(C(=O)NC2CC(CNC(c3c(CCC)nco3)=O)C2)cc2c(n1C)CCOC2 Cc1cc(C(N2CCN(C(c3ccccc3)=O)C3CC23)=O)cc(C)c1 c1(C(=O)NC2CCCCN(C(C=CC(C)C)=O)C2)ccc2ncnn2n1 c1(C(N2CCCC(F)(CNC(CCCC)=O)C2)=O)cc(C)c(F)c(S(C)(=O)=O)c1 N1(C(C(C)SC)=O)CCCC(C)C1CNC(C1COC(=O)N1)=O c1(C(=O)NCC2CC(NC(CSCC)=O)C2)cn(C)nc1C c1(CNC(C=C(CC)C)=O)nnc2n1CCN(C(=O)CCCc1ccccn1)C2 N1(C(C(C(C)C)F)=O)C2CCC1CN(C(=O)CCc1nnc(S)nc1O)C2 N1(c2nccc(C)n2)CC(C(=O)NCCN2CCCCC2)CC(F)C1 N1(C(CCCSC)=O)CC2CCN(C(c3cccc(-c4ccncc4)c3)=O)C2C1 c1(CNC(C2C(C(=O)OC)C2)=O)ncoc1C1CN(C(=O)Cc2cscn2)C1 CC1CCCn2ncc(C(=O)NCCC(C)CCNC(=O)CC3CC3)c21 N1(C(CCC(=O)NCC)=O)CCCC(F)(CNC(=O)C(=Cc2cnc[nH]2)C)C1 C12(CNC(c3c(CC)ccs3)=O)CN(C(C3(C#N)CCC3)=O)CC1CCO2 CCCCC(C)(F)C(=O)NCC1CCCN(C(c2nscc2C)=O)C1 c1(CC(=O)NC(CNC(CCc2cc(C)no2)=O)C2CCC2)ccc(C)c(Cl)c1 c1(NC(=O)Nc2cccc(OC(C)=O)c2)cccc2sc(Cl)nc12 C(=O)(C1=Cc2cc(C)ccc2OC1)NC1CN(C(c2n(CC)cnn2)=O)C2C1C2 C#CC1COCCN1C(=O)Cn1cc(-c2ccc(F)cc2N)nn1 N1(C(CC(=C)C)=O)CCC(C(CO)NC(c2cc(OC)no2)=O)CC1 C1(CC(=O)N(C(CC(CC)C)C)C)CC2(C1)CN(C(c1c[nH]nc1C(F)F)=O)C2 N1(Cc2ccc(C#C)cc2)CC(=O)NCC1(C)C(=O)OCC C1(NC(C(C(C)OC)O)=O)(CC)CCN(C(=O)CC(=O)NCC2CC2)CC1 Cc1c(O)cc(C(=O)Nc2cccc(-c3ccccc3NS(C)(=O)=O)n2)cc1O C(C(C)CCC)(c1nnnn1CC1CC1)NC(CC)CC(N)=O C#Cc1nc(C(=O)NCCC(C)N(C)C(C2CCOC2=O)=O)cs1 C(CCC(N)=O)(C(=O)N1CCC(Cc2cn(Cc3ccno3)nn2)C1)NC(C)=O CC(C)CC(F)C(=O)NC1CN(C(c2ccc(O)c(C(C)(C)C)c2)=O)C(C)(C)C1 C1(C(=O)NCCC(C)N(C(=O)CC(C)(F)F)C)CN(C(N)=O)CCO1 CC1CC(CCNC(=O)C=CSc2nc[nH]n2)CCN1C(c1cc(Cl)n(C)n1)=O C1(NC(CCN(CCCCC)C)=O)C=CC(CNC(=O)C(=O)NC2CC2)C1 Cc1c(NC(C)C)cccc1C(=O)NCc1nc(C2CC2)nn1C C(=O)(C1CCc2nccn21)N1CC2(CCC(CNC(=O)Cc3ccccc3)O2)C1 CCC(C(=O)NCC1(CCNC(=O)C=C2CCC(C)C2)CC1)C1CCOCC1 C1(OCC)CC2CN(C(C3C(C)CN3C(=O)CC3CC=CC3)=O)CC12 C1(CC=C)(NC(C2CCCN2C)=O)CCN(C(=O)C(C)S(C)(=O)=O)CC1 N1(C(CC(C)(C)SC)=O)CCN(C(C2(C)C=CCCC2)=O)CC(C)C1 n1(CCCC)cc(C(=O)NCC(C)NC(c2cscc2CC)=O)nn1 Cc1nc(C)c(C(N2CCCOC(CCNC(C3COC(=O)C3)=O)C2)=O)c(C)n1 C(=O)(C1CCc2ccc(Cl)nc21)NC1CN(C(c2ccc3ccn(C)c3c2)=O)C1 C1(C#N)(C(=O)NC(CN(C(C(CCC)N(C)C)=O)C)C)CCSCC1 n1(CC)cc(CCNC(=O)CCN(C(C2CC(F)C2)=O)CC)nn1 c1(C(=O)NC2CN(C(CC(=C)C)=O)C(C)CC2)cnc2n(c1=O)CCS2 c1(C(=O)OC)ccc(C(=O)NC(CO)C(C)NC(=O)Cc2ccsc2C)o1 C(=O)(C(=O)C(C)(C)C)N(c1ccc(C(c2cn(CCO)nn2)N(C)C)o1)C(C)(C)C CCC(C)CCCC(=O)NCC(C1CCN(C(=O)C#CC2CCC2)CC1)(C)C C1(C)(CNC(C2(CCCC)CC2)=O)CCCN(C(c2ccc(O)cn2)=O)C1 C1(C)(NC(CC=C)=O)CCN(C(=O)C(c2ccccc2C)(C)C)CC1 c1(C(=O)NC2(CNC(c3c(CC)noc3C)=O)CC2)ccc(C)c(F)c1N C1(C)(NC(c2ccn(CC)n2)=O)CCCN(C(=O)CC2CCOCC2(C)C)C1 c1(OC)c(OC)c(CNC2(c3ccccc3)CCOC2)cc2ccccc12 c1(C(C)(C)NC(=O)COc2ccncc2)ccc(O)cc1F C1(C(=O)NC2CCCC2C(N)=O)(COC)C=CCN1C(=O)CC1CCCO1 C1(C(N2C(COC)CC2)=O)C(C)CCN1C(=O)CCCc1cnn[nH]1 N1(C(C2(C(=O)OCC)CC2)=O)CCC2CN(C(=O)C=CBr)CC2C1 Cc1noc(C)c1S(=O)(=O)Nc1ccc(CNC(C2CC(C)CN2)=O)cc1 c1(OC)ccc(C(N2CCCC(C3CCCN3C(c3cc(Br)c[nH]3)=O)C2)=O)cn1 CC1CC(C(=O)NCCC2CCC(=O)N2C)N(Cc2cccc(C(F)(F)F)c2)C1 Cc1cc2c(C(=O)NCC=CCNC(C3CCS(=O)(=O)N3C)=O)cccc2o1 N1(C(C=C(C)C(F)F)=O)CCN(C(C2CC2C(C)(C)O)=O)CC1CO N1(Cc2n(CC#C)ccc2)CCC(NC(=O)C(C)OCC(C)C)C(O)C1 N1(C(C2(C)CCCN(c3cc(C)ncn3)C2)=O)CCc2cc(C#N)ccc2C1 N1(C(C(=O)N(CC(F)Cl)CC)=O)CCCC1(C)C N1(C(CC(=O)OCC)=O)CC2CCCC(NC(=O)C=C3CCCC3)C2C1 C1(CC(=O)NCCC(=O)N(C)C2CC2)CCN(C(=O)Cc2cnn(C)c2)C1 c1(CC)cnc(Cl)nc1N1CCC(F)(CNC(=O)Cc2c(C)nn(C)c2C)CC1 N1(C(C(C(=C)Cl)(C)C)=O)CC(C2CCN(C(c3cc(O)nc(O)n3)=O)CC2)C1 c1(C2(C(=O)NC3CC(CNC(C4CC=CCO4)=O)C3)CC2)ccc(F)cc1F C1(C(N(CC(CNC(CC=CC)=O)C)C)=O)CC(=O)N(C(C)(C)C)C1 Cc1nn(C)c2nc(N3CCOCC(CNC(=O)C(O)C4CC4)C3)c(C#N)cc12 N1(C(c2c(C)n(CC(F)F)nc2)=O)CCC(C)(NC(C2CNC(=O)N2C)=O)CC1 Cc1nc(C(=O)N(Cc2cc(-c3ccccc3)cs2)Cc2cnn(C)c2)cs1 c1(SC)nn(C)cc1C(=O)NC1(C)CC(NC(=O)Cc2ncc(C)s2)C1 C1(C(=O)NC2C(NC(C34CC(C(C)C)(C3)C4)=O)CC2)CC2CCC(C1)O2 CN(C)S(=O)(=O)NCC(=O)NCC1CC(O)CN1C(C1C(Cl)(Cl)C12CC2)=O N1(Cc2nn(C)c3c2CNCC3)CC2COC(C)(C)OCC2C1 S(=O)(=O)(c1ccc(NCC(O)C2CC2)c(C#N)c1)N(C(c1ccccn1)C)C c1(C(=O)NC2CC(C)N(C(=O)CC3CC(C)(C)C3)CC2)cc(C#N)c(F)cc1F CCCC(C#N)C(=O)NCC1CC(NC(c2nc(Br)sc2C)=O)CCO1 C12(C(N(CCCNC(c3c(OC)cc(O)nc3)=O)C)=O)OCCCC1C2(F)F c1(OC)cccc(Cl)c1C(=O)NCC1(C)CCCN(C(=O)CCN(C)C(C)=O)C1 N1(C(CC2CN(C)CC2O)=O)CC2CN(C(c3cccc(=O)n3C)=O)CC2C1 C1(NC(=O)C=C(C2CC2)C2CC2)CC1C1CCCN(C(=O)Cc2nncs2)C1 C1(NC(=O)Cc2cncs2)CN(C(c2c[nH]nc2C(F)(F)F)=O)CCC1CO C(CC(O)C(=O)N1CCC(NC(=O)C(F)CC2CCC2)CC1)SC c1(C(=O)NC2CN(C(c3c(SC)csc3)=O)CC2C)noc2c1CCCC2 c1(CC(=O)NC2CC(CCNC(c3[nH]cc(C)c3)=O)C2)ccc2c(c1)CCCO2 C#Cc1ccc(-c2cnc(OC(F)(F)F)c(C(N3CCCOCC3)=O)c2)cc1 Nc1ccc2ncsc2c1.c1(C=O)sc(Cl)nc1Cl.N12CC(O)(C1)C1CCCN21 C1(CNC(c2cccc(N(C)C)c2)=O)CCN(C(c2snc(C)c2N)=O)C(C)C1 C1(N(CC(=O)NC2CCCCS2)C)CCCC(NC(c2ncccc2Cl)=O)C1 N1(C(C(=O)NCC=C)C)CCC(CN(C(C2CCC(C)O2)=O)CC)CC1 CC(C)(Cc1ccc(Cl)cc1)CC(=O)NCc1cc(Cl)n[nH]1 C1(CCNC(c2c(CC)cno2)=O)COCCN1C(c1cc(C)sn1)=O c1(NC(C(=O)NCCN2CC(c3ncc(Br)cn3)(O)C2)=O)ccccc1C(F)(F)F C(CCCC(=O)NC1CCC(NC(c2ccoc2)=O)CC1)NC(=O)OCC=C C(=O)(C1=C(C#N)CCC1)N1CCC(CCNC(CNC(=O)OCC)=O)C1 c1(-n2c(C)cnn2)ccc(C(N2CC3C(NC(c4ccccc4)=O)C3C2)=O)cc1 C=CC1CCN(CC(=O)NCCC2(O)CCNCC2)C1 C1(NC(C(CC)(C)C)=O)COC2CN(C(C3CCN(C(N)=O)CC3)=O)CC12 Cc1ccc2ncc(C(N3CC4(CCN(C(=O)CCC(C)(C)O)CC4)C3)=O)n2c1 CC(C)C(CC(=O)NCCC1CCOC1(C)C)NC(=O)CN1CCOCC1=O C1(C(=O)NC2CCOCC2C(=O)NCc2cc(O)n(C)n2)(OC)CC(C)(C)C1 C1(CC(=O)NCCCN(C(=O)C=C2CCOCC2)C)COC(C)(C)CO1 C(=O)(C1CCCc2nccn21)N(CC(C)NC(C(COC)C)=O)CC C1(N(C(C2C(C)C2C)=O)C2CC2)CC(NC(=O)CCn2cc(Cl)cn2)C(O)C1 C(C(=O)NCCCC1CCCN1C(c1cc(C#N)cn1C)=O)(C(C)(C)C)SC c1(C(C(=O)NC(CN(C(=O)CCC2CCCOC2)CC)C)(C)C)cccc(C)n1 C1(CNC(C(C)C2CC2)=O)CN(C(c2cccc(C(F)F)c2F)=O)C(C)(C)C1 Cc1ccc(C)c(CCCC(=O)N2CCCC2c2cccnc2F)c1 C(=O)(CCCCCC(C)C)NCC(CO)NC(Cc1cc(C)cc(C)c1)=O c1(-c2ncn(C)n2)ccccc1C(=O)NCCC1CN(C(=O)C2=CCC2)CCO1 CCC(CC)CCC(=O)NC1CCC12CN(C(=O)CCS(C)(=O)=O)C2 CCC(Cc1ccc(C)cc1)N=c1[nH]c2c(c(=NC(C)CCCO)[nH]1)CCC2 O=C(C1=CCOC1)NCCCNC(C1CCCN1CC1CCS(=O)(=O)C1)=O C1(CNC(c2c(C)cccc2)=O)CCC(C)N(C(=O)Cc2ccccn2)C1 CN1CCN(C(=O)C(c2cnn(C)c2)O)CC1C(=O)NCc1cc(C(N)=O)co1 C1(NC(C2C(c3ccc(OC)cc3C)C2)=O)CCCC(N=c2[nH]nc(O)s2)C1 c1(C(=O)NC23CC(C2)N(C(=O)COCC2CCOCC2)C3)cn2c(n1)CCCC2 C(CCO)(CC(C)C)NC(CCCn1cc(CCCCSCC)nn1)=O.C(C)(O)O CC(C)(C)CCC(F)C(=O)N1CC2CC1C2C(N1CCC(N2CCCC2)C1)=O CCCC(CCC)C(=O)NCC1CCN(C(=O)CCc2ccc(N)cc2)C1(C)C N1(C(CC2(N(C)C)COC2)=O)CC(NC(C2C3CCC2CC3)=O)CC1COC N1(C(C(CNC(c2c(C)nsc2)=O)C)=O)CCC(C)(CO)C(O)C1 c1(C(=O)NC2CC(NC(C3N(C)C(=O)CC3)=O)C2)ccc(Cl)c(Br)c1F N1(C(CCC2(C)CCN(C(Cc3n(C)cnc3)=O)C2)=O)Cc2cncnc2C1 c1(C(=O)NCCC2(NC(C3CCC(C)NC3=O)=O)CCC2)ccc2nnnn2c1 c1(C(C(=O)NC(C(=O)OC)C)N(C)CCn2ccnn2)cc(-c2ccco2)on1 c1(CC(C(=O)NCC2N(C(CCOC(C)C)=O)CCC2)C)ccccc1F c1(C(C)(C)C)ccc(CC(=O)NC2CCCN(C(C3CCCSC3)=O)C2)cc1 c1(C(=O)NCCOCCNC(CC(c2scc(C)c2)O)=O)nc(C(C)C)oc1C CC(C)C(C(=O)NCCC(C)CCNC(c1cccnc1OCCO)=O)C(C)C CC1OCCN(C(c2cc(O)cs2)=O)C1C(=O)NCc1nn[nH]n1 N1(C(c2cn(C)nc2C)C(=O)NCCCC(=O)OCC)CCOC(C)(C(F)F)C1 N(C1CCCc2ccc(F)cc21)(CCNC(C1(C)CS(=O)(=O)C1)=O)CCC1CC1 c1(C(=O)NC2CC(C)N(C(c3cnn(CC(F)F)c3)=O)C2)cnc(O)c(Cl)c1 CC1C(NC(N2CCC(c3cnco3)C2)=O)CCN1C.c12cc(ccn1)S2 Cc1oc2cc(C(=O)NCCCC(C)NC(=O)CC(C)n3ccnc3)[nH]c2c1C c1(N(C)CC2CC2(F)F)nc(N2CC(=O)NC(=O)C2)c2c(n1)CCCCC2 c1(C(N(C(C)C(=O)NCC(CC)(CC)CO)CC)=O)c[nH]c2ncccc12 N1(C(C(=Cc2cncs2)C)=O)CCN(C(C23CC(C)(C2)C3)=O)CC1C Cc1ccn(CC(C)C(=O)NC2(CNC(=O)CCc3ccc[nH]3)CCOC2)n1 C1(NC(C(c2n(C)cnn2)(C)C)=O)CN(C(=O)C2=CCC2)Cc2ccnn2C1 C(C(CNC(C1(Cc2cnn[nH]2)CCC1)=O)C(F)(F)F)NC(C(CC#C)C)=O C#CCC(CC#C)C(=O)NC1CC1CNC(=O)Cc1cccc(OC(C)C)c1 CC1CN(C)C(C)CC1NC(C1CC2CC2N1C(C1OC2CCC1C2)=O)=O c1(C(=O)NC(CCC)CCCNC(=O)CC(C)(C)O)scc2c1OCCO2 C1(CNC(CCOC)=O)CCC(F)(CNC(C2(CO)CC2)=O)CC1.C(CC(C)(C)C)N C1(C2CC2)(C(=O)OCC)CCN(c2c(F)cccc2C#N)C1 C(=O)(C(C)CC(C)(F)F)N1CC2C(CC(C)NC(=O)C(N3CCCCC3)=O)C2C1 C1(C(C)(C)C)CC(C(=O)N2CCCN(CC(=O)NC3C4CCCC34)CC2)=NO1 c1(CCC(=O)NC2CCCN(C(c3cncc(C(N)=O)c3)=O)C2)cccc(F)c1 C1(NC(C(C)C)=O)CCC2CN(C(=O)CC34COC(C)(C3)C4)CC2C1 C1(c2cn(C)nn2)OCCCC1NC(=O)CNCC(O)COc1ccc(Cl)cc1 C(O)(Cc1n(CCSC2CNCCC2(C)C)nnn1)(C(F)(F)F)c1ccc(C)o1 N1(C(CC2N(CC)C(=O)CC2)=O)CCC12CN(C(c1ccc(F)cc1)=O)C2 C1(NC(CCCC#CC)=O)CN(C(c2csc(COC)n2)=O)Cc2nccn2C1 c1(OC)ccc2cnc(N3CC(NCc4cc(C)cnc4Cl)C(C)C3)nc2c1 C1(C(N2C(C3CCN(C)CC3)CCC2)=O)CN(C(C2(C)CC(C#N)C2)=O)CCN1C c1(C(=O)NC2CCN(C(Cc3cc(CC)no3)=O)C23CC3)cc2ccccn2c1 C=CC1(C(N2CC(OC)C2)=O)CCN(C(=O)C(F)=CC)CC1 CCC(CNC(=O)C(O)C(C)SC)(CC)NC(c1cnn(C)c1SC)=O c1(C(N2CC(c3ccc(C)cc3)(F)C2)=O)cccc2c1CC(=O)N2 CCN(OC)C(=O)CNC(=O)C(CCNC(=O)C(C)C(C)C)OC N1(C(CNC(C(CC)C)=O)=O)CC(C(=O)NCc2cnc(C)cn2)C2(CC2)C1 Cc1c(C(N2CC(CNC(=O)C(C)(C)N(C)C)CCC2C)=O)oc2ccccc12 C1(NC(c2cnccn2)=O)CC12CCC(NC(C1CN3CCC1CC3)=O)CC2 C1(C(=O)NCCCC2(NC(C3CN(CC(C)C)C3)=O)CC2)CCC(=O)N1 C1(CC(N2CC(CNC(CC3CC(=C)C3)=O)C2)=O)COCC(C)O1 CC(C)CC(C(=O)N1CCOCC1CN(C(=O)C(O)Cn1cncn1)C)N(C)C CC(C)(C)CC(O)C(=O)N1CC2(CCC2NC(c2ccn3c2CCCC3)=O)C1 C1(NC(=O)CN2CC=CC2)CCOC2(CCN(C(=O)CC3CC=CCC3)CC2)C1 c1(C(N2CC3(C(C(=O)Nc4c(OCC)ncnc4)C3)C2)=O)cc(Br)ccc1Cl C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCC(CNC(C1N(C)C(=O)CC1)=O)(C)F N1(C(C=CCOC)=O)CC(C2CC2C(=O)NCc2ccoc2)C1 C1(NC(CNC(CCCCC)=O)=O)CC2(CCN(C(C3CCC(C)CC3)=O)C2)C1 CCC(C)(C)C(C)CC(=O)NC1CCC(NC(C2CCCCC2)=O)CC1 C1(NC(C(CC=C)(C)C)=O)CCCC2CN(C(=O)C3=C(C#N)CCC3)CC12 C1(CC(=O)NCC(C)(C)NC(CC(=C)C)=O)CCCCCO1 c1(C(=O)NCCCCNC(c2cncc(OC(C)C)c2)=O)cscc1S(C)(=O)=O n1(CC(=O)NC2C(NC(C(C(C)C)SC)=O)C2)cnc2cc(C)c(C)cc12 C(=O)(CC(O)CC(C)(C)C)NC1C(OC)CN(C(c2cc(=O)n(C)o2)=O)C1 C(CCC)(CCCNC(c1cc(F)cc(Cl)c1)=O)NC(C1CN(C(C)=O)C1)=O N1(C(C2C=CC(NC(CCC3CC(OC)C3)=O)C2)=O)CCC(N=[N+]=[N-])C1 c1(N(CC(=O)NC2C(NC(C(c3cncnc3)C)=O)C2)C)ccc(Br)s1 C1(CC)CN(CCCOc2cccc(C)c2C)CC(C(F)(F)F)O1 c1(C(=O)NCC2(CN(C(C(C)OC)=O)C)CC2)cn(C)nc1-c1ccncc1 C(=O)(CCC(=O)NC(C1CCN(C(c2cc(C(F)(F)F)cs2)=O)CC1)C)NC N1(C(C(=O)NC2CCC(F)(F)CC2)C2C(C)C2)CCCC2CC1C2(C)C CCCC(c1nccs1)N(C)CC1CC1 N1(C(C(C=CC)O)=O)CC2(CCC(CNC(C3CC3(F)F)=O)O2)C1 c1(CC(=O)NC2CCC(NC(C(C(CC)C)O)=O)CC2)ccc2c(c1)CCCO2 c1(NCCC(C)NC(Cc2nc(CC)sc2)=O)ncnc(O)c1Br C=CCCC(F)(F)C(=O)NC1CC(NC(=O)CC2CC(C)=NO2)CC1O C(c1ccc(F)cc1)=CCC(N1CC(CC(C)NC(C2CC3(CC3)C2)=O)C1)=O Cc1c(C(=O)NC(CC(=O)O)C2CC2)cc(C2CCCC2)n1C C12(C(N(C3CCN(C(c4cc(Cl)cn4CC)=O)C3)CCC)=O)COCC1C2(F)F Cc1cc(Br)c(CNCC2(C)CC(C)C2)s1 N1(C(C(C(C)(C)C)n2ccnn2)=O)CCC2C(CCCN2C(=O)C2=COCC2)C1 C1(NC(C(C(C)C)n2cnnc2)=O)CC2CC(NC(C3(CC4CC4)CC3)=O)C2C1 n1(CC(N2C(C)CCC(CNC(=O)C(F)F)C2)=O)ncc2cc(Br)cnc12 N1(CC(=O)NCC)CCN(C(=O)C(c2ccccc2)OC(C)=O)CC1C.C(C)(C)(C)O Cn1cnc2nc(Cl)nc(N3CC4CC(NC(=O)CCC5CC5(Cl)Cl)CC3C4)c12 c1(OCCCC(=O)N(CCCNC(=O)C(C)c2cncs2)CC)ccc(F)cc1 C1(C(=O)NC(CNC(c2c(C)ccc(Br)c2)=O)C2CC2)CCc2nc[nH]c2C1 C1(CNC(Cc2nc(=N)[nH][nH]2)=O)CN(C(=O)C(F)(F)C2(O)CCC2)CC12CC2 N1(C(CC(=O)NCC)=O)CCN(C(=O)C(C(C)(C)C)C2CCCC2)CC1C(C)C C(=O)(CCCS(N)(=O)=O)N1C(CNC(c2c(C)n(C3CC3)nc2)=O)CC2(CC2)C1 Cc1cc(C)c(C(=O)NCC(C)N(C)C(C2COC(=O)N2C)=O)c(S)n1 N1(C(c2c(OCC)scc2)=O)CCC(C)(CCNC(c2[nH]ccc2COC)=O)C1 c1(OC)c(Cl)cc(-c2c(F)ccc(OC)c2F)cc1C#N C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC1CCC(CNC(C2C(C=C)CC2)=O)C1 C1(C)(CNC(C2(C)CCN(C)C2=O)=O)COCCN(C(C2(CCO)CC2)=O)C1 Cc1cccc2c1CCC2N(C)C(=O)C(C1CCS(=O)(=O)C1)F c1(C(=O)NC(C(C)C)CCN(C(=O)C(F)(F)C2CC2)C)ccc(Cl)c(F)c1N C1(C(=O)NC2CC(NC(C3CC(CCF)C3)=O)C2)CCC(n2ccnn2)CC1 N1(C(CCSCC)=O)CCN2CCN(C(C3CCNC(=O)C3)=O)CC2C1 c1(N2CC3N(C)C(CCC3)CC2)nc(=NC2CCSC2)[nH]c2c1SCC2 C1(C2(O)CN(C(c3n[nH]c(C)c3C)=O)C2)(CNC(c2n(OC)cnc2C)=O)CC1 C1(N(C(C)=O)CC)CCCN(C(=O)CCOCCOC)C1.CCSCC N1(C(c2c(C)ocn2)=O)CC(C)CN(C(=O)CCOCC(F)(F)F)CC1C C1(C(=O)NC2CCCN(C(c3cnc(OC)s3)=O)C2)CCc2cnn(C)c2C1 O=C(CC(O)Cc1ccccc1)NCC1(F)CC(CNC(=O)C(=O)NC2CC2)C1 c1(C(=O)NC(C=CC(=O)NCc2c(C)cc(C)s2)C)c[nH]c2ncccc12 C(=O)(CC(C)C(F)F)N(C(CC(N1CCCC(COC)C1)=O)(C)C)C Cc1cc(CNC(C2CC(NC(C3CC(F)(CF)C3)=O)C2(C)C)=O)cnc1F c1(OC(C(=O)NCC(CNC(CC2(C=C)CC2)=O)(C)O)CC)cccc(Cl)c1 c1(C(N)=O)cc2c(=NC(CCO)c3ccc(CO)cc3)cc[nH]c2cc1Cl Cc1oc(C#N)cc1C(N1CCC(NC(=O)Cc2cscn2)C12CC2)=O c1(C(CNC(C=COCC)=O)NC(=O)CNc2c[nH]nc2C)cccc(C)c1 c1(-c2n(-c3ccn(CC)n3)nc(C3CC=CCC3)n2)cc(C)c(C)cc1Cl c1(OCCNC(C2(O)CC2)=O)ccc(C(F)(F)F)cc1-c1nn[nH]n1 C12C3CCN(CC13)C2=O.c1(C(=O)NCC(CC)OCC)cc(C)c(C)[nH]1 C1(OC)CCCC(C(N2CCCC(CCNC(c3ccc(=N)[nH]c3)=O)C2)=O)C1 C1(CNC(CCOC)=O)CN(C(c2conc2-c2ccccc2)=O)CC12CCC2 c1(COC(CC(C(C)C)c2ccon2)=O)ccc2nc[nH]c2c1F C(=O)(C1CC(=O)Nc2ncccc21)NCC(CNC(c1[nH]cc(C)c1)=O)(C)C N1(c2nccc(OCC)n2)CC(NC(c2c(OC)ccnc2Cl)=O)C2CCCCC12 c1(CC=C)cc(OC)c(O)c(CN2CCCC(C)(C(=O)NCCCO)C2)c1 N1(C(=O)CC2(CCF)CCC2)CCC(F)(C(=O)Nc2ccc(CCO)cc2)C1 C#CC1CC2(CC(C(N3CCCC(N(C)C(c4cc(OC)cs4)=O)C3)=O)C2)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CN(C(Cc2scc(C)c2)=O)CC(O)C1 c1(CN(CC(C)(C)C)C(c2c(CC)cno2)=O)ccc(N(C)C)cc1 C(CC1=CCN(C(c2cccs2)=O)CC1)NC(=O)CC1CN2CCN1CC2 C1(CF)CC12CCN(Cc1ccccc1)CC2.C12CCN1C2 c1(OC)nscc1CNC(c1ccoc1CNC(=O)C(c1cnn(C)c1)C)=O C(C)(C)(CCCNC(=O)C(c1ccc(Cl)s1)=O)NC(C1CC(C(C)C)C1)=O c1(C(N(C2CCOC2)CC#C)=O)cc(Cl)sc1Cl Cc1cc(C(N2CC3CCC(C2)C3NC(=O)CCN2CCCC2)=O)ccc1C#N S(=O)(=O)(CC(=O)NCCC1CCCCN1C(C1CC(C)(O)C1)=O)N(C)C N1(C(c2cn(C)c(=O)cc2)=O)CC(NC(C2CC2CC(C)(C)C)=O)CCC(O)C1 N1(CC2N(C(N=c3ccn(C)[nH]3)=O)CCC2)CC2OCc3cnnn3C2C1 C1(NC(c2scnc2Cl)=O)CCC(CCC(=O)NCc2ncoc2SC(C)C)C1 CC1(C(=O)NCCCCC2CN(C(=O)C(F)(F)c3cscn3)C2)CC1(Cl)Cl C(C(C)C(=O)NCC1CC(NC(C2(N3CCCC3)CC2)=O)C1)SC C(CC(C(=O)N(CC(C(C)C)OC)C)NC(=O)CC1CCSCC1)=CC N1(C(=O)Cc2nccs2)CCN(C2CCN(C(=O)Cc3ccon3)C2)CC1 c1(C(N(C)C)=O)ccc(C(=O)NC(c2ccccc2)CO)nc1 C(=O)(CCCF)NC(C1(C(=O)NC(c2ccsc2)C)CC1)C c1(CC2C(NC(C3CC(c4nn[nH]n4)CC3O)=O)CCOC2)cccc(F)c1Br N1(C(Cn2c(C)nnn2)=O)CCC(C(=O)N(C)CC2(F)CCCC2)C(O)C1 c1(N2CCCC(CNC(c3ccnc(F)c3F)=O)C2)ncccc1[N+](=O)[O-] c1(C(=O)NC2C(OC)CN(C(c3ncn(CC)n3)=O)C2)nnn2c1CSCC2 Cc1ccc(F)cc1CNC(N1CCC(C)C(C(F)Cc2ccccc2O)C1)=O c1(OC)cc(C(N2CCOCC(NC(=O)C(F)CC3CC3)C2)=O)c(Cl)cn1 N1(C(C(=O)NC2CCC(CC)C2)=O)CCc2nc(C)sc2C1 N1(C(CC(=O)OC)=O)CC(NC(c2cnc3cc[nH]c3c2)=O)CC2(CCC2)C1 C1(=O)C(CC)C(=O)NC2C3CC1C(C3)C2(C(=O)NC1COCC1O)OCC C(=O)(C1=CCCOCC1)NC1(C(N2CC(C)(C)CCC2CO)=O)CCN(C)C1 c1(N2C(CN(C(=O)CC3CCCCC3)C)CCC2)nc2cc(F)ccc2o1 c1(CCC(N2C(CNC(C3(C)C(C)C3)=O)C(O)C(O)C2)=O)c[nH]c2ccccc12 c1(C(=O)NCC2(OC)CCN(C(=O)Cc3c[nH]nc3C)C2)nc[nH]c2nccc1-2 c1(OC)cc(Cl)cc(CNC(=O)C(C)(C)OC)c1O.N12CCC(F)(CC1)C2 C1(NC(C2CCCC(F)C2)=O)CCC2CN(C(=O)CCCCC3CC3)CC2C1 C(=O)(C1=CCCN(C(c2cccn(C)c2=O)=O)C1)NC(C#C)C C1(NC(c2c(C)coc2C(C)(C)C)=O)CCN(CC2CC(C)(C)CO2)C(C)C1 CC1(C)CCC(C(=O)NCCCN(C(=O)CCCC2CC2)C2CC2)c2ccccc21 N1(C(C2SCCS2)=O)CCOC2(CCN(C(C34CC5CC3(CO)CC5C4)=O)C2)C1 N1(C(c2cc(CC)[nH]n2)=O)CCC2CC2(NC(c2ccnnc2C)=O)CC1 N1(C(C2CC(=C)C2)=O)CCC(C)C1CNC(c1cnc(Cl)s1)=O C1(C(N(CC)CC2CCCCN2C(=O)CCN2CCCC2)=O)CC2C(C1)C2(C)C C(=O)(C1CCc2nccn21)N1CCC(CNC(c2c(CC)ncs2)=O)C1 Cc1c(C(N2CCC3CC23C(=O)NCc2cccnc2F)=O)[nH]ccc1=O C1(C(=O)NCC(C(C)O)O)CC2(CCN(C(=O)C(F)C(C)(C)O)C2)C1 c1(C(N2C(C)C(NC(=O)C(Cl)=CCl)CCC2)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(c2c(C)cc(CO)o2)=O)CC(NC(c2cc(=O)cc[nH]2)=O)C2(CCCC2)C1 C12(CNC(CCCC#C)=O)CC(CC)(CN1C(=O)CN(C)C(c1ccoc1)=O)C2 c1(C(N2CCC(C)(CNC(CCCCCC=C)=O)C2)=O)ccc(S(N)(=O)=O)cc1 C#CC1CCCCN1C(C1CCCN(C(=O)OC)C1)C(=O)NCSc1ccccc1 C1(NC(C2(CC=C)CCCC2)=O)CN(C(=O)C(C)OC)CCC1C C#CCC(C)(C(=O)N(C)CCO)NC(c1cccc(OC)n1)=O C1(CNC(CCC=CCC=C)=O)CCCC2(CN(C(=O)CC3CCC(=O)N3)C2)O1 Cc1ccc(CN(CCNC(c2ocnc2C2CC2)=O)C2CC2)cc1 CC1CCc2onc(CNC(C3CC34CCCCCC4)C)c2C1 c1(C(=O)NC(CNC(c2c(SC)cc(C)cc2)=O)C)cnn2c1CCCC2C C1(CCNC(CCC2CC(OC)C2)=O)CCC(NC(=O)Cc2cncs2)C1 c1(OCCC#C)ccc(C(=O)NCC2(F)CC(NC(C3CCO3)=O)C2)cc1 c1(C(=O)NC(CCNC(C(C)Oc2ccc(SC)cc2)=O)C)c(C)cccc1C CC(C)C(C#N)C(=O)N(C1C2CN(C(=O)Cc3nc(C4CC4)cs3)CC12)C c1(C(=O)Nc2cc(C)c(NC(=O)CC3CC4CC4C3)cc2)nn(C)c2c1CCC2 Cc1ncccc1C=CC(=O)NCC(C)(C(C)C)NC(=O)CN1CCC(C)C1 c1(CNC(C(=O)N(CC)Cc2ccc(Br)s2)=O)ccc2c(c1F)CCC2 C1(NC(c2c(CC)onc2)=O)CCN(C(=O)COCC2CCOC2)C1(C)C CCS(=O)(=O)CC(=O)N1CCC1CNC(C1CCC(n2ccnn2)CC1)=O Cc1ccc(SCC(=O)NCCCN(C)C(C2CC3(C2)CC3F)=O)cc1C C1(C(=O)NC2CC(C)CN(C(=O)CCCCNC(N)=O)C2)CCC2(CCC2)CC1 C(C(O)CCNC(c1cnoc1-c1ccco1)=O)NC(C1(C(N)=O)CC1)=O c1(C(=O)NC(CC)CN(C(=O)C(c2cccnc2)O)C)ccc2nn[nH]c2c1 C(CC(=O)NCCOC(C)C)(C(C)C)NC(c1cc(C)oc1C)=O C1(NC(=O)C=CC2CC2)CC12CCC(NC(c1ccc(C(F)F)cc1F)=O)CC2 C(C(=O)NCC(C)CCCO)(C(C)C)NC(Cc1c(C)n[nH]c1)=O c1(C(N2CC(=C(CNC(c3c(C)onc3C(C)C)=O)F)C2)=O)nc(O)[nH]c(=O)n1 c1(CC(N2CC(C(C)NC(c3c(C)cccc3C)=O)C2)=O)ccc2nc[nH]c2c1 CC1(C)NC(=O)OC12CCN(c1nc(N3CC4CC3CS4=O)nc3sccc13)C2 CCC(C)(CNC(C1CCN(C(c2c[nH]cc2C2CC2)=O)CC1)=O)C(N)=O N1(C(CCCCC)=O)CCN(C(c2cnn(C3CC3)c2)=O)CC1C(C)C C1(NC(C(C)C2CC2)=O)CCC(O)CN(C(=O)CC2(n3ccnc3)CC2)C1 C1(C(=O)NCC(C)NC(c2cc(C(C)(C)C)ccn2)=O)COC2COCC12 N1(C(c2ccccc2I)=O)CCC(F)(c2cccc(Cl)c2)CC1 c1(S)cccc(OC)c1.C(C(CNC(=O)CC1CC1)CO)NC(C(C)OCC(C)C)=O c1(C(=O)NC2(CNC(=O)C=C(C)C(C)C)CC(OC)C2)ccc(C(C)(F)F)cc1 N1(C(c2ccn(C)c(=O)c2)C(=O)NCCC)CCCN(C)CC1C c1(CC)nc(C(=O)NCC2CCN2C(C2CCCC2OC)=O)cs1 c1(C(=O)NCCC(C)NC(c2ccc(C(=O)OC)s2)=O)cc(Cl)nnc1O N1(C(C(C(C)NC(=O)OC(C)(C)C)C)=O)CCCC2(CCCCO2)C1 C1(CNC(c2c(CC)cno2)=O)C(C)CCN1C(c1cc[nH]c(=N)n1)=O Cc1ccc(C(=O)NCC2(N(C)C(C3CCCN3C(=O)N(C)C)=O)CC2)n1C N1(C(C2(OC)CCCOC2)=O)CC(C2CCN(C(C3C=C(C)CS3)=O)CC2)C1 C1(C(=O)NC2(C3N(C(C4CC(OC)(OC)C4)=O)CCC3)CC2)CC(C(N)=O)=NO1 N(C1CCCn2ccnc21)C(=O)CC1(CO)CC1.C1(=O)C(O)CN1C1CCCC1 C#Cc1ccc(F)c(C(N2CC3CCC2(CNC(=O)CC(C)CCC)C3)=O)c1 N1(C(c2ccc(C)s2)C)C(=O)NC(CC2(C)CC2)C1=O CC12CN(C(=O)Cn3cc(Cl)cn3)C(C(=O)NCCn3cncn3)(C1)C2 c1(OC)ncc(F)c(=NC(=O)c2cncc(-c3cccnc3OC(C)C)n2)[nH]1 N1(C(C)=O)CCC2CN(C(c3cc(-c4ccccn4)[nH]n3)=O)CCC12 c1(COOC)cc(C(N2CC(NC(=O)C(C)COCC)C2)=O)ccc1OC N1(C(Cc2ccc(Cl)c(C)c2Cl)=O)CC2(C1)CN(C)C(=O)C2(F)F C1(OCC)CC2(C1)CC2NC(=O)CC1(CNC(=O)CC2CCSCC2)CC1 C1(NC(C(C)NC(=O)OCC)=O)CCCOCC1.c12cc(ccn1)C(=O)NC2 C1(C(C)C)CN(C(=O)C(O)C(C)C)CCN1C(c1cc(C(N)=O)cn1C)=O Cc1cnncc1C(=O)NC1(CN(C)C(c2ccc(N(C)C)nc2)=O)CC1 O=S(=O)(c1cccc(=NC2CCSC2)[nH]1)NCC1(N2CCCC2)CCC1 Cc1cc(=NCc2ccnc(C#N)c2)[nH]c(NCCN2CCC(N(C)C)C2)n1 CC(O)(C(=O)N1CCOCC(F)(CNC(=O)CCC(N)=O)C1)C(F)(F)F C=CC1COCC1NC(C1(CCNC(C2(O)CCC2)=O)CC1)=O Cc1cccc2c1CCC2NC(=O)NC(c1ccccn1)CCc1cccnc1 C1(NC(CCCOCC=C)=O)CCN(C(c2sc(F)cc2C)=O)C(C2CC2)C1 c1(CN(C(COCCC)=O)C)cc(C)ccn1.C1CCC(=O)NC2CC(C2)O1 c1(CN=c2scc(C(N3CCCC4(CCC4)C3)=O)[nH]2)ccc2c(=O)cc[nH]c2c1 Cc1cc(C(=O)NCC(C)(C)OCCNC(c2cncnc2C(C)C)=O)c(C)s1 CCC(CNC(=O)C=Cc1cnc(C)s1)(CC)NC(c1ccn(C2CC2)c1C)=O c1(C(=O)NCC(CC)NC(c2cncc(OC)c2)=O)cc(Cl)c2ccncc2n1 N1(C(CCN(C(CC(C(CC)C)O)=O)CCCO)=O)CCC2(CCN(C)C2)C1 c1(C(=O)NC(CNC(c2c(CC)ccs2)=O)CO)cc(C)ncn1 N1(C(c2c(CC)onc2)=O)CC2(CCN(C(=O)CCCOC(C)=O)CC2)C1 c1(C(=O)NCC2CCC(F)(CNC(C(C)(C)F)=O)C2)ccc2sccc2c1 c1(C(=O)NCCC2(CNC(C(C)Cc3cnc[nH]3)=O)CC2)csc2cccnc12 c1(C(N2CC(NC(c3cncc(C)c3)=O)C(F)C2)=O)ccc([N+](=O)[O-])cc1Br c1(C(=O)NC2(C)CC(NC(Cn3c(C)nnn3)=O)C2)[nH]cc2c1CCS2(=O)=O C1(CC(=O)NCCC2CCN(C(C34CCC(CC3)C4)=O)C2)CCCS(=O)(=O)C1 N1(C(c2cccc(CSC)c2)=O)CCN(C(=O)C(O)CC(F)F)CCC1C N1(C(C2(CC=C)CC2)=O)CCC(N(C(=O)CCCCN2CCOC2=O)C)CC1 C1(NC(C(=O)NCC)=O)C(C)(C)C(CNC(=O)C=CCN2CCOCC2)C1(C)C C1(C(=O)NC(c2cnn(C)c2)C(=O)NC(C)C)CCN(C)C1=O C(C)(CC(=O)NCC1CCN(C(c2cc(C3CCC3)[nH]n2)=O)C1)SC Cc1ccn2cc(C(=O)NC(C)(C)CCNC(=O)C(C)(F)C(F)(F)F)nc2c1 C1(CNC(CCCn2c(C)nc(C)n2)=O)C2CCC1CN(C(C1C=CCC1)=O)C2 CCCCCCC(=O)NC(C)(C)CNC(c1cc(Cl)cnc1O)=O Cc1cc(O)c(C(=O)NCC(O)CNC(C2CC(=C3CC3)C2)=O)nn1 C(CC(C)C(=O)NCC1C2CN(C(C3CC(=O)N3)=O)CC12)=CC C#CC1(C(=O)NCC(C)C(C)(C)C)CCN(C(=O)C(=O)C2CCCC2)C1 N1(C(=O)OC(c2nccn2C)C)CC2(C1)CN(C(c1ccccc1)C1CC1)C2.OC C(=O)(C(C)CCCC(C)=O)NC(CC(=O)Nc1ccc(OC)cc1)C1CC1 C1(C(=O)NCCCN(C)C(c2cncs2)=O)SCCS1 Cc1o[nH]c(=NC(=O)c2cc(Br)c(C)s2)c1Br C1(NC(C(CCC)CC)=O)CCCCCN(C(=O)CSc2cn[nH]c2)C1 c1(CN2CCC(NC(c3cc(Br)cc(Br)c3)=O)C(O)C2)c(Br)ccc2c1OCO2 CC1CN(C(=O)CC2CCCCO2)CC1NC(=O)CC1C=CCC1 CCS(=O)(=O)CC(=O)N1CCCCCC1CNC(c1cc(O)nc(O)n1)=O c1(C(=O)NCC2(O)CN(C(C(C3CC3)OCC)=O)C2)c(C)n[nH]c1C c1(N2CCC(CSC)CC2)nc(=NC2CCCn3ccnc32)[nH]c2ccsc12 N1(CCNC(C2CCCCS2)=O)CCCN(C(=O)C=C2CCOCC2)CC1 c1(OC)ccc(OC)c(C(=O)NCC2CCC(NC(=O)C(O)c3ccco3)C2)c1 N12CC3(CCOCC3)C1NC(=O)C2C1CCCCC1.Cc1ccc(SC2CCC2)cc1 C=CC(CCC)CC(=O)NC1CCC(CCC(=O)Nc2ccccc2C)C1 C=CCCC(F)(F)C(=O)NCC(C1CCN(C(=O)C(F)CN(CC)CC)CC1)O C(C(C)(C(C)C)NC(c1cccc(NC(=O)OC)c1)=O)NC(C1C(=C)CC1)=O c1(OC)cc(C(=O)Nc2ccc(Br)nc2F)c(NC(c2ccc(Cl)nc2)=O)cn1 C1(C(=O)NC2CC3(CN(C(C=CCC)=O)C3)C2)CC2CCCCC2O1 c1(N2CCC(C3N(C(c4cncs4)=O)CCCC3)C2)nccn2nnnc12 N1(C(C(CCC)=CCC)=O)CC23CCCC2(C1)CN(C(C1CCOC1CC)=O)C3 C(=O)(C1=NOC2COCC12)NC(CCC)CNC(c1cc2cccnc2cn1)=O c1(OC)cc(N)ccc1C(N1CCCC(NC(c2cc3occc3[nH]2)=O)CC1)=O c1(C(=O)NC(CNC(Cc2cc(C)on2)=O)C)noc(C)c1I Cc1c(C(N2CCN(C(C)CO)CC2)=O)cc(F)cc1Cl c1(OC)cc(C=CC(=O)N(C2CCC(NC(=O)C(C)SC(C)C)CC2)C)sn1 CN1CC=C(C(=O)NC2CCC(CCNC(=O)COCc3nc[nH]n3)C2)C1 C1(C2CN(C(=O)CN(C3CCC3)C)C2)(NC(COc2cccc(OC)c2)=O)CC1 N1(C(C(C(CC)O)C)=O)CC(NC(=O)Cn2cnc(C(F)(F)F)c2)C2(CCC2)C1 c1(CC#N)ccccc1C(=O)NCCCC1(C(C2CCCO2)=O)CC1 C(=O)(CC1=CCCC1)NCC1C2N(CCC1)C2=O.c1(CC)cnc(C(C)(C)C)[nH]1 c1(C(N2CCN(C(C3(C)CC(C)C3)=O)CC2C)=O)cn(C)c2c(Cl)cccc12 N12CCN(CC1)C(=O)CC(C)C2.c1(C(N2C(C(C)C)CC2)=O)coc(C2CC2)n1 C12(CC(=O)NCC3C4CN(C(CCc5ccc(C)s5)=O)C3C4)CCC(C)(C1)OC2 C1(C(=O)NCC(Cc2ccccc2C(F)(F)F)CO)(CF)CCOCC1 c1(C(N2CCC(NC(C3CCC(OC)CC3)=O)C(O)C2)=O)cc2oc(C)cc2[nH]1 C1(CN(C(C)C)CC2(NC(=O)NC3(C(F)(F)F)CCCCO3)CC2)CC(=O)N(C)C1 C(=O)(C(C(CC)CC)OC)NCC1(C(=O)NCc2cnc(CC)[nH]2)CC2(CC2)C1 C1(C(N(C)CC2CCCCN2C(=O)Cc2cc(Cl)cs2)=O)CCc2nnnn2C1 CCC(CC)CCC(=O)NC1CC(C)N(C(c2ccc(S(C)(=O)=O)[nH]2)=O)C1 C1(OCC(=O)OC)CCN(C(c2csc(C)c2)=O)C1 Cc1c(C2OCCC2C(=O)NC(C)CCNC(c2cc(CO)[nH]n2)=O)cnn1C N1(C(C(c2cncnc2)C)=O)CCC2CCN(C(=O)C=Cc3cccnc3)C2C1 c1(C(CC(=O)O)NCC2CC3(C2)CC3F)cc(Cl)cc(Br)c1 N1(C(C2C(C)OCCN2C(=O)CC2CCCSC2)=O)CCC(O)C(C)(C)C1 N1(C(CC2CC(NC(c3ccccn3)=O)C2)=O)CCn2nc(CO)cc2C1 c1(CC)ccc(C(=O)NCCC(O)CNC(=O)C2=CCCCO2)cc1CC N1(C(=O)C(C2(O)CCCCC2)(F)F)CCOC(c2cn(Cc3cnns3)nn2)C1 CC1CC(CNC(=O)CCc2cn[nH]c2)CN1C(=O)C=C1CC1 C12CCC3CN(CC13)C2=O.C1(SC)CCCCC1NC(=O)CN N1(c2n(CCCC3N(C)CCC3)nnn2)CC2(CCCCC2)CC1CO C1(CCNC(=O)C(O)CN2CCCC2)CCCN(C(=O)CC2(C3CC3)CC2)CC1 N1(C(C(CC)(CC)c2ccccc2)=O)C2CCC1CN(C(C1(C)CC(F)(F)C1)=O)C2 C1(C(=O)NC(CC(C)NC(C2CC(C)=C(C)CC2)=O)C)CCC2(CC1)CC2(F)F C1(C)(C(=O)NCCC2(C)CCC2)CCCN(C(c2ccccc2C(F)(F)F)=O)C1 C1(CC(N2CC(NC(c3n(SCC)ccc3)=O)C(C)C2)=O)(CC)CCOCC1 N1(C(C(CCC)NC(N)=O)=O)CCC2(CCC2NC(c2coc(Cl)c2)=O)CC1 C#CCCC(O)C(=O)NC1COCC1CNC(c1c[nH]c(=O)cn1)=O c1(OCC)ccccc1-n1cc(C2(C)CN(C(=O)Cc3ccc(Cl)cn3)C2)nn1 N1(C(C(=Cc2cccs2)C)=O)CCC(C(C)NC(C2COC(=O)O2)=O)CC1 C1(NC(C2(C(C)C)CC2)=O)COC2C(NC(c3ccc(N)cc3O)=O)COC12 S(=O)(=O)(c1cccc(Cl)c1C)N1C2CCN(Cc3scc(C)c3)C2CCC1 N1(C(C=C2C(C)(C)CCCC2)=O)CCC2CC2(NC(=O)CCC(=O)N(C)C)CC1 Cc1cc(=NC2CC(CNC(C)C)C2)cc(C)[nH]1 c1(N2CCC(NC(C3CCC3)=O)C2)ncnc2n[nH]cc12 C(=O)(CCN(OC)C(=O)C(CCNC(=O)C(CCOC)N(C)C)OC)NCC N1(C(C2(CCOC)CC2)=O)CCC(C)C(NC(=O)C=Cc2cccnc2C)C1 c1(CNC(N2CC(c3cc(C)c(O)cc3)OCC2)=O)cn2ccccc2n1 N1(C(c2nccc(C)c2)=O)CC(NC(c2cc(CO)[nH]n2)=O)CC12CCCCC2 c1(C(=O)NC2(CNC(c3c(CC)occ3)=O)CCC2)cc2ccc(Br)cc2[nH]1 c1(N(CC(C)OC)C)cc(C)c(S(=O)(=O)NC2CCc3ncccc3C2)cn1 S(=O)(=O)(c1ccc(N2CC3CCC(CC3)C2)c(F)c1)NC1CC(C)CC(C)C1 C1(NC(=O)NC(c2ccc(OC)cc2)C(C)N)CC2(C1)CC(CF)C2 C1(CNC(CN2CC(C)(C)C2)=O)CCCCCN1C(C1CCOC(=O)N1)=O C1(C2CN(C(C=CC(=O)NC3CC3)=O)C2)(NC(C2CC23CCC3)=O)CC1 c1(C(=O)NC(C2CN(C(=O)CSc3cnn(C)c3)C2)C)ccoc1Cl c1(COC)ccc(C(=O)NCCC2(CNC(C3CCC(C(N)=O)O3)=O)CC2)s1 C1(NC(=O)C(F)C2CCC2)CC(F)CN(C(c2cnc(C(F)F)nc2)=O)C1 C(C(CC=C)C(=O)Nn1cnnc1)NC(C1(C#C)CCCC1)=O c1(C(=O)NCCCN2CCNC2=O)nc(-c2cccnc2F)c2ccccn12 C1(NC(C2(COC)CCC2)=O)CN(C(c2ncc(C)cn2)=O)CC1O C12(C(=O)NCC(C)NC(=O)CNC=O)CCCN1S(=O)(=O)CC2 C(N=c1ccnc(NCC2(c3ccccc3)CCCO2)[nH]1)c1c(Br)cn(CC)n1 N1(C(COC)=O)CCC2(C1)CN(C(c1cc3c(s1)CCSC3)=O)C2 c1(C(N2CC(NC(C(C)c3cccs3)=O)C(F)C2)=O)ccc2c(c1)CCN2 Cc1cccc(C(=O)NCC=CCC(=O)NC2(CN(C)C)CC2)c1N C1(CNC(C(C)SCC)=O)CC2CCC1N2C(c1cc(F)cc(F)c1)=O c1(C(N2CCC(N(C(=O)CSCC(N)=O)CCC)C2)=O)c(C)ccc(F)c1N C(CC(=O)NCC1CCNC1=O)(C(F)(F)F)NC(CCOCC#C)=O C(Cn1cncn1)(C(=O)NC1COCC1CO)NC(c1sccc1F)=O C12(C(=O)NCCCN(C(CCCN(C(C)=O)C)=O)C)CCCC(=O)N1CCC2 C1(Nc2nccc(N(CC(=O)NCCOC)C)n2)CCNC(=O)CC1 C(c1ccco1)=CC(=O)NCC(CC)NC(=O)CNC(c1ccc(C(N)=O)s1)=O Cn1cccc1C=CC(N1CCC(O)(CNC(=O)CC2CCS(=O)(=O)C2)C1)=O N1(C(C(F)=CCC)=O)CCC2(CC2)CC1C(=O)Nc1ccc(F)cc1O c1(C(=O)OC(CSC)C)ccnc(OCC(F)(F)F)c1 c1(C(=O)NC2CCC(CNC(c3c(C)oc(CO)c3)=O)C2)cc2scc(Cl)c2[nH]1 C1(C(N(CC)CC2CCCOC2)=O)CN(C(=O)CSCC(F)F)CC1(F)F CC(C(=O)NCC1(CC2CC2)CCCC1)(C1CCC1)NC(=O)CN1CC=CC1 Cc1ccccc1C=CC(=O)NC1CCN(C2CC2)C1 c1(OCC(N)=O)cccc(NC2(c3nnnn3C3CCOCC3)CCCOC2)c1 CC1CC(OC(=O)CN(C)C(C2(F)CCC2)=O)CCC1(C)C c1(COC)ccnc(CNC(=O)C(C)(C2CC2)N(C)C(c2ccc(C#N)[nH]2)=O)c1 c1(CN(C(=O)C=CC=C(Cl)Cl)C)cnn2c1CN(C(C1CC3C=CC1C3)=O)CC2 C1(CC(=O)NC2CC(C)N(C(c3ccncc3F)=O)CC2)CCCC2(CCC2)O1 C(=O)(CC(CC)CC)NCCC1N(C(c2cc(CC)on2)=O)CC(OC)C1 c1(OC)ccc(C)c(-c2nc(Cn3cc(Br)cn3)nn2C2CCCSC2)n1 N1(C(c2ccnc(C)n2)=O)CC2CCC1C(CNC(=O)C(C)CC(C)C)C2 N1(C(c2ccc(OC)cc2OC)=O)CCC2(C1)CN(C(C1CC(C)OC1C)=O)C2 C(=O)(C1=CC2(CCN(C(c3ccsc3Cl)=O)C2)C1)NC1C(O)CCN(C)C1 c1(NC2CN(C)C(=O)C2)cc(=NC2CCC2C2CCC2)[nH]c(C(F)(F)F)n1 c1(C(N2CCC(F)(C(N3CCC(CO)CC3)=O)C2)=O)ccc(CC(F)(F)F)cn1 c1(C(N(C(C)CNC(c2cc(-c3ccccn3)[nH]n2)=O)C)=O)cccc(CO)n1 CCCC(C(=O)N1CCCCCC(NC(c2cc(Cl)cn2C)=O)C1)S(N)(=O)=O N1(C(C(C)OCCOCC)=O)CC(C(=O)NCc2cccc(F)c2C)CC1(C)C N1(C(C(C)CC(N)=O)=O)CCCCCCC1C(=O)NCCN=S(C)(C)=O C(C)(CC(C)N=c1cc(CCOC)nc(SC)[nH]1)NC(CC(CC)(F)F)=O c1(C(=O)NCCCCNC(C2C(C)C2C)=O)cc2ccnn2cn1 C1(CN(CC(C)C)Cc2ccc(OC)cc2)CS(=O)(=O)CCO1 c1(C(CC)C)nc(N(C2CCN(CC3CC3)CC2)C)cc(C)n1 C1(C(N2CCC3CN(C(C=C(CC)CC)=O)CC32)=O)Cc2c(F)cccc2O1 C12(CNC(C3(NC(CC4N(C)CC=CC4)=O)CCCC3)=O)CCCN(CC1)C2 S(=O)(=O)(CCC(=O)NC12CC(C1)N(C(c1cnc(C(C)O)s1)=O)C2)NC c1(C(=O)NC2CCC(NC(c3cnc(COC)s3)=O)C2)ncc(F)cn1 C1(CC)(CNC(C2CC(F)(F)C2)=O)CN(C(C2CC2C2CCCOC2)=O)C1 C12(CC(=O)CNCCC3(CNC(C#CC(C)(C)C)=O)CC3)CCCCC1C2(F)F c1(C(=O)NC(CCNC(C(n2ncc(C)c2)C)=O)C)c(C)nc(C2CC2)nc1O C1(NC(CN2CCN(C)CC2)=O)CCC(C)(C)CC1CNC(C1(CC2CC2)CC1)=O c1(C(=O)NC2CCCN(C(C34CCN(CC3)CC4)=O)C2)ncnc2c1CCC2 C1(N(C(=O)CN(C)CCC)CCC)CCN(C(=O)C(C)C2CCC2)CC1 CONCCC(=O)N1CCC(c2nnc(C)o2)CC1 N=c1nc(N2CCOC3(COCCCO3)C2)[nH]c(=NC2CCNC3(CCC3)C2)[nH]1 C12CN(CCN1C(=O)CCC(=O)N(C)C)C2=O.C1(C)(CC)CCCC1(F)F Cc1nsc(C)c1C(N1CCCC(C(C)NC(=O)CC2COCCOC2)C1)=O c1(CN2CCC(N(C(c3cc(C)sn3)=O)C)C2)ccc2ccccc2c1 C(CC(C(=O)NCCN1CCCOC1=O)NC(C1CCC1C)=O)OC C#CCC(CC#C)C(=O)NC1(CN=c2[nH]nc(C(N)=O)s2)CCCCC1C C1(CC)CN(C(c2sccc2Br)=O)CCC1NC(=O)Cn1cnc(=N)[nH]1 C(CC(=O)NCc1c(CC)noc1CC)(C(F)F)NC(C(C=C)C)=O c1(C2OCCN(C(N(CC)NC(C3CCCC3CF)=O)=O)C2)ccc(F)c(F)c1 c1(C(=O)NCc2ncc(C)o2)cc2c(C)cc(C)c(C)c2[nH]1 C12(CNC(c3c(OCC)csc3)=O)CN(C(=O)COC)C(CF)(C1)C2 C1(C(N2CC(CC(C)NC(c3sc(C)c(O)n3)=O)C2)=O)CCOC(C)(C)C1 c1(CC=O)nc(C)c(C)n1C.N1(C(C(C=C)O)=O)CCCC(c2cncn2C)C1 C(=O)(CC(C(F)(F)F)N1CCOCC1)N1CC(C)(NC(CCNC(=O)OC)=O)C1 N1(C(CN(CCC)C)=O)CC=CC1(C(=O)NCC=CCOC)COC N1(C(CC2CC(=C)C2)=O)CCN(C(=O)CC2CCOC2=O)C2CCCC12 CCCC(C)(C)CC(=O)NC(C)(CNC(c1cc(OC)ncn1)=O)CC(C)C c1(C(=O)NCC2(CNC(c3c(CC)occ3)=O)CCC2)cnccc1C(F)F C1(NC(C(C)NC(COC)=O)=O)CN(C(c2nnc(C3CC3)o2)=O)CCC1C C1(C(C)C)CCC(C(N2CCC2CNC(=O)CSc2ccccc2)=O)C(=O)N1 C1(CC(=O)N(C(C(=O)N2CC(c3cccnc3)C2)C2CC2)C)CCCOCC1 CC(C)C(O)C(=O)N(C)CC1CN(C(c2cccc(C3CC3)n2)=O)C1 N(C1c2ccccc2CC1NCCOC)C(C(=O)NC(CC)C)=O C(=O)(CC(C)CC(C)(C)C)N1CC(CCC=C)(C(=O)Nc2csnc2C)C1 C1(CNC(c2nc(CCC)sc2)=O)CCN(C(=O)CN(C)CC)CCC1(F)F n1(COC)cc(C(=O)NCc2cc(C(N3CC4CC4C3)=O)n[nH]2)cn1 C(=O)(C1CCCc2ncccc21)N(CCN(C(Cc1nc(C)oc1)=O)C)C(C)C C1(OC)CN(C(=O)C=CC2(C)COC2)C(C)(CNC(=O)CCCCSC)C1 n1(C(C(=O)N(CC(CC)NC(C2(c3cc[nH]n3)CCC2)=O)C)C)cc(C)cn1 c1(NC(C2=CCCN(C(C(CCC)CCC)=O)C2)=O)ncc([N+](=O)[O-])cc1F CC1CNc2c(C(=O)NCCCNC(c3ncccc3OC(C)C)=O)cnn2C1 c1(C(=O)NCC2C(NC(C3CC(=C)C3)=O)CCCC2)cn2cccc(Br)c2n1 C1(NC(C2CCc3cnnn3C2)=O)CN(C(=O)Cn2cccn2)C2(CCCC2)C1 c1(C(N(CCC#N)C)=O)noc2c1CC(NC(=O)CN1C(=O)CSC1=S)CC2 c1(NCC(=O)NC(C(=O)OC)Cc2ccccc2)ccc(S(C)=O)cc1 CC1(C)C2(C(=O)NCCSCCCc3cn(C4CCC4)nn3)CCC1(C)C(=O)O2 N1(C(CCC(CC)CC)=O)CCc2sccc2C1CNC(C1C=CCC1)=O C1(C(=O)NCC=CC(N2CC(NC(=O)NC)C2)=O)CCCCNC1=O Cn1cc(C(=O)NCC2(CNC(=O)Cc3nccn3C)CC2(F)F)c(=N)[nH]1 C1(C(N(CCCNC(c2cnc(OC)s2)=O)CCO)=O)CN2CCN1CC2 c1(C(=O)NCC(C)NC(=O)CSCCC(F)(F)F)c[nH]c(=O)c2ccnn12 Cn1cc(C(C(=O)NCC(=O)OCC2CC2)NC(=O)Cn2cnnn2)nn1 C#CC1(C)CCCN(C(=O)COCCOCCc2cccs2)C1 N1(C(C)=O)CCCC(CC(N2CCCC2(C)CNC(=O)C(F)=C(C)C)=O)C1 N1(C(C2(C#N)CCOC2)=O)CC2OCCN(C(=O)C3CC3)C2C1 C(C1c2ccccc2CCN1C(c1cnn(C)c1F)=O)NC(C1(OC)CC1)=O N1(C(c2cc(CCC)n(C)n2)=O)CC2CC(C1)C2NC(c1ccon1)=O C(CC=O)(C(C)C)CC(N)=O.CCCCCC=CCC(=O)N(C)CC O=C(CC(C(F)(F)F)NC(=O)CN1C(=O)CNC1=O)NCC1CCC=CO1 n1(C(C)C)ncc(C(C(=O)NC2CCCC2)N(CC(=O)N(C)C)C)c1F c1(C(N(C)CC2CCCC(NC(COCC=C)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(NC(C2C(C)(C)C2CNC(c2cnnc(O)c2)=O)=O)CCN2CCC1C2 C(=O)(C(CC)CC=C)NCC1(C(=O)NCCCCC#C)CCCC1 N1(C(c2c(CCC)occ2)=O)CCC(C)(C)C1CNC(=O)CCCOC(C)(C)C c1(C(N2CC=CC2C(=O)NC2(C(=O)OCCO)CC2)=O)cnsc1 CCC(C)C(C(=O)NC(CO)C(=O)NCc1ccc(F)cn1)N(C)C C1(C(=O)O)CC(n2cc(CC3(O)CCSC3)nn2)CN1C(C1(C)CCCS1)=O C1(C(=O)NC2C(NC(c3cc(C)on3)=O)COCC2)CCC2(CCC2)O1 N1(C(C(C)OC)=O)CC(F)(F)CC1CNC(c1ccc(=O)n(C)c1)=O c1(NC(C(Cc2cc[nH]n2)NC(=O)C=Cc2cncs2)=O)cc(F)ccc1F N1(CCC2(OCC)CCC2)CC2CCCC(C1)N2C c1(C(N(CC)CC2CCCCN2C(=O)COC)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(c2c(C)n(C3CCOC3)nc2)=O)CCC(F)(CN(C)C)CC1 CN1CCC(C(N2CCCC(CNC(C3(C(=O)OC(C)(C)C)CC3)=O)C2)=O)C1=O N1(C(CN(C(=O)OC)C)=O)CCC(CCNC(=O)C(F)(F)c2ccnn2C)C1 CCC1(C(=O)N2CCOC(COC)CC2)CCCc2ccccc21 C12(C(N3C(CN(C(c4cnc(C)nc4)=O)C)CCCC3)=O)CCC(F)C1CC2 N1(C2N(C(C3CC(C(=O)NO)C3)=O)CCCC2)Cc2ccccc2C1 N1(C(c2nc(C)oc2)=O)CC2(COC(CNC(c3cc4c(nn3)CCC4)=O)C2)C1 c1(C(=O)OC)ccnc(C(=O)NCC(CO)NC(=O)CC2CCS(=O)(=O)C2)c1 c1(OC)ccc(C(=O)NC2CN(CCCCc3ccccc3)CCC2C)c(Cl)c1 C12(C(=O)NCC(C)(CC)NC(C(Br)=C(C)C)=O)CCC(CO1)C2 C1(NC(C(C)C2CCCO2)=O)CC2CC(C1)N(C(C1CCCC1(C)C)=O)C2 C1(NC(CC2CC(=C)C2)=O)(CNC(c2cnccc2OC)=O)CC2CCC1C2 N1(C(CCC=CC(C)C)=O)C2CCC1CC(F)(CNC(c1ccncn1)=O)C2 CCC(O)C(C)(C)C(=O)NCCNC(c1ccoc1C1CC1)=O c1(C(C)C)ccc(CNC(C23CC2CN(Cc2cnc(Br)o2)C3)=O)cc1 C1(C(N(CCN(C(C)C)C(C2CC(S(C)(=O)=O)C2)=O)C)=O)CC(=O)OC1(C)C n1(CC(N2CC3C(CNC(c4c(SC)n(C)nc4)=O)(C3)C2)=O)ccc(C)cc1=O C1(C(=O)NCC2N(C(C)=O)CCC2)CC(=O)C12CCC2 Cc1cccc(-c2nc(C)c(C(=O)NCC3CC(NC(=O)CO)C(O)C3)[nH]2)c1 N1(C(CC(=O)NCC)=O)CC2CC(NC(c3nc(C)ccc3OC)=O)C2C1 C1(C(N2CCN(C(C(C(=C)C)(C)C)=O)CC2CCO)=O)CCC(=O)CC1(C)C N1(C(CC2(N(C)C)CN(C(C(C)CN(C)C)=O)C2)=O)CCC(O)C(C)C1 N1(C(Cc2cc(C)ns2)=O)CC(O)CC1CNC(c1cccc(C(C)(F)F)c1)=O CC1CCCC(C(=O)NC2(C)CCCN(C(C3CCOC3)=O)C2)CC1 C=C=CC(C)C(=O)NCC1(C2CC2CNC(=O)CCc2csc(Br)c2)CC1 C1(C(c2nc(-c3ccc(N)cc3)nn2-c2cccc(Cl)c2C)C)C(C)CCCC1C C1(C)(NC(COCC)=O)CC(C(=O)NCC2CCOC2=O)C1 C(CCF)(C(=O)NCCc1nc(C)cs1)NC(C(C)SCC)=O CCCCC(O)CC(=O)N1CCC(NC(c2ccc(CC)c(F)c2)=O)C1 c1(OC)ccccc1CCO.C12(CCOCC1)CNC(CS)c1n(nnn1)C2.SC CC1=NOC(C)(c2nc(-c3ccccc3N(C)C)no2)C1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(CCOC)N(C(=O)C(C)N2CCCC2)CC1 CC(CS(C)(=O)=O)C(=O)N1CC(C)(C)OCC1CNC(c1ccnn1C)=O C(=O)(CCCS(C)(=O)=O)NC1(C(=O)OC)CCCN(C(=O)C(C)O)C1 N1(C(COCCCCC)=O)CC(NC(=O)CCNC(=O)CC(C)C)C2CC2C1 CC(C)C(C(=O)N1CCC(O)(CCNC(c2ncncc2Cl)=O)C1)NC(N)=O C(C(C)(Cn1cccn1)NC(=O)CCC=CC(C)C)NC(CCOC(C)=O)=O NC(CCF)C(=O)NC(c1ccccc1)C(=O)OCc1ccccc1 CC(Cc1ccccc1)CC(=O)NCC(C)(C)CC1CN(C(c2ccn(C)n2)=O)C1 C(=O)(CCCCCF)N1C(CCNC(C=Cc2ccc(C)o2)=O)CCC1 CN1CCCCC1CC(=O)NCC1CCC1NC(c1cc(Cl)sc1Cl)=O N(C1c2cc(Br)ccc2CC1(C)C)C(=O)NC1C(C)(OC)C1 c1(CC)ccc(CN(C(C2CCC(n3cc(C(C)(C)O)nn3)C2)=O)C2CC2)nc1 C(C1=Nc2ccccc2S(=O)(=O)N1)NC(=O)C(=O)NCCc1c(Cl)cccc1Cl CC1CC(CCNC(c2c(F)cncc2F)=O)CC(C)O1 c1(OC)ccc(-c2cnc(CNC(=O)CCNC(=O)OC(C)(C)C)nc2)c(F)n1 C1(C(=O)NCC2C(C)CCCN2C(C2CCCN2C=O)=O)CCc2n[nH]cc2C1 c1(C(=O)NCC2OCC(C(=O)NCCOCCC3CC3)C2)ccncc1Cl c1(C(C)(C)NC(=O)CC2CC2(F)Cl)ccc(F)cc1 C1(C(=O)OC)CN(C(C2CC2c2ccc(SC)cc2)=O)CC1N N1(C(C(C)N(C(c2ccnn2CCF)=O)CC)=O)CCCN(C(C)=O)CC1 CS(=O)(=O)CCC(=O)NCC1C2CN(C(=O)Cc3cncc(C#N)c3)CC12 N1(C(C2N(C)CC2)=O)CCC2(NC(c3cccc4cncn34)=O)CCCC12 CC1(C)CC(=O)NCC1C(N1CCC(CF)(NC(=O)C(N)=O)C1)=O Cc1cc(C)c(C(N2CC(C)(NC(=O)C(C)OC3CCOC3)C2)=O)s1 c1(CC(=O)NCCCC(C)NC(CN(CCOC)C)=O)ccncc1Cl Cc1cccn2ncc(C(N3CCC(C)(CNC(c4cnc(Cl)s4)=O)C3)=O)c12 N1(C(CC=CC)=O)CC2CC(NC(c3ccnc(C)n3)=O)CC1C2 CC(C)(C(=O)NCCC1CCC(NC(=O)C(O)C(C)(C)C)C1)S(C)(=O)=O Cn1nc2c(c1C(=O)NCCF)CN(Cc1c(C(=O)O)cccc1F)CC2 c1(OCC=C)cccnc1C(=O)NC1CCC(CNC(=O)Cc2ccc(Cl)s2)C1 c1(C(C)(C)C)cc(C(F)(F)F)nc(=NCC2CC23CC3(F)F)[nH]1 CCCC(C)CC(=O)NC(c1ccccc1)CNC(=O)C#CC1CC1 c1(C(C(=O)NC2C(C(C)NC(c3ccn(C4CCC4)n3)=O)C2)O)cnn(C)c1 N1(C(CS(CC)(=O)=O)=O)CCCC2(CCN2C(c2cccc3[nH]ncc23)=O)C1 N1(C(CC2(N(C)C(c3cnc(O)o3)=O)CC2)=O)CC2CC3CC2C1C3 CC1CC(CNC(C2CC3(CCC3)C2)=O)CN(C(=O)Cn2cncn2)C1 C1(NC(C2C(C)(COC)C2)=O)CC2(CCN(C(c3csc(=NC)[nH]3)=O)CC2)C1 C12(CNC(CCC=C(C)C)=O)CC(NC(=O)NC3CCCOC3)(C1)C(C)O2 N1(C(C2C(OC)(OC)CC2)=O)CC(F)CC1C(N1CC(O)(C(=O)N(C)C)C1)=O C1(CCC(=O)NC2C=CC(C(=O)O)C2)CCc2ccccc2C1=O c1(OCCC)cccnc1C(=O)NC(C1CN(C(=O)C(c2ccc(C)s2)C)C1)C C1(NC(C(CC)OCC)=O)CCN(C(c2cnc(CC)nc2O)=O)CC(C)(C)C1 n1(CC)nc(C(=O)NC(C)CC2CN(C(=O)CCc3ncco3)C2)cc1O N(C(=NCc1ccccc1)N1CCC2=C(CCCC2)C1)Cc1cn(CC#C)nc1 N1(C(Cc2n(C)nnc2)=O)CCC2(CCN(C(c3cc(Br)cn3C)=O)C2)C1 Cc1cc(C(=O)Nc2ccc(Br)c(C)c2C(=O)O)c2n[nH]cc2c1 N1(C(=O)CCc2cn[nH]c2)CCCC(CC(N2CCC2CF)=O)C1 c1(C(=O)NCC2CN(c3ncc(F)cn3)C2)cnc(C2CC2)nc1 N1(C(c2n(CC=C)ccn2)=O)CCC2CCN(C(=O)C(C)C#N)CC2C1 N1(C(CCCC=C)=O)CC(C)CN(C(=O)CNC(c2ccc(Cl)cc2)=O)C(C)C1 c1(NC(C(CC)NC(N)=O)=O)nc2c(s1)C(C(=O)O)OCC2 C(CCCN=c1nc(O)c(Cl)c[nH]1)NC(CCC(C)OC)=O C(=O)(C(C(C)(C)C)OC)N1C(C(=O)N(C2CCC3CC23)C)(CC)CCC1 Cc1cccc(C(c2ccccn2)NC(c2snnc2C2CCC2)=O)c1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC1C1CN(C(C3OCCO3)=O)CC21 c1(OC(C(=O)NC2CCCC(NC(CC)=O)C2)(C)C)ccc(F)c(F)c1 C1(N(C(=O)C=CCOC)CC)CC2CCC(C1)N2C(C1(CC2CCC2)CC1)=O C(C(F)(F)C(F)(F)F)OCCC(N1CC(NC(C(c2ccc(C)cc2)C)=O)C1)=O c1(C(=O)NC2C(NC(c3c(C)cc(SC)o3)=O)CCC2)cnc2cccnc2c1 CN1CCCC1(C)C(=O)NC1CCC1CNC(=O)CCc1cncnc1 C(CC(F)F)(C(=O)NCCC1CCCC1)NC(c1csc(O)n1)=O Cn1c(C(N2CCC(C)(NC(=O)C3=NOC(C)(C)C3)CC2)=O)cc2occc12 N1(C(c2cnc(C)o2)=O)CCC(N(C(=O)CN2CCCNC2=O)C)CC1 C1(NC(C2N(C)C(=O)CC2)=O)CCN(C(c2c[nH]ccc2=O)=O)C12CC2 N1(C(c2cncc(OCC)c2)=O)CCC2CCC(NC(=O)C=CCF)C1C2 C(=O)(C(C)(COC)CC)NC(CCCC)CNC(c1cncc(C(F)(F)F)c1)=O N1(C(=O)Nc2c(C)c(C(F)(F)F)ccc2)CCCCC(C)CC1 c1(C(=O)NCC2CCCC2NC(c2c(F)cccc2F)=O)cc(F)nc(F)c1 c1(C(N2C(CNC(C(=O)N(CC)CC)=O)CC(OC)C2)=O)cc2n(n1)CCCO2 n1(C(C)C)ncc(C(=O)NC2(C(=O)NCC(c3cn(C)cn3)O)CSC2)n1 c1(C(N2C3CC(N(C(=O)CC(=O)NC4CC4)C)(C3)C2)=O)ccc2c(c1)NC(=O)CO2 C(=O)(CCCC(F)(F)F)N(CCC(=O)Nc1c(CC)n(C)nc1)CCCO CCCCC(O)CC(=O)N1CC2(C1)SCCC2NC(=O)CC1(CC)CCCCC1 CC1CC=C(C(=O)NCC2C3CCCC2N(C(=O)C(C)C2CCCC2)C3)CC1 N1(C(C(CC=C)C)=O)CCC(F)(F)C(CNC(=O)CC2CCOC2)C1 c1(NC(C2OCCN(Cc3ccc(C)cn3)C2)=O)cnc(C#N)c(C(F)(F)F)c1 Cc1ccnc(C(N2CCC(F)(C(=O)N(C)CCOC(F)F)CC2)=O)c1F c1(N(c2ncnc3[nH]ccc23)C2CNCC(C)C2)ncnc2ncc(Br)cc12 O(NC(=O)C(C)(C)c1csc(C)c1)CCCc1cccc(C(=O)OC)n1 Cc1cc(F)c(F)cc1NC(=O)C(N1CCC(Cc2cccc([N+](=O)[O-])c2)C1)=O Cc1ccnn1CC(=O)NC(CNC(=O)CCc1cn[nH]c1)C1CC1 c1(C(C)=O)cnccc1NC1CN(C(=O)C(C)Cc2ccccc2F)CC1C C(CC1CCOCC1)CN=c1ccnc(NCc2cccnc2)[nH]1 C1(N(C(C2C(C(=O)OC)COC2)=O)C)CCCCC1N(C)C(c1cocn1)=O CS(=O)(=O)c1cccc(C(CO)NC(c2cc(O)cc(O)n2)=O)c1 c1(C(C(=O)NCCCOC)N(C)Cc2ccn(C(C)(C)C)c2)cc(Br)ccn1 c1(C(N2CC(COC)C23CCC3)=O)cnn2c1OCCC2 C(c1cnccc1C)=CC(=O)NC1CC(CNC(CC2C(C)=NOC2=O)=O)C1 FC12CCN(CC1)c1cc(ncn1)N2.c1(SCc2nccs2)ccccc1 n1(CCC(=O)NCC2CC(CNC(C3(CC(F)F)CC3)=O)CO2)cccnc1=O c1(OC)cc(C(=O)Nc2ncncc2C#N)cnc1OC C1(NC(C(=O)NCc2c(CN(C)C)nn[nH]2)=O)CCCN(C(C)(C)C)C1=O Cc1ccc2c(n1)N(C(N1CCOCC1c1cccc(Cl)c1)=O)CCO2 C12(C(N3CCCC(CNC(c4c(OC)nccc4)=O)C3)=O)CCCC1C2(F)F N1(C(=O)C(O)C2CCC2)CCCC(N(CCO)C(C2(Cl)CC2(F)F)=O)C1 CC1(C)CCCC(C(=O)NCC(CC2CC2)C(=O)N2CC=CC2)C1 c1(C(=O)NCc2ccc(CC(=O)OCC)cc2)cc(C2CC2)cc(F)c1 Cc1noc(C)c1S(=O)(=O)NC1CCCCN(S(=O)(=O)c2nccs2)C1 CC1CN(C(c2nncn2C2CC2)=O)CCC1NC(C1CC(N=[N+]=[N-])C1)=O Cc1nc(CO)ncc1C(=O)N(C)CC1(O)CCN(C(C2(C)COC(=O)C2)=O)C1 C1(F)(C(N(C(C(CC)C)C)C2CC2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)C1 C12(C(=O)NCC3C(C)CCN(C(C4CC(OC)C4)=O)C3)CCCCC1C2(F)F C1(CNC(Cc2nc(C(C)OC)sc2)=O)CC(OC)CN1C(=O)CC1CSC1 N1(C(C(OC)OC)=O)CCC(CO)C(NC(=O)CCC2C(=O)NN=C2C)C1 C1(C(C(=O)N(CCN(C(C)C)C)CCS)C)CCCN(C(=O)OC(C)(C)C)C1 C(=O)(C(C(C)C1CC1)N1CCC(CN(C)C)CC1)NCC C(C(C)(C)C(=O)NCC(C)CN(C)C)NC(c1ccc(C)s1)=O C1(C2CCN(C(=O)CN(C(=O)C(C)C)C)C2)(NC(C(C)OCC)=O)CC1 c1(C(=O)NCC(CNC(C=CC(C)(C)SC)=O)(C)F)ccn2cccc2c1 CCCC(C)(O)CC(=O)N1CCC(CNC(C2CCC2)=O)C1 C(=O)(C(C)(C)CC(=O)N(C1CN(C(=O)C(C)C2CCC2)CC12CC2)C)OC C1(C)(CC(=O)NCc2c(C)nsc2)CCN(C(C2(O)CCCCC2)=O)C1 c1(CC)ccc(C(C)CC(=O)NC(C)CC2CN(C(=O)C=CBr)C2)cc1 c1(C(N2CCC(C(C)(C)NC(=O)CC3NC(=O)NC3=O)C2)=O)ccn2c1CCC2 c1(C(=O)NCC2(NC(c3cnsn3)=O)CC2)cc(Br)ccn1 CCCCCC(C)CC(=O)NC(C)CC(C)NC(C1CCN(C)CC1)=O c1(OCCC(=O)N(CC(C)N(C(=O)CCn2cnnn2)C)C)ccc(F)nc1 C1(OC)(CNC(c2conc2C(C)NC(C2CCC(C)O2)=O)=O)CCOCC1 C1(CC(=O)NC(C)C(C)(C)O)CN(C(c2coc(C(F)F)c2)=O)CC12CC2 CCC(CCCC(=O)OC)NC(=O)COCC(=O)NC(c1cncn1C)CO C(=O)(CCCS(N)(=O)=O)NC(C)(C)CSc1c(C(=O)OC)cc(O)cc1 C(C(C)(O)CC(=O)N1CCC(N2CCN(C(=O)CCCC(C)=O)CC2)C1)OC c1(C(C2(n3cnnn3)CC2)N(C(=O)CC2CCNC2=O)C)ccc(CSC)cc1 N1(C(CN(C(C)=O)C)=O)CC2CC(NC(c3ccc(F)cn3)=O)CC1C2 CCCCCC(O)C(=O)NC(C(=O)N1CC(F)C1)C(C)(C)O C1(S(C)(=O)=O)(C(=O)NCC2CN(C(C3N(C(C)(C)C)CC3)=O)C2)CCCC1 C1(CN(C)CC2CCCN(C)C2c2ccnn2C)CCC2CC1C2(C)C N1(C(=O)NC(C(F)(F)F)C2CCOCC2)CC(C2CC2)C(F)(CO)C1 C=C(Cl)C(C)(C)C(=O)N1CCC(CCNC(=O)Cc2n[nH]c(=N)s2)CC1 C1(N(C)C)CCC1NC(=O)NC(CN(CC)CC)C C(C)(CCC(=O)N1CC(C2CCN(C(=O)C(Cl)=CCl)CC2)C1)OCC c1(OC)cc(C(=O)N(C)CC2CCCN2C(C2CCOC(=O)N2)=O)nn1C CC(C)CCC(C(=O)Nc1csnc1C1CC1)NC(c1cc(=O)n(C)cn1)=O C(=O)(C(CCC(N)=O)N(C)C)N(CC(CC)NC(=O)CCCN=[N+]=[N-])CC C(CCCCCC(=O)N1CCC=C(F)C1)NC(CCCCCOC)=O N1(C(=O)COc2ccccc2F)CCCC(N=c2ccnc(C3CC3)[nH]2)C1 C(CC1CC1)(CC(=O)NC1CCN(C)C1)NC(C(CC)=CC)=O C=C1c2ccccc2C(=O)N1CC(N1CCCCC(NC(c2ccco2)=O)C1)=O c1(C(N2CC(CC(C)CNC(=O)CCc3cn[nH]c3)C2)=O)ccnn1C1CCCC1 C1(CNC(CCCNC(=O)OC)=O)CCCCN(C(=O)C(=O)C(C)(C)C)C1 c1(OCC#C)ccc(C(N2CC3C(CN(C(=O)CCC=C(C)C)C)C3C2)=O)cc1 N1(C(C(C)N=[N+]=[N-])=O)CCN(C)C(CNC(C2CCC(O)CC2)=O)C1 CC1(C)CC(C(=O)NCC2CC3CC3C2)CC(C)(C)S1 N1(c2ncc(C(=O)OC)nc2)CCC(CNC(c2cccc(F)n2)=O)C1(C)C N1(CC#CC)CCN(C(=O)CC(COC)NC(=O)CC2CC3CC3C2)CC1 C1(NC(C2N(C(c3c(CC)cc[nH]3)=O)C(C(C)C)CC2)=O)CC2CC1C(O)C2O Cc1cc(O)c(CN2CCCC(CCO)C2)cc1Cl.c12nc(Cl)ccc1C(=O)N2 C#Cc1cccc(CCCNC(c2ncncc2C#N)=O)c1 C1(C(=O)NCC(CNC(=O)C(C)(C)C2CCC2)OC)(C(C)C)CCNC1=O CC1CN(C(c2cc3ccccn3n2)=O)CC(C)C1NC(=O)CC=CC(C)(C)C C1(NC(c2ccc(CSCC)cc2)=O)CCC2CN(C(C3CC3F)=O)CC2C1 N1(C(CCC(=C)Cl)=O)CC2CCC(CNC(c3c(C)coc3C(C)(C)C)=O)(C2)C1 c1(C(=O)NCC(CC=C)NC(=O)C(O)CSC)nccc2ncncc12 C1(N(C(=O)COC(F)(F)F)CCNC(C(C)OCCC(C)C)=O)CCCCC1 c1(OC)cccc(Cl)c1C(=O)NCC(C1CC1)NC(c1cc2n(n1)CCC2)=O N1(C(c2cccc(-c3cccs3)c2)=O)CC2CN(Cc3c(F)cccc3Cl)C2C1 C12(CNC(=O)CN3CCCC3=O)CCCC1CN(C(C1CCCO1)=O)C2 c1(CC(=O)NCC2CCN(C(=O)CC3(O)CCOC3)C2)ccccc1F C1(NC(c2nc(CC)oc2)=O)CC2CC1CN2C(C1(CC)CCC1)=O N1(C(C2CC3CC3N2Cc2cccc(Br)c2Br)=O)CCCC2(CCOC2)C1 C(CC(=O)N1CCCC(C)(C)C1)(C(F)F)NC(C(C1CC1)OCC)=O C1(CC#C)(C(=O)N(C2CCN(C)C2)C)CCN(C(=O)C(C)C2CCCC2)C1 C(=O)(CCC(=O)N(CC(O)CNC(C1CC=CCC1)=O)C)Nc1nnc(CC)s1 c1(C(=O)OC)cccnc1N1CCC(CF)(NC(=O)Cc2cnns2)C1 C(=O)(CC(O)CC(C)(C)C)NCC(C)N(C(CCN(C)C(C)N(C)C)=O)C1CC1 c1(C(=O)NC2(CC)CCCN(C(=O)C(C(C)C)SC)C2)ccc(F)c(F)c1N CCC(CC(=O)NCCOCCOC)NC(C1CCCC(CF)C1)=O C(=O)(C(O)CC(N)=O)N1C(C(=O)NC(C#CCC)(C)C)C=CC1 CC1(C)C(CC(N2CC=C(CO)CC2)=O)CCN1C(C1CCCOC1)=O c1(C(=O)NC(C(C)NC(C(C)(C)NC(=O)OC)=O)C)cc2nnn(C)c2s1 c1(C(=O)NC2CCC(N(C(C3CN(C)C3)=O)C)C2)cccc(-c2ccccc2)n1 C=C(Cl)CC(C(=O)Nc1cnn(CC(C)C)c1)NC(=O)CCC(N)=O C(=O)(C1=CCC(C)(C)CC1)N1C(C)CC(CNC(c2c(COCC)ncs2)=O)C1 C1(C(N(CCOCC=C)C)=O)COC2(C1)CN(C(=O)C(F)C(CC)CC)C2 CC(N=c1[nH]c(=NCc2cnn3ccccc23)[nH]c2c1CCC2)c1ccoc1 C1(CCC=C)(C(=O)N(C2COCC2O)C)CN(C(c2ccoc2C)=O)C1 c1(SCC)[nH]nc(C(=O)NC2CCC(C)(CC(=O)Nc3cccc(C)c3)C2)c1C Cc1c(C(N2CC(C(N)=O)(CNC(C3CCCOCC3)=O)C2)=O)cccc1O c1(C(=O)NC2CCC(NC(C(COC)NC(C)=O)=O)CC2)ccnc2[nH]cnc12 N1(C(=O)Cc2cccc(Cl)c2F)CCC(F)(CN=c2nc(C(F)(F)F)[nH]s2)CC1 N1(C(CCN(C(=O)CC2CC3CCC2O3)CC=C)=O)CCC2CC1C(=O)O2 c1(C(=O)NC(C(C)NC(Cc2cc(OC)cc(F)c2)=O)C)cccc([N+](=O)[O-])c1 C1(C)(C(=O)OC)CC(C(=O)N(CC(O)CN(C)C(C2CC(C(F)(F)F)C2)=O)C)C1 c1(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)ccc2nsnc2c1 C(=O)(C(CCC(N)=O)N(C)C)N1CC(CCNC(c2c(C)occ2)=O)C1 c1(C(C(=O)CCC)O)cccc(C)c1.C1(C(=O)NCCN)CN(S(C)(=O)=O)C1 C(C1=CCN(C(C2CC(C(=O)OC)(OC)C2)=O)CC1)NC(COC(CC)(C)C)=O N1(C(CC(=O)OCC)=O)CC2CC2(NC(c2ccoc2Cl)=O)C1 C(C(=O)NCC1(O)CCC(C)C1)(C(C)(C)C)NC(CC1CCC(C)CC1)=O CCC(C(=O)N(C)Cc1nc(C(C)(F)F)no1)N(C)C C1(C(N2CCN(C(=O)CCF)C(CCO)C2)=O)OCC2CCCC12 Cc1c(C(=O)NCC2C3CN(C(c4cc(Cl)cnn4)=O)CC23)nn2ccccc12 Cc1conc1C(=O)NCC1CC1CNC(c1csc(Cl)n1)=O N1(C(C(CC=C)(C)C)=O)CCC2(NC(c3cccn3C)=O)CCCC12 c1(-c2cc(OC)cc(F)c2F)nc2c(s1)CCN(C(c1cccc(Cl)c1F)=O)C2 N1(C(C(CC)NC(C)=O)=O)CC2(CCN(C(=O)C=CC=C(Cl)Cl)CC2)CC1 C1(C(=O)NC2(CC=C)CN(C(C3CC(OCC)C3)=O)C2)CCCC(O)C1 C1(NC(C(C)=CC)=O)CN(C(=O)Cc2cccc(NC(=O)OC)c2)C2CC12 CC1CN(C(=O)CC2CCCN(C(c3cnc4n3CCC4)=O)C2)C(C)(C)C1 Cc1oc(C2CC2)nc1C(=O)NCC1CCC(NC(=O)CC2CC3CC3C2)CC1 c1(C(=O)NCC(CC(C)C)NC(C(C(C)C)SC)=O)ncc(Br)cc1O c1(CN2C(CNC(=O)Cn3cccn3)CCC2)nc(Br)ccc1F N1(C(C2CCC(C)CC2)=O)CC2CC3CC2C1C3NC(c1cc(F)n(C)n1)=O c1(=O)c(=O)n1C1CC1.C1(C(=O)NC2C(C)C2)(NC(=O)OC(C)(C)C)CC1 c1(C(N(C2CC2)CC)=O)ccnc(SC2CCC(C(=O)OC(C)(C)C)CC2)c1 C1(NC(c2c(C(N)=O)nccn2)=O)CC2CN(c3ncnc4scnc34)CC2C1 C(=O)(C1CCCn2nccc21)NCC1N(C(c2ncn(CC)c2)=O)CC(C)(C)C1 C=C(Cl)C(C)(C)C(=O)OC.C(=O)(CCCCCc1ccc(F)cc1)N1CCC1 c1(C(=O)NCC(N(C(C(C=C)(F)F)=O)C)C2CC2)cnc(O)c(C(F)(F)F)c1 c1(C(=O)NCCN(C(=O)C(C2CCCCCC2)F)CCC)c(C)cc(C)nc1S c1(CNC(c2scc(CNC(C(C3CC3)SC)=O)c2)=O)nn(C)c(=O)n1C c1(N2CCCC(C)(CC)CC2)nc(=NCc2cc(OC)no2)[nH]c2cc[nH]c12 C=C1CCN(C(=O)C(C)CC2CC2)C(C(=O)NC2CCCC2CCO)C1 c1(C(N2CCC(NC(C(CC)CC(C)C)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1N S(=O)(=O)(CCC(=O)NCC1(CNC(c2cncc(C)n2)=O)CCCC1)NC c1(C(N(C2CCN(C(C3CC3Cl)=O)CC2)CC)=O)[nH]c2ccccc2c1C C1(N(C)C(c2cncnc2)=O)Cc2ccccc2N(C(C2C(C)(C)C2(C)C)=O)C1 C1(C(=O)NCC2CC(NC(c3n(C)ccn3)=O)CC2O)CCOCC1(C)C c1(-n2ccc(C(=O)NC(C3CCN(C(c4cn(C)cn4)=O)C3)C)n2)ccc(F)cc1 c1(-c2onc(-c3ncc(C4CCOC4)s3)n2)ccc(COC)nc1 c1(OC)nccc(C(=O)NC2CCN(C(=O)Cc3ccsn3)CC2)c1Br N1(C(C(C)NS(C)(=O)=O)=O)C2CCC1C(NC(=O)CC1SC(=N)NC1=O)C2 C(CCN=c1[nH]c(C)cc(=NCCOC)[nH]1)Oc1cccc(NC(CCC)=O)c1 C1(NC(CCc2ccc(C)s2)=O)CC2CC(NC(=O)CC(C)c3ccco3)C1C2 c1(CC(=O)NC2(C)CC(NC(=O)C(C3CCCO3)=O)C2)ccc(C(F)(F)F)cc1 C1(CC(=O)NCC2C(NC(c3c(C)cc(C(F)F)o3)=O)CC2)CN2CCC1CC2 Cc1ccc(F)c(C(=O)NCC2(F)CCC(CNC(=O)C(C)C3CCC3)CC2)c1 C1(C(=O)NCCCNC(c2cc(C)nn2C(F)F)=O)COc2cc(F)ccc2C1 c1(NC(C2(F)CCN(C(c3cc[nH]n3)=O)C2)=O)cccc2c1CNC2=O c1(C(N2CC3C(NC(=O)Cc4cnc[nH]4)C3C2)=O)cncc2cc(Cl)ccc12 C(N=c1[nH]c(=NCCC#CCO)[nH]c2c1CCC2)C1(OCCO)CCSCC1 c1ccc2c(c1)CCN(c1ccnc(NCc3cnc(C4CC4)o3)n1)C2 C1(CC(=O)NC)CN(C(=O)Cc2nncn2C)CCN1C(=O)CNC(C)=O CC1(C)CN(C(C2CCC23CCC3)=O)CCC1NC(c1n[nH]cc1Br)=O c1(CNC(CC=C)=O)ccc2c(c1)CCCC2NC(C1(S(C)(=O)=O)CCC1)=O S(=O)(=O)(c1ccc(C)c(C(N2c3ccccc3CC2CO)=O)c1)NC C(=O)(C1CCCc2scnc21)N1CC2=C(CN(C(CSCC(=O)OC)=O)C2)C1 N1(C(=O)OC(C)(C)C)CC(CC(=O)NCC2(n3nccn3)CC2)CC1(C)C N1(C(C=CC(=O)NC2CC2)=O)CCC(NC(C2(O)CCCC2)=O)C(CO)CC1 C1(C(N2C(CNC(CCC(=O)NCC)=O)CC2)=O)CCN(C)C(=O)C1 N1(C(C(C)=[SH]c2nc(C)oc2C(=O)O)=O)CCC(C(N)=O)CC1 CC(N=[N+]=[N-])C(=O)N1CC(CC(=O)NCC=Cc2ccccc2)CC1C CC1(C)C(NC(=O)CCC2CCCC2)CC1CNc1ncccn1 N1(C(C(CC(C)C)(C)C)=O)CCN(CCNC(C2CC(C)(C)C2)=O)C2(CCC2)C1 N1(C(C2(COC)CC2(F)F)=O)CCC(O)(CS(C)(=N)=O)CC1 N1(C(CCC#CC)=O)CCCC12CCCN(C(C1CCCN1CC(F)(F)F)=O)C2 CC1(C)CCCC(NC(C2(NC(c3cnn4c3CCC4)=O)CC2)=O)C1 CC1CCC(NC(c2cc(O)nc(Cl)c2)=O)CN1C(c1ccc(C(N)=O)cc1)=O C1(C(=O)NC2CN(C(C=CC=CC)=O)CC(O)CC2)CCn2c(C)nnc2C1 CC(S(=O)(=O)CCCc1ccno1)c1nc[nH]n1 C(=O)(C(C(C)(C)O)NC(=O)C(C)N(C)C)Nc1cc(C)sc1 CC1CN(C(=O)C(C2CCCO2)C2CC2)CCN1C(=O)C=CC1CCOC1 N1(C(c2c(CSC)cccn2)=O)CCN(C(=O)C2=COCCO2)C2(CCC2)C1 C=CCC(CNC(c1ccnnc1C)=O)C(=O)Nc1ccc(F)cc1O N1(C(C(C)C)=O)CCCCC1C(=O)NCC(C)NC(c1csc(C(=O)OC)n1)=O c1ccc(CNC(c2ccc(C3CCCO3)s2)c2nnnn2-c2ccccc2)cc1 N1(C(CCC)=O)CC(NC(=O)Cc2cc(Br)ccc2O)C2(CC2)C1 C(C(C)(C(=O)NCCCCC(C)C)NC(C1CC(F)(F)C1)=O)SC C1(NC(Cc2cnc(C)[nH]2)=O)CCCCC12CCN(C(c1ccccc1)=O)C2 CCC(C)(C(=O)NCC1CN(C)CCN1C(=O)CC1(C(=O)OCC)CC1)C(F)F C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(C)C(CNC(=O)CSC(C)(C)C)C1 c1(C(=O)NCC2CCN(C(c3cc(C)c(Cl)s3)=O)CC2)cccc2ccnn12 C1(CC)CN(C(=O)CC#N)CCC1C(F)(F)F.c12cnc(nc1)CNC2=O c1(C(N(CC(C)NC(C2(C(F)(F)F)CC(F)(F)C2)=O)C)=O)cc(F)cc(F)c1 C1(C(N2CCC(C)(NC(C(c3ccc(C)cc3)=O)=O)C2)=O)CC12CCSCC2 N1(C(C=C(C)C2CC2)=O)CCC(O)(C(C)NC(=O)Cn2cnc([N+](=O)[O-])n2)CC1 C(C(CC(=O)NCC=Cc1ccc(C)o1)OC)NC(C(CC)OCC)=O Cc1ccc(C(=O)NCC2CC2NC(=O)COc2ccc(F)cc2F)c(=O)n1C c1(C(=O)NCC(O)CC2CCCO2)ccc2nnc(-c3ccccc3)n2c1 C12(NC(C(C)C#N)=O)COC(CNC(=O)C(c3ccc(F)cc3)NC(N)=O)(C1)C2 C(CNC(C1CCCN1CC)=O)(C(C)(C)C)NC(COc1cccc(CC)c1)=O C(CC(C)CC)(C(=O)NCCCCS(C)(=O)=O)NC(CC(C(=C)C)OC)=O C1(NC(C2CC(OCC)C2)=O)CC2CC(NC(=O)C(CC)NC(N)=O)CC12 c1(CCC(=O)NC(CNC(CCSCCCC)=O)(C)CC)cncc(O)c1 C(=O)(CCCCCCCC1CC1)N1CC(NC(c2c(CC)cco2)=O)C1 C(C(CNC(=O)C=Cc1ccoc1)C(F)(F)F)NC(C(CCC)N(C)C)=O CCC(CN=c1nc(N(CCCCC(C)C)C)c2ccc(C)cc2[nH]1)C(C)C c1(N(C)CC2CCC2C(F)(F)F)ccc(S(=O)(=O)NC2CC2)cc1Br C(=O)(CC(C(F)F)NC(C1CCNC(=O)C1)=O)NCCOCC(C)C N1(C(CCC2CCC(=O)N2)=O)CCOCCC12CC2 c1(OCCOC)ccc(SC)cc1Cl.N1(CCC(=O)O)CCC(CCCN)C1 C1(NC(CN(C)C(N)=O)=O)CCN(C(C23CC4CC2C3C4O)=O)CC1O c1(C(=O)NCC(C)CN(C(=O)C2=CCCS2)C)cc2scnc2[nH]1 C1(CCNC(c2scc(C)c2)=O)CN(C(c2occ3c2CCC3)=O)CC(C)O1 Cc1ccc2cc(C(N3CCCC3CCCNC(=O)C(=O)NC(C)C)=O)nn2c1 c1(CC(=O)NC(CC)CNC(=O)CCC(N)=O)cc(F)c(OC)c(S(N)(=O)=O)c1 C1(C(N(CC(C)NC(C2COC(=O)O2)=O)C)=O)CCC(=O)N1 CCC(CC1CCCCC1)C(=O)NCCN(C(=O)C(c1cccc(Cl)c1)OC)C N1(C(Cc2c(C)n[nH]c2C)=O)CCCCC(CNC(=O)CSc2nncn2C)C1 N1(C(CCCN(CCCC)CCCC)=O)CCCC(N(C(=O)C(F)F)CC)CC1 c1(C(=O)NCCOC2CCN(C(c3c(C)cn(C)c3)=O)C2)ncc(Cl)cc1O N1(C(c2c(CC)occ2)=O)CC(C2CCCN(C(=O)CC3CCC4CC34)C2)C1 c1(C(=O)NC2C(NC(C3(SC)CCC3)=O)CCCCC2)cnn2c1C(C)CCC2 C1(C(=O)NCCC2CN(C(C(CC)(F)F)=O)C2)CCC(C)(C)OC1 c1(OC)ccc(C(=O)NCCNC(C2(OC)CCSC2)=O)nc1N C1(CNC(C=C(C)C(C)(C)C)=O)CC(O)CN1C(=O)C=CC1CCCO1 c1(C(=O)NCC2CCCN(C(C3(C)CC3(F)F)=O)C2)ccc2cc(F)ccc2n1 O=S1(=O)CCN(CC2CNCC23CC3)C(C2CC2)C1 C(C(C)(C)C=C=C(C)C)(c1nnnn1Cc1ccco1)NCc1n(CC)ncn1 c1(CC)cc(NC(=O)C(CN(C)C)NC(C2COCC2C(N)=O)=O)cnc1C C(=O)(C(CC)(CC)OC)NC(C(C)NC(C1CC(C)(CC)C1)=O)C CC(CC(=O)NC(C)(C)CCNC(=O)CSc1cc2c(s1)CCC2)C(F)F C1(CC#C)CCCCN1C(=O)CC1CCN1C(C1CC2C=CC1O2)=O Cn1cc2c(C(=O)NC(CNC(=O)COC(F)F)C3CC3)cccc2n1 n1(CC)cc([N+](=O)[O-])c(C(N2CCC2CNC(=O)CC2CC3(CC3)C2)=O)n1 c1(C(=O)NC2(CNC(c3c(C)cc(N)s3)=O)CCC2)cc2c(=O)[nH]ccn2n1 C(=O)(CCCC(=O)NC1CC(CNC(=O)CNC(=O)C2CC2)C12CCC2)N(C)C Cc1cnn2cc(C(=O)NCC3CN(C(C4COCCOC4)=O)CC3O)cnc12 C(c1cn(CC(F)(F)CCN(C(C2CCCN2CC(C)C)=O)CC)nn1)=CC c1(CCC(=O)NC2CCN(C(C3CC(=C)C3)=O)C2)nncnc1O CCC(CC)(CC)C(=O)N1CC2CCC1C2NC(=O)C(C)SC c1(NC(C(=O)NC2CC(C(=O)OCC)C2(C)C)=O)ccc(Br)c(C)c1 c1(C(N2CC(C)(C)C(NC(=O)CC3CCOC3)C2)=O)cc2c(cc1N)OCO2 N#CC1(CC(N2CC=C(CNC(C3(C(N)=O)CCC3)=O)CC2)=O)CCOCC1 c1(C(N2CC(CCNC(Cc3scc(C)c3)=O)C2)=O)cc(C)nc(C)n1 N1(C(C2(CNC(C(CSC)O)=O)CCC2)=O)CCCC(C(N)=O)C1 C1(C(N(CCCNC(c2nc(=O)n(C)[nH]2)=O)C(C)C)=O)CN2CCN1C(C)C2 c1(SC)cc(C(=O)NCc2csc(CNC(=O)C(C)(O)C(C)C)n2)ccc1F CC1=C(C(=O)NCC2(C)CC(NC(C3(F)CCC(C)CC3)=O)C2)S(=O)(=O)CCO1 CCCCCC(CC)C(=O)N1CCCN(C(c2cnn3ncccc23)=O)C(C)C1 N12CCC(C)(C(O)C1)C2.c1(C(N(C)C)=O)ncc(C(F)(F)F)cc1C(=O)O C(C(CNC(=O)C(O)CC(F)F)C(F)(F)F)NC(=O)C=Cc1ccccn1 CCCC(C#N)C(=O)N1CCC(NC(C2CC3(CCO2)CC3)=O)CC1C N1(C(C(C(C)(C)C)SC)=O)CCC2CN(C(=O)CCn3cnnn3)CC2C1 N1(C(c2csc(Br)c2)C(=O)NCC)CC(SC)C(C)(C)C1 N1(C(CC(C)CC(C)(C)C)=O)CCC2(CC1)CCN(C(c1cnnn1C)=O)C2 c1(C(C(=O)NCCCOC)N(C(C)CS(C)=O)C)cc(I)ccc1F N1(C(C(C)C2CC2)=O)Cc2[nH]nc(C(=O)NCC(=O)NC(C)(C)C)c2C1 c1(NC(C2CN(C(C(C)=O)=O)C2)=O)cccc(-c2ccn(C)c2)c1 C12(C(=O)NC(C(=O)OCC)(C)C)CC(CO)(CN1C(C1CCC1C)=O)C2 C(=O)(C1Cc2c(Cl)cccc21)NC(CC=C)CNC(=O)C=C(C)C1CCCCC1 c1(C(=O)NCCC(C)N(C)C(c2coc(Cl)n2)=O)ccoc1C(F)(F)F N1(C(C2C3CN(C(C(C)n4cccc4)=O)CC32)=O)CCCOCC1C n1(CC)nc(-c2occc2C)nc1C1CC(=C2CC2)C1 C(=O)(CC1=CCN(C(c2ccoc2Cl)=O)CC1)N(C(CC)COC)C N1(C(c2[nH]cc(S(N)(=O)=O)c2)=O)CC2CCCCC2(NC(c2cc[nH]n2)=O)C1 c1(C(N(C2CCC(NC(=O)C(C)(F)F)CC2)C)=O)cnn2c1OCC2 C1(NC(c2c(CC)cco2)=O)CC2CC1CN2C(c1cnc(C)nc1COC)=O Cc1ccc(CC(=O)NCCCCN(C(=O)C(C)(C)N(C)C)C)s1 CC(N=c1[nH]c(=NCC2(C)CC2(Cl)Cl)[nH]c2c1COC2)c1cccc(O)n1 c1(OCCCOC(C2CSC(C(F)(F)F)C2)=O)cnc2ccccc2c1 c1(CC)nnc(SCC(=O)NC2CC3(CC3)C2)n1N C1(C(=O)NCC2COCC2O)CCCN1C(=O)CN1CCCC1 C1(C(=O)NCC2(O)CC(NC(C3(CC(C)C)CCC3)=O)C2)CCCCC1O C(C1CCC(C)CC1)=C(C)C(=O)NCCNCc1cc(C#N)ccn1 n1(CC#C)c(C)cc(C(=O)NCCCCNC(c2ccc(Cl)cc2CC)=O)c1C N1(C(c2cc(OC)c(Cl)cc2)=O)CC2CCN(C(C3CCS3(=O)=O)=O)CC2C1 Cc1noc(C)c1C(C)CC(=O)NCCC(C)(C)NC(=O)CCc1ncco1 N1(C(c2n(CCC)ncc2)=O)CC(C(=O)N2CCCO2)CCC1(C)C C1(NC(Cc2ccc(CC)cc2)=O)CC(O)CN(C(c2cnc(O)o2)=O)C1 C1(CCC)CN(C(=O)C(O)Cc2cnc[nH]2)CCN1C(C1CCCCC1)=O Fc1cccc(Cl)c1CCc1nc(-c2nccs2)nn1CC1CCOC1 C1(CNC(c2cc(C)[nH]n2)=O)CCCC(NC(=O)C(C)(C)N2CCCC2)C1 N1(C(c2cn(C)nn2)=O)CCC2CCCC12C(N1CCC(C)(F)C1)=O C1(CC(=O)N(C)CCOCCCNC(=O)CSc2nncn2C)CCCCC1C N1(CC=C)C(=S)NC(c2cccc(C)c2I)C(C(=O)OCC)=C1CCl C12(C(=O)NC(c3noc(C)n3)CC)CC(C)(CN1C(=O)C=Cc1cncs1)C2 c1(C(=O)NC(c2c(C)n(C)nc2)C)n[nH]c2c1CC(C)(C)C2 c1(C(=O)NCC(CC=C)NC(C2(C(F)F)CCCO2)=O)ccc(OC)c(F)c1O C1(N(C(C=COCC)=O)C)CC2CCC(C1)N2C(c1cnn2ccsc12)=O N1(C(C(CC)(C)C(F)F)=O)CCC2(CC1)OCCC2NC(c1cnco1)=O c1(C(c2ccccc2)NC(=O)C(F)(F)c2cnccn2)ccc([N+](=O)[O-])c(O)c1 N1(C(C2ON=C(C)C2)=O)CCN(C(c2cc3c(s2)CCCC3)=O)C2COCC12 c1(NC(C2C(c3c(OCC)cccc3Cl)C2)=O)cc(OC)c(C2CC2)c(O)c1 C1(NC(COCCCC)=O)C2CCC1CN(Cc1cc(C)ccc1Br)C2 C1(C(=O)NC2CC2NC(C2(Br)CC2)=O)CCC(CSc2ccccc2)C1 N1(C(CCN(CC)CC)=O)CCCC1(C(=O)NCC(C)CN(C)C)COC c1(C(=O)NCC2CCN(C(CS(CC)(=O)=O)=O)C2)cc2nc[nH]c2cn1 c1(OCC(N2CC(C(C(N3CC(CC(C#C)C)C3)=O)OC)C2)=O)cccnc1 C1(C(C)NC(C2CC(CF)C2)=O)CCN(C(c2cnn(C(F)(F)F)c2)=O)CC1 c1(C(N2CC(CC)C(Nc3ncnc(C)c3Br)CC2)=O)cc(F)c(C)cc1F C1(C(=O)NCc2c(CCNC(=O)CC3=CCCC3)ocn2)CCc2cncn2C1 n1(CC(=O)NC2C(CNC(c3c(C(C)=O)cccc3)=O)C2)ccc(=O)n(C)c1=O C1(C(=O)NCc2c(CN(C(=O)C#CC3CC3)C)cccc2)CCC(C)(O)CC1 c1(-c2cn(C(C(=O)NCCCCC)C)nn2)ccc2c(c1)NC(=O)C2 C1(C(N(CC#CC)C)=O)CN(C(=O)CCc2nccn2C)CC1C c1(C(C)(C)C)ccc(C(N2CC3CC2C3NC(=O)CCC2CCC(=O)N2)=O)nc1 c1(SC)nc(O)c(C(=O)NC2CCC(NC(=O)C3=CCC3)C2)cc1C#N c1(CN2C(c3c(C)cccc3)CCC2)cc2nc(C)cc(-c3ccccc3)n2n1 c1(NC(C2CC(C)N2C(c2cc(C#N)cs2)=O)=O)ccc(CO)c(Cl)c1 C1(C(=O)NCc2cn(C3CC3)nn2)CCN(C(c2cc(C)n(C)n2)=O)C(CC)C1 C1(C)(C(N2CC(NC(CCCCC)=O)C(C)(C)C2)=O)CCCCC1(F)F C1(NC(C2C(C)SCCC2)=O)CCC2(CCN(C(c3cnc(Cl)n3C)=O)C2)C1 c1(C(C)(C)N(C)C(C2CCCCC2)=O)cc(F)c(F)c(Cl)c1F.CC C1(NC(=O)NC(c2nc(C(C)(C)C)cs2)C)CCCCCCC1CO C1(CC)(NC(=O)C=CC2CCOC2)CCN(C(c2ccc(O)cc2OC)=O)CC1 c1(C(N2C3(CNC(c4cc(OC)ncc4)=O)CC(C2)C3)=O)cc(OC)cc(C)n1 c1(NC(C(C(C)C)C)CNC(C2(C)CCCCC2)=O)c(C#N)cccc1[N+](=O)[O-] c1(C(N2CCCN(C(C(CSC)OC)=O)CC2)=O)c2c(nn1C)CCC2 N1(C(C2(C#N)CC=CC2)=O)CC2CCOC2(CNC(C2CCCSC2)=O)C1 C1(CNC(C(F)=CC)=O)(NC(=O)COC(C)(C)CC)CCCCCC1 c1(CCC(N2CCN(C(c3cnc(=N)[nH]c3)=O)CC2)=O)c[nH]c2ccc(F)cc12 C(=O)(CC(CC)C(C)(C)C)N1CCC(N(C(c2ccc(O)cc2F)=O)CC)CC1 c1(C(N2CC(NC(CC3CC(=C)C3)=O)C(SC)C2)=O)ccc(=O)n(C2CC2)c1 N1(C(C(C)(C)C2CCC2)=O)CCC2(CC1)CC(CNC(=O)C1=CC(O)CCC1)C2 c1(OCC)nc(C)ccc1C(=O)N(C1CCN(C(c2ncc(N)cc2Cl)=O)C1)C C(CC(C(C)(C)C)NC(C1C(C(C)=O)C1(C)C)=O)N(C(C(COCC)(C)C)=O)C C(=O)(C(CCS(C)=O)N(C)C)NC(CC)CNC(c1ccn(CC)c(=O)c1)=O Cc1ccc(F)c(C(=O)NCC2(C(N3CCC3CF)=O)CC23CCC3)n1 C=CC1(CC(=O)NC2CCSC2C)CN(C(=O)Cc2cnn(C)c2)C1 c1(C(=O)NC2CCC(NC(c3ccc(CC)s3)=O)C2)ccccc1C(C)C C1(CNC(c2coc(C(F)F)c2)=O)CC(O)CN1C(C1CCCC1C(F)F)=O Cc1noc(C2CC2)c1C(=O)NCC1(NC(=O)CC2(C)CCOC2)CCC1 C1(NC(c2c(CC)n(C)cc2)=O)COC2C(NC(=O)CC3CNC(=O)C3)COC12 Cc1nn(C)c(C)c1CCC(=O)NC(C)(CNC(C1CCCC(F)C1)=O)C1CC1 C1(CCNC(CC=CC=C)=O)CN(C(=O)Cc2cccc(O)c2)CCS1(=O)=O C1(CC(=O)NCC(CC)NC(=O)CN(C)C(c2cccs2)=O)CCCCN1C c1(OCC)cc(C(N2CCC(CC)C2C)C(=O)NCCCSC)ccn1 Cc1nc(NC(CCNC(=O)Cn2cnnn2)C(C)C)cc(SC(C)C)n1 c1(CNc2cc(OCC(C)C)ncc2)cc(Cl)cc(C#N)c1 N1(C(CC(CNC(C=C(C)C2CC2)=O)C)=O)CCn2c(C)nnc2C1 C1(NC(C(C(C)C)C2CCC2)=O)CC2CCCC(C1)N2C(C1CCN1C)=O c1(C(N(C(CC#C)C(=O)NC)C)=O)cccn(CCOC)c1=O c1(CN(C(c2cn(Cc3ccc(Cl)cc3)nn2)C)C)nnc2n1CCCC2 c1(OC)ncc(C(N2CCN(C(C3COCCC3(F)F)=O)CC2C)=O)cc1C C1(CNC(c2ccc(N(C(C)=O)C)cc2)=O)CN(C(=O)CC#N)C2COCC2O1 N1(C(C(C2CN(C(=O)CNC=O)C2)OC)=O)CC2CCC(C1)O2 S(=O)(=O)(c1ccc(NCC2CCCCN2CCO)cc1Cl)NC1C(C)CCC1 CC(C)C(O)CC(=O)N1CCC(C(N2CCC(C(C)(C)O)CC2)=O)C1 C1(NC(C2C(C)CCO2)=O)CCN(C(c2ccc(C(F)F)o2)=O)CCC1(F)F C1(C(=O)NCC2CN(C(c3cnc(COC)s3)=O)CCO2)(CC)CC(C)(C)C1 c1(C(=O)NCC(C2CCOC2)N)noc2cc(C(F)(F)F)ccc12 CCCC(C)(C)CC(=O)NCCCOCCCNC(C1CCN(C)C1CC)=O N1(C(c2nc(COC)oc2)=O)Cc2[nH]nc(C(=O)NC3CCSC3)c2C1 N1(C(Cc2ccc(OCC#N)cc2)=O)CCC2(CC1)CC(=O)NCC2O C(=O)(C(C(=O)N(C(C)(C(=O)Nc1cccnc1C)C1CC1)C)OC)OC C1(C(=O)NC2CCC(C)N(C(=O)Cn3nccn3)C2)CCc2ccnn2C1 C1(CCC)(NC(=O)COc2ccccc2OC)CCN(C(C2CC(F)C2)=O)CC1 C1(c2nnnn2CCCSCC)(Nc2cncc(CC)c2)CSCCSC1 CC1CCN(C(=O)C(C)CCO)CC1NC(C1CCCN1C1CCCC1)=O N1(C(Cn2c(C)nnn2)=O)CCCCC1CCCNC(=O)CCC1CCCOC1 C1(CN(C(C2CC(F)C2)=O)CC)C2CN(C(=O)CC3CCOC3)CC12 C(C(C(C)C)C(C)C)(c1n(-c2c(CC)cccc2)nnn1)NCC1(C)CC1(C)C C1(CNC(=O)CN2CC3CC3C2)CC2(CCC2)CN1C(c1ccc(CO)cc1)=O N1(C(=O)Cc2cc(-c3ccccc3)on2)CCOCC(CNC(C2(Cl)CC2)=O)C1 n1(CCC(=O)NC(CNC(CNC(C(CC)C)=O)=O)CO)ccc(O)nc1=O N(C(=NCCCCC(F)(F)F)NCc1ccc(COC)cc1)CC1(OC)CCOC1 C1(CC(=O)N(CCCNC=O)CCO)CCN(C(c2ncccc2F)=O)CC1 c1(C(C)C)c[nH]cc1C(N1CCC1(C)CC(=O)N(CC(C)O)C)=O CC1CC(C(N2CCCC(CC3CC3)C2)=O)CN(C(C2(Cl)CCCCC2)=O)C1 c1(C(=O)NC(CNC(C2(C)CCCS2)=O)CO)c(C(F)(F)F)ncn1O C1(CC)CN(C(C2CC(O)C2)=O)CC1C(=O)Nc1ccc(F)cc1 C1(C)(N(C)C)CCCN(CCC(=O)NC2CCCC3(C2)N=N3)C1 C1(CNC(c2c(C)nccn2)=O)CC(F)(F)CN1C(c1cnn(C)c1Br)=O Cn1cnc2c1CCCC2C(=O)NCCCCNC(=O)C(C)(C)C1CCOC1 C(F)(c1ccccc1)=CC(=O)NCC(CCOC)NC(=O)C(c1nc(C)cs1)C c1(ONC(=O)Nc2scc(COC)c2)ccc([N+](=O)[O-])c(C)c1 c1(N2CCCC(O)(CNC(c3cncc(OC)c3)=O)C2)[nH]cnc2nc(Br)cc1-2 c1(C(N(C2CCN(C(c3cc(-c4cccs4)on3)=O)C2)CC)=O)nnsc1C c1(CNC2C(C(=O)Nc3cnc(C(F)(F)F)nc3)CCC2)cc2ccncc2[nH]1 c1(CNC(C2C(NC(CCSCCC)=O)C2)=O)ccc2n[nH]cc2c1 c1(N2C(C3CCN(C(C(CCCC)(C)F)=O)C3)CCC2)ncc2c(ncn2C)n1 Cc1cc(CC(=O)OCc2ccn(Cc3cccs3)n2)nc(C)c1 N1(S(C)(=O)=O)CCCC(C(=O)NCC(C2CC2)NC(c2ccon2)=O)C1 C1(CC(=O)NC2CCN(C(CC(C)C(F)F)=O)CC2F)CCC2(CCC2)CO1 C1(C#N)(C(N2CC=CC(C(N3CC(N(C)CC)C3)=O)C2)=O)CCCCC1 C1(C(C)NC(CCC=CC)=O)CCN(C(c2sccc2-n2cccc2)=O)CC1.C CCC(C)(C(=O)OC)NC(C1CC=CCN1C(C1C(C)(C)C1(C)C)=O)=O C(=O)(C(=O)NCCOCCN1CCCC1)NCCC1C(C)C1 CC1CCC(=CC(=O)NCC2CC2CC(=O)NC2(CO)CC(F)(F)C2)CC1 CC1(C)C(C(=O)NC(CNC(c2cncnc2C2CC2)=O)C2CC2)CCS1(=O)=O N1(C(C(COC)N(C)C)=O)CCC(F)C(NC(c2c(Cl)nsc2Cl)=O)C1 C1(NC(Cn2nnc(=N)[nH]2)=O)CS(=O)(=O)CC1NC(=O)CNC(=O)NC1CC1 Cc1[nH]c(NC(=O)CCc2ccccc2)c(C)c1C(N1CC2CC1CN2C)=O O(NC(=O)C(Cc1cc[nH]n1)NC(C1(F)CCCCC1)=O)CC(=C)C C1(CNC(C(C2CCOC2)OC)=O)CN(C(C2CC(F)(CO)C2)=O)CCN1C C1(NC(C(CCC)C)=O)CC2(CCN(C(c3ccc4c(n3)NCC4)=O)C2)C1 C1(Cn2cc(CN(C)CC)nn2)CCCCN1C(=O)Cc1cn(CC(=O)O)nn1 c1(C(=O)NC(CCNC(C(C=C)O)=O)C)cc(F)cc(C)c1N c1(C(=O)NC2(C)CN(C(C(CC)O)=O)C2)ccc(C(=O)OC)n1C N1(C(C(c2ccc(OC)cc2)CC)=O)CC2OCCN(C(c3cc[nH]c3)=O)C2C1 c1(N(C)CC2COC(CNC(=O)C(Cl)=CCl)C2)cc(=O)n(C)cn1 C12(CNC(CCSCCC)=O)CC1CN(C(=O)COc1ccc(C)cc1)C2 c1(C(=O)NC2C(CC(=O)N(CCC(F)(F)F)C)C(O)C2)cn(C)ccc1=O C(=O)(C#CC(C)(C)CNC(=O)C(C)OCC1CC1)N1C(CC)CCCC1 C1(NC(COCCCCC)=O)CCCCCC1NC(C1CCCC(C#N)C1)=O C=CCC(CC(=O)NC(CCO)C(C)(C)C)NC(=O)CCC(C)(C)N(C)C C1(C(=O)NC2CN(C)C(CO)C2)CC(N=[N+]=[N-])CN1C(c1ccc(O)cn1)=O Cc1cc(=O)n(C)nc1C(=O)NC(C)CCCNC(c1n[nH]cc1C(F)(F)F)=O c1(C(=O)OC)cc2c(nc1NC1CCCN(C(=O)C(C)CC3CC3)CC1)CCC2 Cn1nc(C(=O)NCC2(NC(=O)CC3CC(=O)C3)CC2)c2c1CCSC2 N1(C(c2ccn(CC(F)(F)F)n2)=O)CC2CCOC2(CNC(=O)C(O)C2CC2)C1 n1(CCC)cc(C(=O)NC(C)CNC(=O)C(O)C(C)c2ccccc2F)c(C)n1 c1(CC)oc(C(=O)NCCCCNC(=O)C(c2ccc(Br)cc2)O)cc1C CN1CCN(C(C2COCCN2C2CC2)=O)C(CNC(=O)CC2CC3(CC3)C2)C1 CC1CCc2nc(C(N3CCSC3c3ccco3)=O)cn2C1 N1(C(C2CN(C(CC#N)=O)C2)=O)CCCCC1CO C1(C(N2CCCC(CCCC)C2)=O)C2CC3C(C2NC(C2(Cl)CC2)=O)C13 C1(C(N2CCC(CN(C(=O)CCN3C(=O)CCC3=O)C)C2)=O)CC(C2CCC2)C1 CCCC(CNC(=O)CCCCNC(C)=O)C(=O)N(C1CCCNC1=O)C N1(C(c2c(SC)ccs2)=O)CC2CC2(CNC(C2CCS2(=O)=O)=O)C1 N1(C(C(=O)NCCCSC)C2CC2C)CCCC(C)(C)C1 C1(C(=O)NC)CCCCN1CCN(c1ncccn1)C(=O)OC(C)(C)C C1(N(C)C(C23CCCC2C3Br)=O)CCCCCN1C(=O)NC1CCC1 C(C)(C)(CCC(=O)N(C(C)C(C)SC)CC)NC(C=CC(CC)C)=O N1(C(C2CCC3C(C2)C3(F)F)=O)CCC2(C1)CN(C(=O)C(F)C1=CCCCC1)C2 C(=O)(CCC(C)(C)C#N)N1C(CCNC(C(C(C)C)CN(C)C)=O)CCC1 C1(NC(C(F)(F)Sc2cn(C)nn2)=O)C=CCN(C(=O)CC(=O)OC(C)(C)C)C1 N1(c2nccc(NC(CCn3ncc(C)c3)=O)c2)CC(C)OC(C)C1 C1(NC(C(Cc2cn[nH]c2)NC(=O)CCc2cccs2)=O)C2CCCC1COC2 C1(NC(C2C(=C)CC2)=O)CCCCC12CCN(C(c1n[nH]cc1[N+](=O)[O-])=O)CC2 C(=O)(C1CCCc2scnc21)N(CCCNC(c1cc(C(N)=O)no1)=O)C1CC1 c1(NC(C2(Cc3ccccc3)CCNC2)=O)cncc(N2CCCC2)n1 c1(C(C(=O)NCC(C)NC(c2cscc2F)=O)SC)ccccc1 CCCC(CCCNC(=O)CCCF)NC(=O)CC1(C)CCCC1 Cn1c(C(N2CC3CCCC3(NC(C3CCC(O)CC3)=O)C2)=O)cc2sccc12 C(=O)(C1=CCC2CCC1N2C(c1ccc(C)nn1)=O)NC(CC)C(C)(C)C c1(C(=O)NC2CC(CNC(C3(CC#C)CCC3)=O)C2)ccc(C)c(C)c1O N=c1[nH]nc(C(=O)NCc2ccoc2C(F)(F)F)s1 C1(CNC(C(CCSC)OC)=O)CN(C(=O)Cc2cc(C)ccc2F)CC1(C)C c1(C(=O)NC2(CCNC(CCC=C)=O)CC2)cc(F)cc2c1CCC2 c1(C(N2CCC(OCCNC(c3cncc(CC)n3)=O)C2)=O)nccc(OC)c1N C(CN1CCOCC1)(CC(F)(F)F)C(=O)NC(CCCC)(C)C N1(C(CCC=C)=O)CCC(C=C)(C(=O)NCC2CCCCCC2)C1 c1(OC)cc(CCNC(=O)CCCC(=O)C2CC2)cc(OC)c1OC(F)F CC(CS(C)(=O)=O)C(=O)N=c1cc(C2CCNCC2)[nH][nH]1 C1(C)(C(=O)NC2CC(N(C(c3cn(CC)nc3C)=O)C)C2)CCCN(C)C1 c1(C(N2CCN(C(N(C)C)=O)CC2)=O)c(-c2ccc(I)cc2)ccc2c1OCO2 N1(C(c2c(OC)c(Cl)cc(Cl)c2)=O)CCCC(C2(NC(=O)C(C)=C(C)C)CC2)C1 CC(C)C(C(=O)NCC12CCC(CC1)N2C(c1ncccc1N)=O)C(C)C C=C=CCCC(=O)NCCn1ccc(C(=O)N(CC(C)O)C(C)C)c1 N1(C(c2cc(CC)n(C)n2)=O)CC(C(=O)NC2CCN(CC)CC2C)CC(C)C1 c1(CNC2C(C(=O)Nc3c(OCC)ccc(C)c3)C2)c(Br)ccc(OC)c1O C(=O)(CCCCCCCC1CC1)NC1CCN(C(c2cnc(C)s2)=O)C1C1CC1 N1(C(Cn2c(C)ccn2)=O)CC2CCC(C1)N2C(C1CC(F)C1)=O CC1CC(CC(=O)NCCN(C)C(c2cc3cnn(C)c3s2)=O)CC(C)(C)C1 C(=O)(C(C)(C(F)F)c1ccccc1)NC1C(C)CN(C(c2cc(O)nn2C)=O)C1 C1(C)(NC(c2ccnc(C)n2)=O)CCCN(C(c2ccc(C)c(F)n2)=O)C1 Cc1ccc2nc(C(=O)NCCC3CCCN3C(C3CC(=O)N(O)C3)=O)cn2c1 C(=O)(C1(C)CCn2ccnc21)N1CCCC(NC(C(C)n2ccnn2)=O)C1 C1(C(N(C2CC3CC3C2)C)=O)CN(C(c2cc(C3CC3)[nH]n2)=O)CC1(F)F N1(C(CC(C)(F)F)=O)CC2CCN(C(C3(C)CC3Br)=O)CCC2C1 c1(CC(N2CC(n3cc(C4CCCOC4)nn3)C2)=O)c(F)cncc1Cl C(=O)(C(CC(C)C)C(N)=O)NC1CCC(CC(=O)N(CCOC(C)=O)CCO)CC1 C1(CNC(CC2(C)CC2)=O)CC2(CCN(C(C3(F)C(C)(C)C3(C)C)=O)CC2)C1 CC(CC(C)(C)C)C(F)C(=O)NC1CC(NC(c2cc(CO)on2)=O)C1 C1(C(=O)NCC2(C)CCN(C(c3cnc(C)s3)=O)C2)C2Cc3ccccc3C12 C(N=c1[nH]c(N2CCc3[nH]nc(O)c3C2)nc2ccsc12)C1C(=O)NCC1 C1(OC)CN(N2CC3(CC=CC3)C2C(F)(F)F)CC1F c1(OCC=C)cccc(-c2ncsc2C(=O)NCCc2ccncc2Br)c1 c1(OCCC(=O)N(C2C3CN(C(c4n[nH]c(=N)s4)=O)CC23)C)ccc(F)cc1 C(=O)(CC(CC)C(C)C)N1C(CC(=O)NC(C(=O)NC)(C)C)C2CCC1C2 N1(C(c2n[nH]c3c2NCCC3)=O)CCCc2ccccc2CC1 C1(C(=O)NC(C(=O)NCCNC(=O)NCC)N(C)CCF)CC(F)CN1C c1(OC)ccc(CN2CCC(C(N3CCOCC3)=O)C2)c(Cl)n1 Cc1nc2cccc(C(=O)NCC(O)CCNC(c3ncc(N)cc3C)=O)c2[nH]1 c1(N(CCC(=O)OC)CC(N2CC=CC2)=O)cccc(F)c1.C12CCCN1C2=O C1(CNC(C2CC(OC)CC2C(=O)O)=O)COC2(CCC(C)CC2)O1 c1(C(=O)NC(CCNC(C(C)=C2CC2)=O)C)cccc(C2CNC(=O)C2)c1 N1(Cc2cccc(CC)n2)CC(C)Oc2cc(C)ccc21 c1(C(=O)NCC(C)N(C(c2cccnn2)=O)CC)cc(Br)cnc1O C1(CC)CC(O)CCN1C(C1CCN(C(c2c[nH]cc2C2CC2)=O)C1)=O C(=O)(CC(F)(F)C(F)F)NC1(C)CCN(C(CCCn2c(C)csc2=O)=O)C1 CN1CCC(C(N2CC(C(N3CCCOCC3)=O)C(C)(C)C2)=O)CC1=O O=C1CCC(CCC(N2CCC(C(O)CNC(=O)CCCC3CC3)CC2)=O)CN1 c1(Cc2c(OC)nc(C(F)(F)F)cc2)ccnc2cc(C)c(C)cc12 S(=O)(=O)(c1cnn2ccc(N3CCCC(O)CC3)nc12)N(C1(CO)CCOC1)C N1(C(CC2CN(C)C2)=O)C2CCC1CC(N(C)C(C1COC3(CO)CC1C3)=O)C2 c1(OC)ccc(C(N2CCN(C(=O)C(C)n3cncn3)C(C)C2)=O)cc1Br Cc1cccc(C)c1CNC(=O)CC1CC(NC(C2CCC(=O)NC2)=O)C1 C12(C(=O)NCCC(CC)C)CCC(CN(C(=O)C=Cc3cnn(C)c3)C1)C2 c1(C(N2CCCC(N(C(C(C=C)(C)O)=O)CC)CC2)=O)cc2ccsc2n1C C(N=c1[nH]c(=NCCOc2ccc(Cl)cc2)[nH]c2c1COC2)c1c(C)cn(C)n1 N(C1CCCn2nccc21)C1CCCN(C(CC(C)(C)c2ccccc2)=O)C1 CC(C)CC(CNC(=O)Cc1ccc(Cl)nc1)NC(C1CCCC(C(N)=O)C1)=O C12(C(N(CC(CNC(CC3(C=C)CCC3)=O)C)C)=O)C3CC(CC13)C2(F)F C1(CNC(CC=CC=C)=O)CC(NC(c2cc(C)nc(O)n2)=O)C12CCC2 Cc1nc(NCc2ncc(C(C)C)o2)cc(N(CCC(C)(C)C)C)n1 c1(C(C(=O)NCCC2(O)CN(C(c3nc(OCC)sn3)=O)C2)C)cccc(F)c1 CC(CS(C)(=O)=O)C(=O)NCC1CC(NC(=O)CSCc2cccnc2)C1 N1(CC(=O)NC(C)CN(C(=O)C(c2cnccn2)C)C)CCC(=O)NC1=O C1(c2cn(CCN(C(=O)CC(O)c3cnc(Cl)s3)CC)nn2)CCCCCC1 N1(C(C2(Br)C(C)(C)C2)=O)CC2OCCN(C(=O)CNC=O)C2C1 Cc1cc(C)n(CCC(=O)NC(C)(C)CCCNC(=O)CC2CCOC2=O)n1 C1(CC=C)(NC(=O)C(CC)OCC)CCCN(C(=O)CC(Cl)Cl)C1 N1(C(C2C=CCN(C(=O)CCN3CCCCC3)C2)=O)C(CO)CCC12CCC2 C(CNC(c1c(C)oc(C)c1C)=O)(C(C)C(C)C)NC(CC(=O)NCC)=O Cc1c[nH]c(C(N2CCCC(N(C(=O)CSCc3ccccn3)C)C2)=O)cc1=O NS(=O)(=O)c1csc(C(C(=O)NC2CC2(F)F)N(c2ccccc2Cl)CCF)c1 c1(C(=O)NC(C)C(C)NC(c2cccs2)=O)sc2sccc2c1Cl C(C(C(=O)NCC(O)C(F)F)n1cc(Cn2cccn2)nn1)OCC C1(CNC(C(C(C)C)SCC)=O)CCN(C(c2sncc2CC)=O)C1(C)C c1(OC)cc(C(=O)NC2CCOCC2NC(C23CCC(CC2)C3)=O)ccn1 c1(CC)cc(C(=O)N(C)Cc2ccccc2-n2ccnc2C)c(C)o1 c1(C(=O)NCC(C)(O)CNC(C2CC(F)C2)=O)cc(C#N)cs1 c1(OCC)cc(C(=O)NC2CC2NC(=O)C(F)n2ccnc2)oc(=O)c1 N1(C(CCC(C)(F)F)=O)CC2CCC(CNC(=O)CC3CN4CCC3C4)C2C1 c1(C(=O)NC(C(C)NC(C(C)c2ccco2)=O)(C)C)cc(C#N)n(C)n1 C1(N(C)NC(C(c2cnn(C)c2)C)=O)CCCCN1C(=O)CCN1CCOCC1 c1(C(=O)NCCCC(C)NC(C2CCCOC2C)=O)cc(N)cc(F)c1 c1(CCC)noc(CCCC(=O)NC2CCN(C(=O)CCCc3cncs3)C2)n1 N1(C2CN(CC3(CCS(N)(=O)=O)CC3)C2)CC(C(=O)O)CC1=O C1(NC(CC=C)CO)CCCC2(CC1)CC2 CC1CN(S(C)(=O)=O)CCC1N(C(C)(C)C(N)=O)C(=O)CN1CCCC1 C1(C(N2C3C(NC(C4(C)CCN(C)C4)=O)C(C3)C2)=O)CC2(CCCCC2)C1 c1(C(CC(=O)N2CCC(C(F)F)C2)CC2CC2)c(F)cccc1Br N1(C(Cc2cnc(C)s2)=O)CCC(CNC(C2CCCC(=O)N2)=O)C(F)(F)CC1 c1(C(N2CCC(CC=C)(NC(c3conc3CC)=O)C2)=O)cc(F)ccc1F C1(S(C)(=O)=O)(C(=O)NCC(C2CC2)NC(c2c(C)cns2)=O)CCOCC1 C=CCC(C(=O)NCCCCC(=O)NC(CO)CCO)NC(C)=O c1(C(=O)NCC(C2CC2)NC(C(C(C)C)NS(N)(=O)=O)=O)ccc(F)c(F)c1F C(C(C(=O)NCCC(C)(C)N(C)C)C(C)C)NC(C(C)=C1CC1)=O N1(C(c2c(C)oc(Cl)n2)=O)CC2CCC1C(CNC(C1CCS(=O)(=O)CC1)=O)C2 CCC(F)(F)C(C)(C)C(=O)N1CCCC2(NC(c3ccccn3)=O)CCCC12 C1(C)(CC(=O)N(c2ccccn2)C(CC)C)CCOCC1 c1(C(=O)NCC2CN(C(C3CC3F)=O)CC23CCC3)cccc2cc(F)ccc12 C1(NC(CC(CC)C(C)(C)C)=O)CCC2CN(C(c3coc(C)c3)=O)CCC2C1 N1(C(Cc2cc(C)[nH]n2)=O)CCC2(C1)CN(C(c1cc[nH]c(=N)c1N)=O)CCO2 CC(C)CC(C)CC(=O)NC1CN(C(C2CCS(=O)(=O)CC2)=O)CC1C c1(C(=O)NCC2(F)CCN(C(c3cn(C)c(O)n3)=O)C2)ccc(C2CC2)c(F)c1 C1(CCNC(Cn2c(C)ncc2)=O)CN(C(C2CC=CC2)=O)CCCO1 O=C(C#CCNC(C1C2CCC(=O)C12)=O)NOCCCO C1(O)(CNC(=O)CC2COCCO2)CCCN(C(c2cc(F)n[nH]2)=O)C1 C1(NC(C2CCC(CCC(=O)OC)O2)=O)CCN(C(c2cn(C)[nH]c2=N)=O)CC1 C1(NC(c2ccc(C(C)=O)o2)=O)CCN(C(c2cnn(C)c2C(F)F)=O)CC1C c1(C(=O)NCC(CNC(C2CCC3(CCC3)O2)=O)OC)cc2c(Cl)cncc2s1 C1(NC(CC(CC)C)=O)CCC(C)N(C(=O)CC(C)C(F)F)C1 C1(NC(CCC(=O)NC(C)C)=O)CCN(C(=O)CC2COCC(C)(C)O2)C1(C)C c1(NC(C(=O)N(CCCCO)Cc2onc(C(C)C)n2)=O)cccc(N(C)C)c1 Cc1cccc2c(NC(=O)Cc3ccc(Cl)s3)nccc12 N1(C(C(C)OCCC#C)=O)CC2(C1)CN(C(=O)C=Cc1c(C)noc1C)CCO2 C=CCC(C)(C)CC(=O)N1CC(OC)CC1C(=O)NCC(C1CC(C)(C)C1)O CC(C)CCCOCC(N1CCCC1CNC(=O)C(C1CC1)N(C)C)=O C1(C(=O)NCCC(C)NC(=O)C2=CCCS2)CCc2cc(Br)ccc2O1 c1(C(=O)NC2CC(NC(=O)CN3CCC(CO)CC3)C2)ccc2nccnc2c1 C1(NC(C)=O)CN(C(=O)Cc2cncc(F)c2)C2(CCC2)C1 CC12CC(C(N3CC4CC(NC(=O)C=C(Cl)Cl)C3C4)=O)(C1)C1(CCOCC1)O2 n1(CCC(=O)NCC(C)NC(=O)CCC(=O)c2ccc[nH]2)ncn(C)c1=O c1(C(N2CCN(C)CC2CNC(C2COC2)=O)=O)cc(F)cc2ccoc12 Cc1c2c(nn1C)CC(NS(=O)(=O)CC1CC3(CCOC3)CO1)CC2 C1(C(=O)NCC(CCC)NC(c2cc(C)ccc2O)=O)CCc2n[nH]cc2C1 N1(C(c2cnc(C)o2)=O)CC(NC(=O)CCNC(c2ccncc2)=O)C(C)C1 C1(CNC(c2cc(Cl)c[nH]2)=O)C(O)C(O)CN1C(=O)CCC1CNC(=O)N1 c1(CC)nc(-c2cccnc2)nn1C(C1CC(F)(F)C1)C.CC(C)N1CC1 C(CCCCCCO)N(C(C1(CSC)CCOCC1)=O)C Cn1ncc2ccc(CN3C(C(N4CCC(F)(F)C4)=O)CC4CC34)cc12 C1(NC(C2C(C(=O)OCC)CCC2)=O)CN(C(C23COC(CCO2)C3)=O)CCC1C C1(NC(c2c(CC)onc2)=O)CC(F)CN(C(c2cccc(O)c2F)=O)C1 C(CC(C(=O)N1CCCCC1CC(F)(F)F)NC(=O)OC(C)(C)C)=CC.C(=O)OC c1(CN(C)C(C2CCCN(C(C3(C)CCSCC3)=O)CC2)=O)cc(Cl)ccc1F N1(C(CCOC)=O)CCC2(CCCN(C(c3ccc4c(c3)OCCN4)=O)C2)C1 CCCCCCCCCC(C)CCOC(c1cc(-c2c(F)cccc2F)no1)=O n1(CC(=O)NC2C(CNC(C(c3[nH]c(=N)sc3)=O)=O)CC2)cnc([N+](=O)[O-])n1 C1(NC(C(CC)SC)=O)CC2CC(C1)N(C(c1cc(C3CC3)ncn1)=O)C2 c1(NCC(C)CNC(C2CCS2(=O)=O)=O)ncnn2cccc12 c12cccc(c1)C(=O)NCCNC(=O)N2.C(=O)(C(O)CC)N1CC(N(C)CC)C1 O=C(C1=CS(=O)CCC1)NC1(CNC(c2cc(C3CC3)ccc2F)=O)CCOC1 Cc1nc2cc(C(=O)NC3CC(C)(NC(C4CC4C)=O)C3)[nH]c2s1 C1(C)(NC(C(C)N(C(c2cccnc2O)=O)C2CC2)=O)CCC(=O)N(C)C1 C1(OC)(CNC(=O)C=C(C)C(F)F)CCOC1.C1(=O)CCCC2(CCC2)N1 N1(C(C=CC(=O)OCC)=O)CCC(O)C1C(N1CCC=C(C)C1)=O c1(CC)ccccc1COC(C1(CC(F)F)CCC1)=O c1(NC(Cc2cccc(-c3cc(C(C)C)ncc3)n2)=O)cc2ccccc2s1 c1(CNC(CCOC(c2ccc(C3(C(F)(F)F)N=N3)o2)=O)=O)ccccc1Cl C1(NC(c2c(C)scc2)=O)C2CC(CN(C(=O)C(F)CC3CC3)C2)C1CO C1(NC(C2(C=C)CCC2)=O)CC2CCC1(CNC(=O)C=CSC)C2 C1(C(=O)NC(CC)C(C)CN(C)C)CC2CC1CN(C(c1n[nH]c(C)c1O)=O)C2 C(=O)(CCN=C(NCC1CCN1C1CC1)N1CCC=C(c2ccco2)C1)NC C1(NC(c2c(C)cc(CC)o2)=O)CC(O)CN(C(c2c(C)cncc2C)=O)C1 C12(C(N3CC(CN(C(C(C)C4CCCC4)=O)C)OCC3)=O)CC1Cc1c[nH]nc12 c1(OCC(CN2CCC(NC(c3cn(C4CC4)cn3)=O)CC2)O)ccc(F)cc1F N1(C(Cn2cc[n+](C)c2)=O)CCC(F)(CNC(C2CC23CCOCC3)=O)CC1 N1(C(=O)COc2ccc(F)cc2F)CC2CN(C(=O)C3=CCCCC3)CC2C1 c1(C(=O)NCC2CN(C(c3cn(C)nc3)=O)C3C2C3)cc2sc(Cl)cc2s1 C1(C(N2CCC(N(C)C(C3COC(C)(C)C3)=O)C2)=O)CC2CC1C1C2C1(F)F CCC(C)CCC(=O)N1CC2(NC(=O)OC(C)(C)C)CC1(C)C2 C1(C(N2C(Cn3cc(CCCC=C)nn3)CCCC2)=O)CN2CCN1C(C)C2 C(C)(C)(C(c1nnnn1C(C)C(=O)OC)NCc1noc(C)n1)OC N1(C(c2cn(CC)nc2)=O)CCCC(F)(C(=O)NCc2ccnc(Cl)c2)C1 c1(COC(C)C)csc(S(=O)(=O)NC(C)C(c2cccc(Cl)c2)C)c1 N1(C(COCC)=O)CCC(C)(CNC(C2CCN(C)C2)=O)C1 N1(C(C)=O)CC2CCC(N(c3ccc(F)cc3)C(=O)CC3CC3C(=O)O)(C2)C1 c1(C(=O)NC(C2CCN(C(CCOC(C)C)=O)C2)C)ccc(S(N)(=O)=O)cn1 C1(C2(O)CCOCC2)(C(N2CCC3(C(NC(CCC4(C)CC4)=O)C3)CC2)=O)CC1 N1(C(C2CC(C)S(=O)(=O)CC2)=O)CCN(C(=O)C2=CS(=O)CCC2)C2(CCC2)C1 C1(CCOC)(NC(C2CC=CCO2)=O)CCN(C(=O)COc2cccc(Cl)c2)C1 C12(C(N(CC(O)CNC(c3ccc(Br)cn3)=O)C)=O)CC=CCN1CCC2 CC1CCN(C(=O)CCc2cccn2C)CC1CNC(=O)CCC1CCOCC1 N1(C(c2ccnc(S(C)(=O)=O)c2)C(=O)NCCOC)CC2C3CCC(C3)C2(C)C1 c1(C(=O)NC2C(NC(c3c(CC)c[nH]n3)=O)C2)ncnc(O)c1F C1(NC(CC(CC)Cc2ccccc2)=O)CN(c2ncc(Br)c(C)n2)CC2(CC2)C1 C(C(C)(O)CC(=O)NCCN(C(=O)CC1CCC(C)(O)CC1)C)OC C(=O)(C(C)(C)C)N(CC(CC)N1CC(CC(=O)OC(c2[nH]nnc2C)=O)C1)C c1(C(=O)NC2CCCN(C(C(C#C)(C)C)=O)CC2)[nH]nc2ncccc12 CC1=C(C(=O)NC2(C)CC(NC(c3ccnnc3)=O)C2)C(C)(C)CCC1 C1(C(c2cn(C(C)C(=O)NCC3(CO)CCC3)nn2)(C)C)CCOCC1 C1(NC(CCCCOCCC=C)=O)CCN(C(C2CC2CF)=O)CC12CCC2 CC(C)C(F)(F)CCNC(=O)NCC1(C(=O)O)CC1 C1(NC(c2c(OC)cnnc2)=O)CC(C)CN(C(=O)CN2CCN(C)CC2)C1 Cc1ccc(CCC2CCN(CS(Cc3cc(F)ccc3F)(=O)=O)CC2)c(O)c1 c1(C(=O)NC(C)CN(C)C(C2CCC2n2ccnc2)=O)cscc1Cl c1(C2C(=O)N2C)cccnc1.c1(N)cn[nH]c1.n1(CCCC(=O)N)cnnc1 N1(C(C2C(OC)CCC2)=O)C2CC1CN(C(c1ncc(F)cn1)=O)C2 C=CCC(C)C(=O)N1CCCC(CCCCNC(c2cn(C)nc2C)=O)C1 N1(CCC(C)C)CC2(CCC(CNC(=O)CN3Cc4ccccc4C3)O2)C1 c1(C(=O)NCCC(CC)C)cccc2cc(O)ncc12 Cc1cc(C(N2CC3CC2CC3NC(c2sccc2C(C)C)=O)=O)nc(O)c1 c1(CN2CC(C(N(C)Cc3ccccc3)=O)C2)sc(Cl)cc1Br c1(NC(=O)NC2C(SC)CCC2)cnc(C)nc1C C1(NC(CCC2CC(NC(CNC(C3C(C)C3)=O)=O)C2)=O)CN2CCCC1C2 c1(CCC)ccccc1C(=O)NCC(C)NC(C1(C(F)(F)F)CC(O)C1)=O C1(c2n(CC)nnn2)(NCCc2cn(C)nn2)COCCOC1 N1(C(C2OCCC(C)C2)=O)CC(C(=O)NC(CCO)C2CCC2)CC1(C)C N1(C(CCCOC(C)=O)=O)C2CCC1CN(C(=O)C(F)CC1CCCCC1)C2 c1(N2C(CNC(C(C)NC(c3ccoc3)=O)=O)C(C)CC2)ccc(C#N)nn1 N1(C(c2cc(C)cc(Br)c2)C(=O)NC)Cc2ccccc2C(CO)C1 C(=O)(C(C)CC(C)(C)C)NC1CC(NC(CCCN(C(=O)OCC)C)=O)C1 C(C)(CCCCNC(c1cncc(C(F)(F)F)c1)=O)NC(C1CC(C)C1)=O C1(NC(CCCC2C(C)C2)=O)CN(C(=O)Cn2cc(C(F)(F)F)nn2)CC1C c1(C(N2CCC(CC)(NC(=O)C3=CCCC3)CC2)=O)cccc2ncsc12 c1(C(=O)NCC(CC=C)NC(C2CC(CCO)C2)=O)c(C2CC2)nc2sccn12 N1(C(c2cccc(N)c2)=O)CCCCC(NC(C2CCCC3CC23)=O)C1 N1(C(C2CCC(C(=O)OC)C2)=O)CCC(NC(=O)CCNC(=O)C=CCl)C1(C)C C1(CCC)CCCCCCN1C(=O)C(C)C(C)C C1(N(C)C(C2CCC(=O)C2)=O)CCCN(C(c2cn(C)c(C(F)F)n2)=O)C1 O=C(CC(C(F)(F)F)NC(C1CCS1(=O)=O)=O)NCCN1CC=CC1 c1(C(=O)NCC(CNC(CCC#CC)=O)(C)O)nccc(OC)c1C N1(C(c2nc(C)nn2C)=O)CCC(CNC(=O)Cn2nnnc2C)C(F)(F)CC1 C12(C(=O)NCC3CCC(NC(CCCSC)=O)CC3)CC3CC(C(=O)N1)C2C3 c1(-c2cnc(OC)c(F)c2)c(C(=O)NCc2cc(Br)cs2)nn2c1CCCC2 N1(c2scc(C(c3ccccc3)CNC(c3cccs3)=O)n2)CCS(=O)(=O)CC1 c1(C(N2C(C)CN(C(C3CC4CC3C3CC43)=O)CC2)=O)ccc2ncn(C)c2n1 C12CCCN(C1)C2=O.c1(CNC(C)=O)ccc(OC(C)C=O)cc1.CCN C1(C(=O)NCC2CCN(C(c3cc(C)[nH]n3)=O)C23CC3)CCCC(C)(C)CC1 C1(C#N)(C(=O)NCC(CC=C)NC(C2(CO)CC2)=O)CC12CCOCC2 c1(C(N2CCCC(C)(CCO)C2)C(=O)NCCCC)ccc(Cl)c2c1CCC2 CN=c1nc(N2CCOCC2C2CCCO2)[nH]c(=NC(C)c2cnc[nH]2)[nH]1 c1(C(=O)NC(C(C)NC(c2cc(OC)no2)=O)C)coc2ccc(F)cc12 N1(CC)CCCC(C(=O)NCC(F)CNC(=O)CSC(F)F)C1 CCCC(C)CC(=O)N(C)CC1CN(C(=O)C(c2ccccc2F)(F)F)CCO1 n1(CC(N2C3C(NC(C(CC)C(C)C)=O)CC(C3)C2)=O)ccc(=O)c([N+](=O)[O-])c1 CC1CCC(C)N1CC(=O)NCCC1(NC(C2CC=CC2)=O)CC1 C1(NC(=O)Cn2cncn2)CN(C(=O)Cc2cnc(C3CC3)[nH]2)C2(CCCC2)C1 Cc1cc(N2CC3C(NC(=O)Nc4ccc(Cl)cc4Cl)C3C2)n2nc(C)cc2n1 C(C(C)C#N)SCC.C1(C(CN(CC)CC)=O)CC(O)C1 C1(NC(c2c(CC)nns2)=O)CCCC2CN(C(c3sccc3C3CC3)=O)CC12 Cc1nnc2n1CC(C(=O)NCCOCCN(C)Cc1sccc1Br)CC2 c1(OC)cc(NC(c2cnn(C)c2F)c2nnnn2C(C)(C)C)n(C)n1 CCC(C)C(CNC(=O)CCC1CCCN1C(=O)CC1CC(O)C1(C)C)CO C12(C(N3CC(C(C)(C)O)(CNC(CC=C)=O)C3)=O)CC(C1)Oc1ccccc12 N1(C(c2nc(C)nn2C)=O)CCC2CCCNC2C1 C1(NC(=O)Cc2cncnc2)CN(C(c2cccc3[nH]ncc23)=O)C2CCCC12 CC1C=C(C(=O)N(CCNC(C2CCCOCC2)=O)C2CC2)CC1 C(=O)(CCC(C)C)NC(C1CCCN(Cc2ccccc2-n2cccn2)C1)C C(C(=O)NCCC#N)(C1=CCSC1)N(C(C(C)SC)C)C C1(CNC(C23CC(C(C)(C)C)(C2)C3)=O)CCCN(C(C2CCCC2CF)=O)C1 C1(C)(NC(c2c(CC)[nH]cc2)=O)CCCN(C(=O)CCS(=O)(=O)N(C)C)C1 C1(O)(CNC(C(C)(c2cccs2)SC)=O)CCN(C(c2ccc(C)n2C)=O)C1 C1(CNC(CC(C)c2ccco2)=O)CCC(CNC(C2CC(C)CCO2)=O)CC1 C1(C(N2CCN(CC(=O)NCC3CNC(=O)O3)CC2)=O)CCC(F)(F)CC1 Cc1cc(N2CCCC(C(C)(C)CN(C)C)C2)nc(=NCc2cnc(C)[nH]2)[nH]1 C(=O)(C1=CC2(CCN(C(=O)OC(C)(C)C)C2)C1)N(CC(C)O)C(C)C C(=O)(C(C(C)(C)C)NC(C1(C)OCCO1)C(C)C)OCC CC1(C)Cc2ccc(C(=O)NC3CN(C(C4(C5(C)OCCO5)CC4)=O)C3)cc2C1 C(=O)(CC(C)C(C)(C)NC(C1CC(F)C(=O)N1)=O)NC(CCC)C1CCC1 N1(C(C=CC)=O)CCCC(C)(CNC(c2ccc(-c3ccccc3)o2)=O)C1 c1(CC(=O)NCCNC(=O)C2=CCCC2)ccc(-n2cccc2)cc1 n1(CC)ncc2cc(C(N3CCCC3CNC(=O)C(F)=CC3CC3)=O)c(C)nc12 S(=O)(=O)(c1cccs1)NC(C)C(N1CCC2C(NC(=O)CN(C)C3CC3)CC12)=O C(CC(C(=O)N1CC(F)(C(=O)NCC2(F)CCOCC2)C1)OC)OC C(C)(CNC(=O)C(C(C)C)N1CCCC1=O)(CC(C)C)NC(CSCC=C)=O C1(O)(C(C)NC(=O)C(C)c2cccs2)CCN(C(=O)COCC2CC2)C1 c1(C(=O)NC(C(C(C)C)NC(=O)C=Cc2cn(C)nn2)C)cc(Cl)c(Cl)n1C c1(C2(C(c3nnnn3C3CCOC3)NCC3=CCC3)CC2)cccc(C(N)=O)c1 C=CC(C)(CC)C(=O)NCCOCCCNC(=O)CCC(CC)c1ccccc1 CCC(CNC(=O)CCCOc1ccc(F)cc1)N=c1[nH]c(Cl)c(C#N)s1 c1(C(=O)NC2CN(C(CC(C=C)C)=O)CC23CCC3)cc2cccnc2cc1F N1(C(CC(CC)(C)C)=O)CC2CC(NC(=O)CC3(O)CCOC3)C(C2)C1 C(=O)(C1=Cc2ccccc2C1)NC1CC2N(C(C3C(=C)C3)=O)C(CCC2)C1 c1(C(=O)NC2C(CNC(c3ccc(Cn4cccn4)o3)=O)C2)ncccc1F c1(-c2nc(CC(CC)C)nn2C(C)C(C)C)sc2ccccc2c1C CC(C)C(O)C(C)C(=O)NC(C1CN(C(c2c[nH]nc2-c2cnn(C)c2)=O)C1)C C1(C2CCN(C(=O)C=C(CC)CC)CC2)(NC(C(CC)OCC)=O)CC1 N1(C(C(N2CCOCC2)C)=O)CC(=O)CC1C(=O)Nc1ccc(O)cc1 N1(C(C(C)=C(CC)C)=O)CCC(CNC(=O)C(c2cccnc2F)(C)C)(OC)C1 C1(C(N2CCCC(CCC=C)C2)=O)CCN(C(=O)C(C2CCCCC2)=O)C(C)C1 CC1CCC(C)N1C(C)C(=O)N(C)CCNC(=O)Cc1ccc(NS(C)(=O)=O)s1 N1(C(C(C)NC(=O)NC)=O)CCCCC(CNC(c2coc(Br)c2)=O)C1 C(=O)(CC(C)CNC(=O)CN1CCC(F)CC1)N(C(C(CC)C)C)C1CC1 c1(COC)ncc(C(N2CC3CC2CC3NC(=O)OC(C)(C)C)=O)c(=N)[nH]1 C1(NC(C2CC2C(F)(F)F)=O)CC2CCC(C1)N2C(c1nc(Cl)sc1Cl)=O c1(C(=O)NCCC(CNC(C2(C(N(C)C)=O)CC2)=O)O)coc2c1CCCC2 C(C)(C(O)C(F)F)NC(CC1N(C(c2ccc(C)[nH]2)=O)CCC1)=O n1(CC(=O)N(C)CCOc2ccccc2F)ncc2cc(Br)cnc12 c1(C(=O)NC2(CC=C)CCOC2)c(C(F)(F)F)coc1C(=O)OCC C1(C(=O)NC(C=C)C2CCC2)C(C2CC2)CCN1C(c1cn(C)c(C)n1)=O N1(C(c2c(C)nc(O)cc2)=O)CC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C(C2)C1 N1(CCNC(=O)C=Cc2c[nH]cn2)CCC(NC(=O)Cn2cncn2)CC1 c1(OC(=O)NCC(c2ccccc2C)O)ccc(Cl)cc1CN(CCOC)C N1(C(C2CN(C(c3c(CC)ncnc3)=O)CC2F)=O)CC2(C1)CN(C)CCO2 c1(C(=O)NC(C)CNC(C2(Cc3ccc(O)cc3)CC2)=O)cc2cn[nH]c2cn1 C1(OC)CN(C(=O)CN2CC=CC2)CC1NC(=O)C=C1CCSCC1 Cc1[nH]c(CN2CCC(C)(CNC(=O)C(F)C(F)(F)F)CC2)c(C)c1C(=O)O N1(C(C(C)C)=O)CCC(n2cc(CNC(C3(C)C=CCC3)=O)nn2)C1 c1(C(C)NC(c2ncoc2CNC(C2CC2C2CC2)=O)=O)ccccc1O C(=O)(C(CCSC)NC(=O)C(C)=CCC)N(C(C#C)C)CCCC C(=O)(C1COc2ccccc21)NC1CN(C(C2C(C)C(=O)C2)=O)C2C1CCC2 C=C(Cl)CC(C(=O)N1CCN(C(C)C)C(=O)C1)NC(=O)CN1CCCCC1=O Cc1[nH]c(C(N2CC=C(CNC(C3(C)CC(O)CN3C)=O)CC2)=O)c(C)c1C Cc1cccc(C(c2nc(C)cs2)NCc2nnnn2C2CC(F)(F)C2)c1 N1(C(C23CC(C#N)(C2)C3)=O)CCC2CC2(C(=O)NC2CN3CCC2CC3)CC1 C1(CNC(C(C)Cn2ccnc2)=O)CN(C(c2ccnn(C)c2=O)=O)C(C)(C)C1 C(=O)(CCCC(=O)NCCN(C(C1SC2C=CC1C2)=O)CC1CC1)N(C)C N1(C(C(C(C)NC(c2ccnnc2O)=O)C)=O)CC2(CCOCC2)C1 c1(C(=O)NCC2(CNC(C(CC)=CC)=O)CC2)cnc(OC)c(C)c1 c1(OCC)ccccc1OCCCN(C)Cc1cccc(COC)n1 C1(C#C)(C(N(C(C#C)C2CCC2)C)=O)CCN(C(c2n[nH]cc2Cl)=O)C1 c1(C(N(CC(CNC(CSC)=O)O)C)=O)cccc2ccoc12 C1(CNC(C2(F)C(C)C2)=O)CC(C)(C)CN1C(C1CCC(O)C1)=O C1(CNC(CCC(CC)C)=O)COC(C)(C)CN1C(c1cccc(C(C)C)n1)=O C(c1ncc(C)[nH]1)=CC(=O)NC(CC=C)CNC(=O)CSCCCC O=C(N=c1cnn(CC(F)F)[nH]1)C1CCOC(C2CCOC2)C1 c1(SC)cnn(C)c1C(N1CCC(O)(CN(C)C(C2CCCCC2)=O)C1)=O n1(CC)nccc1C1OCCC1C(=O)NC(c1nnnn1C)CC1CCCC1O c1(OC)ccc(C2CC2)c(C(N2CCC(NC(=O)C(C)(C)N(C)C)CC2)=O)c1 C1(NC(C2CC(C)C2)=O)CCCCC12CCN(C(=O)C1CCCc3ncnn31)C2 N1(C(CCC(C)OCC)=O)CCC2(CCC(NC(c3ncc[nH]c3=O)=O)C2)C1 c1(OC)ccc(C(F)F)cc1C(=O)NC(C)CCNC(=O)C=C(C)C(F)F CC(C)C(CCNC(c1cc[n+]([O-])cc1)=O)NC(c1cocc1Br)=O Cc1cccc(COC(c2cccc(CC3CCCCC3)c2)=O)n1 c1(C(N2CC(CC)N(C(=O)CC(C)(C)CC)CC2)=O)cn2c(n1)COCC2 N(C1CCCn2ccnc21)C(C(CC#CC)NC(c1coc(C2CC2)n1)=O)=O C1(NC(c2n3cc(C)sc3nc2)=O)CN(C(C2CCO2)=O)CC1S(C)(=O)=O CN1CCC(F)(CNC(C2CC(C(F)(F)F)CN2C(=O)C(C)(Cl)Cl)=O)C1 C(=O)(C(=O)CCC(C)C)NCC(CC(=O)NC(CC)CC)O Cc1cccc(C)c1NCC(N1CC2CC2(NC(=O)C=CC(F)(F)F)C1)=O C12(C(N3CCN(C(CC(CC)OC)=O)CC3CO)=O)CC3CC(C(=O)N1)C2C3 N1(C(CC(=O)O)=O)CC2C(NC(c3nc[nH]n3)=O)C2C1 N1(C(C(CC)COC)=O)CC(C)(C)OCC1C(=O)N(CCCSC)C C(=O)(C(O)CC(F)(F)F)NCC1(CN(C)C)CC1.CN1CCC2(C1)C(=O)N2 N1(C(C(c2cnn(C)c2Br)C)=O)CC(c2ccccc2)(CO)C(c2ccccc2)C1 N1(C(c2cn(C(COC)C)nc2C)=O)CCC(F)C(NC(c2sccc2F)=O)C1 C1(CNC(c2cc(CCC)[nH]n2)=O)CCCN(C(=O)OC(C)(C)C)CC1 CC(C)CCC(O)C(=O)N1CC(O)CC1(C)C(=O)NCC(C)(C)C(N)=O CC(C(=O)NC(=O)CCc1nc(-c2ccoc2)no1)C(F)F c1(CCC)onc(C)c1NC(C1C2CN(C(=O)CC(=O)C3CCCC3)CC12)=O CC(C)(CC(=O)N1CCCC12CCN(C(C13CCCC1C3(F)F)=O)C2)CC(F)F Cc1ccc([N+](=O)[O-])c(C(N2CC(NC(=O)C(F)C(C)(C)O)C(O)C2)=O)c1 c1(CCCC)ccc(C(=O)NCC(C2CCOC2)NC(c2cccnc2S)=O)cc1 C(C(O)CN(C)OC)n1cc(-c2c(C(=O)OC)cccc2)nn1 C1(CCC)(NC(=O)C2=CCOC2)CCN(C(=O)C=C2CCCC2)CC1 c1(C(N2CCCC(C(C)(O)CNC(=O)C3=COCC3)C2)=O)cnc2[nH]ncc2c1 c1(OC)ccc(C(=O)NC2(C3CCCCN3C(c3cnns3)=O)CC2)cc1 N(C(=NCCCOCC)NCc1cc(C)nc(C)c1)CC(C=C)C c1(C(=O)NCC2C(C)(C)CN(C(c3ccccc3)=O)C2)cc(F)c(N)c(F)c1 CC1(C)C(C(=O)NCC2CC(NC(Cc3ccc(NC(N)=O)cc3)=O)C2)C1(C)C Cc1ccc(C)c(C(=O)NC(C)C(C(C)C)NC(=O)CN2CC(=O)N(C)C2=O)c1 CC(CC1=CCCCC1)NC(C1COCCC1NC(=O)C=C1CCOCC1)=O c1(C(N2CCCCC2CC(N2CC3C(C(=O)O)C3C2)=O)=O)ccc(O)cc1 c1(NC(C2C3(CCN(S(CC#N)(=O)=O)C3)C2)=O)cccc2nc(O)ccc12 N1(C(C2CC(N(C(c3c(C)csc3)=O)C)C2)=O)CCOC(C2CC2)C1 C1(CC)(CC)CN(C(C2CC(C)(NC(=O)C=CCN3CCC3)C2)=O)C1 Cc1cc(C(C(=O)NCc2cccs2)N(C)C(C2CC2)C2CC2)ccc1I N1(C(COc2cccc(C)c2)=O)CCN(C(=O)C2CC2)CC1CC(F)F C12(NC(c3nccc(C)c3)=O)CCOCC1CN(C(c1ccc(C(F)F)s1)=O)C2 CC(C(=O)OC(C)(C)C)C(C)C(C)(C)C.C12CC3(CCC(O3)CNC(=O)OC1)C2 C1(NC(CC2ON=C(CC)C2)=O)(CNC(C2(C3CCC3)CC2)=O)CCCCCC1 O=C(C1=NN(CCO)C(=O)CC1)NC1COC2(CCN(C(=O)C3=CCOC3)C2)C1 Cc1cccc(C2CCCCC2CNC(=O)NC2(n3cccn3)CC2)c1 c1(C(=O)NCC(CC)N(C)C(c2occc2CN(C)C)=O)[nH]cc(C(C)=O)c1C c1(C(N(CC(CC)NC(C2CCCCC2O)=O)C)=O)coc(S(N)(=O)=O)c1 CCCC(C(=O)NC1CCN(C(=O)C(C)N(C)C(=O)OC(C)(C)C)C1)S(N)(=O)=O Cc1noc(C)c1CC(c1nc(-c2ccn(C)n2)nn1CC1CCCCO1)C C(=O)(N=c1cnc(Br)c(Cl)[nH]1)C1N(Cc2c(C(=O)OCC)[nH]cn2)CCC1 C1(C(=O)NCc2c(C)cccc2)CN(C(=O)C(F)CC2CCOC2)CC(C)(C)C1 c1(C(=O)NC2CC(NC(CC#N)=O)C2)cc(F)c(Br)cc1F c1(C(N(CC(CC)NC(C2CSCCS2)=O)CC)=O)cc2c(=O)[nH]ccn2c1 C(C1CCCN1C(C1CCCCC1O)=O)=CC(=O)NCCc1cc(C)[nH]n1 C(=O)(C(CNC(C1(C#N)CC12CCC2)=O)CC=C)N1CCCC(COCC#C)C1 N1(C(CCC2(C)N=N2)=O)CC2CCCC1C2CNC(C1(C)CCCCCCC1)=O N1(C(C2(C)C(C)OCC2)=O)CC2CCC(NC(=O)COC3CC3)(C2)C1 C(CC(C(=O)N1CCC1CNC(=O)Cc1cccnc1Cl)N(C)C)=C(C)C N1(C(C(C)(N(C(=O)CC2CCOCC2)C)C2CC2)=O)CC2COCC2(C)C1 CC1(C)CCN(C(=O)CCC2CCC(=O)N2)C1CNC(C1CC=CC1)=O C1(CNC(C(CC)O)=O)CN(C(=O)C(c2cncnc2)C)CC1(F)F c1(OC)c(C(=O)NC(C)CC(C)NC(c2cc(C#N)cs2)=O)ccc(Cl)c1C c12cnn(c1C)CCNC(=O)NC2.c1(C(=O)OCC)ncsc1NC1CCCO1 CC1(C)OCCC1CCNC(=O)CCOCCNC(C1CC12CCC2)=O C(CCC)(C(=O)N1CCC(O)(C(C)NC(c2nccnc2C(N)=O)=O)C1)=CCC C=CCC(C(=O)N1CCOCC1CNC(=O)CC1CCCSC1)NC(C)=O S(=O)(=O)(c1ccc(N(C2(CCC(C)C)CC2)C)c(Cl)c1)NCC(C)C c1(C(=O)NCC(C)(C)CNC(c2cnc(C3CC3)s2)=O)cc(F)cc(Cl)c1N N1(CCC#C)CCCC2CN(CCc3csc(C)n3)CCC12 N1(C(C(CCOC)OC)=O)CCC2(CCN(C(c3cc(O)cc(C#N)c3)=O)C2)C1 Cc1cncc(C(=O)NC2CCN(C(c3ccco3)=O)C(C3CC3)C2)c1Cl C1(OC)CN(C(=O)Cn2ccnn2)CC1NC(=O)Cn1cc(C2CCOC2)cn1 c1(C(=O)OC)cnn(C)c1C(=O)NC1CC1NC1(C(N2CCCC2)=O)CC1 N1(C(C(CC)n2ccc(C3CC3)n2)=O)CCCC(CNC(C2(CF)COC2)=O)C1 c1(C(c2nnnn2C2CCCC2)N(CCCCC)CC)cnn(-c2cccnc2)c1 Cc1cc(N2CCC(N(C(=O)CCSC(F)(F)F)C)C2)nc(-c2cccs2)n1 c1(C(=O)NC(C(=O)Nc2cccc(C)c2)C)ccc(F)c(C)c1C c1(C(N(CC(C)(C)NC(C(C(C)SC)O)=O)C)=O)ccc(Br)c(C)n1 CC1CN(C(=O)C=Cc2ccnn2C)CCN1C(=O)CCNC(=O)CO C1(C(=O)NCCCC(C)NC(C2CC(CC)(CC)C2)=O)C(F)(F)C12CCC2 N1(C(C(C2CCCN(C(=O)CC3CCC(=O)C3)C2)(C)C)=O)CCOCC2(CC2)C1 C(=O)(C1=C(C)CCOC1)NCC(CCCC)NC(c1cscc1Cl)=O CN1CC2CN(C(C3(CNC(=O)CCc4csnn4)CCCC3)=O)CC2C1 C=C=CC(C)C(=O)NCC(O)CNC(=O)C(C1CCCN(C)C1)(C)C C1(C)(CCC)CCN(C(C2(NC(=O)CC3C=NN(C)C3=O)CC2C)=O)C1 C1(O)(C(N)=O)CN(C(=O)NCc2nc(NC3CCOC3)co2)C1 N1(C(C(CC=CC)NC(C2(C#N)CCOCC2)=O)=O)CC2COC(=O)C2C1 N1(C(c2c(C)ocn2)=O)CC(CNC(=O)C=Cc2ncc[nH]2)OC2CCCC12 C1(NC(c2c(CC)cco2)=O)C2CC1N(C(c1ncc(Cl)cc1F)=O)C2C C(c1c(C)nn(C)c1Cl)=CC(=O)NCC(C)NC(CCc1ccc(C)nc1)=O C(=O)(CC(CC(N)=O)CC(C)C)NCC1(C)OCCN(C(c2cc(CC)[nH]n2)=O)C1 c1(CC(N2CC(O)CCC(NC(=O)COCCF)C2)=O)ccc2nc[nH]c2c1 CC(C(=O)N1CCC(C)(CC(=O)NC(C)C(=O)NO)C1)S(C)(=O)=O c1(CN(C2(C)CCC2)C(C2CC=CCC2)C(=O)NCCCF)ccccc1.CC=O C1(C(N(CC(C2CCCC2)O)C)=O)CCOCC1NC(=O)CC1CCCC12CC2 c1(NC(C2C(NC(c3ccn(C)n3)=O)CC2)=O)ccc2cnn(C)c2c1 c1(C(=O)NC2CC(CNC(C3(CC=C)CCC3)=O)C2)ncoc1C c1(CCCC(=O)N(CC(CNC(C(C)CF)=O)(C)C)C)c[nH]c2ccccc12 C#Cc1cccc(N(C(=O)C(C)C(C)NC(c2cccc(OC)n2)=O)C)c1 N1(Cc2c(OC)c(C)ccc2)CCC2(CCCC2C(N2CCCCC2CO)=O)C1 C=CC(CC)CC(=O)N1CC2CC1CN2C(C1CC2(C1)CC2F)=O Cc1cc(C(=O)NCC(CNC(=O)COc2c(C)nn(C)c2C)CO)c(C)cn1 N1(C(C(CCCC)NC(C2CCC3(CC3)C2)=O)=O)CC2CC(C1)C2(C)C N1(C(=O)C(F)F)CC2CCN(Cc3ccc(-n4ccnc4)c(Br)c3)CC2C1 C1(C(=O)NCC(C2CCC2)OC)CCN(C(=O)c2ccc(C)nc2)O1 N1(C(C2(C)CC=CC2)=O)CCC(C)(CNC(=O)Cn2cnnn2)C1 c1(OCC)c(OC)cc(C(=O)NC2(CO)CN(C(c3conc3C)=O)C2)cc1Cl C1(CNC(c2nc(-c3c(OC)cc(OC)cc3)sc2)=O)Cc2ccccc2O1 N1(C(C)C)CCN(CCC(=O)NCC(=O)CC2CCOC2)CC1 N1(C(C2ON=C(C)C2C)=O)CCC2(CC1)CN(C(=O)CC(C)F)C2 N1(C(C(C)C2CCC2)=O)CC(F)CC1CNC(c1ncccc1C(F)(F)F)=O c1(C(=O)NCC(CNC(c2coc(C(F)(F)F)c2)=O)OC)ccc2cncn2c1 C1(C(=O)NCCC(=O)OCC)CCC(C)N1Cc1sccc1C c1(CNC(C(C2CCC2)OCC)=O)ccc(C(=O)N(CCCN=[N+]=[N-])C)nc1 c1(C(C2CC2)NC(CC)=O)cn(C(C)CNC2CC(C(C)C)C2)nn1 c1(C(N)=O)coc(C(N2CCC(OCCNC(C3CC4(CC4)C3)=O)C2)=O)n1 c1(C(N2CC(C)C(NC(c3cc(F)cc(F)c3)=O)C2)=O)ccc2ncncc2c1 N1(C(C)C)CC2CC(NC(c3cnc(Br)cn3)(C)C)C(C2)C1 c1(N(CC#CC)C)nc(NCC(c2nc(C)cs2)C)c2cnn(C)c2n1 N1(C(C(c2c(C)cncc2)C)=O)CCC(NC(=O)CC2CC(=O)C2)C(C)C1 CCC(CC(=O)NCCC1CC(C(N2CC(c3cc[nH]n3)C2)=O)C1)C1CCC1 c1(NCC(N2CC(CNC(C(CCC)CC)=O)OCC2)=O)ccc2c(c1)CCC2 CCC(CC(F)(F)F)NC(=O)CN(CCOC)C(c1ncn(C(C)C)n1)=O C1(CNC(=O)CCc2ccon2)CCCCC1NC(=O)CC1CCC1 c1(CC)c(C(=O)NCC2(NC(C3CC3F)=O)CC2)oc2ccc(Br)cc12 N1(C(C2(SC)CCC2)=O)CCC(CNC(=O)CCC2OCCO2)C(O)C1 C(=O)(C1=C(C)CCOC1)NC(CC#CC)C(=O)N1CCCC(C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NC(C1(O)CN(C(=O)CN2C(=O)CN(C)C2=O)C1)C CC1(CNC(C2CC2F)=O)CCCN1C(c1nc(Cl)c(Cl)s1)=O C(=O)(C1=NOC(CNC(=O)C(N2CCNC2=O)C)C1)NCC1(C)ON=C(C)C1 N1(C(C2C(C(=O)OC)CCO2)=O)CCC(NC(=O)CCCC(N)=O)C(CO)C1 C1(CCNC(C=C(CCC)C)=O)C(C)CCCN1C(c1cnc(C2CC2)s1)=O C1(NC(C=CCN(CC(F)(F)F)C)=O)CC2(CCCN(C(C3CC3(F)F)=O)C2)C1 C1(N(C(CN(CCC)C(c2conc2C)=O)=O)C)CCOCC1C Cc1ccc(NC(C2CCN(C(c3cnsn3)=O)CC2O)=O)c(Br)n1 N1(C(C2C(=C)C2)=O)CCC12CN(C(=O)C(C)(C)CF)C2 CC1CCc2c(Cl)cccc2C1NC1CCc2ccccc2OC1 C12(OCC)CCC(C(N3CCCC(CCNC(=O)Cn4ccnn4)C3)=O)(CC1)C2 c1(OCC)nc(N2CC(C3CCCN(C)C3=O)CC2)ncc1Cl c1(C(N2CC(N(C(C(OC)OC)=O)C)C2)=O)c(O)nnc(C)c1C N1(C(C=CCC)=O)CCOC(C)(CNC(=O)Cn2nc(C)c(Br)c2C)C1 c1(NC2CCN(C(N3CCc4nc[nH]c4C3)=O)CC2)ccc2c(Cl)csc2c1 CC(CN=C(NCC1CCCN1C)NCC(c1ccc(Cl)cc1)(F)F)C(F)F Cc1nc2c(o1)CCCC2CC(=O)NCCN(C(=O)CC1CC(=O)NC1=O)C N1(C(C=CC(C)=O)=O)CCC(C)C(CNC(c2ncccc2C2CC2)=O)C1 C1(C(=O)NC2CCC(CC(=O)NCc3c(C)ccnc3)C2)CC(C)CC(=O)N1 C12(NC(CSCCCC#N)=O)CN(C(c3ccccc3)=O)CC1CS(=O)(=O)C2 c1(OC)ccc(SC(C2CCC2C)C)c(OC(=O)C(C)N)c1.OC CCCCCC(C)CC(=O)NC(C)(C)CC(=O)NC(C)CCC=C(C)C C1(CNC(COC)(C(C)C)c2nnnn2C2CCC2)CC(C2CC2)=NO1 c1(NC(=O)NC(CC=C)C(=O)OC)nc(OC(C)C)cc(C)n1 C(C1=CCN(C(c2cc(Cl)cc(Cl)c2)=O)CC1)NC(c1c(CSC)nn(C)c1)=O c1(OC)c(CNC(=O)NN(C)Cc2ccc(NCC3CC3)cc2)cccc1F C1(CCOC)CN(C(C2CC=CCC2)=O)CCN1C(=O)COCc1cc(C)on1 c1(C(N(CCNC(COCCC#C)=O)C)=O)cc2nc[nH]c2cc1N c1(N(C)C)ccc(C(=O)NCCc2c[nH]c3cnccc23)cc1[N+](=O)[O-] c1(C(N2CCC(C)C2CNC(c2nn(C)cc2Cl)=O)=O)ccc(F)c(C#N)c1 N1(C(=O)CCC=Cc2ccccc2)CC2C3CCC(O3)C2C1 N1(C(C(C(C)C)SC)=O)CCC2CCN(C(c3cncc(N(C)C)n3)=O)CC12 N#Cc1cc(C(=O)NC2CN(C(c3cnoc3C3CC3)=O)CCC2F)cc(O)c1 c1(OCC(=O)NCC(C)NC(Cc2cc(C)[nH]n2)=O)ccc(Br)c(C)c1 N1(C(C2C(CC(C)C)C2)=O)CCCC(O)(CN(C)C(c2nnc(S)n2C)=O)C1 CCCC(CCCNC(=O)Cc1cnn(C(C)C)c1)NC(=O)CNc1cccs1 C1(C(=O)NC(C2CCCC2)CNC(c2coc(Br)n2)=O)(COC)CCOC1 C1(=O)CS(=O)(=O)N(C(C(C(CC=CCC)=O)CC)=O)C(C)C(CO)N1 CN=C(NCCC1CCCS1(=O)=O)N1CCC(n2ccc(C)n2)CC1 S(=O)(=O)(CCCC(=O)NCC1CCCC1NC(=O)C(C)(C)C1CC1)N(C)C CC1CCN(CC(N2CC(NC(=O)CC3(C(F)F)CC3)C(C)C2)=O)CC1 C1(C(N(C2CCN(C(c3sc(CC)c(C)c3)=O)C2)CC)=O)Cc2cccnc2C1 C1(NC(=O)CCc2ccccc2Cl)CC2CC1CN(C(c1n[nH]cc1Cl)=O)C2 CC1(O)CCC(C(=O)NCC(O)CNC(=O)CC2CC(F)C2)CC1 CC(C)(CC(=O)N1CCCC1CCNC(C1CC1C(F)(F)F)=O)CC(F)F c1(CC(=O)N(CCCNC(CNC(C)=O)=O)C(C)C)c(F)cncc1Cl c1(CC)ncc(C(=O)N(CC(C)N(CC(=O)NCC(C)C)CCOC)C)o1 c1(CNC(C2CN(Cc3ccc(N4CCOCC4)cc3)C2)=O)cc(I)ccc1O CC1CCC(NC(=O)C(C)(C)Cc2ccc(O)cc2)CN1C(c1cnsn1)=O N1(C(CCNC(=O)NC)=O)CCC2CCC12CNC(=O)CN1CCCCS1(=O)=O c1(OC)nccc(N(C(=O)CCC2CCCNC2)Cc2ccc(C(=O)OC)nc2)n1 N1(C(CCC2N(C)CCCC2)=O)CCC(NC(C2(CC(F)F)CC2)=O)C(C)(C)C1 CC1CC(C)N(CC(CCl)N(C(=O)C(C)(C)C2CCCCO2)CC)c2ccccc21 N1(C(C2(C(=O)OC)CC2)=O)CCC(NC(=O)CC2COCC(C)(C)O2)CC(O)C1 c1(C(N(CCNC(CCNC(C)=O)=O)C2CC2)=O)cc(C#N)no1 CCS(=O)(=O)CC(=O)NC1CCN(C(c2cncc(C(C)(C)C)c2)=O)C1C1CC1 C(C(COC)C(C)C)NC(C1C(NC(C(CC)C)=O)CCO1)=O c1(CO)ccc(Br)nc1Cl.C12(CCN(Cc3ccccc3)C1)C(=O)N2 C1(C(=O)NC(C2CCCN2C(c2nn(C)cc2N)=O)C)CCC2(CCOCC2)C1 C(C)(C)(C(=O)NC(C)CC(C)NC(=O)Cn1ncnn1)OC c1(NC(c2ncncc2-c2cccc(F)n2)=O)cc(Br)c(F)cc1F C1(NC(C2CCN(C)C2=O)=O)CCCC12CN(C(=O)C(c1ccc(F)cc1)O)C2 c1(C(C)C)nc(NCc2nnnn2C)cc(N(CCCCCC(C)C)C)n1 CCCCC(F)C(=O)Nc1cc(C2CCCN(C(=O)OC(C)(C)C)C2)nn1C CN1CC(C)(C)CC1C(=O)NCC1(C(N)=O)CN(C(C2(C)CNC(=O)C2)=O)C1 N1(C(CCCCCNC(C)=O)=O)CCC2CCN(C(=O)C=Cc3cnc[nH]3)C2C1 C1(C(=O)NCCCCc2cn(C3CCCC3O)nn2)Cc2ccccc2CN1 c1(CN2CCCC(C)C2C(=O)O)ccc2c(c1)OCC(=O)N2 c1(C(=O)NC2C3CN(C(c4ccc(SC)s4)=O)C2C3)cc2cccnn2c1 c1(NC(C2CCN(C(CC3N(CC)CCC3)=O)C2C)=O)ccc(Cl)c(C)c1 N1(C(Cc2n(C(C)C)cnn2)=O)CC2(CCC(CNC(c3coc(Br)c3)=O)O2)C1 N1(C(CC(C(=O)OC)C)=O)CCC(C2CN(C(C3(CF)CC3)=O)C2)CC1 c1(CNC(c2cnn(-n3cc(C4CC45CC5)nn3)c2)=O)ccoc1C1CC1 C1(CNCCCc2cccc(C(F)(F)F)c2)Cc2ccccc2C1 Cc1cc(C(N2CC(CCNC(C3CS(=O)C3)=O)C2)=O)ncc1Cl n1(CC(C)NC(=O)N(C)CCc2ccccc2)cc(C2CCN(C)C2)nn1 C1(C2CN(C(C3CC3C3CCC3)=O)C2)(NC(C(C)=C(CC)C)=O)CC1 c1(OC)cccc(CNc2ccc(-c3cc(C)cc(O)c3)nc2)c1[N+](=O)[O-] c1(OCC(=O)NCC2(F)CN(C(c3nc(C)oc3)=O)C2)ccc(C)c(C)c1 C1(CNC(C)=O)CCN(CC2CSCCS2)CC1 C1(C(=O)NCCN(C(=O)CCC=C(C)Cc2ccco2)CC)CCOC1C1CC1 C(C#CC(=O)NCc1cccnn1)NC(CCOC(C)C)=O C=CC(CCC)CC(=O)NCCCCNC(=O)CC1CCS(=O)(=O)C1 c1(C(=O)NCC2(CNC(C3C(C=C)C3)=O)CCC2)cc(N)ccc1Br CN1CCCC1C=CC(=O)NC(CCOCCO)C(=O)Nc1cnn(CCO)c1 c1(SC)nc(NC2CCC(C(=O)Nc3cccnc3CO)C2)ncc1F C(C#Cc1ccc(F)cc1)N1CCN(C2CCN(C(C3(C)COC3)=O)C2)CC1 c1(CC(N2CC(NC(C(CCOC)C)=O)(COC)C2)=O)c(F)cncc1Cl C12(CNC(c3cnc(C(C)OCC)s3)=O)CC1CN(C(=O)CCC(C)C)C2 c1(C(CCN(C(=O)C(=O)NCc2cnsc2)C)O)ccccc1 N1(CCCC(C)C)CCC2CN(C(=O)OC(C)(C)C)C2C1 S(=O)(=O)(c1cccs1)NCCNC(=NC)NC(c1cccnc1)C N1(C(CCN(CCC(C)(C)C)C)=O)CCC(C)(NC(=O)C(O)C2CCCC2)C1 C1(CC(=O)NC2(CCNC(=O)CCOC3CC3)CCCC2)CCCC12CC2 N1(C(C(C2CCOCC2)OC)=O)CCC(O)(CNC(c2nocc2Br)=O)CC1 N(C(=NCCF)N1CCC(C(C)C)C1)C(C#C)CC1CC1 C1(C(=O)NCC2CC(F)(F)CN2C(=O)Cc2cccs2)CCc2nnnn2CC1 O=C1NCCCN1CC(N1CC2C(C(=O)NC3CCCNC3=O)C2C1)=O N1(C(c2c(C)n[nH]c2)=O)CC2(C1)SCCC2NC(=O)C(CC(F)F)C1CCC1 N1(c2n(CC=C)c(CC(=C)Br)nn2)CC2CCCCCCC12 C#CCCCCC(=O)NCC(C)(C)NC(=O)CCc1c(F)cccc1Cl C1(CNC(C2CC(CC)C2)=O)CCCN1C(=O)C(F)C1CC1 c1(C(N2CCOC(CCNC(C3(CCF)CCOCC3)=O)C2)=O)ncccc1O C1(NC(Cc2nc(NC=O)sc2)=O)CCCC12CN(C(C13COCC1C3(F)F)=O)C2 C1(NC(C(F)SC)=O)CCN(C(c2ccc(NC(=O)OC(C)C)cc2)=O)C1(C)C CC(O)CN(C)C(=O)OC1C(OOC(C)(C)C)C1.C1(=O)CN1CC1CC1 C1(NC(c2cc(C)c(F)cn2)=O)CN(C(=O)Cc2cnc[nH]2)CC(F)(F)C1 Cn1cc(S(N)(=O)=O)cc1C(=O)NC1CCCN(C(=O)COC2CCOC2)C1 C(CC(CC)C(=O)NC1CCC(CC(=O)NC(CO)C(F)(F)F)C1)=CC CC1(C(N2CCC(C(F)F)C2)=O)CCN(C(=O)C=Cc2ccncn2)C1 C1(C(N)=O)(NC)CCN(C(=O)C(c2cccc(Cl)c2)N)CC1 CC1(NC(C2CC23CC3)=O)CCCN(C(c2sc(-c3ccccc3)cc2N)=O)C1 c1(C(N(CC(C)CNC(=O)C(F)(F)c2cscn2)C)=O)cccn(CCF)c1=O C=CCCCCCC(=O)N1CCC(C(=O)NC(C)(C)C(O)CO)C1 CCCCC(CNC(=O)C(C)(O)CSC)NC(c1ccc(C(N)=O)nc1)=O C(c1ccc([N+](=O)[O-])cc1)=CC(=O)OC.c12cc(C#N)ccc1NC2=O c1(C(N2CC(CC#C)OCC2)=O)ncnc2c1c(Br)cn2C c1(CCC(=O)NCC(C)NC(c2ccc(C3CCCO3)[nH]2)=O)ccc(Br)cn1 C1(C(=O)NCCN(C(=O)CCc2cccc(C)c2)CC)CCCOC1C n1(C(C)C)cc(C(=O)NC(C2CCCCC2)CNC(=O)CNC=O)nn1 c1(C(=O)NCCN(CCOC)C(C2CC2C2CCCC2)=O)ccn2cncc2c1 C(=O)(C(C)N=c1cc[nH]cc1)NC(CCNC(CCN(CC)CC)=O)(C)C C1(CNC(c2c(C)nncc2)=O)CC2CCCC2N1C(=O)CCc1nccs1 C1(C2CN(C(C3CC3F)=O)C2)(NC(CNc2nccc(OC)n2)=O)CC1 c1(CC(=O)NCCCCC(C)NC(C2C(C)C2(F)F)=O)ccc(S(C)(=O)=O)cc1 N1(C(c2cc(C)no2)=O)CC2CCC1CN(C(=O)COC(C)(C)C)C2 N1(C(CCC(C)N(C)C)=O)C2CCC1CN(C(=O)CN1CC(=O)NC1=O)C2 Cc1ccc(C(=O)N(C)CCOCCNC(=O)C(C)C(C)(F)F)c2c1CCCN2 C1(CNC(c2[nH]cc(C#N)c2)=O)CC12CCN(C(=O)CCCN1CCCC1)CC2 C1(C(=O)NCc2cnccn2)CCC2CCCCN12 N1(C(C(C(C)C)OCC)=O)CCN(c2cccc(C)c2)C(=O)C1 c1(C(N(C)C)=O)cn(CC(=O)N(CCc2cn(C3CCCC3)nn2)CCO)nn1 n1(CC)nnnc1C(c1ccc(SC)s1)NC(C)C(=O)NCC(C)C c1(C(=O)NC(C(N2C(CCC)COCC2)=O)(C)CO)cc2ncccc2[nH]1 c1(CC)cc(O)ccc1NC(C1CC=CCC1NC(C12CCCC1C2(F)F)=O)=O Cc1cnc(C(=O)NCCC(C)(C)CNC(=O)CC(C)C2CCCO2)c(F)c1 c1(CCC(=O)N(CC(C)NC(C(C)SCC)=O)CC)cc(Cl)no1 N1(C(C2=CC(C)(CC)C2)=O)CC2=C(C1)CN(C(=O)COC1CC=CC1)C2 N1(C(c2nc(CCC)sc2)=O)CCC2CN(C(c3ccn(C(C)C)c3C)=O)CC12 C1(NC(CCCSC)=O)(CO)CCCN(C(=O)COCC(=O)OC(C)(C)C)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CCC2C(C1)CN2C(c1ncc(Cl)cc1F)=O Cc1ccc(O)c(C(=O)NCC(C)NC(C23CC2CCC3(F)F)=O)c1 N1(C(Cc2nc(C)sc2)=O)CC2CC(C1)CN(C(=O)CCC1(C)CC1(F)F)C2 CCCC(C)CCN(C(CC(N)=O)c1ccccc1)C(=O)C(O)c1ccsc1 CCCCC(CC)C(=O)NCCCN(CCCNC(C1NC(=O)OC1(C)C)=O)C C(=O)(CC1OCc2ccccc21)NC(CCOC)C(C)C C1(c2onc(C(c3ccccc3)OC)n2)(CN)CCCC1C c1(NCC(=O)N(C2CCC(NC(=O)C(C)(C)C)C2)C)ccccc1Cl C1(C(=O)NCC2(CNC(C(CSC)OC)=O)CC23CCC3)CCC(C(N)=O)CC1 Cc1cc(CC(=O)NCc2ncoc2CCNC(=O)C(Cl)=CCl)cc(O)n1 c1(OC)cc2ccc(NC(=O)NC3CCCC(F)C3)cc2cc1OC N#Cc1cc(C(=O)NCc2cc(C(=O)NCCCc3ccco3)on2)cs1 N1(C(C(C2CCN(C(C(C)N(C)C)=O)C2)F)=O)CC(=O)NC(=O)C1 C1(C(=O)NCCC2CCN(C(C3(O)CCC3)=O)C2)CCc2ccccc2S1 c1(C(N2CCC(CN(C(C(CC)(CC)CO)=O)C)C2)=O)csc2cc(Cl)cnc12 O=C1CC(C(=O)NCC2(C(=O)NCC3CCOC3)CC=CC2)NC(=O)N1 c1(CN2CCCN(CCC(=O)OC)CC2)ccc(N(C)C)cc1Cl C(=O)(C1=CCCC1C)NCC1CN(C(Cc2nc(COC)sc2)=O)CC1C C1(C(N2CC3C(CNC(CCCC(=O)N(C)C)=O)C3C2)=O)CN2CCC1(C)CC2 CC1CN(C(c2ccnn2C(F)(F)F)=O)CCCN1C(=O)CC1CC1 N1(C(C(C)(C)c2sccc2Cl)=O)CC2CC(C1)C(CO)C2NC(C1CCCS1)=O c1(C(=O)NCC2CC(NC(c3ccn(CC)c(=O)c3)=O)C2)ccc(C#N)nc1O c1(C(=O)NCC2C(C)(C)C(NC(=O)C3=COCCC3)C2)ccc([N+](=O)[O-])cn1 CCC(C)C(O)CC(=O)NC12CC(C(N3CCCN(C(C)=O)CC3C)=O)(C1)C2 C1(NC(C2C(c3c(OC)cccc3)C2)=O)CN(C(=O)CCCF)CC12CC2 c1(OC)nc(=NC2CC(CNC(C3(C)C=CCCC3)=O)C2)[nH]c2[nH]cnc12 C1(C(=O)NC(C2CCOCC2)C#C)CN(C(=O)CC2(C=C)CCC2)CC12CC2 c1(CN=C(N(C)CC2(OC)CCOC2)NC(C)C)nnc2ccc(C)nn12 C(C)(C)(C(=O)NCCCN(C)C(c1cc[nH]c1C1CCC1)=O)OCCC c1(C(=O)NCCCNC(c2c(C)c(Br)ccn2)=O)[nH]nc2ncccc12 N1(C(C(c2[nH]c(=N)sc2)=O)=O)CCCCC(CNC(=O)CCCCCF)C1 C(=O)(CC(C(C)C)NC(c1cc(OC)ncn1)=O)NC(C=C)COC c1(CC(=O)N(CC(C)O)CCNC(c2c(C)csc2)=O)cccc(C(C)C)c1 C1(C(=O)NC(CC)CNC(c2c(Cl)cnn2CC)=O)CCn2nnnc2C1 c1(OC)ccc2nc(C(F)(F)F)[nH]c(=NCC(CO)OC)c2c1 C(=O)(CC(C)C(F)(F)F)NC(CC#CC)C(=O)NCC1(C)CCC(=O)N1C C1(NC(C2(N(C(C=CCCC)=O)C)CCC2)=O)CCC2CC12 C1(OC)CC2CC1CN(C(=O)C(O)CNC(=O)C(C)C(F)F)C2 CCCC(C)CC(=O)N(C(C)CNC(=O)C(CC)n1cncn1)CC S(=O)(=O)(c1ccc(C(C)=O)cc1)N1C(C(=O)Nc2cc(OC)cc(Cl)c2)CCC1 O=C(C1=NOC2(CCC2)C1)N1CCC2CN(C(C3CCC(F)(F)C3O)=O)C2C1 C1(C(C)NC(c2cc3c[nH]cnc-3n2)=O)CCN(C(c2cncn2C)=O)C12CCC2 C1(NC(CC=C)=O)CCC(NC(=O)C(n2ccc(Br)n2)C)C1 C(C(=O)N1CCCO1)NC(C(CC1CCC1)OC)=O CC1(NC(=O)CCc2ncco2)CCN(C(c2c[nH]c(Br)c2)=O)CC1 c1(-n2cc(CCCC)nn2)nc(CSC)nn1CCc1ccc(OC(C)C)nc1 C(=O)(C(COC)CC)N(CC(CN(C(c1nc(CCC)oc1)=O)C)O)C c1(C(N(C)CC2N(C(CCOC)=O)CCOC2)=O)ccc2ncsc2c1 C(CCCC(CO)NC(=O)C(c1ccc(F)cc1)C(=O)OC(C)(C)C)NC(C)=O N1(CC(=O)NCC(c2ccccc2)N(C)C(C2CCC2(F)F)=O)CCCCC1 CC(C)(C(=O)OC(C)(C)C)CCC(=O)NCC1CCCCC1N1CCOCC1 C12CCCC1NC2.c1(C(=O)NCC(C)C)ccc(C(=O)O)s1 N1(C(C2CC3CCC2O3)C(=O)Nc2ccccc2Cl)CCCC2(CC2)C1 N1(C(c2nc(OC)c(C)s2)=O)CC(NC(C2CCCOCC2)=O)CC1(C)C c1(C(=O)NC2(CNC(CC)=O)CCOC2)cc2cc(C)c(Cl)cc2[nH]1 c1(CC(=O)N(C2CC2)Cc2c(OC)cccc2)cc2ccccc2cc1O C(=O)(C(CC(C)C)C(N)=O)NC1(C(N2CCC(CC(=O)OC)C2)=O)CCCCC1 c1(C(=O)NCCN(CCC)C(c2c(C)nn(C)c2C)=O)cccc2occc12 C1(O)(CN(C(=O)NC(c2cccc(Br)c2)C)C)CCCCC1 c1(CCC(=O)NCC(C)N(C(C2CCN(C(CC)=O)C2)=O)C)ccc(N)c(F)c1 c1(C(N2CCC(CN(C(c3cnc(C)s3)=O)C)C2)=O)cc(O)nc2c1CCCN2 Cc1nc(C)c(C(=O)NCC2(CCNC(=O)C(C)N3CC(C)C3)CC2)nc1C c1(C(=O)Nc2cnc(Br)o2)cccc(-n2ccnc2)c1 c1(C(=O)NC2CCC(C)(CNC(c3n(C)cnc3)=O)CC2)cc(F)cc(F)c1O CC1CN(C(=O)CCn2cccn2)CCC1C(=O)NC1CN(C(N)=O)C1 c1(C(N2C(CNC(C(CC)F)=O)CC(OC)C2)=O)cc2oc(C)cc2[nH]1 C1(C(=O)NCC2(C)CC(C)(C)C2)CC(F)CN1Cc1c(C(=O)OCC)con1 N1(c2ccccc2)CCN2N(CCC3Cc4c(Cl)cccc43)C2CC1 C(CC(CC)C(=O)NCC1CC1CC(N1CCC(N(C)C)C(C)C1)=O)=CC C1(CCOC)CN(C(c2cc(C(C)(C)C)nn2-c2ccccn2)=O)CCS1(=O)=O C1(NC(C=CC=CCC)=O)CN(C(C2CC2C#N)=O)C2CCCC12 N1(C(COc2c(C)cccc2)=O)CC2CC(NC(=O)Cc3ccnn3C)C1C2 Cc1cc(C)c(NC(=O)C(C)NC(c2occc2C)=O)cc1C c1(CC)cc(C)c(C(=O)NCC2CCN2C(=O)CS(=O)(=O)NC(C)(C)C)o1 c1(OC)cnc(Cl)nc1N1CCC(NC(=O)C(c2ccc(Cl)cc2)O)C(C)C1 C(C1CCCCCC1)=CC(=O)NCC1(F)CCN(C(C(CCSC)O)=O)C1 C1(c2n(C(CC)(C)C)nnn2)(NCc2cc(OC)n(C)n2)CCOC1C N1(C(c2scc(C)c2)C(=O)NC2(C)CC2)Cc2ccncc2C1 c1(C(N(C(C)C(=O)NC(c2cc(C)on2)C)CCC)=O)ccc(OC)cc1 CC1CC2(CCC2)CN1C(C1CN(C(=O)C2=CC3C=CC2C3)CC1(C)C)=O C=Cc1cc(C(N2CC(CNC(=O)C(C)(C)C)CC23CCC3)=O)cc(F)c1 C1(NC(CCCC=C)=O)CN(C(c2c(C)coc2C)=O)CC12CC2 N1(C(COCCSC)=O)CC(C)(C)CC1CNC(C1(C)COC(=O)OC1)=O CC1(CNC(=O)NCCCCCc2ccc(Cl)cc2)CCNC1=O CC(C)(C)CC(O)C(=O)NCC.N1(C(C)(C)C)CCN(c2nnc(C(F)F)o2)CC1 C1(C)(C(N(CC(C)CNC(=O)C(c2ccc(Cl)cc2)CO)C)=O)CC2(CCC2)C1 C1(NC(c2cc[nH]n2)=O)CS(=O)(=O)C2CN(C(=O)C(c3cccnc3)O)CC12 N1(C(c2c(OC)csc2)=O)CCN(c2ccccc2C(C)(F)F)CC1 C(=O)(C#CC(C)(C)O)NC(C1CCCN(C(c2cc(F)cnc2O)=O)C1)C C1(NC(c2ccnc(Cl)c2F)=O)CCCN(C(c2c(F)ccnc2Cl)=O)CC1 c1(C(=O)OC)cncc(S(=O)(=O)NC2CCCC3(CCCC3)C2)c1 C1(NCC2C(C)(C)CO2)CC2CC=CCC2C1.c12ccc(cc1)OC2 C=CC(C(=O)N1CCCC1CC(=O)NCC(C)(CO)OC)OC N1(CC)CC(C(=O)NCCC2CC(C(=O)N(C)CCc3ccccn3)C2)CC1=O C12(CNC(C3N(CC)CC3)=O)CCC(CN(C(c3ccnc4c3CCC4)=O)C1)C2 c1(C(=O)NCCC2CSCCN2C(=O)CCc2cnoc2)ccc2ncnn2n1 c1(C(N2CC(O)C(O)C2CF)=O)cc2ccc(Br)c(Cl)c2s1 S(=O)(=O)(c1cccs1)NCC(N1CC(C)C(NC(=O)C(c2cccnc2)C)C1)=O C(O)(CC(=O)NC(=S)NCCCF)(C(F)(F)F)c1ccc(C)o1 Cc1cc(Cl)cc(C)c1C(N1CC(CNC(=O)CCC2CCCOC2)C(O)C1)=O c1(C(=O)NC(CNC(c2c(C)nc(C)o2)=O)C(C)C(C)C)c[nH]c(C)c(Cl)c1=O N1(C(C(C)CN2CCOCC2)=O)CCC(NC(=O)C(N2CCC(O)CC2)C)C1C Cc1nnc2ccc(C(N3CCCN(C(=O)CC(F)(F)F)CC3)=O)cn12 C(=O)(CC(C)CCC)NCC1(O)CC(CNC(c2ccc(CCCCC)o2)=O)C1 c1(C(=O)[N+](C(CN(C(c2ccc(C(O)CF)cc2)=O)CC)C)([O-])NC)cn(C)[nH]c1=N C1(C(=O)O)Cc2nnc(SCCNC(=O)C(O)c3cnc[nH]3)n2C1 N1(C(CNS(CC)(=O)=O)=O)CCCN(C(=O)C=Cc2cscn2)CC1C(C)C c1(C(=O)NC2(CN(C(CS(CC)(=O)=O)=O)C)CC2)ccc2c(c1)CCCO2 O=C(C1=CC(O)C(NC(C2(O)CCCC2)=O)C1)NCCC(O)CCO N1(CC(=O)NCC2C3CN(C(c4cc(C)oc4C)=O)CC32)CCn2ccnc2C1 c1(C(=O)NC2CC(O)(CNC(C(CC=C)(C)C)=O)C2)nc2ccccn2c1F C(=O)(N1OC2CCC1CC2)C1C2N(C(c3c(CC)nc(C)o3)=O)CC(C=C2)C1 CCCC(C(=O)NC(CNC(=O)C(C)NC(C1CCC(=O)N1)=O)CO)NC(N)=O C1(NC(c2n[nH]c(C)c2C)=O)CN(C(c2ccc3c(c2)CCO3)=O)CC(C)(C)C1 C1(NC(CC(=O)NCC)=O)CN(C(c2csnn2)=O)C2CC12 CC1CC(C(=O)N(CCO)CCO)CN(C(=O)CCc2ccnn2C)C1 C1(C2CC2)(C(=O)NCC2C3CN(C(CC4(C)CCCO4)=O)CC32)CCOCC1 c1(C(=O)OCC=CC)ccc(C)nc1NC c1(CC(=O)NCC(C(=O)N(c2scc(C)c2)C)N(C)C)ccccc1C c1(OC)ccc(Br)nc1C(N1CCCC(NC(=O)C(C)(C)OC)C1)C(=O)NC(C)C c1(CC(=O)NC(C(CO)NC(C2C(COC)C2)=O)C)ccc2c(c1)CCCO2 C#Cc1ccccc1CC(N1CCCC(F)(C(=O)NCC(C)(C)SC)C1)=O C1(CC(=O)NCC2(C#N)CCN(C(c3c(C)n[nH]c3)=O)C2)CCC2(CCC2)CO1 Cn1nc(Br)c2nc[nH]c(=NCC3CN(C(c4cc[nH]n4)=O)CCO3)c12 N1(C(C2CCSCC2)=O)CCCC(C2CN(C(C34CCN(C3)S(=O)(=O)C4)=O)C2)C1 CCC(C)C(O)C(=O)NCC(=O)NCCCNC(N)=O N1(C(CC(C)F)=O)CCC2CN(C(c3coc(Br)c3)=O)CC12 c1(C(=O)NC2CN(C(C3(C(=O)OCC)CC3)=O)C3C2C3)cnc(O)n(C)c1=O CC1CCOCC1(F)NC(=O)COC1CCCCC1 CCCS(=O)(=O)CC(=O)NCCC1CCCCN1C(=O)C1=CCCC1 N#Cc1cc(CNC2CN(c3ncnc4[nH]ccc34)CCC2(F)F)cc(F)c1 CCCC(CNC(C1(C(F)F)CCCO1)=O)NC(c1cnc(C(C)C)[nH]1)=O C1(C(=O)NC(C(=O)NCC(=O)NCCOC)C(C)C)CCCCC1(C)C c1(NC)c(C(=O)NCC2CCCCN2C(=O)CCC2CC2)sc2nccnc12 N1(C(CCN(C(C2C=CC=CC=C2)=O)CC)=O)CCOC2CCC12 N1(C(C2(C#C)CCCC2)=O)CCC2(CCN(C(C3(C(C)C)CC3)=O)CC2)C1 C=C(C)C(CC(=O)N1CC2(CO)CC1(C(=O)N(C1(CO)CCSC1)C)C2)OCC N1(C(C(C=C)(C)C)=O)CCCCCC(NC(=O)CSc2nncn2C(C)C)C1 N1(C(C2(C#N)C(C)C2)=O)CCCC2(CCCN2C(=O)C=CC2CCOCC2)C1 C(C(=O)NOCC(N)=O)(c1ccoc1)NC(C1(CCOC)CC1)=O c12ccc3c(c1)C1(CCCC1)Cn3c2=O.Cc1ccc(C)c(C(=O)N(C)CCO)c1 c1(C(N(C2CC3CN(C(C=CC=CC)=O)C2C3)C)=O)cncc2cnccc12 C#Cc1cnn(CC(=O)NCCC2(C(=O)NC3CCOC(C)C3)CC2)c1 N1(C(C2C(C(N)=O)C2)=O)CCC2(CCCC2CNC(=O)C=CC(F)(F)F)CC1 C(=O)(CC(C(F)F)NC(=O)CN1CC(C)(C)C1)N1CC(CC)OCC1CC N1(C(C2C(C)CC2)=O)CCC2(CC2NC(c2cc(O)ncc2Br)=O)C1 CCC(C(=O)NC1C=CC(C(=O)N(C)Cc2cn[nH]c2)C1)C(F)(F)F CN1CC(=O)NC(CC(N2CCC(C)(c3cn(CC(C)(C)C)nn3)C2)=O)C1=O c1(C(N2CC(F)CC(NC(C3C(C)OCC3)=O)C2)=O)cccc2ncnn12 N1(C(c2c(CC)nns2)=O)CCN(C(=O)C(O)P(C)(C)=O)CC1c1ccnn1C N1(C(C2C(CC)OCC2)=O)CC2CCC1CN2C(c1cccnc1OC)=O C(=O)(CS(=O)(=O)C1CC1)NC1C(CNC(C23OC(C)(C)C(C2)C3)=O)CCCC1 c1(CN2C(CC(=O)Nc3ncc(F)cc3F)COCC2)cc(O)ccc1Br N1(C(CC2ON=C(C)C2)=O)CCC(C)(C(=O)N(C)Cc2ccoc2C)CC1 C(=O)(C1CCCn2cnnc21)NC1(C)CCN(C(CSc2n(C)nnn2)=O)CC1 c1(OC)cc(OC)c(CNC2CCC(C(=O)NCCCCl)O2)cc1Br.C(C)(C)O C1(CNC(=O)CC(C(F)F)N2CCOCC2)CCc2ncccc2C1 C1(NC(C(C)OCC#C)=O)CCCCCC1C(=O)NC(c1c[nH]ccc1=O)C c1(C(N2CCN(C(CC3CC(=O)C3)=O)C3C2C3)=O)[nH]c2ccc(F)cc2c1Cl c1(C(N2CCC(O)(C(C)NC(c3ccc(C)nn3)=O)C2)=O)nnn2c1COCC2 CC(C)(C)CCC(=O)C(=O)N1CC2(COC(CNC(=O)CC3CC3(C)C)C2)C1 CC1(C)COCC1C(=O)NCCC1CCN(C(C2(c3cccnc3)CCC2)=O)C1 CC1CCCN(C(=O)C(=O)NCCN(C2CCCC2)C(=O)CC2CC2(Cl)Cl)C1 CCC(C)C(=O)C(=O)N1CCCC(F)(CNC(c2ccc(F)s2)=O)C1 CN1CCc2ccc(NCC3CCCN(S(C)(=O)=O)C3)cc2C1=O N1(C(c2c(COC)cc[nH]2)=O)CC2(CCN(C(C3CCCC4(CC4)C3)=O)C2)C1 C12(CCCCCC1)C(=O)NC2.C(C)(C(=O)OC(=O)C1CC1)C(CC)=O C(=O)(CCCCCN=[N+]=[N-])NCCC(C)(C)NC(c1ccccn1)=O CC1CCN(C(=O)CN2CCN(C(C3(n4cnnn4)CC3)=O)CC2)CC1CO c1(OC)cc(C2(C(=O)N(CCCCCNC(c3cnco3)=O)C)CC2)ccc1C C1(C(c2c(C)cnnc2)=O)C2CC3C1C3C2C(=O)NOCCCC1CC1 CCC(CC(=O)N1CCCCC(CCC(=O)NCc2nncs2)C1)C(C)C O=C(CCC(F)(F)C(F)F)NCC(C1CC1)NC(C1CC1F)=O C1(NC(C(CN(C)C)NC(C#CC(C)C)=O)=O)CCCCC12CC2 C1(COC)(CNC(=O)COCC(C)C)CCCN1C(c1ccoc1Br)=O CC(C)(CO)C(=O)NCCCNC(c1cnn(-c2cccc(Cl)c2)c1)=O.C1CCC1 c1(Sc2cc(OC(C)C)ccn2)c(Br)cc(Br)c(Cl)c1Cl.CC1CC2N(C1)C2 CC(C)(C)C(=O)CCCC(=O)NC1CC2CC(NC(=O)CN3CCOC3=O)C1C2 C(=O)(C(F)C(F)(F)C(F)(F)F)N1C(CC(=O)N(CCOC)C)CCCC1 N1(C(C(=O)NC(C(C(F)(F)F)OC)C)=O)CC2(CCC(=O)N2)C1 c1(C(N(CCC(C)NC(=O)Cc2ccco2)C)=O)nc[nH]c2nccc1-2 N1(C(C(C)=CC)=O)CCC2(CCC2NC(=O)CCc2cccnc2C)CC1 Cc1c(C(N2CC3CCC(C2)N3C(C2CCCC23CC3)=O)=O)cnc2ncnn12 CN1C(=O)CSC1=CC(=O)NCC(O)CCNC(c1ccc(-c2cccs2)s1)=O C1(C(N(C)Cc2cn(CC)nn2)=O)CCC=CC1NC(C1CCCOCC1)=O c1(SCC)nc(-c2ccccc2)sc1C(=O)NC(=O)CCN1CCC(F)C1 C1(CNC(CC(C)(C)O)=O)CCCC2(CN(C(c3noc4ncccc34)=O)C2)O1 N1(C(c2n(C)ccn2)=O)CCC(C)(CNC(C2CCN(c3ccccc3)C2)=O)C1 C=CC(CC)CC(=O)N(CC(=O)NC1CCCNC1=O)CC1CC1 c1(N2C(C(=O)Nc3c(Cl)cc(F)cc3Cl)CC2)ncnc2cnccc12 c1(C(c2cn(CCNC(C3CN(C(C)=O)C3)=O)nn2)=O)cc(Cl)ccc1Cl Cc1ccc(S(=O)(=O)CC(C)NC(C2(c3nnnn3C)CC(C)N(C)C2)=O)cc1 N1(C(c2c(C)c(F)ccc2)=O)CCN(C(=O)CC(C)C)C(C#N)C1 c1(NC2CCCC(NC(c3occ(C)c3)=O)C2)cc(O)nc(O)n1 c1(C(C(=O)NCC(CN(C(C2(CC)CCNC2=O)=O)C)C)C)c(C)nn(C)c1C c1(CC)nnc(CNC(c2ccn(C3CC3)n2)c2nnnn2C2COC2)o1 CCC(C(=O)NCC1CCCCC1NC(C1CC2(CC(=O)N2)C1)=O)C(C)O S(=O)(=O)(c1cccc(Br)c1F)NC1CCCN(C(C=C(C)C)=O)C1 c1(C(N2C(COC)CN(C(c3cc[nH]c3)=O)CC2)=O)[nH]c(C)c(S(N)(=O)=O)c1C Cc1cnc(N2CCC(CC(C)NC(c3cc(C(C)(C)C)[nH]c3C)=O)CC2)nc1 C(CC(=O)NOCC(=O)N(C)C)OCCNC(C1CCN(CC)C1)=O Cc1c(Cl)c[nH]c(=NCC2CN(C(C34CCCCC3C4)=O)CCO2)c1C#N C1(C)(NC(N2CC(C(C)NC(=O)CCn3ccnc3)C2)=O)C2Cc3ccccc3C12 C1(CC(C)NC(Cn2c(C)ccn2)=O)CC2CCC(C1)N2C(=O)Cc1cc[nH]c1 C(CC(O)CC(=O)NCC(C)(C)CC1CN(C(=O)CC2CC2)C1)SC c1(NC(CC2(NC(c3ccc(OC)c(Br)c3)=O)CCC2)=O)cccc(Br)c1C#N c1(C(=O)NC2(COC)CCN(C(=O)CC3CN(C(C)=O)C3)C2)cccc(C)c1F C1(NC(c2cn(CC=C)nn2)=O)CCN(C(c2nnn(C)n2)=O)CC1CC c1(OC)cc(-c2nccn2-c2ccc(C(=O)O)cc2CO)cc(CC#N)c1OC Cc1ccc(C(=O)NCC(N2CCN(C(c3cncs3)=O)CC2)C(F)F)c(C)c1 C1(C(N2C(C)(COC)CC2)=O)CC2CCC(C1)N2C(C1COCC1C(N)=O)=O c1(OC)cc(OC)c(C(=O)N(C)CCN(C)C(c2cc(O)ccc2C)=O)c(F)c1 c1(C(=O)NC(CNC(C(=O)NCC)=O)C2CCC2)cnc(C(F)(F)F)c(Cl)c1 CC1CN(C(c2cnc[nH]2)=O)CC(CCNC(c2n[nH]cc2Cl)=O)O1 C1(NC(CC=C=C)=O)CCC12CN(C(=O)CC1CC(F)(F)C1)C2 C1(CNC(C2CC(S(N)(=O)=O)C2)=O)CCC2(CN(C(=O)COC3CC=CC3)C2)O1 CC1(C(=O)NC2C3CN(C(=O)Cn4cc(C5CCC5)nn4)CC23)CC=CCO1 N1(C(C(CC(C)C)OC)=O)CCC2(CC1)CC2C(=O)NC1COCCC1(F)F C(CCC(=O)NC1CCC1CNC(=O)CC1CCCO1)C1C(C)C1 C1(NC(c2ccc(COC)o2)=O)CCN(C(=O)CCC(C)N(C)C)CC1CO N1(C(C2C(C)(C)COCC2)=O)CCC(C2CCN(C(c3coc(Cl)c3)=O)C2)CC1 CC1(C(=O)NCC2CC2NC(=O)Cn2cnnc2)CCc2ccccc2C1 c1(N(C)C)noc(CNC(=O)C(CNC(=O)CCC2CCCO2)N(C)C)n1 C#CCN(OC)C(=O)C1CN(C(=O)CC2COCC2O)CCO1 C1(Cn2cc(CN(C)C(C3CN4CCN3CC4)=O)nn2)Cc2ccccc2O1 C1(CNC(c2cnn(CC(F)F)c2)=O)CCCN1c1ncns1 C1(NC(CCCCCC)=O)CCSC12CN(C(=O)C(C(C)(C)C)NC(C)=O)C2 N1(C(C=C(CC)CC)=O)CCN(C)CC1C(=O)NC(c1noc(C)n1)C C1(CNC(N(CC(CC=C)O)C)=O)COCCC1(F)F C1(NC(C2CC(OC)CN2C(=O)CCC(N)=O)=O)CCN(C)CC1C N1(C(C=CC=CCC)=O)CCSCC1CCNC(C1COCCN1CCCC)=O N1(C(C=C(C)CNC(C2CCCCO2)=O)=O)CC2CC2C2CC12 C1(NC(COCCC)=O)CCCC1NC(C1(Br)CCC1)=O N1(C(c2[nH]cc(C(C)=O)c2)=O)CC2CC(NC(C3CC(O)C3)=O)C1C2 N1(C(C2N(C(CCC=C(C)C)=O)CCC=C2)=O)CC2(C1)NC(=O)NC2=O CC(C)(C)C(C#N)C(=O)NCCC1(O)CCN(C(C2CCC3(CCC3)C2)=O)CC1 C(=O)(C(C)C(=O)NCC(c1ccccc1)N(C(=O)Cc1c(Cl)cnn1C)C)OC c1(C(=O)NC2CC(NC(=O)C3CC3)CC2O)cnc2c(c1)S(=O)(=O)NC=N2 c1(OC)cccc(CC(O)C(=O)N2CCC(NC(c3ccc(C)o3)=O)C2)c1 CCCCCCC(=O)NC1CN(C(C)C(=O)Nc2cccc(C)c2)CCCO1 C=CCCCC(=O)N1CCC=CC1C(=O)NCC(O)CNC(N)=O CCS(=O)(=O)c1ccc(CC(=O)N(C2CC3CCC(C2)N3C(=O)C(C)O)C)cc1 CC(CCN(C)C)N=c1[nH]c(=NCCc2csc(O)n2)[nH]c2c(F)cccc12 Cc1cc(F)c(C(=O)NCCCCC(C)NC(=O)C(O)CCC(C)C)cc1F c1(C(=O)NCC2C=CC(NC(C3(OC)CCC(C)C3)=O)C2)cnc2ccccn12 C(=O)(CC(C)C(F)F)N1CCC(CNC(C(c2cnn(C)c2)C)=O)CC1 C(=O)(CCCCCCCC1CC1)NC12C(CN(C(C(CC)n3ccnc3)=O)C1)C2 N1(C(c2c(C(N)=O)nccc2)=O)CCN(C(c2cc(Cl)cnc2Br)=O)C(CO)C1 C(=O)(CCC(=O)N1CCCC(NC(=O)C=CC2CC2)C1)N(C)C C1(NC(C(CC)(C)C)=O)CN(C(=O)Cc2n[nH]c(C)n2)C(C)(CC)C1 CC(C(=O)NC1CN(C(=O)C(C)(C)Oc2ccc(F)cc2F)C1)C(C)C(C)(C)C Cn1cnc2c1CCCC2C(=O)NCC1CN(C(c2n[nH]cc2F)=O)C1 C12(C(=O)NCc3c(C)nc(C)s3)CCCC1CCN2C(=O)CC1CCCSC1 n1(CC(=O)NCC23CCC2CCN3C(=O)CC(F)(F)F)nc(O)ccc1=O C12OCCC1C(=O)NC2.C1(C(C)C)CCCC1C(=O)NC(C12CC(CO1)C2)C C12(C(=O)NCC3(C)N(C(CNC(C)=O)=O)CCC3)CC1COC2(C)C.c1ccco1 N1(C(c2c(C)ccc(F)c2)=O)CCc2oc(C(=O)O)cc2C1 CC(CC1CC1)C(=O)NCc1cc(C(=O)NCC2CCN(C)C2)co1 n1(CCC)nc(C)cc1C(N1CCC(NC(=O)CCc2cn(C)nn2)CC1)=O C(=O)(C(C)(C)CC(F)F)N(CC(C)N(C(C(C1CC(F)(F)C1)C)=O)C)C C12(C(=O)NC3CC(OCC)C3)CC(C)(CN1C(C1(CO)CCCCC1)=O)C2 c1(-c2cn(C)nc2)cncc(NC(c2cc(C(C)(C)O)on2)=O)c1 C1(N(C(c2cc(SC)oc2)=O)C)CCC(CNC(=O)CC2CCCC2)CC1 CC(C)C1=NOC(C)(C(=O)NC2CCCC2NC(c2cnc(O)c(F)c2)=O)C1 C1(C(=O)NC(CNC(C2N(C(CCC)=O)CCC2)=O)CO)CCC2(CCC2)CC1 c1(CN(CCS(=O)(=O)Cc2ccc(Br)cc2)C2CC2)ccc(F)c(F)c1 N1(C(C2C(CC)CCO2)=O)CCCN(C(c2ccc(F)c(F)c2C)=O)C(C)C1 N1(C(C(C(C)OC)NC(c2cn(CC=C)nn2)=O)=O)CCn2cc(C)nc2C1 C1(CC)CN(C(c2ccco2)=O)CCC1NC(c1cc(O)nc(O)c1)=O C1(C(=O)NCc2ccns2)(CNC(C(CC)N(C)C)=O)CCCCC1 c1(CC)nc(C)cc(=NCCCCC(C)NC(c2cocc2C)=O)[nH]1 C1(NCCC=CC=C)CCN(C(=O)C=Cc2ccccc2)CC1(C)C C1(C(=O)NCC2N(C(C3(SCC)CC3)=O)CC(C)CC2)CC(C2CCCC2)C1 N1(C(=O)NC2(C3CCCCC3)C(C)(C)C2)CC2COCC2(CN2CCOCC2)C1 N1(C(c2c(CC)cccc2)=O)CC2C=CC1C(C(=O)NCCc1ccccn1)C2 C1(C(=O)Nc2ccccc2OCCc2c(C)n[nH]c2C)CCc2ncccc2C1 c1(C(N(CCCCNC(CC2CC(CC)C2)=O)C)=O)sc(Cl)c(Cl)c1N C(C(C)(C)C(=O)NCCOC1CCN(C(c2sc(COC)nc2C)=O)C1)OCC CCC(C)(C)C(C)CC(=O)NCC1CC(OC)CN1C(c1cc(F)ccc1N)=O c1(C(N2CCC(O)(CNC(C3C(C#C)C3(C)C)=O)C2)=O)ccc2cccnc2n1 c1(NC(C2CC(CCNC(CC(C)OC)=O)C2)=O)cc(C)c(O)cc1C C(=O)(C1=CCCOC1)NCCCc1ncnn1C.C=C1CC2(C1)C(=O)NC2 C1(C(=O)NC(C=C)COC)CCC(CNC(=O)CC2CCCCC2C)CC1 N1(C(c2c(CCC)n(CCO)nc2)=O)CC(NC(=O)C(O)C2CC2)CC(F)C1 c1(C(=O)OCc2nnc(C)n2C)ccc2c(c1)nc(O)n2C c1(CC(=O)NC(C2CCN(C(c3cnc(C4CC4)[nH]3)=O)CC2)C)cncc(F)c1 c1(C(N2CCC(COC3CCN(CC4CC4)C3)C2)=O)ccc2cnoc2c1 N1(C(c2c(CC)ocn2)=O)CC(NC(c2cc(C)cc(F)c2)=O)CCC(O)C1 CCCC(C)(C)CC(=O)NCC1CN(C(C2CCCN2C)=O)CC1C C1(OC)CN(C(=O)C(C)(F)Oc2ccccc2)CC1NC(c1nn(C)cc1C)=O C1(n2cc(CC(OC)OC)nn2)CCC(NC(=O)Cc2cscn2)CC1 Cc1ncc([N+](=O)[O-])n1CC(=O)NC(C1CCCC1)CNC(=O)C1=CCSC1 N1(C(C)=O)CCC(NC(C2CCCN2c2ncccn2)=O)CC1C N1(C(C2CCCCC2)C(=O)NCCC2(C)CC2)CCCC2(C1)CN(C)C(=O)O2 C1(COCC(=O)NCC(O)C2CC2)CCCO1.C12(CC1)C(=O)N2 N1(C(C(C(C)C)NC=O)=O)CC2CCC(C(=O)NC(c3cn(C)cn3)C)(C2)C1 Cc1cc(N2CCC3(CCCOC3)C2)nc(=NCC(C)(C)OCCN(C)C)[nH]1 c1(C(=O)NC2C(CNC(C3C(C)C3)=O)CCC2)ccc(Br)c(C(F)(F)F)c1 N1(C(C(CC)C)=O)CCC(F)(CNC(=O)C(c2ccc(Cl)cc2)(C)C)CC1 c1(C(=O)NC2CC(CNC(C)=O)C2)cc2c(C(F)(F)F)cccc2s1 c1(N(C)CC23CCCCC2C3(F)F)nc(N(C)CC2CCCS2)c2c(n1)CCS2 C(c1cnc(O)nc1O)=CC(N1CCC(O)(C(C)NC(c2nc(C)[nH]n2)=O)C1)=O c1(CCC)[nH]nc(C(N2CC3(C2)CN(C(C2(CO)CC2)=O)C3)=O)c1[N+](=O)[O-] C(C)(C(=O)N(CCNC(=O)CNC=O)CCNS(=O)(=O)CC)OCC#C c1(CN(C(c2cn(CCO)nn2)C(=O)NCCC2CC2)C)ccccc1Br c1(NC(N(CCOC)Cc2ccncc2)=O)cc(Cl)cc(Cl)c1OC N1(C(CS(CC)=O)=O)C(CNC(=O)CCOCC(F)F)CC2CCCC12 C1(C(=O)OC)COCCN(N2CCc3nc(Cl)ccc3C2)C1 n1(CC(=O)NCCC2CSCCN2C(=O)CCCCF)cc([N+](=O)[O-])cn1 C(=O)(CC(CC)C(F)F)N1C(CC(=O)NC(CCC)c2nn[nH]n2)CC(F)C1 C12(OC)CCCC(C(=O)NCC3(NC(=O)C=CSc4nc[nH]n4)CC3)(CC1)C2 c1(C(=O)NC(c2cn[nH]c2)C)csc(C(=O)NCc2cc(Br)cs2)n1 C(=O)(CC(C)(O)c1ccccc1)NCC(C)NC(=O)C(C1CCCCCC1)O C1(CC)C(NC(c2cc(-c3cnn(C)c3)[nH]n2)=O)CCN1C(C1(CC)COC1)=O c1(C(C(=O)NC)N(CC(C)OCc2ccc(F)cc2)C)cccc(OCCCl)c1 Cc1cccc2c1OCC2C(=O)N1CCC(O)(CNC(=O)CN2CC(C)C2)C1 c1(NC(CC2CCCN(Cc3ccc(C#C)s3)C2)=O)cccc(SC)c1Cl c1(OC)ccc(C(CN2CCCC(C)C2)NC(C2(NC(N)=O)CC2)=O)cc1 C1(C(N2C(CCNC(CCOCC#C)=O)CCC2)=O)CCOCC1(C)C c12cn(nn1)C1CN(C1)C2.C1(CC#N)CN(C(=O)Cn2nccn2)C1 c1(OC)ccc(CC(=O)N(C)CC2(Cc3ccc(F)c(OC)c3)CC2)cc1F c1(C(=O)OC)ccc(C(C)C(N2CCN(C(=O)CSCC3CCCO3)CC2)=O)cc1 Cc1ccccc1C(N1CCC(NC(=O)C=Cc2cnccn2)C1)=O N1(C(c2cn(CC)nc2)=O)CC2(CNC(c3cnn(C)c3N)=O)CCC1C2 c1(C(N(CCCNC(c2cnn(CC)c2C)=O)CCO)=O)cnc2sccc2c1 n1(CC(N2CC(C(=O)NCC3CCC(F)C3)SCC2)=O)c(=O)oc2ccccc12 C1(C(=O)NCC2(F)CC(NC(C=CC(CC)=CC)=O)C2)CC2CCC1O2 C(C(C)(C)CC(=O)NC(C)CCNC(C1CC1C1CC1C)=O)OC C#CCC(C(=O)N1CCCC(C(C)C)C1)NC(C1CC(C)(C)C1)=O CC(C)C(O)C(=O)N(CC(O)CNC(c1cc(C#N)on1)=O)C C(=O)(C(C)(C)CCNC(c1sc(C)nc1C)=O)NC(C=C)C1CCC1 Cn1nc(C(=O)NC2(CCNC(C3(C)CCCS3)=O)CCC2)c2cc(F)ccc12 N1(C(C(C)OCC=C)=O)CCN(C2CCN(C(c3ccc(O)cc3)=O)C2)CC1 C1(CC(N2CCC(NC(C(CC)CN(C)C)=O)(CF)C2)=O)CCCCC(=O)N1 c1(C(CC)CC)cc(C(N2CCCC2)=O)on1.C(=O)(CCCN1CCCC1)NC c1(C(=O)NCC2N(C(C3C(C)OCCO3)=O)CCC2)nn(C)c2c(=O)[nH]cnc12 N1(C(c2c(CC)nccn2)=O)CC(NC(=O)CCc2cn(C)nn2)C(C2CC2)C1 CC1(C)CC(CNC(c2cncc(Cl)c2Cl)=O)N(C(=O)Cn2ncnn2)C1 CC(C)(CC(=O)N1CC2CC2(CNC(C2CCCCC2(C)C)=O)C1)C(F)(F)F C=CC(C)(CC)C(=O)NCC1(NC(=O)CN2CCN(S(C)(=O)=O)CC2)CCC1 c1(C(C)C)nc(C(=O)NCC2CN(C(C3(O)CCOC3)=O)C2)co1 C=CCC(C)(C)C(=O)N(C)CC1CCCN(C(c2c(CC)noc2C)=O)C1 Cc1cc(C(=O)N(CC(=O)NOCC2CCC2)C(C)C)c(C)[nH]1 N1(C(C2(C)CCOC2)=O)CCC2C1CCCN2C(=O)Cn1ccc(C(F)F)n1 C1(C(=O)NCC(CNC(=O)CCc2ccoc2)CO)CCc2nc[nH]c2C1 Cc1cc(C)c(C(N2CCCC3OCCC23)C(=O)Nc2ccccc2Cl)cc1C N1(C(c2c(OC)nn(C)c2)=O)C2CCC1CC(CNC(=O)C(F)C(C)(C)O)C2 N1(C(c2cc(COC)no2)=O)CC(NC(=O)CCc2ncccn2)C2CC12 c1(C(N)=O)cccc(CNC(=O)C(N2CCCCC2C2CC2)=O)c1F C1(C(N2CCC(C(N)=O)C2)=O)CC(O)CCN1C(C1CC12CC2)=O c1(C(=O)NC(CNC(CCCC)=O)(C)CO)cnc2c(=O)[nH]ccc2c1 c1(C(N2CCC(NC(c3cc4occc4s3)=O)(CF)C2)=O)cc(=O)cc(Cl)[nH]1 N1(C(CC(=C=C)C)=O)CC2C=CC1C(C(=O)NCC(C1CC1)N(C)C)C2 C1(O)(CNC(C(Cc2cc[nH]n2)NC(C(C)=C(CC)C)=O)=O)CCN(C)C1 N1(Cc2ccc(C(=O)OCC)[nH]2)CCC2C(CCN2C(=O)Cc2cccnc2)C1 c1(N(C)C)cccnc1C(=O)NCCCOCCNC(C12COCC(C1)C2)=O C1(NC(C(C2CCCC2)OCC)=O)CC12CCN(C(c1cc(C(C)C)no1)=O)C2 C(=O)(C1=C(Cl)CCC1)NCC1(C)C(NC(C(C2CCCCCC2)OC)=O)CCC1 c1(C(=O)NC2CN(C(C34CCC(C3)C4)=O)C3CC23)cccc(Cl)c1Br C1(C)(C(N(CCCC(=O)NC2CCCN(C(C)C)C2)C)=O)CCCCC1C c1(COC)ncc(C(N2CC(NC(C3OCCO3)=O)C(O)C2)=O)c(O)n1 CC1CCC(Cl)=C(C(=O)NCCCOCCNC(c2cc(C(N)=O)cs2)=O)C1 C1(CC(=O)N(CC(C)O)C(C)C)CN(C(C2CCCC(O)C2)=O)CC1C c12ccc(cc1)C(C(=O)NCCc1ncc[nH]1)OC2=O.C1(NCC)CC1 N1(C(c2ncn(C(C)N)c2)=O)CCC(C2CCCN(C(=O)C(C)CC)C2)CC1 C1(CC(N2CC(N3CCN(C(C(N)=O)=O)CC3)C2)=O)(C(F)(F)F)CCC(=O)NC1 N1(CC(=O)N(C2CCN(C(=O)C(O)CC3CCCCC3)C2)CCC)CC(C)(C)C1 C1(C(=O)NCCCOCC)C(C2CC2)CCN1C(=O)CC1CCCCC1 N1(C(CCCN(C(c2ccc(C#C)cc2)=O)C)=O)CCC(F)(F)CC1C C(C)(CNC(=O)C=C(Cl)Cl)(CNC(c1cccn1C)=O)OC C(CN=c1[nH]cc(C#N)c2ccsc12)N(C(C(c1ccc(F)cc1F)C)=O)C C1(NC(CC2(N(C)C)COC2)=O)CCOCC1NC(C1COCCO1)=O Cc1cnc(C(=O)NCC2CC(NC(c3n[nH]c(C)c3Cl)=O)C2(C)C)cc1Cl C1(CC)CCCN(C(C2CC(O)C2)=O)C1C(=O)NC1CC2OCCCC12 c1(CC)cnc(C)c(C(=O)NCCOCCNC(=O)COc2ccsc2Cl)c1 CC1CCCc2c(C(=O)NCCN(C)C(c3cccc(Br)c3O)=O)cnn21 C1(CNC(COCCOCC)=O)CC12CCN(C(c1cscc1OC)=O)CC2 c1(SC)nc(CNC(c2ccc(SC)o2)=O)cs1 C1(C(=O)NC2C3CCN(C(c4c(C)n[nH]c4)=O)C32)CCOC2(CCOCC2)C1 c1(NC(C2N(Cc3n(CC)ccn3)CC(O)C2)=O)cccc(C)c1C c1(CNCC2N(C(C(C)S)=O)CCCC2)cccc(Br)c1O N1(C(C(c2ccc(F)cc2)C)=O)CCN(C(C2CCC(=O)O2)=O)C(CC(F)F)C1 C1(C(=O)OC)COCCN(S(=O)(=O)N2Cc3ccccc3C2)C1 C1(C(C)NC(C2(N(C)C)CC2)=O)CCCN1C(c1ccc(Cl)[nH]1)=O O=C(C1=CCCOC1)N1CCC(OCC(=O)NOC2CCC(O)C2O)C1 C1(C(N2CCC(CNC(=O)CCC3(C)CCC(=O)N3)C2)=O)(OC)CCC(C)CC1 C1(C(N2CCC(CN(C(=O)C=Cc3cc[nH]n3)C)CC2)=O)CCc2nn[nH]c2C1 c1(C(C)=O)ccc(=NC2C3CC2CN(C(c2c[nH]cc2Br)=O)C3)[nH]c1C(F)(F)F C1(C(N2C(CN(C(c3nnc(C)o3)C)C)CCCC2)=O)CC(C(C)C)=NO1 C1(C)(C(=O)NC(CC(=O)NCC(NOC)=O)CC2CC2)CC2CCC1C2 CCC(C)(CC)C(=O)NCC1CC2(CC(NC(C3(CC)CCCO3)=O)C2)C1 C12(NC(C3N(Cc4onc(COC)n4)CCCC3)=O)CCC(COC)(CC1)C2 c1(SCC(=O)N(C(C)C)CCNC(c2ccc(Cl)[nH]2)=O)ncnc2[nH]cnc12 N1(C(c2c(CC)nn[nH]2)=O)CCOCC1(C)c1cn(CCC(=O)OC)nn1 C1(NC(CC(C)C2CCCO2)=O)CC2(CCN(C(C34CC5CC3C4C5)=O)C2)C1 c1(NC2CCC(NC(c3c(OC)ccc(Cl)c3)=O)C2)ncnc2ccc(F)cc12 C1(NC(C(CCO)N(C)C)=O)CN(C(c2cccc(F)c2C)=O)CC1(C)C CN1CCN(CC(=O)NC2CCCC2CNC(=O)C=C(Cl)Cl)CC1=O C1(C)(CSC)CN(C(C2(C(=O)OC(C)(C)C)CCOCC2)=O)CC1(F)F C1(CC)(NC(=O)C(F)C(F)(F)F)CCCN(C(=O)CC(C)c2ccco2)C1 C1(C)(CC)C=C(C(=O)N2CCC(CN(C(c3cc(=O)n(C)o3)=O)C3CC3)CC2)C1 CC1C(C(=O)N2CC(N(C)C)C(CNC(=O)CN3CCCCC3C)C2)=NOC1C c1(C(C)C)nccc(=NCC2(O)CN(C(c3occ4c3CCOC4)=O)C2)[nH]1 C(=O)(C1=CC2(CCN(C(=O)OC(C)(C)C)C2)C1)NCCN1CCCC(C)C1 N1(C(=O)C=CCF)CCC(CCC2CCCN2C(c2ccc(C3CC3)o2)=O)CC1 N1(C(CCc2c(-n3cc(COC)nn3)cccc2)=O)CC(C(N)=O)OC(C)C1 c1(C(N2CCCC(C)(NC(CCCC=C)=O)C2)=O)cc2c(OC)ccc(C)c2[nH]1 c1(C(=O)NC2C(C)(C)N(C(=O)CCc3nccs3)CC2)cccc2oc(O)nc12 N1(C(Cn2c(C)cc(C)n2)=O)CCCCCC1CNC(=O)Cc1cn[nH]c1 c1(C(=O)NC2C(CC)CN(C(=O)CCc3cc[nH]n3)CC2)cn2cccnc2n1 CC1CC(NC(C2(C)CCC(F)(F)C2)=O)CCN1C(=O)CC(O)CN(C)C CC(=O)CCCC(=O)N(CCCNC(=O)C(C)NC(C1CCCC1)=O)C c1(C(=O)NCC2(COC)CN(C(=O)CC3OCCC3C)C2)ccc(SC)cc1C CC(CSc1ccccc1)C(=O)NCCN(C(=O)C=CCl)Cc1ccccc1 C(=O)(C(CO)C(C)(C)C)NCC(CNC(c1c(C)cco1)=O)CO C(=O)(C(C)C(C)C(C)(C)C)NCC1(F)CC(CNC(c2cc(C(C)=O)sc2)=O)C1 C1(C)(COC)CC(NC(=O)CCCNC=O)CN1C(=O)CCCCCSC c1(C(=O)NCC2CCCN2Cc2ccccn2)ccc2oc3ccccc3c2c1 c1(C(N2CC3CCN(C(C(C)c4cc[nH]n4)=O)CC32)=O)n[nH]c2c1CN(C)CC2 N1(C(CCOCCCNC(CC2CC(N(C)C)C2)=O)=O)CCCOC(CCO)C1 N1(c2nnc(C)o2)CCC(NC(c2ccnc(-n3cccn3)c2)=O)C(CO)CC1 N1(C(c2c(C)csc2)=O)CC=CCC1C(=O)NCC1COC(=O)N1 c1(C(=O)NC2CCN(C(C(C=CC)O)=O)CC2O)c(C)c(C)c(C)c(C)c1C C1(CNc2ccc(C(=O)OC)c(N)c2)CCn2ccnc2C1 C1(NC(CC(C=C)C)=O)C(C)(C)C(NC(c2ccc(F)c(C#N)c2)=O)C1(C)C Cc1cc(C)c(C(=O)N(CCCCN(C)C(C2(C#N)CC3CC3C2)=O)C)c(S)n1 N1(C(CN(C(C)=O)C)=O)CCN(CCNC(c2cc(C(C)(C)O)ccn2)=O)CC1 C(=O)(CCC1CCc2ccccc21)N1C(CN(C)C(c2cn(C)cn2)=O)CCC1 S(=O)(=O)(c1ccc(NCC(c2ccccc2)F)c(Br)c1)NC(c1cnn(C)c1)C n1(CCC)cc(CNC(=NCc2cnc(C(F)F)nc2)NCC(F)F)c(C)n1 CC(C)CC(C)C(=O)NCC1CCCCCCC1 c1(CC(=O)NCCN(C(c2c(CC)[nH]cc2)=O)C)ccc(Br)nc1 c1(C(N(CC(CCC)O)C)=O)ncc(C(=O)OCC)cc1C.C(C)(C)(C)O Cc1c(C(=O)NCCC2CCC(NC(c3cnsn3)=O)C2)sc(Cl)c1Cl c1(C(N2CCC(NC(C3(F)CC3)=O)C2)=O)c(F)cc(Cl)cc1Br CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1(CF)CCN(C(c2ccncc2C)=O)C1 c1(C(=O)NCCCN(C2CCCC2)C(C2CC(C)(C)O2)=O)ccc(Cl)cc1Cl N1(C(c2ccc(N)c(F)n2)=O)C2CCC1CN(C(C1CCN3CCOCC13)=O)C2 C#CC1(NC(=O)C(C2(C)CC2)NC(=O)CCCC2CC2C)CC(F)(F)C1 c1(C(=O)NCCOCCNC(C(CC#C)O)=O)cc([N+](=O)[O-])nn1C C1(C2(O)CCOC2)(C(N(C(=O)CCCC(C)(C)CC)CC)=O)CCC1 N1(C(C(CC2CCC2)OC)=O)CC(C)C(C)(CNC(=O)C(C)NS(C)(=O)=O)C1 c1(N(CCNC(C)=O)C)nc(N(C)Cc2c(C)cccc2C)nc2scnc12 c1(NC(C=C2CCN(C(c3c(SC)nccc3)=O)CC2)=O)c(F)ccc(Cl)c1F C1(C2(O)CN(C(=O)CCCn3nc(C)cc3C)C2)(CNC(CCC(=C)Cl)=O)CC1 n1(CCCC)ncc(C(=O)NCCC2CC(NC(C34CCCC3C4)=O)C2)c1C CC1C(CNC(=O)C2=CCOC2)CCN1C(=O)CC1CCN(CC(F)F)CC1 C1(NC(Cc2c(C)n[nH]c2)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)CC12CCC2 c1(NC(C(=O)NCC(c2ccccn2)(C)C)=O)cc(F)c(F)cc1N c1(CNC(CCC)(c2nnnn2C(C)C)C2CC2)ccc(F)c(OC)c1 N1(C(C(C)NC(C)=O)=O)CC2(CCN(C(c3c[nH]c4ccc(F)cc34)=O)CC2)C1 N1(C(c2ccc(CC)cc2)=O)CCC2C1CCN2C(c1c(C)n[nH]c1C)=O CCC(C(=O)NC1COCCC1C(=O)NC(C)C(C)C(=O)OC)C(C)C C1(NC(c2cc(CCC)c(C)s2)=O)(CC)CCN(C(C2CN(C)C(=O)N2)=O)CC1 C#CCC(CC(=O)NCC(CCSC)OC)NC(c1cccc(C)n1)=O C1(C(N(CC)CC2CCCN2C(c2coc(Cl)n2)=O)=O)CCC(F)(F)C1 Cc1cc(C(=O)NC2CC(C)(NC(=O)CCCc3nncn3C)C2)ns1 Cc1cc(C)c(C(=O)NC2CC(C)N(C(c3cc(C(F)(F)F)ccn3)=O)C2)cn1 c1(C(N(C(C)CCNC(C2(C)CS(=O)(=O)C2)=O)C)=O)cc(O)c2ccoc2c1 c1(C(C(=O)OC(C2(c3cccc(OC(F)F)c3)CC2)=O)O)ccc(F)c(Cl)c1 Cc1cc(=NC(=O)C(=O)N2CCC(C(C)NC(C3(O)CC(F)(F)C3)=O)CC2)[nH]o1 c1(CC(=O)N(CCC(=O)Nc2cccc(SC)c2)CCO)csc2nc(C)cn12 C(=O)(C1=CCCC(C)(C)C1)NCC(=C)CCNC(c1ccc(C)o1)=O c1(CCC(=O)NC2CC(CNC(=O)COCCF)C2)ccn(-c2ccccc2)n1 c1(CC)cccc(C(=O)NC2(CN(C)C(C3(C)CCC(=O)N3C)=O)CCC2)c1O N1(C(=O)OC(C)(C)C)CC2(C1)C(OC(c1nccn3cnnc13)=O)CCS2(=O)=O C1(C(N(CCNC(c2cnc(N(C)C)s2)=O)CCN(C)C)=O)CCC(=O)N1C1CC1 C1(C(N(C)Cc2cnccn2)=O)CN(C(c2ccc(C#N)n2C)=O)CC12CC2 c1(-c2ccc(C(N(C(=O)OC)Cc3cccn3C3CC3)=O)cc2)cc2ccc(OC)cc2nc1C.CC C1(NC(CCc2c(C)cccc2)=O)C(C)(C)C(NC(c2ccon2)=O)C1(C)C n1(CC(=O)NC(C(C)NC(c2cccc(S)c2)=O)CO)ncc2cccnc12 c1(CC)ccsc1C(N1CCCC1CNC(c1cc(Cn2cccn2)on1)=O)=O c1(OC)noc(C)c1C(=O)Nc1cccc(CNC(=O)C(C)OC)c1 N1(CC)CCCCC1C(=O)NCC(C1CCC1)NC(=O)CCC1CCCC1 N1(C(=O)OC(C)(C)C)CC2CCCC1C2c1ccc(CCN(C)CCCCl)cc1.C(F)(F)F C=CCC(CC(F)F)NC(C1CC(C)CCN1C(=O)C=Cc1cocn1)=O N1(C(C(=O)NCCN(CCC)C(c2ccc(C#N)s2)=O)C)CCC(O)CC1 C1(NC(c2c(OC)nn(C)c2)=O)CC1C1CCCN(C(=O)C=Cc2ccoc2)C1 c1(C(N(C2CN(C(C3(C)COCCO3)=O)CC2O)C)=O)ccn2c1CSCC2 c1(C(=O)NC2CC(NC(C3C(=C)CC3)=O)C2)cc(C(F)(F)F)nn1C1CC1 C1(COC2CN(C(CC=C=C)=O)C2)CCCCN1C(C1CCCN(C(C)=O)C1)=O C1(C(N(C2C(C)COCC2)C)=O)CCCCN(C(=O)CC2CC=CC2)C1 c1(C(=O)NCC2OCCCN(C(c3c(C)occ3)=O)C2)cccc2c1CC(=O)N2 N1(C(C2CC3CC(OC)C3C2)=O)CC2CCCN(C(=O)CCc3nncs3)C2C1 c1(COC)ccc(C(=O)NC2CC(C)(NC(=O)CCNc3ncccn3)C2)s1 C1(C(=O)NCCC=C=C)CC(O)CN1C(=O)C(CC1CC1)OC N1(C(C(C)SCC)=O)CCCCC1CCNC(=O)CC1C=CS(=O)(=O)C1 c1(OC)c(C(=O)NCC(C)NC(=O)C(C(C)C)NC(N)=O)ncnc1C n1(C(C)(C)C)ccc(C(=O)NC2CC2NC(=O)C(C)(O)C2CCOCC2)n1 C1(C)(CC(=O)Nc2cc(C)sc2)CCN(C(c2ccc(C(F)F)o2)=O)C1 C(=O)(C1=CCC(C)CC1)NCC(C(C)C)(C)NC(c1cc(C(F)F)ccn1)=O C12(CNC(c3cc(CC)ncc3)=O)CCC(CC1)N2C(c1cnc(Cl)[nH]1)=O C1(CCNC(C=CC(C)(C)SC)=O)CCN(C(c2coc(C)c2)=O)CCC1(F)F N1(C(c2cc(COC)cn2C)=O)CC(CNC(=O)C(F)OC)C2(CCOCC2)C1 C#CCC(C)(CC)C(=O)NCCc1ccc(CNC(C2(C(C)C)COC2)=O)cc1 c1(OCC(=O)NC2CCN(C(CC)=O)C2)c(C)cc(C)cc1C.C12CCCC1C2 N1(C(Cc2ccn(C)n2)=O)CCOC(C2(O)CC2)C1.c12cccc(c1)CNC2=O c1(NC(C=C2CCN(C(c3cc(C)nn3C)=O)CC2)=O)cc(Br)cc(Cl)n1 N1(C(C(c2n(C)ncc2)O)=O)CCC2(CCCN2C(=O)C=C2CCC2)C1 C1(C(N(CCC(=O)NCCSCCO)CC=C)=O)CC2CC2C1 C1(C(=O)NC(C#N)C(N)=O)CCCC12CCN(C(c1cccc(Cl)c1Br)=O)C2 c1(CC)ccsc1C(=O)N(C1CC(NC(c2cnc(CC(C)C)s2)=O)C1)C C(=O)(CC(C)C(C)C)NC(CC=C)CNC(c1cncc(C(F)F)c1)=O c1(C(N(C2CCN(C(C3(C)CS(=O)(=O)C3)=O)C2)CC)=O)nc(F)ccc1Cl c1(C(=O)NC2CC3CN(C(C4C(=C)C4)=O)CC32)cc([N+](=O)[O-])cc(C)n1 C1(N(C(=O)CCOC2CCOCC2)C)CCCN(C(c2cc[nH]n2)=O)CC1 c1(NC(C23CC(CO2)C3)C)c[nH]c(=O)cn1.n12cc(nn1)C(C)N(C)C(=O)C2 c1(C(=O)NC(C2C(C(=O)NCC(C)(C)OC(C)C)C2)C)cc2ccccn2c1 C1(C)(NC(C(CC=CC)NC(c2c(CC)n(C)nn2)=O)=O)CCC(C)(C)C1 N1(C(CC2C=NN(C)C2=O)=O)CCCC2CN(C(=O)Cc3cnn(C)c3)CC12 c1(C(=O)NCC(C)NC(C2(F)CC=CCC2)=O)ccc2ccc(Br)cc2n1 CCC(C(=O)NCC(C1CCCO1)NC(=O)C=CC(=O)N(C)C)NC(C)=O.O Cc1cc(C(N2CCC(C)C2CNC(c2cn(C(C)C)nc2C)=O)=O)[nH]c1C N1(C(C2(NC(=O)CSCCNC(C)=O)CC(=C)C2)=O)CC(CC)C(O)C1 C1(C(=O)NCC(CCNC(=O)CN2CCC(C)(C)C2)OC)CCOCC12CCC2 c1(C(=O)NC2C(OC)CN(C(c3cn(CC=C)nc3)=O)C2)ncnc2ccsc12 c1(SCC(=O)Nc2c(C)cc(OC)nc2)ccc(F)cc1[N+](=O)[O-] N1(C(CNS(CCOC(C)=O)(=O)=O)=O)CC2CC2(CNC(=O)CC(C)(C)SC)C1 N1(C(C(C)CSC(F)(F)F)=O)CC(NC(C2(F)CCOC2C)=O)C(C)C1 C1(NC(C(c2ccccc2)C2C(C)C2)=O)CCN(C(C2SCCCS2)=O)C(C)C1 C=Cc1cncc(C(N2CCOCC2C(N2CCN(C)CC2CO)=O)=O)c1 N1(C(C)=O)CC(CNC(C2CN(C3CCCCC3)C2)=O)C(C)C1 c1(SC)cc(C(=O)NCCC2(NC(C3CC3c3cccs3)=O)CC2)c(C)o1 CCC(C)C(O)C(=O)N1CCOCC1CNC(=O)CCN(C)CCO C(=O)(C(CC)C(=O)NCCCCNC(C1COCCN1C)=O)OCC C1(CN(C)C(c2cnsn2)=O)CCN(C(C2C3(CC3)C23CC3)=O)CC1 Cc1cc(=O)c(NC(C2CN(C(=O)C(CC(C)C)C(C)C)C3(CCC3)C2)=O)c(C)[nH]1 N1(C(Cc2nc(C)[nH]n2)=O)CCC2CC2(C(=O)N(CC2CCC2)CC2CC2)CC1 CCC(C)(CNC(C1(CC)CCN(C(c2ncccn2)=O)C1)=O)CC S(=O)(=O)(c1ccc(S(=O)(=O)N2CCCCC2)cc1C)N(C1COC(C)C1)CCC C=CCC(C)(C)CCNC(C1CN(C(C2CC(C3CC3)=NO2)=O)CCO1)=O c1(C(=O)NCC2N(C(C(C)(O)C3CCC3)=O)CC2)ccc(Br)nc1 c1(CC)ccc(C(=O)NC(CNC(=O)C(C)CC2CCC2)C2CC2)cc1N N1(C(c2cc(C(F)F)cs2)C(=O)NCCCOC)CC2CC=CC1C2 C1(OC)CCCN(Cc2cc(C3(C)CC3)on2)C1 C1(CN(C)C)CCN(CC(C2COCCO2)=O)C1 O=C1CC(C(N2CCCCC2CNC(=O)COCc2ccccc2)=O)NC(=O)N1 c1(OC)ccc(Br)c(F)c1CNc1cc(Br)cnc1C Cc1cccn2c(C(=O)N(C(c3ccccc3)CNC(=O)C(C)(F)F)C)cnc12 C1(C(=O)NCC(CCC)NC(=O)CCn2ncn(C)c2=O)CCC(=O)N(C)C1 CC1CCCN(C(=O)C=Cc2cscn2)C1CCNC(c1occc1Cl)=O C1(O)(CCNC(C2(C)COC2)=O)CCN(C(C2(c3ccccc3)CCOC2)=O)C1 C1(N(C(CSCC)=O)C)CCC(NC(c2ccsc2CC(N)=O)=O)CC1 N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2cc(C(C)C)n(C)n2)=O)C2CC12 C#CCC(C)(C)NC(=O)C(CN(C)C)NC(=O)C=CCO Cn1ccc(C(F)=CC(N2CCCC2CNC(c2ccc(C(F)F)nn2)=O)=O)n1 c1(CC)ccc(C(=O)NCC(C)N(C)C(c2cccc(C)c2C)=O)c(OC)c1 Cc1cc(C)c(C)c(C(=O)NC2CCCC(N(C(=O)Cn3nccn3)C)C2)c1C c1(OC)ccc(N(C(=O)CC(C)n2cc(Br)cn2)CC(C)C)cn1 C1(C(C)NC(c2ccc(-c3cccs3)s2)=O)CCCCN1C(C1CCC(=O)O1)=O c1(C(=O)Nc2cc(F)cc(Cl)c2O)ccc2[nH]c(=O)ccc2c1 C12CCCC(C1)C(=O)N1CCC1CN2C.c1(NC(=O)CON)ccccn1.CCO C(=O)(C(N=[N+]=[N-])C(C)C)NC(C(C)C)CC(=O)NC(C)(CO)C(C)C C1(N(C(c2nnn(C)n2)c2nnnn2-c2ccccc2)CCO)CCCC=C1Br C1(CNC(C(F)=CCC)=O)CCN(C(=O)CNC(=O)OCC)CC1C C1(C(=O)NC2CC(C)N(c3ccnc(CO)n3)C2)CC2(C1)CC(F)C2 C=C1CN2C(=O)CCC2(C(=O)NC(C)CCN(C)C(C2CC(=O)CC(=O)N2)=O)C1 N1(Cc2nccc(C)c2)CC2(CCC(Nc3ncc(C)c(C)n3)CC2)C1 c1(C(N2CC(CNC(=O)Cn3cnc([N+](=O)[O-])c3)C2)=O)cc2cc[nH]c(=O)c2s1 N1(C(c2cnc(-c3ccc(C)c(F)c3)c(C(F)(F)F)c2)=O)CCn2cncc2C1 C=CCC(CC(F)F)C(=O)N1CCC(NC(=O)Cc2cc[nH]n2)CC1C C1(C(N(CC(O)CO)C(C)C)=O)CN(C(=O)CN2CCCC2)CCC1(F)F c1(C(=O)NC2CN(C(c3c4nnc(C)n4ccn3)=O)C2)c[nH]c2ncnc(O)c12 C1(NC(CCC2(NC(c3c(C)snn3)=O)CCCC2)=O)CCN(C)C1C C1(CNC(C(C)c2cc[nH]n2)=O)CCC(NC(=O)CCC2CCOCC2)C1 CC1(C)C2CCC(C2)C1C(N1CCC2(CC2NC(C2CC3(CSC3)C2)=O)C1)=O C(C(C)C(C)C(=O)N(CC(C)(C)CNC(c1ncccc1OC(C)C)=O)C)OC c1(NC(N(C(C)(C)CCNC(C2C3CS(=O)(=O)CC23)=O)C)=O)ccn2cnnc2c1 c1(CC(N2C(C(C)NC(CCC(C)SC)=O)CCC2)=O)cc2ccccc2s1 c1(NC(Cc2c(OC)cccc2OC)=O)cc(Cl)nc(C#N)n1 c1(N2C3C(CNC(C4C(C)CC5CC5C4)=O)C(C3)C2)ncn(C)c(=O)c1Br CCCC(C)(C)C(=O)NCC1CN(C(=O)CCNC(c2ccccc2)=O)CC1O C1(NC(Cc2c(F)ccc(C)c2)=O)CC2CN(c3ncc4c(n3)COC4)CC2C1 N1(C(c2cnc(C)[nH]2)=O)CCC2(CCCC2NC(c2ccc(F)c(Br)c2)=O)C1 CCC(C)C(O)C(=O)N(CC)Cc1ccccc1CN(C(C1CCOC1)=O)CC C1(CC=C)(NC(=O)COC(C)(C)CC)CCN(C(c2coc(SC)c2)=O)C1 CC1COCC(C(=O)NCc2cccc(CNC(C3(n4ccnc4)CC3)=O)c2)O1 Cc1nn(C)c(N)c1C(=O)NC1(C)CCC(NC(=O)CNC(N)=O)CC1 N1(C(c2cnc(C)o2)=O)CCOC(C)(CNC(C2CC23CC(C)(C)C3)=O)C1 c1(OC)ccc2cccnc2c1C(N1CC(OC)C(F)C1)C(=O)NCCCSC N1(C(C(CC)CC)=O)CCCC2(C1)CN(C(=O)CC1CCC1C(=O)OC)C2 c1(C(C)=O)ccc(C(=O)NCC(CNC(=O)C(C)(C)c2ccno2)OC)c(F)c1 c1(C(N2C(CNC(C3(C)CC(C#N)C3)=O)CCC2)=O)ccc2nc(O)[nH]c2c1 c1(C(=O)NCCN(C(CCc2cc(OC)no2)=O)C(C)C)c(N)ccc(C)c1F c1(CCC)ncc(C(=O)N(C2CCC(NC(=O)COC3CCC3)C2)C)s1 C1(CNC(C(CO)NC(C)=O)=O)(NC(c2oc(CO)nc2C)=O)CCCCC1 N1(C(c2c(C(=O)O)nns2)=O)CCN(C(C2(F)CCC2)=O)C2CC12 C(=O)(C1CCCc2scnc21)NC1C(SC)CN(C(=O)C2=CCCCC2)C1 N1(C(CCCOCCOCC)=O)CC2CC1C2NC(C1CCC(F)CC1)=O c1(C(=O)OC)cc(NCC2CCCC(C)(C)CC2)c(O)c(C)c1 C(CCCC(=O)N(C1CCN(C(c2ncn(C(C)C)n2)=O)CC1)C)OC c1(CN(CC(=O)NC)C)cc(Br)ccc1Cl C(CCC(=O)NC(C(=O)NCCCO)c1ccco1)OCCOC C1(O)(CCNC(=O)C(O)C2CCC2)CCN(C(=O)C(F)=CCCF)C1 C(=O)(C(F)(F)CC1CCNCC1)NC1(C)CN(CCS(N)(=O)=O)C1 c1(-c2n(C)ccn2)ccc(C(=O)NC2C3CC(NC(=O)CC4CCC4)CC23)cc1 N1(C(CCc2c(C)nccn2)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)C2(CC2)C1 CN1CC(C)(C)CC1C(=O)Nc1cccc(NC(c2cnc(C3CC3)s2)=O)c1 Cc1nn(C)c(I)c1C(=O)NC1CCC1NC(c1ccoc1)=O C1(C(=O)NC(C2CCN(C(c3cnns3)=O)C2)C)(N(C)C)CCCC1 n1(CC)cnc2c(NCc3cnco3)[nH]c(=NC3CCOC(C4CC4)C3)nc12 C1(NC(C(Br)=C(C)C)=O)CN(C(=O)C(C2CCC(=O)N2)C)CCC1C(F)(F)F c1(OC)ccc(C=CC(=O)NC2(C)CN(C(=O)C(C)N3CCC3)C2)cc1 C12(CC)CN(C(C3(C)CCOC3C)=O)C(CNC(=O)C=CC(C)(C)SC)(C1)C2 Cc1nnccc1C(=O)N(C)CC1(NC(c2cc(Br)sc2C)=O)CC1 C1(C)(C(N(CCCN(C)C(c2cccc3c2CCS3)=O)C)=O)CC(C2CC2)=NO1 N1(C(=O)OC)CCCC(NCC(C)NC(=O)Cc2cc(C)on2)C1 N1(C(C(C)NC(CC)(C)C)=O)CC2CCC1C(CNC(=O)C(C)O)C2 C(=O)(C(CC(C)C)NC(=O)NC)N1C(CN(C(C(F)=CC)=O)CC)CCCC1 c1(C(=O)NCC(CCNC(c2n(CC)ncc2)=O)O)c(Cl)c(C)nn1C N1(C(CNC(C(OC)OC)=O)=O)CCC(C)(O)C1 c1(CC(=O)NC(C)C(C)NC(=O)CCCCC(N)=O)cn2c(n1)CCCC2 C1(CNC(C2=CCCCC2)c2nnnn2C2CC2)CCc2c[nH]nc2C1 N1(C(CN(C)CC)=O)CCCC12CCN(C(C1CCC3CC3C1)=O)C2 C#CCC(C)C(=O)N(C1CC(Oc2ccccc2)C1(C)C)C(C)C C12CCCC1=C(C)C(=O)N2C(C1CNCCO1)C.CO c1(C(N2CCCCC2c2cn(-c3ccccc3)nn2)=O)nccnc1Br N1(C(CCCN(c2cccc(C=O)c2)C)=O)C2CCC1CC(O)(CO)C2 Cc1cc(=NC(=O)C(=O)NC2CCN(C(=O)C(C)(C)c3cccs3)CC2O)[nH]o1 C1(CC)CN(C(=O)CSC)CCN1C(=O)CCc1nc(F)cc(F)c1 CSC1=C(C(=O)N2CC3(C2)CN(C(c2cccc(C)c2)=O)C3)CCCC1 C(C(CO)C(F)(F)F)NC(CCn1cc(C2(C)CCOC2)nn1)=O C1(C)(NC(C(C)(C2CCC2)NC(CC=C)=O)=O)CC(O)(CO)C1 N1(C(Cc2nc(C(C)C)sc2)=O)CCCC(NC(=O)C(C)CO)C1C CC1CC(CN(CCC(=O)O)Cc2ccc(F)cc2)CCS(=O)(=O)C1 C1(CNC(c2ccc(COC)s2)=O)COCCN1C(c1cc(CF)on1)=O c1(C(=O)NC(c2ccccc2)CNC(C2C(=C)C2)=O)ccc2cc(C)oc2c1 c1(C(N2CCCC(NC(c3c(C)[nH]nc3CO)=O)CC2)=O)cn2cccnc2n1 Cc1nn(CC(F)F)c(C)c1C(=O)NCC(C)(C)NC(=O)C(C)C1CCCO1 Cc1ccc(CC(=O)NC(C(=O)NCC(C)CC2CC2)c2ccoc2)s1 CC(CC(=O)N(CCC(C)(C)NC(c1cnc(CC2CC2)s1)=O)C)CC(C)(C)C C#CC1(C(N2CCS(=O)CC2C)=O)CCN(C(c2nnsc2N)=O)C1 c1(OC)ccc(C(=O)NC(C2CN(C(c3nc(C)n(C)n3)=O)C2)C)cc1F C1(C(=O)NCCc2ncn(CC)c2)N(C(=O)C(C)SC)CC12CCCC2 Cc1cc(C)c(C(N2CCCC2C2(NC(c3sccc3C)=O)CC2)=O)o1 C#Cc1cn(C)nc1C(=O)NC1CCN(C(=O)CCN(CC)CC)C(C)C1 CCCCCCCCNC(c1ccc(NC(=O)CCCOCCOCC)nc1)=O CN1CCN(c2ccc(CN3CC4(CC4CNC(C4(C)CC4)=O)C3)cc2)CC1 c1(N2CC=C(CNC(c3ccc4ocnc4c3)=O)CC2)nc2cccc(F)c2s1 Cc1nc(NC(C2CCN(C(c3ncc(Br)cc3Cl)=O)C2)=O)ccc1Br N1(C(C2(C)CCN(C(C3CCCC(=O)C3)=O)C2)=O)CC2CC(O)CC1C2 c1(C(=O)NCCOC2CCN(C(Cc3c(C)cccc3)=O)C2)ccn(C)c(=O)c1 N1(C(=O)Cc2ccns2)CC2CCC(C1CO)N2C(=O)C(N1CCCC1)C1CC1 C1(C(=O)NCCCN(C(=O)CC2CCC2)C)CCCC12CC2 c1(C(=O)NC2C=CC(NC(=O)OC(C)(C)C)C2)ccc2c(c1)NC(=O)NC2 c1(C(=O)NCC(c2cccc(F)c2Br)F)nc(Br)n2c1CNCC2 c1(NCC23CCC(NC(CC(C)C4CC4)=O)(C2)CO3)cnc2ccccc2n1 N1(C(CC(CC)SC)=O)CCN(C(=O)C(C)=C(C)C)C(c2cccc(OC)c2)C1 C1(CN(C)C(C2(CCNC(=O)Cc3ccns3)CCC2)=O)COCCO1 C1(C(=O)NC2CCC(N(C(c3c(CC)n(C)cc3)=O)C)CC2)CCCC(F)(F)C1 c1(CC)cc(C(=O)NCc2cc(C(=O)NC3CSCC3C)n[nH]2)ns1 c1(N2CCC(C(=O)OC)C2)ccncc1C=CC(=O)OC1CC1.C(=O)C=O C12(C(N3C(C)CC(NC(C4CC4C4CCCO4)=O)CC3)=O)CC3CC1(CO)CC3C2 C(=O)(CCC(=O)N(C)C)N1CC(C(N)=O)(CNC(c2n(CCC)ccc2)=O)C1 c1(C(=O)NC2(C)CC(NC(COCCC)=O)C2)nccn2nccc12 C12(C(=O)NCc3nc(C4CC4)n[nH]3)CCCC1CN(C(=O)C(O)C1CC1)C2 C1(NC(c2c(C)ocn2)=O)CN(C(C2CCC3CC3CC2)=O)C2(CCC2)C1 C1(NC(c2ccc(CC)s2)=O)CC12CCC(NC(=O)C(COC)N(C)C)CC2 C1(C(=O)NCC2(C(N3CC(OCC(C)C)C3)=O)CCC2)CCCC(C)(C)C1 c1(C(N2C(C(C)(C)CNC(c3cnns3)=O)CCC2)=O)ccc(N)cc1Br N1(C(C2N(C(c3cccnn3)=O)CCN(C)C2)=O)CCC2(CNC(=O)C2)C1 c1(C(=O)NC2CC(C(=O)Nc3c(C)nsc3)C2)c(C)ccn1C CC(C(=O)NCC1CC1C(=O)NCCCCO)NC(=O)C1CC1 N1(C(C(C)N(C(C(C)OCC#C)=O)CCC)=O)CC(=O)N2CCCC2C1 c1(C(=O)NC2(C)CCN(C(=O)CSCC(N)=O)C2)cc2ccsc2c(O)n1 C(C(C)(O)C(=O)N1CC(CN(C(=O)CCC2(C)CC2(F)F)C)C1)OC C(CC(CC)C(=O)N(CC(C)CNC(c1cccc(C)c1C(F)(F)F)=O)C)=CC C=CC(C)(CC)C(=O)N1CCCCC(CNC(=O)Cn2nc(C)cc2C)C1 Cc1cc(Cl)ccc1C(=O)N(CC(O)CNC(c1cnc(O)n1C)=O)C C(=O)(C(C)C(C)C(C)(C)C)NCCC1(OC)CN(C(C2(C(=O)NC)CC2)=O)C1 C(=O)(C1=Cc2cccc(Br)c2OC1)N1CC(N(C)C(C23CCC(CC2)O3)=O)C1 c12ccccc1S2.c1(C(=O)NCC2(COCC)COC2)cccc(OC)c1 CC1OC2(C(=O)OC3CC(C)(C)C3CNC(=O)OC(C)(C)C)CC1C2 C1(C(=O)NC2CN(C(CCOCCC)=O)CC(F)C2)Cc2ccc(C)cc2S1 c1(NC2CC(CNC(Cc3cc(COC)on3)=O)C2)cc(=O)n2oc(C)cc2n1 c1(C(=O)NC(c2cccc(N3CCCC3=O)c2)C)cc(O)nc2c(Br)cccc12 N1(C(c2c(C)n(C)cn2)=O)CCC(C2CN(C(=O)C(F)C(C)(F)F)C2)CC1 C1(C(N(C)CCc2ncon2)=O)CNC(=O)CN1C(C1CSC1)=O C(c1ccc(SC)cc1)=CC(N1CC(COC)(CNC(C2CC2(F)Cl)=O)C1)=O c1(C(=O)NC(Cn2cc(-c3cccc(OC)c3F)nn2)C)ccc([N+](=O)[O-])cc1 n1(CC)cc(C(=O)N(C2CCN(C(c3ccc(C(N)=O)o3)=O)C2)C)nn1 c12cc(Cl)ncc1NC2=O.c1(OC)ccc(C(=O)NCc2cnc(C)nc2)cc1 Cc1cc(C(=O)NCC2CC(C(=O)NCCc3cncs3)=NO2)cc(F)c1 CCC(C)(C(=O)NCC1(CNC(=O)CCSc2ccccc2)CCC1)C(N)=O C1(O)(C(C(=O)N(C)CC2(O)CN(C)C2)NC(C(CSC)C)=O)CCCCC1 N1(C(CCCC(=C)C)=O)CCCCC(C2CN(C(C3CCOC3C(C)C)=O)C2)C1 C1(C(=O)NC(C2(C(=O)NC3CCC(F)(F)C3)CC2)C)COCC1(C)C C(=O)(C(O)CCS(C)=O)N1CC(COC)(CNC(C23CCCN2CCC3)=O)C1 C(c1ccncn1)=CC(=O)NCC1C(NC(c2cc(OC)no2)=O)CCC1 C1(CC(N2CC(N(CC(C)C)CCO)C2)=O)CC(C)(C)CN1C(c1cc(F)c[nH]1)=O C1(NC(NC(CC)CCC=O)=NCC(C)F)CCc2cc(OC)ccc2C1.OC Cc1ncc(CN2CCC(CNC(c3cc(C(F)F)[nH]n3)=O)C2)o1 N1(C(c2c(CCC)n[nH]c2)=O)CCN(C(=O)C(C)=Cn2ccnn2)CC(C)(C)C1 C1(NC(C2(F)CN(C(CC3CN(C(C)=O)C3)=O)C2)=O)CCCN(CCO)C1 c1(C(=O)NCC(c2cccnc2)NC(CSCC=C)=O)ccc2c(c1)CC2 N1(C(C2(C)CCCCCC2)=O)CCC2CCC(C1)N2C(=O)Cn1cnccc1=O C1(F)(CNC(c2cc(O)ncn2)=O)CCC(NC(C2CC(CF)C2)=O)C1 c1(C(=O)NCC2C(CNC(c3c(C(C)C)onc3)=O)C2)noc2c1COCC2 C(C(O)C(=O)NC1CC1CNC(=O)Cc1csc(Br)n1)=CCCC CCC(CC)CC(=O)N(C1CCC(NC(C2CSCCS2)=O)CC1)C N#CC1CCCN(C(C2CC2C2CN(C(=O)Cc3ccc(C(F)(F)F)[nH]3)C2)=O)C1 Cc1ccc(F)c(OCCNS(N)(=O)=O)c1 C1(C(N2C3CC(CN(C(C(C=CC)O)=O)C3)C2)=O)CN=C2N=CNN2C1 c1(-n2cc(C3N(C(C(C=C)NC(C)=O)=O)CCCC3)nn2)c(C)cccc1Br Cn1cnc2cccc(C(=O)NC3CCN(C4CCNCC4)C3=O)c12 c1(CC)cc(CC)[nH]c(=NC2CN(C(=O)CC(F)F)CC23CCOCC3)n1 N1(C(C(c2n(C)ncc2)O)=O)CCN(C(=O)CSc2nc[nH]n2)C(C2CCC2)C1 c1(C(=O)NC2CCN(C(C3CCC(N(C)C)CC3)=O)C2)cnc2c(n1)CCCC2 CN1CC2CCCN(C(C3CCOCC3NC(=O)C=Cc3ccncn3)=O)C2C1 C(=O)(CC(C)(C)C)NC(C(=O)N(C(C)C(C)(C)C)CCc1ccccc1)=O Cc1ccc(C(CC(=O)OCC(=O)NC(=O)OC(C)(C)C)NC(N)=O)cc1 c1(C(=O)NCC(C2CCCC2)NC(CSCCC(C)C)=O)cc(N)ccc1F CC1(C)CCCC(NC(=O)CC2CN(C(=O)CCC3CCN(CCO)CC3)C2)C1 C(=O)(C1=Cc2ccccc2C1O)NC(CCNC(C(CC(C)C)C(C)C)=O)(C)C N1(C(C(Cn2cncn2)NC(C=C(C)C)=O)=O)CCCCC1CF N1(C(CN(C(=O)CCOCCCO)C2CC2)=O)CC(O)C2(CCCC2)C1.C(CN)OC C1(NC(=O)NCCOCCCN(C(=O)CCSC(F)(F)F)C)CCC(C2CC2)C1 N1(C(CN(C)C(N)=O)=O)CCN2CCN(C(=O)CCCc3cnn[nH]3)CC2C1 c1(C(N(C)CC2CCC(NC(c3c(C)cccn3)=O)CC2)=O)cnn2ccsc12 C(CN=c1[nH]c2c(C)cccc2o1)NC(CCC1CC(OC)C1)=O c1(-c2onc(COC)n2)sccc1C#N C(=O)(C1CCCc2nc[nH]c21)N1CCCC(CNC(c2n(C=C)ncc2)=O)C1 N1(C(C(c2ccn(C)n2)C)=O)CCC(NC(C2(C)CCOC2)=O)C1 Cc1ccc(C(=O)NCC2CC3CC(C2)N(C(=O)CC(C)(C)O)C3)c2c1CCC2 N1(C(C(C2CCOCC2)OC)=O)CC(O)(C(C)NC(=O)CN2CCCC2)C1 C#CC1(F)CN(C(c2ccc(CNC(C3(CCC)CCC3)=O)cc2)=O)C1 C1(NC(C(C)NC(C)=O)=O)CN(C(=O)CNC(c2cccc(Br)c2)=O)CC1(C)C c1(CCC)cc(C(=O)NCC(CC)(CC)NC(=O)C(C2(O)CCCC2)F)c(C)o1 Cc1c(C(F)(F)F)n[nH]c1C(=O)NCC1CCC(NC(c2cc(Cl)ns2)=O)C1 C(=O)(CCCC(C)(C)C#N)N1CC(O)(C(C)NC(C2C(CC)N(C)CC2)=O)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2(CC2)CC1CNC(=O)C(F)C(F)(F)F C(C1CCn2ccnc21)NCCC1C(O)CCC1 c1(C(=O)NCC(=C)CCNC(=O)C(c2ccc(F)cc2)=O)cnc2[nH]ncc2c1 C(=O)(CN=c1[nH]c(=NCCc2cccs2)[nH]c2ccsc12)N(CC)CC CCS(=O)CC(=O)N1CC(O)CC1CNC(C1CCN(c2cc(O)ncn2)CC1)=O C1(NC(C(C=CC)O)=O)CC2CCC(C1C)N2C(c1cc(O)ccc1[N+](=O)[O-])=O C1(C(=O)NCc2sccc2Cl)CC2CCC(C1)N2C(C1CC(=C2CC2)C1)=O N1(C(c2cc(C3CC3)ns2)C(=O)NCCSC)CCN(CCNC(C)=O)CC1 c1(N2CCC(C(CC)C)CC2)cc(NCCC2CCCCC2O)nc(C)n1 c1(C(N(CCNC(C23CC(CC)(OC2)C3)=O)CCOCCO)=O)cc(F)ccc1Cl CCCC(O)CC(=O)NC(C)CCNC(=O)CCCOc1ccc(Cl)cc1 CC1(C)CC(=O)NC1CNC(=O)C(N1CCC12CCC2)=O N1(C(CC2C(C)(C)C2(C)C)=O)CC2CCCC(C1)N2CCN1C(=O)CNC1=O C1(NC(=O)Cn2ccnn2)CCCC(NC(C2CC3(C2)CC3F)=O)C1 CC(C(=O)OCc1ccccc1)C(=O)N1CCCC1C(=O)OCc1cccnc1 Cc1sc(NC(c2c[nH]nc2OCC(F)F)=O)nc1C(F)(F)F C1(C)(C(N2CCC(CCOC)CC2)=O)CC12CCN(Cc1cc(Br)co1)CC2 C(C)(CNC(C1C=CCNC1)=O)(C(F)(F)F)OC C1(C(N2CCC(O)(CCNC(CCCC#C)=O)C2)=O)CCCC2(CCOCC2)O1 CC1(C)CCc2c(C(N3CCC3CNC(=O)Cn3nnc(=N)[nH]3)=O)n[nH]c2C1 C1(N(C(c2nccn2C)=O)CC)CCN(C(=O)CCc2ccncc2Cl)CC1 c1(C(=O)NCc2c(C(=O)NCCOCC(C)C)cco2)ccnc2cc[nH]c12 Cc1nccc(CCC(N2CC(O)CC2CNC(c2cc(CF)on2)=O)=O)n1 c1(C(N2CC(C(C)NC(=O)CCC(=O)N(C)C)C2)=O)ccc2nccnc2c1 Cc1cc(C(=O)NC(CNC(=O)C(C(C)O)N(C)C)C(C)C)[nH]c1C c1(C(=O)NCC2CCCC(NC(c3ccon3)=O)C2)ccc2sccc2c1 Cn1nc2c(c1C(=O)NC1CC(O)CN(C(c3nncn3C3CC3)=O)C1)CCC2 CC1(C(=O)NCCNC(N)=O)CCCN1C(=O)Cn1cnnc1O Cc1cc(C(=O)NCC(C)(C)NC(=O)Cc2cnns2)c(C)n1-c1ccncc1 C1(C(F)(F)F)CC=C(CSc2ccc(Cl)c(F)c2)CC1 C12(CN=[N+]=[N-])CC3CC(C1)CC(C(=O)Nc1cc(Cl)ccc1C#N)(C3)C2 N1(C(c2c(C)csc2)=O)CCOC2CN(C(c3ccc(N)c(Cl)n3)=O)CC12 N1(C(C(C)N(C)C)=O)CCC2(CC1)CC(NC(=O)CCCCC(N)=O)C2 N1(C(CNC(C=CC(C)C)=O)C(F)F)CCN(C(=O)C(C)O)CC1 N1(C(C(CN(C)C)N(C)C)=O)CC2(NC(=O)CCCCl)CCCC2(F)C1 CCCCC(C(=O)NC1CCN(C(c2ccc([N+](=O)[O-])cn2)=O)C1(C)C)C(C)C N1(C(CC(C)SC)=O)CCN(C)C(C(=O)Nc2cnc(C)nc2C)C1 CC(C)CCC(F)C(=O)NCC1CCC(C(=O)NC(CO)C(C)(C)CO)C1 N1(Cc2n(C)c(-c3cccnc3)nn2)CCCC2(CCS(=O)(=O)C2)C1 CCCCC(CNC(=O)CC1CC2CC2C1)NC(C1(C)C=CCC1)=O c1(OC)cccc(C(=O)NC(C)(C)C(C)NC(=O)Cn2cnc(C(N)=O)n2)c1 C1(OC)CCC(C)(C(=O)NC2CC3C2CCN3C(c2ccc(O)nc2)=O)CC1 C1(NC(C(C)OCCCC)=O)(CF)CCN(C(=O)Cn2cnc(C(F)(F)F)c2)C1 C(=O)(C(C)(CN)OC)SCP(C)(C)=O.C(C(C)NC(=O)COCCOC)OCC CC(C)C(O)C(=O)N(C1CCN(C(c2ccc(-c3ccco3)[nH]2)=O)C1)CCO C(=O)(C(C)(F)C(=O)NC1CN(C(=O)CC2CCCN2C)C1)OCC c1(C(N2CCCC(CC)C2C(=O)OC)C(=O)NCC(=C)C)ccnc(Br)c1OC C(=O)(CC(O)C(C)(C)C)NCC1(NC(c2nc(CC)oc2C)=O)CCCCC1 CC1CC2(CCN(C(=O)CN3CCCC3)CC2)CN1C(=O)CNC1CCN(C)C1 N1(C(C(CCC)NC(C2CCCOCC2)=O)=O)CCC12CC(O)C2 C(=O)(CCP(C)(C)=O)N1C(C(=O)OC)CC(n2cc(CCC3CCOC3)nn2)C1 Cc1c(Cl)ccnc1C(=O)NC1CCC(C)(CNC(c2[nH]cnc2C#N)=O)C1 n1(CC)ncc2cc(-c3nnc(C4CCCCS4)o3)c(C)nc12 c1(C(=O)OC)cc(C(=O)NC(C)C=CC(=O)N(C(C)C(C)(C)C)C)no1 N1(C(C(CC)=CC)=O)CCC(O)(C(C)NC(c2ccn(C)n2)=O)CC1 N1(C(c2ccc(Cl)cn2)C(=O)NCCC)CCSC(C)C1C C(CCC)(C(O)C(=O)N1CC2CC3CC2C1C3)NC(C(C=C)OC)=O c1(C(N2CCC(NC(c3cc(O)nc(Cl)c3)=O)C(O)C2)=O)ccc2cc[nH]c2c1 CC1(NC(C2CCCCO2)=O)CC(C(N2CC(c3ncc[nH]3)C2)=O)C1 N#CC1CN(Cc2occc2Br)CC1N=c1ncnc2[nH][nH]cc1-2 C(=O)(C(C)CC(F)F)NC1(CCCNC(c2nc(C)n(C)n2)=O)CC1 N1(C(C2CCC(C)C2)=O)CC(C2(NC(=O)CCN3CCCC3=O)CC2)C1 c1(SC)ncccc1C(C)NC(C)C(C1CCCCC1)=O C12(NC(C3(OC)CCC3)=O)CC(CNC(=O)COC3CCCCCC3)(C1)OC2C Cc1ccc(C(C)(C)CC(=O)N2CCC(NC(C34CC(C(=O)O)C3C4)=O)CC2)cc1 C(=O)(C(C)C(C)C1CCCCC1)N(CCCN(C(=O)OCC)C)C.C(CO)N c1(C(N(CCCN(C(C(C(CC)O)(C)C)=O)C)C)=O)cc2c(cc1F)OCO2 C1(CN(C(c2ccc(OC)o2)=O)C)CCCCN1C(=O)CCCC1CCCO1 c1(C(=O)NC(C2CN(C(C3CCCN3C3CC3)=O)C2)C)cc(C(N)=O)co1 C1(CNC(CCCC=C)=O)CN(C(=O)CN(c2ncccn2)C)CCC1C N1(C(CCC=CC)=O)C(CNC(=O)CC(C)CCCCC)CC2CCCCC12 O=C(CCCn1ccnc1)NC1CCC(C(N2CCC(n3cncn3)C2)=O)C1 C1(NC(C(CSC)C)=O)CN(C(=O)CCCCCN(C)C)Cc2ccnn2C1 C1(C(N(CCCN(C(CCCOC)=O)C)C)=O)CCCN2CCCC12 N1(C(c2cc(OC)ncn2)=O)CCCCC(CCC(=O)N(C(C)CO)C)C1 Cc1cc(C(N2CCC2CNC(c2cccc(CCN(C)C)c2)=O)=O)nc(C)c1 c1(OC)ccccc1C(C)CC(=O)NC1CC1NC(=O)CSC(F)F c1(C(N2C3CN(Cc4ccc(OCC#C)cc4)CC32)=O)ccc(=O)n(C)c1 c1(C(=O)NCC(c2ccccc2)NC(C2C(C#C)C2)=O)cc(Cl)c(Cl)cc1C c1(C(=O)NC2CC(CNC(C34CCCN(CC3)C4)=O)C2)cc2ccnc(Cl)c2s1 C(=O)(CC(C)C(C)(C)C)NC1C(C=C)CN(C(=O)COc2ccccc2)C1 CCCCC(C)(F)C(=O)N1CC(F)CC1CN(C(=O)CC(C1CC1)C1CC1)C C(=O)(C1=CC2(CCOCC2)C1)N1CCC2CCN(C(C(CCC(C)C)O)=O)CC21 N1(C(CCC#C)=O)CCCC(O)(CNC(c2ccccc2Cn2ccnc2)=O)C1 C1(C(=O)NCC=CC(=O)NC2CC(C)C2)CCCC12CCC2 c1(-c2cc(CNC(CCCC=C)=O)n[nH]2)cc(C)ccc1[N+](=O)[O-] c1(C(N(CC(C)N(C(C(C)SCC)=O)C)C)=O)cnc2cc(C)ccn12 N1(CC(=O)NC(C)C)CCCC(NC(C2CN(C(C)C)CCO2)=O)C1C O=C1OCCC12CN(C(c1ccc(F)cc1)c1cnc(-c3ccc(F)c(F)c3)s1)C2 C(=O)(C(C(=O)N1CCC(NC(C2CC(N(C)C)C2)=O)C1)C(C)(C)C)OCC c1(NC(=O)COC(=O)CC(C(F)F)c2cccc(F)c2)ncc(Cl)cc1[N+](=O)[O-] N1(C(CC)=O)CSCC1C(=O)NCC1CC1NC(=O)COCCCF C(=O)(CCCCN(C(=O)C(C)c1ccco1)C1CC1)N(CC#C)CCO N1(c2nc(CC)cc(CC)n2)CCN(C(C2CCCCN2C)=O)CC(C)(F)C1 C(=O)(C1=COCCC1)N(CCCN(C)C)CCNC(C1(C(C)(F)F)CCOCC1)=O c1(C(N(C(C)C(=O)N(C(C)CC(N)=O)C)CC)=O)nc(O)sc1C N1(C(c2[nH]c(=NCC)sc2)=O)CC(C2CCCN(C(C3(C)C=CCCC3)=O)C2)C1 CN1CCC2(CCN2C(=O)C2=CCN(C(c3ccc(CO)nc3)=O)C2)C1 CCCCC(O)CC(=O)NC1(C)CCN(C(c2cc(C#N)no2)=O)C1 C1(C(N2CC(CNC(C3CCC(OC)CC3)=O)C(O)C2)=O)CN(C)CCN1C C=CC1(CC(=O)NC(C)CC2CN(C(C3CC=CCC3)=O)C2)CCOCC1 N1(C(CCSC)=O)CCN(C(c2cc(F)ccc2F)=O)C(C)CC1C C1(C(N2CC(OC(C)C)C2)=O)CCN(C(C2CCCCC2)=O)CC1O C1(CNC(CCc2cc(C)no2)=O)CCCC2CN(C(=O)CC(C)N(C)C)CC12 C=C(C)CC(C)C(=O)NCC1N(C(c2cc(OC)ccc2F)=O)CCC1(C)C Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CCC=CBr)c(O)c(C)n1 c1(C(C)(C)C)ncc(C(=O)NCCC2CC(NC(=O)CCNC(=O)CO)C2)[nH]1 c1(OC)c(Cl)ccc(C(N2CCCC(CN(C)C(C3CCCO3)=O)C2)=O)c1F C(=O)(C#CC1(C)CCCO1)N(CCC)CCNC(c1cc(C(F)F)cc(Cl)c1)=O Cc1cccc(CC(=O)NCC(C)N(C)C)c1.c12cn(nn1)CC(=O)N2 N(C(=NCC(OCC)OC)NCC1CC1(F)F)C(C=C)C N1(C(C2CC=CCC2)=O)CC2CN(C(=O)C(c3ccccc3F)(F)F)CC(C1)O2 c1(C(N2CCCC2c2ccnc(C)c2)C(=O)NCCCOC)cncc(Cl)c1C c1(C(N2CC(C)(NC(CCC=C)=O)C2)=O)ccc(F)c(C)c1Cl N#Cc1cn[nH]c1C(N1CCCC(N(C(=O)C=CSc2ccccc2)CCO)C1)=O C1(SCCNC(c2ccc(N(C(=O)OCC)C)cc2)=O)COc2ccccc2C1 CC1OC(=O)NC1C(=O)N(CC(O)CNC(c1nnn(C)c1C(F)(F)F)=O)C Cc1cc(C(N2CCOCC2CNC(c2cnn3c2CCC3)=O)=O)cc(C)c1N c1(C(N2C(CCNC(CCOCCC)=O)CCCC2)=O)ncc(F)cc1N C(=O)(C(CC(C)C)C(C)C)N1C(C2(NC(c3cc(C)no3)=O)CC2)CCC1 c1(CC)ccc(Oc2nc(C3CN(C(C4(CO)CCCC4)=O)CCO3)n[nH]2)cc1 Cc1cc(C(=O)N(C2CCC(NC(=O)C(O)c3ccco3)CC2)C)ccc1O N1(C(C(C)(O)C(F)(F)F)=O)CCc2ncc(NC(c3cnc(Cl)s3)=O)cc2C1 C(C(CC(C)C)C(=O)NC(CNC(C1CC1C)=O)C1CC1)OC N1(CC)CC(C(=O)NCC2CCCN(C(C3CNC(=O)N3)=O)C2)CCC1=O N1(C(C(=O)NCCCCCNC(c2nn(CC)c(O)c2)=O)C)CCP(C)(=O)CC1 C(c1ccccc1)=CCC(=O)NC1CCN(C(c2cccc(CO)c2)=O)C1 c1(C(=O)NC(CC)CNC(c2cc(C(C)(C)C)on2)=O)cc(C)nc(C)n1 c1(C(=O)NC(CC=CC)CO)cc(CNC(=O)Cc2ccc[nH]2)nn1C C1(CCC)CN(C(=O)C#CC(C)(C)C)CCN1C(=O)C(C)P(C)(C)=O c1(CC)cccc(CC)c1CC(=O)NC1CCN(C(=O)CC2CC3(CC3)C2)C1C CC(C)(CO)C(=O)NCc1ccc(C(=O)NC2CCC2O)cc1 N1(Cc2cnc(SC)nc2)CC2CCC(C1)N2C(c1ccc(C)cc1O)=O Cc1ccc(F)cc1NC(=O)C(C)(C)NC(=O)CCc1ccccn1 N1(C(CC2CCCN(C(C)=O)C2)=O)CCCC(CCNC(=O)CSC(=N)N)CC1 C1(CNC(c2ccnc(Cl)c2F)=O)CC2(CCN(C(=O)CSC3CC3)CC2)CO1 C12(NC(c3cnc(C)s3)=O)CCCCC1N(C(=O)COCC1CCOC1)CC2 C(=O)(C1SCCc2sccc21)NCCCOCCN(C(C(CC)(C)CC)=O)C N1(C(c2c(OCC=C)cccc2)=O)CCCC(C2CC2NC(=O)CNC(N)=O)C1 N1(C(Cc2c(OC)csc2)=O)CC2CCC1CN2C(=O)C(c1ccc(Cl)cc1)=O c1(C(N2CC(NC(C(CC)C)=O)CC(C)(C)C2)=O)c[nH]c2nccc-2c1C C1(NCC(=O)Nc2cc(C)no2)CCN(C(c2cc(C)n(C(C)C)n2)=O)CC1C N1(C(c2ccc(CNC(Cc3c(C)n(C)cn3)=O)o2)=O)CC2C3C=CC(O3)C2C1 N1(C(CC2CCC(C)(C)C2)=O)CC(NC(=O)CC2(n3cncn3)CC2)CC(F)C1 C(=O)(C#CC1(C(F)(F)F)CC1)NCC(C(C)C)NC(C(C)(C1CC1)NC(C)=O)=O c1(C(=O)NCCc2cnc(NC(c3c(C)nc(Cl)cc3)=O)s2)c(F)cc(Br)cc1Br c1(-c2nc(C3(C#C)CC3)on2)cc([N+](=O)[O-])cnc1O C(C(C)(C)C(=O)NCCCCCCN(C)C(c1nc(C)sc1C)=O)NC(C)=O c1(OCC)ccc(C)cc1C(=O)NC(C)CC(C)NC(c1nnn(C)n1)=O S(=O)(=O)(c1[nH]c(=NCc2ccc(C#N)cc2)ccc1Br)NCC(C)CO c1(C(=O)NC2CC(NC(CCCC=C)=O)C2)cc(N2CCCC2=O)ccc1Cl C1(c2nnnn2CC(F)F)(NC(C(CC)O)C)CCCSCC1 C(=O)(CC(C)(C)C#N)NC1CN(C(CS(=O)(=O)NC(c2cn(C)nc2)=O)=O)C1 CC1CC(CNC(=O)C(C2(O)CCCC2)F)CN1C(C1(O)CC1)=O Cc1nc(C(C)C)ccc1C(=O)NC(CNC(=O)Cc1cccnc1F)C1CC1 c1(C(C)C)cc(C(N2CC(O)(CNC(=O)CC3CC4CC4C3)C2)=O)ns1 CC(C)CC(C(=O)N1CC(S(C)=O)C1)ONC(=O)C1(C2(C)CCCN(C)C2)CC1 Cn1nnc(C(=O)NC2CCOCC2C(=O)NCC(F)Cl)c1N N1(C(CCCSCC)=O)CC2CC1CC2CNC(c1cccc(Cl)c1O)=O CC1CN(C(=O)Cc2cnccc2Cl)CCN1C(=O)C(C)OCCN(C)C c1(OC)ccc(C)c(C(=O)NCC(CNC(=O)C(C)C(C)(C)C)OC)c1N Cc1cnc(C(=O)NC(C)C(CO)NC(c2ccnc(C(C)(F)F)c2)=O)c(C)c1 Cc1ccc(CC(=O)NCCNC(=O)C2=NOCC2)cc1Br c1(C(=O)NCCN(C(c2ccccc2C)=O)CC)cnncc1C(F)(F)F c1(C(=O)NC(c2ccccc2)C(C)NC(C2CCC(C)O2)=O)ccc2cnoc2c1 CCC(C)C(C(=O)N1CCCC1(C(N1CC(C)(C(N)=O)C1)=O)CC)N(C)C C(=O)(CCCC(=O)C1CC1)N1CC2C(CNC(Cc3c(C)scc3)=O)(C2)C1 CN1CCC2CN(C(=O)C3=CCCN(C(=O)CC4CC5(CC5)C4)C3)CC12 C1(C(=O)NC2CCC(C)(NC(C3CS(=O)C3)=O)CC2)CC1C1CC(F)(F)C1 N1(C(c2ccc(CNC(C(C)N3CCCC3)=O)o2)=O)CCOC(C)(C)C1 C#CC1(O)CCN(C(=O)NCCN2C3CCC2COC3)C1 N1(C(C2(C)CC(C)(C)C2)=O)CC2CCCC(C1)N2C(=O)C(C)(C)c1cncnc1 Cn1nccc1CC(=O)NC(CNC(C1(CC(F)F)CC1)=O)C1CC1 CC(C)CC(O)C(=O)NCCCCn1ccnc1C N1(C(CCOCCCOC)=O)CCCC(C2CCN(C(=O)C(C)O)CC2)C1 CC1(C)C(CNC(=O)COC2CN(C(=O)C#CC3CC3)C2)CC1O N1(C(c2cncc(C)c2)=O)CCC2(CCCN2C(c2sccc2C(F)F)=O)C1 Cc1ccc(NC(C2COCCN2C(=O)Nc2cc(O)no2)=O)nc1 c1(C(=O)NCCC2CC(C)C2)cncc(CNC(C2(C)CNC(=O)C2)=O)c1 c1(C(C)C(F)(F)F)cccc(NC(C2CCCN2Cc2cccs2)=O)c1 c1(C(=O)NC)ccc(S(=O)(=O)N2CCCCC2CNc2cc(Br)ccc2Br)cc1 c1(NC(C23CCCC2C3(F)F)c2n(C)nnn2)cccc(N=[N+]=[N-])c1 N1(C(c2ccc(=NC)[nH]c2)=O)CC2(CC(NC(=O)C(C)NS(=O)(=O)CC)CO2)C1 c1(C2C(SCC(=O)NC(C)(C)CNC(C3COCCO3)=O)C2)ccc(C#N)cc1 N1(C(CCCC#C)=O)CCC(NC(c2cc(I)c[nH]2)=O)C(CO)CC1 C1(C(=O)NC(C2CCCCC2)C#C)(NC(C2C(C)(C)C2(C)C)=O)CCN(C)C1 c1(OCC(=O)NCC23CCC2CN(C(=O)C(Cl)=CCl)C3)c(F)c(F)cc(F)c1F c1(C(=O)NCCC2C(C)CN(C(=O)C(C)(C)Cl)C2)cc2ncccn2n1 c1(OC)cc(F)cc(C(=O)N(CC(C)CNC(C2CCCCN2N=O)=O)C)c1N N1(C(C(CN(C)C)O)=O)CCCN(Cc2cn(C3CC3)nn2)CC1 C1(C(=O)OC)CN(Cc2cccnc2OCc2ccccc2)C(CO)CO1 CCCC(F)C(=O)NC(C1(C(=O)NC(c2nn(C)cc2O)C)CC1)C N(C1CCCOc2c(F)cccc21)C(c1ccc(CC)s1)C c1(C(N2CC3CCN(C(c4nc(Br)cs4)=O)CC3C2)=O)cc(Cl)cc2cc[nH]c12 c1(C(Cc2ccn(C)n2)=O)nc(Cl)nc2c1ncn2C.C1(O)CCCCC1(C)C=O c1(C(N2C(C)CCN(C(=O)C(C)(F)F)CC2)=O)sc2cccc(Cl)c2c1Cl C(CC(C)(C)CNC(C1CC(Cl)(Cl)C1)=O)NC(c1nc(CCC)oc1)=O C1(CCCNC(=O)CSC(F)(F)F)(CNC(C(C)OC2CCOC2)=O)CCCC1 C(c1c(F)ccc(Cl)c1F)=CC(=O)NC12C(CCN(C(C(CC)=CC)=O)CC1)C2 C1(CCC)CN(C(=O)Cc2ccc(Cl)s2)CCN1C(=O)C(C)Cc1ccnn1C CC1CN(C(C2(C)CCC2)=O)CC1NC(=O)CN(C1CCC1)C N1(C(C(C=C)O)=O)CC(OC)CC1CNC(c1ccc(OCCC)cc1)=O C1(CNC(C(C)SCC)=O)C(C2CC2)CCN1C(=O)COCC(F)F C(N=c1ccn(C2CCCCC2)[nH]1)c1c(N)n(C2CCOCC2)nc1 CC(C)CC(C(=O)NC1CCOC1)ONC(c1cnn(C(F)F)c1)=O N1(C(c2cn(C3CCOC3)nn2)=O)CC2CCC1CN2C(=O)C(O)CC(F)F CC(C)C(F)(F)CNC(=O)CCOCCNC(=O)CCC1OCCO1 C(=O)(CCCCNC(=O)C(F)C(C)C)NC(c1nccn1C)CC C(=O)(CC(C(F)F)n1ccnc1)NCCCC(C)(C)NC(CN(CCC)C)=O c1(C(N2CC(C3(NC(CCc4n[nH]c(=N)s4)=O)CC3)C2)=O)ccc2cncn2c1 c1(C(=O)NCC(CSC)OC)ccc2c(n1)OCCO2.C1(C(=O)NC)CCCN1C=O N1(C(C2CCCN(c3nc(C)cc(C)n3)C2)=O)CCC2(N(C)CCO)CCCC12 c1(CSC)cccnc1C(=O)NCC1N2CCC(CC2)C(=O)N1.C(C)=O.C1CC1 C1(C(=O)N(Cc2ccc(C(N(C3CCCC3)CC#CC)=O)o2)CC)CC2(CC2)C1 N1(C(C2(N(C)C)CC2)=O)CC2CC(C(=O)NC3CC34CCC4)(C2)C1 C(=O)(CCCc1ccccn1)NCCC(C)N(C(CCOC(C)C)=O)C c1(C(N(C2CCC(NC(C3CCCSS3)=O)CC2)C)=O)cccc2c1OCO2 N1(C(C2C(COC)C2)=O)CC2(CCC(CNC(c3nc(C)c(C)[nH]c3=O)=O)O2)C1 N1(C(C2C(C)(C)COCC2)=O)CC2CC(CNC(=O)C3=CCC3)CC1C2 CC1OC2(c3cn(C4CCOCC4(C)C)nn3)CC1(CO)C2 C1(C(N2CC(NC(c3cn(CCOC)nn3)=O)C(C)C2)=O)CN=C2N=CNN2C1 CS(=O)(=O)c1ncc(C(=O)NCC2(F)CCC(NC(=O)C#CC3CC3)C2)s1 c1(NC(C)=O)ccc(C(=O)NCC(C)(C)NC(c2c[nH]c(Br)c2)=O)nc1 CCCCCC(O)CC(=O)NCc1nc(C(=O)N(C2CCCC(C)C2)C2CC2)co1 C1(NC(C2(CC#C)CCOCC2)=O)CCN(C(=O)C=Cc2ccccc2)C(C)C1 c1(C(C(=O)Nc2cccc(C(C)F)c2)NC(C2CC2(Cl)Cl)=O)c(C)cccc1Br N1(C(c2cc(CCC)oc2C)=O)CCC(NC(=O)CC2(C)OCCO2)C(CC)C1 N1(c2c(-c3ccccc3)cnc(C)n2)CCCC2(CCN(C(=O)CC3CC3)CC2)C1 C1(C(=O)NC2CC(CCNC(c3ccc(C(N)=O)[nH]3)=O)C2)CCc2nncn2C1 C(CCCC(=O)N(CC(O)C1CCC1)C)N(C(C1C(C(=O)OC)CC1)=O)C C(=O)(C1CCN(C)c2ccccc21)OCc1cncc(C)c1 C12(C(=O)NCCCN(C(c3c[nH]c(C)c3)=O)CC)CC1COC2(C)C c1(C(=O)NC2C(CNC(c3c(C)coc3)=O)C2)cc([N+](=O)[O-])c2nsnc2c1 C1(CC)CN(C(=O)C(C)(C)CN(C)C)CCN1C(=O)C(F)=CC1CC1 C(CC(C)(C)C(=O)NCC1CC1c1ccco1)NC(CC1(C)CCOCC1)=O C(=O)(C#CC(C)(C)C)NC(CNC(C1CCN(CC(C)C)C1)=O)(C)C1CC1 C(=O)(CC1=CCCCC1)N1CCC(CC(=O)NC(C#C)(C)C2CCCC2)C1 N(C(=NCc1ccc(Br)cc1F)NCC(C)(C)C1CC1)C1C(C)C1 C1(C(N2C(CNC(COCC(=O)NC)=O)CCC2)=O)CCCC2(CCC2)C1 Cn1cncc1C=CC(=O)N(C1CCC(NC(=O)Cc2cnoc2)CC1)C c1(OCCC)ccccc1C(=O)NCCN(C(=O)C(C)(C)C)C N1(C(C2(CC)CC2)=O)CCSC(C(N2CCC(N3CCCC3)CC2)=O)C1 c1(OC)c(C(=O)NC2CCN(C(C3CCC3F)=O)CC2)cccc1C(F)F Cc1[nH]nc(C(=O)NCCC2CCCN(C(=O)C(C)(C)c3cnc[nH]3)C2)c1Br S(=O)(=O)(c1cc(C(F)(F)F)ccc1N1CCn2ncnc2C1)N(C)Cc1cscn1 C(=O)(C#CC1CCCO1)NC1CCN(C(c2c(Cl)sc(C)c2C)=O)C1 C1(C(CNC(=O)Cc2ccno2)NC(=O)CNC(=O)C(F)(F)F)CCCCC1 N(C1CC(C)(C)CCc2ccccc21)C(C)C(c1ccccc1)O Cc1nnc(CCNC(=O)C=CCC(C)(C)NC(=O)CCCc2ncco2)n1C c1(C(=O)NC(CCC)CNC(C2CCS(=O)(=O)C2)=O)ccc2nn[nH]c2n1 Cc1cccc(C2CC2)c1C.N1C(NCc2cccs2)=NCc2cccc(c2)C1 N1(C(Cc2ccc(C)o2)=O)CC2CC1CN(C(=O)C=CSc1nc[nH]n1)C2 C1(CC=C)COCC1NC(C1CCC(NC(C2CC(C)C2)=O)C1)=O C(C#Cc1ccccc1Cl)N1CCC(N(C(=O)C(O)C(C)(C)CC)CCC)C1 c1(C(=O)N(C)C)ccc2cccnn12.Cc1oc2cc1-c1csc(n1)NC2=O Cc1cc(F)c(C(N2CCCC(NC(c3ccc(O)cc3C)=O)CC2)=O)c(Br)c1 c1(NC(C(CCF)NC(=O)OC(C)(C)C)=O)cc(Cl)ccc1F c1(CN=C(NCC2C(C)C2)NC2CCC2)nn(C)c2ccccc12 c1(C(=O)NCC2CCN2C(=O)C(O)CC2CCCCC2)nc2cccnc2s1 CC(CNC(=O)CN(C)C)CC(=O)N1CC(S(C)=O)C1 C1(CNC(c2scc(OC)c2)=O)CCN(C(=O)Cn2cncn2)CC1O N1(C(=O)Cc2ccc3cccnc3c2)CCSCc2ccc(Br)cc21 Cc1cc(NC(C2(F)CC=CCC2)=O)cc(C(C)C)c1 N1(C(C)=O)CCCC(c2nc(C3CC3)nn2C(C2(C)CC2)C)C1 C12(NC(CN(CCC)C)=O)CCCC(CN(C(c3ccc(C(N)=O)o3)=O)C1)C2 C1(COC)CN(C(=O)C(O)c2ccsc2)CCN1Cc1ccccc1 c1(C(CN(CC)CC2CCCN2C(C)C)(C)C)ccc(C(F)(F)F)cc1 c1(CCNC(=O)Nc2scc(C(=O)OC)n2)c[nH]c2cc(C)ccc12 N1(C(CC(CCC)C)=O)CC2CCCC1(CNC(c1ccc(C)cn1)=O)C2 C1(C(=O)NCC(CNC(C2(C(C)C)CNC(=O)C2)=O)(C)C)CC(C2CC2)=NO1 c1(COC(CC=C)CNCc2ccc(C)o2)ccc(F)cc1 N1(CC(=O)NCC2CN(C(C(CCC)O)=O)CC2O)OC(C)(C)CC1=O C1(CC(=O)NC(CC#C)CC)CCCN(C(=O)C(C)(C2CC2)OC)C1 C1(C#N)(C(N2CC(n3cc(CNC(CCOC(C)C)=O)nn3)C2)=O)CCCO1 c1(C(=O)NCC(Cn2cc(C(N3CCCC3)C)nn2)OC)snnc1C1CC1 N1(C(C(F)=CC)=O)CCCC12CCCN(C(=O)CCOC1CCCCC1)C2 C1(CCNC(Cc2ncc(CC)[nH]2)=O)CC(F)(F)CN1C(C1C=CC=CC=C1)=O CCCCC(CC)CC(=O)N(C)CCOCCNC(c1cc(C#N)ccc1O)=O C(CCC(F)(F)F)(S(CC1CCC(C)CC1)(=O)=O)C1CC1 C(=O)(CC1=CCN(C(c2coc(C(C)C)n2)=O)CC1)NC(c1onc(C)n1)C c1(NC(=O)COCCCN(C(C2CC(F)(F)C2)=O)CC2CC2)cc(O)ccc1Cl c1(OC)ccc(C(N2CCC(CN(C)C(C3CCOC3C3CC3)=O)CC2)=O)nc1 N1(C(c2c(C)con2)=O)CCC2(CCCCN(C(C3CC3C3CC3C)=O)C2)C1 C(N=c1ccnc(NCc2nn(C)c(OCCC)c2C)[nH]1)C1(CCC)CCC1 C1(CC(=O)NC2(CCNC(c3ncn(C(C)(C)C)n3)=O)CC2)NC(=O)NC1=O C1(COC)(NC(=O)CN(C)CC2(F)CC2)CCN(C(=O)CC(C)CN(C)C)C1 c1(CNC(CC2N(C(CN3C(C)CCC3)=O)CCC2)=O)ccc(C(N)=O)nc1 c1(-c2cn(C(C)C(=O)NCC3(CF)CCNC3=O)nn2)ccc2cnccc2c1 C(CC(C)(O)CC)NC(C(CN(C)C)NC(C(C)OCCC#C)=O)=O c1(CC(=O)NC2CC(CNC(C(C)NS(C)(=O)=O)=O)C2)cn2c(n1)CCCC2 N1(S(c2cn(C)nc2)(=O)=O)CC2C3CCC(O3)C2C1.c12ccccc1[nH]c(=O)[nH]2 C(C(=O)Nc1cccc(Br)c1)(C(C)CC(C)(C)C)NC(C1CC(C)CC(C)C1)C C1(C)(CC)C=C(C(=O)N(CC(C)NC(c2ccc(OCCF)cn2)=O)CC)C1 C12(NC(c3cccnc3O)=O)CCCN(C(C3CCOCC3)=O)CC1C2 c1(C(=O)NC(CN(C(=O)CN2CC(C)C2)CC)C)cnn2ccc(Cl)c(F)c12 C1(C(N(C2CC3(CC3)C2)C)=O)CC2C=CC1N(C(C1(N(C)C)CCCCC1)=O)C2 n1(CC(=O)NCCC2N(C(C(C)(O)C3CCC3)=O)CCCC2)cnc([N+](=O)[O-])n1 N1(C(C2C(OC)C2)=O)CCn2ncc(CNC(=O)C(C3CCCCC3)O)c2C1 C1(C(=O)NCCC(=C)CNC(=O)CN2CCCCC2=O)CCCC(C#N)C1 C1(NC(c2c[nH]nc2-c2cccs2)=O)CCN(c2cc(C3CC3)ncn2)CC1F c1(C(=O)NC2CCN(C(CSC)=O)C(C3CC3)C2)c2c(nn1C)CCSC2 c1(C(N2CCC(C)C2CNC(=O)CCCC(F)(F)F)=O)cccn2ncnc12 c1(CNC(C(n2c(C)ncc2)C)=O)ncccc1C(=O)N(CCO)CC1CC1 CC(C)CC(C(=O)NC1CC(C)(C)C12CC2)NC(c1cccc(O)n1)=O C1(C(N(CCNC(=O)CC2CCCC2)CC)=O)CC2CC1CC2(F)F CC(C)C(F)(CNC(C1CCN(C)C(=O)C1)=O)C(=O)NCCC1(C)CCOCC1 C(=O)(CS(N)(=O)=O)NC(c1ccccc1)CC1(NC(=O)OC(C)(C)C)CCOC1 N1(C(C(C=C)OC)=O)CCC(O)CC1C(=O)NCC1(C2CC2)CC1 C(CCC(C)(C)C(=O)N1CC(C)=C(C)C1)NC(C1CN(CC)C(=O)C1)=O c1(C(=O)NC2C(NC(CCC(CC)CC)=O)C2)cn2c(n1)CCC(C)C2 Cc1n[nH]c(C)c1C1CC(NCC(=O)N(C)C)C1 C1(CNC(c2c(CC)nc[nH]2)=O)CC2(CCC2)CN1C(C1CC1[N+](=O)[O-])=O C(C)(c1ccccc1C)=CC(=O)NC(CNC(C(CCSC)O)=O)CC(F)(F)F N1(C(c2c(C(C)=O)ccs2)=O)CC(NC(C2(C)CCCO2)=O)C2CCCCC12 c1(C(C)=O)nc(C(=O)NC(C2CCOC2)CNC(=O)Cc2n[nH]c(C)n2)co1 C1(C(=O)NC2CC(CNC(C(CC)O)=O)C2)CCCCN1C1CC1 C1(N2C(=O)CCC2)CCCN(CCC(N2CCC(Oc3ccccc3)CC2)=O)C1 C(C(CC1CC1)C(=O)N(CCCN=[N+]=[N-])C)NC(C(C)N(CC)CC)=O C1(CC)C(NC(=O)CCCOC(C)C)CCN1C(=O)CN1CCNC(=O)C1 N1(C(C(C)=NOCC#N)=O)CC=C(C(=O)NCC(C)(C)CCCO)C1 CCCC(C)(CC)C(=O)NCC1CCN(C(c2cc(C)no2)=O)C(C)C1 C(CC(C(=O)O)NC(=O)CC1CC2CC2C1)SC c1(OC)cc(C)c(C(=O)NCC=CCNC(C2CCCC(F)C2)=O)c(C)c1 C(=O)(C(O)C(C)C)N1C(CN(C(C2CCC(C(N)=O)CC2)=O)CC)CCC1 C(CC(C(=O)NCC1CSCCO1)NC(c1cc(C)[nH]c1C)=O)SC N1(C(C2CCN(CC)C2)=O)CCCCC(C(=O)NCCCC(C)C)C1 N1(C(C=C(C)C)=O)CCCC(CCC(=O)NCC2(CO)CCCO2)C1 N1(C(CCCC2C(C)C2)=O)CC(C2CN(C(c3ccc([N+](=O)[O-])cc3)=O)C2)C1 C1(C(N(C2CC(NC(C3(CC(F)F)CC3)=O)C2)C)=O)CCCCC1F CC1CCCC(CNC(C2(N(C(=O)C=Cc3cncs3)C)CC2)=O)CC1 C1(NC(C(CCSC)O)=O)CN(C(=O)C(C2CCS(=O)(=O)CC2)(F)F)CCC1O c1(C(=O)NC2CN(C(CCC(C)C)=O)C(C)CC2)cnc2c(F)cccc2c1 c1(NC(C=CCC(C)(C)NC(C2C(C(C)C)CCC2)=O)=O)cn(C)nc1C#N c1(NC(C(=O)N(CC)Cc2cccc([N+](=O)[O-])c2)=O)ccc2oc(O)nc2c1 c1(-c2c[nH]nn2)ccc(Cl)cc1O.O=C(C1=CCOC1)N.C12CCCCN1CC2 C1(CNC(C(CC)NC(C)=O)=O)C2CN(C(=O)CCn3ccnc3)CC12 C(c1cc(F)c(F)c(F)c1)=CC(N1C(CNC(COCC#C)=O)CCCCC1)=O N1(C(C2CCC(NC(=O)CCc3cscn3)C2)=O)CCCc2occc2C1 CC1C(NC(C2CC2c2nccn2C)=O)CC2CCC1N2C(c1cn[nH]c1)=O N1(C(COCCC(C)C)=O)CC2CCCC2(NC(C2CC(CCO)C2)=O)C1 C1(NC(c2cc(F)c[nH]2)=O)CCN(C(c2ccc(CO)cc2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC12CC1CN(C(C1(C)CCC1)=O)C2 S(=O)(=O)(c1c[nH]ccc1=NC1CCCC(C)C1)N(CCC)C C(N=C(NCC1(C)CCCCC1)NC1CCCSC1)c1n(C)ncc1 N1(CC)CCCN(C(C2CC2C(C)NC(c2cc(C)n(C)c2C)=O)=O)CC1 CCC(C)(C)CCNC(C1CCN(C(=O)C(C)c2ccco2)CC1)=O C(=O)(NNC(=O)COc1cccc(C#N)c1)NC1C(C(=O)NCC)CCC1 S(=O)(=O)(c1ccc(C(=O)NCCCNC(=O)C(C)=C(C)C)cc1)COCCC c1(C(N(CC(=O)NC2CN(C(C)C)C(=O)C2)C)=O)ccn2ccnc2c1 c1(C(=O)NCC2N(C(C3C(=O)NCC3)=O)CCC2)cc2c(Cl)nccc2o1 CCCC(C)(CC)C(=O)N1CCC(N(c2cc(CC)nc(C)n2)C)C1 N1(C(CCCc2ccc(SC)cc2)=O)CC(NC(=O)C=CC(F)(F)F)CC(O)C1 C(C)(C(CC(=O)N1CCCCC1C1(O)CC1)NC(c1c[nH]c(=N)c(C)c1)=O)OC C1(NC(C=CC(C)(C)NC(C2CC3C(C2)C3(C)C)=O)=O)CC2CC(O)C1C2 C1(CC#N)CN(C(c2cc(O)nc(O)c2)=O)CCN1C(c1cc(Cl)cs1)=O C1(C(=O)NC2CCC(NC(c3c(C)cno3)=O)C2)COc2ccccc2C1 N1(C(C(CC)CO)=O)CCCC2CN(C(c3ccc(OC)cc3O)=O)CC12 C=CC1(NC(C2CN(C(=O)CCN3CCCC3=O)CC2F)=O)CCOCC1 c1(C(N2CCN(C(CC3C(C)C3)=O)C(CF)C2)=O)ccc2c(c1)nc(O)n2CCO N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC2(C1)CN(C(C1CC3CC3C1)=O)CCO2 c1(CC(=O)NC(C2CCCCC2)CNC(c2csnn2)=O)ccccc1C(F)(F)F c1(C(N(C2CCCN(C(=O)CC(C)F)C2)CC)=O)[nH]nc([N+](=O)[O-])c1Cl c1(C(C)=O)nc(C(=O)NC(CNC(=O)C(C)Cc2ccco2)C(C)C)cs1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(NC(c2csc(C3CC3)n2)=O)C(O)C1 N1(C(C2(NC(C)=O)CCCC2)=O)CCC(NC(=O)CC2CC2(C)C)C(O)C1 C1(NC(c2onc(C)n2)=O)CN(C(c2scnc2C)=O)Cc2nccn2C1 c1(N2C(CN(C)C)CCCC2)nc(C)c([N+](=O)[O-])cc1Cl Cc1cc(C(=O)NCC(C)CC(=O)N2CC(C)(F)C2)c(C)[nH]1 S(=O)(=O)(c1ccc([N+](=O)[O-])c(F)c1)N(CCC(N1CCC2CCOCC2C1)=O)C C1(C)(C(=O)NCC2(CC)CC(C)(C)C2)CN(C(C2CC(C)(C)C2)=O)CC1C CC1(NC(=O)CCCC2CCC2)CC(NC(=O)C(C)(C)c2ccccc2)C1 C1(N(C(C2N(CC)CC2)=O)CC)CCCN(C(=O)C(C)O)C1 c1(C(=O)NC2C(CNC(CS(=O)(=O)NCC)=O)CC2)cnn2c1OCC(C)C2 N1(C(=O)C(c2ccc(O)cc2)O)CC2CCN(C(=O)CCc3cscn3)C2C1 C1(NC(c2cc3oc(Cl)cc3[nH]2)=O)CCC2CN(C(=O)CCC3CCC3)CC2C1 CCCCCC(C)CC(=O)NCC(C)(CO)NC(=O)C(c1cccn1C)=O Cc1cc(C(=O)NCC2CN(C(c3cccnc3O)=O)CCCO2)c(O)nc1C C(=O)(C(C)CCC)NCCCN1CCC(NC(c2nc(CCC)sc2)=O)C1 CC1C(C(=O)N2CC3CCC(C2)C3NC(C23C(=O)C4CC2C3C4)=O)=NOC1C N(C1CCCn2nccc21)C(CC1CCCN(C(Cc2c(C)ccs2)=O)C1)=O Cc1cc(C(=O)N(C2CCCN(C(C3CCCN3C3CC3)=O)C2)C)cc(C)c1N CS(=O)(=O)c1cc(C(N2CC3CC(NC(C4CCOC4)=O)CC2C3)=O)ccc1F c1(OC)cn(CC(=O)N(CC(O)CNC(c2ncc(F)cn2)=O)C)c(C)cc1=O C1(COC)(CNC(=O)C(C)Cn2cccn2)CCN(C(C2CCNC2=O)=O)CC1 N1(C(C(CCC)OC)=O)CC(NC(=O)CSCC(F)(F)F)CC12CCCC2.C(C)(=O)N N1(C(c2c(CC)ncs2)=O)CCC(C)(C)C1C(N1CCC(CC2CC2)CC1)=O c1(C(=O)NCC(CCCC)NC(C)=O)ccc2c(c1)C(=O)N(C)C2=O n1(CC(C)C)nccc1CNC(c1cnc(C2CC2)o1)c1nnnn1C c1(CC)cc(C(=O)NC2CCC(C)N(C(=O)C=CI)C2)cc(O)n1 N1(Cc2c(OCC(=O)O)cc(Br)cc2)CCCC2(C1)OCCCO2 C1(C(=O)NCC2CC(F)CN2C(=O)C(C2CCOCC2)O)CC2(CCC2)C1 c1(CC(=O)NCCCn2cc(CCCCOC(C)=O)nn2)ncc2c(n1)CCC2 C1(NC(=O)C=Cc2ccoc2)CC(NC(=O)CCCN2CCCCC2)CC1O C1(C)(NC(C(C)N(C)C)=O)CN(C(=O)C(C)(C)c2ncco2)C1 C1(OCC)CCN(C(C2CC2C(=O)Nc2cc(OC)nn2C)=O)CC1 C1(CC(=O)NCC2(C(C)NC(c3c(C)noc3)=O)CC2)CN2CCN1CC2 C1(CNC(C=CC(C)C)=O)C=CCN1C(=O)C(n1ccc(Sc2nncs2)n1)C C1(OC)CCC2(C(N3CC(F)(CNC(C4CC4Cl)=O)C3)=O)CC12 CCC(CC)C(CO)CN=c1[nH]c(=NCc2cc(Br)cs2)[nH]c2cccc(F)c12 C1(c2n(C(C)(C)C)nnn2)(Nc2cccc(O)c2)CCC2(CCCOC2)C1 C(CC)(C(=O)NCC1(COC)CN(C(c2ccc(C(C)=O)[nH]2)=O)C1)=CC C=CCC(C)C(=O)NCCCN(C(c1ccnn1C1CC1(F)F)=O)CC CS(=O)(=O)CC(=O)NCC1(C(N)=O)CN(C(c2cnn[nH]2)=O)C1 C(C(C(C)(C)C)NC(=O)Cc1nccs1)NC(C1(C(=O)OC)C(=C)CC1)=O c1(C(N(C)CCNC(C2CCCN2N=O)=O)=O)ccc(Cl)cc1Cl c1(C(N)=O)cccc(C(=O)NC2CC(NC(c3ccc(C(F)F)cc3)=O)C2)c1F C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(c2cc3ncccc3s2)=O)CCC1(C)C CC1CCC(C(=O)NCCN(CC(C)O)C(c2csc(Br)c2)=O)CC1 N1(CC(=O)N(CC(CC)NC(=O)C(C)n2cccn2)C)CCNC(=O)C1 c1(C(C)=O)cc(Br)c(C(=O)NCCC2CCCCN2C(=O)OC(C)(C)C)s1 C12CC3CCC1CN3C(=O)N1CCN2C(=O)C1.c1ccccc1.COC c1(NC(C2(C)CCN(C(CCOC)=O)C2)=O)cccc(C)c1C(F)(F)F C#Cc1cccc(C(N2CCOCC(C(=O)N(CC(C)COC)C)C2)=O)c1 NS(=O)(=O)c1cc(C(=O)NCCCCCCNC(=O)CC2=CCOCC2)co1 Cc1ncc([N+](=O)[O-])c(NC2CC(CNC(=O)CSCC(F)(F)F)C2)n1 c1(C(=O)NC2CC(NC(c3cc(CC)c(O)cc3)=O)C2)ccc(Cl)c(C)c1OC C1(N(C)C(c2occc2Cl)=O)CC2CCC(C1)N2C(C1CCn2ncnc2C1)=O N1(C(Cn2c(C)c(Cl)cn2)=O)CCCN(C(C2CCC2C#N)=O)CC1 Cc1cc(C(=O)N(C2CN(C(=O)CCCc3cnccn3)CC2F)C)c(C)cn1 C1(C(=O)NC2CCC(NC(c3ccc(O)nc3)=O)CC2)(COC)CCC(=O)N1 CC1CN(CC(=O)NC2CCCOC2)CC1C(=O)NC(C)(C)C c1(C(=O)NCC(C)N(C(C2C(C=C)C2)=O)C)ccc(C)c2cccnc12 Cn1cc2c(C(N3CCC4(C3)CN(C(=O)CC(F)F)CCO4)=O)cc(F)cc2n1 C1(C(=O)NC2(c3nc(C)on3)CC2)C2CCN(C(=O)C#CC(C)(C)C)CC12 C1(NC(CCc2n(C)ncc2)=O)CCC2CC1CN2C(c1occc1Cl)=O C1(N(C)C(c2cn(C(C)(C)C)cn2)=O)CCCCC1NC(=O)C1=C(Cl)CC1 CCC(C(=O)NCCN(C(C1CC1C(F)(F)F)=O)C(C)C)SC C(C(C(C)C(C)C)NC(C1OCCO1)=O)NC(C1(CCC=C)CC1)=O CC(C)CC(C(=O)NCCC1CCN(Cc2ccnnc2Cl)CC1)C(N)=O C1(C(N2CCN(C(C=Cc3c(C)cccc3F)=O)CC2)=O)Cc2c(F)cccc2O1 c1(CNC(C2CCC(COC)C2)=O)ccc2c(c1)CN(C(=O)CCOC(C)=O)C2 C=CCCCC(C(=O)N(CC(C1CC1)OC)C)NC(=O)C(F)C(C)(F)F C(CN=c1ccc(S(=O)(=O)N2CCNCCC2C)c[nH]1)c1ccn(C(C)C)n1 C1(CC=C)(C(=O)NCCCC(C)(C)NC(=O)C(C)C2(N(C)C)CC2)CCOCC1 C1(C(N2CCCC(N(C)C(c3cccnn3)=O)C2)=O)CCCC12CCOCC2 c1(C(=O)NC(C2CCN(c3ncccn3)C2)C)cccc(P(C)(C)=O)c1 C1(CN(C(c2ccc(OC)cc2)=O)CC)CCCN(C(=O)C(C)C(F)F)C1 N1(C(CC2(CSC)CC2)=O)CCC2(C1)CN(C(C1(Br)CC1)=O)C2 Cn1ncc(C(=O)Nc2ccc(O)cc2)c1C(N)=O S(=O)(=O)(c1ccc2[nH]c(=NC3CCN(CC(C(C)C)C)C3)sc2c1)NC1CCCC1 c1(N(C(c2c(C)cccc2Cl)=O)CC2CNC2)ncc2c(n1)NC(=O)C2 C1(CNC(=O)NC(CC)C2CCC2)CCC(c2ccccc2)O1 N1(c2nnc(C)s2)CCCC(CNC(c2coc(Cc3ccccc3)n2)=O)CC1 C1(C(=O)NCC(C)(C)Cn2cc(CO)nn2)CNCC12CCS(=O)(=O)CC2 Cc1cccc(C(=O)NC2CC(NC(C3(C)CC=CC3)=O)CC2O)c1F c1(C(=O)NCCN(C(C2(C(F)(F)F)CC(=C)C2)=O)CC)cc(Cl)nnc1O C1(NC(C(CC=C)N(C)C)=O)CCC12CCN(C(=O)CC(C)F)CC2 C(=O)(CCCC(C)NC(C1CCC(=O)N1)=O)NC(C(=O)OC)CO C1(C(=O)NCC(C(C)C)N(C)C)CC1C1CN(C(c2cccnc2S)=O)C1 CC(CC1CCCC1)C(=O)NC1CCN1CC(=O)NC1CC1 c1(COC(c2cnc(C(F)(F)Cl)o2)=O)ccncc1Cl c1(N(CCN(C=O)C)C)ncnc2ccc(O)cc12.CCO C(=O)(C1CCc2cc(OC)ccc21)NCCCNC(C(CCC)C)=O CC1(C)CC(CNC(=O)CSCc2cccs2)CN1C(=O)C1=CCOC1 N1(C(CCN(C(C)C)C)=O)CC(NC(=O)COc2ccsn2)CC(C)C1 CC(C(=O)N1CCCC(CC(=O)NCC2(CN=[N+]=[N-])CC2)CC1)S(N)(=O)=O C1(CC(=O)OCC)CCCN(C(C2CCC(=O)N2c2cn[nH]c2)=O)C1 c1(C(=O)Nc2cncc(C(F)C(F)F)c2)ccc2ccc(O)nc2c1 C(=O)(C1=CC2CCCC12)N1C(CNC(C2(C)CCN(C(C)=O)C2)=O)CCC1 c1(C(N2CCCC(CCNC(C(CC)C(C)O)=O)C2)=O)ncc(C#N)cc1C c1(NCC(N2CC(C(C)NC(C3(C)C(CC)CCC3)=O)C2)=O)cccc(C#N)c1 c1(C(=O)NCC(C)N(C(=O)C(F)C(C)(C)O)CC)cc(C)c2c(O)n[nH]c2n1 c1(C(C)C)ccc(OCC(=O)OC(C)(CC2CC2)CO)cc1 c1(C(=O)NCC2OCCN(C(C(CCCC)O)=O)C2)nc(Br)c2ccccn12 c1(C(=O)NCC2N(C(c3n(CC(C)C)ncc3)=O)CCC2)cn(C)c(C(F)F)n1 C1(CC(=O)NCCCC(C)NC(c2ccsc2Cl)=O)CC2CCC1O2 C1(C(=O)NCCC(CCC)C)Cc2c(cnn2C)N(C(=O)OC(C)(C)C)C1 c1(C(N2CCC(CNC(C=C(C)Cl)=O)C23CCC3)=O)cc2ccccc2nc1O C(=O)(C#CC1(C(F)(F)F)CC1)NC(C)CCCNC(c1nccnc1N)=O CC1C(NC(C2C(F)(F)C23CC3)=O)CCN1C(=O)CN1CCOC1=O C(=O)(CCCNC(=O)NC)NCCN(CC)CC.c1(C(=O)N)cnn(C)n1 c1(NC(C(c2ncccc2Cl)N2CC(n3ncc(C)c3)C2)=O)c(C)cccc1C N1(C(C(C2CN(C(C3CN(C)CCO3)=O)C2)OC)=O)CCc2cccc(O)c21 c1(C(=O)NCC2C(OCC)CN(C(C3CCSCC3)=O)C2)cc(Cl)ccc1N C(=O)(CC(C)CCCCC)N1C(C=C)CN(C(=O)CCC(C)N(C)C)CC1 C(=O)(C1=CCCCCC1)NC(C)(CNC(C1CC2CCC1O2)=O)C1CCC1 C=CC(CC)CC(=O)N1CC2C(N(C)C(c3ccc(C(C)(F)F)nc3O)=O)C2C1 CCCCCC(C)(CC)C(=O)NCC(C(C)C)NC(c1nncs1)=O C(CC(F)(F)CO)n1cc(COC(C)C(=O)NC2CCCCC2)nn1 C1(NCCNC(C(C)NS(C)(=O)=O)=O)(NC(=O)CC2CCOC2=O)CCCC1 N1(C(c2cnn(CCC)c2Cl)=O)CCC(O)C(NC(=O)Cc2nonc2C)C1 N1(C(COC2CC(NC(CN3CC(=O)NC3=O)=O)C2)=O)CC2(CCCC2)C1 CC(C)CCC(F)C(=O)N1CCOCC(C(=O)NC(CC(C)C)C(N)=O)C1 N1(C(c2cccc(CC)n2)=O)CCN(C(C2SCC=C2C)=O)CC1CCO CCCS(=O)(=O)C(C)C(=O)NC1CCC1CNC(c1ccc2c(c1)OCC2)=O N1(C(CC#N)=O)CCC(NC(C2CCC(F)C2)=O)CC1 C12CC3CCCC3N1C2=O.C12(CC(C3CC4C=CC3C4)=O)C3C4C5C3C1C5C24 Nc1cccc(Cl)c1C(=O)NC1CC1NC(c1ncoc1C1CC1)=O c1(C(=O)NC2C(NC(c3cn(CCC)nc3)=O)COC2)nccnc1N N1(C(C23C(CN(C(C)=O)C2)C3)=O)CCOC2CN(C(=O)CCCOC(C)C)CC12 N1(C(CC(CCC)C)=O)CCC=C(C(=O)N2CC3(C2)CC3(F)F)C1 c1(C(=O)NC2CN(C(C3CC(O)CCN3OC)=O)CCO2)cccc2c1CCC2 C12(CNC(C3CCOC3)=O)CC(C1)C(NC(=O)C(F)(F)c1ncccn1)CO2 CC1(C)CCCN(C(C2CC3CC3C2)C(=O)NCc2ccco2)C1 C1(NC(COC(CC)C)=O)COCCN(C(=O)C(F)(F)c2ccccn2)C1 c1(OC)cc(C(=O)NCC(C2CC2)NC(=O)CCC=C(C)C)ncn1 c1(C(N2CCCCC2CO)=O)ccc(I)cc1Cl C(=O)(CC(C)(C(F)F)N(C)C)N1C(C)CCC(NC(c2c(C)cc(F)cn2)=O)C1 Cc1[nH]c2ncnc(NCC(C)N(C)C(c3ccnc4c3CCC4)=O)c2c1C C(=O)(CC1CC(=O)Nc2ccccc21)N1C(CNC(CNS(N)(=O)=O)=O)CC1.C C1(C(N2C(CNC(c3ccsc3Br)=O)CCC2)=O)CC12CCOC2 N1(C(C(C)NC(N)=O)=O)CCC(NC(c2cc(F)cnc2O)=O)C(O)C1 N1(C(C2CC(OC)(OC)C2)=O)CCC(NC(=O)C(C)Cc2ccco2)C12CCC2 N1(C(CCC=C)=O)CC2CCCC(C1)N2C(=O)C(C)C(C)CCC N1(C(c2c(C)c(Cl)ccn2)=O)CC2CC(C)N(C(C3CC(C(F)(F)F)C3)=O)C2C1 c1(C(=O)NC2CN(C(c3c(C)n(C(C)C)nn3)=O)C2)cccc2cccnc12 c1(OC)ccc(C(N2CC(O)(CNC(C3CC34CCC4)=O)C2)=O)c(O)c1 C1(CNC(C2C(C(C)C)CCC2)=O)CCC2(CN(C(c3cc(N)ccn3)=O)C2)O1 N1(C(C(COCC)C)=O)CCCC(CNC(c2csc3nccn23)=O)CC1 C(=O)(C(CNC(c1ccc(C)c(O)c1)=O)CC(C)C)N1C(CSC)COCC1 CCCCC(F)C(=O)N1CCN(C(c2cccc(C=C(F)F)c2)=O)C(CO)C1 Cn1cc(C(=O)NCC2(CNC(=O)Cc3ccc(F)cn3)CC2)c(=O)n(C)c1=O N1(C(CC2CCN(C)C2=O)=O)CC2(CC2)CC1CNC(c1csnc1Cl)=O N1(C(CCn2ccc(C)n2)=O)CCC2(CC(NS(=O)(=O)CCBr)C2)C1 C=C1CCC(C(=O)NCC2CN(C(=O)C(C3CC3)OC)CC2C(F)(F)F)CC1 CCC(C)CC(C(=O)N1CC(C(N)=O)C2(CC2)C1)NC(=O)CCCC1CCCO1 Cn1cc(NC(c2ccc(-c3ccccn3)nc2)=O)cc1NC(=O)NCC1CC1 CC(c1ccc(F)cc1)=CC(=O)NCC1(C)CCN(C(=O)CCn2cccn2)C1 C(C(C(C)C(C)C)NC(=O)CC12CCC(CC1)OC2)NC(COCC(=O)NC)=O c1(C(N2CC3(CCC(C(=O)NC(C)C4CC4)O3)C2)=O)ccc2[nH][nH]c(=N)c2c1 C(CCO)(C(=O)NCC(O)CNC(=O)Cn1ccc(Br)n1)N(C)C C(=O)(C1CCc2c(Cl)cccc21)N1CC(NC(c2ccc[nH]2)=O)(CO)C1 c1(C(=O)NCC(CN(C)C(C2CCCS2)=O)(C)C)cc(Cl)c(Cl)c(Cl)c1 CCC(C)CC(C(=O)NC1CCCC(C)(C)C1)NC(=O)C=CCOCCOC c12nnc(-c3ccc(Cl)cc3)cc1SCCC2=O.c1(CCCOC)cncn1C NS(=O)(=O)N1CCC(C(=O)NCCC(O)CNC(C2CC3CCCCC23)=O)CC1 c1(CC)ccc2cc(C(=O)NC3CCC(N(C(=O)CC(C)F)C)CC3)ccc2c1 c1(C(=O)NC(C)CN(c2ncc(C#N)cc2F)C)ccc2nc[nH]c2c1 c1(C(N2C(C(C)NC(C3CC4C=CC3C4)=O)CCC2)=O)ccc(O)cc1F Cc1cc(C(=O)NC(C)(C)CNC(C2CC(F)C(=O)N2C)=O)cnc1C(F)(F)F O(NC(=O)CN=c1nc(N2CCC(CC(=O)N(C)C)CC2)c2sccc2[nH]1)CC CC(C(F)C(=O)NC1CC2(CCCN(C(=O)CC(C)(C)C(F)F)C2)C1)C(F)(F)F C1(NC(CC2COCC(C)(C)O2)=O)CC2CCC(C1)N2C(c1ccc(O)cc1)=O c1(C(=O)NCCCN(C(=O)C(C)C(C)C)CCC)ccnc2c1CCC2 c1(C(=O)NC(CCNC)C(C)C)cn(CCOC)c(C)cc1=O C1(NC(C2CCC(CC(=O)OC)C2)=O)CCCCCN1C(=O)COCC(C)C c1(C(=O)NC(CCNC(C(C)OCCC#C)=O)C)ccnn1CCCC C1(NC(c2ccc(CC3CC3)nc2)=O)CCN(C(=O)C(F)=CC2CC2)CC1CO C(c1ccc(F)cc1)=CC(=O)NCCOCCN(C(C1(F)C(C)C1)=O)C CC#CCCCC(=O)NCC1CCC(C)N(C(c2coc(C(=O)OC)n2)=O)C1 c1(C(N2CC(O)(CNC(Cc3n(C)ncc3)=O)C2)=O)c(C(F)(F)F)cncc1F C1(NC(CC2(C(=O)OC)CC2)=O)CCCC2CN(C(C3(NC(C)C)CC3)=O)CC12 c1(CCC(=O)NCC(C)NC(C2CC2C(C)(F)F)=O)nc(O)c2ccccc2n1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C(=O)COC(F)F)CCC1C1CC1 c1(C(=O)NCCCN(CC)Cc2cncnc2)ccccc1CO C(=O)(CCS(=O)(=O)c1cc(Cl)ccc1Cl)N1CCC(C)CC1C(F)(F)F C1(CC=C)(CNC(C2CC2CCOC)=O)CCCN1C(=O)Cc1c[nH]nc1O C1(C)(CC)CC(NC(c2ccc(CNC(=O)C(O)C(C)(C)C)o2)=O)CCO1 c1(OC)nc(C)cnc1C(N1CC(O)(CNC(C2COC(=O)N2)=O)C1)=O c1(NCCCc2c(C)cccc2)ncccc1S(=O)(=O)NC1CN(C)CC1C c1(C(=O)NCc2cc(C)cc(Br)c2)cc2cc(-c3cccc(C)c3O)ccc2[nH]1 c1(OC)ccc(NC(C2CC(F)CN2C(c2ccc(O)cc2Br)=O)=O)c(C)c1C N1(CC)N=C(C(=O)NCCC2(C)CCN(C(C3CC(C)CCO3)=O)C2)CCC1=O N1(C(C=CC=CCC)=O)CC(N(C(=O)CCC2CC2(F)F)C)C(C)(C)C1 CC1CC(NC(=O)C(C)O)CN(C(=O)CCc2ccccc2O)C1 C(CCCCC(=O)NC(C1CC1)C1CC1)N(C(C1C(C)CCC1)=O)C CCC(CC)C(=O)NCC1CN(C(c2ccc(N)cn2)=O)C2CC12 C1(NC(=O)NC2CC(C(F)(F)F)(OC)C2)CCCCC1(F)F C(=O)(C1c2c[nH]nc2CCC1C)N1CCC(NC(C(CC)(C)OC)=O)C1C c1(C(=O)NCC2(OC)CCN(C(=O)CSc3cccs3)C2)cc(Cl)c(C)cn1 c1(C(=O)NCC2C(NC(C(C3CCCC3)SC)=O)CC2)cc(CO)n(C)n1 C(=O)(C(CNC(=O)C(C)(C)OC1CCCC1)CC(C)C)N1CCC(COCC)C1 N1(C(C=CCN(C)CC)=O)CCC(C)(C)C1CC(N1CCN(CCO)C(=O)C1)=O c1(C(N2CCCC(CN(CCOC)CC)C2)C(=O)NC)nc(Cl)ccc1Cl Cc1cc(C(C2CC2)NC(=O)C(=O)NC(C)CCc2ccccc2)cc(C)c1 c1(CN(C2CCN(C(C3(COC)CCC3)=O)CC2C)C)cn2cc(C)ccc2n1 c1(N2CCN(CC)C(C)(C)C2)nc2cc[nH]c2c(=NCc2c(C)nnn2C)[nH]1 c1(C(N2CC(N(C(CC(C)C(F)(F)F)=O)C)C2)=O)cc2n(c1)CCS(=O)(=O)C2 Cc1c(C(=O)NC2CC2CNC(c2ccc(F)cc2)=O)cnn1C1CCC1 C(=O)(C1=CCOCC1)N1CCC(CN(C(C(CC)NC(C)=O)=O)C)CC1 c1(C(=O)NC2CN(C(CC(C=C)(C)C)=O)CC(C)C2)cccc2c1CCOC2 c1(C(C)C(=O)NC23CCC(C(C)NC(C)=O)(CC2)C3)ccc(S(N)(=O)=O)cc1 c1(CC(=O)NCCC(C)N(C)C(C2CC2(Cl)Cl)=O)c[nH]c2ncncc12 N1(CCNC(CCOCC)=O)CCN(C(c2ccc(C3CC3(F)F)cc2)=O)CC1 c1(C(=O)NC2CCC3(CC2)CC3)ncnc(N2CC3CC3C2)c1F.CCOC C=CCC(CC)N=c1nc(N2CCC(CC(C)CO)CC2)c2sccc2[nH]1 c1(NC(=O)NC(c2ccccc2F)C(C)C)nnc2n1CCC(C(F)(F)F)C2 N1(c2cc(C(C)=O)ncn2)C2CCC1CC(CNC(=O)Cc1c(C)noc1C)C2 c1(CNC(=NCc2ccc(OC)cc2)NCC2=CCOCC2)ccc2sccc2c1 CC1(C)CCCC1CCNC(=O)CN(C(=O)CC1OCCCO1)CC1CC1 N1(C(c2c(OCC=C)cccn2)=O)CC2(C1)SCCC2NC(C12COCC1C2)=O C1(S(N)(=O)=O)(C(N2CCC(C(Cn3cc(CN(C)C)nn3)F)CC2)=O)CCCC1 C12(C(=O)NCCCN(C(=O)CC3COC4CC3C4)C3CC3)CCCN(CCC1)C2 CCC(CCCC(=O)NC1CCSC1)NC(c1ccc(N)cn1)=O C#CC(C)(C)C(=O)NCC(C1CCCN(C(c2sc(CC)nc2C)=O)C1)(C)O C=C(C)CCC(=O)N(C1CCN(C(C2(CC(C)C)CCC2)=O)C1)CCC N1(c2nccc(OCC)n2)CCC2(CCCC2CNC(c2ccc(Br)o2)=O)CC1 c1(C(=O)NCC2CCN(C(C3N(CC)CCCC3)=O)C2)c2c(nn1C)CCC2 N1(C(c2c(OC)csc2)=O)CCC(CNC(c2n[nH]cc2[N+](=O)[O-])=O)C(F)(F)C1 Cc1ccnc(O)c1C(=O)NC1CCC(NC(=O)C(N2CCNC2=O)C)C1 n1(CC(=O)NC2CC(NC(c3cnccc3Br)=O)C2)cc([N+](=O)[O-])cn1 C1(NC(c2c(CC)scc2)=O)CCN(C(c2[nH]cnc2COC)=O)CC(C)(C)C1 C1(C(N2CCC(NC(c3c(SC)csc3)=O)CC2)=O)CCCC(C#N)C1 C(=O)(CCC(C)C)NC(C(=O)NC(CC(=O)OC)C1CC1)c1ccco1 c1(C(N(C)CCNC(C2CCCOC2C2CC2)=O)=O)c(Cl)ccc2ncccc12 N1(C(c2cn(C)nc2C)C(=O)NCCCCCC)CCc2ccc(OCC)cc21 CC(CCNC(=O)CCCCCNC(=O)CNC=O)C(C)(C)C N1(C(C2CCC(C)C2)=O)CCCC(C2(NC(C3(C)CC=CCC3)=O)CC2)C1 CCC(C)C(=O)C(=O)NCC#CC(=O)NCC1(C)CCCC1O c1(N2CC(CN(C(C(CC)=CC)=O)C)OCC2)nc(Cl)nc2c1CCOC2 C1(C(=O)NCCOC2CCCC2)CC=CCN1C(=O)CCC1CCCOC1 N1(C(C(C)Sc2ccccn2)=O)CC2CC1CN2C(C12CC3CC1C2C3O)=O N1(C(C(C=CC)O)=O)CCOCC(C(=O)NC(c2ccc(O)nc2)C)C1 CCC(CC)CCCC(=O)N1CCC(N(C(=O)C(C)(F)F)C)CC2(CC2)C1 C(=O)(C1=CC2CCCC12)N1CC(CC=C)(NC(c2c(N)cnn2C)=O)C1 C1(CSC)CCCN1C(=O)CC1C(NC(=O)C(n2ccc(C)n2)C)CC1O c1(C(N2CCCC(NC(c3c(N)cn(C)n3)=O)C2)=O)cccc2c1C(=O)NC2=O C1(C(=O)NC(C(C)NC(COCC(=C)C)=O)C)CN2CCCN1CC2 C(C(C)CC(=O)N1CC(CCO)(NC(=O)C(C)Sc2ccco2)C1)OC c1(C(N2CCC3(NC(C(CC)CC)=O)C(CC2)C3)=O)cnc2ccccc2c1 C(C(C)(C)C(=O)NCCC1CCC(NC(C2(C)CC=CC2)=O)C1)OC CC1CN(C(=O)CCC2CCCCC2)CC1CCNC(C1CC=CCC1)=O C1(CC=C)CCCN(C(=O)COCC(=O)NCC)CC1.c1cnc(C(F)(F)F)nc1 C1(NC(CCNC(C)=O)=O)CCCC(NC(=O)C(C2CC2)C2CC2)C1 Cc1coc(C)c1C(=O)NCC1(CNC(=O)CC2C=CCC2)CC12CCC2 C1(CNC(=O)Cc2cccs2)CC2(CCC2)CN1C(C1C2CCCOC12)=O c1(OCC)cc(C(N2CCOC(CNC(=O)Cc3csc(=N)[nH]3)C2)=O)ccc1C CN1CC2CCN(C(C3(CNC(c4cc(CO)ccn4)=O)CC4(CC4)C3)=O)C2C1 c1(OC)c(COC(C2(C(=O)OC)CCNCC2)=O)cccc1Br C1(C(=O)NCC(N(C(CCC(=O)N(C)C)=O)C)C2CC2)CCCS(=O)(=O)N1 C1(NC(CCC)=O)CC(CNC(=O)NC(=O)C(C)SCC2CCCO2)C12CCC2 C1(CNC(C2C(CC)C2)=O)CN(C(=O)CCCCN2CCCC2)CC(C(C)C)O1 CCCCC(C(=O)N1CCC(C)(C(=O)NC2CN(C(C)C)C2)CC1)C(C)C N1(C(C2N(C(C3ON=C(CC)C3)=O)CCOC2)=O)CCOCC2(CC2)C1 c1(OC)ccc(CN2CC3(CC3)CC2C(=O)Nc2cccc(C)c2O)c(C#N)c1 N1(C(CC2CN(C)C2)=O)CCC(NC(C2CCCCC2C(C)(C)C)=O)C2(CCC2)C1 C1(C(C)=O)C(C(=O)NC2CC(O)(CNC(c3ccc(CN=[N+]=[N-])o3)=O)C2)C1(F)F C1(C(N2CC(C(C)NC(c3nn(C)c(Cl)c3Cl)=O)C2)=O)CC2CCCCN2C1 N1(C(CCOCCOCC)=O)CCC(NC(=O)CCCC(C)=O)CC(C)(C)C1 c1(SC)cccc(CC(=O)NCC23CC2CN(C(C2(F)CCOCC2)=O)C3)c1 c1(OC)ccnc(C(=O)NCC2CCN2C(C2CC3C=CC2C3)=O)c1OC c1(C(=O)NCCCN(C(C2(C)CCCCC2C)=O)CC)ccc(F)c(C(F)F)n1 c1(OC)c(C(=O)NC2CN(C(=O)C#CC3(C)CC3)CC23CC3)ccnc1Cl N1(C(C2(COC)C=CCN2C(=O)C(CO)OC)=O)CCC(C)(C2CC2)C1 c1(OC)ncc(C(=O)NCC2CC(F)(F)CN2C(c2cc(C)sn2)=O)cc1C N1(C(CCOC(C)=O)=O)CC=C(CNC(C2C(C)(C)C2(F)F)=O)CC1 C1(Cl)(C(=O)NCC(CC)NC(c2scnc2C)=O)CC1(C)C C1(NC(CC2CCN(C)CC2)=O)CCC2CN(C(=O)CC3OCCO3)CC2C1 c1(NC(C2C(C(N3C(COCC)CCCC3)=O)C2)=O)ccc(C2CC2)cc1I C(CCOC)(C(=O)NCCn1ccnc1C)NC(C1(COCC)CC1)=O c1(C(C)O)ccc(C(=O)NC2CC(CNC(=O)Cc3cn(C4CC4)cn3)C2)cc1 N1(C(CCCONC(=O)OCC)=O)CCC(C)(C)C(CNC(C2C3COCC23)=O)C1 C12(NC(C=CSC)=O)CCCCCC1N(C(c1ccc3ccnn3c1)=O)CC2 C1(NC(c2c(CC)nc[nH]2)=O)C=CCN(C(=O)C(c2cccc(OC)c2)O)C1 C(C(CC(C)C)C(=O)N1CCCOC(CN(C)C)C1)NC(C(CC)NC(C)=O)=O CCC(COC)C(=O)N(CCCCCCNC(C1CCCCC1)=O)C C(=O)(C1CCOc2c(F)cccc21)N1CCC(NC(C2(CSC)CC2)=O)C(O)C1 CC1CCN(C(C23CCC(C2)OC3)=O)CC1CNC(c1ccncc1Cl)=O C(=O)(C1=COCC1)NCC1(CNC(CCc2cc(C(C)C)no2)=O)CCCC1 N1(C(CC2(NC(C)=O)CC2)=O)CCCN(C(C2CC3CCCCC23)=O)C(C)C1 c1(C(N(C(C)C)CCN(C)C(C2C(C)C2C)=O)=O)coc2ccc(Br)cc12 c1(C(=O)NCC2(C)C(C)CN(C(=O)CC3CC3)C2)ccc(S(N)(=O)=O)cc1F N1(C(C(C(CC)C)N(C)C)=O)CCCN(C(=O)CCNS(=O)(=O)CC)CC1C N1(C(C2(N(C3CC3)Cc3nnc(CO)s3)CCC2)=O)CCCC1NC(N)=O c1(C(N2CC(C)(NC(C3OCC4CCCC34)=O)C2)=O)cnc2c(F)cccn12 C1(NC(c2ccn(CC)n2)=O)CC(C)CN(C(c2ccoc2)=O)C1 N1(C(C2CCC(C)CC2)=O)CCC2(CCCCC2NC(c2sccc2F)=O)C1 c1(CC(=O)N(CCCCCC)CCNC(=O)C=CC(C)C)ccc(OC)nc1 N1(C(CC(n2c(CC)ncc2)C)=O)CC(NC(=O)CC2(CSC)CC2)C(C)C1 c1(C(=O)NC2CC(CNC(c3c(C#C)cnn3C)=O)C2)scc2c1OCCO2 Cc1oc(-c2ccsc2)cc1C(=O)NCCCn1cc(C2CCOCC2)nn1 N1(C(C2OCCN(CC)C2)=O)CCC2CCN(C(c3c[nH]nc3C)=O)CC12 c1(NC(C2CCN(S(=O)(=O)C(F)F)CC2)=O)ccc(OC(F)F)cc1C c1(CCCC(=O)NC2(CNC(C3CCC(CC)C3)=O)CCC2)cc(F)ccc1F N1(C(C2(O)C(C)(C)C2)=O)CCC2CN(C(c3c[nH]c4ncccc34)=O)CC2C1 Cc1cc(O)ncc1C(=O)NCc1cc(C(=O)N(C2CC3CC3C2)C)n[nH]1 CC(C)CC(O)C(C)C(=O)NCCOC1CN(C(c2ncccc2C2CC2)=O)C1 Cc1ccn2cc(C(=O)NC3CCCC4CN(c5ncns5)CC34)nc2c1 c1(C(=O)NCCCCCN(C(c2cc(OCC)n[nH]2)=O)C)sc(CO)nc1C N1(C(CCN(C)CCO)=O)CC(NC(c2ccc([N+](=O)[O-])s2)=O)CC(O)C1 N1(C(C(C)OC)=O)C2CCC1(CNC(=O)Cc1cc(C)ccc1Br)CC2 N1(C(CCC(C)OCC)=O)CCN(C(c2ccnn2C(C)(C)C)=O)C(CCO)C1 N1(C(c2c(OCC)cncc2)=O)CCOC(C)(CNC(C23CCCC2C3(F)F)=O)C1 N1(C(CCNC(C)=O)=O)CCCC(C2CC2NC(C2(C#N)CC23CCC3)=O)C1 c1(NCCNC(=O)CSCC(N2CCSCC2)=O)cc(=O)cc[nH]1 C1(CNC(CCC)=O)CN(C(=O)Cn2nc(C(F)(F)F)cc2Cl)CCCO1 CC(CCCCNC(=O)CCCc1cnn[nH]1)NC(=O)CCC1CC1 C1(C(=O)Nc2cccc(NC(C3CCN(C)CC3)=O)c2)CC2CCCC2C1 c1(CC(N2CCC3(C2)CN(C(C24COCC2C4)=O)C3)=O)nc2ncccn2n1 N1(C(c2cc(NC)cc(C)c2)=O)CCN(C(=O)CCCCNC(N)=O)C2CCC12 c1(OCC)ccc(C)cc1C(N1CC2CC(NC(=O)CCn3cccn3)C2C1)=O N1(C(c2c(C)n(C(C)C)cc2)=O)CC(NC(C23CCCC2C3)=O)CC(C)C1 Cc1cn2nc(C(=O)NC3CCN(C(c4sncc4C)=O)CC3F)cc2c(=O)[nH]1 CCC(N=c1nc(N2CCOC(c3nc(C)cs3)C2)c2c([nH]1)CSC2)C1CCC1 C1(CCCC)C(=O)NCCN1C(=O)CC1CCN(CC2CCN(CC)CC2)CC1 c1(C(=O)NC2CCC(NC(CSCCC)=O)C2)ccc2c(c1)CC(C)(C)C2 N1(C(C=CCN(C)C)=O)CC(C2CN(C(=O)CC3CCCC34CC4)C2)C1 C1(NC(c2ncc(CC)s2)=O)C(C)CCN(C(=O)CN2CCCCC2)C1C C12(Nc3nccc(OC)n3)CCCC1N(C=O)CC2.C1(C2CO2)CCCC1.OC CC(CN(C)C)CCC(=O)NC1(C)CC(NC(=O)C2=NOCC2)C1 c1(N2CC(C(C)C)SCC2)nccc(=NCCc2nnc(Br)n2C)[nH]1 c1(OC)c(CC(=O)NC2CC2CNC(=O)C(C)(C)CF)cccc1F c1(C(=O)NCC(C)NC(c2nncn2C)=O)ccc2c(c1O)CCCC2 c1(SC)cc(C(N2CCC(NC(c3cncc(N)c3)=O)C2)=O)ccc1Br C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC2C(NC(C3CCCN(CCC)C3)=O)C(C2)C1 C(=O)(C1=CCCCC1C)N(CC(=O)NCC(C)S(C)(=O)=O)CC N1(C(=O)OC(C)(C)C)CCC1CC(=O)NCC1CC(C(C)(C)C)C1 c1(C(=O)NCC2C(NC(CC(=O)NCC#C)=O)CCC2)cscc1S(C)(=O)=O C(=O)(CCCC(=O)OC)NC1(C(N2CC(C(C)OC)C2)=O)CC(F)C1 CCC(CC)CCCC(=O)NCC1CC2CCC(C1)N2C(=O)C(C)NS(C)(=O)=O C1(C(N2C(C(=O)NCc3cnc(C)nc3)CCCC2)=O)CC2C(C1)C2(C)C c1cc2c(c(Cl)c1)[nH]c(=O)[nH]2.C(C)(C)(C)OC(=O)NCC1CC1.CC(C)COCC Cc1ccccc1C(C)CC(=O)NCCNC(c1c(Cl)n[nH]c1C)=O CCC(C)CCCCC(=O)NCC(C(N1CCOC(C)(C)C1)=O)N(C)C c1(C(=O)NC(C2CCCN2C(=O)CC2CC2)C)ccc(Br)cc1 c1(CC)ccccc1C(CNC(=O)C(C)CCOC)NC(=O)CC(C)(C)C c1(C(N2CCCC(CN(C(=O)CC3C=CCC3)C)C2)=O)ccc(=O)n(CCO)c1 N1(C(c2c(C)ccc(C)c2)=O)CC(NC(C2C3CCCC23)=O)CC12CCCCC2 c1(OCCOC)ccc(C(=O)NCCC(O)CNC(C2CC2CF)=O)c(Cl)c1 C1(C(=O)NCC(CC(C)C)NC(c2ccc(OC)cn2)=O)CCc2nnnn2C1 N1(C(=O)NC)CCCN(C(c2cnc(O)cc2C)C(=O)NCCCSC)CC1 N1(C(Cc2ncn(C)c2)=O)CC2(C(N3CCC(N4CC=CC4)C3)=O)CC1CCO2 c1(CCC(=O)Nc2cncc(C(C)(C)C)c2)c(F)cc(Br)cc1F CN1CCCC1CC(=O)NC1CCCC1NC(c1cncs1)=O N1(C(c2cccc(C)c2OC(F)F)=O)CCOC2CS(=O)(=O)CC12 C1(CNC(C(C2CCCC2)OCC)=O)CC2CCC1N2C(=O)CCCCC#N C(=O)(C1CSc2ccccc21)N(CC(C)O)CCNC(c1ncccc1N)=O CC(C)(C)C(=O)C(=O)N1CC2(C(N3C4CC(NC(c5ccccc5)=O)(C4)C3)=O)CC1CO2 C1(CNC(=O)NC2CC(NC(C3CCSC3)=O)C2)CCCC(C(F)(F)F)C1 N1(C(C2CC2F)=O)CCC2(CCCC2C(N2CCCC3CCCCC23)=O)C1 N1(C(c2cc(C)n(C)n2)=O)CC2CCN(C(C3CC3(Cl)Cl)=O)CC(C2)C1 N1(C(C(C)CO)=O)CCC(O)(Cn2cc(-c3cncc(Cl)c3)nn2)C1 C12(NC(CCCNC(=O)OC)=O)CCC(C(=O)NCCCC3(C)CC3)(CC1)C2 C1C(F)(F)CCC(=O)NCc2cn1nn2.C(CC(C)C)OCCCSC Cc1ocnc1CC(=O)NC1CC(CCNC(=O)C(n2ccc(Br)n2)C)C1 C1(C(N2CC(C(N)=O)(CNC(c3n(CC)ccc3)=O)C2)=O)NC(=O)OC1C C1(NC(c2cc[nH]c2)=O)CN(C(C2CC3CC2C3)=O)CC12CCC2 C1(N(C)C(C2(c3ccc(F)c(F)c3)CC2)=O)CC2CCC(C1)N2C(=O)C(C)(C)O C=CCC(CC)C(=O)NCCCC1CCCN1C(C1CCC(C)(C)CC1)=O O=C(C1=C2CCN=C2NC=C1)N1CC2C(CNC(C3(CC4CC4)CC3)=O)C2C1 C1(F)(CNC(CC=CCC)=O)CCC(CNC(C2(C)CCOCC2)=O)C1 Cc1cn2c(=O)c(C(=O)NC(C)CNC(c3ccn4ncccc34)=O)cnc2s1 CCC(CN(C)C)CC(=O)NCC1CCCCN(C(=O)C=Cc2cn[nH]c2)C1 Cc1c(F)ccc(Cl)c1C(=O)NCCN(C)C(c1occc1F)=O c1(C(=O)NC(C(C(C)C)C)CNC(=O)CSC(C)(C)C)ncnc2ccsc12 c1(SC)cncc(C(=O)NCC(O)CNC(=O)C(N2CCSCC2)C)c1 Cc1coc(C)c1C=CC(N1CC(O)CC1CNC(=O)CC1CC1(C)C)=O c1(C(=O)Nc2c(C(=O)Nc3c(C)n[nH]c3)scc2)sc(Cl)nc1C c1(C(N(C)CCNC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)=O)cc2n(c1)CCCNC2=O C=CCCCCCCC(=O)N(C(C)C(=O)NOCCC(C)O)CCN(C)C c1(C(c2nnnn2C(C)C)NCC(CSC)C)c(C)cnn1COC c1(-c2onc(Cc3ccc(Cl)cc3)n2)ccc2sccc2c1 N1(CC)CCN(c2ccc(NC(=O)CC3CCCCCO3)cc2)CC1 C1(C(N(C)C)=O)CC2CC1CN(C(N)=O)C2.C1(C)(CC(=O)N)CCC1 C(=O)(C(CC)(CC)OC)NCC1(O)CC(NC(C2CC(C#C)(O)C2)=O)C1 C1(NC(C2C(C)C2C)=O)CCN(C(=O)Cc2cccc(C3CC3)c2)C1C(F)F N1(CCC(=O)NCCC2(O)CN(C(C3(C#C)CC3)=O)C2)C(=O)CCC1=O Cc1nc(C)n(CC(=O)NC2CCC(C(F)C(=O)NCc3cnn(C)c3C)C2)n1 n1(CCOC)cccc(C(=O)NCC2CC(C)N(C(=O)C(C(C)C)SC)C2)c1=O C(=O)(CC(CC(C)C)NC1CC12CCC2)NC(c1nc(C)oc1C)C C1(C(C)C)(CO)CCN(C(=O)C(C2CCCC2)NC(c2cc[nH]c(=N)n2)=O)C1 CCCC(C(=O)NCC1(CNC(C2(CO)CCCO2)=O)CC1(F)F)NC(N)=O C(C=O)(C1=NOC2CC12)N(C)CCCCF.c1(C(F)(F)F)cccc(C2CCC2)c1 N1(C(C2(CC(=O)OC)CC2)=O)CC2CC3CC2C1C3NC(=O)CS(=O)(=O)C1CC1 CC1CN(C(=O)CC(CC2CC2)NC(=O)COCC(F)F)CCO1 C(CC(CNC(c1cnco1)=O)NC(=O)C(C)CSCc1ccccc1)OC CC1(C(N2CCC(CF)(NC(=O)COCC3CCOC3)C2)=O)CCNC1=O c1(NCC(N2C(CC(=O)NC(c3nc(=O)o[nH]3)C)CC2)=O)ncccn1 Cc1cc(C)c(NC(=O)NCCS(=O)(=O)C2CC2)c(C)c1 N1(C(C2C(COC)C2)=O)CCC(N(C(=O)Cn2nc(C)cc2C)C)C2(CC2)C1 N1(C(C(CC)C#N)=O)C2CCC1CC(C(=O)NC1CCC13CCCC3)C2 Cc1ccc(CNC(C2CC(NC3(F)CN(C(=O)OC(C)(C)C)C3)C2)=O)cc1 N1(C(CN2CCC(C)(O)C2)=O)CCCC2(CCCN2C(C2SCCS2)=O)C1 c1(CNC(=NCCC)NCc2nc(C)cs2)cc(=O)n2ccccc2n1 CC1CCC(CNC(C2NC(=O)OC2C)=O)CN1C(=O)C=CC1CC1 n1(CC(=O)NC2C(CNC(Cc3cccc(OC)c3)=O)C2)ccc(O)nc1=O C1(C(=O)NC)CC(O)CN1C(=O)C(C1CCCN(C(=O)CCCCOC)C1)C CC1CC(Nc2nccc(-n3ccnc3)n2)CCN1C(=O)CC1CCC(O)C1 C1(CC=C)(C(=O)N(C)CC2CCCC3CC23)CCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 C1(Cn2cc(C(C)OCC)nn2)CCC(NC(c2cnc(NC)cn2)=O)CC1 CC1(C)CC(NC(=O)C2=CCSC2)CN1C(c1cnn(CCO)c1N)=O CC1(C)CC(CC(N2CCOC(CNCC3CC34CCOC4)C2)=O)CO1 C1(CC(=O)OCC)CC(CNC(=S)Nc2ccc(OCC)cc2)=NO1 O=C1CCC(CCC(N2CC(O)(CNC(=O)CC3CSC3)C2)=O)N1 Cc1cc(C)c(NC(C2CC(CNC(=O)CC3CCCO3)C2)=O)c(C)c1 c1(CC)cc(C(N2CCC(CCNC(c3nn[nH]c3Cl)=O)CC2C)=O)c(C)nn1 N1(C(c2c(C)ccs2)=O)CCC(NC(C2CCCN(C(N)=O)C2)=O)CC(C)(C)C1 CCC(C)CC(C)C(=O)NC1(CC=CC(=O)NC2CC3CC2CC32CC2)CCC1 c1(C(N2CCC3(C(NC(C(CC)C)=O)C3)CC2)=O)nn(C)c2c1COCC2 c1(C(c2n(CCCSC)nnn2)NCC2(C)COC2)cc(C(F)(F)F)ccc1Br N1(C(c2ccc(C)c(F)c2)=O)CC(NC(=O)C2=CCOC2)CC12CCCCCC2 Cc1ccc2oc(C(N3CC4CC(C3)C4(F)F)C(=O)NC3CCOC3)cc2c1 CCC(C)(CCNC(=O)C(C)C(F)F)NC(C1SCCS1)=O c1(C(=O)OCC)cccc(-n2cc(CCN(C(=O)Cn3cnnc3)C)nn2)c1 c1(C(=O)NCC(C(C)C)NC(Cn2ccc(C)n2)=O)cn(C)c(C)n1 C1(SC)CN(C(=O)C(F)(F)c2cn[nH]c2)CC1NC(=O)C(N)=O C(=O)(CC(F)(F)c1ccc(Br)nc1)OCCCOCOC Cc1ccc(C(N2CCCCCC2C(=O)NCc2cnccc2Cl)=O)c(F)c1 c1(C(N(CCN(C(c2cncc(NC)n2)=O)CC)CC)=O)nc(C)ccc1F C1(CC(=O)NC(CNC(C(CCOC)C)=O)(C)C)CSc2ccccc2O1 C1(O)(C(C)NC(C2(C)CC2)=O)CCN(C(=O)CCN(CC(F)(F)F)C)CC1 c1(NC(C(=O)NC2CCN(Cc3ccn(CC)n3)C2)C)ccc(Cl)cc1Cl N1(C(C(c2cccnc2)C)=O)CC2CCC(C1)N2C(c1cnc(O)n(C)c1=O)=O C1(CNC(CSC)=O)CCC(C)N(C(=O)CC(C)n2cccn2)C1 N1(CC(=O)NCCCn2cc(C(c3ccccn3)O)nn2)CCCS1(=O)=O Cc1c(C(=O)Nc2cncnc2-n2cccn2)sc2c(Br)csc12 c1(C(=O)NC2CCC(C(N(C)CCN3CC=CC3)=O)C2)cc(Cl)cc(Cl)c1 Cn1cc(OCC(=O)NCC2(NC(c3ccnn3C(C)(C)C)=O)CCOC2)cn1 N1(C(CCOCCCOC)=O)CCCCC(N(C)C(C2C3CC4C(C3)C24)=O)C1 Cc1ccc(C(=O)NCCC2CN(C(=O)Cc3cc[nH]c3)CC(C)O2)cc1C Cn1cnc2sc(C(N3CC4CC(NC(=O)C5=COCCC5)C(C4)C3)=O)cc12 C(=O)(CCCCCN(C)C)NC1CC(N(C(C2(OCC)CCC2)=O)C)C1 N1(C(C2(CCC)CCN(C(=O)Cc3cnn(C)c3C)C2)=O)CC(OC)CC(C)C1 C1(C(=O)NC(CC=C)C(=O)OCC)CC(C)(C)CN1C(c1cnccc1C#N)=O C1(C(N(C2CN(C(=O)C(C)(O)C(F)(F)F)CC2(C)C)C)=O)CCC2(CCC2)CC1 C1(O)(CN(C(c2c(CC)[nH]c(=N)s2)=O)C)CCCN(C(C2CC=CCO2)=O)C1 Cc1cc(C(N2CCOC(C3(C)CC3)C2)C(=O)NC2CC2)cc(C)c1 c1(C(=O)NC2CC2CN(c2cc(Cl)ccn2)C(C)=O)ccc(F)c(C2(C)CC2)c1 C(=O)(CC(C)(C)C(F)(F)F)NC1C(CNC(CN2CC(C)(C)C2)=O)CCC1 C1(Cc2cn(N(C(CC3CCC(C)C3)=O)C)nn2)CCC(CO)CC1 c1(C2CCN(C(c3cccc(C(CC)C)c3)=O)C2)ccc(OC)c(OC)c1 c1(-c2onc(C(C)OCC=C)n2)nnn(C)c1C CC(C)CC(O)C(C)C(=O)N1CC(OCC(=O)NCC(C)C(=O)OC)C1 c1(C(N(C2CN(C(=O)Cc3cccc(F)c3)CC2F)C)=O)cccc(F)c1Cl C(=O)(CCCCCN=[N+]=[N-])N1C(C(=O)NC(C=C)(C)C)CN(C)CC1 N1(C(C(COC(C)C)NC(=O)CC(C)CN(C)C)=O)CCC2(CCCCC2)C1 Cc1cc(C(N2CC(C(=O)NCC3(C)NC(=O)NC3=O)C3(CC3)C2)=O)c(O)nn1 C1(CNC(=NCCC=C)NCCc2ncccc2Cl)COc2ccccc2O1 N1(C(Cc2nnc(C)o2)=O)CC2CC1C2NC(c1ccsc1Cl)=O c1(NC(CC2(C=C)CN(C(=O)CCCCCCC)C2)=O)ccc2ccncc2c1 C(=O)(C1=CC2(CCN(C(=O)C(C)CC3CCC3)C2)C1)NCC(CC(=O)OC)O c1(C(=O)OC)ccc(COc2cc(O)nc(SC)n2)cc1F N1(C(c2cc(OCC)n[nH]2)=O)CCCCC(NC(C2CC2(C)C(F)(F)F)=O)C1 Cc1cccc(C(O)C(=O)N(CCCNC(c2ccc(Cl)s2)=O)C2CC2)c1 c1(NC(C2CN(C(C(C(C)C)CN(C)C)=O)CC2(C)C)=O)cccc2ccoc12 c1(C(N2CC(C)C(NC(=O)C3=CCCSC3)CC2)=O)ccn2c1CSCC2 c1(C(N2CCC(CCNC(C3NC(=O)OC3)=O)C2)=O)cccc2c1COCCN2 c1(C(N2CC(NC(c3nn(C)c(Cl)c3)=O)C(CO)C2)=O)cn(C)c(=O)n1C N#Cc1ccc(NNC(=O)NCc2cccc(F)c2Br)cc1F c1(C(N(C(C(=O)OCC)C2CC2)C)=O)nc(CC)c(C)cc1C#N c1(C(N(CC(CC)NC(=O)C(COC)OC)C)=O)ccccc1Br Cc1sc2ncnc(NC(CNC(=O)CCc3cncs3)C3CC3)c2c1C N1(C(COCC(C)C)=O)CCN(C(c2ccc(C(C)C)cn2)=O)C(CC(F)F)C1 Nc1cccc(F)c1C(N1CCC(C(N2CCOCC2)=O)CC1)=O C1(CC)(NC(c2ccc(C3CC3(F)F)cc2)=O)CCN(C(=O)C(O)C2CC2)CC1 Cc1ccc(C2(C(c3cccs3)CNC(=O)C(C)(C)C3CCC3)CC2)c(F)c1 c1(C(N2CCC(NC(C(CC)=O)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 CCCC(C(=O)N(C)CC1CCCN1C(=O)C(CC)c1ccccc1)OC C1(NC(C(CC(C)C)OC)=O)CCC2CN(c3ccnc(CO)n3)CC2C1 N1(C(Cc2c(C)ccnc2)=O)CCN(C(c2cccnn2)=O)C2CCCCC12 CC1CN(C(=O)Cn2cccnc2=O)CC1CNC(=O)Cc1nc[nH]n1 c1(CC(=O)NCCCN(CCC)CC)cccc(F)c1.c1(C=O)cc(O)n(CC)n1 Cc1cc(C#N)ccc1C(=O)N(CC(C)(C)C(=O)NCC1CCN(C)CC1)C C=Cc1cncc(C(N2CC(C)(C(N3CCCCCC3)=O)C2)=O)c1 C(CN=c1nc(N2CCC3(CCOC3)C2)c2sccc2[nH]1)N1CC(SC)C1 C1(CC)(NC(=O)C(C)S(N)(=O)=O)CCN(C(C2CC2c2ccncc2)=O)CC1 C(=O)(CCC(CC)OC)N(CC(=O)NCc1n(CCC)ncc1)C(C)C C(CCC)(CC(=O)NC(CO)C(=O)N(C)C)NC(C(CCC)OCC)=O Nc1ncccc1C(N1CCCC(CNC(c2ccnc(C(F)(F)F)n2)=O)C1)=O C(CCCCC(=O)NCC1OCCC1C)NC(C1(CCC=C)CC1)=O N1(C(CC(=O)NCC)=O)CCC(C(=O)NCCSC(C)(C)C)C1C C1(C(N2CCCC(C(C)NC(c3c(C)scc3)=O)C2)=O)CC(C)(C)OC(C)(C)C1 c1(C(=O)NCC2(F)CC(NC(C=C(C)Cl)=O)C2)ccc2c(c1)NC(=O)CN2C C1(CC(=O)NCCCCNC(C2(C)C(C)(C)C2)=O)COCC1(C)C c1(C(N2C(CNC(C(CCC)SC)=O)CN(C)CC2)=O)cc(F)c(N)cc1OC c1(C(N2CC(C(=O)Nc3c(C#N)cc(CC)s3)C2)=O)ccc([N+](=O)[O-])c(C)c1 c1(OC)ccc(C(=O)NCC2C(C)CCCN2C(c2csnc2Cl)=O)c(F)c1 c1(OC)nc(C(=O)NC(C)CC(C)NC(=O)C=Cc2ncc[nH]2)ncc1F c1(-c2cccc(C(N3CC4CC(F)(F)CC4C3)=O)c2)cccc(S(=O)(=O)NC)c1 c1(C(=O)NC2(C)CCN(C(C3(c4ccccc4)CC3)=O)C2)[nH]nc2ncccc12 C(=O)(C1=CCCC(C)(C)C1)NCC(C)CN(C)C(c1cc(CO)[nH]n1)=O c1(C(=O)NCCC(CNC(C(C)OCCCCCC)=O)O)cc2oc1=NC=CC=2 C1(C(=O)NCCCN(OC)C)(NC(=O)CN2C(C)CCC2C)CCC(C)(C)C1 c1(C(=O)NC(CC)(CNC(c2ccncc2O)=O)CC)cc2oc(C)cc2[nH]1 CC(C)CCOC(C)C(=O)NCCN(C)C(C12CC(C1)C2)=O c1(C(=O)CC2N(C(C(C)SCC)=O)CCC2)cnc(O)c(C(C)(C)N)c1 C1(NC(C(C)C2CC2)=O)CC(C)N(CC(O)CCc2ccccc2)C1 C(=O)(C1CCCc2ccccc21)NCC1CC(NC(c2csc(Cl)n2)=O)C1 c1(C(N2CCC3CN(C(C(COCC)C)=O)CC32)=O)coc2ccc(OC)cc12 c1(SC)cc(C(=O)N(C)CCN(C(=O)Cc2cnn(C)c2C)C(C)C)c(C)o1 C1(C(=O)NCC2CCC(C(=O)NCCN(C(C)C)C(C)C)C2)CCOCC1C C(CCCCC(=O)N(CC(C)(C)O)C)N(C(c1c(OC)scc1)=O)C CC(C)C(CC(=O)NCCc1nc(CO)n[nH]1)NC(=O)CCC(C)(C)F c1(C(N2CCCC(C(=O)NCCOC)C2)C(=O)NC(CC)C)sc(=O)n(C)c1Cl N1(C(CNC(C(CC)C)=O)=O)CC2CCC(N(C)C(C3CCN3CC)=O)C2C1 C12(C(N3CC(C)C(NC(C4CCN4C(C)(C)C)=O)C3)=O)CCCN(CC1)C2 C1(CN(C(=O)CCSC(F)(F)F)CC(=O)NC2(F)CC(NS(C)(=O)=O)C2)CCCCO1 c1(N2CC(CN(C(C(CCCC)C)=O)C)OCC2)cc(C(N)=O)ccc1[N+](=O)[O-] c1(OC)cc(C(=O)NC(C)CC(C)NC(=O)CC2(O)CCCCC2)ccc1Cl Cn1ccc2c(-c3nc(CCN(C)C)nn3C3CCS(=O)(=O)C3)ccnc12 c1(CNC(c2n(CC)nnn2)c2cc(C(F)(F)F)ns2)cnc2n1CCC2 c1(CC(c2cn(Cc3nnc(C4CC4)o3)nn2)O)cccc(I)c1 N1(C(C2CC(=C)C2)=O)CCN(C(=O)CNS(=O)(=O)CC)C(CCC)C1 c1(C(=O)NC2CC(NC(c3ccc(C(F)(F)F)[nH]3)=O)C2)ncoc1Br c1(OC)ccc(C#CC(=O)N2CCN(C)CC2CC(=O)OC)cc1 Cc1cc(C(=O)NCC2CCCN2C(c2cccc(F)c2)=O)cc(Br)c1 CC(C)(CO)C(C1CC1)NC(c1ccc(Br)cc1)=O CC1(CC(=O)NC2CC(NC(=O)CC3CCCOC3)C2)CCCCC1 CC1CCN(C(=O)CCOC2CCC2)CCN1C(c1coc(C(F)F)c1)=O n1(CC)c(CNC(C2(CF)CCN(C(C3C4CCC(F)C34)=O)C2)=O)nnc1O Cc1nc2cc(CC(N3CC(CN=c4ncc(I)c[nH]4)C(C)C3)=O)ccc2o1 CCCC(O)CC(=O)NCC1(C)CCN(C(C23CC(C(C)C)(C2)C3)=O)CC1 C(N=c1[nH]c2ccc(O)cc2s1)C1CCN(C(c2cnc(F)c(F)c2)=O)CC1 N1(C(c2ccc(-c3nc(=N)s[nH]3)cc2)=O)CCCC2(COCCN2)C1 C1(N(C)C)CCC(C(=O)NCCNC(=O)CCc2cnoc2)C1 c1(C(=O)OC)ccnc(C(=O)NC2C3CN(C(C4CC(C)(C)O4)=O)CC23)c1 N1(C(CC(C)SC)=O)CCN(C(=O)C=C(C)Cl)CC1CF c1(C(=O)NC2(C3CCCCN3C(c3ccc(Cl)cn3)=O)CC2)csc2nnsc12 CCCC(=O)C(=O)N1CCCC(C(=O)Nc2oc(C)nc2C)C1 c1(NC)nc(C)ccc1C(N1CC(CNC(=O)CCC2CCOC2)C(C)C1)=O C1(O)(CNC(Cn2cc(C(N)=O)nc2)=O)CCN(C(=O)CCn2cnnn2)C1 C1(CNC(CCNC(C)=O)=O)CN(C(c2ccc(C3CCCC3)cc2)=O)C2CC12 Cc1nnc2n1C(C(=O)N1CCN(C(c3ccc(O)nc3)=O)CC(CO)C1)CC2 Cc1noc(C)c1CCNC(C1(NC(=O)CCc2nncn2C)CC1C)=O CC(CN=c1ccc(Br)c(S(=O)(=O)N2CCCOC(CCO)C2)[nH]1)C(C)(C)C C1(NC(C(C)NC=O)=O)CCCN(C(c2c[nH]c(=S)cn2)=O)C1 C1(CCC(=O)NC(c2cn(C)nc2)C(=O)NCCCC2CCC2)CC(C)(C)CO1 C(=O)(C(F)(F)C(F)F)N1CC(CN(C(=O)COCC2CCOCC2)C)OCC1 Cc1cccc(C(=O)NC(C)CC(C)NC(C2CCC=CCC2)=O)c1[N+](=O)[O-] C=CC(CCC)CC(=O)N(CCC(=O)Nc1ccc(O)cc1CC)CCO c1(C(N2CCC(C(=O)N(CC(F)F)C)CC2)C(=O)NCCC)nn(C)c(C)c1Cl c1(C(=O)O)cc([N+](=O)[O-])ccc1CN1CC2CCCC(C1)C2C(=O)OC N(C1CCCn2ccnc21)C(c1cccc(NC(CC(=O)OC(C)(C)C)=O)c1)=O C1(CNC(c2ccncc2F)=O)CCCC2(CN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)O1 C1(C(N(C)CC2N(C(C(C)CCO)=O)CCC2)=O)CCN2CCOCC12 c1(NCC(=C)Br)nc[nH]c(=NCc2ccccc2C(C)C)c1C CCCCCC(O)CC(=O)N1CC(CC(C)NC(C2CCC2C)=O)C1 N1(C(C2C=C(C)CS2)=O)CC2(C(N3CCC4(CSC4)C3)=O)CC1CCO2 c1(NC)ccc(-c2cncc3sc(C(N4CCCC(C)C4)=O)cc23)cc1[N+](=O)[O-] c1(CC)ccc(C(=O)NCC2CC(NC(c3occc3C)=O)C2)c(C)n1 c1(C(=O)NC(C)C(C)NC(c2sccc2Br)=O)ccc(O)c(F)c1 c1(CNC(C(CC)C)=O)cccc2c1CN(C(C1(C)CC=CCC1)=O)C2 c1(OC)cc(C(=O)NC2CC(CO)N(C(c3cc(O)n(C)n3)=O)C2)c(Cl)cn1 c1(C(=O)NCCCN(C(=O)CCCCN(C)C)CC)ccccc1[N+](=O)[O-] c1(C(N2CC(Cn3cc(C(C)(C)C)nn3)OCC2)=O)c(F)ccc2c1OCO2 c1(C(=O)NCCC(C)NC(c2ccc(-c3ccncc3)cc2)=O)cccc(=O)o1 N1(C(c2ccc(C#C)cn2)=O)CC2(CCCC2NC(C2(CC=C)CC2)=O)C1 c1(OCC)ccc(CC(N2CCCC2CCCNC(C2CNC(=O)C2)=O)=O)nc1 C1(CNC(CC(CC)SC)=O)CC2CCC1N2C(C12CC(F)(C1)C2)=O N1(C(CC=CCC)=O)CCC(C)C1CNC(C1(CC2(CF)CC2)CCCC1)=O C1(C(N(CCCN(C(C(COC)(C)O)=O)C)C)=O)CCOCC12CCCC2 C1(NC(COCCSC)=O)CCC2CN(C(c3cnn(C4COC4)c3)=O)CC2C1 C(=O)(CCS(C)(=O)=O)N1CCC(N(C(=O)CCC2CC2)CC)CC1.c1(C)ccccc1 c1(C(N2CCC(C)(CNC(CC=C(C)C)=O)C2)=O)ccc2c(c1O)CCCC2 c1(OC(C)C)cc(C(=O)N(C)C)ccc1NC(C1CCC(F)(F)CC1)=O N1(C(C2N(CC)CC2)=O)CCN(C(=O)Cn2nnc3ccccc23)CC(C)(C)C1 Cc1cc(C)c(C(N2CCC3(NC(C45CC(C)(C4)C5)=O)CC3C2)=O)c(C)n1 Cc1ncncc1NC(C1CC(F)CN1C(=O)CC1CC2CCC1C2)=O C1(C(=O)NC(C)(C)CC=CC(=O)NC2CCCC2C(C)(C)C)(OC)CCOCC1 CN=c1ccc(C(N2CCC(O)(CCNC(=O)CC(C)N(C)C3CC3)C2)=O)c[nH]1 C1(NC(C2(CC#C)CCCCC2)=O)CCN(C(=O)CN2CC=CC2)CC12CCC2 C1(CNC(CC(C)C2CC2)=O)CCC12CCN(C(c1ccc[nH]1)=O)CC2 c1(C(C)C)ncc(C(=O)NCCCC(C)NC(=O)C(F)(F)C2CCOCC2)o1 N1(C(C2(NC(=O)CCC(F)(F)F)C(C)(C)C2)=O)CC23CCC2(COC3)C1 C1(c2cccc(OC)c2)CCC2(CCN(c3ncccc3F)C2)C1 C(=O)(C(CO)C(C)(C)C)N1CCCN(C(c2c(C)n(CCO)nc2)=O)CC1 c1(C(=O)NC2CCC(CCNC(Cc3c(C)occ3)=O)C2)cc(O)ccc1F c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CCC2)cnn2c(=O)cc[nH]c12 C(C1OCc2ccccc21)NC(=NCC=C)N(C)Cc1ccon1 C(CC1CC1)(C(=O)NCC(=O)NC1CC(CO)(CO)C1)NC(C)=O CC(CC(=O)NCC1(CNC(C2(NC(N)=O)CCC2)=O)CCC1)C(F)F C1(C)(CC)CC1C(=O)N(CC(C)C)CC=CC(=O)NC.c1(CC(=O)OC)ccoc1 CC(CC(F)F)C(=O)N1C2CCC(C2)C1CNC(c1cnn(CC2CC2)c1)=O C12(CNC(c3cccnc3C(F)F)=O)CCCCC1CN(C(c1cn[nH]c1)=O)C2 N1(C(CCCCSC)=O)CCCC1C1CCCN1C(C1CC2(CCCC2)C1)=O c1(C(N2CC(C)C(NC(C3CC(F)(CO)C3)=O)C2)=O)cnc(N)c(Br)c1 c1(NCCC(C=C)(C)C)ncc(S(=O)(=O)N2C3CCC2CC(C(N)=O)C3)cc1Cl C(C(CC(=O)NCC(C)(C)N(C)C)NC(C1CC(F)CN1C)=O)OC c1(C(N(C(C)CNC(=O)C=CC2CCOCC2)CC)=O)ccnnc1C C1(C(=O)NCCC=C=C)CC(C)CN(C(=O)CSc2nc[nH]n2)C1 N1(C(C(CCSC)O)=O)Cc2ccnn2CC(NC(=O)Cc2ccccc2C)C1 c1(CCC(N2CCC(O)(c3cn(CC(=O)OC)nn3)C2)=O)cc(F)ccc1Br CC1CC(C(=O)NCC2(NC(=O)CC3CCC(C)(C)O3)CC2)CCO1 CCC(C)CCCC(=O)N1CCOCC1CC(=O)NCCCN1CCCC1 N1(C(CCOCC)=O)CCC(C(C)C(=O)NC(C)C#N)CC1 c1(CNC2C(SCC)CCC2)cc(F)c(Cl)c(F)c1 c1(C(=O)OCCN(CCNC(c2cnoc2)=O)CCl)csc([N+](=O)[O-])c1 Cc1cccnc1C(N1CC(NC(c2ccc(-c3ccncc3)s2)=O)C2CC12)=O C1(NC(CC(C)(C)O)=O)CC2CN(C(c3cnc(Cl)s3)=O)CCN2C1=O N1(C(c2cc3ccccc3o2)=O)CCn2c(-c3cncc(Br)c3)nnc2C1 C12(C(=O)NCC=CCC(=O)NCCOc3ncccn3)CCCCC1C2 C=CCCCCC(=O)N1CC(CNC(=O)C(C)(C)c2csc(C)c2)C2(CC2)C1 C12(CNC(C3(NC(N)=O)CC3)=O)CCCC1CCN2C(c1cnc(C(F)F)s1)=O N1(C(C(c2cccc(N)c2)(C)C)=O)CCC2(CCCN2C(C2CCCC2)=O)CC1 N12CCN(CC1)C1CCN(C1)C(=O)C2=O.C1(CS(C)(=O)=O)CCCCN1C1CC1 N1(S(c2c(C)noc2C)(=O)=O)CCN(N2CC(F)(F)CC2CC#N)CC1 N1(C(Cc2cc(OC)no2)=O)CCC2C(C1)CN2C(=O)CSC1CCCCO1 N1(C(C2CCCN(C)C2)=O)CCN2CCN(C(C3CC4CC4C3)=O)CC2C1 C12(NC(CSCCNC(C3(CC)CC3)=O)=O)CCCC1OCC2 C(=O)(C1CCc2cccnc21)C(=O)CCn1ccc2cccnc12.C1(N)CC1N C1(CNC(C(COCC)C)=O)CCC2CN(C(=O)Cc3ccc(Cl)cn3)CC12 c1(NC(COCCCOC)=O)ccc(CNC(=O)CCCc2cccs2)c(F)c1 C1(NC(c2c(CC)cns2)=O)CCC(NC(c2cnc(Cl)n2C)=O)CC1 c1(CNC(c2c(CC)c[nH]n2)=O)nc2c(s1)CN(C(c1sccc1CC)=O)CC2 N1(C(c2cccc(C)c2)=O)CC2C3CCC(C2C1)N(C(=O)CN1CCCC1=O)C3 Cc1ccc(SCC(N2CC(NC(c3nnccc3C)=O)CC2(C)C)=O)c(C)c1 N1(C(c2c(CC)con2)=O)CC(NC(c2occc2C)=O)C(C)C1 N1(C(c2cnc(CC)s2)=O)CC(CNC(=O)CCc2ccoc2)C(O)C1 c1(C(N2CC(F)(CNC(C(C(C)C)NS(C)(=O)=O)=O)C2)=O)nc(C)c(C)nc1C c1(NC)cc(C(=O)NC(C)CCNC(c2c(C)cccc2C)=O)cc(Cl)n1 C=C(C)CC(C(=O)NCc1csc(CNC(C2(C(C)(C)O)CC2)=O)n1)OC CC1(C)CCCC(C(=O)NCC2COCCN(C(C3(C(F)F)CCCO3)=O)C2)C1 C12CCCN(C1)C(=O)OC2C.CC(=O)NCC1CC1 c1(C(=O)NC2CC(NCc3cc(OC)c(Br)cc3)C2)ccc2cccc(F)c2n1 N1(C(c2c(C)nn(CCO)c2)=O)CC(NC(=O)Cc2c(Cl)cnn2C)CC(C)C1 c1(N(C(c2c(OC)cccn2)=O)CC2(F)CCCNC2)ncc(F)c(C)n1 CC(C)CC(C)(CO)NC(C1CCN(C(c2cn(C3CC3)nn2)=O)C1C)=O C(C(C)C(C)C(=O)NC(C)CCCNC(C1CC(c2ccccc2)O1)=O)OC Oc1ccc(Nc2c(CN(c3ccncn3)C3CCC3)cc(Cl)nc2)c(F)c1 N1(CC(=O)NC(Cc2ncn(C)c2)C(=O)O)C(=O)NC(C)(C2CC2)C1=O C#Cc1ccc(CNC23CCC(Nc4cc(C)nc(C)n4)(CC2)C3)cc1 N1(C(c2c(C)cncc2)=O)CCC(NC(=O)C(C)SC(F)(F)F)C(C)(C)C1 CC1CN(C(=O)C(=O)Nc2ccoc2)CC1CNC(=O)C(N1CCSCC1)C C(=O)(C1=C(C#N)CCC1)NCC1(C(=O)NC(C(=O)NCC)C)CC(C)(C)C1 N1(C(CCC2CCC(C)O2)=O)CCc2c(ncn2C2CC2)C1 Cc1ccc2c(C(N3CCCC4(C3)CN(C(C3COC(=O)O3)=O)C4)=O)c[nH]c2c1 CC(CC(=O)NCC(O)Cn1cccn1)C(C)(C)NC(=O)CCN=[N+]=[N-] C1(NC(c2c(Cl)ccc(C)c2)=O)CC2CC(C1)N(C(C1(C#N)CCCO1)=O)C2 CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CC(C)(NC(=O)CC2CCCCC2O)C1 C1(C(=O)NC2CN(C(=O)C(c3ccc(C)cc3)(C)C)CC2F)(CC)CC(F)(F)C1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(c2cc(C(C)C)no2)=O)c(C)o1 c1(C(=O)NCC(C)NC(C(CCC)C)=O)cccc2nc(C)nn12 CCC(CC)C(F)C(=O)N1CC(C)(C)CC1CC(N1CCCCC1CC(=O)OC)=O CC(C)(C)CC(=O)NC1(CF)CN(C(C2CC(=C3CCC3)C2)=O)C1 c1(CC(=O)NC(CN(C(C2(OCC)CCOC2)=O)C)C)cnccc1C N1(C(=O)COc2ccc(CN3CCOC3=O)cc2)CCC(F)(F)C(O)C1 n1(CCCC(=O)NCC2(OC)CN(C(C=CCC)=O)C2)nc(C)nc1C C(C(C)(F)C(C)(C)F)(c1nnnn1CCCF)Sc1ccc(OCC)c(OC)c1 N1(C(c2c(C)n[nH]c2)=O)CCN(C(=O)CC2CCCC(C)(C)C2)CC1CO c1(OCC)ccc(C(=O)NC23CC(NC(=O)CC4OCCC4(C)C)(C2)C3)cc1C C(=O)(CC1CCc2ccccc21)NC(C)CNC(c1cnc2c(ccn2C)c1)=O c1(OC)ccc(CCC(C)C(=O)NCC2CCCC(CO)C2)cc1 O=C1CC(C(=O)N2CCN(C(C3CCCN3CC(F)(F)F)=O)CC2CF)=NN1 c1(COC)csc(C(=O)N(Cc2cn(C(C)C(=O)O)nn2)CC2C3CCCC23)c1 c1(C(N2CC(NC(C3(C4CCCO4)CCCC3)=O)C2)=O)cc2c(nn1)CCOC2 c1(NCc2nn(C)c(Cl)c2)ncccc1S(=O)(=O)N1CCCC(c2ncc[nH]2)C1 c1(NC(C2C(n3cc(CCCC)nn3)CCC2)=O)c(C)cnnc1O C=CCC(CC(=O)NCc1cnnn1C)NC(C1(C#N)CCCOC1)=O C(CNC(=O)C=Cc1cccc(OC)c1)(CC(F)(F)F)NC(C(C=CC)O)=O Cn1ccc2nc(C(N(S(=O)(=O)c3ccoc3)CC3CCCN3)=O)ncc12 N1(C(c2ccc(OC)cn2)=O)CCC(c2cn(-c3cncc(Br)c3)nn2)C12CC2 c1(OCCOC)cccc(C(=O)NC2CCC2CNC(c2cc(=O)cc[nH]2)=O)c1 C1(NC(CCC#N)=O)CC2(NC(=O)Cn3cc(Br)cn3)COC1C2 N1(C(C2(CC)CC2)=O)CCC(O)(C(C)NC(=O)CCCNC(=O)OC)C1 N1(C(CC=CCCCCC)=O)CCC(C)(F)CC1.C1CC(=O)N=CC(=O)N1C C1(OC)CCN(C(=O)CC(C)(C)n2cc(CCS(C)(=O)=O)nn2)CC1 CC1CN(C(N2CCCC2CC2CC2)=O)CCN1C(=O)Sc1ccc(F)cc1F C1(C(N2CC(CNC(=O)C3=CCCC3)C(O)C2)=O)CCCCC1(F)F c1(NC(=O)CC2CCCN2C(c2ncc(F)cc2F)=O)ccnc([N+](=O)[O-])c1 c1(C(N2C(C(=O)NC3C(CC=C)CCCC3)CCC2)=O)cc(C)c(C)nn1 C1(NC(C23CCC(OC)C2C3)=O)CC2CCC1CN2C(=O)C(C)(C)Br CC1CC(CNC(=O)CCc2cnoc2)CCN1C(=O)CC1CCCC(F)(F)C1 CCC(C)CC(=O)C(=O)NC1CC2CC(NC(c3csc(F)c3)=O)CC12 N1(C(C(c2ccc(C)cc2)C2CC2)=O)CCC2CCC(C1)N2C(=O)CN(C)C C1(CNC(C(C2CC2)SC)=O)(NC(c2cc(C#N)c[nH]2)=O)CCCCC1 C1(NC(C2CC23CCOCC3)=O)CC12CCN(C(c1cc(F)cs1)=O)CC2 C1(C(=O)NC2CCC2O)CC12CCN(C(=O)Cn1cc(CO)nn1)CC2 C12(NC(c3cn4c(n3)SCC4)=O)CCOCC1CN(C(C1CCCCS1)=O)C2 n1(SCC(CC#N)O)ccc2cc(C(=O)O)ccc12 C#Cc1ccc(C(=O)NC(CNC(c2scnc2C2CC2)=O)CCCC)c(F)c1 C1(NC(c2nc(CC)oc2)=O)CCCCN1C(=O)C(C)C#N.C1(NCC)CCCC1 c1(CC)nc2ccccn2c1C(=O)NC1CC2(C1)CC2NC(=O)CCC1CC1 c12c(nnn1C)C2N1CCSCC1.N1(CC)CCN(C2CCCC2O)CC1 C1(C2(NC(C3C(O)CCN3C(c3cscc3C)=O)=O)CC2)(OC)CCC1 c1(C(=O)NC2C(NC(COc3c(OCC)cccc3)=O)C2)c(C)cccc1N c1(C(=O)Nc2ccns2)ccc(-n2cc(CNCCO)nn2)cc1 CCC(C(=O)N(CC(CO)NC(C12CC(C(=O)OC(C)(C)C)(C1)C2)=O)CC)C(C)C N1(C(c2cc(C#N)no2)=O)CCCC2CN(C(C3(n4cncn4)CC3)=O)CCC12 c1(C(N2C(CNC(c3ncn(CC)c3)=O)C=CC2)=O)cc(O)cc(F)c1 C(=O)(CCCCC(F)(F)F)NCC12OCC(NC(c3n(CC)ncc3)=O)C(C1)C2 C12=C(Cl)N=CNC1=NCC(C1CC1)N(C)C2=O.c1(N)ccc(C(N)=O)o1.CO C(=O)(C1=CCCCCC1)N1CCCC(C(=O)NCc2ncsc2C)(CC)C1 Cc1ccc(C(=O)NCC2CCCC2NC(=O)CCc2ccon2)c([N+](=O)[O-])c1 CCCCC(CC(=O)NCCCC(=O)NO)NC(=O)C(C)CN(C)C c1(C(N2CC(CNC(COC)=O)C(C)C2)=O)ccc2ncn(C3CC3)c2c1 c1(C(=O)NC(C(CO)NC(CCNC(C)=O)=O)C)ccc([N+](=O)[O-])cc1Cl C=CC(CCC)CC(=O)NC1CCC(C)N(C(=O)CCc2cnc(C3CC3)o2)C1 CC(C)(C#N)CCC(=O)N1CCCC1C(=O)NCC1(c2ccccc2)CC1(C)C N1(C(=O)Cc2cn3ccccc3n2)CCC2CN(C(C3CCS3(=O)=O)=O)CC2C1 N1(C(CCn2cnc(=N)[nH]2)=O)CC(NC(=O)CCC2CCOCC2)C(C2CC2)C1 CN1CCC2CCN(C(=O)CCN(C(=O)CCC3CCCCO3)CCO)C2C1 c1(CNC(CC(C)CF)=O)cc(O)nc(CNC(c2ccsn2)=O)n1 N1(C(C2CC(N(C)C)C2)=O)CCC(C)(C)C(C(N2CCC3(CCC3)C2)=O)C1 C(C(CN(C)C)C(=O)N(C1CC2CCC1C2)CC(=O)OC(C)(C)C)NC(C)=O N1(C(c2cc(C(C)C)no2)=O)C2CCC1CC(CNC(=O)C(C(C)C)NC=O)C2 c1(C(=O)NC(C(C)NC(C(CC#C)CC#C)=O)C)ccc2nnc(C)n2c1 C=CCC(CC(=O)NOCC1CC1)NC(=O)C1=NOC2COCC12 C1(NC(=O)NC(CCCC)CCC)C2CCC1CC(CO)C2 C1(CNC(c2c(C)noc2)=O)CC2(CCC2)CN1C(C1CCS1(=O)=O)=O N1(C(C2N(C(CC=CC)=O)CCOC2)=O)CC2(CCCO2)C1 CC1(C)CC(CC(N2CC(F)(F)C2C2CC2)=O)CN1C(=O)CC(=O)NC1CC1 N1(C(C2(C)CC(C)C2)=O)CCN(C(=O)CCc2cccc(O)c2)C(CCO)C1 CCCC(CCC)=CC(N1CCCC1CNC(=O)CCCCN1CCCCC1)=O C1(C(=O)NC2(C(N3CCCCCCC3)=O)C(C)C2)CCCC12CCC2 C(=O)(C(C)(C)C1=CCN(C(=O)C2=COCC2)C1)NC1C(C=C)CC1 C(=O)(CCCCC#N)NC(CCC)C(=O)N1CCC(N2CCC2)C1 CC1(C)CN(C(=O)C=Cc2ccccc2)CC1NC(=O)COCC(F)F CC(C(=O)NC1CC2CC1N(C(c1cc(O)nc(O)n1)=O)C2)C(C)(C)C c1(OC)ccccc1C(C)C(=O)N(CC(O)CN(C)C(c1cccnc1N)=O)C c1(C(N(C2CCN(C(C3CCCS3)=O)C2)CC)=O)oc(Br)cc1C Cc1nc(C2CC2)sc1C(N1CC(F)CC1CNC(=O)CC(=O)NC1CC1)=O Cc1nc2c(C(=O)NCC(C)(CC(C)C)NC(c3nn[nH]c3Cl)=O)ccnc2[nH]1 N1(Cc2nc(C)sc2C)CCC2CCC(C1)N2C(c1cc2ncccc2[nH]1)=O C1(C(=O)NC(C#C)(C)C2CCC2)CCOCC1NC(C1CCCN1C=O)=O C(=O)(N=c1cc(Br)[nH][nH]1)C1C2CN(CC)C1C2.c12ccccc1CNC2=O N1(C(c2ccc(C)cc2F)C(=O)NCC)CCC2(CC1)COC(=N)N2 c1(CNC(C2N(c3ncc(N(C)C)cn3)C3C(C2)C3)=O)cccc(F)c1Br C(=O)(C1=CCC(F)(F)CC1)NC(C(C)C)(C)CNC(=O)C(C)N(C)C C1(NC(CCOCC)=O)COC2(CCN(C(c3ncnc(C)c3C)=O)C2)C1 N1(C(C(C)C)=O)CC(C(=O)NCCC2CCCO2)C(C)(C)C1 C(CC(=O)NC(C1CC1C(=O)NC1CC1(C)CN(C)C)C)=CCC Cc1cc(C(=O)NCCC2(O)CCN(C(=O)CCc3cccc(O)c3)C2)nn1C c12cccc(c1)NC2=O.C1(SC)C=CCN(C(=O)CCCCN(C)C)C1 N1(C(Cn2ncc(C#C)c2)=O)CCC(N=[N+]=[N-])(C(=O)N(CCC)CC)C1 C(=O)(CCC(CF)CF)N(C1CCN(C(C2(C(F)(F)CC)CC2)=O)C1)CC#C N1(CC(N2CC(CNC(c3ccoc3)=O)C(F)(F)C2)=O)Cc2ccccc2C1 C1(NC(c2ccc(C#C)nc2)=O)CN(C(=O)C(O)CCC(C)C)CC(C)(C)C1 C(=O)(C(F)CC1CCCC1)NCCCN(C)C(c1ocnc1C1CCC1)=O N1(C(c2cccc(OC)c2)=O)C2CCC1CC(CNC(=O)C(C)(C)F)C2 c1(C(N(CCCNC(CCS(C)=O)=O)C2CC2)=O)ccc(F)c2c1CCC2 c1ccc(CCCSCc2nnnn2C2COC2)cc1.C1(C)COC1 N1(C(C(Cc2cnc[nH]2)NC(CC)=O)=O)CC(OCC)CC(C)C1 c1(NC(CC(C)N(C(c2cn(CCC)nn2)=O)C)=O)ccc(C)nc1O CP(C)(=O)c1csc(=NCC(C(F)F)Nc2ccccc2)[nH]1 N1(C(C(CC)(F)F)=O)CCC2(CC(NC(=O)COCCc3ccccc3)CO2)C1 c1(C(C)C)c(NC(=O)NCc2ccnnc2)cnn1-c1ccccn1 c1(C(=O)NC(CNC(C(CC#C)C)=O)(C)C(C)C)cc(Cl)c(Cl)cc1OC C1(NC(CCC2C(C)C2)=O)CN(C(c2cc(C)n(CCO)n2)=O)CC1C1CC1 c1(C(=O)NCC(C)CN(C)C(c2c[nH]c(C#N)c2)=O)nc2n(c1Br)CCC2 c1(CC(N2C(CNC(C(F)=CCC)=O)C(C)CC2)=O)cccc(Br)c1C Cc1c(NC(C2CCC2CNC(c2c[nH]c(C(N)=O)c2)=O)=O)cccc1F CC1=NN(CCC(C)C)C(=O)C1CC(=O)NCCNC(C12CC(C)C1C2)=O c1(OC(C)C)cc(C(=O)NC(CNC(c2ccon2)=O)CO)ccn1 CCC(CC(=O)N1CC2(CC2)CC1C(=O)NC1CCC(=O)N(C)C1)C(F)F c1(C(N2CCCC(CCNC(c3cc(C)n(C)c3)=O)C2)=O)ncc2ccccn12 c1(OC)ccc(N)cc1-c1cccc(CN2CCCC2C)c1 N1(C(C(N2CCOCC2)C)=O)CC2CCN(C(c3ncc(Cl)cc3O)=O)C2C1 c1(C(=O)NCCC2(O)CCN(C(C3(C)CCOC3)=O)C2)sc2cccnc2c1Cl C(CN=[N+]=[N-])(C(=O)NCCCC(C)C)NC(C(CC)n1ccnc1)=O N1(N2CCCN(C(C)=O)CC2)CCCCC(C2CN(C(=O)OC(C)(C)C)C2)C1 Cc1[nH]c(C)c(C(N2CC(CCCCNC(C3CCCN3N=O)=O)C2)=O)c1C C1(C2(NC(=O)Cc3ccsn3)CC2)CCCN1C(C1CCSCC1)=O C1(C(N2CC(C(C)NC(=O)CSCCN(C)C)C2)=O)CC12CC(C)(C)C2 CC1CCn2c(-c3nc(CCN(C)C)nn3-c3cccc(C(F)(F)F)c3)cnc2C1 c1(C(C(=O)NCC2C(NC(COCC(=C)C)=O)CC2)C)ccccc1F C1(C(C)NC(C2CC(CC(F)F)C2)=O)C2CN(C(=O)COCCF)CC12 C(=O)(CC(C(=O)NC(C)CCN(C)C(c1ccnc(C2CC2)c1)=O)N(C)C)OC C1(CC)CN(Cc2ccncc2-c2c(C(F)(F)F)nn(C)c2OC)CC(C)S1=O CC1(C)C(C(=O)N(C2CCCC2)CCCOCC2CC2)C1(C)C C1(O)(C(N2CCC(N(C)C(c3ccnn(C)c3=O)=O)C2)=O)CCCC(C)(C)CC1 N1(C(C(CC)N(C)C)=O)CC(NC(=O)Cc2nc(C)sc2C)C(C2CC2)C1 c1(C(C(=O)NC2CC2)N(C)C(c2ccc(C(N)=O)cc2)=O)cc2cccnc2[nH]1 Cc1cccn(CC(=O)NC23CC(NC(C4C(F)(F)C45CCC5)=O)(C2)C3)c1=O C12(C(=O)NC(C3CCCN3C(=O)C(CO)N(C)C)C)CC(C)(C1)OC2(C)C C(=O)(CCCCCC#N)NC1CC(C)(C(=O)NC2C(C)OCC2)C1 c1(CN2C(CNCc3cnc(CCC)o3)CC2)cnc(Cl)cc1Br Cc1cnn(C)c1-c1cn(CC2CN(C(C3C4CC(=O)CC34)=O)CCO2)nn1 c1(-c2nc(CCCO)n(CC(F)F)n2)ccc(Cl)cc1O N1(C(c2c(C)non2)=O)CCC(C(C)(C)C)(CO)C1.c1(C(=O)NC2CC2)coc(C)n1 C1(CC)CN(C(c2cc(CNC(=O)C(C)C3(O)CCC3)cs2)=O)CC(=O)N1 C1(CC)OCCCC1C(=O)NCCCOCCNC(=O)CCCN(C)C CN1N=C(CC(=O)NC2CC3(C2)CC(CNC(c2cc(C#N)on2)=O)C3)CC1=O N1(C(c2ccc(CCC)[nH]2)=O)CCCC(CO)(NC(c2cc(COC)no2)=O)C1 C#CC1(O)CCCN(C(=O)CN(CC(C)C)C(c2ccc(C(C)=O)o2)=O)C1 c1(NC(C2CCCC2)CSC(F)(F)F)cccc(CC(F)(F)F)n1 C1(Nc2cc(NCc3ccc4c(c3)OCO4)nc(C)n2)CCOC12CCCCC2 Cc1ncc(C(=O)NCCC2CSCCN2C(c2csc(Cl)n2)=O)n1C O=C(C1CCCn2ccnc21)N1CCC2CN(C(C3CC3c3cccs3)=O)C2C1 S(=O)(=O)(CC(=O)NCCC1(NC(=O)CCn2cc(C)cn2)CC1)NC c1(N2CCC(CC=C)(NC(C3CC3(C)CC)=O)C2)ncn(C)c(=O)c1Br c1(C(N2CC3C(CNC(Cc4cc(C)no4)=O)(C3)C2)=O)c[nH]c2ncc(F)cc12 N1(C(C(c2cnn(C)c2)C)=O)CCOC2(CCN(C(=O)Cn3ncnn3)C2)C1 c1(C(=O)NCC=CCNC(C(C(CC)O)(C)C)=O)c[nH]c2ccc(C#N)cc12 N1(C(CCC)=O)CCCCC1CCC1(C2CCCN2C(c2ccns2)=O)CC1 C1(NC(C=C(C)C(F)F)=O)CCN(C(=O)C(F)C(F)(F)F)CC1(C)C C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C)N(C(C2CC(OC(F)(F)F)C2)=O)CC1 C1(C(N2C(C)CC(O)C2)=O)CCC2(CN(Cc3cccc(O)n3)C2)O1 Cc1cc2[nH]c(C(=O)NC(C)(C)C(C)NC(=O)Cc3nnc(C)o3)cc2o1 c1(C(N2C(CNc3cccc(C(N(C)C4CC4)=O)c3)CCC2)=O)nccnc1Cl c1(NC(c2ncc(C)cn2)C)ncc(C)cc1S(=O)(=O)NC1CCS(=O)(=O)C1C c1(C(=O)NC(C(C)(C)NC(C2C(C(=O)OC)CC2)=O)C)cc2ccccc2cn1 Cc1ccc(C)c(C(=O)CCC(=O)NC2CCC2NC(c2nnsc2C)=O)c1 N1(C(C2(CCC)CC2)=O)CCC2CN(C(c3cc(N)c(F)cc3F)=O)CCC2C1 C(C(C)(O)CC(=O)NCC1(C(N2CCCC(C)C2CCO)=O)CCCCC1)OC C(=O)(C(C)(C)C(F)(F)F)OCCNC1(c2ccc(C)cn2)CCC1 c1(CC(=O)Nc2c(OCCCC(=O)OC)cccc2)cc(=O)n(C)cc1Br Cc1oc(C(N2CCC(O)(CN(C)C(c3cnn(C)c3)=O)C2)=O)cc1CO c1(CCC(=O)NCC(CNC(COCCOCC#C)=O)F)nccn1C c1(-c2n(C(C=C)C)nc(-c3cccnc3)n2)cc2c(C)ccc(F)c2[nH]1 c1(C(=O)NCCOCc2ccccc2)cc2c(cc1F)NCCC2 C(=O)(C1=CCC(C)(C)CC1)NCC(C(C)C(C)C)NC(C1CC(OC)C1)=O N1(C(C=C(COC)C)=O)CCCC(CC(N2CCC(CC3CCC3)C2)=O)CC1 c1(C(C)=O)ccc(N(C)Cc2cncn2C)cc1 N1(C(CCS(C)(=O)=O)=O)CCCC12CN(Cc1c(Cl)ccc(Br)c1F)C2 CN1C(=O)NCC1C(=O)NC1CC(F)(CNC(C2CCCC2)=O)C1 c1(OC)cccc(Cl)c1CC(=O)N(C1CN(C(c2csc(C(F)F)n2)=O)C1)C C1(NC(c2ccc(OC)o2)=O)CC2(C1)CN(C(=O)C(CO)N(C)C)C2 c1(C(=O)NC2CCC(NC(c3cnc(C(F)F)s3)=O)C2)cnn2cccnc12 c1(C(N2C(CCN(C)C(C3C4CC(=O)CC34)=O)CCCC2)=O)cccc(Cl)c1F c1(C(=O)NCC(=O)NCC2(SC)CCC2)cccc(C(=O)Nc2cccnc2)n1 Cc1cc(NC2CN(C(c3csc(CC(C)C)n3)=O)C2)n2ncnc2n1 C12(C(=O)NC3CCN(C(C4(c5cc[nH]n5)CCC4)=O)C3)CC(C3CCCC3)(C1)C2 c1(C(N(CC(C)CNC(C2CC2C)=O)C)=O)ccc([N+](=O)[O-])cc1Br C(CC(C)C)(C(=O)N1C2CCC(C2)C1CO)NC(COCCC)=O c1(C(=O)OC)cc(NC(c2snc(-c3ccccc3)c2Cl)=O)cc(SC)c1C c1(CC(N2CCC(N(C(C3C(=C)C3)=O)CC)C2)=O)ncccc1F N1(C(c2c(OC)ccs2)=O)CCC(C)C1CNC(=O)Cc1csc(S)n1 N1(C(C=CCCC)=O)CCN(C(c2ccc(CCC)cc2)=O)C(C)C1C C1(NS(CC(C)OCC)(=O)=O)CCS(=O)(=O)C2(C1)CC(C(=O)O)C2 c12nc(cs1)CN(C)C2=O.C(C(C)(C)CNC(=O)COCC)OCC(=O)NC C(=O)(C1c2c[nH]nc2CN1C(c1ccc(C(N)=O)o1)=O)N1C(C(C)O)CC1 C1(C(=O)NCC(O)CNC(=O)Cn2ncc(Cl)c2C)(OCC)CCCCCC1 c1(C(=O)NC(CC(C)NC(c2ncn(CC)c2)=O)C)cn2nc(OC)ccc2n1 C(CC(C)OC(C)C)NC(C1(NC(CN(C2CC2)CC)=O)CCCC1)=O C(=O)(C(F)C(C)(C)O)NCCOC(C(=O)N(CC(C)C#N)CCOCCO)(C)C c1(OC)ccc(CN2CC(C)CC2C(N2CCC(OC3CCC3)CC2)=O)cc1Br CCCC(C)(C)C(=O)NCCC1(NC(C2CCOC2c2cccnc2)=O)CCC1 C(=O)(C(F)(F)CC1CC1)N(CCCN(C(C(COC)N(C)C)=O)C)C c1(CC(=O)NCCN(C(=O)C(c2ccccc2F)C)C(C)C)c(F)cccc1Cl CC1CN(C(c2cc(O)cs2)=O)CCN1C(c1csc(Br)c1)=O c1(C(N(CCNC(c2c(OC)ccnc2O)=O)C(C)C)=O)cc2nnn(C)c2s1 Cn1nc(C(=O)NCCC2(CNC(C3CCC(C)O3)=O)CC2)cc1C1(Cl)CC1 C1(CC)C(NC(c2cccnc2O)=O)CCCN1C(=O)CC1CCC2(CC1)CC2 c1(OC)c(CN(C(=O)CCN2CCOCC2)C(C2CCCC2C#N)=O)cccc1Br C(=O)(C1=CS(=O)(=O)c2ccccc21)NC1C(C)(C)CN(C(=O)C(O)C(F)(F)F)C1 c1(CNC(C(c2ccc(C)o2)N)=O)ccc2c(c1)C(=O)N(C)C2 CC1(C)CCCC(C(=O)NCCCCCNC(=O)COc2cccc(O)c2)CC1 Cc1cccc(C(N2CCC(N(C)C(C3CCCN3N)=O)C2)=O)c1N Cc1cncc(C(=O)NCCOCCN(C(=O)C2=CCCC2C(F)(F)F)C)c1C CCCC(C#N)C(=O)NC(C)(C)CN(C(=O)CSCC(C1CCCCC1)=O)C CC(C)CCC(C(=O)N1CC(O)(CO)C1)NC(=O)CCN(C)C N1(C(CCCCC)=O)CC(C(N2CC(n3ccnc3)C2)=O)CC12CCC2 C1(C(C)NC(c2c(CC)nc(C)s2)=O)COc2ccccc2O1 c1(NC(C2C=CC(NC(CCc3ccc(OC)cc3)=O)C2)=O)ccnc(Cl)c1C Cc1nn(C)c(C(F)F)c1C(=O)NCC1CCC(NC(=O)C(C)C#N)CC1 c1(CC)ccccc1C(CNC(=O)C=CCO)NC(C1(C)CCCN1C)=O CCCCCCCCC(=O)N1CCC2(CCCN2C(C2CCC(C)C2)=O)C1 c12cc(Cl)cnc1N2.C(CNC(=O)NCC(C(=O)OC)C)(CC(C)C)OC CC(C(c1nnnn1CSc1ccccc1)NC1CC=CCC1)C(C)(C)C N12CC(CCC(O)C1)NC(=O)C1C(C1(F)F)CC2=O.c1c(F)cncc1Cl.CC C(C(Cl)C(C)(F)F)N1CC(C)C1=O.COC(=O)NC(=O)COC.C=CC c1(C(N2CC(O)(C(C)NC(C(C)=CC3CC3)=O)C2)=O)cc(C(N)=O)cn1C c1(N2CCC(NC(CC)=O)CC2)cc(NCC2(C)CC(C)C2)nc(C(F)(F)F)n1 Cc1nn(C)c(C(=O)NC2CCCN(C(C3CCCC(CF)C3)=O)C2)c1Br N(C(=NCCF)N(C)CC12CCC(CO1)C2)CC(c1cnn(C)c1)OCC CCCCCC(F)C(=O)N(C(C)C(=O)NCC1CC1CN(C)C)C1CC1 c1(NC(C2CCN(C(C3C(C)(C)C3)=O)CC2O)=O)ccc2c(c1)OCC(=O)N2 N#Cc1c[nH]c2ncnc(N3CCC(N4CCOCC4)C(O)C3)c12 CC1CCC=C1C(=O)N1CCN(C(c2ccncc2)=O)CC1c1cccnc1 c1(C(=O)Nc2c(C)cnc(F)c2)ccc2[nH]cc(-c3cc(CO)cc(F)c3)c2c1 Cc1cc(F)c(C(N2CC3CCC3(NC(=O)C#CC(C)C)C2)=O)cc1F c1(C(=O)NCCN(C(=O)C(C)(O)c2ccccc2)CC)ccnc(O)c1 CC1CC2CCC(C(N3CC(C4(NC(=O)CN5CCOC5=O)CC4)C3)=O)CN2C1 CC1(C)Cc2[nH]nc(C(N3CCC(NC(C4CNC(=O)C(C)(C)C4)=O)C3)=O)c2C1 Cc1ccccc1S(C)(=O)=NC(=O)c1coc(=O)c(Cl)c1 c1(C(=O)NC(CC)CNC(=O)C(F)(F)C(F)F)ccnc2c1cnn2C c1(CNC(CCNS(CC)(=O)=O)=O)nc(NC(C2CCCN2C(C)C)=O)cs1 Cn1ccc2cccc(CN3CCC3C(=O)Nc3ncc(Cl)nc3C(N)=O)c12 C1(CNC(C(C)OCCOC)=O)CN(C(=O)COCCOCC)C2(CCOCC2)C1 C1(Cl)(C(=O)NC(c2occ(C(N(CC(CCC)C)C)=O)n2)C)CCCCC1 N1(C(c2ccc(OC)c(OC)n2)=O)CCCN(C(=O)C(=O)NCC2CC2)C(C)C1 N1(C(C(C(CC)CC)OC)=O)Cc2n[nH]cc2C1C(=O)NCC(C)CC1CC1 c1(C(N(C2CN(C(c3c[nH]cc(C)c3=O)=O)C2)C)=O)cc(S(C)(=O)=O)cnc1O N1(C(CC(C)(C)C)=O)CC(C(=O)NCCNC(N)=O)C2(CC2)C1 c1(C(=O)NCC2CN(C(C3(C=C)CCC3)=O)CC2C)cc(Cl)ccc1F c1(C(=O)NC2CCN(C(=O)C(F)(F)CO)CC2F)cccc2cncn12 C1(C(N2CCC(C(C)C(=O)NCc3cc(CO)ccn3)C2)=O)CN(C)CCN1C CC(C(=O)NOCC(=O)NCc1ccc(F)cc1F)C(C)(C)C C1(C(N(C(CNC(c2c(C)oc(CO)c2)=O)C)C)=O)C2(CCC2)C12CCC2 C(=O)(N=c1cc(Cl)n(C)[nH]1)C1C2(CCN(C(c3c(SCC)nccc3)=O)C2)C1 C(=O)(CC(C(F)F)NC(C1CC2(CCC2)C1)=O)N(CCCC)C Cc1ccc(C=CC(=O)NC(CCN(C)C(C2CCS(=O)(=O)N2)=O)C(C)C)cn1 N1(C(c2c(O)ncc(CC(=O)OC(C)(C)C)c2)=O)CCC(O)CC12CC2 c1(C(N2CCC(O)(CNC(CC(CCC)O)=O)CC2)=O)nc2cc(O)ccc2[nH]1 Cc1ccc(F)c(C(c2nnnn2CC(F)F)NCc2nn(C)c(Cl)c2Br)c1F C1(COC)CN(C(c2csc(C3CCCNC3)n2)=O)C1(C)C.C1CN1 N1(C(=O)Cc2cc[nH]c2)CC2(CCN2C(c2cc(O)ccc2Br)=O)C1 c1(C(=O)NC2CCN(C(C3N(CC)CC3)=O)C2C)ccc2nc(O)oc2c1 C1(c2n(C)ncc2)CN(C(c2cnsc2)=O)CC1NC(=O)CC1CCC=CCC1 CC1C2C(CCN2C(c2cc([N+](=O)[O-])ccn2)=O)CN1C(=O)C(O)C(C)(C)C C#CCC(C)C(=O)N(C)CC1C2CN(C(C3CCC(C(C)C)CC3)=O)CC12 Cc1cc[nH]c1C(=O)NC1CC(NC(C2CC(OC(C)C)C2)=O)C1 N1(C(CN(CCC#C)C)=O)C2CCC1C(F)C(NC(=O)C(C)(COC)CC)C2 C1(C(=O)NCC2N(C(CNS(CC)(=O)=O)=O)CC2)COC2(CCC2)CO1 c1(N2C(C(=O)N(C3COCC3OC)C)CC(OCC)C2)cc(N(C)C)nc(C)n1 N1(C(C2C(CC(C)(C)C)C2)=O)CC2CC(C(=O)NC(C3CCCO3)CO)CC2C1 c1(C(N(CCCNC(c2nn(C)c(Cl)c2Cl)=O)C)=O)coc2c(F)c(Cl)ccc12 C1(O)(C(C)NC(C2CCCO2)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1 c1(CNC(c2ccc(C)cc2Cl)CC)cc(C)nc2c1CCCC2 CC12CN(C(=O)CCOC3CC3)CC1CN(C(=O)C(c1ccc(Cl)c(F)c1)F)C2 c1(CC(=O)N(CC(CNC(C(C)CN(C)C)=O)O)C)cc2cc(Cl)ccc2[nH]1 c1(C(N2CC(CCOC)C(=O)CC2)=O)nccn2cnnc12.C1(=O)CCO1 C1(N(C)C(c2cc(C(F)F)[nH]n2)=O)CCC(CO)CC1.C123CC1CCN2C3=O C(C)(C)(CCCNC(c1cnn(-c2nccs2)c1)=O)NC(C(F)=CC)=O C1(C(N(C)CC)=O)CCN(C(c2cn(C(C)(C)C)nc2C)=O)CC1(C)C CCCC(C)CCCC(=O)NC(C)CNC(c1cc(N)cc(O)n1)=O c1(OC)cccc(C(N2CCCC(C(C)C)C2)C(=O)NCCOC)c1 N1(C(C2(CC#C)CCC2)=O)CCC(NC(c2ncsc2C)=O)C(CO)CC1 c1(CNC(C(C2CCOC2)NC(c2c(CC)nn[nH]2)=O)=O)nnc2n1CCC2 c1(CC)cccc(C(N2CC3CCC3(CNC(=O)C(C)(COC)OC)C2)=O)c1O C1(C(=O)NCCCCOCC)CCCC1NC(=O)CC(=O)N(C)C C1(NC(C(COC)OC)=O)CCCC12CCN(c1ccnc(C#N)n1)CC2 C12(C(N(C)CC=CC(F)(F)F)=O)CCCC1CCN2C(C1CCC1)=O Cc1ncc([N+](=O)[O-])n1CC(=O)NCC(F)CNC(=O)C(C(C)C)n1cncn1 C1(NC(c2c(C)nccn2)=O)CN(C(=O)C(C)n2cccn2)C2(CCC2)C1 C1(C)(CNC(c2occ(NC(C3CC(C(C)C)C3)=O)c2)=O)CC2(CC2)C1 c1(N2CCN(CC(=O)N(C(Cc3n(C)ncc3)=O)CC)CC2)nc(F)c(F)cc1F c1(CN2CC(CC)CC3(C2)CC3)cc2nc(OC)ccc2[nH]1 CC1(C)CC(CNC(C2CCOCC2)=O)N(c2nnc(C(F)(F)F)s2)C1 c1(C(N2C(C(C)C(=O)NC(C)(C)CN(C)C)CCC2)=O)cc(Cl)c(N)cc1F c1(CN2C(C(=O)Nc3ccc(Cl)nc3I)COCC2)cc(F)c(I)c(F)c1 C1(OC)CC2(CCC(NC(C3CC4CCCC(C3)N4C(C)=O)=O)CC2)C1 c1(OC)ccc(CN2CC3(CC(CC(N4CCC(C#N)CC4)=O)C3)C2)cc1C C1(C2CCN(C(c3n[nH]cc3Cl)=O)C2)(NC(c2nnn3c2CSCC3)=O)CC1 c1(C(N(C)CC2N(C(C3(CC)COC3)=O)CCC2)=O)cc(NC(C)=O)ccc1F c1(CC)ncc(C(=O)NC(CCN(C)C(c2nn(C)cc2C)=O)C(C)C)c(O)n1 CC1CN(C(=O)C(N2CCCCC2)=O)CC(C)N1CCc1cccc(F)c1 c1(C(=O)OC)cccc(C(=O)NC2CC(C)(NC(C3CCOCC3C)=O)C2)c1 c1(C(C(=O)NCC(C)NC(C(COC)OC)=O)C)cc(C)cc(C)c1 CCC1=C(C(=O)NCCC2CCC(NC(=O)COCCOCC)C2)SCCO1 c1(OC)ccc(COC(C2CCCCN2C(=O)Nc2ccccn2)=O)c(CO)c1 C1(NC(c2c(CC)oc(C)c2)=O)CCCN(C(=O)Cc2c(C)cccc2F)CC1 c1(CCC)ccc(C(=O)NC2CC23CC(NC(=O)Cc2cc(C)oc2C)C3)cc1 C(=O)(C(CC(C)(C)C)OC)N1CC(CC)N(C(c2cc(C3CC3)on2)=O)CC1 C1(CCNC(C(CC)=CCCC)=O)CN(C(C2(C(N)=O)CCC2)=O)CC1C C1(N(C(=O)CC2(C)CCC2)C)CN(C(c2ncnc(O)c2F)=O)CCC1O N1(C(CN(C)Cc2c(I)cn(C)n2)=O)CCC(Cc2sc(O)nc2O)C(F)(F)C1 CN1CC2C(CCCN2Cc2ccc3c(c2)OCC3(C)C)C1=O C12CCCN1C(=O)c1ccc(s1)C2.N1(NC(C2CC23CC3)=O)CCCC1 C=CC1CCCCN1C(=O)CC1CC(C)(C)CN1C(=O)C(=O)C(C)CC c1(SCC)cccc(C(=O)NC2CCC(NC(=O)C(F)OC)C2)c1 C(=O)(C(C)(C)n1cc(Br)cn1)NC(C1CN(C(C2(C(C)=O)CCC2)=O)C1)C c1(NC(C)C)ccc(C(=O)N(CC(O)CN(C(=O)C(C)C2CC2)C)C)cc1 C1(CNC(c2nc(C(C)(C)C)oc2)=O)CN(C(=O)CCc2ccsc2)CCO1 c1(C(=O)O)cnn2c(-c3ccc(N4CCC(n5ccnc5)CC4)cc3)ccnc12 c1(CC(N2C(CNC(C(C3CC3)OCC)=O)CC(OC)C2)=O)ccc(C)c(C)c1 N1(C(C2C(=C)C2)=O)CCN(C(C2(C)CCC2(C)C(=O)OC)=O)C2(CC2)C1 N1(C(C2CCC(N(C)C)C2)=O)CC(NC(C2CCCCC2)=O)C(CC(C)(C)C)C1 C1(C(=O)NCCNC(C2C(=C)CC2)=O)CCOC2(CCOCC2)C1 C(CN=C(NCCF)N1CCC(CSC)CC1)C1CCN(C)C1 N1(C(CCS(C)=O)=O)CCC(C)(CNC(c2ccc(Cl)s2)=O)CC1 C[S+](C)CCC(O)C(=O)N1CCN(C(c2ncccn2)=O)C(CC(F)(F)F)C1 c1(C(=O)NCc2cccs2)nn2c(c1-c1ccc3nc(O)oc3c1)CCCC2 C1(C(=O)NCC2CCN(C(C(c3cccc(Cl)c3)C)=O)CC2)CCCNS1(=O)=O C1(C)(CC(=O)NC(CC)CN(C(=O)CC2CC(C(C)(C)C)C2)CC)CCCCC1 CC(=NO)c1cc(C(N2CCC(CCNC(c3cnsn3)=O)C2)=O)cnc1O c1(CC(=O)NC(CCOC)CNC(=O)C(C)(Cl)Cl)c(OC)cccc1Cl C1(CNC(C2C(CNC(c3c(C)cns3)=O)CCC2)=O)OC(=O)CC1(C)C C1(C(=O)NCCN(C(=O)C(C)C(C)(C)O)CC)CCCC(C)(C)CC1 C1(NC(c2c(C)oc(CO)c2)=O)CCN(C(=O)CSS(C)(=O)=O)C(C)C1 c1(C(C)=O)cc(C(=O)NC2COCCC2NC(=O)CCC2CCOC2)ccc1O n1(C(CC)C(C)O)cnc2c(N3CCC(CS(N)(=O)=O)C3)ncnc12 C(=O)(C1c2ccccc2C2CC1C2)N1C2CN(C(C(CC#C)O)=O)C(CC2)C1 C(=O)(CC(C)C(C)(C)NC(c1cc(O)ccc1F)=O)N1CC(CC)C1 C#CCCCCCCC(=O)N(C(C)CNC(c1cccc(-n2cccn2)n1)=O)C C1(CC(=O)N(CC(c2ccccc2)NC(=O)Cc2csnn2)CC)COCCN1C.CO N(C1CCCc2occc21)C(=O)CC1CCN(C(c2cc(Cl)c(Cl)cn2)=O)CC1 c1(C(N2CCC(N(C(=O)Cc3ccccc3)CC)C2)=O)ccc(S(C)(=O)=O)c(C)c1 N1(C(c2c(NC(=O)NCCCn3cnnn3)cc[nH]2)=O)CCOCC1CO N1(C(c2cncc(OC(C)C)c2)=O)CC(NC(=O)CCn2ccnn2)CC1(C)C C(N=c1nc2c(ncn2C(C)C)c(NCc2cccc(N)c2F)[nH]1)c1c(C)ccs1 C#CCCCCCC(=O)NC(CN(C)C(C1(O)CCCCCC1)=O)CC c1(C(N2C(CO)CC(NC(c3cc(CF)on3)=O)C2)=O)ccc2ncncc2c1 CCCCC(F)C(=O)N1CCC(C(C)NC(=O)CCn2ccnn2)C1 c1(OC)ccc(C)c(C(=O)N(C)CCNC(=O)C(C)C2CCCO2)n1 Cc1nc2c(N3CCC4(CCN(C(=O)C(C)N5CCC5)C4)C3)ncnc2s1 c1(C(=O)NCC(C)N(C(c2ccc(O)cn2)=O)CC)ccc(C)c(Cl)c1Cl C(CC(C(=O)N1CC2CC1(CNC(=O)Cc1ccco1)C2)NC(C)=O)SC c1(C(=O)NC2CN(C(CCc3ncc(C)[nH]3)=O)C3C2C3)cccc(P(C)(C)=O)c1 c1(C(C)C)cccc(CC(=O)NCC2CN(C(c3ccc(C#N)s3)=O)C3CC23)c1 C(=O)(N=c1[nH]onc1-c1ccccc1F)N1C(CCOC)CCCC1 C1(N(C(CCC)C(=O)NCCN=[N+]=[N-])CC(=O)OC)CCC(F)(F)CC1 N1(C(C(C)NC=O)=O)CCC1(C)C(N1CCC(c2nn[nH]n2)C1)=O N1(C(C2C(CCC)C2)=O)CCC(CNC(c2cnc(N(C)C)cn2)=O)CC1C c1(C(N(CC(C)NC(C2(c3cccs3)CCCC2)=O)C)=O)cnn2ncccc12 Cc1cccc(C(N2CCCC(CN(C(C34CCCC3C4)=O)C3CC3)C2)=O)c1Cl N1(C(C(c2cc(C)oc2C)C)=O)C2CCC1C(NC(c1cn(C(C)C)nn1)(C)C)C2 C(CC(C(C)C)NC(c1cnc(CC)cn1)=O)N(C(C(C)(C)OCC)=O)C N1(C(CCCN(C)C(c2ccc(=N)[nH]n2)=O)=O)CCC2CCCC2C1 C=C(C)C1OCCC1C(=O)NCC1(C)CCN(C(=O)Cc2nnc(O)s2)CC1 c1(CCC(=O)NCC(CNC(C(C2CC2)OCC)=O)(C)O)cc(C(C)=O)c(C)o1 C1(C(N(CCCCOC)C)=O)CC(C)CN1C(c1nscc1C)=O c1(NC(C2N(Cc3c(OCC)nccc3)CC(F)C2)=O)cccc(Cl)c1O C(c1ccccn1)=CC(=O)NCCCC(C)NC(c1n(COC)ncc1)=O C=CCC(C)(C)C(=O)NCC(C)(C)NC(c1ccc(C(F)(F)F)s1)=O c1(OC)ccccc1NC(=O)NC1CCN(Cc2cccc(Br)n2)CC1 c1(C(N2CC(OC)(CNC(C3(C)CCCNC3=O)=O)C2)=O)ccc(C#N)cc1O c1(C(=O)NCC(C)(C)NC(C2C(C)C2)=O)ccc(N2CCC(O)C2)cc1 C1(C(N(C)CCN(C)C(C2CCCNS2(=O)=O)=O)=O)CN(CP(C)(C)=O)C1 c1(C(=O)NCC2CN(C(C(CCC)C)=O)CC2(C)C)ccc2nc[nH]c2c1 C(=O)(C(CC(F)F)NC(=O)CC1CC2(CC2)CO1)NCc1occ(C)n1 C(C)(CCN=c1[nH]c(=NC2CCn3nnnc3C2)[nH]c2cc[nH]c12)OC c1(C(=O)NCC(C)N(C(c2c(C)nns2)=O)C)cc2c(cc1F)NCCC2 N1(C(C(CC)CC)=O)CCOCC(CNC(c2cnn(CC3CC3)c2)=O)C1 CC(CC(C)(c1nnnn1C1CCCC1)NCC1CC(C(=O)N(C)C)C1)C(F)F C1(CNC(CCC(=C)C)=O)CN(C(C2CCC3CC3CC2)=O)CCC1(C)C C1(C)(C(N(CCNC(C2N(C(C)=O)CC(O)C2)=O)C2CC2)=O)CCCS1(=O)=O c1(-c2n(-c3ccc(OCC)cc3)nc(C(C)OC)n2)cc(Br)cnc1COC N1(C(C(C)Oc2ccn(C)n2)=O)CC2(C1)CC(C)(C)C2 C1(CCC)(NC(=O)C=CC2CCCO2)CCN(C(=O)CC2CCCS2(=O)=O)CC1 c1(NC(=O)NC2CNCC2F)cc2cnccc2[nH]1 c1(C2N3CCC(C3)OC2=O)ccc(F)cc1C.c1(OC)cccc(SC)c1 c1(C(N(C(C)C2CC2)C2CC2)=O)coc(CNC(=O)C(C)(C)C2CCOC2)c1 Cc1cc(C(N2CC(O)(CCNC(=O)C(C)(F)C(C)(C)F)C2)=O)ccc1[N+](=O)[O-] N1(C(c2c(OC)scc2)=O)CC(NC(C2CCCOC2C)=O)C(C)C1 Cc1ccc(CC(N2CC(CC(=O)NCc3ccc(Cl)cc3)C2)=O)cc1 C(=O)(CCS(=O)(=O)C(F)(F)F)NCC(CNC(=O)Cc1cscn1)O N1(C(CC2(C=C)CC2)=O)CC(NC(c2ccc(C)c(OCC)c2)=O)CC(F)C1 c1(C(N(C(C)CCNC(=O)Cc2ccco2)C)=O)nccc2cnn(C)c12 C1(CNC(C=CCCC(C)C)=O)CCCN(C(=O)C(C(C)C)c2ccccc2)C1 Cc1cc(C(=O)C(C)NC(=N)N)c(C)n1-c1nccs1.c1(CN)nc(CO)nn1C c1(COC)ccc2c(Br)cccc2c1.C1CCNC(=O)N1C N1(C(c2cn(CCC)nn2)=O)CCC2(CC1)CN(C(C1CC1C(N)=O)=O)C2 N1(C(C)=O)CCC(C(N(C(=O)C(F)(F)F)C2CC2)C)CC1 Cc1nn(C)c2c(NCC3CC4(CC4)C3)nc(=NC3C(C)CCC3C)[nH]c12 C=CCC(C(=O)NCC1CN(C(=O)CCC2CC(F)(F)C2)CC1O)NC(C)=O C1(CNC(C=C=C(C)C)=O)CCN(C(=O)CC2CC=CCN2C)CC1O C(CNC(=NC)NCc1ccn(C2CCC2)n1)(C(C)(C)C)SC C#CC1(C(=O)NCCOCCN=[N+]=[N-])CCN(C(=O)CC2CC3CC3C2)CC1 CCC(C(=O)NCCCCn1cc(C2(O)COC2)nn1)Sc1ccccc1 Cc1nn(CC(c2ccccc2)=O)c2nc(NC3CCN(C)CC3)ccc12 c1(C2(NC(c3nnnn3C3COC3)C3(CS(C)(=O)=O)CC3)CC2)ccc(Br)cc1 C1(C(N2C(C)CC(CNC(=O)C(C)(C)CF)C2)=O)CCC(N=[N+]=[N-])C1 C(C(C)C(=O)N(C)C1CC1)N(C(CCN(C(CCC)C)C)=O)C C1(C(=O)NCCOC(=N)O)C=CCN(C(C23CCC(C2)C3)=O)C1 N1(C(c2c(C)cc[nH]2)=O)CCN(C(=O)CCc2ccccn2)C(C)CC1C c1(C(=O)Nc2c(C(=O)OC)c(Cl)cc(F)c2)cc(O)nc2[nH]c(=N)ccc12 N1(C(CN(C(=O)C=Cc2cc[nH]n2)CCC)=O)CCC(F)(F)C(F)C1 C1(C(=O)NCC#CCNC(CCC(c2cc(C)sc2C)=O)=O)CCC2C1C2(F)F Cc1nc2cc(C(=O)NC3CC4CN(C(=O)C(C)S(C)(=O)=O)CC4C3)ccc2s1 C1(N(C(C(C)C)=O)CC(=O)NCCC2(O)CC2)CCC12CCNCC2 c1(C(N2CCC(C(F)F)(CNC(c3c(C)con3)=O)C2)=O)nnc2n1CCCC2 C1(C(=O)NCC2(C(=O)NC(C)CF)CC23CCC3)CC2CC(=O)C1C2 N#Cc1ccc(SCCC(N2CC3(CNC(C4C5CCC45)=O)CCC2C3)=O)cc1 C1(CC)(CO)CCCN(C(C2C=CC(NC(=O)Cc3cccc(C)c3)C2)=O)C1 C1(C)(N(C(CCN(C)C)=O)C2CC2)CCCCC1C(N1CC(O)(c2cc[nH]n2)C1)=O N1(C(C#CC)=O)CC2(CC2)CC1C(=O)NCC(c1ccc(F)cc1)O C1(NC(c2c(CC)cno2)=O)CCCC(NC(=O)C(C2CCOCC2)C)C1 c1(CNC(CCOC)=O)cccc(CN(C)C(C2(N=[N+]=[N-])CC2)=O)c1 C1(n2cc(C(COC)(C)O)nn2)CCN(CC(C2CC23CCCC3)=O)CC1 N1(C(C2CC(CC)C2)=O)CCN(C(c2ccc(C)c(C)n2)=O)CC1CCO c1(C(N2CCN(C(c3cnc(CC)s3)=O)CC2CO)=O)cnn2c1CC(C)CC2 Cc1ccnc(C(C)(C)C(=O)NCC(C(C)(C)C)NC(=O)CC2CC2(Cl)Cl)c1 C1(C(=O)NCC(=O)OCC#C)C=CCN(C(=O)CC2COCCO2)C1 CN1CCC(C(=O)NCC2(C(=O)NCCCOCC3CC3)CC2)C1 C=C(Cl)CCC(=O)N(CCNC(=O)CC=Cc1ccccc1)Cc1ccccc1 Cc1ccnc(C(=O)NC(C)(C)CCN(C)C(c2cncn2C)=O)c1F N1(c2c(OC)cncn2)CC(C2CCCN(C(c3ncoc3C(F)(F)F)=O)C2)C1 N1(C(C2N(C)CCC2)=O)CC2CC(NC(=O)C(c3cccc(F)c3)O)CC2C1 N1(C(C=CCOC)=O)CC2CCC2(CCNC(c2sc(C(C)(C)C)nc2C)=O)C1 c1(C(=O)NCC#CCNC(C(CCC)c2cccc(Cl)c2)=O)ccc(F)c(N)c1 C(N=c1[nH]c(C(=O)OC)nc(=N)[nH]1)C1CN(C(Cc2c(OC)c(F)ccc2)=O)C1 N1(C(COC(C)C)=O)CCC(NC(=O)COc2ccc(C(C)C)cc2)C(O)C1 c1(C(N(C(CC=C(C)C)C(=O)O)Cc2ccccc2)=O)ccc2cncn2c1 N1(C(COCC)=O)CCC(N2CCC(NC(c3sccc3COCC)=O)C2)CC1 C=CC(C)(C)C(=O)N1CC(CN2CCC(n3cc(C4C5COCC45)nn3)C2)C(C)C1 C1(C(C)(C)OC)(NC(=O)CC2CC2(Br)Br)COC1 c1(OC)nsc(C(=O)NC2CC(CO)N(C(=O)Cn3cnnc3O)C2)c1Br C1(C(=O)NCCCN(C(c2n[nH]c(C)c2Cl)=O)CCO)COCC(C)(C)O1 c1(C(=O)NCCSCC(=O)NCC(CCOC)O)ccc(C2CNC(=O)C2)cc1 Cc1cnc(CCCC(=O)N(CCNC(=O)C(C)NS(C)(=O)=O)C(C)C)o1 CCC(CC)CC(=O)N1CCOCC(NC(=O)CCc2ccc(C)c(Cl)c2)C1 C1(CC(=O)N(C2CCC(NC(CC(=C)C)=O)CC2)C)CN2CCN1CC2 Cc1scnc1C(N1CC(C)(CCC(=O)N(C)CCN(C)C2CC2)C1)=O CCCCC(CCCC)C(=O)NCCOCCCNC(c1c[nH]c(=N)o1)=O CCC(C(=O)N1CCC1C(=O)NCC(C)COCC1CC1)OC C1(CCNC(c2c(COC)cco2)=O)CN(C(c2cc(C)cs2)=O)CC(C)O1 N1(C(=O)C(F)Cl)CC2CCN(C(c3ccc4ncnn4c3)=O)C2C1 N1(C(C2CC(SC)C2)=O)CC2(CCC(NC(=O)CC3CC(=O)NC(=O)C3)CC2)C1 CCC(F)(F)CC(=O)NC1CCCN(C(c2[nH]c(C)c(C)c2C)=O)CC1 N(C1CCCc2c[nH]nc21)C(CCCCN(C(C(CC)C#N)=O)C)=O C1(C(N(C2(C(=O)NC(c3cccnc3)CO)CC2)C)=O)CCCC1C1CC1 CCC(C(=O)N(CC(C)(C)CNC(C1(OC)CC(C)C1)=O)CC)N1CCCC1=O Cc1ccnc2nc(C(=O)NCC3CC3NC(=O)CC(C)C)nn12 C1(C(=O)NCCN(C(C2CN3CCN2C(C)C3)=O)CC)CC12CCOC(C)C2 Cc1cc(Cl)cc(C)c1C(N1CCN(C(=O)C(=O)NCC(F)F)CC1C)=O c1(C(N2CC(CC(C)NC(=O)C(N3CCCCCC3)C)C2)=O)cccc(F)c1F C(=O)(CC(O)C(C)C)N(C1CCN(C(=O)CN(C(=O)C(C)C)C)CC1)CCCC Cc1nn(CC(F)F)cc1C(=O)NC1CCCC1CNC(=O)C(C)n1cncn1 N1(C(CN2CCC(C(C)(C)O)C2(C)C)=O)CCC2(CCC2)C1.c1(CN)ccccc1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(C(C)NC(c1cc(CO)on1)=O)CO c1(CC(=O)NC(C(C)NC(C2(CSC)CC2)=O)C(C)C)cncc2ccccc12 c1(C(N(C2CCN(C(C3OCCN(C(C)C)C3)=O)CC2)C)=O)cc2sccc2s1 N1(C(C(N2CCCCCC2)C)=O)CCC(C)(CCNC(C2(C)CC=CC2)=O)C1 CC(C)CC(C(=O)N1CCC(C(C)(C)NC(=O)C(CN(C)C)N(C)C)CC1)N(C)C Cc1cc(C(=O)NC(C2CCCN2C(=O)C(C)C(C)C)(C)C)nn1C Cc1cc(Br)cc(Cl)c1NC(=O)C(C)Sc1ccc(N2CCC2)cc1 C1(C(=O)OC)CCN(c2nnc(CNC(C34CC(C)C3C4)=O)n2CC(C)C)CC1 c1(C(=O)OC)cc(N2CCC(NC(=O)CCC(F)(F)F)CC2C)nc(COC)n1 c1(C(=O)NC2(CNC(C3(CC)CCOC3)=O)CCC2)ccc(C(C)(C)C)c(Cl)c1 C1(NC(c2c(C)c(C3CC3)on2)=O)CCCCN(C(c2cnoc2C(C)C)=O)C1 N1(CC)CC(NC(c2csc(C(=O)NCCOC(C)(C)C)n2)=O)CCC1=O c1(OC)ccc(CC(=O)NC2CCCN(C(=O)COC3CC(F)(F)C3)C2)c(F)c1 C(=O)(C1=Cc2ccccc2C1O)NCC1(CNC(CC(CCCCC)C)=O)CC1 C1(C)(OC)CCN(C(c2cccc(C)c2F)C(=O)NC2COC2)CC1 c1(C(N(CCNC(CC=CC=C)=O)C)=O)cncc(C(=O)OCC)c1.C(C)(C)C C1(NC(CCCOC)=O)CCCCCN(C(=O)Cc2ccc(OC)cc2)C1 N1(C(CCOCCN(C)C)=O)CCCC(CNC(=O)CCN2CCC(C)(C)C2)C1 c1(C(=O)NCC2CCCCN(C(C)=O)C2)coc(S(=O)(=O)N2CCCC2)c1 c1(CCC)cc(C(=O)NCC(C)(CC)NC(=O)CCCc2nc(C)cs2)ccn1 N1(C(CCC(N)=O)=O)CCC(CNC(c2ccc(O)nc2)=O)C(F)(F)C1 N1(C(C=C(CC)C)=O)CCCC(C)C1CNC(c1cc(C(F)F)nn1C)=O C1(NC(c2cc(C(F)F)ncn2)=O)C=CCN(C(C2(CF)CCOCC2)=O)C1 N#Cc1ccc(S(=O)(=O)Nc2ccc(SCC(n3ccnn3)=O)cc2)cc1 c1(N(C(CCN(C(=O)C(O)CC(N)=O)CC=C)=O)CC)cnn2c1OCCC2 C(C(=O)NCC(CO)NC(=O)CCCc1ccncc1)(C(C)C)SCC c1(COC)cccc(CC(=O)NCC2CCCN(C(c3c(C)n[nH]c3C)=O)C2)c1 CC1COCC(C(=O)NCC2CC(NC(c3coc(Cl)n3)=O)C2)O1 c1(C(N(C(C)C)CCN(C(=O)Cc2cnn(C)c2)C)=O)csc2nnsc12 C1(C(N(CC(CC)NC(C23CC(C(F)F)(CO2)C3)=O)C)=O)CCCCC1F c1(C(=O)NC2(COC)CN(C(c3cc(CC)c(C)s3)=O)C2)n[nH]c2c1CCSC2 c1(COC)nsc(CCCOC(C2C(C)CC2C)=O)n1 C1(CNC(CCOCCOCC)=O)CC2CCCC2N1C(=O)CC1CCC2CC2C1 C1(CNC(C(CC)n2cncn2)=O)CC(OC)CN1C(c1ccc(C(F)F)s1)=O c1(N(CCCCN(C(Cc2c(C)nc(C)s2)=O)C)C)cnc(C#N)cn1 N=c1nc(N2CCC(F)(c3ccccc3)C2)[nH]c(=NCC2(CO)CC=CC2)[nH]1 C1(NC(CC=C=C)=O)CCCCN(C(c2ccc(NCCS(C)(=O)=O)s2)=O)C1 CCC(CNC(C1CC12CCC2)=O)(CC)NC(c1ccsc1Cl)=O C1(C(=O)NC2(CC(C)C)CC2)CC2(CCN(C(=O)CC3CC4CC4C3)C2)C1 C1(CNC(C(CC)F)=O)CN(C(=O)CCCNS(C)(=O)=O)CCC1C(F)(F)F C1(CNC(c2cc(C)ncc2)=O)CC2CN(C(=O)C(C(C)C)OCC(C)C)CC12 N1(C(=O)Cc2cn[nH]c2)CC2C(c3ccc(Br)cc3)(C1)CS2(=O)=O S(=O)(=O)(c1ccc(NCc2cn(C)nc2Cl)nc1)NCC(C(C)O)C N1(C(C(=O)OCC)=O)CCC2(CC1)CC(NC(c1c(Br)cnn1C)=O)CCO2 CC1CN(C(C2CC2(C)C)=O)CCCN1C(=O)CCCc1c(F)cccc1F C1(CC=C)(NC(c2cncc(Cl)c2)=O)CCN(C(C2CCC(=O)N2)=O)CC1 c1(C(N(C2CN(C(c3n[nH]c(C)c3C)=O)C2)C)=O)cnc2cccc(C)n12 N1(C(c2nc(CC)oc2)=O)CCC(NC(=O)C(F)=C(C)C2CC2)C(CO)C1 C1(C)(NC(C)=O)CCN(C(C2CCC2NC(=O)Cc2ccnc(O)c2)=O)C1 c1(C(=O)NCC(CN(C(c2cc(SC)oc2)=O)C)C)cc2c([nH]1)CCCC2 C(=O)(CC(C)C(F)(F)F)NC1CCC(CCC(=O)NC(C)Cn2ccnc2)C1 c1(C(=O)NCC2(F)COCCN(C(CSCC#C)=O)C2)ccc2c(c1)N(C)CC2 C1(C(C)NC(c2ccc(Nc3cccc(C(F)F)c3)cc2)=O)OCCOC1(C)C C12(C(N(C3CCN(C(c4cnc(Cl)s4)=O)CC3)C)=O)CC(C)(C1)OC2(C)C C(C(C)C(C)C(=O)NCC(C)(C1CC1)NC(=O)Cc1cncc(C)c1)OC Cc1cc(C(=O)NC2(C)CN(C(C3C=CC=CC=C3)=O)C2)nn1C(C)(C)C C1(NC(CN(C(CCSCCC)=O)C2(C(=O)OC)CC2)=O)CC(C#N)C1 CN1CC2C(C(=O)NC3CCCC(CC(=O)NCCC4CC=CC4)C3)C2C1 Cc1nn(C)cc1-c1cn(C2CCC(CNC(=O)C(C)(C)CC3CCC3)C2)nn1 C(=O)(C(O)C(C)(C)C)N1CCC(CC(N2CCC(OCC#C)C2)=O)CC1 CC1(C(=O)NC(CC2C(CNCCN3CC(C(N)=O)C3)C2)=O)CCCC1O n1(C2(CCO)C(c3cn(C(C)CNC4CCCC4O)nn3)C2)cc(C#N)cn1 Cc1nnc(O)c(C(N2CCC(NC(c3ccnnc3O)=O)C(F)C2)=O)c1C C1(CNC(=O)C(O)C(F)F)CCCCN(C(=O)Cc2ccc(O)cc2)C1 Cc1c(F)cc(CN2CCCC2C(=O)Nc2c(F)ccc(F)c2F)cc1F C1(n2cc(C(C)NC(C3CC(CO)C3)=O)nn2)C=CCC(CN(C)C)C1.C(N)=O C1(C(N(C)CC2CCCN2C(C2(F)CCC2)=O)=O)CC(C)(C)CO1 N1(C(c2ccc3c(c2)CCC3)=O)CCC2(CCCN2C(=O)CCC(F)F)CC1 N1(C(COCCC=C)=O)CC2CC1CN(C(c1c(Cl)sc(C)c1C)=O)C2 c1(NC(N2CCC(c3ccc(OC4CC4)nc3)C2)=O)cc(F)ccc1I C1(CNC(C(C)Sc2ncccn2)=O)CC2CCC1N2C(=O)CCN1CCCC1 c1(NCc2ncc(C)nc2)nc(=NCCc2nncs2)[nH]c2c(C)nn(C)c12 C1(NC(CCNC(C)=O)=O)CC(NC(c2n[nH]cc2Br)=O)C12CCC2 C1(N(C(=O)Cn2ccnn2)C)CC2CCC(C1)N2C(C1CCCC(C)(C)C1)=O c1(C(N2CC(N(C(CC(C)n3cccn3)=O)C)C2)=O)cn(C)c(C(F)F)n1 C(CNC(c1ccc(Cl)cc1)=O)(CC(=O)NC(c1ccncc1)C)OC C=CCC(C(=O)N1CC(NC(=O)C(C)C)C1)NC(C)CC(=O)OC C1(NC(C(C(=O)OC)C)=O)C2CC1CN(C(C1CC(=O)NC1(C)C)=O)C2 C1(O)CCCN(C(=O)COCCC(C)C)C1.C(=O)(CCOC)NCCOCCC c1(C(=O)NC2CC(CNC(C3CC(C)C3)=O)C2)cccc2cccc(O)c12 c1(C(=O)OC)ccc(CC(=O)NC2(CCCNC(C3CC34CC(O)C4)=O)CC2)cc1 Cc1cc(C(N2CC(CCNC(c3cn[nH]c3)=O)C(C)C2)=O)ccc1Br N1(C(C(C)n2cccn2)=O)CCC2(CC1)CC2CNC(C1CC2C=CC1C2)=O C1(C(=O)NC(C)CCCCNC(=O)C(=O)C=C=O)CC2(C1)CC1(CCC1)C2 c1(C(=O)Nc2c(C(=O)NC)nccc2)ccc(C)nc1-n1cncn1 c1(CNC(C2(F)CCN(C(CCCC#C)=O)CC2)=O)cc(F)cc(C#N)c1 C1(NC(=O)NC2CN(C(C)=O)C2)CCC2CC2C1 C1(NC(CCN(c2ccccc2)C)=O)CC2CC1N(C(C1(C)CCC(=O)N1)=O)C2 c1(C(=O)NC2(CNC(C3C(C)(C)CC3)=O)CCCCC2)ccc2c(c1)CCOC2 C1(C(N(C2C(C)CC2)C)=O)CC1C1CN(C(c2coc(C(N)=O)c2)=O)C1 C#CCC(C(=O)N1CCC(CN=[N+]=[N-])CC1)NC(=O)CC(C)c1ccco1 C(=O)(C(C)(C)n1ccc(C2CC2)n1)NCCCN(C(C1C(C)CC1)=O)CCO n1(CC(=O)NCCC2CCCN(C(C(C)C(C)(F)F)=O)C2)ncc2ncccc12 CC(C)C(C)(O)C(=O)N1CC(NC(c2cnc(S)n2C)=O)C1 C(=O)(CCCCCNC(=O)C(O)C1CC1)NCCCCCC C(=O)(C(C)(C)S(C)(=O)=O)N1CC(O)(C(C)NC(c2cncc(OC)n2)=O)C1 N1(C(C(CC)COC)=O)CCC2CCN(C(=O)C#CC3(C)CC3)C2C1 C1(CNC(C2CCNC2=O)=O)CN(C(=O)Cc2cc[nH]c2)CCC12CCC2 C12(C(=O)NC3(CC=C)CCOC3)CCN(C(c3c[nH]nc3C)=O)CCC1C2 C1(NC(Cc2onc(C)n2)=O)CC2(CCCN(C(c3ccnc(Cl)c3O)=O)C2)C1 n1(CC)nc(C(=O)NC(C#N)C(N)=O)cc1C.N12CCC(CC1)C2=O c1(C(=O)NC2C(CN(C(=O)CC3CC=CC3)C)CC2)ccn(C2CC2)n1 N1(C(CCc2c(C)ncs2)=O)CCC2(CC1)CC(NC(=O)CN1CCC1C)C2 CCC(C)(C)CC(=O)N1CC2CCC1C2NC(c1ccc(F)c(C)c1)=O c1(C(=O)NC2(C)CCN(CCC(=C)C)C2)cc(C)nc(O)c1 c1(C(=O)NC(C(C)NC(c2c(CC)nccc2)=O)C)ccc(CN(C)C)c(Cl)c1 c1(CC(=O)NC(CC)CNC(=O)CC2CCC3(CC3)CO2)csc2nc(C)cn12 N1(C(C2CCN(C(=O)Cc3cc[nH]n3)C2)=O)CC2(CCC1CO)CC2 N1(C(C2(CCC)CC2)=O)CCC(O)(C(C)NC(=O)CN2CCC(=O)NC2=O)CC1 C1(CNC(CCn2c(C(C)C)ncc2)=O)CC(C)CN(C(C2(C#N)CC2)=O)C1 C1(C(=O)NCCCN(CCCNC(C2CC=CCO2)=O)C)COC(=O)N1 C1(C(=O)NC2CN(C(CCC(=O)NCCC)=O)CC2C)CC2(C1)CC(F)C2 C12(NC(=O)CCCCN3CCCCC3)CCC1CN(C(=O)C1=CSCCO1)C2 c1(C(=O)NCC(CC(F)(F)F)NC(=O)CCc2ncc[nH]2)ccc([N+](=O)[O-])cc1 N1(Cc2ccc(OCCC)cc2C)C(=O)CCN(CC2CCC(=O)N2)C1=O c1(C(=O)NCC2(OC)CN(C(=O)C(F)n3cccn3)C2)cc2cccc(C)c2[nH]1 Cc1cc(C(=O)NC2CCN(C(=O)C(C)(C)C(F)F)C2C)c(Cl)cc1Cl C(c1nc(C)c(C)[nH]1)=CC(=O)NC1CCN(C(C(CC)C)=O)C1 c1(NC(=O)Nc2sc3c(c2C(=O)N=c2cc[nH][nH]2)CCC3)cc(I)c(F)cc1F N1(C(CCCSC)=O)CCN(C(N)=O)CC1.N1(C(CNC)=O)CCN(C(=O)C(C)CO)CC1 N1(C(C(C)=C(C)C)=O)CCCCCC1C(=O)NCC1CCCC1 c1(C(=O)NC2CC(NC(c3n(CC)ncc3)=O)C2)ccc2c(c1C)NC(=O)C2=O C(CCCN=c1cc(C)c(S(=O)(=O)NC2COC(C)(C)C2)c[nH]1)=CC c1(NC(C2CCN(C(CNC(COC)=O)=O)CC2)=O)nc(OC)nc(OC)n1 N1(C(C2CC2CC)=O)C2CCC1CC(NC(C1(CC)COC1)=O)C2 c1(C(N(CCC(C)NC(C2C(CC)OCC2)=O)C)=O)ccc2c(c1)nc(C)n2C C(C(N=[N+]=[N-])C(=O)N1CCC(N(C(=O)CC2(OC)CCC2)C)C1)OCC c1(C(=O)NCC(CO)NC(Cc2c(C)nn(C)c2Cl)=O)cccc([N+](=O)[O-])c1 c1(OC)cc(C(=O)NC(C)C(CO)NC(C2CCC2C#N)=O)[nH]n1 N1(C(Cn2ccc(C)n2)=O)CCC(C(O)CNC(c2oc(C)nc2C)=O)CC1 C1(C(=O)NC2(C(=O)NCc3n(CC)cnc3)CSC2)CCC(C)(C)CC1 C1(NC(c2c(C(C)C)ccs2)=O)CCCC(NC(=O)CC(C)n2ccnc2)C1 CC1(CO)CC(O)CN1C(=O)CCOC1CN(C(c2ccoc2Cl)=O)C1 CCC(CC(=O)NCCCCNC(c1cnn(CC)c1Br)=O)C(C)(C)C C1(NC(C(COC)OC)=O)CC2CC(C1)N(c1ccnc(C3CCC3)n1)C2 C1(CCNC(C2C(OC)CC2)=O)CN(C(C2CN(C(C)C)C2)=O)CC(C)O1 Cn1cc(C(=O)NC2CCC2CNC(c2ccccc2F)=O)n2cncc2c1=O C1(C(C)NC(c2c(CC)ocn2)=O)CCCCN1C(=O)CCc1csnn1 C1(C2CC2)(C(=O)NCCC2CCCO2)CN(C(C2CC3CCC3C2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CCN(C(=O)CC(C)O)C(C)C1 N1(C(c2ccc(CC)o2)=O)CCC(F)(C(=O)NC2(C)CCC(O)CC2)CC1 c1(C(C(=O)NC(C)C)N(C)Cc2ccccc2Br)ccc(Br)cc1F c1(CNC(CCCn2cc(-c3ccc(=N)[nH]c3)nn2)=O)cccc2c1OCC2 CC1CCC(CNC(c2sc(F)cc2Cl)=O)CN1C(=O)CNC=O c1(C(N2CCC(CC=C)(C(=O)NC3CCCC3COC)C2)=O)cnn(C)c(=O)c1 Cc1ccc(C(N2CC(NC(=O)C(c3cccnc3)C)CC2C)=O)cc1Cl N1(C(=O)CCC2CC2)C2CCC1C(NC(C1(c3cncc(Br)c3)CC1)=O)C2 N1(C(c2cc(CCC)n(C)n2)=O)CCCOC(CNC(=O)C=CC=CCC)C1 C(C)(CN=c1[nH]c(Cl)nc(C(C)C)c1C#N)N(C)C.Cc1nn2c3sc2cc13 c1(C(=O)NC(CCNC(c2c(COC)cc[nH]2)=O)(C)C)nc(Cl)sc1C Cc1cc(=NCC2CCCN(C(=O)C(C)SC(F)(F)F)C2)nc(O)n1C(C)(C)C C1(CC(=O)NC(CC)(CC)C2CC2)C2CCC(C2)N1C(c1ccc(=N)[nH]c1)=O N1(C(c2cn(C)nc2)=O)CC2CCN(C(c3ccc4cccnc4n3)=O)C(C2)C1 C(=O)(CCC(C)(C)C#N)NC1CCCCN(C(c2cc(CC)cc(F)c2)=O)C1 C1(CNC(C2CC(CC)(CC)C2)=O)(NC(c2cccc(N)c2)=O)CCOCC1 c1(NC(=O)CC2COCCN2C(c2nc(Br)cs2)=O)nc2cc(Cl)ccn2n1 C(CC(C(F)F)N1CCC1)NC(=O)C(c1cccnc1)C1CCCCN1 c1(N(C(C)(CCOC(C)C)c2nnnn2CC(F)F)CC)ccccc1C(N)=O CC(CC(=O)NCCOC1CCN(C(=O)C=CC2(C)CCOCC2)C1)C(F)(F)F C(CC(=O)NC1(C)CCSC1)(C(F)(F)F)NC(c1cc(CCC)[nH]n1)=O c1(CNC(c2n(CCCCCC)nnn2)c2cnnn2C)cc(C)ccc1Cl C1(C(=O)NC2(CF)CCN(C(C(C)NC(CC)=O)=O)C2)CCCC2C1C2(F)F N1(C(c2cncc(COC)c2)=O)CCN(C(C2(OC)CCCCC2)=O)CC1CF N1(C(CCc2cnc(C)o2)=O)CCC(C(=O)NC(c2cncs2)C)C(C)(C)C1 CC(C)(CC(=O)NCC1CC(F)CN1C(=O)CC(O)c1ccccc1)C1CCCC1 C=C(C)CC(C(=O)N1CC(N2CCCCC2)C1)N(C)CCOCCC(=O)NC CC1CN(C(c2cc[nH]c(=N)c2)=O)CCC1NC(c1cc(Cl)nnc1O)=O C1(N(C(c2sc(CCC)c(CC)c2)=O)C)CCN(C(c2cc[nH]n2)=O)CC1C c1(C(=O)NCC2N(c3nnc(C)s3)CCC2)cc(F)c(F)cc1F S(=O)(=O)(CC(C(F)(F)F)NC(=O)N(C1CCCC1)Cc1ccco1)N(C)C C(c1nccs1)=CC(=O)NCC1CC1CNC(C1CC1C(F)F)=O C1(F)(CNC(C=CC=CC)=O)COCCN(C(c2ncccc2C2CC2)=O)C1 C1(C)(CNC(c2c(C(C)C)ocn2)=O)CN(C(=O)CN(C2CCSC2)C)CCO1 C1(NC(c2[nH]cc(C(N)=O)c2)=O)CC(O)CN(C(=O)CCCc2ccncc2)C1 CN1CCN(C(=O)CCSC(F)(F)F)C(CNC(C2CC23CCSCC3)=O)C1 N1(C(c2scc(OC)c2)=O)CC(NC(=O)C2=C(C)CC2)C(C2CC2)C1 C1(CC(=O)NCCC(=C)C)C2CCCC2N1C(=O)CC12CCCC1C2 N1(C(c2c(C)scc2)=O)C2CCC1CN(Cc1ccc(O)c(O)c1)C2 Cc1c(C(=O)NC(C2CCOC2)CNC(c2ccoc2C2CC2)=O)cncc1F N1(c2cc(N(C)Cc3ncc(Br)cn3)nc(C(C)C)n2)CCC2CN(C)CC2C1 N1(C(c2c(SCC)cncc2)=O)CCC(NC(=O)CC2CCCSC2)C(F)C1 C1(F)(CNC(CSCCC#N)=O)CC(CNC(C2CCC(C(F)(F)F)C2)=O)C1 c12ccc-1cc2.C(=O)(C(C)CF)NC(C(C)N)C.C(=O)CSC(F)F Cc1nn(C)cc1C(=O)NCCC1CN(C(=O)CNC(c2ccco2)=O)CC1C c1(C(=O)OC)cccc2nc(CN3CCNC(=O)C3C(=O)O)[nH]c12 N1(C(C=C(C)I)=O)CC2CC2(NC(c2nnsc2C(F)F)=O)C1 c1(C(N(CC(CN(C(CCN(CC)CC)=O)C)O)C)=O)ccc(CN(C)C)nc1 N1(C(CNC(CC(C)OC)=O)=O)CCCC(C)(F)C1 C(=O)(CCCCC(C)C)NCC(CC(F)(F)F)NC(c1nn(CC)c(O)c1)=O C1(C(N2CCC(CCNC(c3nnc(O)cc3O)=O)C2)=O)Cc2ccccc2S1 n1(C(C)C)cc(CC(=O)NCCC2CCC(NC(=O)C=CCN3CCC3)C2)cn1 C(CC(C)C(=O)NCC1(NC(=O)Cc2nncn2C(C)C)CC1)OC C1(C)(CC)C=C(C(=O)NCCCN(C)C(C2CCCN2c2ncccn2)=O)C1 c1(CNC(c2c(N)c(Br)c(Br)cc2F)=O)nc2cc3c(cc2[nH]1)OCO3 C1(CNC(c2cc(C)nn2C)=O)CCC(C)(C)CN1C(=O)C(O)CC(N)=O c1(C(=O)NCC(CC2CN(C(COCC#C)=O)C2)(C)C)cc2ccc(Cl)cc2o1 c1(NC(c2cccs2)C)ccc(S(=O)(=O)N2CCCC2C2CCCOC2)c(Cl)c1 Cc1cc(F)sc1C(N1CC(CNC(=O)CNC(c2cccc(O)c2)=O)C(C)C1)=O N1(C(C2CCC(O)CC2)=O)CCCC(C(N2CCN(CC3CC3)CC2)=O)CC1 C12(CCC13CCC3)C(=O)N2.c1(OC)cnn(C)c1-n1cc(COC(N)=O)nn1 c1(OC)cnc(C(=O)NC(c2cccc(Cl)c2Cl)CNC(=O)C(C)CO)c(F)c1 c1(C(=O)NC(CNC(C(Br)=C(C)C)=O)C2CC2)ccc(C#N)[nH]1 C12(C(=O)NC3(C)CN(C(=O)CC4CCCOCC4)C3)CCCC1C2Br c1(NC2CCCN(CC)C2)nc(C)cc(=NCC2(C(F)(F)F)CCCC2)[nH]1 N1(C(CC(C(=C)C)O)=O)CCC(N(C)C(c2cnc3ccccc3c2)=O)C2(CC2)C1 c1(OC)cnc(SC)[nH]c1=NC1CCCN(C(=O)Cc2cnn(C)c2)C1 N1(C(CC)C)CCN(C(=O)C=CCN(C)C(c2sccc2OC)=O)CC1 c1(C(N2CC(NC(C3(C=C)CCC3)=O)C(F)CC2)=O)cc2c(F)cc(C)cc2[nH]1 c1nc(NCc2ccns2)cc(C2(C3CCCCO3)CCC2)n1 c1(C(CC)=O)cc(C(=O)NCC2=CCN(C(=O)CCCNC(N)=O)CC2)ccc1F CCC(CC(=O)NCNC1(CN)CCCCC1)CC(F)(F)F c1(C(N(C2CCN(C(c3csc(C4CC4)n3)=O)C2)C)=O)cc2occc2n1C C1(C(N(C2CC3(CC3)C2)C)=O)CCN(C(=O)c2cnnc(O)c2)O1 C1(CNC(c2n(CC)ccn2)=O)CC(C)CN(C(c2ccc(=N)[nH]c2C)=O)C1 CC1(C)C2CCC(C(=O)NC3CC3CNC(c3cnc(O)c(F)c3)=O)C1C2 c1(C(=O)OC)cccc(S(=O)(=O)Nc2ccco2)c1.C12CC3(C1)CN(C3)C2=O C1(NC(CCC)=O)CC2CCC1C(NCCCC1CC1)C2 C(=O)(C1=NOC(C)(C)C1)NC1(CO)CCN(C(Cc2c(C)nc(C3CC3)s2)=O)C1 O(NC(=O)C(Cc1ccncc1)NC(=O)C(C1(O)CCCC1)F)CC#C n1(CC(=O)NC(CN(C(C2C(OCC)C2C)=O)C)C)cc[n+](C)c1 c1(C(c2cncn2C)NCCNC(CN(C(C)=O)C)=O)ccccc1 CCCC(C)(CC)C(=O)N1CC2(COC(CNC(=O)C(F)(F)C3(O)CCC3)C2)C1 c1(CC)cnccc1C(=O)N(C1(CC(=O)N(C)CC)CC1)C C12(CCOCC1)C(=O)NC2.CCC(C(=O)NC12CC(C)C1C2)C1CCOCC1 N1(C(C=CCC)=O)CC2CCC(NC(c3coc(C(F)F)c3)=O)CC2C1 c1(C(=O)NC23CC(CNC(C4(OC)CCC4)=O)(C2)C3)ccc2ccccc2c1O C(C1CCCC1)=CC(=O)N1C(C)C1=O.c1(C(CNC(CC)=O)O)cn(C)cn1 Cc1ccsc1CC(=O)NC(C1CCOC1)CNC(=O)Cn1nnnc1C N1(C(C2CC(OC)C2)=O)CCC(N(C)C(c2cnc(C)[nH]2)=O)C1 C1(COC)(NC(=O)C(C)CCc2cccc(F)c2)CCN(C(=O)C(C)C(C)C)C1 c1(-c2cn(CC)nc2)c(Cc2scc(C(N3CCCC3(C)C)=O)n2)cccc1Br CCS(=O)(=O)c1cnc(O)c(C(=O)NC(C)CCCCNC(=O)CSCC#N)c1 N1(C(C=CCOC)=O)CC2CCOC2(CNC(C2CC2c2cnccc2C)=O)C1 C1(C=O)CCOC(C)C1.C(CCC(=O)NC1CC(N)C1)ONC(=O)OCCOC c1(C(=O)OC)cccc(Cl)c1NC(c1ccc(C(N2CCCC2C(N)=O)=O)[nH]1)=O C1(C(=O)NC(CO)C(=O)NCC2CCOC2)C2CCCC12 C(=O)(CCC(C)(C)c1ccccc1)NC1(C)CC(NC(Cn2ncn(C)c2=O)=O)C1 C1(CC(=O)NCC(C)(C)CNC(=O)COc2ccccc2)CCC(=O)NC1 Cc1cccc2cc(C(=O)NCCC3(CNC(c4n[nH]c(=N)s4)=O)CC3)oc12 C1(CNC(C2CCS(=O)(=O)CC2)=O)CCCCN(C(=O)CCc2ccc(O)nn2)C1 c1(OCC(N2CCC(CNC(CCC=CC)=O)CC2)=O)cccc2ccccc12 C(=O)(CCC(C)(C)C)N(C)CC1CCN(C(c2ccc(=O)n(C)n2)=O)CC1 Cc1cc(C)c(C(=O)NC2(CNC(C3CCC(C)CC3)=O)CCCCCC2)cn1 N1(C(C2(CCCC)CCC2)=O)CC(C)OC2(CCN(C(=O)CNC(=O)OCC)C2)C1 c1(OC)cccnc1C(=O)NC1CN(C(C2CCS2(=O)=O)=O)C1 C(=O)(C#CC1(C)CCCO1)N1CCC(C(C)C(N2CCC(CO)C(C)C2)=O)CC1 c1(C(=O)NCc2ccc(NC)cc2)cccc2c1OCCN2 N1(C(C=NOC)=O)CCC2(CC1)C(NC(c1ccnnc1Cl)=O)CS(=O)(=O)N2C C1(C)(C(N2CCN(C(C(C)(C)C)=O)CC2)=O)CC2CCC1O2 C(=O)(C(O)CC(C)C)NCCCN1CCC(NC(CCC=C=C)=O)C1 N1(C(c2ccc(CO)[nH]2)=O)CC(C2(NC(=O)CN(C)C(=O)OC)COC2)CC1=O c1(C(=O)OCC)ccsc1CNC1CCCC1NC(C1OCCC1C(F)(F)F)=O C(=O)(C(C)(C)CCC#N)NC1C(C(F)(F)F)CCN(C(CC(CC)OC)=O)C1 c1(-c2cc(C)c(F)c(C)c2)ncn2c1CN(C(=O)C(C)(C)CCl)CC2 CC1C(C(N2CCN(C(=O)CS(C)(=O)=O)CC23CCC3)=O)OC2CCCCC12 Cc1ccc(CC(=O)NC(CNC(c2cc(O)ncn2)=O)C2CCC2)cc1C c1(OCCC(C)C)cccc(NS(=O)(=O)C(C)CN2CCNCC2)c1 c1(NC(c2cc(CNC(C(C)OCCC=C)=O)on2)=O)ccc(C2CC2)nc1 CCCCCC(F)C(=O)NC(Cn1ccnn1)C(=O)N1CC(CO)(OC)C1 N1(C(C(C(C)O)C)=O)CCC2(CCN(C(=O)C=Cc3ncc[nH]3)CC2)C1 C1(C(N2CC(CNC(c3cnc(OCC)s3)=O)(OC)C2)=O)CC(C2CCCC2)C1 N1(C(CC(C)Nc2cccnc2-n2nccn2)=O)CCN(C(C2CC2)OC)CC1 c1(OC)ccc(Cl)c(C(N2CC(NC(=O)C3=CCCSC3)CCC2C)=O)n1 Cc1cc(C=CC(=O)NC2CCN(C(=O)CC3CC(F)(F)C3)CC2)on1 C1(CC=C)(C(=O)NCc2csc(CNC(=O)C(CO)OC)n2)CC=CC1 C(=O)(C(C)S(C)(=O)=O)N(C)CC1CCCN(C(c2cc(C)nn2C2CCC2)=O)C1 C(=O)(CC1=CCOCC1)N1CCC(CNC(C(C)OCCCC)=O)C1 CCC(CC(=O)NC1(C(=O)NC(c2ccccn2)CO)CCOCC1)C1CC1 c1(C(c2nnnn2CCCSC)NCC(CC)CC)cc(Cl)ccc1OC C1(O)(CN(C(=O)C#CC2CC2)C)CCN(C(C2CC3CC3C2)=O)CC1 C1(C(=O)NCC(C(CC)C)C)CN(C)CCN1C(=O)C(C1CC1)SC N1(C(C2CCC(OC)CC2)=O)CCCCC(CNC(C2COCCN2C)=O)C1 C(C(C)(O)CCOC)NC(C1N(C(C=CC=CC)=O)CC=C1)=O C(=O)(C1=CCCCO1)NCC(C)N(C(=O)CSC(F)(F)F)CC c1(C(N2C(C(N(CC(C)C)CCC)=O)CC(O)C2)=O)cc(F)cc(Br)c1 C1(NC(C2(N=[N+]=[N-])CC2)=O)CC(O)CN(C(=O)CCc2cncs2)C1 c1(-c2cn(CC3(C4CN(OC)C(=O)C4)CC3)nn2)cc2c(C#N)cccc2[nH]1 C1(C(N(C)CCn2cc(C(C)(C)C(N)=O)nn2)=O)C2CNC(=O)C12 c1(CNC(C23CCCC2C3)C(=O)OC)ccc(C(F)(F)F)c(OC)c1 C1(c2ccccc2)(C(=O)NCC2(NC(C3(Br)CC3)=O)CC2)CCCCC1 CC(O)(CNC(=O)CC(CC1CC1)NC(C1CC(=C2CCC2)C1)=O)CCO c1(C(=O)NC(CC)CNC(c2cnc(S)n2C)=O)cccc(OC(F)F)c1OC C(=O)(CCN=c1[nH]c2ccccc2s1)NC(CCNC(C(CC)SC)=O)C C1(CC(=O)NCC(C)CN(C)C(c2ccnc(N(C)CCO)c2)=O)NC(=O)NC1=O Cc1cc(C(=O)NC(C)(C)CN(C)C(C23CCC(C2)C3)=O)c(C)[nH]1 CC(CF)C(=O)N(CCNC(=O)CCCc1ncco1)C1CC1 C1(NC(COCC(=C)C)=O)CCCN(C(C2C(C)C2C)=O)CC1 C1(CC)CCCCCN1C(=O)Nc1ccc(-c2ccc(C)c(N)c2)cn1 C1(CNC(=O)CNC(c2cscn2)=O)CCCCN1C(=O)C=C(C1CC1)C1CC1 CN1CC(=O)N(CC(=O)NCCN(C(=O)CN(C2CCCC2O)C)C)C1=O C1(C(N(CCN(C)C(C2(F)CCCC2)=O)C)=O)CC(S(C)(=O)=O)C1 C1(C(N(C)CC2CCN(C(c3n[nH]cc3F)=O)CC2)=O)CCC(F)(F)CC1(C)C N1(C(c2cc(NC)nc(Cl)c2)=O)CCCC2(NC(C3CCCC3O)=O)CC2C1 N12CC(C(C)C1)NCC2=O.c1(C(CC)CC)ccccc1 c1(CC)nc(O)c(C(=O)N(C2CCC(NC(=O)CCOC3CCC3)C2)C)cc1C N1(C(C2(OC)CCC2)=O)CCN(C(=O)C(CC(C)C)NC(N)=O)C2(CC2)C1 C(C(CC(F)(F)F)NC(C1CC(=O)NC(C)C1)=O)NC(C1(SC)CC1)=O C(C)(CCN=c1nc(C(F)(F)F)[nH]s1)NC(c1c(C)ccc(C)c1)=O C1(c2ccc(C)nc2C)NC(=S)N(CCc2ccco2)C2=C1C(=O)OC2 C1(CNC(C(C)NC(=O)NC)=O)CC(C(C)C)CCN1C(=O)Cc1ccsc1 c12ccc(cc1)C(=O)NC2.C1(NC(C(C)SC(F)(F)F)=O)CCCC(C(N)=O)C1 C1(CC(=O)NCc2c(OCCN(CCOC)CC)cccc2)CCC(C)(C)CO1 CN=c1nc(NCC(C)Oc2cccc(C#N)c2)[nH]c(=NCCS(C)=O)[nH]1 C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCC(N(C(CCCC=C)=O)CCC)C1 CC(C)CC(C(=O)NCC(O)CNC(c1cn(C2CC2)cn1)=O)C(C)C N1(CC)N=C(C(=O)NC2CCC2CNC(c2ncccc2N(C)C)=O)CCC1=O c1(C(N2CCC(NC(c3n(CC)nc(C)c3)=O)C2C)=O)nc(Cl)ccc1N c1(CC)nc(=NC2(c3nnnn3C(C)CC)CCC(C)(C)CC2)s[nH]1 Cc1[nH]nc(C(N2CCOCC2CNC(=O)CCCN(C)C(C)C)=O)c1N N1(C(c2cn(C=C)nc2)C(=O)NC2CCC2)CCN(C)C(=O)C1CC(C)C S(=O)(=O)(c1cnccc1N1CCCC(C(C)(C)N(c2scc(C)n2)C)C1)N(C)C C(=O)(C(Cc1ccoc1)NC(=O)C(C)CSC)NCC1(CCOC)CC1 c1(OC)cccc(Cl)c1NC(C1CCN(c2nc(SC)ncc2Br)C1)=O C1(CNC(=O)CCc2cccs2)CC2CC(C1)N(C(=O)Cn1cnnc1)C2 C1(C(=O)NC(CNC(c2ccc(-c3ccccc3)[nH]2)=O)C2CCC2)CC2CC2C1 C(=O)(C1=CCCN(C(C2CCC(=O)CC2)=O)C1)Nc1c(OC)nccc1 c1(COC)cc(C=O)cs1.C12CCC1C2.C1(CNC=O)CCC(C(=O)N)C1.OC c1(C(=O)NCC2C3N(C(C(C)CF)=O)CC(CC3)C2)cc2cccc(F)c2o1 c1(C(=O)NC2CN(C(C=CCOC)=O)CC2C2CC2)cc2cccc(F)c2o1 c1(N2C(C)CC(CNC(c3c(C)nn(C)c3)=O)C2)ccc([N+](=O)[O-])cc1Br C12(NC(C=NOC)=O)CCC(CNC(c3ccc(C(C)C)nc3)=O)(CC1)OC2 Cc1ncc(C(=O)NCC#CCNC(=O)CCC2CCCN(C)C2)c(C)n1 C1(C(N2CCN(C(CC(CC)SC)=O)CC2CCO)=O)CCn2c(O)nnc2C1 N1(C(c2ccc(=NCC)[nH]c2)=O)CC2(CCN(C(C3(CC(F)(F)F)CC3)=O)CC2)C1 C12(C(=O)NC3C(C)CN(C(C4CCOC(C)(C)C4)=O)C3)C3C4C1C1C2C3C41C#N C1(NC(C(C)CNC(C23CC(F)(C2)C3)=O)=O)CNC(=O)C1(C)C C12(NC(c3c(C(C)C)sc(Cl)n3)=O)CCCN(C(=O)CC3(N(C)C)CCC3)CC1C2 c1(C2C(C(=O)NC3CC(N(C(=O)Cn4cncn4)C)C3)C2)ccc2c(c1)CCO2 Cc1nc(NCCN2CCOCC2C)cc(N2CCCC(C#N)C2)n1 CC1(C)CCC(C(=O)NCC2(F)CC(CNC(c3ccc(OCF)cc3)=O)C2)OC1 c1(-c2ccc(CN3CC(O)(C(=O)NC(C(=O)OC(C)C)C)C3)o2)ccc(Cl)cc1 C1(CNC(C(F)=CC)=O)(N(C(C2CCN(CC(F)(F)F)C2)=O)CC)CCCCCC1 C1(C(F)(F)F)(NC(c2cn(C3CCNCC3)nn2)=O)CCNCC1 c1(OC)ccc(C(=O)NC2CCCN(C(c3csc([N+](=O)[O-])c3)=O)C2C)cc1F C1(NC(c2c(OC)ncc(F)c2)=O)CN(C(=O)C(=O)NC2CC2)CC12CCOCC2 c1(NC2CC2)ccc(CO)c2oc(C)cc12.C1(C(=O)OCC)CN1CCNC(C)=O N1(C(CC(C)n2cccn2)=O)CCCC(C2CC2NC(C2(C)CC2)=O)C1 c1(CCCC)ccc(C(=O)NC(C)CC(C)NC(=O)CCCC2CC2)cc1 Cc1n[nH]c(C)c1C(=O)NC1CCCC1CC(=O)NC1CCC(N(C)C)CC1 N1(C(C(CC=CCC)C)=O)CCC(C)(C)C(NC(=O)CNC(c2ccsc2)=O)C1 c1(C(=O)NC2CC3CC(NC(C(C)CC(N)=O)=O)C2C3)cnn2cc[nH]c(=O)c12 c1(C(=O)NCCc2cn(C3CC3)nn2)ocnc1CNC(=O)C(O)C1CCC1 c1(C(=O)NCC2C(NC(CNC(CCCCC)=O)=O)CC2)cc(O)nc(C)n1 N1(c2nc(SC)nc(C)c2)CCC2(NC(=O)C=CC=C(Cl)Cl)CCCCCC12 Cc1ncc(Cl)c(C(=O)NCC(C2CC2)NC(=O)C(O)C(F)(F)F)n1 C1(C(=O)NC2(CNC(C(C)CC3CCCC3)=O)CCCC2)CC2CC1CC2(F)F c1(C(C)=O)ccc(N2CCCC(CCNC(=O)C(C)=CC3CC3)C2)nc1 C1(C(=O)NC2CCC23CN(C(=O)CCSc2ccccc2)C3)CC2CCC(C1)S2 c1(C(C)(C)C)ccc(C(N2CCCC2CN(C(c2csc(Cl)c2)=O)C2CC2)=O)cn1 CN1CCCC1C=CC(=O)NC(C1(O)CCCCC1)C(=O)NCCN1CCCC1 C(=O)(C(C)C(C)NC(=O)CCc1ccccc1Br)NC(CC(=O)OC)C1CC1 c1(OC)nc(NC2CC(C)N(C3CC3)C(Cc3csc(O)n3)C2)c2ncsc2n1 C=CC(F)(F)C(=O)NCC(c1ccc(C)cc1)NC(c1ccnn1CCC)=O c1(-n2c(C(c3ccn(C)n3)NCC(CO)OCCO)nnn2)ccc(F)cc1 c1(NC(c2c(NS(CC(=O)OC)(=O)=O)ccs2)=O)cnc(OC)c(F)c1Cl c1(C(N2C(C3(O)CN(C(CCCC(C)C)=O)C3)CCC2)=O)cccc2occc12 N1(C(C2C(=C)C2)=O)CC2CCC1CN2C(=O)CNC(=O)CC C1(CC)CN(C(=O)C(=O)NCc2nc(C3CC3)cs2)CCN1C(C1CC1)=O N1(C(C2(F)C(C)OCC2)=O)CCCC2(C1)CN(C(c1ccccc1F)=O)CCO2 C1(C(=O)N(Cc2ccccc2)CC)CC=CCC1C(=O)OC.n1(CCC)nccc1N N1(C(C(c2cc(C)sc2)(C)C)=O)CC2CC(NC(C34CC(C)(CO3)C4)=O)CC1C2 CCC(C)CCN=c1[nH]c(=NC(CC(=O)NC)C2CCC2)[nH]c2c1CCCCC2 C1(O)(C(N2CCC(O)(CCNC(C=C(CC)C)=O)CC2)=O)CCCC(C)(C)CC1 N1(C(C2C=C(C)CS2)=O)CCC2CN(C(=O)C3=C(Cl)CC3)CCC12 N1(C(c2c(C)oc(-c3cccs3)n2)=O)CCCC12CCN(C(=O)C(C)CF)C2 C(=O)(C1=CNC2=NCCCN12)N1CCCC(N(C(CCCCC)=O)C)C1 C(=O)(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C(C)C)NCCNS(CC)(=O)=O C1(CN(C(C2(C(=O)OC)CC2)=O)C)CCCCC1C.c12cc([nH]n1)CNC2=O c1(NCc2n(CCC)ccn2)ccc(S(=O)(=O)N2CCC(N(C)C)C2)cn1 C(C(CN=c1[nH]c2ncc(Cl)cc2s1)C(F)(F)F)NC(=O)OC(C)(C)C C12(CNC(=O)Cc3cscn3)CC(NC(=O)C(F)C(F)(F)F)(CCO1)C2 N1(C(c2cc(CC)on2)=O)CC2CCC1C1CN(C(=O)C(F)=CCCF)CC21 C(=O)(CS(=O)(=O)CC)N1C(CNC(=O)C(C)NC(N)=O)CC(OC)C1 C1(C(=O)NCCCC(C)NC(=O)CC2CCC(=O)NC2)CN2CCN1CC2C CCC(CCC(=O)Oc1cccc(C)c1)NC(c1cc(C2CC2)n[nH]1)=O CCCCCCC(CC)C(=O)N1CC2CC(C1)N(c1c(F)cccc1[N+](=O)[O-])C2 C(=O)(CCCC(F)(F)F)NC(C)CN(C)C(c1ccc(O)cc1O)=O CN1CCCC(C(N2CCC(C(O)CNC(C3(CO)CC3)=O)CC2)=O)C1 C1(C(N2CCC(CCCO)C2)=O)(COC)C=CCN1C(c1sc(O)nc1C)=O CCCCCCCC(O)CC(=O)N1CCOCCC1C(=O)NCC C(C(=O)N1CCC(C(=O)NCCn2cnnn2)O1)=CCCN=[N+]=[N-] C1(NC(c2c(SC)cn(C)n2)=O)CC12CCN(C(c1[nH]c(C)nc1C)=O)CC2 C(CC(C)C(=O)NC(CN(CC1(CC(=O)OC)CCC1)CC)CC(C)C)=CCC C(=O)(CS(=O)(=O)CC(=O)NC(CNC(=O)CC1CC2(CC2)C1)C1CC1)OC C1(C(N2CC(CCNC(C3(C#N)CCCC3)=O)(OC)C2)=O)CCCCC1(F)F N1(C(COCC(C)C)=O)CC2(CCCC2)C1C(=O)NCCN1CC=CC1 CCC(C)CCCC(=O)NCC1(C)CN(C(c2cc(C)c(N)cc2F)=O)CCO1 c1(OC)cc(C(=O)NCCCCNC(=O)CCc2ncccc2OC)cc(C)c1 C1(NC(C=CCCC(C)C)=O)CC12CCN(C(=O)CCC1CC1C)C2 NS(=O)(=O)c1ccc(CCC(N2CCCC2CNC(C23CSC(C2)C3)=O)=O)cc1 C(=O)(C(C)CCC(C)(C)C)N(CCNC1CN(C(=O)C2=C(C)CC2)C1)CC N12CCC3(CCN(C3)C(=O)C3(COC3)C1=O)C2.c1(CC)cnncc1C c1(C(=O)NC(C(=O)N(CC=C)CCC)C2(O)CCC2)cscc1CC C1(NC(Cc2scc(C)n2)=O)CCCCN(C(=O)CC(=O)NCC(F)(F)F)C1 C12(CNC(C3CC(C)(O)C3)=O)CCC1CN(C(c1cccc(F)c1Br)=O)C2 CCS(=O)CC(=O)N(CCC(=O)NCC1COCCOC1)OC C(=O)(C1=CC2C=CC(C1)C2)N1CCN(C(c2c(C)occ2)=O)CC12CC2 c1(C(=O)NC2CCCN(Cc3c(OC)cccc3O)CC2)cccn2ccnc12 c1(C(=O)NC2(CCNC(C3CCC(C)S3)=O)CCC2)cc2cccc(Cl)c2o1 CCC1CCN(C(=O)OCC2CC(=O)N(C(C)C)C2)c2ccccc21 c1(CNC(C(C)(O)C2CC2)=O)ccc(CNC(=O)Cc2ccc(Cl)cn2)nc1 C(CCC(O)C(=O)NC1CC1C(C)C)NC(c1c(C)n[nH]c1C)=O Cc1ccnc(C(N2CCC3(CC3NC(=O)CCOCCN(C)C)C2)=O)c1N c1(N2CCC(CCC)C2)nc(=NCCCCCOC)[nH]c2c1COC2 C1(CC(=O)N(CCC(C(C)C)NC(C(CCC)C)=O)C)CCn2cncc2C1 C12(C(N(C)CC3(NC(c4ncccc4N(C)C)=O)CC3)=O)CCCN(CC1)C2 c1(N2CC(C)(NC(C3CC4CCCC34)=O)C2)ccncc1C#N C(=O)(C(C)CS(C)(=O)=O)NCC1OCCN(C(C2CC(C#C)(O)C2)=O)C1 Cc1ncc(C(=O)NCCC2(O)CN(C(=O)CC3CCCC(C)C3)C2)c(C)n1 C(=O)(CCCCCOC)N(C1CCN(C(c2ccc(OC)cc2F)=O)CC1)CC C1(N(C(CCCOCC)=O)C)CCN(C(=O)Cc2c(OC)cccc2Cl)CC1C CN1CCN(C(C2C=CCN(C(C3(C)CCCCC3)=O)C2)=O)CC1=O C(=O)(CC(C)C(=O)N1CCC(CF)(NC(=O)CS(N)(=O)=O)C1)OC c1(CC(=O)NC2C(NC(c3cc(C(=O)OC)sc3)=O)C2)c(Cl)cncc1Cl c1(C(C)C)ccc(C(N2CCC(NC(=O)C(C)C(C)(C)C)C(CO)C2)=O)cc1F N1(C(=O)OC)CC2CCC(C(=O)Nc3cccc(OC)c3C)C2C1 C1(C(N(C2CCCN(C(C(CCC)N(C)C)=O)C2)CCO)=O)CC(=O)C12CCC2 Cc1nc2ccccc2nc1C(=O)NC1CN(C(c2ccccn2)=O)CC1O C1(NC(=O)CC2(c3ccno3)CC2)(CO)CCN(C(=O)C=CCN2CCCC2)CC1 c1(C(c2nnnn2CCCOCC)NC(CCCC)(C)C)cc(C(C)C)c(C)s1 C1(NC(C=CC(N)=O)=O)CCN(C(=O)C=Cc2ccc[nH]2)CC12CCC2 Cc1ccc(C(=O)NC2CN(C(=O)C(O)CF)CCC2c2ccccc2)cc1N CC1=C(C(=O)N2CCCC2CNC(c2ccc(C(F)F)cc2Cl)=O)CCCC1 C#Cc1cccc(-c2nc(C(=O)OC)cs2)c1.C1(Cc2ccccc2)CCN1 C1(CC)(OC)CN(C(C2CC(N(C(=O)CCC3CC3(F)F)CC)C2)=O)C1 C(C(C)(C)CCCC)N(C(=O)COCC(=O)OC)C(C1CC1c1ccccc1)=O c1(CC(=O)NCC2N(C(c3scc(S(N)(=O)=O)c3)=O)CC2)ccc2oc(O)nc2c1 C(C)(CCC(=O)N(C1(C(=O)NC2CC2c2cnn(C)c2)CC1)C)OCC N1(C(C(=O)NCc2cc(C)sc2Cl)=O)CCNC(=O)C1c1cccs1 C(=O)(CCCCCOC(C)=O)NC1CCN(C(c2c(CC)cco2)=O)C1 c1(C(N2C(CNC(C(C3CCC3)OC)=O)CC(F)(F)C2)=O)ccc2nc[nH]c2c1 CCC(CC(=O)NC1CC(OCC(N2CCN(C)CC(O)C2)=O)C1)C(F)F N1(C(c2n(CCOC)ncc2)=O)CC(NC(C2OCCC2COC)=O)C(O)C1 C(C(=O)NCc1c[nH]nc1C(=O)NCC1CCCSC1)(C(C)C)OC C1(NC(c2n(C)c(=O)ccc2)=O)CCC2(CC1)CCN(C(=O)CC1CC(F)C1)C2 CCC(C)C(C(=O)NCCOC1CCN(C(=O)C#CC(C)C)C1)N(C)C C1(NC(c2ccc(C(C)=O)o2)=O)COCCC1NC(=O)C(C)=C1CCCC1 c1(OC)ccc(C)c(NC(=O)C(CC2CC2)NC(=O)CCN2CCOCC2)c1 Cc1ccc(C(N2CCC(O)(CN(C(=O)C(C)c3cncs3)C)C2)=O)n1C N1(C(Cc2c(C)nc[nH]2)=O)CCN(C)CC1CNC(c1cc(N)cnc1Cl)=O Cc1cc(N)cc(C(=O)NCC(CNC(C2CCCN2C)=O)CO)c1F COn1cnc(C)c1C(=O)NCC1COCCN1C(c1cnc[nH]1)=O C(=O)(C1Cc2ccccc21)NC1CCC(C)(NC(CCc2onc(C)n2)=O)CC1 C(=O)(C(C)CN(C(=O)CCC=C(C)C)C)N(CCCO)CC Cn1cc(CCCN(c2ccccc2Cl)CC2CCCC2)nc1-c1ccccn1 c1(C(=O)NC(C(C)NC(c2cscn2)=O)C)c(Cl)c2ccccc2n1C C1(C(=O)NC2CCC(NC(COc3c(C)cccc3)=O)CC2)CC2CCC(C1)C2 c1(C(=O)NCC(CNC(c2cnc(O)o2)=O)O)c(F)cc(Cl)cc1Br C#CCCCCCCC(=O)NC1CCC(CC(=O)NC2CCC(C)(C)C2)CC1 C(=O)(CCC(C)(C)C)N(C1CCCN(C(C2C(F)(F)C23CC3)=O)CC1)CC CC1CCC=C1C(=O)N1CCC(F)(CNC(=O)CN(C)C(c2cccs2)=O)CC1 N1(CC(N2CCC(NC(c3cn(CCOC)nc3)=O)C2)=O)CCCCCC1 c1(C(=O)NCC2CC(COC)CN2C(=O)CCn2cnnn2)ncc(F)cc1C C1(C)(CNC(C(C=C)O)=O)CN(c2nc(C3CC3)ns2)CCO1 C1(N(C(C2C(C(=O)OC)C2)=O)C)CCN(C(=O)C(c2ccc(C)cc2)F)CC1 c1(C(C)C)cc(C(N2CC3C(CNC(C4CCOC4)=O)C3C2)=O)n(C)n1 N1(C(c2cc(SC)oc2)=O)CC2CCC1C(CNC(=O)Cn1cc(N)cn1)C2 c1(C(=O)NC(c2ccnn2C)C(=O)NC2C(C)CCCCC2)cccn2cncc12 c1(NC(C2CCCC(NC(c3ccc(Br)cc3O)=O)C2)=O)cc(Cl)ccc1CO c1(C(=O)OC)cccc(C(=O)NC(C)(C)CCCNC(C23COCC(C2)C3)=O)n1 O(NC(=O)C(C)NC(c1ccc(C(C)=O)o1)=O)CCCC=C c1(CNC(c2ccn(C)c2)=O)ccc(C(=O)NCC2CCC(F)(F)C2)cc1 C1(NC(C2C(C)C2C)=O)CCCN(CCc2cc(Cl)cc(Cl)c2)C1C CC1CCCCN(C(=O)C(C2CCNCC2)F)C1 c1(C(N(C(CNC(C(C)COc2ccccc2)=O)C)C)=O)nccc(N)c1Cl C12(OC)CCC(C(=O)NC3CC3NC(=O)CC(C)c3ccccc3)(CC1)C(=O)C2 C1(O)(CN(C(Cc2cc(C)no2)=O)C)CCN(C(c2ccccc2Cl)=O)C1 C1(CNC(c2nn(C)c(F)c2)=O)CN(C(c2ccc[nH]2)=O)C2CCN1C2 C1(CNC(c2ncc(C)cn2)=O)CC2(CC2)CN1C(C1CCCN1C(C)C)=O C1(C(=O)NC(C2CCOC2)C#C)CCCCCN1C(c1[nH]ccc1COC)=O C1(C(N(CCCCNC(Cn2cc(C(C)O)nn2)=O)C)=O)CC12CCOCC2 C1(C(=O)NCC(CN(C(c2c(CCC)occ2)=O)CC)(C)C)CCCNS1(=O)=O N1(C(c2cc(F)cs2)=O)CC(NC(C2(CO)CC2(F)F)=O)C(O)C1 c1(C(=O)NC2CCC(C(=O)Nc3nc(C)c(C)s3)C2)ccc2c(c1)CCC(=O)N2 C(=O)(C1=CC(C)(CC)C1)NC1C2CN(C(C3N(S(CCC)(=O)=O)CCC3)=O)C1C2 c1(C(N(C(C)CCNC(c2ccc(C(F)F)o2)=O)C)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NC(CC)CN(C(=O)CNS(N)(=O)=O)CC)cc(C)n(C(C)C)n1 N1(C(C(C)(C)CO)=O)CCOCC(CNC(=O)CN2CCCCCC2)C1 c1(-c2cc(C)c(-c3ncc(C(F)(F)F)cc3CO)cc2)cnc2ccccc2n1 CC1(C)CC(C)(CNC(c2cnc(O)c(F)c2)=O)CN1C(=O)CC1CS(=O)(=O)C1 CC1CCCn2ncc(C(N3CCC(C(C4CCCNC4=O)=O)CC3C)=O)c21 C1(CNC(C=C(CCC)C)=O)CN(C)CCN1C(C1CC1CCOC)=O C(C(=O)N=S1(=O)CCC2(NC=O)CCCN2CC1)N1CCC(OC)CC1 C(=O)(C1=NNC(C(F)(F)F)C1)NCC1N(C(C=C(C)C(C)(C)C)=O)CCC1 C(C1CCCC1)=C(C)C(=O)NC(C1(O)CN(C(=O)C=CC(=O)NC2CC2)C1)C C1(NC(c2ccc(C#N)s2)=O)C2CC3C1C3C2C(=O)NCC1CC2CCC2C1 N1(C(C(=O)NC(CCNC(C2CCC(CC)O2)=O)(C)C)C)CCCCC1=O Cc1cc(C(=O)NC2CC(NC(=O)CC#N)CC2O)c(Br)cc1F C1(NC(C2C(=O)NCCC2)=O)CCCC12CCCO2 C(C(=O)NCC1CC(NC(=O)CCCC(F)(F)F)C1)(C(C)C)(C(C)C)NC(C)=O c1(C(N2CCC(C(C)C(=O)NCCC(=O)N(C)C3CC3)C2)=O)c[nH]nc1[N+](=O)[O-] c1(C(=O)NC2CC(CNC(C(C=C)(C)O)=O)C2)cccc([N+](=O)[O-])c1OC C(=O)(CCCCCCN=[N+]=[N-])NCC(CC(C)C)NC(=O)C(C)CCN(C)C C(CN=c1[nH]n2cc(C)nc2s1)C1CCN(C(C(CCCOC)C)=O)CC1 N1(C(CCS(CC)=O)=O)CC2(C1)CN(C(=O)Nc1ccc(SC)cc1)CC2C(=O)O Cc1cc(Cl)nc(Cl)c1C(=O)NCC1CN(C(c2cnnc(O)c2)=O)C1 C#Cc1cncc(C(=O)N(CC(C)NC(c2cnc(-c3ccncc3)s2)=O)C)c1 CC(C)(C)CCC(F)C(=O)NC1CC2(C1)CC2NC(=O)Cc1cccc(C#N)c1 c1(C(=O)NC2(CNC(C3CC34CCC4)=O)CC2)ccc(Cl)cc1O c1(C(N2C(CNC(=O)COC3CC=CC3)CCC2)=O)cn2c(n1)SCC2 C1(NC(CCCc2scc(C)n2)=O)CCN(C(=O)COC2CCCC2)CC1O Fc1ccc2c(c1)CCC(CNC1CCCCNC1)O2 N1(C=O)CCOC(CC2(C(N)=O)CCC2)C1.C1(C(=O)NC2CC2)(C(=O)N)CC1 c1(NC(C2(F)CCN(c3cc(C(=O)O)ncn3)C2)=O)ccc(Br)cc1 CC1(CC(=O)NCc2cnc(C3CC3)[nH]2)CCN(C(C2(F)CCOC2)=O)C1 c1(C(n2cc(CN(C(Cc3c(C)nn[nH]3)=O)C)nn2)C)ccc(Cl)cc1 n1(CC)ncc(C(=O)COC(=O)CC2CCCC2C)n1 C(=O)(C(CC1CCOCC1)NC(=O)C(C)n1cccn1)NCC1(SCC)CCO1 C(=O)(C1=NOC2(CCC2)C1)NCC(C(C)(C)C)NC(C(CC=C)CC)=O c1(CCC)cnc(Nc2c[nH]nc2C(=O)Nc2cc(C)c(C)[nH]2)nc1 N1(CC(=O)N(C2CCN(C(C3COCCOC3)=O)C2)C)CCCCC1=O CN1CC(C)(C(N2CCCCC(NC(=O)CCCc3cncs3)C2)=O)CC1=O c1(OC)cc(NC(=O)C(c2ccc(CC(C)CO)cc2)C)c(Br)cn1 Cc1cccc(C)c1NC(=O)C(=O)N(CCC(C)NC(=O)C=CC1CCOC1)C N1(C(C2C(C)C2C)=O)CC(NC(c2ccc(F)c(O)c2)=O)C(C)(C)C1 c1(NC(C2CCN(C(CCNC(C)=O)=O)C2)=O)ccc(Br)c(F)c1 N1(NC2CC3(C(C(=O)NC(c4cc5ccccn5n4)=O)C3)C2)CCC2(CCSC2)C1 C1(NC(CCCn2cc(-c3cn(CCC)nc3)nn2)=O)CCCC2CCC12 c1(CC(=O)NC(C)CCN(C(=O)C(C)C2CCC2)C)cccc(Br)c1F CCCC(C(O)C(=O)N1CCCC1)NC(C1CCCN1CC)=O Cc1cc(CNC(=O)Cn2ccnn2)cc(C)n1.C1(CNC(C2CC2)=O)CCCO1 C#Cc1ccc(C(=O)NC2CC(F)(CNC(C3(C#C)CCCC3)=O)C2)c(F)c1 c1(C(N2CC3C(CNC(c4c(C)cco4)=O)(C3)C2)=O)cc(Br)cnc1F C1(CC(=O)NCC2C(C(=O)NCc3nnc(CC)o3)CCO2)CCCC2CC12 N1(C(CCOCC)=O)CCN2C(=O)C(NC(c3nccc(Cl)c3F)=O)CC2C1 C1(C(=O)NCc2cccc(CO)n2)(NC(c2c(C)nns2)=O)CCN(C)C1 C1(CNC(C(c2cccc(C)n2)C)=O)CN(C(C23CCC(CC2)O3)=O)CCN1C C1(CNC(C2C(CCC)C2)=O)CCCCN(C(=O)Cc2cccnc2)C1 N1(C(c2ccc(Br)cc2)C(=O)NC(CC)(C)C)CCC2C(C(=O)OC)C2C1 C1(C(=O)NC(c2ccc(Cl)s2)C)CN(C(c2ccc(Br)cc2)=O)CC(F)(F)C1 N1(C(CC(CC(C)C)C)=O)CC23CCCC2(C1)CN(C(=O)CCC1CCOC1)C3 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CCCC(N(C(=O)CC(C)C(F)F)C)C2C1 CCCC(O)CC(=O)NCC(c1ccccc1)NC(=O)Cc1ccc(SCC)o1 c1(-c2oc(C(=O)NCC(C#C)C)c(C)n2)ccc(Cl)c(Cl)c1 C12(C(=O)NCC3(C)C(C)CN(C(CN(C(C)C)C)=O)C3)C3C4C1C1C2C3C41C Cc1cc(C(=O)NC2(C(=O)NC(C(F)(F)F)C3CC3)CSC2)on1 N1(C(CCC(N)=O)=O)CC2OCCN(C(c3cc(F)cc(F)c3Br)=O)C2C1 c1(C(N2C(CNC(C3C(CN(C)C)C3)=O)CC2)=O)cn(C)c(=O)nc1O CCCCC(=O)NCC1(O)CC(CNC(C2CCN(c3nccn3C)C2)=O)C1 C(C)(C)(CCC(=O)NCC(c1ccc(F)cc1F)NC(=O)CC1CCOC1)OC C1(C(=O)NCC(CC)(C)NC(=O)Cc2cn(C)nc2C)CCc2nncn2CC1 C1(NC(C(CCNC(C2CN(C)C(=O)N2)=O)O)=O)Cc2cscc2C1 Cc1onc(-c2ccsc2)c1C(=O)NC(CNC(C1CNC(=O)N1)=O)C1CC1 c1(N(C)C)cccc(C(=O)NCC(C(C)(C)C)NC(C2(C(C)(F)F)CCC2)=O)c1 C1(NC(c2c(Br)cn(C)n2)=O)CCN(C(c2ns[nH]c2=O)=O)CC1CO N1(C(CCOCC)=O)CCC(CNC(c2cscc2OC)=O)C(C)C1 C1(C(N(CCC(C)NC(C2CCCCC2O)=O)C)=O)CC(C)(C)OC(C)(C)C1 Cc1c(C(N2CCN(C(=O)C3=C(C#N)CCC3)C3CC23)=O)sc2nccn12 c1(C(=O)NCCC(CNC(C2(C=C)CCOCC2)=O)=C)ccc2ccncc2c1 C1(C(=O)NC2CC(CCOC)C2)CCOCC1NC(c1cc(F)n(C)n1)=O c1(OC)cncc(C(N2CCC(NC(=O)CSC(C)(C)C)C2C2CC2)=O)n1 N1(C(c2cc(CC)on2)=O)CCCC(N(C(=O)CCc2cc(C)nn2C)C)C1 c1(OCCNC(c2c[nH]c(C(=O)OC)c2)=O)ccccc1C(N1CCCCC1)=O C=CC(C)(O)C(=O)NCCN(C(c1cn(-c2ccccc2)nn1)=O)CC CC(C(C)(C)NC(=O)CCOc1ccccc1)NC(c1cc(C2CC2)cs1)=O c1(CNC(c2cccc(CC)n2)=O)ccc(CNC(=O)C(F)C(C)(C)O)c(F)c1 C#CC(C(C)OC)NC(=O)C(C1CC1)N(C(=O)CCn1cncn1)C c1(CC(=O)N(C(C)C)CCNC(=O)C(O)C(F)(F)F)ccc2ccoc2c1 N1(C(C(C)=C2CC2)=O)CCC2(CC1)CC2CNC(=O)CCc1cccnc1F c1(OCC)ccccc1C1(NC2CCCC(F)C2)CC1 Cc1nnc(NC2CCN(C(C3CNC(=O)CC3(C)C)=O)C2)c(C#N)c1C O=C(CC1OCCc2ccsc21)NCC1CC2CCC1N2C(C1(F)CC=CC1)=O C1(C)(CCN(C)C(c2ccn(CCn3cccn3)n2)=O)CN(CC2CCCO2)C1 C=CCN=C(NCC(C)C(F)(F)F)NC1CC(OC(=O)N(C)C)C1 N1(C(=O)CCc2cnc(O)[nH]2)CC2(C1)CN(C(c1ccncc1C(F)(F)F)=O)C2 c1(NC(C2N(C(C3CC(C)(C)C3)=O)CC3(CC3)C2)=O)cccnc1[N+](=O)[O-] C1(OC)CN(C(=O)NC2CC(F)(F)C2C)CCC1(CO)OC c1(OC)cc(C)c(C(=O)N(CCNC(=O)C(C)(C)CC2CC2)C2CC2)c(C)c1 CCC(CC)C(C(=O)N(CCCCCNC(c1cc([N+](=O)[O-])ccn1)=O)C)OC C12(CNC(C3(CCCC)CC3)=O)CCC(CN1C(c1cc(C)ccc1F)=O)C2 C12(C(=O)NC(CNC(CCC(=O)OCC)=O)CC(C)C)CC1COC2(C)C Cc1ccc2ncc(C(=O)NCC(F)CNC(C3CCCN(C)C3)=O)n2c1 Cc1cncc(C(=O)NC(CNC(=O)Cc2ccc(C(N)=O)cc2)C(C)C)c1C C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(CNC(n2ncc(C)c2)=O)(C)C)C1 c1(C(=O)NC2CCN(C(C3(C)CNC(=O)C3)=O)C2)nnc(O)c(Br)c1O Cc1cc(C(N2CCC(F)(C(=O)Nc3cc(F)cnc3O)C2)=O)c[nH]c1=N C1(C(N2CC(C#C)C2)=O)CN(C(C2CCC(C#N)CC2)=O)C(C)(C)C1 Cn1ncc(NC(c2cnon2)=O)c1-c1cn(CCCCC2CCC2)nn1 N1(CC2(C)CCOCC2)CC(=O)N(Cc2csc(Cc3ccccc3)n2)C1=O N(C1CCc2cccnc21)C(C1CN(C(c2ccc(C)nc2C)=O)CC(F)C1)=O C(C(C)(O)C(F)F)NC(c1cc(CNC(c2c(C)non2)=O)oc1)=O Cn1c(C2CC2)nc2cc(NC(=O)CNC(c3ccc(Cl)cc3)=O)ccc12 C(CCC(C)C)(C(=O)NC1CCC12CN(C(C13CC(C)(CCO1)C3)=O)C2)NC(C)=O N1(C(CNC(c2cc(OC)ncc2)=O)=O)CC2CN(C(c3ccco3)=O)CCC12 N1(C(C2CCN(C(CC)=O)C2)=O)CCC(F)(CNC(C2CCOC2(C)C)=O)CC1 N1(C(C2CCC(C)CC2)=O)CCN(C(=O)C(c2ccc(Cl)s2)=O)C(CO)C1 Cc1cc(C(N2CCC2CNC(=O)Cc2ccccc2C(N)=O)=O)ncc1CO c1(CC(=O)NCC(O)CNC(=O)Cc2cccs2)cc[nH]n1 c1(C(N2C(CNC(CNC(c3ccco3)=O)=O)CCC2)=O)ccn2cccc2c1 C1(C)(CC)CCN1C(C1(F)CN(C(=O)C(C2CC2)OC)C1)=O CC1(CO)CCN(C(C2CCN2Cc2cc(Br)c[nH]2)=O)CC1O C1(C(N(CCCCN(C(c2cn(CCC)nc2)=O)C)C)=O)C2CCCCCCC12 c1(C(=O)NC(CC)CNC(c2ccc([N+](=O)[O-])s2)=O)cc2cc(F)ccc2o1 CC1(C)CCC(C(=O)NCC2CN(C(c3cc(C#N)c[nH]3)=O)CCO2)C1 C1(NC(c2ncccn2)=O)CCCN(C(c2cc3cccnc3[nH]2)=O)CC1F N1(C(C2N(C)C(=O)NC2)=O)C2CCC1C(CNC(c1ccnc(Cl)c1Cl)=O)C2 C(c1cscn1)=CC(=O)NC1CC(CCNC(C(C)NC(C2CCCC2)=O)=O)C1 O=C(CCC1CCc2ccccc21)NCC1(CNC(C23CC(F)C2C3)=O)CCC1 c1(C(=O)NC(CNC(C(CC(=C)C)C)=O)CC(C)C)cc2ccc(C)cc2[nH]1 c1(CC)ccccc1-n1cc(O)c(C(N2CC3(CCC3)C2)=O)n1 CC1(C#CC(=O)NC2CCC(NC(=O)CCCC(N)=O)CC2)CC1 c1(OC)ccc([N+](=O)[O-])c(N2CCC(CCNC(=O)CCN3CCCCC3)C2)n1 CCCCC(O)CC(=O)NC1CC(CC(N2CCNC(=O)CC2C)=O)C1 N1(C(Cn2nnc(-c3snc(C)c3N)n2)=O)CCC(S(=O)(=O)C(F)F)C1 c1(C(N)=O)cccc(OCCOC)c1.C12CC1CN(CC)CCNC2=O c1(C(=O)NCCCN(C)C(c2nncn2C2CC2)=O)cc(C(c2ccco2)=O)c[nH]1 C(C1=CCN(C(c2c(C(F)(F)F)n[nH]c2C)=O)CC1)NC(C1(C)CC(=C)C1)=O C1(CNC(c2cc(SC)c(C)o2)=O)CC2(CC(NC(c3cnn(C)c3Cl)=O)C2)C1 Cn1ccc2c(C(N3CC(NC(=O)C(O)C4CCC4)CC3(C)C)=O)cnc(O)c12 C1(C(=O)NCC(=O)NC)CCCCC1NC(=O)CC1CCC(C)CO1 C(N=c1[nH]c(=NCCC2(C)CC2(Cl)Cl)[nH]c2c1CCCCCC2)C1(C)CC(C)C1 C1(NC(C(c2ccncc2)C)=O)COCCN(C(=O)CCC(C)N(C)C)C1 C1(NC(C2C(C)CCN2C(C2OC3CCC2C3)=O)=O)CC(F)(F)C1(C)C C(CC(C)C(=O)NC1CN(C(C2(CNC(c3cccs3)=O)CCC2)=O)CC1C)=CC C(=O)(C(C)C(C)S(C)(=O)=O)NC(C1OCCN(C(c2cccc(C)n2)=O)C1)C N1(C(c2c(CC)nc(C)[nH]2)=O)CC2N(C(c3nc(C)ccc3F)=O)CCC2(C)C1 c1(NC(C)=O)ccc(C(N2CC(CNC(c3ccon3)=O)C(C)(C)C2)=O)cc1F Cn1cnc(NC(C2(C)CCN2C(=O)C(N)=O)=O)c1 C1(CC(=O)NC2C(C)CCN(C(C3CCC4CC4C3)=O)C2)Cc2ccccc2N1 C1(C(=O)NCC2CNC(=O)O2)CC2CC1CN(C(=O)C(O)C1CCC1)C2 N1(C(CCC(C)C)=O)CCC(CNC(C2CCCS2(=O)=O)=O)C(O)C1 C1(CC=C)(NC(=O)COCCC(C)C)CN(C(C2CCOC2C(F)(F)F)=O)C1 Cc1nc2cc(CN3CCC4CN(C(c5cncc(F)c5)=O)CCC34)ccc2o1 c1(C(=O)NC2CCN(C(C3C(C)(C)CO3)=O)C2C2CC2)cnc2cc[nH]c2c1 CCCCC(=O)NCC(C)C(=O)NCC1(C)CC1(C)C N1(C(c2c(OC)scc2)=O)CCC2(CC1)CC2NC(C1(C)CC1C)=O N1(C(CC(CC)(F)F)=O)CCN(C(=O)C(C)c2ccsc2)CC2CCCCC12 c1(C(=O)NCC(CCCC)NC(C2(C(C)C)CCCO2)=O)ccc(C)c(O)n1 O(NC(=O)C(F)C1(CNC(C2(C3CC3(C)C)CC2)=O)CC1)C(CC)C n1(CC)ncc(C(=O)NCC2CCN2C(C2(C)CC(C)C2)=O)n1 C1(C(=O)NCCC2CCN(C(CCC=C)=O)CC2(F)F)CCn2c(C)nnc2C1 CC#CCC(C(=O)OCC)c1nccn1C.C12(CCOCC1)C(F)(F)C(=O)O2 N1(C(C(=O)N(C)C)=O)CCC2CCN(C(C3CCc4nc(C)cn4C3)=O)CC2C1 N#CC12CC(C(N3CC(NC(C4CC(n5cnnc5)C4)=O)C(O)C3)=O)(C1)C2 CS(=O)(=O)c1ccc(CC(N2CCC(N(S(=O)(=O)CCBr)CCO)C2)=O)cc1 c1(C(=O)NC2CCCCN(C(c3cc(F)c[nH]3)=O)C2)ccn2ccccc12 c1(OCCN(C(C(c2ccnn2C)NC(C(C)NC(N)=O)=O)=O)C)cnn(C)c1 c1(OCC(=O)NCC(C)N(C)C(C2CCCN2C=O)=O)ccc(S(N)(=O)=O)cc1 c1(OCC)ccc(NC(C2C(C(C)C)C2c2csc(Br)c2)=O)c(C)c1 Cc1ccc(O)cc1NC(c1cncc(-c2cn(C)nc2C)n1)=O c1(CNC(c2cc(C)sc2)=O)cccnc1CNC(C1COCCN1C)=O c1(C(C)C(=O)NC23CC(CNC(c4nn[nH]c4Cl)=O)(C2)C3)ccccc1F N1(C2CCN(C(C3C(C)C3)=O)C2)CCC(NC(=O)COc2cnn(C)c2)CC1 CCC(CNC(C1(NC(c2c[nH]c(=N)o2)=O)CC(O)C1)=O)CC(C)C c1(NC(CC(C)F)=O)cc2sccc2s1.C12CCC(F)(C1)CNC2=O N1(Cc2ccn(CC(C)C)n2)CCOC(C)(CNC(=O)C(c2cnn(C)c2)C)C1 CCCC(C(=O)NCC1(F)CC(NC(=O)CC(C)OC)C1)OCC C(=O)(C(CC(C)C)OC)NC1(CC(NOCC)=O)CC1.C1(=O)CCCN1 C(C1=CCN(C(c2ccns2)=O)CC1)NC(Cc1cn(C(C)(C)C)nc1)=O CCC(C)C(C(=O)NCC1(CCOC)CC1)NC(=O)C(C)C(F)F C(C(C(=O)NCC)NC(=O)C(CC)OC)OCC.CC(O)CN(C)C O=C(CCCCCNC(=O)C(F)C1CCOC1)NCc1cncc(Cl)c1 c1(CC)cc(Cl)ccc1C(=O)NC1CCC(NC(c2cnc(C)n2C(F)F)=O)C1 Cc1noc(N)c1C(=O)NCC1CCCC1NC(=O)Cc1ccnc(O)c1 C1(CC)(NC(=O)CC(C)N(C(=O)C(C)(O)C2CCC2)C)CCCC1 N1(C(C(C(C)C)O)=O)CCCC(O)(CN(C)C(c2cn3ccnc3s2)=O)C1 c1(C(C)C(=O)N(C2CC(NC(c3cnns3)=O)C2)C)cccc(O)c1 CC(C)(C(=O)NC(c1ccccc1)CNC(c1ccc(C(F)F)s1)=O)C(F)(F)F Cc1nc(O)[nH]c1C(=O)N(CCCOCCN(C)C(c1oc(CO)nc1C)=O)C N1(C(CC2CCC(C)CO2)=O)CCN(C(C2CCSC2)=O)C(CCO)C1 CC(C)(C)CC(CO)NC(=O)CCN(C(C1CC=CC(O)C1)=O)CC1CC1 Cc1cc(CCC(=O)NCC2CCN(Cc3ccsc3)C2)no1 c1(C(=O)NCC2C(C)(C)C(NC(C3CS(=O)(=O)C3)=O)C2)cn2cccnc2n1 C1(CC)CCN(C(c2nnc(S)n2C)=O)C1C(=O)NCCCC(N)=O c1(C(=O)NC(c2c(OCCC)cccc2)C)cc(Br)cnc1O C(c1ncccc1C)=CC(=O)NC(CNC(C1N(C(C)=O)CCCC1)=O)C(C)C C1(CNC(C23CC(C(C)C)(C2)C3)=O)CN(C(c2ncc(Cl)cc2Cl)=O)CCN1C C1(C)(CNC(C2(CCC)CC2)=O)CCCN1C(c1sc(C)nc1C)=O CC(C)(F)CCC(=O)N1CCC(CNC(c2ncnc(O)c2Br)=O)C12CC2 CCC(CC)C(F)C(=O)NCCCCCC(=O)NCC1C(C)(C)C1(C)C c1(C(=O)NC2(CNC(=O)C=CCn3cncn3)CCC2)cc2c(Cl)nccc2s1 Cc1sc(S(N)(=O)=O)cc1C(=O)NCC(C(C)C)NC(c1ncncc1F)=O N1(C(CC(CCC)CC)=O)CCC2(CCC2)C(NC(=O)C(COC)OC)C1 c1(C(=O)NC2C(NC(c3ccc(C)o3)=O)CC2)cccc(C2CC2)c1Cl C1(C(N2CC3(C(NC(CCCC(=C)C)=O)CCS3)C2)=O)CCC(C2CCCO2)O1 Cc1nc(C)n(CCNC(c2cc(CNC(C3CC(C4CC4)C3)=O)nn2C)=O)n1 C1(C(=O)NC2CCCC(NC(c3csc(CO)n3)=O)C2)CCn2ccnc2C1 c1(C(=O)NCC(=C)CCNC(C2CC2F)=O)cnc2n1CCOC2 C1(CCOC)CN(C(c2ccnn2C(C)CC)=O)CCN1C(=O)Cc1cnns1 C1(NC(CC2(OC)CCC2)=O)CCN(C(=O)CCOC(C)C)CC12CC2 c1(C(=O)NCCCCNC(c2c(CC)[nH]c(=N)s2)=O)c(Br)ccc2c1OCO2 C1(C(=O)NCC2C(CC(C)(C)C)C2)CCCC(NC(=O)CCc2cnoc2)CC1 C1(CNC(CCCCSC)=O)CC(C)(C)CN1C(=O)Cc1sccc1Cl C(=O)(C(C1=CCCSC1)N1CCCC1CF)NC(C)C c1(NC(=O)NC2C(CNC(c3n[nH]c4c3CCC4)=O)C2)ccc2ccccc2c1 c1(C(=O)NCC(C)N(C(c2c[nH]c(=NCC)s2)=O)C)cccc(S(N)(=O)=O)c1 Cc1ccc(C(C)C)c(C(N2CCCC(NC(c3ccsc3C#N)=O)C2)=O)c1 Cc1cc(F)cnc1C(N1CC(F)CC1CN(C(=O)CC1=CCCC1)C)=O Cc1ccc(O)nc1CNC(=O)C(C1CCCO1)NC(c1ncn(C)n1)=O c1(C(=O)NCCCN(C(=O)C(O)CC(F)F)C)cc(Cl)c(N)cc1F N1(C(C=Cc2c(C)nccc2)=O)CCCC2C1CCCN2C(c1cn[nH]c1)=O Cc1c(Cl)ccc(C(N2CCC(F)(CNC(=O)CC(O)CN(C)C)C2)=O)c1O CC1CC(NC(=O)CC23CCC(CC2)C3)CN(C(c2cn(CCO)nn2)=O)C1 c1(N2CCC(CCCCNC(COC)=O)CC2)nc(Cl)nc2nc(Cl)n(C)c12 Cc1c(C(=O)NC2CC2CNC(=O)C(F)(F)CC2CC2)cccc1O CC1(CCC(=O)NC2C3CC2N(C(=O)CN2CC4CC4C2)C3)CCC(=O)N1 c1(C(N2C3C(N(C(C=CC)=O)C)CC(C3)C2)=O)cc(OC)c(OC)cc1[N+](=O)[O-] N1(C(c2sc(Cl)cc2Cl)C(=O)NCCCOC)CC(N(C)C)C(C)(C)C1 c1(C(=O)NCC2(NC(c3cc(N)c(Cl)cc3)=O)CC2)cc2nn[nH]c2cc1F c1(C(=O)OC(C)(C)C)c(C#N)cnc2c(Cl)cccc12.CC1(C)CCCOC1 n1(CC(=O)NCC2C=CCN2C(=O)C(C2CCCCC2)O)cnc(C(F)(F)F)c1 CC1CC(c2cn(CCO)nn2)CN1c1ccc(C(=O)NS(C)(=O)=O)cc1 C1(N(C(=O)CCCOC)CC)CCCC(NC(=O)CSCCN(C)C)C1 S(=O)(=O)(c1ccc(CC(=O)NCC(C)NC(=O)CNC(=O)CN(C)C)s1)NC C12(C(N3CC(CF)C3)=O)CCCC1N(C(=O)C(COCC)OC)CC2 CCCC(C(=O)NCC1C(CC)CCN1C(c1cc(F)c[nH]1)=O)N(C)C C1(NC(CCNC(COC)=O)=O)CN(C(c2csc(=N)[nH]2)=O)CC12CCOCC2 c1(N2CC(O)(C(C)NC(c3cc(CCC(=O)N(C)C)on3)=O)C2)snc(Cl)c1C#N n1(CCC(=O)NC(CNC(C2(CC=C)COC2)=O)(C)C2CC2)ccc(O)nc1=O C(CCC)(C(=O)NCC1CCC1NC(=O)C(c1ccc(F)cc1)CC)=CCC C1(C(N2CC(C=C)C(NC(c3cccn3C3CC3)=O)C2)=O)CCCC(C)(C)CC1 N1(C(C2(c3ccc(OC)cc3)CC2)=O)CCC(O)(CN(C(=O)CCC#N)C)CC1 c1(C(=O)NCC2N(C(c3cc(C)ns3)=O)CCN(C)C2)cccc(C#CCO)c1 C1(NC(C(=Cc2cccs2)C)=O)CC(F)CN(C(=O)Cn2cnnc2O)C1 CCCCCCCCC(=O)N1CCC(C)CC1C(=O)N(C1CC(C)(C)C1)C c1(CC)nn(C)cc1S(=O)(=O)NC1(CO)CC(OC)C1.c1(O)ccccc1 c1(C(N2CC=C(C#N)CC2)C(=O)Nc2ccc(OC)cc2)cc(F)cc(Br)c1 c1(C(=O)NCCC2OCCN(C(C(CCC)OC)=O)C2)c(F)cc(C#N)cc1F C(=O)(CC(O)C(Cl)(Cl)Cl)N(CC(C)CNC(c1cnn(C)c1C(F)F)=O)C NS(=O)(=O)c1cccc(C(=O)NC2CN(C(=O)C(F)=CCCF)CC2O)c1 C(=O)(CC(C=C)CCC)N1CCC(C(CO)NC(C2C(CC#C)OCC2)=O)CC1 C1(C(N(C(CNC(c2cnc(C(C)O)s2)=O)C)C)=O)CCNC(=O)C1 N1(C(C(CCC)(C)CC)=O)CC2CCC(NC(=O)C(CC)N(C)C)CC2C1 C(=O)(CC1CCc2ccccc21)N(CCNC(c1ccc(F)c(C)c1N)=O)CC N1(C(C2(O)CCCN(C(C)=O)C2)=O)CC2CN(C(=O)C3=NOC(C)(C)C3)CC2C1 c1(C(=O)NC(CCNC(C2(COC)CC2)=O)(C)C)cn2cccc(F)c2n1 CC1(C)OCCC1C(=O)NC1CC(NC(c2cc(C#N)c[nH]2)=O)C(O)C1 CC1(C)CCCOC1C(N1CCCCCC1C(=O)NC(CCO)C(C)(C)O)=O C1(CC(=O)N(CC(CC)(C)OC)C)CCCCN1C(=O)CCn1ccnc1 c1(C(=O)NC(CC)(CNC(c2c(O)noc2C)=O)CC)cc2nc(Cl)ccc2s1 N1(C(c2cncc(NCC)c2)=O)CC(O)C(O)C1CNC(c1ccnnc1)=O S(=O)(=O)(CC(=O)NC(C)C(C(C)C)NCc1cc(CC)[nH]n1)NCC c1(CC)cnc(C(N2CCC(C)C2C(=O)N(C)Cc2nc[nH]n2)=O)nc1 N1(C(C(C)SCC)=O)CC2(C(=O)NCCCc3nc(C)no3)CC1CO2 c1(C(N2C(C)CC(NC(C3CC(SC)C3)=O)C2)=O)cc(Cl)cc(F)c1N CCCCC(C(=O)NCC1CC(NC(C2(CF)CC2)=O)C1)NC(N)=O c1(C(=O)NCCN(CCC)C(C)=O)ccc(OC(C)CC)c(Cl)c1 c1(C(N(CC(C)NC(=O)C(COC)OC)CC)=O)ncc(Br)cc1N C1(C(C(N2CC(=CCC)C2)=O)NC(=O)CSc2cn[nH]c2)CC=CCC1 N1(C(C(CC)F)=O)CCN(C(=O)C(C)N(C)C)CC1CCO c1(C(N2CC(C)CC(NC(c3ccc(CC)s3)=O)C2)=O)cccc2[nH]ncc12 C=CCC(C(=O)NC(C)(C)C)NC(=O)NC1CCCN(CC(=O)OC)C1 C12(CNC(c3nc(C4CC4)cs3)=O)CCC(CC3CC3)(CC1)CO2.O=C1CSN1 c1(OC)ncnc(N2CCC(C(C)NC(=O)C(C)Cc3ccco3)CC2)c1OC Cc1c(C(=O)NC2CC2NC(C2(O)CCCCC2)=O)oc2ccc(Cl)cc12 c1(C(=O)NCC2C(NC(c3c(C)cn(C)n3)=O)C2)cc(F)cc2cccnc12 c1(OCC)cccc(CC(=O)NCC(O)CNC(=O)CCn2ccnc2)n1 CC1CN(c2ccnc(NCC(c3ccc(O)cc3)(C)C)n2)CC1N(C)C C1(N(C(=O)CC2CCCOCC2)C)CCCN(C(=O)CCCc2cnn[nH]2)CC1 Cc1ccn2c(C(=O)NC3CCCC3CNC(c3nc(O)sc3C)=O)cnc2c1 c1(C(N2C3CN(C(c4n(C)cc(Br)n4)=O)CC32)=O)ccc2[nH][nH]c(=N)c2c1 Cc1cc(NC(c2cscn2)=O)ccc1NC(=O)C(C)N(C)C C(=O)(C(CC(C)C)Nn1c(C2CCCC(Cc3ccc(F)cc3)O2)ncc1)OCC C(c1ccc(Cl)s1)=CC(=O)NCCOCCNC(C1CCC2CCC12)=O N1(C(C(C2CN(C(CC(C)(C)C3CC3)=O)C2)O)=O)CC2CCC(C1)C(=O)N2 C1(NC(=O)NC(CN(C)C)CO)CC(=O)N(C(C)(C)C)C1=O C1(NC(CCOCC)=O)C2CCCC1CC(NC(c1cnn(CCF)c1)=O)C2 c1(OC)ccc(C)cc1C=CC(=O)NC(CCN(C)C(C1(C)CC1)=O)C(C)(C)C c1(CC(=O)NC(CC)COC)ccc(OCc2ccccc2)c([N+](=O)[O-])c1 C(=O)(C(CC#CC)NC(c1cc(C)c[nH]1)=O)NCC1(CCC=C)CC1 C(=O)(C(C(C)C)NC(C1(CNC2(CC3CCC3)CC2)CC1)=O)OCC C1(NC(c2nccc(C)c2)=O)CC2CN(C(=O)C(C)C3CCOC3)CC12 C(=O)(N=c1[nH][nH]c(C)c1Cl)c1nc(-c2c(OCOC)ccc(F)c2)c(F)cc1 c1ccc(C(C)(C)C)cc1.C1(C(=O)NCCOCCCNC=O)CCCN1N=O C(CCCCCCC1(OC)N=N1)n1cc(CSC)nn1 c1(C2C(O)CCC2)ccccc1-c1cccc(C2CN(C3CC3)CCO2)c1 N1(C(C=CC)=O)CCC2(CCCCN(C(=O)COCC3CCCCO3)C2)C1 C1(NC(CCC2N(C(C(CC(C)C)O)=O)CCC2)=O)CN(C)C(=O)C12CC2 C1(c2non2C2CN(c3nnnn3C)C2)CN(CC2(C3(C)CC3(C)C)CC2)CCCO1 CC1C(=O)N(CC(N2CC(CCCCNC(c3cccnn3)=O)C2)=O)C(=O)C1C C12(C(CNC(=O)C(N)=O)NC(c3ccn(C4CCC4)n3)=O)CCC(CC1)C2 Cc1cccc2[nH]c(C(=O)NC3CC3CNC(=O)C=Cc3cccnc3)cc12 C(CNC(=O)C(C(C)C)OC)(C(C)(C)C)NC(c1c(COC)cc[nH]1)=O C1(C(=O)NC2(C)CCCN(C(C(C(COC)C)C)=O)C2)CCC2(C1)CC2(F)F CCCCC(C)C(=O)NCC1OCCC1C(=O)NCc1nn(CC)nc1C N1(C(c2c(CC)nns2)=O)CCCC(C)C1CNC(C1CC(n2ccnn2)C1)=O C(=O)(C(C)(C)C1=CCN(C(=O)Cc2c[nH]nc2C)C1)NC(CCN(CC)CC)C C(CCCC(C)NC(c1ccc(-n2cnnn2)cc1)=O)NC(c1c(C)nn[nH]1)=O c1(NCc2ccc(C(=O)OCC)cc2)cc(N(CC(C)C)C)nc(CCOC)n1 C1(C(=O)NC(C2CN(Cc3noc4c3CCCC4)C2)C)CCC(C2CCCO2)O1 c1(CNC2CC(C(=O)NC3CC3(F)F)C2)cc(Cl)cc(Cl)c1O c1(C(=O)NC(c2cn(C3CCOC3)nn2)C)ccc2c(=O)ccoc2c1 c1(C(N2CCN(C(c3c(C)n(C)cn3)=O)CC2CCO)=O)ccn2ccnc2c1 N1(C(c2cc(C#N)[nH]c2)=O)CCCC(NC(C2(O)CCCCCC2)=O)CC1 c1(N(CCNC(c2oc(C)nc2C)=O)CC)ccc(C#N)c([N+](=O)[O-])c1 C1(C(=O)NCCN(C(=O)C(CNS(C)(=O)=O)N(C)C)C)CCCC(C(F)(F)F)O1 N1(C(C(C)CC(F)F)=O)CC2(CC(C(=O)NCC3(CO)CCC3)CO2)C1 C1(C(=O)NC2(C)CC(NC(C=Cc3ccc(C)cn3)=O)C2)Cc2ccccc2C1 C1(CN(C(C(CC)N(C)C)=O)C)CCCCN1C(=O)CN(C)C(=O)OC(C)(C)C c1(C(=O)NCC(CC)NC(C(CCCC)CC)=O)c[nH]c2ncc(Br)cc12 N1(C(C(CC)C)=O)CCC(C)CC1CNC(=O)C=CC(C)(C)C C1(NC(C2CCCCS2)=O)CN(C(=O)C=C2CN3CCC2CC3)CC1C1CC1 CCC(CC(=O)NC1CC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C1)C1CC1 n1(CCC)nc(C)cc1C(N1CCCC1CN(C)C(C1CCCC1OC)=O)=O c1(C(C(=O)NCC)N(CCOC)CC2CC2)nc(Cl)cs1 c1(NC(C2CCCN(C(c3cnc(C)s3)=O)CC2)=O)ccc(Cl)c(C#N)c1Cl C#CC1(C(N2CCCC2CNC(=O)C=Cc2nc(C)co2)=O)CCCC1 C1(C(=O)NCCOC2CN(C(=O)C(F)=CC3CC3)C2)CCCN1c1ncccn1 c1(C(=O)NCC2(F)CN(C(C3C4CCC34)=O)C2)cccc(C(F)(F)F)n1 c1(NC(C(c2ccccn2)C)=O)ccc2c(c1)OCC(=O)N2 C=CCC(CC(=O)NCC1CCCCS1)NC(C12CC(C)(CCO1)C2)=O N1(C(c2n(C)nnc2)=O)CCC2(CCOCC2C(N2CC(F)C2)=O)CC1 C1(CCCNC(C2(C(C)C)CC2)=O)CCCN1C(=O)C(C)Cn1ccnc1 Cc1ccc(CC(N2CCCC2CNC(C2CC23CCC3)=O)=O)cc1[N+](=O)[O-] c1(C(CC)NC(c2n(CCC)nnn2)(C)Cc2cnccn2)ccc(Br)cc1 c1(OCC)ccc(C(=O)N(CCC(C)NC(=O)C=CC2CCCC2)C)cc1Cl C(=O)(CC(CC)C(C)(C)C)N1CCC(C#C)(C(=O)NCC2C3CCCC23)CC1 C1(C(=O)NC2CCCN(C(C(C)c3ccco3)=O)C2)CCn2cnnc2C1 N1(C(C2C(C)C2C)=O)CC(NC(c2cn(CC3CC3)nn2)=O)CC1(C)C C1(NC(C2(OC(C)=O)CC2)=O)CCOCC1C(=O)N(C1(CCO)CC1)C N1(C(CC)=O)CCc2ccc(S(=O)(=O)N3CC(Oc4ccc(O)cc4)C3)cc21 C(=O)(C(N=[N+]=[N-])C(C)C)N(C1(C(=O)NC(C(=O)NC)C)CC1)C c1(OC)cc(CCC(=O)N(CCCNC(=O)CC2CC2C)C2CC2)ccc1Cl C(CNC(c1cc(C2CCC2)nn1C)=O)(C(C)C(C)C)NC(CSC)=O C(c1cn(C(C)(C)CC(=O)N(C(C)Cc2ccccc2)C)nn1)=CC(C)C c1(CC2CCN(CC=C(C)C)CC2)cc(F)c(C)c([N+](=O)[O-])c1 C1(N(C(c2ccc(CC)[nH]2)=O)C)CN(C(=O)Cc2ccnc(OC)c2)CC12CC2 Cc1cccc2oc(C(=O)NC(C3CCN(C(C4(C)CNC(=O)C4)=O)C3)C)cc12 N1(C(C2CCCN(C)C2)=O)CCCCC(NC(c2cc(Cl)ccc2F)=O)CC1 c1(Cc2cc(NC(C)C)ns2)cccc2cccnc12.C12(CCCO1)CC(=O)N2 c1(C(N2CCC(C(C)NC(C3(CCC=C)CC3)=O)C2)=O)cc(C)c(OC)c(C)c1 N1(C(CCN2CCC(C(=O)OC(C)(C)C)CC2)=O)CCn2cc(CO)nc2C1 C1(CC(=O)NCCC(COC)(C)O)CN(C(c2c(CO)n[nH]c2C)=O)CC12CC2 N1(C(c2c(C)ncs2)=O)CCCC(F)(CNC(=O)C(c2ccccc2)F)C1 C1(CC(N2CCC(N(C)CC)C2)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1C c1(NC(c2c(C(=O)OCC)cccc2F)=O)ccc2c(c1)C(=O)OC2(C)C N1(C(c2c(N)cncn2)=O)CC2CC(C1)N2C(=O)C1=CCOCC1 c1(C(=O)NC2C(O)CCN(C(C3CC(C)C3)=O)C2)cc2c(F)cc(F)cc2[nH]1 C(=O)(C1=CC2CCCC12)NCCCCCCNC(Cc1c(OC)nccc1)=O CN1CCC(C)(C(=O)NCC(F)CNC(c2ccc(CC3CCC3)cc2)=O)CC1 C1(NC(c2nc(C)nc(O)c2)=O)CC2CC(NC(C3CC4(CCC4)C3)=O)C2CC1 C1(O)(C(CN(C(=O)C2=CCC2)C)(C)C)CCN(C(=O)C(=O)Nc2ccccc2)C1 C1(C(=O)NCC(N(C(c2cccc(C)n2)=O)C)C2CC2)CC2(CCCCC2)C1 CS(=O)CCC(O)C(=O)NCCCOCCCNC(=O)CN1CCOC1=O c1(C(=O)NC2(CNC(c3ccc(CCO)cc3)=O)COC2)cc(F)c(Cl)nc1Cl C(=O)(CCCC(=O)NC1CC(CNC(=O)COc2cnn(C)c2)C1(C)C)NC CCC(C(=O)NCC(C(C)C)NC(=O)Cc1nc[nH]n1)C1CCOCC1 C1(C)(C(=O)NCC2(C)CCN(C(=O)CCCCC3CC3)C2)CC(C2CC2)=NO1 c1(CNC2CCC(C(=O)Nc3ccc(CC)cc3O)C2)c(O)ccc(F)c1F c1(N2CC(NC(CCCCSC)=O)C(C)(C)C2)nc(C)nc2scc(C)c12 C12(CNC(C)=O)CCC(CNC(=O)C=Cc3cncnc3O)(CC1)OC2 c1(C(N2CCC(NC(c3c(C)cnnc3)=O)C2)=O)csc2c1CCC(C)C2 c1(C(=O)NC2CCCN(C(c3n(C(C)C)ncc3)=O)C2)cnc(O)c(Br)c1 CC1(C)CC(C(N2CCC3CC23)=O)CCN1C(c1ccncc1O)=O c1(CC(=O)NCC(CC)NC(=O)C(O)CSC)cc2nc[nH]c2cc1Br C1(C(=O)OC)CN(C(=O)C=Cc2cscn2)CC(C(F)(F)F)O1 N1(C(C=C(C)C(F)F)=O)CCC(NC(=O)CSc2ccc(O)cc2)C(C)(C)C1 c1(C(=O)NC(CNC(C2C(=C)C2)=O)CCCC)cc(OC)cc(F)c1 c1(C(=O)NC(C(=O)NC(c2nnc(O)o2)C)(C)C2CCC2)ncc(F)cn1 c1(C(=O)NCCCC(C)NC(CCC#C)=O)ccc2c(n1)NCC2 Cc1cc(F)c(C(N2CC3CC2CCN3C(=O)C=CC2CCCCC2)=O)c(F)c1 C(=O)(N=c1cc(OC)n(C)[nH]1)C1C(CC)CN(C(C2CC2CCOC)=O)C1 C1(NC(c2onc(C)c2C)=O)C2CCC1N(C(=O)C(c1cnn(C)c1)C)C2 N1(C(c2c(OC)cc(N)cc2)=O)CC(F)(F)CC1(C)CNC(C1CNC(=O)C1)=O c1(CCC(=O)NCC(C)NC(C2CCc3ccnn3C2)=O)ccc(F)c(F)c1F N1(C(C(C)C#N)=O)CCC(F)(F)C(NC(=O)COc2cccc(F)n2)C1 C#Cc1ccc(C(N2CC(NC(C3CCSC3)=O)C(Cc3ccccc3)C2)=O)cc1 CC1CN(C(c2ccccc2Br)=O)CCN1C(C1CCC(CN(C)C)CC1)=O S(=O)(=O)(c1cc(C(=O)N(C(C)CNC(c2ccc(SC)o2)=O)C)co1)NC c1(C2(C(=O)NCC(CO)NC(=O)CC3(O)CCC3)CC2)ncco1 CC1CCN(C(=O)Cn2cnc(=N)[nH]2)CC1C(=O)N(c1cccc(Cl)c1)C C(=O)(C(Cc1ccccc1C)CC)NC(C(C)NC(C1(COC)CC1)=O)C c1(NC(CC2CCCN(C(CCOC)=O)C2)=O)c(Cl)cccc1[N+](=O)[O-] C=CC(C)(C)CC(=O)NCCCCn1cc(CO)nn1.N12CC(CC1=O)C2 c1(C(N2C(C(C)NC(CC3(C=C)CC3)=O)CCC2)=O)cnc(N(C)C)c(Cl)c1 c1(CCOC(c2c(C(=O)OC)ccs2)=O)c(OC)ccc2ccccc12 N1(C(C(C=C)OC)=O)CCCC(CCNC(c2occc2C(C)=O)=O)C1 CC1(C)CN(C(C2CCC(=O)NC2)=O)CC1CNC(=O)COCC1CCC1 N1(C(C(C=C)(C)O)=O)CCCOC(CNC(c2ccc(Br)c(O)n2)=O)C1 N1(C(c2c(COC)noc2)=O)CCC(CNC(=O)CC2CCC(C)(C)O2)C12CC2 N1(C(C(C)NC(CC)=O)=O)CCCC2(CC(NC(=O)CCC3CCOC3)C2)C1 N1(C(c2cc(CC)on2)=O)C2CCC1CC(NC(=O)C(=Cc1cccn1C)F)C2 c1(CNC(C2(CCC)CC2)=O)cccc(C(=O)NCCc2cncn2C)n1 CCC#CC(C)(C)NC(c1cnc(CNC(=O)C(O)CSC)nc1)=O CC1(C)C2CCC1(C(=O)NC1CN(C(c3conc3C3CCC3)=O)CC1F)C2 N1(C(=O)OC)CC2(CCN(C(C3CC3C(C)(F)F)=O)CC2)c2cc(F)c(Br)cc21 c1(CCCSCC)nc(-c2cc(C)sc2C)n(C2CCOC2)n1 c1(OC)ccccc1C(=O)NC1COCCC1NC(c1cccc(CSC)c1)=O CC1(C)CC(c2cn(-c3c(F)cccc3F)nn2)CN(C(=O)C(O)C(F)F)C1 C1(CNC(C(C)O)=O)CC(O)(CNC(=O)CCN2CCOCC2)C1 CC1CCN(C(=O)Cc2ccsn2)C(C(=O)NC2(C3CCCCO3)CC2)C1 C1(CNC(CSCC#C)=O)CC2(CC2)CN1C(c1ccc(Cl)c(C(F)(F)F)c1)=O C1(NC(CN(CC#C)C(C2C3(CC3)C23CC3)=O)=O)(CO)CCC(C)(C)C1 C(=O)(CC(C)(C)OC)N1CCC(CCC(=O)N(C(CC)C)C)C1 C(=O)(CCCCCNC(C1CCCC(=O)C1)=O)NC(CC#C)C(N)=O c1(CN(C(CC2(OC)CC2)=O)Cc2ccccc2)ccccc1C c1(C(N2CCC(NC(C(C#C)(C)C)=O)C2C)=O)nn(C)c2c(=O)[nH]cnc12 N1(CCNCCCN(S(CC)(=O)=O)C)CCN(c2ccnc(CO)n2)CC1 Cc1cc(C(C)C(=O)NCC2CCN(C(c3ncncc3F)=O)C2)cc(F)c1 N1(C(C2CC(NC(CCCN(C(C)C)C)=O)C2)=O)CCCC2(CC(O)C2)C1 C1(C(N2CC(CCC#C)C2)=O)CCN(C(=O)C(C)(C)O)CCO1 C(=O)(C1=CC2C=CC1C2)N1CCCCC(N(C(C(CCCC)C)=O)C)C1 N1(C(C2N(C)CCC2)=O)CC2CC1CN2C(=O)C(c1cccnc1)O CCCCCC(O)CC(=O)NC(CO)CCCNC(=O)C=C(CC)CC N1(C(C(C=C)O)=O)CCCCC2(C1)CN(C(c1cnc(C3OCCO3)s1)=O)C2 Cc1oc(C2CC2)nc1CNC(=O)C(N1CCCC(c2cccs2)C1)=O c1(CC)c(C(=O)NCC2(C)CCN(C(=O)CC3CC4(CC4)CO3)C2)nnn1CC C1(NC(c2ncc(C)nc2)=O)CN(C(=O)CCc2nccs2)CCC1C C(=O)(C1CNC(=O)c2ccnn21)NCCN(C(=O)C(F)C1=CCCCC1)CCC N12CCC(C1)C(=O)C1CN(C1)C(=O)C2=O.N12CCC1CC2.C(=O)(CC1CCC1)OC C(=O)(C1=CCC2(COC2)OC1)NCC(CC)NC(=O)C(C)NS(=O)(=O)CC C1(C)(C(=O)NCC(C)(C)CNC(=O)C(CO)NC(c2ccco2)=O)CC2CC2C1 C1(CNC(c2cn(C)nc2C2CC2)=O)CC2CCC1N(C(=O)CC1OCCO1)C2 C1(NC(CN(C(COC)=O)C)=O)CCN(C(=O)CSCC(N)=O)C12CC2 CC1(C)CCN(C(C2CC3(CCC3=O)C2)=O)C1C(=O)NCc1ccco1 C(C1=NOC2CN(C(c3cc(C(=O)OC)sc3C)=O)CC12)NC(CC=CC=C)=O c1(OC)cc(C(=O)NC(C)(C)CCCOc2ccc(F)cc2)c(F)cc1Br C1(=CC(=O)N(C2CCN(C(C3CCC(=O)N3)=O)C2)CCC)CCCCC1(C)C N1(C(C2(n3cc(CCCCCCC)nn3)CC2)=O)CC(CC(=O)O)OCC1(C)C c1(C(N2C(CC)C(NC(=O)COC3(C)CCC3)CC2)=O)ccc(F)c(C(F)F)c1 c1(C(N2CCC(NC(C(COC)OCC)=O)(CF)C2)=O)cn2c(n1)CCC2 C1(C(=O)NCCC(C)N(C(c2ccc(CC)[nH]2)=O)C)CCOC(C)(C)C1 C1(COC)CN(C(c2cccc(Br)c2Cl)=O)CCN1C(c1c(I)ccnc1F)=O C=CCCCCCC(=O)NCC1CCN(C(=O)C(c2ccccc2Br)O)C1 N1(C(COCCCC)=O)CCCC(C)C1CCNC(=O)CC(F)(F)F C1(CC)CC(CC(=O)OC(c2ccc(Br)cc2)C(C)(F)F)CCO1 Cc1cc(NCC2C3CN(C(C4(O)CCC(C)CC4)=O)CC23)ncc1[N+](=O)[O-] C12(OC)CCCCC(C(N3CCC(NC(=O)Cn4cnnn4)C(F)C3)=O)(C1)C2 C1(C(=O)NC2(COC)CN(C(=O)CC(C)C(C)C)C2)CCc2nnnn2C1 C1(CC(=O)NCCCNC(c2ccc(C(F)(F)F)c(Cl)c2)=O)CCCC(F)(F)C1 N1(C(c2c(C(C)C)nns2)=O)C2CCC1CC(NC(c1cnn(CCF)c1)=O)C2 C=CCCCC(=O)NCc1ccc(CNC(=O)CCc2ccc(OC)cc2)o1 C12(CC)CN(C(c3cnccc3C)=O)C(CNC(=O)C(F)C3CCOC3)(C1)C2 Cc1nc2cc(C(N3CCC(CO)(NC(=O)C(F)=C4CCC4)CC3)=O)[nH]c2s1 c1(C(=O)OCc2cccnc2)cc(S(=O)(=O)N2CC(N3CCNC3=O)C2)c[nH]1 C1(CCNC(C(C)N(C(=O)Cc2ccsn2)CCC)=O)CC(=O)N(C)C1 O=C(C1=CS(=O)(=O)CCC1)N1CCN(C(C2CC=CC2)=O)C(c2ccncc2)C1 Cc1ccnc2sc(C(=O)NCC(C)NC(=O)C(F)(F)C(O)C(C)C)c(C)c12 Cc1cc(N)ccc1C(N1CCCC1C1CCCN(C(=O)Cc2cnoc2)C1)=O c1(C(=O)NC(CCNC(C2N(C(C)C)C(=O)CC2)=O)C)nnn2c1CCCCC2 N1(C(C(C=C)OC)=O)CCCC2(CCC2NC(c2cnc(C(C)C)o2)=O)C1 CCCC(F)C(=O)NCCC(CNC(C1CC(C)(CC)C1)=O)OC CCCC(C)(CCC)NC(C)C(c1ccc(F)c(F)c1)O c1(C(=O)NCC(CC)(C)NC(=O)CCc2nc(C)c(C)[nH]2)cc(Cl)cnc1O C1(C(=O)NCc2occ(C(=O)NC3(C(C)(C)C)CCCC3)n2)CCC=CCC1 c12ncc(cc1Br)c(=O)n2C(C)C.C1(COC)CCCN1C(=O)C(C)SC1CC1 c1(OC)cccnc1C(F)(F)C(N1CCC(O)(C(N)=O)C1)=O N1(C(C(C)(C)NCCC)=O)CC2C(C(N3CCC(C(F)(F)F)CC3)=O)C2C1 c1(C(C(=O)Nc2c(C)cccc2C)N(CC=C)C(C)C)cc(C(F)F)cc(C)c1 C(C)(CCCCNC(c1csc(C2CC2)n1)=O)NC(c1n(CC)ccc1)=O C(N=c1[nH]c2c(c(=NCCCC(C)CO)[nH]1)CCC2)c1cnc(CC)s1 c1(OC)ccc(OC)c([N+](=O)[O-])c1C(=O)NC1CC1C(=O)Nc1ccsc1 C(C)(CCC(=O)N1CCCC1C(=O)NC(C)CC(C)C)OC c1(C(=O)NCCC2CC(NC(=O)C=Cc3cnc[nH]3)C2)cc2n(n1)CCNC2=O c1(CC)nc(=NCc2cccc(CNC(C3CC3C3CC3C)=O)c2)s[nH]1 c1(N2CC3C(CNC(C(C(CC)CC)C)=O)C3C2)nccc2c(C)cccc12 C1(CNC(CCc2nc(=N)[nH][nH]2)=O)(NC(=O)CC2CCCC(O)C2)CCCCC1 C(c1ccc(C)cc1)=CCC(=O)NC1C(NC(c2c(CC)noc2)=O)CCCC1 c1(C(N(C2CCC(NC(C3(CC#C)CC3)=O)C2)C)=O)cccc2c1CCCC2 C12(NC(C)=O)CCCCCC1OCC2.c12nn(C)c(Cl)c1CCCN(C)C2=O C1(NC(CC(C)C2CC2)=O)CC2(CCN(C(=O)Cc3ccc(O)nc3)CC2)C1 c1(C(=O)NCC(C)(C)NC(C2C(C(C)C)OCC2)=O)ccnc2ccnn12 C(=O)(CC(=O)NCC1CC1NC(C12COCC1C2)=O)OC(C)(C)C c1(C(N(CC(C)N(C(C2CCC(C)O2)=O)C)C)=O)nn(C)cc1S(N)(=O)=O c1(C(C(N2CC=CC2Cn2cc(CC3(O)CCC3)nn2)=O)OC)ccc(F)cc1 N1(C(c2ccn(COC)n2)=O)CC=CCC1C(N1CCC=C(C)C1)=O C1(C(=O)NC2CCC(NC(C3CC=CCC3)=O)CC2)(COC)CC=CCC1 c1(C(CNC(C=C(C)CNC(=O)CCCn2ccnc2C)=O)=O)cnc(C)[nH]c1=N CC(C)C1=NOC(C(=O)N(C2CN(C(=O)C=CBr)CC2(C)C)C)C1 c1(-n2cc(CC(C)C(=O)O)nn2)cccc(C(=O)NC2(C(C)(F)F)CCOC2)c1 Cc1cccc(C(O)C(N2CC(CNC(=O)Cc3cn(C)cn3)C(O)C2)=O)c1F C1(C(=O)NCCC(C)NC(C(C(CC)C)O)=O)CCc2cc(F)ccc2O1 N1(C(c2sc(C)c(O)n2)=O)CC2CN(C(c3c[nH]nc3C3CC3)=O)CC2(C)C1 C(=O)(CC(O)CN(C)C)NC(CN(C(c1cn(CC=C)nn1)=O)CC)CC OC1(c2cn[nH]c2)CCNCC1.n12nccc1C2 C(CCCCC(=O)NC1CCCC(N(C)C(c2cc[nH]n2)=O)C1)NC(C)=O C(C(C)(C)CC(=O)N(C1CN(C(=O)Cc2ccnn2C(C)C)CC1(C)C)C)OC CC1CCC(=O)N1.C1(C(=O)N(C)C)(CN)CC2(CC2)C1 CC1CN(C(c2cc(C3(C)CC3)n[nH]2)=O)CC(C)C1NC(c1coc(CO)c1)=O C=CC1CCN(C(=O)C(CCSC)NC(C2CCC(=C)CC2)=O)C1 C1(O)(C(C(=O)NC2CC(CC(=O)NCCN(CCO)CC)C2)F)CCCC1 C1(CNC(C(=O)NCC2CN(C(=O)OC(C)(C)C)C2)=O)CC(=O)NC1=O c1(C(N(C(C)CCNC(C2(C(C)(F)F)CC2)=O)C)=O)ccn2nnnc2c1 C(=O)(CC(C(F)(F)F)OC)N1CCN(C(CS(=O)(=O)NC)=O)CC1c1cn[nH]c1 c1(C(=O)O)cccc(S(=O)(=O)N2CC3C(C(=O)N(C4CC4)Cc4cccnc4)C3C2)c1 C12(C)CN(C(C)(C)C1)C2=O.C(CCC(=O)NNC(=O)OC)OCC.C(=O)NCCO CC(C)C(C)(F)CNC(C1C=CCN1C(=O)CC(=O)OC(C)(C)C)=O c1(CN(C=O)Cc2c(C)n3c(s2)cnc3)ccc(F)c2c1CCC2 C1(NC(C2C(C=C)C2)=O)COCC1CNC(C1(COC)CCC1)=O C1(C(=O)NC(CCO)C(F)F)(CC)CCCN(C(=O)COCCCN=[N+]=[N-])C1 C1(C(C)NC(N(CC(=O)OC)CC)=O)(CNC(=O)CCC(=O)OC)CCOCC1 C(CCCC(=O)NCC1(C)CCCOC1)N(C(COC)=O)C C#CC(C)(C)C(=O)N1CCCC(N(CCF)C(c2ccc(OCCO)cc2)=O)C1 C1(C(=O)NCC(C)(O)CNC(=O)CC2CCOCC2)CCOC(=O)N1 Cn1c(C(=O)NC2CC23CC(NC(=O)Cc2ccc(F)c(F)c2)C3)ccc1C#N c1(CC(=O)NC(CCNC(CNS(CC)(=O)=O)=O)C)cc(C)[nH]n1.C1CO1 N1(C(CCNC(=O)OCC)=O)CC(C(=O)NCC2C(CO)C2(F)F)CC1(C)C c1(CCC(=O)NC(CSCC)C(=O)NC(C)Cc2cn[nH]c2)ccnc(C)n1 C1(C(=O)NC(CCC)CO)CCC(C(=O)N(CCc2c(C)n[nH]c2C)CC)CC1 CC1(C)C(NC(C2CC23CCSCC3)=O)CCN1C(C1C=CCC1)=O C(=O)(C1=Cc2ccccc2C1)N1C(CC(N2CC3(CCC3)CC2CO)=O)CCC1 C1(O)(CC(=O)NCC2(CCNC(C3CC4CC3C4)=O)CC2)CCCC1 C12C3CCCN(C3C1(C)C)C2=O.Cc1nnc(CC(=O)NCCn2ccnn2)o1 N1(C(c2c(OC)cccn2)=O)CCc2sc(C(N3CCC(C)C(F)C3)=O)cc2C1 CCC(C)(C)C(=O)N(C1CCC(NC(c2nc(C(F)(F)F)cn2C)=O)CC1)C C(=O)(C(F)(F)C(O)C(C)C)NC1CCN(C(CCSCCCC)=O)C1 c1ccc(N2CCOCC2)nn1.CCC(C)C(C)NCC(=O)O N1(C(C2(C=C)CC2)=O)CCC(N(C)C(c2cc(C(N)=O)[nH]n2)=O)C1 CC(C)(C)CCC(F)C(=O)NC(C1(CNC(C23CC2C3)=O)CC1)=O CC(Cn1cccn1)C(=O)N1CCC(CCNC(C2CC(C(F)(F)F)C2)=O)C1 N1(C(C(CCC)O)=O)CCN(Cc2ccccc2)C(CNC(c2cnn[nH]2)=O)C1 C#CCCCC(C)C(=O)NC(CCNC(=O)C(C)(C)CNC(C)=O)C(C)C C1(NC(=O)Nc2c(OC)cc(OCCN(C)C)cc2)CCCC1C1CCCC1 CC1CN2CCN1C(C(=O)NCC1CC(F)(CNC(=O)CCC3(C#N)CC3)C1)C2 C#CCCCCC(=O)NCCCOCCNC(C1CCN(S(C)(=O)=O)C1)=O C1(NC(c2ccc(C(C)O)cc2)=O)CN(C(c2coc(C3CC3)n2)=O)CC1(C)C C(=O)(CC(CC)N(C)C(c1ccc(C#N)s1)=O)NC(C1CCCO1)CC C1(CC)CCN(C(=O)CCOCCCOC)C1CNC(=O)CS(C)(=O)=O N1(C(c2nnn(C(C)(C)C)n2)=O)CCCCCC1CNC(c1coc(Cl)n1)=O N1(C(C(=O)NCC)=O)CCCC(C)C1CNC(=O)C(C)(C)c1ccccc1 C1(C)(C(=O)NC(CNC(c2[nH]c(=NC)sc2)=O)CC(C)C)CCCCNC1=O N1(C(CC=C(C)C)=O)CCCN(C(c2cccc(Cl)c2OC(F)(F)F)=O)CC1C n1(CCC)cc(C(c2nnnn2C(C)(C)C)NCCn2cc(Cl)cn2)cn1 C12(C(=O)NC(CC)CN(C(=O)CC3(C)CCCCC3)CC)CC3CC1C2C3(F)F c1(C(N2CCN(C(Cn3ccc(C)n3)=O)CC(O)C2)=O)cnc2nccnc2c1 C(=O)(C1CCCc2c1ncn2C)N1CCCN(C(c2[nH]cc(C)c2)=O)CC1CO CCCC(C(=O)NCC=C1CCN(C(c2nn(C)cc2N)=O)CC1)NC(C)=O C1(CNC(C(C=C)C)=O)CCCC12CCN(C(=O)C(C1CCCSC1)SC)CC2 c1(NC(CC)(CNC(=O)CC(C)N(C)C)CC)ncc2cccnc2n1 N1(C(C(C)(F)F)=O)CCC2(CCC(C(N3CCC(O)CC3)=O)O2)CC1 c1(C(=O)NCC2CC(NC(C3C(=C)CC3)=O)C2)cnoc1C(C)C C1(C(N2C(C(N3CCC(OC(C)=O)C3)=O)CCCC2)=O)CC(C(C)C)=NO1 CC(C)(C)CC(O)CC(=O)NCc1ccc(Cl)cc1OCCO c1(C(=O)NC23CCN(C(C4N(C)CCOC4)=O)CC2C3)ccc2cnoc2c1 N1(C(=O)OC)CSCC1C(=O)N(CCCCNC(=O)CCOc1ccccc1)C C(CCN(C)C(C1(C)CC2CCC(C1)S2)=O)(C(C)(C)C)NC(CNC(CC)=O)=O c1(C(=O)NC(C2CCCN2C(c2coc(C3CCC3)n2)=O)C)ccc(F)c(O)c1 N1(C(c2c(C)cc(C)o2)=O)Cc2ccnn2CC(NC(=O)C(C)CF)C1 n1(CCOCC)nc(CSCC)nc1-c1ccn(-c2c(C)n[nH]c2C)n1 c1(C(N2CCCC(CO)(NC(C3CC(O)C3)=O)C2)=O)ccn2nccc2n1 c1(C(N(CC(C)NC(c2c(C)occ2)=O)C)=O)nccc2c1[nH]c1ccccc21 CC(C)C(O)C(C)C(=O)NC1(CNC(=O)C2=COCCC2)CCCCC1 CC(C)C(C(=O)OCc1ccsc1)c1ccc(F)cc1.C12CC(C(O)C1)NC2=O N1(C(CC(C(C)C)OCC)=O)CCC2OCCN(C(c3ccc(CC)s3)=O)C2C1 C12(CNC(C(C)OCC)=O)CCC(CC1)N2C(c1cc(N)nc(Cl)c1)=O Cc1ccc(C(=O)NC2CC(C(=O)NC(C3(CO)CC3)C)C2)cc1C C(CC1=CCN(C(=O)CC(C(F)(F)F)n2ccnc2)CC1)NC(C(C)OCC)=O c1(C(N(CCCCCNC(=O)Cc2cnc[nH]2)C)=O)nc2ccccc2cc1Cl C1(NC(CC2(OC)CC2)=O)CCCCN(C(C2CN(C)CCO2)=O)C1 C1(C(=O)NC2(C)CN(C(C3C(CN(C)C)C3)=O)C2)C(F)(F)C12CCC2 CC1CN(C(c2c[nH]nc2C(C)(C)C)=O)CC(C)N(C(=O)C2=CCC2)C1 C(c1nc2ccccc2s1)=CC(=O)N(CC1N(C(C(C(C)C)F)=O)CCC1)CC CN1CCC(C)(C(N2CC=C(CNC(=O)CC3CC(CC4CC4)C3)CC2)=O)C1=O N1(C(c2c(C#N)cc(F)cc2)=O)CCC2C1CCCN2C(C1CCC(O)CC1)=O c1(CC(N2CCC(CCNC(=O)C=Cc3cscn3)C2)=O)ccccc1C1CC1 C1(CN(C(C2(C#C)CC2)=O)C)CN(C(c2c[nH]c(=N)s2)=O)CC12CC2 c1(C(=O)NC2CN(C(c3c(C)cc(C)nc3)=O)CC23CC3)ccc2cc[nH]c2c1 C1(NC(CN(C(=O)Cn2cccn2)C(C2CC(N)C2)C)=O)CCCCC1(C)C CC(C)C(C)CN(CCC(=O)NCCN(C(c1coc(Br)c1)=O)C(C)C)C CC1(NC(=O)CCc2ccncc2)CCCCC1C(=O)NCC1(CCO)CCC1 C(=O)(C1=CC2(CCOC2)C1)NCCCCCCNC(c1cnc(CC)nc1C)=O C#CCC(C)C(=O)N1CCCC(N(CCO)C(c2cnnc(O)c2)=O)C1 N1(C(C(C=C)(C)O)=O)C2CCC1CC(CNC(=O)CC1CCOC(C(C)C)C1)C2 C1(CC)CCCCC1C(=O)NCC1(CN(C(=O)CCN2CCCCC2=O)C)CC1 C1(CN(C)C)CCN(C(=O)OC(C)(C)C)C1(C)C.c12ccc(F)nc1CNC2=O c1(C(=O)NCC=CC(=O)NCCNC(CC(C)C)=O)ccc(Br)cc1 c1(C(=O)NC2C(NC(CNC(CN(C)C)=O)=O)COCC2)cc2occc2[nH]1 C1(c2n(C)nnn2)CCN(C(=O)CC2CC(Oc3ccccc3)C2(C)C)CC1 c1(C(=O)NCC2(C)N=N2)ccc([N+](=O)[O-])c(NCc2ccccc2)c1.C1CC1 N1(C(CC2CCCC(C)O2)=O)CCC(C)(C)C1C(=O)NOCC(F)(F)F c1(C(N(C2CCN(C(c3cncc(CO)c3)=O)C2)C)=O)ccc(F)cc1C1CC1 c1(C(=O)NCCC(O)CNC(C2CC2F)=O)ccc(OCC(F)(F)F)nc1 Cc1nc(CC2CC2)sc1C(=O)NC(C)CCNC(C1(C(F)F)CCC1)=O c1(C(N2CC(OC)C(NC(c3ccncc3O)=O)C2)=O)ccnc2c1CCC2 C1(C)(CNC(C(C)CN(C)C)=O)CCC(NC(=O)Cn2ccc(C3CC3)n2)CC1 CCC(C)(C)CC(=O)NC1C=CC(CC(=O)NC2(C(N)=O)CCCCC2)C1 c1(C(C)Nc2n[nH]c(-c3ccccn3)n2)ccc2c(c1)OCCO2 C1(CNC(c2c(C)scc2)=O)CN(C(=O)CCC2CC2(F)F)CCC12CCC2 C(C(O)C(C)c1ccccc1)CCN1C(=O)C(C)N(C(=O)COC)CC1.C(N)(=O)OC N1(C(c2cc(C)n(C)c2)=O)CC(C)N(C(C2CCN(CCO)C(=O)C2)=O)CC1C c1(C(N2C(CNC(CC(CC)CN(C)C)=O)CCC2)=O)nc2ccccc2o1 c1(C(N2CC3C(CNC(=O)Cn4cc(CO)nn4)(C3)C2)=O)ccc(Cl)cc1O C1(NC(c2n(CC=C)ccn2)=O)(CO)CCCN(C(c2cncc(OC)n2)=O)C1 c1(C(N2CC3C(CNC(c4c(CC)ocn4)=O)C3C2)=O)c[nH]c(=N)c(C)c1 C(=O)(C1SCc2cccnc21)N1CC(C)C(n2cc(-c3cnsc3)nn2)C1 c1(C(=O)NCC(CC=C)NC(c2ccc(CC)nc2C)=O)noc2c1COCC2 c1(C(N(C(c2ccccc2)CNC(CNC(CCC)=O)=O)C)=O)cc(C#N)no1 C1(NC(C2CC(CC)C2)=O)CCCC(NC(c2ccccc2OC(F)F)=O)C1 c1(C(CC)C)ccccc1OCC(=O)N(C)CCN(C)C(c1c[nH]cc1Br)=O C#CCC(C)(CC)C(=O)NCCCC1CCN(C(=O)CS(=O)(=O)C2CC2)CC1 N(C(=NCCCF)N1CCC(OC(F)(F)F)C(C)(C)C1)CC1CCC(CC)O1 CCCC(CC)C(C(=O)NC1COC1)N1CCCC(Cn2ccnn2)C1 c1(C(C(=O)NC(CC2CN(C(C(C)=C(CC)C)=O)C2)C)C)cnn(C)c1 c1(OCC)ccc2c(c1)C(NC(=O)Nc1cc(CSC)ccc1O)CCS2 C1(C(C(CCC=CC)=O)=O)CN(C(=O)Cn2nc(N)cc2C)CC1C1CC1.NC CCC(CC(=O)NCc1nn[nH]n1)NC(c1cn(C)nc1C)=O C(CCCC(C)C)N(C(C1N(C(C(COCC)C)=O)CSC1)=O)C c1(CC)nn(C)c(CC)c1NC(=O)NCCN1CC(C)CC1CC c1(C(=O)NC2C3(CC(NC(C)=O)C3)C2)ccc(C)nc1Cl N1(C(CCC(C)SC)=O)CCCC2C1CCN2C(=O)CN1CCC(C(N)=O)CC1 N1(C(C(C)NC=O)=O)CC(C)(C)CC1CC(=O)NCCCc1ncn(C)n1 c1(CN2C(C(=O)Nc3ccc(F)nc3)CCC2)ccc(F)c(CO)c1F C1(C(N2CC3C(C)C3C2)=O)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCN1C c1(C(N(C)CC2(NC(=O)Cc3cnnn3C)CCC2)=O)cc2n(n1)CCCC2O C(=O)(C(C1CC1)N(C(=O)C(F)n1ccnc1)C)NCCSCCOC N1(C(C(C)OCCCCCC)=O)CC2(CC(NC(=O)C(N)=O)C2)C1 c1(NC(C2OCCN(C(Cn3ccc(C)n3)=O)C2)=O)ccc2nnsc2c1 c1(C(=O)NCC2C(F)(F)CCN(C(C3(C#C)CC3)=O)C2)cc2cccc(F)c2s1 C1(NC(c2cnc(COC)s2)=O)CC(F)CN(C(=O)C=Cc2ccccc2)C1 CCC(C(=O)NC(c1cccnc1)C(=O)NCCN1CCNC1=O)C(F)(F)F CCCCCCC(C)C(=O)N1CC2CC1(C(N1CCCC1C1CCOC1)=O)C2 c1(C(N(CCCN(C)C)CCNC(C2(C)COC2)=O)=O)ccc(O)nc1 C(=O)(CCCC(=O)NCCCOCCNC(=O)C(c1ccc(F)cc1)CO)NC c1(SC(C)C(N2CCOC(CNC(C3CC3(C)C)=O)C2)=O)ccc(F)cc1 C12(CS(=O)(=O)NC3CN(C)C(c4ccccc4)C3)CCCN(CC1)C2 C(CCCCCNC(c1csc(C(F)(F)F)c1)=O)NC(CCC#C)=O CCCCC(CC)CCC(Cn1c(NC2CC2)nnc1-c1cc(Br)cn1C)CC C(=O)(CCCC(F)(F)F)N1C(CNC(CCCC(=O)NCC)=O)COC(C)(C)C1 c1(C(=O)NC2(CC(=O)N(C(C)CS(C)=O)C)CC2)ncccc1O C1(C(N2CC(C#C)C2)=O)CCN(NC(C2(CC=C)CC2)=O)CC1(C)C N1(C(c2cc(C)on2)=O)CC2(CCOCC2C(=O)NCc2cnccn2)C1 c1(C(=O)NCC(C)NC(=O)C=Cc2ccncn2)cc(N)cc(O)c1 C1(NC(C2OCCN(CC)C2)=O)CN(C(=O)CS(=O)(=O)CC)C2(CCOCC2)C1 C1(C(=O)NC2C(NC(CCc3cccc(OC)n3)=O)C2)CC2(CCOCC2)CO1 N1(C(CC=C(C)C)=O)CCCC2CN(C(c3cccc4c[nH]nc34)=O)CC12 C1(CCCNC(=O)CCN2CCC2)CCCCN1C(c1ccccn1)=O c1(C(N2CCOCC(NC(C(C)n3ccnc3)=O)C2)=O)c([N+](=O)[O-])cnn1C C1(O)(C(C)NC(c2nc(C)[nH]n2)=O)CCN(C(c2ccc(CO)cc2)=O)CC1 c1(NCCC(C2CC2)NC(=O)CCCC(=O)NCCC)nnc(C)c(C)c1C#N c1(CN2C(CC(=O)Nc3cccc(F)c3)CCC2)ccc(CO)cc1 C(c1cccc(F)c1F)=CC(N1C(C)C(NC(C2(F)CCC2)=O)CCC1)=O N1(C(c2c(C#N)scc2)=O)CC2CC(C1)N(C(C1CCCC1C(F)F)=O)C2 N1(C(Cc2c(C)ccs2)=O)CCOCC(CNC(=O)CCCC2CCCC2)C1 CC1(C)CCC(NC(=O)CC2C3CCC(C3)N2C(=O)C(O)C2CCC2)CC1 N1(C(CSc2n(C(C)C)cnn2)=O)CC2CC2(CNC(c2ccccn2)=O)C1 C#CC(CC(C)(C)C)NC(C1CN(C(C2(CC)CCOC2)=O)CCN1C)=O c12ccccc1C(=O)NC(C)CNC(=O)C21CC1.c1(C(C)=O)cn(C2CC2)nn1 CC1CN(C(=O)C(N)=O)CC1C(F)(F)F.c12cnc(o1)-c1ncc(s1)CNC2=O C1(NC(c2cc(CC)on2)=O)CN(C(c2cccc(OCCO)c2)=O)CC1F C(=O)(CCC(=O)N1CC2CC1C2NC(=O)C(C)Cn1ccnc1)c1ccc(C)s1 O=C(N=c1ccn(CCN2CCCC2)[nH]1)c1ccc(-c2ccc3c(c2)OCO3)nc1 c1(C(N2CC(N(C(=O)C#CC3CC3)C)C3(C2)CC3)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(C2(CCNC(CC3(CC)CC3)=O)CC2)=O)CCCC1C(C)C N1(C(c2c(OC)ccs2)=O)CCC2(CCC2)C(NC(=O)CC2CC2)C1 c1(C(=O)NCC2C(c3n(C)ncc3)C2)c(Cl)ccnc1F c1(C(=O)NCCCCN(C(CCSCC)=O)C)c(NC(C)=O)cccc1C C1(CCNC(C2C(OC)CC2)=O)CSCCN1C(c1cc(C(C)C)no1)=O CC(C)CC(O)CNC(Cc1ccccc1)Cc1ccccc1Br Cc1nc(CNC(c2nccnc2N)=O)oc1C(=O)NCC1CNC(=O)O1 C1(CN(C)C(C2(CO)CCCC2)=O)CCN(C(C2CC2C(C)(C)C)=O)CC1 Cn1nccc1C(=O)NC1CC(CCNC(=O)CC2CC(=O)C2)C1 c1(C(N2CC3C(N(C(=O)Cc4ccc(F)cn4)C)C3C2)=O)cc(F)cc(Cl)c1N CC1(C)CCC2(CC1)CC2C(N1CC(NC(c2cc(Cl)ccc2N)=O)C1)=O C1(CN(C(CN(C)C)=O)C)CCCN1C(c1cnn[nH]1)=O c1(CC(=O)NCC(CC)NC(c2cc3n(c2)CCC3)=O)ccc(OC)cc1Cl c1(O)ccc2ccccc2c1Br.c1(N)cc2c(Cl)cncc2o1.CN1CC1 N1(C(C(=O)NCCCC(N)=O)=O)CCCC(F)(F)C1 c1(C(=O)NCC(C2CCC2)OCC)ccc(S(=O)(=O)NC)o1 C(C)(CSC)(C(=O)NCC1CCCN1C(=O)C(c1ccc(F)cc1)CO)OC N1(C(Cc2ccc(C)cc2)=O)CCCC(NC(c2c(C)ncnc2O)=O)CCC1 CCCCC(C)(F)C(=O)NCC1CN(C(=O)C(C)(C)C(C)(F)F)CC1(C)C c1(NC(=O)NC2(CN3CCCCC3)CCOC2)cc(-c2ccncc2)ccc1F N1(C(C2(CC)CCNC2=O)=O)CC(NC(=O)NC)CC2(CCC2)C1 CCC(CC(C)C)C(=O)N1CCC(OCC(=O)NC(C)(C)C(C)(C)C)C1 c1(CC(=O)NC2CCC(NC(C(C)(C)c3cccnc3)=O)C2)cc(O)nc(O)n1 N1(C(CC2(N)CCS(=O)(=O)C2)=O)CCc2c(F)cc(C(=O)O)cc2C1 C1(C(N2CCC(CNC(CCCN(C)C)=O)C2)=O)CC(=O)N(C2CCCCC2)C1 CN1CCC(=O)NC2CN(C(=O)Cc3csc4cccc(Cl)c34)CCC12 N1(C(CN(C(=O)C(C)(C)C)CC#C)=O)CCC(N(C(=O)CNC(C)=O)C)C1 C(=O)(CC(C)CCC(=O)N1CCN(CCCNC(=O)CCF)CC1)OC c1(OCC)cccc2c1OCC(NC(=O)CS(=O)(=O)C1CCCC1)C2 c1(C(N2C3(C(N4CC(CC)SCC4)=O)CC(C)(C2)C3)=O)cccn2ccnc12 C12CCC3(CC1)CN(CCO3)C(=O)CNC2=O.N1(CC#C)CCCC1.C1C(=O)N1 Cc1nncn1CCCNC(=O)C(CC1CC1)NC(c1csc(=N)[nH]1)=O N1(C(CCCOCC=C)=O)CCC2C(C1)CN2C(=O)C(F)C1CC1 Cc1ccc(NC(=O)CC2CCCN2C(c2c[nH]c(=S)cn2)=O)cc1O N1(C(Cc2cccc(OC)c2)=O)CCC(C)(NC(=O)Cc2csc(CO)n2)CC1 c12ccccc1C(=O)c1c[nH]cc1C(=O)NCCCNC2=O.C(C)(C)(C)S.CC C12(C(=O)NCC(C(=O)NCC(=O)OC)N(C)C)CC(C#N)(C1)C2 c1(C(=O)NCC(CC(=O)NCC(CCC)(C)O)C2CCC2)ccc(C)c(C)n1 C1(CNC(C2CCC(C)CC2)=O)C2CCCC1N(C(C1CCS(=O)CC1)=O)C2 Cc1nc(O)nc(O)c1CCC(=O)NC12CC(NC(C3CC(O)C3)=O)(C1)C2 Cc1cc(C)c(C(=O)NC(C)CNC(C2CCC(C)(C)OC2)=O)cc1Br c1(OC)cc(C)cc(C(N2CC3(CCN3C(C3CCCCC3O)=O)C2)=O)c1C c1(C(=O)NC(C)CCCCNC(=O)CCC2CCOC2)cnc2[nH]ccc2n1 N1(C(C2(CC)CCNC2=O)=O)CC=C(CCNC(=O)CC2CCSCC2)CC1 c1(N2CCN(C)C(=O)C2)nc(NCC2C(=O)NCCC2C)c2ncsc2n1 c1(C(=O)NCC#CCNC(C=CC(CC)C)=O)cnnc2ccccc12 c1(C(N2CCCC(NC(CCCC(C)C)=O)C2C)=O)cc(O)nc2ccccc12 N(C(=NCCc1ccccn1)NCc1ccc(C)o1)Cc1ccc(OC)nc1 C12(CNC(CCCOCCOCC)=O)CC(CC)(CN1C(C1(C3CC3)CC1)=O)C2 CC(C#N)CNC(=O)C(c1ccoc1)NC(=O)CN(C)C(N)=O Cc1ccc(C(N2CCN(C(C3CC(O)CN3C(N)=O)=O)CC2)=O)cc1O c1(C(=O)OC)cc(OC(F)F)c(OC(=O)C(CC)CCC)cc1OC(F)F C1(CN(C(=O)CCc2cn(CCc3ncon3)nn2)C)C2Cc3ccccc3C12 N1(C(=O)COC2CC=CC2)CC2(C1)CN(C(c1ccc(Cl)nc1Cl)=O)C2 C(c1cccc(F)c1)=CC(=O)NCC(CCOC)NC(C1(CCOC)CC1)=O N1(C(c2c(C)nccn2)=O)CC2CCC(C1)C2N1CCC(C)OC(C)C1 c1(CN2CC(CC(C)O)C2)cn(CCN(C)C)cn1 c1(C(=O)NC(CN(C(C(F)=C(C)C)=O)C)C)csc(S(C)(=O)=O)c1 N1(C(c2c(CCC)nns2)=O)CCN(C(c2ncnn2CC)=O)CC(O)C1 N1(C(CNC2CC(C)(CC)OCC2)=O)CCc2cc([N+](=O)[O-])ccc2C1C C1(CC(=O)NCC2CCC(NC(c3n(CC)c(O)nc3)=O)C2)CCC(C)(C)CO1 c1(OC)coc(C(=O)NCC(C)(O)CNC(C2CC(CC(C)(C)C)C2)=O)cc1=O Cc1cc(C2(C(=O)NCc3cc(C#N)ccn3)CC2)cc(C)c1 C(=O)(CC(C)C(=O)OC)NC(CC)C(=O)NC(c1ncc[nH]1)C C(CC(C)(C)C(=O)N1CCC(C)(NC(=O)CCS(C)=O)C1)OC O(NC(CCO)CC(C)C)N(CC)CC.CCCCO C1(CC(=O)NC2C3CC(CNC(C(CCC)O)=O)(C3)OC2)CCN(OC)CC1 C1(C2CC2)(COC)CN(C(=O)C(c2ccoc2)NC(C2SCCS2)=O)C1 C1(C(N2C3C(CNC(CCCOC)=O)CC(CC3)C2)=O)CC(C)(C)OC(C)(C)C1 Cc1ccc(OCCC(=O)OCCC2(O)CCCNC2)c(Cl)c1 N1(C(CN(CCC#C)C)=O)CC2CCN(C(c3nc4ccccc4[nH]3)=O)CC2C1 C(=O)(CCC(=O)NCCCC(C)NC(=O)C(c1ccc(C(F)F)cc1)C)OCC Cc1[nH]c(C#N)cc1C(=O)NC1CC(NC(C2(Br)CC2)=O)C12CCC2 c1(C(=O)NC2CN(C(CCOCC#C)=O)CC2C)ccc(F)c(COC(C)C)c1 Cc1ncnc(C)c1CC(=O)NC1CC(C)CN(C(C2COC(=O)N2C)=O)C1 c1(C(=O)OCC)nnn(C2CCN(CCN3CC(C)CC3)CC2)c1C(F)(F)F C(=O)(C(C(C)C)Nc1cncnc1)N(CCCNC(CN(S(CC)(=O)=O)C)=O)C c1(C(N(C2CC(C(=O)NCCc3ccncn3)C2)C)=O)cncc(CO)c1 Cc1nc(C(=O)NCC2(NC(=O)Cn3nnnc3C(C)C)CC2)ccc1C#N C(CCC(O)CO)N(C(=O)CC(O)CNC(=O)COC1CC1)C C1(CNC(CNC=O)=O)CCC12CCN(C(=O)C=Cc1ccc(O)c(O)c1)CC2 c1(NCC2(O)CN(C(c3c(SC)scc3)=O)C2)ncnc2c1ncn2C C(C)(C)(C(C)CC(=O)N(C)CCOC(F)F)NC(c1n(CC)ccn1)=O c1(C(=O)NC2C(NC(CCc3ccc(C)cc3)=O)CC2)ccc(O)c([N+](=O)[O-])c1 CC1CCC=C1C(=O)N1CCC(NC(c2cc(=O)cc[nH]2)=O)C12CC2 c1(NC(c2ccc(CNC(Cc3c(C)ncs3)=O)s2)=O)cnc(N(C)C)nc1 N1(C(c2c(C)nc(CC)o2)=O)CCC(C2CC2NC(=O)C(C)C2(O)CCC2)CC1 c1(C(=O)NCC(C(C)C)NC(C2CCCN2N=O)=O)cccc(C(C)(C)C)c1 C1(N(C(c2c(C)nn(CC)c2C)C(=O)NC2CC2)C)CS(=O)(=O)C12CCOCC2 n1(CC)nc(C)c(C(=O)NC2CC3CC(CO)CC23)c1C(F)(F)Cl C1(C(=O)NC2CCCC(NC(C3C(OCC)CCCC3)=O)C2)CC2CCC1CC2 N(C(=NCC1COCCOC1)N1CCC2(CCOCC2)CC1)C(C=C)C N1(C(C(n2cc(C)nc2)(C)C)=O)CCC(NC(=O)C=CC2CC2)C(F)C1 CCCN=C(NCC(CO)C(C)(C)C)NC(C1C(C2C(C(=O)OC)C2)CC1)=O c1(OCCC)cc(OC)ccc1C(=O)NC1CN(C(=O)C(C)C)CC1C(F)F [N-]=[N+]=NC1(CNC(c2[nH]ccc(=O)c2O)=O)CCN(C(=O)CC23CCCC2C3)C1 c1(OC)cccc(C(C)(C)C(=O)N(CC(C)NC(=O)C(C)(C)OC(C)=O)C)c1 c1(C(N(CCNC(Cn2ccc(C)n2)=O)CC2CC2)=O)ccc(C2CC2)nc1 c1(OC)sccc1C(N1CCC(C(=O)NCC2COCC2O)C1)=O c1(OC)cccc(OC)c1C(=O)N(C(C1CCCCC1)C(C)C)C C12(NC(CCCOCC)=O)CCCC1N(C(C1CC1c1ccccc1Cl)=O)CC2 c1(C(N2CC(NC(Cc3c(C)noc3)=O)C(F)CC2)=O)cc(C#N)ccc1Br C1(C(=O)NC2(C)CC2)CC(F)CN(C(c2cccc(C(C)(C)C)c2)=O)C1 c1(C(=O)NCC(CC(=O)N(C2CCOC2C)CC)(C)C)coc2ccccc12 c1(C(N2CC(CN(C(c3cc(C)nc(Cl)c3)=O)C)C2)=O)nccc2ccsc12 c1(C2C(NC(C3(N4CCCC4)CC3)=O)CC2)nc(S)n[nH]1 c1(C(=O)NC2CC(C)N(C(=O)CC(C)(C)F)C2)cc([N+](=O)[O-])cc2ccccc12 c1(COC)nc(C)ncc1C(N1CC2(NC(C3CCOC3)=O)CCC1C2)=O C(=O)(C1=CCCN(C(C2CCC(=O)C2C)=O)C1)NC(c1c(C)nns1)C N1(C(c2c(C)c(C3CC3)on2)=O)CCC2(CC2NC(c2cnccc2Cl)=O)C1 N1(CC(=O)Nc2cccc(Br)c2)CCCCNCC(F)(F)C1 C(=O)(C(F)C(C)CNC(=O)CC1(N(C)C)CC1)N1CC(C(=O)OCC)C1 C1(CCO)CCC(C)(C)CC1.C=CC(CC1CC1)CCNCC=C CN(CCOc1ccc(Cl)cc1Cl)N1CCn2c(-c3cccnc3)nnc2C1 N1(C(c2c(C)nccc2)=O)CCC(F)(F)C(NC(c2cc(F)c(F)cc2F)=O)C1 C(=O)(C(CC1CC1)CC1CC1)NCC(CC)NC(=O)C(C)(C)c1ccnn1C N1(C(C(C)NC(COC)=O)=O)CCCC(NC(=O)C=CC=C(Cl)Cl)C1C C1(NC(c2cc(C)nc(O)n2)=O)CCC2CN(C(=O)C(C)(C)O)CC2C1 N1(CC)C(=O)CCC1CC(=O)NC1CC(CNC(=O)CSc2ccncc2)C1 c1(CC(=O)NC(CNC(c2c(C)nc(C)[nH]2)=O)C2CC2)ccc2c(c1)CC(C)O2 c1(C(=O)NCC2(C)N(C(CNC(CC)=O)=O)CC(F)(F)C2)cc(S(C)(=O)=O)oc1C CN1CCC(CC(=O)NCC2CC(NC(C3COCC3(C)C)=O)C2)CC1 c1(C(=O)NC)ccc(C(=O)NC2CN(C(C)C(=O)NC(C)C)CC2(C)C)cc1F CN1CCN(C(C2(CNC(C3CC=CCC3)=O)CCC2)=O)CC(O)C1 C1(C(=O)NCC(CO)C(C)C)(CNC(Cn2ccc(C)n2)=O)CCCCC1 N1(C(C)CC2CNc3ccccc3O2)CCC2C(C1)NC(=O)CCN2C CCCC(C(=O)OC)C(=O)NC(C)(C)CC(=O)NC1CCCCC1CCO C(=O)(N=c1nc[nH]n1C)C1N(Cc2c(OC)cc(Br)cn2)C2C(C1)C2 C1(CNC(Cc2c(C)occ2)=O)CC(NC(C23CC(C)C2C3)=O)CCO1 Cc1ccc2cccc(C(=O)NCCC3CCCCN3C(=O)C=CS(C)=O)c2n1 CC1CN(C(=O)COc2ccc(O)cc2)C(C)CN1C(=O)CCC(F)F c1(C(=O)OC)cc2c(Br)cccc2c(N2CCOC(CCN)C2)n1 C1(CCC)(CNC(C2CC(OC)C2)=O)CCN(C(c2nnn(C)c2C)=O)C1 c1(CC(=O)NC2CCC2NC(c2cncn2C(F)(F)F)=O)conc1C(C)=O C12(CNC(c3n[nH]cc3Br)=O)CCC(CC1)N2C(=O)CC1CCC1 S(=O)(=O)(c1ccc(C#N)c(NC(c2nccs2)C)c1)NCCn1c(CC)ncc1 C1(NC(C(CCC)OCC)=O)CCCN(C(=O)C(C)=CC(C)(C)C)C1C N1(c2nnc(C)s2)CCC(C2CCCN(C(C3CCC4(C3)CC4(F)F)=O)C2)CC1 Cc1cc(C)c(NC(=O)C(N2CCC(N(C)C(C)C)CC2)=O)c(C)c1 C#CC1CN(C(C2C(CC)CCN2C(=O)Cc2cn(C)nc2C)=O)CCO1 N1(C(c2cncc(SCC)n2)=O)CCN(C(=O)Cn2cccnc2=O)C(CO)C1 C1(NC(CCCOCC=C)=O)CC2(C1)CC(NC(C1(c3cc[nH]n3)CC1)=O)C2 C1(CNC(C2C(C=O)C2)=O)(CO)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1.COC C1(CC(=O)N(C2CCN(C(c3nc(CC)oc3)=O)C2)CCO)COCC(C)(C)O1 C1(C)(C(N(C2CCN(C(=O)Cc3ccc(C(=O)OC)cc3)C2)CC)=O)CCOCC1 N1(C(C23CCC(NC(c4cc(C)on4)=O)(CC2)C3)=O)CC(=O)NC(C)(C)C1 N1(C(c2c(C)n(C)cc2)=O)C2CCC1CC(C(=O)NC1COCC1N=[N+]=[N-])C2 N1(C(C(CCC)OCC)=O)CCC(F)(C(=O)NCCN2CCC(OC)C2)CC1 c1(C(=O)NCC(CNC(C(C2CCC2)OCC)=O)CO)cc(C)ccc1C C(=O)(CN=c1ccc(C#N)c[nH]1)NCC1(NC(CC(C)N(C)C)=O)CCC1 c1(C(CC(N2CC3(C2)NC(=O)N3)=O)C)ccc(C(N)=O)cc1.C(C)(SC)SC C1(CNC(C2(C)C=CCC2)=O)CCCCN1C(c1sccc1SC(F)F)=O Cc1c(C)c(-c2c[nH]c(=NCc3cnc(Cl)c(F)c3N)s2)c(C)c(C)c1C N1(C(C2(CC#C)CC2)=O)CCCC(F)(C(=O)NC(c2noc(C)n2)CC)C1 C12(C(N3CC4C(CC)(C4)C3)=O)CC(C)(CN1C(C1CCC(O)CC1)=O)C2 C(=O)(C(C#N)C(C)(C)C)NC1(CN(C(C=C2CCC(C)CC2)=O)C)CC1 N1(C(C(C)NC(c2ccoc2)=O)=O)CC2CC(NC(c3ccn(C)c3)=O)C1C2 c1(CN2CCCC(C(=O)NC(C3CCOC3)CC)C2)ccc(Cl)cc1OC C1(CC(=O)NCC(=O)N(CC=C)C(C)C)OCCO1 CC(CCO)CN=c1nc(N2CCCC3(CCCC3)C2)c2sccc2[nH]1 C(CC(C)N=c1nc(C#N)[nH]cc1C)NC(C1CCCN(CC)C1)=O c1(-n2cc(CNC(c3ccc(Br)s3)C)nn2)cc(F)ccc1Cl C1(NC(c2cncc(OC)c2C)=O)CN(C(=O)CC(F)F)CC(C)(C)C1 C=CCCCCCCC(=O)NC1CCC2CC1CN2C(=O)CSC(C)(C)C CCCC(CC(=O)NC1CCC(O)CC1)NC(=O)C(O)CN(C)C N1(C(=O)NC2C(C)N(C)CC2)CCCCC(CN=[N+]=[N-])C1 c1(OC)cnc[nH]c1=NCCc1cc(Br)no1 C1(F)(CNC(=O)C=Cc2ccco2)CCCN(C(C2CC23CC3)=O)C1 c1(C(N2CCN(C(C3(CC=C)CCOC3)=O)CC2)=O)nc(C(C)C)ncc1NC n1(CCC)ncc(CNC(=O)CSCC2N(C)CCCC2)c1C.C1(C)CCCOC1 C1(NC(CC(C)(C)OC)=O)CN(C(=O)CC2(O)CN(C(C)(C)C)C2)CC12CC2 N1(C(c2cc(CC)c(F)cc2)=O)CC2=C(C1)CN(C(C1CCN1S(C)(=O)=O)=O)C2 Cc1cc(C(=O)NCC(C)N(C)C(c2cc(-c3ccccn3)[nH]n2)=O)ncc1Cl C1(COC)CC(CNC(=O)C(C)Cc2cccc(Cl)c2)N(C(=O)CCF)C1 C1(C2CC2)(NC(c2cnn(CCC)c2C)=O)CCN(C(=O)CC(=O)N(C)C)C1 c1(C(=O)NCC(C)N(C)C(C2CCCSC2)=O)cc(Br)ccc1Cl c1(CCCCC)oc2ccccc2c1CNC(C1COC(=O)N1C)=O.C1C(=O)O1 C1(C(=O)NC2C(NC(c3nc(COC)sc3)=O)CCC2)CCCN(CC(C)C)C1 C1(NC(CC(C)c2ccco2)=O)(CNC(=O)C(O)Cn2cncn2)CCOCC1 c1(C(=O)NC2CN(C(C=C(CC)C)=O)CC2C)cnc(OC)c(C(F)(F)F)c1 c1(C(N(CC(C)NC(C2(F)CC=CCC2)=O)CC)=O)coc2c(F)cccc12 C(CC(C)CC)(C(=O)NOCc1ccccc1)NC(c1cc(CC)on1)=O C1(C(=O)NC2C(NC(C(F)=C(C)C)=O)COCC2)CCc2ccnn2C1 N1(C(=O)NCc2cccc(OCCCCC)c2)C2CCC1(C(C)O)CC2 C(CCc1ccccc1)(C(C)NC(c1ccco1)=O)NC(C=C1CCC(C)C1)=O N1(C(c2c(COC)cco2)=O)CCOC(C(=O)NC2CCCC2OC)C1 Cc1cc(=NCC(=O)NCCS(=O)C(C)(C)C)[nH]c(C(F)(F)F)n1 CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc[n+]([O-])cc2)=O)C(F)(F)C1 c1(N(C(=O)C(C)Cc2ccco2)CCC)ncnc2n[nH]c(C)c12.C(CC)(CC)N N1(C(C(C)C2CC2)=O)CC2(CCCCN(C(=O)Cc3ccnc(Br)c3)C2)C1 Cc1cc(C=CC(=O)NCC2CC(F)(F)CN2C(=O)CCF)ccc1C(F)(F)F c1(C(N2CC(CNC(C(C)(CO)OC)=O)(OC)C2)=O)cc(C)cc2ccncc12 C#CCCCC(C)C(=O)N1CCC(CN(C)C(c2c(C)cncc2C)=O)C1 c1(CC)ccc(OCC(=O)NCCC2CCN(C(c3c[nH]nc3F)=O)CC2)cc1 Cc1nc(O)[nH]c1C(=O)NCC1CCCCN1C(C1CCCCC1)=O C(=O)(CS(=O)(=O)C(C)C)N1CC(n2cc(CN(C3CC(C)(O)C3)C(C)=O)nn2)C1 C=CCC(CNC(c1cc(C)cc(C)n1)=O)C(=O)NCC(Cl)C(C)(F)F c1(C(=O)NC2CCN(C(=O)C=CC3CC3)CC2)cncc(Br)c1Cl c1(C(N2CCC(N(C(=O)CCC(=O)NC)CC#C)CC2)=O)cc(F)ccc1CC N1(C(C(C(C)C)SC)=O)CCCC2(CCC2NC(=O)Cc2cnn(C(C)C)c2)C1 C(C(C)CC(=O)NC(Cn1cncn1)C(N1CCCOCC1)=O)OC C1(C(N(C2CCCN(C(C3(C)CC(F)(F)C3)=O)C2)C)=O)CCS(=O)(=O)N1C c1(CN2CCC(NC(C)CC3CC3C3CC3)C2)cccc(Cl)c1 CCCCC(F)C(=O)N1CC(CNC(C2(C(F)F)CCCO2)=O)C2(CC2)C1 c1(C(N2C(CN(C(C3OCCN(CC)C3)=O)C)CCC2)=O)cnc2scc(C)n12 CC(C)(C)CCCCCC(=O)N1CC2CC(C1)CN(C(=O)CC1CCCCO1)C2 O=C(CCCc1cnn[nH]1)NCCC1CC1C(=O)NC1(CSC)CCOC1 CN=c1cc(C(=O)NC23CCN(C(c4oc(SC)cc4C)=O)CC2C3)cc[nH]1 c1(C(N2CCN(C(CCCC=C)=O)C(C(F)F)C2)=O)nc2ccccc2o1 c1(N2CCN(C(C)C(N)=O)CC2)ncnc2c1ncn2CC(O)CO C(=O)(C(C(C)C)Sc1ccccc1Cl)NC(CNC(C(CC=CC)C)=O)C1CC1 c1(C2(C(=O)NCCC(=C)CNC(C3CCC(C)C3)=O)CC2)ccc(Br)cn1 N1CC(N=c2[nH]c(=NC)[nH]c(=NCCCCCF)[nH]2)CC1=O.N1(CCC)CCCC1 C1(c2n(CCCOC)nnn2)(NCc2noc(C)n2)CC2CCC(C1)O2 CCCC(C)CC(C(=O)NCC(C)C)N(C1CCCCCCC1)C c1(C(=O)Nc2ccc(NC(C3CC=CCC3)=O)nc2)cc(Cl)ccc1Cl c1(CNC(N)=O)ccc(C(N2CC(NC(C3CCCCC3)=O)C3CC23)=O)cc1 C(=O)(C1=NOC2COCC12)N1CC(C(=O)NCCCCO)C2(C1)CC2 C1(CC(=O)NCC(C)NC(c2cnc(N3CCOCC3)s2)=O)CC(C)OC1C Cc1noc(CCC(=O)NCC(C)NC(=O)C(=O)NCC(F)(F)F)n1 Cc1ccc(C#N)cc1OC(C)C(=O)Nc1ccccc1C(c1ccccc1)=O CC1=C(C(=O)N2CC(NC(c3ccc(C4CCC4)nc3)=O)CC2C)CCO1 C1(C(=O)NCCN(C(CC)C)C)C=CC(NC(=O)Cc2cncs2)C1 N1(CCNC(Cc2c(C)nc(S)s2)C)CCOCC1(C)C C(CC(C(C)(C)C)NC(C1(C)CCOCC1)=O)N(C)C(c1cc(=O)cc[nH]1)=O C(CC(C)C(=O)NCC1CC1NC(c1ccnc(N)c1)=O)=CCC c1(NC(C)C)ccc(C(=O)N(C(C)CNC(=O)CCn2ccnc2)C)cc1F C1(NC(c2cocn2)=O)CC2CC1CN2C(=O)CCc1ccccc1Cl C(C(=O)N1OC2CCC1CC2)C12C(CN(C(C3(CCCF)CC3)=O)C1)CC2 N1(C(C(C)C(C)(C)C)=O)CCC2(CCC(NC(=O)CC3C=CCC3)C2)C1 Cc1cc(C(=O)NCC(CC2CC2)C(=O)NCc2ccc(C)s2)nc(O)n1 CCCC(CCCNC(=O)CCc1ncc[nH]1)NC(C1(CN(C)C)CC1)=O N1(C(C(c2ccc(C)cc2)=O)=O)CCN(C(=O)CC2OCCC2C)C(C)C1 Cc1cc(NC(C2CCCCC2NC(C2(C)CC(CF)C2)=O)=O)cc(O)c1 C1(C(N2CC3CC(NC(CC(C(C)C)C)=O)C3C2)=O)CC2(C1)CC(F)(F)C2 c1(C(=O)NC(C)CCCNC(=O)CC2CC(N(C)C)C2)ccnc(CN(C)C)c1 C12(CNC(=O)CCc3cc(Cl)cs3)CC1CN(C(=O)CC1CCOC1=O)C2 C1(C(N(CCNC(C2CCC(=O)C2)=O)C2CC2)=O)CCc2ncc(Br)n2C1 c1(OC)noc(C)c1C(N1CCCC(CCNC(=O)CC2CCCN2C)C1)=O c1(CNC(C=CC(CC)C)=O)csc(NC(=O)CC2COC(=O)C2)c1 CCCC(C(=O)NCc1ccc(CN(C(=O)CC2C=CCC2)C)cc1)NC(N)=O N1(C(C2CN(C(C)=O)C2)=O)CC2CCN(C(C3CC(C#N)C3)=O)C2C1 c1(C(N2CCC(C(C)(C)NC(CC(CCC)C)=O)C2)=O)ccc2nc(C)cn2c1 C1(C(=O)NC2CCN(CCC)C2)CC2CN(C(C3CCCC(OC)C3)=O)CC2C1 c1(C(=O)NCCC2(NC(CN(CC)CC)=O)CCC2)cc(CO)oc1C C1(NC(C(C(C)(C)C)NC(C2N(CC)CCOC2)=O)=O)CN2CCC1(C)CC2 N1(C(CC2(CC(=O)OC)CC2)=O)CC2CC(NC(=O)C3=NNC(C(F)(F)F)C3)C2C1 N1(CC)CC2(NCCc3nc(COC)c(Br)s3)CC1(c1ncno1)C2.CCOC N1(C(CCn2c(C)ccc2C)=O)CCC(CNC(=O)CC(C)C2CC2)CC1C C1(F)(C(N(C)CC2OCCN(C(C3CC(CC)C3)=O)C2)=O)CCS(=O)(=O)C1 C1(C(=O)NCC2(C(N)=O)CC2)C2CC1N(C(=O)COC(F)(F)F)C2 N1(C(CCCOCCC)=O)CCCC(OCC)C1.N12CCC(O)C1C2=O c1(OC)cc(N)ccc1C(=O)NCC1CCC(CNC(=O)C(C)CC(F)F)CC1 N1(C(C)=O)CCN2CCOCC2C1.c1(N2CCCCC2)ncnc2cc(C)[nH]c12 N(C(=NCc1ccc(F)cc1CC)NC1CCOc2cc(OC)ccc21)C(CC)C c1(NC(C(C)Cc2ccncc2)=O)ccc2nnc(C(F)F)n2c1 N1(C(=O)NCC(C2(CCOC)CC2)C)CCCC(CN(C)C)CC1 C1(NC(c2nc(COC)sc2)=O)CC2CC(NC(=O)CC(C)SC)CC2C1 N1(C(Cn2cnc(C(N)=O)n2)=O)CC(C2CN(C(c3cscc3F)=O)C2)C1 Cc1cnc(C(=O)NC(C2CCCCC2)CNC(=O)Cn2ccnc2C)c(F)c1 n1(CC(=O)NCC2C(C(=O)NC3CC(C(C)(C)O)C3)CCO2)cccnc1=O C1(COC)(NC(C2CCOC2C)=O)CCN(C(C2(N=[N+]=[N-])CC2)=O)CC1 N1(C(CCN(CC)CC)=O)C2CCC1C(NC(c1c(F)cncc1Br)=O)C2 N1(C(C(C)NC=O)=O)CC2CN(C(c3cn(C4CCC4O)nn3)=O)CC2C1 N1(C(C(C)C(C)(C)C)=O)CC2CCN(C(c3c[nH]cc(F)c3=O)=O)CC2C1 c1(C(C)C)cc(Nc2ncnc3c2cnn3C)cc(F)c1F c1(CC(=O)NC(CNC(C2C(CCC)C2)=O)(C)CO)sc(C)cc1Br n1(C(COC)C)nc(C(C)C)nc1C1CC1c1cccc(OC)c1 C(=O)(C1CCc2nccn21)NCC1C(CC)CCN1C(C1CC(C)(C)CO1)=O N1(CCc2ccc(C(=O)O)cn2)C(=O)c2ccccc2C1=O.C1(S)CC1C(F)(F)F c1(C(N(C(C)CNC(c2cnc(OC)s2)=O)CC)=O)cn2cc(Cl)cc(Cl)c2n1 C1(CNC(c2ccn(C)n2)=O)CCCCCN1C(=O)COCC1CCCC1 C1(C(=O)NC(C(CC)C)CO)C2CC(O)C(C2)N1C(c1ccsc1C#N)=O CC1CN(C(C2CC3(C2)CC(C)(C)C3)=O)CC(C)C1NC(=O)C1=COCCC1 C(=O)(C(C)(C)CNC(C1(C#N)CC(C)C1)=O)N1CC(OCC#C)C1 c1(C(=O)NCC(CC=C)NC(c2n[nH]cc2Cl)=O)ccc(C(C)(F)F)nc1O CC1=C(C(=O)Nc2ccccc2)C(c2ncoc2C(C)C)NC(=S)N1CCF c1(C(=O)NC2CCC(NC(c3c(C)nn(C)c3)=O)C2)c[nH]cc(F)c1=O C(CCNC(=O)CCCOCn1cc(Cc2ccc(N)cc2)nn1)(C(C)C)OC C1C(C(C)C)O1.C1(=O)CC(C)N1.C1(C(N(CC)CC)=O)CC12CC2 N1(C(C(C)N(C(c2c(CC)nn[nH]2)=O)C2CC2)=O)CCC(C)OC(C)C1 N1(C(CCCC)=O)CCCC12CCCN(C(=O)C(F)C(C)(C)O)C2 Cn1ncc2c(C(N3C4CCC3CC(NCc3cccnc3Br)C4)=O)cccc12 C(C(C)(C)CCNC(C1CCOC1C1CC1)=O)NC(CCNC(C)=O)=O N1(C(CN(C(C(CC)CCOC)=O)CCOC)=O)CCc2nncn2CC1 c1(SCC)ccc(C(=O)NCC2(F)CCC(NC(C3(F)CCCOC3)=O)C2)cc1 N1(C(C2OCCN(CC)C2)=O)CCCOC(CCNC(C2CCCC2)=O)C1 CCC(C)(CC)CN=c1nc2scnc2c(NCC2(C)CCCCO2)[nH]1 N1(C(C(CC)F)=O)CCC(CCCCCNC(C2CCCN2N=O)=O)CC1 C1(C(N(CCNC(C2C=CCCC2)=O)CC)=O)CC2CCC(C1)O2 C(=O)(C1=CC2(CCOC2)C1)NCC(CC)(CC)C(=O)NC1CN(C)CCC1O N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)CC(C)C2CCCCC2)CC(CO)C1 C1(NC(C2N(CC)CC2)=O)CCCC2CN(C(c3cn(CC)nc3C)=O)CC12 c1(C(=O)NC2(CCNC(C3C(CC)C3)=O)CC2)cc(C(=O)OC)ccc1[N+](=O)[O-] C1(NC(C2N(C(C)=O)CCCC2)=O)CN(C(=O)Cc2ccns2)CC(C)(C)C1 c1(C(=O)NCC(CN(C)C(C2COCCOC2)=O)O)cn2c(n1)CCC2 CCCCC(C)(F)C(=O)N1CCCC(CN(C)C(c2cc(C)nc(O)c2)=O)C1 Cc1cc(C(N2CC(O)C(C3CC3)C2)=O)cc2ccsc12 O=C(NNc1ncc(I)cn1)C1CCCN(C(C2CCCO2)=O)C1 c1(NC2CC(NC(c3nc(CC)oc3)=O)C2(C)C)cc2nncn2c(C)n1 c1(OC)ccccc1C1CNCCN1C(N1CCC(C(C)(C)O)C1)=O C1(OC)CCC2(C(=O)N(CC(=O)NCC3CC3)Cc3ccoc3)CC12 N1(C(c2c(C)n(C3CC3)nc2)=O)CCC(CNC(=O)C(F)CC2CC2)C(F)(F)C1 c1(C(C(=O)NCCOC)N(C)CC2CC2)nncn1C CC1CCCC(C)N1C(C1CCN(C(c2coc(C(C)(C)C)n2)=O)C1(C)C)=O C1(C(=O)NCC(C)C2CC2)(NC(Cc2c(C)occ2)=O)CCN(C)C1 Cc1ncc(C(=O)NCC2(C(C)(C)O)CN(C(C3(C)CC3(F)F)=O)C2)s1 c1(C(N2C(C)CN(C(C3C4CN(C)CC34)=O)C(C)C2)=O)cccc2nc(O)oc12 N1(C(c2c(N)ccc(C)c2)=O)C(C)CC2CN(C(C3(C)CC3(Cl)Cl)=O)CC12 C1(CN(C)C(C2(NC(=O)C=CC3CCOC3)CCSC2)=O)CCCC2CC12 C(=O)(CCCCCNC(C1C2COCC12)=O)N1CC(=CCC)C1 C1(NC(C(=O)NC(C)C)=O)CCN(C(c2cc3nnn(C)c3s2)=O)CC(O)C1 CC#CCCCC(=O)N1CC(C(N)=O)(CNC(=O)C(C)(F)F)C1 C1(NC(=O)C(F)n2ccnc2)CCN(C(C2CC2(Cl)Cl)=O)CC1 C1(C)(C(=O)NCCC2N(C(Cc3n(C)nnc3)=O)CCC2)CCCC(F)(F)C1 c1(C(=O)NC(CNC(C(C)=C(C)C)=O)CO)cc(F)ccc1Br c1(C(N(CCCCNC(C2C(CC)CCCC2)=O)C)=O)ccc(Cl)c(O)c1 CCCCCC(O)C(=O)NC(C)CNC(C1(Cc2cnn[nH]2)CCCC1)=O C1(NC(C2(c3n(CCC(N4CC(C)C4)=O)nnn3)CC(O)C2)=O)(CO)CCCCC1C CC1(C(=O)NC2CC(C)(NC(=O)Cc3ccc(CO)cc3)C2)CC(C2CC2)=NO1 C1(C(N(C(C(N2CCC(CCO)C2)=O)C2CC2)C)=O)C2(CC2)C12CC2 N1(C(CCc2onc(C)n2)=O)CCCC(C)C1CCNC(=O)COC1CCC1 CC1C(NC(=O)C(N2CCCC2=O)C2CC2)CCCN1C(=O)CCC#N C1(C(=O)NC(C)C(CO)NC(C2COCCO2)=O)(COC)CCCCO1 C(=O)(CC(C)C(=O)c1ccccc1)NC(CNC(c1c(OC)ccs1)=O)C C1(C(=O)OC)CC(NCc2cccc(OCc3cccnc3)c2)CCO1 CCCCC(C)C(=O)NCC(O)CNC(=O)C(C)Cc1c(C)noc1C Cc1ccc(C(N2CCN(C(=O)Cc3sc(O)nc3O)C3CC23)=O)c(=O)n1C S(=O)(=O)(c1nc(N2CCCC(C(F)(F)F)CC2)ccc1Br)NCC(C)(C)C1CC1 c1(CC)c(C(=O)NCC23CC(NC(=O)C=CCO)(CCO2)C3)sc2ccccc12 N1(C(c2cnn(CC(F)F)c2)C(=O)NCCOC)CCC2(CCOCC2)C1 C1(CCNC(C2CCC(C)O2)=O)CN(c2ncnc3c2CCO3)CCS1(=O)=O c1(NC23C(CN(C(=O)Nc4cnnn4-c4ccccc4Cl)C2)C3)nccc(Br)c1O C(=O)(CC(O)CC(C)(C)C)N1CCC(CC(C)C(c2ccccc2Br)=O)CC1 N12CCCC(C)(C1)NC2=O.c1(C(=O)NCCCCOC)ccc(N(C)C)cc1 C1(CCOC(N2CC(CC(=O)OC(C)(C)C)(OC)C2)=O)CCc2ncnn2C1 CN1CCN(C2CN(C(=O)CCn3cc(COCc4nccs4)nn3)C2)CC1 CC(C)C(N=[N+]=[N-])C(=O)NC1CC1CNC(C1CCOC1c1ccnn1C)=O C1(NC(=O)C(Cl)=CCl)CCCCC12CCN(C(=O)Cn1cccn1)C2 C1(CNC(Cc2cc(C)cc(F)c2)=O)CCN(C(=O)Cc2ccon2)CC1(F)F N1(C(CCC)=O)CCC(C2CCCN(C(c3nc[nH]c3C(C)(C)C)=O)C2)C1 CCC(CC(=O)NCCSC)NC(c1ccnnc1C)=O CC1CC(C(N2CC(C3(NC(=O)C#CC4CC4)CC3)C2)=O)CCS1(=O)=O C1(C(=O)NC2(C)CC(NC(=O)C3=CCCC3)C2)CCCC(F)(F)C1 N1(C(C(CC)(C#N)CC)=O)CCC2(C=C(C(=O)NC(C)CCC3CCCC3)C2)C1 C1(C(N2CCC(OCCNC(=O)CCC3OCCO3)C2)=O)CCC2(CCC2)CO1 C1(C(N2CC(CNC(Cc3nc(CCCC)sc3)=O)C2)=O)CC(=O)N(COC)C1 N1(C(C(CCC)CC)=O)CCCC(C)(C)C1CNC(C1(C(F)F)CCCCC1)=O c1(C(=O)NC2CC3N(C(C(CCOC)C)=O)C(CC3)C2)ccc2oc(O)nc2c1 N1(CCC)C(=O)CCC1C(=O)N(C(C)CNC(C1CC(C#N)C1)=O)C C1(CN(C)C(c2cocc2Br)=O)CCN(C(c2scnc2C2CC2)=O)C1 S(=O)(=O)(CC(=O)NCC1CN(C(=O)COC2CCOCC2)C2CC12)N(C)C c1(C(N)=O)ccc(C(=O)NCC2(F)CC(NC(=O)CSCC(F)(F)F)C2)cn1 c1(C(N(CCC)CCNC(=O)C(C)CC)=O)noc(C)c1I c1(OC)coc(CN(C2CCCN(C(=O)CCN3CCC3)C2)C)cc1=O CCC(C(=O)NCC1C(C)CCN1C(=O)C(c1nncs1)N(C)C(C)=O)C(C)O C(=O)(C(C)(C)COCC)N(CCC)CCNC(C1CC=CCC1)=O c1(C(N2CCN(C(=O)CC3CC3)CC2CC2CC2)=O)cc2cccnn2n1 c1(N2C(C)(CNC(C3CCC(OC)CC3)=O)CCC2)cc(=O)n(C(C)C)c(O)n1 N1(C(C2=CCC(NC(C3(C)CCCC3)=O)C2)=O)CCN2CCC1CC2 N1(C(C(C)O)=O)CCCC2C1CCN2C(c1cccc(NC(N)=O)c1)=O C1(C(=O)NCC(CNC(COCCC)=O)C)CCc2nccn2CC1 C1(NC(C(C(CC)C)C)=O)CC2(CCC(NC(C3CC(=O)CCO3)=O)CC2)C1 N1(C(C2C(=C)C2)=O)CCCC(N(CCO)C(c2cncc(O)c2)=O)C1 n1(CC(N2CC(N(C(CCCC)=O)C)C(O)C2)=O)sc2ccccc2c1=O N(C(=NCCCCl)NCC(O)C1CC1)CC1CN(C(CN(C)C)=O)C1 C1(CNC(C2OCCO2)=O)CC(F)CN1C(c1ccnc(N2CCOCC2)n1)=O N1(C(C(C)NS(CC)(=O)=O)=O)CCCN(C(c2ccc(N)cc2F)=O)CC1C Cc1ccc(C=CC(=O)NCC2(C(N)=O)CN(C(C34CC(C3)C4)=O)C2)cc1Cl C1(CNC(c2cc(C)on2)=O)CCN(C(=O)C(c2ccc(C(C)C)cc2)(C)C)CC1 N1(C(C(C(C=C)C)C)=O)CCC2(CC1)CN(C(=O)CC1COC3CC1C3)CCO2 N1(C(C)=O)CC2CCC1C(N=c1[nH]c(=NCCC3CC3)[nH]c3ccccc13)C2 C1(C(=O)NCCOc2ccc(Cl)c(Br)c2)CC2(CCN(C(c3ccns3)=O)CC2)C1 c1(CC)ccc(CC(N2CC3(CCC3NC(=O)C(C)SC)C2)=O)c(Cl)c1 N1(C(Cc2cn(CC)nc2)=O)CCCC(C)(CNC(=O)C(SC)SC)C1 c1(N2CC=CC(NC(CC(=C)C)=O)C2)c(F)cc([N+](=O)[O-])cc1F N1(C(c2c(CCC)nco2)=O)CC(NC(c2ccncc2O)=O)C(C2CC2)C1 c1(CCC(=O)NCC(CN(C(C(C(C)C)C)=O)C)C)ccc2c(c1)CCCO2 C(CC(C)C(=O)N1CC(CCNC(c2cnsn2)=O)(OC)C1)=CCC C1(C(CNC(C(C)(C)C)=O)F)CCN(C(c2cc(-c3ccccn3)c[nH]2)=O)CC1 C(=O)(C1=CC2(CCOC2)C1)N1C(CNC(CCC(=C)Br)=O)COC(C)(C)C1 S(=O)(=O)(c1nc(N2CCC(C)(F)CC2)ccc1Br)NC(C)COCC1CC1 O=C(N=c1cc(-c2cccc(C(F)(F)F)c2)[nH][nH]1)c1cocn1.N1CCC2CC2C1 C(=O)(C1=CCC(F)(F)CC1)NC1CCC(CNC(C2=C(C)OCC2)=O)C1 C1(NC(=O)COC2CCOCC2)COCCN(C(=O)CC2CC(F)(F)C2)C1 C1(CC(=O)NC(C)CCNc2nccc(-n3ccnc3)n2)(COC)CCOCC1 CCCC(C)CC(=O)N1CC(OCCNC(C23CCC(CC2)C3)=O)C1 N1(C(=O)Cc2ccsc2)CCCN(Cc2cc(Cl)cc(F)c2F)C(CO)C1 c1(CC)nc(C(=O)Nc2nc(CC(=O)NCCN3CCOCC3)cs2)co1 c1(CNC(C)COc2ccc(F)cc2)c(-n2cccn2)cccc1F CCCCS(=O)(=O)N1CCCC(CNC(c2cnc(-n3cncn3)nc2)=O)C1 C1(C(=O)NC(CN(C(c2ccsc2OC)=O)CC)C)CN2CCCN1CC2 C1(NCc2c(C)ccc(C)c2)CC2(C1)NC(=O)NC2=O C1(c2cn(C)nc2)CC(N(CCC(C)(C)CO)CCCO)CCS1.n12cc-1nn2 CC(C)(C)C1CC(=O)N1.C1(C)(NC(C2CCC3CC3C2)=O)CCNC1=O c1(NC2C(O)CCN(C)C2)ncc(F)c2c(N)cccc12 C1(C(=O)NC2(C)CC(NC(C(c3ccc(Cl)cc3)C)=O)C2)CC2C=CC1CCC2 C12CC=CC(C1)n1cc(nn1)COC2=O.C(=O)(C(F)(F)F)OC.C12CCN1C2=O c1(C(=O)NC(C(C)C)CNC(=O)CN2CCC(C)(O)C2)cccc(F)c1Br C(=O)(C1=C(C2CCC2)N(CC)C(=S)NC1c1ncsc1C(C)C)OCC c1(C(=O)NC(C2CCN(C(=O)CSc3nncn3C)C2)C)ccn2ccnc2n1 c1(C(=O)NCCN(C(Cc2c(C)occ2)=O)CC(C)O)c[nH]c(C#N)c1 c1(C(N(C)CCN(C)C(C2CC(C)(F)C2)=O)=O)ccc(-c2cnnn2C)cc1 n1(CC)nccc1S(=O)(=O)NC(C1CCS(=O)(=O)N1)(C)C c1(C(=O)OC)cc(Cl)cc(NC(=O)Cc2cc(C)cc(C#N)c2)c1Cl CCCC(C(=O)NCc1nc(C(=O)N(CC(C2CCC2)OC)CC)co1)OC N#CC1(C(=O)OCCSCCC(F)(F)CO)CCCOC1 c1(C(N(CC(CNC(C(C)OCCCC)=O)C)C)=O)c(C)nn(C)c1OC C1(CCC)(NC(CCCC=C)=O)CCCN(C(=O)C(CC)n2ccnc2)C1 C(=O)(CCCC(F)(F)CO)N1CC2C(CNC(c3cn(CC(C)C)nc3)=O)C2C1 CC1(C)CN(C(c2ccc(C3CC3)o2)C(=O)N(CC(F)F)CCO)C1c1ccncc1 n1(C(C)C)cc(C(N2CC(O)(CN(C(=O)C(C)(C)c3cccnc3)C)C2)=O)cn1 Cc1ccsc1C=CC(=O)OCCOC1(OCc2ccccc2)CCC1 C#CCCCC(C)C(=O)N1CCOC(C(N2CCN(C(C)CC)CC2)=O)C1 C1(COC)(CNC(C2CCCC2O)=O)CN(C(=O)C2CC2)C1 C1(CNC(CC2CN(C)C2)=O)CCC2(CCN(C(c3ccsc3SC)=O)CC2)O1 C(=O)(CCCCc1ccc(Cl)cc1)N(C(C)CNC(C1CC1CN(C)C)=O)C C1(C(=O)NCC(=O)NCc2cn[nH]c2)CCCCN1C(=O)C(O)CN1CCCC1 c1(OCCS(CC=C)(=O)=O)ccc([N+](=O)[O-])c(O)c1 C(C(C(=O)N(CCNC(=O)CC(C)CC)CCOCCO)C(C)(C)C)OCC=C N1(C(CCCCCC)=O)CCC2(CC2)CC1C(=O)NC1CCCOC12CCC2 N1(C(C2C(C(N)=O)CC2)=O)CC2C(CN(C(c3cnsc3)=O)C3CC3)C2C1 c1(C(=O)NC2(CCCOCC)CC2)ccc(C(C)=O)o1.C12CCC1C(=O)N2 C(C)(C(=O)NC1CCC(NC(C2CC3CCC2CC3)=O)C1)(C(C)C)NC(C)=O CC(CCCNC(c1ccncc1)=O)NC(=O)CNC(=O)CC1CCCCO1 N1(C(c2c(C)cc[nH]2)=O)CC2CCCC2(NC(c2c(OC(C)C)c[nH]c2C)=O)C1 C12(C(N(CCC)CCNC(C3C(C)(C)C3(C)C)=O)=O)CCCC1C2(F)F C=CCC(CC=C)NC(=O)CC1CCCC1NC(c1occc1C(C)C)=O N1(C(C2C(NC(c3cn(C4CC4)nn3)=O)CCC2)=O)CCN(C2CC2)C(=O)C1 CCCN=C(NCC1CC2(C1)CC21CCC1)N1CCN(CC(C)C)CC1 N1(C(C)C)N=C(C(=O)NC2(C)CC(NC(=O)C3=CC4CCCCC34)C2)CCC1=O N1(C(CCSC)=O)CCCC1C(c1ccon1)N(C(=O)CC1CC1)C C(C(=O)NOCc1cccnc1)(c1ccnn1C)NC(C(C)c1ccsc1)=O c1(C(=O)NCC(O)CO)ccc2c(c1)CCN(C(c1c(F)cccc1Br)=O)C2 N1(C(c2c(C)n(C)cn2)=O)CCN(C(=O)CC2CC2C2CC2)CC1C1CCCC1 c1(C(N2CCOC3CCCC23)=O)ccnc2c1CCC2.c12ccccc1NC2=O N1(C(c2sc(Br)nc2Cl)C(=O)Nc2ccc(F)cc2)CCOC2(CCC2)CC1 CCC(C)(C(=O)NC1CCCN(C(c2cc(C)c(C)[nH]2)=O)CC1)C(N)=O c1(C(N(C2CCOCC2)CC#C)=O)cnc(CNC(=O)CC2COC(=O)C2)nc1 c1(OC)ccc(C(C)NC2CN(C(N)=O)CC2NC(=O)OC(C)(C)C)c(F)c1 C1(CNC(C2N(C(Cc3nnc(C)o3)=O)CC(O)C2)=O)CCCCC1(F)F c1(C(N2C(CNC(c3ccccc3C(F)(F)F)=O)CC2)=O)nnc2ccccn12 C12(C(=O)NC3CC(C)(CNC(C4(C)CCN(C)CC4)=O)C3)CC=CCN1CCC2 Cc1nn(C)cc1C1=NOC(C(N2CC3CC(O)C2C3C(=O)O)=O)C1 C1(NC(C(CC)OC2CCCC2)=O)CCCCC1NC(c1ccnnc1)=O C(C(C(=O)N1CCC(C(N2CCC(CC(C)(C)C)CC2)=O)O1)N(C)C)N(C)C c1(OC)nc(C(=O)NCC2CCCC2NC(=O)CC2CCCC2O)co1 N1(C(CN(CC(C)(C)C)C)=O)CCC2CC2(C(N2CCCCC(C)(C)C2)=O)CC1 C1(NC(C(C)OCCC=C)=O)CN(C(c2nc[nH]c2C(F)(F)F)=O)CC12CC2 N1(C(c2nc(C)n(-c3ccccc3)n2)=O)CCCC(CCO)CC1 C1(CC)CCN(C(c2cnnc(O)c2)=O)C1C(=O)NCCN1CCCOC1=O C1(CNC(C(C)OCC(C)C)=O)CC2CCC1N2c1nnn(C)n1 C1(N(C(=O)CC2C3CN(C(=O)CCCC#N)CC23)C)C2CCCCCC12 c1(CC)cc(C)c(C(=O)NC2CCCC2C(=O)NC2(CSC)CC2)o1 C1(C(N(CC(C)(C)NC(c2cc(C#N)no2)=O)C)=O)CCc2cncn2C1 CC1C(C)N(C(=O)COCCNC(=O)CS(C)(=O)=O)CCN1C C1(c2cn(C)nc2)CC(NCCS(=O)(=O)CC2CC2)CCO1 C12(NC(c3ccncc3)=O)CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC1C2 c1(C(=O)NCCC2CCN(C(C(COC)(F)F)=O)C2)cc2c(C)nn(C)c2s1 CC1(C)CCC(C(N2CCC2CNC(c2ccc(Oc3ccccc3)o2)=O)=O)O1 c1(C(=O)NC(CC(C)NC(C2(SC)CCC2)=O)C)snc(C)c1N C1(NC(C=C(CC)C)=O)C2CC1CN(C(=O)Cc1nnc(C(F)F)o1)C2 C1(CN(C(c2c(NC)nccc2)=O)C)CN(C(C2CC3CCC2O3)=O)CC12CC2 C1(C(=O)NCCCNC(=O)CCC2CCOC2)CCCN(CC(F)F)C1 C1(C(C)C)N(C(=O)C(n2cc(CCNS(C)(=O)=O)nn2)C)CC12CCC2 CCC(CCCO)NC(C1C2CC1N(C(C1(OC)CCC(C)C1)=O)C2)=O C1(C(N2C(C(=O)O)CC(Cl)C2)=O)Cc2ccccc2NC1=O CC(C)CCC(=O)NCC1(F)CC(CNC(c2conc2C(F)(F)F)=O)C1 c1(CCCC(=O)Nc2cccc(NC(CCC(C)SC)=O)c2)ccc(C)c(C)c1 N1(C(CC(CC)C)=O)CCC2CCCC12C(=O)NC1CC2(CCCCO2)C1 c1(SC)cccc(F)c1C(=O)NC1CCN(C(c2nncn2C2CC2)=O)CC1C C1(C(=O)NCC2(C(C)(C)O)CN(C(CSC)=O)C2)C(C)OC(C)C1C C(C(C(=O)N1CCOC2(C1)CN(C(c1cncc(CO)c1)=O)C2)C(F)(F)F)OC N1(CC#C)CCN(C(=O)C(C)C(C)NC(c2occc2COC)=O)CC1=O C(=O)(CC(C)(C)C(F)F)N1C(C)CC(CC(N2CC3CCC3(CO)C2)=O)C1 C1(NC(CCS(=O)(=O)NC)=O)CC2CC(C1)N(C(c1cc(C)c(C)s1)=O)C2 C12(CC(=O)NCC(C)(C)NC(c3cc(Br)n[nH]3)=O)CCCC1C2 C(=O)(C(CCC(=O)O)C1CCCCC1)N1CCC(N(C(C)(C)C)C)C1 C=CCCC(C)C(C(=O)NCCCF)N(C(C)(C)CC)C C1(C(=O)NC(C)(CNC(C2(C(F)(F)F)CC(O)C2)=O)C2CC2)OCC2CCCC12 N(C1c2ccccc2OCC1O)Cc1c(C)nn(CC(C)C)c1C c1(C(N2C(C)(C)CC(NC(C3CCCC4(CC4)C3)=O)C2)=O)ccc2c(c1)COC2 CC1C(NC(=O)CS(N)(=O)=O)CC2CCC1N2C(=O)COCc1ccccc1 C(=O)(C1CCc2c[nH]nc21)NCC1CCC(NC(c2c(OC)ccc(C)n2)=O)C1 C(=O)(C1=C(Cl)CCC1)N(C1CCN(C(C2CCC(NC(CC)=O)C2)=O)CC1)CC c1(C(=O)NC2(C(C)C)CCNCC2)ccc2c(c1)ncn2C C(=O)(C(F)C(C)CNC(c1cc[nH]c1)=O)N1CC(C#CC)C1 C1(CNC(C=CC)=O)(NC(c2cc(-c3ccccc3)nn2C)=O)CCCCC1C C1(C(N2CCN(C(C34C(C)OC(C)(C3)C4)=O)CC2CO)=O)CCc2nn[nH]c2C1 C(=O)(C(=O)C(C)CC)NCc1ccc(CNC(CCC#C)=O)cc1 Cc1ccc(C=CC(=O)NCC2COCCN2C(C2CCCN2C(C)C)=O)nc1 c1(C(N2C(C)CC(NC(=O)CC3CCC(=O)N3)CC2)=O)nccc2ccccc12 n1(CC(N2CCC(NC(CCC)=O)C2(C)C)=O)ccc2cc(F)ccc12 C1(=O)CCCN(C)C(=O)C2(CCC2)N1.C1(CC(C)C)(NC(C)=O)CC1 C1(C(NOCC(C)(C)C)=O)CCCCCC1NC(=O)CCC1CC1(F)F C1(CC(=O)NCC2(NC(c3ccoc3Cl)=O)CC2)CCC(O)C1 C1(CC(C)C)(C(=O)NCC(CC)NC(=O)CC2CCCO2)CCCCC1 C1(C(=O)NC2CCC(CNC(=O)CC(C)n3cccn3)CC2)(CC)CNC(=O)C1 C1(CC)(CC)CN(N2CC(OC)C(C(C)C)C2)CCS1=O C1(C(C)C)CN(C(=O)C(C(C)O)NC(C2CC(=O)NC(=O)N2)=O)CC(=O)N1 Cc1ccc(C(=O)NCC2CC2CNC(=O)CCC(C)C)c([N+](=O)[O-])c1 C1(c2n(CCOC)nc(C(C)OC)n2)CCc2n[nH]c(C)c2C1 N1(C(c2ccnc(OC)n2)=O)CC(NC(C2CC(OC)C2)=O)C2CCCC12 CCC(C)(COC)C(=O)NCC(C)(C1CC1)NC(=O)CCCCCN(C)C c1(C(=O)NC2C3CN(C(CNC(CNC(C)=O)=O)=O)C2C3)ccccc1S(C)=O CC(C)(F)C(C)(F)C(=O)NC(C)CC(=O)NCC(F)Cl C1(NC(C(C)NC(COC)=O)=O)CCC(C(=O)NC2CCC(C)CC2)CC1 C(=O)(CCCCCC1CC1)N1CC2C(NC(C(C(C)C)SCC)=O)(C2)C1 c1(C(=O)NCC(CNC(c2cccc(C(C)C)n2)=O)F)cnc(O)c([N+](=O)[O-])c1 C12(CNC(C(C)OCC)=O)CCCCCC1N(C(=O)CN1CCCS1(=O)=O)CC2 c1(C(C)NC(C(C2CN(C(C(CSC)OC)=O)C2)O)=O)ccccc1F c1(C(=O)NC2CC(CCC(N)=O)C2)cnn(CCNC(C2CC2F)=O)c1 C1(C(=O)NC2(CCCC)CC2)CCN(C(c2cccc(COC)c2)=O)CC1C c1(C(=O)NCCC2CCN(C(c3c(C)ocn3)=O)C2)ccc(=O)n(CC(C)O)c1 N1(C(C2C(C(=O)NCCNCCO)C2)=O)CCc2cc(F)ccc2C1 C(C(C)(O)CC(=O)N(C1CCCN(C(C2CC(O)(C(F)(F)F)C2)=O)C1)CC)OC C(CCC(C)C(=O)NCC1(F)CCN(C(c2cc(O)ccc2O)=O)C1)OC N1(C(CC(C=C)(C)C)=O)CCC2CN(C(c3nnn(C)c3C(F)F)=O)CCC2C1 Cc1nnc2c(C(=O)NC3CC(NC(=O)Cn4cccn4)C34CCC4)nccn12 C(=O)(CCC(=O)NC1CC2(C1)CC2NC(=O)OC)NCCC.C1(=O)CC2CC2N1 C(=O)(C(F)C(C)(F)F)NC1(C(=O)NCC(COC)(C)CO)CC(O)C1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(=O)C(O)C(C)C)CC1O N1(C(c2cnc(C)n2C)=O)CCC(CO)CC1C(=O)N(C1CC1(C)C)C C1(C2CN(C(=O)CC3(O)CCOC3)C2)(NC(=O)CC2CCCOCC2)CC1 N1(C(c2c(CC)onc2)=O)CCC(C2(NC(=O)CC3(C#N)CCC3)CCC2)CC1 C1(NC(C2C(C)(C)COC2)=O)CC(CNC(c2cnccc2Cl)=O)C12CCC2 C(CC(=O)NOC(CO)C(C)C)N(C(CNC(C)=O)=O)C1CC1 N1(C(C2CC2CF)=O)CCCC2(CCCN2NC(C2CN(C(N(C)C)=O)C2)=O)C1 C1(C(=O)NC(C)CCNC(c2ncccn2)=O)(CO)CC(C)(C)C1 c1(CC)ccc(F)cc1C(N1CCCC1CNC(C1CCCC12CC2)=O)=O C1(C(=O)NCC(CCNC(C2(N3CCCC3)CC2)=O)OC)CC2C(C1)C2(F)F c1(NC2CC(NC(C(c3cccc(Cl)c3)N(C)C)=O)C2)nc2ccc(N)cc2s1 C1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)CCC2)COc2cc(F)ccc2O1 C1(NC(c2nc(C)sc2C)=O)CCCC(C(=O)NCC2CC2CO)CC1 C1(N(C(COCCCCC)=O)C)CC2CCC(C1)N2c1nnco1 N1(C(CC2(OCC)CC2)=O)CCC(C=CC(=O)NC(C)Cc2ncn(C)n2)CC1 N1(C(C2CC(CC)(CC)C2)=O)CCOCC1CN(C(=O)C(C)C1CCOC1)C c1(C(=O)NCC(CNC(c2cnnc(O)c2)=O)F)ccc(-c2ccco2)nc1O N1(C(CN2C(C)CCC2)=O)CC2CC(NC(=O)C=Cc3cccs3)C(C2)C1 c1(C(N(C(C)CNC(=O)C=NOC)CC)=O)ccc(OC)cc1OC Cc1nc(-c2ccc(Cl)cc2)sc1NC(=O)C(=O)NC1CCC(C)C1 c1(NCC2CC(NC(C3C(C)OCC3)=O)C2(C)C)ncc(C#N)cc1F S(=O)(=O)(c1cccc(F)c1)NCC(=O)N(CCNC(c1c(C)ncnc1)=O)C N1(C(C(C)CN(C)C(C2(F)CC2)=O)=O)CC(O)(C2CC2)C1 c1(C(=O)NC2(CC=C)CN(C(c3cc[nH]c3)=O)C2)csc2nccn12 Cn1ccc(C(=O)N(C2(C(=O)NC3CC(C(C)(C)C)C3)CCC2)C2CC2)n1 C(=O)(C(C(C)(C)C)C1CCC1)N1CCN(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC1 N1(C(C(C)=C(C)C)=O)CC2(CCC2NC(C2CCCN2C(c2cccs2)=O)=O)C1 C(=O)(CCCC(F)(F)F)N(C1CCCCN(C(c2ccc(C(F)F)o2)=O)C1)C C(=O)(C(CNC(=O)CC1COCC1O)C(C)C)NCC(C#C)CC1CC1 N1(C(c2ccc(CC(C)C)cc2)=O)CC2(CC2)CC1C(=O)NCc1ncccn1 CCCCCCCC(=O)NCc1cnc(CC)s1 N1(C(C2(C=C)CCC2)=O)CC2CC(NC(C3(C(F)F)CC3)=O)CC2C1 S(=O)(=O)(c1cccc(Cl)c1)NCC(N1CC(NC(c2n(C)c(Cl)c(Cl)c2)=O)C1)=O c1(OC)ccc2c(C(N3CCN(C(=O)C=CS(C)=O)CC3C(C)C)=O)csc2c1 C(=O)(CCC=C(C)C)N(CCC(=O)N(CCCC)CC)C1CCCC1 C1(c2ccccc2)(C(=O)NC(C(C)C)CNC(=O)C(C)CF)CC(F)(F)C1 C1(C(=O)N(CCCCO)C)(COC)C=CCN1C(=O)CC1CCCSC1 N1(C(C(C)CC(F)(F)F)=O)CC2CN(C(=O)CCCCc3cnc[nH]3)CC2(C)C1 c1(C(=O)NC(CNC(c2c(C)scc2)=O)C(C)(C)C)ccc2c(c1)OCC2 C12(C(=O)NCC(C)OCC=C)CC(CN(C(C3(C#N)CC3C)=O)C1)C2 C(=O)(C1CCc2c[nH]nc21)NCC(C)(C)OCC(=O)NC1CC2CCC1C2 c1(C(N2C(CNC(CN(CCC#C)C)=O)C=CC2)=O)cc(Cl)cc(Cl)c1Cl C1(CNC(C(C)(C)n2cc(Br)cn2)=O)CCN(C(=O)CC(F)F)CC1O c1(C(=O)NC2CC(O)(CNC(CS(N)(=O)=O)=O)C2)ccc([N+](=O)[O-])cc1 Cc1nc2cc(C(=O)NC3CCCCC3NC(=O)CCCS(N)(=O)=O)cnc2s1 O=C(NNC(=O)c1cccc(I)c1)C(=O)Nc1cnn(-c2ccccc2)c1 CC1(C)CCC(c2nc(-c3sccc3S(N)(=O)=O)no2)CC1 O=S(=O)(c1cccnc1N1CCN2CC(F)CC2C1)NCC1CCNC(=O)C1 C(=O)(C1SCCc2ccccc21)N1CCN(C(C(C(C)C)OC)=O)CC(C)(C)C1 CN(C1c2cc(Cl)cc(Cl)c2CC1O)C(=O)NCc1ccoc1 C1(OCCNC(CC=CC)=O)CCN(C(=O)C(F)C2CC2)CC1 Cc1c(Br)ccc(F)c1C(=O)NC(C)CNC(c1cc(F)c(F)cc1N)=O c1(CC)ccc(N)c(C(N2CCCN(C(c3nn(C)nc3Br)=O)CC2)=O)c1 C1(C(F)(F)F)(C(N(CC(CC)NC(c2snc(O)c2Cl)=O)C)=O)CCCCO1 c1(CSC)nc(-c2ccsc2)nn1C(C1CCC1)C1CC1 CCC(C)(C)C(O)C(=O)N1CCCCC(CNC(C2(N=[N+]=[N-])CC2)=O)C1 C1(C(=O)NCC(CNC(C(CC)n2ccnc2)=O)(C)O)CCC([N+](=O)[O-])CC1 Cc1ccc(NC(=O)NCC2CCC(C)(C(=O)OC(C)(C)C)CC2)cc1CO C1(C(=O)NCC(C)C(C)(F)F)CCN(C(c2ccccc2CC#N)=O)CCO1 N1(C(c2ccc(OC)o2)=O)CCN(C(C2CC(=O)N(OC)C2)=O)CC(C)C1 C(N=c1[nH]c2ccc(F)cc2o1)C1CC(C)N(C(c2cc3c(s2)CCC3)=O)C1 C1(C)(C(=O)NCCn2cc(Cn3ncc(C)c3)nn2)COCCOC1 CC1=CC(C)C(C(N2CCCC2CCC2CCCO2)C(=O)NC2(C)CC2)CC1 Cc1cc(NC(C2CCN2C(C2(C#N)CC23CCC3)=O)=O)cc(C)c1C c1(C(=O)NC(CCCNC(C2(COC)CC2)=O)CO)cc([N+](=O)[O-])cn1C N1(C(C(C)OCC#C)=O)CCC(C2(O)CN(C(C3(n4cncn4)CC3)=O)C2)CC1 C=CC1(CC(=O)NCC2CC(NC(=O)C3=CCOCC3)C(O)C2)CCCCC1 Cc1cc(C(=O)NC2C3CC2N(C(=O)C=Cc2ccc(Cl)cc2)C3)c(O)nn1 N=c1nc(C(=O)Nc2cccc(C3CCCN3)c2)c2ccc(C(F)(F)F)cc2[nH]1 N1(C(CN(C(=O)C(=C2CCCCC2)F)CCC)=O)CC(OC(C)=O)CC(C)C1 c1(C(=O)NC2C(NC(C3C(C)C3C)=O)C2)cnc2ccncc2c1 CCC(C)(C)C(C)CC(=O)N(C(C)CNC(=O)C=Cc1ccco1)C c1(NC(=O)NCC2(OC)CCN(C)CC2)cccn2nc(C)nc12 Cn1cc(C2CC2NC(=O)CC2CCN2C(C2(n3nccn3)CC2)=O)cn1 N1(C(C2CCC(C(C)C)CC2)=O)CCCC(C)(CNC(=O)CCc2cnoc2)C1 S(=O)(=O)(c1cccs1)N1C(NC(c2ccccc2C(F)(F)F)=O)C=CC1 CC1(C(=O)NCCC2CN(C(C3CC4CCC4C3)=O)C2)CCC2(CC1)CC2 N1(C(COC)=O)C(C)CC2CN(C(c3nc(Br)sc3Cl)=O)CC12 N1(C(C(C)c2cc[nH]n2)=O)CCC(CNC(=O)CC2CC3(CCC3)CO2)C(O)C1 c1(C(N2C(CC)CCC2)=O)cncc(Cl)c1.C12CC1C(=O)NC2(C)C c1(OC)ccc(CC(N2CC3(C2)CN(C(c2ccccc2Br)=O)C3)=O)cc1Br N1(C(C)C(N2CCN(c3cc(F)ccc3F)CC2)=O)CC2(CN(C(N)=O)C2)C1 c1(OC)cc(CNC(C2CC(NC(=O)CCC(C)(C)C)C2)=O)ccc1Cl Cc1ccnc(Cl)c1C(=O)NCC1=CCN(C(C2CC2(C)C(C)C)=O)CC1 c1(C(=O)NCC2N(C(C(CC)C#N)=O)CC(OC)C2)cc2c(Cl)nccc2s1 c1(C(=O)OC)ccc(C(N2CCC(CF)(NC(=O)Cc3ccco3)C2)=O)cc1C C1(C(N(CCNC(C2(CO)CC(F)(F)C2)=O)CC)=O)CCC2(CCC2)CO1 CC12CCC(C(N3CCCC(C)(NC(=O)CC4CCS(=O)(=O)C4)C3)=O)(CC1)CO2 C(=O)(N1OC2CCC1C2)C1C(CC)N(C(c2ccc(C)c(N)c2)=O)CC1 C12(NC(=O)C(F)F)COCCC1CN(C(C1(c3cc[nH]n3)CCC1)=O)C2 C=CC(C)CC(=O)NC(c1ccccc1)CNC(c1cc(CN(C)C)c[nH]1)=O c1(C(N2CC(C(C)NC(c3ccc(CSCCC)o3)=O)C2)=O)cc(Cl)nn1C.N Cc1nc2ncnn2c(C)c1C(=O)NCC1=CCN(C(=O)CSCC(C)C)CC1 C1(NC(C(CN(C(C2=CCN(C)C2)=O)C)(C)C)=O)CCC2(CCCC2)C1 Cc1cccc2cc(C(=O)NC3CCC(NC(=O)CC4C=CCCC4)CC3)oc12 c1(OC(C)C)nccc(C(=O)NC2CCC(NC(C3CC(C(F)F)C3)=O)C2)c1F C1(C(=O)NCc2snc(C)n2)CN(C(C2CC(=O)NC2=O)=O)CC12CCC2 C(C(C)(C)CN=c1nc2sccc2c(NC2CC2(C)c2cccs2)[nH]1)SCC C(=O)(C1=CC2(CN(C(=O)C(C)C(F)(F)F)C2)OC1)NCC1C(CC)C1 C1(O)(C(N2CCS(=O)CC2)C)CCCN(C(=O)C(=O)NCC2CC2)C1 C1(C(N(CCCN(C)C(c2ncccn2)=O)C2CCC2)=O)CC12CCCC2 N(C(=NCCc1ccc(Cl)cc1)NC(C)CC(F)(F)F)CCCn1c(C)ncc1 CC(C)C(CC(=O)N1CCCN(C(C)C)CC1)NC(=O)Cc1cnn(C)c1 c1(NC(C(CC(=C)Cl)N)=O)ccc2c(c1)C(=O)N(C)C2 N1(C(c2cn(CCOC)nn2)=O)CCN(C(=O)C(F)(F)C2CCCC2)CC1CF CCC(C)CCCC(=O)N1CCCC1C1(C(=O)NCCOC(F)F)CC1 c1(OC)ccccc1C(C(C)NC(=O)CC#N)NC(=O)CSC(F)F N1(C(C(F)=CC)=O)C2CCC1CC(NC(c1ccc(-c3ccncc3)o1)=O)C2 C1(CCNC(CCSC)=O)COCCN1C(=O)C(C)NS(=O)(=O)Cc1cccs1 c1(C(=O)NC(C)CN(C)C(C2CCCCN2N=O)=O)cc2ccccc2[nH]c1=N C12(CNC(Cc3c(C)n(C)nc3)=O)CCC1CCN2C(=O)C1=CCSC1 C1(NC(CCN(C(CCC)C)C)=O)CN(C(c2ccc(O)nn2)=O)C2(CCC2)C1 N1(C(C2(C=C)CCC2)=O)CCC2CN(C(c3c(S(C)(=O)=O)cnn3C)=O)CC2C1 N1(C(CN(C)CC2CC2)=O)CCCC1C1(CNC(=O)C=CC(F)F)CC1 Cc1ccn(C)c1C(N1CCC(N(C)C(c2cnn(C)c2N)=O)C1)=O C(=O)(CCCCCC(C)O)NCC(CCNC(c1c(C)nc(CC)o1)=O)O C(=O)(CC1=CCN(C)CC1)NC(c1nc(-c2ccncc2)no1)C CCC(C(=O)NCCC1CC(C)=NO1)N(C(=O)C=C1CCOCC1)C N1(C(c2cccc(C(=O)NC)c2)C(=O)NC2CC2)CC(O)CCC1C c1(C(=O)NC2CCN(c3cccc(F)c3)CC2)cc(Cl)cc2c1OCCNC2 Cc1oc(C)c(C(=O)NCc2csc(C(N3C(CO)CC3CO)=O)c2)c1C c1(C(=O)NC(CC)CNC(C2(n3cccn3)CCCC2)=O)c[nH]c2ccccc12 C1(NC(c2ncc(OCC)nc2)=O)CCC2CCN(C(C3C4CC5C(C4)C35)=O)C1C2 c1(CC(=O)NCCN(C(C(CC#C)O)=O)C(C)C)c(Cl)cccc1Br CON1CCC(C(=O)NC2CCCC2NC(c2cc(Cl)cnc2C)=O)CC1 c1(OC)cc(C(=O)NCC2CCC2NC(=O)C(C#N)C2CC2)cnc1C(F)(F)F Cc1nc(C)c(C(=O)N(C(CNC(C2CCOC(=O)N2)=O)C2CC2)C)nc1C N1(CC(N2C(C(CCC)C)CCC2)=O)CCN(C(c2cc(CC)ncn2)=O)CC1 c1(OC)ccccc1-n1nnnc1C1(NCC(C)(C)COC)CN(C)CC1C CCCCC(CN(C(=O)CC1CCN(C(C2(C3CC3)CC2)=O)C1)C)CC C=CCCC(=O)NC(C1CC(n2cc(C3(OC)CCCC3)nn2)C1)=O c1(CC(=O)NC(CNC(C2ON=C(C)C2)=O)C2CC2)ccc(F)cc1Br c1(CCNC(C(N2CC(C(C)=O)C2)=O)=O)c(C)[nH]c2ccccc12 N1(C(C2C(=C)CC2)=O)CCCC(N(CCF)C(c2cc(C)c(C)s2)=O)C1 CC1CC(CNC(=O)CCN(C(=O)CCC2CCC(=O)C2)C)=NO1 Cc1cccc(CNC2CC2C(=O)NCCSc2ccccc2)c1Br C(C)(CNC(=O)CN1CCCCC1)(CC(C)C)NC(c1cncc(C)n1)=O c1(OC)cc(-c2ccc(-c3nccn3CCCN3CCOCC3)cn2)ccc1C Cc1cc(O)ccc1-c1cn(CCC(=O)N(C)CC2CCCC2)nn1 Cc1nn(C)c2nc(C(=O)NCC3CCN(C(=O)C=CC(C)C)CC3)cc(O)c12 N(C1CCc2cc(C#N)ccc21)C(=O)NC(C)CCC(F)(F)F N1(C(C(CCF)NC(c2ncc(OC)nc2)=O)=O)CC(S(C)(=N)=O)C1 c1(C(=O)NC2(CNC(C3COCC(C)O3)=O)CCCCC2)ccnc(F)c1F C1(NC(CSc2cccc(C)c2)=O)CCC12CN(C(C1CCCC3(CC3)C1)=O)C2 N1(C(CC(C)(C)C(F)(F)F)=O)CC=C(C(C)(C)C(=O)NCCc2ccsc2)C1 C(C)(N=c1cc(Cl)c(O)n[nH]1)C1CCCN(C(C2N3C(C)CN(CC3)C2)=O)C1 C(=O)(C(C)(C)C(F)(F)CC)N(C)CCN(C(CCC=CC)=O)C C12(NC(c3c[nH]nc3C(F)F)=O)CCCC1NCC2 C1(N(CC(C)C)C(C2C(CC)C2)=O)CCN(C(c2ccc(C)o2)=O)CC1 Cc1cccc(Cl)c1NC(=O)CC1CCN(C(=O)C(C)Nc2ccccn2)C1 C1(NC(CCC(Cn2cc(CNC(C)=O)nn2)(F)F)=O)CC2CCC1CC2(F)F n1(CC)cc(C(=O)NCCC(O)CNC(=O)C(=O)NC2CC2)c(CC(F)(F)F)n1 N1(C(c2cccc(CC)c2F)=O)CCN(C(c2nn(CC)cc2Cl)=O)CCC1C c1(C(=O)NCC(C2CCCC2)NC(C(c2cncnc2)C)=O)ccncc1Cl N1(C(c2cc(C)no2)=O)CCC2(C=C(C(=O)NCC3CC34CC4(F)F)C2)C1 N1(C(C2C(NC(C34CCC(CC3)C4)=O)COC2)=O)CCCC(CCO)CC1 O=C1CCC(CC(N2CCC(C(=O)NC(CO)C3CC3)(CO)C2)=O)CN1 C1(C(=O)NCc2cc(C(N3CC(OC(N)=O)C3)=O)on2)CCCC2CC12 Cc1sc2ccccc2c1C(=O)NCC(C)CNC(=O)C(=O)NCC(F)(F)F C1(CNC(=NC)NCCCN2CCOCC2)CCCC1C1CC1 Cc1c(F)ccc(C(N2CCC2CNc2cccc(-c3ccccc3)n2)=O)c1Cl c1(C(=O)OC)cnc(N2CCC(NC(=O)CCc3cnc(C)s3)CC2C)cc1C c1(OC)c(F)cc2nc(N(C)Cc3ccc(F)cc3C)sc2c1F Cc1oc(C)c(C(N2CC3CC(NC(c4ncoc4C(C)(C)C)=O)C2C3)=O)c1C c1(C(=O)NC2CN(C(C3(C(C)C)CCC3)=O)CC2F)cc(Cl)c(Cl)nc1Cl c1(C(N2CCN(C(C(C)C(C)O)=O)CC2)=O)cc(S(=O)(=O)N(C)C)cnc1O C1(CN(C(=O)CC#N)C)CCCCN1C(=O)Cc1ccc(Cl)s1 c1(OCC)nccc(C)c1C(N1CCC1CCNCCCN1CCC(C)CC1)=O n1(CC(N2C(C)(CNC(C3CC3C(F)F)=O)CCC2)=O)cc(S(C)(=O)=O)cn1 c1(CN(C(C2C3CN(C(C4CN(C)C4)=O)CC23)=O)CC)ccc(C)c(C)c1 c1(CC(=O)NCCC(CCNC(C=CC(C)C)=O)C)cccc(Cl)c1F N1(C(C(C)C2CC2)=O)CCC2(CC1)CC(NC(c1ccc(O)cc1F)=O)CCO2 CC1(C)C(CO)CCN1C(=O)C(=O)NCC1(C#N)CC1 C1(O)(n2cc(CCC3CN(C(c4ccn(CCCC)n4)=O)C3)nn2)CCOCC1 C1(NC(C2(NC(C)=O)CC2)=O)COC2(C1)CN(C(C13CCCC(CO1)C3)=O)C2 C1(NC(N2CCC(O)(c3cccc(F)c3)C2)=O)CCc2scnc2C1 C1(C(=O)NCCC(C)(C)NC(CCNC(COC)=O)=O)CN2CCC1(C)CC2 CC1(C)CC(CNC(c2cc(F)cc(F)c2)=O)CN(C(=O)CC2(O)CCCC2)C1 c1(C(=O)NC2C(OC)CN(C(C(F)=CC)=O)C2)cc(C)n(C(C)C)c1C C1(C(N(C)CC2CCC(NC(CC3C(OC)CC3)=O)CC2)=O)CC12CCSCC2 C1(CCOC)CN(C(=O)CC2CCCO2)CCN1C(c1csc(C(C)=O)c1)=O C(=O)(C(F)C(C)(C)O)NC1C(NC(CCCOCC)=O)CCCC1 c1(C(=O)NC(CNC(C(C(CC)O)(C)C)=O)CO)cc(C)c2c(O)n[nH]c2n1 c1(COC)nc(N2CC(CCNC(=O)C(C)(C)C)(OC)C2)cc(Cl)n1 C(CCCCCC(=O)NC(CC(=O)OC)C1CC1)NC(CCC(C)OCC)=O CC(C)C(C)(C)C(c1nnnn1C1CCCC1)NC(C1CCC1)C c1(CC(C)NC2CCCN(Cc3cccc(C(F)(F)F)c3)C2)cnccc1C#N C12(C(=O)OC)CCCC(C(=O)NCCCNC(=O)CC3CCCCCC3)(CC1)C2 c1(OC)ccc(C(N2CCC(CNC(=O)C(F)CC3CC3)C2)=O)cc1Br N1(C(c2c(C)cco2)=O)CC(C(=O)NCc2cc(Cl)cc(Br)c2)CC(F)C1 C1(C)(C(=O)NC(c2cc(C)on2)C)CCN(C(c2conc2C)=O)C1 C1(C(N(C(C)CNC(c2ccn(CF)n2)=O)C)=O)CCc2n[nH]cc2C1C c1(C(=O)NCC2CC(O)(CNC(c3cnn(C)c3F)=O)C2)cnc2n1CCCC2 c1(NCCC(=C)C)ccoc1C(c1nnnn1C1CCOC1)OC n1(CC)c(=NC(=O)NCc2ccccc2C(C)(F)F)sc2ccccc12 c1(C(=O)NCC=CCNC(CC(C=C)C)=O)cccc(OC)c1C Cc1oc2ncnc(O)c2c1C(=O)NC1CC1C(C)C.c12ccccc1N(C)C2 C1(NC(c2c(OC)scc2)=O)CN(C(c2ccc(C(C)C)s2)=O)CC12CCCC2 C#CCCC(=O)N1CC(O)(C(C)NC(C2(C)CC2(F)F)=O)C1 C1(C(NOCC(c2ccccc2)C)=O)CC=CCN1C(C1CCCOCC1)=O CCC(CC(C)C)C(=O)NCC1CCC2(CN(C(=O)Cn3nnc(=N)[nH]3)C2)O1 C#CCC(C)C(=O)N(C)CCN(C(=O)CN1CC2C=CC1C2)C(C)C C(C)(CO)(C(=O)NCc1ocnc1C(=O)NC1CC(O)C(F)C1)OC c1(OC)ccc2c(CCC(=O)N(CC(C)NC(=O)C#CC3CC3)C)c[nH]c2c1 Cc1cccc(C(c2cc(Cl)cnc2-c2cncc(F)c2)=O)c1O CC(C)(CNC(=O)NCC1CC(C#N)C1)C#CBr c1(C(=O)NCC(CO)NC(=O)CCc2cnoc2)cc2n(n1)CCCC2O C(CS(=O)(=O)Cc1cccc(NC(=O)C(=O)N2CCC2c2ccc(Cl)cc2)c1)OC C1(C(C)C)(C(=O)NCCCOCCC(=O)NC(C(C)C)c2ncc[nH]2)COC1 CN(CCCC(=O)NCC1CC(CNC(c2cncc(O)c2)=O)C1)N=O N1(C(C(C(C)C)SCC)=O)CCC(C2CCN(C(c3cc[nH]n3)=O)C2)CC1 N1(C(CSCC#C)=O)CCC(CCNC(c2ccc(F)cc2)=O)CC1C CC(CC(N)=O)C(=O)N(CC(C)O)CCNC(c1ccn(CC#N)n1)=O CC1OC2(C(=O)NCC3CC(O)(CNC(=O)COCC4CC4)C3)CCC1CC2 C1(CNC(C2N(C)CCCC2)=O)CC2COCC2N1C(c1ccc(N)c(F)c1)=O CCC(C)(C)C(O)C(=O)N1CCCCCC(NC(C2CC(=C3CC3)C2)=O)C1 c1(N2CC(=C(CNC(C3N(C)CCC3)=O)F)C2)nc(Cl)nc2c1CCC2 CCC(CC(=O)NCC(CNC(C1(C)CCCCO1)=O)S(C)(=O)=O)C(F)F Cc1cc(C(N2CC=CC(C(=O)N(C)CCc3ncon3)C2)=O)cc(F)c1 N1(C(Cn2ccc(C)n2)=O)CCCC(C)(CNC(=O)CCN2CCC(F)C2)C1 Cc1ccc(CC(=O)N(C2CCCC2)CCNC(=O)COCC(C)(C)C)o1 C(CCCC1CCC1)NCCC(CO)C1CCC1 CC1(C(=O)NCC(c2ccccc2F)NC(C2CCOC2)=O)CC2(CC2)C1 n1(CC)ccnc1C(c1nnnn1C1CC1)NCC=C.C1C=CCO1 CC#CCC(C)N=c1[nH]c2c(c(=NCc3cn(C4CC4)nn3)[nH]1)COC2 Cc1ccc2cc(C(N3CCC(CCN=c4[nH]cncc4I)C3)=O)[nH]c2c1 N1(C(c2c(C)cno2)=O)CCC(C)(CNC(C2CCOC(=O)N2)=O)CC1 N1(C(C(c2cccc(OC)c2)C)=O)CCC(NC(=O)C(C)=C(C)C)C2(CCC2)C1 C1(NC(=O)NCC(c2ccc(OC)cc2)N(C)C)COC2(COC2)C1 c1(C(=O)NCCN(C(C(CC=C)C)=O)CCC)coc(C#Cc2ccccc2)c1 c1(C(=O)NCCOCCC(=O)NCc2cc(C3CC3)no2)cccc(CO)n1 c1(C(N(C)CCN(C)C(C2CC23CC3)=O)=O)cc2cc(Br)sc2s1 c1(N2C(CCCNC(C3(CCC)CC3)=O)CCC2)ncc([N+](=O)[O-])cn1 C1(C)(CC)CN(C(c2ccc(C)cc2F)C(=O)NC2CCCC2)CCO1 c1(C(=O)NCC(CC)NC(=O)C(C)CCc2ccccc2F)cnccc1C#N n1(CC)ccc(=NC(=O)CC2(CNC(c3cnn(C)c3OC)=O)CC2)[nH]1 c1(C(N(C2CN(C(c3csc(CS(C)(=O)=O)n3)=O)C2)C)=O)cnn2c1OCCC2 C1(CNC(CC=CC=C)=O)CCCC(NC(=O)CN2CC(C)C2)C1 n1(C(C)C)cc(Br)cc1C(=O)NCC1CC(NC(c2ncccc2N)=O)C1 c1(CC(C)OC)nc(-c2cc(Br)cs2)n(-c2ccn(C(C)C)n2)n1 CC(C)C(C(C)NC(=O)Cc1ccccc1Br)NC(=O)C=Cc1cocn1 C1(C(N(CCC(=O)NC2CC3CCC2O3)CCO)=O)CC(C2CC2)=NO1 N1(C(C(C(C)(C)C)N(C)C)=O)CCC2(CNC(=O)CCN3CCCC3)CCCC12 N(C(=NCCc1ncccc1C)N1CCC(C)C2(CCC2)C1)CCC(=O)NC C1(C(N(c2cccc(CC)c2)C)=O)CN(C(C2CCCC(=O)C2)=O)CC(C)(C)C1 N1(C(COCC)=O)CCCC2(CCCCC2NC(=O)C(C)Oc2cccnc2)C1 C(C(=O)NCCN(C(c1cnc(C2CC2)[nH]1)=O)C(C)C)(C(C)C)SCC c1(C(=O)NCC(=CC(=O)NC(COCC)C)C)ccc(O)cc1 C1(C(=O)N(Cc2c(C)ncs2)CCc2ccc(Cl)cc2)CN(C)C(=O)N1C(C)C N1(C(CC(C=C)CC)=O)CCC2CCC(C1)N2C(C1CCC(=O)N(C2CC2)C1)=O c1(C(=O)NC(CNC(c2cccc(OC)c2N)=O)CO)cc2cccc(C)c2o1 c1(CN2C(C(N3CC4CC4C3)=O)CC2)cc(Cl)c2c(c1)OCCO2 c1(C(C)=O)ccc(C(=O)NCc2cc[nH]c2C(=O)N(C)CCc2ccccn2)[nH]1 c1(C(=O)NC2CCCN(C(=O)CO)CC2)ccc2nncn2c1 N1(C(C(CC)N(C)C)=O)CCc2ccccc2C(NC(=O)CSC(=N)N)C1 c1(C(=O)NCC(CC)(CC)NC(c2ccc(CO)cc2F)=O)c(C)cccc1Cl c1(N(C)C)cc(C(=O)NC2CCCC(CNC(=O)C3=NOCC3)C2)ccn1 CC(C(C)(C)C(=O)NOCC(F)(F)F)NC(c1ccn(C)c1)=O C1(CC)CN(C(C2(CC)COC2)=O)CCC1NC(=O)C(O)C(C)C c1(NC(C2(F)CCN(Cc3ccc(C)nc3)C2)=O)cccc2c1OCCO2 c1(OC)ccc(S(=O)(=O)N2CCCC(CC(=O)Nc3cccc(CO)c3)C2)cc1 CCCCC(C(=O)NCCCC(N1CC2CC1(C(F)F)C2)=O)C(C)C C(=O)(C#CC1(C)COC1)NC(CC(C)C)C(=O)N(CC(F)Cl)C C=CCC(C)(CC)C(=O)NC1CCOC1C(=O)NC(C(=O)OC)C1CC1 CCCCC(C(=O)N1CCC(NC(c2sncc2Br)=O)C1(C)C)N(C)C c1(CN(CC(C)C)CC2CCCO2)cnc(-c2cccs2)s1 CC1(C)CCC(CNC(=O)C(c2cccc(F)c2)O)(NC(c2cocn2)=O)CC1 C12CCCCN(C1)C2.C1(C(=O)NC(=O)C(c2ccccc2)F)C=CC=CC=C1 C(=O)(C(C)C(=O)NCC1CC(C(=O)NCC#CCCO)CO1)OC C#CCCC(C(=O)N1CCC(F)(CO)CC1)NC(C1CC2C=CC1O2)=O C1(NC(C2CC(C#C)(O)C2)=O)CC(C(=O)Nc2ccc(F)c(C)c2)C12CCC2 CCCCC(C(=O)N(CCNC(=O)Cc1nc2c([nH]1)CCCC2)CC)C(C)C CC(C)P(=O)(CC(=O)NCC#CCNC(C1CCS(=O)(=O)C1)=O)C(C)C N1(C(CNC(c2ccsc2)=O)=O)CCCCCC1CO.C1(C=O)CC(F)(CO)C1 c1(C(=O)OC)ccc(N=c2scc(-c3cnn(C)n3)n2C2CC2F)cc1 c1(C(=O)NC2C(NC(=O)COc3ccccc3)CC2)cccc2nonc12 Cc1cscc1C(N1CCCC1C1CCOC1)C(=O)N(C)C.C1CN1 c1(OC)cc(C)c(C(=O)NC2C3CCC(C3)N2C(=O)CCCOC(C)C)cn1 c1(C(=O)NCC2N(C(CC(C)(O)C3CC3)=O)CC2)cccc2c1CCS2(=O)=O C(=O)(C1CCCc2cccnc21)N1CC2CN(C(C(CC)(C)CO)=O)CC(C1)O2 c1(C(=O)OCC(CC)(C)OC)ccc(C(F)(F)F)c(I)c1 N1(C(C(=O)NC(C)C)=O)CC2(C1)CN(C(C1CC(C(F)(F)F)C1)=O)CC2CO N1(C(C2(C)CCOC2)=O)CCOC(C(=O)NCC(c2ccco2)O)CC1 CN1CCc2[nH]nc(C(=O)NC3(CNC(C4CC4C4CCCCC4)=O)CC3)c2C1 N1(C(c2cccc(C)n2)=O)CCC(C)C(CNC(=O)C(C)CF)C1 Cc1ncc(C(=O)NCC2=NOCC2)c(Br)c1Cl C1(C(N(C(C(C)C)C)C2CC2)=O)CN(C(=O)Cc2cnsc2)CCC1(C)C C(=O)(C1=CCN(C(=O)COCCCN=[N+]=[N-])C1)N(C1C(C)CCCC1)C C(C(C)CC(=O)NCC1CCCC1NC(c1c[nH]nc1Br)=O)OC C12(CNC(CCC(C)OC)=O)CCC(CC1)N(C(c1sccc1Cl)=O)C2 C1(C(=O)N(C)CC2CCCN(C(=O)C=CS(C)=O)C2)(OC)Cc2ccccc2C1 Cc1cc(CNC(C23CC(CO2)N(C(c2ccsc2C)=O)C3)=O)cnc1C C(=O)(C(F)C(F)(F)F)NC(CN(C(C1OCCC1C(C)C)=O)CC)C N1(C(CCC(N)=O)=O)CC(CNC(c2nscc2Br)=O)C2(CC2)C1 c1(C(=O)NC2(CCCNC(=O)CCCc3cccs3)CC2)ccn2cncc2c1 Cc1ccc2c(c1)CN(C(c1cccc(NCc3cccc(O)c3F)c1)=O)CC2 c1(C(=O)NCC2(F)CN(C(CC(=O)OCC)=O)C2)ccn2cncc2c1 C1(NC(CC=C(C)C)=O)CN(C(=O)CCc2cnc[nH]2)CCC1C(F)(F)F Cc1cc(C(=O)NC(CNC(C2CC(=C3CC3)C2)=O)C2CCC2)c(F)cc1Cl CC1(C)C(NC(=O)Cc2ccsn2)C2CCCN(C(=O)CC3CCCCCC3)C12 CN1CC2C(C(=O)NCC3CN(C(=O)CC4(C(F)(F)F)CCC4)C3)C2C1 C1(CCC)CCC(C(N2CCCC2CCNC(C2CC2(F)F)=O)=O)CC1 C1(NC(C(C)(C)C#N)=O)CN(C(c2ncncc2F)=O)CC1(C)C C1(NC(C2CC(C)OC2)=O)CC2(CCCCN2C(=O)CCc2ccncc2)C1 c1(N2CCC(C)C(NC(c3c(CC)ccs3)=O)C2C)ncc2ncn(C)c2n1 N1(CC2N(CC3(C(C)(C)O)CC3)CCC2)CCC(C#N)C1 CCCCC(CC)C(=O)NC(CNC(=O)C(C)n1ccnc1)(CC)CC c1(C(=O)NC(C2CCCC2)CNC(=O)COCCCF)ccc2n[nH]cc2c1 CCCCC(C)C(=O)N1CCCC1(C(=O)NCc1n[nH]c(C)n1)C(C)C CC(C)(C(=O)NCC(O)CNC(C1(C#N)CCN(C)CC1)=O)S(=O)(=O)C1CC1 CCC(C)C(=O)NCC(N1CCC(N(C(=O)C(O)CN(C)C)C)C1)=O c1(C(=O)OC)nc2sc(C)cn2c1NC(=O)NCC1(C(O)C(C)C)CC1 C1(NCC2OCCN(C3C(F)(F)CCC(F)(F)C3)C2)COc2ccccc2C1 N1(C(CC(=C)C)=O)CCCCC1CCN(C)C(c1ccc(NC(C)C)cc1)=O CCC(CNC(=O)C(F)Cc1ccccc1)(CC)NC(=O)CN1CSCC1=O O=C(C1=COCC1)NC(CNC(C1CCC(Cc2ccccc2)CC1)=O)CO S(=O)(=O)(c1ccc(Cl)cc1)CC(=O)NCCCNC(=O)OC(C)(C)C C1(CCOC)(C(=O)NC(C2CCCC2)C)CCN(C(=O)CC2CCCCO2)CC1 c1(C(=O)NCC23CC(NC(C4C(C)SCCC4)=O)(C2)C3)c(Cl)nc2ccccn12 C(=O)(C1CCCn2ccnc21)NC1CN(C(c2ccnc(C)c2C)=O)CC1C C=C(C)CC(C(=O)N1CCC(O)C1C(=O)N(C1COCC1O)C)OC N1(C(c2cn(C)nc2)=O)CCOCC1CCNC(c1cnc(C(=O)OC)cn1)=O c1(C(=O)OC)cnc(C)[nH]c1=NC(C)CNC(c1ccc2c(c1)COB2O)=O C(=O)(CC(O)CC(C)(C)C)NC(CC(C)NC(COCC(=O)OC)=O)C C(=O)(C(CN(C)C)C(C)C)NCC1(C)N(C(c2cc(C)n(C(F)F)n2)=O)CCC1 C(CCCC)(C(=O)NCC(O)C(C)CC)NC(CCC=CCC=C)=O C(=O)(CCN=C(NCc1cccc(OC)c1C)NC(C)C(F)(F)F)NC c1(OC(C(=O)Nc2cc(C(=O)OC)sc2)(F)F)ccccc1F N1(C(CC(=O)N(C)C)=O)CCCC2(CCC(NC(=O)Cc3cn(C)cn3)C2)C1 C(CN=[N+]=[N-])(C(=O)N(C)CCn1ccnc1)NC(c1n[nH]c(C)c1C)=O C1(C(C)(C)C)CC(NC(=O)CC2CC(NC(C3CCSC3)=O)C2)C1 c1(NC(N2CCCC(NC(c3n(CC)nnc3)=O)C2)=O)ccc(F)cc1C C#CC1(C(=O)NC2CCN(CCCO)C2)CN(C(=O)CN(CC(C)(C)C)C)C1 Cc1nc2c([nH]1)C(C(=O)N1CCN(C(=O)CC3CCC3)CC1CC1CC1)CCC2 C1(C(C)(C)C)CC2(CC(NC(C3(CNC(C4CC5(CCCC5)C4)=O)CC3)=O)C2)C1 C1(CNC(c2cnc(C(C)C)[nH]2)=O)CCCCCN1C(C1CCCOC1)=O C(N=c1[nH]cnc(Cl)c1C(C)C)C1CCCC(NC(C(=O)NCCOC)=O)C1 c1(C(=O)NCCCN(C)C(C2CNC(=O)N2)=O)cc2n(c1)CCSC2 C1(CN2C(COC)CSCC2)CCn2nnnc2C1 c1(CCC)ccc(C(=O)NCC(O)CNC(=O)Cc2cc(C)[nH]n2)s1 C=CCC(C)C(=O)NCc1ccc(C(F)C(F)F)cc1 Cc1csc(C(c2nnnn2C2CCOC2)NCCCC2CCC2)n1 c1(CNC(C(CC2CN(C(CCC3C(C)C3)=O)C2)F)=O)cccc2cccnc12 c1(-c2c(C(C(N(OC)C)=O)(C)C)ccs2)ccccc1S(=O)(=O)C(F)F N1(C(CCOCCNC(C2(C(C)C)COC2)=O)=O)CC(C)C(C)C1C CON(CCC(=O)N1CCOC2CCC12)C(=O)C1CC(C)CO1 c1(OC)ccncc1CNC(C1(C(C)NC(C2CCC(=O)C2)=O)CC1)=O c1(OCC)cnc(C(=O)NC(c2nccn2C)C(C)C)nc1 c1(OC)cccc(CN2CC(C(C)NC(c3cccc(OC)c3)=O)C2)c1 C12CCOC1CN(CCN1CC=CC1)C2=O.C1(OCC(=O)NC)CCOCC1 Cc1csc2ncnc(N3CCC(NC(C45CCCC(C)(C4)OC5)=O)CC3C)c12 CC(CC(=O)Nc1ccc(NC(C2(C(N)=O)CC2)=O)cn1)CC(C)(C)C C=CC1CN(C(=O)C(C)(C)CO)CC1NC(=O)C(c1ccc(F)cc1F)(C)C C1(C(=O)NCC(Cn2cc(CCN(C)CC)nn2)(F)F)(C(F)F)CCCC1 c1(CC#N)ccc(S(=O)(=O)NCC2CC2F)cc1 N1(C(=O)NCC(N2CCOCC2)C(C)C)CCCCC1Cc1ccccn1 c1(C(N2CCC(C(NOC3CC(=C)C3)=O)(CC(=C)C)C2)=O)cc(C)c(F)cn1 N1(C(CCC(=C)C)=O)Cc2ccnn2CC(NC(=O)C(C)OC2CCCCC2)C1 C(CNC(=O)COC(F)(F)F)(CCNC(c1csc(Cl)n1)=O)OC C(=O)(C(CC(F)F)C1CCC1)N1CC(NC(CCOC(C)C)=O)C(C)C1 CC1(C#CC(=O)NC(CO)C(N2CC3CC(N(C)C)C2C3)=O)COC1 Cc1cc(C(=O)NC2(CO)CN(C(=O)C(C)Oc3ccccn3)C2)cc(F)c1 C1(C(F)(F)F)(CNC(c2ccc(Sc3ccco3)o2)=O)CCCC1 c1(C(=O)NC(CC)CNC(=O)C(c2ccc(Cl)cc2)CO)ccc2nc[nH]c2n1 S(=O)(=O)(c1cc(F)ccc1OCC(F)F)NC(C(N1CC(NC)C1C(C)C)=O)=O C(=O)(C(O)CCNC(C1CC(OCC)C1)=O)NCC=C CON=CC(=O)NC(c1cnn(C)c1)C(=O)NCCn1cnnn1 c1(C(=O)NCCC2CCC(NC(c3ccc(C)s3)=O)C2)ccc(N)nn1 C1(CNC(C)=O)CC2CCC(C1)N2N1CCC(OC(c2ccccc2)=O)C1 c1(C(C)C)ccc(C(N2CCCCC(NC(=O)C=Cc3ncco3)C2)=O)c(F)c1 N1(C(c2cncc(C)c2Cl)=O)CC2CC(NC(c3n[nH]cc3[N+](=O)[O-])=O)CC1C2 S(=O)(=O)(c1ccc(I)cc1)N1C(C(N2CCN(C)CC2)=O)CCCC1 c1(CC(=O)NCC(CC)C)csc(NCC(c2ccccc2)OC)n1 c1(CNC(CN(C2CCC2)C(C)=O)=O)noc(C(C)C)n1 c1(C(=O)NCC2(NC(C(C)OCC#C)=O)CCCCC2)cccc2c1CCCN2 CC(CC(F)(F)F)C(=O)NC1CCCN(C(c2nccc(C(F)F)n2)=O)C1 c1(C(=O)NCC(C)N(C(=O)C=Cc2ccc[nH]2)C)nc2c(Br)cncc2[nH]1 Cc1nc2cnn(C)c2cc1C(=O)NCC1COCCN1C(c1c[nH]c(=N)s1)=O C(=O)(C1=Cc2ccccc2C1)N1CCC(Cc2ccc3nc(C)[nH]c3c2)CC1 C12(C(=O)NCC3C(NC(C4CC(C(C)(C)C)OCC4)=O)C3)CCC(CC1)C(C)O2 CC(C)CC(O)C(=O)NCCCCNC(=O)CC(C(F)F)N1CCOCC1 N1(C(C(CCCOC)NC(c2cc[nH]n2)=O)=O)CCOCC2(CCC2)C1 c1(CC)cc(C)[nH]c(=NCC2CC(CNC(=O)Cn3ccc(=O)n(C)c3=O)CO2)n1 N1(C(C2C(C=C)C2)=O)CCN(C(=O)CCOC2CC2)CC1c1ccnn1C C(=O)(CCC(C)C)NC1(CNC(c2c(CC)[nH]cc2)=O)CCCC1 C(c1ccc(F)c(F)c1)=CC(=O)NC(CNC(C1CC(O)(CC#C)C1)=O)(C)CC C(C(F)(F)CC(=O)Nc1cc(CC)ncn1)N(C1CC1)Cc1c(OCC)cccc1 N#Cc1ccc(C(=O)NCC(=O)NCC2CC2NC(=O)C2=NOCC2)cc1 Cc1ccc(F)c(C(=O)NCCC(C)N(C)C(C2CCC(N=[N+]=[N-])C2)=O)c1N c1(CC)nn(C)c(Cl)c1C(=O)NC(C)CC1CN(C(=O)C=CI)C1 C1(C(=O)NC2CC(C(N3C(CSC)CCC3)=O)C2)CC(F)CN1C C(=O)(C1=CC(O)CCC1)NCC1(F)CCC(CNC(=O)CCc2cccnc2)C1 c1(CC)nc(NC(=O)C(=O)NCCC23CCC(CC2)C3(C)C)c2n1CCCC2 CC1CCN(C(C2(CCO)CC2)=O)CC1NC(=O)Cn1cccn1 C(=O)(C(C)N(OC)C(=O)CCCNC(=O)CCCC(C)OC)OC c1(C(C)=O)ccc(C(=O)NC(C)CNC(C2CC2C)=O)[nH]1 CC1(NC(c2ccc(C(F)F)s2)=O)CCCN(C(=O)C(F)(F)C2(O)CCC2)C1 C1(CC(N2C(CCNC(CC3N(CC)CCC3)=O)CCC2)=O)CCCOCC1 N1(C(C(C2CC2)SC)=O)CCCCC(CCC(=O)Nc2ncccc2F)C1 C(c1c(Cl)cccc1Cl)=CC(=O)NCC=CCNC(CSCCC#N)=O C(=O)(CC(F)(F)C(C)C)N1CCC(CCN(C(c2nc(C)n(C)c2C)=O)C)CC1 CS(C)(=O)=NCC(=O)N1CC(F)CC1CNC(=O)CCNc1ccccc1 c1(C(=O)NCCC2OCCN(C(CCC(C)(C)C)=O)C2)cnc2ccnn2c1N c1(C(=O)NC(CC=C)C)cnc(C(C)(C)C)cc1OC Cc1ccncc1CC(=O)NC1CC(CNC(=O)CCCN(C)C)C1 N1(C(CCNC(COC)=O)=O)CCCC12CCN(C(C1CN(C(N)=O)C1)=O)C2 C1(C(=O)NC(CC)CNC(c2ccc(=N)[nH]c2Cl)=O)CCn2c(C)nnc2C1 c12sc(cc1OC)C(=O)NCCCN(CC)C(=O)C2.C1(C2CC2)CCCC1.C#CC C1(NC(=O)CCC2CCN(C(c3ccnn3C3CC3)=O)C2)C2CCCOC12 C1(CC)(CNC(C(=O)OC2(CF)COC2)C2CC2)CCCCO1 C(CCS(C)=O)(C(=O)NC(CNC(c1ccnnc1)=O)CC(F)(F)F)N(C)C CC(C)(CCCCNC(=O)C#CC1CC1)NC(c1coc(CO)c1)=O Cc1cc(N)c(C)nc1C(N1CCC(NC(=O)CC2CCN(C)C2)C(O)C1)=O C#CC1(C)CCCN(C(C2(CC)CCCN2C(=O)COCCCOC)=O)C1 C1(NC(c2nc(OC)oc2)=O)CC2CCC(C1)N2C(c1oc(C)nc1C)=O C1(CC(=O)NCC2CCN(C(c3ccc(=O)oc3)=O)C2)CCCC(C(F)(F)F)C1 Cc1cc(Br)cc2cc(CN3CCC(N(C)C)C3)oc12 N1(C(CCCCC(C)=O)=O)CCCC2NC(=O)CC12 Cc1conc1C(=O)NCCOCCCNC(=O)C(c1ccnn1C)C c1(C(=O)NC2C(NC(C(COC)N(C)C)=O)CCCC2)cc(Cl)cc(F)c1N c1(CN(C)C)cc(C(=O)NCCOCCN(C)C(c2ncoc2C)=O)sc1C N1(C(c2c(CC)nc(C)[nH]2)=O)CC(C)N(C(=O)C(F)CC(C)(C)C)CC1C N1(C(C2C(C(C)O)C2)=O)CCC2(CCN(C(=O)CN3CCC(F)C3)C2)C1 c1(OCC=C)ccc(C(=O)NCC2CC(NC(C3C=CCC3)=O)C2)cc1 C1(C(C(N2CC(NC(CSS(C)(=O)=O)=O)(CO)C2)=O)O)CCCCCCC1 c1(OC)cccc2c1OCC(C(=O)N1CC(NC(=O)C(C(C)C)N(C)C)C1)=C2 Cc1c(C(=O)NC2CCC2NC(c2ccsc2)=O)cnc2c(Cl)cccc12 CC(C)C(CN(C)C)C(=O)N1CCN(C(c2cnn(C(C)(C)C)c2)=O)CC1CF C1(NC(CCOCCSC)=O)CCC2(CC1)CC2NC(=O)Cc1csc(C)n1 Cc1nn(CC(N2CCCC(O)(CNC(C3CC3C)=O)CC2)=O)c(C)c1C=NO CCC(C(=O)N(CCCNC(=O)Cc1nncn1C)C)N(C)C Cc1cccn2cc(C(=O)NC34CC3CN(C(=O)CCN3CC3)C4)nc12 C1(N=[N+]=[N-])(C(N2CC(CC(C#C)C)C2)=O)CCN(C(c2cc(C)n(C)c2)=O)C1 C(=O)(C1CCCc2scnc21)NC(CNC(c1cnc(C)s1)=O)CC(C)C c1(CC(=O)N(C(C)Cc2cccs2)Cc2ccco2)cc(C2CC2)on1 Cc1sc2cc(F)ccc2c1CCNC(CC(O)CF)=O C(=O)(C(C)(C)CCCNC(c1cc2cccn2cn1)=O)N1C(COC)C=CC1 C(=O)(C(C(C)(C)C)NC(C1CC(C)(C)CN1C)=O)N(CCC(F)(F)CO)C c1(C(=O)NC(C(C)C)C(C)NC(=O)CN2CCCCC2)ccc2nccnc2n1 CCCC(CCC)C(=O)N(C)CC1COCCN1C(c1csc(C(F)F)c1)=O c1(CCNC(NC2C(F)C2)=NCC2CCCCC2)ccc(F)cc1F C1(N(C)CCO)CCCCN(C(=O)C2=COCCO2)C1=O CC1CN(C(C2CCN(C(=O)C3CC3)CC2)=O)CCN1c1ccc(C2CC2)nn1 Cc1nc(N2CC(NC(c3cccc(F)n3)=O)C(C)C2)c2cc(Br)ccc2n1 c1(NC(CNC2CCN(C(c3ccc(OC)cn3)=O)C2)=O)cc(C)c(Cl)cc1F C(CC(O)C(=O)NC(CNC(c1cncnc1)=O)C1CC1)N(C)C c1(CC)cc(C(=O)NC2(CNC(=O)CC3CC3)CCCCC2)ncn1 Cc1oc(S(N)(=O)=O)cc1C(=O)NCC1CC(NC(=O)C2=NOCC2)CCO1 C1(C(N2C(C)(C(=O)NC3C=CC(C(=O)OC)C3)CCC2)=O)CCOCC1(C)C Cc1nc(C)n(CCCC(N2CC(NC(=O)Cc3c(C)noc3Cl)CC2C)=O)n1 N12CCC(CC1C)CNC(=O)C(C1CC1)CC2=O.c1(CC=C)cccc(CO)c1 N1(Cc2c(C(F)(F)F)cc3c(c2)CCC3)Cc2ccccc2C12CCOCC2 C1(NC(CC2C(C)CCO2)=O)CCCC2CN(c3cc(Cl)nc(C4CC4)n3)CC12 C1(C(=O)NC23CC(NC(C(C)CO)=O)(C2)C3)CCc2cnn(C)c2C1 N1(C(C(C2(O)CN(C(c3ccc(C)nc3)=O)C2)F)=O)CCC2(CCC2)C(O)C1 c1(OC)cncnc1C(=O)N(C(C)C(=O)NCC1COCC(C)O1)C C(N=c1[nH]c(C(F)F)nc(=N)[nH]1)C1CCC(NC(Cn2ncc(C(N)=O)c2)=O)C1 c1(C(N2C(COC)COCC2)=O)cnc2n[nH]c(-c3ccc(F)c(F)c3)c2c1 c12cccc(c1Cl)OC(=O)CN(CCOC)C2=O.C(C)(C)OC N#Cc1cc(S(=O)(=O)N2CC3C(C2C(=O)NC2CCC2)C3C(=O)O)ccc1F c1(C(=O)NCCCOC)ccc(NC(c2cncn2C)=O)nc1 N1(C(CC)C(=O)N(CC(CC)NC(=O)CC2(O)CCC2)C)CCc2ccccc21 C1(OC)CC(CCNC(C2CCCN2C)=O)N(C(=O)COCCCN=[N+]=[N-])C1 N1(C(c2nc(OC)nc(O)c2)=O)CC2CC1CN(C(C1CCOC(C)(C)C1)=O)C2 C1(CNC(C(CC#C)C)=O)CCC2(CC1)CCN(C(=O)CN(C(=O)C(C)C)C)CC2 c1(CNC(C2(C)CCN(C)C2)=O)cc2n(n1)CCN(C(=O)CC1CCCOC1)C2 N1(Cc2cncc(F)c2)CCC2CN(c3ccn4nccc4n3)CCC12 CC(=O)C(C)CC(C)C(=O)NC(C(=O)NCC(O)C(C)(C)O)C1CC1 c1(C(=O)NC(CC)CNC(=O)C(C)c2cncs2)cccc(C(F)F)c1OC N1(C(c2sc(CC)c(C)c2)=O)CCN(C(=O)CC2CCC2)C(CC(F)F)C1 CCC(C)CC(C(=O)NCC1CN(C(N)=O)C1)NC(c1cc(C#N)oc1C)=O C1(NC(C=C(C)I)=O)CS(=O)(=O)C12CCN(C(C1CC1C(C)O)=O)CC2 N1(C(=O)C2=CCC(F)(F)CC2)CCC2C(CCCN2C(=O)Cc2csc(Cl)c2)C1 n1(C(CC)CC)nc(-c2cccc(Cl)c2)nc1CN1CC(O)CCO1 C1(O)(CNC(c2[nH]c(=NC)sc2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 C12COC(C)(C)CN1CC(=O)N2.Cc1ccccc1COc1ccccc1 C12(CNC(CCOCCC)=O)CC(CO1)N(C(=O)Cc1nnc(S)n1C)C2 Cn1ncc2c(N3CCN(C(C4CC=CC4)=O)CC3CCO)ncnc12 c1(CC)cc(NC(=O)C(Cn2cncn2)NC(=O)CC#N)ccc1F c1(C(C)(C)C)c[nH]cc1C(N1CCC(N)C1)=O.c1(C2CCOC2)cn(C2CC2)nn1 N1(C(c2c(SC)snn2)=O)CCN(C(=O)Cc2ccoc2C)C2CCCCC2C1 N1(C(c2ccccc2C(N)=O)=O)CCC(N(C(=O)Cc2cccc(O)c2)C)CC1C c1(NC(c2scnc2-c2ccncc2F)=O)c(F)ccc(Br)c1F C1(NC(C(c2ccc(C#N)cc2)C)=O)CCN(C(C2CCCN(C)C2)=O)CC1F C(C)(CCCC(=O)N1CCOC(CC(N)=O)C1)NC(C(n1c(C)ccn1)C)=O CCCC(C(=O)N1CCCC1C(C)NC(c1cc(C(N)=O)[nH]n1)=O)S(N)(=O)=O C(C1=CCN(C(C2CCOC2)=O)CC1)NC(C(CCN(C)C)O)=O C1(N(C(c2c(OC)n[nH]c2)=O)C)CCC2CN(C(=O)C3=CCCCC3)CC12 N#CC1CCCCC1NC(c1ncc(Br)cc1C(F)F)=O C(=O)(CCC(C)(F)F)NC(C)C(C)(C)NC(=O)COc1ccc(C#N)cc1 C1(C(C)C)(NC(=O)NCCC2C=CC(NC(C)(C)C)C2)CCOC1 N1(C(=O)OCC)CCC(NC(=O)COC(c2ncccc2Cl)=O)CC1.NCC N1(C(C2CC3CC2(c2ccc(F)cc2)C3)=O)CCC(O)C(O)C1 CCCC(CCC)CC(=O)NCC1(CNC(=O)C(O)C(C)C)CCCC1 CC(CNC(=O)NCC#CC1CC1)CC(F)F C1(C(=O)NCCCN(C(C(F)=CC)=O)CCO)C(c2ccncc2)C1(C)C c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(C3CCOCC3)O)C2)cc(F)c1 C1(C(=O)NCCCNC(C2(C)CS(=O)(=O)C2)=O)COc2cc(F)ccc2O1 C1(F)(CNC(c2ccc(Br)o2)=O)CC(NC(C2CC(CCF)C2)=O)C1 N1(C(COC(CC)(C)C)=O)CC(O)CC1(C)C(=O)NC1CC(O)C(O)C1 c1ccc2scc(Br)c2c1.Cn1cc(N(C(=O)NC(C)(C)C)C(=O)C2CC2)c(C#N)n1 CC12CCN(CC1)CC(=O)N2.C1(CCSC)CCOCC1.C1(N)CCCCC1 CC1CC(NC(c2scnc2C(F)(F)F)=O)CN(C(c2cnn3c2OCC3)=O)C1 N1(C(c2nc(C(F)(F)F)nn2C)C(=O)NCCOC)CCOCC12CCSC2 CC1CN(C(C23CCC(C(=O)Nc4cnc(F)c(Br)c4)(CC2)C3)=O)CCC1=O C1(C(N2C(C)CN(C(c3nc(C(F)(F)F)cs3)=O)CC2)=O)CC2CC1CC2(F)F C1(C(=O)NCCCOC)CC2CN(C(=O)CCCSC)CC2C1 CCC(F)(F)CC(=O)NCC(C1CCCCN1C(=O)C(O)Cc1cnc[nH]1)(C)C O=S(=O)(Oc1cnc(Br)c(F)c1)c1cccc2ncccc12 c1(C(CC)C)ccc(C(=O)NCCNC(c2sc(-c3ncc[nH]3)nc2C)=O)cc1 C12(C(=O)NC3C(C)(C)OCC3)CC(CO1)N(C(=O)Cc1ccccc1F)C2 C1(=O)C(CCOC)NC(=O)C(COCC)N1.c1ccc(C#N)o1.C(CO)OCC Cc1nn(C)cc1C(O)C(=O)NCCCN(CCO)C(c1ccc(Cl)s1)=O N1(C(c2c(C#C)c[nH]n2)=O)CC(C)N(C(=O)CCCS(N)(=O)=O)CC1C C=CCC(CC(C)C)C(=O)NC(Cn1cncn1)C(N1CCOCC(C)(C)C1)=O Cn1cc2c(n1)CC(C(=O)NC1COCCC1NC(c1c[nH]nc1F)=O)NC2=O C1(C)(CC)CCN1C(=O)CC1(NC(=O)CC(C)C2CC2)CC1 C1(NC(C2CC2c2cnc[nH]2)=O)CCN(C(=O)Cc2ncc(Cl)s2)CC1F c1(C(=O)NC2CC(CNC(C=CC)=O)C(O)C2)cccc2c1OC(F)(F)O2 C1(C(N2C3C(NC(c4ccc(OC)s4)=O)CC(C3)C2)=O)CC2(C1)CC(C)(C)C2 c1(NC(c2c(F)ncc(-c3c(C)nc(C)s3)c2)=O)ccc(Cl)nc1Br Cc1cc(C=CC(=O)NCC2CCN(C(=O)Cn3nccn3)C2(C)C)on1 c1(NC(C2CC(=C)CN2C(c2cc(Cl)ccn2)=O)=O)cccc2nsnc12 C(C(F)(F)C(C)(C)O)N(C(=O)CCC1CCCCN1C(=O)CSC)CCC(C)C N1(C(C2(c3ccncc3)CCC2)=O)CCN(C(C23CC(F)(C2)C3)=O)CC(O)C1 c1(C(N(C)C)=O)cc(S(=O)(=O)Nc2ccc(OC(F)F)c(C#N)c2)cn1C C1(CC#C)CCN(C(=O)C(CNC(=O)C(C)N(C)C(=O)CC)N(C)C)C1 c1(CNC(=O)Nc2cscn2)cc(OC2CCOCC2)ccn1 Clc1ccc(Br)c2c1C(N=c1[nH]c(=NCC3CC3C3CCOC3)[nH]c3ccsc13)CC2 C#Cc1ccc(CC(N2CC(NC(C3(C=C)CCCC3)=O)CC(F)C2)=O)cc1 N1(C(CC2(C=C)CCOCC2)=O)CCOCC(F)(CNC(=O)CC(C)SC)C1 N1(C(C=CC)=O)CC(OC)CC(NC(=O)CSc2cccs2)C1 CC1=C(C(=O)NCC(C)NC(c2cccc(-n3cnnn3)c2)=O)C(C)(C)CCC1 C1(NC(Cc2ccc(C)s2)=O)CCCN(C(=O)Cn2cc(C#N)cn2)CC1 C1(C(N2CCC(N3CCCCC3)CC2)=O)C(O)CCN1C(C1CC1F)=O C1(CC(=O)N(CCN(C(=O)CC2CC(=O)NC2=O)CC)CC)CCS(=O)(=O)C1 c1(C(C)C)c(C)sc(NC(=O)C(=O)N(C)CCC2COCCO2)c1C(N)=O N1(C(CC(COC)C)=O)CCC(F)C(NC(=O)CCOC2CCCCC2)C1 C1(C(C)C)CC(O)CN1C(c1c[nH]nc1CNC(C1COCOC1)=O)=O C#Cc1ccc(C(=O)NC2CCC(C)N(C(=O)C=C3CCOCC3)C2)c(F)c1 C1(OC)CC2(C(=O)NCCCN(C(=O)CCC3CCOCC3)C)CC12 CC1CN(C(=O)C(C)(O)C(F)(F)F)CCCN1C(=O)Cc1cc(F)c(N)cc1F N1(C(c2cnc(CC)[nH]2)=O)CCC(C)C1CNC(c1ccccn1)=O Cc1ncc2c(n1)CCC(C(=O)NC1CN(C(c3nc(C)n(C)n3)=O)CC1C)C2 c1(C(N2CC(CC(C)NC(=O)C(C)N(C)C)C2)=O)nc[nH]c2ncnc1-2 c1(CC)c(C(=O)N(CC(C)NC(C2OCCC2(C)C)=O)C)cnn1CC(C)C C1(NC(c2c(C)nn[nH]2)=O)COC2(CNC(=O)C(C)OCCN(C)C)CC1C2 C(C)(C(=O)N1Cc2ccccc2CO1)C1CC(NC(CC(C)SC)=O)C1 c1(NC(C2(c3cn(C(c4ccc(C5CC5)cc4)C)nn3)CCC2)=O)cnncc1O C1(C(=O)NCCn2cccn2)(CNC(C(C)OCC=C)=O)CCCO1 n1(CC)ccc(C(=O)NC(C)(CNC(=O)CC2CCC(C)(C)O2)C2CC2)cc1=O C#CC1(C(=O)N(C2CC(C)(C)C2)C)CCN(C(=O)C(N)=O)CC1 Cc1cc(Cl)c([N+](=O)[O-])cc1C(=O)NCCc1ccc2ccccc2c1 C#Cc1cccc(C(=O)NCC2CC(F)(CNC(=O)C=C3CCC(C)C3)C2)c1F C1(O)(C(C(=O)N(C2CCOCC2)CC#C)F)CN(C(=O)CCC2CC2CC2CC2)C1 CCCCCCCCC(=O)NCC(C)CC(=O)N(C1CC(O)C1(C)C)C c1(C(N2C3CCC(NC(C4C(=C)CC4)=O)(C3)C2)=O)ccc2ccn(C(C)C)c2c1 CC(CN(C)C)CC(=O)N1CCCC1CN(C)C(c1ccccn1)=O CC1(C)CCC2(CC1)CC2C(=O)NC1CN(C(=O)C(F)OC(F)(F)F)C1 C(=O)(C1Cc2ccccc21)NC1CC2CN(C(c3c(NC)cncc3)=O)CC2C1 S(=O)(=O)(c1cc(C)ccc1C)NC1CCCN(C(c2cc(C)[nH]c2)=O)C1 C1(NC(C(CCSC)NC(C(C)NC(=O)OC)=O)=O)CC2CCCC2C1 C1(CN(C(C2(OCC)CCC2)=O)C)CCN(C(=O)Cc2cc[nH]c2)CC1 C1(CC)(NC(=O)CC2CC=CCC2)CCN(C(c2cc(C)cnc2N)=O)CC1 N1(C(COCC(C)C)=O)CC2CC(NC(=O)CC3(C)CCOC3)CC2C1 Cc1cc(N2CCC3(CNC(=O)C3)C2)ncc1S(=O)(=O)NC(C)(C)CO C12(NC(C(CC)COC)=O)CCCC1(F)CN(C(c1cnc(OC)c(C)c1)=O)C2 c1(CC)n[nH]c(CC)c1CC(=O)NC1CCN(C(=O)CC2CCC(O)C2)CC1 N1(C(CC=C=C)=O)CCC(C(C)CNC(c2ccccc2)=O)CC1 C1(C(F)F)(CNC(C2CCN(CC)C2)=O)CCN(C(c2coc(C(N)=O)c2)=O)C1 c1(C(=O)NCC2(F)CC(NC(C3CC(C)C3)=O)C2)sc2cccnc2c1Cl C(C1=NOC2CN(C(=O)Cc3cccnc3Cl)CC12)NC(C(C#C)(C)C)=O C1(C(=O)NCC2(NC(c3cnc(C4CC4)s3)=O)CCCCC2)CCC2(CCC2)O1 Cc1cc(C(=O)NCC(c2ccccc2)CN)n2ncc(C#N)c2n1 Cc1nccn1C(C)C(=O)NCc1nc(CNC(=O)C(C)O)cs1 N1(CCCNC(C2(N(C)C(C3CC(O)C3)=O)CC2)=O)CCOCC1 N1(C(CN(C(C)C)C(c2ccc(CO)o2)=O)=O)CCCCCC1C c1(CNC2(c3n(CCOC)nnn3)CCN(C)CC2)nn(C)c2c1COCC2 C1(C)(C(N(CC=CC(=O)NCCC2CCN(C)C2)C)=O)CCCN1C c1(CC(=O)NC(CC#C)C(=O)NCc2cnn(C(C)C)c2)ccc(C#N)cc1 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)C2=CC3CCCC23)CC(C)(F)C1 c1(C(CC)(CN(C(c2cc(Br)c(C)s2)C(=O)NCC)C)CC)cccc([N+](=O)[O-])c1 C=C1CC2CCC(C1)N2C(=O)C(C)C(C)NC(c1ccc2occc2c1)=O Cc1nc2c(C(=O)NC3CN(C(=O)CC(=O)NCC4CC4)CC3C)ccnc2[nH]1 C(C(=O)N(C)Cc1sccc1C)(C(C)(C)C)NC(C1C(CC)C1)=O N1(C(C2N(CC)CC2)=O)CC(C2(NC(C3CCN(C)CC3)=O)CC2)C1 c1(C(N(CCNC(=O)C(C)Sc2ccccc2)CC)=O)cc(OC)c(F)c(F)c1 CC(CNC(=O)CC=CCNC(=O)CN1CCCCC1=O)C(C)(C)C c1(C(N(CCN(C(C2(C)COCCO2)=O)CC)CC)=O)cnc(O)c(C)c1 C1(C(N2CCCN(CCNC(C3(C#N)CC3)=O)CC2)=O)CCC2CCCCN12 N1(C(c2ccc(C#C)cc2)=O)CC2CC(NC(=O)CN(CC=C)CCO)CC1C2 C1(NC(CCSC)=O)CN(C(c2ccsc2Br)=O)C2(CCOCC2)C1 c1(C(N2CC(O)(C(C)NC(=O)CSc3nc[nH]n3)C2)=O)c(F)ccc(F)c1N C1(C(=O)NCC(CN(C(C(C)OC)=O)C)C)CCCC(F)(F)C1 N1(C(CC(=C)C)=O)CCCC1C1CCCCN1C(=O)C1=C(C)CCCC1 C1(NC(c2ncn(CC)c2)=O)CCOCC1NC(C1(Br)CC1(C)C)=O c1(C(=O)NC2CC3CC(NC(C(CCCC)O)=O)C2C3)cc(OC)cc(Cl)c1F c1(OC)cc(F)c(C(c2nnnn2C)NCC2CCS(=O)(=O)C2)cc1Br C1(CC(=O)N(CC(C2CCCCC2)O)C)CC2(C1)CN(C(c1cn[nH]c1)=O)C2 C1(C(=O)OCC)CCC2(CC1)CC(O)C2.N1(C(C(=O)NCC)=O)CC=C(CO)CC1 N1(C(C2CCN(C(=O)CCCCC3CC3)C2)=O)CC2C3CCC(C3)C12 C(C(F)C(=O)N1CCCC1CC(c1ccco1)O)C1CN(C(C2CC2(F)Cl)=O)C1 c1(C(=O)NCCCCCCNC(C2(CC)CCNC2=O)=O)ccc2nsnc2c1 N1(C(Cc2cccc(OC)n2)=O)CCCC2CCN(C(c3cnoc3C)=O)CC12 N1(c2c3scc(C)c3ncn2)CCCC(C2CC2NC(c2ccnc(O)c2)=O)C1 C1(C(=O)NCCC(C)(C)F)C(C2CC2)CCN1C(=O)C(F)C1CCCC1 C12(OC)CCCC1CN(c1nc(-c3ccc(OC(C)=O)cc3)no1)C2 c1(OC)ncnc(C(N2CCN(C)CC2CNC(=O)CN2CC=CC2)=O)c1F O=C1CCC(CCNC(=O)NC2CC2c2cccs2)C1 c1(CC(=O)NCCCNC(C2(C)CCCCO2)=O)ccc(C#N)cc1F c1(CNC(C=C(C)C(F)F)=O)ccc(CN(C)C(c2cncnc2O)=O)cc1 C1(N(C(=O)C(F)CC2CCC2)C)CCCN(C(=O)CCc2ncco2)C1 c1(OC)ccc(C(N2CCCCC2C(N2CCC2(C)C(C)C)=O)=O)cn1 N1(C(C2N=C(C)SC2)=O)CCCC(N(C)C(C2CC3(C2)CC3F)=O)C1 c1(CCCC)nc(C(=O)NCCC2CC(NC(C3CCS3(=O)=O)=O)C2)cs1 N1(C(COc2c(C#N)cccc2)=O)CCN(C(C2SCCCS2)=O)C2COCC12 C1(C(=O)OC(C)(C)C)CCCN1C(N1C(C(C2CCCO2)C)CC1)=O C12(CNC(CSCCOC)=O)CC1CN(C(=O)C(F)n1cccn1)C2 c1(CC(N2CC(CC=C)(NC(=O)CCC#CC)C2)=O)csc2c1CCCC2 c1(C(N2CCN(C(C3CCOC3)=O)CC2C(F)F)=O)[nH]c2ccc(F)cc2c1Cl C(CCCC(C(=O)NC(c1cn(CC)cn1)c1nnnn1C)C(C)C)(OCC)SC C1(CNC(CCc2cc(C)no2)=O)CN(C(=O)CCC2CC2(C)C)CCO1 C1(NC(CCOCCOC)=O)CCN(C(c2ccc(C)cc2)=O)CC1O N(C1CC2(CCN(CC(F)(F)C(F)F)C2)Oc2ccccc21)Cc1scc(C)c1 Cc1cc(C(=O)NCCOc2ccc([N+](=O)[O-])cc2)c(N)c(C)c1 C1(NC(C2CC(C)(CC)C2)=O)COC2(CCN(C(=O)Cc3cnns3)C2)C1 CC1(C(=O)NCCCCCNC(=O)COCC2(F)CC2)CCS(=O)(=O)CC1 N1(C(C2CCN(C(CSC)=O)C2)=O)CCC2CC(c3ccc(F)cc3)C2C1 c1(C(N(C(CNC(CCCCC#C)=O)C)CC)=O)cc(C)nc2ccc(Cl)cc12 C1(C(C)(C)C)CN(C(c2ccc(=N)[nH]c2)=O)CCN1C(=O)CN1CC2CCC1C2 c1(CN2CCC(CNC(c3cn(C4CCOC4)nn3)=O)C2)ccc(Cl)cc1 Cc1nc(C(N2CC(CCCCNC(C3(CO)CC3(F)F)=O)C2)=O)c(C)o1 C(=O)(CCS(=O)(=O)CC(C)C)NCC1C(CNC(c2c(C)cc(C(F)F)o2)=O)C1 C#CCC(C)(C)CNC(=O)C(O)CCNC(C1(C)CNC(=O)N1)=O CC1CN(C(C2CCC(=O)O2)=O)CCC1CNC(c1cc(Cl)ccc1Cl)=O C1(=CC(=O)NC2(CCCNC(C3CC(F)(CF)C3)=O)CC2)CCCCC1 C1(SCC)CCC2C(C1)C2(F)F.CCN=C1NCc2cc(no2)CN1 N1(C(C(C)C(C)(F)F)=O)CCN(C(c2ncn(C)n2)=O)C2CCCC12 CC(C)C(CNC(c1n[nH]c(O)n1)=O)NC(C1(F)CCCC1)=O N1(CCCNC(C23C(CN(C(c4ccncc4)=O)C2)C3)=O)CCS(=O)CC1 C1(NC(C2CCN(C(C)=O)CC2)=O)CC2CCC(C1)N2C(c1ncon1)=O C(=O)(C(F)CC(C)(C)C)N(C(C1CCCCC1)CNC(=O)C(c1ccccn1)O)C C(=O)(CCCC(=O)NOC(C)(C)C)NCC1CC(NC(C=CSC)=O)C1 c1(C(=O)NCC2C3N(C(C=C(C)Cl)=O)C(CC3)C2)c(F)ccc(O)c1F Cc1onc(-c2ccncc2)c1C(N1CCC1CNC(=O)C(O)CC1CC1)=O c1(N2CC(C)S(=O)CC2)nc2ccc(S(=O)(=O)NCCSCCF)cc2s1 c1(C(N2CCCC(NC(C3C(C#N)C3)=O)C2)=O)cncc2nc[nH]c12 c1(-n2ncc(C(=O)NCC(O)CNC(C3CC3C(F)F)=O)c2)ccccc1F C(=O)(CC(C)(O)C(F)(F)F)N1CCCC(F)(CNC(CN2C(C)CCC2)=O)C1 N1(C(C2C(c3c(C)cc(F)cc3)C2)=O)CC2CCC1CN2C(=O)C1=CCCOC1 Cc1nc(N2CCC2(C)C(N2CCC(C(F)(F)F)C2)=O)c2c(n1)CCC2 C(CS(=O)(=O)CC(=O)NCC1COCC1NC(C1CCC(=C(F)F)CC1)=O)OC C1(C(N2C(C)CN(C(c3ccsc3)=O)CC2)=O)CC12C1CC3CC(C1)CC2C3 c1(C(N2CC(C)C(NC(c3cnc(S)[nH]3)=O)C2)=O)ccc2nc(O)nc(O)c2c1 C1(NC(c2n(CC)ncc2)=O)CC(NC(=O)COCC(F)F)CC1O c1(C(=O)OC)ccc(Br)cc1NC(c1cc(-c2ccc(Cl)nc2)[nH]n1)=O Cc1cc([N+](=O)[O-])cc(Br)c1NCC1(c2ccccc2)CC1(C)C CC1CCc2[nH]nc(C(=O)NCC34CCCC3CN(C(=O)CSC3CC3)C4)c2C1 C1(NC(c2cc(=O)cc[nH]2)=O)CN(c2nc(Cl)ncc2Br)CC2(CCC2)C1 CCC(CC)C(C)C(=O)Nc1cnc(C(C)C)nc1C(C)(C)C C1(CC)(CC)CC(NC(=O)CC2(OC)CC2)CN1C(c1cc(OC)no1)=O CC1Cc2ccc(F)c(Br)c2CN1C(C1CN(C)CC1C(F)(F)F)=O CC1=C(C(=O)N2CCC(CO)C(NC(=O)C(C)(C)N(C)C)CC2)C(C)(C)CCC1 C(CC(C)C)(C(=O)N1CC2(CC(NC(=O)CC3CCCN(C)C3)C2)C1)NC(C)=O N1(c2nnc(-c3c(C)c[nH]n3)n2CC2CCOC2)CCC2(CCCN2C)C1 c1(C(CC)=O)ccccc1C(=O)NCCN(C(=O)C(c1c(C)noc1C)C)C N1(C(=O)CCc2ncccn2)CC2CCN(C(c3ccc4c(c3)CC4)=O)C2C1 C1(C)(C(N(CCCNC(c2cnn(CCN(C)C)c2)=O)CC)=O)CCCCC1 CC1(C)Cc2cc(C(=O)NC3C4CC3N(C(C3CC(C(F)(F)F)C3)=O)C4)sc2C1 C1(C(N2CCC(NC(Cc3n(C)ncc3Cl)=O)C2)=O)CCc2nnc(O)cc2C1 c1(OC)cc(C(=O)NC2CCC(CNCc3ccnc(F)c3Cl)CC2)ccc1O c1(-c2scc(C(N(CC(C)(C)CNC(C3CCC3(F)F)=O)C)=O)n2)ncccc1F C(=O)(CCCS(=O)(=O)N(C)C)NCC1N(C(C(CC)O)=O)CCC(C)C1 N1(C(COCC#C)=O)CC(=O)NC2CN(C(=O)CSCC(=O)OCC)CCC12 CC(O)CCCCCC(=O)NC1COCCC1NC(c1cnc(Cl)[nH]1)=O C1(C(N(C2CCCC2)CCNC(c2cc[n+]([O-])cc2)=O)=O)C(F)(F)C12CC2 C1(NC(C(C2CCOCC2)C)=O)CCCCN(C(=O)CC2CCOC(C)(C)C2)C1 Cc1cccc(F)c1CC(=O)NCC(CC(F)(F)F)NC(=O)C=CC(C)C C1(CNC(C(C(C)(C)C)O)=O)CN(C(c2cn3cccnc3n2)=O)CCC1(C)C C(=O)(NN1CCc2ccccc21)C1(C)CCC1.N1CCCC1C1CCCNC1 C(=O)(C(=O)N=c1cc(C)o[nH]1)N1CC(C)(CNC(C(C=C)O)=O)C(C)C1 c1(C(=O)NCCNC(=O)Cc2ccc(Br)nc2)cccc(CN(C)C)n1 Cc1noc(Cl)c1CC(=O)NC1CC(CCNC(=O)C=CCn2cncn2)C1 C1(C)(C(N2CC(COC)OCCC2)=O)CC(c2ccccc2Cl)=NO1 C1(OC)(CNC(=O)C(F)F)CCN(C(c2c[nH]cc2C(F)(F)F)=O)C1 n1(C(C(C)C)C)nc(-c2ccc(Br)cn2)nc1C(c1ccc(F)cc1)C N(C(=NCc1cc(Cl)n(C)n1)NC1CCCC1)NC(C)=O.C1(C(N)=O)(C)CC1 Cn1c(C(N2CC3CC3(CNC(=O)Cc3ccc(O)cc3Cl)C2)=O)cccc1=O CCC(CC)(CCNC(=O)C(C)OC(C)(C)C)NC(=O)Cn1ccc(C2CC2)n1 C1(CNC(C2OCCN(C)C2)=O)C2CCC(C2)N1C(=O)CCCN1CCCC1 c1(C(=O)NCCCCN(C(=O)CNC(=O)C(F)C2CCC2)C)ccccc1 Cc1nc(CNC(c2ccc(O)nn2)=O)oc1C(=O)NCc1nc(C#N)cs1 C1(CNC(C(COC)NC(C)=O)=O)CCCCCN1C(=O)C(C)=C1CC1 C1(c2n(CCSCC)nnn2)(NC2CCC(C(=O)NC)CC2)COC2(CCCC2)C1 CCCCCCC(C(=O)NCCCN1CCCC(N(C)C)C1)NC(C)C CCC(CCC(=O)NC(C)COC)NCCCC1(C)CC1 C=CC(C)(CCOC)C(=O)NC1CCCC1C(=O)NCc1nc(C)ccc1C CC(C)CCC(=O)C(=O)NC1CCCCC1CNC(=O)Cc1nccs1 c1(C(=O)NC2CCN(CCCC3CCCCC3)CC2)nc2ccccc2o1 c1(N(C)C)ccc(C(=O)NC2CCC2CNC(c2ncoc2C(F)F)=O)cn1 N12CCC(O)(C1)CCCC2=O.C(=O)(CCCc1cccs1)NC(C)(C)C c1(OC)cccc(Cl)c1CN1CC(C(O)CO)C1 n1(CC(=O)NCCC2CCCN2C(=O)CC2CCCC2O)cc2ccccc2n1 c1(CC)ncc(C(N2CC(CNC(C3CC3C(F)(F)F)=O)C(C)C2)=O)c(C)n1 N1(C(CCC=CC(C)C)=O)CCOC(CCNC(C2CC2C(N)=O)=O)C1 CCCCC(C)(C)NC(=O)CONC(C1(C)OCCO1)=O CCC(C)(O)C(=O)NC1CCC(CNC(c2cncc(N3CCCC3)n2)=O)C1 CC(C)(C)S(=O)(=O)CC(=O)NCCC1(C(=O)O)CC12CCC2 c1(C2C(C(=O)NCCN(C(C)C)C(c3nsnc3O)=O)C2)cccc(F)c1 N1(C(CC(CC)(C)C)=O)CCCC2(CCCN2C(=O)C#CC2CCOC2)C1 N1(C(CN(C2CC2)CC)=O)CC(C(N2CC[Si](C)(C)C2)=O)C(C)C1 c1(NCC(C)CNC(c2cc(S(N)(=O)=O)c[nH]2)=O)nc(Cl)nc2c1ncn2C N1(C(C(C)Sc2c(C)n[nH]c2C)=O)CCOCC(NC(C2(C)CC2(F)Cl)=O)C1 c1(C(N2CCN(C(c3c(=O)ccn(C)c3)=O)CC2)=O)cc([N+](=O)[O-])c(Cl)cc1Cl C1(C(=O)NCC(CNC(C(C)(C)C(N)=O)=O)O)CC2COCC(C1)C2 CC1CC(NC(c2c[nH]cc2Br)=O)CN1C(=O)Cc1sc(O)nc1O c1(C(=O)NC2C(NC(c3ccc(Cl)cc3O)=O)CCCC2)onc2ccccc12 O=C(CCC(F)F)NC1CC(CCNC(c2cccc(N3CCOC3=O)c2)=O)C1 CC1=CCC(C(N2CCCC(C(=O)NCC3(S(C)=O)CC3)C2)=O)CC1 C1(NC(CCNC(=O)C=CCl)=O)CCN(C(c2cnns2)=O)CC1O C(=O)(C(F)(F)CCNC(=O)C=C1CCC1)NCc1cn(Cc2nc(CC)sc2)nn1 c1(C(=O)OCC)coc(C(=O)NCC=CCNC(C2CCC(N(C)C)C2)=O)n1 N1(C(CCC(=O)OC)=O)CCCOC(CNC(=O)C(C)(C)N2CCCC2)C1 Cc1ccc(C#N)c(NC(C2CN(C(C3(CO)COC3)=O)CC2C)=O)n1 c1(C(C(C)NC(c2cccc(-c3n[nH]c(C)n3)c2)=O)OC)ccc(F)cc1 N1(C(C2(C=C)CCCCC2)=O)C2CCCC1CC(NC(=O)C(O)c1ccco1)C2 CC1CCc2c(F)cccc2C1NC(C1CC(=O)N(c2cccc(Br)c2)C1)=O C1(CC(=O)NCc2nc(CNC(C3C(=C)C3C(C)=O)=O)sc2)CCC(=O)NC1=O CCCC(C(=O)NCCc1cc(C(N2CCC(O)(C(C)C)C2)=O)no1)OC C1(CN(C(=O)Cn2cc(Cl)cn2)C)CCCN(C(C2CCC(N(C)C)C2)=O)C1 c1(OC)ccc2c(c1)NC(=O)C2NC(=O)C(N)Cc1ccc(Cl)s1 c1(C(=O)NC(CC)CNC(=O)CC2CC(F)(F)C2)cccc2ncc(Br)n12 C(=O)(C1=CCCOCC1)N1C(CNC(=O)Cc2ccn3cncc3c2)CC(F)C1 C=CCC(CC=C)C(=O)N1CC2CCC1C(NC(c1ccccc1Cl)=O)C2 C1(C(N2CCC(OC3CCCC3)C2)=O)Cc2cc(Br)ccc2O1 c1(C(N2C(C)CCC(NC(C3(CC=C)CC=CC3)=O)C2)=O)cc2n(n1)CCNC2=O n1(C(C(=O)NC(CNC(CCC(=O)NC)=O)C(C)C)C)c(C)cc(O)cc1=O C1(C(=O)NCCS(C)(=N)=O)CCOCC1NC(C1CCNC1=O)=O C1(C(=O)NCC2C(NC(CCC#C)=O)CC2)CCS(=O)(=O)N1 N#Cc1cnc(NC(=O)CC2CC3CC3C2)c(F)c1.N12CCCC(C1)C2=O C#Cc1c[nH]nc1C(=O)NOCC(N1CC(C(N)=O)(Sc2ccccc2F)C1)=O C1(C(N2CCC(N(C(=O)C(F)=C3CCCC3)CC)C2)=O)CC(C)(C)OC1(C)C C1(C#N)(C(=O)NCCn2ncc(C(=O)NC(c3csnn3)C)c2)CC2CC2C1 Cc1ncnc(C)c1CC(=O)NC1CCCC1NC(C1(C)C=CCC1)=O c1(C(N2CCC(CNC(=O)CCCc3nccs3)C2)=O)c(Cl)ccc(Cl)c1O Cc1cnn(C)c1C(=O)NCC(CC1CC1)CO c1(C(N(CC(C)C(N2CC=C(CO)CC2)=O)C)=O)cc[nH]c2nccc1-2 Cc1ncn(Cc2cn(CC(C)NC(C3CC4CCC3O4)=O)nn2)c1C c1(-c2ccc(COC)cc2)c(-c2cncs2)[nH]c2c(Cl)cccc12 CN=c1cc(C(N2CCC(F)(C(=O)NCC(O)CC(C)C)C2)=O)cc[nH]1 c1(C(=O)NCC(CN(C(CCC(C)OC)=O)C)O)cccc2nc(C(F)F)sc12 C1(NC(=O)Nc2c(OCC)cc(C)s2)CCCN(C2CCCCO2)C1=O N1(C(C2CN(C(C)=O)C2)=O)C(C(=O)NCc2nccs2)CC2CCCCC12 C1(C(=O)NCC2(CO)CCCC2)(CC)CCCN(C(=O)C(C)C(=O)OC)C1 Cc1cc(C)c(C(N2CCCCC2C2(NC(c3nc(O)c(C)s3)=O)CC2)=O)[nH]1 Cc1cc(Cl)c(C(N2CC(C)(C)CC2CNC(c2nc(C)c(C)s2)=O)=O)cc1C c1(C(=O)NC2CC(NC(=O)C(F)C3CCC3)C2)ccc(-c2cscn2)nc1 c1(NC(=O)NC(=O)NCC(=O)NCC(C)N(C(C2C(C)C2)=O)C)ccccc1 c1(C(=O)NC(CNC(C(CCC)C(C)C)=O)CC)ccc(O)cc1[N+](=O)[O-] Cc1cc(=NCC(C)(C(C)C)NC(c2[nH]c(C)nc2C)=O)[nH]c(Cl)n1 Cc1nc2cncc(C(N3CCC(CN(C)C(C4C(C)C4(F)F)=O)C3)=O)c2[nH]1 C1(C(=O)NCC2CC(C(C)C)C2)CCC(C)(C)N(C(C2CCCC(C#N)C2)=O)C1 c1(C(N2C(CN(C(c3c(C)coc3C)=O)C)COCC2)=O)cccc(Cl)c1Cl N1(C(CSCC)=O)CCC(C(C)C(=O)NC(c2nc(C)cs2)(C)C)CC1 C(=O)(CC(C)(O)C1CC1)NC1C(NC(c2cn(CCOC)nc2)=O)CCC1 N1(CC)CCCCC1C(=O)N(CC(=O)NC1CC(C#N)C1)CC1CCOC1CC C1(C(=O)NCC(=O)NCC(C2CCC2)NC(c2ccncc2)=O)CCCOCC1 c1(C(N2C(C(N(CCC(F)(F)F)CC)=O)C(C)CC2)=O)cnc(C)[nH]c1=N CCCC(CC(C)C)C(=O)NCC1CCN(C(c2c(C)cnnc2O)=O)C1 c1(OC)cncc(C=CC(N2CCC(O)(C(C)CNC(=O)C3=CCCC3)C2)=O)c1 c1(C(N(CCN(C(C2C(OCC)CCC2)=O)C)C(C)C)=O)cccnc1CC Cc1cc(C)c(CC(=O)NCCCNC(C2CCN(c3cnn(C)c3)C2=O)=O)s1 N1(C(C(C)=CC2CC2)=O)CC2CCN(C(C3CN(CP(C)(C)=O)C3)=O)C2C1 C1(C(=O)Nc2cc(F)cc(F)c2Br)CCC2(CN(CC(N3CCCCC3)=O)C2)O1 c1(C(=O)NC2CCC(NC(C(C)OCCOC)=O)CC2)ccc2c(n1)CCCC2 C1(O)(CN(CC(=O)Nc2cc(F)ccc2F)C)CCCN(C(=O)CS(N)(=O)=O)C1 C1(C)(C(=O)NC2CCC(NC(c3cc(C)nc(O)c3)=O)C2)CCCCC1(F)F c1(CC)cc(N)ccc1Cl.c1(C(CN(C(C)=O)C2CC2)=O)cnn(CC)c1 CC1CN(C(c2ncc(C3CC3)cc2F)=O)CCC1N(C)C(c1nonc1N)=O C#CCC(CC(F)F)C(=O)NC1CCCN(C(c2cc(C)ccc2CC)=O)CC1 N1(C(C)=O)CCCCC1C1CCCN(C(c2cc(C3(C)COC3)no2)=O)C1 c1(C(N2CCC(N3CCCC(SC)CC3)C2=O)=O)c2c(nn1C)CCCC2 Cc1cc(CC(N2CCC(NC(C3CCCS3)=O)C2)=O)nn1C C1(C(=O)NC(CC)CNC(c2nc(C(F)(F)F)cs2)=O)CC(=O)N(C)C1 C(=O)(C1SCCc2sccc21)N1CCC(NC(C2(C)CC3(CCC3)C2)=O)C1 c1(NC(C(N2CCCCC(CO)C2)c2oc(C)c(Br)c2)=O)cccc(Cl)c1C c1(C(=O)NCC(COC)NC(=O)C(c2cncnc2)C)cccc(OC)n1 Cc1ccc(C(=O)N(CC(O)CNC(c2cnccn2)=O)C)c2ccccc12 S(=O)(=O)(c1cc(Cl)cc(Cl)c1)OCCN(C(C1(NC)CCCC1)=O)C C(=O)(CCCC(=O)NC1CC1NC(=O)C=CBr)Nc1c(C)cccc1 N1(C(CCSCC)=O)CCC2(CC1)CCN(C(=O)C(C)(C)C(C)(C)O)C2 Cc1cc(CNCC2COCCN2C(=O)Cn2cc(C)cn2)cc(C)c1 N1(C(C(C)N(C(c2c(CCC)n[nH]c2)=O)C2CC2)=O)C(CO)CC2CCCC12 C(=O)(C1CCCc2nncn21)N(CCN(C(C(C#C)(C)C)=O)C)C(C)C C1(CNC(C(C)N(C)C)=O)CC(NC(=O)CC(=O)NCC(F)(F)F)CCO1 C(=O)(CCCCCCNC(C1CCC(F)C1)=O)N(C(C)C1CC1)CC c1(C(=O)NCC2(OC)CCN(C(=O)COC(C)C)C2)cnc2cc(C)ccn12 N1(CC)CCN(CC(=O)N(C2CN(C(=O)CC3C=CCC3)CC2O)C)CC1 CCC(CNC(=O)C(C)(c1ccccc1)OC)(CC)NC(c1coc(CO)c1)=O c1(-n2c(C)nnn2)ccc(C(=O)NCC2C3CN(C(C4CC(F)C4)=O)CC23)cc1 Cc1cc(CC(=O)NCC2CN(C(=O)CCn3cccn3)CCO2)cc(F)c1 c1(NCCS(CC)(=O)=O)cc(=NC(C)c2nc(C)oc2C)[nH]c(C)n1 C(C(CNC(=O)C=Cc1ccc(Br)o1)C(F)(F)F)NC(C(CC#C)C)=O C12CCC1NC(=O)C1(CC1)OCC(=O)N2C.C1(N(C)C)CCCC1 C=Cn1nccc1C(=O)NC(CNC(=O)Cc1ncc(C)s1)CC(C)C C1(NC(c2ccn(CCOC)n2)=O)CN(C(=O)C(C)(C)CC#N)CCC12CCC2 C=C[Si](C)(C)COC(c1ccc(N2CC(N)C23CCC3)cc1)=O Cc1cc(OCC(=O)NCCCC2(NC(C3(C4CCCO4)CCC3)=O)CC2)no1 NC1CCCCN(CC(N2CCC(C(=O)O)C2)=O)C1=O C1(C(N2C(CNC(c3cc(F)c[nH]3)=O)CCCCC2)=O)CCn2c(O)nnc2C1 C1(C(N(C)CC2(OC)CCC2)=O)CN(C(c2ccccc2COC)=O)CC12CC2 N1(C(C(C)C2CC2)=O)CCC(CCC(=O)NCCCCc2ncc[nH]2)C1 N1(C(COC)=O)CCCC2(CCN(C(=O)C(F)CC3CCCC3)CC2)C1 N1(C(c2n(C)ccc2)=O)CC2CC2(NC(C2CC(C(F)F)C2)=O)C1 C(=O)(C(C)(C)C(=O)NC1C2CN(C(c3cc(C(C)(C)C)oc3C)=O)CC12)OCC c1(C(=O)NC2CC(C)(NC(C(CCCC)CC)=O)C2)cnn2cccc(C)c12 c1(C(N(C)CC2CCN(C(C(=O)NCC)=O)C2)=O)cnn(C(C)(C)C)c1Cl c1(C(N2CC(CNC(C(C(C)O)(F)F)=O)N(C)CC2)=O)cccn2ncnc12 CC1(C)C=C(C(=O)N2CC(CCCCNC(c3cc4sccc4s3)=O)C2)C1 c1(C(N2CC3C(NC(C(C)n4ccnc4)=O)(C3)C2)=O)cc2ccncc2o1 c1(-c2scc(C(=O)NC3CN(C(=O)Cc4nnc(O)s4)C3)n2)ccccc1O C1(OC)CN(C(=O)COC(F)(F)F)C(C)(CNC(c2ccoc2C(F)(F)F)=O)C1 NS(=O)(=O)c1cnn(-c2ccnc(N3CCC(C(=O)NC4CCC4=O)CC3)c2)c1 c1(C(N(C2CCN(C(C3CCCO3)=O)C2)CC)=O)ccc(F)cc1F Cc1cc(F)c(S(=O)(=O)N2CCN(C)c3ccc(OC(F)(F)F)cc32)c(Br)c1 c1(C(COC(C2CCN(c3ccccc3)S2(=O)=O)=O)=O)ccccc1[N+](=O)[O-] c1(C(N(CCCCCCNC(C2(C3CC3)CC2)=O)C)=O)cnn2ccccc12 c1(SC)nn(C)cc1C(=O)NCCC1(O)CN(C(c2cn(C3CC3)nn2)=O)C1 C1(C(N2C(C(C)C)CCOCC2)=O)CN(C(=O)C2=CCC(C)CC2)CC12CCC2 c1(C(=O)OCC)ccccc1C(N1CC2CC2(C(=O)NCc2ccccc2)C1)=O c1(CC(N2C(C(C)(C)NC(c3scc(C)c3)=O)CCC2)=O)ccc2nonc2c1 C1(CCNC(c2ccncn2)=O)CSCCN1C(c1ccnc(F)c1)=O C1(C(=O)NCC(C(C)C)NC(C=CC=CC)=O)CCn2ccnc2C1 Cn1cc(CN2CCC(CC(=O)NCCc3sc(O)nc3O)C2)c2cccnc12 Cc1cc(C)c(C(=O)N(C)CCOCCNC(=O)CCC2CCC(=O)NC2)s1 c1(C(N2CCC(NC(C3ON=C(C)C3)=O)C2C)=O)ccc2occ(C)c2c1 O=C(C1=CCCOCC1)NC1CN(C(c2c[nH]nc2-c2ccoc2)=O)C1 c1(C(=O)NCCC2C(CC)CC2)cc2cccc(Cl)c2cn1 c1(C(=O)NC2C(NC(C(C)CC(C)(F)F)=O)CCCC2)ccc2c(c1)CNC2=O C(=O)(C1=CCC(F)(F)CC1)NC1CC2(CN(C(C3C(c4cn(C)nc4)C3)=O)C2)C1 C1(NC(CC2(C=C)CN(C(C3(C(C)C)COC3)=O)C2)=O)CC2CCCC(C1)C2 Cc1cc(C(=O)NCC(C)NC(c2nc3ccccc3s2)=O)c2c(O)n[nH]c2n1 N1(CC)CC(CNC(C2CCCCC2CNC(=O)C(O)c2ccco2)=O)OC1=O C(=O)(C1CCCCc2ccccc21)N1CC(NC(c2c(CC)scc2)=O)C1 N1(C(C(C)CC(N)=O)=O)CCCCC2(CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 C12(NC(c3cc(C)ncc3)=O)CCCC1N(CC(C)CC(C)C)CC2 C1(NC(=O)C(=O)NC(C2(O)CCCCC2)C2CCC2)CCc2nnnn2CC1 C1(OC)CN(C(c2cc(CN(C)C)on2)=O)CCC1CO.C12CC(C1)CC(=O)N2 C1(N(C(CC2(OC)CN(C(c3ccc(CC)cc3)=O)C2)=O)C)CCN(C)C(C)C1 CCCC(C)CC(=O)NCCOC1CN(C(=O)C(C2CCC(=O)N2)C)C1 C(CCC1CC1)(C(=O)NCC1COCC1O)NC(C(C)n1cccc1)=O C(=O)(N1CCC(C(=O)NC2CC(n3ccnn3)C2)O1)C1C(C)(C)CCO1 C(C1=NOC2CCCC12)NC(CN(CC#C)C(c1ccc(C)cc1C)=O)=O C1(NC(C(=O)NCC2CCCCC(=O)N2)=O)CC2CSCC(C1)C2 N1(C(c2n(C)ncn2)=O)CC2CCCC1C2CNC(C1(C)CC1C(F)(F)F)=O C1(NC(c2c(SC)n(C)nc2)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC1(C)C C(CC(C(C)(C)C)NC(c1csc(C(N)=O)n1)=O)N(C)C(c1[nH]cnc1C#N)=O CCCCC(C(=O)NCc1ccc(F)cc1O)NC(=O)C(C(C)(C)C)OC C(C(C(=O)NC(CCO)C1CC1)C(C)C)NC(c1n(CC)ncc1C)=O C1(O)(CNC(C2(CSC)CC2)=O)CCN(C(c2cc(C(F)F)on2)=O)C1 CC1(C)C(NCCc2ccc(O)cc2Br)CCN1C(=O)OC(C)(C)C C(=O)(CCCC(=O)OC)N1CCC(C)(C(=O)NC(CCC)c2ccco2)C1 C1(C)(C(=O)NCC2CN(C(c3cc(C)c(Cl)s3)=O)CC2(C)C)CCCCNC1=O Cc1cccc2[nH]cc(CC(=O)NC3CC3CNC(c3cn(C)nn3)=O)c12 N1(C(c2ccc(OC)nc2C)=O)CCN(C(=O)C=CC2CCCC2)C2(CCC2)C1 CC1CN(C(=O)CC2(C#N)CC2)C(C)CN1C(=O)CN1CCCC1=O c1(C(N(CCCCCCNC(=O)C(O)c2ccco2)C)=O)ccc2nc[nH]c2n1 C1(C(=O)Nc2ccc(Br)cc2F)CN(Cc2cncs2)CC(F)(F)C1 CC(CN=c1[nH]c(=NCCC2CCCC2(F)F)[nH]c2c1CCCCC2)N(C)C C1(COCC)CCCC1N=c1[nH]c(=NCc2cccc(C)c2F)[nH]c2ccsc12 C1(CC(=O)NC(COC)(C)CCO)C2CCC(C2)N1C(c1ccc(CO)cc1)=O N1(C(C2(C=C)CCC2)=O)CC(NC(=O)CC2CCOC2)C(C)(C)C1 c1(CCO)ncccc1CNc1ccccc1OC1CCC1 C1(C(=O)NCC2CCN2C(=O)C=CC2CCC2)CCCN(c2ccccn2)C1 C=CCCCCCCCC(=O)NC(CNC(c1cnc(C2CC2)o1)=O)CC=C N1(C(C2C(C)(C)C2)=O)CC(NC(C2CCN(CC(F)(F)F)CC2)=O)CC1CO c1(OC)ccc(C(=O)NCCNC(=O)COCc2ccc(C(=O)OC)cc2)nc1 c1(C(N2CCC(C(C)NC(=O)Cn3ncnn3)C2)=O)ccc(Br)cc1O c1(C(N2CC(OCCNC(C3CC(C)C3)=O)C2)=O)ccc2nc(C3CC3)[nH]c2c1 c1(C(N2CCC(N(C(c3cnc(C)[nH]3)=O)C)CC2)=O)cnc2c(F)cccn12 C1(C(=O)NCCCN(C)C(c2cccc(C3CC3)n2)=O)OC2CCC1C2 C1(CC)(NC(c2cc(COC)[nH]n2)=O)CCN(C(c2ncc(C)cc2F)=O)CC1 c1(C(N2CCOCC(NC(=O)C(F)C3CCC3)C2)=O)cc(=O)n2ccccc2n1 C1(NC(c2ccc(Cl)o2)=O)CCC2CCN(C(=O)C3=CCS(=O)(=O)C3)C1C2 Cc1ccc(NC2CCCCC2N2CCCC2)cc1C(C)(C)C c1(CN(C)CC2CCC(F)(F)CC2)c(O)cccc1C#N C(c1ccncc1)=C(C)C(=O)NC1COCC1CNC(C1(N(C)C)CCC1)=O c1(C(N2CC3N(C(c4c(CC)occ4)=O)C(CC3)C2)=O)cc(S(C)(=O)=O)oc1C c1(OC)ccc(C)cc1C=CC(=O)NC1CC2CN(C(c3ccsc3)=O)CC2C1 CCC(C)CC(N=c1[nH]c2c(C)cc(F)cc2s1)C(=O)O c1(OC)ccc2c(C(=O)NC3CC3(C)C(C)C)n[nH]c2c1F C(c1cc(Cl)ccc1Cl)=CC(=O)NCC1C2CN(C(C(C)(C)OC(C)=O)=O)CC21 CC1(C)CC(O)CN(C(C2CCN(C(=O)CN3CCCCC3=O)C2)=O)C1 c1(OCC)cccc(NC(C2C(O)CCN2Cc2ccc(COC)o2)=O)c1 Cc1nn(CCC(=O)NC(C)CNC(=O)CC(O)CN(C)C)c(C)c1[N+](=O)[O-] C1(N(C)C(c2cn(C)cn2)=O)CC2CCC(C1)N2C(c1ccc(C#N)o1)=O c1(C(C)NC(C)(CNc2ncccn2)C(C)C)cc(Cl)ccc1[N+](=O)[O-] c1(C(=O)NCC(C(C)C)NC(c2csc(Cl)n2)=O)ccc(-n2cnnn2)cc1 CC(C)CC(C)(CNC(C1(C)CCC1)=O)NC(C1CN(S(N)(=O)=O)C1)=O c1(C(=O)NC2(C)CN(C(c3c(OC)n[nH]c3)=O)C2)cc2n(n1)CCCC2O C1(CNC(C=CCC)=O)C2CCC(C2)N1C(=O)CCN1CCCCC1=O C#Cc1ccnc(C(=O)NCC(O)C(=O)NCc2cc(C)cc(F)c2)c1 c1(C(N(C)Cc2c(OC)cc(C#N)cc2)=O)ccc2cc(C(=O)OC)ccc2c1 c1(C(N2CC(NC(C3C(C)C3)=O)CC23CCC3)=O)ccc(S(C)(=O)=O)cc1N C1(C(N(CCCC#C)CCO)=O)CCCC(NC(=O)CC2CCC(=O)N2)C1 C(=O)(CCCc1cccs1)NC(C1CC1C(=O)NCC1(c2cnn[nH]2)CC1)C CC1CS(=O)CCN1C(=O)CNC(=O)CNC(C1CCCC(=O)CC1)=O C1(C(N(C)CCOCCC(=O)NCc2ccnc(O)c2)=O)CC2(CCC2)C1 c1(C(N2CC(O)CC(NC(C3CCN(C)CC3)=O)C2)=O)ccc(S(N)(=O)=O)o1 C(=O)(CC(C)CC(C)C)N1CC(CC(C)NC(Cc2cc(CC)no2)=O)C1 c1(C(CC)C(=O)NC(C)CCNC(C2CC2F)=O)ccc(OC)cc1 c1(C(=O)NC(CN(C(=O)C(C)OCC(F)(F)F)CC)C)c[nH]c2nccc-2c1C C(CC(C(N)=O)NC(c1cc(CNC(=O)Cn2ccnn2)nn1C)=O)OC C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(NC(c2cncc(C#C)c2)=O)C1(C)C c1(C(CCC)NC(=O)N(C2CC2)Cc2ccn(C)c2)cnn(C(C)CC)c1 C(C(=O)N(CCC(=O)N(C1CC1)CC1CCCC2CC12)OC)SC c1(C(=O)NC(C(n2ncc(C)c2)C)C)cccc([N+](=O)[O-])c1Br C12(NC(Cc3ccc(C)s3)=O)CCCC(NC(=O)C=C3CCN(C)CC3)(C1)C2 C#Cc1cccc(C(=O)N(C)CC2CCCCN2C(=O)C=CC(=O)N(C)C)c1F c1(C(N2C(CN(C)C(C3CC(C#N)C3)=O)CCC2)=O)cccnc1OC(F)F C(CN=c1[nH]c(=NCc2ccc3c(c2)OCO3)[nH]c2c1CC(C)CC2)=C(C)C C(N=C(NC1CC1)N1CCC(Br)=C(C)C1)c1cc(OC(CC)C)ncc1 C1(F)(CNC(CNC(C(CC)C)=O)=O)CCC(NC(c2cnn(C)c2)=O)C1 C1(CC)CN(C(c2cc(Cl)sc2Cl)=O)CC1NC(=O)CC(C)N(C)C N1(C(CC(CC)(F)F)=O)C2CCC1CC(CNC(C1CC13CCOC(C)C3)=O)C2 Cc1occc(=O)c1OCC(=O)NCC(C)(C)NC(=O)C=C1CCC1 C(=O)(C(F)C(C)CNC(=O)CCCN(C)C(C)C)N1CC(CCC)OCC1 N1(C(Cn2c(C)cnc2)=O)CC(NC(=O)CCc2cn[nH]c2)CC1C c1(CC)ncc(Cl)c(C(=O)NC2(C)CCN(C(=O)Cc3ccn(CC)n3)C2)n1 N#Cc1ccccc1C=CC(N1CC(NC(=O)Cc2ccsc2)C1)=O C(=O)(CCC(=O)C1CC1)N(CCCN(C(C=CC)=O)C)C CC(O)CCCCCC(=O)NCCN(C(=O)CC(C)CF)C c1(C(N2CC(C)(c3cn(CC=C)nn3)OCC2)=O)cc2c(nc1O)CCCC2O c1(-c2cn(CC(CCNC(CCOC)=O)(F)F)nn2)ccc(Cl)c(F)c1F CC1CC(C(=O)NCC2(CNC(=O)C(F)=CC3CC3)CCOCC2)CCO1 N1(C(CC(=O)OCC)=O)CCCC(F)(CNC(C2CCC(O)C2)=O)CC1 C1(CNC(C=COCC)=O)CCC2(CCN(C(=O)COC3CC3(F)F)CC2)CO1 C(CCC(C)CC(=O)NC1C2CC1N(C(c1cncc(C)c1Cl)=O)C2)=C(C)C CCCCC(CNC(=O)CCC(C)N(C)C)NC(c1cc(OC)n[nH]1)=O Cc1[nH]nc(Cl)c1C(=O)NC1CC(CNC(C2CCCCN2C)=O)C1 C(C(C)(C)CC(=O)NCCc1n[nH]cc1C(=O)N(C)CC1(O)CCC1)N(C)C CC(C)C#CC(=O)NC1(CCNC(=O)C(C)CC2CCCO2)CCC1 c1(C(=O)NCCNC(c2c(OC)ccc(CO)c2)=O)c(C)cc(=O)oc1C.C(C)(=O)N N1(C(C2C(=C)C2)=O)CCC(C2(NC(=O)CCC(C)CC)CC2)CC1 N1(C(c2ccc([N+](=O)[O-])s2)C(=O)NCC=C)CCCC1C1CCCCO1 C12(C(=O)NC(CC)(CNC(=O)C=CC(C)(C)C)CC)CCCN1S(=O)(=O)CC2 c1(C(=O)NCc2ccc(CNCC(C)O)cc2)c([N+](=O)[O-])cnn1CC(F)F C(CCC)(C(=O)N1CCCC1C1CCCN(C(c2n[nH]cc2Cl)=O)C1)=CCC C(=O)(C(C(C)C)C(C)C)N1CC(COC)(NC(=O)C(c2ccccn2)C)C1 CC(CNC(=O)Cc1csnn1)C(=O)N=c1ccn(C(F)F)[nH]1 C(=O)(C(C)(C)CCNC(c1cnn2c1OCC2)=O)NCc1c(CC)c[nH]n1 CCC(C)(C)C(=O)NC(C1CCCN1C(=O)CCc1cc(C)no1)C N1(C(=O)Cc2ccccc2NC(C2CCC3(CC2)CC3)=O)CCC2(CCCO2)C1 C(CCN(C)C)(C(=O)N1CC(N2CCOCC2)C1)NC(c1cc(CCC)on1)=O N1(C(c2c(C)nn(CC(=O)O)c2)=O)CCC(C2CC2)C1CNC(C1(SC)CC1)=O C(C(C)(CC(C)C)NC(=O)C(=Cc1ccc(Br)o1)C)NC(C1(C#C)CC1)=O c1(N2CC(COC)OC(C)(C)C2)ccc(S(=O)(=O)N(CC(O)C(N)=O)C)cc1Cl C1(C(N2CCC(NC(CC(=C)C)=O)C2C(C)(C)C)=O)COCC2(CCC2)O1 c1(C(=O)NC2CCN(C(C(C)(C)OC)=O)CC2C)c(F)ccc(C#N)c1F C(=O)(C(COC)(CC)CC)NCC(C(=O)NCC(C(CC)C)C)(C)CC Cc1nn(C)c(Cl)c1CC(N1CC(NC(C2(C3CC3)CC2)=O)CCC1C)=O CC1C(NC(c2ccoc2Cl)=O)CC2CCC1N2C(c1nnn2ccccc12)=O c1(CNC(N(C(C(CC)C)C)CCO)=O)nnc2ccccn12 N1(C(c2c(C)csc2C)=O)CC2CCC2(CNC(c2cc(F)c[nH]2)=O)C1 Cc1ncn(O)c1C(=O)NCC(O)CCNC(c1n[nH]c(C(C)(C)C)n1)=O N1(CC(=O)NCC(CC)NC(=O)CC(c2cccc(OC)c2)C)CC2CCC1C2 CCCCCC(C)CC(=O)NCc1ccc(N2CC(C)OC(C)C2)nc1 c1(C(C)=O)c[nH]c(C(=O)NCC2CC(O)(CNC(c3cncn3C)=O)C2)c1 C(c1cncc(O)c1)=CC(=O)C(=O)Cn1ccc(C(F)(F)F)n1.N N1(C(C=CCC)=O)C2CCCC1CC(NC(=O)C(C)c1cccs1)C2 Cc1sc(Br)c(C(=O)NCC(C(C)C)NC(=O)Cc2nc[nH]n2)c1C Cc1ccn2ncc(C(=O)NC3(CNC(C4CC5CCCCCCC45)=O)CC3)c2c1 Cc1nnc(N2CCCC(CNC(C3CC3(C)C)=O)C2)nc1C C1(CNC(C(CN(C)C)NC(CN(CC)CC)=O)=O)CC(C(N)=O)=NO1 C1(c2nnnn2C)(N(C(C)CC(C)O)Cc2ncc(C)s2)CCN(C)CC1 C1(OC)CCCC(NC(C2(CC3CCC3)CC2)=O)C1.C12CN(C1)C2=O N1(C(c2c(C)nc[nH]2)=O)CCCC(C2CN(C(c3sccc3C(C)(C)C)=O)C2)C1 c1(C(=O)NC2(CNC(C34CC(F)(C3)C4)=O)CC2)c[nH]c(=O)c2ccnn12 C1(NC(CCOCCOC)=O)CC(N=c2nc(CC3CC3)[nH]s2)C12CCC2 CC1CCN(C(=O)C=C2CCCC2)CC1CNC(=O)C(O)CC1CC1 C12(C(=O)NCC(C3CCCC3)NC(c3ccnc(C)n3)=O)CC(C)(C1)OC2C C1(CC)CCN(C(C2CCC2C#N)=O)C(C(=O)N(C2CCC(=O)N(C)C2)C)C1 Cc1nc(C(=O)NCCC2CCN(C(C3(N(C)C)CC3)=O)C2)co1 N1(C(C2(O)CCCC2)=O)CCOCC(NC(C2(F)CCOC2)=O)C1 C1(CC(=O)NCCNC(Cc2c(C)nc(C)s2)=O)COCC(C)(C)O1 C(=O)(CCCC(F)(F)F)N1C(CNC(CC2OCC(C)(C)OC2)=O)COCC1 c1(OC)c(C(=O)NC(CNC(c2ccccc2O)=O)C2CC2)nc(O)nc1O c1(C(=O)NCCC2CCN(C(C3(CO)CCCO3)=O)C2)ccnc2nccnc12 c1(CNC(N2CCOCC2C2CCNCC2)=O)cccc(C2(F)COC2)c1 C(CC(CC)C(=O)N1CCCC1CNC(=O)C(C)(C)c1ccno1)=CC N1(C(c2ccc(Br)cc2F)C(=O)NC(C(=O)OC)C)C2CCC1CN(C)CC2 c1(C(N2C(C(C)NC(CCCOC)=O)CCCC2)=O)cccc2ccncc12 CC(C)CCCCC(=O)NCc1c[nH]nc1C(=O)NC1CCCCCC1CO CC1(C)CN(C(=O)C=Cc2cccc(F)c2)CC1CNC(c1ccnnc1O)=O C(=O)(C(C)S(=O)(=O)C(C)C)NC(CCOC)CNC(c1cnn2c1OCCC2)=O C1(C(N(C(CC)COC)C)=O)CC(NC(C2CC(OC)C2)=O)C(O)C1 Cc1cc(=NCc2cc(C(F)(F)F)cc(Br)c2)[nH]nc1-c1ccccc1 C1(N(C(=O)CCCn2cccc2)C)CN(C(=O)C(O)Cc2cnc[nH]2)CC1(C)C C=CC1(C(=O)N(C)CC2(C)CCCO2)CCN(C(c2cccc(C)c2C)=O)CC1 N1(C(CN2CCC(C)CC2)=O)CCC(C2CC2)(NC(=O)CCC(F)(F)F)C1 N1(C(C2(OC(F)F)CCNC2)=O)CCC2(CCc3ccccc3C2=O)C1 C1(C(=O)NC2(CNC(c3c(C(C)C)ocn3)=O)CCOC2)CCC12CCC2 C=CC(C)(C)CC(=O)N1CCSCC1C(=O)NCC1COCCN1C C1(C)(C(=O)NCCNC(C(CC=CC)C)=O)CCCC(F)(F)C1 C(C(COC)N(C(=O)CN(C(=O)C(=O)C(=O)CN1CC=CC1)C)C)OC.N CC1(C)OCc2cc(C(=O)NCCCNC(=O)C3=COCCC3)ccc2O1 C(=O)(C(C)CCN(C)C)N1CC(C)(NC(C2C(C)C2)=O)C1 C1C(CO)(CO)NC(=O)N1C.N1(C(C)COC2CCOC2C)C(=O)CCC1=O N1(C(C)C(F)(F)F)CCC2CC(C(N3CCC(O)C(C)C3)=O)C2C1 c1(C(=O)NCC(CO)NC(CSCC)=O)ccc(=O)n(Cc2cccc(C)c2)n1 c1(CC(=O)NC(C(C)NC(c2c(NC)nccc2)=O)C)cnn2c1CCCC2 CC1NC(=O)CCC1CNC(=O)C(Cc1cn[nH]c1)NC(=O)CC1CC(=O)C1 N1(C(C2(P(C)(C)=O)CC2)=O)CCCC12CCCN(C(C1CCCOC1)=O)C2 C1(O)(CNC(C2CN(C(N)=O)C2)=O)CCN(C(c2sccc2CC#N)=O)C1 CCC(F)(C(=O)OC)C(=O)NCCCCCCN(C(=O)CCCC1CC1)C CC1CC(NC(c2c[nH]c(=N)o2)=O)CCN1C(=O)CNS(=O)(=O)N(C)C c1(SCCC(=O)NCCCN(C(C2C(C)C2)=O)C2CC2)nnnn1C1CC1 Cc1cc(C(N2CC(NC(=O)COCC3CCCC3)CC(C)C2)=O)c(N)c(Cl)n1 c1(C(N2CCN(C(CCC(=O)NC)=O)C(C)C2)=O)ccc(P(C)(C)=O)cn1 O=C(N=c1ccn(C2CN(Cc3cn[nH]c3)C2)[nH]1)c1ccc(Cl)cc1Cl c1(CC(=O)NCC(CC)(C)NC(=O)CC2CCCO2)cccc(F)c1 C(CC(C)C)(C(=O)NCC(C)(C1CCC1)NC(c1cc(C2CC2)n(C)n1)=O)OC C(=O)(CC1=CCCC1)N(CC(C)CNC(=O)CN(C)C(N)=O)C N1(C(c2c(C)cccc2)=O)CCOCC(C)(CNC(c2csc(Cl)n2)=O)C1 C1(NC(c2cccc(C3CC3)c2)=O)C2CCN(C(C3(F)CCCCC3)=O)CCC12 Cc1nc(Br)sc1NC(C1C2CN(C(=O)C=CC(=O)NC(C)(C)C)CC12)=O c1(OC)cc(CN(C2CN(C(=O)CCc3ccoc3)C2)C)cc2c1OCO2 C1(NC(c2c(C)nns2)=O)CCC2CN(c3ncc(F)cn3)CC2C1 N1(C(C(CNC(CCCCC)=O)(F)C(C)C)=O)CCC2(CNC(=O)O2)C1 Cc1nc(CCC(=O)NCCN(C(C2CCC(C)C2)=O)Cc2ccccc2)[nH]c1C N1(C(C2(C(=O)NC)CCC2)=O)CCC2CCN(C(c3cc(=O)cc[nH]3)=O)CC2C1 C1(C(=O)NC(CNC(CN(C)CC)=O)C)COCCN1CC C1(CNC(c2c(C)cc[nH]2)=O)CN(C(C2CCCCN2C)=O)CC1(C)C C1(C(=O)NCC(CCOC)NC(c2cncc(N3CCCC3)n2)=O)NC(=O)OC1C C1(CNC(c2ncn(C)n2)=O)COCCN1C(C1CC(CF)C1)=O CC(C)(CN=c1ccc2ncc[nH]c-2n1)NC(c1ccc(C(=O)N(C)C)cc1)=O N1(C(N=c2[nH]n(C)c(C(F)F)c2)=O)CC2COCC(C1)C(=O)N2 Cn1cc(C(N2CCC3OCC3C2)=O)c(O)nc1=O c1(C(=O)NC2C(C)CN(C(=O)CCC3CCC3)CC2)ccc(P(C)(C)=O)o1 CCCC(CC)CC(=O)N1C2CCC1CC(NC(=O)CC1COC(=O)N1)C2 C1(CNC(CC2(C=C)CCC2)=O)COC(C(F)(F)F)CN1C(=O)Cc1ccon1 Cc1nc(O)nc(C)c1C(N1CCC(C)C(N(C(=O)C(C)NC=O)C)C1)=O c1(CCC)c(C(=O)NCC2(F)CN(C(=O)C(C)CO)C2)[nH]c(C)c1C(C)=O N1(C(C2C(NC(Cc3c(C)nsc3)=O)COCC2)=O)CC(O)C(O)C1CO c1(C(N2C(CN(C(=O)CC3CCCC3)C)CCCC2)=O)c(Cl)ccc2c1OCO2 C#CCCCC(=O)NC(c1ccc(CN(C)CCO)cc1)=O.C12CCN(CC1)C2 C(CC(=O)NC1(C)CCCC1(F)F)(C(F)F)NC(CCCOC(C)C)=O C#CCCCC(=O)NCC(C)(CC)NC(c1ncoc1CCCC)=O N1(C(c2c(C)cc(CNC(CCC=C)=O)o2)=O)CC(=O)NCC1C(N)=O c1(C(N2CCCC(NC(C=CC=CC)=O)C2C)=O)ccc2nn[nH]c2c1 C(=O)(C(C)(C)S(C)(=O)=O)NC.N12CC(CC1C)NC2=O.n12cc(cn1)C(CC)C2 c1(C(=O)NCc2cc(C(N(C(C)CCO)C)=O)n[nH]2)cncc(CO)c1 c1(C2(NCC(=O)N(C)C=O)CNC2)cccc(Cl)c1.c1(C)noc(C(N)=O)n1 n1(CCN2CCC(CCc3ccc(F)cc3)C2)cnc2c1CCCC2 N1(C(COC(C)=O)=O)CCOCC12COCCN(C(c1cc(CO)c(C)o1)=O)C2 CC1CCC(C(N2CCCCC2CS(=O)(=O)NC)C(=O)NCC2CCOC2)CC1 c1(CNCCCCN2CCCC(NC(C)=O)C2)nc(O)c2c(C)c(C)sc2n1 C(c1cc(F)c(F)c(F)c1)=CC(=O)NC(C(C)C)CCNC(C1CN(C)C1)=O c1(C(=O)NC2(CNC(c3ccn(CCC)n3)=O)CCC2)cc(Cl)ccn1 C1(NC(CCC(=O)NC)=O)CC(F)CN(C(c2ccc(CCN(C)C)cc2)=O)C1 C1(NC(c2c(C)ncc([N+](=O)[O-])c2)=O)CCCC1N=c1cc(C(C)C)nc(Cl)[nH]1 c1(CC(=O)NC2C(CNC(c3ccc(C)nc3N)=O)CC2)nc2ccccc2[nH]1 N(C(=NCCc1cn(C)nn1)NCC1CC1)C(c1ccc(F)c(F)c1)C Cc1nc(Cl)ccc1CC(=O)NC1CCC(C)N(C(c2sccc2Cl)=O)C1 c1(C(N2CC(O)(C(C)NC(CCNC(C)=O)=O)C2)=O)c(C)noc1C(F)(F)F C(=O)(CCC(C)(F)F)N1CCC(C(C(C)C)NC(c2c(CC)scn2)=O)CC1 Cn1nc(C(F)(F)F)cc1CC(N1CC(CNC(C2(NC(N)=O)CC2)=O)C(O)C1)=O Cc1cc(C(=O)NC(C)CC(=O)N(C2CC(C)(C)C2)C)n(C)n1 c1(C(=O)NCCN(CC(C)O)C(=O)COc2ccsc2)cc2ccccc2nn1 c1(COC)n[nH]c(-c2cn(C(C)C(=O)NCCC(N)=O)nn2)n1 N1(C(CC(C)C(F)F)=O)CC2OCCN(C(c3cc(=O)c(O)c[nH]3)=O)C2C1 c1(OC)cc(C2(C(=O)O)CCCC2)c(OC)cc1S(=O)(=O)NCC(C)C#N Cc1nc(C2CC2)ccc1C(N1CCCCC(NC(c2coc(Cl)n2)=O)C1)=O CCC(C)C(O)CC(=O)NCC(C)(CC)C(=O)N(C)Cc1ccc(O)cc1 C(N=c1[nH]c(N2CCOC(CO)C2)nc2c1COCC2)c1c(C)c(Cl)c(Cl)cc1 c1(C(N2CC(SC)C(NC(=O)C=C(C)C(F)F)C2)=O)cc(C)c2nc(C)cn2c1 C1(NC(CCSC)=O)CCCCN(c2nc(Cl)ncc2F)C1 N1(C(=O)OCC)CCC(N=c2nc(CC(C)C)[nH]s2)CC1 c1(C(=O)NC(CCNC(C(CC2CCCC2)OC)=O)(C)C)cccc2scnc12 CC1CN(C(=O)C=Cc2cc[nH]n2)CCC1NC(c1cc(CO)ccn1)=O N1(C(c2ccc(CSCCC)o2)=O)CC2C(CN(C(=O)C=C3CCC3)C)C2C1 N1(C(C2(CCC=C)CCCC2)=O)CCN(CCCNC(=O)C(=O)NC2CC2)CC1 c1(-c2cccc(NC(N3C(CS(=O)(=O)NC)CC3)=O)c2)nnc2n1CCCCC2 c1(C(N2C(CNC(c3c(C)nc(CO)s3)=O)CCC2)=O)nc2n(c1Cl)CCCC2 C12(CC)CN(C(=O)C(F)=C3CCCC3)C(C(=O)Nc3c(OC)ccnc3F)(C1)C2 C(C)(C(=O)NNC(=O)c1ccncc1)n1cc(-c2cccc(C(=O)OC)c2)nn1 C1(NC(c2c(CC)cccc2)=O)CN(C(c2cnc(OC)nc2C)=O)C(C)(C)C1 C1(CN(C(=O)C(C2CCOCC2)OCC)CC)CCCN1C(C1C=CCCC1)=O C1(C(=O)NC(CCC)C)CCN(C(c2ccnc(C)n2)=O)C(C)(C)C1 c1(C(N2CC(NC(C3(O)COC3)=O)CC(F)C2)=O)c(O)cc(=O)n2c1CCCC2 c1(C(=O)NC(CCCNC(CC(CC)OC)=O)C)cc(=O)c2cc(Cl)ccc2[nH]1 C1(NCC)CCC(c2nnnn2C(C)(C)CC)(NCCC2CCCOC2)CC1 C(=O)(C(C(C)C)N(C)C)NC1(C(N(C(CCSC)C)C)=O)CC1 c1(-c2cc(C(N(C)CCO)=O)cc3c2cc[nH]3)cccc2c1OC(F)(F)O2 N1(C(CN(CCC#C)C)=O)CC2(C(N3CCCCC3CCO)=O)CC1CO2 C1(CCC(=O)NCCC(C(=O)OC)C)CCCCN(C(C2(Cl)CCCCC2)=O)C1 C1(CC)C(NC(=O)C(O)CC(C)C)CCCN1C(c1cnc(Cl)s1)=O CC1(C)CC(NC(=O)CC2CC2)CN(C(=O)COCCOc2ccccc2)C1 C1(CC=C)(C(N2CC(O)(C(C)NC(c3cnoc3CC(C)C)=O)C2)=O)CCCC1 C1(C2CC2)(C(N2CCC(CC#C)(C(=O)NC(C)CS(C)(=O)=O)C2)=O)CC(=O)C1 c1(OCC=C)ccc(C(N2CC(NC(c3oncc3CC)=O)CC2C)=O)cc1 C1(CNC(C(c2ccco2)NC(c2c(C)n(C)cc2)=O)=O)CCCC12CCC2 c1(C(=O)OCC)n[nH]c(=NC2CC(CCNC(C3(c4ccncc4)CC3)=O)C2)s1 C1(O)(C(C(=O)NCC(N2CCC(O)C2)=O)NC(c2c(C)csc2)=O)CCCCC1 CN1CCCC(c2cn(CCCN(C(c3c(Br)n[nH]c3Br)=O)C3CC3)nn2)C1 c1(C(=O)NC(C(C)NC(C2ON=C(CC)C2)=O)CO)cc2ccccc2c(O)n1 CC1CCN(C(c2cccc(CF)c2)=O)CC1CNC(=O)C1=CCOC1 N1(C(CN(CCC#C)C)=O)CC2CCC2(CC(=O)NCC(O)CN(C)C)C1 c1(CNC2(CC(=O)Nc3cc(-c4ccccc4)no3)CCC2)cc(O)nc(O)n1 N1(C(COCC=C)=O)CCC(C)(NC(=O)CSCC(c2ccc(F)cc2)=O)C1 C1(C)(CNC(CSCC)=O)CCCN(C(c2cncc(C3CCCCC3)c2)=O)C1 N1(c2n(CC(C)OCCOC)c(CO)nn2)CC2CCOC(=O)C2C1 c1(N2CCC(C)(OC)CC2)nc(N2CC(C)SC(C)C2)c2ncccc2n1 Cc1ccc(NC2CC2)c(C(=O)NCC(F)CNC(C2CC3C(C2)C3(C)C)=O)c1 C1(n2cnnn2)(CNC(=O)OC(C)(C)C)CCCCC1.c12conc1CS2 N1(C(c2n(C)ccc2)=O)CCN(C(c2scnc2C2CC2)=O)CC(C)(C)C1 C1(C)(CCNC(c2ccc(C)s2)=O)CCN(C(C2(Cl)CCCCC2)=O)C1 N1(C(CC2CC(C(=O)OC)C2)=O)CCC(NC(C2C(C3CC3)C2(F)F)=O)C(O)C1 C(c1nc2ccccc2[nH]1)=CC(N1CC2(CN(C(=O)CC3CC(F)C3)C2)C1)=O C(=O)(CC(O)CCSC)NC1(CF)CCN(C(Cc2cc(OCC)ncc2)=O)C1 c1(C(=O)NCC2(C(C)(C)O)CN(C(C(CCC)(C)O)=O)C2)cc2c(s1)CCOC2 C1(C2CC2)(C(=O)NCC(CN(C(c2nncc(OC)c2)=O)C)O)CC=CC1 N1(C(c2cc(C)c(Cl)s2)=O)CCC(CNC(C2CC(N(C)C)C2)=O)C12CC2 N1(C(c2n(CC)cnn2)=O)CCCC1C1CCCN1C(c1c(Cl)n[nH]c1C)=O Cc1oc(Cl)nc1C(=O)NCC1(F)CCN(C(=O)C(C)Cn2cccn2)C1 C(=O)(CC1=NN(C)C(=O)C1)NCC(C)NC(=O)Cc1ccc(F)cc1[N+](=O)[O-] CC(C)(CO)C(CO)NC(=O)CNC(=O)CNC(C1(F)CCOC1)=O CC(C)C(CCC(=O)NC(C1(O)CCCCC1)C)NC(c1ccc(F)cn1)=O C1(C(=O)NCC(CCCC)NC(CCC=C=C)=O)CC2(C)CCCN2S1(=O)=O C(=O)(C1=CCSC1)NC(c1n(C)ncc1)C(=O)NCC1(C)CC2CC2C1 c1(N(C(C)CCNC(c2scnc2C2CCCC2)=O)C)ccc2nncn2n1 c1(C(=O)NCC(C)NC(C(CCCC)c2ccccc2)=O)cccc2[nH]ncc12 CC1CCCC=C1C(=O)N(C)CC1CC(F)CN1C(=O)CCc1ccnc(Cl)c1 c1(CC(C)C(=O)N2CCC(CCNC(=O)C(F)=C3CCC3)C2)ccc(F)cc1 C(=O)(C1=NOC2(CCN(S(=O)(=O)c3cc(Br)c(F)cc3F)C2)C1)N(C)CC#N c1(C(=O)NCC(CNC(=O)CCCC(F)F)O)c(Br)ccc2n[nH]cc12 C(N=c1[nH]c(=NCC2OCCC2(C)C)[nH]c2cc[nH]c12)C1(CSC)CC1 N1(C(c2c(CC)nco2)=O)CCOC2(CCCN(C(=O)CCn3ccnn3)C2)C1 c1(C(N(CCCNC(c2[nH]cc(CC)c2)=O)C)=O)oc2ccccc2c1Cl C(=O)(C(F)CCC(C)(C)C)NC(C(=O)NCC(CCCC)CCC)C(C)COC c1(CC(=O)Nc2cccc(C(C)C)n2)csc(=NCc2cccc(CO)n2)[nH]1 C1(NC(c2c(CC)cno2)=O)COC2(CCN(c3ncc(C)c(O)n3)C2)C1 CN1CC(NC(=O)CCN(C(C23CC(C#N)(C2)C3)=O)C2CC2)C2(CC2)C1 c1(C(N2CC(O)CC(NC(COCCCC#C)=O)C2)=O)cc2c(n1C)CCOC2 C12(CNC(=O)C3CC3)CC1CN(C(c1ccnc(C(F)(F)F)c1)=O)C2 c1(C(=O)OCC)nc(C(N2CCC(CNC(C3CC(C)(C)C3)=O)C2)=O)c(C)s1 C1(C(N2C3CC(CNC(=O)CCC4CC4)C2CC3)=O)COc2ccccc2C1 N1(CCS(=O)(=O)N(C2CCC(C)CC2)CCO)CCC2(CC1)COC(CC(=O)O)C2 CCCCCCOC(C)C(=O)N(CCCN(C(=O)C(C)CN(C)C)C)C(C)C N1(C(CCc2c(C)ncs2)=O)CCCC12CCN(C(C1CC1C)=O)C2 Cc1cncc(C(=O)NC(CNC(=O)C(F)CC2CCCC2)CO)c1 C1(N(C(=O)CC2CC2(Cl)Cl)C)CN(C(C2CC(=O)C2C(C)(C)C)=O)CC12CC2 CC(CC(=O)N1CCN(C)C(CNC(c2cc3scnc3[nH]2)=O)C1)P(C)(C)=O Cc1scc(C(=O)NC2(CCC(=O)NC(C)C(O)C(C)C)CCCC2)c1C N1(c2nc(C)cc(CC)n2)CCC2(CCCCN(C(c3ccc(F)s3)=O)C2)C1 C1(CN(C)C(c2csc(CO)n2)=O)CCN(C(c2cscc2C2CC2)=O)C1 C12(NC(c3c(CC)nn(C)c3)=O)CCN(C(c3c(Cl)cnn3C)=O)CCC1C2 C1(CC)CCN(CC(N2CCCCC2C2(NC(C3CSC3)=O)CC2)=O)CC1 N1(C(C2(C)CCCC2)=O)CCC2(CCCC2C(=O)Nc2nnc(C(C)(C)C)o2)C1 C1(CC(N2C(C)COCC2)=O)OCC2CN(C(C3CCSCC3)=O)CCC12 c1(C(=O)NC2CCCN(C(c3cc(C(C)=O)on3)=O)C2)cc2ccncc2s1 N1(C(CC)=O)CCCCC1C(=O)N(C)CCN(C(=O)C(O)C1CC1)C(C)C CC1(NC(c2scnc2C(F)F)=O)CCC(NC(C2(C)CCOCC2)=O)CC1 c1(OC)cccc2c(C(=O)NC(C)CN(C(=O)CCc3ccoc3)C)coc12 Cc1cccnc1CC(=O)N(CCCCNC(C1CC2CC1CO2)=O)C c12ccc(cc1O)C1CC1C2=O.C(C(C)=O)COCC.C(COCCOCCOC)N C1(C(=O)NC2C(CNC(c3nc(OCC)sn3)=O)COC2)CCc2nn[nH]c2C1 CC1CN=C(N2CCN(C(c3nc(Cl)sc3Cl)C(=O)NC3(C)CC3)CC2)S1 C12(CNC(c3c(COC)ccs3)=O)CCC(CC1)N2C(c1sc(O)nc1C)=O Cc1c(C#N)sc(C(=O)NCCCOCC2CCOC2)c1C#N C12(C(=O)NCC(CNC(C(C)CCc3ccccc3F)=O)C)CCCC1CCC2 N1(C(CC(C)NC(COCCSC)=O)=O)CC(C)(C)OCC1C C1(CNC(C=CC=CC)=O)C2CCCC1N(C(=O)CN1C(=O)CCC1=O)C2 CC(C)(C)C(CNC(=O)C=CC=C(Cl)Cl)NC(C1CCOC(C2CC2)C1)=O c1(CC(=O)N(CC(CNC(CCN(C(CCC)C)C)=O)C)C)ccccc1F CC1CN2CCN1C(C(N1CC3(CC3)CC1CNC(=O)Cc1nccn1C)=O)C2 C1(C(=O)NCC2CN(C(C3CC3c3ccnc(O)c3)=O)C2)(CF)CC(F)(F)C1 N1(C(C(C(CNC(C(CCCC)(F)F)=O)C)F)=O)CCC2(COC(=O)N2)C1 c1(C(N(CCCCC(=O)NC(C(CCC)C)C)C)=O)cc[nH]c2nccc1-2 S(=O)(=O)(c1ccc(NCC2CCOC(C)C2)c(Br)c1)NCCC N1(C2CCN(C(C(N3CCC(C)CC3)C)=O)C2)CCC(NC(=O)CCF)CC1 C1(C(=O)NCC(CC)C#N)CCN(C(C2CC(C)(C)CO2)=O)CC1 N1(C(CCCOC(C)C)=O)CCC(C(C)NC(=O)CC2(N(C)C)COC2)CC1 c1(C(=O)NCC(CNC(CC(CC)OC)=O)O)cnn2cccc(C)c12 C(c1cnccc1C)=CC(=O)NCC(CNC(C1(SC)CCC1)=O)CO Cc1cc(N2CCC(CC(F)F)CC2)ncc1S(=O)(=O)NC(CO)C1CCC1 Cc1ccc2nc(C)cc(C(N3CCC(O)(CNC(=O)C(O)C(F)F)C3)=O)c2c1 c1(OC)n[nH]c(C(=O)NC2CC(NC(=O)Cc3cncc(C)c3)C(O)C2)c1Cl c1(C(=O)NCC2CCC(NC(=O)CCc3ncc[nH]3)C2)cnn2c1CC(O)C2 c1(C(=O)OC)n[nH]c(=NC2CC23CCC(NC(=O)CCC(=O)N(C)C)CC3)s1 N1(C(C(c2ccc(C(F)(F)F)cc2)(C)O)=O)CCC(F)(CNC(=O)C=C(Cl)Cl)C1 C=CC(CCC)CC(=O)NCCOCCN(C)C(c1cc(C)nn1CCC)=O CC1(C)OC(C)(C)C1C(=O)NCC1CCC(NC(c2ccc(O)nc2Cl)=O)C1 CC1CSCCCN1C(=O)CCCCNC(C1(NC(N)=O)CC1)=O Cc1cc(F)ccc1C(=O)NCC(C(C)(C)C)NC(=O)CC1CNC(=O)N1 c1(C(=O)NCC(CNC(C2CC(CC)OCC2)=O)C)cccc2nonc12 N1(C(CC(C(C)C)O)=O)CCC(C2CCOCC2)(CNC(c2ccoc2Cl)=O)C1 c1(N2CC(F)CC(NC(c3cccc(C(F)(F)F)c3)=O)C2)ncnc2sccc12 N1(C(CCNC2CN(C(C3CCC(CC)CC3)=O)C2)=O)CC(C)(CO)CC1(C)C Cc1c(C(=O)NCC2CCCN(C(=O)C=CCBr)C2)cccc1O c1(OCC(=O)OC2CCCC(C)C2)csc2nnsc12 Cc1nn[nH]c1C(=O)NCCOCCNC(=O)C(C1CCOCC1)F C#CC1(F)CCN(C(C2CC2CNC(c2csc(C(C)=O)n2)=O)=O)CC1 C1(CNC(=O)C(Cl)=CCl)CCN(C(c2cc(C(=O)OC)n[nH]2)=O)C1C C1(CCCNC(=O)Cc2ccccc2F)(NC(C(CC)O)=O)CCCCC1 CC#CCC(C(=O)NC1CC(O)(CO)C1)NC(c1ccoc1C)=O c1(C(N(CCC(=O)NC(C)CCC2CC2)CC=C)=O)ccoc1CC c1(OC)nc(C(=O)NCC2(NC(C3CCN3C)=O)CC2)sc1C Cn1nc(CNC(C2(CF)CCN(C(c3cc[nH]c3)=O)C2)=O)n(C)c1=O c1(C(=O)NCC#CCNC(C(CCCC)O)=O)nnc(O)c(Br)c1O N1(C(C#CCNC(c2ncnc(C)c2C)=O)=O)CCOC2COCC2C1 Cc1ccc(C2CCC2C2CCCNC2)c(C)c1.C(=O)C(F)Cc1ccccc1 n1(C(C)C(F)(F)F)nc(-c2cncs2)nc1-c1cnn[nH]1 CC(CC(=O)N(C)CCC1CCN(C(C2CCCC2C)=O)CC1)CC(F)(F)F c1(C(=O)NCC2CCCCN2C(=O)CC2CC(F)C2)cn2ccccc2n1 c1(CC)cccc(CC)c1C(=O)NCC1CCCCN1C(=O)C(C)C1(O)CCC1 Cc1cccc2c1OC(C(N1CCC(CCNC(C3(O)CC(F)(F)C3)=O)C1)=O)C2 c1(C(=O)OC)cc(OC)cc(C(=O)NCc2cncc(C3CC3)c2)c1C n1(CC)nc(C)c(C(=O)NCCC2CC(NC(=O)CC3COCCO3)C2)c1C c1(NC(c2csc(-c3ccnc(C4CC4)c3)n2)=O)cc(F)c(O)cc1Cl CC(CS(=O)(=O)c1ccc(F)cc1)C(=O)N1CCC(NC(=O)CC2CC2)C1(C)C c1(C(N2CCC(N(C(=O)CC3(CC(=O)OC)CC3)CC)C2)=O)cnc(C)[nH]c1=N Cc1sc(S(N)(=O)=O)cc1C(=O)NCCN(C(c1cc(CO)[nH]n1)=O)CC1CC1 c1(C(=O)NCC(CC=C)NC(=O)CCC2CC2(F)F)cc(Cl)cc(Cl)c1Cl CC1(C)C(NC(=O)CN2CCCC2=O)CCN1C(C1CCC=CO1)=O C=CC1CN(C(C2CN(C(=O)CSC3CC3)CC2CCC)=O)CCO1 c1(CC)ccc2c(CC(=O)NC3C4CN(C(c5csnc5C)=O)CC34)coc2c1 c1(C(=O)NC2CC(CNC(C(CC=C)C)=O)C2)cccc(O)c1[N+](=O)[O-] C1(OC)C=CCN(C(=O)CSS(C)(=O)=O)C1.n12cc(nn1)COCC2 C1(NC(C=CC(C)(C)C)=O)CCOC(CNC(C2CCCN2C=O)=O)C1 C=Cn1nncc1C(=O)NCC#CCNC(c1cscc1OC)=O c1(C(=O)NCC(CNC(CC(C(=C)C)O)=O)OC)sccc1S(N)(=O)=O c1(C(N2CC(n3cc(CCC4CC4)nn3)C(O)C2)=O)cc2cnccn2c1 C1(C(=O)NCCCNC(CN(C)C(=O)NC2CC2)=O)(CO)CCC1 C(=O)(CC(C(F)(F)F)n1cccn1)N(CCC)CCNC(=O)Cc1nc(C)cs1 CCC(C)(C(=O)NC(C)C(CO)NC(=O)C=CC=C(Cl)Cl)OC N1(C(CCCCC=C)=O)CCC(N=[N+]=[N-])(CO)C1.C1(N2CC2=O)CCOCC1F C1(C)(C(=O)NCCN(C(Cc2scc(C)n2)=O)CCOCCO)CCOCC1 c1(OC)nc(C(=O)NC(C)(CNC(=O)C(C)N(C)C)CC(C)C)cc(O)n1 C1(OC)CC(CNC(=O)CN2CCCNC2=O)N(C(=O)CCc2ncccn2)C1 C1(C(=O)NC2CCN(C(C(C)Oc3ccccc3F)=O)C2)CC2(COC(=O)N2)C1 N1(C(CCn2ncn(C)c2=O)=O)CCC(F)(CNC(c2cc(Cl)c[nH]2)=O)CC1 CC1CCC(C(=O)NCCC2CC=CCC2)N1C(C1CC1C1CC1)=O C=C(C)CC(C(=O)NCC(C)CN(C)C(C1(OC)CCCCC1)=O)OC C=C1CCN(Cc2ccc(OCC(F)(F)F)c(F)c2)C(C(F)(F)F)C1 Cc1nc2c([nH]1)CC(C(N1CC(NC(c3scc4c3CCCC4)=O)C1)=O)CC2 C1(O)(CCNC(CSCC)=O)CCN(C(=O)C=Cc2ccc(F)nc2)CC1 C1(C(=O)NC(C2CCN(C(C(C)n3cncn3)=O)C2)(C)C)CCCC2(CCC2)C1 Cc1sc(=O)n(CCC(=O)NCC2(F)CC(NC(C3CCCSC3)=O)C2)c1C Cc1ccnc2nc(C(N3CCC(O)(CNC(C4CC5CCC5C4)=O)C3)=O)nn12 c1(SCC(=O)NCC(CO)NC(C(C)c2ccco2)=O)ccccc1Br N1(C(C2OCCN(C(C)C)C2)=O)C2CCC1C(CNC(c1nncn1C)=O)C2 c1(N(CCCC)C)cc(N2CCOC(C3CC3)C2)nc(C)n1 CCC(C)(CCC(C)C)C(=O)NCCCN(C(=O)Cc1sccc1Cl)C c1(NCc2c([N+](=O)[O-])scc2)ccc(S(=O)(=O)NCC(O)Cn2cccn2)cn1 c1(OCC(=O)NC2C(NC(c3c(C)cc[nH]3)=O)C2)ccccc1[N+](=O)[O-] c1(CC)cnc(-c2ccc(C(C)NCCc3ccco3)cc2)nc1 C1(NC(C2(CCNC(c3scc(OC)c3OC)=O)CC2)=O)CC(C)(C)C12CCC2 C(CC(=O)C1CC1)OCCN(C(COCC(=O)NC)=O)C.C(CC)OC C1(C(=O)NC(CCC=C)C)CN(C(=O)COCCOC)CCN1C c1(C(=O)OCCC2CC(C)(C)NC2=O)c(Cl)cc(OC(F)(F)F)cc1Cl C(=O)(C1=C(C)CCCC1)NCC(CN(C(c1c(COC)cco1)=O)C)C c1(OC)ccc(Cl)c(F)c1C.C(CC(C)N(C(=O)Cc1nc[nH]n1)C)OCC(=O)N c1(NCC2C(F)COCC2)nccc(=NCCc2cccnc2Br)[nH]1 C(C(CN(C)C)N=c1cc[nH]c(=NCCCC2CCOC2)[nH]1)OC C1(CC=CC(=O)N2CCC2)(NC(c2cc[nH]c2C)=O)CCCC1.CCSC C(C(=O)N(C(C)C(=O)NCCN(CCCN(C)C)C)C)(C(C)C)OC C(C1=NOC2CCCC12)NC(COC1CN(C(C(CC)SC)=O)C1)=O c1(CC)cc(C(=O)NC2CCCC2NC(=O)C(C)C(C)(C)O)ccc1C c1(C(=O)NC(C)(CNC(c2cnco2)=O)Cn2cccn2)ccc2ccsc2c1 c1(C(=O)NCC(=C2CN(C(C(C#N)=CC3CC3)=O)C2)F)ccc2ccccc2c1O CC1(C)CCC(C(=O)NC2CC(O)C2)(NC(C2CCC(=O)O2)=O)C1 C1(C(N(C2(C#C)CC2)C)=O)(CNC(=O)C(C)C2(O)CCC2)CCCO1 CCC(C)(CC)C(=O)N1CC2(CCN2C(c2cc(C(=O)OC)on2)=O)C1 C(Cc1ccc(Cl)cc1)(C(C)(C)C)NCCCN(c1ccn(CC=C)n1)C C1(O)(C(=O)NCC2(F)CCN(C(CC3(C)CC3(F)Cl)=O)CC2)CN2CCC1CC2 C1(CC(=O)NCCOCCN(C(=O)CN(C)C2CC2)C)CC(F)(F)C1(F)F c1(C(N2CC(N(C(CC(C)SC)=O)C)C2)=O)cccc(CC(F)(F)F)c1 C1(C(=O)NCC(C)N(C(=O)CC2CCCCC2(C)C)C)Cc2cccnc2C1 C1(OC)CCCC(CNC(=O)C(C2CCCN(C(=O)CC3(C)CCC3)C2)(C)C)C1 C1(NC(C(C)OCCCC)=O)CCCCC1CNC(=O)C(c1ccccc1)F C1(C(=O)NCC2CCCCN2C(=O)Cc2sccc2Cl)Cc2nccn2C1 N1(C(CC(=O)OCC)=O)Cc2n[nH]cc2C1C(=O)N(C(C)C(N)=O)C C1(C)(NC(C2C(C=C)C2)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 C(N=c1ccc(Br)c(S(=O)(=O)NCC2CC2C)[nH]1)c1ccc(C)cc1F C1(OC)CC(NC(c2cccc[n+]2[O-])=O)CN(C(c2ncc(F)cc2C)=O)C1 N1(c2c(CC)ncc(F)c2)C(C)CCC(C(=O)O)C1C CCC(CCCC(=O)NC1CCC(NC(C2(COC)CC(=O)C2)=O)CC1)OC N1(C(c2ccc(C)c(Cl)c2)=O)CCOCC12CCN(C(C1(Br)CC1)=O)C2 N1(C(Cn2c(C)cc(C)n2)=O)CCC2CCN(C(=O)CCC=CC(C)C)CC12 C(c1ccccc1C)=CC(N1C(CC(=O)NCC(CSC)(C)C)CCCC1)=O C(=O)(C1=NOC(C)(C)C1)N1CC2C(CNC(CC(CC)CN(C)C)=O)C2C1 C(C(F)(F)CC(=O)OC(C)(C)C)NC(=O)NC1C(OC)CCC1 Cc1ccc(CN2CCCC(CC(=O)NCC3(O)CCCC3)C2)cc1 CCN(CC(C)NC(=O)OC(C)(C)C)N1CC(CC)C1 C1(NC(C(=Cc2ccco2)C)=O)CCCN(C(c2cc(C)n(C3CC3)n2)=O)C1C N1(CC)CCN(CCNC(=O)C(c2ccsc2)NC(C2CC3C=CC2C3)=O)CC1 C(=O)(C1=CCCCC1C)NC1CN(C(c2c(C)nc[nH]2)=O)CC12CC2 c1(CC)c[nH]nc1C(=O)NCC(C)N(C)C(C1(n2ccnc2)CCC1)=O c1(C(N2C(C(C)NC(=O)Cc3cccn3C)CCCC2)=O)nccc2occc12 CCS(=O)(=O)c1cccnc1CNn1c(C(N=c2cc(Br)n(C)[nH]2)C2CC2)nnn1 c1(OC(CC)C(c2cc(F)ccc2F)=O)ccc2c(c1)CCNCC2 c1(CC)[nH]c(Cc2ccccc2)cc1C(N1CC(C(=O)NC2SCCS2)C1)=O C1(CC)CSCCN1C(=O)OC(C)(C)C.C12CCN(C1=O)CCO2 C1(O)(CC(=O)NCC(C)(C)OCC(=O)NC2(CC#C)CC2)CCOCC1 N1(C(c2cnn(CC)c2Br)=O)CC2CN(C(=O)C(C)C(F)(F)F)CCC12 C(=O)(C(O)CC(F)(F)F)N1C(CCC(C)(C)NC(=O)CCC2CC2)CCC1 C1(C(=O)NCCCC(=O)N(CC(CC)C)CC)CC(O)C(F)C1 c1(CC(=O)NCC2(O)CC(C(=O)NC3(CSC)CCC3)C2)cc(C)ccc1C C1(NC(CC)=O)CCCCCC1C(=O)NCC(C)(C)C(=O)NC c1(CC)cccc(C(=O)NCC(C(=O)NC(C2CCOC2)C)N(C)C)c1 N1(Cc2cnn(C(C)C)c2F)CCC(O)(CO)CC1 CCCC(C(=O)N(CC(O)CN(C)C(C12CCC(CC1=O)C2)=O)C)C(C)C C(=O)(C(CC(C)C)C(N)=O)N1CCN(C(c2c(C)nc(=N)[nH]c2)=O)CC1C(C)C C(=O)(CC1=CCCCC1)Nc1c(C)ccc(C)c1.N12CC(C1)NC(=O)CC2 Cc1cc(C(N2CC(CNC(C3(C)CCN(C)C3)=O)C(C)(C)C2)=O)cc(C)c1F C(C(=O)NCC(C)NC(c1cnc(Cl)c(Cl)c1)=O)(C(F)(F)F)OC(C)=O Cc1ncc(C(=O)NC2CCN(CCNC(=O)C3=CCCOCC3)CC2)c(=N)[nH]1 C1(C(N2CC(C)(NC(C3CC3c3cnn(CC(=O)O)c3)=O)C2)=O)CCCC(F)C1 CC(C)C(C(=O)N(CCCNC(c1cnn(C)c1)=O)CC1CCCC1)C1CCC1 CCCCCCCCOCC(=O)NC1CC1NC(=O)CCc1nnc(C(F)F)o1 O=C1NCC(C(N2CCC2CNC(=O)C(=O)NCC(F)(F)F)=O)N1 c1(CC(=O)NCCC(C)NC(C2(N(C)C)CCCSC2)=O)cc(F)ccc1O c1(CNC(C(C2CCN(C(CC3(OC)CCC3)=O)C2)F)=O)ncccc1Cl C1(C2CC2)(C(=O)NC(C#C)C2CCC2)CN(C(c2cc[nH]c(=N)n2)=O)C1 C(=O)(C(C)(F)C(=O)N1CCCC(N(C)C(c2ccc(C)cc2)=O)C1)OC n1(C(C)C2CC2)nc(-c2ccccc2)nc1C1CC1C1CC1 Cc1ncc(Cl)cc1C(=O)NC1CN(C(=O)C(C)(C)c2ccns2)CC1O C1(CNC(=O)Cc2cccnc2)CC2CCC(C1)N2C(=O)CN1CCOCC1=O CC(C)(O)C(=O)NC1(C(=O)NCCC2CC(F)(F)C2)CC(CO)C1 C(CC(C)C(C)(C)C)NC(CC(CNC(C(C)OCC=C)=O)C1CCC1)=O c1(CC)cc(C)c(C(=O)NC2(C)CCN(C(C3(C(=O)OCC)CC3)=O)C2)o1 N1(C(CSC)=O)CCN(C(c2c(N)sc(C)c2C)=O)CC1c1cn[nH]c1 N1(C(C(C)C)=O)CCN(C(=O)CC(=O)NC2CC2)C(c2cccc(Cl)c2)C1 c1(OC)ccc(Cl)cc1S(=O)(=O)N(C)CC1CCN(C(c2sccc2Cl)=O)C1 c1(C(=O)NC(C(=O)NCCC)C)ccc(Oc2ccc(Cl)cc2)cn1 C=CC1(C(N2CC3CC(C2)N3C(=O)CCC#CC)=O)CCCCC1 C12(C(N(C(C)C(=O)NCCc3ocnc3CO)C3CC3)=O)CCCC1CCC2 C1(C(=O)NCCCN(C(=O)CC(c2ccccc2)OC)CC)CCC(C)(C)CC1 Cc1cn2ccc(C(=O)NCC3(F)CC(NC(C4CCCCC4C)=O)C3)cc2n1 N1(C(C(CC)O)=O)CC2(CCC(CNC(c3cc(Cl)c(Br)c(Cl)c3)=O)O2)C1 c1(CN(CCC)CCNC(=O)CCNC(=O)CC2C(C)C2(F)F)cc(C)nn1C N1(C(C2C(C)CCC2)=O)CCCC1(C)C(N1CCCC1C#N)=O N1(C(C2C(C)C2)=O)CCC(NC(c2ccc([N+](=O)[O-])cc2Cl)=O)C(F)(F)CC1 C(=O)(C(C#N)C(C)(C)C)OC1CC(NC(COc2cc(C)c(O)nc2)=O)C1 C(C1(C)CCc2cc(Br)ccc21)NC(CC1CC(C)(C)CCC1C)C(=O)O Cc1c(F)ccc(C(N2CC(NC(C3CC3C)=O)C(C)C2)=O)c1F C(=O)(C1=CC(O)C(O)C(O)C1)NC(C(Cc1ccc(C(C)C)cc1)N(C)C)=O C1(NC(C(C)OC)=O)(CNC(c2[nH]c(C)nc2C)=O)CCCCC1 c1(Nc2nc(C)nc(N3CCC4CCN(C)CC34)c2)ccc2c(c1F)CCNC2=O C1(C)(C(N2CC(F)(CNC(COCc3cc(C)no3)=O)C2)=O)CC(=O)N(C)C1 c1(N2C(C)(C(=O)Nc3cc(C)cc(Cl)c3)CC2)ncnc2occc12 CCC(CC(=O)NCCCCC(=O)N1CCC(CO)C1)OC c1(OC)nc(Cl)ccc1C(=O)NCC1(C)CCCN1C(=O)C1CC1 C(CN=[N+]=[N-])(C(=O)N1CCCC1CCCO)NC(C(SC)SC)=O N1(C(c2noc(CC)c2C)=O)Cc2ccccc2C(NC(c2nccn2C)=O)C1 N1(C(CC=C(C)C)=O)CC2CCN(C(C3COC4(CCC4)C3)=O)C2C1 N1(C(c2cc(CC)c(C)cc2)=O)C2CCC1CC(N(C)C(c1coc(C)c1)=O)C2 N1(C(c2nc(OC)nc(O)c2)=O)CC(C)(C)CCC1CNC(c1nocc1C)=O c1(C(=O)NC2(CC)CC2)conc1C(C)NC(=O)CC(C1CC1)C1CC1 CC(=O)CC(C)(C)C(=O)NCC1CCCN1C(c1cnn(CCC(C)C)c1C)=O c1(NC(c2cc(C(CC)C)no2)=O)nc2c(s1)CS(=O)(=O)CC2 c1(C(=O)NCC(C)(C)NC(CC(C)F)=O)nc2ccccc2cc1Cl CC1CCN(C(=O)CCC2CCCO2)CCC1c1ccccc1.CCCS(C)(=O)=O N1(C(c2c(C)c(Br)no2)=O)CCN(C(c2ccccn2)=O)CC1C(C)C N1(C(CC2(NC)COC2)=O)CCC2(CC1)CC(NC(=O)C(C)n1cccn1)CO2 c1(C(=O)NC(C2CN(C(c3ccnc(S)c3)=O)C2)C)ccc2c(c1)COCO2 CCN=C(NCC(=O)Nc1ccc(NC(=O)OC(C)(C)C)cc1)NCC c1(C(=O)N(CCO)C2CC2)ccc(-c2ccncc2)cc1F CC1CN(C(C2(c3ccccc3F)CC2)=O)CC1CNC(=O)C(C)NC(N)=O C1(CNC(CCNC(N)=O)=O)CN(C(=O)C(O)C(F)F)CCC12CCC2 c1(NS(CCCC)(=O)=O)c(F)cccc1C#N.C12CCN(C1)C2=O N1(C(C2OCCN(CC)C2)=O)CC2CCCC2(CNC(=O)C(F)(F)CO)C1 N1(C(c2c(COC)scc2)=O)CCC2(CC(NC(=O)C(Cl)=CCl)CO2)C1 CCC(C(=O)NC(C1CCCN1C(c1cccc(Cl)c1F)=O)C)C(C)C C1(CNC(CC2(CC)CCC2)=O)CC(C(=O)NCC(C)(O)CN(C)C)=NO1 C1(C(=O)OC)CN(C(c2cc(Br)co2)C(=O)Nc2c(C)cccc2C)CC(=O)N1 C1(CNC(CC(C)(C)C)=O)CC2COCC2N1C(c1cccc(Br)c1)=O Cc1c(C(=O)NC2CC2NC(c2ncoc2-c2ccco2)=O)cncc1N C1(CC)CN(c2ccnc(NCc3cc(C)cc(F)c3)n2)CC(C)(C)O1 n1(C(C)CNC(=O)N(C)C)cc(C2CC(N(C(=O)C(C)N(C)C)C)C2)nn1 N1(C(C(C2CCC(=O)N2)C)=O)CC2(C1)CN(C(c1ccsc1C(F)F)=O)CCO2 c1(C(N(C)Cc2c(C)ccs2)=O)coc2c1CN(C(=O)C(c1cnn(C)c1)O)C2 c1(C(N2CC(CCNC(=O)Cc3cocn3)OCC2)=O)ccc(F)c2occc12 c1(C(=O)NCC2C(C)(C)N(C(c3sc(F)cc3Cl)=O)CC2)ccnc2[nH]cnc12 c1(OC)cccc(C(=O)NC(C(=O)NC(C)COC(C)C)c2ccco2)c1 N1(C(C(C)OCCCC)=O)C(C(=O)NC2CN(CC)CC2C)CCC1C(C)C C1(C(=O)NC2C(C)CCN(C(C(CC)(C)CC)=O)C2)Cc2ccccc2O1 N1(C(c2cnc(CCC)s2)=O)CCC(NC(=O)COCc2nc(C)no2)C1CC C#CC1CCC(C(=O)NCCCC2CCCN2C(c2cc(SC)c(C)o2)=O)CC1 C1(C(N(C(CO)CCS(C)(=O)=O)C)=O)Cc2ccncc2C1 C(N=c1[nH]c2cccnc2s1)C1(CNC(CCCCOCCC=C)=O)CC12CCC2 N1(C(C2CCCN(C(C3C(C)OCC3)=O)CC2)=O)CCCC2C1CCN2C C(=O)(C(C)C(=O)NCC=CC(N1CC(C)(C)C1C(=O)OC)=O)OCC C1(NC(=O)NCCOC2(C#N)CCC2)CCC2C1C2(F)F C(=O)(CCC(=O)NC(C)CC(C)NC(=O)CCOC1CCOC1)NCCC C(=O)(C(C)(O)CCC)N1CCCC(N(C(Cc2nc(CC)sc2)=O)CCF)C1 C1(C(C)(C)C)CCN(C(=O)CC2CC23CC3)C(CNC(=O)C2=CCCCC2)C1 c12cc(ccc1[N+](=O)[O-])N1CCCC(CC1)N2C(=O)CCC1CC1.CCOCC c1(C(=O)NC2CN(C(C3(OC)CCC(C)C3)=O)C2)c(C)cc(C)cc1O c1(CCNC(=O)CCC2(NC(c3ccon3)=O)CCCC2)ccc(F)cc1 C1(C(=O)NC2CCC(NC(c3c(C)nn(C)c3)=O)C2)CC(C)CC(C)(C)C1 CCCC(O)CC(=O)NCC(CC)NC(c1cc(Br)ccc1N)=O N1(C(C(C)CC(F)F)=O)CCC(CNC(=O)CC(C)(C)C)C(C2CC2)C1 CC(C)CC(O)C(=O)NC12CC1CN(C(=O)CCc1ccccc1Cl)C2 C1(C(=O)NC(C(=O)OC)Cc2[nH]cnc2C)OCCCN1C(=O)OC(C)(C)C C=CCCCC(C(=O)N1CCC(C)(CCO)CC1)NC(c1ncccc1C)=O N1(C(c2c(C(C)NC(=O)C(C)(F)C(C)(C)F)noc2)=O)CCC2CN(C)CCC12 C(=O)(C(C)CCC(C)(C)C)NCCC(=C)CNC(c1ccc(F)cc1Cl)=O C=CCC(C(=O)NCC1C(CNC(C2(F)CC(COC)C2)=O)C1(F)F)N(C)C c1(OC)cccc(C(=O)NC2(C(=O)N(C3CC3C)C)CCC2)n1 Cc1cc(C(=O)NC2CCC(NC(C3(C#N)CCC3)=O)C2)c(C)n1-c1ccon1 N(C1CC(C)(C)Oc2ccc(F)cc21)C(=O)NCCS(CCOC)=O C12(C(=O)NCCC(Cn3cc(C(COC)(C)O)nn3)F)CCCCC(F)(C1)C2 c1(C(N(C(C)CCN(C(=O)CC2CCCO2)CCO)C)=O)cc(C2CC2)on1 C(C(=O)N(C)C)(C(C)O)NC(=O)CN(C(c1c(C)ccs1)C(=O)NC1CC1)C C1(CNC(c2n(CC=C)ccc2)=O)CCCCC1NC(c1ccoc1C1CC1)=O CC#CCCC(=O)NC1CC1NC(=O)CCOCC(F)(F)C(F)F N1(C(c2cnc(OCC)nc2)=O)CCC(C)(C)C1CNC(c1ccnn1CC)=O Cc1cc(C#N)c(O)nc1NC(N1CC(C)c2ccccc21)=O C1(CCNC(C2(CC=C)CCC2)=O)CCN(C(=O)C(C)OCC2CC2)CC1(F)F Cc1ccc(OCC(=O)N(C)CCNC(C2CCC(=O)O2)=O)cc1 CCCC(C(=O)NCC1CCCCC1NC(=O)C(F)OC(F)(F)F)NC(N)=O N1(C(Cc2ccc(C(=O)OC)nc2)=O)CCN(C(C2COCC2O)=O)CC1CO CCC(O)C(C)C(=O)NC1CC(NC(=O)C=C(C)c2ccccc2)C1 N1(C(C2CCCC(NC(COCCCCC)=O)C2)=O)CCC12CC(COC)C2 C(C(=O)NCCN(C(=O)CCc1ccncc1)C)(C(C)C)NC(COC)=O c1(C(N2CCN(C(c3c(Cl)ncc(C)c3)=O)C(C)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 Cc1ccsc1C(=O)NCC(CO)NC(=O)CSCC1CCCO1 C1(NC(CCSC(=N)N)=O)CC2CC1CN2C(=O)C(=O)Nc1ccc(F)cc1 CCC(Cc1cccc(C)c1)N=c1ccc2ncc[nH]c-2n1 C(=O)(C1CCCc2ncnn21)N1CCC(N(C(c2ccnc(C(C)C)n2)=O)C)C1 C1(C(=O)NCCOCCN(C)C(c2cc(C(C)(F)F)n[nH]2)=O)CCC=CCCC1 N1(C(C(C)(C)C2CC2)=O)CCC2CCN(C(C34CC(F)(C3)C4)=O)C2C1 CC(O)CC(=O)N1CC(NC(c2cc(C(F)F)[nH]n2)=O)C1 N1(Cc2cn(-c3ccnc(C(=O)O)c3)nn2)CCCN(C2C(C)CC2)CC1 N1(C(C2(CC(C)C)CC2)=O)CC2CC(C1)CN(C(C1CCCC(C)(C)O1)=O)C2 N1(C(C(C)CN2CCOCC2)=O)CC2CC1C2NC(c1cn(CC(N)=O)nn1)=O C1(C(C2(O)CCC2)C)CCCCN1C(=O)C(C#N)=CC(=O)N(C)CC1CNC1 Cc1cccc(C(N2CCCC2C(C)(C)CNC(C2CC23CCOC3)=O)=O)c1F c1(C(=O)OCc2ccc(OC3CCCCC3)nc2)ncc2c(n1)CCOC2 N1(C(c2cnc(NC(C)=O)o2)C(=O)NCC=C)CC2CCCCCC2C1.C(C)(C)(C)O N1(CCC(=O)Nc2cn(-c3ccc(C)cn3)nn2)CCS(=O)C(C)(C)C1 c1(C(N(CC(CNC(C(C)SCC)=O)C)C)=O)ncc2n1CCCC2 CC1(C)CCCCC(C(=O)NC2CCC(NC(=O)CSCC(F)(F)F)CC2)C1 C1(C)(C(N2CCC(=CCNC(c3c(C)nn(C)c3)=O)CC2)=O)CCCCC1C C(=O)(NNc1cccc(Cl)c1)C1C2CN(c3ccnc(OCCOC)n3)CC21 CCC(CC)(CCNC(c1ccco1)=O)NC(=O)C(c1nc(F)ccc1Cl)C C(=O)(CC1OCCc2sccc21)OCc1nc(CC)on1 C1(C(N(C2CC(NC(C3(F)CCOC3)=O)C2)C)=O)CCN(C2CCSC2)CC1 C1(C(N2CC3C(C(=O)OC)(C3)C2)=O)C2C(CN1C(c1sccc1OC)=O)C2(C)C c1(OC)nc(C)cc(=NCC(O)CNC(c2cc(CN(C)C)c[nH]2)=O)[nH]1 n1(CC(=O)NC(CNC(C(=O)Nc2ccc(N)cc2)=O)CO)cc(Cl)c(O)nc1=O c1(C(=O)NCC(CCOC)NC(c2cnc(SC)nc2)=O)cccnc1N(C)C N1(C(COC(C)C)=O)CCC(C(N2CCC(c3nn[nH]n3)C2)=O)(CF)C1 N1(C(C2COCC(C)O2)=O)CCCCC(CC(N2CC(N(C)C)C(C)C2)=O)C1 CC1(C)CCC(C(N2CCCC2C2(C(=O)NC3CCOC3)CCC2)=O)CO1 c1(C(=O)NC2C(CNC(C3CCC(C(N)=O)CC3)=O)C2)cc2c(F)cccc2[nH]1 c1(C(N(CCC(C)NC(c2c(C)cc(O)nn2)=O)C)=O)cc2ccccc2s1 Cc1nc2cnn(C)c2cc1C(=O)NC1(CNC(=O)C(O)C(F)(F)F)CC1 C1(CCCNC(CC#N)=O)CCN(C(C2CC2(F)F)=O)CC1 c1(C(=O)NCC2(CNC(C3CCN(C)CC3)=O)CCC2)ccc([N+](=O)[O-])cn1 C1(CN(CC(F)(F)F)C(=O)NC(c2nc(Cl)ccc2Cl)C)CCC(N=[N+]=[N-])CC1 c1(CN2CC(CC(=O)NCC=C)OCC2)cc(Br)cc(F)c1O CCC(C)CC(=O)NCC1CC(C(N2CC(C)(C)C2C(C)C)=O)C1 C#CC(CC)(CC)NC(c1ccn(CCNC(=O)C(C)(C)C=C)c1)=O Cc1ccnnc1C(=O)NC1CC2(C1)CC2C(=O)NCCC(O)C1CCC1 C1(CNC(C(CC)O)=O)CC12CCN(C(c1cccc(CO)n1)=O)CC2 Cc1cc(F)ncc1-c1noc(-c2ccc(-n3cccn3)cc2S(N)(=O)=O)n1 N1(CCC(C2CC(=O)CS2)O)CCC(C)(CCC(=O)NC2C=C(C)CS2)CC1 c1(NC(C(=O)N(C)CC2CC(CC(C)C)C2)=O)nnnn1C1CC1 N1(C(C(C=C)O)=O)CC2CN(Cc3ccccc3)CC(C1)C2C(=O)OCC C1(CNC(c2cn(C(C)C)nc2)=O)C(C)CCN1C(c1ccc(C(F)F)cn1)=O c1(NC(=O)C=CC(F)(F)F)ccnc(NCC(F)F)c1 c1(C(N2CCC(C3CCCN3C(=O)CC3CC=CC3)C2)=O)coc(Cl)n1 C1(CC=C)(NC(=O)C(O)COC)CCCN(C(=O)Cc2ccc(CC)cc2)C1 c1(C(=O)N(CCO)Cc2ncon2)cnc(C(F)(F)F)cn1 c1(C(N(C2CCN(C(C3(CC)CCC3)=O)C2)CC)=O)nc(C)sc1C c1(OC)ccc2cccc(C(=O)NC3(c4nn[nH]n4)CCN(C(C)=O)C3)c2c1 C12(C(=O)NC(C3CCN(C(CCC(C)OC)=O)CC3)CO)CCCC1C2(F)F N1(C(C(C)OCC)=O)C(C(=O)NC2CCC(F)CC2)CCC1C C(=O)(C#CC1(C)CCCO1)N1CC2CC(NC(c3nn(CC)c(C)c3)=O)CC2C1 CC1(C)CCCC(C(=O)NC(C2CCCC2)CNC(=O)C2CC2)CC1 C1(CNC(c2cccc(C)c2C(=O)O)=O)(CO)CC12CCOCC2 N1(C(CC(C)(F)F)=O)CCCC(CO)(NC(c2cc[nH]n2)=O)C1 C1(C(=O)NCc2ccc(C(=O)NC3CC(F)C3)s2)C2CCC(F)(F)C12 c1(C(N(CCC(C)NC(c2c(C)oc(C)c2C)=O)C)=O)cccc2ncn(C)c12 C1(c2ccoc2)C(=O)N1.C(C(=O)NCCCOCCN(C)C)=CCOC O=C(C#CC1(O)CCCCC1)NCC1C=CCN1C(c1ccc(Br)cn1)=O C1(C(=O)NCC(C)NC(=O)CNC(=O)C2CC2)CCc2nncn2C1 C(=O)(C(C)C(F)(F)C(F)F)NC1CC(N(C(c2cc(CC)n(C)n2)=O)C)C1 N1(C(CCCOC(CCC)=O)=O)CCCCC1CCNC(=O)C(CC)NC(N)=O n1(CC)cnc(C(=O)NCCCC(C)NC(c2ccoc2Br)=O)c1 C1(CC(=O)N(CCC(C)NC(=O)CC2(CO)CC2)C)CCCCC(=O)N1 N1(C(CN(C(C)=O)C)=O)CCC(NC(=O)CC2CC3(CCC3)C2)C(O)C1 S(=O)(=O)(CCC(=O)NCC(=O)NC1CC1)NC(=O)CN1CCSCC1 C(=O)(C1CCCc2scnc21)N1CC2(C(NC(c3c[nH]c(Br)c3)=O)CC2)C1 C(=O)(C1CCc2c(Cl)cccc21)NCCN(C1CCCOCCC1C(=O)OC)CC C1(C2CCN(c3nnccc3C#N)C2)(NC(CCCCC#C)=O)CC1 C12(C(N3CCC(O)(CC)C3)=O)C(NC(=O)Cc3cn(C)nc3C)C3CC1C2C3 N1(C(C(C)(C)SC)=O)CCN(C(c2cc(C)c(C)[nH]2)=O)CC(O)C1 c1(C(=O)NCCC2CCCN(C(C(C=CC)O)=O)C2)cc2cccc(C)c2s1 C=CCC(C(=O)N1CC(CCNC(=O)C#CC(C)(C)C)C(C)C1)C(C)C C(=O)(C1(C)CCc2ccccc21)N1CCN(c2cc(OC)c(F)cc2)CC1 c1(C(=O)NCc2nc(CNC(c3nn(CC)c(C)c3)=O)sc2)cc([N+](=O)[O-])c[nH]1 C(=O)(C(CC(C)C)ONC(c1cnn(C)c1C#N)=O)N(CCNC(C)=O)C C1(NC(c2c(COC)scc2)=O)CCC12CCCO2 CC(C)C(C)C(CNC(=O)C(C)CC1CCC1)NC(=O)C=C(Cl)Cl C(=O)(C(C(C)C)C1CCC1)NC(COCC)C(=O)NC(C)Cc1cncnc1O c1(C(N2CCC(OCCNC(CSC=S)=O)CC2)=O)ncn2ccccc12 c1(NC2CN(Cc3c(F)ncc(C)c3)CC(C)C2)ncnc2cccc(F)c12 C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NCCNC(Cc1c(C)n(C)nc1)=O Cc1ccc(C(C)C(=O)N(C(C)C(=O)NCc2nc(C)ns2)C)o1 CCCCC(CC(=O)N(CC(O)CO)C(C)C)NC(c1cccc2[nH]ccc12)=O c1(NC(C2CC(C)CN2C(C2(C3CC3)CC2)=O)=O)nc(Br)c(Br)cc1Br C1(C(N2CC(OCCNC(c3csc(O)n3)=O)C2)=O)CCCCC12CC2(F)F CC1Cc2cccc(C(N3CCCC3CN(C(=O)C=CC3(C)COC3)C)=O)c2O1 C1(C#N)(C(N2CCC(OCCNC(c3c(C)ncs3)=O)C2)=O)CC(C)C1 N(C1CCCn2ncnc21)C(C(C1CC1)NC(c1cc(C#N)sc1)=O)=O c1(OC)ccc(F)cc1-c1cncc(CN2CCN(c3cc(Br)ccc3C)CC2)n1 C(=O)(C(C)CS(C)(=O)=O)OC.C12(NC(=O)NCC3CC3)CCCN1C2=O N1(CC(=O)NC(CC(C)NC(c2cc(C(=O)OC)sc2)=O)C)CC(=O)NC1=O CC(C)CS(=O)(=O)CCC(=O)N1CCC(C)C(NC(C2CC(C)OC2C)=O)C1C N1(C(CCCCSC)=O)CCN(C(c2cc(C(C)C)[nH]n2)=O)CC(O)C1 N1(C(CC(=C)C)=O)CCC2C(CCN2C(=O)CC2CSc3ccccc3O2)C1 CN=c1nc(C(N2CCC(OCCNC(c3cccc(C)c3)=O)C2)=O)cc(C)[nH]1 C1(C)(C(N2CCC(CNC(c3ccc(CCC)s3)=O)C2)=O)CC(C)=NO1 c1(CC(C(=O)N(CC(C)N(C(C2(C(C)=O)CC2)=O)C)C)N(C)C)cccc(F)c1 C1(CC(=O)O)(CNC(C2C(OC)CC2)=O)CC=CCC1 c1(CN(C(C(C2N(CC)CCC2)(C)C)=O)C)sc(-c2ccc(Cl)cc2)nc1C CCCC(CCC)NC(=O)CCCN(C(=O)COc1ccccc1)C C1(NC(CC2ON=C(C)C2)=O)C=CCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 N1(C(CN(CCOC)C(C2CC(C)C2)=O)=O)CCC(O)(C(F)F)C1 c1(N2CCC(N(C(c3ccc(OC)nc3)=O)C)CC2)nc(C)nc(O)c1C C1(C(=O)NCc2nn(CC)nc2C)CC(C)(C)CCN1C(=O)CCn1ccnc1 S(=O)(=O)(c1ccccc1)NCCC(=O)N(C(C)CNC(C1CC2CCC1C2)=O)C c1(OCC(=O)NCCC(C)N(C(=O)CC2CC(=O)NC2=O)C)cncc(Cl)n1 C1(NC(C2C(Cc3ccc(C)cc3)CCC2)=O)CCC(C)N(S(C)(=O)=O)C1 Cc1nc(CC(C)C)oc1C(=O)NCCCN(C)C(c1cn(CCN(C)C)nn1)=O C(=O)(N=c1nc2cc(Cl)ccn2[nH]1)C1C(C)(C(F)F)C1 N1(C(CCCC=C)=O)CCN(C)CC1C(N1CCN(C)C(CC)C1)=O N1(C(c2n[nH]c3c2CN(C(C2(N(C)C)CC2)=O)C3)=O)CCc2ccc(F)cc2C1 c1(CC(=O)N(C(C)CN(C)C(c2n[nH]cc2Br)=O)C)ccc2c(c1)CCO2 N1(C(COCCC(=O)OC)=O)CCC(NC(=O)CC(C)n2cccn2)C12CC2 C#CC1(C(=O)NCC2(C(N)=O)CN(C(C3CCOC(C)C3)=O)C2)CCCC1 C(C(O)CC(F)(F)F)ONC(c1oc(C)c(CO)c1)=O c1(CC)nc(C(=O)NC(C2CCOC2)CC(=O)O)c(C)o1 n1(CCC#C)cc(NC(c2n[nH]cc2Br)c2nnnn2CCCOC)cn1 N1(C(CNC(CCC)=O)=O)CC(NC(=O)CC2(OCC)CC2)CC1(C)CC Cc1ccc(N(C)C(N(C(=N)N)C(c2ccc(Cl)cc2)c2ccccc2)=O)cc1 CN1CC(NC(=O)CC2CCCCN2C(c2cc(CO)on2)=O)CCC1=O N1(C(c2c(C)nns2)C(=O)NC2CCOC2)CCC(CCCCC2CC2)CC1 N1(C(c2nc(C)oc2)=O)CCOC2(CCN(C(C3(C)CC3C(F)(F)F)=O)CC2)C1 N1(C(COCCCCCC)=O)CCC(CO)(NC(=O)Cc2cc(CC)no2)CC1 Cc1cc(N(C=O)C2CC2)c(C)cc1C(C)(C)C.N1(C(=O)O)CC(C#N)C1 C1(C(N2CCC(NC(C3(OC)CCC3)=O)C2)=O)(CC)CCC(F)(F)CC1 C1(O)(CC(=O)N(CCOC)C(C)C2CC2)CCN(C(c2coc(OC)n2)=O)CC1 CCCCCC(O)C(=O)NC(CCC)C(=O)N(C)Cc1cncnc1 C(=O)(C(CO)NC(C1COCC1C(N)=O)=O)N(CCCN(C)C)CCO CC1CN2CCCCC2CN1C(c1ccc(NC(c2ccco2)=O)cc1)=O C1(C(=O)NCC2(C(N3CCC(CC=C)C3)=O)CCCC2)CSCC(=O)N1 N1(C(C=C(C)Cl)=O)CCC(O)(CNC(=O)CCC2CC2CC2CC2)C1 c1(NCC(CNC(c2n(CC)ccc2)=O)O)ncc2c(c1C#N)CCC2 C(=O)(C(C(C)(C)C)C1CC1)NC(C)CNC(c1cccc(CC#N)c1)=O c1(OC)c(F)ccc(F)c1C(=O)NC(CCNC(=O)COc1ccon1)C(C)C C#CCC(O)C(=O)NCC1CCCN1C(c1cnc(-c2cccc(F)c2)s1)=O c1(CNC(C2CCNC23CC3)=O)cc(F)ccc1C1CC1 CC1CC(N(C)C(c2cncc(CNC(=O)C(C3CCCCC3)O)c2)=O)CCO1 C(=O)C(C)C(C)(F)F.N1(C(c2cn(CCOC)nn2)=O)CCCC(c2n(C)cnn2)C1 CC1=C(C(=O)NC2CN(C(=O)CC3CC4C=CC3CC4)CC2C)C(=O)OC1(C)C C1(NC(CC2C(C)C2)=O)CS(=O)(=O)N(C)C12CCN(C(C1CCNC1=O)=O)CC2 C(=O)(C1CCCn2nccc21)NCC1(OC)CCN(C(C2(F)CCCC2)=O)CC1 C=C(C)CC(C)C(=O)N1CC=C(CNC(=O)COC2CCOCC2)CC1 N1(C(CS(=O)(=O)NC(C)(C)C)=O)CCC2(CCC2)C(NC(c2cc(Cl)cs2)=O)C1 c1(C(C)=O)ccc2nc(NC3CCOC3)cc(C)c2c1 c1(C(=O)NCC(C)NC(C2CCCN2C2CC2)=O)cnn2c1OCC2 C1(C)(C(=O)NC(CC=C)(C)C)CC(O)CN1C(c1ccsc1OC)=O C(=O)(C1=CCCN(C(c2cc[nH]c2C)=O)C1)N1CCC(=C)CC1 C1(C(=O)OC)CC(=O)N(C)C1C(=O)NCC1CCCN1C(c1nnccc1C)=O CCC(CN(C)C)CC(=O)N1CCCCC(NC(=O)C(COC(C)(C)C)N(C)C)C1 CC(C)C(O)C(F)(F)C(=O)N1CCC(CNC(=O)CC2CC(F)(F)C2)C(O)C1 c1(C2(C(=O)Nc3cn(CC(N4CC(C=O)C4)=O)nn3)CC2)ccccc1F.CO CCC1=NOC(C(=O)NCCNC(=O)C(C)n2ccnn2)C1 N#Cc1ncc(NCC2(F)CC(NC(c3ocnc3C3CC3)=O)C2)nc1C#N Cc1ncc(NC(C2CCCC(NC(=O)CC3(N(C)C)CCC3)C2)=O)cc1F C1(CC(=O)NC2C3CC2N(C(c2cnn4ccsc24)=O)C3)CCC2(CCC2)O1 CCCCCCC(C)CC(=O)NCCOC1CCN(C(C2CCCSS2)=O)C1 c1(OC)ccnc(C(N2CC(NC(=O)C=C(C)c3cccs3)C(F)C2)=O)c1F c1(N2CC(O)C2)nc(N2CCCC(Cc3ccccn3)C2)ncc1Cl c1(C(=O)NC2(C3CN(C(C4(CC)CCNC4=O)=O)C3)CC2)ccnc2c1CCO2 Cc1cc(=NC(=O)C(=O)N2CCCC2CN(C)C(C2(C)CCC3CC3C2)=O)[nH]o1 C(=O)(C=C1SCC(=O)N1C)N(C(C)CNC(C1CCC(C(F)(F)F)O1)=O)C N1(C(C(C)NS(CC)(=O)=O)=O)CCC2(C1)CN(c1ncc(C)cn1)C2 CC(CS(C)(=O)=O)C(=O)NC1CN(C(C2(CCF)CC2)=O)CC(C)(C)C1 c1(CNC(C(CC)N(C(=O)CC2=CCCC2)C)=O)ccc(F)c(O)c1 Cc1nc(Cl)ccc1C(N1CC(NC(C2CCNC2=O)=O)C(C)C1)=O Cc1ccc(CN2CCC2(C)C(=O)NC2CCS(=O)(=O)C2)c(F)c1 [N-]=[N+]=NCCCCCC(=O)NCCn1cc(C(=O)NC2CC23CCC3)nn1 N1(C(c2cnc(C)s2)C(=O)NCc2ccccc2Br)CCCOCC12CCCC2 Cc1cc(C(=O)NC2CC2NC(C2(C)CCCCC2)=O)c2n[nH]cc2c1 S(=O)(=O)(c1ccc(F)cc1)NC(c1cc(C)nc(SCCSC2CC2)n1)C N1(C(C)C)C(=O)COCC1C(=O)NCCCCCNC(=O)CC(O)C1CCCC1 N1(C(C(=O)Nc2ccc(C)nc2)=O)CCCC(c2ccccc2)C1C CC1(C(=O)NCC2CCC2NC(c2cc(Cl)ns2)=O)CC=CCC1 c1(NC)ccc(C(N2CCC(CNC(=O)CN3CC(C)C3)CC2)=O)cc1F c1(OC)c(C(=O)NCCN(C)C(C2CCC(F)C2)=O)[nH]c2ccccc12 C1(CCC)CN(C(c2ocnc2C)=O)CCN1C(C1CCC1C(F)F)=O C1(CNC(c2ccc(NC(c3cn[nH]c3)=O)cc2)=O)Cc2cc(F)ccc2O1 CCN=c1[nH]c(C)c(C(=O)NC(c2ccccc2)CNC(C23CCC2C3)=O)s1 c1(NC(c2n(CCOC)nnn2)c2ccnn2C)cnc(O)c(C(C)C)c1 C=C1CC2CC1CN2C(C(=O)NC1CCC(N(C)C)CC1)c1ccco1 N1(C(c2cc(F)cc(Br)c2)=O)CC2CC(C1)CN(C(C1(Cl)CC1)=O)C2 CC1(CNC(c2csc(-c3cnccn3)n2)=O)CCc2ccccc2O1 C1(CNC(C(C)O)=O)CCC2(CO1)CC(NC(=O)Cc1sccc1Cl)C2 C1(C(=O)NC(CC)(C)CNC(c2cc3c(s2)CCC3)=O)Cc2ccccc2O1 N1(C(C2C(C(C)(C)C)C2)=O)CCC2(CC1)CN(C(=O)C1Cc3ccccc31)C2 C(CNC(=O)C(=O)NCC(c1ccsc1)C)(CC(=O)NCC(F)F)OC CN1CCCCC1C(N1CC2CC1C2CNC(C1(C)CS(=O)(=O)C1)=O)=O Cc1cc(NC(c2c(CNC(c3sccc3C#N)=O)nnn2C)=O)cc(F)c1 N1(C(CCc2n(C)ncc2)=O)CCC(C2CC2)C1CNC(=O)CC1(C)CCCO1 C1(CC(N)=O)CN(C(C2CCCN2C(c2cnn3c2CCC3)=O)=O)CC12CC2 N1(C(CC(C)(F)F)=O)CC2(NC(C3CC3C3CCC3)=O)CCC1CC2 N1(C(CC(C)C2CC2)=O)CCC(F)C(NC(c2ccc(C(N)=O)s2)=O)C1 CC1CCC(CNC(=O)C(=O)NC2CC(c3ccccc3)C(C#N)C2)CS1(=O)=O C=CC1(CC(N2CCCC2CNC(c2cnc(CCC)nc2)=O)=O)CCOCC1 N1(C(=O)OC(C)(C)C)CCC1CN(O)Cc1cc(Br)no1 CCCC(C(=O)NCC1CCCN(C(=O)C=CC(=O)NC2CC2)C1)OCC CC(CC(=O)N(CCNC(C1COCC1C(N)=O)=O)CC1CC1)C1CCCC1 Cc1cc(C(=O)NCC2CC2CC(N2CCC(C)(C)C2)=O)c(F)c(Br)c1 CC1(C)CCN(C(=O)CCn2cccc2)CC1CNC(c1coc(C2CC2)n1)=O N1(C(CCc2c(C)cccc2)=O)CC2CCOCC(C1)N2C(=O)CC(F)(F)F C(=O)(C(C)(C(C)C)OC)N1CC(CC=C)(NC(=O)Cc2c(C)nn(CC)c2C)C1 c1(C(=O)NCC2CC(NC(C3OCC(C)(C)C3)=O)C2)cncc2cc(Cl)ccc12 C1(C(=O)NC2CC(CCC(=O)NC(C3(O)CCC3)C)C2)CC2CC1CC2O C(=O)(CCCCC(=O)N1CC2CC2(C(=O)NCc2cccc(Cl)c2)C1)OC Cc1cccc(C(=O)C(N2CC3C(NC(c4cn(C5CC5)cn4)=O)C3C2)=O)c1 CC(CC(C)NC(c1cnc(-c2cccs2)o1)=O)NC(C1(N(C)C)CC1)=O C1(C)(CNC(c2cn(CC=C)nn2)=O)CCN(C(c2ccc(C(C)=O)s2)=O)C1 Cc1nc2cc(C(N3CCC(C#N)(NC(c4ccc(Cl)nc4)=O)C3)=O)ccc2s1 C(=O)(CCCCCN(C(=O)COCC1CCOC1)C)N1CCC(C)C1 Cn1cnc2c1CN(C(=O)C(O)CCCNC(c1ccc(O)cc1F)=O)CC2 N1(C(c2cccc(C)c2)=O)CCC2(CC1)CC2C(N1CCS(=O)CC1C)=O C=CCC(C)(CC=C)NC(c1occc1CNC(=O)C=CC1CCCCC1)=O N1(C(c2c(C)csc2C)=O)CCCC2(CCN(C(=O)CC3CCCOC3)C2)C1 c1(-c2occ(C(=O)OCc3cn(C(C)C)nc3)n2)ccc(F)cc1 c1(C(=O)NC2(C)CC(NC(c3cncc(N)c3)=O)C2)occ2c1CCCC2 c1(C(N(C2CN(C(C(CC)n3ccnc3)=O)C2)C)=O)ccc(OC(C)CC)cc1 c1(C(N2CCCCC2C2CCC2)C(=O)Nn2cncn2)cccc2ccncc12 N1(C(C(CC)C)=O)CCC2(CCOCC2)C(NC(c2nc(C)sc2C)=O)C1 C(N=c1ccc(S(=O)(=O)NCC2CC3(CCC3O)C2)c[nH]1)C1CC(C(C)C)C1 C1(CNC(C2(C)C(C)C2)=O)CN(C(C2CC(C)(O)C2)=O)CC1O c1(OC)cc(C)ccc1CNCCc1csc(Br)c1 c1(C(=O)NCC(CN(C(=O)C(C)(C)C2CC2)C)O)cc(-n2ccnc2)ccn1 C(C1C(C(=O)NCc2cccc(NC(=O)CN3CCC(CO)C3)c2)C1(C)C)=C(C)C C(CC(CNC(=O)CCC=C(C)C)NC(=O)CCC1CCOC1)OC S(=O)(=O)(c1ccc(N2CCC3(C2)CN(C)C3)c(Br)c1)NC1CC(C)NC1=O N1(C(C(C)C)=O)CC2CC2(C(=O)NC(CO)CCC2CC2)C1 C=C(Br)CC(C)(C)C(=O)NCC1CCC(N(C)C(C2CC2(C)C)=O)CC1 Cc1nc(C(N2CCCC2)CNC(=O)Cc2cnn(C)c2)n[nH]1 C1(CNC(C2(CC)CCCC2)=O)CCN(C(=O)CCCCN(C)C)CCC1(F)F C(CNC(c1cn(C)nn1)=O)(CC(=O)N1CCCC1(C)C(C)(C)C)OC C1(CNC(C2CC(=O)OC2)=O)CN(C(=O)C(=O)NCC(F)(F)F)CC12CC2 C1(CC(=O)NC(C(=O)NCCc2cnc(C)s2)C)CCC(=O)CC1 N1(CC#N)CCC(COC(c2nn(CC(F)(F)F)cc2Cl)=O)CC1 n1(CC(=O)NCC(C)NC(C2CC3CCC3C2)=O)ccc2ccccc2c1=O N1(C(C(CC(C)C)ONC(C2CN(C)CCO2)=O)=O)CC2(CCOC2=O)C1 N1(C(C2CC(C#C)(O)C2)=O)CCC(C)N(C(=O)CC2CC2(C)C)CC1 n1(CC)c(C)nn(CC(=O)NCC(C)NC(=O)CSc2ccccc2)c1=O N1(C(Cc2c(C)scc2)=O)CC2(CCCN(C(C3(NC(N)=O)CC3)=O)C2)C1 C1(C(=O)NC(C#C)C(C)C)C=CCCN1C(=O)CSC(F)(F)F c1(-c2ccc(C3C(C)CN(C)C3)cc2)nccc(=NC2COc3ccccc32)[nH]1 CCC(O)CC(=O)N=c1cc(C2CCCCN2C(c2ccc(COC)s2)=O)[nH][nH]1 CC1=CCC(C(=O)NC(C)(C)C(=O)NCCNC(=O)C2CC2)CC1 C1(C(=O)NCC(=O)NCCC(=O)OCC)OCCC1COC C1(C(=O)NCC(COC)NC(c2ncn(CC)n2)=O)CCOCC1(C)C C1(NC(C2CCC(F)(F)CC2)=O)CC2CC(C1)N(c1nncs1)C2 c1(C(=O)NC(C(=O)NC(CN(C)C)CO)CC2CCC2)ccc(O)cn1 N1(C(CCc2c(C)ncs2)=O)CC(NC(c2cnn(CC3CCC3)c2)=O)CC(C)C1 CC1CC(=O)NC(C(=O)NCC23CC(NC(C4C5CCCCC45)=O)(CO2)C3)C1 CC(C)C(O)C(=O)N1CCC(N(C(=O)Cn2cc(C3CC3)nn2)CCO)C1 c1(NC(C2(C)CCN(C(=O)CC3(O)CCCCC3)C2)=O)ccc(Cl)cc1O C(=O)(CCCCCn1cnnn1)NCC(CCNC(C1N(C(C)=O)CCC1)=O)O C1(C(=O)NCC(NOCCC(=C)C)=O)CCNC(=O)C1 C1(NC(CC(=O)N(C)C)=O)CN(C(=O)Cc2cc(F)ccc2Br)CCC1F C1(CNC(CCC(=C)Br)=O)CC(C)CCN1C(c1n[nH]c(CC)c1Cl)=O CC(O)C(C)C(=O)NCC(C)NC(C1(C)CCNC1=O)=O C1(CNC(Cc2c(OC)cccc2F)=O)CC12CCN(C(=O)C(C)CF)CC2 Cc1ccc(F)c(O)c1C(=O)NCC12CC1CN(C(=O)CN(C1CCC1)C)C2 c1(C(=O)NCC23N(C(C4CCN(C)CC4)=O)CCC2CC3)cncc2c1CCC2 c1(C(=O)NCC2(CNC(C3CCOC3)=O)CC23CCC3)cnc(O)c(F)c1 c1(C(=O)NC2CN(C(c3n(CCC)ncc3)=O)CC2SC)cccc2nccn12 N1(C(c2n[nH]c(CC)c2C)=O)Cc2occ(C(N3CC(O)CCC3C)=O)c2C1 C12(C(=O)NCC(CC(C)C)(C)C)CC3CC1C2C3(F)F n1(C(CC)CC)nc(C(=O)N(CC(O)CNC(=O)CCNC(=O)CO)C)cc1C Cc1ccccc1Oc1nc(CSc2ccc(Cl)cc2)no1 C1(C(N(CC(=C)C)CC(=C)C)=O)CN(C(c2cc(OC)n(C)n2)=O)CC1(C)C N1(C(c2cccc3nc(C)nn32)=O)CCOC2(CCCN(C(=O)CCC#N)C2)C1 c1(CNC(C2(NC(N)=O)CC2)=O)ccc(C(N2CCCC2C(N)=O)=O)s1 C=C(C)C(C)(C)C(=O)N(CC(CO)(CO)NC(=O)CNS(=O)(=O)CC)C CC12CCC(CCn3cc(CC4CCCC4CNCCC#N)nn3)(CO1)C2 O=C(C#CC1CCCOC1)NC1CCC1CNC(c1ccn(CC(F)(F)F)n1)=O CC1(C)CC(NC(=O)CC2(C)CCN2C(=O)Cc2cc[nH]c2)C(C)(C)O1 Cc1c(C(=O)NC2C3CN(C(c4ccoc4)=O)CC23)cnn1C(C)(C)C C12(NC(C3=NOC(C)(C)C3)=O)CN(C(=O)CCC3CC3)CC1CS(=O)(=O)C2 Cc1ncnc2c1CC(C(=O)NCC1CC(C)N(C(=O)C(=O)NC3CC3)C1)CC2 C1(CN(C(C2CCN(CC(C)C)C2)=O)CC)CCN(C(=O)Cc2ccon2)C1 c1(C(=O)N)ccc(OC)c(OC)c1.C1(C(N(CC=C)C)=O)CCN(C(=O)COC)C1 c1(C(=O)NCCCN(C)C(C2CC23CCCOC3)=O)cncc2c1CCCC2 c1(CNC(CCCOC)=O)ccc(CCNC(C2OC3CCC2C3)=O)cc1 CC(C)C(O)(C(=O)NC1CCN(C(C2(CCF)CCC2)=O)CC1)C(F)(F)F c1(CN(C(=O)CCc2ccncc2)Cc2ccccc2)ccc(Br)cc1 C1(C(=O)NCC2C(NC(c3cocc3Br)=O)CC2)CCCCO1 CCCC(C(=O)N1CCC(C)CC1)C(C)C.c1(CC(C2CCCN2)=O)ccc([N+](=O)[O-])cc1.N c1(C(=O)NC2C3N(C(C4C(C(=O)OCC)C4)=O)C(CC3)C2)cc2c(F)cccc2s1 CCN=C(NCCN1CCCC1)NCc1cc(C)no1.C12CC1C2 C1(N(CCCNC(C(CC)C)C)C(c2cncs2)=O)CCN(C(=O)C2CC2)CC1 c1(C(N(CC(=O)N(CC(C)NC(CN(CCOC)C)=O)C)C(C)C)=O)ccsc1 C(=O)(CC1=CCCC1)NCc1cc(C(N(CC(C)OC)C2CC2)=O)no1 N1(CC)CC(C(N2CC(CC(C)NC(=O)CC3(O)CCCC3)C2)=O)CCC1=O C(CC(O)C(=O)NCCCC(C)NC(c1ccc(-c2csnn2)cc1)=O)SC C(=O)(C(C)(C)CCC#N)NCN(C(C(=O)NC)C)C(=O)OC(C)(C)C c1(C(N(C)CC2OCCN(C(CCC#C)=O)C2)=O)cc(F)cc2ccccc12 N1(C(C(c2ccnn2C)C)=O)CCC(NC(c2cc(C3CC3)ns2)=O)C(F)C1 Cc1cc(C)c(C(N2CC(NC(c3nn(C)cc3[N+](=O)[O-])=O)C(O)C2)=O)c(N)c1 C1(NC(C2(CC=C)CCCCC2)=O)CC(OC)CN(C(=O)C=C(C)C(C)(C)C)C1 C1(CCC(=O)NCC(C2CCCC2)NC(c2cnc(C)[nH]2)=O)CCCCN1C c1(CC)nc(C)c(C(=O)NC(C2CCN(C(C3CC(CC(F)F)C3)=O)CC2)C)o1 N1(C(c2onc(COC)n2)=O)CCC(F)(F)C(CNC(=O)C=CI)C1 C1(C(N(CCCNC(=O)C(C)(C)OC)CC)=O)Cc2cc(Cl)ccc2C(=O)O1 CCCCC(O)CC(=O)N1CCCC(C(N2CCC(C)(CN(C)C)C2)=O)CC1 C1(C(N2C(c3n(C)cnc3)CCC2)=O)(CO)CC(F)(F)C1 c1(C(=O)NC(COCC)C(=O)NC2CCCC2(F)F)ncncc1Cl N#Cc1nc(Br)cnc1NC(C1CC1NCc1ccc(Br)[nH]1)=O C1(C(=O)OC)CCSC12CN(C(=O)NCC1(C)CCCC(F)(F)C1)C2 c1(CC(=O)NC(CNC(C(CC=CC)C)=O)(C)CC)ccc(F)cc1C c1(CNc2ccc(NC(c3c(C)ccs3)=O)cn2)cc2ncccc2[nH]1 C1(NC(c2c(C)nn[nH]2)=O)(CNC(=O)Cc2ccc(F)cc2)CCCCC1C N1(C(c2c(CC)non2)=O)CC2(C)CC1(C(=O)NC1CCN(C(C)C)C1=O)C2 N1(C(COC2CN(C(c3cc(C)ncc3)=O)C2)=O)CC2C=CCC(C2)C1 C#CCCN=C(NCc1nc(CC(F)(F)F)no1)N1CCC(OC2CCCC2)C1.C(C)C C(c1ccc(C#N)cc1)=CC(N1CC(N2C(=O)CC(NC(C=CCC)=O)C2)C1)=O c1(CC)cc(NC(c2cccc(CNCc3cc(C)ccc3O)c2)=O)ccc1O C=CC1(C(=O)NC2(CO)CN(C(=O)COC3(C)CCCC3)C2)CCC1 c1(OCC)cccc(C=CC(=O)NCC(C)N(C)Cc2ccc(Cl)nc2)c1 c1(NC(CCC)=O)ccc(Oc2nccc(C(F)(F)F)n2)c(Cl)c1 c1(NC2CC(C(=O)NCC3(c4ccccc4)CC3)C2)ncncc1C(=O)O C1(NC(=O)C(F)CC2CN(C(=O)Cn3ccccc3=O)C2)CCn2ccnc2C1 N1(C(CSC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)CO.C12CN(C1)C2=O c1(OC)ccccc1C(C)C(=O)N1CC(N(C(=O)CC(O)c2ccccc2)C)C1 c1(C(N(C)CCc2nccs2)=O)conc1CNC(=O)C(O)C1CCCC1 CCCCC(O)CCC(=O)N1CCCOC(CNC(=O)C(CC(C)C)C(N)=O)C1 C1(NC(C(CC=CC)C)=O)CCC12CCN(C(=O)CNc1ccccc1Cl)CC2 N1(C(CCC=CCC=C)=O)CC2CC(NC(=O)C(CC)NC(N)=O)CC1C2 C1(F)(C(=O)NC(C2N(C(c3c(C)nc[nH]3)=O)CCC2)C)CCN(C)CC1 C1(C)(C(=O)NC(CN(C(c2cc3ncccn3n2)=O)CC)C)CC(C(C)C)=NO1 N1(C(C(CC#C)(C)NC(=O)CC2CC(=C3CC3)C2)=O)CCC(C)C(F)(F)C1 C(C(COC)CC(=O)NC1(C(=O)NCc2cc(F)ccc2F)CSC1)OC c1(C(=O)NC2CCC(N(C(CSCCC(C)C)=O)C)C2)cnn2c1CCC2 Cc1cc(F)cc(C)c1C(N1CC2CN(C(c3ccc4ccoc4c3)=O)CC12)=O c12cn(C)nc1SCc1nnc-2o1.Cn1ccc(-c2cccs2)n1 C1(NC(c2cc(Cl)cs2)=O)CCN(C(=O)C=Cc2cncc(O)c2)CCC1CO c1(C(N2CCCC(CN(C(C3CCN(C)C3)=O)C)C2)=O)cc2ccsc2n1C c1(C(=O)NCC2OCCN(C(c3c(C)oc(C(C)C)n3)=O)C2)ccnc(O)c1F C1(CNC(c2cc(CC)n(C)n2)=O)COCCN(C(C2C(F)(F)C23CC3)=O)C1 c1(C(=O)OC)ccc2c(c1)C(C1CCOCC1)CN2Cc1nc2ccccc2s1 N1(C(c2nc(C)[nH]n2)=O)C2CCC1CN(C(C1CCCC(F)C1)=O)C2 CN1CCN(C(=O)CN2CCOC2=O)C(CNC(=O)CC2(CO)CC2)C1 c1(C(=O)NC2CC(NC(Cc3ncc(C)[nH]3)=O)C2)cc(N)nc(Br)c1 CCC(C)CCCC(=O)NCC1CC(NC(C)=O)C1.C1(=O)COC(=O)CN1 C1(CC)CC(C(=O)OCC(N2CCCC2c2ccc(F)cc2F)=O)CCC1=O CC1(C(=O)NC2CCN(C(c3ccoc3C3CC3)=O)CC2)CC2(C1)CC(F)(F)C2 c1(C(CF)NC(=O)NC(C(CC)C)CO)cccc2ccccc12 C1(C(=O)NCC(C(C)C)NC(C2OCC2(C)C)=O)(OC)CCSCC1 C(c1ccccn1)=C(C(=O)NCC(CNC(c1cscc1Cl)=O)OC)C CC(C)CCC(F)C(=O)NC1(C(=O)NCC(c2ccsc2)C)CC(F)C1 CC1=NOC(CC(=O)N(C(C)C(=O)NC(c2ccc(C)s2)C)C)C1 C1(C(=O)NCC2(C3CC3)CC2)COCCN1C(C1CCC2CC12)=O C1(C(N(C2CCN(C(c3sc(C)cc3C)=O)C2)CC#C)=O)CN(C)CCO1 Cc1ncnc(NC2(CNC(=O)COCC3CC3)CCOCC2)c1C#N C(CCC)(C(=O)NC1CCCC1NC(=O)CSc1ccc(OC)cc1)=CCC C1(N)(C(N2CCCC(C(N(c3ccccc3)C)=O)C2)=O)CC(O)C1(C)C C1(NC(c2n(CC#C)ccc2)=O)C2CC(O)C1N(C(c1cnc(SC)n1C)=O)C2 c1(CC(=O)NCCCC(C)NC(C2CC3(CC3)CO2)=O)cnc2ccccc2c1 N1(C(=O)Cc2ccsc2)CCC2CN(C(c3c(Cl)cncc3Cl)=O)CCC2C1 C1(CC)CN(C(=O)CCCC2CCCC2)CCC1NC(=O)CSC1CCCC1 C1(CC(=O)NCCOCCC(C)C)CC2(CC2)CN1C(=O)CC1CCOCC1 C1(n2cc(CNC(c3cnc[nH]3)=O)nn2)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 C1(CC=C)(C(=O)NC(C)Cc2nc[nH]n2)CN(C(=O)CCOCC)C1 Cc1nc2cc(C(N3CCN(C(C4CC(CCO)C4)=O)C(C)C3)=O)cnc2[nH]1 C1(CC(N2C(C)(CNC(=O)C(O)C(F)F)CCC2)=O)CC2C=CC1CC2 C1(C(=O)NCC2C(C(=O)NCCCCN=[N+]=[N-])CC2)CCC2(CC1)CC2 c1(C(=O)NCC(CN(C(CCc2c(C)nn(C)c2)=O)C)C)[nH]ccc(=O)c1C c1(C(N2C3C(NC(CC(C)C(F)F)=O)C(C3)C2)=O)cc2ccc(F)cc2cn1 C1(C(=O)NC2C(C(N(CCOCC=C)C)=O)CC2)CC(=O)NC(=O)N1 c1(OC)cc(C(=O)NCC(O)CN(C(=O)Cc2cc(C)sc2C)C)cc(F)n1 N1(C(c2ncc(CC)s2)=O)CCOC(C(C)NC(=O)C(=O)NCC2CC2)C1 C(=O)(C1=CCCSC1)NC(=O)N(C)C.c1(C2C(C)N2C(C)=O)ccccc1 N1(CCOCC(=O)Nc2cnc(C)s2)CCC(C)CC1 c1(CC)c(C(=O)NC2CC(F)CN(C(c3cc4n(n3)CCC4)=O)C2)cccc1F C(C(=O)N1CCC1CC)(c1ccoc1)NC(C1C(=C)C1)=O Cc1nnccc1C(=O)NC1CC(F)(CNC(=O)C(C)C(C)C2CCCCC2)C1 c1(OC)ccc(C(=O)NCC2CC(NC(=O)C3=CSCCO3)C2)cc1F C1(C(=O)NC2(C(=O)NCC3(C#C)CCC3)CC2(C)C)CCCC(=O)CC1 CC(CC(C)(F)F)C(=O)NC1(CO)CCN(C(C2(F)CC2)=O)C1 C1(CN(C(c2cc(F)cs2)=O)CC)CCCCN1C(c1cnc(NC)cn1)=O CC(CC(F)(F)F)C(=O)NC1C2CC3C(C2)C13C(N1CC2CC2(CO)C1)=O C(=O)(CS(=O)(=O)c1ccccc1F)NCC1(NC(=O)CCc2ncccn2)CC1 N(C1CN(C(=O)C(F)CC2CC2)CCc2ccccc21)C(Cc1nnc(C)s1)=O c1(C(=O)NCC2CCCC2NC(=O)C(F)(F)C(F)F)ccc(O)c(F)c1F C(CCC(C)(C)C)(C(=O)NCC1CC1)N1CCCC(c2nc(C)c(C)s2)C1 CN(OCC(F)(F)F)C(=O)CC(CNC(C1(C#N)CCOCC1)=O)C1CCC1 c1(-c2c(NC(c3cc(C)c(F)cn3)=O)cccc2)cnc2c(c1)NCCO2 CC1(C)C2CC(O)(C(N3CC(C(F)(F)F)C(O)C3)=O)CC12 CC(C)(CNC(=O)C(c1ccoc1)NC(c1cn(C(F)F)cn1)=O)CO CC1NC(=O)CCC1CNC(=O)C(CN=[N+]=[N-])NC(c1cncn1C)=O C(=O)(CC(O)CCSC)NC(CCCC)CNC(c1ccc(C)cn1)=O C1(C(=O)NC(C=C)C2CC2)CCCCCC1NC(c1cc(C)cc(C)n1)=O Cn1cnc(N2C3CCC2C(CNC(c2nccnc2C(N)=O)=O)C3)c(Br)c1=O CC1CN(C(c2cccc(N)n2)=O)CCC1NC(=O)CN1CC(=O)NC1=O C(=O)(C(O)CC[S+](C)C)N1CCC(C)(NC(C2CCC(OC)CC2)=O)C1 c1(C(N2C(CN(C(CCCC#CC)=O)C)CCCC2)=O)nc(Cl)c(=O)[nH]c1N N1(C(C2(CC=C)CCC2)=O)CCC(NC(=O)Cc2cccc(SC)c2)C(C)C1 C1(NC(C(CCC=C)NC(=O)Cc2cnn(C)c2)=O)CCn2nnnc2C1 C(=O)(C1CCCc2nnn(C)c21)N(C)CCC1CCCCN1C(=O)C(N)=O C#CCCC(C(=O)NCC(CC)CC)NC(c1cc(Cl)cn1C)=O Cc1nc(C(=O)NCC(C)(CO)NC(C2CCCCC(=O)N2)=O)ccc1Br CCC(C)(CO)C(=O)NCCC1CN(C(c2cc(C)nc(OC)n2)=O)C1 c1(OCCCC(=O)NCC(CC)NC(=O)CCCN(C)C)ccc(F)c(F)c1 C(c1c(Cl)ccc(Cl)c1Cl)=CC(N1CC2CCN(C(C=CSC)=O)CC21)=O c1(C(=O)NCCC23CC2CCN3)cccc2c1CCS2(=O)=O C#Cc1cc(COC(=O)CSc2ncccn2)cc(O)c1 C(C)(C)(C(=O)N1CCC1CNC(c1c[nH]c(C(N)=O)c1)=O)NC(=O)OC c1(C(=O)NC2CC(C)(NC(c3n(C)nc(O)c3)=O)C2)csc2ccc(F)cc12 C1(COC)(CNC(=O)Cc2cc[nH]n2)CCN(C(=O)CC2CC=CC2)CC1 C1(C(=O)NC2(C)CCC(NC(CC=CC)=O)CC2)Cc2cccnc2C1 C(CCSC)(C(=O)NC(C)CNC(=O)CS(C)(=O)=O)OC CC(CC(=O)NCCC1(CNC(C2(C#N)CC2)=O)CC1)C(C)(C)C c1(C(=O)NCCC(N2CCC(CC(=O)NC)C2)=O)ccccc1O C(=O)(CCCCCC#N)N1CCC1CNC(c1cccc(N2CCC(C)C2)c1)=O c1(C(N2CC(C)C(NC(=O)C(C)(C)CF)C2)=O)cn(C)c(=O)cn1 C1(CNC(C(CC2CC2)NC(C(C)SC(C)C)=O)=O)CC2(CC2)C(=O)O1 c1(NC(CC)CC#N)[nH]c(=NC2CCN(CC3CC3)CC2)nc2scnc12 c1(CC(=O)NCC2(O)CCN(C(C3CCN(C)C3=O)=O)C2)ccc2c(c1)COC2 c1(OC)ncc(C(=O)NCCCCC(C)NC(=O)C(C)Cn2ccc(C)n2)cn1 N1(C(CCC)=O)CCCC2(CCN(C(=O)C(c3cccc(OC)c3)O)C2)C1 Cc1noc2ncnc(N3CCC(CC(N4CCN(c5ncccn5)CC4)=O)C3)c12 C1(C(=O)NC2CN(Cc3ncccc3C(=O)O)CC2C)(OC)CCOCC1 N1(C(C#C)=O)CCCC(C)(C(=O)NC2CCC(n3cccc3)CC2)C1 Cn1nc(C(=O)NC2CC(F)CN(C(C3CC3(F)F)=O)C2)c2cc(F)ccc12 C1(NC(c2scc(OC)c2)=O)CC2CCC(C1)N2C(=O)Cc1ccc(F)cc1 CN1CCC(N(C)C(C2C=CCN(C(c3cc(=N)[nH][nH]3)=O)C2)=O)C1=O C1(N(C(c2ccc(OCC)nc2)=O)C)CCCN(C(c2sncc2CC)=O)CC1 CCN=C(NCCOc1ccccc1)NCCC1(C)CC1(F)Cl n1(CCCC)nc(C(C)OC)nc1-c1c[nH]ccc1=O Cc1cc(C(=O)NC2CC2NC(=O)CCC2CCC(=O)NC2)n(C2CCC2)n1 C12(NC(=O)Cn3ncnn3)CCN(C(c3cc4ccccn4n3)=O)CCC1C2 c1(C(N(CCCN(C(C(C(C)C)NC(C)=O)=O)C)C)=O)ccc(C#N)c(O)c1 C1(CC(N2CC3CSCC3C2)C(=O)NCC(=C)C)CCC(F)(F)CC1 CON(CCC(=O)NC1CCCCC1N=[N+]=[N-])C(=O)c1cc(Cl)cs1 c1(OC)ccc(C(C)C(=O)N2CC(NC(c3c(C)cccc3O)=O)C2)cc1Br C(C)(CCC(=O)NCC(C)(C)OCCNC(=O)C(c1cccc(Cl)c1)C)OCC C(=O)(CCCS(C)(=O)=O)NCC1C2CN(C(C3(COC)CCCCC3)=O)C1C2 c1(OC)ccc(Cl)c(C(=O)NC2CC2NC(=O)CCNC(C)=O)c1 C(=O)(CCC(=O)NC1CC(NC(=O)CC2(NC)CCCC2)C1)Nc1nnc(C)s1 C1(SC)CCCC1NC(c1ccc(CNC(c2ccoc2C(C)C)=O)s1)=O C(C(C)CNC(C1CC(NC(C2(F)CCC2)=O)C1)=O)OCC C1(C(=O)NC(c2ncc(C)[nH]2)CC)CC(C)(C)CCN1C(c1csc(Cl)n1)=O C1(CC=C)(C(N2CC(CO)CC2CO)=O)CCN(C(C2CC(N(C)C)C2)=O)C1 C=CC1(CC(=O)OC)CN(C(=O)NCc2ccccn2)C1 N=S1(=O)CCC(CC=O)CC1.C1(C(=O)O)CCCNC1c1ccccc1 c1(C(=O)NCC(C)N(C)C(C2OC(C)(C)OC2(C)C)=O)ccc2c(n1)COCC2 C1(CN(C(c2c(C)cc[nH]2)=O)C)CN(C(=O)C(C)Cc2cnc[nH]2)CC12CC2 O=C(C1=COc2ccccc2O1)NCC1CC(O)CN1C(=O)Cc1ccc(Cl)s1 Cc1ccc2nc(C3CC3)[nH]c2c1.C12CCCC1C(=O)N2.c12cnoc1CNC2 C1(NC(C2CC(SC)C2)=O)CCN(C(=O)CC2(C(F)F)CC2)CC12CCC2 c1(C(N2CCN(C(C3CC(CCC)OCC3)=O)CC2C)=O)cc2cccnc2[nH]1 N1(C(CN(C(COC)=O)C)=O)CCC(NC(c2cnc(O)n2C)=O)C1C(C)(C)C c1(C(=O)NCC(CNC(C2(N3CCCC3)CC2)=O)OC)ncsc1Br c1(C(=O)NCCC2CN(C(c3cc(F)cc(Br)c3)=O)C2)coc2c1CCCC2 C(C(C(=O)NCCN1CC2CC2C1)NC(C1CN(C)C1)=O)OCC c1(C(N2CCCC(N(C(=O)C(F)OC(F)(F)F)CCF)C2)=O)ccc2nsnc2c1 C(=O)(C#CC(C)(C)C)NC(CCOC)C(=O)N1CC(NC(N)=O)C1 C(=O)(C(=O)CC(=O)c1ccsc1)N1C(C(C)NC(=O)CSC2CC2)CCCC1 n1(CCC=C)nc(-c2ccoc2)nc1CCC(F)F N1(C(=O)Cc2cc(Cl)ccc2Br)CCC2C1CCN2C(=O)C(F)F c1(C(N(CCC)CCNC(C2CC2(C)C)=O)=O)cc(=O)c2ccccc2[nH]1 C(=O)(C(COC)CC(C)C)N(CCC)CCNC(C1(C(=O)NC)CCC1)=O CC1CN(C(=O)CC2(C(F)(F)F)CC2)CC1NC(=O)Cn1cc(Br)cn1 CCCCC(O)CC(=O)N1CC=CC1C(N1CC(C)(C#N)C1)=O C1(NC(c2nc(C(N)=O)sc2)=O)CN(C(=O)CC2CC(=O)C2)CCC1O N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCC2CCCN(C(=O)COCCOC)C2C1 C1(C(=O)NCC(C)NC(C2N(C(=O)OC)CCC2)=O)CC(C)(C)CO1 c1(C(=O)OC)cccc(CN(C)CC2CN(C(C3CC(=O)N3)=O)CCO2)n1 c1(NC(=O)NC(C)C(c2ccc3c(c2)OCO3)O)cc(C#N)cc(Cl)n1 C1(CNC(c2ncn3c2CCC3)=O)CC2(CCN(C(c3ccsc3)=O)CC2)CO1 CCCC(C(=O)NC(C)CN(C)C(C)C)NC(c1cc(CC)sn1)=O C1(C)(CNC(C(CC=CCC)C)=O)CCN(C(c2cc(F)n[nH]2)=O)CC1 c1(C(N(C)CC2CCCN2C(c2ncc(N)cc2Cl)=O)=O)cc2c(o1)CCCC2 c1(C(N2C(CCNC(=O)COc3cccnc3)CCC2)=O)nnn2c1CSCC2 c1(OC)cc(C(=O)NCCNC(=O)Cc2cccc(C(F)(F)F)n2)n(C)n1 C(CCN(C(=O)COc1ccc(C(C)C)cc1)C)(C(C)C)NC(C(C)OC)=O c1(C(=O)NCC2N(C(CN(C3CC3)CC)=O)CCOC2)cc2c(cn1)COCC2 N1(C(c2cn(C)nn2)=O)CCC(C)(CNC(=O)CC2C=CS(=O)(=O)C2)C1 n1(CC)ccnc1C(=O)NCCOCCCN(C)C(C1(CCOC)CCC1)=O CC1CN(C(=O)C(N2CCC(O)CC2)C)CC1CNC(c1cc(CO)n(C)n1)=O CCC(F)(F)CC(=O)N(C)CC1CCCN(C(c2cccc(C(=O)OC)n2)=O)C1 c1(CNC(CCN(CC#C)C(C2CCOC(C)C2)=O)=O)ccc(F)c(C)c1 CC1C(NC(=O)C(c2ccc(F)cc2)F)CCN1C(=O)C1CC1 C#CCCC(O)C(=O)NCCc1ocnc1CNC(=O)CC(C)(C)OC CC(C)CC(C(=O)NCC1CC(C)CN(C(=O)C(N2CCNC2=O)C)C1)C(C)C N1(C(c2c(N)ccc(OC)c2)=O)CCC2(CC1)CC2NC(=O)CCc1nncs1 C1(CNC(=O)NCC(Cn2c(C)ncc2)C)C2CCCCC12 CCCC(C(=O)NC(CO)C(=O)N1CC(N2CCOC2=O)C1)NC(C)=O c1(C(N2CC3C(CNC(C4CC45CCC5)=O)(C3)C2)=O)ccc(F)c2ccncc12 Cc1ccc(CC(N2CCC(NC(=O)C(C)C(C)C)C2C(C)(C)C)=O)cn1 C(=O)(C1Cc2ccc(F)cc21)N1CCC(NC(c2n[nH]c(CC)c2[N+](=O)[O-])=O)C1 N1(C(C(C2CCOCC2)C)=O)CCN(C(c2cc(Cl)ncc2N)=O)CC1C Nc1c(C(=O)NCCN(C(C2CN3CCC2C3)=O)CC2CC2)cc(Cl)cc1F C1(N(C(=O)C=CSc2nc[nH]n2)CC)CCN(C(=O)CCc2cc(Cl)no2)CC1 Cc1nc(C(=O)N(C2CCCC2)CCNC(=O)C=C2CCC(C)CC2)c(C)s1 C(N=c1nc(N2CCSC(C(C)C)C2)c2c([nH]1)CCS2)C1CCN(CC)C1 C(C(=O)NCCCCn1cc(CNC(C)=O)nn1)(C1(NC)CCC1)OCC C1(CC(N2C(CC(=O)NCC3COC(=O)N3)CC2)=O)CC2CC2C1 N1(C(CNC(CC)=O)=O)CCc2nc(CNC(=O)CCOC3CC3)sc2C1 C1(C(=O)NCC2(c3onc(C)n3)CCC2)CNCc2ccnn2C1 c1(N(CC(C)NC(CSc2c(OCC)cccc2)=O)C)ncc2cccnc2n1 C#Cc1cnc(C(N2CCC(O)CC2C(=O)N(C)CCSC)=O)c(C)c1 c1(CC)cnoc1C(=O)NC(C)(C)C(=O)NC(C)CCn1cncn1 C1(C(N2CC(C)C(N(C)C)C2)=O)CCN(C(c2ccns2)=O)C1(C)C N1(C(CCC(C)=O)=O)CC2CCN(C(c3scnc3C(F)(F)F)=O)CC2C1 Cc1cc(C(N2CC3C(CC(=O)N(C4CCOC(C)(C)C4)C)C3C2)=O)nc(C)n1 c1(C(=O)NCC2CCN2C(c2ccc(C(F)F)o2)=O)ccc(-n2ccnc2)nn1 CCCCC(F)C(=O)NCCCN(C(=O)Cc1ccoc1C)C c1(C(=O)NCCN(C(c2cncc(C)c2)=O)C)cc2c[nH]nc2s1 c1(CC)nccnc1C(N1CCN(C2CCN(C(C3CC(=O)N3)=O)CC2)CC1)=O c1(C(=O)NCC2C(NC(C=Cc3c(C)ccs3)=O)C2)nn2cccnc2c1Br C=CCC(C)(C)C(=O)NC1CCCN(CCc2ccc(C(=O)OC)nc2C)CC1 CCCCS(=O)(=O)NCC(=O)N(C1CCN(C(=O)C(CCSC)N(C)C)C1)C c1(C(N2CCN(C(=O)CSC3CC3)CC2CCO)=O)cncc([N+](=O)[O-])c1 N1(C(C2CCCCN2Cc2ccc(-c3ccccc3Cl)o2)=O)CCOCC(O)C1 C(=O)(CCC(C)(C)N(C)C)NC(CCN(C(CCC(=O)NCCC)=O)C)C c1(C(N2CCC(C(C)NC(=O)C(C)C3CCC3)CC2)=O)cccc2c1C(=O)CC2 c1(CC(N2CC(O)(CNC(C(CC)(C)C(F)F)=O)C2)=O)ccc2c(c1)CCN2C S(=O)(=O)(c1ccc(F)cc1F)N1CCN(c2c(S(C)(=O)=O)ccnn2)CC1 C1(NC(c2cnc(CC)s2)=O)CCC2CN(C(=O)Cc3nonc3C)CCC2C1 N1(C(C(CC)(C)CO)=O)CCC2(C=C(C(=O)N(C)CCc3ccncc3)C2)C1 c1(NC2(CNC(CC3CC(C)(C)OC3)=O)CCCCC2)ccccc1[N+](=O)[O-] Cc1cccc(CN2CCCC(C(=O)Nc3cnnc(Cl)c3)CC2)c1Br c1(C(=O)NCC(CNC(C(CCCC)(C)F)=O)C)c[nH]c2ccc(Cl)cc2c1=O n1(CC)c(S(=O)(=O)NC2CCCC3(C(C)C)CC23)cnc1C c1(S)ccc(C(=O)N(C2CCC(N)C2)C)cc1.c1(CC(=O)NC(C)=O)scnc1C c1(C(=O)NCC(C(N2CC(O)(COC)C2)=O)OC)ccc(F)c(C)c1 c1(C(C)C)nc(NCC2CC2)cc(N2CCCC(CNC3CCC(=O)N3C)C2)n1 c1(-c2c(OCC(=O)OC(C(C)C)C(=O)N(C)C)cccc2)ccc(F)cc1Cl C1(NC(=O)CC2CC2)CCN(C(=O)COc2ccc(F)cc2Cl)CC1F c1(C(N2CC(CNC(C(CCC)F)=O)C(F)(F)C2)=O)nc(C)c(C)nc1C C1(NC(C(COC)C)=O)CCCN(C(=O)C=Cc2scnc2C)C1C Cc1nc2c(C(=O)NC3CCC(NC(C4CC4(F)Br)=O)CC3)cccc2o1 CC1CCC(C)(C(=O)NCC=C2CCN(C(C3CCO3)=O)CC2)C1 CCCC(C)(O)C(=O)N1CCCOC(CNC(=O)CCCc2ccc(C)cc2)C1 C(C)(CCC(=O)NC(C(=O)NCCCc1n[nH]c(C)n1)C(C)OC)OCC C(C(C)(C)CC1CN(C(c2cnn(CCO)c2)=O)C1)NC(C(C)OCC1CC1)=O Cc1cc(C(=O)NCC2CN(c3ccnc(-c4nccs4)n3)CCO2)ncc1F N1(C(CCC=C)=O)CCN(CCCCCNC(C2(C)CC(F)C2)=O)CC1 S(=O)(=O)(c1ccc(N2CCC(C)C2)c(Br)c1)N1CC(C)=C(C)C1 C#Cc1ccc(CC(=O)NCC(CC2CC2)C(=O)NC2CC(F)C2)cc1 C1(CN(C(=O)CC2CCNC(=O)C2)C)CCCCN1C(c1cnc(C2CC2)[nH]1)=O c1(C(N2CCC(CNC(C(C)SCCCC)=O)C23CC3)=O)cnc([N+](=O)[O-])n1C CC1CCCCC1(CNc1ncnc(O)c1Br)NC(c1ccncc1F)=O C=Cc1cnn(C)c1C(=O)NCC1CCN1C(=O)C(C)Oc1cccnc1 c1(C(C)C)ccc(SCC(=O)NC2CN(C(c3cc(F)n(C)n3)=O)C3CC23)cc1 CN1CCC(C2(C(=O)N(CCCNC(=O)C(C)(C)CC(F)F)CCO)CC2)CC1 CCC(C)(CNC(=O)C(c1cccs1)NCC(=O)OC)C(C)O O=C(N=c1ccnc2[nH][nH]cc1-2)C12CC1CN(Cc1ncccc1Cl)C2 C1(CC(=O)N(C2CC(C#N)C2)CC(=O)NCC(C)CO)CCCNC1=O C1(C(=O)NCC2N(C(C(C)(C)OCCC)=O)CC2)CCN(CC(=O)NCC)CC1 c1(OC)ccc(F)c(CN2CCCC2C(=O)NCc2cc(C#N)ccc2Br)c1Br C1(C(=O)NCc2n[nH]c(C)c2C)CN(C(=O)CC(C)F)C2(CCC2)C1 CS(=O)(=O)c1sccc1C(=O)NC1CCCN(C(C2C3CC4C(C3=O)C24)=O)CC1 C(=O)(N=c1[nH]onc1-c1ccccc1)NCCCC(C)O C1(CC(N2CCC(COC)(NC(=O)C3=CCC3)C2)=O)CC(=O)c2ccccc2C1 c1(C(=O)NC(C2CCN(C(=O)C(O)C3CCC3)CC2)C)ncc(Cl)cc1F CC1(C)CC(O)CCN(C(=O)C(CC(F)F)NC(C2OCCC2(C)C)=O)C1 c1(C(=O)NC(C(=O)NCc2cnc(CC)s2)CC2CCCC2)cccc(C)c1F N1(C(c2cccc(CC)c2)=O)CCC(NC(=O)CN2CSCC2=O)C(C)C1 Cc1c[nH]c(C(=O)NCC2(O)CC(CNC(=O)C(=Cc3cscn3)F)C2)c1 C1(NC(c2c(C)occ2)=O)CCCCCC1NC(=O)C=C(C1CC1)C1CC1 CC1=C(C(=O)NCC2CCCC(CNC(c3cc(C4CC4)[nH]n3)=O)C2)CCC1 C(=O)(C#CC1(CC)COC1)OCC.C12(C3CCCO3)CN(C1)C(=O)CCN2CC N1(C(C2(CC)CCCC2)=O)CCC(N(C)C(c2ccnn2C2CCC2)=O)C(C)C1 C1(C(=O)NCCCn2c(C)ncc2)CCOCC1NC(c1cc(F)c[nH]1)=O c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)C(C)CC2)ccc(=O)n2c1CCCC2 c1(C(=O)NC(CNC(C(c2c(C)nn(C)c2)O)=O)C2CC2)sc2nccn2c1C c1(SC)ccc(Cl)cc1NC(c1sccc1I)c1nnnn1C(C)(C)C CCC(F)(F)C(C)(C)C(=O)NC1CC(CNC(c2coc(CS(C)(=O)=O)n2)=O)C1 CCC(C)(C)CCCC(=O)NC1CCC(NC(c2n[nH]c(C)c2F)=O)C1 C(CC(F)F)(C(=O)NCC(C)(C)CCC=C)NC(CCOCC#C)=O C(=O)(C(C)(O)C(C)C)N1CCCC(CN(C(=O)C(c2c(C)noc2C)C)CC)C1 CCCCC(CNC(C1(F)CC1(Cl)Cl)=O)NC(=O)CC1CC(F)(F)C1 C1(C(=O)NCC(C)(C2CC2)NC(=O)CCn2cnnn2)CC2(CCOC2)C1 c1(CC)cnoc1C(=O)NC(C(=O)NCCNC(=O)NCC)C1CCOC1 C1(O)(CN(C(c2cc(CC)[nH]n2)=O)C)CCCN(C(=O)CC(C)C2CCCC2)C1 C1(C)(C(=O)NC(c2ncc(C)cn2)C)CC(O)CN1C(=O)Cc1nc(=N)[nH][nH]1 CCC(CC(=O)NCC1CN(C(=O)CCF)CC1C(F)(F)F)c1ccccc1 C#CCC(CC(=O)N(CC(C)CCC)C)NC(=O)CCc1ccccn1 C1(CC)CN(C(=O)Cc2ccc(OC)nc2)CCN1C(C1CC(C2CC2)=NO1)=O C(C(C)(O)CC(=O)N(CCC(=O)NC1(n2ccnn2)CC1)OC)OC C1(CNC(c2cn(C)nc2)=O)(CNC(C2CCCC2CF)=O)CCCCC1 C1(C(=O)NCC(C)(C2CCC2)NC(C(CCC)O)=O)Cc2nnsc2S1 N1(C(CCCC(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCc2cncc(F)c2)C1 N1(C(C2CC3CCC2C3)=O)CCCC(CNC2N(C(C)(C)C)CC2)C1 C1(NC(C=CCOCCOC)=O)CN(c2ncc(C#N)cc2F)CC2(CC2)C1 N1(C(C(c2ccc(C(=O)O)o2)C)=O)CCCCC1Cc1cn(CCN(C)C)nn1 C1(C(=O)NCC23N(C(c4c(C)csc4)=O)C(CC2)CC3)OCC2COCCC12 CC(CCNC(=O)C(O)C(C)(C)C)N=c1[nH]c2ccc(Br)cc2o1 C1(CC(=O)NC(CCNC(C(C(C)C)C#N)=O)(C)C)CCC2CC1C2(C)C c1(CC)ccc(S(=O)(=O)N2CCOC3CN(C(C45CC(C4)C5)=O)CC23)cc1 Cc1cnc(C(=O)NCC2CC(O)(CNC(=O)Cn3cncn3)C2)cc1Br c1(C(=O)NCC(CC)(CC)NC(C2C(CC)C2)=O)cn2c(n1)CCCC2C C1(Cc2nc(CCc3ccccc3)on2)CNCC12CCOCC2 c1(CC(C)C(N2CC3(NC(c4cc(Cl)no4)=O)CCC2C3)=O)ccc(F)cc1F c1(-c2ccccc2)cccc2nc(CNc3ccn4ncnc4c3)cn12 C(C1=NOC2(CCC2)C1)NC(C(C1CN(C(c2ccn(C)c2)=O)C1)O)=O CC#CCCCC(=O)N1CCCC(C)C1CNC(C1(c2cccnc2)CCC1)=O C(=O)(CCCC(=O)C1CC1)NC(CNC(CC1(OCC)CCC1)=O)(C)CO C(=O)(C(C)(C)CC(F)F)N1CC(C)C(C)(CNC(c2ccoc2)=O)C1 N1(C(CC)=O)CCC(N(C)C(c2csc(C)n2)=O)CC1 CCC(C)(C)CC(=O)NC(c1ccccc1)c1nnc[nH]1 Cc1nn(C(F)F)c(C)c1C(=O)Nc1cnn(-c2ccccn2)c1C N1(C(C(C)(C)c2nccs2)=O)CCC(CO)C(NC(=O)CCC2CCCC2)C1 c1(CNC(C2N(C(c3cc(C)on3)=O)CCCC2)=O)ccc(C)c(O)c1 Cn1cc2c(n1)CCC(C(=O)NCC1CC(F)CN1C(=O)C1CC1)C2 C(CC(COC)N=c1nc(N(C)Cc2scnc2C)c2ncccc2[nH]1)OC c1(C(=O)NC(C(C)C)C(C)NC(=O)CNS(=O)(=O)C2CC2)ccc2nonc2c1 C=C1CCN(C(=O)COCC(C)(C)C)C(C(N2CC(CO)C2(C)C)=O)C1 c1(CC)cc(CNC(CNC(C)=O)C(C)(C)C)ccn1 CCCC(CC)CC(=O)N1CCC(NC(=O)C(=O)N=S(C)(C)=O)C(F)(F)CC1 C1(NC(c2c(CC)cccc2)=O)CCN(C(c2csc(C)c2)=O)CCC1CO c1(C(=O)NC(C(C)NC(C=C(CCC)C)=O)(C)C)cc(OC)cc(Cl)c1F c1(C(C)C)nnc2n1CCN(C(=O)CCNC(c1ccc[n+]([O-])c1)=O)C2C Cn1c(C(=O)NCCN(C(=O)C(O)C(F)F)CC2CCCC2)cc(Cl)c1Cl C1(C(C)O)COCCN1N1CCC(c2nc3ccc(C)cc3[nH]2)CC1 c1(C(=O)NCCNC(C(C(C)C)C#N)=O)cc2c(Cl)cccc2[nH]1 c1(CC(=O)NC(C(C(C)C)NC(=O)COC2CC(F)(F)C2)C)ccc(O)c(F)c1 c1(CN(CCC)CC2CC3(CCCO3)C2)ccc(C2CC2)c(F)c1 N1(C(c2ccc(C)s2)=O)CCC(O)(CN(C(=O)CC2CCCS2(=O)=O)C)C1 C1(CNC(CSC)=O)CN(C(=O)C(c2cccs2)SC)CCC12CCC2 C1(NC(CSCCC)=O)CCCC2CN(C(=O)CN3CCCC3C)CC12 c1(C(=O)NC2COCCC2NC(C2CCCO2)=O)c(F)cc(F)c(O)c1F c1(CC(=O)NCC2C(NC(C3CCN(CCC)CC3)=O)C2)c(C)nc(O)nc1C c1(C(=O)NC2CC(N(C)C(c3ncc(Cl)cc3Cl)=O)C2)c(F)cc(Cl)cc1F CCCCC(=O)C(=O)N1CCCC(NC(c2oc(C(F)F)cc2C)=O)C1 N1(C(c2nc(C)c(C)[nH]2)=O)CC2CCC1C(CNC(=O)C(O)(C1CC1)C1CC1)C2 C1(C2CCN(C(C3CC3Cl)=O)CC2)(NC(CCc2n(C)cnc2)=O)CC1 C1(O)(CNC(c2cc(F)cs2)=O)CCCN(C(=O)C(C2CCCCC2)F)C1 c1(OC)cccc2c1OC(C(=O)NCC1CCN(C(c3csc(CO)n3)=O)C1)C2 N1(C(C2N(C(CCC)=O)CCC2)=O)CCC12CN(C(=O)C=CSC)C2 CC(C)(F)CCC(=O)N1CCC(c2cn(-c3ccccc3)nn2)C1C(C)(C)C C=C(C)C1CCC(C)=CC1CC(=O)N(C1CN(C(c2cc(C)nc(C)c2)=O)C1)C Cc1cccc(N)c1C(=O)NC(C1CCN(C(=O)Cc2csc(Cl)n2)C1)C C1(SC)CN(C(=O)C=Cc2ccc(C)o2)CC1NC(c1c(C)csc1Cl)=O CC(CC(C)(F)F)C(=O)NC1CCCN(C)CC1 C1(C(C)(C)CNC(=O)Cc2cocn2)CCN(C(c2cnnn2C2CC2)=O)CC1 C(C#Cc1cccnc1)NC(C1N(C(C(C(C)C)OCC)=O)CCC1)=O N1(Cc2c(OC)ccc(Cl)c2)CCCC2C(NC(=O)C=C(C)C)C(C)(C)C12 C(=O)(C(C)(C)C)NC(C)C(=O)NC1CCC(CNC(c2ccns2)=O)C1 N1(C(c2cc(C)c(C)nn2)=O)CCCN(C(=O)Cc2cc(Cl)ccc2Cl)C(C)C1 C(=O)(C1CCCn2c(C)nnc21)N(CCNC(C(CC)CC(F)F)=O)C(C)C C1(C(=O)N(C)CC2(O)CCN(C(=O)C(c3cncn3C)O)C2)(OC)CCCCC1 c1(OCC)ccccc1CCC(N1CCC(C)(NC(C2CCS2(=O)=O)=O)C1)=O N1(C(CNS(C)(=O)=O)=O)CCC(O)C(NC(=O)Cn2cccn2)C1 C1(C(N2CCC(=C)C2)=O)C2CC1N(C(=O)CCC1CCOC1)C2 C1(CC)CN(C(c2cc(C)cc(F)c2)=O)CCN1C(=O)Cc1ccsc1C C1(CNC(CCC(C)C)=O)COCCN(C(C23CCN(CC2)C3)=O)C1 C1(CC)CN(C(c2ccn(CC)c(=O)c2)=O)CCC1NC(=O)C1=CCCO1 C12(C(=O)NC(CCOC(C)C)CO)CCCCN1CCC2 c1(C(N2CC(NC(CCCOC)=O)C(O)C2)=O)cnc2n1CC(C)CC2 Cc1cn2cc(C(=O)NCC3(C)CCCN(C(=O)CC4(O)CCOC4)C3)nc2s1 C(C(CC(C)C)NC(=O)C(C)n1cnnn1)NC(c1ccc(CC)s1)=O CC1(NC(C2(C)CCCN2C(=O)C=Cc2ccsc2)=O)CCOC1=O c1(OC)cc(C(N2CC(NC(C3COC(=O)O3)=O)C(C)C2)=O)nc(Br)c1 c1(N(C(COC(=O)CCC=O)C)C(C)=O)cc(F)c(N)cc1F.C1(OC)CCC1 Cc1cc(C(=O)NCC2CCN(C(=O)C(c3ccccn3)O)C2)ccc1N C(CCS(C)=O)(C(=O)NCCN1CCC(NC(=O)CCC2(C)CC2)CC1)N(C)C C1(C(C)(C)OC)CCCCCCN1C(=O)C(O)CCCOC C1(C)CCN(C=O)CC1.C1(N(C(=O)COCCSC)CCOC)(CO)CCCCC1 CS(=O)(=O)c1cccc(-c2cccnc2NC(c2csc3ccccc23)=O)c1 C1(C(=O)NC(CC)(CNC(=O)CCOCCN(C)C)CC)CC(C(C)C)=NO1 C12(NC(C(C)Cc3ccco3)=O)CCC1CN(C(=O)Cc1ccc(Cl)c(F)c1)C2 c1(C(=O)NCC2(NC(C(C)NC(CC)=O)=O)CC2)[nH]ccc1C N1(C(=O)NCC2=NOC(C)C2)C2CCC1CC(C(F)Cn1cc([N+](=O)[O-])cn1)C2 CC(C(C)(C)C(=O)N1CCC(C(C)(C)C)C1)NC(=O)CCOCC(F)F C1(CNC(CCCC#CC)=O)CN(C(c2cc(C)cnc2N)=O)CC2(CCC2)O1 C=C1CCC(C(=O)N(CCNC(=O)C(C2CCCCC2)N(C)CC)CC)CC1 C1(NC(C(CC)N(CC)CC)=O)(CF)CCN(C(C2(C(F)(F)F)CC2)=O)C1 C12CCN(CC1)C(=O)CCSCC2C.C(=O)(COCC(C)C)NC(=O)OCC CCC(C)C(C)C(=O)N(CC(C)NC(=O)Cc1cc(C)[nH]n1)C N1(C(C(C)NS(CC)(=O)=O)=O)CC2(CCC(CNC(=O)CC3(C(F)F)CC3)O2)C1 C(CC(C)C)(C(=O)NCCOCCN(C(=O)CC(C)n1ccnc1)C)OC C#Cc1ccc(CN(C)C(c2c(Br)cnn2Cc2noc(CC)n2)=O)cc1 c1(C(=O)NCC(C)CNC(=O)CCc2nccn2C)coc(C#N)c1 C12(NC(CC(=O)OC)=O)CCN(C(c3ccc(N4CCCCC4)cc3)=O)CC1C2 C(C(=O)NCC1CC1NC(c1[nH]c(C)cc1C)=O)(C(C)(C)C)OC C1(C(=O)NC2(C)CC(NC(C(C3CC3)OCC)=O)C2)(OC)CC(F)(F)C1 C1(OC(C)C(N2CCCC2C2CCN(C(c3csc(Cl)n3)=O)C2)=O)CCCCC1 C(CC(C)(C)CN=c1[nH]c(=NC(C)c2cn(C)cn2)[nH]c2c1COC2)OC c1(OC)cc(C(=O)NC2CCOCC2C(=O)N(C)Cc2ccncc2F)nn1C CCC(C(=O)N1CC(F)CC1CNC(c1ccc(Br)s1)=O)C(F)(F)F c1(C(C(=O)N(CCN(C(=O)Cc2nccn2C)CC)CC)N(C)C)cncn1C CC1SCCC1NC(c1ccc(-c2ccco2)[nH]1)=O N1(C(C)=O)CCOCC(C(=O)NCc2cccc(I)c2)C1 C1(NC(c2csc(Cl)n2)=O)CN(C(c2csc(Br)n2)=O)C2CC12 C1(NC(C(C)OCC=C)=O)C2COCC1CN(C(c1cc(C)ccn1)=O)C2 c1(C(N(C(C)CNC(c2cccc(OC)c2)=O)CC)=O)cc(C)n(C2CC2)n1 c1(C(N2CCCCC(NC(C(C)N3CCC3)=O)C2)=O)cc(F)c(F)cc1Cl CCCC(C(=O)OC)C(=O)N1CCCC1C1CCN(C(c2cnn(C)c2C)=O)C1 C(C1CCCN1C)=CC(N1CCC(CN(C(=O)Cc2cc(C3CC3)on2)C)C1)=O c1(C(N2CCCN(C(C3(CO)CC(F)(F)C3)=O)CC2)=O)cnn2cnnc2c1 c1(C(N2CCC(C(CO)NC(c3n(CC)nnc3)=O)CC2)=O)cc(C)nc(C)c1 CC(=O)CCCCC(=O)NC(CC(=O)NC1(C2CCCCC2)CC1)CC(C)C C1(COC)CC2(CCN2C(=O)C=CCC2(NC(C3CCN(C)C3=O)=O)CCC2)C1 N1(C(C2CCCCC2)=O)CCC2C1CCN2C(C1(c2cccc(Br)c2)CC1)=O C1(NC(c2cc(C)c(C)s2)=O)CCC2(CCCN2C(=O)COCC(F)(F)F)CC1 c1(C(N2CC(C(C)NC(CCC(C)OCC)=O)C2)=O)ccc([N+](=O)[O-])c(O)c1 C(N=c1ccnc(C2CCC2)[nH]1)C1CN(C(C(CO)NC(N)=O)=O)CC12CC2 N1(C(CC2CC(=C)C2)=O)CCC2(NC(=O)CS(=O)(=O)NCC)CC2C1 C1(C(N2CC(n3cc(CNC(C(C(C)C)OC)=O)nn3)C2)=O)CCC2(CCC2)CC1 c1(CC)cccc(F)c1C(=O)NCC(CNC(C1(C(F)F)CCOCC1)=O)OC C12(CC)COC(C(=O)NCC=CCNC(=O)CN(C3CCCC3)C)(C1)C2.C(C)=O c1(C(=O)NC2(C)CCN(C(CC(CC)C3CC3)=O)CC2)cnc2[nH]c(=N)sc2c1 N1(C(CCNC(COC)=O)=O)CCCCCC1C(N1CC(CO)C(C)C1)=O C#Cc1ccc(CC(N2CC(NC(C3CCC=CCCC3)=O)CC2C)=O)cc1 N1(C(C(C)(C)CCl)=O)CCC2CC2(C(=O)Nn2cccn2)CC1 CC1(C)CCCCC1=CC(=O)NC1(CCNC(=O)CCN2CCC(F)C2)CCC1 c1(C(=O)NCC(=C2CN(C(c3n(CC)ncc3Cl)=O)C2)F)cc2occc2[nH]1 c1(OC)cc(C(=O)N(CC(O)CN(C)C(c2nccn2C(C)C)=O)C)cc(C)n1 c1(C(N2C(C(=O)NCc3cocn3)CCCC2)=O)cccc(O)c1O c1(C(=O)NCC(C)N(C)C(c2cc[n+]([O-])cc2)=O)cccc(CO)n1 c1(OC)ccnc(OC)c1C(=O)N(C)CCNC(=O)Cc1cccc(F)c1F C(CCCC(=O)N(C(C)(C(=O)N1CCC1(CC)CC)C1CC1)C)OCC CC(CCNC(=O)CCC1CCN(C)CC1)CCNC(C1CC12CC(O)C2)=O Cn1ncc(C(=O)NCC2(C(=O)NC3CC4(CCC4)C3O)CC23CCC3)c1C#N N1(C(c2nc(C)sc2)=O)CCCCC1C(=O)Nc1ccc(O)cc1 N1(C(C2CC(=C)C2)=O)C2CCC1CN(C(=O)CC(CC)(C1CCC1)NC(C)=O)C2 C(CC(N)=O)(C(=O)NC1(CO)CCC1)NC(c1ncn(C(C)C)c1)=O C(c1cn(CCC2(O)CCN(C(C3CCOC3)=O)C2)nn1)=CC c1(C(c2nnnn2CC2CC2)NCC(CC)(CC)SC)nccc2ccccc12 C1(NC(CCCCC)=O)CC2(C1)CC(NC(C1CCN(C(C)C)CC1)=O)C2 c1(C(=O)NCC2CC(F)(CNC(C(C3CC3)SC)=O)C2)cc(O)ccc1[N+](=O)[O-] c1(C2(C(C(C)C)NC(C3CC3C(F)(F)F)=O)CCC2)ccnn1C C1(NC(C2CCCS2)=O)CC1C1CCCN(C(c2cncc(Cl)n2)=O)C1 CCCC(C(=O)NCC1(O)CC(NC(=O)Cc2cnns2)C1)OC(C)(C)OCC Cc1nc2cc(C(=O)NCC3C4CN(C(C56CC(C)(C5)C6)=O)CC34)ccc2n1C O=C1CC(C(=O)NC2CC(O)CN(C(C34CC(CO)(C3)C4)=O)C2)=NN1 C1(CC)CN(C(=O)C=CS(=O)(=O)CC)CCC1NC(=O)C(C)(C)C(F)(F)F C1(C(=O)NCCC2CCC2)COC2(C1)CN(C(=O)C=C1CCOCC1)C2 c1(C(=O)NCc2ccc(C(C)NC(C(CCC)O)=O)cc2)ccc2n[nH]cc2n1 C12(C(N3CC(C)C(NC(C4CCS(=O)CC4)=O)C3)=O)CC(C)(C1)OC2(C)C c1(C(C(C)C)NC(CC(C)OC)=O)ccc(CNC(c2cnn[nH]2)=O)cc1 c1(OC)cc(C(=O)NCC(C)NC(=O)C(C)C(F)F)cc(OC)c1OC CCCC(F)C(=O)NC(Cc1ccco1)C(=O)NCC1CCC(=O)N1 C1(c2cnn(C)c2)(C(=O)OCCC#CC)CCCO1 CON1CCC(C(=O)NC2CN(C(=O)CSc3cccc(C)c3)C2)CC1 C(CC(C)N=c1[nH]c(C)c(CC(c2ccc(Br)cn2)=O)s1)OC CC1(C)CC(CCO)(CNC(=O)N(c2cnccn2)CCN2CCOCC2)C1 C(=O)(C#CC(C)(C)C)NC1C(C(=O)NC(CC#C)C(=O)OCC)CCCC1 c1(C(=O)NCc2ccc(C)cc2Cl)nccc2c1NCCC2 c1(C(C(N2CCC(C(C)NC(c3n(CCC)ncc3)=O)C2)=O)O)ccc(F)cc1 c1(C(N2CCCC(NC(CCCOC(C)=O)=O)CC2)=O)coc2c(Cl)cccc12 C(=O)(C(C)(C)C(C)(F)F)NCC1N(C)CCN(C(c2ccc(O)c(CO)c2)=O)C1 C1(CNC(C2C(C=C)OCC2)=O)(NC(=O)CC2CNC(=O)C2)CCCCCC1 N1(C(C2C3(CC(NC(c4n(C=C)ncc4)=O)C3)C2)=O)CCC(CO)C12CC2 C1(C(=O)NCc2c(C(=O)NC(C3CSC3)C)n[nH]c2)CC2CC(=O)C1O2 C(=O)(C#CC1CCCOC1)N1CCN(C(c2ccc(F)cn2)=O)CC1CC1CC1 N#Cc1cscc1C(=O)NCCNC(=O)CC1(O)CCCCC1 O=C(C1CSc2ccccc21)NC1CC2CN(C(C3CCCC34CC4)=O)CC12 C1(C(N2CCCC2CN(C)C(C23CCC(CC2)C3)=O)=O)(CC)CCOCC1 Cc1ccc(F)c(O)c1C(=O)NCCNC(c1cccnc1N(C)C)=O C1(CNC(CC2(NC(C)=O)CC2)=O)CCN(c2ccncc2)C1 c1(OC)ccc(C(N2CC3CCC3(CNC(c3ccoc3C)=O)C2)=O)c(Cl)c1 c1(C(=O)NC2C(NC(COCC#C)=O)COCC2)cc(OC)c(OC)c(Cl)c1 C1(NC(C2C(OCC)CC2)=O)CN(C(c2cnncc2O)=O)C(CC)(CC)C1 C1(C(C(=O)N(CCCCCNC(C2(O)COC2)=O)C)O)CCCCCC1 C1(N(C(c2c(COC)cco2)=O)C)CCCCN(C(c2cc(OC)ns2)=O)C1 C1(C(=O)NCC2C(C)(C)C2)CN(C(c2nccnc2Cl)=O)CCC1(F)F N1(CCCC(=O)OC)CCCC(NCC(C)(C)CN(C)C(=O)OC(C)(C)C)C1 c12ccc(cc1[N+](=O)[O-])CCC(=O)N2C.CC(CC(N)=O)c1noc(C2CC2)n1 c1(CC(=O)NC2CN(C(c3c(CC)c[nH]n3)=O)CC2CC)cncc(C#N)c1 N1(CC(CN(C)C2CC2)O)CCCC1c1ccsc1 C(C(=O)NCC1CCC(F)(F)CC1)(C1=NOC2(CCC2)C1)N1CC(C#C)C1 C1(CNC(c2c(OC)cc(C)s2)=O)CN(C(c2cnc(C)[nH]2)=O)CCCO1 N(C1CCOc2ccc(Cl)cc21)C1C2CN(C(C(C(C)(C)C)CO)=O)C(C2)C1 c1(C(=O)NC2C(C)CCN(c3cc(CC)nc(CC)n3)C2)cccc2sccc12 N1(CCC(C)(C)C)CCCCC1C1CCCN(C(c2ccc[nH]2)=O)C1 c1(CNC(CC)=O)ccc2c(c1)CCC2NC(=O)CCCC1CCCCC1 C#CC1CN(C(=O)C(CC)CCOC)CCN1C(=O)C(=O)NOC c1(C(=O)NCC(CN(C(c2cc(CC(C)C)on2)=O)C)O)ccc(C(N)=O)nc1 n1(CC(=O)NCCN(C(c2ccc(C#N)s2)=O)CC)nc2n(c1=O)CCOC2 C1(n2ccnc2)(CC(=O)OC)CN(C(C2CC2c2ccoc2)=O)C1 Cc1ccc(C(=O)NC2CCN(C(=O)C(F)C(C)C)CC2C)c2c1CCCN2 S(=O)(=O)(c1ccc(N2CCC(OCC(N)=O)C2)cc1Br)NCC1(C)CCOC1 c1(NCC(=O)N(C2CCN(C(=O)Cc3ncnn3C)C2)CC)ccncc1.C(=O)NC c1(CC(=O)NC2CC2NC(C2C3CC4C(C3=O)C24)=O)ccc(Cl)c([N+](=O)[O-])c1 N1(C(CNC(CCc2n(C)cnn2)=O)=O)CCC(NC(=O)CC2CC2)CC(O)C1 N1(C(c2cc(CC)ncc2)=O)CCOCC(C(=O)NCC(C)(O)C2(C)CC2)C1 C12(C(F)(F)F)CCN(C1)c1nnnn1C2.C1CCOCC1.CC.SC c1(OC)ccc(F)c(C(=O)NCC2CCCCC2NC(C2CC(OC)C2)=O)c1F C1(Cn2cc(-c3c(C)nsc3)nn2)CCCCN(C(=O)CN(C(C)C)CC2CC2)C1 Cc1nc(CNC(C2CN(CCC(=O)O)CC2O)=O)ccc1Br c1(CC(=O)NCC(CC(C)C)NC(=O)CN2CCCC2=O)cccc([N+](=O)[O-])c1 CCC(C#N)(CC)C(=O)NC1CC(NC(=O)C(F)n2ccnc2)C1 CC(C)CC(C)(O)C(=O)NC1CCC(CC(=O)NC2(C)CS(=O)(=O)C2)C1 c1(C(=O)NC(CNC(C2CC(SC)C2)=O)C2CC2)ccc(N)c(C)c1Cl N1(C(c2[nH]nc(OC)c2Cl)=O)CCCC(NC(=O)CN2CCCCC2)CCC1 c1(C(=O)NCC=CCNC(C(CCC)C)=O)cnc(C)nc1COC C(C)(C(=O)NCCCc1nccs1)(C1CCC1)NC(C(C)c1cc[nH]n1)=O Cc1cc(C)c2cc(C(=O)NOCc3cn(-c4ccc(Br)cn4)nn3)[nH]c2c1 C1(C(=O)NCC2CN(C)C2)CCCCN(C(=O)COc2cnn(C)c2)CC1 C1(CNC(c2cccn2C(F)F)=O)CCC(F)(CNC(C2OCCO2)=O)C1 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(=O)CC1CCS(=O)(=O)C1 N1(C(CN(C)C2CC2)=O)CC2(NC(=O)Cc3coc(C4CC4)n3)CCC1CC2 C(=O)(C(C)C1CCC1)NCC(=CC(=O)NCC1(COC)CC1)C N1(C(C)=O)CCC(CCNC(=O)COCCF)CC1C.C(CC(C)C)O C1(CNC(C2OCCN(CC)C2)=O)CN(C(=O)C(C)=O)CCN1C C1(OCC#C)CCN(C(C2CC(COc3cnc[nH]3)CO2)=O)CC1 c1(CC(=O)NCCOCCn2cc(-c3ccccc3F)nn2)ccc(Cl)c(Cl)c1 C(=O)(C1=COCCO1)NCCC1(NC(=O)CSc2nc[nH]n2)CCCC1 C1(C(N2CCN(C(c3cnsn3)=O)C3CCCC23)=O)CCc2cc(F)ccc2O1 C(=O)(C1=CC2CC=CCC12)NC1(CO)CN(C(CCOCCOC)=O)C1 C1(NC(c2c(OC)c[nH]n2)=O)CC(C)CN(C(=O)C(C)Cc2cnn(C)c2)C1 Cc1cnn(C)c1CC(=O)NC1CCOC(CNC(c2cc(C#N)no2)=O)C1 Cc1nn(CC(=O)NCc2cc(C(=O)NC(C3CCCC3)CO)n(C)n2)c(=O)o1 C1(NC(CCCSC)=O)CC2CCC(C1C)N2C(C1CCN(CC2CC2)CC1)=O C1(N(C(CC(CC)C)=O)C)CN(C(C2(F)CC2)=O)CC1(C)C N1(C(C2CCC(C(=O)OCC)CC2)=O)CCc2sc(-c3ccnn3C)cc2C1 c1(OC)ccc(Cl)cc1C(=O)NC1CC2CCC1N2C(=O)CC1CCC(=O)N1 c1(C(N(CCC(C)NC(c2nccc(OC)c2C)=O)C)=O)cc2c(ncn2C)[nH]1 C(=O)(NNc1ccc(CC(C)C)cc1)C1(CCn2cc(CC=C)nn2)CCCCC1 CC1(NC(=O)C(CC(C)(N)CO)c2ccccc2)CCN(Cc2ccc(Cl)cc2)C1 N1(C(C2C(C)C2)=O)CCC2(CC1)CC(C(=O)Nc1ncc(C(C)(C)C)[nH]1)C2 N1(C(=O)NC(CCCC#C)C)CCC2(CCOC2=O)C1 N1(C(C2CCN(C)C2)=O)CC(NC(=O)CC2CN3CCC2CC3)CC2(CC2)C1 C1(N(C(=O)Cn2ccnn2)CCC)CCN(C(c2cnn(CC)n2)=O)C1 C1(C(N2CCCC(CCNC(CC(C)(C)OC)=O)C2)=O)CCOC(=O)CC1 C1(N(C(C=Cc2c(C)ccs2)=O)C)CN(C(c2sccc2C(C)C)=O)CC12CC2 N1(C(c2cc(OC)n(C)n2)=O)CCCC(CC)C1C(=O)NC(c1ccsc1)CO C1(N)CCC2CN(C(=O)CC)CCC2C1.C=CC(C)(CC)C(=O)N Cc1ccc(CCC(=O)NC(C)CCN(C)C(C2(Br)CC2(F)F)=O)cc1 N1(C(C2(OCC)CCC2)=O)CCc2[nH]nc(CNC(=O)Cc3csc(C)c3)c2C1 C1(C(=O)NCC2C(NC(=O)COC3CCCOC3)C2)COC2COCC2O1 c1(C(=O)OC)nc2ccccc2nc1N(C)Cc1c(F)cccc1F C1(NC(C=CC(C)(C)C)=O)(NC(=O)CNC(=O)NCc2ccco2)CCOC1 Cc1nn2cc(C(=O)Nc3cccc(NC(C4CCCC(=O)N4)=O)c3)nc2s1 CC(=Cn1ccnn1)C(=O)N1CC2CCCC2(NC(=O)Cn2c(C)csc2=O)C1 c1(NCCc2c(C)nccn2)[nH]c(=NCc2nnc(CO)s2)nc2scnc12 C1(NC(C(F)OC)=O)CC2CC(C1)CN(C(c1cscc1C(=O)OC)=O)C2 c1(C(N(CC(C)NC(CC)=O)C)=O)ccccc1Sc1ncoc1C1CCC1 c1(C(C)C)ccc(C(=O)NC2CCC(C(N3CCC(CO)C3)=O)CC2)c(Cl)n1 C12(CNC(C(C)(C)c3ccncc3)=O)CC(CN1C(c1cccnn1)=O)C2 C1(CC(=O)N(C(C)C)CCN(C(=O)CSCc2ncc[nH]2)C)CCCC(F)(F)C1 N1(C(c2cc(OC)n[nH]2)=O)CCC2(NC(=O)CCn3ccnn3)CC2C1 C1(C(=O)Nc2cnn(C)c2C(C)C)(CC)CCCN(C(c2ccnnc2C)=O)C1 c1(CC(N2CCN(CCNC(C3CC3C3CC3)=O)CC2)=O)ccc2c(c1)CC2 c1(N2C(CNC(=O)CCc3ccccc3)CCCC2)ncnc2c(Br)cccc12 CCC(CC)C(C)C(=O)NC(C)CNC(=O)C(O)(C(F)(F)F)C1CC1 C1(N(C(=O)CN2CCCC2=O)C)CCCN(C(=O)COCC2CCCO2)C1 C(CC(=O)NCCCCN(CCCNC(C1(NC(N)=O)CC1)=O)C)SC S(=O)(=O)(c1cnn2ccc(=NCCOC3CCOC3)[nH]c12)N1CC(C)(OC)C1 Cc1cc(O)c(Cl)cc1C(=O)NC(CNC(c1c[nH]nc1C)=O)C(C)C(C)C N1(C(=O)NC2C(c3onc(CC)n3)C2)CCNCC1C1CCCC1 CC1(C)CC2(CO1)CN(C(=O)NCC1CCOCC1F)C2 O=C(C#CC1CC1)NCc1ocnc1C(=O)NC1CC=CCC1 Cn1cc(C(=O)NCCCCNC(=O)CCc2c[nH]c(C(=O)OC(C)(C)C)c2)cn1 C(=O)(C(C(C)(C)C)N(C)C)NCC(CC(=O)NCCCC(C)C)C1CCC1 N1(C(C(C)=C(C)C)=O)CC(NC(C2CC23CCCC3)=O)C2(CCS(=O)(=O)CC2)C1 c1(C(N2CC=CC(NC(C3(c4cccs4)CC3)=O)C2)=O)cc(C2CC2)nc(Cl)c1 C1(CNC(CCOC2(C)CC2)=O)CC2COCC2N1c1cc(=O)n(C)cn1 c1(C(N2C(CCNC(Cc3n(C)ccn3)=O)CCC2)=O)ccn2c(O)nnc2c1 N1(C(c2c(C)cc[nH]2)=O)CC2CCCC2(NC(c2cc(F)c(F)c(Cl)c2)=O)C1 C1(NC(C=C(C)Cl)=O)C2COCC1CN(C(=O)Cc1ccn3ccnc3c1)C2 C1(CCC)CN(C(=O)CCCc2cccs2)CCN1C(c1cnc[nH]c1=N)=O c1(C(N(C)CC2CN(C(c3cnn(C)c3)=O)CCO2)=O)cc2cc[nH]c2cn1 N1(C(C(CC=C)NC(=O)C(F)=CCC)=O)CC2NC(=O)OC2C1 C#CC1CCC(CNC(=O)C(Cc2cn[nH]c2)NC(c2cc(OC)n[nH]2)=O)CC1 c1(C(N2C(CN(C(=O)C3=CCSC3)C)CCCC2)=O)cnc2cc[nH]c2c1 N1(CCC(=O)NCC(F)CNC(C2CC3CC3C2)=O)C(=O)CCC1=O C1(C(=O)NCC(CC(=O)NC)C)CC(O)CCN1C(C1CNC(=O)C1)=O C(=O)(C1=NNC(=O)CC1)N1CCC(O)(C(CNC(CC=CCCCCC)=O)C)C1 C1(NC(CCc2ncc(C)[nH]2)=O)CCC(C)N(C(=O)Cc2cnc(C3CC3)[nH]2)C1 c1(N(C(C(C)C)CO)C)ccc(S(=O)(=O)NC2CCC(N(C)C)C2)cc1C#N C1(CNC(c2c(C)coc2C)=O)CC2CCC1N2C(C1COC(=O)O1)=O N1(C(C)=O)CC2CCC(C1)N2C(=O)CNC(c1cscn1)=O c1(NC(=O)NCC2CS(=O)C2)cccc(Oc2ncccn2)c1 N1(C(C2(F)C(C)C2)=O)CCC(NC(C2CCN(C(c3ccoc3)=O)CC2)=O)CC1 C(CCSC)(C(=O)NCC1(O)CCCOC1)NC(COCC)=O N1(c2nc(OC(C)C)c(Br)cn2)CCCC(C2CN(C(=O)CCC3CC3)C2)C1 n1(CC)cc(C(=O)NCC(CO)NC(c2cc(C(C)C)oc2C)=O)c(C)n1 C12(C(=O)NCCCNCCC(=O)NCC(C)(O)CO)C(=O)C3CC1C2C3 CCC(C(=O)NCc1nc(C2CCN(C(=O)CSc3cccs3)CC2)n[nH]1)CO C(=O)(C1=NNC(=O)CC1)NC(C1CCCN(C(C2(COC)CC=CC2)=O)C1)C N1(C(C(CC)F)=O)CCCC2(CCN(C(=O)Cn3cc(S(C)(=O)=O)cn3)C2)C1 Cc1cc(C(=O)NC2(C(=O)NCCCOC(C)C)CCCC2C)cnc1C c1(C(C(=O)OC)N(C)C(C2CC=CC2)=O)cccnc1 c1(C(C)C)cccc(C(N2CCC(N(C(=O)C(N3CCC(O)CC3)C)C)C2)=O)n1 C1(C(F)(F)F)(C(=O)NC2CCC(NC(c3nc(C)oc3)=O)CC2)C(C)(C)C1(C)C c1(C(=O)NCC2N(C(C(COC)OC)=O)CC=C2)c(Cl)cc(Cl)cc1Cl C#CCC(C(=O)NCCC(O)C(C)C)NC(=O)CCC1(C)CC1 c1(CC)nc(C)c(C(=O)NCCn2ccc(C(=O)NC3(Cl)CC3(F)F)c2)o1 N1(Cc2csc3ccc(Br)cc32)CCOC2(CC3CCC2C3)C1 O(NC(=O)C(CC(N)=O)NC(c1ocnc1CCC)=O)CC=C C1(CC)C(C(=O)NCC(C)(C)C2(O)CCC2)CCN1C(c1cn(CCO)nn1)=O c1(C(c2nnnn2C2CCOC2)NC(CCSC)(C)C)cn(C)nc1Br C#CC(C(C)OC)NC(c1sccc1CNC(=O)C1CC1)=O C(=O)(C1=CC2(CCN(C(c3cc(O)ccc3C)=O)C2)C1)NCC(C#C)C(C)C c1(NCCN(C(=O)CSc2ccncc2)C)ccc(Cl)c(Cl)c1 c1(OC)cccc2c(C(=O)NCC(C)(Cc3ccccc3)C(C)O)cnn12 N1(CCCCNC(=O)CC2CCCOC2)CCCN(C(c2ccccn2)=O)CC1 CCCCCC(=O)NCC(N1CC(F)CC1CN(C)C(c1ccc(SC)s1)=O)=O C1(C(=O)NCCN(C(c2ccn(C(F)(F)F)n2)=O)C2CC2)OC2CCC1C2 C(=O)(C(C)S(N)(=O)=O)NCC1(OC)CN(C(C2CC(=O)NC(=O)C2)=O)C1 N1(C(=O)CC2CCN(C(c3cc[nH]n3)=O)C2)CCC(CF)CC1 C1(C(N(C)CC2CCN(C(=O)CSC3CCS(=O)(=O)C3)C2)=O)C2CC3C(C2=O)C13 C(=O)(CCCC(=O)N(C)CC1CCCN1C(C1CCC=CO1)=O)NC N1(C(C(C)OCCCC)=O)CCCC(NC(=O)CCc2ccn(C)n2)CCC1 N1(c2n(CC(c3ccc(Cl)cc3)C)nnn2)CCc2c(F)cc(Br)cc2C1 CC(C(C)(C)N1CCOCC1)NC(C1CCCN1CC(c1ccccc1)O)=O C1(C(=O)NC(C)C)CC2(C1)CC(C(=O)NOC1CCCCC1)C2 C1(CN(C(=O)NCC2CCC(C)CO2)C)CC12CCOCC2 CCC(C)C(C(=O)N(CCCCN(C(=O)C#CC(C)(C)O)C)C)N(C)C(C)=O c1(C(=O)NCC2(OC)CN(C(=O)CC3CC=CCC3)C2)cnc2c(C)cccn12 N1(CC(=O)N(C2CN(C(=O)CCCS(N)(=O)=O)C2)C)CCCC2(CC2)S1(=O)=O C(=O)(C(CC(C)C)C(C)C)N1CCC(COC)(NC(c2cn(CCO)nn2)=O)C1 CC(CO)(CO)C(=O)N1CCNC(C(=O)Nc2ccccc2-c2ccccc2)C1 C(=O)(C1CCCn2cncc21)NCC1CCC(NC(Cc2c(C)cnn2C)=O)C1 N1(C(=O)C=Cc2cccs2)CC2CCC1C1CN(c3ncncc3Br)CC21 C1(CNC(=O)CCC2CCCC2)CN(C)CCN1C(C1C(C(=O)OC)CC1)=O CCCC(CCC)CCCC(=O)N(CC(O)CNC(c1ccnc(F)c1N)=O)C c1(C(N2C(CNC(C(COC)(C)OC)=O)CC2)=O)nc(Br)c2n1CCCC2 c1(C(=O)NC(C2CCN(C(c3n(C)ccc3)=O)C2)(C)C)ccc2[nH]ccc2n1 C1(C)(NC(C(OC)OC)=O)CCN(C(c2c(F)cncc2Br)=O)CC1 Cc1nccc(C(=O)NCCC2CCCCN2C(C2CCC(O)C2)=O)n1 CC(CCNC(C1CCC(CNC(=O)C(C)(C)n2ccnn2)CC1)=O)C(F)(F)F C1(C(=O)NC2CCC(CNC(C(C(=O)OC)OC)=O)C2)CC2CCC1C21CC1 c1(CC)cc(C(=O)N(C)CCN(C)C(c2cc(C3(C)CC3)n[nH]2)=O)ncn1 c1(C(=O)NCCCN(C(=O)CS(=O)C(F)(F)F)C)cccc2[nH]nc(O)c12 C(N=c1[nH]c(=NCCc2cncs2)[nH]c2c1CCCCC2)C1CC(C)OCC1 N1(C(C2C(C(C)(F)F)C2)=O)CCN(CCOCCO)CC1.c12nncn1CCN2 C(=O)(C(C)(C(C)C)OC)NC1C(NC(COC)=O)CCC1.C1CC(OC)C1 c1(N(CCC#C)C)ncnc2c1ncn2C1CC(O)(C(F)(F)F)CO1 C1(C(=O)NC(c2ccns2)C)COCCN(C(c2nc[nH]n2)=O)C1 Cc1c(C(N2C(C(=O)Nc3cnn(C)c3C(C)C)CC2C)=O)cccc1F C1(C(N2CCC(N(CCC)C(c3cccc[n+]3[O-])=O)C2)=O)CCC2(CCC2)C1 N1(C(Cc2nc(COC)sc2)=O)CC(NC(c2ncccc2C)=O)C2CC12 N1(C(CCOC(CC(C)C)C)=O)C2CCC1CN(C(=O)CCC(F)F)CC2 O=S(=O)(c1ccc(F)c(F)c1F)N1CCC2CCCCC2C1c1ccccc1OC CC(C(=O)N1CC=CC1C(=O)NCC(=O)N1CCCO1)C(F)(F)F C(=O)(C(C)S(N)(=O)=O)N1CCN(C2CCN(C(Cn3c(C)ncc3)=O)C2)CC1 CC(C)(C)C(O)C(=O)N1CC2C(C(N3CC4(CCC4)C3)=O)C2C1 CCS(=O)CC(=O)NC(c1ccc(Cl)n1C)c1nnnn1CC(F)F c1(CC)ccsc1C(N1CCC(CCNC(=O)CN2CC=CC2)C1)=O n1(CC)cnc2nc(=NCC3CC3(C)C)[nH]c(NCCNC3(CO)CCSCC3)c12 C(=O)(C1CCc2cccc(O)c21)NC1CC(F)(CNC(c2cc(C)nn2C)=O)C1 CCCN=C(NCC1(CC(F)F)CCC1)N1CCCC(CSC)C1 C1(Cc2ccccc2)C(=O)O1.CCCC(C1CCC1)NC(=O)CC c1(OC)ccc(N(C(=O)NCCC(O)CO)C(C)C)cc1N(C)C C(=O)(CCC(C(C)C)NC(=O)CCP(C)(C)=O)NC(c1nn[nH]n1)CC C1(CC(=O)NCCC2N(C(CC#N)=O)CCC2)CCC2(CC1)CC2 N1(C(CNC(CCC)=O)=O)CCOCC1CCNC(=O)CC(C)n1cccn1 CCC(CC)C(C)C(=O)NCC1CCN(C(=O)Cc2ccc(=O)n(C)c2)C12CC2 C12(CS(C)(=O)=O)CCCC(CN1CCNc1nc(C)cc(OC)n1)C2 c1(CC(C(=O)NCC(C)N(C)C(C2(C3CCCCO3)CC2)=O)C)ccccc1C S(=O)(=O)(c1cnc(NCCN(C)CCO)c(Cl)c1)N1CC(CC)SCC1 Cn1cnc2cncc(C(=O)NCC(C3CC3)NC(c3cc(=O)n(C)o3)=O)c12 c1(C(=O)NCC(CC)(C)NC(=O)C(F)CC2CCC2)cc2occc2n1C C1(C(N(CCS(=O)(=O)NC)C(C)C)=O)CCC(n2cc(C(O)C(C)C)nn2)CC1 N1(C(CC(CC)C)=O)CCC2(CC2NC(C2CC23CCSCC3)=O)C1 Cc1c(C(=O)NCC2C3CN(C(=O)C(F)C(C)C)CC23)nc(O)c2ccccc12 c1(C(=O)NC2CN(C(c3sc(C)c(O)n3)=O)CC(O)C2)cnc2sccn2c1=O c1(C(N2CCC(C(C)C(=O)NCCCN3CCCC3=O)C2)=O)c(C)csc1C C=CC1CCCCN1C(=O)C(F)CC1CN(C(c2c[nH][nH]c2=N)=O)C1 C1(CC)(NC(=O)Cn2nccn2)CCCN(C(C2CC2c2ccncc2F)=O)C1 C1(C(=O)NCc2c(CCNC(CN(C)C3CC3)=O)ocn2)CCc2c[nH]nc2C1 c1(N2CC3N(C(C4CC4c4ccccc4)=O)C3C2)ncnc2cc(Br)sc12 C1(C)(NC(c2cc(-c3cn(C)nn3)on2)=O)CCN(C(C2CCC(=O)C2)=O)CC1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2ncn(C(C)C)n2)=O)ncc1F N1(C(c2nc(Cl)ccc2F)=O)CC2CCN(C(C3(CO)CC3)=O)CCC2C1 CC(C)C(C(=O)NCCN(C1CCCC1)C(C1CCC(F)C1)=O)C1CCC1 c1(C(N2C(C(C)NC(=O)COCC(C)(C)C)CCC2)=O)ccc([N+](=O)[O-])c(Cl)c1 N1(C(c2c(C)cc(F)cn2)=O)CC2CCOC2(CNC(=O)CC2CCOC2)C1 c1(C(=O)NC(CC=C)CNC(c2cn(C(C)(C)C)cn2)=O)ccc2nn[nH]c2c1 C1(N(C(c2cccnc2)C(=O)Nc2nncn2C)C)CCN(C(=O)CNC=O)C1 N1(C(c2cnc(C)[nH]2)=O)CC2C(NC(=O)CC(C)CC(C)C)CS(=O)(=O)C2C1 CCC(C)C(O)CC(=O)NCC(C)(C)CC(=O)N1CCCC(CO)C1 CC1(C2CCN(Cc3cn(Cc4ncc(Br)cn4)nn3)CC2)COC(=O)N1 CCC(C(=O)N1CCC(C(C)NC(c2cc(-c3cnccn3)[nH]n2)=O)C1)OC c1(OC)ccc(C(=O)N(C)CC2CCCN2C(=O)CC(C)CF)cc1O Cc1cc(N)cc(C(N2CCCC(NC(c3cnn(C(C)C)c3F)=O)C2)=O)c1F c1(CC(=O)NCC2(C)CC(NC(c3cn(CCC)nc3)=O)C2)c(Cl)cccc1Cl c1(OC)cc(C(=O)N(C(C)CNC(=O)C=C(C)C(F)F)C)cc2cn(C)nc12 C(=O)(C(C)(F)C(C)(C)F)NCc1cn(CCNC(C2ON=C(C(C)C)C2)=O)nn1 c1(OCCC(=O)OC2CCCC2OCCC(Cl)Cl)ccccc1 c1(OC)cc(NC(c2ccc(NC(c3cc(Cl)cc(I)c3)=O)nc2)=O)cc(O)c1 CCC(C(C)(F)F)NC(C1(C)CCN(C(C2CC(OC)C2)=O)C1)=O C1(NC(c2ccc(CCCC)cc2)=O)CN(C(=O)C(O)CSC)CC1(C)C Cc1ccnc(C(=O)NCC2CCCN(C(c3ccc(C(F)(F)F)nc3)=O)C2)n1 C(=O)(C1=CC(O)CCC1)N(CC(C)NC(c1ccc(NC(C)=O)cc1)=O)CC c1(OC)ccc(C(=O)NCC(C)NC(=O)C=C(C)C)cc1-n1c(C)ccc1C c1(OC(=O)OCC(CO)OC)ccc(OC(F)F)cc1 O=NN1CCCC1C(=O)NC1CCCCC1CNC(=O)CCCC1CCCO1 CC1CCCN(C(=O)CNS(N)(=O)=O)C1CNC(=O)C(F)CC1CCOC1 N1(C(c2ccc(-c3ccco3)[nH]2)=O)CCN2C(=O)NCCC2C1 C#CCCCCC(=O)NC1CCN(C(c2[nH]ccc2COC)=O)CC1F c1(C(=O)NCC2N(C(C3CC(C)OC3)=O)CC2)nc(-c2ccccc2)ncc1Cl C1(C(N(C2CCN(C(=O)Cc3cccc(Br)c3)CC2)C)=O)CC12CCOC2 C#CC1CN(C(=O)CCCSCC)CCN1C(=O)C=Cc1ncc(C)[nH]1 c1(C(=O)NC2CCC(n3cc(-c4cc(C)sc4)nn3)C2)cc(Cl)cc(Br)c1 CC1=C(C(=O)NCC2CCC(C(=O)NC3CSC(C)C3)C2)CCCO1 CCC(CC)CCCC(=O)NC(C)(C)C(N1CCOC(CC)(CC)C1)=O NS(=O)(=O)c1scnc1C(N1CCCC1c1cn(Cc2ccncc2)nn1)=O C(=O)(CCCC(C)=O)NC(CC=C)C(N1CCOCC12CC2)=O N1(C(CC(C)N(C)C)=O)CCOC2(CCN(C(=O)C=CBr)CC2)C1 N(C(=NCC1CCC1)N1CCC(C2CCOC2)C1)Cc1cn(CCN(C)C)nc1 C(=O)(C#CC1(C)COC1)N1CCC(CC=C)(NC(c2cc(C)c(Br)s2)=O)C1 c1(C(=O)OC(N)=O)[nH]c(C)c(C(=O)CN(C(c2ccc(Br)cc2)=O)CC)c1C C1(C(=O)Nc2ccc(C(N)=O)nc2)CC2CCC(C1)N2C(=O)CCc1cn[nH]c1 C(N=c1[nH]c2cccc(C)c2o1)C1(NC(Cc2c(C)nn(C)c2)=O)CCCC1 c1(C(N(CCNC(C2(COC)CC2(F)F)=O)C2CC2)=O)ccc(CO)cc1OC O=c1cc(C(F)(F)F)nc2ccc(N3CCCCC(N4CCOCC4)C3)nn12 CC(C)C1=NOC(C(=O)N(CC(=O)O)Cc2cn(Cc3csc(Cl)n3)nn2)C1 C1(C(=O)NC(C)(CNC(c2csc(C#N)c2)=O)C2CC2)C2(CCC2)C12CCC2 C1(C(=O)NC2(C3N(C(CC(C)OC)=O)CCC3)CC2)COC2COCC12 Cc1ccc(C)c(CC(N2CCN(C(C3CCCN3C)=O)C(CC3CC3)C2)=O)c1 N1(C(C2(CC#C)CCCO2)=O)CC2(C1)CN(C(=O)COC1COC1)CC2CO N1(C(CCCCCC#C)=O)CC2CN(C(c3nn(CCC)cc3Cl)=O)CC2(C)C1 CC(C)(CCC(=O)NC1CC2CC1N(C(c1csc(Cl)c1)=O)C2)[N+](=O)[O-] O=C1CCC(C(=O)NC2C3CCC2N(C(c2nc(C4CC4)ncc2Cl)=O)C3)=NN1 CC1(C)CCN(C(C2CCSCC2)=O)C1C(N1CC(N2CCCC2=O)C1)=O C1(CNC(C2C(C)(CC)C2)=O)CCN(C(C2CCCN(C)C2)=O)CC1C N1(C(c2n(CC)cnn2)=O)CC2CCC1C(CNC(c1cnc(O)n1C)=O)C2 CCCCCCC(C)(CC)C(=O)N1CCC(N(CCC)C(c2n[nH]cc2F)=O)C1 N1(C(c2c(C)nccc2)=O)CCN(C(c2ccnn2C)=O)CC(O)C1 CC1(C)CCC(F)(F)CC1N1CCN(C(c2cc(O)cc(Cl)c2Cl)=O)CC1 c1(OC)ncccc1CN(C(=O)COC)Cc1nc(-c2cccs2)oc1C C(c1ccsc1Br)=CC(=O)NCC1COC(=O)N1 c1(C(N2C3C(CNC(c4c(COC)scc4)=O)C(C3)C2)=O)cc(Cl)cc(Cl)c1N C(=O)(CC(O)CN(C)C)N(CCOC)CCNC(C1CCC(C)CC1)=O CC(C1CCCCC1)=CC(=O)NC1CCCC(N(C)C(c2nocc2C)=O)C1 N1(C(C(C)OCc2ccccc2)=O)CCCCC(NC(c2cc[nH]n2)=O)C1 C1(C(C)NC(c2c(C)nsc2)=O)CCCN(C(C2(C(F)F)CC(O)C2)=O)C1 c1(CCOC)ccc(F)cc1C(=O)NC1(CCO)CCCCC1 C(CC(C)C(=O)NCC1C(CNC(=O)CNC(=O)NC2CCCC2)C1(F)F)=CC c1(C(=O)NCCN(C(C2(c3oncc3C)CC2)=O)CC)ccnc2ccccc12 c1(NC(c2ccc(OCC)c(Cl)n2)=O)cc(Cl)c(C)cc1Cl c1(C(=O)NC2C(NC(C=C(C)Cl)=O)COC2)cccc(C#CCO)c1 C(CCCCC(=O)NNc1cccc(Cl)c1)n1cc(CCN(CC)CC)nn1 N1(C(CC2C(C)C(=O)CC2)=O)CCC2CCC(NC(c3ccc(CO)o3)=O)C1C2 C1(C(N2CCCC(N(C(=O)Cn3ncnn3)C)CC2)=O)CC2CC1C1CC21 C1(N(C(C(C)n2cncn2)=O)C(c2cccnc2)C2CCCCO2)CC2CNC1C2 CN1CC(C)(C(N2CCCC(n3cc(C4(CO)CC4)nn3)CC2)=O)CCC1=O c1(C(=O)NC2CCC(CCNC(CCOCC#C)=O)C2)c(F)ccc(F)c1Cl c1(N2C(CNC(Cc3cncc(C)c3)=O)CN(C)CC2)ncnc(C)c1Br CCCC(C)(C)C(=O)N1CCC(CC(=O)NCCC(N)=O)C1 C1(C(=O)NC(C(C)C)C(C)(C)CO)CCc2ccccc2C1O c1(COC)ccoc1N(C(C1CCSCC1)C(=O)NCCSC)C c1(-c2c(C(=O)Nc3c[nH]nc3Br)nccc2)ccc2nc[nH]c2c1 N1(C(C(C)(C)N)=O)CCOCC(C(NC[Si](C)(C)C)=O)C1 C(=O)(C(C)(C)C(=O)N(C)C)N1CCC(NC(CCc2onc(CC)n2)=O)(CO)C1 N1(C(c2cc(COC)on2)=O)CC(C)CN(C(=O)C(F)n2cccn2)C(C)C1 Cn1nnc(CNC(c2ncn(C)n2)=O)c1C(N1CC2(CSC2)C1)=O N1(C(c2c(C)nccn2)=O)CCC2CC2(C(=O)N(C(C)(C)CO)C2CC2)CC1 c1(OCC)cc2c(cc1C(=O)NC13CC(C(N4CCOCC4)=O)(C1)C3)OCCO2 c1(NC(C(=O)NCC2(c3cc(C)on3)CCC2)=O)ccc(C2CNCCO2)cc1 Cc1nc(C(=O)N(C)CC2CCCN(C(=O)CC3CCC3C)C2)n(C)n1 C1(NC(c2cccc(C)c2)=O)CN(C(c2nn(C)nc2Br)=O)CCC1O N1(C(c2c(CCC)n[nH]c2)=O)CCC(C(=O)NCC2CCC(F)(F)C2)C12CCC2 C1(C(=O)OC)CCCCC1C(=O)NCCC(C(C)C)NC(C1CC2CC2C1)=O CC1CC2(CC(C(=O)NC(C)C(C)NC(C3CCCCNC3=O)=O)C2)C1 N1(C(c2c(C#C)c[nH]n2)=O)CC(CNC(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 N(C(=NCc1ccc(N(C)C)cc1)NC(C)CCC(=O)OCC)C(C=C)C Cc1cc(C(=O)NC2CC2CNC(c2cc(CC(C)C)[nH]n2)=O)ccc1C1CC1 c1(C(=O)NCC(C)CNC(=O)COCC2(F)CC2)coc(C(F)F)n1 C1(C(=O)OC)(CNC(=O)CN(C(c2c[nH]cc2C)=O)C2CC2)CC=CC1 Cc1cc(C(=O)NC2CCC(CNC(C3CN(C)CCO3)=O)C2)ccc1Cl N1(C(C(CC2CN(C(CCOC(C)C)=O)C2)F)=O)CCCCN(C)CC1 Cc1oc(C2CC2)nc1C(N1CCC(N(C(=O)C(N)=O)CCO)CC1)=O c1(C(C(=O)N(CCCNC(=O)CCc2ccn(C)c2)C)=O)ccc(C(N)=O)cc1 N1(C(=O)COC2COC2)CCOC2(CCCN(C(C3CC4(C3)CC(F)C4)=O)C2)C1 N1(C(CCNC(COC)=O)=O)CC2CN(C(c3onc(Br)c3C)=O)CCC12 c1(CC)ccc(C(=O)NCC2CN(C(C3(OC)CCCOC3)=O)CCO2)nc1 c1(C(=O)NC(C(C)NC(=O)CCc2cncs2)C)c[nH]nc1-c1ccsc1 C(C(CO)(CO)NC(c1cnn(C)n1)=O)N(C(CC1C(C)C1)=O)C O=C(C1CCc2nccn21)NCCC1CN(C(=O)CCC2=CCCCC2)CCO1 C(=O)(C(F)CCC(C)(C)C)NCC(C)(C)OCC(=O)NC1(C#C)CC2CCCC12 CCC(C)C(O)C(C)C(=O)NCC1(OC)CN(C(=O)CC(C)CC)C1 C12(C(N3CC(O)(CCNC(c4cccc(Br)n4)=O)C3)=O)CCC(CC1)C2 C=CC(C)(O)C(=O)N(CC(C)C(=O)N(CCCC)C)C C=CCC(C(=O)NC1COCC1O)NC(c1nc(C)sc1C)=O c1(C(=O)OCC)cc(C(=O)N(C(C)CCNC(=O)C(=O)NC2CC2)C)on1 N1(C(Cc2cc(C(C)C)no2)=O)CCCC(CNC(C2CCCC2(C)C)=O)C1 Cc1ccnc2ccc(C(=O)N(O)Cc3cn(-c4cc(Cl)cc(Br)c4)nn3)cc12 N1(C(c2ccc(C)cn2)=O)CCCN(C(C2CCC(C#N)CC2)=O)CC1C c1(C(=O)Nc2c(C(=O)NC)cccn2)cn(C)c2ccc(C3=CCOC3)cc12 C1(O)(CN(C)C(c2coc(CO)c2)=O)CCN(C(=O)Cc2cn(C)cn2)CC1 Cc1cc(Br)cc2cc(C(=O)NC3C4CCN(C(=O)C(C)C#N)C34)[nH]c12 C12(CC(=O)N(C)Cc3ccccc3F)CCC1CN(C(c1ncccc1N)=O)C2 C1(O)(C(C(=O)N(C)CCC2CCCC2)F)CN(C(C2(F)CCCC2)=O)C1 N1(CC#CC)CCC(C2CCCN(C(C3CCC=CCC3)=O)C2)C1 N1(C(c2c(OC)ccs2)=O)CCC2(CCC2)C(NC(=O)C(C)(CC)OC)C1 N1(C(CC=CC)=O)CCC2CCN(C(c3ccc4c(c3)C(=O)NC4)=O)CC12 c1(NC(C2CCN(Cc3cncc(OC)c3)C2)=O)ccc(C)c(OC)c1 c1(C(N(CCCCNC(CCC#CC)=O)C)=O)cc(F)cc(F)c1Br C(=O)(C(C)C(C)n1cccn1)N(CC(=O)NCC1(NC(c2ccsc2)=O)CC1)C c1(C(N2CC(C)(CNC(c3ccc(SC)nc3)=O)C2)=O)cc(C#N)ccc1Cl c1(CC(C(=O)NCCN(C(=O)CCC2CCOC2)CC)C)ccc(OC)cc1 S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)N1C2CC(NC(C(C)=O)=O)CC1CCC2 c1(NC(C2COC(C)(C)C2)(c2n(CC)nnn2)C)cccc(C2CCCCO2)c1 c1(C(=O)OCC)c(NC(=O)CC2CCCN2C(=O)C(C)CC(N)=O)sc(C)c1C Cc1cc(C(=O)N(CC(C)O)CCNC(C2CC(C)(C)CO2)=O)ccc1[N+](=O)[O-] O(NC(=O)C1=NN2CCC(C)N=C2N1)N(CC(C)NC(=O)OC(C)(C)C)CC C1(CNC(CSC)=O)CCN(C(c2cc(Br)cn2C(C)C)=O)CC1(F)F c1(NCc2c(F)ccc(N)c2)cc(=NCC(=O)N2CCCC2)[nH]cn1 N1(C(C(=O)NC)CC(C)C)CCOC(C)(C)C1(C)C N1(C(CC(N)Cc2cccc(F)c2)=O)CCC2(CCO2)CC1 N1(C(=O)C2=CCCOC2)CCCC2(CCCN2C(C2CCC3(C2)CC3(F)F)=O)C1 C1(CNC(C2N(N=O)CCC2)=O)CC2CCC1N(C(C1CC(=C3CC3)C1)=O)C2 C(=O)(C(C)C(C)S(C)(=O)=O)N1C(CN(C(c2c(C)n(C)cc2)=O)C)CCC1 N#Cc1ccc(O)c(CN2CCCC(C(=O)NCc3cnc[nH]3)C2)c1 C1(C(CNC(=O)C(c2ccc(F)cc2)F)NC(c2ccon2)=O)CC2CCC1C2 Nc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(-c3c4c(nn3C)CCC4)cc2)c1 CCC1=NOC(C(N2CCC(N(C(=O)CC(F)(F)F)CC)C2)=O)C1 c1(C(=O)NC2C(CNC(C(C)O)=O)C2)c[nH]c(Br)c1 c1(C(CCCC)C)nc(-c2cnn(C)c2)nn1CCCn1ccnc1 c1(C(=O)NC2C(NC(C(C)O)=O)C2)cn(C)nc1-c1cccs1 c1(N(C)C)cccc(C(=O)NC2(CNC(=O)COCCF)CCCC2)n1 Cc1n[nH]c(C)c1C(=O)N(C1CCCN(C(=O)C(C)OCCC(C)C)C1)CCO c1(C(=O)NC2CCC(CNC(=O)CCCCCl)CC2)n[nH]c2ccccc12 N1(C(=O)CC2COC(C(F)(F)F)C2)CCCC(N(c2cc(O)ncn2)CCO)C1 CN=c1nc(N2CCN(C)CCN(C)CC2)[nH]c(=NCc2cc(C)cnc2O)[nH]1 C1(COC)(NC(=O)CC(C)n2cccn2)CCN(C(=O)C(C)(C)c2cnsc2)C1 C(CC(C(=O)N1CC(N2CC(F)C2)C1)NC(=O)CC(C)n1cccc1)SC CC(=O)CC(C)(C)CC(=O)N1CC(NC(=O)C=Cc2cn[nH]c2)CC1C C1(NC(C(N)=O)=O)CCC(NC(=O)CCc2cccnc2)CC1 C=CCCC(CC(C)C)C(=O)N1CCC(C2(NC(=O)CC3CSCCS3)CC2)C1 Cc1ccc(CN2CCCCC2)c(O)c1.N12CCCCC1(C)C(=O)NCCC2=O N#Cc1ccnc(NCc2ccccc2-n2nccn2)n1 N1(C(c2cnc3ncccn23)=O)CCCC2(CCCCN2C(=O)CC(Cl)Cl)C1 C(=O)(C1=NN(C)C(=O)CC1)NC1C(CNC(CCCC(=O)N(C)C)=O)C1 N1(C(C2(C#N)CCOC2)=O)CC(CC(N2CCCC(O)(CO)C2)=O)C2(CC2)C1 C(=O)(C(F)CCC(C)(C)C)NC1C(CC(=O)N(CC(CC)O)C)CCCC1 N1(C(c2cn(C)c(=O)n2C)=O)CCCC(C2CN(C(=O)C(F)n3ccnc3)C2)C1 c1(C(N(C(C(N2CC3(N(C)CC3)C2)=O)(C)C2CC2)C)=O)cnn2ccc(Cl)c(F)c12 C1(CNC(=O)Nc2cccc(C)c2)CN(C(C2CCCC2)=O)CC12COC2 N1(c2ncn(C)c(=O)c2)CC(NC(c2cc(Cl)nc(Cl)c2)=O)CC(C)(C)C1 C(=O)(C(CCC1CC1)NC(C1C=CC=CC=C1)=O)N1C(C)(CCO)CC1 c1(C(C)NC(CN(C(=O)CCc2ccn(C)n2)CCC)=O)ccnc(C)n1 c1(C(N(CC(C)NC(CCCOc2c(C)cccc2)=O)C)=O)cnccc1C#N CCC(C)CCCC(=O)NCCOCCNC(=O)Cn1cc(C2CCOC2)cn1 CCCCCC(C)CC(=O)NC(C)CCC(=O)NCC1CC(C#N)C1 c1(C(=O)NC(CN(C(C(F)=CCC)=O)C)CC)ncc(C#N)cc1Cl c1(CC(N2C(C3(O)CN(C(CCC=C)=O)C3)CCC2)=O)ccnc(C)c1 c1(C(=O)NC(C(C)NC(c2c(NC(C)=O)cccc2)=O)CO)cccc(C)c1C Cc1cc(C)c(CC(N2CCC(N(C(=O)C(C(C)C)c3ccncc3)C)C2)=O)s1 c1(C(N2CC(CCO)(NC(C3SC4C=CC3C4)=O)C2)=O)ccc(C(F)F)cc1 C1(OC)CCn2cc(C(N3CCC4CN(C(=O)COC5CC5)CC4C3)=O)nc2C1 C1(NC(CC2(C)CC2)=O)CCN(C(=O)CCCC2(C)NC(=O)NC2=O)C12CCCC2 n1(CC(=O)NCc2c(C)cncc2)ccc(=O)c2ccccc12 c1(C(=O)NCC(C)N(C(c2cc(OC)nn2C)=O)C)nc(C)c(C)cc1N N1(Cc2nn(C)c(=O)n2C)CCC2(NC(C3CC3(C)C)=O)CCCC12 N1(C(C(CC)C)=O)CC(C(=O)NCC(F)(F)C(C)C)C(C)C1 C1(O)(CNC(C(CNC(c2nccc(CC)c2)=O)C)=O)CCC(C)(C)C1 c1(OC)cc(C(=O)OCC(c2ccnn2C)O)c2c(c1)CCC2 c1(C2(C(c3n(CCCC)nnn3)NC(C)C(C)C)CCC2)ccccc1Br N1(C(CC23C(CN(C(C(CC=CCC)C)=O)C2)CC3)=O)CC2(CCN(C)CC2)C1 c1(C(C(=O)NCCN(C(C(C(C)C)F)=O)C(C)C)(C)C)ccc(Cl)cc1F c1(NC(COCc2cn(CCC(C)C)nn2)=O)ccccc1C(N1CCCC1)=O CCC(C)(CCC(C)C)C(=O)N1CC2C(NC(=O)C(=O)C3CC3)C2C1 N1(C(Cc2n(C)ccn2)=O)CCC2CN(C(C3CCCCC34CC4)=O)C2C1 c1(CC)nc(=N)[nH]cc1C(=O)NC1(CCO)CN(C(=O)CSC)C1 N1(C(COc2c(N)ccc(C(F)(F)F)c2)=O)CCc2c(Cl)cccc21 c1(C(N2CCC(NCCCCCC)C(C)C2)=O)ccc([N+](=O)[O-])cc1 c1(OC)ccn2ncc(C(=O)NCC3CC(NC(=O)CCCN=[N+]=[N-])C3)c2c1 C1(NC(CCCOCCOC)=O)CC2CC(NC(=O)C(F)(F)CN(C)C)C2C1 C1(CCNC(=O)CSC(F)(F)F)CCCN1C(=O)CCc1nncs1 c1(CC(=O)NC2C(CNC(=O)CC3CCC3)CCC2)cccc2ccoc12 C(CCCCC(=O)NC1CC(O)CN(C(c2cccc(C)n2)=O)C1)NC(C)=O S(=O)(=O)(c1ccccc1)NCC(C)NC(=O)N=c1ncn(C2CCCC2)[nH]1 N1(C(C(C)Oc2cccnc2)=O)CCC(NC(=O)CC2CCC(C)C2)C(C)C1 N1(C(Cc2nc(C)c(C)s2)=O)CCC(NC(C2(CF)COC2)=O)C(C)(C)C1 C(=O)(C(C)(O)CC(C)C)N1CC(O)(C(C(N2CCC(OCC)CC2)=O)F)C1 N1(C(C(=Cc2ccco2)C)=O)CCC(C)(NC(c2ccn(C)c2)=O)CC1 N1(C(C=C(CCC)CCC)=O)CCC(CC)CC1C(=O)NCCC(O)C(F)(F)F C1(CNC(c2c(C)nn(C3CC3)c2)=O)CN(C(=O)CCCC2CC2C)CC1(C)C C1(C(=O)NCC(CC)C#N)CCC2CCC1N2C(=O)C=Cc1cnn(C)c1 N1(C(C2(CC#C)CCCC2)=O)C2CCC1C(C)C(NC(C1CC1CCC)=O)C2 C1(N(C(CCSC(C)(C)C)=O)C)CCCCC1N(C(=O)C(C)NCCC)C N1(C(c2nc3ccc(C(=O)O)nn3c2)=O)CC(S(=O)(=O)CC(F)(F)F)C1 C(=O)(CCCC(=O)NC(C)C)NCC(CCOC)NC(C1CC2CC2C1)=O N1(C(c2c(OC)cnnc2)=O)CC(CNC(C2(C)CCC2)=O)CC(C)C1 C#CCC(C)(C(=O)N(C)CCOCCOC)NC(C1CCC2CC1CO2)=O Cc1cnccc1CC=C1CCN(C(c2ccncc2F)C(=O)NCC(F)F)C1 N1(C(C2(CC(c3ccccc3)C)CCCCO2)=O)CCOC2(CCN(OC)C2)C1 CCCC(C(=O)OC)NC(=O)NC1CCC(C(=O)OC)C1 N1(C(C2CCCN(CC)C2)=O)CC2CCCC2C1C(=O)N(CCCC(=O)NC)C c1(COC(C(COC)OC)=O)cccc(F)c1 N1(C(C2(C=C)CCC2)=O)CCC2(CCCCN(C(=O)C(C)(C3CC3)OC)C2)C1 CC(C)(C)CCC(=O)N1CCC(c2cn(-c3ccc(F)cc3Br)nn2)CC1 c1(C(N2CC(C)C(CNC(=O)C3=CCCCCC3)C2)=O)[nH]cc2c1CCS2(=O)=O CON(CCC(=O)NCC1CCC2(CC2)CO1)C(=O)C1CCS1(=O)=O C1(C(N(C2CC(NC(c3n[nH]cc3F)=O)C2)C)=O)CCCC1n1cccc1 N(C(=NCCCC1CCOC1)NCC1CCOC1)Cc1c(=O)cc[nH]c1 c1(C(N2CCC(N(CCC)C(c3nncn3CC)=O)C2)=O)cc2sc(Cl)cc2[nH]1 N1(c2nnc(COC(C)C)s2)CCC(c2cccs2)CC1 c1(N2CCC(CCNC(c3sccc3F)=O)C2)nc(O)c2ccccc2n1 c1(N(C)Cc2nccc(C)c2)ccc(S(=O)(=O)NCCC2CC2C)cc1Cl C1(CC(=O)N(CC(N)=O)CC2CC2)CCCC1CNC(c1csc(F)c1)=O CC1(C)CC(NC(c2cc(Cl)ccc2N)=O)CN1C(C1CC2C(C1)C2(F)F)=O O=S(Cc1cccnc1Br)CCCCc1ccccc1Br C(=O)(CCC#Cc1ccccc1)N1C(CCNC(CCCCCOC)=O)CCC1 c1(C(N(C(c2ccccc2)CNC(C(CC)C)=O)C)=O)cc2cccnc2cn1 C1(C)(CNC(C2C(NC(C3N(C)CC3)=O)C=CCC2)=O)CCCC(=O)N1 C(=O)(C(CC(C)(C)C)OC)N(C)CC1CCN(C(c2n(CCC)ccc2)=O)C1 C1(C(N2C(CCNC(C=CCCC=C(C)C)=O)CCC2)=O)Cc2nnc(C)n2C1 C1(NC(c2c(C)cn(C)n2)=O)CC(C)CN(C(C23CCCN2CCC3)=O)C1 Cc1c(C(N2CC(NC(=O)C(C)O)C(C)C2)=O)[nH]c2c1CCCC2 C(CN=c1cccc(S(=O)(=O)N2CCC(CCO)CC2)[nH]1)N1CCC(C)C1 C1(NC(c2n(C(CC)(C)C)nnn2)c2ccsc2)CCOC2(CCOC2)C1 C1(C(=O)NC2C(NC(C(C)c3cc[nH]n3)=O)CCC2)CC2(C1)CC1(CC1)C2 c1(C(=O)OC)[nH]c(=NC2CC3CN(C(c4c(OC)noc4C)=O)CC23)sc1C Cc1nc(=O)c2c(C)c(C(=O)NC3COCC3NC(=O)CC(C)F)sc2[nH]1 N1(C(C(CC)C(C2(CCn3ccnc3)CCCC2O)=O)=O)C2CCC1CC(CO)C2 c1(CC)ccc(C(=O)NC2(CNC(C3CCN(C)C(C)C3)=O)CCOC2)cc1F S(=O)(=O)(c1c[nH]ccc1=NCCOCCF)NCCN(CC(C)C)CC c1(C(C)CC(=O)N(C)CCN(C(=O)CCc2cc[nH]n2)C)ccc(F)cc1 CCC(C)CCCCC(=O)N1CCCC(NC(=O)COc2cccc(Cl)c2)C1C N1(C(C(C)OC)=O)CCC(OCCNC(=O)NCCc2nnc(O)s2)C1 N1(C(CCCn2cc(CC(=O)OCC)nn2)=O)CCCC1(C)CN1CCNC1=O C1(C(=O)NC(C(C)(C)CO)CO)CCCCCCN1C(=O)CSC(F)F C1(OC)CC(CNC(C2(N3CCCC3)CCC2)=O)N(C(c2[nH]c(C)cc2C)=O)C1 CCN=c1[nH]cc(C(=O)NCC2CC3CN(C(C4(C)CCCCO4)=O)CC23)s1 n1(CC)nccc1C=CC(=O)N(CC(O)CN(C(=O)C(C)O)C)C C(CC(C)C(F)F)NC(C(CC1CCCC1)NC(C(C)NC(C)=O)=O)=O C1(NC(c2c(OC)noc2C)=O)COC2(CCN(C(=O)CSc3nc[nH]n3)C2)C1 c1(C(=O)NC(C)CCNC(C2CCCC2O)=O)cnc2ncnc(O)c2c1 C(=O)(CCC(C)C)NC1(CNC(=O)C(C2(C)CCCCC2)OC)CC(OC)C1 CCC(CC)C(C)C(=O)N1CCC(CN(C(=O)CCSC(F)(F)F)C)C1 c1(NC(C2N(C(C3(CC)CCOCC3)=O)C(C3CC3)CC2)=O)ccc(C)c(Cl)c1 c1(C(=O)NCc2cc(C(=O)NC(c3ncnn3C)CC)on2)cn(C)c(C)n1 c1(CCC(=O)NC2(CCNC(c3n(CC)ccc3)=O)CCC2)cccnc1Br C1(O)(CNC(=O)CCn2cnnn2)CCCN(C(c2c[nH]c(Br)c2)=O)C1 N1(C(C2CN(C(C)C)C2)=O)CCCC(C2CN(C(c3ccnnc3)=O)C2)C1 C(=O)(C(C)(O)C(F)(F)F)Nc1nc(OC)c(C(=O)N(C)CCCl)cc1 c1(C(=O)NC(CCC)CNC(=O)CCc2ncc(C)[nH]2)c(C)cccc1O c1(C(=O)NCC(C)NC(c2cccc(C(C)C)n2)=O)cc(F)c(O)c(Cl)c1 N1(C(CCC(CC)=O)=O)CC2CC(NC(c3ccnc(C)n3)=O)CC1C2 N1(C(CC=CCC)=O)CC(NC(c2c(C(C)C)cccc2C)=O)CC12CCOC2 N1(C(COCCC)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC1C NS(=O)(=O)c1cc(C(=O)NCC2CCN2C(=O)CC2CCOC2)c(Cl)o1 N1(C(C2(C#C)CCC2)=O)CCN(C(c2cc(F)ccc2Cl)=O)C(CC(F)(F)F)C1 c1(CC(=O)NCCC(=C)CNC(C2CC2(F)F)=O)ccc2c(c1)CCCS2(=O)=O C1(CC(=O)NCC(CNC(C2(C#N)CCCC2)=O)F)CC2C=CC1CC2 O=S(=O)(c1cccnc1NC1CC1)N1CCC(OC2CCC2)CC1 c1(C(C(=O)NC(C2CN(C(=O)CCOCC3CC3)C2)C)N(C)C)ccccc1 C12(C(C)NC(c3coc(CNC(=O)CC(=O)N(C)C)n3)=O)CCC(CO1)C2 N(C(=NCCCCCC1CC1)NCc1cnc(O)c(F)c1)C(c1cccs1)C C1(NC(C(c2cccnc2)C)=O)COCCN(C(=O)CSC(F)F)C1 C1(NC(C(C)(CO)OC)=O)CN(C(c2ccsc2C(F)F)=O)CC2CC12 C12(NC(CSCC=C)=O)COCCC1CN(C(c1cn(CCO)nc1C)=O)C2 c1(C(=O)OC)cc(CC(N2CC=CC(NC(=O)C(C)OC)C2)=O)ccc1Cl N1(C(Cn2ccc(C)n2)=O)CC(C(=O)NCc2n[nH]cc2C)C(C(C)C)C1 Cc1[nH]nc(CO)c1C(=O)NCCN(C1CCCC1)C(=O)C=Cc1cccnc1 C(=O)(C1=NOC(C)(C)C1)N1CC(C(C(N2CC(C)=C(C)CC2)=O)O)C1 C=CCCC(C(=O)NCC(O)CN(CC)CC)NC(=O)C(CO)OC C(=O)(C(C(=O)NCc1cn(CCNC(C2(F)CCCOC2)=O)nn1)C1CC1)OCC N(C(=NCCCCn1ccnc1)N(C)CC1CCC(F)(F)CC1)C(CC)C c1(C(N(C2CN(C(=O)CC3(O)CCC3)CC23CC3)C)=O)ccc(N)c(Br)n1 c1(CCNC(N)=O)nc(-c2ccccn2)nn1-c1ccccc1F C(CO)(C(C)NC(C1(Cl)CC1)=O)NC(C(C1CC1)SC)=O c1(C(=O)NCC(C)N(C(c2ccnc(C(C)C)n2)=O)C)c(N)cccc1Cl C1(CNC(=O)CCc2cccnc2C)CCC(C)(NC(CC(=O)NCC)=O)CC1 C1(C(N(CC(=O)N(C2C(C)CCCC2)C)C)=O)C2CCC(C2)C1C c1(C(=O)NCCCCNC(C2CCS(=O)(=O)N2)=O)ccc(=O)n(CC(F)(F)F)c1 C1(NC(c2ccncc2F)=O)CC2CN(C(c3cccc4c3COC4)=O)CC2C1 C1(C(=O)NCC(N(C(C(C(C)C)C)=O)C)C2CC2)CC(F)(F)CCC1(C)C CC1(C)CCN(C(=O)C2=C(Cl)CCC2)C(C(N2CCCCC(F)(F)C2)=O)C1 Cc1ccc2oc(=NCCC(C)(C)NC(c3cccnc3F)=O)[nH]c2c1 C(=O)(C(C(C)C)n1cnnn1)NC(CN(C(C(CC)Sc1ccccc1)=O)CC)C C(=O)(CCCCCCCCC1CC1)N1CCN(C(C2C(=C)CC2)=O)CC1CO C1(NC(C=Cc2cc(OC)ns2)=O)CN(C(=O)C(C)(F)F)CC12CCOCC2 N1(C(c2c(CC)occ2)=O)CC(F)(F)CC1C(=O)NCCN1CC2CC2C1 c1(OCC)ccc(C(=O)Nc2nnc(CO)s2)c(-c2ccnn2C)c1 C#CC1CN(C(=O)C(C2CCC2)NC(=O)C=NOC)C1 N1(C(CC=CC=C)=O)CCC2(CC1)CC2NC(=O)CC(C)(C)C(=O)OC(C)(C)C C1(CC=C)(NC(c2cc(C)ncn2)=O)CCN(C(c2c[nH]nc2CC)=O)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)C(c2ccncc2)C)ccc2ocnc2c1 Cc1c(C(N2CCC(NC(=O)C(C)(C)F)C(CO)CC2)=O)[nH]c2c1CCCC2 N1(C(C=CC=CC)=O)CCC(C(N2CCC(CCCO)C2)=O)CC1 c1(C(=O)NC2CC3(CN(C(c4c(C)nn[nH]4)=O)C3)OC2)ccc2[nH]nc(Cl)c2c1 CC1(O)CCC(CC(=O)NCCCCCNC(=O)Cn2cccc(O)c2=O)CC1 CCC(C)(C)C(=O)C(=O)N1CCC1C(=O)NCC1SCCS1 c1(CC(=O)NC2CCN(C(CCCC(C)=O)=O)C(C)C2)c[nH]c2cc(C)ccc12 N1(C(CSC)=O)CC2(C1)C(NC(c1oc(C)nc1C)=O)CCS2(=O)=O C1(NC(c2c(C)ocn2)=O)CCCCC12CCN(C(=O)C(C)(C)C1CCC1)CC2 C(C(C)CN=c1nc(-n2cccn2)cc(C)[nH]1)NC(c1ccc(OC)c(Cl)n1)=O N1(C(C(N)Cc2cnc[nH]2)=O)CCC2(CC=CCO2)CC1 N1(C(CCN(C)C)=O)CCCC(C)(NC(c2cnccc2C(F)(F)F)=O)C1 c1(CCC(=O)NC2C3CN(S(=O)(=O)CCBr)CC23)ccc(C(F)(F)F)cc1 CCC(CC(=O)NCc1nc(C(N2CCC(CCO)C2)=O)c(C)o1)OC c1(C(=O)NC2C=CCN(C(c3cc(F)ccc3F)=O)C2)cccc2c1CCC2 C1(NC(c2cc3n(c2)CCC3)=O)CCN(C(C2CCSCC2)=O)CCC1CO C1(NC(=O)C=CCNC(c2cnc(Cl)[nH]2)=O)CCN(C2CC2)C1=O CCC(F)(F)CC(=O)NC(C12CCC(CC1)C2)CNC(c1cnoc1C)=O c1(CC(=O)NCCN(C(c2cc(CCCCC)[nH]n2)=O)C)noc2ccccc12 CC(C)(C)C(C(=O)OCC(=O)Nc1cc(Br)ccc1F)C(=O)O C1(COC)CC(CNC(=O)CC2CC(CF)C2)N(C(c2nn(C)cc2C)=O)C1 N1(C(C2N(C(c3c(OC)noc3C)=O)CSC2)=O)CCC2C(C1)C2(F)F C123COCC1CN(C2)C3=O.C1(C(=O)OC)CCC(NC(C2CCCC2C)=O)C1 C12(C(=O)NCC3CC3NC(C34CC3COC43CCC3)=O)CCC(O)(CC1)CC2 Cn1ncnc1-c1cn(CC2CC(CNC(C3(Br)CC3(F)F)=O)C2)nn1 N1(C(C2CCC(N(C)C)C2)=O)CCCN(C(C2(N(C)C)CCC2)=O)CC1 C1(C(=O)NC(C2N(C(c3c(CC)nco3)=O)CCC2)C)CC(C2CCCC2)C1 n1(CC)nc(C)cc1C(=O)NCC(=O)NC(C)CC1CCC1 c1(CCC(=O)N(CCCNC(C2CCCCC2O)=O)C)cc2ccccc2[nH]1 CCC(C)CCCC(=O)N1CC(OCCNC(=O)Cc2cc(C3CC3)no2)C1 c1(C(=O)NCCC2CCC(NC(C3(C)C(C)C3)=O)C2)ccc(CO)c(Cl)c1 C(CC(C)(C)C)(C(=O)N1CC(C)CC1C(=O)N(C12CC(C1)C2)C)OC c1(CN(C(c2nc(CC(C)C)co2)C(=O)NCCSC)C)ccc(SC)cc1 C1(CCN(CC(C)C)C(=O)C=CC(C)(C)NC(=O)OC)CCCCC1.C(C)(C)C C12(C(N3C(CNC(c4c(C)n[nH]c4)=O)CC4(CC4)C3)=O)CCCC(=O)N1CCC2 C(=O)(C1CCCn2ncnc21)N(C1CCN(C(c2cc(C)c(C)[nH]2)=O)C1)CC C1(C)(CC)C=C(C(=O)NCC=CC(=O)NCCc2ccc(F)nc2)C1 c1(OC)ccc(C=CC(=O)N(CCNC(c2ccc(C#N)[nH]2)=O)CC2CC2)cc1 C1(NC(C2CC23CCOCC3)=O)CCSC12CN(C(c1cnn(CCO)c1)=O)C2 Cc1nn(C)c(C(N2CCC(NC(=O)C(c3ccccc3)NC(N)=O)C2)=O)c1F c1(C(N(CC(C)CNC(=O)Cc2ccn(C)n2)C)=O)ccc2nnn(C)c2c1 c1(C(=O)NC23CC(NC(C4C(C#C)C4)=O)C(OC2)C3)cc(S(N)(=O)=O)ccc1C c1(C(C)NC(C2CC(NCc3cn(C)nn3)C2)=O)ccc(C#N)cc1F C(=O)(C1CCc2cc(F)ccc21)NC(C)CNC(C1C2COCC12)=O C1(NC(CCc2nc(C)c(C)o2)=O)CN(C(C2CCOC2C2CC2)=O)CC1(C)C N1(C(C=Cc2ncc(C)[nH]2)=O)CC(NC(=O)C(C)CF)CC(C)(C)C1 N1(C(Cc2ccn(CC)n2)=O)CC2CC(NC(C3(C4CC4)CC=CC3)=O)C(C2)C1 C(=O)(CC(CNC(C1CN(CC(C)(C)O)CCO1)=O)CC(C)C)OC C1(NC(C2C3CN(C(C45CSCC4C5)=O)CC23)=O)CCn2cnnc2C1 C1(NC(C(c2cccc(Br)c2)OC)=O)C2CC1CN(C(C1CCSC1)=O)C2 c1(CC(=O)NCCOC2CN(C(C(C)C3CCC3)=O)C2)c[nH]c2ncccc12 CC1=C(C(=O)NC2CN(C(c3ccccc3C3CCC3)=O)CC2C)CCCC1 CC(C)CCCC(=O)NCCCC(=O)NCC#CC#CCO c1(C(=O)NCC2(NC(c3c(OC)cnnc3)=O)CCC2)cc2cc(F)ccc2[nH]1 C(=O)(C(C(C)C)n1cc(C)nn1)N(CCC(C)NC(C(C=CC)O)=O)C c1(SC)ccc(C(=O)NC2CCCC2CNC(=O)COC(C)C)cc1[N+](=O)[O-] c1(NC(C(n2cc(Br)cn2)C)=O)cccc(NC(C2CC(F)(CO)C2)=O)c1 C1(NC(Cc2ncc(CC)[nH]2)=O)(CNC(=O)Cc2ccoc2)CCCCC1C N1(Cc2ccc(C(N(C3(C(=O)NC)CC3)C)=O)s2)CC2CC(CO)C(C2)C1 c1(N2CCN(C(c3c(OC)nc(C)s3)=O)CC2)snc(Cl)c1C#N c1(CC(=O)N(C2CCN(C(C3CCN(C)C3)=O)C2)CC)cn(C)nc1C C=C1CCN(C(=O)CC2(OC)CCC2)C(C(=O)N(C2CCOC(C)C2)C)C1 CCC(CCCC(=O)N1CCCN(CC)CC1)NC(=O)CC1CN(C(C)=O)C1 c1(C(N2CCN(C(C(C#C)(C)C)=O)CC2C2CCCC2)=O)ncn2ccccc12 C(c1cccn1C)=CC(=O)N(CCN(C(=O)CC1CCC1(C)C)C(C)C)C C1(C(=O)NC2(CNC(CCOC(C)C)=O)CCCCC2)CCCC2(C1)CC2(F)F C1(NC(=O)NC2CC2)CC12CCN(C(c1nnc(C3CC3)s1)=O)CC2 C(=O)(C(C)(F)C(F)(F)F)NC1C(C)(C)CN(C(c2ccc(Br)cn2)=O)C1 C(CCN(C)C)(C(=O)NC(c1ncn(C)n1)C)NC(C1CC(=C)C1)=O C1(CNC(C2(NC(Cc3n(C)ccn3)=O)CSC2)=O)CCC(F)(F)C1 C1(C(N2CCN(c3cc(OC)ncn3)CC2)=O)CC(=O)N(C)C1c1cccs1 CC1(C)CCC(F)(F)CC1NC1(CO)CCC(C(=O)O)C1 Cc1cc(NC(c2ccc(C#N)o2)c2nnnn2CC2CCCO2)cc(C)c1O c1(C(=O)OC(=O)N(CCC(=O)OC)C(=O)C2CC2)cccc(F)n1 c1(C(N(C2CCN(C(C3CCSCC3)=O)C2)C)=O)cncc(N)c1 n1(CC)ccc(=NC(=O)C2CC(O)CCN2C(=O)C2=CCSC2)[nH]1 Cc1nc(C(C)(C)C)[nH]c(=NC2CC23CC(C(=O)CC(C)(C)C)C3)c1F c1(C(N(CCCN(C(=O)CC2CCCN2C2CC2)C)C)=O)cccc[n+]1[O-] C1(C(F)CF)CN(N(CC2CCCCO2)Cc2ccccc2)C1 c1(C(CC)C(=O)NCC(C)CN(C)C(c2cn(C)nn2)=O)cccc(Cl)c1 C1(N(C(C(C=C)OC)=O)CC2CC2)CCCN(C(=O)CC=CC)C1 c1(C(=O)NCCC(=O)OC)ccc(-n2cc(C3CC=CCC3)nn2)cc1 c1(C(C(N2CCOC(CNC(=O)C(F)(F)CO)C2)=O)O)ccc(Cl)cc1F c1(C(N2C(CNC(C(CCN(C)C)O)=O)CC(O)C2)=O)cc2c(s1)CCOC2 c1(COC)nc(Cl)cc(=NCCCC(C)NC(=O)Cc2cnc(C3CC3)s2)[nH]1 C1(OC)CCCCC1C(N1CC2CC1C2NC(=O)CN1CCCS1(=O)=O)=O C1(C)(COC)CC(NC(c2cnc(O)c(C)c2)=O)CN1C(=O)CC1CC(C)=NO1 C1(C(N2CCCC(CC)(NC(=O)C=Cc3ccoc3)C2)=O)CC12CCCCCC2 CCCCC(C)(F)C(=O)N1CCC(NC(c2cc3occc3[nH]2)=O)C(CO)CC1 c1(C(c2n(CCCC)nnn2)NC2CC2C2CCC2)ccc(F)c(C2CC2)c1 C1(C(=O)NC(CC)CO)CCOC1CNC(=O)Cc1csc(C)n1 c1(C(=O)NC2CCN(C(C3CC(CC)C3)=O)CC2)ccc(S(C)(=O)=O)[nH]1 c1(CC)ccc(C(N2CC(NC(c3ccc(N)c(N)c3)=O)C2)=O)c(C)n1 N1(C(C23N(C(C4CCCO4)=O)CC(C)(C2)C3)=O)CCOCC2(CC2)C1 C1(C(=O)NCC(C)(CO)NC(c2n[nH]c3c2COC3)=O)CC2CC1CC2O Cc1sc(C(=O)NCC(C)(C)CNC(C2CC3CCC2O3)=O)nc1Br N1(C(C2CCC(C)(C)C2)=O)CCCC(F)(CNC(=O)Cn2cnnc2O)C1 c1(OC)c(C(CO)NC(=O)NC2(CO)CC=CC2)cccc1Br C(=O)(C1COc2c(F)cccc21)N1CCc2c(cnc(C(=O)OC)c2C#N)C1 c1(CC)nnc(O)c(C(=O)NC(C)CCNC(C2COCC(C)(C)O2)=O)c1CC C1(N(C(=O)CC(F)F)C)CCCN(C(c2cscc2-c2ccccc2)=O)C1 C(C(C)(C)C(=O)NCCNc1ccc(CN2CCCC2)o1)N(C)C C(=O)(CC(O)(CCC)CCC)N1C(C2CCN(C(CCC(=C)Cl)=O)C2)CCC1 C=CCC(C)(C)CN=C(NC1CCCC1)N1CCN2C(=O)OCC2C1 c1(OC)ccc(C=CC(=O)NCC2CCN2C(C2CCCCC23CC3)=O)cc1F c1(CC(N2CC(OC)(CNC(C3CC(OC)C3)=O)C2)=O)coc2cc(Cl)ccc12 C1(NC(c2ccc(CC)[nH]2)=O)CC2(C1)CC2C(=O)N(C(C)CC(C)C)C c1(C(=O)NC(c2ccccc2)C(C)NC(=O)C=C2CCC2)ccn(C)c(=O)c1 c1(CC2CCN(C(CCCC#C)=O)CC2)ccc(C)c(C)c1.C1(=O)CCN1C1CC1 c1(C(=O)NC2C(OC)CN(C(=O)C(C)(CO)OC)C2)n[nH]c2c1CC1CC21 CCCC(C)(O)C(=O)NC(C)CN(C(=O)COc1ccccc1CC)C C1(NC(c2c(C)cc[nH]2)=O)CCC(n2cc(C3C=CC=CC=C3)nn2)CC1 C1(CCC)CN(C(=O)C=CC(C)CC)CCN1C(c1cn(C)nc1Br)=O c1(CN(C(c2n(CCC)ncc2)C(=O)NCC2CCCO2)C)ccccc1CO N1(C(C2CNC(=O)N2)=O)CC2(CC(NC(=O)C(c3ccccc3)N3CCCC3)C2)C1 C1(CCNC(c2ccns2)=O)(NC(CC2N(C)CCC2)=O)CCOCC1 S(=O)(=O)(c1cccc(C(F)(F)F)c1)NC1CC(C(N2CCC(CO)C2)=O)C1 N1(C(c2n(C=C)ncc2)=O)CCCC2(CCN(C(=O)C3=CCCCO3)C2)C1 C1(NC(C2C(CC)CCN2C(c2ccncc2F)=O)=O)CC2CCC(C1)N2C Cc1ccc(F)c(COC(c2cccc(-c3ccc(O)cc3)c2)=O)c1 c1(C(=O)NCCC2CCCN(C(C(C)OCC)=O)C2)ccc2c(ccn2C)c1 Cc1ccc(NC(c2cc(F)ncc2NC(c2ccc(Cl)c(I)c2)=O)=O)cc1F C1(NC(Cc2c(C)n(C)nc2)=O)CCN(C(c2cccc(CO)n2)=O)C1(C)C c1(OC)c(C(N2CC(CNC(=O)CC(C)OC)C2)=O)cc(F)cc1F C(=O)(C#CC1CCOCC1)N1C(CNC(c2c(C)ccc(F)c2)=O)C(C)(C)CC1 CC1CN(C(C2(C)CCN(C)C2)=O)CCC1C(=O)N(C)CC1CN(C)C1 c1(-c2ccc(C3(COC)CC3)cc2)ccc(-c2cn(CC3CC3(Cl)Cl)nn2)cc1F C1(CNC(C2(CNC(c3n(CC)ccn3)=O)CCCC2)=O)CCC2(CC1)CC2 N1(C(CC2CCN(C(c3c(CCC)[nH]cc3)=O)C2)=O)CCC(OC2CC2)CC1 C1(OC)CN(C)C(C)(C(N2CCN(CCCNC(=O)CCC(=O)NC)CC2)=O)C1 c1(C(=O)NCC(CC)(C)NC(C2CC2CF)=O)ccc2nccc(C)c2c1 N1(C(C(CC=C)OC)=O)CCC(F)CC1C(=O)NCCC(O)C(=O)OC Cc1ccc(C(=O)NCC2CCC(C)CN2C(=O)CSCCC(C)C)c(C)c1 C1(CNC(C2(C(N)=O)CC2)=O)CC(C(=O)NCc2cccc(O)n2)=NO1 N1(C(C(C(CC)O)(F)F)=O)CC=C(CC(=O)NC(c2nccs2)C)CC1 CC1CC(=O)NC(C(N2CC(C)(NC(=O)CCOc3ccccc3F)C2)=O)C1 c1(NC(c2nnnn2CCOC)(C2CC(=C)C2)C)ccc(OC)c(Br)c1 C=CCC(C(=O)N1CCCC1C=CC(N1CCC(OC)C1C)=O)NC(C)=O c1(C(=O)NCc2ccc(C(=O)NC3CC(F)(F)C3)cc2)ccc(=O)n(CCO)c1 C1(O)(C(=O)NCC2(C(F)F)CCN(C(c3cc(C)no3)=O)C2)CCCC(C)CC1 C1(C2CCN(C(=O)Cc3ccsn3)CC2)(NC(c2cc(CC)c(C)cc2)=O)CC1 C1(C(=O)NCCC(C)OC)CC2CCN(Cc3ccc(O)c(CO)c3)CC12 C(=O)(CC(=O)NCC(Cc1ccccc1)N(C(C12CC(F)C1C2)=O)C1CC1)OC O=C1Nc2c(C(N3CCC3C(=O)Nc3cccnc3Cl)=O)cccc2C1=O c1(C(=O)NC(CN(C(C(C)CO)=O)C)C)cc2cccnc2[nH]1 C1(C(=O)NC(c2ccsc2)C)CC(F)CN1C(c1ccc[n+]([O-])c1)=O CC1=CC(C(=O)NCCOCC(=O)NCCOC2CCOC2)SC1 c1(C(=O)NC2CCN(C(C3CC34CC4)=O)C2)n[nH]c(C2CC2)c1Br Cc1ccccc1-c1ccc(N2CCC(S)C2)cc1.C(=O)(C(O)C(C)C)N1CCCCC1 C(=O)(C(F)C(F)(F)F)NC(C(=O)N(C1C(C)C1)C)CO CCCCC(C)(F)C(=O)NC1CCOC1C(=O)NCc1ncn(CC)n1 CC(C)C1=CCC(NC(=O)C(C)(C)C(C)NC(=O)CCC2CC2(C)C)CC1 c1(C(=O)OC)cc(C(N(C2CCN(C(=O)CC)CC2)CCO)=O)c(C(=O)O)o1 c1(C(=O)NCC(CNC(c2nc(C)sc2C)=O)(C)C)cc(F)cc(F)c1N N1(CC(N2C(CN(C(=O)C(C)(C)NS(C)(=O)=O)C)CCCC2)=O)CCCCS1(=O)=O N1(C(C2CCN(CC)C2)=O)CC2CCC(C1)N2C(=O)Cc1c(C)cnn1C N1(C(CCOC)=O)CCC2(CC1)CCN(C(=O)CC1CC(C)(C)OC(C)(C)C1)C2 c1(C(C(=O)NC2(CC=C)CN(C(C3CC3COC)=O)C2)C)ccc(C)cc1 C(=O)(C1=CC2CCCC12)NCC1(NC(CCC(N)=O)=O)COC1 C1(C(N2C(CN(C(COC)=O)C3CC3)CCC2)=O)C(C2CC2)C1(F)F c12ccc(cc1C(F)(F)F)NC(=O)C2.C1(C(=O)NCC)(C(C)C(=O)OC)CC1 c1(C(C)=O)[nH]c2ccccc2c1C(=O)NCCN(C(=O)C1CCc2c[nH]nc21)C CC1(C)CN(C(C2(C)CCCO2)=O)CC(CNC(c2ncn3ccccc23)=O)O1 C(CC(CNC(=O)CCCc1cccs1)NC(=O)C(C)NS(C)(=O)=O)OC CN1N=CC(CC(N2CCC(OCC(=O)N(C3CCOCC3)C3CC3)C2)=O)C1=O C1(NC(C(C)O)=O)CCC2(CC1)CCN(C(C1CCCN1S(C)(=O)=O)=O)CC2 c1(C(N2CC(OC)(CNC(C3CC4(CC4)C3)=O)C2)=O)cnn2c1CC(C)CC2 N1(C(C(C2(O)CN(C(c3c(C)coc3)=O)C2)F)=O)CCCC(N(C)C)C1 c1(-n2cc(C(=O)NC3CCN(CC)C3)nn2)ccc(C)cc1F CCC(CC(C)C)C(=O)N1CCOCC1CNC(C1(OC(C)C)CCC1)=O Cc1nn(C)cc1CC(=O)NCc1ncoc1C1CN(C(c2ccn(C)n2)=O)C1 c1(C(=O)NC2CCC(N(C(c3c(COC)cco3)=O)C)C2)sc(C)cc1C c1(C(N2C(CNC(C(C)(C)OC)=O)CN(C)CC2)=O)ccc2nc(O)n(C)c2c1 c1(C(N(CC(CN(C)Cc2ccc(Cl)cc2Cl)O)C)=O)cncc2ccsc12 C(=O)(C(CCc1ccccc1)N1CCOC(CCO)C1)NC(c1ccccc1)C C12(C(=O)NCC(C3CCCCC3)NC(C(CC)SC)=O)CCC(N=[N+]=[N-])C1C2 c1(OC)cc(CN2CC3(CC3)CC2C(=O)Nc2cc(Br)ncc2F)cc(Br)c1 c1(N(CCNC(=O)C(C)N(C(C2CCCC2)=O)CC)CC)ncnc(Cl)c1C#N C1(NC(CCC(=O)NCC)=O)CN(C(=O)COc2cncc(Cl)n2)CC(F)(F)C1 c1(C(=O)NCC2N(C(c3ccc(C)cc3)=O)CCCC2C)ccc(N)c(F)c1F C=CC(C)CC(=O)N(CC(C)N(C(=O)C(F)CC1CCCC1)C)C N1(CC(N2CC(CS(C)=O)C2)=O)CCC2(CC1)CC(O)CNC2=O c1(C(=O)N(C2CC(C(=O)NC)C2)C)ccc(NC(CC2C(CC)CC2)=O)o1 C#CC1CC2CCC1N(C(c1coc(CNC(c3ccc(F)c(O)c3)=O)c1)=O)C2 c1(CC)ccc(C(=O)NCC23CC2CN(C(=O)CCC2CC(F)(F)C2)C3)cn1 CC(C)(Cc1ccccc1)C(=O)NCC1CCCCN1C(c1cc(CF)on1)=O Cc1c(CC(=O)NC2C=CC(NC(=O)CNc3ccccn3)C2)cnn1C n1(CC)cc(Cl)c(C(=O)NC(C2CCN(C(C3SCC=C3C)=O)CC2)CO)n1 C(=O)(CC(C)(C)CNC(=O)CCc1ccncc1)NC(C(C)C)(C)C C1(C(N2CC3(C2)CN(C(C2(CO)CCC2)=O)C3)=O)CCn2nnnc2C1 c1(C(=O)NCC(C2CCOC2)NC(CCCCC#C)=O)ccc2nn[nH]c2c1 N1(C(c2scc(OC)c2OC)=O)CCC(C)N(C(=O)CC2SC(=N)NC2=O)CC1 C(=O)(CCC(=O)NCC(N1CCCCC1)(C)C)NC1C(NC(=O)OCC)CC1 CC(C)CC(C(=O)NCC(F)C1CCC1)NC(C1CN(C2COC2)C1)=O N1(C(C(CCC)NC(C)=O)=O)CC2CCC1C(NC(C13CCC(CC1)OC3)=O)C2 CC1CN(C)CC(C(N2CC3CC(CNC(c4ccc(N)c(N)n4)=O)C3C2)=O)O1 c1(-c2onc(C)n2)ccc(C(=O)NC2(CN(C)C(c3ncoc3C)=O)CC2)cc1 C(CCCC(C)(C)C(=O)NNC(=O)C1CCC(F)(F)C1)NC(C(C)OC)=O CC(CC(=O)NCCCC1CCCN1C(=O)CN1CCCCC1=O)C(F)F C1(CN(C(C(C)Cn2cccn2)=O)C)COCCN1C(=O)C=Cc1cccs1 C1(C(=O)NC(CC2CN(C(c3ccc(C)s3)=O)C2)C)CCC(=O)N1C N1(C(c2cc(C)oc2C)=O)CCC(F)(CNC(=O)CNC=O)CC1 c1(OC(c2nn(C)c3c2COCC3)=O)cc(F)c([N+](=O)[O-])cc1F c1(CC(=O)NCC2(C(=O)NC(C(COC)C)C)CC2)ncccc1F c1(C(=O)NC(C)CNC(c2cc3c(ncn3C)s2)=O)ccc(F)c2cccnc12 C(=O)(C(C)CC(C)(F)F)N1CC(CCC)N(C(=O)C(=O)NCC2CC2)CC1 N1(C(CNC(CCCCC)=O)=O)CCOC(C(=O)NCC2(COC)CCC2)CC1 N1(c2nnc(CC)n2CCn2cnnn2)C2CCCC1CNC2 CC(C)(S(C)(=O)=O)c1cn(CCNC(C2(C)CC=CCC2)=O)nn1 c1(C(N(CC(C)NC(CCC#CC)=O)C)=O)c(OC)ccc(Cl)c1F N1(C(C2C=CCC2)=O)CC2(C(N3CC4(C3)CC4(F)F)=O)CCC1CC2 N1(C(C(C=C)(C)CC)=O)CCCN(C(=O)C(CCSC)OC)CCC1 C1(C)(C(=O)NCCC2(O)CN(C(C3(C#N)C(C)C3)=O)C2)CS(=O)(=O)C1 CC1CCCCC1(CNC(=O)C1=CCCCC1)NC(=O)COCP(C)(C)=O c1(CN2C(C)(C(N3CCC(C)(OC)C3)=O)CCC2)ccc(Br)cc1I C1(NC(C(C(C)O)C)=O)CS(=O)(=O)CC1N=c1ccnc(C2CC2)[nH]1 C1(C(=O)NCC(C(C)(C)C)NC(c2c(N(C)C)ccnc2)=O)CC2(CC2)CN1C N1(OC)CCC(NCc2n[nH]c(COc3ncc(Br)cn3)n2)CC1 C1(C)(CNC(c2c(CC)[nH]c(=N)s2)=O)COCCN(C(=O)CC(F)(F)F)C1 C(=O)(CCC(C)CN(C)C)N1CC(C(CCNC(c2cnc(SC)s2)=O)O)C1 Nc1ccc(S(=O)(=O)N2CCCC2c2nc(C(=O)O)co2)c(F)c1 CN1CC2CC(C1)N2C(C1CCN(C(=O)c2nonc2N)O1)=O C(=O)(CC=C(Cl)Cl)NC1(C)CC(NC(c2[nH]cc(C(C)=O)c2)=O)C1 Cc1ccc(C(N2CCCC2CC(=O)Nc2cccnc2F)=O)c(Br)c1 N12CC3(CC(C3)CC(=O)NCC(C)C1=O)C2.C1(NCCSCCOC)CC1(F)F c1(OC)cc(C)cc2cc(C(=O)OCc3cc(I)ccc3F)sc12 C1(C(N2CCN(C(C(F)=CC)=O)C(CS(C)(=O)=O)C2)=O)CCn2c(O)nnc2C1 N1(C(c2cc(C(=O)OC)cc(F)c2)C(=O)NCCC)CCCCC12CCOC2 CC(C)CC(O)C(=O)NC1CCN(C(C2CC(O)CN2C)=O)CC1 C1(CC(=O)NOCCF)CCCC(NC(=O)CC2CC(=O)NC2=O)C1 c1(C(=O)NCc2ccc(OC)cc2)ccc2c(C)c[nH]c2c1 c1(C(=O)NC2C(C(C)(C)C)N(C(C3COC(=O)N3)=O)CC2)ccc2snnc2c1 c1(C(=O)NC2CCC(CC(N)=O)C2)cc2ccc(Br)cc2c(=O)o1 C#Cc1ccnc(C(N2CC3(C2)CN(C(=O)CN(c2ccccc2)CC)C3)=O)c1 c1(CNC(CC2CC(C)C2)=O)ccc2c(c1)CCCC2NC(c1cncnc1)=O c1(C(N2CC(C)(C(=O)Nc3cnc(C)c(Cl)c3)C2)=O)c(F)ccc([N+](=O)[O-])c1C C(=O)(C1CCCc2sc(C)nc21)N1CC(CNC(C(CC)O)=O)(OC)C1 CCN(OC)C(=O)C(C)N(C)C(C1(F)CC=CCC1)=O c1(C(=O)NC2(CC=C)CCN(c3ncncc3Br)C2)cccc2nc(C)[nH]c12 Cc1ncnc(N2CCC(CNC(=O)C3=CCCC3)C23CC3)c1Br NC(Cn1cccn1)C(=O)NCC1OCCO1 N1(OC)CCC2CN(Cc3ccccc3)C2C1.C1(C)(C)CCNC1 C1(CNC(C2C(C(=O)OC)C2(C)C)=O)CC2(CO1)CN(C(c1cnco1)=O)C2 C1(CNC(C(CC)NC(C)=O)=O)CN(C(=O)CCCC2CCC2)C2COCC2O1 c1(OC)cccc(C(=O)NC2CC(NC(C3C(C)C3C)=O)C2)c1C N1(C(CC(COC)COC)=O)CCN(C(C2CCC(=O)C2)=O)C2CS(=O)(=O)CC12 c1(NC(C2C(C(=O)NCc3nc(C)c(Br)s3)C2)=O)cccc2ccccc12 N1(C(C2C(C(=O)OC)C2)=O)CC2CC1C2NC(=O)CCc1ccncc1 CC(C)(C)C1=NOC(C(N2CCC(F)(CNC(C3C4(CC4)C34CC4)=O)C2)=O)C1 C1(C)(C(=O)NC2C=CC(CC(N3CC(SC)C3)=O)C2)CCOC1C C(C(CC(=O)N1CCC1C)C1CCC1)NC(C1(COC)CCC1)=O N1(C(c2cc(C(N)=O)oc2)=O)CCCCC(CNC(C2CSCCS2)=O)C1 c1(C(=O)NC2CN(C(C3CC(SC)C3)=O)CC2C(F)F)ccnn2ccnc12 C1(CC(=O)NC)CN(C(=O)CNC(c2ccsc2)=O)CCN1C(=O)CC(C)C(F)F n1(CCC(=O)NC2(C)CC(NC(CCC(C)OC)=O)C2)ccc(O)nc1=O c1(CC)cc(F)ccc1C(=O)NC1CN(C(=O)Cc2csc(Cl)c2)CC1O C(=O)(C(O)CC(C)(C)C)N1CCN(C(COCc2n(C)ccn2)=O)CC1CCO c1(Nc2ccc3oc(Sc4n(C)nnn4)cc3c2)cc2c(cc1F)NC(=O)CC2 c1(N(C)C)nc(Cl)c(C(=O)NC2(CNC(=O)Cc3ccc(O)nc3)CCOC2)s1 C(=O)(C(CCCC)NC(c1csc(C)c1C)=O)NCC(=C)C(F)(F)F C1(C(=O)NCc2n(C)ccn2)Cc2ccccc2CN1c1ccnc2ccnn12 C1(C(=O)NCC(CC=C)NC(c2cncc(COC)c2)=O)CCCC(C)O1 n1(C(CC)C)ccc(=NC(=O)c2coc(CNC(C3(CC(=O)OC)CC3)=O)c2)[nH]1 N1(C(C2(CC=C)CCOCC2)=O)CC2CC(NC(C3CC(=O)N(C)C3)=O)C2C1 N1(c2n(CC(C)OC)c(C3CC3c3ccc(F)cc3F)nn2)Cc2ccccc2C1 CC1CN(C(=O)CCNc2nccs2)CC2(CCN(C(=O)C3=CCSC3)CC2)O1 c1(C(N2C3C(NC(C(=O)NCCOC)=O)C(C3)C2)=O)cc(S(N)(=O)=O)n(C)c1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NCC(c1ccncc1)C)CCC1CC1 C#CC1(NC(=O)C(C)N(C(=O)COCCF)C2CC2)CCCCC1 C1(CCNC(c2c(C)snc2)=O)CCCCN1C(=O)CSc1cccc(Cl)c1 C(c1ccc(Br)s1)=CC(=O)NC(C)C(CO)NC(C1CC1C(F)F)=O C(=O)(C(C)C(C)N(C(=O)CNC(=O)COC)C)N(CC)CC.C(C)C CC1CC(NC(C2CC3CCCC23)=O)CN1C(=O)C(c1ccccn1)O Cc1cc(F)ccc1CNC(C1CC(NC(c2ncccc2Cl)=O)C1)=O C1(C(=O)Nc2ccc(O)cc2)CC2OCCC2N(C(=O)C2=COCCC2)C1 Cc1cc(C(=O)NCC2(Cc3cn(CCN4CCOC4=O)nn3)CC2)cc(C)c1 N1(C(COCCOCC#C)=O)CC(F)CC1C(=O)NCCCCCO C(C(C)(O)CNC(C1CCOC1CNC(c1ncsc1NC)=O)=O)SC C12(NC(Cc3c(Cl)cn(C)n3)=O)COCCC1CN(C(c1cn[nH]c1)=O)C2 C(=O)(C(CC(C)CC)NC(=O)CN(C)C(C)=O)NC(CC#C)C(N)=O Cc1nc2ccc(C(=O)NCCCCNC(c3cc4cccnn4n3)=O)cc2o1 C(=O)(C(CCC(C)(C)C)NCC1COCCN1)OCC N1(C(C(C)SCC#C)=O)CCC(NC(c2cnn(CCO)c2CC)=O)C1CC N1(C(CC(C2CC2)NC(C(CC)C#N)=O)=O)CCCC(N=[N+]=[N-])C1 O=S(=O)(c1c(F)cc(Cl)cc1Br)NCC(C(F)(F)F)OC(F)(F)F CC(CC(=O)N(CCCNC(C12CC(C)C1C2)=O)CCO)c1ccccc1 N1(C(CCC#CCOCOCC(C)O)=O)CC(=O)Nc2ccccc21 C1(C(=O)NC(CCCC=C)C2CC2)CC(N=[N+]=[N-])CN1C(c1cc[nH]n1)=O C1(NC(=O)NCc2sc(Cl)cc2Br)CC2C3C=CC(O3)C12 c1(OCC)c(F)ccc(C(=O)N(C)CCNC(=O)CSCC2CCCO2)c1F N(S(=O)(=O)N1CCCC1C(=O)O)Cc1c(F)ccc(OC)c1F N1(C(C2(C(=O)OC)CC2)=O)CCC2(CC1)CCN(C(=O)CCC(F)F)CC2C N1(Cc2c(OC)cc(I)cc2)CCC2CN(C(c3cc(O)nc(O)n3)=O)CC12 c1(C(N(CC(C)N(C(Cn2c(C)nnn2)=O)C)C)=O)cc2n(n1)C(C)CCC2 C(C(N=[N+]=[N-])C(=O)N(C)CC1CCCN1C(C1(O)CCSCC1)=O)OCC N1(C(c2ccc(CCCC)cc2)=O)CCC(NC(=O)C(C)=CC2CC2)C(O)C1 c1(C(=O)NCCCN(C(=O)Cn2cc(C3CC3)cn2)C)cc(F)c2[nH]nnc2c1 c1(C(N(C)COC(C)(C)C)=O)cc(-c2ccco2)no1.C12CC1NC2=O c1(C(=O)NC2(C)CN(C(c3nncc(C)c3)=O)C2)ccc2ccn(C)c2c1 c1(CCC(=O)NC(C2N(C(C(C)Cn3ccnc3)=O)CCC2)C)ccc(F)cc1 c1(C(N(CCCNC(=O)CCOC)CC)=O)cc(SCC)cc(Cl)c1 Cc1cccnc1CC(=O)NCC1(C(=O)NCCCCO)CCCC1 C1(C(=O)NC(CSC)(C)CO)CC(F)(F)CN1C(c1cncc(C#N)c1)=O CCC(CC)C(=O)NCCCCN(C)C(C1C2CCCC12)=O c1(C(=O)NC2CCC(C)N(C(=O)Cn3ncn(C)c3=O)C2)cc2n(c1)CCCC2 C1(NC(C=CCCC)=O)CC(OC)CN(C(C2(c3ccc(Cl)nc3)CCC2)=O)C1 C(=O)(C(C)C(C)n1cccn1)NCCN(C(c1csc(C)c1N)=O)CC c1(OC)ncccc1SCC(=O)NCCOCC(=O)NC(C)C C(=O)(CC(C)CC(C)(C)C)N1CC(C(=O)Nc2cn(CC)nc2)C(O)CC1 CC1CC2CCN1C2=O.C(C(F)(F)C(F)F)OCC(=O)Nc1ccsc1 C1(CCO)(NC(=O)CCN(C(=O)CC2CCCOC2)CCO)CCOCC1 c1(C(=O)NCC(CC)NC(=O)CN2CCCCC2=O)cc(C)c(C)c(C)c1 Cc1c(CC(=O)NC23CC(CNC(=O)CC4CCC(F)(CO)C4)(C2)C3)ncn1C C#Cc1ccc(CC(CNC(=O)Nc2c(C)ccnc2OCC)CO)cc1 C(CN=c1[nH]c2cc(Cl)ccc2s1)N(C(=O)CN1C(=O)NC(C)(C)C1=O)C(C)CO Cc1ncccc1CCC(N1CC2CC2(CNC(C2CCSC2)=O)C1)=O N1(C(c2n(OC)cnc2C)=O)CCCCC(NC(c2ccc(Cl)cc2Cl)=O)CC1 O=C(C1CCCc2ncnn21)NC1CCN(C(=O)C(F)=CC2CC2)C1C1CC1 CN1CC2(CCN(C(=O)Nc3cc(I)ccc3F)C2)CC1(C)C c1(N2C(C(C)(C)CNC(C34CCC(CC3)C4)=O)CCCC2)cnc(C#N)cn1 c1(C(C2(OC)CCCC2)N(C(C)CC(=O)OC)C(=O)C(F)(F)F)ccc(F)cc1 CC1(C)COC(C(N2CC(OCCNC(=O)CCC3CCCCC3)C2)=O)C1 CC(CC(C)(C)C)C(=O)NC(CC(F)F)C(=O)NCCCC(=O)NO N1(C(C2(CC#C)CCC2)=O)CC(NC(C2CC(C#N)C2)=O)C2(CCC2)C1 N1(C(C2CCC(C)C2)=O)CCOC2(CCN(C(=O)C=CC(=O)OC(C)(C)C)CC2)C1 c1(C(=O)NCC2CCCCCO2)c(F)cc(O)cc1F C(=O)(CS(=O)c1ccc(N)cc1)NC(c1c(CC)n(Cc2ccccc2)nc1)=O c1(C(=O)NCC(CNC(C2(c3cccc(C)c3)CC2)=O)F)nc[nH]c2ncnc1-2 c1(OC)ccnc(CC(=O)NC2CCN(C(c3ccc(NC(C)C)nc3)=O)C2)n1 CCCCCCC(CC)C(=O)NC(C)C(C)NC(c1ccc(C2CC2)nc1O)=O N1(C(c2ccc(CC)s2)=O)CCCC(O)(CN(C)C(C2CCN(C)C2)=O)C1 c1(OC)cc(CNC(C2CC3CC3N2Cc2ccccc2SC(F)(F)F)=O)ncn1 N1(C(CCCOCCOCC)=O)CC2CCC1CN2C(c1cc(O)nn1C)=O CC1(C(=O)NC2COCCC2NC(C23CCC(CC2)O3)=O)CCS(=O)(=O)CC1 C(=O)(CCCC(=O)N(C)C)N(C1CCN(C(C2C=C2C)=O)CC1)CC C12(CNC(c3ncc(OC)cn3)=O)CCCC1N(C(=O)C(C)S(C)(=O)=O)CCC2 c1(SC)ccc(C(=O)NCCCC(C)NC(c2cc(CN(C)C)c[nH]2)=O)c(Cl)c1 C(CCS(=O)(=O)N1CC(F)CC1CC(=O)O)N(C)C C1(C(=O)NC(CC)C(C)C)CC2CCCC2N1C(=O)C=C1CCCCC1 c1(C(=O)NC(CC)CN(C(=O)CCCSC(C)(C)C)C)cc(OC)nc(F)c1 CCC(C)C(O)C(C)C(=O)N1CCCC(CNC(=O)COC(C)(C)O)CC1 C(C)(CCC(F)(F)F)NC(CNC(CNC(c1nc(OCC)oc1)=O)=O)=O CC1CN(C(=O)C(c2ccccc2F)N(C)C)CCN1C(=O)OC(C)(C)C C1(NC(CN(CC(O)CC(C)C)C(COC)=O)=O)CCC(NC(c2nc[nH]n2)=O)CC1 N1(CC(=O)NCCC(CNC(CN(C)CCO)=O)O)C(=O)CCC1=O C1(c2nn[nH]n2)(C(=O)NC2CC(n3cncn3)C2)CCCC1 N1(C(c2ccc(N(C)C(c3nc(C(C)=O)sc3)=O)cc2)=O)CC(C)OC(C)C1 C1(C)(CC)CC(C(N2CCC(F)C(NC(=O)CSCCOC)C2)=O)CCO1 c1(NC(=O)NCCC2(C(=O)O)CC2)cc(F)cc2c1OCCC2 C(=O)(CCCC(F)(F)C(F)(F)F)N(C)CC1(NC(C2Cc3nccn3C2)=O)CC1 C1(NC(c2coc(Cl)n2)=O)CCC2CN(c3nccc(-n4ccnc4)n3)CC2C1 Cn1c(C(=O)NC2CC3(C2)CN(C(C2CC(=O)NC(=O)N2)=O)C3)cc2sccc12 N1(C(C(C(C)C)N=[N+]=[N-])=O)CC2(C1)CN(C(c1cccc(O)n1)=O)CC(C)(C)O2 N1(C(CNC(CCC)=O)=O)CC(CNC(=O)CC2CN3CCN2CC3)C(F)(F)C1 C(=O)(C(C(=O)N(C)CC1CN(C(=O)C(c2ccccc2)F)C1)C(C)C)OCC C1(NC(=O)C=Cc2cnc[nH]2)CCN(C(C2(c3ccno3)CC2)=O)C12CC2 c1(C(=O)NCCCC2(NC(c3cc(C)nnc3)=O)CC2)[nH]cc2c1CCCC2 N1(C(C2N(C(C)C)CCC2)=O)CCOCC1CNC(c1ccc(N(C)C)cn1)=O CN1Cc2ccc(C(N3CCC(N(C(=O)CN4CC=CC4)C)C3)=O)cc2C1 N1(C(c2nc(CC)sc2N)=O)CCCC(CNC(c2cnn[nH]2)=O)CC1 CC1=NOC(=O)C1CC(=O)NCCC1(O)CN(C(=O)C(n2cc(Cl)cn2)C)C1 CC1CCN(C(=O)CC2CCC(=O)N2)C(CNC(c2cccc(N)n2)=O)C1 CC(C)(C)C(O)C(=O)N1CCCC1CNC(=O)C=Cc1ccc(C(F)(F)F)cc1 CC(C)(C)CCCC(=O)N1CC2CC2(CNC(c2cccnc2OC(F)F)=O)C1 N1(C(c2ncccc2F)=O)CCC2CC(C1)CN(C(=O)CC1CC=CC1)C2 C1(C(N(C2CCN(C(Cc3ccc(C)s3)=O)CC2)C)=O)CCC2(CCCO2)CC1 CC1CN(C(=O)C(C2CCCO2)NC(=O)C#CC(C)(C)O)C(C)CO1 c1(C(=O)NCC(C)(CO)NC(C)=O)c(F)ccc(OCF)c1F C12(C(=O)NCCSCCCCCO)CC(CN(C(=O)CCC3CCCCO3)C1)C2 CC(O)CCCCCC(=O)NC1(CNC(=O)CCn2cccnc2=O)CCC1 N1(Cc2n(C)nc(C(F)(F)F)c2)CCC(NC(C2CC=CC2)=O)CC(C)(C)C1 CC1C(=O)NC(C)CN1C(=O)C(n1cc(C2(NS(C)(=O)=O)CCCOC2)nn1)C c1(C(=O)NC2CCN(C(c3nc(C)oc3C)=O)C(C)C2)c(C)ccc(C)c1O N1(C(=O)OC(C)(C)C)CCC(N(CC(CC)(F)F)C)CC1 N1(C(C2C(CNC(C3CCCCC3)=O)CCC2)=O)CCC(O)(CC=CCO)CC1 C#Cc1cc(F)c(C(N2CCOC(CNC(C3(CC)CC3)=O)C2)=O)c(F)c1 C1(OC)(OC)CCC(CN2C(=S)N2)C1.c1(NC(C)=O)cccs1 C1(C(C(=O)N(CCNC(=O)CCc2cc(OC)no2)CC)OC)CCC(F)(F)CC1 N1(C(CN2CC(CC)C2)=O)CCCCCCC1C(=O)NC(C)CC1(O)CCC1 CN1CCCC1CCC(N1CC(C(C)(C)O)(CNC(C2CNC(=O)N2)=O)C1)=O C(=O)(C(CC(F)F)N(C)C(c1cn(C)nc1OC)=O)NC1C(C=C)OCC1 CCC(CC(F)(F)F)NC(c1ccccc1-c1ncnn1C)=O N1(C(c2c(OC)n[nH]c2)=O)CC2CN(C(C34CCC(CC3)C(C)O4)=O)CC2C1 N1(C(C=NOC)=O)CCN(CCN(C)C(C2CCS(=O)(=O)N2)=O)CC1 c1(NC(=O)COc2ccc(C34CC(CC)(C3)C4)cc2)cc(OC)cc(OC)c1.CS C=CC(CC)C(=O)NCC=CC(N1CCC(C(N)=O)C1)=O N1(C(CC2N(C(CC(C)n3ccnc3)=O)CC2)=O)CCC(F)(F)C(C)C1 N1(C(c2c(CCC)[nH]cc2)=O)CCCC(C2CC2NC(C2CCCS2)=O)C1 C1(NC(c2c(OC)scc2)=O)CC(NC(C2CCSCC2)=O)C12CCOCC2 c1(C(=O)NC2CC3CCC(C2)N3C(=O)CCOC2CC2)ccc(F)c2occc12 CC1(C)C(C(=O)NCC2CCC(NC(c3cnn4ccsc34)=O)C2)CCS1(=O)=O C1(F)(C(N2CC(CNC(C3(S(C)(=O)=O)CC3)=O)C2)=O)C2CCCCC12 c1(C(=O)NCC2C(NC(CCCOCCC)=O)C2)ccnc(NC(C)(C)C)c1 CN1CC(O)CCC1C(N1CC(C(=O)N(CC(F)F)C2CC2)C(C)(C)C1)=O c1(C(=O)NCCN(C(c2cc(CCC)on2)=O)CC)nnc(O)c2ccccc12 Cc1c(C(=O)N(c2cccc(Br)c2)Cc2ccccc2)cccc1O c1(C(N2C(CCCNC(c3c(C)csc3)=O)CCC2)=O)ccc2sc(C)nc2c1 c1(N2CCC(N(C)CC)C2)nc(=N)[nH]c(=NCC(C)(CC)c2ccncc2)[nH]1 C1(NC(c2c(C)ccc(C)c2)=O)CC2(CCC(NC(=O)C(O)C3CCC3)CC2)C1 C(=O)(CC1CCc2ccccc21)NCC1(COC)CN(C(=O)C(C)(C)SC)C1 c1(C(C(C)NCC(=O)Nc2ccc(COC)cc2)O)ccc(C)c(C)c1 Cc1nn(CCF)cc1NC(=O)C(C)(C1CC1)N(C)C(C1CC1(C)C)=O N1(C(C(CCOC)N(C)C)=O)CC(CC(=O)NC2CC3CCCC3C2)C2(CC2)C1 C1(C(=O)NC(C)(C)CCCNC(c2ncccc2O)=O)CCc2ncsc2C1 C1(C2CCOCC2)(C(N2CCC(N(C(=O)C3=CCCS3)CCC)C2)=O)CC1 N1(C(c2nc(COCC)sc2)=O)CCC(O)(CN)C1.C1(=O)CN1.C(C)C c1(CN(C(C(=O)NC2C(C)CC2)=O)C)ccc(Br)cc1 c1(CNC(=O)C(=O)N(C(c2ccc(N(C(C)=O)C)cc2)C)C)cc2c(s1)CCC2 c1(C(N2CC(NC(C3(C)CCNC3=O)=O)(CO)C2)=O)nc2ccccn2n1 C1(C(N2C(C(C)C)C(C)(C)C2)=O)CCCCCN1C(=O)C(C(C)O)N(C)C N1(C(c2cnc(OCC)s2)=O)CCN(C(=O)C(c2cncn2C)O)CC1C(F)F C1(CNC(CCCNC(C)=O)=O)COCCN(C(=O)C2=CCOCC2)C1 N1(C(C2(N(C)C)CC2)=O)CCC(NC(c2cc(=O)cc(Cl)[nH]2)=O)C(CO)C1 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)C(C3CC3)SC)C(C)C2)=O)o1)NC CC1Oc2ccc(CNC(=O)CCN3CCCC3=O)cc2NC1=O c1(NC(CCC2CCN(C(C(C)(C)C3CCC3)=O)C2)=O)cccc(N=[N+]=[N-])c1 N1(C(C2C(c3n(C)ncc3)OCC2)=O)CCCC(Cn2cccn2)C1 Cn1cc(NC(=O)C(Cc2cn[nH]c2)NC(=O)C(C#N)C(C)(C)C)c(O)nc1=O c1(C(=O)NCC2C(C)CCN2C(C2COC(C)(C)O2)=O)ccc2nn[nH]c2c1 C1(NC(c2n[nH]c(C)c2Br)=O)CCN(C(C2OCCO2)=O)CC1C C1(C(=O)NC(C)CF)(CNC(=O)Cn2cc(Cl)cn2)CC12CCC2 N1(CCC)C(=S)NC(c2ccccc2I)C(C(=O)OC(C)(C)C)=C1C1CCNC1 N1(Cc2cccc(C(C)C)c2)C(=O)CN(CC23CC(C2)C(C)O3)C1=O Cc1ccncc1C=CC(=O)NCC1(C)CN(C(c2cn(C)nn2)=O)CCO1 C(CC)(CCCC(=O)NCCCC1CCCCO1)NC(c1cnc(CC)s1)=O N1(c2nnc(CCC)s2)CC2CCCN(C(c3nc(C4CC4)cs3)=O)C2C1 c1(CC)csc(C(F)(F)C(=O)NC(C)CCNC(=O)CCn2ccnc2)n1 C1(COC)(CNC(=O)C(N2CCSCC2)C)CN(C(C2(F)CCC2)=O)C1 c1(NC(c2cccc(Br)c2O)c2n(CC)nnn2)cccn2ncnc12 Cc1cccn(CC(=O)NC(C)C(C)NC(=O)C=Cc2ccc(C(N)=O)o2)c1=O n1(CCC)c(CN2CC(C(C)NC(C3COC(=O)O3)=O)C2)nnc1C c1(OC)cc(Br)cc(CN2CCC(NC(c3cc(B(O)O)co3)=O)C(F)C2)c1O C1(C)(CNC(C(C)(C)NC(C)=O)=O)CN(C(C2CCCN2c2nccs2)=O)CCO1 CC1CN(C(=O)Cc2cccc(F)c2)CCC1NC(=O)CC1CC(=O)NC(=O)C1 CC(C)(F)C(C)(F)CNC(=O)CCc1nnc(-c2cccs2)n1-c1ccccc1 C1(OC)CCCC(CC(=O)NCCn2cc(NC3CC3CC(C)(C)C)nn2)C1 c1(OC)cncnc1C(=O)N(C1CC(NC(=O)CCc2nncs2)C1)C C(=O)(C(C)CS(C)(=O)=O)NCCc1c(CNC(CC(C)O)=O)nco1 C1(C#N)(C(=O)NC(CCOC)CNC(=O)CSCc2ccccc2)CCCCC1 N1(C(CC2C(CC)C2)=O)CCCC(N(C(c2ccnn2C2CC2(F)F)=O)CC)C1 C1(NC(c2c(NC)nccc2)=O)CC(O)CN(C(=O)C(C)(C)c2ccnn2C)C1 c1(CC)cnccc1CNC(=O)C(CCF)NC(=O)C(CC)N(C)C N1(C(c2c(CC)cc[nH]2)=O)CC2COCC2(C(=O)NCC(C)(F)C(C)(C)F)C1 Cc1ncc(F)c(N2CC(C(=O)Nc3cnn(C4CCOCC4)c3C)C2)n1 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(NC(c2c(C)cc(N)c(C)n2)=O)C(C)C1 N#Cc1ccc2cc(CNc3nc(C(N4CCCC(F)C4)=O)cs3)[nH]c2c1 CCC1(C)CN1C.c1(C(=O)NC2CCCC2)cn(C)nn1 c1(OCC(=O)NCC(CC=C)NC(C2(CF)CCC2)=O)ccccc1[N+](=O)[O-] c1(C(N(C(C)CN(C(=O)Cc2cccc(O)c2)C)C)=O)cnc2ccnn2c1 C(=O)(C1COc2ccc(F)cc21)NC(=O)NC(C(C)(C)C)CCN1CCOCC1 N1(C(CCn2ccc(C)n2)=O)CCC2C(CCN2C(c2csc(C#N)c2)=O)C1 Cc1[nH]nc2c1CCC(C(=O)NCC1(F)CCC(CNC(C3CCC3)=O)CC1)C2 C(=O)(C(C)C(=O)N1CCC(N(C(c2cccnc2S)=O)CC2CC2)C1)OC CCC(C(=O)NCC1(C(N2CC3(CCC3O)C2)=O)CCCC1)C(C)(C)CC C1(C2CC2)(NC(C2OCCN(C)C2)=O)CCN(C(C2(CO)COC2)=O)C1 N1(C(c2c(CC)cno2)=O)CCCC(CC2CCN(C(=O)C3=CCCC3)CC2)C1 CCC(CC)CC(c1nnnn1C1CCC1)NC1COC(CC)C1 CCC(CC(=O)N1CCN(C(=O)C=CCn2cncn2)C(C(C)C)C1)CC(C)C C(C(=O)NCCOCCC(=O)NCC1(C)CC(C)=NO1)(C(C)C)SC c1(OCC(=O)NCC2(NC(C(C)N(C(C)=O)C)=O)CCOC2)cc(F)cc(Cl)c1 c1(C(N2CC(C)C(NC(=O)Cc3ccc(O)c(O)c3)C2)=O)cc(O)c(O)c(O)c1 CCCC(C(=O)NC(C1CCCC1)CNC(=O)C(F)(F)C(O)CC)S(N)(=O)=O c1(OC)ncc(C(=O)NC(CO)C(C)NC(=O)C(c2cccc(Cl)c2)C)cn1 c1(CC(=O)NCCCNC(C(C)N(C)C2CC2)=O)ccc(C(=O)OC(C)(C)C)cc1 C#CCC(O)C(=O)NC(CC1CCOCC1)C(=O)N(CCC1CC1)CC1CC1 N1(C(C=C(CC)CC)=O)CCC2(NC(=O)Cn3cccn3)CCCCCC12 C1(C(=O)NCC2CN(C(=O)CN(c3ccccc3)C)C2)(OC)CCSCC1 CCCCCCCC(=O)N1CCC(NC(=O)Cn2nc(C)oc2=O)C1CC N(C(=NCCNS(=O)(=O)C(F)F)N1CCC2(CC2)C1)C(C=C)C C1CC(S)CCO1.C(CN(C)CCN(C)C)OC N1(C(CSC)=O)CCC2(CCCCC2NC(C2CCNC2=O)=O)C1 C1(CNC(C2C(C)OCCO2)=O)CCN(C(=O)C2=CCCC2)CC1c1ccccc1 c1(C(C(=O)N2CC(CCCCNC(C(C)OC)=O)C2)(C)F)ccc(F)cc1 C1(C(N2C(CCNC(C3(C)CC=CC3)=O)CCC2)=O)CCn2nccc2C1 N1(C(c2c(CCC)nco2)=O)CCCC12CCN(C(c1cnc(C)nc1C)=O)C2 C1(NC(C2OCC3COCCC23)=O)CCC2CCN(C(c3sccc3F)=O)C1C2 c1(C(=O)OC2CN(C(=O)OC(C)(C)C)CC(F)C2)cnc2cc(Cl)ccn12 Cc1sc(S(N)(=O)=O)cc1C(N1CC(NC(c2cn(C)[nH]c2=N)=O)CC1C)=O C(=O)(CCCCCC(=O)OC)NCC1CCN(CCCNC(C(C=C)O)=O)C1 CCN=c1[nH]cc(C(=O)NCCN2CCN(C(C3(C4CC4)CC3)=O)CC2)s1 C(=O)(CCC(C)(C)NC(c1csc(CO)n1)=O)N1CCC(C)(N(C)C)C1 c1(CSCC(=O)NCC(C)NC(COC2(C#C)COC2)=O)c(C)noc1C c1(-c2ccc(C(c3n(CCSC)nnn3)NCc3snnc3C)o2)ccccc1Cl C(C(C)N=c1nc(C#N)[nH]cc1C)N(C(C1(O)CCC(C)CC1)=O)C c1(CN(C)Cc2ccc(Br)cc2)c(Cl)ccc([N+](=O)[O-])c1Cl.C12CN(C1)C2=O Cc1cc(C(=O)Nc2nccn2Cc2ccc(Br)s2)nc(C)n1 C1(C(N2C(C)C(NC(=O)C=C3CCN(C)CC3)CCC2)=O)Cc2cccnc2C1 c1(C(N2C(C)(CNC(C(CCC)C#N)=O)CCC2)=O)cc(Cl)c(C)cc1OC c1(CNC(C2N(C(Cc3nc(C)on3)=O)C3C(C2)C3)=O)n[nH]c2ccccc12 C1(CC=C)(NC(c2ccc(Cl)o2)=O)CC2CCC(C1)N2C(c1cc[nH]c1CC)=O C(N=C(NC(C)CC(C)C)N1CCOC(c2ccc(Cl)s2)C1)c1ccc(C)cn1 C=CCCC(C)NC(=O)C(CO)NC(=O)CC1CC1 N1(C(C(CC=C)(F)F)=O)CC2(C1)SCCC2NC(=O)CN(C(=O)COC)C c1(OC)oc(C)nc1C(N1CCC(NC(=O)C(c2c(C)noc2C)(C)C)C1)=O C(CCCC(=O)N1CCC(N(C)CCN2CCOC2=O)C1)N(C)C(N)=O c1(OC)ccnc(C(N2CCN(C(c3cccnc3F)=O)CC2)=O)c1OC C12(C(=O)NC3CN(C(C4CC=CCC4)=O)C3)CCCN1S(=O)(=O)CC2 N1(C(CC)C(=O)O)CCOc2ccccc21.N12CCC3CC(C3C1)C2=O c1(CNC(c2n(CCCSCC)nnn2)C2CCC2)cccc(C)c1 Cn1c(C(N2CCC(C(=O)NCCS(C)(=N)=O)C2)=O)cccc1=O N1(C(C2CC(C#N)C2)=O)CCCC(NC(C2CC2c2ccccc2Cl)=O)C1 C1(NC(=O)CC2(CO)CC2)CCCC12CN(C(=O)CCCn1ccnn1)C2 C(CC(C)(C)CC(=O)NC(CNC(c1cccc(OC)c1)=O)CC(F)(F)F)OC c1(OCC(C)C)ncc(C(=O)NC2(C)CC(NC(C3(F)CCOC3)=O)C2)cc1Cl C(=O)(C(F)CCC(C)(C)C)NCC1(C(N2CC(F)(F)CC2C)=O)CC(=C)C1 CCC(C)CCCC(=O)N1CC(NC(=O)Cc2cncnc2)CC1(C)C Cn1cc(C2C(NC(=O)OC(C)(C)C)CC2O)cn1.c12nc(cs1)CCOC(=O)N2 N(C(=NCC1CC12CC2)N1CC2CN(S(=O)(=O)c3ccccc3)CC2C1)C(C)C c1(C(=O)NC(CC=C)CNC(=O)CC(C)C(=O)OC)noc2cc(Br)ccc12 C1(C(=O)NC2CC(CCNC(c3ccc(C4CC4)nc3)=O)C2)CC12CCCCC2 c1(C(N2CCC(OCCNC(CC(CCC)C)=O)C2)=O)c([N+](=O)[O-])cnn1C N1(C(c2c(OC)ccs2)=O)CC2CC2(NC(c2ccccc2N(C)C)=O)C1 CC(CCN=c1nc(Oc2ccccc2)cc[nH]1)NC(=O)CC(C)(C)C(F)F C1(C(N2CCC(O)(CCNC(C(=O)NCC)=O)C2)=O)CCCCC12CC2 N1(C(CC(C)SC)=O)CCC(NC(=O)C(c2ccccc2)NC2CCCC2)CC1 c1(OC)ccc(Br)cc1CC(N1CCOCC(NC(c2ncoc2C)=O)C1)=O Cc1nc(C2CC2)ncc1CC.c1(C(c2nnnn2C2CC2)N)cc(Cl)ccc1Br C1(C)(C(=O)NCC(CNC(C2(C(=O)OC)C(=C)CC2)=O)C)Cc2ccccc2C1 n1(CC(N2CC(C(C)NC(c3c(C)c[nH]c3)=O)C2)=O)c(=O)oc2ccccc12 N1(C(COc2c(CC)cccc2)=O)CCC2(CCN(C(=O)C(C)C(C)CC)C2)C1 C1(C(=O)NC2CCOC2(C)C)(CC)CCCN1C(C1CCCN1C(C)C)=O c1(OC)ccc(C(=O)NCC2CCCN2Cc2cncc(OC)c2C)cc1C c1(C(=O)NC(CCOC)CNC(C2CCC(=O)N2)=O)oc(Br)cc1C CCCCC(CC)CC(=O)NCC(C)(CO)NC(=O)Cc1cn(C)nc1C C(C(F)(F)C(=O)NC1CCN(C2CCN(C(=O)COCCSC)CC2)CC1)OC C(C(=O)Nn1nnc2c1CCCC2)C1N(C(c2c(OC)scc2)=O)CCOC1 c1(N2C3CN(C(C(C)NC(C)=O)=O)C(C3)C2)nc(C(C)C)cc(C)n1 CC(C(=O)NC(C)C(CO)NC(=O)Cc1ccc(C(F)F)cc1)C(F)F c1(CC(=O)NC(C2CN(c3nccc(C#N)n3)C2)C)cccc2ccccc12 c1(C(=O)NC2CC(CNC(CCCSCC=C)=O)C2)cc(C)sc1-n1cccc1 N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CCOCC(NC(C2CC3CC2C3)=O)C1 C(=O)(C(CO)NC(c1sccc1F)=O)N(CCCn1ccnc1)C c1(C(C)=O)ccc(C(=O)NCC2(CNC(c3cc(C)ccc3F)=O)CC2)cc1F C12(NC(CCCCOc3cccc(C)c3)=O)CC(c3ccccc3)(C1)C2(F)Cl Cc1cn2nc(NC(=O)CCSc3ccccc3Cl)sc2n1 C(CCN(C)C(C1(CO)CC(C)(C)C1)=O)(C(C)C)NC(C(C)SCC)=O C=CC(C)(CCOC)C(=O)N(C(CNC(c1cnn2ccn(C)c12)=O)C1CC1)C C1(C(N2CCC(CNC(C(c3cnccn3)C)=O)C2)=O)CC12CCCC2 N1(C(c2c(C)[nH]c(=NCC)s2)=O)CC2CCC(CCN)CC2C1 C1(NC(=O)COCC(F)F)CC2(CCN(C(=O)C(CC(F)F)C3CCC3)CC2)C1 C(c1cncc(C)c1)=CC(=O)NC1C(CC)N(C(C2CC(C)C2)=O)CC1 C=C1CC2(C1)CC(C(N1CCC(C(C)NC(=O)C(C)(C)OCC)C1)=O)C2 C(=O)(C1CCOc2ccc(F)cc21)N1CCC(C)C1C CC1CC(C(=O)NCC2(NC(C3CC(O)C3)=O)CCCCC2)CC(=O)N1 c1(C(N2C(CNC(C(CCCC)C)=O)C(C)CC2)=O)cc2c(F)ccc(F)c2s1 CC(C)S(=O)c1ccc(C(=O)NCC2CCC2NC(C2CCC(C)CC2)=O)cc1 N1(C(c2ccn(C3CC3(F)F)n2)C(=O)NCCCCCC)Cc2cncnc2C1 N1(CC2(O)CCN(C(Cc3ccc(CCCCC)cc3)=O)C2)CCC(O)C(F)C1 C1(C(N(CC(CNC(C(C=CC)O)=O)(C)C)C)=O)CC2(CCC2OC)C1 C12CCCCC1C(=O)N1CC(C1)O2.c1(CNC(CCOC)=O)cnccn1 N1(CCc2nnc(-c3ccc(OC)c(Br)c3)o2)CCCc2ccccc21 Cc1cc(C(=O)NC2CCC2NC(=O)CCC(N)=O)cc(S(N)(=O)=O)c1C C1(NC(CCOCCN(C(=O)C2=NNC(=O)C2)C)=O)CC(CO)C12CCC2 c1(C(=O)NCC=C2CCN(C(C3CC(C)(C)C3)=O)CC2)nc(O)nc(O)c1F N1(C(C(c2ccc(CC)cc2)C)=O)CC2CCC(C1)N2c1nc(Cl)ncc1F CCC(CCC(=O)N1CC(c2ccccc2)(NC(=O)CCCC(C)C)C1)OC C(=O)(CC(C)C(C)(C)NC(=O)C(C1CCC1)OC)NCC1N(C(C)=O)CCC1 N1(CCC)C(=O)CCC1C(=O)NC(CNC(=O)Cc1cn(CC)nn1)C(C)(C)C C1(N(C(=O)C(C)=CC2CC2)CC)CCN(C(c2sccc2OC)=O)C1 CC(C)(N=[N+]=[N-])C(=O)N1CCC1C(=O)NCC1Cc2nccn2C1 C1(CNC(C(=O)N(C)C)=O)CN(C(c2ccc(C#N)cn2)=O)CCC1C(F)(F)F N1(CC(=O)NCC)CCCN(CCC2(C(F)(F)F)CCNC2)CC1=O C1(CS(C)(=O)=O)COCCN1C(c1ncc(C(F)F)s1)=O N1(C(C=Cc2ccc(=N)[nH]c2)=O)CC2(CCN(C(C3(CF)CC3)=O)C2)C1 c1(N2CC(CC)N(Cc3cccc(OC)c3)CC2)ncnc2scc(C)c12 N1(C(=O)C(c2ccn(C)c2)C)CC2OCCN(C)C2C1.C(C=O)NC(C)C C(C(CC(C)C)C(=O)NC(C)Cc1cccs1)NC(C(n1c(C)ncc1)C)=O N1(Cc2onc(CC(=O)NCCOC)n2)CCCC(CNc2ccccc2C)C1 N1(C(C(C)C)=O)CC2CC1C2C(=O)Nc1cn(C)nc1C(F)(F)F Cc1cc(C(=O)NCC2CCCC(NC(=O)Cc3ccsn3)C2)cnn1 C1(CNC(CNC(CC)=O)=O)C(C)CCN1C(c1csc(C)n1)=O N1(C(C(C)Oc2ccccc2O)=O)CCC2C(CCN2C(c2cncs2)=O)C1 C1(O)(CN(C(C(CC)=CC)=O)C)CCCN(C(=O)CC2SC(=N)NC2=O)C1 C(=O)(C(F)C(C)CNC(C12CC(CO)(C1)C2)=O)N(C)Cc1c(C)ncs1 C(CC1=CCN(C(=O)CCCC(=O)OC(C)(C)C)CC1)NC(C(C)NS(C)(=O)=O)=O Cc1[nH]nc(C(=O)NCCCN(C)C(C2COCC2(C)C)=O)c1[N+](=O)[O-] N12CC(CC1=O)C(=O)NCC(C)(C)OCC(=O)N1CC2C1.C1(CF)CC2CCC1O2 N1(C(C(C)SCCCC)=O)C2CCC(C2)C1CNC(c1cc(C)n(C)c1C)=O c1(C(=O)NCCCN(C(CCCC(C)C)=O)CCO)ccc2c(c1)COC(=O)N2 C1(NC(C(c2c(C)cccc2)(C)C)=O)CC2CCC(C1)N2CC1CCCOC1 C1(C)(CNC(c2cc(CNC(CC=CCC)=O)no2)=O)NC(=O)NC1=O N1(C(CCc2scc(C)n2)=O)CCOCC(NC(C2(F)CCOC2)=O)C1 c1(-c2ccc(OCOC)cc2)ccc2[nH]c(C(=O)NC3(C)CCCCC3)nc2c1 N1(C(C2(C#C)CCC2)=O)CC2CCN(C(c3nc(Br)c[nH]3)=O)CC2C1 N1(C(Cn2cnc(=N)[nH]2)=O)CCC(O)C(NC(C2CCNC2=O)=O)C1 C(=O)(CCC(CF)CF)OCC(=O)O.Cc1ccc2cc1NC(=O)C(=O)N2 O=C(CS(=O)(=O)C1CC1)N1CC(CNC(C2(Cl)CC2(F)F)=O)C(F)(CO)C1 C1(C(=O)NC2CC(C)N(Cc3cccc(F)c3Cl)CC2)CCC2CCCCN12 C(=O)(C1=CCCSC1)N(C1CN(C(C2CC(=O)C23CCC3)=O)CC1(C)C)C C1(C(=O)NC2CC3(CN(C(C(F)=C(C)C)=O)C3)C2)C2Cc3cc(Cl)ccc3C12 CC(C)CCC(O)C(=O)N1CCCC(O)(CN(C(=O)CCc2ccccc2)C)C1 O(NC(=O)CCCC(C)NC(c1c(C)cccc1O)=O)CC(=O)OCC c1(C(=O)NCC(CC)(CC)NC(C(F)=CC)=O)cc(Cl)cc([N+](=O)[O-])c1O c1(C(=O)NCC(C)NC(Cc2ccc(CCC)cc2)=O)ncc(C)cc1F N1(C(C2C(C(C)(C)C)OCCC2)=O)CC2(CCCN(C(C3CCC3)=O)C2)C1 c1(CNC(C2(CSC)CC2)=O)cn(C2CCN(C(=O)CC3CC3)C2)nn1.C1CCC1O c1(CC)c(C(=O)NC(C)CNC(C2(C)CCCCO2)=O)cccc1F CC1(NC(c2ccnn2C(C)(C)C)=O)CCN(c2ncc(Br)cn2)C1 c1(CC(=O)NCC2(CC(=O)N(C3CCCC3O)C3CC3)CC2)ccccn1 C=CCC(C(=O)N1CCC(CF)(NC(c2nncn2C)=O)C1)NC(C)=O O=C(CC1=NNC(=O)C1)NCCC1CC(NC(=O)CC2CCCOCC2)C1 N1(CC(N2CCN(C(c3n(C)c(S)nn3)=O)C3C2C3)=O)C(=O)NC(C)(C)C1=O c1(C(N(C)CC2OCCN(C(Cc3cc(C)nn3C)=O)C2)=O)cccc(C)c1C C(=O)(C(CC(C)C)n1ccnc1)OCc1scc(C(=O)OC)n1 c1(C(=O)NC2CCN(C(c3c(CC)con3)=O)C2C(C)C)cnc2nccn2c1 N1(C(C2(CNC(C3COCC(C)O3)=O)CC(=C)C2)=O)CCN(C)CC(C)C1 CC1(C)C(NC(=O)COc2ccc(Br)cc2F)C2CCOC12 N1(C(C(C)OC)=O)CCC(C2(NC(=O)CNC(c3ccc(C)s3)=O)CC2)C1 N1(C(CCC(C)OC)=O)CCC(CNC(c2ccc(C(N)=O)o2)=O)C1(C)C CCCC(C(=O)OC)C(=O)NCC1CC(C)(C)CN1C(C12CCC(C1)C2)=O c1(CC)cscc1C(=O)NC1CC(C)(NC(=O)C(C)OCC2CCCCO2)C1 CC1CC(NC(c2cccnn2)=O)CN1C(=O)CCCc1ccncc1 N1(C(C(COCC)NC(c2ccc(Cl)o2)=O)=O)CCOC(CF)C1 C=CC(C)(C)CCN=c1nc(N2C3C=CCC2CCC3)c2c(F)cccc2[nH]1 c1(C(N2CCC(CN(C(CC(C)c3ccco3)=O)C)C2)=O)cnn(C)c1F N1(C(CCC2CN(C(C3N(C(C)=O)CCC3)=O)C2)=O)CC(C)NC(=O)C12CC2 Cc1cccc(C)c1-n1cc(C2CC2CN2CCCC2c2ccc(F)cc2)nn1 CCCCCC(O)CC(=O)N1CC(n2cc(Cn3cncn3)nn2)(C(=O)OC)C1 C(C(C(=O)NC1CCCC1SC)C(C)(C)C)NC(c1cc(OCC)n[nH]1)=O N#Cc1ccc(NC(C2CCN(C(c3ccc(C(N)=O)cc3)=O)C2)=O)s1 N1(C(C2N(C)CC(O)C2)=O)CCN(C(C2CC2c2ccccc2)=O)C(CO)C1 c1(OC)cccc(C(C)N(c2cccc(C)c2)C(c2ccco2)=O)c1 CC1COCCC1N(C)C(C1CCN(C(c2cc(N(C)C)ccn2)=O)C1)=O c1(C(N2CCN(CCF)CC2)=O)cc2c(s1)CCN(Cc1c(F)cncc1F)C2 N1(C(C(C)(C)OC)=O)CCN(C(=O)C(C)(C)C(N)=O)CC12CCC2 C1(C2CCCN(C(c3ccc(Cl)[nH]3)=O)C2)(NC(CCC=C(C)C)=O)CC1 C(=O)(C1CCc2ccccc21)NC(CN(C(=O)CSc1nc(C)no1)CC)C N1(C(=O)C=CBr)CC2CCCC(NC(C34CCCCC3OCC4)=O)C2C1 Cc1cc(CNC(C2CN(C(=O)CCCC3CCC3)CC2C)=O)ccn1 c1(C(=O)NC(CC(C)NC(c2cc(O)ncn2)=O)C)ncc(Br)cc1Cl C(=O)(C1COc2ccc(Cl)cc21)NC1(CNC(CC2OCC(C)(C)OC2)=O)CC1 C(=O)(CC(C)C(C)C(C)C)N1CCC(C)(NC(C2(OCC)CCCC2)=O)C1 C(=O)(CC1COc2cc(OC)ccc21)N(C1CCCN(C(C=COCC)=O)C1)C C(CC(O)CC(=O)NC1CCCC1NC(C1(C)CCOC1)=O)SC c1(CNC(C2(C(C)C)N(C(C3C(OCC)C3C)=O)CCC2)=O)ccc(C)cc1O c1(C(=O)NC(CNC(c2nc(C)nn2C)=O)C)cn2ccn(C)c(=O)c2n1 C(=O)(C1COc2ccc(Cl)cc21)NCC1(NC(=O)CCc2cccnc2F)CC1 N1(CCCCNC(C=CCOC)=O)CCCN(C(=O)CC(C)(C)OC)CC1 C1(C(N2CCC(C(C(=O)N(C3(C)CC3)C)F)C2)=O)CC(=O)NC(=O)C1 c1(C(N(CC(CC)NC(C2CSCCS2)=O)C)=O)ncoc1-c1cc(C)no1 c1(CN(C(=O)C(N)Cc2ccco2)C)nc(C(F)(F)F)no1 N1(C(C=COCC)=O)CCC2OCCN(C(c3cccc(N)c3)=O)C2C1 N1(C(c2cc(OC)ns2)=O)CCN(C(C23COCC2C3)=O)CC1C Cc1cncc(C(N2CCC(O)(CNC(C3CCC3C(F)(F)F)=O)C2)=O)n1 C1(CC)C(NC(=O)C(C)N(CC)CC)CCN1C(C1CCC(=O)N1)=O c1(C(N2CCC(NC(=O)C=Cc3cn[nH]c3)C23CC3)=O)cc2cccc(Cl)c2s1 C(=O)(C1=CCC(C)(C)CC1)NC1C(CNC(C(C)C(C)(C)C)=O)CC1 C1(NC(C2C(C)CN(C(C3COC(=O)N3C)=O)CC2)=O)CCn2ncnc2C1 C1(N(C)C(c2cc(CNC(C3CCCC3O)=O)[nH]n2)=O)CCSCC1 c1(C(=O)NC(CNC(CCNC(C)=O)=O)C(C)(C)C)cc(Cl)ccc1C C#CCC(CC#C)C(=O)NCC1CCC(NC(=O)CC(=O)NCC2CC2)C1 C1(NC(c2cccc(C)c2)=O)CC2CC1CN2C(C1(c2cccc(C)c2)CC1)=O Cn1cc(C(=O)Nc2cccc(NC(=O)Cc3nc[nH]n3)c2)c(C2CCC2)n1 CC1CCC(C(c2nnnn2C)NCc2sccc2Br)CC1 C=C1CCC1(C(N1CCC1CNC(=O)Cc1cnn(C(C)(C)C)c1)=O)C(=O)OC C(=O)(CC(CN(C)CC)CC)N1C(CNC(CC2(C(=C)F)CCC2)=O)CC1 C(CC(O)C(F)(F)F)NC(C1(OC)CCN(C(c2cc(SC)oc2)=O)C1)=O C(CNC(c1oncc1C)=O)(CC(C)C)NC(C(C)SCCCC)=O N#Cc1ccc(NCC2(c3ccc(Br)o3)CC2)nc1 C12(CNC(CC=CC)=O)COCCN1C(=O)CN(C(=O)CCCCCCC#N)C2 c1(SCC2N(C(C(C)C)CN3CC4CC4(CO)C3)CCC2)ccc(F)nc1F C=CC(C)(CCOC)C(=O)NCCc1ocnc1CNC(c1ccn(CC)n1)=O CC(C)(C(=O)NCC1(C)CCN(C(=O)C(F)(F)C(F)F)C1)C1=CCSCC1 c1(NC(C2(C)CCN(Cc3c(C)cccc3)C2)=O)cc(F)c(Cl)nc1Cl S(=O)(=O)(C1CCN(C(=O)CC2(C(=O)N(C)C)CCCC2)CC1)N(C)C C(CCC(C)(C)NC(=O)CN1CCSCC1)NC(CCCOCCC)=O c1(C(NOCCCC(=C)C)=O)cccc(Oc2ccccc2C)c1 C(C(CNC(=O)COc1ccc(Cl)cn1)C(F)(F)F)NC(C(CC)OCC)=O Cc1n[nH]c(=NCC2(CNC(c3cc(C4CC4)[nH]n3)=O)CC2)s1.C1CC1 C=CCN=C(NCCc1cccc(C#N)c1)NCCC1CCS(=O)(=O)C1 c1(C(=O)NC(CCOC)CNC(=O)C(C)(C)C)ccc2c(c1)NC(=O)C(C)S2 CCC(C(=O)NCCOCCCNC(c1ccc(-c2ccco2)o1)=O)OC c1(CC(C)C(=O)N2CCC(N(CCO)C(c3n[nH]cc3Br)=O)C2)ccccc1F CC(CC(F)F)C(=O)N1CCCC1C(C)NC(=O)COCc1ccncc1 N1(C(Cn2ccc(C(=O)OC)n2)=O)CC(NC(=O)CSc2cccs2)C(C)C1 c1(NC(=O)NC(C2CCCCC2)CN2CCN(C)CC2)cnc(Br)cc1O N1(C(C(=CC2CCCC2)C)=O)CC2CC2(NC(=O)Cc2ccc(Cl)cn2)C1 Cc1[nH]c(=N)ccc1C=CC(=O)NC1CN(C(C2(Cl)CC2)=O)CC1(C)C C1(C2CC2)(NC(c2coc(C3CC3)n2)=O)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 c1(C(=O)NC(CNC(c2cc(C)no2)=O)C(C)C)cccn(C)c1=O C(=O)(C(C(C)(C)C)c1ccccc1)N1CC(F)(CN(C)C(c2ccc(Cl)s2)=O)C1 C1(CNCc2cc(CCOC)on2)OC(=O)CC12CCC2 C1(NC(c2cnsn2)=O)CCCCN(C(C2C3(CC3)C23CC3)=O)CC1 C1(CNC(CSCC(=O)OC)=O)CCC(NC(=O)C(c2cccc(F)c2)O)CC1 c1(OCC(=O)N(CCCNC(c2cnc(Cl)s2)=O)C)ccccc1C(C)(C)C O=C(NNc1ncnc2sccc12)c1coc2c(F)cccc12 C1(C(=O)N(CC(O)CNC(=O)COc2ccsc2)C)(CC)CCCCC1 Cc1c(Cl)nc[nH]c1=NCC1(O)CCCN(C(C2CCCN(S(C)(=O)=O)C2)=O)C1 c1(C(N2CC(CCCNC(=O)CN3CC4CC4C3)OCC2)=O)nccc(Cl)c1O c1(OC(C(=O)NCC(CC)(C)NC(=O)CC2(C)CC2)C)ccccc1Br c1(CNC2(c3cn(C)nc3)CC2)ccnc(P(C)(C)=O)c1 N1(C(=O)CC2=CCCC2)CCC2CCCN(C(c3ccc(CO)cc3F)=O)C2C1 C1(OC)(CNC(c2ccc(C(F)F)o2)=O)CCN(C(=O)C2CC2)C1 c1(OC)ccc(F)cc1CC(=O)NC1(C)CCCN(C(c2cc(Cl)sc2Cl)=O)C1 N1(C(C(=O)CC2CCCCC2)=O)CCCC12CCN(C(C1CC=CCO1)=O)C2 C1(C(=O)NCc2c(C(=O)NC3CC(C(C)(C)C)C3)[nH]cc2)C(C)(C)C1(C)C n1(CC(=O)NC2C(C)CN(CCC(C)(C)O)CC2)ccc2ccccc12 N1(C(CC(C)C)=O)CCC(C2CC2)(CNC(C2CC3(C2)CC(F)(F)C3)=O)C1 c1(C(N2C(C)C(NC(c3csc(C4CC4)n3)=O)CC2)=O)cnc2ncccc2c1 C1(CC(=O)NCCC(N2C(CC(C)C)COC2)=O)CCN(C)CC1 C1(C(F)F)(CN(Cc2scc(Br)c2Br)CC2CC2)CCCCO1 c1(C(N2CCC(NC(C34CCCN3CCC4)=O)C(O)C2)=O)cncc2sccc12 C#CCC(C)(C)C(=O)NCC1(F)CCC(NC(c2cc(C3CCC3)on2)=O)C1 c1(C(=O)NCCCN(C(=O)C(O)CC2CC2)CC)cn(C)c(C)cc1=O N1(C(C(C)=C2CCC2)=O)CCC2(C1)CN(C(=O)C(C)c1ccon1)C2 C(S(=O)(=O)c1ccccc1)c1c(CN(C(=S)NC(C)C)CCCOC)cccc1 CCCC(C)(CCC)C(=O)NCC1(F)CCN(C(C2(C)CCOC2)=O)C1 C(=O)(C(CC)CCCCCC)N1CCC(CC=C)(NC(C2CCCCC2)=O)C1 C#CCC(C)(C(=O)NC1COCC1N(C)C)NC(C1CC2(CC(=O)C2)C1)=O c1(C(=O)NC2C(C)CCN(C(C(CC)SC)=O)C2C)c(C)ccc([N+](=O)[O-])c1C N1(C(CN(CC(C)(C)C)C)=O)C2CCC(C2)C1C(N1CCOCC12CC2)=O C#CCCCCCC(=O)NC(CO)C(C)NC(C1CC(Cl)(Cl)C1)=O Cc1cc(-c2ccccc2NC(C2(O)CC2)C)ccc1OC(F)F C1(C(N(C(CNC(CS(CC)(=O)=O)=O)C)C)=O)CCc2nc(O)nc(O)c2C1 N1(C(C(CSC)(C)C)=O)CC2CS(=O)(=O)CC2(NC(c2cc(C)c[nH]2)=O)C1 CC(CC(C)(F)F)C(=O)NC1CCN(C(c2ccnc(-c3ccccc3)n2)=O)C1 C(c1ccc(O)cc1)=CC(N1C2(CNC(C3CC34CCOCC4)=O)CC(C1)C2)=O C(=O)(CC(C)C(F)(F)F)NCC1(C(=O)NCc2c(C)noc2CC)CC(=C)C1 C#Cc1ccc(CNC(C2CN(C(=O)C(C)CC=CCC)CCO2)=O)cc1 Cc1ccc(NC(=O)C2=CCN(C(C3C=CCC3)=O)C2)c(O)n1 CC1CC(NC(=O)NC(Cc2ccccc2Cl)CO)CC(C)S1(=O)=O C1(CC=C)(NC(=O)C(C)CF)CCN(C(c2cc(NC(C)=O)ccc2C)=O)CC1 CC1(NC(c2nncn2C2CC2)=O)CCCN(C(c2c(F)cccc2F)=O)C1 c1(C(=O)NCC2N(C(C(C(CC)C)OC)=O)CC3(CC3)C2)cnc2ccccc2c1 Cc1cc(C(N2CCN(C(c3nocc3C)=O)C(C3CC3)C2)=O)cc(O)c1 N1(C(CSCC=C)=O)C2CCC1CC(NC(c1cc(Cl)cnc1C)=O)C2 c1(OC)c(Cl)ccnc1NC(=O)NC(CC(=O)OC(C)(C)C)C1CC1 C1(N(C(C(CC#C)O)=O)C)CC2CCC(C1)N2C(=O)C(F)C(CC)CC CCCC(C(=O)NC1CCCC1NC(c1nc(C)oc1C)=O)NC(C)=O N1(C(CC2(C)CCOC2)=O)CCN(C(C2(N3CCCC3)CC2)=O)C2CCCCC12 Cc1ccc(C(=O)NCC(C)N(C)C(c2cc(-c3ccco3)c[nH]2)=O)s1 c1(CC(N2CC(C)C(NC(c3cncc(Br)c3)=O)C2)=O)ccc2nonc2c1 C1(CNc2ccc(OCC)cn2)CCCC(O)(c2nccn2C)C1 c1(CN2CC(C(=O)NC3CC3F)OCC2)cc2cnccc2[nH]1 N1(C(C(COC)N(C)C)=O)CCC2(CCN(C(c3nc(O)c(C)s3)=O)CC2)C1 C12(CNC(c3c(C)ccnn3)=O)CC(NC(=O)CC3CC3)(C1)C1(CCOCC1)O2 C1(CCOC)CCN(C(c2ccc(-c3ccc(F)cc3)cn2)=O)CC1 C1(CC(=O)NC2CN(C(C(c3ccccc3)OC)=O)C2)CC=CCC1 c1(Nc2cccc(OC)c2)cc(NC(=O)C(O)CC(C)C)c(F)cc1F Cc1ccc(OC(C)C(=O)NC2(CNC(c3scnc3C)=O)CCOC2)cc1 CC1CN(C(c2nc(Br)ccc2F)=O)CCCN1C(=O)C(C)S c1(OC)ccc(C(N2CCN(C(=O)C3=CCCOC3)CC2)=O)c(OC)c1Cl c1(C(N(c2ccc(N(S(C)(=O)=O)CCO)cc2)C)=O)ccc(Cl)cc1[N+](=O)[O-] CC1CN(C(=O)C=Cc2ccncn2)CCC1CNC(C1(O)CCOCC1)=O N1(C(CCSC)=O)CCC(NC(c2cc(Cl)c(C)cn2)=O)C(F)C1 O=C1CCC(C(=O)NCC=CCC(=O)NC2C3(CC3)C23CC3)CN1 CC1CN(C(c2cc(C3CC3)[nH]n2)=O)CC2(CCN(C(=O)CCS(N)(=O)=O)C2)O1 C1(CN2CC(CCO)(OC)C2)CCN(C(=O)CC(C)C(C)C)CCC1CO Cn1nc(C(N2C3CCC2CC(NC(=O)CN2CC=CC2)C3)=O)c2c1CCOC2 C1(CNC(CCCNC(CN2CCC(C)C2)=O)=O)CCC(F)(F)C1 c1(C(N2CC(CC=C)(C(=O)NCC3CCCS3)C2)=O)cnc[nH]c1=N c1(-n2ccc(NC(C3CC4OCCC34)=O)n2)cc(F)ccc1F.CC12CCCN1C2 C1(C)(NC(C(CC#C)(C)NC(=O)CC2(C)CCOC2)=O)CCCC(C)(C)C1 N1(C(CSCC)=O)CCC2CN(C(=O)CN(S(=O)(=O)c3ccccc3)C)C2C1 CCCCC(C)C(=O)NCC1CC(C)N(C(=O)COCc2nccs2)C1 c1(OC)ccncc1CNC(c1nnnn1C(C)(C)C)C12CC(CO1)C2 N1(C(C(CC)NC(C)=O)=O)CC(C)CCC1C(=O)N(C(CO)C(C)C)C N1(C(c2ccc(C)cc2)=O)CCCC(CNC(C2(C)CCCCO2)=O)CC1 C1(N(C(=O)Cn2cnccc2=O)C)CC2CCC(C1)N2C(=O)Cn1cnnc1O c1(C(=O)NC2(C)CN(C(c3n(CCOC)ncc3)=O)C2)cc(C)cc(Br)c1 c1(NC(c2cncc(-c3cc(C)c(C)nc3)n2)=O)cnn2cc(Br)ccc12 c1(OCC)ccc(C(=O)NCC2(NC(=O)CSc3nc[nH]n3)CCOC2)cn1 c1(CC)c(C(=O)N(C)CC2COCCN2C(=O)C(CSC)OC)cnn1C CC(CC(F)(F)F)C(=O)NC1CN(C(c2ccc(N(C)C)cn2)=O)CC(F)(F)C1 c1(NC(C(=O)N(CCCc2ncco2)C)=O)ccccc1N1CCCC1 C1(COC)(NC(=O)CCC(=O)N(C)C)CCN(C(c2cc(C(F)F)no2)=O)C1 C(=O)(C(O)CC(N)=O)N(CCNC(c1c(CC(=O)OC)scc1)=O)C c1(N(C(=O)CCCCCO)C2CC23CCNCC3)ncnc2[nH]cc(I)c12 n1(CC=C)nc(-c2ccc(N)cc2)nc1CCc1cnc[nH]1 C1(CNC(c2cc(C)[nH]n2)=O)CCCC(NC(c2ccnnc2O)=O)C1 C1(CC)CC(C(=O)NCCCOCCCO)CCN1C(C1C2CCC(F)C12)=O N1(C(C(COC)N(C)C)=O)CCCC(N(C(=O)Cc2ncc(C)s2)C)CC1 c1(C(N2CC(OC)(CNC(c3cncnc3)=O)C2)=O)cccc(CF)c1 c1(OC)ccccc1S(=O)(=O)Nc1cc(-c2ccncc2C)n(C)c1 Cc1cn2c(=O)c(C(N3CCC(C(N4CCC(=O)C(C)C4)=O)CC3)=O)cnc2s1 c1(NC(C(C)NCCc2cn(CCN(C)C)nn2)=O)ncccc1F C1(NC(CCc2nc(C)sc2)=O)CC(NC(c2cnoc2C2CC2)=O)CC1O N1(C(C2(C#N)CC(=O)C2)=O)CCCC(C(=O)NCc2ncccc2F)CC1 Cc1coc(C)c1C(=O)N(C1CCN(C(=O)C(C)(F)F)C1)C C1(C(CNC(C(COCC)C)=O)(C)C)CCN(C(=O)C=CC2CCOC2)CC1 C1(C(=O)NC(C#C)CC(C)C)C(C)OCCN1C(=O)C#CC(C)(C)O N1(C(C2CCC(C)(C)O2)=O)CCCC(C)(C)C1CNC(=O)COC1CC(F)(F)C1 c1(C(=O)NC2CCC(CNC(=O)CSc3cccc(Cl)c3)C2)cc(F)ccc1O C1(C(N(CC(CC)(O)CC)C)=O)CC2(CC(NC(C3CC(C(C)C)=NO3)=O)C2)C1 c1(C(=O)NCC(C)NC(=O)CC2CCCCC2)c[nH]c2cc(Br)ccc12 C(C)(C)(CCCNC(=O)Cn1cnnn1)NC(CN(C(COC)=O)C)=O C(=O)(CCC[N+](=O)[O-])NC1(CC=C)CN(C(C2CCC(=O)N(C(C)C)C2)=O)C1 CN1CCC(C(N2CCC2CF)=O)C1=O C1(C)(NC(C(CCN(C)C)O)=O)CCN(c2ncc(F)cn2)CC1 N1(CCNC(C2C(CC)C2)=O)CCCN(C(c2cc(C#N)oc2C)=O)CC1 C(=O)(C1=CCCCC1C)NCCOC(CNC(C(C(=O)OC)C)=O)(C)C c1(C(N2CC(F)(CNC(C3C(C)(C)CO3)=O)C2)=O)cc(O)nc(O)c1 n12cc(nn1)C1(F)CN(C1)C(=O)CC2.C1(C(=O)OC)CC(C(=O)O)C1 N1(C(C2(C)CC2(Cl)Cl)=O)C2CCC1CC(NC(=O)CCc1ccc[nH]1)C2 C(C)(C(=O)Nn1nnc2c1CCCC2)N.C(=O)(C(CCC)C(=O)OC)CCC c1(C(N(c2cc(OC)ncn2)CC2CNCCO2)=O)c(F)ccc(C)c1Br c1(C(=O)NC2CC(NC(=O)OC(C)(C)C)C2)c(Cl)cncc1Cl.c12cnc([nH]1)C2 N1(C(c2cc(C)nc(O)n2)=O)CC(C(=O)NCC2([Si](C)(C)C)CC2)CC12CCC2 C1(F)(CNC(CC(=O)NCC#C)=O)COCCN(C(c2ccnc(O)c2)=O)C1 C(=O)(C1=C(C)CCC1)NC(C(=O)NCCC1(OC)CCC1)CCN(C)C C(c1cc(Cl)ccc1Br)=CC(=O)NCC1C(C(=O)OC)CCC1 Cc1ccc(C(=O)N(C)CCN2CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)c(N)c1 c1(CC(COc2ccc(F)cc2)NC(CC2C(C)C2)=O)ccc2c(c1)OCO2 C(=O)(C1=CCC(F)(F)CC1)N1CCCCC(CNC(c2c(Cl)cc(C)nc2)=O)C1 c1(C(C)OCC)nc(-c2coc(Cl)n2)n(Cc2cccs2)n1 c1(C(=O)NC2COCCC2NC(=O)C(F)(F)CO)cccc2occc12 C1(CNC(c2nc(C(N)=O)sc2)=O)CN(C(C2(O)COC2)=O)CC(C(F)(F)F)O1 N1(C(c2cccc(NC)n2)=O)CC2(CCOCC2)CC1CNC(=O)CC1CSC1 C(CN=C(NCN(C)C)NCC(c1ccc(F)cc1F)(C)O)Nc1ccccc1 C1(Cc2nc(COCC)nn2-c2cncc(C)c2)CCCCC1(C)C C1(C(=O)NC2C(CNC(CSCC(N)=O)=O)C2)CC(=O)N(C2CC2)C1 C(=O)(CCCCCC(C)(C)C)N(C1C2CN(C(C3CC34CCSCC4)=O)CC12)C c1(CC(O)CN2CCC(O)(c3cccc(Br)c3)C2)ccc(Br)cc1 c1(C(=O)NC2CN(C(C(C)=CC3CC3)=O)CC(O)C2)cc2oc(C)cc2[nH]1 c1(CC)nc(C)c(C(=O)NC(CO)C(C)NC(C2(c3ccccc3)CCC2)=O)o1 N1(C(CN(CC#C)C(c2cn(C3CC3)cn2)=O)=O)CC2(C1)CN(CC)C2 C1(C2CC2)(C(=O)NCC2N(C(C3CC3F)=O)CC(O)C2)CC=CC1 c1(C(C2CCCCC2)C)cc(Br)ccc1F.C1(=O)CNC(=O)NCCN1C C(C)(CC(C)NC(=O)C(O)CC1CCOCC1)NC(C(C)OCOC)=O c1(C(=O)NCC(C2CC2)NC(C(c2ccc(C)cc2)C)=O)c(F)ccc(C)c1F C1(NC(C(CC)CC(F)(F)F)=O)CCC2(CC1)CCN(C(=O)CC(C)(C)O)C2 Cc1cc(=O)c(-c2ccccc2)nn1CC(N1CCN(CC(C)(C)O)CC1C)=O N12CCC(C3CCOCCN3C(=O)C1CC=CC)CC2.C(C)(C)(C)OC(=O)NC N1(CCCC(=O)NCCN(C(C2CCSCC2)=O)CC)Cc2ccccc2C1=O N1(C(c2nn(C)c(C#N)c2)=O)CC(C2CN(C(=O)CC3CC4(CC4)CO3)C2)C1 c1(OCC(C)C)ccc(CC(C)C(=O)NC(c2ccc(Br)s2)C)cc1 c1(OC)ccc2c(c1)CC(C(N1CCCN(C)CCC1)=O)O2 c1(CC)ccc(C(C)CC(=O)NCCCCn2cc(C(C)C(=O)OC)nn2)cc1 C(C(O)CC(F)(F)F)N(c1cc(C(F)(F)F)cnc1C)CC c1(C(N2CC3(C(NC(C=C4CCN(C)C4)=O)CC3)C2)=O)c[nH]c2c(F)cccc12 c1(CN(C)C)ccoc1C(=O)N(C(CNC(=O)C(F)n1cccn1)C1CC1)C C(C1=NOC2CN(C(=O)COc3ccccc3)CC12)NC(c1ccnc(C)n1)=O c1(C(=O)NCCCOCCNC(CC=C)=O)nscc1Br c1(CN2CCN(C(CCc3c(C)c[nH]c3C)=O)CC2)cc(O)ccc1O C(=O)(C1CCCn2ncnc21)N1CCC(C2(NC(CCC(=O)NC)=O)CC2)CC1 CCC(CC1CCCC1)C(=O)NCC(O)CCSC C1(C(=O)NC2(C(C)NC(CNC(=O)OCC=C)=O)CC2)CC12CCCCC2 C1(C(N2C(C(C)(C)NC(c3cnc(O)o3)=O)CCC2)=O)CC2C=CC1C2 C1(C(=O)Nc2ccc(-c3n(CC)ncn3)cc2)CC2CCC1C(O)C2O c1(C(N2C(C)CC(NC(c3nc(CCC)sc3)=O)C2)=O)cnn2ncccc12 C1(CC(=O)N(CCCCCSC)CCNC(C2CN(CC)C2)=O)CCNC(=O)C1 C(=O)(C1=C(F)CN(C(C2CCC2C#N)=O)CC1)N(C(CC#C)C)C C(=O)(C(F)(F)C(F)(F)F)NCC1CN(C(Cn2c(C)cnc2)=O)CC1C Cc1cc(C(=O)NC2CCCC2CNC(=O)CC2C=CCCC2)n(C)n1 CC(C)C(O)C(F)(F)C(=O)NC1C=CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 Cc1ccc2nc(C(=O)NCC3CCCN3C(=O)C=CC(=O)N(C)C)ccc2c1 c1(OC)cn(C)c(C(=O)NC(C)CCCNC(=O)C(C)=C2CC2)cc1=O C(C(CC(=O)N1CCC1CC(C)C)NC(=O)Cc1ccncc1)OC N1(CC(N2CC(O)(C(C)(C)CNC(=O)COCC3CCC3)C2)=O)CCS(=O)CC1 C1(N(C(=O)CC2CCCCC2)C)CCOC(C(C)(C)C)C1 N1(C(C2CN(C)C2)=O)CC(NC(=O)Cc2cc(Cl)cc(Cl)c2)C(F)(F)C1 N1(C(C2CC(OC)C2)=O)CCC(C2CCN(C(=O)CCS(=O)(=O)N(C)C)CC2)C1 CC(c1ccccc1C)=CC(N1CCC1CNC(C1CSCCS1)=O)=O CCCCC(F)C(=O)NC(CN(C)C)C(=O)NC(CC)C(C)C N1(C(c2ccc(I)c(F)c2)=O)CCC2C1CCCN2C(c1cc(Br)ccc1I)=O C#Cc1ccc(C(=O)NC(CNC(C2(C)CNC(=O)C2)=O)CC(F)(F)F)cc1 N1(C(C2(CNCc3ccc(C)c(C(F)(F)F)c3)CC2)=O)CCC(=O)N(C)CC1 CCC(CCC(=O)N1CCC(N2CCC2)CC1)NC(c1n[nH]cc1Cl)=O CON(CCC(=O)N(c1cc(C)cc(C)c1)C)C(=O)C1CC1F C1(C#CC(=O)N2CC(CC(=O)NCCC(O)C(=O)OC)CC2(C)C)(CC)COC1 C1(NC(c2nc(C)sc2C)=O)CC2CC(C1)N(C(=O)CC1CCCCC1(C)C)C2 C(CN=c1nc(N2CCC=C(F)C2)c2c([nH]1)CCCC2)C1CN(C)C1 C1(C2(O)CCNC2)(NCC(CCCC)c2ccccc2)CCC1 N#Cc1ccc(CN(C(c2ccc(Cl)cc2)CO)CC2CC2)nc1 C1(COC)(CNC(c2cnc(C3CC3)s2)=O)CN(C(=O)C(C)(C)O)C1 CC1CN(C(=O)CCNC(C2CCC2)=O)CC(C)C1NC(=O)CSc1ccnn1C c1(C(=O)NC2CCCC(NC(c3ccc(C)nc3)=O)C2)ncc(Br)cc1F C1(C)(NC(CC2CCCN(C(Cc3nc(C)[nH]n3)=O)C2)=O)CCC(O)CC1 C(CCO)(C(=O)NCCC1(NC(=O)CCCOc2ccccc2Cl)CC1)N(C)C c1(O)cccc2c1OC(C)(C)C2.N1(S(CC)(=O)=O)CC2CCC(C1)N2C(=O)CC1CC1 C1(CCNC(=O)CCc2cnco2)(NC(=O)C=Cc2ccsc2)CCOCC1 CN1Cc2c(NC(=O)NCc3csc4c3CCC(C)(C)C4)cccc2C1=O CC(C)C(O)C(=O)N(C1CCN(C(=O)COCC2(S(N)(=O)=O)CC2)C1)CCO C1(C(N2CC(F)(CNC(Cc3c(C)con3)=O)C2)=O)Nc2ccccc2C1(C)C C(=O)(C(F)C(CC)CC)NCC1CCC(NC(C(CCC)NC(C)=O)=O)C1 CC(C)(C)C(O)C(=O)NCC12CC(NC(C3(C(F)(F)F)CCCCO3)=O)(C1)C2 CC1CC(NC(=O)CCCn2c(O)nnc2O)CN1C(=O)CC1CCCO1 C#CC(C)(C)C(=O)NCC(=C1CN(C(=O)C(C)CN2CCOCC2)C1)F C#Cc1cccc(C(=O)N(C2CCC(NC(c3cnn(CCC)c3)=O)C2)C)c1Cl CC1C(NC(c2ccco2)=O)CCCN1C(c1ccoc1I)=O c1(C(=O)NC2(C)CN(C(C3COCC(C)O3)=O)C2)cc(F)c(F)c(F)c1N c1(C(N2C(CN(C(=O)C(F)C(F)(F)F)C)CCCC2)=O)ccc2c(n1)CCC2=O c1(C(N2CC(CCNC(=O)C(C)C)(OC)C2)=O)ccc(NC(=O)C(C)(C)C)cc1 c1(CN(C2CCCNC2)CCO)nccc(C2CC2)n1 N1(C(CC(C)OC)=O)CCN(C(=O)CNC(c2nn(C3CC3)cc2Cl)=O)CC1 N1(C(c2c(CC)ncs2)=O)CC(NC(C2CCC(C)(C)CC2)=O)C(C)(C)C1 N1(C(COCCCOC)=O)CCN(CC(C)NC(=O)CC2CC(C)=NO2)CC1 c1(CC)nc(=NC(CCN(C(=O)C(O)Cc2ccccc2)C)C(C)C)s[nH]1 N1(C(C=CC2CCN(C(C3(C(C)C)COC3)=O)CC2)=O)CC(=O)N(C)C(C)C1 c1(C(=O)NC2CC3N(C(CCC=C(C)C)=O)C(CC3)C2)ccc2nc(Cl)nn2c1 c1(N(C(C)CS(C)(=O)=O)C)nc(=N)[nH]c(=NCCN2CC=CC2)[nH]1 c1(C(=O)OC)ccc(C(=O)OC(c2ccccc2F)C)cc1C(F)(F)F N1(C(c2c(OC)ccc(O)c2)=O)CCC2CN(C(=O)C(C)CC3CCC3)CC2C1 C(=O)(C1=NNC(=O)CC1)N1CCC(NC(C(C)(C)C2CCCC2)=O)CC1C1CC1 C1(C)(C(=O)NC(CNC(c2cc(CC)on2)=O)Cc2ccccc2)COCCO1 CC1CCOC1C(=O)NCCNC(=O)COc1ccccc1 C1(C(=O)NCC2(C(=O)NCC3CSC3)CC2)CC1C1CCC1 Cc1ccc(NC(=O)Cc2ccc(C#N)nc2)cc1OC(C)C N1(C(C(C)N(C)C(=O)OC(C)(C)C)=O)CCN2C(=O)CCCC2C1 c1(C(N2C(CC)CN(C(=O)C(C#N)CC)CC2)=O)csc2ccc(C)cc12 S(=O)(=O)(c1cnc(NC2CCc3c(Cl)cccc32)c(Cl)c1)NCC1(C)CCOC1 c1(N2CC3CN(C(c4c(C(=O)OC)cccc4)=O)C3C2)nc(C)nc2ccsc12 c1(N(CCN(C(CC(c2ccc(Br)cc2)NC(C)=O)=O)C)C)ccc(O)nn1 N1(C(C)C(=O)NC2CC(C)(C(=O)OCCOC(C)(C)C)C2)CCCCCC1 N1(C(C(CC)SC)=O)CCC(C)C(N(C(=O)Cc2ccc(C)o2)C)C1 Cc1cc2ncc(C(N3CCC(C(C)(C)NC(c4cncn4C)=O)C3)=O)cc2[nH]1 C(c1ccccc1)=C(CC)C(=O)NC1(NC(=O)OC(C)(C)C)CC(F)(F)C1 N1(C(C(CC)SC)=O)C2CCCC1CC(NC(C1CC3CCC1O3)=O)C2 c1(C(C)=O)cc(C(=O)NC2CN(C(C3CCOC(C)C3)=O)CCC2C)ccc1C c1(C(N2CCC(CNC(C(CCC)C#N)=O)C2)=O)ccc(Br)c([N+](=O)[O-])c1 C(=O)(CC1CN(C)c2ccccc21)NC(CCNC(CCNC(=O)NC)=O)C c1(NC(CN(C(CC(CC=C)OC)=O)C)=O)ccc2nncn2c1 CC1CCC(CNC(=O)Cn2cccn2)N(C(=O)CN(C)C(c2ccoc2)=O)C1 Cn1ccc2c(NCC3CCCN3Cc3cc(I)ccc3O)ncnc12 CC1C(C(=O)NC2CC(CC(C)(C)C)C2)CCN1C(c1cccc(O)c1)=O N1(C(C(C)N(C(c2c(C)cccn2)=O)C)=O)CCc2c(C#N)cccc21 N1(C(CCOCC#C)=O)CC2CCN(C(C3CC4C=CC3C43CC3)=O)C2C1 CC1CN(C(=O)COCc2ccnc(C(F)(F)F)c2)CCCN1C(C1CC1F)=O CCCCC(CNC(c1cccc(N(C)C)c1)=O)NC(C1CCC(=O)N1C)=O c1(NC(C2CCN(C(=O)OC)C2)=O)ccc(C(NC)=O)cc1.c1(N)ccc(I)cc1 c1(N2CCC3(CCN(C(c4ncccc4Br)=O)C3)C2)ncnc2cccc(F)c12 C(=O)(C(C)NC(C)(C)CC)NCCN(C(C=CC)=O)CC(C)O C1(N(C)C)CCCN(C(=O)C(N2CC(O)CC2CN)=O)C1 Cc1nc(C(=O)NCC2CCCN2C(c2ccc(Cl)c(O)c2)=O)cc(O)n1 c1(CCC(=O)NCC(C)N(C(c2cnn(CC)c2C)=O)C)ccc(OC)cc1F CCC(CC)C(C(=O)NCC1CCN(C(=O)C2=NNC(=O)CC2)C1C)OC CC1=C(C(=O)N(C(C)(C)CC(N2CCCOCC2C)=O)C)COCC1 C1(NC(C(C)CO)=O)CCC2CN(C(C3CC(n4cnnc4)C3)=O)CC2C1 C1(C(=O)NC(CC)CNC(=O)CCc2cc[nH]n2)CCC2(CC1)OCCO2 N1(C(c2occ(CN)n2)C(=O)NC2CC(F)(F)C2)CCCN(S(N)(=O)=O)CC1 C=CC(O)C(=O)NC1CC(CNC(=O)CNC(=O)OC)C1 C(=O)(CCCSCCNC(=O)C(C)OCOC)NC1CC(C(=O)NC)C1 C(=O)(C(COC)NC(c1cc(C(C)=O)c[nH]1)=O)N(CCCCC)C C1(NC(C2CC23CC3)=O)CCCC12CCN(C(c1cncc(O)c1)=O)CC2 N1(C(CCC(C)N(C)C)=O)CC2CC1CN(C(c1cnn3c1CCC3)=O)C2 C12(C(C)C)CCN(C1)C2.c1(CNC(c2cn(C)cn2)=O)ccc(Cl)nc1 c1(C(=O)NC2CN(C(COCC)=O)C(C)(C)C2)coc2c(Cl)cccc12 C1(C(=O)Nc2cc(F)ccc2Br)CCC2(CN(Cc3ccc(I)c(F)c3)C2)O1 c1(C(N2CC(C)C2C(N2CCC(N(C)CCO)C(C)C2)=O)=O)cn2cccc(Cl)c2n1 n1(CC(=O)NC2CCC2NC(C2CSCCS2)=O)cccnc1=O C=C(Cl)CC(C(=O)NCc1ccnn1C)NC(c1cc[n+]([O-])cc1)=O CC1CN(C(C2CCS(=O)CC2)=O)CCN1C(C1(C(F)F)CCCO1)=O C(CC(C(=O)N1CCC(n2ccnn2)C1)NC(c1cc(C)[nH]n1)=O)OC C=CCC(CC(C)C)C(=O)NCC1CN(C(c2coc(Br)c2)=O)CC1C c1(-c2ccc(NCc3nc(C)oc3)nc2)ccc2c(cnn2C)c1 C1(C)(NC(=O)NCC2CC(C)(C)COC2)CCC(=O)NC1=O N1(C(C)=O)CCC(C)(CC(=O)NCCSCC2CNC(=O)O2)C1 c1(-n2cc(CC(C(=O)NCCc3n(C)cnc3)O)nn2)ccccc1Cl CC1(NC(c2cc(C(N)=O)co2)=O)CC(NC(C2CSC2)=O)C1 C1(CCC(=O)NCCC(C)NC(C2(P(C)(C)=O)CC2)=O)CCC(O)CC1 CC(CN(C)C)CC(=O)NCC(c1ccccc1Cl)NC(=O)CCC1CCC1 CC1(C)CN(C(=O)C2=CCSC2)CC1CNC(=O)CCCOc1ccccc1Cl c1(C(=O)NCC(C)(C2CC2)NC(=O)CC2CC=CCC2)cc(C(N)=O)co1 N1(N(C(c2cccc(F)c2)CCO)C)CCCCC1CCCN.C C1(C(=O)NCCCC(F)(F)F)(COC)C=CCN1C(=O)CNC=O Cc1nc(C)c(CC(=O)N(CCCNC(c2cn(C(C)(C)C)cn2)=O)C)s1 CC1(C)CC(NC(=O)COCC2CCOC2)CN1C(c1ccon1)=O c1(OC)ccc2c(c1)CCC2C(=O)NC(C)(C(=O)O)C1CCOCC1 N1(C(C(C)S(C)(=O)=O)=O)CCN(C(=O)CC2(C3CC3)CC2)CC12CCC2 C1(NC(c2cc(CC)c(C)s2)=O)CN(C(=O)CCC(C)SC)CCC1C(F)(F)F N1(C(C=CCN(C)CC)=O)CC2(CCN(C(=O)C(C)(O)CC(C)C)C2)C1 C1(C(=O)NC(CNC(c2c(C)nncc2)=O)(C)C(C)C)CCC2(CC1)CC2 c1(OCC)ccccc1C(N1CCCC1C1(NC(c2coc(SC)c2)=O)CC1)=O C1(C(N(CCO)CC)=O)CCOC1CNC(c1cc(C)cs1)=O CC(C)(CCC(=O)NC1CCCC(C(=O)NCc2cccc(O)n2)CC1)[N+](=O)[O-] c1(C(=O)NC2C(C)CCN(C(c3ns[nH]c3=O)=O)C2)ccc2c(c1)NCCC2=O C(=O)(C(C)(C)C(C)NC(C1CC2(C1)CC2(F)F)=O)N(CC(COC)(F)F)C Cc1c[nH]cc(C(=O)NC2CCCN(C(=O)CN3CCCC3CO)CC2)c1=O N1(C(c2ccc([N+](=O)[O-])s2)=O)CCC2CCN(C(C3CC4(CC4)CO3)=O)C2C1 Cc1cc(Br)cc(F)c1NC(C1CC(NC(=O)C(Cl)(Cl)Cl)C1)=O C(CCC(CCC)NC(c1coc(Cl)n1)=O)NC(C1C(=C)CC1)=O C1(CNC(C2CCN(C(CC)=O)C2)=O)CN(C(c2ncc(F)cn2)=O)CC1(C)C C1(CNC(CCC=C)=O)CC2CCC(C1)N2C(=O)CN1CCOCC1=O C1(c2c(OC)c([N+](=O)[O-])c(F)cc2)C2=C(C(C)N(C)C2=O)N(C)C(=O)N1C C#Cc1cc(C(N2CCC(NCCCC3(C)NC(=O)NC3=O)C2C)=O)ccc1C CCCS(=O)(=O)C(C)C(=O)N1CC2CCCN(C(c3cscc3C)=O)C2C1 C1(NC(CC2CC(N(C)C)C2)=O)CC12CC(NC(c1ccnnc1)=O)C2 N1(C(C(C(=O)OC)C)=O)CCCC2(CCN(C(c3cccc(Cl)c3C)=O)C2)C1 O(NC(=O)C(F)C1CCN(C(C2CC=CCC2)=O)C1)CCC CN(C)C(=S)NCC(=O)NC1CC(Cl)=NO1 CCN=c1[nH]c(C(=O)NC(CNC(=O)Cc2cccs2)C(C)C(C)C)cs1 C1(NC(C(CCCC#C)C)=O)CN(C(=O)CC2(O)CCOCC2)CCC12CCC2 c1(NC(C2CC2Cl)C)cc(C)c(S(=O)(=O)N2CCC=C(F)C2)cn1 CC(CN(C)C)C(=O)N(C1CC(NC(c2c[nH]c(=N)s2)=O)C1)C C1(CCC=C)(C(=O)NC(c2nc[nH]n2)C)CN(C(c2c[nH]nc2OC)=O)C1 C(CO)(CCCCNC(c1cnn(CC)c1)=O)NC(C=CCCC)=O O=C1CN(Cc2ccnc(OCC(F)(F)F)c2)C(=O)N1CCC1CCCO1 c1(C(=O)NCCN(C)C(c2c[nH]nc2C2CCCO2)=O)cccc(F)c1Cl c1(C(=O)NCC2N(C(c3cc(C)n(CC)c3C)=O)CC2)cc2cccn2c(O)n1 N1(C(COCCCC#C)=O)CCC2(CC1)CC2NC(c1c(C)csc1Cl)=O C(C(=O)NC1CCCCC1NC(c1csc(C(F)(F)F)c1)=O)(C(C)C)OCC N=C1NC(=O)C(CC(N2CCN(C(C3(c4ccc(Cl)nc4)CC3)=O)CC2)=O)S1 CC(C)(CC(=O)Nc1cccc(Cl)c1)NC1(F)CN(C(=O)NC2CCCCC2)C1 CCCCCCC(F)C(=O)NCC1CC(NC(=O)C=CC)C(O)C1 c1(C(=O)NC2CC(C)CN(C(C3CC=CC3)=O)C2)c(F)ccc2nc[nH]c12 C(=O)(C(C)C(C)(F)F)NC(CCNC(CCC(C)=O)=O)C C(=O)(CCC(C)(F)F)N1C(C(N2CC(C)C2C(=O)O)=O)C(C)C1 c1(C(=O)NC2CCCC(NC(c3ccc(F)cc3)=O)CC2)ccccc1[N+](=O)[O-] C1(C#CC(=O)NC(C2CCN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)C)(CC)CC1 c1(OC)cc(C(=O)NCC2CN(C(=O)C(C)(F)F)C2)ccc1OCCC(C)C N1(C(c2nccc(CC)c2)=O)CCCCC(NC(=O)COc2cccc(C)c2)C1 N1(C(C=CCC)=O)CCCCC(CNC(=O)C(CC2CCOCC2)OC)C1 CC1=CCN(C(=O)CCC2(NC(C3CC34CC4)=O)CCC2)CC1 C=CC1(c2cn(Cc3nncs3)nn2)COCCN1C(=O)CC1CCN(C)C1 c1(C(=O)OC)ccc(NC(C2CC2NC(c2ccc(OC)cc2I)=O)=O)c(C)c1 C1(NC(C=CCOC)=O)CCC12CCN(C(=O)CC(C)n1ccnc1)CC2 C1(C(=O)NCC2CC(NC(c3c(C)n(C)nn3)=O)C2)CC2(CCC2)CO1 N12CCC(CC1)CN(CCC)C2=O.C(C)(C)(C)NC(=O)CC C12(CNC(C(c3ccc(Cl)s3)C)=O)CCC(CC1)N(C(=O)CC1CCC(=O)N1)C2 CN1CCC(C(N2CC(N3CCNC3=O)C2)=O)(NC(=O)C2=CCSC2)C1 c1(-n2ncc(C(=O)NC(C)C(C)NC(c3cncn3C)=O)c2)cccc(F)c1 N1(C(c2ncc(NC)nc2)=O)CC2CCC(C1)N2C(=O)Cc1coc(C)n1 N1(C(c2n(CC)ccn2)=O)CC(NC(c2nncs2)=O)CC1(CC)CC c1(OC)ccc(C(F)(F)F)cc1NC(C1CCCN1C(=O)C(F)CC1CC1)=O N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC2CCC(C1)N2C(C1(C#N)CC1(C)C)=O C12(CNC(COC(CC)C)=O)CC(NC(c3ncc(Cl)cc3F)=O)(C1)C(C)(C)O2 c1(C(N(C2CN(C(c3coc(CO)c3)=O)CC2O)C)=O)ccc(OC(F)F)cc1 Cc1nc(C(=O)NC(C)C(C)NC(=O)Cn2cc(CO)nn2)c(C)s1 c1(NC(=O)NC(C)CN(C(=O)CNC(=O)CC2CCCC2)C)csc(Cl)c1 C(CCCCCOC)(C(=O)NNCC1CCOCC1)N1CCC(C#C)(O)C1 c1(C(=O)NC(C2(O)CN(C(C3C(C)C3)=O)C2)C)cccc2sncc12 C1(NC(CCNS(C)(=O)=O)=O)CCN(C(=O)C=Cc2ncc[nH]2)C12CCC2 c1(C(=O)NC(C)(C)CNC(=O)Cn2nccn2)cccc(Oc2ccccc2)c1 N1(C(C(=O)NC(CC)(C)C)c2cccs2)CCN(Cc2ccco2)CC1CSC C(=O)(C(O)P(C)(C)=O)N1C(CNC(CCC(c2cc(C)sc2C)=O)=O)CCC1 C(=O)(C(C)CC(C)(C)C)NC(C(=O)N(CC(C)C#N)C)(C)C C1(NC(=O)COC2CCN(C(c3ccc(C(F)F)o3)=O)C2)CCC=CCCC1 c1(CC(=O)NCC23OCC(NC(C=CC=CCC)=O)(C2)C3)cc(F)ccc1Cl C12CN(CC13CC3)C2=O.C1(CN(C(=O)CC2CCC2)C)C(C#N)C1(C)C C1(NC(=O)Nc2cccc(OC)c2)CN(C(=O)C(C)n2cncn2)CC1C#N C1(NC(CCC(=C)Br)=O)CC(F)CN(C(=O)C(C)OC(C)=O)C1 N1(CC(C(=O)NCC#N)N(C)C(c2ccc(Br)cc2)C2(C)CC2)CCCC(C)(C)C1 C1(NC(C(C)(C)C(N)=O)=O)CCC2CC1CN2C(c1cnn2ccccc12)=O C1(NC(C(CC=CC)CC)=O)CC2CCC1CN2C(=O)Cc1cc(F)ccc1O N1(C(c2cn(CC(F)(F)F)cn2)=O)CC(NC(C2(Br)CC2)=O)CC(O)C1 C(C(C(C)(C)C)NC(=O)COCCc1ccc(Cl)s1)NC(CC(=O)NCC)=O C1(CC(=O)N(C)Cc2ccon2)CN(C(=O)C(C)(O)C2CCC2)CCO1 Cc1cc(N)c(C(=O)NC(CNC(C2CCCC(F)(F)C2)=O)C2CCC2)cc1C N1(C(CC(CCC)CC)=O)CC2CC(C)N(C(=O)COC(F)(F)F)C2C1 C1(C(=O)NCC(CNC(c2ccc(OC)s2)=O)(C)OC)CCN(C)C1C Cc1cc(C(N2CC3C(C(=O)N(c4ccccc4)CCO)C3C2)=O)c(Br)cc1F N1(C(CCCNC(C)=O)=O)CCC2(CC(C(=O)NC(C)CC(F)(F)F)C2)C1 C1(C(=O)NCCC2(C(=O)NCC(C(CC)C)C)CC2)CCCCC1(C)C c1(C(=O)NC2(CNC(C3CCC(C)CC3)=O)CCC2)ccc(=O)n(CCF)n1 CC(CCCCNC(=O)C=CCN1CCOCC1)NC(C1(CO)CCOCC1)=O CCCCC(C(=O)NC(c1ccccc1F)C)NC(=O)CC(=O)NC C(C)(CC(C)NC(c1occc1Br)=O)NC(CSC(C)C)=O C1(CNC(N2CC(c3n(C)ncc3)S(=O)(=O)CC2)=O)CCCC2(CCCC2)C1 N1(C(CCc2c(C)noc2)=O)CC2CN(C(c3c[nH]c(Br)c3)=O)CCC12 CCC(C)C(C)CN1C(C2CC2)C1=O.c1(NCC(=O)O)ccc(C2CC2)nn1 c1(C(=O)NCC(CC(=O)NCC2(O)CCCC2)OC)cc(O)ccc1C N1(C(c2n(C)ccc2)=O)CCN(C(c2cc(C(F)F)ccc2F)=O)CC(O)C1 C1(NC(C(C(C)C)SC)=O)CCN(C(c2cc(C3CC3)nc(O)c2)=O)CC1F C=CCCC(F)(F)C(=O)N1CC2(CCC2NC(c2cc(C3CC3)ccn2)=O)C1 N1(C(CCNC(=O)C=CCl)=O)CCCC12CCCN(C(=O)CC(F)F)C2 CCCCC(O)C(=O)NCC1CCC1NC(c1csc(Br)c1C)=O N1(C(C2CCN(CC)C2)=O)CCC(CN(C)C(C2CC2c2ccncc2)=O)CC1 c1(CC)cccc(C(=O)NCC2(CO)CCN(C(c3ccc(=N)[nH]n3)=O)C2)c1C C(=O)(CCCC(=O)N1CCC(C(=O)N(C)CCc2ccncc2)C(C)C1)OCC Cc1cccc(C(=O)NCC(C)C(=O)NO)c1F.C12CC(C1)NC2=O CCCCC(C)CCC(=O)NC(CNC(=O)CNC(c1ccoc1)=O)CCC CCCCC(O)C(C)C(=O)NCC1CC(C(N2CCC23CCCSC3)=O)=NO1 c1(N2CC(C)C(O)C(C)C2)ccc(S(=O)(=O)NCCc2cnccn2)cc1Cl Cc1c(C(N2CCN(C(=O)CC3CCC(=O)NC3)C(CF)C2)=O)cncc1Cl CCCCC(C)(F)C(=O)NCC(C)CN(C(=O)C(N1CCCCCC1)C)C C1(C(N(CCC(C(C)(C)C)NC(=O)C#CC2CC2)C)=O)CN(CP(C)(C)=O)C1 c1(C(N2CC(CNC(C(C)C3CCOC3)=O)N(C)CC2)=O)ccc2[nH]ccc2c1 Cc1ccc(C(=O)NC2CCC2NC(c2nccn2C(C)C)=O)c(Cl)c1 N1(C(c2occ(C)c2C)=O)C2CCC1CC(CC(C)NC(=O)C1=CCCS1)C2 C(C(C)CN=c1nc(C(C)C)[nH]s1)SCC.c12ccccc1C(=O)NC2 N1(C(C2CC(CCC)C2)=O)CCC(NC(c2ncsc2C)=O)C(F)C1 C1(c2ccccc2)(NC(C2C(C#N)C2)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)C1 Cc1nc(C(=O)NC2CCCC2NC(=O)CC(C)(C)C)nn1C Cn1nc([N+](=O)[O-])cc1C(=O)NCC1(NC(=O)Cc2ccc(Cl)c(F)c2)CC1 c1(C(=O)NC2CC(F)(CNC(C3C(C)(CC)C3)=O)C2)ccc2cccnn12 CC(C)CC(CC(=O)NCC1(CO)CCCC1)NC(=O)C(C(C)O)N(C)C C1(S(C)(=O)=O)(C(=O)NCC2N(C(CNC(C(CC)C)=O)=O)CCC2)CC1 Cn1ncc(C(=O)NC(Cc2cc[nH]n2)C(=O)NCCCn2cnnc2)cc1=O C1(O)(CNC(C2(C(C)C)CC2)=O)CCCN(C(c2c(C(=O)OC)cccn2)=O)C1 c1(CNc2c(C(=O)Nc3ccc(-n4cccn4)cc3)scc2)cc(O)cc(F)c1 CC(C)CC(C(=O)NCC#CCNC(=O)CCc1ccccc1Br)C(C)C N1(c2c(OCCC)nccc2)CC(C2CCCCN(C(=O)CC3CC3(Cl)Cl)C2)C1 Cc1ccc(C)c(SCC(=O)NCCN(CC(C)O)C(c2ccccc2Cl)=O)c1 C1(OC)CC(CC(N2CC(O)(CN(C)C(c3ccc(C)s3)=O)C2)=O)C1(C)C C(=O)(C1=CCC(C)(C)CC1)NCC1CCC2(CN(C(C(COC)O)=O)C2)O1 C1(NC(C2N(C(C)=O)CCC2)=O)CCCN(c2nnn(C)n2)C1 Cn1nc(C(F)(F)F)c(CNCCCNC(=O)CC2(C)CC2F)c1Cl C1(CC(=O)NCC(Cn2ncc(C)c2)C)CCCC12NC(=O)NC2=O c1(CC(C(=O)NCC(C)N(C(=O)CC2CCNC2=O)C)(C)C)cc(F)ccc1F O=C(C1Cc2ccc(Cl)cc21)NCC1CCN(c2cc(-c3cccs3)ncn2)C1 C1(O)(CNC(CC(C)C2CC2)=O)CCCN(C(C2(C)CCC(=O)N2)=O)CC1 C(=O)(CCS(=O)(=O)N(C)C)NC1CCC(CNC(c2ccc(C)cn2)=O)C1 C(=O)(CC(C)C(F)(F)F)NCC(CNC(=O)CNS(C)(=O)=O)OC C(=O)(C1CCc2cc(F)ccc21)NC1C2CCN(C(c3cn(C)[nH]c3=N)=O)C2C1 c1(C(=O)NC2CC(NC(c3cncc(O)c3Cl)=O)C2)cc(C(F)F)ccc1Cl C1(CC)C(NC(=O)CC2COC(=O)N2)CCN1C(=O)CSC(F)(F)F C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(c1ccc3nsnc3c1)=O)C2 c1(CC)cc(C(=O)NC2CC3(C2)CC3NC(=O)CC2OCCCO2)sc1C C1(OC)CN(C(C2(O)CC2)=O)CC1C(N1CCN(CC(N)=O)CC1)=O C1(CC(=O)N(C(C)COCC)C)CC(O)C1(C)C.C1C(=O)N1CC#C Cc1ccc(C(N2CC(F)CC2CN(C)C(C2(F)CCCOC2)=O)=O)cc1F N1(C(c2ccc(N(C)C)cn2)=O)CCCCC(NC(=O)CCC2CCC2)C1 N1(C(c2n(C=C)nnc2)=O)C2CCC1CC(CNC(=O)C(C)OCC)C2 N(C(=NCCc1cccnc1-n1cccn1)NCC(C(C)C)C(C)C)C(CC)C N1(C(C(OC)OC)=O)CCC(C)C1CNC(C1CCCN(C(C)C)C1)=O C(=O)(CCC(C)(C)NC(N1CCC(SCC)CC1C)=O)OCC c1(C(=O)NC2CC=CC2)cc(C(N2CCCC(CCOC(C)(C)C)C2)=O)ccn1 N1(C(c2cc(C)ncn2)=O)CCC2(CCCN(C(=O)CN3CCCC3C)C2)C1 C=CCC(CC=C)C(=O)NCCC1CCN(C(=O)C(=O)Nc2ncc[nH]2)C(C)C1 N1(C(c2cc(C)no2)=O)CCOC2(C1)CN(C(=O)CC(C)N1CCCC1=O)C2 Cc1oc(C#N)cc1C(N1CCC(CC(=O)NCCC2CC(C)(C)CO2)CC1)=O c1(C(=O)NCCC(C)N(C(CC2CC(=C)C2)=O)C)cc(C)cc(C)c1N C#Cc1ccc(C(=O)NCCN(C(=O)C=C(CC)CC)C)c(F)c1Cl Cc1cc(O)ccc1C(=O)Nc1ccc(-n2ncnc2C)cc1 c1(C(=O)NCC23C(CN(C(C(=O)NCCOC)=O)C2)C3)nn(CC)cc1[N+](=O)[O-] C1(C#N)(NC(C(C2CCCN(C(c3ccc(C)cn3)=O)C2)C)=O)CCOCC1 c1(CC)cc[nH]c1C(=O)NC1CC(NC(C2(CSC)CCCO2)=O)C1 c12ccccc1C(=O)N(C)C2c1ccccc1.C1(CC(CO)N)CCOCC1 c1(C(=O)NCC2CN(C(C(CC)SC)=O)CC2C)cccc2c1OCC2 N1(C(CCN(C(C2COCOC2)=O)CCO)=O)CCC(CC2CC2)CC1 N(C1CCOc2ccc(Cl)cc21)C(=O)Nc1c[nH]c2cc(F)c(F)cc2c1=O c1(C(N2CC(C)N(C(=O)CCC3CNC(=O)N3)CC2)=O)cnn2ncccc12 c1(C(N2CC3CN(Cc4c(C)c(O)ccc4)CC32)=O)ccc2ccccc2n1 c1(C(C)C(=O)NC2CCC(O)CN(C(=O)CNC=O)C2)ccc2c(c1)OCCO2 c1(CC(=O)NC(C2CN(C(C=CC=CC)=O)C2)C)coc2cc3c(cc12)CCC3 c1(C(=O)NCC(CN(C)C(c2cccnc2)=O)(C)C)cc(=O)cc(Cl)[nH]1 S(=O)(=O)(c1cccc(F)c1)NCC(=O)NC(CCN(C(=O)CCCF)CC)(C)C C1(C(=O)NCc2ccc(O)cc2)CC2CCC1N2C(=O)C1CC1.c12nn[nH]c1N2 C=CC1CN(C(=O)NC2CCCCC2C2CC2)CCC1CC(=O)O CC1(NC(C23CC(F)(C2)C3)=O)CCN(C(c2c[nH]cc2Br)=O)C1 c1(NC(=O)Cn2cnnn2)cc(CNC(=O)CCC2CCCCO2)on1 C1(C(N(CC(C)NC(C2(C)CC(=C)C2)=O)CC)=O)CC2CC1C1CC21 c1(OC)ccc(CN2CC(NC(c3c(OC)cccc3Br)=O)C(O)C2)cc1OC C(CCN=c1nc2ncn(C)c2c(NCCN2CCC3CC23)[nH]1)(C(C)C)OC Cc1cccc2c1OC(C(=O)NCC1(NC(c3sc(N(C)C)nc3Cl)=O)CC1)C2 Cc1cc(O)c(CNC2CC(NC(c3cc(=O)cco3)=O)C2)cc1Cl Cc1ccc2c(c1)CCN2C(=O)CCS(=O)(=O)Cc1cnccc1.CC(C)C(O)C1CC1 C=CCCCCCC(=O)NCC1CC(C)(C)CCC1NC(=O)CN1CC2CC2C1 c1(C2C(CC)N(Cc3ccccc3)CC2)ccn2nccc2n1 Cc1cc(C(N2CC(NC(=O)CC(C)c3ccco3)C(C)(C)C2)=O)nnc1O c1(C(N(CCCNC(C2CCS(=O)(=O)C2)=O)CCC)=O)cc([N+](=O)[O-])sn1 N1(C(C(COCc2ccccc2)OC)=O)CCC(NC(=O)C2=CSCS2)C1(C)C C(=O)(C1CCc2cccnc21)NC1CCC2(CCN(C(C(C)O)=O)C2)C1 N1(C(CC2CCN(C(CCCOC(C)(C)C)=O)C2)=O)Cc2n[nH]cc2C1CO N1(CCC(=O)N(CCCNC(=O)CCc2scnc2C)CCC)CCC(C)CC1 N1(C(c2c(C)c(Cl)cnc2)=O)CCC(NC(=O)CCC(C)C)C(CO)CC1 N#Cc1ccc(Cl)c(CN2CCCC(CCNC(c3ncccc3Cl)=O)C2)c1 C(N=C(NCC12CC(CCO1)C2)N1CCCC(F)(F)C1)c1n(C)ncc1 C(=O)(C1CCc2snnc21)NC(CN(C(C(CC(CC)C)C)=O)C)(C)C CC(C)CCCCCC(=O)N(C(C)(C(=O)N1CCC(C2CCCO2)C1)C1CC1)C CN1CC2CCN(C(C3CCCCN(C(=O)CC4OCCC4(C)C)C3)=O)CC2C1 Cc1nc(NC2(COC(C)C)CC3CCC2C3)cc(=NC(=O)c2cnoc2)[nH]1 c1(C(N2CC(CC(C(=O)N(C(CC)C)CCO)F)C2)=O)cncnc1C C1(NC(c2cnc(C3CC3)s2)=O)COC2CN(C(C3(O)CCSCC3)=O)CC12 N1(C(c2ccc(C=C)cc2)=O)CC(C2CN(C(=O)CN3CCC(C)CC3)C2)C1 N1(C(c2nnc(C)s2)=O)CC(CNC(C2CCCN2S(C)(=O)=O)=O)C2(CCC2)C1 C1(N(C(C=C(CC)CC)=O)CCF)CCCN(C(C2C(C(F)F)C2(C)C)=O)C1 c1(OC)nc(=NC2CCC3(CC2)CN(C(=O)C(C)=C2CC2)CCO3)nc(OC)[nH]1 N1(C(c2c(C)ncs2)=O)CCC2(CCC2CNC(C2COCCO2)=O)CC1 c1(C(=O)NCC2CC(NC(C(CC)OC3CCCCC3)=O)C2)cccc(NC)n1 c1(CC(N2C(CC(=O)N(C(C)(C)C)CCO)CCC2)C(=O)O)ccc(F)cc1 C1(NC(c2c(OC)oc(C)n2)=O)CCC2CN(C(C3CCCO3)=O)CCC2C1 N12CCC3CCCC13C2=O.c1(COc2ccc(OC)cc2)cc(O)cc(=O)o1 S(=O)(=O)(c1c[nH]c(C(=O)O)c1)N(C)CC1CC(OC2CCOCC2)C1 c1(-n2cc(C(N(C(c3nc(Cl)sc3Br)=O)CC)C)nn2)ccnc(CO)c1F C1(CC)CN(C(=O)CCCN=[N+]=[N-])CCC1NC(=O)CC1CCS(=O)(=O)C1 C(C(CC(=O)NC1CC(CNC(C2CC(n3cnnc3)C2)=O)C1)C(F)F)N(C)C CCC(F)(F)C(C)(C)C(=O)NC1CC1NC(=O)C(C1CCOC1)OC C1(CNC(CC(CC)C2CCC2)=O)CN(C(c2ccnc(Cl)c2N)=O)CCCO1 C1(CNC(c2c(OC)c(Cl)ccc2)=O)C(C2CC2)CCN1C(=O)C1=NOCC1 N1(C(C2(CC3CCCOC3)CC2)=O)CCC(O)(CNC(C)=O)C1.C1(=O)CON1 c1(C(=O)NCCCN(C(=O)C(C)(F)F)C(C)C)cc2ccccc2c(=O)o1 c1(C(=O)NCC(CNC(CCC(C)OCC)=O)O)cc2nc(C)[nH]c2cc1F C(=O)(CCC(C)CN(C)C)N(CCCNC(C1CN(C(C)=O)CCO1)=O)CC N1(C(Cn2c(C)cc(C(F)F)n2)=O)CC2(CCN2C(=O)COC2CCOC2)C1 C(C)(CC(=O)NC1CC1NC(c1cc2cc(Cl)ccn2n1)=O)(C(F)(F)F)N(C)C Cc1cc(C=CC(=O)NCC2CCCN(C(=O)C(O)C(F)F)C2)ccc1Br Cc1cc(F)cnc1C(=O)NCCC1CN(C(C2(C(F)(F)F)CC2)=O)C1 c1(CC)cc(OC)cc(C(=O)N(CC(C)NC(C2(O)CCCCCC2)=O)C)c1 N1(C(C=CCOCCOC)=O)CCN(C2CCCC2NC(C2CC23CCC3)=O)CC1 N1(C(CSCCOC)=O)CCC(C(=O)NCc2n[nH]c3c2CCC3)C12CCC2 C1(C(N(CCCCN(C(C(C2CCCCC2)OC)=O)C)C)=O)CCOC1C C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1(C)CCN(C(N2CC(C)CC(C)C2)=O)CC1 C1(CNC(CN(C(C)C)CCF)=O)CCOC(C(C)C)C1 C1(CNC(C(C)c2cc[nH]n2)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1O C1(C(N2C(C)CN(C(C3CC(F)(F)C3)=O)CC2)=O)C(O)C(=O)N(C)C1C c1(CC)nn(C)c(C(=O)NC2CC2CNC(c2cccc(C(C)(C)C)n2)=O)c1Cl C1(C)(C(=O)NCC2(C(C)C)CC2)CCCN(C(=O)Cc2cnn(C)c2)C1 CCCC(CCC)C(=O)NCC1CC1CNC(C1(COC)COC1)=O c1(N2C(COCC)CCC2)nc2ccc(OC(F)F)cc2s1 C1(NC(=O)Cn2ccnn2)C2CC1N(C(C1CCC1C(=O)OC)=O)C2 c1(C(N2CCN(C(C(CCC)(C)C)=O)CC2CF)=O)ccc2c(c1)NCC2 Cc1nc2ccc(C(N3CC(NC(C4CC=CCO4)=O)CC(C)C3)=O)cc2s1 C1(NC(C2CCCN2C(c2nccs2)=O)=O)CC2CCC1(CO)C2 N1(C(Cn2c(C)nc(C)n2)=O)CCC(CNC(c2nocc2Cl)=O)C(C)C1 c1(OC)ccc(C(N2CC(N(C(=O)CCC(C)OC)C)C2)=O)c(Cl)n1 C(N=c1[nH]c2c(c(=NCC3(CCOC)CC3)[nH]1)CCCC2)c1c(CC)nccc1 C1(CC#C)(C(N2CC(=CCCCNC(c3nncn3CC)=O)C2)=O)CCOC1 N1(C(c2cnc(Cl)[nH]2)=O)CC(NC(C2(c3cc[nH]n3)CCC2)=O)C(F)C1 C(CC(C(=O)NCC(F)(F)C(C)C)NC(=O)Cc1ccc(C)nc1)SC C#Cc1c[nH]nc1C(=O)N(C1(CC(=O)NC2CCC(CN(C)C)C2)CC1)C C=C(C)CC(C(=O)NCC1CC(C)C1)NC(=O)CC#N c1(C(NC(C)(C)C)OC(N2CC(c3cc(CC)on3)C2)=O)ccccc1F C12(C(N(CCCN(C)C)CCNC(C(C)OCC)=O)=O)CC(C)(C1)OC21CCC1 c1(-c2nc(-c3cc(OC(F)F)ncc3F)on2)ccc2cnccc2c1 N1(C(CCC2CC(C)C2)=O)CC2CCN(C(=O)CN3CCCCC3=O)CC2C1 N1(C(c2c(C)cnn2C)=O)CCN(C(C2CC(=O)N(CC(C)C)C2)=O)CC1C N1(C(CC2CN(C)C2)=O)CC2CCN(C(=O)CCCCc3c[nH]ccc3=O)CC2C1 C1(C(=O)OC)C2CCC(C2)N1C(C1(CC(=O)N(CCC=C)CCOC)CC1)=O Cc1[nH]c(C#N)cc1C(=O)N(C(C)CNC(=O)C1=NNC(C(F)(F)F)C1)C Cc1c(Br)csc1C(=O)NC12CC(NC(=O)CC3(C)CC3)(C1)C2 CC12CCC(NCc3cccc(OCc4ccccc4F)c3)(C1)NC2=O c1(C(C(=O)NC(c2ccc(Cl)cc2)COC)=O)ccc2c(c1)-c1ccccc1C2 C(CC(C(=O)NC1(CO)CN(C(=O)COC2CC=CC2)C1)NC(C)=O)SC n1(Cc2nc(C(CC)CC)nn2-c2nccn2C)cnc2ccccc12 C(=O)(CC(C)(C)C1CCCCC1)N1C(CNC(C2N(C(COC)=O)CCC2)=O)CC1 c1(C(=O)NC2(C)CC(NC(CCCOCCOCC)=O)C2)ccc2cnccc2n1 C1(C(N(CC#CC)C)=O)CCCC(NC(c2cccc(C)c2F)=O)CC1 c1(C(=O)NCC(CNC(=O)CCCc2cccc(Cl)n2)O)ccc(O)c(F)c1F CC1CN(C(c2cc(Cl)no2)=O)CC1NC(c1cn(CC2CCOC2)nn1)=O C(=O)(CC(CN(C)C)C(F)(F)F)NC(CNC(CNC(=O)NC)=O)(C)CO.C1CC1 c1(C(N2CC3(OCCN(C(CCCC=C)=O)C3)C2)=O)cc(S(C)(=O)=O)ccc1Cl C(=O)(C1COc2ccccc21)NCC1CN(C(c2cc(C)on2)=O)CC1(F)CO CC(C)(C)CC(O)C(=O)NC1CCOC1C(=O)NC1CCN(CCF)C1 c1(NCC(=O)NC(C)(C)C)ccc(-c2ccc(CN)s2)cn1 C1(C=O)CC(O)CN1N(C)C.C(=O)C(C)(C)C1(O)CN(C(=O)C2CC2)C1 C1(CNC(C=COc2ccc(OC)cc2)=O)N(C(=O)COC2CC2)CCC1(C)C CCC(C)C(O)CNC(=O)NCc1c(Cl)cnn1C C#CC1(NC(=O)CC(C(F)(F)F)NC(=O)C(c2ccccc2)C)CC2CCCC12 c1(C(N2CC3C(NC(C4CC(c5nncs5)C4)=O)(C3)C2)=O)ccc(Cl)c(F)c1F c1(C(N(C(CNC(CCCC)=O)C2CC2)C)=O)cc(C)ccc1F CCC(Cc1ccccc1)C(=O)NC1(COC)CN(C(=O)C=CS(C)=O)C1 c1(OC)cccc(NC(C2CC(F)CN(S(=O)(=O)CCCCCl)C2)=O)c1Br C(C(COC)CC(=O)NCCCCN(C)C(C1CN(C)CC1C(F)(F)F)=O)OC c1(C(C)C)ccc(C(=O)NC23COC(C2)C(NC(=O)C(F)C(C)(C)O)C3)cc1Cl c1(C(N(CCCCNC(C2CCC2C(N)=O)=O)C)=O)ccc(F)c(CO)c1 CC(=NOCC#N)C(=O)N(CC(C)C(=O)NC1CCC1)C(C)C(C)C CC(C)CC(CNC(C1CCN(C(N)=O)CC1)=O)NC(=O)CCc1cccnc1Cl C(=O)(C(CC1CCC1)C1CC1)CCCn1cc(C(=O)N)nc1.CCCCC1CC1 CCS(=O)CC(=O)NC(C)C(C)(C)NC(c1ccoc1CC(N)=O)=O N1(C(C2N(CC)CCC2)=O)CC(C)(C)CC1CC(=O)NC1CC(OC)C1 C1(C(C(=O)NC(c2ccc(C)s2)C)C)CCN(C(C2(CO)CCC2)=O)CC1 CCCCCCC(C)CC(=O)NCC(F)CNC(c1c[nH]nc1[N+](=O)[O-])=O C(=O)(C1SCCc2ccccc21)NC1CCC(NC(c2cnc(CC)[nH]2)=O)CC1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC(C)CC1CN(C(=O)CC(C)(C)C)C1 C1(C(=O)NC(C2CCN(C(c3cncnc3)=O)C2)C)C2COCC12 c1(CC)c(C(N2CCC(CO)C(NC(=O)C(C)(C)C#N)C2)=O)oc2ccccc12 CCC(C(=O)NC(CCNC(=O)CCn1cncn1)C(C)C)C(C)(C)CC C1(C(=O)OC)CCCCN1C(=O)Cn1cc(-c2cn(CCCC(=O)O)nn2)cn1 CC(C)CC(C)CN=C(NCc1ccco1)NC1CCc2nnnn2CC1 c1(OCC=CC)ccccc1CC(N1CC(NC(C23CCC(C2)C3)=O)C(O)C1)=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(NC(CCCOCC=C)=O)COC1 c1(C(=O)NC(C)(C)CCNC(=O)CSCCC#N)ccc2nsnc2c1 C1(CNC(CC2N(C)CC=CC2)=O)CN(C(C2(CN(C)C)CC2)=O)CCC1(C)C c1(C(=O)N(CCNC(C23CSCC2C3(F)F)=O)C2CC2)ccc([N+](=O)[O-])s1 Cc1c(Cl)ccnc1C(N1CCOCC1CCNC(=O)C(F)C1CCC1)=O c1(C(=O)NCCCN(C)C(c2cccc(NC(N)=O)c2)=O)nnc(S)n1C N1(C(C=CC2(C)COC2)=O)CCCC12CCN(C(=O)Cn1ncc(Br)n1)C2 C1(NC(CNC(C)=O)=O)CCCN(C(=O)C=Cc2sc(Cl)nc2Cl)CCC1 N1(C(Cc2n(C(C)C)cnn2)=O)CCN(C(c2cc(C#N)cn2C)=O)C(C)C1 Cc1nc(C(=O)NC2CC2NC(C2CCC2C(=O)OC)=O)c(C)n1C1CC1 S(=O)(=O)(c1cc(OC)ccc1C(C)C(=O)OC)N1CCCC(COC)C1 C=C(Cl)C(C)(C)C(=O)NCC(F)CNC(=O)C(c1ccc(F)cc1)(C)O Cc1nc2c(C(=O)NC(C)C(CO)NC(=O)C(C)(C)C3CCOC3)ccnc2[nH]1 Cn1ccc(C=CC(N2CC(O)(C(F)C(N3CCCCC3C(C)(C)O)=O)C2)=O)c1 n1(CC(=O)NC(CCNC(C(N2CCSCC2)C)=O)(C)C)nc(C)nc1C C(=O)(C#CC1CCCC1)N1CC(NC(C(C2CCOCC2)OCC)=O)(COC)C1 c1(C(=O)NC23CC(C2)N(C(c2ccc(F)cc2F)=O)C3)ccc2nonc2c1 Cc1cc(C)n(C(C)C(=O)NCCN(C(=O)Cn2ccnn2)C2CC2)n1 Cc1nc(CC(=O)NC2CCN(C(=O)Cn3nnnc3C3CC3)C2)sc1C CN(CCC(=O)Nc1ccc(Br)cc1)N1CCCCC(O)C1 C(=O)(C1=CC2CCC=CCCC12)OC.c1(CC)cc2c(s1)NCC2=O C1(CNC(C2(CC#C)CC2)=O)CCCCN1C(c1cnc(C(C)=O)s1)=O CC1(C)CN(C(C2CC(O)CN2C(C2(C#N)CCOC2)=O)=O)CCC1CO c1(C(C)C)cc(C(=O)NC2CCCCC2NC(C2CCCN2C)=O)c(C(C)C)[nH]1 NS(=O)(=O)CCC(=O)NC1CN(C(c2cccc(N3CCOC3=O)c2)=O)C2CC12 N1(c2nc(N3CCOC(C)(C)C3)cc(C)n2)CC(=O)N2CCCCC2C1 C1(NC(c2ccnc3[nH]ncc23)=O)C2CCN(C(c3cc(Cl)no3)=O)CCC12 c1(CC)oc(C)cc1-c1nc(-c2cccnc2)nn1C1CCC(C)(C)C1 N1(C(c2c(C)scc2)=O)CC(CNC(C2CCNC(=O)C2)=O)CC(C)C1 Cc1ccc(F)cc1NC(C1C2CCC(C2)C1NC(c1cc(F)n(C)n1)=O)=O c1(C(=O)NCC2C3CCCC2N(C(=O)C2=CCCC2)C3)cc2cc(Cl)ccn2n1 C1(NC(C(CC)O)=O)CC2CCC1CN(C(=O)Cc1ccc(Cl)c(Cl)c1)C2 c1(C(N2C(CNC(=O)Cn3ccc(C)n3)CC(OC)C2)=O)ccn2nccc2n1 CC1(C(=O)NC2CC(NC(c3ccc(CC4CC4)cc3)=O)C2)CCCCO1 C#CC1CC2(CC2)CN1C(C1CC(C)CN1C(=O)Cc1ccc(C)nc1)=O c1(SCCCC)ccc(Cl)cc1C(=O)NCC(CCOC)NC(=O)CC(C)F N1(C(=O)CO)CCCC2(CCN(C(C3(Cc4ccccn4)CC3)=O)CC2)C1 N1(C(c2cnc(C(=O)OC)s2)=O)CCCN(C(=O)C=Cc2cncs2)C(CO)C1 c1(C(=O)NCC2(NC(C(CC)C#N)=O)CCCC2)cc2c(ccn2C)s1 CCCC(C)(CC)C(=O)NC1CC(C(=O)N2CCC(c3nc[nH]n3)C2)=CC1O C12(CNC(c3nccc(C)c3)=O)CCC1CCN2C(c1cc(N(C)C)ccn1)=O c1(C(NOCCCC)=O)[nH]ccc1C(=O)NC.C12CCCC1CNC2=O Cc1ccc(F)c(C(=O)NC(C2(O)CCCCC2)C(N2CC3CC(C)C3C2)=O)n1 N1(C(C(C)N(C)C)=O)CCC(CO)(CNC(c2cc3[nH]ccc3s2)=O)CC1 CCCS(=O)(=O)CC(=O)NCC(C1CCCC1)NC(C1CCC(CC)NC1=O)=O c1(CCC(=O)N(CCCNC(C2CNC(=O)N2)=O)CC)cc(F)cc(F)c1 c1(C(=O)NC(CCNC(C2C(C)CC2C)=O)(C)C)cncc2sccc12 N1(C(c2c(CC)nco2)=O)C(C(N2CC3(CCCCC3)C2)=O)C2CC(O)C1C2 CC1CS(=O)(=O)CCCN1C(=O)C(C1C2CC3CC(C2)CC1C3)N c1(C(N2CC(CCOC)C(C)C2)C(=O)NCC(=C)C)ccc(CC(C)C)cc1 N1(C(C2C(C)(CC)C2)=O)CCC(O)(CN(C(=O)CCOC2COC2)C)CC1 CSC=CC(=O)NCC1(O)CN(C(=O)C=CCN2CCC2)C1 C(C)(CO)(C(=O)NCC1CC1CNC(c1cc(-c2csc(C)n2)c[nH]1)=O)OC c1(NCCC2CCC(NC(CC)=O)C2)ccc(C#N)cc1[N+](=O)[O-] Nc1c(C(=O)NC2CC3CC(NC(C4(F)CC=CC4)=O)C2C3)sc2nccnc12 C1(NC(c2nc(COC)oc2)=O)CC2CC1CN(C(=O)Cn1cccnc1=O)C2 c1(C(=O)NC2CC(Nc3c(C(=O)OC)cnc(C)n3)C2)ccc(C)c([N+](=O)[O-])c1 C(=O)(C1CCCc2nc[nH]c21)N1CCCN(C(c2[nH]ccc2C2CC2)=O)CC1CO CC1CC(NC(N2CCN(CC(=O)N(C)CCSc3cccs3)CC2)=O)CCO1 c1(COC)ncsc1C(=O)NC(C)CCCNC(c1cn[nH]c1)=O C=Cc1cncc(C(=O)NC2(C(=O)NC3CC(O)C3O)CC2(C)C)c1 N12CCCC(C1)n1cc(cn1)C2=O.c1(C(=O)OCC)cnc(C)n1CCOC c1(OC)cc(C(=O)NC2CC(F)(CNC(=O)C(C)n3cccn3)C2)ccc1C N1(C(CN(C)C(N)=O)=O)CCC(C2(NC(C3CN(CP(C)(C)=O)C3)=O)CC2)C1 C#CC1CN(C(C23CCCCC2C3(F)F)=O)CCN1C(c1nc(CC)oc1C)=O CC1C(NC(C2CCS(=O)CC2)=O)CCCN1C(C1CC2C=CC1C2)=O CCCC(C(=O)N1CC(CS(C)=O)C1)NC(c1cnn(C)c1Cl)=O C1(C(C)C)CCc2sc(C(N3CCOC(CNC(=O)C(F)F)C3)=O)cc2C1 C(CNC(=O)CCCN1C(=O)CNC1=O)(C(C)C(C)C)NC(c1cnc(C)o1)=O C(=O)(C1Cc2ccccc21)NC(C(CC)C)C(=O)NC.C1(=O)C(C)(C)O1 c1(CN2CCC=C(C(=O)NCCOCCSC)C2)ccc2oc(O)nc2c1 c1(C(=O)NCC(C)NC(C2(CCO)CC2)=O)cn(C)nc1C1CCOC1 c1(C(=O)NC(C(=O)NCCc2onc(C)n2)C2CCC2)ncnc(C)c1C N1(CC)CCCC1CNC(=O)CNC(=O)CNC(=O)CC1OCCCO1 C1(N(C(=O)C2=CCCS2)C(=O)CC(=O)OCC)CCCN(CCC(C)C)C1 CCC(C)CC(C)C(=O)NCC#CC(=O)NCc1nnn(C)n1 C(=O)(C1CCCc2ncnn21)N1CC(N(C(C2=C(C)OCCC2)=O)C)C2(C1)CC2 CCCCS(=O)(=O)NCC(=O)NC1(CO)CN(C(=O)C(c2cncnc2)C)C1 c1(C(=O)OCC)cccc([N+](=O)[O-])c1NCC(N1CC2C(CC(=O)OC)(C2)C1)=O N1(C(C2CC(C(=O)OC)C2)=O)CCC2CN(C(c3c(O)nnc(C)c3C)=O)CC12 N1(CCNS(CC)(=O)=O)CCC(C)(NC(C2CCC(c3ccccc3)C2)=O)CC1 c1(C(N(C2CC(OCC)C2)C)=O)cnc(CNC(c2cc(O)cs2)=O)nc1 C(C(C)(C)O)(C1CC1)NC(CCN(C(C=CC)=O)C)=O C1(NC(c2[nH]cc(C)c2)=O)CC2(C1)CC(CNC(C1CC3CC3C1)=O)C2 C(=O)(CCCC(C)CC)NC(CCC#C)C(=O)N1CCC(C)(CC)C1 c1(C(=O)NCC2CN(C(C(C(CC)CC)C)=O)C3C2C3)[nH]c2ccccc2c1Cl C12(NC(c3c(CC)onc3)=O)CCC(C(=O)NC3CCCC(COC)C3)(CC1)C2 N1(C2N(C)C(=O)NC2)CCN2CCOCC2(CO)C1 C1(NC(CCCOC)=O)CCN(C(=O)CCN2CCCCC2=O)CC1F C(CC)(CCCO)NC(CC1(NC(CCOCCC)=O)CCC1)=O N1(C(C(n2cc(C(C)(C)OC)nn2)C)=O)CC(=O)CC(C)C1 Cc1cccc2c(C(=O)NCCC(O)CNC(C3CC(O)CN3C)=O)n[nH]c12 C12(CNC(c3ncn(CC)c3)=O)CCC(CN1C(C1CCN(C(=O)NC)CC1)=O)C2 NS(=O)(=O)c1cc(Br)ccc1NC(=O)CCCC(F)F N1(C(c2ccc(C#C)cc2F)=O)CC(NC(C2CC2(C)C)=O)CC12CCCCC2 c1(OC)cc(C(=O)NCC2C=CCN2C(c2cnn(CCO)c2)=O)cc(F)c1F O(NC(=O)C(O)Cc1ccccc1Br)CCC1CN(C(=O)OC(C)(C)C)C1 CC1(C(N2CCC(C(CO)NC(=O)CC3CC3)CC2)=O)CCNC(=O)C1 N1(CC)N=C(C(=O)N2CCN(C(C3CC3c3cccs3)=O)CC2)CCC1=O N1(C(c2c(C)coc2C)=O)CCC2(C1)CN(C(=O)CCc1cnccn1)CCO2 C(C)(N=c1nc2c(cnn2C)c(NC23CCC(CO)(CC2)C3)[nH]1)c1cc(C)on1 N1(C(c2ccc(C#N)[nH]2)=O)CCC2(CC(NC(c3cccnc3O)=O)CO2)C1 c1(C(=O)NCC2(CNC(C3CN4CCC3C4)=O)CCCC2)cnc2n1CCOC2 c1(CC)nccnc1C(=O)NCC1CCC1NC(=O)C(c1ccccc1)SC Cc1noc(C)c1CC(=O)N(C(C)(C)CN(C(=O)C(C)SC(F)(F)F)C)CCO C(CC(C)C)(C(C)NC(Cc1ccc(C)cc1)C(C)C)OC N(C1CCc2ccccc21)(CC(=O)OC(c1ccc2nc(O)oc2c1)=O)CC c1(SC)cc(C(N2CCC(CO)C(NC(C3(C#N)CCCC3)=O)C2)=O)ccc1F C(=O)(C(C)(C)C(O)C(C)C)N1CCC2CN(C(CCCCCOCC)=O)C2C1 C1(F)(C(C2CCC2)NC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)C#CC(C)C)C1 c1(SC)ncc(C(N2CC(O)CC2CNC(=O)COC(F)(F)C(F)(F)F)=O)cn1 c1(C(N2C(C)CC(CC(=O)N(CCCC(=O)OC)C)C2)=O)cnc(O)c(C)c1 N1(C(C(CC(C)C)O)=O)CCC2CN(C(C3CCc4nncn4C3)=O)CC12 C1(NC(c2cccc(COC)c2)=O)CS(=O)(=O)CC1NC(c1cnn(CC)c1)=O C1(CC(=O)N(CCNC(CSC)=O)CC2CCC2O)CCC(O)C1 C1C(n2cc(CSC)nn2)C(=O)c2cn(nn2)SCCC(O)CN1.CCSCC n1(C2CCN(C(c3c(C(N4CCC(C)C4CO)=O)cco3)=O)C2)ccc(O)nc1=O c1(C(C)C)ccc(C(=O)NC2(C)CC(NC(C3(O)CCC3)=O)C2)cc1.C1C(=O)N1 c1(CCC)[nH]ccc1C(=O)NCC1(O)CC(NC(=O)CNC2CC(CC)C2)C1 c1(C(N2CCCCC(CNC(CN(C)CC)=O)C2)=O)nc2ccccc2nc1C C1(NC(C2(C)C(C)C2)=O)CN(C(=O)CCc2ccnc(Br)c2)C(C)(C)C1 N1(CCCNC(=O)NCC2C3COCC23)CCc2ccccc2C1 Cc1cc(Cl)c(F)cc1NC(=O)CN1CCOCC1.C12CC1C(=O)N2 C1(O)(C(=O)NCc2scc(CNC(Cc3ccn(CC)n3)=O)n2)CCOCC1 c1(N(C)CC2CCOC2C)cc(C)c(S(=O)(=O)NCC2CC(CC)C2)cn1 C1(C(N2CC(C(=O)OC)(OC)C2)=O)CCN(S(=O)(=O)C(F)(F)F)CC1 S(=O)(=O)(c1cn(C)cn1)NCC(N1CC(CNC(C2(C#C)CCC2)=O)C(C)C1)=O Cc1ccncc1C(=O)NCc1cnn(C)c1C(N1CCC(C(C)(C)O)C1)=O C1(NC(C2(CO)CC(NC(c3cccc(O)c3F)=O)C2)=O)CCN2CCC1C2 S(=O)(=O)(c1ccc(C)c(C)c1)n1c(-c2cc(C(N3CCCCC3)=O)[nH]n2)ncc1.CS N1(C(C2(OCC)CCC2)=O)CC2CC2(NC(c2ccc(CN3CCCC3)o2)=O)C1 CCC(C(=O)NCCCCCn1cc(-c2nccn2C)nn1)NC(N)=O O=C1Cc2cc(C(=O)N(CCCNC(c3cnccn3)=O)CCO)ccc2CN1 N1(C(c2c(CC)cccc2)=O)CCCCC(NC(=O)C(C)N(C)C(C)=O)CC1 c1(NC(C23C(CN(C(c4ncn(C)c4)=O)C2)CC3)=O)cccc(F)c1C#N c1(OC)ccc(C)c(C(=O)NCC(CO)NC(C2COCC2(C)C)=O)n1 Cc1cnccc1CN(C(=O)C(Cn1ccnn1)NC(=O)CN1CCOC1=O)C C1(OC)CCC(C)(C(N2CC(O)(CNC(=O)C(=O)N(C)C)C2)=O)CC1 N1(C(c2cccc(I)c2)C(=O)NCCC(=O)OCC)CCOCC2(CCC2)C1 c1(C(=O)NC2CCN(C(C(C(C)C)n3cc(C)nc3)=O)C2)ccnc2cc[nH]c12 N1(C(C=CC(=O)OCC)=O)CCN(C(c2ncc(F)cc2F)=O)C(C#N)C1 N1(C(c2ncn(C)n2)=O)CCC(C)(C)C1CNC(=O)CN1C(=O)CCC1=O n1(C(C)C)ncc(C(=O)N(C2CCCC2)CCNC(c2coc(Cl)c2)=O)n1 n1(Cc2ccc(C)cc2)cc(Br)c(=NC(=O)Nc2cc(F)c(I)c(F)c2)[nH]1 C(=O)(C#CC1CCCCC1)N1C(C)CCN(C(=O)Cn2nc(Cl)ccc2=O)CC1 c1(Cn2c(C(=O)NC3C(CNC(C4(CC)CCC4)=O)C3)cnn2)ccc(Cl)cc1 C1(NC(C2N(C(=O)OC)CCC2)=O)CCC(C)N(C(=O)C2=CCCCC2)C1 N1(C(c2n(CC)ncn2)=O)CC(C)CN(C(C2CC(CF)C2)=O)C(C)C1 c1(C(C(=O)NC2CCC2)N(C)Cc2c(Cl)cccc2Cl)nc2c([nH]1)CCCC2 N1(C(C(C)CC(F)F)=O)CC2CC(C1)CN(C(=O)C=Cc1cccc(CO)c1)C2 c1(CCC)noc(CCCC(=O)NCC2COC(CNC(=O)CCOC)C2)n1 CC1(C)CC(CC(N2CC(CO)(NC(c3cnc[nH]3)=O)C2)=O)CO1 C1(C(=O)NCCNC(C)=O)CCC=CC1NC(=O)COC1CCCOC1 n1(CC)ncc2cc(C(N3CC4CCC3CN4C(c3cc[nH]c3)=O)=O)c(C)nc12 N1(C(CCCC)=O)CCCC(NC(c2cnc(C(C)(C)C)[nH]2)=O)CC1 N1(C(C(C)=C(C)C)=O)CCc2sc(CNC(c3nc(C)ccc3F)=O)nc2C1 N1(C(C2(C)CCCC2)=O)CC2CCC(C1)C(NC(C1CCCC(F)C1)=O)C2 C(Cc1ccccc1)(C(=O)NNC(=O)OCC1CC1)N(C)C(=O)OC(C)(C)C C(=O)(CCCCCC(C)O)N1CCC(NC(c2cc(OC)c(C)cc2)=O)(CF)C1 CC1CN(C(c2cccnc2SC(F)F)=O)CCC1CNC(c1csnc1Cl)=O Cc1cc(C)c(CC(N2CC(O)CC2CNC(c2coc(C(F)(F)F)c2)=O)=O)s1 c1(OCC#C)ncccc1C(=O)NCC(CO)NC(=O)C(C)CC=C C(CC(C)C(=O)NC(CC1CC1)CC(=O)NC1CC(Cl)(Cl)C1)OC N1(C(C=C(CC)C)=O)CC2(CCCC(CNC(=O)CCSc3n[nH]c(C)n3)O2)C1 C1(N(C(C(C)SC)=O)CC2CC2)CCN(C(C2(C3CC3)CCC2)=O)CC1 N1(C(C(CCNC(=O)C=Cc2ccco2)OC)=O)CCN(C)CC1C N1(C(Cc2c(C)cccc2)=O)CC2CCN(C(C3CCOCC3(C)C)=O)CC12 c1(OC)cccc(I)c1C(N1CC2(CC(NC(c3ncnn3C)=O)C2)C1)=O N1(CC(=O)N(CCC(C)NC(=O)C=C2CCC2)C)CCCC(C(F)(F)F)C1=O c1(C(N(C(C=C)C)Cc2ccccc2)=O)cccc(-c2cncn2C)c1 C1(Cn2cc(CCNC(C)=O)nn2)CCCN(C(=O)CCCc2nc(C)cs2)C1 c1(CC(=O)NCC(C)(C2CC2)NC(=O)C=C2CCCC2)c(F)cncc1Cl C1(NC(c2n[nH]c(C)c2C)=O)CCCCCC1NC(=O)CN1CCCC1CO c1(C(=O)NC2CCCCN(C(Cc3c(C)nc(C)s3)=O)C2)cccc(N=[N+]=[N-])c1 N1(CCNC(C2C(C(=O)OC)CC2)=O)CCN(C(C2(CO)CCCO2)=O)CC1 N1(CCC)CC2CCC(C1)N2Cc1ccc(O)cc1 C1(C(CNC(C=C(C)C(C)(C)C)=O)C)CCN(C(C2(CF)COC2)=O)CC1 CC(C)CC(O)C(=O)N1CCC(NC(=O)Cc2ncn3c2CCC3)C12CC2 c1(C(=O)NCCN2CCCCC(C(C)(C)O)C2)ncc([N+](=O)[O-])cc1Cl C1(NC(C2N(CC)CCC2)=O)CCOCC1NC(=O)CCC(F)F Cc1cc(C(C)N(C(=O)C=CCNC(C2CCNC2=O)=O)C)no1 c1(C(N2CC(COC)(NC(=O)CC3C=CCC3)C2)=O)nnn(C2CC2)c1C N1(C(C23C(CN(C(C(C)CBr)=O)C2)CC3)=O)CCc2sccc2C1 c1(C(N2CCC(CCNC(c3cncc(C(C)=O)c3)=O)C2)=O)ccc(N)cc1F CCCCC(C)C(=O)N1CCC(C(CO)NC(=O)CCC2CCCC2)CC1 CCC(C)CCC(=O)NC1CN(C(=O)Cc2cc(C(C)C)no2)CC1O C=CCCCC(C(=O)N1CCCC(CCF)C1)NC(c1n[nH]cc1C#C)=O C1(NC(Cc2n(C)ccn2)=O)C2CCCCN(C(C3CCCCCC3)=O)C12 c1(OC)cc(C)c2cc(C(=O)NCC3(NC(=O)CC=C(C)C)CCOC3)[nH]c2c1 CCCCCCCCC(=O)N1CCC(O)C(NC(=O)CSS(C)(=O)=O)C1 C1(NC(c2c(OC)csc2)=O)COC2C(NC(c3ccnc(C)c3C)=O)COC12 c1(C(=O)NC(C)CN(C(=O)CC2(Oc3ccc(F)cc3)CC2)C)ccccc1Cl C1(CNC(C(COC)SC)=O)COCCN(C(=O)COc2ccccc2C#N)C1 CC1CC(CNC(=O)CC(C)(C)c2ccccc2)CCN1C(c1nccn1C)=O C(=O)(CC=C(Cl)Cl)NCC(C(=O)N(C)CC1CCSC1)N(C)C C1(C(N2CC(F)(CC#N)C2)=O)CC2(CCSCC2)CN1 N1(C(C(C)NC=O)=O)CC2CCN(C(c3ccc(I)cc3)=O)C2C1 C1(NC(CCCCCSC)=O)CCCC12CN(C(=O)C(C)OCC1CCCO1)C2 CC1(C)CCN(C(c2cnc(Cl)cn2)=O)CC1CNC(c1cccc(Cl)c1)=O N1(C(CC(=O)NC)=O)CCCCC1CCCNC(c1cn(C(C)(C)C)nc1C)=O C1(CNC(CCn2cc(CC3N(C)CCN(C)C3)nn2)=O)CCc2nncn2C1 C(CN=c1[nH]cnc(Cl)c1F)C(C1(C2CCCO2)CC1)=O CCCCC(C)NC(=O)CCC1CCN(C(=O)COC2CCC2)C1.OCC C(=O)(CC(C)C(F)(F)F)N1C(C(N2CC(=C)C2)=O)CCCCC1 c1(C(=O)NCC2CCCN(C(CC3CCC(C)C3)=O)C2)cc(O)cc(C#N)c1 N1(C(C2CC(C)(CC)C2)=O)CCC2CCN(C(c3cc(Cl)cs3)=O)C2C1 c1(C(=O)NC(c2ccccc2)CNC(C2C(C)C2)=O)ccc(F)c2[nH]ccc12 N1(C(C(C(C)NC(=O)COC2CCC2)C)=O)CC2(CNC(=O)C2)C1 N1(C(c2cc(C)c(C3CC3)cc2)=O)CC(O)C2(CCOCC2)C1 C1(C)(CNC(=O)NC2C(NC(CSCC)=O)CCCC2)COc2ccccc2O1 c1(C(=O)NCC2(F)CCCN(C(CCC=C)=O)C2)nccn2nc(C)cc12 C(=O)(C(C)CC(F)F)N(CC(=O)NCc1cnc(COC)[nH]1)C c1(C(=O)NC(CC(C)C)CNC(=O)CC(C)(C)C2CC2)cc2c[nH]nc2s1 n1(CC)nnnc1C1CC(c2nnnn2C)N1.c1(CO)csc(SCC2CC2)n1 CC(=O)CCCC(=O)N1CCC(C)C(NC(c2c(Cl)cnn2C)=O)C1 N1(C(CCC#CC)=O)CC2CN(C(C3OCC4CCCC34)=O)CCC12 c1(C(N2CC3C(CNC(C4CC4(F)F)=O)C3C2)=O)nnc(O)c2c1CCCC2 c1(OCCC(=O)NCC2(C(=O)NC3CC(SC)C3)CCC2)ccccc1Cl c1(CC)ccc(C(=O)NCC2(NC(=O)CCc3ccc(Br)cn3)CC2)cc1 c1(C(N2CCC(n3c(C(=O)OCC)ncn3)C2)=O)cccc(C(F)(F)F)c1C c1(C(N2CC(CC=C)(C(=O)Nc3cnccc3OC)C2)=O)cn2cc(C)sc2n1 c1(C(=O)NC2CC(C)N(C(=O)Cc3cc[nH]c(=N)c3)C2)cnc2ccnn2c1O c1(C(C(=O)N(CC(C)CNC(C2CC2(C)C(F)(F)F)=O)C)F)ccccc1 N1(C(c2c(OC)csc2)=O)CCC(C)(C)C1C(=O)NCC1(C)CC(O)C1 c1(COC)nc(=N)[nH]cc1C(=O)N(CCCN(C(=O)CCCCCSC)C)C C1(C(=O)NC(C(CC)C)CO)CC12CCN(C(=O)C(c1cccc(O)c1)C)CC2 c1(C(C)C(=O)NC23CC(NC(=O)Cn4ccnn4)(C2)C3)ccc(F)c(F)c1 CC1CN(C(=O)Oc2cnncc2NC(C)(C)C)CC1(C)CO Nc1cc(C(=O)NCC2(C(=O)Nn3cc(-c4ccccc4)nn3)CC2)cc(F)c1 N1(C(c2c(OC)n[nH]c2)=O)CC(NC(=O)C(F)(F)C2CCCC2)C(O)C1 c1(OC)ccccc1S(=O)(=O)N1CCC(N(c2ccnc(C(F)(F)F)n2)C)C1 c1(C(=O)NCC2(OC)CN(C(=O)CSC(C)(C)C)C2)csc2c1CCCC2 N1(C(CCOCC(C)C)=O)CCCC(CNC(=O)C(C)SCC2CC2)CC1 C(=O)(CCCCCF)NC1CCC(C(=O)NCCNC(C2N(C)C(=O)CC2)=O)CC1 CC1CN(C(=O)CCC2(C#N)CCC2)CC(C)CN1C(c1cnc(N(C)C)o1)=O C1(C(=O)NC2C(NC(c3cc(C#N)[nH]c3)=O)C2)Cc2ccccc2C1 C1(CC(=O)NC(C)CNC(C2CCC(F)CC2)=O)CC2(CCCC2)CO1 N1(C(CCCCC=C)=O)CC2CC(C)N(C(=O)CCc3cnc[nH]3)C2C1 C(=O)(C(CO)C(F)(F)F)N1C(Cn2cc(CCCCC)nn2)C=CC1 CC1(C)C(C(N2CCCC(NC(c3coc(Br)c3)=O)C2)=O)C1(C)C N1(C(N(C)C)=O)CCC2(CC1)CC2(C)NC(=O)CC1CCCCN1 c1(C(=O)NC2CCN(C(Cn3ncc(C)c3)=O)C2)cc2cccnn2n1 C(=O)(CCC(C(C)C)NC(=O)CCNC(C)=O)NCC(=C)CC N(C1CCc2ccc(O)cc21)CC1CCN(C(=O)NC(C)(C)CC(C)(C)C)C1 C1(CN)CC12CCN(C(c1cc(C3CC3)on1)=O)C2 c1(C(c2nnnn2-c2cccc(OC)c2)NC(CC)CSC)sc(C)nc1C C1(C(=O)NCc2ccccc2)CNCC12CCCCCC2.O=C1CS(=O)(=O)N1 C(CC1CCC1)(C(=O)N(C1CN(C(=O)CCc2nc[nH]n2)C1)CCO)NC(C)=O CC1(F)CN(C(c2ccc3c(c2)CCCN3)=O)CCN(C(C23CC(F)(C2)C3)=O)C1 n1(CC(N2C(C)CN(C(c3n[nH]cc3Br)=O)CC2)=O)cc2ccccc2n1 C1(C(N2CCC(C)(CNC(=O)Cc3ncccc3C)C2)=O)(COC)CCOCC1 c1(NC(C(Cc2ccoc2)NC(c2c[nH]c(=N)o2)=O)=O)ccc(C2CC2)cc1 C1(CC(=O)NC2CC(N(C(=O)CC3C=CCCC3)C)C2)CCCNC(=O)C1 c1(C(CC)O)cn(CC2CCCN2C(=O)CN2CC(N(C)C)C2)nn1 C(=O)(C(C)S(=O)(=O)C(C)C)NCC1(O)CCN(C(Cc2cc(C)sc2C)=O)C1 C1(NC(C2(CNC(C)=O)CC2)=O)COC2(CCN(Cc3ccccc3)C2)C1 N1(C(C(C)OCC#C)=O)CCC(C=C)(Nc2cccc(C)c2Br)C1 CC1CCc2cc(C(=O)NC3CC(NC(=O)C(F)n4cccn4)C3)ccc2N1 C(CC(O)CO)N(C(=O)NC(C)C(F)F)CCO C1(C(=O)NCC(n2cc(-c3cnc(C)s3)nn2)C)CCC2CCCCC2C1 Cc1cc(C(=O)N(C2CN(C(C3CC3C3CCCO3)=O)C2)C)sc1C N(C(=NCCn1cc([N+](=O)[O-])ccc1=O)N1CCC(CNC(C)(C)C)C1)CCOC CC(C)CCCC(C)C(=O)NC(C)(C)CC=CC(=O)N(C1(CO)CC1)C N1(C(CCc2cc(C)n(C)n2)=O)CCC(NC(C2CCCC2O)=O)C1(C)C C1(C(=O)NCCOCCN(C(C2C(C(=O)OC)OCC2)=O)C)CC1C1CCCC1 C1(C(=O)NC2CCCC(CNC(Cc3n(C)ncc3Cl)=O)C2)CCC(C)(C)OC1 c1(NCC(C)OC(F)F)ccc(S(=O)(=O)N2CCCC3(CCC3)C2)cc1Br N1(C(CCC(=O)NC)=O)CCC(C(N2CCC(C)(CN(C)C)C2)=O)C(O)C1 c1(C(=O)OC)ccc(S(=O)(=O)N2CCCC(C(F)(F)F)C2)s1 C1(CNC(C(CSC)OC)=O)CCCCN(C(C2(C)CCC3CC3C2)=O)C1 N1(Cc2cn(CC(=O)OCC)nn2)CCCN(C(C2CC23CCCC3)=O)CC1 N1(C(C(=O)N(c2ccc(C#N)cc2)CCS(N)(=O)=O)=O)CCc2ccc(Cl)nc2C1 C(CC(=O)NCCCSCCO)N(C(=O)CC1(C)CCC1)CC C(=O)(C1CCCc2nn(C)cc21)N(C(C)C(=O)O)C C1(O)(C(CNC(c2n(CC)nnc2)=O)C)CCN(C(=O)CCC2CC(F)(F)C2)C1 N1(C(Cc2c(C)ccs2)=O)CCC(NC(=O)CCc2nccn2C)C12CCCC2 CCC(CC(=O)N1CC=CC(C(N2CCC(CC3CC3)CC2)=O)C1)C(C)(C)C N1(C(CNC(CCC(C)C)=O)=O)CC2CC(NC(C3(O)CCSCC3)=O)C2C1 CCC(C(=O)N(C)C)(c1nnnn1CCCF)Nc1cc(OC)ns1 C(=O)(CCCCC(F)F)N1CC(COC)(NC(C2CC=C(C)CC2)=O)C1 c1(C(=O)NCC2C(NC(=O)Cc3cocn3)COC2)ncc2cc(Cl)ccn12 O=C(CC1OCCc2ccsc21)NC1c2ccc(Br)cc2CC1C(F)(F)F C1(CC(N2C(C(=O)OC)CC2)=O)CN(CC2(C(=O)OC)CCC2)CCO1 N1(C(C2CC(C)(C(=O)OC)C2)=O)CCN(C(c2cccc(=O)o2)=O)C(C)C1C C1(NC(c2ccnc(S)c2)=O)CCN(C(c2occc2-c2cnn(C)c2)=O)CC1 Cn1cc2cc(C(N3CCSCC3C(=O)Nc3cnccc3Br)=O)ccc2n1 CC1(C)CN(C(=O)CSCC(N)=O)CC(CNC(c2cc(C(F)F)ncn2)=O)O1 C12(CNC(=O)CCN3CCCC3)CC1CN(C(=O)C(Cc1cccc(Cl)c1)=NO)C2 N1(C(Cc2c(CC)con2)=O)CCC(CC)(NC(=O)CC2CCC(F)(F)C2)CC1 C1(NC(c2cncc(C(F)F)c2)=O)C2CCC1N(C(c1cc(C3CC3)ns1)=O)C2 c1(C(N(C)Cc2cc(OC)ns2)=O)ccc(S(=N)(=O)N(C)C)cc1 c1(C(N2CC(CNC(c3ccc(F)c(F)c3)=O)C2)=O)ccc2c(c1)COCO2 O=C(O)CCC(C(=O)O)NC(c1ccc(Cl)c(F)c1F)=O N1(CC(=O)NCCN(C)C(c2csc3cncn23)=O)CCC(=O)NC1=O C#Cc1ccc(C)c(NC(C2CCCN(C(=O)CC3CCC(=O)N3)CC2)=O)c1 N1(C(=O)NCCO)CCCC(Cc2cn(C3CCN(C(F)F)CC3)nn2)C1 CC(C)CN=C(NCC12CCC(CC1)C2)N1CC2CC(C1)c1cccc(=O)n1C2 C1(CCNC(C2(C)CCCC2)=O)CCCN(C(C2(CF)CC(F)(F)C2)=O)C1 c1(C(=O)NCC(C2CC2)NC(C(c2c(C)n[nH]c2C)C)=O)cnn2cnnc2c1 Cc1nc(O)nc(C)c1CC(=O)NC1CCCC1NC(C1CC12CCCCC2)=O CC1CCCN(C(=O)C(=O)NCC2(N(C(=O)Cn3cnc(=N)[nH]3)C3CC3)CC2)C1 c1(N(CCS(=O)(=O)NC)C)nc(N2CCC3(CC(OC)C3)C2)c2ccsc2n1 N1(C(C(=O)NCCNC2CCOCC2)C2CCC2)CCc2ccccc21 C1(C(N(CCC(C)(C)NC(c2ccnnc2O)=O)C)=O)C2Cc3ccccc3C12 C1(CN(c2ccc(C(N)=O)[nH]2)C)CN(C(C2CCCN(C(N)=O)C2)=O)CCO1 c1(C2C(=O)NCCCC(C)O2)cccc(Cl)c1.C(C(=O)NCC(=O)NC)OC C1(CNC(Cc2c(C)cccc2)=O)CCC2(CO1)CC(NC(=O)CC1CC1)C2 C12COCCN1C2=O.C1(CC)CC(NC(=O)CCC(=O)NC2CC2)C(O)C1 c1(C(C)(C)C#N)cc(C(=O)O)cc(CN2CCOCC2)c1 Cn1ncc(I)c1NC(c1nc(C(C)(C)C)c(Br)s1)=O c12nc3ccc(cc3[nH]1)N2.C1(c2nnnn2CCC2CC2)(OC)CC(CSC)C1 N1(Cc2ccc(OC)nc2)CCC2(CC1)CC2C(=O)Nc1ccns1 N1(C(c2cc(C)cc(N)c2)=O)CC2CN(C(=O)CCC3CCN(C)CC3)CC2C1 C=C(F)C1(CC(N2CCC2CNC(=O)Cc2ccc(O)c(Cl)c2)=O)CCOCC1 CC(C)(C)C(CO)C(=O)N1CCCC(NC(=O)Cc2nc([N+](=O)[O-])n[nH]2)CC1 N1(C(C2C(C)C(=O)C2)=O)CCC(C)(NC(c2cc(C(F)F)ncn2)=O)C1 c1(C(C(=O)NCC=C)N(C(C)C(=O)OC)C)c[nH]c2ccc(OC(C)C)cc12 N1(C(Cc2c(Cl)cn(C)n2)=O)CCC(NC(C2COC(=O)N2)=O)C2(CCC2)C1 c1(CNC(CC(C)C)=O)ncccc1C(=O)NCc1cnn(CCO)c1 N1(C(C)=O)CCOCC(F)(NCCNC(=O)CCCCC(N)=O)C1 CC1(C)CCC(CCN2CCOC(C3CN(C(=O)N(C)C)C3)C2)CC1 Cc1ncoc1C(=O)NCC(C1CC1)NC(=O)CC1CCN(C)C1 CCC(C(=O)N(CCC(=O)NC)C)NC(=O)C(C)CO N1(C(C(C2CCN(C(C3CN(C(C)=O)C3)=O)C2)(C)C)=O)CCn2cncc2C1 C1(CC(=O)OC)C(=O)NCCN1C(=O)NCC1(CN(C)C)CCCCC1 S(=O)(=O)(c1cc(Cl)ccc1Cl)N1C2CC(N3CCN(CC=C)C(=O)C3)C(C2)C1 N1(C(CCCN(C)C)=O)CCCC(CN(C(=O)C(c2ccccc2)=O)C)C1 C1(C(N2CC(OCC)C2)=O)CCN(C(c2ocnc2C2CC2)=O)CCO1 N1(C(CCC(C)OCC)=O)CCC(C)(C(=O)NC(C(O)CO)C2CC2)CC1 c1(C(=O)NCC(CN(C)C(C23CCCC2CCC3)=O)O)c(O)cc(F)cc1F N1(C(c2ccc(C)o2)=O)CC2CCCC2(NC(=O)CSCc2ccccn2)C1 C(=O)(CCS(N)(=O)=O)NC1CCN(C(Cc2c(C)noc2)=O)C1C(C)C c1(C(N2CC(CCC)C(C(=O)NCc3cnccc3C)C2)=O)ncc(F)cc1F N1(C(C23CCC(OC)(CC2)C3)=O)CCN(C(=O)CN2CCOCC2=O)CCC1C CSC1=C(C(=O)N2CCC(CNC(=O)C(F)F)C(C)C2)CCCC1 N1(C(CC2CC(CC)C2)=O)C2CCC1CN(C(=O)COc1ccc(F)cc1O)C2 c1(NC(c2cccc(C)c2F)c2n(CCC)nnn2)cc([N+](=O)[O-])c(C)cc1C c1(C(=O)NCCCOCCNC(C(C)SC)=O)cnc(C(F)F)nc1 c1(C(N(CC(CN(C(=O)C(F)n2ccnc2)C)O)C)=O)cc2cc(Cl)ccc2[nH]1 C1(C(=O)NCC2(O)CCN(C(c3cnc(N)c(Cl)c3)=O)C2)CCc2ncnn2C1 N1(C(C(=O)NC(CC)(C)C)c2cnc[nH]2)CC=C(C(=O)OC)C1 C(=O)(CCCS(=O)(=O)N1CCCC1)NCc1c(Cn2cc(COC)nn2)cccc1 c1(C(N(C)CC2CN(c3nc(OC)c(Br)cn3)C2)=O)cc(Cl)c(F)cc1F C(=O)(CCCCCC(=O)NCC1CCN(C(C2CCC2C)=O)CC1)OCC C1(NC(CC=CCC)=O)CC2CCC1CN(C(c1cc3c(ncn3C)[nH]1)=O)C2 N1(CC)CC(CNC(C2CCCC(CNC(C3CCCCC3O)=O)C2)=O)OC1=O c1(C(N(c2ccccc2F)CCC(=O)OC)=O)cnc(O)c(Br)c1C C=CCC(CC(C)C)C(=O)NC1CCN(c2cc3nncn3cn2)C1 C1(C(=O)NC(C)C(C)(C)C)CC(F)CN1C(=O)OC(C)(C)C C1(=O)C(C)(C2CCC2)N1.N1(CC(=O)NC(C(C2CC2)OC)C)CCSCC1 CC(C)C(O)C(=O)N(C1CCCC1)CCCNC(=O)Cc1cnccn1 n1(C(C)C)cccc1C(=O)NCC1CC1CC(=O)NCC(C)(C)CC1CC1 C1(C(=O)NC2C(C(C(=O)N(CC=C)C)(C)C)CCCC2)OCCCC1(C)C c1(C(=O)NCC(C)NC(c2cc(-c3ccccc3)no2)=O)cc(O)c(F)cc1N c1(CCC)[nH]ccc1C(=O)N(CC(C)NC(=O)CNC(c1ccsc1)=O)CC C1(C)(C(=O)NCCCC(C)(C)OC)CC(O)CN1C(C1CC(N=[N+]=[N-])C1)=O N1(C(c2c(C)occ2)=O)CC(NC(=O)C(C)(O)C(C)C)CC(F)C1 C1(c2n(-c3c(CC)cccc3)nnn2)(NCCOC2CCOC2)CCN(C)CC1 CCC(C)C(O)C(=O)N1CCC(CNC(=O)COc2c(C)ncnc2C)C1(C)C N1(C(C2(CC)CCCO2)=O)CCC(C(N2CC(O)(COC)C2)=O)CC1 c1(C(=O)NC2CCCC(NC(c3cccnc3S)=O)C2)ccc2oc(S)nc2c1 N1(C(c2cn(C(COCC)C)nc2)=O)CCC(C)(C(=O)Nc2cncnc2)CC1 C12(C(N(C(c3ccccn3)CC)C)=O)CC(CO1)N(C(=O)OC(C)(C)C)C2 Cn1nc(C(N2CC(OCC(=O)NC3CCC(CO)C3)C2)=O)cc1C1CC1 C1(C(=O)NCC2CCN2C(=O)Cc2cc(Br)cs2)CC2(CCC2O)C1 Cc1csc(C(C)C(=O)NCCN(C2CCCC2)C(=O)Cn2cncn2)n1 c1(C(=O)NC2CN(C(CCC(=C)Cl)=O)C(CO)C2)cc(F)c(F)cc1Br C(C(N=[N+]=[N-])C(=O)NCC1CCCC1NC(c1ccc(=N)[nH]c1Cl)=O)OCC c1(C(N2C(C)CN(C(=O)C#CC3CCC3)C(C)C2)=O)ccnc2cc(Cl)ccc12 N1(c2n(CC(=O)N(CC)CC)c(C(C)C)nn2)CCS(=O)(=O)C(C)C1 C1(CC)CN(C(N2CC(OC(C)(C)C)C(C)(C)C2)=O)c2ccccc2O1 N1(C(c2ccncc2Br)=O)CC2CCC(C1)N2C(=O)Cc1ccncc1 c1(C(N2CCN(C(c3cncc(OC)c3)=O)CC2)=O)ccc2ncsc2c1 c1(OCCO)ccc2c(c1)CN(c1ncnc(Cl)c1F)C2 N1(C(c2cccc(Cl)c2)C(=O)NCCCC2CC2)Cc2ncsc2C1 C1(O)(CC(=O)N(C(CNC(CSc2n(C(C)C)cnn2)=O)C)C)CCCCC1 C(=O)(C(O)C1=CCCCC1)NCc1ccc(CN(C(CCC(C)C)=O)C)cc1 N1(C(C(C)=C(CC)C)=O)CC(C)(C)OCC1CNC(C1CCCC(F)(F)C1)=O O(NC(=O)N(CC(=O)OC)CC)C(C=C)C C1(C(=O)NC2(c3nnnn3Cc3cc(Cl)ccc3F)CCN(C)C2)CCC2(CCC2)C1 C1(CNC(C(F)=CCC)=O)CC(NC(C2CN(CC(F)(F)F)C2)=O)C12CCC2 C1(C(=O)NC)CCN(c2cc(NCCO)ncn2)CC1.C12CCN(C1)C2=O N1(C(C23CCN(C(CNC(=O)OCC)=O)C2CCC3)=O)CCC(O)CC(C)(C)C1 Cc1c(C(=O)NC(C)CNC(=O)C(N2CCCCC2=O)C)c(Cl)nn1C C1(C(=O)NCC2(C(=O)NCC3CCC3(F)F)CC(=C)C2)CCCOCC1 C(=O)(CCCC(C)(C)NC(=O)C(CC1CC1)OC)NC(CC)CCCO c1(OC)nc(C(=O)NCC(C2CCCCC2)NC(=O)CC(C)(C)O)cc(O)n1 N1(C(CN)=O)CCC2(CC2C(=O)Nc2cccc(O)c2Cl)C1 N1(C(C2N(C(CC3CC(=O)C3)=O)CC(O)C2)=O)CC2CCC(O)C2C1 Cc1cccc(C(=O)NCCNC(=O)Cc2cccnc2O)c1 c1(C(N2CC3C(CNC(c4cocn4)=O)C3C2)=O)ccc(F)cc1OC(F)F C(=O)(CC(C)C(F)F)N1CC(NC(CCN(CC)CC)=O)C(C)C1 C1(NC(c2c(OC)cccc2F)=O)CCOC2(CCN(C(=O)CC3CC3)CC2)C1 c1(OC)ccc(NCc2csc(-c3ncc[nH]3)n2)cc1NC(=O)C(F)(F)F C1(CCNC(c2nccc(CC)c2)=O)C(C)CCCN1C(=O)C=CBr Cc1ccc2c(=O)c(C(=O)NC3C4CN(C(=O)C(O)CC(C)C)CC34)c[nH]c2c1 N#Cc1cc(C(=O)NCCn2cc(C(=O)NCCC(O)CO)nn2)cs1 Cc1cncc(C(=O)NC2CCCC2NC(=O)C(O)CCN(C)C)c1C C1(c2ccccc2)(NC(C(C)N(CCC2CCCC2=O)C2CC2)=O)CC1(C)C N1(C(C(COC)C)=O)CCC(C)(C)C1CC(=O)Nc1ccc(Cl)c(OC)c1 c1(C(=O)NCCN(C(=O)CCCCC(C)C)CC)ccc2c(c1)C(=O)OC2 C1(NC(=O)CSc2ccccc2)CC2(C1)CN(C(c1ccc(Cl)c(Cl)n1)=O)C2 C1(C(N(CCNC(c2ccc(NC(C)C)cc2)=O)C)=O)COC(C)(C)CO1 C1(C2CCCN(C(C3(N4CCCC4)CCC3)=O)C2)(NC(c2c(C)nsc2C)=O)CC1 C1(C(=O)NC(C)C(CO)NC(=O)Cc2n[nH]c(=N)s2)CCCC2(CC2)C1 c1(C(=O)NC2C(CNC(C(C)(C)c3cc[nH]n3)=O)CCC2)cccc2ccnn12 C#CC1CN(C(c2ccc(F)cc2F)=O)CCN1C(=O)CCOCCCN=[N+]=[N-] N1(C(Cc2c(C)ocn2)=O)CCC2CN(C(=O)C(C)C3=CCCC3)C2C1 N1(C(c2c(CC=C)cccc2)=O)CC2(CCCC2)C1C(=O)NCC1CC=CCC1 C(C(Cc1ccccc1)CC(C)C)N1CC(NC(=O)OCC)C(C)C1 Cc1cnccc1C=CC(=O)NCC1CCC1NC(=O)C(c1cccnc1)O C1(NC(C(C)(C)c2cnsc2)=O)CC2CCC(C1F)N2C(c1cncs1)=O C(=O)(CCCN(C)N=O)N1C(C2(NC(C(COC)(C)C)=O)CC2)CCC1 C1(NC(c2cnc(Cl)s2)=O)CCOCC1NC(C1CC12CC2)=O c1(OC)ccc(CC(N2CC(NC(=O)CN3CCCC3=O)C3CC23)=O)cc1Cl N1(C(CCCN(C)N=O)=O)CCN(C(c2c[nH]c(=N)s2)=O)C2CCCCC12 CC(C)(O)C(F)C(=O)NCCOCCNC(=O)CN1CCNC(=O)C1 C(=O)(C(C)(C)C(F)F)NCCN(C(=O)CC1CCC(C)O1)CCOC C1(C(=O)NC(C2CCOC2)CC)CCC(C)N1C(c1cccnn1)=O c1(NCC(=O)NC(CNC(Cc2c(C)occ2)=O)CO)cccc(C#N)c1 c1(C(N2CC(O)(C(C)NC(C(C(C)OC)N(C)C)=O)C2)=O)c(N)cc(C)cc1F c1(C(=O)NC2CC(c3ccccc3)(NC(C(C)C)=O)C2)cc(O)cc(C#N)c1 C(=O)(CC1=CCOCC1)N1C(C(N(CC(c2nn[nH]n2)C)C)=O)CN(C)CC1 C1(NC(Cc2c(OC)cncc2)=O)CC2(CCN(C(=O)C(C)c3ccco3)C2)C1 CC(C(=O)NCCNC(c1ccc(C(F)(F)F)c(O)n1)=O)C(F)(F)C(F)F C12(NC(C(CCSC)O)=O)CCC(C1)N(C(c1ccsc1SC)=O)C2 N1(C(c2c(CC)c[nH]c2)=O)Cc2nccn2CC(NC(=O)C(C)SCCCC)C1 C(=O)(CCC(C)(C)C)NC(CNC(C(CCC)c1ccc(Cl)cc1)=O)C1CCC1 c1(C(=O)NCC2CCCCN(C(C3(C4CC4)CC3)=O)C2)noc2cc(F)ccc12 C#Cc1cccc(C(C(=O)NCCCF)N(C(c2ccccc2)CSC)C)n1 C1(NC(CCSC)=O)C2CC3C1C3C2C(N1CC(F)(F)C1C1CC1)=O C(=O)(C(C)C(O)C(C)C)N1CCC(C2N(C(c3c(C)cn(C)n3)=O)CCC2)C1 CCC(C(=O)NC(C)C(CO)NC(c1ccnc(C(C)(C)C)n1)=O)C(C)(C)CC C12(NC(CSC)=O)CCCN(C(C3CN(SC(F)(F)F)C3)=O)CC1C2 Cc1ncc(CNC(=O)C(C2CCCCC2)NC(=O)CC2CC2(C)C)s1 N1(C(c2nc(C)sc2C)=O)CC2CC(NC(c3cccc(F)c3)=O)C1C2 C1(c2n(C)ncc2)CN(C(=O)CCc2cc[nH]n2)CC1NC(c1ccsc1)=O CN1CCC(CCNC(C2CC=CCN2C(c2ccn(C)c2)=O)=O)CC1 CC1CN(C(c2ccc(-c3nn[nH]n3)cn2)=O)Cc2ccccc21 c1(C(=O)NCC(C)(C)NC(C(CC)n2cccn2)=O)ccc2snnc2c1 C12CCC(C(=O)O)N(C1)C(=O)N2.c1(N(C(C)(C)C)CC)nc2sccn2n1 C#CCCCC(=O)N1CCC(CO)(NC(c2ccc(C3CCOC3)cc2)=O)C1 c1(OC)cccc(C)c1C(C(=O)NC1CC(F)(F)C1)N(C)Cc1cc(C)ccn1 C(=O)(C1Cc2ccc(Cl)cc21)N(C(c1ccc(S(C)=O)cc1)C)CC1CCC1 C(=O)(CCC(C)(C)F)N1C(CNC(C2C(OC)CCC2)=O)C(C)CC1 C1(CCC)CN(C(=O)CCCNC(C)=O)CCN1C(C1CC(=C(F)F)C1)=O N1(C(c2cnc(OCC)s2)=O)CCN(C(=O)CCc2ccon2)C(C2CC2)C1 N1(C(Cc2c(C)noc2)=O)CCC(NC(=O)CC(F)F)C(F)(F)CC1 N1(C(c2ccc(=O)n(C)c2)C(=O)NC)CCC2CCC(O)CC2C1 c1(C(=O)NC(C(CO)NC(C(CO)N(C)C)=O)C)nn(CC(F)(F)F)cc1Cl c1(C(N(CCC(C(C)C)NC(C2CCC(F)C2)=O)C)=O)ccc2nc(O)[nH]c2c1 C(=O)(CCCC(=O)N(C)CCN(C)C(c1cnc(CC(C)C)[nH]1)=O)OCC N1(C(Cc2c(C)c(Cl)ccc2)=O)CCN(C(=O)COC(F)(F)F)C2CCCC12 c12cc(on1)CCC(=O)NCC(C1CCOC1)NC2=O.C1(CC)(OC)CCCC1 C1(C(=O)NCC2CCN(C(c3c(C)ocn3)=O)C2)CCc2nn[nH]c2C1 N1(C(CCCCCCSC)=O)CCC2CCC(C1)N2C(c1cccn(C)c1=O)=O c1(C(N2C(CN(C(C(COCC)C)=O)C)CCC2)=O)cnnc(C)c1C C1(NC(C(CC=C)C)=O)C2CC3C(C2)C13C(=O)N(C)Cc1cc(C)on1 N1(C(C)=O)CC2CC2(C(=O)NC2(CNC(=O)C(C)SC(F)(F)F)CCC2)C1 C1(C(N2CC3(CC(NC(c4cnn(C)c4N)=O)C3)C2)=O)CCCC2(CCC2)C1 C(=O)(C(CCO)N(C)C)NCC1(CNC(C(C)OCC2CC2)=O)CCCC1 C1(C(=O)NCC2CN(C(c3coc(Cl)n3)=O)CCO2)CCCCS1(=O)=O Cc1ncc(C(=O)NC2CC(C)N(C(c3ccc(C(C)(F)F)cc3)=O)C2)cc1N C(CCN=c1ccnc(NCC2CC(=O)N(CCOC)C2)[nH]1)N(CCC)CCC C(=O)(C(CCOC)OC)NC1C(CNC(CC(=O)NCC#C)=O)COC1 C(=O)(C1=CC2CCCCCC12)NCC1CN(C(c2c(OC)cc(C)s2)=O)C1 C(=O)(CS(C)(=O)=O)N(C1CCN(C(C2CCCN(C(=O)CC)C2)=O)CC1)CC#C c1(C(N2CCC(C(=O)NC(CO)C(C)O)(CC)CC2)=O)cc2ccccn2c1 c1(NC(=O)NC(CC)CSC)cccc(OCCN(C)C)c1 Cn1[nH]c(C(F)F)nc1=NC(=O)NCc1cccc2c1OCCO2 c1(C(N2CC(CC(C(=O)NC3CC4CC(=O)C3C4)F)C2)=O)cc2cccn2cn1 C=CCC(C)(CC)C(=O)NCCC1(O)CN(C(c2ccc(=N)[nH]n2)=O)C1 c1(C(=O)NCC(C)(CNC(=O)C(N)=O)OC)cnn(C(C)C)c1N C(N=c1[nH]c(=NCC=CBr)c2sccc2[nH]1)C1(c2ccccc2)CCC(=O)N1 C1(NC(CCC(C)NC(=O)C(O)C(F)(F)F)=O)CCCC(C)(C)C1 c1(COCC(=O)NCC(C)NC(C=CC)=O)ccccc1C CC1(C(=O)NC2CC(CNC(C3CCNC3=O)=O)C2)CCCCC1(F)F CON1CCC(C(=O)NC2(CCNC(c3cnn(CCO)c3C)=O)CCC2)CC1 c1(OC)ccc(F)cc1C(=O)NCC1(O)CCN(C(=O)C2=C(Cl)CCC2)C1 c1(OC)ccc(C(F)(F)F)nc1C(N1CC(OC)CC1CNC(=O)CCF)=O c1(C(=O)NCCC2CCCCN2C(C2COCCO2)=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(COc2ccc(SC)cc2)=O)CCC(NC(c2ccnnc2O)=O)C(F)C1 N1(C(COCC(C)C)=O)CCCC(CNC(=O)Cc2cncnc2O)CC1 Cc1coc(C(N2CCC2CNC(C2CCOC2c2cccnc2)=O)=O)c1C N1(C(c2c(SC)cn(C)n2)=O)CCC(F)(F)C(CNC(c2ncsc2C)=O)C1 S(=O)(=O)(CCCN=c1[nH]c(=NC(C)COCC)[nH]c2ccsc12)NCCCC CC1OCCC12CN(c1nccc(=NCc3ccc(C(F)F)cc3F)[nH]1)CCO2 C12(NC(c3ccc(CCC)s3)=O)CCCCCC1N(C(C1CCCCS1)=O)CC2 c1(C(=O)NC2C3CN(C(CC4ON=C(CC)C4)=O)C2CC3)nccn2nccc12 CC1CN(C(=O)C=C2CCC2)CC1CNC(=O)CSc1cccc[n+]1[O-] O=C(CS(=O)(=O)C1CCCC1)N1CCC(C2CCCN2C(c2cccnn2)=O)C1 C1(C(N2CCC(c3ccc(Br)cc3)C2)=O)CC(O)CN1C(c1cc(Cl)c(Cl)s1)=O Cc1c(C(N2CCC2CNC(C2C(Cl)(Cl)C23CC3)=O)=O)ccn1CC1CC1 c1(C(C)C)ccccc1CC(=O)NCC(C)(C1CC1)NC(c1sccc1Cl)=O CC1CC(NC(=O)Cc2ccccc2)CCN1C(=O)Cc1ccsc1 N1(C(Cc2cccc(-c3ccc(C#C)cc3)c2)=O)CCC2(CC1)CC(C(=O)O)C2 C1(CC(CC)C)CN(C(=O)CC(CC2CC2)NC(=O)CC2COCC2O)CCO1 c1(C(CC)(C)C)cccc(CC(=O)NCC2CCC(NC(=O)CS(C)(=O)=O)C2)c1 C1(C(=O)NC(C)CNC(c2ccc(C(F)F)c(F)c2)=O)CN2CCN1C(C)C2 C1(C)(CNC(CC2(CSC)CC2)=O)CCN(C(=O)CCCc2n[nH]c(=N)s2)C1 c1(CNC(C(C(C)C)O)=O)ccc2c(c1)CCN(C(C1CCCN1C(C)C)=O)C2 C1(C(=O)NCC(C2CCN(C(c3nc(C)n(C)n3)=O)CC2)O)CCC12CCCO2 N1(C(c2c(C)ncn(C)c2=O)=O)CC2COCC(C1)C2NC(=O)Cc1cccs1 C1(O)(C(C)NC(C(C)NC(=O)OC)=O)CN(C(=O)CC2CCCO2)C1 c1(C(N2CCCC(CN(C(C(CC3CC3)OC)=O)C)C2)=O)cc(C)ccc1C C1(C(N2C(C)CC(NC(C3CC(=C)C3)=O)C2)=O)CCC(C)=C(C)C1 C1(CC(=O)NCCCC(C)CO)CCN(C(c2ncc(F)cc2N)=O)C1(C)C CC1(CNC(=O)COCCCN(C)C)CCC(C(=O)NCC2COCC2CF)O1 N1(Cc2nc(=NC)[nH]c(C(F)(F)F)c2)CC2OCc3cnnn3C2C1 c1(N(C(CCC)=O)C)c(C)nc(C)n1C c1(C(=O)NC2CC(C)N(C(=O)CCC(F)F)CC2)ccc2oc(O)nc2c1 CC1=CC(C(=O)NCC(C)=CC(=O)NCCc2ncn(C)n2)SC1 N1(C(C(C)(C2(C)CC2)OC)=O)CCN(C(=O)CNC(c2ccco2)=O)C(CF)C1 C1(NC(c2cccc(N3CCCC3=O)c2)=O)(CO)CCN(C(c2ccoc2)=O)C1 C(CCCCCC(=O)NCc1cc(C2CC2)on1)NC(c1nn(CC)nc1C)=O c1(C(=O)NC(C(C(C)C)NC(CN(C(COC)=O)C)=O)C)ccc(C)cc1SC C#CC1CCC(N(CCOc2ccc(C(C)(C)C)cc2)C2CC2)C1 Cc1nc(C(N2CC(c3cccc(F)c3)CC2C)C(=O)NC2CCC2)sc1C Cc1ccc(C(=O)NCC(C2CCCN(C(=O)C(C3CC3)C3CC3)C2)(C)O)cc1 N1(C(C(C2CC2)OC)=O)CC(C)(C)OCC1CNC(c1cc(C)c(N)cn1)=O C1(C(N(C2CN(C(C(C)(C)OC(C)=O)=O)C2)C)=O)CCCC(C(N)=O)C1 c1(CC)ccccc1SCC(=O)NCC(C1CCOC1)NC(c1n[nH]c(C)n1)=O C1(C(C(=O)N(CC(C)O)CC)C)CCN(C(=O)C(N)=O)C1.C(=O)(CO)N O=C(C1=CCCS1)NC(CNC(c1cncc(F)c1)=O)C1CC1 N1(C(CCCC)C(=O)Nc2ccccc2)CC=CCC2(CCCC2)C1 c1(CNC(C2CC2NC(c2ccc(Br)s2)=O)=O)cnc(O)nc1O c1(NC(CC2(C)CN(C(C3CCC(CC)CC3)=O)C2)=O)cc(Br)c(O)cc1Br C1(C(=O)NCCOCCC#C)C(CC)CCN1C(=O)C(C1CCOCC1)F C1(CNC(CC(C=C)C)=O)CN(C(c2cn(CCC3CC3)nn2)=O)CC(C)(C)C1 c1(CNC(CNC(COCC)=O)=O)nnc2nc(C)cc(C)n12 C=C1CC2(C1)CC(C(=O)NC(CCNC(c1ccnn1C1CC1)=O)C(C)C)C2 C1(C(N(CCOCCN(C)C(c2cocn2)=O)C)=O)CC1(F)F N1(Cc2ccnc(C)n2)CCC2CN(Cc3cc(Cl)ccc3OC(F)F)CC2C1 C1(CC(=O)N(CC#C)C(C)C)(N(C)C)COC1 c1(NC(N(CCC)CC)=O)ccc(Oc2cccc(C)c2)cc1C(C)C c1(C(=O)NC(C)CN(C)C(c2cncn2C)=O)ccc2c(c1F)CCC2 C(C(C)(C)CC(=O)NC(CC1CC1)CO)NC(c1n(C(C)C)ccn1)=O c1(C(N2C(C)CC(NC(C3(C(F)F)CCCC3)=O)C2)=O)ccc(Cl)c(F)c1 c1(SCCNC(c2n(C)nnn2)CC2CCC2)cccc(Cl)c1 c1(NC(C(C(C)NC(c2cc3n(n2)CCO3)=O)(C)C)=O)ccc(O)c(=O)cc1 S(=O)(=O)(c1ccc(N(C)CCN(C)C)c(Br)c1)NCC(C)CCCO N1(C(CC2(C)CC2)=O)CC23CCCC2(C1)CN(C(C1CCCC(=O)N1)=O)C3 C=CCC(CC(C)C)C(=O)N(C1CN(C(=O)C(C)CC=Cc2ccccc2)C1)C CCC(CC(=O)NC1CCN(C(=O)Cn2ncn(C)c2=O)CC1F)C(F)F c1(-c2cc(CC(=O)NC(c3ccccc3)CO)ncc2)cc(F)c(F)c(F)c1F N1(C(CN(C(C)=O)C)=O)CC2CCC(CNC(=O)Cc3cn(C)cn3)C2C1 N1(C(Cn2c(C)ncc2[N+](=O)[O-])=O)CCCC2C1CCN2C(=O)Cc1cnsc1 C1(CNC(C=CC(C)(C)SC)=O)CN(C(=O)C(C(C)C)n2cnc(C)c2)CCO1 C1(NC(c2ncn(C(C)C)n2)=O)CN(C(=O)CCCNC(N)=O)CC(C)(C)C1 Cc1cc(C(N2CCN(C(=O)CCCn3ccnn3)C(C)C2C)=O)cc(F)c1C C(N=c1[nH]cnc2ccsc12)C1CCCCN(C(CC2(C)CC2(Cl)Cl)=O)C1 N1(C(CCCC(=O)N(CC)CC)=O)CC(NC(=O)C(O)C(C)C)C2CCCCC12 C1(C(=O)NCC2(CNC(C(C)CC3CC3)=O)CCCC2)CC(=O)N(O)C1 c1(C(=O)NCC2CC(OC)CN2C(=O)CCC2CC2)ccc(C)c2ncccc12 Cc1cn(CC(=O)NC2CC3CC(NC(=O)C(C)C(C)C)CC23)c2ccccc12 CC1CN(C(c2ccc(C(N)=O)o2)=O)CCC1NC(=O)CC(C)C1CCCO1 C1(C(=O)NC(C2CN(C(c3n[nH]c(C(C)(C)C)n3)=O)C2)C)CC=CCC1 c1(NC(C2CC(=C)CN2CCc2c(O)n[nH]c2C)=O)ccc(F)nc1F O=C(C1=C(Cl)CCC1)NCC1CCCCN(C(=O)COC2CC(F)(F)C2)C1 c1(-c2cccc(C)c2)cc(=NC(=O)CC(C)C2CC2)[nH][nH]1 c1(C(=O)NC(C)CN(C(=O)CN2CCCC2CO)C)cncc(OCC(F)F)c1 C1(CNC(=O)Cn2ncnn2)CC(F)CN1C(c1ccc(-n2cccc2)nc1)=O C1(CNC(Cc2cc(C)ns2)=O)CC2(CO1)CN(C(=O)C=C(Cl)Cl)C2 C1(CC(C)NC(c2ccc(O)nc2)=O)CCN(C(C2(C(F)F)CCCO2)=O)CC1 C1(CNC(C(C2CCOCC2)C)=O)CN(C)CCN1C(c1cnc2n1CCC2)=O Cc1ccc(F)c(C(=O)NC2CCC2NC(C2(CO)CC23CCC3)=O)c1 N1(C(c2cc(C(C)C)on2)=O)CCCCC1.n1(C)cc(CCN(C)CCO)nn1 c1(C(N2C(C)C(NC(=O)CC3CCOC3)CC2)=O)ccc2c(c1)CC2 N1(C(c2c(C(C)C)cccc2)=O)CCC2(CC1)CC2NC(C1(C)CC=CCO1)=O C1(NC(CS(=O)(=O)NC)=O)CN(C(c2cc(Cl)cnc2C)=O)C(C)(C)C1 c1(C(N2CC(CC=C)(NC(c3ccc(F)s3)=O)C2)=O)c(OC)nsc1OC c1(C(N2CC(C)C(CNC(=O)C#CC3CC3)C2)=O)cc2ccoc2cc1F C(C1c2ccccc2CC1C)Nc1cc(OC)nc(OC)n1 C12(NC(C3CC=C(C)CC3)=O)CCC(CN(C(=O)CCn3cnnn3)C1)C2 N1(C(CC(CC)SC)=O)CCN(C(c2cn(CCO)nn2)=O)C(CCO)C1 CC#CCC(C(=O)N1CCCC(C)(N(C)C)C1)NC(C1CN2CCN1CC2)=O c1(NC(C2N(C(C(CCCC)O)=O)CC(O)C2)=O)ccnc(S(C)(=O)=O)c1 CCC(C)(CCC(C)C)C(=O)NC1CCN(C(=O)CC2(O)CCOCC2)CC1C C1(C2CCN(C(C3CC3[N+](=O)[O-])=O)C2)(NC(=O)C=CC2CCCCCC2)CC1 N1(C(c2c(OC)ncnc2C)=O)CCN(C(=O)Cc2c(C)noc2C)CC12CC2 Cc1ccc(C(=O)NCC=CCNC(=O)CC(C)N(C)C)c(F)c1C C1(c2cn(C3CCC(C(=O)N(C4CCC4)CC4CCC4)C3)nn2)(OC)CCCCC1 c1(C(=O)NCCC(C(C)C)NC(=O)C2=NOC(C)C2C)ccc(S(N)(=O)=O)cn1 C1(NC(c2c(CC)nc[nH]2)=O)CCOC12CCN(C(C1CCCOCC1)=O)CC2 N1(c2sc(C#N)c(Cl)n2)Cc2ccccc2C(CNC(c2cnc(Cl)cn2)=O)C1 Cc1cc(C(=O)NCC2C(O)C(O)CN2C(C2CCS(=O)(=O)C2)=O)cc(F)c1 N1(C(C2C(C)(NC(C3CC(C)(O)C3)=O)CCCC2)=O)CCC2CC1C(=O)O2 C1(C(=O)NC(C2OCCN(C(c3ncc(OC)cn3)=O)C2)C)CNC(=O)CC1C CC1CN(C(c2ncccc2Br)=O)CCC1CNC(C1(C#N)CCCC1)=O c1(C(=O)OC)cccc(C(N2CCCC2C(C)NC(=O)C(C)COC)=O)c1O Nc1cc(Cl)nnc1C(N1CCC(O)(CNC(c2c[nH]c(C(F)(F)F)c2)=O)C1)=O C(=O)(C(C)(C)C(=O)N(C)C)NC1CC(CNC(C(C2CC(F)(F)C2)OCC)=O)C1 c1(OCC)ccccc1-c1cccc(CN2CC(C)C2CO)c1 c1(OC)cc(C(=O)NCC2(O)CN(C(C3(NC(C)=O)CC3)=O)C2)cc(F)c1 Cc1ccc2c(c1)CC(C(N1CCN(C(C3CC4CCC4C3)=O)CC1)=O)S2 CC1CN(C(C2CCCC2)=O)CCC1CNC(=O)C(C)(C)C1CC1 c1(C(C)NC(Cn2c(C)ncc2)=O)ccc(CNC(=O)C(O)C2CCCC2)cc1 N1(C(C2CC(C)OC2)=O)Cc2nccn2CC(NC(C23CCCC(C2)OC3)=O)C1 c1(C(=O)OC)ccc(N(C(=O)CC2CCCN2C(=O)CO)C)c(SC)c1 CCC(C)CC(=O)C(=O)NCC1CN(C(=O)CCS(N)(=O)=O)CCC1C C(=O)(C(F)C(C)(C)O)NC(C)(C)CCCNC(c1csc(C(F)(F)F)n1)=O n1(CC)ccc(C(=O)NC(C)(CNC(=O)C=CC2CC2)C(C)C)cc1=O C(CC1=CCN(C(=O)CC2=CCCCC2)CC1)NC(C1CC2(CC(=C)C2)C1)=O c1(NC(c2n(C(C)C)nnc2)=O)cccc(-n2cc(CCN)nn2)c1 c1(NC(c2c(C)ccc(OC)n2)c2nnnn2C(C)(C)C)nc2ccccc2o1 N1(C(CCCCC2CN(C(=O)CC3CCCN3C)C2)C)CCCC1C(C)(C)C Cc1c(NC(c2c(-c3ccc(C(C)(C)C#N)cc3)cnn2C)=O)cc(F)cc1Br c1(C(N(CCCCNC(C(CC)c2cccnc2)=O)C)=O)ncnc(O)c1Cl C1(C(N(CC(=O)N(CCC(=O)NC)C)CC)=O)CC(=O)N(OC)C1 c1(CN(C(C(=O)OCC)CC)C2CC2)c(Br)cc(OC)c(F)c1F N1(C(CCC#C)=O)CC(NC(=O)CCNC(c2ccc(F)cc2)=O)C(F)C1 N1(C(c2c(CC)cno2)=O)CCOC(CCNC(c2cscn2)=O)C1 CC1(C)CN(C(C2CC2Cc2ccccc2)=O)CC1NC(C1CCCO1)=O C(=O)(C1CCCc2c[nH]nc21)NC12CCCN(c3nc(C#C)c(C)cn3)CC1C2 CCCCCC(=O)NC1CCCC(NC(=O)C(C)C#N)C1 CC(C(=O)NC1(CNC(=O)Cc2cnsc2)CCCCC1)C(C)C(C)(C)C N1(c2snc(C(=O)OC)n2)CCC(C2CC2)(CNC(C2CCC3(CC3)C2)=O)C1 c1(CC(=O)NC2(CCC(=O)NC3CCN(C)CC3)CCCC2)ccc(Cl)c(Cl)c1 C(CC(C)(C)C(=O)NC1CCN(C(c2nccn2C)=O)CC1CO)OC O=C(C#CC12CC3CC(CC(C3)C1)C2)N1CCC2CCN(C(=O)C(F)F)CC2C1 C(=O)(C(C)(C)CCCNC(c1cnc(C)n1C)=O)NC(CC)C(O)C(C)C N1(C(c2ccc(C(F)(F)F)s2)C(=O)NCCC)CCN(Cc2ccccc2)CC1 N1(C(c2c(CC)cns2)=O)CCC(F)(C(N2CCC(O)(CC)C2)=O)C1 c1(CCNC(=NCC=C)NCCC2(C)CC2(F)Cl)ccc2c(c1)OCCO2 c1(C(N(CC(O)CNC(c2ccccn2)=O)C)=O)sccc1S(C)(=O)=O c1(NC2(c3nnnn3CCCF)C(CC=C)CCC2)ccc(NC(=O)OC)cc1 C(=O)(C1=C(C)OCCS1)N1CCC2C(NC(c3nn(CC)c(O)c3)=O)C2C1 N1(C(=O)Cc2cccc(Cl)c2F)CCC2(CCN(C(C34CC(F)C3C4)=O)C2)C1 NS(=O)(=O)c1ccc(NCCOCCF)cc1Br C1(OCC(=O)NC(C(=O)NCc2ccoc2)C2CCCO2)CC=CC1 c1(CNC2(c3nnnn3CC)C(CCC)COCC2)cccc(F)c1OC(F)F C1(C(C)C)CN(C(C2CCC=CCC2)=O)CCCN1C(=O)C(C)NS(C)(=O)=O Cc1ccc2cc(C(N3CCN(C(=O)Cc4cncnc4)C(C)C3)=O)ccc2n1 c1(C(=O)NCC(C)N(C(=O)CCC2CCCN2C)C)ccc(N)c(Br)n1 C1(O)(CN(C)C(C2(CS(C)(=O)=O)COC2)=O)CCCN(C(C2CCCCN2C)=O)C1 C(=O)(CC(C)C(F)(F)F)N1C(CC(=O)NC(CCC)CCO)COCC1 CCC(C)CC(C)C(=O)NCCCN(C(=O)CN1CCCC1=O)C1CC1 c1(C(=O)NC(C=CC(=O)NC2C(OC)C(O)C2)(C)C)nc(=N)cc[nH]1 c1(OCC(CCCC)O)cc(F)c(F)cc1Cl C(CC(=O)N1CCCCC1CNC(=O)C1=CSCS1)(C(F)(F)F)OC C1(CNC(C2CC=CCO2)=O)CN(C(c2sccc2F)=O)C2CCCC2O1 Cc1cccc2c1CN(C(C1CC3(CCC3)CN1C(=O)COCC1CC1)=O)C2 c1(C(=O)NCCC2(C)CCN(C(c3c(C)nsc3)=O)C2)c(F)ccc2n[nH]cc12 C12(NC(CCCC#C)=O)CCCC1N(C(c1ccnn1CCF)=O)CCC2 O=C1COC(C(=O)NCC(C2CCCC2)NC(C2CCSC2)=O)C1 N1(C(c2n[nH]c(C)c2Cl)=O)CCCC(C)C1CNC(C1CCC(=O)O1)=O c1(C(N2C(CNC(c3cc(N)c(Cl)nc3)=O)CCC2)=O)cccc(Cl)c1[N+](=O)[O-] CCC(Cc1ccccc1C)C(=O)N(C)Cc1cc(C#N)cs1 Cc1cc(C(N2CC(C3(NC(=O)COCCOCCO)CC3)C2)=O)cc(Cl)n1 c1(N(CC(=O)NC(c2cccc(OC)c2)CO)C)cn(C)c2ccccc12 c1(CNC(C2(C)CCCS2)=O)cccc(C(=O)NCCN(CCO)CCO)n1 C1(CNC(CCC2(C)CC2)=O)CN(C(c2cncc([N+](=O)[O-])c2)=O)C2(CCC2)C1 C1(CC(=O)N(CCCNC(c2csc(CC(F)F)n2)=O)C(C)C)CCCS1(=O)=O CN=C(NCC1SCCS1)NCC(C)(O)CC1CC1 c1(CC)nsc(CNC(=O)CSCCNC(=O)Cc2cncnc2)n1 CCC(C)C(C(=O)NCC(CO)NC(C1(C)CC=CCC1)=O)NC(C)=O C(C)(CCC(=O)N(C1CCN(C(C2CC2F)=O)CC1)CCO)OCC C(c1cccs1)=CC(=O)NC1CCCC1NC(=O)CCc1ccncc1 c1(C(=O)NC(CCN(C(C=CC=CC)=O)C)C)ccc2ccn(CCCC)c2c1 c1(NC(C(C2CC2)NC(C2(CCC=C)CC2)=O)=O)cc(F)ccc1OC CP(C)(=O)c1ccccc1C(N1CCC(NC(=O)COCC(=O)OC(C)(C)C)C1)=O C1(CC(=O)N(CCOCCCNC(C2CCC(CC)O2)=O)C)CCCCC1(C)C C1(CNC(C2CC2Br)=O)CCCCN1C(=O)CCc1cccc(O)n1 c1(C(N2CCC(C(N3C4CN(C)CC3CC4)=O)O2)=O)cccc2c1cnn2C C#CC1CCC(C(N2CCC(C)(CCNC(C3CC(O)C(F)C3)=O)CC2)=O)CC1 C1(NC(C2CCn3nnnc3C2)=O)CCCCCN(C(c2ccc(Cl)o2)=O)C1 C1(F)(CNC(CCC2C(C)C2)=O)CCN(C(C2(c3nccs3)CC2)=O)C1 C1(CC)(CNC(=O)C(CO)NC(=O)C(C)c2cc[nH]n2)CCCC1 C(CNC(c1[nH]ccc1CNC(C1CCC(=O)N1)=O)=O)(C(C)(C)C)OC c1(C(N(C2CCN(C(COCCCC)=O)CC2)C)=O)cc(CC)cc(F)c1 N1(CCNC(C2(N3CCOCC3)CCCOC2)=O)CCOc2ccc(Cl)cc2C1 CC1(CC(N2CCC(C#N)C2)=O)CCN(C(=O)CC2CCCO2)C1 C=CC1(C(=O)NC2CC3(CCC3)C2O)CCN(C(=O)CCCOC(C)(C)C)C1 c1(C(=O)NC(c2occ(C(N3CCC(C)(CCC)C3)=O)n2)C)cccc(C)c1F C(CN=C(NCC(C)Cc1cccc(C)c1)NCC1CCCC1OC)SC N#CCCCCC(=O)NCC12CC1CN(C(c1ccc(C(F)(F)F)c(F)c1)=O)C2 C1(CC(CO)NC(N2CC3CC3C2)=O)CCC(F)(F)CC1 c1(C(=O)NC2CCC(NC(c3nnn(C)c3N)=O)CC2)cc2ncccc2[nH]1 C(=O)(CCCC(C)(F)F)NC1CCCN(C(CCCc2nc(C)sc2)=O)C1 N1(C(C(C)Cc2ccc(F)cc2)=O)CC(C)(CNC(c2cocn2)=O)CC1(C)C c1(N(S(C)(=O)=O)C)cccc(C(=O)Nc2ccccc2CN2CC(O)C2)c1 N1(C(c2cc(C(=O)OC)cn2C)C(=O)NC2COC2)CC2CC=CCC2C1 N1(C(C(c2cccc(F)c2)C)=O)CC(NC(c2cnn[nH]2)=O)CC12CCOCC2 C(=O)(C(C)(F)CC1CCCC1)N(CCCNC(c1sccc1F)=O)C C1(C(=O)NC2CC(=O)OC2)C2CCC(C2)N1C(c1ccnc(C(F)F)c1)=O C(=O)(C(CCOC1(CC#C)CCC1)NC(=O)Cc1ncoc1C)NCCO Cn1cc(S(N)(=O)=O)cc1C(=O)NCC1(F)CCC(CNC(=O)CS(N)(=O)=O)C1 C12CN(CC1C)C2=O.C1(CCNC(CSCC(C)C)=O)CCC(=O)N1C1CC1 C1(NC(C(C=C=C)C)=O)CCC2(CC1)CC(NC(c1ccc(COC)s1)=O)C2 c1(-c2scc(NC(C3CC4(C(C(=O)OCC)C4)C3)=O)n2)c(OC)cccc1Cl C1(NC(=O)CS(=O)(=O)C2CC2)CCC2(CCN(C(c3csnn3)=O)C2)C1 C#CC1(C(=O)NCc2ncccc2Cl)CCN(C(=O)C(c2ccc(C)o2)C)CC1 CCCC(C)C(=O)NC12CC1CN(C(=O)CC1CCCC1(F)F)C2 c1(C(N2CCOCC(NC(c3c(C)cc(C)s3)=O)C2)=O)ccc(F)c(O)c1F c1(C(=O)NCC(C)N(C(c2n(CC)ncc2)=O)C)ccc(C)c(O)n1 C#Cc1cnn(C)c1C(=O)NC1CC2CC1N(C(=O)CCC1CCOC1)C2 c1(OC)ccc2c(c1)CC1(CC1)CN(N1CCOCC1CC1CC1)C2 CC1(C(=O)NC2CCCCC2NC(C2(C3CCC3)CC2)=O)CC(C#N)C1 C1(CC(=O)OC(C)(C)C)CN(C(=O)OC2CCCC2c2ccccc2)CC1(C)C CC1CN(C(c2ccc(O)nc2)=O)CC(CCNC(=O)CC2OCCC2(C)C)O1 c1(CNC(=O)OC(C)(C)C)ccnc(N2CCCC2)n1.C12CCOC(C1)C(=O)N2 CCC(C)C(C(=O)NCc1nc(CNC(=O)COC(C)CC)cs1)NC(C)=O c1(OC)cc(CC(=O)NC2CCC(CNC(C34CSCC3C4)=O)C2)on1 Cc1ccc(CNC(=O)C(C2CCN(C(c3csc(C)c3C)=O)C2)C)cc1C S(=O)(=O)(c1cnc2ccccc2n1)NC1CCN(c2cc(C)nn2C)C1 CCC(C(=O)NC(C)(CNC(c1nc2cccnc2s1)=O)C(C)C)C(C)(F)F C1(C(=O)OC)CC2(CCN(C(C34CCN(C3)S(=O)(=O)C4)=O)CC2)CO1 N1(C(C=C(C)C(C)C)=O)CCN(C(c2cnn[nH]2)=O)C(CC(F)(F)F)C1 C1(CNC(C(C=CC)O)=O)COCC2(CCN(C(=O)Cc3coc(C)n3)CC2)O1 CCC(C)CC(C)C(=O)NC1C=CCN(C(C2(c3ccncc3)CC2)=O)C1 C(=O)(C(C)C(O)C(C)C)N(C(CNC(C(COC(C)C)NC(C)=O)=O)C)C N#CC1(NC(c2ccc(O)c(F)c2)=O)CCN(C(=O)C=Cc2ccc(Br)cc2)C1 N1(C(C2(NC(C3CCC(C)O3)=O)CC2(C)C)=O)CC2CCC1C(O)C2O N1(C(c2c(C)cccn2)=O)CCCC(C2CN(C(c3cn4c(n3)SCC4)=O)C2)C1 c1(CC(=O)NC2(C)CCN(C(CCCC=C)=O)C2)cn2c(C)cncc2n1 C1(CNC(C(CCC)OCC)=O)CC2COCC2N1C(=O)C(O)CCSC c1(C(=O)NC(C(C)C)CNC(=O)C2CC2)cc2c(cc1F)OCC(=O)N2 C(CC(C)(C)CC(=O)NC1CCN(C(c2nc(O)[nH]c(=O)n2)=O)CC1C)OC N1(C(c2c(C)cn(C)c2)=O)CCN(C)CC1C(=O)NCCCC1(O)CCC1 C1(NC(COC2(C)CCCC2)=O)CCOC(CNC(=O)CC2(O)CCCOC2)C1 Cc1c(C(=O)NC(CNC(c2coc(C(F)F)n2)=O)CO)[nH]c2ccccc12 c1(C(N)=O)cccc(C2(NC(=O)C(=O)NC3(C4CCCO4)CCCC3)CC2)c1 O=C1CCC(CC(N2CCC(N(C(=O)C(=O)Nc3ncc[nH]3)CCO)C2)=O)N1 C1(NC(C(COC)OC)=O)CCC(CN(C(=O)CCc2ccc(F)cc2)C)CC1 c1(OC)ccn2cc(C(=O)NC(C)CCCNC(=O)CC(C)N(C)C)nc2c1 c12cc(ccc1Br)C2NC1CCOC1(C)C.c1(COCC)nnnn1C C1(C)(C(N2CCC(CN(C)C(c3ncoc3C3CC3)=O)C2)=O)CNC(=O)C1 c1(OC)nccc(Br)c1C(=O)NC1CCC(N(C(=O)CS(C)(=O)=O)C)C1 c1(CC(C(=O)NC(C)CC2CCC2)NC(=O)CSC(F)F)ccccc1 Cc1cccnc1C(F)(F)C(=O)NC12CC(NC(=O)Cc3sc(S)nc3C)(C1)C2 O=C(C1CCc2ccc(Cl)nc21)NC1CCN(C(c2cccnc2O)=O)CC1 C=CCCCCCCCC(=O)NCC(C(C)C)NC(C1OCC2CCCC1C2)=O C1(C(=O)NCC(CN(C(C(CCC)F)=O)C)(C)C)CC(C(C)C)=NO1 c1(C(N2C3(C(N4CC(OC)C4)=O)CC3CC2)=O)ccccc1C#N N1(C(C(c2cncnc2)C)=O)CCCC(N(C(=O)CC2C=CS(=O)(=O)C2)C)CC1 C(C(=O)N1CC2COCC2O1)C1N(C(CCC(C)(F)F)=O)CCC1 c1(OCC(=O)NC2(CNC(C3C(C)CCC3)=O)CC2)nn(C)cc1Br Cc1c(CCNC(N2CCCCC23CCSC3)=O)sc2ccccc12 CC1CCC(C)C1NC(=O)C(c1cccnc1)NC(=O)CC1(N(C)C)CCC1 N1(C(C(C)Cc2ccccc2)=O)CCC2CN(C(=O)C3=CCCS3)C2C1 N1(C(C(C)N(C(c2cnc(Cl)n2C)=O)C2CC2)=O)CC(CO)C1(C)C c1(C(=O)NC23CCN(C(c4n(CC)ccn4)=O)CC2C3)cc(C)c(F)cc1F C1(CC)CN(C(c2c(C)n[nH]c2C)=O)CCN1C(C1CCS(=O)(=O)C1)=O N1(C(Cn2nnc(=N)[nH]2)=O)CC2(CCC2NC(C2CC=CCC2)=O)C1 C1(CC(C2CCCCC2)NC(=O)CC2CCCCCC2)CCCCN1C(C)=O c1(CC(=O)OC(C)(C)C)c(F)cc(N)cc1F.CC1CC(=O)N1C(C)(C)C C(=O)(C1OCCn2ccnc21)N1CCC(C)(NC(Cc2ncc(C)[nH]2)=O)CC1 C12(CNC(C(N3CCCC(O)C3)C)=O)COC(CNC(=O)CC3(C4CC4)CC3)(C1)C2 C(C(=O)N(C)OCc1ccccc1)(C1(C)CC1)NC(C(C=CC)O)=O N1(C(c2c(C)ccnn2)=O)CCCC(C2CCN(C(=O)C3=CC(C)(C)C3)C2)C1 C1(NC(CC(CN(C(CCNC(C)=O)=O)C2CC2)C2CCC2)=O)CCCC2(CCC2)C1 c1(CNC(C(C=C)O)=O)ccc(C(C)NC(c2ncoc2-c2cccs2)=O)cc1 C1(C(N(CC)Cc2ccn(CC)n2)=O)CCN(C(=O)Cc2cccc(C)n2)CC1 c1(OC)cnc(C(F)(F)F)cc1C(=O)NCC1CCN(C(c2cccn2C)=O)C1 c1(C(=O)NCC(CCOC)NC(C2(O)CCCC2)=O)cc(S(N)(=O)=O)cs1 c1(CN2CCC(NC(Cn3ncc(C)c3)=O)C(F)C2)cccc2c1OCCO2 O=C(CCCN1CCCC1)NCC1CC1NC(c1sccc1Cc1ccccc1)=O C1(NC(C(C(C)C)O)=O)CCN(C(=O)CC2CC=CCN2C)C1(C)C C1(C(N(C2(C(=O)NCCSC)CC2)C)=O)CCC(F)(F)C1 N1(C(c2c(C)ccc(C)c2)C)C(=O)C2CC3(CCCCC3)CN2C1=O C1(C(=O)NC2(C)CS(=O)(=O)C2)CC2(CCN(C(=O)CCC(CF)CF)C2)C1 c1(CNC2CCC(C(=O)Nc3n(CC)nnn3)OC2)ccc(I)c(O)c1 C1(NC(C(CCC2CCC2)NC(c2cnncc2O)=O)=O)CCCC2(CCC2)C1 n12cc(cc1C1CC1)S(=O)(=O)N2C.c1(SCC)c(F)cccc1F C1(C)(CCNC(CSCCN(C)C)=O)CCN(C(c2nocc2Cl)=O)CC1 c1(C(N2CCC(CC=C)(NC(c3cc(Cl)ns3)=O)C2)=O)cc2n(n1)CCC2 C1(C(N2C(C)(CCO)CC2)=O)CC(=O)CN1C(=O)C1=C(Cl)CC1 C1(NC(CCCOCC=C)=O)CCN(C(=O)Cn2nc(C)nc2C)CCC1(F)F c1(CC2CC(C(N(CCN(C)C(c3ccccc3)=O)C)=O)C2)ccccc1 N1(C(COC2(C)CCOCC2)=O)CC(F)(F)CC1(C)CNC(C1CCNC1=O)=O c1(-n2c(C)ccn2)ccc(OCN2CCN(C(C3C4CCC(F)C34)=O)CC2)cc1 Cc1nc2cc(C(N3CC=CC(NC(C4CC(=O)N4)=O)C3)=O)cnc2[nH]1 N1(C(CC)(C)C)CCC2(CCCN(CC3CCC(C(=O)OC)OC3)C2)C1 CCC(CNC(=O)Cc1ccc(C2CC2)nc1)C(=O)O c1(C(N2C(CCNC(Cn3c(C)cnc3)=O)CCC2)=O)ccc2ccccc2n1 N1(C(C=CCCC=C(C)C)=O)CCCC(O)(CNC(=O)C(N2CCCCC2)C)C1 Cc1cc(F)c(C(N2CCOCC2CN(C(=O)Cc2scnc2C)C)=O)cc1F Cc1nc(C=CC(N2CC(C)(NC(=O)CCc3cncs3)C2)=O)cs1 CC1C(C)N(C(=O)C=Cc2nccs2)CCN1C(c1ccc(Cl)cc1)=O N1(C(CC(C(F)F)NC(CCC2(C#N)CCC2)=O)=O)CCC2(CC1)CC2C#N c1(C(=O)NC2CN(C(c3c(C)ncs3)=O)C2)cc2c(nc1O)CCCC2O CC1(C)CC(NC(c2ccc(N3CCCC3)cc2)=O)CN1C(C1C=CCC1)=O C1(Nc2c(C(=O)NC(COC)C)cccn2)CCCN(C)C1=O C(=O)(C(CO)C(C)(C)C)NCCC(=O)NCC(CCC=C)O N1(C(C2CC(OCC)C2)=O)CC2(C1)CN(C(c1ccc(N)cc1C)=O)C2 N1(C(C2N(C)C(=O)OC2)=O)CCC2(CC(NC(=O)Cc3csnn3)C2)C1 CCC(C(=O)N1CC2(C1)CN(C(=O)Cc1csc(C(F)(F)F)n1)C2)C(C)C C1(C(=O)Nc2c(C(C)C)nc(Br)s2)Cc2ccccc2O1 c1(C(N2C(C3(NC(C(C4CC4)SC)=O)CC3)CCC2)=O)ccnc2cc[nH]c12 C1(CNC(C(CC)NC(N)=O)=O)CCN(C(c2cc(C)ccc2N)=O)C(C)C1 C1(C(N2C3CCN(C(Cc4nnc(C)s4)=O)CC3C2)=O)CCC2(CC1)CC2(F)F Cc1cc(C(N2CC(NC(=O)CNS(N)(=O)=O)CC(F)C2)=O)nc(C(F)(F)F)n1 C1(CNC(Cc2c(C)nc(SCC)s2)=O)CN(C(C2C=CCC2)=O)CC12CCC2 CCC(CCC(=O)NCC1C(C(N2CCC(C)C2)=O)C1(C)C)OC C(CN=C(NCC(=C1CCCC1)F)NC(C1CCCO1)C1CCOC1)C(=O)C1CC1 c1(C(=O)NC2CN(C(C(=O)N(C)C)=O)C(C)(C)C2)nccn2nccc12 N1(C(COCCSC)=O)CCCC1C(C)(C)CNC(=O)C(C)Sc1nncn1C N1(C(C(C)N(C(C)=O)C)=O)CCCCC1C(=O)NC1(C)CC(CO)C1 N1(C(C(C=C)O)=O)CC(C(=O)N(CC(=O)NC(C)C)C)C(CC)C1 c1(OC)cncc(C=CC(N2CCC(Oc3ccc(F)cc3F)C2)=O)c1 C12(CC(=O)NC3(CF)CCN(C(c4[nH]ccc(=N)n4)=O)C3)CCCCC1C2(F)F C(=O)(C1=C(C)OCCS1(=O)=O)NC1CCCN(C(CCSC)=O)CC1 C(C(=O)NC1CCC2(CC2)C1)(C(C)(C)C)NC(C(C=C)CC)=O N1(S(CC)(=O)=O)CCCC1C(=O)NC(C)CCNC(C1CCO1)=O N(C(=NCCc1ccc(Cl)c(C)c1)NCC1(OC)CCOC(C(F)(F)F)C1)CC C(=O)(CC(CC)SC)NCc1cn(CC(=O)NCCC)nn1 O=C1CC(CCNC(C2(O)CCCC2)CCO)C12CCC2 C1(CNC(C(CC#C)O)=O)CCN(C(=O)Cn2ccc(O)nc2=O)C12CC2 N1(C(C2(C#C)CC2)=O)CCC2(CC1)CC2CNC(C1CCn2ncnc2C1)=O c1(CC(=O)NCC(C)NC(CCCNC(=O)OC)=O)ccc(OC(F)F)c(F)c1 N1(CCC=C(CC)C)CCCN(Cc2noc(-c3oc(C(C)C)nc3C)n2)CC1 C=CCC(C(=O)NCCCOCC1CC1)NC(N1CCCCCC1)=O N1(C(CN2C(C)CCC2C)=O)CCN(c2ccccc2)CC1C C1(NC(C(CC=CC)NC(=O)CCOC)=O)C2CCCC1CC2 c1(C(=O)NC2CN(C(C3CCN(C(CC)=O)C3)=O)C2)ccc(C(C)(C)C)cc1N NC1CCc2cc(Cl)ccc21.n1(CCCSC)nnnc1C1(N)CC(C(N)=O)C1 c1(C(=O)NCC(CC)NC(c2c[nH]cc(F)c2=O)=O)ccc(Br)c(C)c1F C1(NC(c2ccc(COC)cc2)=O)CCCCCN(C(c2ccc(F)s2)=O)C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)(C)C2CC2)ccnc2[nH]cnc12 CC(C)(C)CC1CN(C(=O)C(C2(O)CCC2)NC(=O)Cc2ccns2)C1 N1(C(c2c(C)cns2)=O)CCCC(C)(NC(=O)C=CCN2CCCC2)C1 C1(C(=O)NCC2C(C(=O)NC(CSC)(C)CO)CCCC2)CCCC(C#N)C1 N(C)(S(=O)(=O)N(C)C)C1CCN(C(CCC=CC)=O)C1.c1(N2CC2)ccccc1F Cc1c(C(=O)NCCc2nc(C3CCCO3)n[nH]2)nnn1-c1cccc(Cl)c1 c1(C(N2CCCC(C(C)NC(C3CCC3(C)C)=O)C2)=O)cn2cccnc2n1 CCCC(C)CN(C(=O)C(C)=CCNC(c1cc[nH]c1CC)=O)C CC(C)CS(=O)(=O)CC(=O)NC1CCCCCN(C(=O)Cc2ccoc2)C1 CNS(=O)(=O)NCC(=O)NC1CC(F)(CNC(=O)CN2CCCCC2)C1 C1(NC(c2cc(C)ns2)=O)CC(C2CCN(C(=O)CC3CN4CCC3CC4)C2)C1 N1(C(c2c(C)nco2)=O)CC2=C(C1)CN(C(c1ccccc1C#N)=O)C2 C1(CCC(=O)NCC(CC)OC)CCCCN(C(=O)CCCC(C)C)C1 N1(C(C(F)OC)=O)CCC(c2ccccc2)(NC(=O)CCN(C)CCO)C1 c1(C(=O)NCC2OCC(C(=O)OC)C2)ncccc1NC(C)=O C1(C(N2CCCCC(NC(C=COCC)=O)C2)=O)Cc2cc(C)ccc2S1(=O)=O C1(C(N(CCCC)CCOC)=O)CC2CC2N1C(c1cccc(=O)o1)=O N1(C(COCC)=O)C2CCC1C(CO)N(C(=O)COC(F)(F)F)C2 N1(C(=O)CSC(F)(F)F)CC(C2CN(C(c3cccc(F)c3Br)=O)C2)C1 C(=O)(CCNC(C1(C(F)(F)F)CC1)=O)NCCNC(C1(CCOC)CC1)=O C1(NC(Cc2cc(COC)on2)=O)CCCCN(C(C2(C(F)(F)F)CC2)=O)C1 C12(C(=O)NC(C)(C)CCCNC(=O)CSc3ccc(F)cc3)COCC1C2(F)F C1(C(=O)NC2CC(NC(C(Cc3cn(C)nc3)O)=O)C2)CCCS(=O)(=O)C1 c1(C(=O)NCC2(F)CCC(NC(C3(OC)CS(=O)(=O)C3)=O)C2)cc2c(s1)CCC2 N1(CCNC(C(C)Sc2ccccn2)=O)CCCN(C(=O)Cc2cncs2)CC1 CC12C3C4C1C1C2C3C41C(N1CCC(NC(C2CCCN2C2CCCC2)=O)C1)=O N1(C(CN(CC)CC)=O)CCCC(C2CCCN2C(=O)Cn2[nH]cnc2=N)C1 c1(CC(=O)NC(COC)(C)CC(=O)O)cccc(S(C)(=O)=O)c1 Cc1cc(Cc2noc(-c3nc(Oc4cccc(F)c4)ccc3C)n2)cc(O)c1 N1(C(C(CCC)NC(=O)C(F)OC(F)(F)F)=O)CCCc2ccccc21 c1(-c2cn(CC(C)NC(c3ccn4ncnc4c3)=O)nn2)cc(Cl)c(Cl)c(Cl)c1 C1(N(C(C(C2(C)CC2)NC(C2C(=C)C2)=O)=O)C)CC(C)(C)C1 c1(OC)c(C(N2CCCC2CN(C)C(c2scnc2Cl)=O)=O)cccc1C C(=O)(C1=CS(=O)(=O)CCC1)NCC1(NC(C(C)(C)OC)=O)CCCCCC1 C1(C(=O)NC2CC(CNC(CCCOC)=O)C2)CCC(C)(C)C1 C12(CNC(Cc3c(C)ocn3)=O)CCCC1N(C(c1cc(Br)c[nH]1)=O)CCC2 C=CCC(CC)C(=O)N1CC(C=C)(CC(=O)NC2CN(C)CC2(C)C)C1 c1(C(N2C(CC)CN(C(C3CC3C(F)F)=O)CC2)=O)ccc2c(c1)CCN2C CCCC(C(=O)OC)C(=O)N1CCCCC(N(C)C(c2cn(CC)nc2C)=O)C1 C1(C(=O)NC2C(C=C)CN(C(c3occc3C(C)C)=O)C2)CCc2ncnn2C1 N#CC1CN(C(=O)CCc2ccc(O)cc2)CC1NC(c1cnco1)=O c1(OCC)ccc(C(=O)NC2CC(NC(=O)CCn3cccnc3=O)C2)cn1 N1(C(C(C)N(C)C)=O)CCC2(CCC2)C(NC(=O)Cc2cc(Cl)n(C)n2)C1 C1(C)(C(=O)NCCC2CCC(NC(CC3C(C)(C)C(O)C3)=O)C2)CC2CCC1C2 N1(C(C(=O)NCCOC)=O)CC(NC(=O)C=Cc2ccc(C3CC3C)o2)CC(O)C1 c1(C(N2CC(CCNC(CCOCCC)=O)OCC2)=O)cc2c(C)cccc2o1 O=C(C1=C2CCN=C2NC=C1)NCC1CCCSCC1 C1(C(=O)NC(CC(C)C)C(=O)N2CCCC2)CCC2COCCC2C1 CC1CCC(NC(=O)C=CC(C)(C)C)CN1C(C1CC(=O)C12CCC2)=O c12ccc(cc1)OC(=O)N2.c1(OC)cnc(CNCC(C)N=[N+]=[N-])o1 Cc1ccc(-n2cccc2)c(C(=O)N(C)Cc2cn(Cc3ccccn3)nn2)c1 c1(CNC(=O)NC(c2ccc(C)c(F)c2)C)c(C)nc2cc(O)nn2c1C N1(C(C2=CCC(C)CC2)=O)CC2CC(C)N(C(=O)CC3CC(=O)NC(=O)C3)C2C1 c1(C(=O)NC2C(CNC(=O)Cc3ccc(F)cn3)CCC2)cccc(F)c1O C1(CCNC(c2n[nH]cc2CNC2CC2)=O)CCCSC1 C1(CC(N2C(CNC(c3cc(OC)n(C)n3)=O)CC(F)C2)=O)CCC(C)(C)CO1 c1(C(=O)NCCC(C)(C)NC(Cc2cnc(C)o2)=O)sc(=N)[nH]c1C Cc1cc(N)c(C(=O)N(C)CCNC(=O)Cc2cccc(C)c2Cl)c(F)c1 c1(C(=O)NC2CCC(N(C(=O)C=CC(F)F)C)C2)ncc(F)cc1F N1(CCN(C(CCC(=O)N(C)C)=O)C)CC(NC(c2ccccc2)=O)CCC1=O N1(C(C)=O)CCC2(NC(=O)NCCCc3cccc(N(C)C)c3)CCCCC12 N1(C(C2(COC)CCC2)=O)CC2CCC1C(NC(=O)C(F)(F)CC1CC1)C2 C1(C(C(=O)NCC(CNC(C(C)CN(C)C)=O)c2cn[nH]c2)O)COC(C)(C)O1 C1(C(=O)OC)(C(N2CCC2c2cccc(F)c2)=O)CC(O)C12CCC2 C1(C(N(C2CC(NC(Cn3ccc(C)n3)=O)C2)C)=O)CC(F)C(=O)N1 N1(C(C(C)=CC(C)(C)C)=O)CCCC(C)(C(N2CCNC(=O)C2CCO)=O)C1 Cc1ccc(Br)c(CC(=O)NCC2COCCN2C(=O)C=C(Cl)Cl)c1 C(CC(C(=O)NOCCN(C)C)NC(=O)CC(O)CN(C)C)SC C1(NC(CC2(CSC)CC2)=O)CC(CC(=O)NCCN2CCCCC2=O)C1(C)C Cc1csc(C(=O)N(CCCNC(=O)C(C2CCCCCC2)O)C)c1Br c1(CCC)cc(C(=O)N(CC(C)(C)NC(C2CCN2CC)=O)C)ccn1 N1(C(C(=O)Nc2ccc(OCCC)cc2)C)CCN(C)CC1C#N CC(C)C(CCN(C)C(C1(C)CC(F)C1)=O)NC(=O)CCOCC1CC1 c1(C(N2CCC(NC(=O)CC3CCCC3)C2)=O)c(F)cccc1Br c1(SC)cc(C(=O)NC(C)CC2CN(C(C3(F)CCOC3)=O)C2)ccc1[N+](=O)[O-] C1(CCC)CCC(C(=O)NCC(C)NC(C2(n3nccn3)CC2)=O)CC1 C1(CNC(C(C)(F)F)=O)CCN(C(c2nccnc2Cl)=O)CC1 C1(NC(C(CSC)O)=O)CCN(C(c2ccc(C3CC3)c(Cl)c2)=O)CC1(C)C N1(C(C(CC)COC)=O)CCCC12CCN(C(c1ccc3c(c1)CCC3)=O)CC2 C1(C(=O)NC2CCC2CNC(C23CC4CC2C3C4)=O)CC2(CCC2)CO1 CC(C)(O)C(F)C(=O)N1CCC(CO)(NC(c2ccnc(C(F)(F)F)c2)=O)C1 S(=O)(=O)(CC(=O)NC1(CNC(=O)CC2CC(F)C2)CCCC1)NC C(=O)(C(C(C)C)C(C)C)NCCN(CCC)C(c1nc[nH]c2ncnc1-2)=O c1(CC)cc(Cl)ccc1C(=O)NC1(CO)CCCN(C(c2cnn(C)c2C)=O)C1 c1(OC)cccc(-n2cc(CNC(N3CC(N4CCOCC4)C(C)C3)=O)nn2)c1 c1(-c2cn(C(C)C(=O)N3CC(Cc4ccccn4)C3)nn2)c(Br)c(C)nn1C C1(NC(c2c(C)ccc(C)n2)=O)CC2CCC(C1C)N2C(=O)CCc1cnoc1 N1(C(c2c[nH]c(=NC)s2)=O)CCC(NC(=O)C(C)S(N)(=O)=O)C(F)C1 C1(C(=O)NC(C(=O)OCCCC)C)CN(Cc2cnc(Cl)cc2OC)CCC1O C(c1ccc(C(N)=O)cc1)=CC(N1CC=CC(NC(c2cnn(C)n2)=O)C1)=O N1(C(C(C=C)(C)C)=O)CC(C(=O)NCC(N2CCOC(C)C2)=O)C(C)(C)C1 N12CCC3(CCCN3C(=O)C(CC3CC3C)C3N(CCOC)CC(C3)C1=O)C2 C(CC1CCOCC1)(C(=O)NCC(CO)N(C)C)NC(CCC1CC(OC)C1)=O C(C(CC1CC1)C(=O)N1CCCC(OC)C1)N(C(c1cc(CC)sn1)=O)C1CC1 C(=O)(CC(C)(C)C(F)(F)F)NC1C(C)CCN(C(c2c(Cl)cn(CCC)n2)=O)C1 c1(CN2CCC(CN(CC=C)C(=O)NC(C)CC)CC2)ccc(Cl)c(F)c1 N1(C(c2n(CC#C)ccc2)=O)CCC(NC(=O)Cc2nocc2C)C(CO)C1 CC(CC(=O)NC1(CC(=O)NC2CCC=CCC2)CCC1)C(F)F c1(C(=O)NCC(CC(=O)N2CCC2CO)OC)ccc2cc[nH]c2c1 N1(C(Cc2cccc(NC(=O)OC)c2)=O)CCC(C2CCN(C(=O)CO)C2)C1 N1(C(C2C(C)OCC2)=O)CCN(C(c2cnoc2)=O)CC12CCC2 C1(C(=O)NC2CC(n3cc(-c4n(C)ccc4)nn3)C2)C2CC3C(C2)C13 c1(C(C(N2CCN(C(C3N(CC)CC3)=O)C3C2C3)=O)=O)c[nH]c2cc(F)ccc12 N1(C(C2CC=C(C)CC2)=O)CCC2(CCN(C(=O)CCCC(C)(C)C)C2)C1 c1(C(N(CC(CC)NC(=O)C(C)n2cnnn2)C)=O)cn(CC)nc1C C(=O)(CCCC(C)(F)F)N1CCCC(CCNC(c2c(C)cc(F)cc2)=O)CC1 c1(CC(=O)NCC2(NC(CC3C(C)(C)C(O)C3)=O)CC2)ccc2cccnc2c1 c1(CN(C(C2CC2NCc2ccsc2Br)=O)CC)ccccc1Cl c1(CN2CCC(O)(C(=O)Nc3c(Br)ccc(C)n3)C2)ccc2c(Cl)ccnc2c1 c1(C(N2C(CN(C(=O)CCCF)C)CCCC2)=O)ccc2c(n1)CCCC2 c1(NC(C2C(NC(C3C(C(=O)OC)C3)=O)CCCC2)=O)ccc(N(C)C)c(F)c1 C1(C(=O)NCC2(OCC)CCC2)CC(O)CCN1C(c1csnn1)=O c1(C(=O)NC2CCN(C3CC3)CC2)coc2ccc(Cl)cc12 S(=O)(=O)(CC(=O)N1CCCC1C(C)(C)CNC(=O)C(c1ccc(C)s1)C)NCC C#CC1(O)CC(C(N2CCC(C(C)NC(=O)CNC(=O)CN(C)C)C2)=O)C1 C1(NC(Cn2c(CC=C)nnc2S)=O)CCCCN(C(=O)CCC(=C)C)C1 c1(OC)ccc(C(=O)NCC2(O)CCCC2C)c2ccccc12 N1(C(C(C)SC(F)(F)F)=O)CCC(CNC(C2(C)CC(F)(F)C2)=O)C12CCC2 c1(N2C(=O)CCC2)cccc(NCC2CCC3(C2)CC3(F)F)c1[N+](=O)[O-] C(CCCC(=O)N1CC(C)(NC(=O)C(C)OCC(C)C)C1)OCC c1(C(c2nnnn2Cc2cnc(Cl)s2)NCC)cn2ccnc2s1.c1ccccc1 C1(NC(C(C=C)O)=O)CCCCC1NC(C1(Cc2ccccc2F)CC1)=O CCCC(CCC)CC(=O)NC12CCC(C1)N(C(c1cc(Cl)ccc1F)=O)C2 C1(C(=O)NCC2CCCC2)CC2CCCCC2N1C(C1CC(O)C1)=O C(C1=CCN(C(C2COC(=O)C2)=O)CC1)NC(C1(C(F)(F)F)CC(=C)C1)=O CC1OCC2(CCN(C(C3(Br)CC3)=O)CC2)C1NC(=O)CC1(O)CCC1 N1(C(c2cn(CC)nn2)=O)CCC2(CCN(C(c3ccnc(C(F)F)c3)=O)C2)C1 C1(C(=O)NC(C#C)C(C)OC)CCOCC1NC(C1(CC#C)CCCO1)=O C1(C)(CNCCn2cc(CC3(O)CN(C(C(C)SCC)=O)C3)nn2)CSC(C)=N1 C(=O)(CC(C)(C)CN(C(C1CCCSC1)=O)C1CC1)N1CC(CS(C)=O)C1 C#CCCCCC(=O)N1CCCN(CCCCNC(=O)Cc2cnsc2)CC1 N1(C(c2c(C)coc2)=O)CCN(C)C(C(N2CCOC(C3(C)CC3)C2)=O)C1 N1(c2nnc(COC)s2)CCOCC12COCCN(C(=O)CN(C)C(C)=O)C2 Cc1nc(C(N2CCOCC(F)(CNC(=O)C=C3CCC3)C2)=O)c2ccccn12 Cc1cc(C(=O)N(C2CCN(C(c3cn[nH]c3)=O)CC2)C)nc(O)n1 N1(C(=O)OC(C)(C)C)CCC2CCC12C(=O)NCc1cc(C(=O)O)on1 N1(C(c2ccc(-c3cn(C)nc3)cn2)=O)CCCCC(CNC(=O)C=CCO)C1 c1(C(N2CCC(O)(C(CNC(C(C#C)(C)C)=O)C)C2)=O)cc(C(N)=O)ccc1F N1(C(C(=O)NCC)=O)CCN(C(=O)CCCN2CCCCC2)CC1CF N1(C(C(COC)N(C)C)=O)CC2(CCC2)CC1C(=O)NC1(CF)CC1 Cc1c(CC(=O)OCC2CC(=O)N(Cc3ccccn3)C2)nc(Br)n1C CCC(C(=O)NC1COCCN(C(=O)Cc2conc2C)C1)C(C)(F)F Cc1cc(S(=O)(=O)Nc2cncc(NCCN3CC4CCCC4C3)c2)c(F)cc1Cl C(C(CCNC(CC1CC1C1CC1)=O)NC(=O)CCNC(=O)OC)NC(C=C)=O N1(C(C2(CCNC(CC=C)=O)CC2)=O)CCCN(C)CC1C C1(C(=O)NC2C(CO)CCN(C(C=CC)=O)C2)CC2CC1CC2(F)F C(=O)(C1=CCCC1C)N1CC(F)(CNC(C2(COC)CC=CCC2)=O)C1 C1(C)(NC(C(C2CCN(C(Cc3cc(C)[nH]n3)=O)C2)C)=O)CCN(C)C1 C(=O)(C1Cc2ccccc21)NCC(CC(C)C)C(=O)NCc1ccnc(Cl)c1 Cc1cc(F)cnc1C(=O)N(C1CN(C(=O)CCC2(C)CCC(=O)N2)C1)C C1(O)(CC(=O)N(C(C)(CNC(=O)C(C)(C)N2CCCCC2)CO)C)CCOCC1 C(C(C)(O)CC(=O)NC(CNC(=O)Cn1cc(C2CC2)cn1)C(C)(C)C)OC N1(C(C(=O)NCCOC)=O)CC2CC(NC(C3(COC)CCCC3)=O)C1C2 C1(N(C(C(C)NS(CCC)(=O)=O)=O)C)CN(C(=O)CCCC(C)C)CCC1O N1(C(C(C2CCC(C)CC2)CC)=O)CCN(C(=O)OC(C)(C)C)CC1CO c1(C(N(CCCCNC(c2n(CC)ncc2)=O)C)=O)cccc2c1COC2 N1(C(Cc2c(C)non2)=O)CCCC(F)(CNC(c2sncc2Br)=O)C1 C1(NC(c2n(CC)ccc2)=O)CCC(C)N(C(=O)CCCC#N)C1 Cc1nc2ccc(CN3CCC(C(=O)NC(c4nccn4C)C)CC3)cc2o1 c1(C(=O)NC(C2CCN(C(CCC=C(C)C)=O)C2)C)[nH]cc2c1CCC2 c1(C(N(CCC2(C)CCCN2)CC)=O)ccc2oc(O)nc2n1.C(CCCl)N C(=O)(CCCCNC(=O)C1CC1)N(CC(CC)NC(=O)CCC1CCCCO1)C N#Cc1ccc(F)c(CN2CC(O)(CNC(c3nc(Cl)sc3Cl)=O)C2)c1 C1(CNC(c2c(C)n[nH]c2)=O)CCCCC1NC(c1ncccc1Br)=O c1(OCC)ccc(N)c(C(N2CC3(NC(=O)CN4CCN(C)CC4)CC2C3)=O)c1 c1(CN2CCC(NC(CC(C)n3cccn3)=O)CC2)cn2ccccc2n1 C(=O)(C(CCN(C)C)NC(c1c[nH][nH]c1=N)=O)N1CC(O)(COC)C1 C1(C)(C(C(=O)NC2CC2)N(C2CCOC2)CCN(C)C)CCCC1 CS(=O)c1ccc(C(=O)NCCCN(C(C2(C)CCNC2=O)=O)C2CC2)cc1 C(C(CC(F)(F)CNC(=O)NCc1noc2c1COCC2)OC)OC c1(OC)nn(C)cc1C(=O)NC(C1(O)CCN(C(C2CCCN2C)=O)C1)C c1(NC(C2N(Cc3c(C)c(Br)ccc3)CC(O)C2)=O)cc(Br)ccc1[N+](=O)[O-] Cc1nn[nH]c1C(=O)NC1CCCC1NC(=O)Cc1nocc1C(C)C N(C1CN(C(=O)CO)Cc2ccccc21)C(c1cn(C)nc1-c1ccccc1)=O C1(OC)CN(C(=O)CC2OCCC2(C)C)CC1NC(=O)CCCc1nncn1C c1(CN(C)Cc2ccccc2F)ccc(CN2CCCC2=O)cc1 C(C1c2ccsc2CCN1C(c1ccc2cccnn12)=O)NC(C(N)=O)=O N1(C(C2(COCC)CC2)=O)CCC=C(CNC2CCC(=O)NC2=O)C1 C1(C(=O)NCC(=O)NC(CCNC(C(C)c2cncs2)=O)(C)C)CCS(=O)(=O)C1 N1(C(C(C)OC)=O)CCC=C(C(=O)NC2CC(C(C)=O)C2(C)C)C1 c1(CC)cc(N)c(C(=O)NC2CCCN(C(C3CNC(=O)N3)=O)C2)c(F)c1 C(=O)(CCC(=O)N(C)C)NCC1(C(C)(C)O)CN(C(C2C(OCC)C2C)=O)C1 C(=O)(CCC(C)(C)O)NCC(C1CCN(C(C(OC)OC)=O)CC1)(C)C c1(C(=O)NC2CN(C(C=CC=CC)=O)CC2C)cccc2c1OCCCO2 C1(C(=O)NCCN(C(C2=C(C)CCCC2)=O)CCN(C)C)Cc2ccc(C)cc2S1 C(=O)(C(C#N)C(C)(C)C)N1CCC(CCNC(c2cc(COC)on2)=O)C1 C(C(C)(C)C(=O)N1CCCC(N(C(=O)CSc2cn[nH]c2)C2CC2)C1)OC(C)(C)C C1(CC(=O)NCC(=O)NC2CN(C(=O)CN3CCOCC3=O)C2)CCC1C1CC1 C1(COCCNC(N2CC(C(=O)OCC)C2)=O)CCOCC1 c1(C(=O)NCC2(OC)CN(C(c3cc(=O)n(C)o3)=O)C2)cc(C(F)F)ccc1F c1(C(=O)NC(C(C)NC(C(C)(C)NCC)=O)C)cc(OC)c2ccccc2n1 Cc1sc(-n2cnnn2)c(C(N2CCC(C)(CNC(=O)C=C3CCC3)C2)=O)c1C CC(C)C(C)CC(=O)N1CCC(Cc2cn(-c3cccnc3-n3ccnn3)nn2)C1 c1(C(N2C(C)CCC(NC(c3ncc(F)cc3F)=O)C2)=O)cccc2c1CCN2 C1(COC)CN(C(=O)C(O)CN2CCCC2)CCN1C(=O)C(F)CC(C)C CC(C)C(C(=O)NCCN(C)C(C1CCCN1Cc1ccsc1)=O)n1cncn1 N1(C(C(COCC)(C)C)=O)CCCCC(C(N2CCN(CC3CCC3)CC2)=O)C1 C1(C)(CN(C(C2(CC#C)CC2)=O)C)CCCC1NC(c1noc(CC)c1C)=O N1(C(C(C)O)=O)CCCC(C2CCCN(C(c3cc4cc(F)ccc4[nH]3)=O)C2)C1 c1(C(=O)NC2(CNC(C(CC(C)C)O)=O)CCCCC2)onc2ccccc12 c1(C(=O)NC(C)CNC(=O)CC2C(C)(C)C2(C)C)c[nH]nc1[N+](=O)[O-] c1(C(C(=O)NC2CCC2)N(CCF)CC)cnc(C(C)C)[nH]1 c1(C(N2CC3C(CNC(C(CCC=C)(F)F)=O)(C3)C2)=O)c(F)cc(C#N)cc1F C(CC(N)=O)(C(=O)NCC12CCC(CC1)CC2)NC(C(n1ccc(C)n1)C)=O Cc1ccccc1C1(NC(C2CC2C(=O)NCc2cnncc2O)=O)CCC1 c1(NC(CC)C(C)(O)CC)ccc2c(C)nn(-c3ccccc3)c2n1 CC(C)C(C(C)C)C(N)C(=O)NCC1(CN2CCOCC2)CC1 C1(OC)(CNC(=O)NC(C(F)(F)CO)C2CC2)CCCS(=O)(=O)C1 c1(C(=O)NC(CCCNC(c2nnn(C)n2)=O)(C)C)ccc(C#CC2CC2)cc1 C1(CNC(c2c(C)snn2)=O)CN(C(c2cc(Cl)ncc2N)=O)C2COCC2O1 N1(C(c2cc(COC)oc2C)=O)CC2CC(NC(=O)Cc3cccnc3)C(C2)C1 C(=O)(C(C)(O)C(C)(C)C)N(CCC(C)NC(c1c(C)c(Cl)cnc1)=O)C c1(C(N(C2CCN(C(c3cnccc3Cl)=O)CC2)CC#C)=O)c(C)cccc1O C(=O)(CC1=CCOCC1)NC1CN(C(c2c(C)nn(-c3ccccc3)n2)=O)CC1O N#Cc1ccc(OCC(N2CC(CO)C3CC23)=O)cc1.c12cccc(c1)C(=O)N2 c1(CC(=O)NCC2(CNC(C3(O)CCSC3)=O)CC2)coc(C(F)F)n1 C1(C(=O)NCC2C(NC(C3N(C)CC(F)C3)=O)CCCC2)CC2COCC2C1 c1(OC)cc(C(=O)NCCCN(C(=O)CC2CCC(C)O2)CCO)ccc1C c12ocnc1NC2.C1(NC(=O)NOC2CCOC2)C=CCOC1 C1(C(=O)NCC2(OC)CN(C(=O)C=CCN(C)CC)C2)CCc2nnnn2CC1 c1(NC(C(c2cccs2)NC(C(C)=CC(C)(C)C)=O)=O)ccc(Cl)nc1 CN1CCC(CCC(=O)NC2(CNC(C3CCC3(F)F)=O)CCCC2)CC1 C1(C(=O)O)CC(NC(=O)CC2(OC)CC(NC)C2)CN1C(=O)CCSCC C1(CNC(=O)OC(C)(C)C)CCC(CNC2CCN(S(=O)(=O)C3CC3)CC2)CC1 c1(C(N2CC(NC(c3ncc(C)nc3)=O)C(F)C2)=O)c(Cl)ccc(Cl)c1F N1(C(C(C)=C2CCC2)=O)CCC(CCC(=O)N2CC(CC(F)F)C2)CC1 C1(C(N2C(C)CC(CNC(CCc3onc(C)n3)=O)C2)=O)CC2(CC2)CN1C C1(C(=O)NC2C(NC(c3ccc(OC)nc3)=O)CC2)CC(C2CC2)=NO1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CC2CC(C1)N2C(=O)Cn1ccnn1 C1(C2CCN(C(=O)CC3CC3)C2)(NC(=O)C(O)CC(F)F)CC1 C1(C(N(CCCN(C)C(C2(CO)CCCCC2)=O)C)=O)CCCC(=O)CC1 c1(C(=O)NC2CN(C(C34CC(COCC)(OC3)C4)=O)CC2C)cc(F)ccc1O c1(C(=O)NC2(CC(=O)NC(C3CCC3)C)CC2)cn(C)cc1C(F)(F)F C(C1CCCCC1)=CC(=O)NCC(CNC(CC1CCN(C)C1)=O)(C)O N1(C(c2c(CC)noc2C)=O)CCC2(CCC(NC(=O)C=Cc3ccoc3)C2)C1 N1(C(c2nc(C)n(C)c2)=O)CC2CCC(C(=O)NCC3CCCC(C)(C)C3)(C2)C1 Cc1cc(C(=O)NCCC(C)N2CCCC2)c2cccc(O)c2n1 C(=O)(C(C)(C)CN(C(=O)Cc1cc(C)on1)C)NCC(C(C)C)OC C(=O)(C#CC1CCOCC1)N1CCC(C(C(N2CCOCC(C)C2)=O)F)C1 C(=O)(C1CCc2snnc21)N(C1CC2CN(C(COCCCCCC)=O)CC21)C C1(N(C(C2CN(C)C2)=O)CC2CC2)CCN(C(=O)C=Cc2ccc[nH]2)CC1 C(=O)(C(C(C)C)SC)NC(C(=O)N1CC(F)(CC(=O)OC)C1)Cn1cccn1 C1(NC(C(C)(C)n2cnnn2)=O)CCOCC1NC(c1cnn(C(C)(C)C)c1Cl)=O c1(C(N2CC(N(C(c3c(C)onc3)=O)C)C2)=O)ccc2[nH]ccc2c1F C(CC(C)C)(C(=O)Nc1ccc(CN2C(CC3CC3)CCC2C)cc1)OC(C)=O C1(N)(NC(=O)COCC(=O)NCC2C=CCCC2)CCOC1.C(COCC)OC S(=O)(=O)(c1ccc(NC2CCCCC2)c(F)c1)NC1(C2C(OC)CCO2)CC1 N1(C(C=CCCC(C)C)=O)CC2(C1)CN(C(c1occc1C1CC1)=O)CC2CO c1(C(=O)OCC)c(NC(C2(C)CC(NC)CCO2)=O)sc2c1CCC(C)C2.O Cc1noc(C)c1-n1nc(-c2cncs2)nc1Cn1nnc(-c2ccsc2)n1 C1(C(N2CCCC(CNC(C3(C)CS(=O)(=O)C3)=O)C2)=O)CCc2nccn2CC1 Nc1ccc(C(=O)NC2(CNC(C3CCCOCC3)=O)CCC2)c2cnccc12 C1(C(=O)Nc2ccc(C(C)NC(C(COC)OC)=O)cc2)SC2C=CC1CC2 C1(NC(C=C(CNC(C(CC)N(C)C)=O)C)=O)COC2(CCC2)C1 C#CC1C(C(=O)NC2CN(C(c3c[nH]nc3C3CC3)=O)CC2CCC)C1(C)C c1(C(=O)NC2(C)CC(NC(CC3C(C)(C)C(O)C3)=O)C2)c[nH]c2cccc(F)c12 C1(CC)(CNC(=O)CC(C)F)CCN(C(c2cn(C)nc2C2CCC2)=O)CC1 c1(C(N2CC(CN(C(CC(CC)C)=O)C)C2)=O)cnc(Cl)cc1Cl C=C(CNC(=O)CCN1CCC(F)C1)CCNC(c1c[nH]cc1C(C)(C)C)=O c1(CCC)nc(C(=O)NCC(C)(C)CNC(=O)Cc2nc[nH]n2)co1 c1(C2N(C(C34CC(C(F)(F)F)(C3)C4)=O)CC2)ccc(-c2nn[nH]n2)cc1 C1(C(=O)NCCC2CCN(C(C(C)(C)CC3CC3)=O)CC2)CC2C(C1)C2(F)F CC1CN(Cc2c(-c3c(C(=O)NC(C)(C)C)cc(F)cc3)cncc2)CC(C)O1 C#CC1(C(=O)NCCOCCOCCNC(C2C3CCCC23)=O)CCC1 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NCC1(F)CC(NC(C(C)N(C)C)=O)C1 c1(CNC(NC(C)CC2CCN(C3CC3)CC2)=S)csc2ccc(Cl)cc12 C1(NC(CN2CC(C)(OC)C2)=O)CN(C(=O)CC(C)n2ccnc2)C2(CCC2)C1 c1(C(N2CCC(F)(CNC(c3cc(C)oc3)=O)C2)=O)c(S(N)(=O)=O)cnn1C c1(OC)ccc2ncnc(NC3CCCCC3C(=O)NC3CC3(F)F)c2c1 C(=O)(C(O)CN(C(=O)CCOC1CCCC1)C)NCC(C)CC1CC1 CCCCC(C)C(=O)N1CCC(CNC(=O)C(=O)NCCOCCCC)CC1 C1(N(C)C(C2CCC(=O)N2)=O)CCCCC1N(C(=O)C=CSCc1ccco1)C c1(C(N(CCCCC)C(C)C)=O)cc(C)n(C2CCCOC2)c1C C(=O)(C(F)C(=O)N1CC(OC)C(NC(c2ccc(O)nc2)=O)C1)OCC Cc1nnc2n1CCN(C(=O)C#CCNC(C1CC3CCC1CC3)=O)C2 N1(c2ccnc(NCCCCC(CC)C)n2)CCC2(CCCN(C)C2)C1 N1(C(CC(COC)NC(=O)C2=NOCC2)=O)CC2(CCC2)CC1C c1(-c2c(C)cc(=N)[nH]c2)nn(C)c2c1C(NC(=O)Cc1cccc(F)c1)CC2 Cc1cc(C(=O)NC(C2CCCN(C(=O)CCP(C)(C)=O)C2)C)c2nccn2c1 C1(NC(COC)=O)CCC2(CC1)CCN(C(c1n[nH]c(C)c1Cl)=O)CC2 CCC(C)C(C(=O)NCC(C)C(C)(C)C)NC(=O)OC(C)(C)C c1(C(N2CC3C(C(N4CC5(CCCCC5)C4)=O)(C3)C2)=O)ccc2c(c1)CCC2 n1(CC(=O)N(CC(=O)NCC(C)(C)c2cccs2)C2CCC2)cnnc1O C(C(CC(C)C)C(=O)NCCCC1C=NNC1=O)NC(CCC(C)=O)=O C=CCCC(O)CNC(=O)CCC1(NC(C2C3CCCC23)=O)CCC1 C1(NC(=O)Cc2ccoc2)CC(O)CN(C(c2cnn(CCO)c2)=O)C1 C=C1CC2(C1)CC(C(=O)NC(C)C(CO)NC(=O)CS(=O)(=O)Cc1cccs1)C2 c1(OC)ccc(CN2CC(C)CC2C(=O)Nc2ccc(C(C)C)nc2)c(Cl)n1 c1(CC)sc(C(=O)NCC2(F)CC(NC(c3cn(C4COC4)nn3)=O)C2)cc1C C1(C(=O)NC2(CC=C)CCCC2)CC(NC(c2ccc(=N)[nH]c2)=O)CCO1 c1(OC)ccnc(C(=O)NC2CCN(C(c3ccc(C(F)(F)F)[nH]3)=O)C2)c1 c1(C(N(CC(CN(C)C(c2nc(Cl)cs2)=O)O)C)=O)cccc2c1OCCC2 C(C(C)(C)CCNC(=O)C(C)(C)c1cnn(C)c1)NC(C1CCC(C)C1)=O c1(CNC(C2(F)CCCCC2)=O)ccc2c(c1)CN(C(=O)C#CC1CCCO1)C2 CC1CN(C(C2(Cc3ccc(O)cc3)CC2)=O)CCCN1C(C1CC1(Cl)Cl)=O C1(SCC(=O)NCCCNC(=O)CCc2ccc[nH]2)CCOC1=O C1(C(=O)NCC2(F)CC(CNC(C3CC(F)(F)C3)=O)C2)(CC)CCNC1=O Cc1nc(NC(=O)NC2CC(Cn3cccn3)C2)oc1C C1(NC(C2C(OCC)C2)=O)CCN(C(=O)Cc2nnc(O)s2)CCC1(F)F c1(CCCCC)nc(-c2ccnc(C)c2)n(C2CCOC2)n1 C1(NC(=O)COCC2CCCC2)CC2(CCN(C(c3ccc(Cl)nn3)=O)CC2)C1 C12(C(=O)NCC(CNC(c3cc(N)cc(F)c3)=O)CO)C3CC(CC13)C2(F)F C=CCC(C)C(=O)NCCCCN(C(=O)Cc1nc(C)c(C)[nH]1)C N1(C(C)=O)CC(C(N2CC(C(C)NC(=O)C(C)c3ccco3)C2)=O)C1 c1(C(C)C)ccnc(C(c2nnnn2C(C)C)NC(c2cccc(Cl)c2)C)n1 CC1CN(C(c2cnc(O)s2)=O)CCCN1C(c1cn(CCF)nn1)=O N#Cc1ccc(NC(c2cccc(NCc3ccc(O)c(F)c3F)c2)=O)c(O)c1 c1(CC)ccccc1CN(C)CC1CCCCN1S(=O)(=O)CC(C)O c1(CCC(=O)NCC2C(CNC(C(C)(C)CO)=O)C2)ccc2ccccc2c1 CC1c2c[nH]nc2CCC1C(N1CCOC(CN(C(=O)CSC(F)(F)F)C)C1)=O c1(C(=O)NC2C(CNC(c3cc(F)cc(Cl)c3)=O)CC2)ccnc2ccccc12 Cc1noc(C)c1C(N1CC(CNC(c2ccoc2C2CC2)=O)C(O)C1)=O N1(C(C(C(=O)OCC)F)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)CC)CCO2 N1(C(c2c(F)ccc(OC)c2)=O)CC(C)OC2(CCN(C(=O)C(C)(C)OC)C2)C1 c1(SCCCC)cccc(C(N2CC3CC3(NC(C3CCN(C)CC3)=O)C2)=O)c1 C1(CNC(N2C(C(C(=O)OC)(C)C)CCC2)=O)CC=C(C)CC1 C#CCC(C(=O)N(C1CCC1)CCOC)NC(c1ccn(CCF)n1)=O C12(NC(CCC=C=C)=O)CCCCC1N(C(c1cncc(C(N)=O)c1)=O)CC2 C1(CC#C)(C(N2CC(C)(CF)C2)=O)CCN(C(C2OC3CCC2C3)=O)C1 c1(OC)cc(C=CC(=O)N(C)CC2CCCN2C(c2csc(C(N)=O)n2)=O)sn1 Cc1ccc(F)c(C(C(=O)NC(c2ccccc2)C)N(CC(F)Cl)C)n1 c1(OC)cc(=NC(=O)CC2(CNC(=O)CC3(C)CCOCC3)CCC2)[nH]n1C N1(C(C(C)Oc2ccc(F)c(F)c2)=O)CC2CCCOC2C1 N1(C(c2n[nH]cc2I)=O)CC2COC(C1)C2O N1(C(CCCc2onc(C)n2)=O)CC2CC(NC(C34CCCC(C3)OC4)=O)C1C2 Cc1cc(F)c(C(=O)NC2CC3CN(C(=O)CN4CCCCC4)CC3C2)cc1Br c1(NC(CC)Cn2ccc3ccccc3c2=O)cc(Br)cc([N+](=O)[O-])c1 c1(OC)nc(C)ccc1C(N1CCC(CO)(NC(C2C(C)(C)C2(F)F)=O)CC1)=O C12CCN(CC1)C(=O)CC(N)Cc1noc2n1.CC(C)(F)F c1(OC)ccc(NC(=O)C(CC(C)=O)NC(=O)CCOCC(F)(F)F)cc1C C1(F)(CNC(=O)CSCC(F)(F)F)CCC(NC(=O)C2CC2)C1 C#CCCCCCCC(=O)N1CCC(C)C(CNC(c2cnn(C)c(=O)c2)=O)C1 CCCC(CC1CC1)C(=O)NCC1CCC1NC(=O)C(OC)OC c1(N(C)C)cnc(C(=O)NC(C)(C)CNC(C2CC2c2cnnn2C)=O)nc1 C1(CC(C)NC(=O)C(C)(O)C2CC2)CCN(C(=O)C(F)CC2CC2)CC1 C(=O)(CC(C)(C(F)F)N(C)C)N1CCC(NC(c2cnc(C(C)OC)s2)=O)CC1 CC(C)(C)CC(F)C(=O)N1CCCC(CC(=O)NCCC(O)CCO)CC1 C(=O)(C#CC1CCCCC1)N1CCCC(NC(C(CN(C)C)(C)C)=O)C(F)C1 c1(C(=O)NCC(C2CCC2)NC(=O)C(O)C2CC2)n[nH]c2c1COCC2 c1(OC)ccc2c(c1)CCC2N=c1[nH]c(=NCC(C)CN(C)C)[nH]c2c1COC2 c1(C(=O)NCC2CN(C(C3C(C)C3)=O)C2)ccnc(CN(CC(F)(F)F)C)c1 CCC(CC)CC(=O)NC12CCN(C(=O)Cn3nc(C)cc3C)CC1C2 C(=O)(C1COc2ccccc21)NCCN(C(=O)C(C)(C)Cc1ccccc1)CC C(C(CC(C)C)C(=O)NC1CC(O)(CNC(c2cccc(CC#N)c2)=O)C1)OC C(CC(CNC(c1cc(C(N)=O)co1)=O)NC(=O)CC1CC(OC(C)=O)C1)OC c1(CN2CC3(C(C(=O)Nc4c(OCC)ncnc4)C3)C2)ccnc(F)c1Cl CC(CCCN=c1ccc(C(F)(F)F)n[nH]1)NC(=O)Nc1cc(Cl)on1 c1(C(N2CCCCC(NC(C(CC)F)=O)C2)=O)cnc2ccccc2c1C N1(C(C(C)OCC2CC2)=O)CCOCCC1C(=O)NCC=CC1CC1 c1(CCC)cc(C(=O)NC(CNC(=O)CC2CCCCC2)CC)no1 CC1=C(C(=O)N2CCN(C)C(C)C2)CCO1.c12ccccc1CC(=O)N2 c1(CC(N2C(C)CC(C(=O)NCC3(OCC)CCC3)C2)=O)ccc(Cl)c(F)c1 C1(CNC(c2nc(SC)sc2)=O)CC2CCC1N2C(=O)CSCc1nccn1C c12cnc(s1)CNC2=O.C(C(C)(CNSC)OCCC(=O)OC)SCC.C1CO1 N1(C(C2CN(C)C2)=O)CC2CC2(NC(=O)CCCc2nccs2)C1 C1(NC(CC2CCCC(C)C2)=O)C2CC3C1C3C2C(=O)NCC(C)(C)F N(C(=NCCC1CCCO1)NCCc1cnccn1)CC(c1ccc(C)cc1)O c1(C(=O)NCC(CC(C)C)NC(C2(N(C)C)CC2)=O)coc2cc(F)ccc12 N1(C(C(C)(C)OC)=O)CCC(C)(CC(=O)N(C)CC2CCC(C)CC2)C1 n1(CC(=O)NC(C2CN(C(=O)COc3ccc(Cl)nc3)C2)C)cccnc1=O C1(O)(CNC(C2(CC)CC2)=O)CCCN(C(C2CC(O)(c3ccncc3)C2)=O)C1 C1(NC(C(CC)NC(N)=O)=O)CC2(C1)CC2NC(=O)C(COC(C)(C)C)N(C)C c1(NC(N2CC(C)(C)C(Cc3ccccc3)CC2)=O)ccc2c(c1)CCOC2 c1(C(C(C)C)NC(N(CCCCCC=C)C)=O)c(C(F)(F)F)cccc1C Cc1nsc(C)c1C(N1CC(CCCCNC(C2CCCCN2C)=O)C1)=O N1(C(CC(=O)OCC)=O)CC(NC(=O)C(C)OC)C(C)C1 c1(N2CC(C(C)NC(=O)CCC(F)(F)F)C2)cc(C(F)(F)F)ncc1[N+](=O)[O-] C#CC12C3C4C1C1C2C3C41C(=O)NC1CC(F)CN(C(=O)C(C)NC(C)=O)C1 C(C)(C(CC(=O)N1CCCCC1C)NC(=O)CCN(C)CCO)OC C1(CC(=O)NC(C)C(C)(C)NC(c2cc(N)ccc2F)=O)Cc2ccccc2O1 C1(C(=O)NCC2CC23CC3)CC2CCCC2N1C(c1ccccn1)=O n1(CC)cccc1C(=O)N(CCNC(C1CCCN1C1CCCCC1)=O)C1CC1 C1(CNC(=O)CC2CC(F)(F)C2)CC(F)CN1C(=O)C(F)CC1CCOC1 C1(O)(CNC(CCC(C)OCC)=O)CCCN(C(=O)COCCCN(C)C)C1 C1(CC)CN(C(=O)CC2CCCOC2)CC1C(=O)NCC1(CC(C)C)CC1 c1(C(N2CCC(C)C2CNC(=O)CCc2cocn2)=O)cc2n(n1)CCO2 c1(C(=O)NCC(C)N(C(C2CCN(C)C2)=O)CC)cccc2occ(Br)c12 CC1CCC=C1C(=O)NCC1CC1C(=O)NCCCOCC1CCC1 N1(C(C(C)(c2ccccc2)OC)=O)CCC(CNC(=O)CC(C)(C)C2CC2)CC1 N1(C(CC(CCC)O)=O)CCCC2(CCN(C(C3(C)CC3C)=O)CC2)C1 N1(C(C(c2cn(C)nc2)(C)C)=O)CC2C(CNC(c3ccc(CF)cc3)=O)C2C1 c1(OC)c([N+](=O)[O-])ccc(CNC(=O)C(=O)NCC2CCCC(F)C2)c1O CC(C)=C=CC(=O)NC12CC(CNC(C3CC3(F)Cl)=O)(C1)C2 c1(C(=O)NC(C(C)(C)C)CNC(c2scnc2C(F)(F)F)=O)cc(F)cc(Cl)c1 c1(OC)ccc(F)c(CNCc2ccn(CC(C)C)n2)c1F C1(C(N(C)CCNC(=O)Cc2ccccc2)=O)Cc2nncn2C1 C1(CC(=O)N(CCNC(=O)CCCC(F)F)C2CC2)Cc2ccccc2C1 c1(CCNC(N2C(C)(COC)CC2)=O)cccc(N(C)C)c1 c1(CC)[nH]ccc1C(=O)NCC(C(=O)NCCN1CC=CCC1)N(C)C c1(C(N(C2CCN(C(=O)C=C(C)C3CC3)C2)CCC)=O)cc(OC(F)F)ns1 N1(C(CCC(CC)OC)=O)CCOC2CCN(C(c3ccc(F)s3)=O)CC12 c1(SC)ccccc1CC(=O)NCCNC(=O)CNC(C)=O.C1CC(C)N1 Cc1cc(CN2CCOC(CC(=O)NC3CNC(=O)C3)C2)ccn1 N1(C2CCCN(C(C(C)O)=O)C2)CCN(C(c2cc(=O)n(C)cn2)=O)CC1=O C(CN=C(NCC(CO)C1CC1)N1CC(O)C(C)(C)C1)OCCOC C1(C(=O)NCC23OCC(NC(C(C)OC)=O)(C2)C3)CC2CCCC2C1 CC1(C(=O)NCC(O)CCNC(=O)C=CCF)CCCCO1 C(=O)(C(C(C)(C)C)C1CCC1)NCC(C)CN(C)C(C1CC(=O)NC(=O)C1)=O C1(c2n(C)ncc2)CN(C(C2OCCCO2)=O)CCN1C(=O)C(N)=O N1(C(CN2CCC(C)CC2)=O)CC2CC(C(N3CCC(CO)CC3C)=O)(C2)C1 c1(C(=O)NCC2C(CNC(=O)CCCn3ccnn3)C2)ccccc1OC1CC1 Cc1cccnc1CCC(=O)NCC(C)NC(c1ccccc1CC#N)=O N1(C(CN(C(CC(COC)(C)O)=O)CC2CC2)=O)CCN(C)CC(O)C1 c1(C(=O)NC2CC(NC(CCS(C)=O)=O)C(O)C2)c(N)cccc1F C(CC(=O)NC(C1CCN(C(c2c[nH]c(=N)s2)=O)C1)(C)C)(C(C)C)OCC CCCCC(C)C(=O)NCC(CC(=O)NCC(F)(F)C(F)F)OC CC(C)CC(C(=O)NC1(C2CCCN2C(c2ccnnc2S)=O)CC1)C(C)C C(=O)(C1=CC2CCCC12)N1CC2C(NC(CCc3cc(OC)no3)=O)(C2)C1 n1(CCNC(C(C2CCN(C(C=CC(CC)C)=O)C2)C)=O)cnccc1=O CC(N=c1nc(N2Cc3ncsc3C2)c2cccc(F)c2[nH]1)c1cnn(C)c1 C1(C(NOCC(=O)OCC)=O)CC(N=[N+]=[N-])CN1C(C1CC(CF)C1)=O C1(C(N(CCNC(Cc2cccc(SCC)c2)=O)C)=O)CC2COCC2C1 N#CC1(CCNCc2cnn(-c3ccc(F)cc3)c2)CCNC1 N1(C(C2CC(OCC)C2)=O)CCCC2(C1)CN(S(C)(=O)=O)C2 C1(C(=O)NCCNC(CCC=CC)=O)CC(c2cccc(Cl)c2F)=NO1 N1(C(COC2CN(C(C3C(C)OCC3)=O)C2)=O)CCOC(C(C)(C)C)C1 c1(C(=O)NC2(OCC#C)CC2)ccc(C2CC2)cc1.C12COC(C1)CNC2=O c1(C(=O)NCCC(=O)NC(C)C)cnc(CNC(C2(C)CCCC2O)=O)nc1 C(c1cc(F)cc(F)c1)=CC(N1CCC(NC(CC(=O)NCC)=O)C1(C)C)=O Cc1cc(C(=O)NC2(C)CCN(C(=O)C(F)C3CC3)C2)c2cccc(C)c2n1 C(C)(CCCCC(=O)OC)NC(CN(CCCCC)C)=O CC1(NC(=O)CCSC(F)(F)F)CN(C(=O)CCc2cscn2)C1 c1(OC)cc(CNC(=O)CN(C(=O)C(n2ccc(SC)n2)C)CC(C)C)ncn1 C1(NC(c2c(CC)ncnc2)=O)CCC2CN(C(=O)CC(=O)OC(C)(C)C)CC12 N1(CC(N2C(C(=O)NC3CCN(C)C3=O)CC=CC2)=O)C(=O)CCCC1=O c1(C(N(C2CN(C(c3c(C)c(Cl)ccn3)=O)C2)C)=O)ccc2c(n1)CCCN2 C1(C(=O)NC2CC(CO)C2)COC2CN(C(=O)CC3CCOC3)CC12 c1(C(=O)NC(C2CN(C(=O)CCc3cn[nH]c3)C2)C)cc(C(F)(F)F)cs1 N1(C(C(C(C)C)N(C)C)=O)CCOCC(NC(C2(c3cccnc3O)CC2)=O)C1 C1(CNC(COCC)=O)CCCC1C(=O)N(C)Cc1ccn(CC)n1 C1(C(N(C(CC)C)C)=O)CC2CCN(C(=O)CNC(C3CCCC3)=O)CC12 c1(C(N2CC3C(NC(CCC(CC)CC)=O)(C3)C2)=O)ccc(F)c(S(N)(=O)=O)c1 C1(C(N(CCNC(C(CC)n2nccc2C)=O)CCOC)=O)COC(C)(C)CO1 O=C1CN(C(=O)CCS(=O)(=O)N2CCCC2)C2CCN(C(=O)C(O)C3CC3)CC2N1 C#CCC(C)C(=O)N1CC2(NC(c3sc(OC)nc3C)=O)CC1C2 C(=O)(CCC(=O)N(C)C)N(C)CC1N(C(C2N(C(C)=O)CSC2)=O)CCC1 N1(C(C(C)CN(C)C)=O)CCCC1(C)CNC(C1(n2cnnn2)CC1)=O N1(C(C(C)OCCN(C)C)=O)CCCC1(C)CNC(=O)C=Cc1ccn(C)c1 c1(NC(C2CC(NC(C=CCOC)=O)C2)=O)cc(Cl)cc(Br)c1C Cn1cc(S(=O)(=O)NCCNC(CCC(=O)O)C(=O)O)cn1 c1(C2CC2)ccn(C)n1.c1(CCC(=O)N2CCC(=O)N(C)C2)cccnc1 c1(C(N(CCNC(C(CC#C)C2CC2)=O)C)=O)ccc(F)cc1C#N C1(C(=O)NCC#CCNC(CN2CC(CC)C2)=O)(C(C)C)CCCO1 c1(OC)ccc(C(=O)NCC(F)CNC(=O)CCc2ncc[nH]2)cc1C1CC1 C(=O)(C1Cc2c(Cl)cccc21)NC(CNC(c1ccc(CC#N)cc1)=O)C1CC1 C#Cc1cncc(C(=O)NCC2CCC(C)N(C(=O)C#CC(C)(C)C)C2)c1 N1(C(C(C)OC(c2c(C)onc2)=O)=O)CCC(C)N(C(=O)OC(C)(C)C)CC1 N1(C(CC2(N(C)C)CCC2)=O)C2CCC(C(=O)NC34CC3CN(C)C4)C1CC2 c1(C(=O)NC(c2ccccc2)CNC(=O)CCC2CCCO2)ccn(C2CC2)n1 c1(CNc2c(C(=O)OC)c(OC)ns2)ccc(CN(C)C)nc1O N1(C(c2cccc(NC)n2)=O)CCC2CN(C(c3cncnc3)=O)CCC12 c1(C(=O)NC2C(NC(=O)C3=CCOC3)CC2)csc2ccccc12 CCC(CCCC(=O)NCc1ncccc1O)NC(=O)Cc1ccn(CC)n1 C1(C(=O)NC2C(NC(C(Cc3ccsc3)NC=O)=O)C2)CC2CC1C1CC21 C1(=CC(N2CC(C)N(C(=O)CS(C)(=O)=O)CC2)=O)CCCCCC1(F)F N1(C(c2cncc(SCC)n2)=O)CCCCCC1CNC(C1CCSCC1)=O c1(C(N2CC(C)C(NC(C3CC(C)(C)C3)=O)C2)=O)ccc([N+](=O)[O-])cc1N c1(CCCNC(C(=O)NCC(c2cncnc2)C)=O)c(F)cccc1F C1(NC(Cc2c(OC)nccc2)=O)CCC2(CC1)CN(C(C1CC(C)=NO1)=O)C2 C1(NC(C=C(CC)CC)=O)CC(O)CN(C(=O)Cc2cnccc2C)C1 N1(C(C=Cc2n(C)cnc2)=O)CC(C2(NC(=O)Cc3ccc(Cl)cc3)CC2)C1 c1(C(=O)NC(CNC(c2c(C(C)C)ocn2)=O)C)nn(C)c(Cl)c1Cl C1(Nc2c(C)noc2C(N)=O)CC2CCC(C1)O2 C(C)(C(C)CC)(c1ccccc1)NCc1cn(CCC=C)nn1.C(C)(C)S C1(CNC(NC2C(C)C2)=NCCN2CCCC2=O)CC2CCC(C1)N2C CCC(C(=O)N(C)CCN(C(c1cnn(-c2cccc(F)c2)c1)=O)C(C)C)C(C)O CCC(CC(F)F)C(=O)N1CC2(CCC2)CC1CNC(c1cnc(S)nc1)=O C1(NC(C(c2ccccc2)OCC)=O)CC2C(NC(C3CC3CC(C)C)=O)C2C1 C1(C(=O)NCCCC(=O)N(C)C)CCC2CCC1N2C(=O)C=C1CCC1 c1(CC)[nH]nc(C(=O)NCCCOCCNC(=O)CCNC(=O)CO)c1Cl c1(C(=O)NCCC2CCCN(C(C(C3CC3)OCC)=O)C2)cncc(N)c1C c1(NC(CCCC)COC(c2ccc(C)cc2Br)=O)ncnc2cccc(F)c12 n1(CC(N2C(CCNC(C(F)=CC)=O)CCCC2)=O)cc(Br)c(O)nc1=O C12(NC(C3C4CC4C4CC34)=O)CCC(CC1)N(C(=O)CCCN1CCCC1)C2 C1(CC(=O)N(CC(C)C)CC#C)CCN(C(C2CC3(CC3)CO2)=O)CC1 C(c1ccc(Br)cc1F)=CCNC(c1ccc(Nc2n[nH]c3c2CNC3)nc1)=O Cc1cccn2cc(C(=O)NCC=C3CCN(C(=O)COCC(C)C)CC3)cc12 C1(C)(COC)CCCC1NC(=O)CC1CCCN1C(=O)C(C)C1CCC1 C(=O)(C1=NOC2COCC12)NC1CC(NC(=O)Cc2ccc(Br)cc2)C1 Cc1cc(CC(N2CC(O)(CNC(=O)CCOc3ccccc3)C2)=O)ccc1O N1(C(C(=Cc2cccs2)C)=O)CCC(NC(=O)CC2CCCN2C(C)C)C(O)C1 c1(C(=O)NC(CNC(c2c(C)cccc2)=O)C2CC2)ccnc(C)c1N CC(C)(C)CC(O)CNC(C1CCCN1C(C1OC2CCC1C2)=O)=O c1(N2CC(NC(c3cnn(C(C)C)n3)=O)C(C)(C)C2)ncc(Br)cc1[N+](=O)[O-] CCC(O)C(C)C(=O)N1CC(CNC(=O)C(F)(F)CC2CC2)C(C)C1 C1(C)(C(N2CC(CNC(C#CC3(CC)CC3)=O)N(C)CC2)=O)CC(C(C)C)=NO1 C(=O)(C(F)C(=O)N1CCCCC1CCNC(c1cnc(S)n1C)=O)OCC CC(C)(C(=O)NC1CC(NC(c2ccc(Cl)c(C3CC3)c2)=O)C1)C(N)=O N1(C(c2nn(C)cc2Cl)C(=O)NCC=C)CCCC2(F)CCCC12 N1(OC)CCC(CNC(=O)Nc2ncc(Nc3cccc(F)c3)s2)CC1 N1(C(C(CC)OC2CCCCC2)=O)CC(NC(c2csc(Cl)c2Cl)=O)C(C)(C)C1 CCS(=O)c1ccccc1C(=O)NCC1CCN1C(=O)CC1CCCCC1 C1(CN(C(CCNC(=O)OCC)=O)C)CCN(C(c2ccc(OC)o2)=O)CC1 S(=O)(=O)(c1ccc2[nH]c(=NC3COC(C)(C)C3)ccc2c1)NCCCC(C)O c1(C(=O)NCCN(C(C2CC2C2CCCO2)=O)C2CC2)c(Cl)ccc(Cl)c1O N1(C(c2ncoc2C)C(=O)NC(CC)C)CCCCCC1c1ccccc1 c1(NCCC(=O)NC(CC)CNC(C2CCC3(CC3)C2)=O)oc(C)nc1C#N C1(CNC(COCCCN=[N+]=[N-])=O)CC(C(=O)NCCS(C)(=O)=O)=NO1 N1(C(CN(C(c2cc(CC)[nH]n2)=O)C)=O)CCN(C(c2cc(C)[nH]c2C)=O)CC1 Cc1cccc(Br)c1C(C(=O)NC1CSC1)NC(=O)CC1OCCC1(C)C N1(C(CC(C=C)C)=O)CCN(C)CC1C(=O)NCCCN1CCC1 C1(NC(c2nc(C)[nH]c2C(F)(F)F)=O)CN(C(c2cncnc2C)=O)CC12CC2 C1(C(N2CCC(CNC(c3ccnc(C)n3)=O)C2)=O)CC2COCC2C1 N1(c2ccnc(C(CC)C)n2)CCC2(CCN(C(=O)CCc3cncn3C)C2)C1 N1(C(c2cccc[n+]2[O-])=O)CCCC2(CCN(CC=C(Cl)Cl)C2)C1 C(C(F)C(=O)NC1(CO)CN(C(=O)CC2OCCCO2)C1)N(CC)CC C(=O)(C(C)(C)C(=O)N(CC(C)N(C(=O)CC1CCC(=O)N1)C)C)OC N1(C(C2CC(CNC(c3cccc(C)c3O)=O)OC2)=O)CCOC(C)(C)C1C Cc1cc(C)c(NC(C2CCCCC2NC(c2ccc(F)c(Br)c2)=O)=O)cc1Br c1(C(N2CCC(C)(OC)C2)=O)cnn2cccc(-c3cc(C)cnc3F)c12 C1(NC(C(COCC)NC(C2CCC(=O)N2)=O)=O)CC(CO)C12CCC2 C12(NC(C3N(S(CC)(=O)=O)CCC3)=O)CC1CN(C(=O)CCSCC(N)=O)C2 Cc1nc2cc(NC(C3CCC(NC(c4n[nH]c(C)c4C)=O)CC3)=O)cnc2[nH]1 CCS(=O)(=O)CC(=O)NCCCCC1CCN(C(c2cccc(C)c2Cl)=O)CC1 C1(NC(Cc2cn(C)nc2)=O)C=CCCC1C(N1CCC1C(C)O)=O c1(C(C(=O)NC)N(C2CCN(CC)C2)C)ccc(Cc2cccs2)cn1 CC1=NN(C)C(=O)C1CC(=O)NC1CC(NC(=O)C=CC=C(Cl)Cl)C1 c1(C(N2CCN(CC(=O)NC(C)C(=O)O)CC2)=O)cc(F)cc(F)c1 C1(C(N(C)C)=O)CCC(C(=O)NCC2COCCN2C(c2ccc(C#N)o2)=O)CC1 c1(CC)cc(C(N2CCCC(NC(c3ccc(SCCO)cc3)=O)C2)=O)sc1C Cc1nc(=N)[nH]c(=NCC2(c3ccc(Cl)cc3)CC2)[nH]1 CCC(CC(=O)N1CCCC(O)(CNC(=O)CN2CC3CC3C2)CC1)C(C)C c1(C(=O)NC(CCCNC(C2(CCC=C)CCCC2)=O)C)cccc(O)n1 C1(CCC)CN(C(=O)CC(C)SC)CC1NC(c1cc(C(CC)CC)no1)=O c1(SC)ccc(O)c(C(=O)NCC2CCCN2C(C2CCC(N(C)C)CC2)=O)c1 CC1C(C(=O)Nc2nnccc2C(F)(F)F)CCN1C CCC(C(=O)N1CCC(N(CCO)C(c2coc(COC)n2)=O)C1)C(F)(F)F N1(C(C2(OCC)CC2)=O)CCC2(CCCN(C(C3COCCC3(F)F)=O)C2)C1 N1(C(C(C(C)C)NC(C)=O)=O)CCC(C2(NC(=O)C#CC(C)(C)C)CC2)C1 C(=O)(C(CC(C)(C)C)N1CCC(CC2OCCO2)CC1)N(C1CC(SC)C1)C c1(C(=O)OCc2cc(C(=O)OC)cc(Br)c2)cc2cc(Cl)ccn2n1 C=CCC(CNC(c1cncn1C)=O)C(=O)NC1CC(C(C)O)C1 C1(NC(c2scc3c2OCCO3)=O)COC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 N1(C(=O)CC2CSCCO2)CCCC2C1CCCN2C(=O)CCc1nc(O)n[nH]1 c1(N2CC(COCCOC)OCC2)ccc(S(=O)(=O)NCC(CO)OC)c(Br)c1 Cc1cc(C(=O)NCCCCCCNC(c2cc(C)c(C)o2)=O)c(C)cc1Br N1(C(C(=O)NC(CC)(C)C)CC(C)C)C2CCC1c1ccccc12 C(C)(CNC(C1(N2CCCC2)CC1)=O)(CC(C)C)NC(Cc1c(C)n(C)cn1)=O C(CC(C(=O)N1CCC(C)(CC(=O)N(C)Cc2cscn2)C1)OC)OC N1(C(CC(C)OC2CC2)=O)CCC(OC(c2ccccc2)=O)CC1 CN1CCC(O)(C2(C(=O)NCC(C3CCC3)NC(C3(C4CC4)CC3)=O)CC2)CC1 C1(NC(CC=C=C)=O)CCCCC12CCN(C(C13CCC(CC1)C(C)(C)O3)=O)C2 c1(CC(=O)N(C)CCN(C(=O)CC2CC=CC2)C)ccc(Br)c(F)c1 c1(C(=O)NCC(C)CN(C)C(c2ccc(CO)c(F)c2)=O)n[nH]cc1[N+](=O)[O-] CC1CN2CCN1C(C(=O)NC(C)CNC(c1ccncc1)=O)C2 C12(C(=O)NCCCCNC(CCC(C)(C)C#N)=O)CC3CC(C1)CC(C)(C3)C2 c1(CC(=O)NCC2(C#N)CC2)n[nH]c2cc(C3=CCNCC3)ccc12 Cc1ccc(C(=O)NC2CN(C(=O)CCSC3CCCC3)CC2C)c2c1CCC2 c1(NC)c(C(=O)Nc2cccc(C3CC3)c2)cccc1F C1(C(=O)NC(C2CCOC2)CNC(CCOCC)=O)(OC)CCSC1 N1(C(CCC=CC)=O)CC(C)(C)CCC1CNC(C1CCN(C)C(=O)C1)=O C(C(=O)N1CCC(NC(C2(C)CCC(OC)CC2)=O)C(F)C1)(C(C)(C)C)OCC CC1CC(CNC(N2CCC(C(N3CCCC3)=O)C2)=O)=NO1 c1(C(N2CC3C(CNC(C4CC4F)=O)C3C2)=O)nncc2ccccc12 C1(OCC=C)CCN(C(C2CCN(C(=O)CCn3ccc(C)n3)CC2)=O)CC1 N1(C(CN2CC(C)(C)C2)=O)CCCCC1CCCNC(C1CCCCCC1)=O N1(C(C(C(C)OC)NC(=O)C=CC(F)(F)F)=O)CCCC(CCO)CC1 C1(C(N2CC3C(CC)(C3)C2)=O)CN(C(C2CC3C=CC2C3)=O)CCC1(C)C c1(CC(=O)NCC2C(NC(c3c(C)cc(CO)o3)=O)CCC2)cc(F)ccc1O N1(C(CN(C)C(=O)C2CC2)=O)CC(NC(C2CCCC(=O)N2)=O)CC1(C)C C1(NC(c2c(C)nns2)=O)(CNC(=O)Cc2ccco2)CCOCC1 n1(CCCC(N2CC(CC)(NC(C3CCN3S(C)(=O)=O)=O)C2)=O)nc(C)cc1C c1(C(=O)NCC(CNC(=O)CCCCC2CC2)F)ccc(C(F)F)c(F)c1 N1(C(=O)C2=CC(O)CCC2)CCC2(C1)CN(C(C1(CC3CC3)CC1)=O)CCO2 c1(OC)cc(C(=O)NC(CNC(=O)C(O)C(C)(C)C)CO)c(F)cc1N N1(CC(=O)NC(C)CCN(C)C(C2CCC2C(F)(F)F)=O)CCOCC1 C12(C(=O)NC(CCCNC(c3ncc(OC)cn3)=O)C)CCCC1CCC2 C(C(C)(C(=O)NC1CC1NC(=O)Cc1nc(C)sc1C)OC)OC c1(CC)ccc(C(N2CC(CC(C)NC(=O)Cc3nocc3COC)C2)=O)cc1 C1(NC(CCSc2n(C)ccn2)=O)CCCN(C(c2ccncc2F)=O)C1 CCCCC(CC)CC(=O)NCCC(C)(C)C(=O)N(C1CC(OC)C1)C CC1CCOCCN1C(c1[nH]ccc1CNC(=O)CCCC1CC1)=O S(=O)(=O)(c1ccc(NCCCN2C(=O)CCC2=O)c(F)c1)NCC(CC(C)C)O c1(C(N2CC(C)(NC(c3cn(CCOC)nc3C)=O)C2)=O)ccc2[nH]ccc2n1 C1(CNC(Cn2c(C)c(Cl)cn2)=O)CC2(CO1)CN(C(C1(CCF)CC1)=O)C2 C(=O)(C1c2c[nH]nc2CCC1C)OC(C(C)C)C(=O)NCC1CCCC1 C1(C(=O)NC(C)CN(C)C)CN(Cc2ccc(C(=O)O)o2)CC(F)(F)C1 C1(CCOC)CN(C(C2(C(N)=O)CCC2)=O)CCN1C(=O)C(O)CN(C)C C(CCCCC(=O)NC1CN(C(c2cc(C(C)C)on2)=O)CC12CC2)OC C1(CCN(C(C=C(C)Cl)=O)C)CCN(C(=O)C(c2ccc(F)cc2)C)CC1 C1(C)(C(=O)NCC2CC3(CC(NC(C=C(CCC)C)=O)C3)C2)CC2(C1)CC2(F)F C1(NC(N(CCCOCC)CC)=O)CCCN(c2ccc(C#N)cc2)C1=O C=CC1(C(=O)NCCc2n[nH]c(C)n2)CCN(C(=O)CC2CCSC2)CC1 c1(C(=O)OC)cc(Br)cc(Br)c1NC(C1CC2CC2N1C(C1CC=CCC1)=O)=O C1(NC(CC(C=C)C)=O)CCN(C(=O)Cc2c(N)nc(C)nc2O)CC(C)(C)C1 C1(O)(CNC(C2CC2C(F)F)=O)CCCN(C(c2cccc(F)c2Cl)=O)C1 C1(O)(CN(C(C(C)=C2CC2)=O)C)CCCN(C(=O)Cc2cn(C)nn2)C1 S(=O)(=O)(c1ccc(NCC2COCCN2C)c2cnccc12)NC(CCOC)C N1(C(c2ncc(Cl)s2)C(=O)NCCSC)CCCOC(C)C1 Cc1cc(NC(=O)C#CCNC(=O)C(C2CCOCC2)O)cs1 c1(C(N2C(CNC(C3C4COCC34)=O)CC2)=O)cccc2sncc12 N1(C(C(C)Oc2ccccc2)=O)CCOc2ccc(-c3cscc3C#N)cc21 N1(C(C2CC2NC(C(C)SCC)=O)=O)CCC2(CC1)CNC(=O)N2 c1(CC)cc(F)ccc1C(=O)NC1CN(C(=O)Cc2cc(Cl)cnc2C)C1 CC(CC(C)NC(=O)Cn1nccn1)NC(C1CCC2CC12)=O C1(C(N2C(C)CCC(NC(=O)Cc3cnn(C)n3)C2)=O)Cc2ccncc2C1 c1(C(=O)NCC(N)=O)ccc(NC(=O)Nc2ccccc2)cc1 C(=O)(CC(O)CC(C)(C)C)NCC(C)(Cn1cccn1)NC(C(COC)C)=O N#CC1(C(=O)NC2CCC(CNC(C3(C4CCC4)CC3)=O)CC2)CCOCC1 n1(CC)c(C(c2nnnn2CC2CC2)NCC2CCCO2)nc2ccccc12 c1(C(=O)NCC(C)CN(C(=O)C(CO)N(C)C)C)coc(C(F)F)c1 CC#CCC(C(=O)NCc1nc(C)ns1)NC(C1CN(C(N)=O)C1)=O C(=O)(CCCCC(F)(F)F)NC1(C2CCN(C(CNS(N(C)C)(=O)=O)=O)C2)CC1 N1(C(C(C(C)OC)N(C)C)=O)CCN(C)CC1C(=O)NCC(O)C(F)F C1(C(=O)NC(C)(CNC(c2cc3sccc3[nH]2)=O)CO)CCCC12CCOCC2 c1(CC)cnc(C(C)NC(=O)NC2(n3ccnn3)CC2)s1 N1(C(CC(CC)C)=O)CC2CCN(Cc3cccc(Cl)c3OC(F)(F)F)C2C1 c1(C(=O)NC(CC(C)NC(C2CCC(C(=O)OC)C2)=O)C)nccnc1OC C1(CN(C(=O)C2=CCCS2)C)CCN(C(=O)CCC2CCCN2C)CC1 c1(C(=O)NCC2CCN(C(c3c(OC)ccs3)=O)CC2O)cccc2c1COC2 CCCCCCCCCC(=O)NCC(C)(C(C)C)NC(=O)CCC(C)(C)[N+](=O)[O-] C1(C(=O)NC(CCC(C)(C)c2nn[nH]n2)=O)Cc2cccnc2C1 c1(N(C2CCN(C(C)=O)C2)C)cc(C(=O)NCC(CSC)O)ccc1O Cc1cc(C(=O)NCCCN(C)C(C2CCCCC2O)=O)c(O)nc1C N1(C(C(C)OCC2CC2)=O)CCCC(C(C)(C)C(=O)Nc2cccc(CO)c2)C1 C1(C(N(CC)Cc2ncc[nH]2)=O)CN(C(=O)Cn2c(O)nnc2O)CC1F c1(NCC(C)OCC=C)cc(Br)ccc1S(=O)(=O)NCc1cc(Br)cs1 C1(NC(CC2(C)CCCC2)=O)CN(c2nnc(C(F)F)o2)C2CCCCC12 C(C)(CCC(=O)N(C)Cc1ccon1)NC(C1N(CC)CCC1)=O C1(NC(C(CC=C)NC(C)=O)=O)CN(C(=O)Cn2ccnc2C)C(CC)(CC)C1 c1(N(C)C)cc(F)c(Br)cc1-n1nc(C2CCC(F)(F)CC2)nc1-c1cnsc1 C(C(CC(C)C)NC(C(CC)F)=O)NC(c1ncc[nH]1)=O CC(C)(CCC(=O)O)NC(=O)C(C1CCOCC1)c1cn(-c2ccccc2)nn1 c1(C(=O)NCC2(C)CCN(C(C(COC)(C)O)=O)C2)cc2c(cc1Cl)OCCO2 C(CO)(CCCCNC(C1CC2(C1)CC21CC1)=O)NC(c1cc(CC)nn1C)=O C1(C(N2CCC(NC(CCCC)=O)CC2)=O)CN2CCN1CC2C N1(C(c2ccc(C)nc2)=O)CC(NC(=O)CCC2CCC(C)O2)C2(CCCC2)C1 C1(C(=O)NC(C=C)C2CC2)CN(C)CCN1C(=O)CC=CC(C)(C)C C1(NC(=O)NC)CC(C)CN(C(c2n[nH]c(C)c2Br)C(=O)NC2CCOC2)C1 N1(C(C2C(C)OCC2)=O)CCC2(CC1)CCN(C(c1ccnn1C1CC1)=O)CC2 N1(CCCCCNC(C2CC(C)OC2)=O)CCN(C(=O)C(CO)N(C)C)CC1 CC(C)(C)CC(O)CC(=O)NC1CCC(NC(c2csc(C(F)(F)F)c2)=O)CC1 c1(C(N(C(CNC(CC(CC)CN(C)C)=O)C2CC2)C)=O)cc(C)c(C)nc1C C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCCC1OCCN(C(C=CCOC)=O)C1 c1(CCC)sc(C(=O)NC2(C)CC(NC(c3cccc(N)c3)=O)C2)cc1CC CCC(C)CCC(=O)NC1(C2CN(C(c3sccc3SC(F)F)=O)C2)CC1 CC(F)(F)C(F)C(=O)NCCCC(O)C(=O)NC1CCCC1CF c1(Cn2cc(C(C)NC3CC3c3ccc(Br)s3)nn2)cccnc1OC(F)F C1(C(=O)NCC2CC2(F)F)C2CCC(C2)N1C(=O)CC1OCCCO1 c1(C(=O)NCCC2N(C(C3C(C)C3)=O)CCSC2)nn(C)c2ccc(Br)cc12 N1(C(c2[nH]nnc2-c2ccccc2)=O)CCCCC1C1CCCN1CC(Cl)=CCl Cc1cc(CN2C3CCC(C3)C2C(=O)NCC2CCCO2)c2ccccc2n1 C(CCCC(=O)N1CCCC(CNC(=O)CC(C)(O)c2ccccc2)C1)SC C1(C(=O)NCC2N(C(C(CC(C)C)O)=O)CCOC2)C2CCC1(C)C2(C)C C12(CNC(c3c(C)nc[nH]3)=O)CCCC1CN(C(C1CC13CCC3)=O)C2 CC1CC(C(=O)NCCCn2ccnc2)N(C(c2ccccc2O)=O)C1 C1(O)(C(C)NC(CS(CC)=O)=O)CCN(C(C2(n3ccnc3)CCCC2)=O)CC1 C1(C(=O)OC)CN(C(=O)C(=O)Nc2ccccc2Br)CC1(C)COCC(C)C C1(C(=O)NCC(c2cccc(O)n2)O)CC2CC2N1C(C1CC2CCC1O2)=O c1(C(=O)NCC(C(C)C)(C)NC(C2COCCOC2)=O)cccc2sncc12 N1(C(c2cn(CCCC)nc2C)=O)CCN(C(c2cocc2C)=O)C(C)C1C C1(C#N)(C(=O)NCC(C)NC(c2c(C)ccc(C(F)(F)F)c2)=O)CC12CCCC2 c1(C(=O)NC2C=CCN(C(c3nc(COC)[nH]n3)=O)C2)c(C)oc(C)c1C CC1CC(NC(=O)CCc2cncn2C)CN(C(=O)CC2(C#N)CCC2)C1 N1(C(C2N(C)CC(C)(C)C2)=O)CC2CCC(C1)N2C(=O)C1=CSCCO1 CCC(CC(=O)N1CCCC1(CNC(c1conc1C(C)C)=O)COC)SC C1(NC(CN(C2CCC2)C)=O)CCCN(C(=O)CSc2n[nH]c(=N)s2)CC1 c1(C(=O)NC2CCN(C(=O)Cn3ncnn3)C2)ncc2[nH]ncc2n1 Cc1cccc(Cl)c1CC(N1CC(O)(C2CCCN2C(=O)C2=CSCS2)C1)=O N1(C(C=C(C)C(F)F)=O)CCS(=O)(=O)C(CCNC(c2cc(C)c[nH]2)=O)C1 C(c1ccc(=N)[nH]c1)=CC(N1CC(C(C)NC(=O)CC2CC(=O)NC2=O)C1)=O N1(C(c2cccc(C)c2C)=O)CC2(CCN(C(C3(C)CC4CC4C3)=O)C2)C1 Cc1ccccc1C(N1CC(F)CC1CNC(c1ccc(Cl)cn1)=O)=O C1(C(=O)NC(c2ccc(F)cc2)C)CN(C(c2ccc(Br)s2)=O)CCS1 C1(CNC(N(C2CCc3ccccc32)CC)=O)CCc2[nH]c3ccccc3c2C1 CC(C)C(CCC(=O)N1CCN2CCCC2C1)NC(C1COC(=O)N1C)=O N1(C(Cc2n(C)cnc2)=O)CCC(c2ccccc2)(CNC(=O)C2=CCC2)CC1 c1(NC(=O)C(F)CC2CCCCC2)cccc(F)c1F.C12CCN(C1)C(=O)N2C c1(CC)cnc2ccccc2c1C(N1CC(NC(=O)C2=COCC2)CC1C)=O CC(C(=O)NC1C(C(F)(F)F)C1C(F)(F)F)C(C)(C)c1ccccc1 C1(NC(c2ccc(C(N)=O)o2)=O)CCSC12CN(C(c1c(F)cccc1Cl)=O)C2 N1(C(N=NN(C)C)=O)CCC(NC(=O)Cc2ccccc2O)C(CO)C1 C1(N=[N+]=[N-])(C(=O)NC2C(OC)C(O)C2)CCN(C(c2nc(Cl)oc2C)=O)C1 CCCCC(F)C(=O)N1CC(C2CN(C(=O)C(O)C3CC3)CCO2)C1 C(C(C)(C)C(=O)N1CCCC(CCC(=O)NC(c2ccoc2)(C)C)C1)N(C)C CCCCC(CC(=O)NCc1[nH]c(C)nc1C)NC(=O)C(C)(C)Cl C1(CNC(C(c2ccncc2)C)=O)CN(C(C2CCCCC2)=O)CC(C)(C)O1 C1(CNC(c2c(C)occ2)=O)CCC(N(C)C(C2CC2OC(C)(C)C)=O)CC1 C12(CCC(C)(C)C1)CN2.C1(=O)CC(=O)O1.C(C)(C)(C)CCSC(C)C C1(CNC(c2ccc(OC(F)F)nc2)=O)CN(C(c2n[nH]cc2I)=O)CCO1 CC(O)C(C(=O)NCC1C2CN(C(C3(N(C)C)CCOCC3)=O)CC12)N(C)C C=C1CC2(C1)CC(C(=O)NC(C1CCN(C(C34CC(CO3)C4)=O)C1)C)C2 Cc1[nH]cc(C(N2CCC3(CC3NC(C3CCN(C)C3)=O)C2)=O)c(=O)c1Cl N1(C(C(CC(C)C)C)=O)CCC2C(CCCN2C(c2cc(C#N)c[nH]2)=O)C1 C(C(CO)(CO)NC(c1cncc(C)n1)=O)N(C(C(C)(C)OCC)=O)C N1(C(CCn2ncc(C)c2)=O)CCC(NC(C2(F)CCCC2)=O)C(C(N)=O)C1 C1(C)(CC)CCC(C(=O)NC2CC(CNC(=O)C=C(C)c3ccco3)C2)O1 c1(C(=O)OC)c(F)cc(NCc2cc(Br)c(O)nc2C)cc1Br n1(CCCOC)nnnc1C(c1cc(C(F)F)cs1)NCC1CCC1(F)F c1(C(=O)NCC(CNC(CCN(C)CC)=O)O)ccc(F)c(S(N)(=O)=O)c1 C(CNC(=O)C(C)(C)c1cccnc1)(C(C)(C)C)NC(C(c1ccc(C)o1)C)=O c1(NC(N2CCC(CC3CCCO3)C2)=O)csc(Cc2nn[nH]n2)n1 CC1C(NC(=O)C=Cc2cscn2)CC2CCC1N2C(c1ccc(N)cc1)=O N1(C(C2C=CC(NC(Cc3c(C)nn(C)c3)=O)C2)=O)CCN(C)CC1C1CC1 CC1(CNC(C2CC3(CC3)CO2)=O)CCCN1C(C1CC12CC2)=O N1(C(c2n(CC)ncc2)=O)CCC=CC1C(=O)NCc1ncco1 c1(OC)cc(CNC(=O)COCc2cn(C3CC4CCC3CC4)nn2)cc(Cl)c1 c1(CC(C(=O)OC)NCc2cccc(Cl)c2OC)c[nH]c2ncccc12 CC(C)(CC(F)F)C(=O)NCC(CC1CCCC1)C(=O)NCCC1CC(C)(C)C1 c1(N(C(c2cn(C)cn2)C(=O)NCCCF)C)ccc(C#N)cc1F c1(C(=O)NC(CN(C(=O)Cn2cc(Br)c(C)n2)CC)C)cncc(C)c1C CCCC(C)CCCOC(c1ccc(-n2cc(Br)cn2)nn1)=O c1(CCCOCC)nc(-c2cccc(N)n2)nn1-c1cccc(C)n1 CCCCC(F)(F)C(=O)NCC1(O)CC(C(=O)N=c2ccn(C(C)CC)[nH]2)C1 Cc1cc(C(N2CCCC2CCNC(=O)CN2CC(C)(C)C2)=O)cn(C)c1=O C1(NC(c2cn(C)nn2)=O)CCC(CNC(=O)CCn2cccnc2=O)CC1 C1(C(N2CCC2CNC(=O)C(C(C)C)NS(C)(=O)=O)=O)(OC)CCCCC1 CC(C)CC(O)C(=O)NCC(C)(C)CNC(=O)C=C1CCC(C)C1 C1(C(=O)NCC2(COC)CCC2)CCCN(C(=O)C(F)CC2CCC2)C1 c1(C(N2CCC(F)(CNC(C3C(CC)CCO3)=O)C2)=O)c(OC)ncnc1OC c1(C(=O)NC(CCNC(C(CC)(CC)OC)=O)(C)C)csc2ncnc(O)c12 C(=O)(C1=C(C)OCCC1)NC(CC=CC)C(=O)Nc1cn(CC)nc1C c1(C(=O)NCC2C(NC(c3c(C(N)=O)nccn3)=O)CCC2)n[nH]c2c1CCC2 C(C(C)C(C)C(=O)NC(C)(C)CNC(c1ccc(CN(C)C)[nH]1)=O)OC Cc1nc(C(=O)NCC2CN(C(=O)C3=CCCOC3)C3CC23)ccc1C(F)(F)F Cc1cc(C(=O)Nc2cc(Cl)nnc2Cl)n2nc(C(F)(F)F)cc2n1 N1(C(CC(c2c(F)cccc2F)C)=O)CCC(C)C(NC(c2csnc2C)=O)C1 C1(O)(CC(=O)N(C2CC(C(=O)NC(C(C)C)C3CCC3)C2)C)CCCCC1 c1(C(N2CCCC(CC=C)(NC(C3COC(C)C3)=O)C2)=O)ccc(C)c(Cl)c1F N1(C(C2CCCCC2(F)F)=O)CCC2(CCN(C(C3CCCS3)=O)C2)C1 c1(NCC(C2CCN(C(C)=O)CC2)CO)ncnc2sc(C(F)(F)F)nc12 C1(C(=O)NCCSCCOC)(SC)CN(C(=O)CCCF)C1 C1(C(N2CCC(C(C(=O)NCCNC(=O)NC)(C)C)C2)=O)CCCC(=O)CC1 N1(C(CCOCCC)=O)CC2CCC(C(=O)NCC(=O)NOC)(C2)C1 N1(C(Cc2c(OC)c(Cl)ccc2)=O)CC(NC(C2CC2C)=O)CC(C)(C)C1 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)C(CCOC)OC)CC(C)C1 c1(C(=O)NC2CC(CNC(C(CC=C)C)=O)C2)cc(C)c(F)cc1Cl Cc1cc(NC(C2CC2NC(c2cc(Br)cnc2O)=O)=O)c(Br)cc1F c1(CC)nc2c(C(=O)NC(CO)C(C)NC(=O)CCn3cncn3)ccnc2[nH]1 N1(C(c2c(OC)nn(C)c2)=O)CCCC(C)(CNC(C2CCS(=O)(=O)N2C)=O)C1 C1(NC(CCc2cnn(C)n2)=O)CCC2CCN(C(=O)CSc3ccccc3)C12 N1(C(c2cnn(C(C)C)n2)=O)CCCCC(CCC(=O)NCCC(C)(C)CO)C1 C=CCCCC(C(=O)N1CCC(OCC(C)C)C1)NC(c1cccnc1NC)=O N1(C(C(c2cn(C)nn2)NC(=O)C#CC(C)(C)C)=O)CCC2C(C1)C2(F)F CCC(C(=O)NCC(=O)N(C(COC(C)C)C(=O)NCc1ccco1)C)N(C)C N1(C(CC=CCC)=O)CC(OC)CC(C)C1.C12(CC=CCC1)C(=O)NC2 C1(N=[N+]=[N-])(C(N2CC(C)OCCC2)=O)CCN(C(=O)CN2C(=O)CNC2=O)C1 N1(C(COCCC=C)=O)C(CC(=O)NCC(F)Cl)C2CCCC12 C1(F)(C(N(C2CC(C(=O)OC)C2)C)=O)CN(C(c2ncn(C(C)C)n2)=O)C1 C1(NC(c2cc(CNC(C3C(C)CC3)=O)on2)=O)CC(O)C(F)C1 c1(CCC(=O)NC(C)CCNC(C2(F)CCC2)=O)csc2ccccc12 N1(C(c2snc(C)c2N)=O)CCC2CC1CN2C(C1CN(c2nncs2)C1)=O CCCCC(C(=O)NCCC(C)CCO)NC(c1nn(C)cc1C)=O C(CO)(C(C)NC(=O)CC1(O)CN(C(=O)CSc2nc[nH]n2)C1)SC c1(C(=O)NC(c2scc(C)n2)C(F)(F)F)ccc(CC(C)C)nc1 C(=O)(C(C(C)C)S(=O)(=O)C1CCCCC1)N(c1cnn(OC(C)=O)c1)CCC C1(C(=O)NC(C(C)C)CNC(=O)Cc2cnn(C(C)(C)C)c2)CC2CC(=O)C1C2 c1(C(=O)NC(CN(C(C2C(CCC)CCC2)=O)C)C)nc2ccccc2[nH]1 Cc1c(C(=O)NCC(C)(O)CNC(=O)COCCN(C)C)c[nH]c1C#N N1(C(Cc2c(C)scc2)=O)CCN(C)CC1C(=O)NCC(C)N(C)C C(C(CC(C)C)C(=O)N1CCC(OCC(=O)NC(C)(CO)CCF)C1)OC C1(C)(CC)CN(C(C2CCCN2C(c2cc(C#N)cn2C)=O)=O)CCO1 C1(C2(NC(C(c3cnn(C)c3)C)=O)CC2)CCCN1C(=O)C(F)=CC1CC1 C1(NC(CCSCCCC)=O)C(C)CN(C(c2nc(=N)cc[nH]2)=O)CC1C N1(C(C(C)SCCCC)=O)CCC(F)C(NC(c2nocc2C(C)(C)C)=O)C1 N1(CC2(C)ON=C(C)C2)CCCC(N(C)C(=O)OC(C)(C)C)CC1 C1(CC(=O)NCC2CC(CNC(C3(F)C(C)C3)=O)C2)CCCCN1C C12(NC(c3ccc(COC)[nH]3)=O)CCCC1N(c1nccnc1F)CC2 C(=O)(N=S1(=O)CCC2(CCN(C(=O)C3=CCC3)CC2)C1)c1ccc(OC)c(Cl)n1 N1(NC(C(CC#C)C2CC2CC(C)(C)C2CCCC2)=O)CC(S(N)(=O)=O)C1 N1(C(C2CC=C(C)CC2)=O)CCC2C1CCCN2C(c1ccc(Br)cn1)=O C1(C(=O)NCC(CNC(C(c2cccc(OC)c2)O)=O)C)CN2CCN1CC2C N1(C(CC2CCC(C#N)C2)=O)CCC2(C1)CN(C(=O)C=C(Cl)Cl)C2 CC(O)C(F)(F)C(=O)N1CCC(C(F)CNC(c2cnccn2)=O)CC1 CCC(C)(CC)C(=O)NC1CN(C(=O)C=CCOC(C)(C)C)CCC1C N1(C(N2CCS(=O)CC2)=O)CCCC2(CCCN2C(=O)C(C2CCOCC2)F)C1 c1(NC(CC)CCCO)nc(C)cc(=NC2CCn3ncnc3C2)[nH]1 Cc1nc(NC(C2(F)CN(C(C3CC4(CCC4)C3)=O)C2)=O)nc(Cl)c1Br C1(C(=O)OCC)(C(=O)NCC(C)C2CCC2)CC(C)=C(C)C1 C1(CNC(=O)C=C2CCOCC2)CN(C(C2(C(F)F)CC2)=O)CC12CCOCC2 c1(OC)cc(C(=O)N(CC(C)CNC(=O)C=C(C)C2CC2)C)ccc1C#N C1(NC(C(N(C(c2ccc(COC)o2)=O)C)C2CC2)=O)CC(O)CC(C)(C)C1 c1(C(N(C)CC2(NC(C(c3ccccc3)OC)=O)CC2)=O)cnc(O)c(F)c1 N1(C(C2(CC#C)CCC2)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)CC12CCC2 c1(-c2c(-c3n(CCC(C)C)ccn3)nn(C)c2)cc(O)c2cnn(C)c2c1 c1(C(=O)NCC(C)(CC(C)C)NC(C2C(C=C)C2)=O)cnn2c(C)cc(C)nc12 C1(NC(C2(OC)CCC2)=O)CC2CC1N(C(=O)CC(C)c1cccnc1)C2 CN1CC(C)(NC(=O)C(=O)NCC(c2ccccc2)N(C)C)CCC1=O c1(OC)c(C)cc(C(=O)N(CCCNC(=O)C(Cl)=CCl)CCO)cc1C c1(C(=O)NCC2(O)CN(C(=O)CCc3cnn[nH]3)C2)noc2c1CCCC2 C12(NC(C=CCNC(C(C)(O)C3CCC3)=O)=O)CCN(CC1)C2 CC(C)(C)CN=c1[nH]nc(S(=O)(=O)Cc2csc(Br)n2)s1 C(C)(CC(C)(C)O)NC(CC1N(C(CCOCCOC)=O)CCC1)=O C(=O)(C1=CC2(CCN(C(=O)Cc3ccnc(O)c3)C2)C1)NC1C(O)CCN(C)C1 c1(CNC(C2C(NC(c3[nH]c(=N)sc3)=O)CCO2)=O)cccnc1F N1(C(CCCCSC)=O)CCCC(NC(=O)Cc2sccc2C)CC1 CC1C(NC(=O)Cc2cnsc2)CCCN1C(c1cnc2n1CCC2)=O C1(NC(CNS(N)(=O)=O)=O)CN(C(c2cccc3scnc23)=O)C2(CCOC2)C1 C1(C(=O)NC2(C(C)=O)CC2)CC(NC(=O)C(c2cncnc2)C)C(O)C1 N1(C(C(CCC)N(C)C)=O)C2CCC1CC(CNC(C1(C)CCCC1C)=O)C2 Cc1scc(CNC(=O)C(C)CNC(=O)CC2CCC(=O)N2C)c1C C(=O)(CCCC(=O)NCC(CO)NC(=O)C(c1ccccc1F)O)OC(C)(C)C C12(NC(C(C)O)=O)CCCC1N(C(=O)C(C)S)CC2 c1(C(=O)NCCC(CNC(=O)C(C)S(N)(=O)=O)OC)cc(F)ccc1C(C)C CC1CCN(C(c2cnc[nH]2)=O)CC1NC(=O)Cn1ncn(C)c1=O N1(C(C2(C)CSC2)=O)CCC(NC(=O)COC2CCCOC2)C(F)C1 C1(C(=O)NC(C)CCCNC(c2ccc(Cl)c(N)c2)=O)CCc2nc[nH]c2C1 N1(C(C2(C=C)CCC2)=O)CC(NC(C2CCCN2C(=O)C2CC2)=O)C(COC)C1 CC1CC(n2nc(-c3cc(Cl)ccn3)nc2C2CC2)CCO1 c1(C(=O)OC)cccc2c(C(=O)NC3CCCCC3C(C)C)cccc12 CC1(C)CCCCC1NC(=O)NCc1nccn1-c1ccccc1 C1(C#N)(C(=O)NC(CCNC(C(c2c(C)nn(C)c2)C)=O)C)CCOCC1 CC(C)(C)CCCCNC(C1(NC(=O)CSc2nc[nH]n2)CC1)=O c1(CC(=O)NCCC2CN(C(C3CCS(=O)(=O)C3)=O)C2)ccc2ccoc2c1 c1(C(=O)NCC(COC)NC(C(CC)COC)=O)cccn2nccc12 N1(C(C(COC)O)=O)CCCN(C(=O)Cc2ccc(Br)c(F)c2)CC1C c1(NCC2(C)CCCN2C(c2cc(C)sc2)=O)nc2c(cc1C#N)CCOC2 O=C1CCC(CC(N2CCCCC2Cc2cn(Cc3ccccc3)nn2)=O)CN1 Cn1ncc(C(=O)NC2CCCC2CNC(=O)CC2CCC(=O)NC2)c1C1CC1 C(=O)(C(=O)C(C)(C)C)NC1(C(N2CCC(CC)C2)=O)CCCCC1 CC(C)CC(CCO)NC(C1CCN(C(c2ccoc2)=O)C1)=O C1(C(=O)OC)Cc2c[nH]nc2CN1C(=O)C(O)CC(F)(F)F C1(C(=O)NC2CC(C)(C(=O)NCC3(CO)CCCO3)C2)CC2(CCC2)CO1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC(CF)C2)=O)cc2ccsc2n1C N1(C(c2cc(CNC(C3C(C)CCC3)=O)on2)=O)CC(CO)C(O)C1 C1(C(=O)NC(CCCC)CNC(C2CCCC3CC23)=O)CCCCS1(=O)=O C1(NC(c2ccccc2C(F)F)=O)CN(C(=O)C(F)CC2CC2)CCC1O Cn1ccc(C(C)(C)C(=O)NCC2CC(NC(c3cc(CN(C)C)on3)=O)C2)n1 C(c1c(F)cccc1F)=CC(N1CC(C)(NC(C(C(CC)C)C)=O)C1)=O C1(C(N2CC(OC)CC(NC(C3CC(=C)C3)=O)C2)=O)COc2ccc(Cl)cc2C1 c1(C(=O)NCC(C)CNC(C2CC3(CC3)CO2)=O)ccc2c(c1)NC(=O)C2(C)C c1(OC)cc(C(=O)O)ccc1CN1CCOCC1CC(=O)NCCCCN(C)C c1(OC)ccccc1N(C)C(C1(O)CCN(C(=O)Cc2ccccc2)C1)=O c1(C(=O)NCC2N(c3nccc(C)n3)CCC2)c(Cl)ccc2c1OCO2 c1(C(=O)NC(C(C)C)CNC(=O)CC2CC2C(F)(F)F)cnn2c(=O)cc[nH]c12 Nc1cc(Cl)ncc1C(N1CC(CNC(=O)CCn2cc(Cl)cn2)C2(CC2)C1)=O C(CC(=O)NCc1cncc(C#N)c1)(C(F)F)NC(C1(C)N(C)CCC1)=O c1(CCC(N2C(C)CC(CNC(C=C(C)C)=O)C2)=O)ccc2ccn(C)c2c1 C(=O)(CC(C)(C)C(F)F)NCC1CN(C(C2(O)CCCNC2)=O)C1.CO C1(NC(C2CC(=C)C2)=O)CC2CN(C(C3CC(F)(F)CS3)=O)CCN2C1=O c1(-c2nc(-c3c(OC)nccc3)nn2C)cc2ccccc2s1 CS(=O)(=O)c1ccc(C(=O)NCC2CN(C(c3cnc[nH]3)=O)CCO2)cc1F Cc1ccn(C(C)C(N2CCC(CCNC(c3ccoc3C3CC3)=O)C2)=O)n1 Cc1cc(N2CCN(CCNC(=O)C(c3ccccc3)C)CC2)c(F)cc1[N+](=O)[O-] c1(C(N2CCC(N(CCC)C(C3CCC(O)C3)=O)C2)=O)nnn2c1CCCCC2 c1(C(N2CC(NC(C34CCCCN3CCC4)=O)C2)=O)cnc2ncc(Cl)cn12 C(=O)(CCS(C)(=O)=O)NCC(CO)NC(C1CCCN(C(C)C)C1)=O C1(NC(C2CCOCC2)=O)CCN(Cc2csc(Br)n2)C1 C1(C(N(CC(CC)(F)F)C)=O)CC2CN(C(=O)C(O)CCN(C)C)CC2C1 n1(CC)ccc(=NC(=O)C(CCSC)NC(C2CCOC2C(C)C)=O)[nH]1 c1(NCC)ncc(C(=O)NC2CC3(NC(=O)CC4CC4(C)C)COC2C3)cc1Cl c1(C(C)C(=O)N(C)CC2COCCN2C(=O)CO)ccc(Br)cc1F c1(C(=O)NC2CCC(Nc3ncc(OC(C)C)cn3)C2)c[nH]c2ccc(O)cc12 CC(O)CC(C)CN=c1[nH]c(=NCC2(C3(n4cc(Br)cn4)CC3)CC2)[nH]c2cc[nH]c12 N1(C(C(C)(F)F)=O)CCCCCC1C(N1CC2(CO)CC2(CO)C1)=O c1(NC(N2C(C)(c3ccccc3)CC2)=O)c(F)cc(Cl)cc1Cl C1(O)(Cc2cn(C(C)C(=O)N(N3CCCCS3(=O)=O)C)nn2)CCC(C)(C)CC1 C1(NC(C(C)SC)=O)C2CC(CN(C(=O)CCC3CCC3)C2)C1c1ccccc1 Cc1ccc(-n2cc(C(C)NC(c3cncc(F)c3Cl)=O)nn2)c(F)c1 c1(C(=O)NC2CC(NC(C3(C(C)(C)C)CCCC3)=O)C2)cnc(Cl)cc1N CC1(C)CC(C)(CNC(=O)Cc2csc(Cl)c2)CN1C(c1cccc(CO)c1)=O C1(C(N2CC(O)CC2c2ccccc2)=O)CC(c2ccccc2F)=NO1 N1(C(C(=O)NC(C(=O)OC)C)C(C)CC2CCOCC2)CCn2nc(C)cc2C1 c1(OC)cc(OC)c(C(=O)N(CC(C)O)CCNC(C2CC=CC2)=O)cc1Cl C1(CNC(C(CC=C)CC)=O)CC(O)C(O)CC1C(=O)N(CC(F)(F)COC)C C12(C(=O)NC(C(C)NC(c3cscc3Br)=O)C)CC3CC(CC(C3)C1)C2 C#CC1CN(C(=O)C(C)C(O)C(C)C)CCN1C(=O)CC1CCCN(C)C1 N1(C(C(CC)NC(C)=O)=O)CC2CC1CN(C(=O)CCNC(=O)CO)C2 N1(C(C2CC(OC)C2)=O)CCC2(CCC2)C(CNC(c2cccs2)=O)C1 CCC(CC(=O)NC1(C(N2CCC23CCOCC3)=O)CC1(C)C)C(C)C C1(C(N(C2CCN(C(=O)Cc3cc[nH]n3)CC2)CCOC)=O)CCS(=O)(=O)CC1 C(=O)(C1CCCn2ccnc21)N1CC(NC(c2nn(C)c(Cl)c2Cl)=O)C1 N1(C(CCSCCC)=O)CC(CNC(=O)CCC2(C#N)CCC2)CC1C C1(C(=O)NCC(CC)NC(c2nc[nH]c3nccc2-3)=O)CC2(COC(=O)N2)C1 O=[N+]([O-])c1cccc(Oc2ccc(-c3noc(Cc4ncccn4)n3)cc2)c1 C1(O)(C(=O)NC(C)CNC(C2CC2C2CCC2)=O)CCCC(C)(C)CC1 c1(C(=O)NC(C2CCN(C(=O)Cc3ccccn3)CC2)C)ccc(P(C)(C)=O)cc1 c1(NCC(CC(C)(C)C)OC)ccc(S(=O)(=O)NC2COCC2F)cc1C#N C(=O)(C(C)(C)CCC#N)NCC1CC(NC(c2c(C)nc(C3CCCO3)s2)=O)C1 C1(C)(C(=O)NC(COCC)C(=O)Nc2cccc(C)c2)CCNC1=O N1(C(N2CC3(CC(OC)C3)C2)=O)CCn2cccc2C1 C1(NC(c2cn(CC)nc2C)=O)CN(C(C2(CO)CCCO2)=O)CCC1(C)C N1(C(=O)COCC2CC2)CCN(C(=O)CCc2cscn2)C(CCO)C1 C1(C(N(C)CC2CCCN(C(c3cn(C)nc3Cl)=O)C2)=O)CCCS(=O)(=O)C1 CCCCCC(F)C(=O)NCCn1cnc(C(=O)NC2CCC(F)CC2)c1 N1(C(C)C(=O)NC(C2CCCN2C(c2ccsc2)=O)(C)C)CCC(O)CC1 n1(CCC(=O)NC(CN(CC)CC)C)cnc(C)cc1=O.C1(C=O)CCOCC1 N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCC1C(NC(c1c[nH]nc1C(F)F)=O)C2 c1(OC)ccc2c(c1)C(C)(C)N(c1cc(NCCN(C)C)nc(C(C)C)n1)CC2 N1(C(CC2(C(=O)OCC)CCCC2)=O)CCC2(CCN(C(c3cnns3)=O)C2)C1 C1(CN(C(=O)Cc2cccnc2)C)CC(F)CN1C(=O)C(F)CC1CCCCC1 N1(C(C2N(Cc3cccc(OC)n3)CC(F)(F)C2)=O)CCc2nc(Br)sc2C1 C(CCC(C)C)(C(=O)Nc1cnccc1CO)NC(C(CC#C)O)=O C1(C(=O)NCCN(OC)C)CCCN1NC(=O)C1COCC(C)O1 N1(C(CC(COC)C)=O)CCC(NC(c2cc(OC(C)C)ccc2N)=O)C(F)C1 CON1CCC(C(N2CCCCC2CC(N2CC(CC(F)F)C2)=O)=O)CC1 N1(C(c2cc(C)oc2C)=O)CC2(CO)CC1(C(N1CCCC(C)(F)C1)=O)C2 C12(C(N3CCCC(C(C)NC(c4nocc4Cl)=O)C3)=O)CCC(CC1)CC2 C1(CN(C(C(CSC)OC)=O)C)CCCN(C(c2cccc(C(=O)OC)n2)=O)C1 CC(C(=O)NC(Cc1cn(CC2(C(C)(F)F)CC2)nn1)CC(=O)O)C(C)(C)C c1(C(=O)NC2C(NC(C(N)=O)=O)CCOC2)ccc(Br)c(O)c1 c1(CNCC(=O)N(CC(C)N(C(C(C)=CC2CC2)=O)C)C)ccc(C#N)cc1 CC1CCN(C(C2CNC(=O)CC2(C)C)=O)C(C)C1NC(C1CN(C)CCO1)=O C1(CNC(C2ON=C(C)C2)=O)(NC(c2ccsc2Cl)=O)CCCCC1C c1(OCC)cccc(OC(C)C(=O)N(C)CC2CC2C)c1 N1(C(C2CN(CC)C(=O)N2)=O)CCC(O)C(NC(c2ncc(C)cc2C)=O)C1 c1(C(N2CCC(NC(C=C(C)C3CC3)=O)C(F)C2)=O)c(F)ccc(O)c1O n1(CCC)ccc(C(=O)NC(C)(C)CC=CC(=O)N(C)CC2COCCO2)n1 Cc1coc2c(C(=O)NCC3(O)CCCN(C(=O)CC4CC5CC5C4)C3)cccc12 C1(C)(NC(CC)(CCOC2(C)CS(=O)(=O)C2)c2nnnn2C)CCC(C)(C)CC1 C=CCC(CC=C)C(=O)N1CCC2C(NC(=O)COC(C)(C)C(F)(F)F)CC12 CC(C)CC(C)(CNC(=O)Cn1ncn(C)c1=O)NC(C1CC2CC1CC2O)=O c1(C(C2CCCC2)N)ccc(NC(=O)N(CCO)CC2CC(F)(F)C2)c(F)c1 N1(C(c2cc(CC)[nH]n2)=O)CC(C)(C)CC1CNC(=O)C(C)CSC(F)(F)F C(CCCCC(=O)NC1CCC(NC(c2cc(C3CC3)[nH]n2)=O)CC1)=CCCC C1(NC(CN(C(CC)CO)C)=O)CCC(C)(OC)C1 c1(OC)ccc(F)cc1C=CC(N1CC(CC(C)NC(=O)C(C(C)C)OC)C1)=O C=CCC(C(=O)NC(C1CN(C(=O)CNC(=O)NCC2CCCC2)C1)C)C(C)C C1(C(=O)N(C)CC2(O)CCN(C(c3c(C)nsc3C)=O)C2)(OC)CCCSC1 C1(C(N2CCC(N(C(=O)C=CC3CCOC3)C)CC2)=O)(CC)CCCCC1 N1(C(c2c(CC)noc2)=O)CC2CCCCC2(NC(=O)CC2CCC(=O)N2CC)C1 N1(C(CC(C)SC)=O)CC2N(C(c3nn4cccnc4c3Cl)=O)CCC2(C)C1 S(=O)(=O)(c1ccc(C#N)c(NCc2csc(=N)[nH]2)c1)NC(CC)COC CC(CC(=O)NC1CCN(C(=O)C(O)C(F)(F)F)C1C)C(F)(F)F S(=O)(=O)(c1cccc(NC(=O)CC2(n3cccn3)CC2)c1)Oc1cc(C)on1 c1(Cc2n(CC)c(NCP(C)(C)=O)nn2)cc(F)cnc1Br Cc1ccc(CC(N2CC(NC(c3c(C)coc3C)=O)C(O)C2)=O)cc1C c1(C(=O)NCC(C)N(C(CN(C(=O)OC)C)=O)C)csc(-c2cn[nH]c2)n1 c1(C(=O)NC2COCCN(C(c3ncc(Cl)cn3)=O)C2)ccc2[nH]nc(Br)c2c1 CCCC(CC)C(=O)N1CC(CC(=O)NCC2SCCS2)CC1(C)C CCCCC(O)CC(=O)NC1CC(CNC(C2CC2c2ccc(C)cc2)=O)C1 C1(CC)CCCC1(C)C(=O)NCC1CN(C(c2ccnn2CC(C)C)=O)CCO1 C=C(Cl)CCC(=O)N1CCCC1C(C)(C)NC(c1cc(C(F)(F)F)n(CC)n1)=O C(=O)(C1=C(F)CN(C(=O)CC2C=NN(C)C2=O)CC1)NC(CCC)(C)CC C(CCCCC(=O)NCCCCC(=O)N1CCC(c2ccco2)C1)SC N1(C(C(CC)SC)=O)CC2(CNC(c3cc(C(C)C)on3)=O)CC2(C(F)(F)F)C1 Cc1c(F)cc(NC(C2CCC2C(=O)Nc2nc(Br)cs2)=O)cc1Br C(CC(Cl)=CC(=O)N(CCCNC(c1cocn1)=O)CCO)N(C)C N1(C(CN(C(C)=O)C)=O)CCCC(C2CC2NC(c2scc3c2OCCO3)=O)C1 C1(C(N2CCC(CC)C2)=O)CCN(C(=O)Cc2ccoc2)C12CC2 c1(C(=O)NC2CC(C)NCC2)ccc(Cl)c(S(=O)(=O)NC2=NCCCC2)c1 c1(C(C(=O)NCC(CC)NC(=O)CNC=O)CC)ccc(OC)c(OC)c1.C(C#N)OC c1(C(N2C(COC)CC(F)C2)C(=O)NCCSC)sc2ccc(Cl)cc2c1C S(=O)(=O)(c1cccnc1N1CCCC(F)C1)NC1(c2scc(C)n2)CC1 C(=O)(CC(C=C)CCC)NC(C(=O)NCC(C#C)CC1CC1)Cn1cncn1 c1(-n2ccc(NC(c3nc(COC)oc3)=O)n2)ccc(O)cc1 CCCC(C)(CC)C(=O)NC1CCCN(C(c2noc3ncccc23)=O)CC1 N1(C(c2ccc(C)c(C(F)(F)F)c2)=O)CCCC12CCN(C(C1CC1CF)=O)C2 c1(C(=O)NCCOCCNC(C(C(CC)O)(F)F)=O)cn2cccc(Cl)c2n1 Cc1ncnc(C)c1C(=O)NCCCNC(c1cc(Cl)c(Cl)s1)=O CC1CN(C(c2ccc(F)c(F)c2)C)CCN1C(=O)CCCN1CCCCC1 C1(NC(C(C)NC(C)=O)=O)CCN(C(c2cnoc2C2CCC2)=O)CCC1CO n1(CC)cc(S(=O)(=O)N2CC(SC(C)C)C2)cn1.N12CCC(C)(C1)C2=O C1(NC(N2CC(n3ncc(C(=O)OCC)n3)C2)=O)CCC2(CCC2)OC1 CCCC(C)(CC)C(=O)NC1CCCCC1NC(=O)Cc1cc(C)cs1 N1(C(c2c(OC)n(C)nc2C)=O)CCCC2(CCN(C(=O)C(C)(O)C3CC3)C2)C1 c1(C(=O)OC)cc2c(cc1NC(C1CCN(CC(C)(C)O)CC1)C)OCO2 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CC(O)C1C2NC(C1OCCC1C)=O C1(NC(CC(=C=C)C)=O)CC2COCC(C1)N2C(=O)C(C)OC1CCOC1 c1(NCC2(CNC(c3ncc(C)nc3)=O)CCC2)ncc2c(n1)COC2 N1(C(C(CC)NC(c2ccn(CC)c2C)=O)=O)CCC2(CCC2)C(O)C1 N1(CC(N2CCC(C3CCCCO3)C2)=O)CCC(F)CC1 N1(C(c2ccc(CC)cc2N)=O)CCC2(CC1)CC2NC(=O)C(C)(C1CC1)OC C1(Cn2cc(CC(OCC)OC)nn2)CCC2(CCOCC2)O1 c1(CC)cc(C(=O)NC2CCN(C(C3C=CC=CC=C3)=O)C2CC)cc(F)c1 CC1(O)CCCN(C(C2CCC(CNC(c3cc(F)ncc3Br)=O)CC2)=O)C1 N1(C(c2ccc(OC)s2)=O)CCC(NC(=O)CCSc2ccccn2)C(C)C1 CC1CCN(C(C23CCC(CC2)C3)=O)CC1CC(=O)Nc1cn(C2CC2)cn1 C1(C(=O)NC(CCC)CO)CN(C(C2CN(C(C)=O)C2)=O)CC(C)(C)C1 c1(C(N2CCC(NC(CC(C)(C)O)=O)C23CCC3)=O)cc(F)c(C#N)c(F)c1 c1(C(N(C2CN(C(CC3C(C)CCO3)=O)C2)C)=O)cc2oc(Br)cc2s1 O=C1CC(C(=O)N2CCCCC(CNC(=O)C(C)(C)N3CCCCC3)C2)=NN1 c1(C(=O)Nc2ccc(-c3cccn(C)c3=O)s2)n[nH]c2c(F)cccc12 c1(NCC(=O)NCC(C)NC(=O)CCCc2cnccn2)ccc(C(N)=O)cn1 c1(CNC(NCC2CCCC(OC)C2)=NCCN2CCC2)n[nH]c2ccccc12 C(N=c1[nH]cnc(Cl)c1C(=O)OC)C1CCC(NC(c2nc(CC)sc2)=O)C1 c1(CC)cc(C(=O)NC(CNC(c2c(OC)cccc2Br)=O)CC)cc(O)n1 c1(C(C(=O)NCC=C)N(C2CCC(C)C2)C)ccc(C)c(I)c1 C(=O)(C1CCCn2cnnc21)NC1(CNC(C2(N=[N+]=[N-])CC2)=O)CCC1 CON1CCC(C(N2CC(C)(C)CC2C(=O)N(C2CCCC(C)C2)C)=O)CC1 C1(CNC(C(CC)(C)C)=O)(NC(=O)CCC(=O)c2cnn(C)c2)CC2CCC1C2 C(=O)(CCC(C)(C)C#N)N1C(CC)CN(C(c2cc(OC)ccc2O)=O)CC1 c1(CNC(c2n(CC=C)nnn2)c2cncn2C)ccc(-c2nnc(O)o2)cc1 c1(C(N(C(=O)C(N2CC(N)C(O)C2)c2ccccc2)C)C)ccc(F)cc1Cl c1(C(=O)NC(CN(C(=O)Cc2nonc2C)CC)C)cncc(NC(C)C)n1 C(CC1CC1)(CC(=O)NCc1cn(C2CC2)nn1)NC(c1c[nH]c(=N)o1)=O N1(C(CCCCOCC)=O)CCC2CN(C(=O)CN=S(C)(C)=O)CCC2C1 C#CCC(O)C(=O)C(CCNC)=O.c1(CC2CC2)cccnc1.C12(CCC1)C(=O)N2 c1(C(N2CC(NC(c3scc(OC)c3)=O)C(OC)C2)=O)ccc2c(c1)NCC2 Cc1cc(C(N2CCCN(C(c3ccoc3)=O)CC2C(C)C)=O)cc(C)c1F O=C(C1=CC(O)C(O)C(O)C1)Nc1ccc(N2CCC(=O)NC2=O)c(C(=O)O)c1 C1(CC(=O)NCc2ccc(C(=O)NC(CSC)(C)C)o2)CCC(C)CO1 C(C)(C)(CC(F)C(=O)N1CC(C)CC(O)C1)NC(C(CC=C)CC)=O N1(C(=O)OC(C)(C)C)CC2(CCC2)CC1CNC(C1CCC(N=[N+]=[N-])C1)=O c1(OC)cc(COC(=O)C(c2ccc(Br)cc2)OC)c2c(c1)CCC2 c1(CN(c2n(CCC=C)c(-c3cnn(C)c3)nn2)C)cc(F)cc(Br)c1 C[Si](C)(C)c1ccc(-c2cscc2C(=O)Nc2cnn(CCO)c2)cc1 C(=O)(C1=COCCO1)N(C1CCCCC1)CCNC(c1cc(C(C)C)n(C)n1)=O c1(NC(CSC)C)cc(C)c(S(=O)(=O)NCC2CCCC(F)(F)C2)cn1 C1(C(N2CC(OCCNC(=O)CCC3CCCCC3)C2)=O)CC2(C1)CC(F)C2 N1(C(=O)COCC2CC2)CCC2CN(Cc3ccccc3)CC12 CCCC(CCCNC(=O)CC1CCCC(C)(C)C1)NC(c1c[nH]nc1SC)=O Cc1ccc(C=CC(=O)N(C2CCC(NC(=O)Cc3ccoc3)C2)C)o1 Cn1cc2cc(C(=O)NC3CC(O)CN(C(=O)C4=NOCC4)C3)ccc2n1 C(c1cnc(O)nc1O)=CC(N1C(C)C(NC(c2nn[nH]c2Cl)=O)CC1)=O Cn1c(I)cc2c(N(C3CNCC3F)Cc3cncc(F)c3)ncnc12 CCCCC(=O)C(=O)NCC(O)C(=O)NC(C(C)C)C1CC1 Cc1cc(=O)n(C)nc1C(=O)NC(C1CCCC1)CNC(=O)C(CCO)N(C)C N1(C(C(C)NC(=O)CC(C)(C)C)=O)CCC2(C1)CN(C(=O)C(=O)NC(=O)C1CC1)C2 Cc1cc(=NCC2(N(C)C)CCC2)[nH]c(N2CC(OC(C)C)CC(F)C2)n1 C1(NC(COCCSC)=O)CC=CCC1C(=O)NCC1=CCCCC1 C(C(=O)NOC(C)C)(C1CCCC1)NC(c1cc(CC)no1)=O C1(CNC(C(=O)N(C2(C)CC(O)C2)C)=O)CCC(NC(=O)C2CC2)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(=O)NCC2CC2)ccc(F)c(F)c1 c1(CNC(C(CC#C)NC(=O)Cc2cnc(C)s2)=O)ccc(F)c(C)c1 CC1CCC2(CC1)CCN2C(=O)CC1CN(C(C2CC2C(C)C)=O)CCO1 C1(CNC(CNS(CC)(=O)=O)=O)CCC2(CCN(C(=O)C(C)C)CC2)O1 c1(OCC)cc(C(=O)N(CCN(C)C(c2ccnc(O)c2)=O)C(C)C)cc(F)c1 C1(CC(=O)NC2CC3(CC(C)(C)C3)C2)C(=O)Nc2ccccc2S1(=O)=O CC(C)CC(C)CC(=O)N1CCC1CNC(c1cc(=N)[nH]cc1Br)=O C1(NC(C(N2C(C)CCC2C)C)=O)CC2CCC(C1C)N2C(c1ccnn1C)=O N1(C(C2(CC=C)CN(C(C3CCCCN3C)=O)C2)=O)Cc2ccccc2C1 Cc1cccnc1C(=O)N(C1CC1)CC1CCCN1C(C1CC12CC2)=O C1(C(N(CC(CC)NC(=O)Cn2ncn(C)c2=O)C)=O)CCC(=O)N(CC)C1 N1(C(c2c(C)n[nH]c2)=O)CC(CNC(=O)C(F)OC(F)(F)F)CC1(C)C N1(C(c2cc(CC)on2)=O)CC2CCC1(CNC(C1CCCC(C)CC1)=O)CC2 C(=O)(C(CC(=O)OC)NC(C)=O)N1CC(CC=C)(NC(=O)CCCCF)C1 C1(NC(CC#N)=O)CC2(C1)CC(NC(C1(c3cncnc3)CCCC1)=O)C2 C(CN=c1[nH]nco1)C1N(C(C2C(C)OCC2)=O)CC(O)C1 N1(C(C2(CC=C)CC2)=O)CCCC(C2CN(C(=O)CC3=NNC(=O)C3)C2)C1 C(=O)(C(CC1CCOC1)NC(c1ccc(OCC2CC2)s1)=O)OCC C1(NC(=O)CC2CC(F)(F)C2)Cc2ccccc2C1NC(=O)Cc1cscn1 N1(C(C(C2CCC2)OC)=O)CC(CO)(NC(c2cc(C(F)(F)F)cs2)=O)C1 N1(C(C(C(C)C)SC)=O)CCC2(CCN(C(c3cc[n+]([O-])cc3)=O)C2)C1 CN1CC(C)(NC(C2(F)CCN(C(C3CCC(F)CC3)=O)CC2)=O)CCC1=O c1(CNC(C2(CCNC(C3C(CC)CCC3)=O)CCC2)=O)cc(C)c(C)o1 c1(OC)ncc(C(=O)Nc2sc(C)nc2C)cn1.c1(C2CC(=O)N2)ccc(F)cc1 c1(C(N(CC(C)N(C)C(c2cccc(-n3cccc3)n2)=O)C)=O)cncc(O)c1 c1(C(N2CCCC(CCNC(C(C)n3ccnn3)=O)C2)=O)ccc(F)cc1F c1(C(N(CCCNC(C(CC)C(C)C)=O)C2CC2)=O)cc(F)c(OC)c(Cl)c1 C1(C(=O)NC2(C)CCN(C(c3n(CC)nnc3)=O)C2)Cc2nccnc2C1 N1(CCC(=O)NC2CC(C)(NC(C3C(C)C3C)=O)C2)C(=O)C2CCCCC2C1=O C=Cn1nncc1C(=O)NC1CC(CNC(c2cnc(O)o2)=O)C1(C)C N#CC1(C(=O)NC2CC(F)CN(C(=O)COCc3ccncc3)C2)CCCCC1 C(=O)(C1=CCC(C)(C)CC1)NC(C)C(CO)NC(=O)Cc1csc(Cl)c1 CC1CN(c2ccc(NC(N3CCC(C)(CO)C3)=O)cn2)CCN1 N1(C(c2c(C)nc(O)s2)=O)CCC2(CC1)CC2C(N1CCC1c1nncn1C)=O c1(CN2CCN(C(c3n(C)cc(Br)n3)=O)C3C2C3)ccc(C#N)c(F)c1 N1(C(CN(CCOC)C)=O)CCCCC1CCC(=O)Nc1ccnn1CC(C)C C#CCCCC(=O)NCC(c1ccccc1)CNC(c1ccc(OC)cc1)=O C12(CNC(C)Cc3ncn(C)n3)CNCC(=O)N1CCOC2 c1(NCC2(O)CCN(C(CCn3ncc(C)c3)=O)CC2)ncnc2scc(C)c12 C(=O)(CCC(C)(C)NC(C1CCN(C)C1)=O)NC(CC)CO C1(O)CCCC1OC.c1(C(CNCCC)=O)ccccc1 C1(NC(C(=O)NCCOc2cc(F)cc(F)c2)=O)CCC2(CC1)NC(=O)NC2=O N1(C(CCCC2C(C)C2)=O)CCC(CC(=O)NC(C)CC(=O)N(C)C)C1(C)C C(=O)(C1=NOC2COCC12)NC1CC2CC(NC(C3C(CC)C3)=O)CC21 c1(CC(C(=C)C)OC(=O)CC2CCCCC2C)cccc(OC)c1 c1(C(C(=O)N(CC(C)C(=O)O)C)N(CCOCC)C)cc(C)ccc1C Cc1noc2ncc(C(=O)NC(C)CNC(C3(F)CCOC3)=O)cc12 C(=O)(C(CC(N)=O)NC(=O)C(C)C1CCOC1)Nc1cnc(C(C)C)nc1 C12(C(=O)NC(CN(C(=O)Cc3c(C)n[nH]c3C)CC)C)CCCC1(C(N)=O)C2 c1(C(c2n(CCC)nnn2)NCc2c(C)nn(C)c2Cl)cc(C)ccc1C(F)F C1(CC(=O)NCC2C(NC(C3CC(=O)C3)=O)CC2)CC2C=CC1C2 Cc1cnc(F)cc1C(=O)NC1CCN(CCNC(C2CC2C)=O)CC1 C(=O)(C(F)C(=O)NCC1(C(=O)NC2(C)CC(O)C2)CC(C)(C)C1)OCC c1(C(=O)NC2C(C)CN(C(c3cc[nH]c3)=O)C2)c(F)c(F)c(Br)c(F)c1F C1(NC(C2CC(CNC(Cc3cn(CC)nc3)=O)OC2)=O)CCCCCCC1 c1(-c2cc(C(=O)NC3C(NC(c4cc(C)sc4)=O)CC3)n[nH]2)ccc(C)c(C)c1 N12CCC(CC13CC3)C2.c1(OC)ccc(-n2cc(CCC(C)(C)CO)nn2)cc1C N1(C(C2N(CC)CCOC2)=O)CCC(F)(CNC(c2cn(C)cn2)=O)CC1 C1(C(N(CC(=O)NC2CC3CCC2O3)C2CCC2)=O)CN2CCN1CC2 CC1(CC(=O)NCC2CC(CO)CO2)CCCNC1 c1(-c2nc(C(CCC)C)nn2C(C)COC)ccc(C)c(C(F)(F)F)c1 C(=O)(CCC(C)OC)N(CC(C(N1CC(C)(CC=C)C1)=O)C)C C=C(C)CN=C(NCCN1CCC(C)(C)C1)NC1CCC(c2ccc(Br)cc2)C1 N1(CC)CC(C(=O)NCC#CCNC(=O)CN(c2cnccn2)C)NC1=O N1(CC(=O)NC2C(CNC(=O)CCCc3cc(Br)cs3)C2)C(=O)CCC1=O C1(C#N)(C(N2CCC(N(C(=O)CC3CCCCO3)C)C2)=O)CC12CCOCC2 C1(C(=O)NC2CCC(OC)C2)CCCN(C(C2(CC3CC3)CC2)=O)CC1 C(N=c1cc(NCCc2ocnc2C)nc[nH]1)C1(CC)CCC1 C1(N(c2cncc(C)c2)c2cc(C)ncn2)CCNCCC1C N1(C(N2CCC(C(=O)NC3CCCC(c4ccccc4)C3)C2)=O)CCCC12CC2 C(CCCN=c1[nH]c(=NCCC(C)SC)c2sccc2[nH]1)c1ccc(OC)cc1 c1(C(CNC(=O)C=CCO)NC(C(CN(C)C)(C)C)=O)ccc(F)cc1F c1(NCCN2CCCC(C(C)NC(=O)CCc3cncs3)C2)cc2c(s1)CCC2 c1(N(C)C(C2(CN)CC2)=O)c(F)cc(Cl)cc1Br S(=O)(=O)(c1ccc(C)c(Cl)c1)N1CC2CCN(Cc3cccc(OC)c3)C2CC1 C(=O)(CC(C(F)F)NC(C1C(C)C1C)=O)NCC(C(=O)NC)(C)C N1(C(C(C2CCCOC2)OC)=O)CC(C)(C)CC1CNC(C1(O)CCCCC1)=O N1(C(C(C)=CCC)=O)CCOC(C(=O)NCCn2ccnc2C)CC1 CC1CC2CCC(C(N3CCN(C(=O)C=Cc4cccnc4)CC3)=O)CN2C1 CCC(C#N)C(=O)N1CCC(CC)C1C(=O)NOCCC(C)C Cc1c(C(=O)NCC2COCCN2C(C2CCNC(=O)C2)=O)cccc1Br N1(C(CC2C(C)CCO2)=O)CC2N(C(c3ccn4ccnc4n3)=O)CCC2(C)C1 CC(CC#N)C(=O)NCCNC(=O)CCn1cncn1 c1(C(N(CCCOCCN(C(=O)CCCSC(C)(C)C)C)C)=O)ccc(Cl)cc1 c1(OC)cc(OC)cc(C(=O)Nc2ccc(CC3CCCO3)c(C)c2)c1 C1(CNC(CCC)=O)CN(C)CCN1C(=O)C(c1ccc(OC)cc1)O C1(NC(c2c(CC)n(CC)nc2)=O)CCCN(C(=O)CC(=O)OC(C)(C)C)C1C C12(CC(=O)NCC(COC)(C)C)CCC1CN(C(=O)CCCC1CCCC1)C2 Cc1nc(C(C)(F)F)ccc1C(=O)NC1C2CC1N(C(c1c[nH]nc1F)=O)C2 CC1(C)CC(CC(=O)NCC2CC(O)C23CCC3)N(C(=O)CN2CC3CC3C2)C1 C1(CCNC)CC(F)(F)C12CCC2.C12CCCCN1C2(C)C c1(OCC)cc(C(=O)NCCC(O)CNC(=O)C(C)COC)ccc1C C1(NC(Cn2c(C)ccn2)=O)CC2CCC(C1C)N2C(c1cnc(C2CC2)s1)=O N1(C(CCNC(=O)NC)=O)CCOCC1CCN(C)C(C1CN(S(C)(=O)=O)C1)=O CC(C(=O)N1CCOC(CNC(=O)CC=C(Cl)Cl)C1)S(C)(=O)=O CN1CCC(C)(C(=O)NC(CCF)C(=O)Nc2ccc(N(C)C)nc2)C1 Cn1cnnc1CC(=O)NCCc1ocnc1CNC(C1(C(N)=O)CC1)=O CC(C)C(CNC(=O)CCc1cnccn1)C(=O)NCCCN1CCC1 S(=O)(=O)(c1cccnc1NC1CCCC2(CC2)C1)NC1CCC2C(C)(C)C1C2 C12(C(=O)NC(C)C(C)NC(c3ccnnc3N(C)C)=O)CC(C1)C(C(F)(F)F)O2 C1(CC(=O)NCC2(CCNC(CCNC(N)=O)=O)CCC2)CNC(=O)O1 c1(CNC(C(C)OCC#C)=O)nc2c(s1)CN(C(c1[nH]cnc1C)=O)CC2 Cc1cc(NC(c2nnnn2CCCF)CCC2CCCC2)cc(Cl)c1 Cc1cc(Cl)c(C(N2CCN(C(C3CCCS3(=O)=O)=O)C(C3CC3)C2)=O)cc1N N(C(=NCC=Cc1ccc(F)cc1)NCC1CC1)C(C1CCC(F)CC1)C c1(C(N2C(C)CCC(NC(C(c3cccnc3)C)=O)C2)=O)n[nH]c2c1CCOC2 CC(CSC)CC(=O)N(CCNC(=O)C(C)NC(=O)C(C)(C)C)C1CC1.C(C)C N1(C(c2c(C)cco2)=O)CC2(C1)CN(C(C1CC1C1CC1C)=O)CCO2 c1(C(N2CCCN(C(C(COC)C)=O)CC2C)=O)cc2c(cc1Cl)NC(=O)CO2 Cc1ccc(Br)c(NC(=O)NCC2CC23CCOCC3)c1 c1(NC(C2C(C(=O)Nc3c(OC)ccc(Cl)c3)C2)=O)cc(Cl)c(Cl)cc1O N1(C(CC(C=C)C)=O)CC2CCC(C1CO)N2C(c1ccc(C)cc1C)=O C1(C(=O)NCC2(C(C)(C)O)CN(C(C3(F)CCCC3)=O)C2)CC12CCSCC2 C1(NC(C(c2ccccc2)OCC)=O)CCC2CN(C(=O)C(C)(C)C)CC12 C#CCC(CC#C)C(=O)NC(CN(C)C(c1cccc(OC)n1)=O)CC c1(C(=O)NC2CC2)ccc2oc3ccccc3c(=O)c2c1.O=C1CN1 C1(C(N2CC(CN(C)C(c3cnnc(O)c3)=O)C2)=O)(CC)CCCCC1 C1(NC(C2(COC)CCC(=O)N2)=O)CCCN(C(c2cccnc2OC)=O)CC1 C(=O)(C1=CCC(NC(=O)C(C)(C)N2CCCC2)C1)N(CCCC(=O)OC)C c1(C(N(CC(CC)NC(c2ccc[nH]2)=O)CC)=O)ccc(F)c(CC2CC2)c1 c1(OC)cncc(-c2csc(NC(=O)C(CCC3CCC3)OC)n2)n1 C(=O)(C1=CCCCC1P(C)(C)=O)NC(C1N(C(CCCNC(C)=O)=O)CCC1)C C1(NC(c2nn(CC)c(O)c2)=O)CN(C(=O)C=CCN2CCOCC2)CCC1C N1(C(CNC(CCC)=O)=O)CC(NC(=O)C(CO)c2ccccc2)CC(F)C1 C1(C)(NC(Cc2c(OC)cccc2)=O)CCCN(C(=O)Cc2ccsn2)C1 Cc1cc(Cl)c(Cl)cc1CN1CC2CC(C1)N2C(=O)C=Cc1ccc(Cl)cc1 c1(CC)ccc(OC(C2CCN(C(=O)CC3(CO)CC3)CC2O)=O)c(OC)c1 C1(C)(C(N2CC(C)C(NC(C3(C(F)(F)F)CCCC3)=O)C2)=O)CC2(CCC2)C1 C1(C(=O)NCC2(F)CN(C(c3c(CC)oc(C)c3)=O)C2)CCC2(CCC2)O1 CC(C)CCC(C(=O)N1CC(C)(O)C1)N1CCC1CNC(=O)OC(C)(C)C C1(NC(c2n(C)ncc2Cl)=O)CN(C(=O)Cc2ccn(C(F)F)n2)C2(CCC2)C1 C1(OC)CC(C)N(C)CC1C.C=CC(CC)C(=O)N1CC=CC12C(=O)NC2 c1(CCC(=O)NC2(CNC(c3c(C(C)C)nco3)=O)CCC2)cccc(Cl)c1 C(=O)(CC1=CCCCC1)NC1C(NC(c2cccc(C(C)C)c2)=O)CCC1 N1(C(C(CC(=C)C)NC(c2cccc(F)c2O)=O)=O)CCn2ncnc2C1 CCC(CCC(=O)NCCC1CCCCO1)NC(=O)C1CC1 C(CC(=O)N(C1CC(C(N)=O)C1)C)N(C(c1cc[nH]c1)=O)CC C#CC1(C(N2CCC(CCN(C)C)C2)=O)CN(C(c2ccc(O)nn2)=O)C1 Cc1onc(Cl)c1C(N1CCOC(CCNC(=O)C(C)(C)C2CCOC2)C1)=O Brc1[nH]nc2ncc(-c3nc(CC4CC4)nn3C3CCOC3)cc12 N1(C(C(C(CC)CC)OC)=O)CCCC2(C1)CN(C(C1CCC3(CC3)C1)=O)C2 N1(C(C=C(CC)CC)=O)CC2(CCN2C(=O)COCP(C)(C)=O)C1 Cc1ccc2c(n1)OCCN(S(=O)(=O)Cc1cc(Cl)ccc1Cl)C2 CCC(C(=O)N1CCCC1C(C)NC(=O)C(n1nccc1C)C)n1nccc1C C1(CCC(N2CC(O)(CN(C(CCCOC)=O)C)C2)=O)C(=O)NN=C1C C1(CC)CN(C(c2cc(C)c[nH]2)=O)CCN1Cc1ccc(C)cc1 N1(C(C(C)CN2CCOCC2)=O)CCN(C(C2CCC(=O)NC2)=O)C(CCO)C1 N1(C(C2CC(C)(NC(C(C)N=[N+]=[N-])=O)C2)=O)CCC12CCCSC2 N1(C(c2ccc(C(C)=O)cc2)=O)CCCC(C)(C(=O)N(C)C)C1.C(C)(C(=O)OC)N N1(C(CC2(C)CC2)=O)CCCC1C(C)(C)CNC(C1(C(F)(F)F)CC(O)C1)=O c1(C(=O)NC(C(C(C)C)NC(CSCC=C)=O)C)ccc(Cl)c(Cl)c1C C(=O)(C(O)C(O)C(=O)OC(C)(C)C)OC.C123CC(CO1)N(C2)C(=O)N3 c1(C(C(=O)NC(C)C)N(C)Cc2scc(C)n2)ccc(CO)cc1 c1(CCCC=C)cn(C2CC3(C(=O)NCCSCC4CCCO4)CC23)nn1 N1(C(c2c(C)c[nH]n2)=O)CC2CC(NC(=O)CC3(N(C)C)CCC3)CC1C2 N1(C(C2CN(C(CC3CC(C)C3)=O)CC2F)=O)CC2COCC2(C)C1 c1(OC)cc(C(=O)NC2CCCC(CNC(=O)CCOC(C)=O)C2)cc(F)c1 Cc1cc2ccc(C(N3CC(C4CN(C(=O)CN(S(C)(=O)=O)C)C4)C3)=O)cn2c1 C1(C)(OC)CC2CN1C(=O)O2.c1(CC(=O)OCC2CCC2)ccnn1C C#CCCCCCC(=O)N(CCNC(c1cccc(Cl)c1C)=O)C1CC1 N1(C(CCC(C)OC)=O)CCCC(C2CCN(C(c3c(C)cnn3C)=O)CC2)C1 C#Cc1ccc(F)c(C(=O)NCCOC2CN(C(C3(C)CCCC3(F)F)=O)C2)c1 CC(C(=O)N(CCCCNC(=O)CN(C)C1CC1)C)C(C)(C)O C1(F)(C(=O)OC)CC2CC1(c1nc(-c3cc(C4CC4)nn3C)no1)C2 C#CC1(C(=O)NC2C3CN(C(C)=O)CC23)CN(C(C2C3CCC(=O)C23)=O)C1 CN1CCN(C(c2cnc(C(C)(C)CF)o2)=O)CC1CN(C(=O)C(F)(F)F)CCl C1(CNC(c2cc(C)sn2)=O)CN(C(=O)CC(C)(C)C2CC2)CC(C)(C)O1 C12CN(CCO1)C(=O)c1csc(c1)CNC(=O)C2.CCC(CC)n1ccnc1 Cn1ccc(CNC(=O)C(CC2CC2)NC(=O)CCc2ccn(C)n2)n1 c1(C(N2CC3N(C(COC)=O)C3C2)=O)cc2c(C)snc2s1 Cc1cc(C(=O)NCC(C2CC2)N(C(=O)Cc2cn(C)cn2)C)cnc1C C1(NC(C2(C(=O)OCC)CC2)=O)CN(C(c2ccc(C)nn2)=O)CC1C1CC1 C1(NC(C(C)N(CC)CC)=O)C2COCC1CC(NC(C1(SCC)CC1)=O)C2 C(=O)(C1CCCn2nccc21)NC1CCN(C(c2cc(CCO)on2)=O)C1 c1(C(N2CC(O)(CNC(CCCOC)=O)C2)=O)cc(N)cc(C)c1F Cn1ncc2ccc(C(=O)NCCCNC(c3ccoc3C(F)(F)F)=O)cc12 CCCCCCCCNC(=O)CC(CNC(C1CCC(C)(C)OC1)=O)C1CCC1 n1(CC(=O)N(C(C)CNC(C2CCN2C)=O)C)ccc(O)nc1=O c1(C(=O)NC(=O)CSCCc2ncc[nH]2)ccc(C=CC(=O)NCC2CC2)o1 c1(-c2cn(CC3N(C(CC)=O)CCC3)nn2)cccc(-c2nn[nH]n2)c1 c1(C(c2cn(CC(F)(F)F)nc2)N)c2c(nn1C(F)(F)F)CCC2.C1CC1 Cc1cccc(C)c1CC(N1CCC(CF)(NC(=O)C(F)=CCCF)C1)=O n1(CC(=O)NC(CC(C)NC(=O)CC(O)CN(C)C)C)ccccc1=O CCCC(CC)CCC(=O)NC1CC(CO)N(C(=O)C(C)OCC(C)C)C1 n1(CCN(C(=O)CCc2cn(C)nn2)CC)cc(CNc2csnc2C)nn1 C(CN=c1ccc(C(=O)NCC2CN(C(C3CCCC3OC)=O)C2)c[nH]1)OC C1(C(N2C(Cn3cc(C=CC)nn3)C=CC2)=O)CCC2(CCOCC2)O1 C(CC1CCC1)(C(=O)NC)OC.[nH]1cc(C2(C)CCCC2)nn1 C12(NC(c3ccnc(F)c3F)=O)CCCCCC1N(C(=O)Cn1ccnn1)CC2 C1(NC(C2CCC(=C)CC2)=O)CC2(C1)CC(NC(=O)Cn1cnnn1)C2 C(=O)(CCS(N)(=O)=O)N1C(CC)C(C(=O)NCC2CSCCO2)CC1 c1(C(N(CCCn2cc(CCCC(=O)OC)nn2)C)=O)sc2ccccc2c1C C1(NC(C2N(C(=O)C=Cc3ccncc3)CCN(C)C2)=O)CCn2nccc2C1 Cn1c(O)nc2ccc(C(=O)NC(CNC(C3CC34CC(O)C4)=O)CO)cc12 C1(NC(c2c(CCNC(Cn3c(C)cc(C)n3)=O)n[nH]c2)=O)CC(C)CC(C)C1 Cc1ccc(C(F)(F)F)cc1C(=O)NC1CCCC1(C)NC(=O)C(C)(C)C(C)O C1(C(N2CC(F)(CNC(c3ccc(F)c(F)c3)=O)C2)=O)C(F)(F)C12CCC2 C(=O)(C(F)(F)C(F)(F)F)N1CC(CN(C(=O)C=Cc2cc(F)cc(F)c2)C)C1 c1(C(N2C(CNC(C3(CCC)CCC3)=O)CCC2)=O)ccc(Cl)cc1O CN=c1[nH]cc(C(=O)NCCNC(=O)Cc2cccc(C(F)(F)F)c2)s1 CCCCC(O)C(=O)N(C1CCN(C(c2ccc(N)c(O)c2)=O)C1)CC c1(C(=O)NCC(C)N(C(C(C(C)C)c2ccc(F)cc2)=O)C)cccc(=O)n1O c1(C(=O)NCC2C(NC(CCc3ccc(C)s3)=O)C2)ccc2oc(C)nc2c1 c1(N(C)CCF)ccc(S(=O)(=O)NC2(C3CCCC3)CCC2)cn1 C1(C(=O)NC(C(C)(C)NC(CCn2c(C)csc2=O)=O)C)CN2CCN1C(C)C2 C1(C)(C(=O)NCCCN(C(=O)CC2CCC3CC23)CC)CCOCC1 C1(C)(NC(C)Cc2cccc(C(C)NC(=O)NC3CCC3)c2)NC(=O)NC1=O c1(C(=O)NC(C2CCCN2C(C2CNC(=O)N2)=O)C)coc(-c2ccccc2)n1 c1(C(=O)OC)cncn1CC(=O)N(C)CC1CCCN1C(=O)C(C)OC N1(C(Cc2cn(CC)nn2)=O)CC2(CC2)CC1CNC1(C(=O)NC)CC(O)C1 C(=O)(CS(=O)(=O)CCO)NCC1C2CN(C(c3ccn(C)c3)=O)CC21 CC(C(=O)NC(C1CCN(C(C2(C#N)CCCCC2)=O)CC1)(C)C)C1=CCCC1 C=CC1CC(NC(=O)CC2CCN(C(=O)C(C)C(C)C)CC2)CCO1 CCC(CC(F)F)C(=O)N(C1CCN(C(=O)CCSCC(N)=O)C1)C C1(=O)CCCCCN1C.C1(C(=O)NCCCNC(=O)NCCC)COCCO1 C1(CCNC(c2ccnc(CNC(C3CCC4(CC4)C3)=O)c2)=O)CCCC2CC12 c1(CC)ccc(C(=O)NC2(C(=O)NCCC(=O)NO)CC2(C)C)cn1 c1(OCC)ccc(CNC(C2CCS(=O)(=O)CC2)(C)C)c(F)c1F N1(C(CCNC(COC)=O)=O)CCCCC(N(C(=O)C(C)(C)CO)C)C1 C(=O)(C1CCOc2ccc(Br)cc21)NC1(CO)CN(C(CCC#C)=O)C1 Cc1cnc(C(=O)NCC2CCCC(NC(c3[nH]c(C)nc3C)=O)C2)cn1 c1(OC)ccc(CNC(C2CCC(Nc3cnc(Cl)c(Br)c3)CC2)=O)cc1OC N1(C(c2cc(CCCC)oc2C)=O)CCCC(C)C1Nc1ncncc1OC c1(N2CCCC(C(C)NC(c3ccc(C)nn3)=O)C2)cc2nnc(C)n2cn1 C(=O)(CC(C)CC(=O)NCC1(C)CCCN1C(C1CC2(CCCC2)CO1)=O)OC c1(CC)cc2cc(OC)c(OC)cc2nc1CNC(=O)C=CC(N)=O c1(C(=O)NC(C2CCN(C(=O)Cn3cccc3)CC2)C)c[nH]c2nccc-2c1 c1(C(N(C2CCCN(C(=O)CC(C)F)C2)CC)=O)n[nH]c2ccccc12 c1(-c2cn(CC(=O)NCCNC(C)=O)nc2)ccc(NC(=O)OC(C)C)c(N)n1 C1(C(N(C(C=C)C2CC2)C)=O)CC(O)(CNC(=O)CC2CCSC2)C1 C12(NC(CCc3ccc(C)o3)=O)CC1CN(C(=O)CC1CCOC1=O)C2 c1(CC(C(=O)NC(C)CNC(=O)CC2(O)CCC2)F)ccc([N+](=O)[O-])cc1 c1(NCC=C)cccnc1C(N1CCC(NC(=O)C(C(C)O)N(C)C)C1)=O C(CC(C)C)(C(=O)N1CC2CC1CN2C(c1csc(C(F)(F)F)n1)=O)NC(C)=O C1(CCNC(CCOC(C)=O)=O)CC(OC)CN1C(c1nccnc1C)=O C1(NC(c2c(C)nc(O)s2)=O)CS(=O)(=O)CC1CNC(C1CCN(C)C1)=O N1(C(C)=O)CCN(C(C2(NC(=O)C=CC(F)F)CCC2)=O)C(C)C1 C(=O)(C1=CC2(CCOCC2)C1)NC1C(CNC(c2cn(CC)nc2)=O)CCCC1 c1(C(N2CCCC(N(C(C3CCC3C(F)F)=O)CC)C2)=O)ccn(C)c(=O)c1 c1(C(=O)NC2C(CNC(C=CS(C)=O)=O)CC2)nnc2ccccc2n1 C1(NC(c2c(CNC(c3ccnc(CO)c3)=O)n[nH]c2)=O)CCC2CCCC1O2 C=CCC(C(=O)N(CC(=O)NOCCN(C)C)CC1CCCC1)OC Cc1ccc(C)c(C(=O)NCC2CC(NC(C3(C)CCCS3)=O)C2)c1N C(=O)(C(C)(C)C(C)NC(=O)CCC(=O)N(C)C)NC1CC(CC)(CC)C1 c1(C(=O)NC2C(NC(c3ncn(C(C)(C)C)c3)=O)CCC2)ccc(Cl)c(Cl)c1O Cc1sc2nc(CCNC(N3CCOC(C)(C4CC4)C3)=O)nc(O)c2c1C C(CC(C)(C)C)(C(=O)NCC1CN(C(=O)C(C2(O)CCCCC2)(F)F)C1)OC Cc1ccc(C(=O)NCCCN(C(=O)Cn2cc(C3CCOC3)cn2)C)s1 C1(OC)CC(C(=O)NCc2ccc(O)cc2)N(C(c2ccc(F)cc2)=O)C1 c1(C(=O)NCC(CNC(=O)CCc2cnc[nH]2)CO)cccc2c1NCCC2 c1(OCC(=O)NCC(C2CC2)NC(CC(C)(C)O)=O)cc(F)cc(F)c1 C(CCC(=O)NCC(C(C)C)NC(=O)CSc1ccccc1)=CC(C)C.C(CN)S c1(NC(C2(C)CCN(C(CCOCC)=O)C2)=O)cc(C)cnc1C CC(C)CCCC(=O)NCC1CC1NC(=O)C(CC(F)F)C1CCC1 c1(C(=O)OC)cnc(C(=O)N(CC(C)NC(=O)CC2CCC(C)C2)C)cn1 CON(CCC(=O)NC1CCN(C(C)(C)C)C1)C(=O)C1CCN(OC)CC1 N1(C(CC2C(C)CCCC2)=O)CCC2(NC(C3CCCC(=O)N3)=O)CCCC12 c1(C(N2C(CNC(Cc3nc(C(C)OC)sc3)=O)CC2)=O)ccc(C#N)s1 C1(NC(=O)CCC2CCOC2)Cc2ccccc2N(C(c2ccc(Cl)nc2)=O)C1 C(=O)(CCCC(=O)c1ccccc1N)N(C(C)=O)C(c1ccccn1)c1ccccc1 N1(C(C(c2ccc(C)o2)C)=O)CCN(C)CC1CNC(C1CCCCCC1)=O N1(C(C(COC)C(F)(F)F)=O)CCCC2CN(C(C3(n4ccnn4)CC3)=O)CC12 N1(C(CCSCCCC)=O)CCCN(C(=O)OC(C)(C)C)C(c2ccccc2)C1 N(C1CN(C(C2CCS2(=O)=O)=O)Cc2ccccc21)C(c1c(NC)nccc1)=O Cc1cc(N2CC(CCO)OC(C)(C)C2)nc(=NC(C)CC(C)(C)C)[nH]1 c1(C(=O)NCCC(C)NC(C(C)(C)OCC)=O)cc(N)c(C)c(N)c1 C1(NC(C(C=CC)O)=O)C=CCC(C(=O)NCC2(F)CCN(C)C2)C1 N1(C(c2c(C)nns2)=O)CCC(C)C(CC(=O)N(C2CC(O)C2)C)C1 N1(C(C(CC)C)=O)CCC(Oc2cc(C)cc(F)c2)CC1 C1(CNC(CC=C)=O)CN(C(=O)CCC(C)N(C)C)CC1(C)C c1(OC)cc(C(=O)NCCNC(=O)C#CC(C)(C)C(C)(C)C)c([N+](=O)[O-])cc1OC c1(C(=O)NC2CN(c3nccc(C(C)C)n3)CC2O)ccc([N+](=O)[O-])nc1 N1(C(C(c2cccnc2)C)=O)C2CCC1C(CNC(=O)CC1CC1)C2 C12(C(=O)NCC(CC)NC(c3csc(COC)n3)=O)CCC(CC1)CC2 CC1(CNCC(O)CNC(=O)CC=CCN)CCC1 c1(C(=O)NC2CCCCN2Cc2cnc[nH]2)ccc(F)c([N+](=O)[O-])c1 c1(C(N2CC(NC(=O)C#CC3(C)CC3)CC(OC)C2)=O)cc(N)c(F)cc1F C12(C(=O)NC3C4CN(C(C(C)OCCC=C)=O)C3C4)CCC(N(C)C)(CC1)CC2 CCC(C(=O)NCC(C1CCCC1)NC(C1(c2n[nH]c(C)n2)CC1)=O)NC(C)=O C#Cc1ccc(C#N)c(NC(=O)NC(c2cnnn2C)CC)c1 CN=c1nc(N2CCC(OCCC(C)C)CC2)[nH]c(=NC2CCCSCC2)[nH]1 C1(N(C(C2(CCCF)CC2)=O)C)CCCC1C#N.C1(C(=O)NCC)CC(CF)C1 c1(C(=O)NC2(C)CN(C(C3CCC(NC)C3)=O)C2)noc(C)c1C c1(OC)cnccc1C(=O)NCC(N1CCC(C2CCCCN2)C1)=O C=CCCCCCCC(=O)NCC(CC(=O)NC(C)CCOC)C1CCC1 C12CN(CC3(CCC3)C1)C(=O)N2.c1(CN)cc(=NCC2CC(=O)NC2=O)[nH]cn1 CC(CCNC(=O)CCNS(C)(=O)=O)N=c1[nH]c(C2CC2)nc(=N)[nH]1 Cc1ccc(C(N(C)S(=O)(=O)NCc2noc(C3CCCO3)n2)C)c(C)c1 CC(O)C(C)(C)C(=O)N1CC=CC(NC(=O)CCC2CCCCO2)C1 Cc1c(Cc2cn(C(C)C(N3CCCOCC3)=O)nn2)cnn1C(C)(C)C C1(CC(=O)NCc2ncn(CC)n2)CC(NC(=O)C(C)C)C1(C)C C#CC(C)(C)C(=O)NCC1CCCN1C(c1cnc(C(C)(C)C)[nH]1)=O C=C=CC(C)C(=O)NC1(C(=O)NCCC23CC(CO2)C3)CC1(C)C c1(C(=O)NC2CCN(C(Cc3ncc(CC)[nH]3)=O)C2)ccc(C(C)C)c(F)c1 c1(C(=O)OCC)cc(Br)cc2c1CCN2C(=O)OCC1CCC(C)CC1 c1(N(C)CC)nc(N2CCCC(CC3CCCO3)C2)c2c(n1)CCCCC2 C(N=c1[nH]cc(CCNC(c2cc(CO)on2)=O)s1)c1cccc(OCC=C)c1 N1(C(c2cc(C(N)=O)cc(C)c2)=O)CC2CCC(CNC(c3cccs3)=O)C2C1 N1(C(CNC(C(=O)OC)C)C(F)F)CCN(C(c2ccccc2)=O)CC1 C1(C(=O)NC2(CNC(C(c3ccc(C)s3)C)=O)CCC2)CC(C)(C)SC(C)(C)C1 C1(C(=O)NC2(C#C)CC2)CCCCC1(C)NC(=O)CC1CCN(C)CC1 c1(CC)ccc(CNc2cc(Nc3ccc(C4CC4)c(C)c3)ncn2)c(F)c1 Cc1coc(C2CC2)c1C(N1CC=CC(NC(=O)CCCN(C)C(C)C)C1)=O N1(C(c2ccc(CC)[nH]2)=O)CC23CCCC2(C1)CN(C(c1cc(C#N)no1)=O)C3 c1(C(=O)NCC(CC)(CC)NC(=O)C(F)=C2CCC2)cc([N+](=O)[O-])cnc1N S(=O)(=O)(c1ccc(NCc2ccc(C#N)cn2)c(Br)c1)NCCCCCCC=C C1(C(=O)NC(C)C(O)C(C)C)(CNC(C(CO)OC)=O)CC2(CC2)C1 c1(C(N2CCCC(Cn3ccnn3)C2)=O)cnc2n[nH]c(Br)c2c1 c1(OC)nccc(C(=O)NCc2cc(C(=O)NC(C)C(C)n3cncn3)n(C)n2)n1 c1(CC(C)C)cc(NC(c2ccc(-n3cccn3)cc2)=O)n(-c2ccccc2)n1 c1(SC)ccc(OCC(=O)N(CCCCCNC(c2ccoc2Cl)=O)C)cc1.C1(C)CC1 N1(C(C(CC)(C)O)=O)CCCC(C2CCN(C(c3c[nH]nc3C3CC3)=O)CC2)C1 Cc1cc(C(N2CCOCC2CN(C)Cc2ncc(C)o2)=O)cc(Cl)c1 Cc1ccc(C(N2CCCCCC2CNC(=O)C(F)CC2CC2)=O)cc1F CCC(C)C(O)C(=O)N(C)CC1CCN(C(c2ccc(-n3ccnn3)cc2)=O)C1 N1(C(Cc2cnc(C)[nH]2)=O)CC2(CCC2NC(C2CCC(N(C)C)CC2)=O)C1 C1(NC(C2CC(CC)C2)=O)CCC(O)CN(C(=O)CC=Cc2ccccc2)C1 C1(NC(c2cncc(C#C)c2)=O)(CNC(C2CC3CC3C2)=O)CC2CCC1CC2 C(=O)(C1CCc2nccn21)NCC1(O)CCCN(C(CNC(C)=O)=O)CC1 C1(C(N(C2CCN(C(C3(CF)CC3(F)F)=O)CC2)CC)=O)CCn2nncc2C1 C(=O)(C1CCCn2c(C)cnc21)Nc1cccc(CNC(CSCCCC)=O)c1 C1(C(=O)OC(C)(C)C)CCS(=O)(=NC(=O)CC23CCCCC2C3(F)F)CC1 CCCC(C)CC(=O)NCCCCC(CO)NC(=O)Cc1cncnc1 c1(OC)cc(C(N2CCC(C)(NC(=O)COCC3CC3)CC2)=O)cc(F)c1 Cc1c(Cl)sc(Cl)c1C(=O)OCC(C)NC(c1ccccc1)=O C1(CNC(C(C)(C)N(C)C)=O)CC2CCC(C1)N2C(C12CCC1C2)=O c1(C(=O)NCC(C2CC2)NC(c2n(C)c(Cl)c(Cl)c2)=O)c(F)ccc(Cl)c1N C1(C)(C(=O)NC2CC(N(C(=O)CCC3CCCC3)C)C2)CCOCC1 CCC(C)(CCC(C)C)C(=O)NCC(C)CNC(=O)C(C)(C)c1sccc1Cl n1(C(C=C)C)nc(-c2ccccc2C)nc1C1CCC(F)CC1 CS(=O)(=O)C(C(=O)NC1C2CCC1N(C(=O)COc1ccc(Cl)cc1)C2)C1CC1 c1(C(=O)NCCCN(C(=O)CCCc2sccc2C)CC)cn2cccnc2n1 c1(OC)cc(N(C)CC2CCCN2C(C2CC2(C)C(C)C)=O)nc(OC)n1 C(=O)(C(F)C(F)(F)F)NC(CCSCC)C(=O)NC1CCCC1C1CC1 Cc1cc(CC(=O)NC(CNC(=O)C(C)c2ncco2)C2CC2)n[nH]1 C1(Cn2cc(CCSC)nn2)CN(C(c2sc(C)nc2Br)=O)CCO1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(C)CNC(c1ccc(C(C)(C)C)cc1)=O c1(C(C)C)nc2cc[nH]c2c(=NCCN(CCCOCCNC(=O)C(C)C)C)[nH]1 C(=O)(C#CC1(C)CCCO1)N1CCN(C(C(C)C)=O)CC1c1cccc(Cl)c1 Cn1cc(C(=O)NC2CN(C(=O)CC3CCOC3)C(C)(C)C2)c2cc(F)ccc12 C1(C)(C(N(CCS(=O)(=O)NC)C)=O)CN(C2CC2)C1=O.C(C)(C(=O)O)SC c1(CN(c2ccnc(C3(N)CCC3)n2)C(c2ccco2)=O)ccc(F)c(F)c1 C(=O)(C1=NOC(C)C1C)NCC(C)NC(c1c(OC)ccnc1O)=O Cc1csc2cc(C(=O)NC3CC4CN(C(c5ccnnc5O)=O)CC4C3)[nH]c12 CCC(COC)C(=O)NC(CC1CC1)CC(=O)N(C(C)COC)C N1(C(C23CC(CN2C(C2CC24CCOCC4)=O)C3)=O)CCC2(CC1)CC2NC1CC1 CC1CC(NC(C2CCO2)=O)CCN1C(c1ccc(CN=[N+]=[N-])cc1)=O N1(C(C(CNC(COC)=O)C)=O)CC(O)CC1CO C12(C(=O)NC(C)CC(N)=O)CC(CCO1)N(C(=O)CC1CCCCN1C)C2 N1(C(c2cc(CC(C)C)[nH]n2)=O)CCC2CCN(C(=O)CSC(F)(F)F)C2C1 C(=O)(C(C)C(C)(C)C)NCCC1(O)CCN(C(c2c(SC)snn2)=O)C1 C1(NCCOCC(F)(F)F)CCCCN1C(C(C)SCC)=O c1(C(=O)NCC(CC=C)NC(=O)CC2CSCCS2)cc(OC)c(OC)c(Cl)c1 C1(C(=O)NCC(CC(C)C)NC(=O)CCCCCF)CC2CC2CC1C CCCC(O)CC(=O)NC(C)CN(CC(=O)NCc1csc(CC)n1)C C(CCNC(=O)CCn1cccn1)(C(=O)NCCc1nc(C)cs1)OC CC1CCN(C(c2occc2CNC(c2ccc[n+]([O-])c2)=O)=O)C1CO C1(NC(=O)Nc2ccc3nc(N)c(Br)n3c2)CCOC2(CCCOC2)C1 C1(NC(c2c(SC)nn(C)c2)=O)CCN(C(=O)CC2(C)CCC2)CC1F C12(C(=O)NC3CN(C(c4c(CC)csc4)=O)C(C)C3)CCC(OC)(CC1)CC2 C(=O)(C(C)C(C)C)NC(C1(C(NOC)=O)CC(=O)C1)=O C(=O)(C(C)C1=CCCC1)N1CC2C(NC(C(C)C(C)(C)O)=O)C2C1 CC1=C(C(=O)N2CCN(CC3CN(C(C4CCOC(C)(C)C4)=O)C3)CC2)CCC1 N1(C(C=C(CC)CC)=O)CC(CNC(=O)CCCN2CCOC2=O)C(C(F)F)C1 C1(NC(CNc2cccc(C(N)=O)c2)=O)C2Cc3ccccc3C12 N1(C(C2(C(=O)OC(C)(C)C)CC(=O)N(O)C2)=O)CC(C(F)(F)F)OC2(CCC2)C1 N1(C(C2(N3CCOCC3)CC2)=O)CC2(CCC2)CC1C(=O)NCCN1CCCC1 CCC1=NOC(CC(=O)N(C2CCCN(C(=O)C3=CCC3)C2)C)C1 N1(C(c2n(CC)ccn2)=O)CCC2CCC(C1)N2C(c1coc(C#N)c1)=O CC1CN(C(c2ncccc2N)=O)CC1C(N1CCC(CC(N)=O)C1)=O N1(C(CCSCC(=O)OC)=O)CC(NC(C2(OC)CCC2(C)C)=O)C(C2CC2)C1 O=C(CC1=CCCCC1)NC1CCC(NC(C2CC3(C2)CC3F)=O)CC1 C12(C(N3CCC(N(C(c4nnn(CC)c4C)=O)C)CC3)=O)CC1COC2(C)C C1(C(=O)NCC2CCC(C(=O)NC(C)(C)C(N)=O)C2)CC=CC(O)C1 C1(NC(Cc2ccc(C)s2)=O)COC2(C1)CN(C(=O)CCCc1n[nH]c(=N)s1)C2 CC(F)(F)CCC(=O)NC1CCC(NC(C2CCOC2c2nccn2C)=O)CC1 C(=O)(C1CCCc2sccc21)N1CC(CNC(C=C(C)c2ccsc2)=O)OCC1 C(=O)(C1Cc2cccc(Cl)c21)NCCCNC(Cc1ccn(C(C)C)n1)=O N12CCc3c(c(nn3C)SC(CCC)C1=O)C2.C(C)(=O)OCC c1(C(=O)NC2C(C)CCN(C(c3cc[nH]c(=N)c3)=O)C2)cnc(S(C)(=O)=O)s1 CC(C)(C)CC(O)CC(=O)N1CCCC(C)(NC(=O)CCOCC(F)(F)F)C1 c1(C(N2CCCC(CNC(c3[nH]c(CC)c(Cl)n3)=O)C2)=O)cc(C)c(F)c(C)c1 C1(C(=O)NC2C3(CN(C(C45CC(C)(C4)C5)=O)C3)CC2)CC(c2ccccc2)=NO1 Cc1cc(C2CC2)ncc1C(N1CCC(O)(C(C)NC(C2CCCS2)=O)C1)=O C1(CNC(c2ccnc(CSC)c2)=O)CCN(CC2(c3cc[nH]n3)CC2)CC1 C1(CCNC(C2CC(C(C)(C)C)C2)=O)CN(C(=O)CCCC2CC2)CCO1 N1(C(Cc2c(C)non2)=O)CCCC2CN(C(=O)CC3CSCCO3)CCC12 CC(C)C(O)C(C)(C)C(=O)N1CCC(NC(C2CCC(N(C)C)CC2)=O)C(O)C1 c1(CNC(C2CC(=C)C2)=O)c(NC(c2cc(Br)cnc2C)=O)cccc1C(=O)O CC(C)C(CCNC(c1cc(CO)on1)=O)NC(=O)CSc1nnc(S)n1C C(=O)(NN1Cc2ccc(Br)cc2C1=O)c1ccc(C#C)cc1C(F)(F)F c1(CN=C(NCC(CC)(C)C)NC2CCCC2)cccc(C)c1O CC(Cc1cccnc1)N=c1[nH]c(=NCC2CCCCN2C)c2ncccc2[nH]1 C(=O)(CCCCCCCS(C)(=O)=O)NC(C)C.C12CCCN1CCCN2 C1(SC)CC(c2ccccc2)CN(C(c2cnn(C3CCCNC3)c2)=O)C1 C(CCNC(C1CC1c1ccccc1F)=O)(C(C)C)NC(C(COC)C)=O c1(CC)cc(C(=O)N(C)CCNC(C2CC3C=CC2C3)=O)cc(C)c1 C1(C(=O)NC2CCC(CNC(c3ocnc3C(F)F)=O)CC2)SC2C=CC1CC2 CC1C(NC(=O)CSC(F)(F)F)C(C)CCN1C(=O)CC1CC1(Cl)Cl C(=O)(CCCCCN(C(=O)C(c1ccccc1)F)C)NCc1n(CCC)ncn1 CC(C)(C)C(O)C(=O)NC1CC1C(=O)NCCc1ccco1 N1(C(C=CC(=O)N(C)C)=O)CC2(C1)CN(C(=O)CCc1cnco1)CC2CO Cn1c(CNCc2cccc(C3(C)CCO3)c2)nc2cccc(Cl)c12 N1(C(CC=CC=C)=O)CCN(C(c2ncc(Cl)cc2Cl)=O)CC1C(F)(F)F c1(C(=O)NCCC2C(C)CN(C(c3ccc(O)nc3)=O)C2)c(F)cncc1Cl C1(N(C(=O)NCc2ncc(CC)s2)CC2CCOCC2)CCS(=O)(=O)C1 C(CCCCCCCO)=CC(=O)NCC1CN(C(c2cc(NC)nc(Cl)c2)=O)C1 c1(N(C(N(C)CC2(C)CCCCC2)=O)C)ccnc(CO)n1 CC(C)(C(=O)N1CCC1CNC(=O)CC1CCC(C2CC2)O1)c1ccc(Cl)s1 N1(C(C(C)NC(CC)(C)C)=O)CCC(O)(C(C)NC(=O)CCCn2ccnn2)C1 C1CC2CCC(C1)N2N(c1ncccn1)C.C1(C=O)(N(C)C)CCOCC1 C1(C(=O)NC2CC(C(=O)N(C(c3ccncn3)C)C)C2)CC(C)(C)CO1 Cc1cccc(C)c1S(=O)(=O)N(C1CS(=O)(=O)CC1O)C N1(C(COCC)=O)CCCCCC(NC(=O)CSc2ccc(C(C)C)cc2)C1 c1(C(N2CCC(Nc3cn(CC4(C)CCCCC4)nn3)C2)=O)cnc(O)c(Br)c1 Cn1cc(NC(=O)CC2CC(NC(c3csc(Cl)n3)=O)C2(C)C)c(C#N)n1 C(=O)(C1=CCCN(C(C2CCOC2(C)C)=O)C1)NCC(CC(C)C)OC Cn1c(C(N2CC3CC3(NC(c3cc(C#N)no3)=O)C2)=O)cnc1[N+](=O)[O-] c1(CC)cccnc1C(N1CCC(C(C)CNC(C2(CF)CC2)=O)CC1)=O C(=O)(C1(C)CCn2ccnc21)NCC(C)(C1CC1)NC(=O)Cn1cc(CO)nn1 c1(C(=O)NCC(CNC(CCCCC)=O)OC)ccc2cnc(C)cc2c1 C1(NC(C=CCN(C)CC)=O)C=CCN(C(c2coc(C3CCCC3)n2)=O)C1 c1(C(C)=O)ccc(C(=O)NC2CN(C(=O)CCN(CC(F)(F)F)C)C2)c(F)c1 N1(C(c2c(SC)cnn2C)=O)CCN(C(c2ccccc2OC(F)F)=O)C(C)C1 N1(C(Cc2c(C)ocn2)=O)CC2CCC(C1)N2C(=O)CCN1CCCS1(=O)=O c1(C(=O)NCCCCN(CCCNC(C(C2CC2)OCC)=O)C)ccc(C)nn1 C1(C(=O)NC(CC=CC)C(=O)N2CCCC2CNC(N)=O)CCOCC1(C)C N1(C(C(=O)NC2(C)CC2)C(C2CC2)C2CC2)CCOC2(CCC2)C1 Cc1ccc2cc(C(N3CCN(C(=O)CC(O)C(C)C)CC3CF)=O)cnc2c1 N1(C(c2cc(=NC)[nH]cc2)=O)C2CCCC1CN(C(c1cc(C)nnc1O)=O)C2 c1(C(=O)NCC(CNC(C(CC)NC(C)=O)=O)F)ncc(C(F)(F)F)cc1Cl C1(CC(=O)NCC2(C(C)C)CCC2)C2CN(C(=O)C(C)(C)C3CCC3)CC12 c1(NCC2CCC(NC(C3C(=O)NCC3)=O)C2)ncc([N+](=O)[O-])cc1Br c1(C(=O)NCC(C)CNC(=O)C=CC2CCCO2)cc(N)c(F)cc1Cl N1(C(C2(C3CCCO3)CCC2)=O)CCCC1C(=O)NC1COCC1COCC CCN=C(NCC)N1CCC(NC(=O)NC)C1.c12cc(c(C)c(Br)c1)NC2=O C(=O)(C(F)(F)C(O)c1ccccc1)NCC1N(C(CC=C)=O)CC(O)C1 CN1CCOC(C(N2CCC(N(C(=O)CNc3ccc(Cl)nc3)CCO)C2)=O)C1 N1(C(C(N2CC(c3cn(C)nc3)OCCC2)=O)=O)CCc2ccc(O)cc2C1 c1(CC)cc(C(N2CC(C(=O)NC3CCN(CCOC)C3)(CC)C2)=O)ns1 n1(CC)nc(C(C)C)cc1C(=O)OC1CCN(C2CNC2)C1=O CCC(C)(C(=O)NC(C)CN(C)C(c1cc(Cl)cc(Cl)c1)=O)C(N)=O C1(C(N(C(CO)CO)C)=O)CCCN(C(=O)C(c2ccccc2)O)CC1 C1(OC)CN(C(C2CC3CC3C2)=O)CC1NC(=O)CCc1nnc(C)n1C N1(C(C(CCC)NC(N)=O)=O)CC2CC(C1)N(C(c1cc(C)nc(Cl)c1)=O)C2 N1(C(C2(C#C)CCN(C(c3cc(C)oc3C)=O)C2)=O)CCOCC(C)(C)C1 CCC(C)CCCCC(=O)N1CC2(CCCN(C(=O)CC(C)(O)COC)C2)C1 CCC(O)C(C)C(=O)N(C1(CC(=O)NC2CC(C)(O)C2)CC1)C c1(CC(=O)NCC2N(C(c3n(C(C)C)ccc3)=O)CCOC2)cc(O)nnc1O N1(C(C2(CC)CCN(C(C(CCC)N(C)C)=O)C2)=O)CCN2CC(O)CC2C1 C(CC(C)C(=O)N1CCCCC1CNC(c1sc(OC)nc1Cl)=O)=CC CCC(CNC(=O)CCCCN(C)C(C1CC(OC2CC2)C1)=O)CC(C)C CCCCCCC(C)CC(=O)N(C)CC1(O)CN(C(=O)C(C(C)C)OC)C1 c1(C(N(C2CCCN(C(c3ccon3)=O)C2)C)=O)cc([N+](=O)[O-])ccn1 C(=O)(C(C)(C)C(c1nnnn1CCCF)NC1CCCC1SC)OC c1(C(N2CCN(C(c3c(C)n[nH]c3)=O)CC2C#N)=O)cc(C)c2cc[nH]c2c1 C1(NC(C(C)C#N)=O)CC2CCC1(C(=O)NC1CCC(C(C)O)CC1)C2 N1(C(C(CC=CC)C)=O)CCCC(C(=O)NCC(CC(C)C)N(C)C)CC1 c1(OC)c(C(=O)NC(C)CC2CCN(C(=O)CC(C)C)CC2)cccc1C CC(C)C(C#N)C(=O)NC(Cc1cnn(C)c1O)C(N1CCOCC(O)C1)=O CC1Oc2ccccc2N(CC(=O)Nc2cccn(C3CCSC3)c2=O)C1=O C1(CN(C(C(C)OCCN(C)C)=O)C2CC2)(NC(c2cnn[nH]2)=O)CCOCC1 N1(C(CC2C(C)=NOC2=O)=O)CCCC(N(C)C(c2cc[nH]c2)=O)CC1 C(=O)NC(CC)=O.C1(C)C(=O)NCC(=O)NCC(=O)N1.C1(NC)CCCC1 n1(CC)c(C(=O)NCCC2CCCN(C(c3ccncc3Cl)=O)C2)cnc1O c1(C(=O)NC2(c3ccccc3)CCN(C(=O)C3CC3)C2)ccc2c(c1)CCOC2 N1(C(CC(C(C)C)C)=O)CCC2(CC1)CCN(C(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O)C2 c1(CC(C2(OCC)CCC2)N2CCCC2)nncn1C CCCCC(C)C(=O)NCC1(O)CC(CNC(C2(C)CS(=O)(=O)C2)=O)C1 N1(c2ccnc(NCc3ccc(OC)cn3)n2)CCCC(C)(OC)C1 N1(C(C(C)C2CCOC2)=O)CC2CCCC1C2CNC(=O)CN(C)C(=O)C1CC1 C(C)(C(C(C)C)NC(c1ncoc1CC(N)=O)=O)NC(c1c(CC)con1)=O O=C(C(O)CC(F)(F)F)NCC(CC(=O)NCc1ncc[nH]1)C1CCC1 CC(C)CC(S(=O)(=O)ONc1ccc(C(N)=O)cc1)c1ccccc1 CC(C)C(C(=O)NC12CC(C(N3CCC3C#N)=O)(C1)C2)NC(C)=O C12(C(N(C(CNC(C(c3c(C)cccc3)C)=O)C)C)=O)COC(CCO1)C2 CC1CC(NC(=O)C=Cc2ncc[nH]2)CN(C(=O)CC(C)(C)C)C1 C(C)(C)(CCCCNC(=O)C(C)=CC1CC1)NC(c1nc(CCC)sc1)=O C1(C(=O)NC2(CNC(CCC(C)N(C)C)=O)CC2)CCCCCS1(=O)=O C1(F)(CNC(=O)C=Cc2cnccn2)CCCN(C(=O)C(O)C(F)(F)F)CC1 N1(C(c2c(C)nsc2)=O)CCC(CCCNC(=O)COC2CC2)CC1 C(c1cnn(C)c1C)=CC(=O)NC1CCC(N(C(c2ccc(SC)cc2)=O)C)C1 c1(CN(CCC)Cc2ccc(N3CCOCC3)cc2)cccc(OC)c1Cl C(=O)(C(CNC(=O)C(F)C(C)(C)O)C(C)C)NCC1(CCC=C)CC1 C1(C(=O)NC2(CO)CCCN(C(CC=CC)=O)C2)CC2(CCCC2)CO1 N1(C(CNC(c2ccc(C(=O)NC)nc2)=O)=O)CCN(C(=O)C(C)O)CC(C)(F)C1 C(CCC(C)(C)C(=O)NCCc1nc(C)no1)NC(c1ncn(CC)n1)=O c1(CNC(COCC(=C)C)=O)cc(O)nc(CNC(=O)C(C)C(C)C)n1 c1(CC2(CSC)CC2)nc(-c2oc(Br)cc2C)n(CCC2CC2)n1 c1(C(=O)NCC(CNC(CCSCCC)=O)C)cncc2[nH]ccc12 C#CC1(NC(C2(CNC(C3CC(C)CCO3)=O)CCC2)=O)CCC(C)CC1 C1(CNC(=O)C=Cc2nccs2)CC(O)CN1C(=O)C1=CCCS1 C1(c2nc(C3ON=C(C(C)(C)C)C3)on2)CCc2nnnn2CC1 c1(CN2CCCC(C(C)NC(c3c(SC)nccc3)=O)C2)c(Br)ccc(Cl)c1Cl c1(C(N2CCC(CN(C)C(C3CC3(Cl)Cl)=O)C2)=O)ncncc1N Cc1cc(F)ncc1C(=O)N(CC(C)CNC(=O)CSCCC(F)(F)F)C C1(CC(=O)NC(CCC=C)C)N(C(c2cc(CC)ncn2)=O)CCC1(C)C c1(CNC(C(N2CCCC(CCC=C)C2)=O)=O)c(C)sc(C)c1C CC12C3C4C1C1C2C3C41C(=O)NC1CCC(NC(c2cc[nH]c2)=O)C1 N1(C(CNC(=O)OC)=O)CC(F)CC1CNC(=O)CCC1CCCOC1 C1(NC(C(C(C)NC(CC2C(C)C(=O)CC2)=O)C)=O)CC(=O)N(C)C1=O Cc1sc(S(N)(=O)=O)cc1C(N1CC(NC(=O)CS(N)(=O)=O)CC1C)=O C(CCCC(=O)N1CCC(C)CC1C(=O)Nc1cc(Cl)cnc1O)(OC)OC N1(C(C2CCC(CC)O2)=O)CC2(CC2)CC1CNC(=O)C(C)CSC Cc1cc(=NCC2(C(N)=O)CCOCC2)[nH]c(=NCc2ncoc2C(C)C)[nH]1 c1(C(=O)NC2CCC(NC(c3cnc(C)s3)=O)C2)ccc(N2CCCC2=O)cc1 Cc1cc(F)ccc1C(N1CCC1CNC(C1CN(C)CCN1C)=O)=O O=C(C1CCc2nccn21)NCCCCC1CCN(C(c2coc(Cl)n2)=O)CC1 CC1OCCCC1C(=O)NCCN(C(=O)C=C(Cl)Cl)C1CC1 c1(C(N(C)CCN(C)C(C2(C3CCC3)CCC2)=O)=O)nnn2c1CSCC2 C1(CC)CN(C(=O)C(C)(F)F)CCC1NC(C1CCN(c2nc(C)cs2)CC1)=O c1(NC(c2cnc(F)cc2C(=O)Nc2cscn2)=O)ccc2ccccc2n1 CC1(CCO)CCN(C(=O)NCC(F)F)CC1.C12CCN(C1=O)CC2 C1(C(c2n(CC(=C)C)nnn2)NCc2sccc2Br)CCC2(CC2)C1 C1(C(C)C)CCOCCN1C(=O)CCC(=O)NC(c1ccc(C#N)cn1)=O C(C(CNC(c1cc2n(c1)CCC2)=O)S(C)(=O)=O)NC(CNC(=O)NC)=O N1(C(C(F)=C(C)C)=O)CCN(C(=O)C(c2ccc(F)cc2F)C)C(C2CC2)C1 c1(OCC)ccnc2sc(C(=O)NCC34CCCC(CN)(C3)C4)cc12 c1(SC(CC)CO)ccc(NC(=O)C(=O)N(C(c2cccnc2)C(C)C)C)cc1 C12(C(=O)NCCC(C)NC(CCSC)=O)CC3CC(C1)C(=O)C(C3)C2 c1(OC)ccc2cccc(NC(=O)NCC(c3ccccc3C)C)c2c1 C1(CNC(C(CC)N(C)C)=O)CN(C(=O)Cc2ccc(OC)cc2Cl)CCCO1 CC(C(=O)N1CCC(CCNC(=O)CC2CC2c2cccnc2)CC1)C(F)F C(=O)(N=c1ccn(C2CCC2)[nH]1)c1c(C(C)NC(=O)CCCN(C)C)noc1 Cc1cccc(C(C(=O)NCC(F)F)N(C)CC2COCCO2)c1F C1(C(=O)NC(C)(CNC(c2ccccc2)=O)Cn2cccn2)CN2CCN1CC2 C(=O)(CC(CC(C)C)NC(=O)CSC(F)(F)F)NC(CC=C)(C)C(F)F N1(C(c2c(OC)nsc2OC)=O)CCC2CN(C(C3CCOC3)=O)C2C1 N1(C(CC2C(C)=NNC2=O)=O)CC2CCOC2(CNC(c2cc(Cl)c(Cl)[nH]2)=O)C1 CCC(CCC(=O)N(C(C)CC(N1C2CSCC1C2)=O)C)OC c1(C(N2CC(CC=C)(NC(=O)CCCc3cccs3)C2)=O)c(C)ncn1O N1(C(C(CSC)C)=O)CCOC2(CCN(C(=O)CCC3CCC(=O)N3)C2)C1 C(=O)(N1OC2CCC1C2)C1N(C(c2sccc2F)=O)CCCCC1 c1(CCC(N2CCC(N(C(C=CCCCCC)=O)C)C2)=O)ccc(Br)c(F)c1 C(CCC1CCC1)(C(=O)N(C1CCC1C)C)NC(COC)=O C(=O)(CC(CN(C)C)CC)NC1CN(C(C(CC)=CCCC)=O)C1 C1(CN(C)C(C2CC2[N+](=O)[O-])=O)C2CN(C(=O)Cc3nccn3C)CC12 c1(CN2CC(F)(C(=O)NC3CC(C(=O)OC)C3)C2)c(C)cccc1Br N1(C(c2c(CC)con2)=O)CC(CCNC(c2c(C)noc2C)=O)C(C)C1 N1(C(Cc2scc(C)c2)=O)CCOCC1CN(C(=O)CC1CC(C)(C)CO1)CC c1(C(=O)NC(C(=O)NCCC=C=C)CCC2CC2)cc(C)n(C)c1C C1(CC(=O)NCC#CCNC(=O)CCC(=O)c2ccncc2)CCCCCCC1 Cc1cc(=NCC2CN(C(C)C)C2)[nH]c(N2CCOC(c3cccc(Cl)c3)C2)n1 c1(C(N2CCC(c3c(CNC(C4C(C(C)O)C4)=O)c[nH]n3)C2)=O)cnn(C)c1Cl N1(C(C(C(C)C)CN(C)C)=O)CC2CCCC(N(C(=O)C=CC3CC3)C)C2C1 C1(C(N(CCN(C(=O)CCNC(=O)C=CCl)CC)CC)=O)CCCCN1CC c1(C(=O)NC(CN(C(CCC=C=C)=O)C)CC)sc(C#N)cc1Cl C(CC(C(C)(C)C)NC(=O)CCn1cc(Cl)cn1)N(C(=O)CC1(C)CC1)C C(=O)(C1Cc2ccccc21)NC12CCC(C(N3C(C(CC)C)CCC3)=O)(CC1)C2 C(=O)(CCCC(=O)N(CC(C)NC(=O)C(C)OCCC(C)C)C)OCC N1(C(C2(CC)CC2(F)F)=O)CC(C)CN(C(c2cc(C)cc(O)c2)=O)C(C)C1 c1(CN(C(CNC(c2ccc(OCC)cc2)=O)=O)CC)cc(F)c(F)c(F)c1 Cc1nc(=N)[nH]cc1C(=O)NCCC(C)CCNC(=O)C(C)(O)c1ccccn1 C1(NC(c2n(C)c(Cl)cn2)=O)CC12CCC(C(=O)NC(C)(C)C)CC2 CCCCC(CNC(=O)CCc1ncccc1C)NC(C1CC2(CC2)CO1)=O C(=O)(C(C)(C)C(C)O)NC(CC=C)CNC(=O)CC=CCCCCC c1(C(N2CC3N(C(CC#N)=O)C(CC3)C2)=O)noc2cc(F)ccc12 C(=O)(CCCS(C)(=O)=O)N(CC(O)CN(C)C(c1cn(C2CCC2)nn1)=O)C c1(C(=O)NCC2N(C(C(=O)NCC3CC4C=CC3O4)=O)CC2)c(F)cccc1F C1(CNC(CCNS(C)(=O)=O)=O)CCC(F)(CNC(=O)Cn2ccnn2)C1 c1(C(=O)NCC2(CO)CCN(C(c3nccc(C)n3)=O)C2)ccc2[nH]ccc2n1 N(C(=NCCCCl)NCCN1CC2(COC2)C1)CC(C)C(F)F C1(NC(CC(C)=CC(=O)NCC2(C)CSC(C)=N2)=O)CC(C)(C)CN1C C1(C(N2CCC(CC=C)(NC(=O)C(c3ccncc3)C)C2)=O)CC12CCSCC2 CC1=C(C)CC(C(=O)NCCCC2CCN(C(C34CC(CO3)C4)=O)CC2)CC1 Cc1cc(C(=O)N(C(C)CCNC(C2(C(F)(F)F)CCCCO2)=O)C)c(C)o1 c1(C(N2C(C(N3CCC(N(C)C)C3)=O)CC2)=O)ccc2nc(Br)sc2c1 C1(C(N(C2CCC(NC(c3cc(OC)n(C)n3)=O)CC2)C)=O)CCC(F)(F)CC1 N1(C(C(C(C)(C)O)F)=O)CCC2C(CCN2C(c2cc(C#N)ccn2)=O)C1 N1(C(C2CC(C)OCC2)=O)CCCC(CNC(=O)C=Cc2cncs2)CC1 C1(CNC(C(F)=CCC)=O)CN(C(=O)CCOC2COC2)CCC1C(F)(F)F CC1CN(C(c2cc(Cl)n(C)n2)=O)CC(C)CN1S(C)(=O)=O c1(C(=O)NC(CCNC(c2ccc(OCC#C)cc2)=O)C)ccc(C)nc1OC C(=O)(CC(Cc1ccco1)NC(c1cc(COC)[nH]n1)=O)NCC1(C=C)CCC1 N1(C(c2ncn(CC)c2)=O)CCC2C(C(=O)Nc3cn(C)nc3O)C2C1 N1(C(C2CCCOCC2)C(=O)NCCCC(=O)OCC)CC2CCC(O)C2C1 c1(C(N2CC3C(CNC(c4c(COC)noc4)=O)C3C2)=O)cc2c[nH]nc2s1 c1(C(=O)OCC)sc2cnccc2c1NCC.C(CC(C)C)NC(=O)C(CN)OC C1(C(N(C2CCN(C(=O)CC3CC3(C)C)C2)CC)=O)CC(F)(F)C1 CON1CCC(CC(=O)NCC(C)CNC(C2(C)CC3CC3C2)=O)CC1 Cc1sc(O)nc1C(=O)NCC(C1CCOC1)NC(=O)C=C(Cl)Cl Cc1csc(C#N)c1CN1CCC(N)(CO)CC1 N1(C(C2(C#N)CC2)=O)CCC2CC(C(=O)NCC3(C4CCCCO4)CC3)C2C1 C(=O)(C(C)C(=O)N1CCCC1C1CCN(C(=O)COC2CCOCC2)CC1)OC Cc1ccc2c(c1)C(C(=O)NC(C)CCCNC(=O)COc1ccccc1)C2 Cc1nn(CC(=O)NCC2CC2NC(c2ccn(C(C)(C)C)n2)=O)cc1Br Cc1cc(C)n(CCC(N2CCOC(C(C)NC(=O)C=Cc3cnc[nH]3)C2)=O)n1 c1(C(=O)NC23C(CN(C(CN(CC)CC)=O)C2)C3)cc(Br)c2ncccc2c1 N1(C(CC=C)=O)CC(C(=O)NC2CCCCC2)C2(CCC2)C1 n1(CCC(N2C(C(N3CC(C(=O)OC)C3)=O)CC2)=O)nc(C)cc1C C(=O)(CC(C(F)(F)F)n1ccnc1)NCCCN(C(=O)Cc1cnoc1)C(C)C c1(C(C)C)cc(C(N2CCC(O)C(NC(C3C(C)(C)C3(F)F)=O)C2)=O)ccc1O C1(c2nc(-c3ccc(NC(C)=O)cc3)on2)CC2CC1N(C(=O)C(C)(C)F)C2 c1(OC)c(C(=O)NCC2CCCC2NC(=O)CCCNC(C)=O)c(C)nn1C c1(OC)c(F)ccc(F)c1C(=O)N(C)CC1(O)CCN(C(C2CC2C)=O)C1 C12(C(=O)OC)CC3CC1C2C3C(N1CCCC(c2ccon2)C1)=O N1(C(c2c(CC)ccs2)C(=O)NC2CCOC2)CCC(c2ccccc2)C(O)C1 C1(CN(C(CC2CN(C)C2)=O)C)CN(C(c2cccc(O)n2)=O)CC1O Cc1cc(C(N2CCCCCC2CNC(C2CCN(C)C2)=O)=O)c(C)c(C)c1 N1(C(C2CCN(C(c3c(CC)cno3)=O)CC2)=O)CCCC(C)(N(C)C)C1 c1(C(=O)NC2CC(CNC(c3cnc(COC)s3)=O)C2)cc(=O)n(C)cn1 N12CC3(CC(CO3)C(=O)NC3CC(C3)CC1=O)C2.C(CCC(C)(C)C)OC CCC(CC(C)C)C(=O)N(CC(C)(C)CNC(=O)CC1CCCCC1O)C C(=O)(CC(C)CNC(C1CSCN1C(C1CCS(=O)CC1)=O)=O)OC C1(CNC(c2cnc[nH]2)=O)CCN(C(C2CCc3nncn3C2)=O)CC1C1CC1 N1(C(CCC2(C)CC2)=O)CCC(CO)(CNC(=O)CC(C)(O)C2CC2)CC1 CCC(CN(C)C)C(=O)N1CCC(C(=O)NCC(=O)NCC)C1C CC1SCCCC1C(=O)NCC1(C(N2CC(F)C2)=O)CCCCC1 C1(N(C(c2cccc(N(C)C)n2)=O)C)CCCN(C(C2(Br)CC2)=O)CC1 C(c1ccc(F)cc1)=CCC(=O)NC1CCN(C(C2(CC)CC2)=O)CC1 c1(C(N2CCC(NC(C(C)Oc3cccc(F)c3)=O)C2)=O)csc2ccncc12 c1(C(=O)Oc2c(C)cc(C(=O)OCC)o2)ccc(F)cc1OC(C)(C)C c1(N2CCC(CNc3scc(C)c3)C(C)C2)ccc(S(=O)(=O)N(C)C)cn1 c1(C(=O)NCCOCCN(C(=O)C2=CCCC2)C)cccc(N)c1 C1(CNC(CC(=O)OC(C)(C)C)=O)CCCN(C(C2(C)CC2Br)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)NC1C(C)(C)CCN(C(CC2CC(C)C2)=O)C1 C=C(Cl)CC(C(=O)NCC(=O)NCCO)NC(c1ncnc(C)c1C)=O c1(CNC(C2(CC)CCC2)=O)ccc(C(=O)NCCCN2CCC2)o1 Cc1nc(C(=O)NC2CN(C(C3CC(=O)NC(=O)N3)=O)C2)ccc1[N+](=O)[O-] c1(C(c2nnnn2C2CC2)NC(c2occc2Br)C)ccc(Br)s1 Cc1n[nH]c2cc(C(=O)NC3CCCCC3NC(C3(C)CCCS3)=O)ncc12 S(=O)(=O)(c1ccccn1)N1CCN(C(c2cccc(SC)c2)=O)C(C(F)(F)F)C1 C1(C(=O)NC2(CC=C)CC2)CC=CC(n2cc(C3CCC3)nn2)C1 CC(C)(O)C(C(=O)NCc1n[nH]cc1C1CC1)NC(=O)CC1CCOC1=O C1(C(=O)NC(C2(O)CN(C(c3ccn(O)c(=O)c3)=O)C2)C)CC2(CC(=O)N2)C1 C1(CCC)CN(C(=O)C(CC)CCC)CCN1C(=O)Cc1ccc(C)cc1C c1(C(=O)NC2CN(C(C3CC4OC3C3CC43)=O)C2)c[nH]c2c(Br)cccc12 N1(C(C(CC=C)NC(C)=O)=O)CC(O)CCC1C(=O)NCC1CN(C)CCN1C c1(C(C(N2CC(CCNC(c3c(OC)ccnc3)=O)C2)=O)C)ccc(F)cc1F C1(C(N2CCC2CF)=O)CCC(O)CN1C(c1cc[nH]c1)=O CN1CCC(c2ccccc2)(C(N2CC3CC3(CNC(=O)C(C)(F)F)C2)=O)C1 c1(OC)nccc(NC(N2CCCC(c3nnc(C)o3)C2C)=O)c1Br C(=O)(CCCC(C)C)NC1C(CNC(c2c(CC)n(C)nn2)=O)CCC1 C1(C(=O)NCc2nnc(CC)s2)CC(C)CN(C(C2OC3CCC2C3)=O)C1 c1(C(N2CCCC(C(=O)Nc3cccc(F)c3Cl)CC2)=O)c(F)cc(Br)cc1Br C(CC(C)C(=O)NCCOC1(CNC(=O)Cc2cccs2)CCOCC1)=CCC c1(C(C)(C)C)ccc(C(C)(C)NC(c2ccc(CN=[N+]=[N-])cc2)=O)cc1 C(=O)(C1(C)CCCc2ccccc21)N1CC(N(C(=O)C(=O)NC(C)(C)C)C)C1 c1(C(=O)NCC2C(NC(c3c(CC)nccn3)=O)CCC2)c(C)ncnc1O C1(O)(C(C)NC(=O)C=CC(C)(C)N(C)C)CCN(C(c2c(C)n[nH]c2C)=O)C1 C1(C(=O)NC(C(C)C)C2CC2)CSCCN1C(=O)Cn1ccccc1=O C12(NC(=O)Cc3csc(-c4ccccc4)n3)CCN(C(c3ccsc3)=O)CC1C2 C12(NC(C3CC4(C3)CC3(CCC3)C4)=O)CCCCCC1N(c1ccncn1)CC2 C1(=CCNC(CC=C)CC)CCN(C(=O)OC)CC1 c1(C(N2CC(NC(=O)CCS(C)=O)CC(OC)C2)=O)ccc(Cl)c(Cl)c1N c1(C(N2CC(CC(C)NC(c3cnn[nH]3)=O)C2)=O)cc(Cl)c(Br)[nH]1 C(=O)(C1=CS(=O)(=O)CCC1)NCC1N(C(C2CCOC2)=O)CCC(C)C1 C1(NC(C2(CC)CC2)=O)COCC1CNC(=O)CC1(C2CC2)CC1 Cc1ncc(NC(C23CCC2CN(C(=O)CSc2ncccn2)C3)=O)nc1Br CCC(=O)CCC(=O)N(C(C)C(=O)NCc1ccc(F)c(C)c1)CC O=C(CCC(=O)c1ccncc1)NCC1CC(NC(C2CC3CCCC23)=O)C1 C1=CC(=O)Nc2ccc1cc2.C(C(C)(C)CC1CC1)NC(C(C)OCCOC)=O CCCCC(O)C(=O)NC(c1ccc(CNC(=O)CN(C)C(=O)N(C)C)cc1)C C(=O)(C(C)(C)CC(=O)N1CC(C(=O)NC(C)CCC(F)(F)F)CC1(C)C)OC c1(C(N(CC(O)CN(C(=O)C(C#N)=CC2CC2)C)C)=O)cncc(C(F)(F)F)c1 CC1CC(CNC(=O)NCC(c2cccc(Br)c2)c2ccccn2)CC(C)(C)C1 C1(C(=O)NCC(CO)NC(c2c(CC)nc[nH]2)=O)CC(C(C)(C)C)=NO1 CC1CN(C(C2Cc3ccncc3C2)=O)CCC1N=c1ccnc(Cl)[nH]1 C(CC(C(C)(C)C)NC(=O)C(C)OCCC(C)C)N(C(CN(C1CC1)CC)=O)C c1(C(=O)NC2(CO)CN(C(C(c3cn(C)nc3)=O)=O)C2)cccc2nc(O)[nH]c12 CN=c1nc(N(C)CC2(OC)CCC2)[nH]c(=NCCc2cscn2)[nH]1 c1(CCC(=O)NC2C(NC(c3c(SC)ccs3)=O)CC2)nc(O)c2cnn(C)c2n1 c1(-n2cc(CNC(C3CCCC(=O)O3)=O)nn2)ccc(Cl)cc1Br C1(NCc2c(C)oc(-c3ccccc3)n2)CCCOC12CCNCC2 N1(C(=O)OC)C2CCC1CC(c1nnnn1-c1ccccc1)(NC1CCC1)C2 CC(CNC(c1nnc(O)nc1O)=O)C(F)C(=O)N1CCC1(CO)CO C(C)(CC(=O)N(CC=C)OC)NC(C)=O.C1C(=O)N1CC#C C(=O)(C(O)CCC(C)C)NC(C(=O)NCC(=C)C)CCC1CC1 N1(C(CCS(C)(=O)=O)=O)CCC2(COC(CNC(c3c(Cl)cccc3Cl)=O)C2)C1 c1(OCC(N2C(C(C)NC(=O)C(C)(C)C(F)F)CCC2)=O)nn(C)cc1[N+](=O)[O-] CC1(C)C=C(C(=O)NC2CCN(CCNC(=O)CC3CC(C)(C)C(=O)N3)CC2)C1 N1(C(C2CCC(CC)O2)=O)CC(NC(=O)Cn2ccc(C)c2)C2CCCC12 N1(C(c2c(OC)cncc2)=O)CC2(C1)CN(C(=O)C(C)(C)SC)C2 CCCC(Cc1ccccc1)(c1nnnn1CCCF)NCCc1cscc1Br c1(C(=O)NC2CC(C)CN(C(=O)C=C(Cl)Cl)C2)oc2ccccc2c1Cl c1(C(=O)NC(CNC(CCC)=O)CC(F)(F)F)ccn2c(Br)cnc2c1 c1(C(N(C)CC2CCN(C(CC(C(=O)OC)C)=O)C2)=O)cc([N+](=O)[O-])c(C)s1 c1(C(C(N2CC(NC(C=CCCC)=O)C(OC)C2)=O)(C)C)c[nH]c2ccccc12 N1(C(c2cnc(C)nc2)=O)CCC2(C1)CN(C(=O)CC(C)(C)CN(C)C)CCO2 c1(Cc2n(CC(C)C)c(N3CCc4ccccc43)nn2)ncn2ccccc12 C(=O)(C(C)(C)CCS(C)(=O)=O)N1CC2C(CN(C(C(C)O)=O)C)C2C1 c1(C(=O)NC(C2CCN(C(C(C(C)C)(C)O)=O)CC2)C)cnc2cccnc2c1 CC1(N(C(=O)CCc2cnoc2)CC(=O)NCc2ccncc2)CC(O)C1 c1(C(N2CCC(O)(CCNC(C=CSC)=O)C2)=O)cnc(=NCCF)[nH]c1 CN1C(=O)OCC12CN(C(c1cn(CCNC(c3c[nH]nc3[N+](=O)[O-])=O)cn1)=O)C2 S(=O)(=O)(c1ccc2c(c1)OCCO2)C(C(=O)CN)=O.N1Cc2ccccc2-c2ccccc21 N1(C(C(=O)Nc2nnc(OC)s2)=O)CC(F)(F)CC1CN C(=O)(C(F)(F)NCc1cn(Cc2ccc(Br)s2)nn1)NCCC(=O)O c1(NC(CC)CNS(C)(=O)=O)ccc(S(=O)(=O)CC)cc1 CC1C(NC(c2ccc(C3CC3)o2)=O)CCCN1C(=O)CCC1CCCC1 c1(NC(c2ccc(CNC(C(C)NC(C)=O)=O)o2)=O)c(O)cccc1Cl CC(C)C(CNC(=O)C=Cc1ccc[nH]1)C(=O)NC(c1cncn1C)(C)C N1(C(C2C(=C)CC2)=O)CCN(C(C2CN3CCN2CC3)=O)CC1C(F)F N1(C(C2(C)C(C)CCC2)=O)Cc2ccc(CNC(c3ccc(Cl)cc3)=O)cc2C1 C1(CNC(C2(OC)CCCC2)=O)CC(F)CN1C(=O)Cc1ccsc1Br Cn1nc(C(=O)NC2CC2NC(C2(NC)CCOCC2)=O)cc1C(F)F C1(O)(CN(C)C(c2n[nH]cc2Cl)=O)CN(C(=O)C(C)(O)C2CC2)C1 c1(CCC(=O)NCC2CCN(C(=O)C(F)CC3CCC3)C2)ccccc1Cl N1(C(CN2CCC(OC)C2)=O)CCCC(C)C1CCNC(=O)CCC(C)(F)F C(=O)(CC(C)C(=O)OC)NC(C(=O)NC(CCC)C1CCCC1)Cn1cncn1 CC(C)C(C(=O)N1CCCC1)NC(=O)CC(C)O C1(CC)CCN(C(=O)C=CCO)CC1NC(=O)C(CC)N(CC)CC C1(C(=O)NCCCCl)CC12CCN(C(=O)OC)C2.C(=O)C(F)(F)F CC(C)(C)C1=NOC(C)(C(N2CC(O)(CCNC(c3cc[n+]([O-])cc3)=O)C2)=O)C1 C=C(C)CC(=O)NCCN(C(=O)Cc1cc(Br)cs1)CCOCCO N1(C(CC2CN(C(c3ccc(Br)cc3)=O)C2)=O)CCC(O)C(O)C1 n1(CC)cc(C(=O)NC2CC2NC(=O)Cc2csc(-c3ccccc3)n2)c(C)n1 c1(NCC2C(c3cn(CC)nc3)OCC2)nc(C(F)(F)F)ccc1C#N CC1CN(C(c2ncc(C(F)F)s2)=O)CCC1NC(c1conc1C1CC1)=O c1(C(N(C(C2CC=CCC2)C(=O)NCCC(=O)OCC)C)C2CC2)cnn(C)c1 c1(C(NNC(=O)NCCCOCC(C)C)=O)cc(Cl)cc(Cl)c1 N1(NCCOCCN(C(N=c2c(C)c[nH]cc2)=O)C)Cc2ccccc2C1=O C(=O)(CC(C)(F)F)NC1(C(NOCC(=C)C)=O)CC(F)C1 Cc1nc(O)sc1C(N1CCC(CC(=O)NC2CC(CO)N(C)C2)C1)=O Cc1cc(C)c(C(=O)NCC(O)CN(C(=O)C=Cc2cn(C)cn2)C)[nH]1 C1(C2CN(C(=O)Cn3cccc(C)c3=O)C2)(NC(c2c(C)nccc2)=O)CC1 C=CC(C(=O)NC1CC(NC(=O)CSCC(F)(F)F)C1)OC C12(CNC(C3=CC(C)(CC)C3)=O)CCCC1N(C(c1csc(C(F)F)n1)=O)CC2 C1(C(=O)NC(CC)(C)CNC(=O)C=Cc2scnc2C)CCC(O)CN1C C1(CC)CCOC1C(=O)NC1CC(C)(NC(=O)CCc2ccoc2)C1 N1(C(C2CCN(C)C2)=O)CCC2C(C1)CN2C(c1ccc(-c2ccco2)o1)=O c1(OC)ccc(-n2nnnc2C2(NCc3ncc[nH]3)CCCC2CCF)cc1Cl c1(C(N2CCC(C(=O)NC(CC#C)CC)C2C)=O)cccc(C#N)c1 c1(N(C)CC2CCCN(C(c3cnc(C)[nH]3)=O)C2)ncnc(C)c1C#N N1(C(c2nc(C(C)NC(C(CC)C#N)=O)oc2)=O)CC2(CCC(C)OC2)C1 C1(OC)CC(NC(=O)Nc2ccccc2OC2CCNCC2)C12CCCC2 N1(C(C(C)=C(CC)C)=O)CCN(C(=O)CP(C)(C)=O)CC1c1ccnn1C N1(C(c2cc(CC)nn2C)=O)CCC2(CCCN2C(C2CCCN2C)=O)C1 C12(C(N(CC)CC)=O)CC(CO1)N(C(=O)CC1(O)CN(C(=O)OC(C)(C)C)C1)C2 S(=O)(=O)(c1cccc(=NCC(C)NS(C)(=O)=O)[nH]1)N1CCC(CC)C1 Cc1cc(Br)cnc1C(N1CCC(C)(NC(=O)CN2CCOCC2)CC1)=O N1(C(C2CCCOCC2)=O)CC23CCCCC2(C1)CN(C(C1CCCOC1)=O)C3 CCC(O)C(F)(F)C(=O)N(C)CC1CCCN1C(C1CC(CC(F)(F)F)C1)=O C(C(C)C(C)C(=O)NC(C)CNC(c1cnc(N(C)C)cn1)=O)OC C1(NC(CCOCCC)=O)CCCC1CNC(=O)Cc1cnns1 CCC(Cc1ccccc1)CC(=O)NCCNC(=O)C(C)(C)n1cccn1 N1(CC(=O)NCCOc2ccc(C#C)cc2)CC(C)OC2(CCCOC2)C1 C1(NC(C2(CC)CC2)=O)CC2CCC1CN2C(C1CCCN1C1CC1)=O O=C1CCC(n2ccnc2-c2cccc(-c3cccc(Cl)c3)n2)CN1 CCN=c1[nH]c(C)cc(=NCCNC(=NCCCC)NCC(C)(C)C)[nH]1 C1(C(=O)NCCC2(O)CN(C(C3(C(C)C)CCC3)=O)C2)CC(C2CC2)=NO1 C1(C(=O)NC(CC)(CNC(c2cccnc2N)=O)CC)CN2CCC1CC2 N#CC1CCCC1N=c1[nH]c(=NCCc2ncccc2C(F)F)[nH]c2c1SCC2 N1(C(C2CC(=O)CC23CCC3)=O)CC(C2CCN(C(C3CC34CCC4)=O)CC2)C1 N1(C(CSCCCC)=O)CC(NC(=O)CC(CC)C2CCC2)C2(CCOCC2)C1 c1(OC)ncc(C(=O)NCC2(F)CC(NC(c3csc(Cl)c3)=O)C2)s1 CC1(C)COC(C(=O)NCC2(NC(=O)CCOCCN(C)C)CC2)CO1 c1(CC)cc(C(=O)NC2CCN(CC(CC)CC)C2)no1 Cn1ccc2cccc(C(N3CCC(CO)(NC(=O)Cn4cccn4)C3)=O)c12 C=CC1(CC(=O)NC(CNC(C2CC2C2CC2)=O)CO)CCOCC1 c1(C(=O)NCC(C)(C2CCC2)NC(C(C=C=C)C)=O)ccc(OC)nc1Cl CCCCCCCCNC(=O)CC1CCCCN1C(C1CC1c1ccccc1)=O c1(N2CCN(C(c3c(OC)csc3)=O)C3(C2)CC3)ncnc2cc(F)ccc12 N1(C(c2cc(SC)oc2)=O)CCCCC1CN(C(=O)CNS(N)(=O)=O)C1CC1 CN1CCCCC1CCC(=O)NCC(C1CCC1)NC(=O)C1=CCOC1 c1(CNC(NC(=O)NC2(Cc3ccccc3)CC2)=S)ccc2c(c1)OCO2 c1(C(=O)NCc2cc(C(N3CC(CC#C)OCC3)=O)sc2)cc(C#N)oc1C C1(N(C)C(C2CC2[N+](=O)[O-])=O)CCC(CNC(C2(O)CC2(C)C)=O)CC1 CC1(C(N2CC3CC2C3NC(c2cnn(-c3ccccc3)c2)=O)=O)COC(=O)C1 N1(C(CC(CC2CC2)NC(c2c(C#N)ccnc2)=O)=O)CCn2nccc21 C1(NC(=O)NCC(O)Cc2cccc(F)c2)=C2C=C(Br)NC(=NC=N1)C2 CCCCS(=O)c1ccc(CC(=O)N(CCCCCO)CC)cc1 Cc1ccc(C(N2C3CCC2C(C(N2CCC(CO)C(O)C2)=O)C3)=O)cc1C N1(C(c2c(CC)nco2)=O)CCC2C(C1)NC(=O)CN2C(c1ncnn1CC)=O C1(C(=O)NC2CC3(C(NC(c4c(OCC)cccc4)=O)C3)C2)CC(=O)NC(C)C1 C(=O)(C1=COCCC1)NCC(C1CCN(C(C(CCOC)C)=O)CC1)O Cc1nc(Cl)ncc1NC(C1C=CCN1C(C1CCCS1)=O)=O c1(OC)cc(OC)c2c(c1)N(C(N1CCCNC(=O)CC1)=O)CCC2 C#CCCCC(=O)N1CC2CC1(CNC(c1cc(-c3ccccc3)ncn1)=O)C2 CC(C)C(C)CC(=O)N1CCC(C(C)NC(=O)Cc2cc(O)nnc2O)CC1 C=CCC(C)C(=O)NCC1CN(C(=O)COC(C)C)CC1OC c1(C(=O)NCCC2CCCN(C(C3CC(O)C3)=O)C2)cnc2cc(Br)ccn12 CC(C)(CCCNC(c1cc(-c2ccoc2)on1)=O)NC(C1CC2CCC1O2)=O Cc1cnc(C(C)NC(C2CCCC2CNC(c2csnc2Cl)=O)=O)nc1 CCC(C)(C)CCCC(=O)NCC1CCN1C(c1cncc2ccsc12)=O n1(CC2C(C(=O)SC3CC3)C2)nc(C)c(C(=O)NC2(CCCOC)CC2)c1C C(=O)(C(O)CC(N)=O)N1C(C(=O)NCC(CSC)(C)C)CSCC1 C(=O)(C(O)C(C)CC)NCC1CC(NC(CC=C)=O)C1 c1(C(C)N(C(C)CCC(=O)OCC)C(C=CC)=O)ccc2c(c1)OCCO2 c1(C(N2CC(C3(NC(C(C)SC(F)(F)F)=O)CC3)C2)=O)cc2c(cc1N)CCC2 C1(C(N2CCN(C3CCC(OCC(=O)O)CC3)CC2)=O)CCc2nc[nH]c2C1 N1(C(CCC(=O)NC)=O)CC2(CCC2)CC1C(N1CCC1C(=O)NC1CC1)=O C1(C(=O)NCCC2(NC(c3ccncc3C)=O)CC2)(COC)CCOCC1 Cc1nccnc1CNC(=O)C(C)(C1CCC1)NC(=O)C=CC(C)C C=CCCCC(C)(C)C(=O)N(C)CC1(NC(=O)C(C)n2cnnn2)CC1 N1(C(CC2(COC)CCCC2)=O)CCC(C)(CNC(=O)C(C#N)C2CC2)CC1 N1(C(C)=O)CCOC(C(=O)NCCC2(NC(c3ccon3)=O)CC2)C1 C#Cc1cccc(CC(N2C(CC(=O)NCc3ccc(C)s3)C3CCCC23)=O)c1 N1(C(C2CC3(CCO2)CC3)=O)CCN(C(=O)CC2(COC)CC2)CC1C N1(C(C(CSC)O)=O)CCCC(C(=O)N(C)Cc2cccc(C)n2)C1 c1(OC)ccnc(C(N2CC(C)(CNC(c3nn(C)cc3SC)=O)C2)=O)c1 N1(C(=O)Cc2csnn2)CCC2CC12C(=O)NC1CC1c1ccsc1 c1(NC(C)=O)ccc(C(N2CCC(O)(C(C)NC(C3COCCO3)=O)C2)=O)cc1 N1(C(c2ccc(C)cc2N)=O)CCCC2CN(C(=O)COC3CC3)CCC12 C1(F)(C(N2CCC(NC(CC)=O)C2)=O)CCN(C(C2CCCO2)=O)C1 C1(C(N2CCC(OCC(=O)NC3(C)CC(O)C3)C2)=O)CC2CCC1CC2 C1(C#N)(C(=O)NC(CC)CN(C(c2coc(C(=O)NC)c2)=O)CC)CCC(=O)CC1 C1(NC(CCSC)=O)CCCC(CC(=O)N(CCn2cncn2)C2CC2)C1 C1(C(=O)NC(C)Cn2cccn2)CCCCC1CNC(c1ccns1)=O CC1=C(C(=O)NCCC(C)(C)NC(=O)CCC2CC(C)(C)CO2)SCCO1 CC(C)(C(=O)NCC1CC(F)(CNC(=O)C=Cc2ccc(O)cc2)C1)C(F)F N1(C(CSC)=O)CCC2(CC2C(=O)NCC(CSC)OC)C1 C=Cc1ccc(C(=O)NC2CC3CC2N(C(=O)C(c2cncn2C)O)C3)cc1 C12(C(=O)NCC3C(CNC(c4nc(CC)oc4C)=O)C3)CCC(=O)N1CCS2 CON=CC(=O)NCC(CNC(=O)C=CCOC1CCOCC1)OC c1(CN(CCCCC=C)C(C)=O)ccc(C)c(C)c1.C1(CC)CN1 C1(C(=O)NC(C)CNC(C2CC3CCCC(C2)C3)=O)CC(=O)c2ccccc2O1 C1(NC(c2conc2C(F)(F)F)=O)COCCN(C(C2CC(C3CC3)=NO2)=O)C1 C(=O)(CS(=O)(=O)CC(=O)OC)NCC(C1CC1)NC(C(CCOC)OC)=O C(CCCC(=O)N1CCOC(C(=O)NC2CCN(C3CC3)C2)C1)(OC)OC CC1=C(CNC(=O)C#CCNC(=O)CCC(N)=O)CCC1 CC1(C(=O)NCCc2ccccn2)CC12CCN(C(=O)COc1ccccc1)CC2 c1(CNC(CN2CCN(C(C3(CC)CC3)=O)CC2)=O)cc(C)cc(F)c1 CC(C)S(=O)(=O)CC(=O)NC1CC2CN(C(C3(CC4CC4)CCC3)=O)CC2C1 C=CCC(CC)C(=O)NC12CC(NC(=O)Cc3cc(C)ccc3F)(C1)C2 c1(C(N2CC(CNC(C3CC4(CC4)C3)=O)OCC2)=O)ccnc(N2CCCC2)n1 C(=O)(C1=NNC(=O)CC1)NCC(=C)CCNC(=O)CCOCCN(C)CC C=C(C)CCCC(=O)NC(C)CC(C)NC(c1ccc(-c2cc[nH]n2)cc1)=O CC1CC(C)(C(=O)NC(C)(C)CN2CCN(C(=O)C(C)(C)CC#N)CC2)CCO1 N1(C(CCC)=O)CCCC(C(N2CCC(NC(=O)C3=NOCC3)CC2)=O)C1 CC(C)(C)C#CC(=O)N1CCC1C(=O)NCC(C1CCCC1)N(C)C C(=O)(C(CO)C(C)(C)C)NC1CN(C(CS(N2CCC(C)CC2)(=O)=O)=O)CC1O C1(C(=O)NC2CCC2CNC(=O)C(C)(C)C)(OCC)CCCC1.C1(=O)C(C)N1 C(C(=O)N1CCCC(C(C)N)C1)(C(C)C)c1nc(C)sc1 c1(C(=O)NCC2(O)CN(C(c3cccc(N)n3)=O)C2)c(F)ccc(Br)c1F N1(C(CSCCC(C)C)=O)Cc2occ(NC(c3cnn[nH]3)C3CC3)c2C1 CC1(NC(=O)CNC(c2ccoc2)=O)CCN(C(c2ccc(Cl)cn2)=O)CC1 c1(OC)cccc2c1OCC(C(N1CCCCCC1CCO)=O)C2 C(=O)(C(C)C(C)(F)F)NC(C(C)NC(C(C(C)C)O)=O)CO C1(C(=O)NC(C)Cc2cn[nH]c2)COC(CNC(=O)Cc2ccc(Cl)s2)C1 C=CC1(C(=O)OCC2CCCCCC2)CCCC1 c1(C(N2CC3C(CNC(c4c(C)cccc4)=O)(C3)C2)=O)cncc(O)c1Cl C1(CNC(C2(OC)CCSCC2)=O)CCC(C)CN1C(=O)COCC1(F)CC1 c1(C(=O)NCCC(N)=O)ccc(-c2cn(CCCCF)nn2)cn1 N1(C(CCSCC)=O)CC(NC(c2ccc(C)c(OC)c2)=O)CC1(C)COC c1(N2CCC(CNC(c3cnc(OC)s3)C)C2)cccnc1Cl c1(C(=O)NCC(CN(C(C2(CC#C)CCC2)=O)C)C)ccn(CCO)c(=O)c1 c1(C(N2C3C(CNC(c4cnc(O)s4)=O)C(C3)C2)=O)cc(Cl)ccc1Cl N1(C(CC(C)(C)OC)=O)CCN(C(c2cc(C)ccc2N)=O)C(CC(C)(C)C)C1 Cn1ccc(C=CC(=O)NCCCCNC(c2ccc(Cl)o2)=O)c1 CC(N=c1[nH]c(=NCC(CO)C2CCCCC2)[nH]c2c1CCC2)C1(NC)CCC1 c1(-n2c(C(=O)NC(C)CCNC(=O)Cn3cccc3)cnc2)ccccc1F N1(C(C(CCC)N(C)C)=O)CC2CCCC(CNC(c3cnns3)=O)C2C1 N1(C(C2CCCC(NC(C(C)(C)CF)=O)CC2)=O)Cc2cccc(C#N)c2C1 O(N1CCC(CC(=O)NC(CNC(=O)C=CCN2CCC2)CO)CC1)CC C1(C(N(CCNC(C(C(C)C)NC(=O)OC(C)C)=O)C)=O)CC2CCC1CC2 c1(C(=O)NC(CN(C(c2ccn(CCCC)n2)=O)C)CC)cccc(C)c1CC CN1CC=C(CC(=O)NCC(O)CCNC(c2ccc(C#N)c(Cl)c2)=O)CC1 CCC(CCCC(=O)NCC(C)CC1CC1)NC(c1sccc1C)=O CC1CC(C)CN(CCCN2CCN(C(C(=O)Nc3ccsc3)C3CC3)CC2)C1 N1(C(C(C=C)(C)C)=O)CCC(C(F)(F)F)C(NC(=O)C(c2cncn2C)O)C1 C1(CN(C(CC2(COC)CC2)=O)C)CCCCN1C(=O)C(C)CNC(=O)OC Cc1nnc2n1CCC(C(=O)NC1CCC(NC(C3(C(C)(F)F)CC3)=O)CC1)C2 C1(C)(C(N2CC(C(N)=O)(CNC(C3ON=C(C)C3)=O)C2)=O)CCCCNC1=O C1(C(=O)NC2C(C)(C)C2C(=O)NCC(F)(F)F)CCC2(CC2)C1 C1(C(=O)NC(C(C)NC(c2ccc[nH]2)=O)CO)CC(C)(C)C(C)(C)C1 C(N1CCCC(c2ccncc2)CC1)c1nnc(CC)s1 Cc1cc(=NC2CCCC2C#N)[nH]c(=NCc2cccc(S(C)(=O)=O)c2)[nH]1 N1(C(c2c(OCC)ccs2)=O)CCC2CC1CN(C(C1COCC(C)(C)O1)=O)C2 C(=O)(C(C(C)O)N(C)C)NCCCN(CCC)C(C1CCC(=O)O1)=O c1(C(=O)NC2CCCN(C(CC(CC)OC)=O)C2C)cnc2[nH]c(O)nc2c1 c1(CC(=O)NCC(CNC(C(CN(C)C)(C)C)=O)F)ccc2cccnc2c1 C1(COC)(CNC(C2CC(N)C23CCC3)=O)CCN(C)CC1 C1(CC(=O)N(C2CCN(c3nnc(C(C)(C)C)s3)CC2)CC)CCCS(=O)(=O)C1 c1(CC(=O)NCC(N(C(CC=C(C)C)=O)C)C2CC2)coc2ccc(C)cc12 N1(C(c2c(C(C)C)occ2)=O)CC(NC(c2cncc(N)n2)=O)C(C)C1 C1(NC(CCOC(C)C)=O)CC2C1CCN2C(c1ccnc(S)c1)=O C(=O)(C(=O)CCC(C)C)N(C1(C(=O)C(=O)O)CC1)C.C(CCN)N(C(C)=O)C N1(C(c2c(NC)cnnc2)=O)CC(NC(=O)C2=CCN(C)C2)CC1(C)C C1(C(=O)NCC2(CN(C)C(C3CC3(Cl)Cl)=O)CC2)OCC2CCCC1C2 Cc1cc(C(=O)NC(C(N2CCCCC2CCO)=O)c2ccco2)nnc1O C1(OC)(CNC(c2cnsc2C)=O)CCN(C(C2(C#N)CC2(C)C)=O)C1 C(=O)(C1=CCS(=O)(=O)C1)N(CC(CNC(C(CC)(C)C#N)=O)(C)C)C c1(-c2cc(C(=O)NCC=CCNC(C(=O)NCC(F)(F)F)=O)on2)cccc(Cl)c1 N1(C(c2n(CC)ccn2)=O)CCCC(O)(CNC(=O)Cc2ccncc2Cl)CC1 c1(C(=O)NC(CNC(c2n(C)ccn2)=O)(C)CO)cc(Br)cn1C C(=O)(C1CCc2nccn21)NC(C)(CO)C(=O)NCCC1(O)CCCCC1 C1(CNC(=O)CC2CC=CC2)CN(C(c2ccn3cccc3c2)=O)C2(CCC2)C1 N1(C(CC2(COC)CC2)=O)CC(NC(c2c(C3CC3)cnn2C)=O)C(SC)C1 N1(C(C2(CNC(=O)Cc3ncccc3OCC)CC2)=O)CCC(C)C(CO)C1 c1(C(=O)NC2CC(NC(C34OCC(C(C)C)(C3)C4)=O)C2)cc(C2CC2)nc(O)c1 c1(C(=O)NCC2N(C(C(C)SC(C)C)=O)C3C(C2)C3)ccnn2ccnc12 C(=O)(CCCCCOC)N1CC2C(c3cn(CCOCC)nn3)(C2)C1 C(C)(CCC(=O)c1cccs1)NCCOCCOCC=C C1(CCC)(C(=O)NC2CC2NC(c2ccccc2OC(F)F)=O)CCNC1=O c1(CC(=O)NC(C2CCN(C(=O)CC3CCC4CC34)CC2)C)cc(Cl)sc1Cl c1(C(CC(=O)NCC(C)NC(CCN(C(C)=O)C)=O)C)c(C)n[nH]c1C Cc1nccn1CCCC(=O)NCC(C)CN(C(=O)CCN1CCCCC1)C C1(NC(C(C(CC)C)O)=O)CCSC12CN(C(c1cnc(N)c(N)c1)=O)C2 C(=O)(CCCCCSC)N1CCC(N(C(c2cc(C)sc2C)=O)CC)C1 CCC(CC(=O)NCC1(OC)CN(C(c2cnn(C)c2OCC)=O)C1)C(C)(C)C c1(C(=O)NCC(C)(C)NC(C2CCC23CCCO3)=O)cccc(N)c1Br C1(C(=O)NC2(CC=C)CN(C(=O)CCc3nccs3)C2)CCCOC1C Cc1coc(C(c2nnnn2Cc2nnn(C)n2)NC2(C)CC2(C)C)c1 C=CCC(CC=C)C(=O)N1CCC(C(F)(F)F)C(CNC(=O)CC(C)C(C)C)C1 CC1CN(C(C2(C#N)CCCOC2)=O)CCN1C(C1CNC(=O)C1)=O C(=O)(CS(=O)(=O)CCC)N1CCN(C(C(C=C=C)C)=O)C(C(F)F)C1 CN1CCCC2CN(C(C3CC4(C3)CC3(CNC3)C4)=O)CCC12 c1(C(=O)NCc2c(Nc3cnc(Br)cn3)cccc2F)ccc([N+](=O)[O-])c(O)c1 N1(C(C(C=C)C)=O)CCC2(CC1)CC2CNC(C1CC(OC)C1)=O c1(C(=O)NCCC(=C)CNC(c2cnoc2CC)=O)c(Br)c(C)nn1C c1(NCC2(C)N=C(C)SC2)ccc(S(=O)(=O)NCc2c[nH]nc2C(C)C)cc1Br N1(C(c2c(C)occ2C(=O)O)=O)CCCC(C(C)C)CC1 Cc1[nH]cc(C(N2CCCC(C)(CNC(c3ccc(O)cn3)=O)C2)=O)c(=O)c1Cl O(NC(=O)C(C)(C)CCNC(c1c[nH]c(=NC)s1)=O)CC(=C)Cl CCC(C(=O)NC(CNC(c1ncccn1)=O)C(C)C)C(C)C C1(C(N2CCC(NC(=O)C3=CCCCC3)CC2)=O)CC12CCc1ccccc12 C12(NC(C3CCN(C)CC3)=O)CCCN(C(c3cnc4n3CCS4)=O)C1C2 c1(OC)ccc(C=CCSC)cc1S(=O)(=O)NC1CCCN(C2CCCC(C)C2)C1 CCC(O)C(C)(C)C(=O)NC1CC(CCNC(=O)C(C)(C)c2ccccn2)C1 CC1CN(C(=O)C=Cc2cnccn2)CC(CCNC(c2cc(Cl)c[nH]2)=O)O1 Cc1cc([N+](=O)[O-])cc(C(N2CC(NC(=O)CSc3cccs3)CC2(C)C)=O)n1 C1(c2ccccc2)(N(C(=O)CC2CC=CC2)C)CN(C(=O)C=C2CCSCC2)C1 C1(C(=O)Nc2c(O)ncnc2O)C2CC(F)C(C2)N1C(c1ccco1)=O c1(C(=O)NC2C(c3cn(C(C)C)nc3)C2)c(N(C)C)cccc1C(F)F c1(NC(N(C(c2ccccc2Cl)CC)C)=O)cc(-c2ccccc2)nn1C(C)C c1(C(=O)NC(C)C(C)NC(=O)Cc2ccn(C)n2)c(F)cc(F)cc1Cl C(N=c1nc(N2Cc3c[nH]nc3C(C)C2)c2c([nH]1)CSC2)c1c(CC)cncc1 c1(CC(N2CC(CN(C(C(C)CN(C)C)=O)C)C2)=O)cccc(C(F)F)c1 CC1(CCNC(c2cccn2C2CCCC2)=O)CCN(C(c2ccsc2)=O)C1 n1(CC(=O)NC2(C)CCN(C(C3C(C)CCC3)=O)C2)ccc2cc(F)ccc12 c1(C(N(CCCN(C)C(C2(C)CCCCO2)=O)C)=O)cccc2nsnc12 N1(C(c2cc(F)c(C)c(F)c2)=O)CCc2c(cccc2[N+](=O)[O-])C1 C1(NC(C(=O)N(C(c2ccc(F)c(Cl)c2)C)C)=O)CCNC2(CCCCC2)C1 C1(C(F)(F)F)(NC(=O)CC2CCC2NC(=O)C(F)F)CCOCC1 c1(NC(C2C(NC(C3CC(C)(C)C3)=O)C2)=O)ccc(F)cc1 C1(C(=O)O)CN(C(c2cc(Br)ncc2F)=O)CC12CN(Cc1ncco1)C2 N1(CC(=O)NC2(CCO)CN(C(c3ncn(C)n3)=O)C2)CC(=O)NC1=O N1(C(C=C(CCC)C)=O)CC(NC(C2CCC(C)O2)=O)CC1CO C(=O)(C1CCCc2cccnc21)N1CCN(C(CC2(C)CCC2)=O)CC1CCO O=C(C=NN1CCCCC1)N1CC2CC(C1)O2 CC1=C(C(=O)NCC2CCN(C(c3cn(C)nc3C(C)C)=O)CC2O)CCO1 c1(NC(C(N2C(CNC(C(C)=O)=O)CCC2)=O)=O)cccc2ccccc12 C(CS(=O)(=O)c1ccc(C(=O)NC2CCCC2N(c2ccccc2)C)cc1)OC CCC(C)(C(=O)N1CC2CN(C(c3c(Cl)n[nH]c3C)=O)CC2C1)C(F)F c1(OC)ccc2c(c1)OCCC2NC(=O)CC(=O)Nc1nccs1 CC1OCCCC1C(=O)NCCN(C(=O)C(C1CC1)NC(=O)OC(C)(C)C)C C(C(C)(C)CNC(C1(n2cccn2)CCCC1)=O)N(C(=O)C(O)C1CCC1)CC CCC(CNC(=O)CC1CC2(C1)CN(C(C1CC1C(=O)OC)=O)C2)C(C)(F)F CC(C)CCC(=O)C(=O)NC(CCN(C)C)C(=O)NC(C)(C)CCCF C12(NC(C3CC(OCC)C3)=O)CCCC1CN(C(c1cccc(F)c1Cl)=O)C2 C1(C(=O)NCC(C(CC)C)C)CN(C(C2(C)C=CCCC2)=O)CC(C)(C)C1 c1(OC)cc(OC)cc(C(=O)NC2CN(C(=O)CCc3nc(=N)[nH][nH]3)CC2C)c1 C(CC1CCc2ccccc21)NC(=NCC)NCc1nc(O)c2c(n1)CCOC2 Cc1ccnc(C(C)(C)C(=O)NCCCN(C(=O)CC(=O)NCC(F)(F)F)C)c1 C1(CC#C)CN(C(C2(C)CCN(C(=O)CN3CCCC3C)C2)=O)CCO1 C12(C(=O)NC3CN(C(c4cn(C5CCC5)nn4)=O)C(F)C3)CCC(CO)(CC1)C2 N1(C(C=C)=O)CCC(C(=O)NCC2CC(F)(F)C2)C(O)C1 N1(C(c2cn(CC)nc2)=O)CCCCC2(CCN(C(=O)C(=O)N(C)C)C2)C1 CC1(C(=O)NC(CNC(c2csc(COC3CCC3)n2)=O)C2CC2)CCCC1 Cc1occc1C(N(C(c1csc(C2CCC2)n1)C(=O)NC(C)(C)C)C(C)C)=O c1(-c2cc(C(N(C3CC(C(N)=O)C3)C)=O)n[nH]2)ccccc1F C1(CNC(c2cnc(C)s2)=O)CN(C)CCN1C(C1CC2(CC2)CO1)=O C=CCCC(C(=O)NCc1ccccc1CO)NC(=O)C(C)N(CC)CC C12(NC(c3c(C(C)C)cnn3C)=O)CCCC(CN(C(c3n[nH]cc3Cl)=O)C1)C2 N1(C(C(C)(C)OC(C)=O)=O)CCCC(F)(CNC(=O)C=CC2CCCC2)C1 Cc1cnnc(O)c1C(N1CCC(C)(CNC(=O)CC2(C)CCOCC2)C1)=O CCCC(CC)C(=O)NCC(O)CCNC(c1cnc(CC(C)(C)C)s1)=O CCC(C)(O)C(=O)NCC(C)C(=O)NCCC12CC(CCO1)C2 N1(C(COCCC=C)=O)CCC(C)C1CNC(c1coc(C)c1)=O N1(C(C23N(C(C(CC)(COC)CC)=O)CC(C2)C3)=O)CCN2C(=O)CCC2C1 C(=O)(C1=NOC2(CCC2)C1)NC(C(C)C)C(=O)NCC(C1CCCC1)C CCC(CC)C(F)C(=O)NC1CCCC1CNC(=O)CCc1ncc[nH]1 C(C)(CCC(=O)NCC(C1CCCCC1)NC(=O)CSC(F)F)SC c1(C(F)(F)F)csc(CNC(C2CCOC2)Cc2nn[nH]n2)n1 Cc1ccc(CC(=O)NC(Cc2ccccc2)CCNC(C2CC2(Cl)Cl)=O)cn1 O=C(C#CCNC(C1CCCO1)=O)NC(C(N)=O)C1CC1 c1(C(=O)NCCCCC(C)NC(C(C(C)C)NC=O)=O)cccc(Br)c1N N1(C(c2nncc(CCC)c2)=O)CCC(CO)(NC(c2cc(CO)[nH]n2)=O)CC1 CON1CC(C(=O)NC2CCCC2C(=O)NCCC(C)(C)N(C)C)CC1=O c1(C(=O)NCC(C)(C2CC2)NC(=O)CCC2CC2(F)F)cc2cccc(F)c2o1 C(C(=O)N(C(C)CNC(c1ncc(OC)cn1)=O)CC)(C(C)C)SCC CC#CC1CCN(C(=O)CC2CN(C(c3csc(C#N)c3)=O)CC2C)CC1 c1(C(=O)NCCCC2(NC(C3CC=CC3)=O)CC2)cnn(CCO)c1 c1(C(N2C(C)(CNC(C3(C)CCCO3)=O)CCC2)=O)cc(O)c2ccsc2c1 CC1(CNC(C23CCCC2CCC3)=O)CCCN(C(c2ncnc(O)c2F)=O)C1 C1(NC(c2c(CNC(COC(C)(C)C)=O)n[nH]c2)=O)CC(=O)NC(=O)N1 C1(C(=O)NCC(C)(C)NC(C2CCC(CC)O2)=O)CC(C)(C)C(C)(C)C1 C12(C(=O)NC3CN(C(C(CO)N(C)C)=O)C(C)CC3)CC3CC(C1)CC(F)(C3)C2 C1(OC)CC(NC(=O)CCC=Cc2ccccc2)CN(C(=O)C(C)CO)C1 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NCC(CCSC)OCC C1(CN(C(C2CC(SC)C2)=O)C)(CNC(C)=O)CC1(F)F C12(NC(CCCC(=C)C)=O)CCCC1N(C(=O)CN1CCCNC1=O)CCC2 C1(CC=C)CCCC1NC(c1coc(COC)n1)=O.c12ccc(o1)CNC(=O)CC2 N1(C(c2c(C)nccn2)=O)CCC2(CCC2)C(NC(C2CCOC2C2CC2)=O)C1 N1(CC(=O)NC(C)C(N2CCCCC2)=O)CCC(CCCCCN2CCC2)CC1 N1(C(c2n(CC#C)cnn2)=O)CCC2CCCC12C(N1C2CSCC1C2)=O Cc1nn(C(C)(C)C)c(C)c1C(=O)OCC1CN(C)CC1C(F)(F)F N1(C(Cc2ccc(SC)o2)=O)CCCN(CCCCNC(C2CCSC2)=O)CC1 N1(c2nc(C)cc(C(=O)OC)n2)CC2CCC1CN2Cc1ccc(C)cc1 CN1CCCC(CN(C)C(C2CCC2CNC(=O)Cc2cnsc2)=O)C1 CC1(NC(c2cc(O)ncn2)=O)CCCN(C(=O)C=Cc2ccccc2)C1 c1(C(N2CC(C)C(NC(c3coc(Br)n3)=O)C2)=O)cccc2c1NC(=O)CC2 CC1(C)CCC(CC(=O)NCCn2cc(CNC(=O)C(O)CC3CC3)nn2)CC1 c1(C(N2CCC(CC=C)(NC(=O)C=CCF)CC2)=O)cc(Cl)cc(F)c1F N1(C(c2n(C(C)C)ccn2)=O)CCC2(CCCCC2NC(=O)C(C)CF)C1 CCC(C(=O)N1CC2CC1CN(C(C1(SC)CCC1)=O)C2)C(C)(F)F c1(C(=O)NCCN(CCCN(C)C)C(c2cc(Cl)c[nH]2)=O)ccc(CO)cc1 C(=O)(C(C)C(C)C(C)(C)C)NCCN(C(=O)C(C)(C)OC)CC S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(C(N)=O)s1)NCC(CC)N1CCCC1 CC(C)C(C(=O)N1CCC2CN(C(c3ccnn3CCF)=O)CC12)C(C)C C1(C)(CC)C=C(C(=O)NCCCCC(CO)NC(=O)CCc2c(C)noc2C)C1 N1(CCc2cn(CC)nc2)CCOC(C)(CNC(C2(C)CCNC2=O)=O)C1 c1(C(=O)NC(C)CCCNC(C2CCC(F)C2)=O)cnc2nccn2c1 C1(C(=O)NCCN(C)C(C23CCCC2(C(N)=O)C3)=O)CCC(C)(O)CC1 c1(NC(COCc2onc(C)n2)=O)ccc2c(c1Br)OC(F)(F)O2 n1(C2C(C(=O)NC(C(=O)OC)C)C2)cc(C2(O)CC2)nn1 CP(C)(=O)c1ccnc(-c2noc(-c3ocnc3CS(C)(=O)=O)n2)c1 N1(C(C2(C#C)CCCC2)=O)CCN(C(=O)C2=NNC(=O)CC2)CC(C)C1 C(=O)(N=c1[nH]oc2ccc(Cl)cc12)NC1CN(C)C(=O)CC1 C(CN=c1cc(C)c(S(=O)(=O)N(CC(N2CCCC2)C)C)c[nH]1)C1C(C)C1 C#CC1(C(=O)NCC2CC(CSC)C2)CCN(C(=O)CNC(=O)CC)C1 c1(C(=O)NCC23CC(C2)C(NC(c2cscc2Cl)=O)CO3)cc(O)nc(O)n1 C(=O)(C(O)CC(N)=O)NC(CNC(C=C(CCC)CCC)=O)(C)Cn1cccn1 CCC(CC)C(F)C(=O)N1CC(O)(C(F)C(=O)NCC2CCC(OC)C2)C1 O=C(CS(=O)(=O)Cc1cccs1)NCC12CC1CN(C(C1C3(CC3)C13CC3)=O)C2 C1(CN(C(CSCC#C)=O)C)CN(C(C2CC2c2ccccc2Cl)=O)CCO1 N1(C(C2N(C)CC2)=O)CCC(O)(CNC(=O)CC2CSC2)CC1 c1(C(=O)OCC2CC(NCC)C2)cc(F)ccc1CC C1(C#N)(C(=O)NCC(C(C)(C)C)NC(CC2C(C)(C)C2(C)C)=O)CCSCC1 C1(CNC(CN2CCC(C)C2)=O)COCCN(C(c2cc[nH]n2)=O)C1 Cc1ccc(-c2cc(C(=O)NCCC(C)NC(c3occc3C)=O)no2)c(C)c1 c1(C(=O)NC2C(C(=O)Nc3c(C(=O)OC)n[nH]c3)C2)cc(C)c2cc[nH]c2c1 n1(CC2C(NCC3CC3)CN(C(C3CCC(OC)CC3)=O)C2)c(C(F)F)cnc1O C(C1CN(C(=O)CC2C=CCC2)Cc2ccccc21)NC(c1scc(OC)c1)=O CC1CCOC1C(=O)NCC1(CNC(c2cc(C3CC3)ns2)=O)CC1 C1(CC)CN(C(=O)Cc2ccnn2C)CC1C(=O)NCC(C)(C)C1CCC1 C1(N(C(=O)CCn2cccnc2=O)CC)CCCN(C(=O)CC(C)(C)C#N)CC1 C1(F)(CNC(c2c(C)nc(C(C)C)o2)=O)CCCN(C(c2ccc(Cl)cc2)=O)C1 C1(CC)COC(C)(C)CN1C(C1CC2CCC(C1)N2C(=O)CC(C)(C)C)=O c1(C(N2CC(CN)C(n3ccnn3)C2)=O)cccc(C(F)(F)F)c1F C=CCCCCCC(=O)NCCN(C)C(C1(COC)CC(=C)C1)=O c1(C(N(CC(C)(C)NC(c2cc(CC)sn2)=O)C)=O)cncc(OC)n1 c1(COC)cc[nH]c1C(N1CC(C(C)NC(c2c[nH]nc2C2CCOC2)=O)C1)=O C1(C(N2CCC(CC(=O)NCCC(=O)OC)C2)=O)CC12CCOC2 C(=O)(C1CC(NCC(=O)NCc2ccc(OC)cc2)c2ccccc21)OC C1(CC(=O)NCCCCNC(CCOCC(C)C)=O)CCC(O)C1 N(C(=NCCc1ncccc1C)NCC1C=CCC1)C(C=C)C CCC(C(=O)NCC1(C)CN(C(c2ccnn2CCF)=O)CC1C)C(C)(F)F c1(C(=O)NCCN(C(C(CC)=CC)=O)CC(C)O)ccc2cccnc2c1O c1(CC)ncccc1NC(c1nnc(-c2ccccc2)n1-c1ccccc1Cl)=O c1(OC(C)C(=O)NCCN2CCN(C(=O)C(C)(Cl)Cl)CC2)ccc(F)cc1F N1(C(C(CCC)NC(C2(c3ccno3)CC2)=O)=O)CCC(F)(CF)CC1 c1(CC)cccc2c1OC(C(=O)OC(c1ccc(OCCOC(C)C)cc1)=O)C2 C1(CNC(C=C(COC)C)=O)(OC)CCN(C(C2(Cl)CC23CCC3)=O)C1 Cc1oc(Cl)nc1C(=O)NC1(NCC(C)(C)N(C(=O)Cc2cc[nH]n2)C)CC1 Cc1cccc2nc(CNC(C3CCCN(CCCC4CCCO4)CC3)=O)cn12 N1(C(C)=O)CCCCC(F)(F)C1.N12CCCC(C1)C(C)CC2=O CCCCC(CCCC)C(=O)N1CCC(N(C(=O)C=CS(C)=O)C)C1 C1(NC(CSC)=O)CN(C(C2(NC(C)=O)CCOC2)=O)CC2(CCC2)C1 C1(C(N2CCC(=CCNC(COC3(C)CCC3)=O)CC2)=O)CCCC1P(C)(C)=O C(=O)(C1=NNC(=O)CC1)N1CCC(C)C(NC(C2(c3ccno3)CCC2)=O)C1 N1(C(CCc2n(C)ccn2)=O)Cc2[nH]nc(C(N3CCOC4CC34)=O)c2C1 C(=O)(CC(CN(C)C)CC)NCC(CC(=O)NCc1c(CC)con1)O CON(CCC(=O)N(C1CS(=O)(=O)C1(C)C)C)C(=O)CC1CC(=O)NC1=O C(=O)(C1=CC(O)CCC1)NCCOCCNC(c1ccc(CC)c(N)c1)=O N1(C(C2C(C)OCC2)=O)CCCCC(CNC(=O)COc2cccnc2Cl)C1 C(c1c(F)cccc1F)=CC(=O)NC1CC(NC(=O)CC2(O)CC2)C12CCC2 C(=O)(C1SCc2cccnc21)NC12C(CN(C(C(C)=CC)=O)C1)COCC2 Nc1ccc(Br)c(C(=O)NCC2CCC(NC(=O)CC3(CO)CC3)C2)c1 C1(c2ccccc2)CCN(CCCc2nc[nH]n2)CCO1 C1(N(C)C(C2(S(C)(=O)=O)CC2)=O)CN(C(=O)C(c2cccn2C)=O)CC1(C)C C(=O)(C#CC(C)(C)O)N(C1CCN(C(C(C=CC)O)=O)C1)C c1(C(C2CN(C(C3C(C(=O)OC)C3)=O)C2)CNC(c2cc[nH]c2)=O)ccccc1 c1(C(=O)Nc2cccc(CNC(C=CS(C)=O)=O)c2)ccc2n[nH]cc2c1F CC1CN(C(=O)CCC2(N3CCCC3)CCCC2)CCO1 C(=O)(C(O)CC(C)(C)C)N(CC(C)NC(c1cnccc1C#N)=O)C N1(C(C2(CF)CCC2)=O)CC(NCc2ccc(Cl)cn2)CC(F)C1 c1(C(=O)NCCC2CCCCN2C(=O)CCc2nccs2)ccc(F)c(C2CC2)c1 c1(N2C(C)CC(NC(c3ccc(CN(C)C)o3)=O)CC2)ncn(C)c(=O)c1Br CC1CC(NC(C2(NC(C3CC(F)(F)C3)=O)CSC2)=O)CCS1 C(=O)(C(F)C(C)(C)O)NC1CC2(C(NC(c3ccc(C(CC)=O)cc3)=O)C2)C1 C(=O)(CCC(C)(C)OC)NCCC(C(C)C)NC(CCC(=O)NCC)=O N1(C(CC2(OC)CN(C(=O)CC3CCCSC3)C2)=O)CCC(=C(F)F)CC1 CC1(CO)CN(C(C2CC(O)CN2Cc2ncc3cn[nH]c3n2)=O)CCC1O Cc1ccc(C(=O)NCC2CCCCN(C(c3c(C)noc3C)=O)C2)c(Cl)c1C CC(C)C(C)(O)C(=O)NC1CCN(C(c2ccc(Br)nc2N)=O)C1C C1(CNC(C(COCC)(C)C)=O)CCN(C(c2nccnc2SC)=O)CC1O C1(C(=O)NCCOCCCNC(c2cncc(OC)n2)=O)CCC(=C(F)F)CC1 c1(C(c2cc(Br)cc(Br)c2)=O)ccc2c(-c3cn[nH]c3)cccc2n1 Cc1cc2c(C(=O)NC3CC(NC(c4cc[nH]c4C4CC4)=O)C3)nccn2n1 c1(OC)ncc(C(=O)NC(C)C(C(C)C)NC(=O)Cc2ccoc2)c(C)n1 N1(C(CCn2cc(CCOC(C)=O)nn2)=O)CCC(O)(CSc2ccco2)C1 N12CCC(F)(F)C(C1)C(=O)Nc1cc2ncn1.N1(OC)CCCC(C)C1C C(=O)(C1=C(N)CCC1)N(CCCOc1cccc(C)c1)C c1(OC(C2C(C)(C(=O)OCc3ccc(F)cc3)C2)=O)ccc(F)c(C#N)c1 C1(NC(c2cc(SC)oc2)=O)CN(C(=O)CC2CCCC23CC3)CC1(C)C Cc1nc(C(F)(F)F)oc1C(N1CCCC1CN(C)C(C1CCCOC1)=O)=O CCC(C(=O)N(CCCCNC(C1CCC(=O)N1CC)=O)C)C(C)(F)F c1(C(=O)NC2CN(C(C=C(C)Cl)=O)CC2C2CC2)cn2cccc(C)c2n1 c1(C(N2C(CNC(C(CCC)OCC)=O)CC3CC32)=O)ccnc2c1ncn2C N#Cc1cccc(NC(C2C3CN(C(c4cc(F)c(Cl)cc4Cl)=O)CC23)=O)c1Cl C(CN(C)C)(C(=O)NCC1(O)CCCC1)NC(C(C)OCC#C)=O C1(CNC(C(c2cn(C)nc2)O)=O)CC2(CCC2)CN1C(=O)CC1CC(C)(C)C1 C=CC(C)(CCOC)C(=O)N1CCC(F)(CNC(=O)CC(C)C(F)F)CC1 Cc1nn(C)c2sc(C(N3CCC(NC(C4(C5CC5)CC4)=O)CC(O)C3)=O)cc12 N1(C(c2c(CC)ocn2)=O)CC2CC(C(N3CCC3C3CCCC3)=O)(C2)C1 C(c1cccc(Cl)c1)=C(C)C(=O)N(CCCCNC(C1(C#N)CCCOC1)=O)C c1(C(N2CC(C(C)NC(C3CC(=C)C3)=O)OCC2)=O)ccc2c(Cl)nccc2c1 C1(C(=O)NC2CC(C)(NC(c3c(N)cn(C)n3)=O)C2)CC(=O)NC1(C)C Cc1cn2nnc(C(N3CCN(C(=O)CCc4cncs4)C(C)C3)=O)c2c(O)n1 c1(C(=O)NCCCN(C(=O)CCC2CCCN2C)CCC)ccc(C)nc1OC N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(NC(c2cncs2)=O)CC(F)C1 c1(NC)ccc(C(N2CCN(C(=O)C#CC(=O)N(C)C)CC2C(F)F)=O)c(Cl)c1 c1(NC(C2C(C)C2)=O)ccccc1C(=O)NC1CCS(=O)(=O)C1 N1(C(c2ccc(C(C)=O)o2)=O)CCC(CCNC(=O)CCSC2CCCC2)CC1 CCC(CO)CN=C(NCCC(=O)NC1CCCCO1)NCc1cccc(F)n1 c1(C(C(=O)OCC2C(C(=O)O)C2)(F)F)ncccc1F C=CCC(C(=O)NCC1(F)CC(NC(=O)C(c2ccccc2)=O)C1)NC(C)=O C=CCC(C)(C)C(=O)NCC1CCCCN(C(=O)C(C)CC(N)=O)C1 n1(CC)cnc2[nH]c(=NCC3CC3(C)C)nc(N3CCC(CC(C)C)(CO)C3)c12 C1(OC)CC(OC)CN(C(C2CCC(Cl)C2)=O)C1 N1(C(c2cc(C)nc(C)c2)=O)CC(NC(c2[nH]cc3c2CCC3)=O)CCC(O)C1 C1(C)(CNC(C(CN(C(CC2CC(=C)C2)=O)C)C)=O)CCCC(=O)N1 c1(CC)nocc1CN(C(=O)C(C1CCOC1)NC(=O)CC(=O)N(C)C)C N1(C(c2cc(OC)c(C)cc2)=O)CC2CCCC(NC(C3CCSCC3)=O)C2C1 C1(=O)CCOCCCN1.C1(C(=O)OC)CC1C(=O)NC1CCC1.C(C)=O c1(C(N2CC=CC(NC(C3C(C)(C)CC3)=O)C2)=O)ccc(C#N)c(O)c1 c1(C(=O)NC(C2CCCN(C(c3scnc3Cl)=O)C2)C)cc([N+](=O)[O-])nn1C c1(N2CC(NC(c3cc(C(F)F)on3)=O)(CO)C2)ncnc2ccc(O)cc12 c1(C(CC(N)=O)NCc2cnc(C3CC3)o2)ccc(Cl)cc1 N1(C(C(CC)O)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C)(C)c1ccno1)C2 C12(C(=O)NCc3nc(C)c(C)s3)CCN(C(=O)C=CC(=O)N(C)C)CC1C2 c1(C(N2CCOCC2CC)C(=O)NCC=C)ccc(C)c(C)c1 c1(C(=O)NC2CCN(C(c3nc(C)oc3C)=O)CC2)cnc2ccccn12 N1(C(C(C)OCCCC)=O)CC2(C)CN(C(c3cc(CCC)on3)=O)CC2(C)C1 c1(C(=O)NCC(CC)(C)NC(=O)C(C(C)C)C(C)C)ccn2cc(C)nc2c1 c1(C(N(C2(CC(=O)NCC3(CC=C)CC3)CC2)C)=O)cnc(N)cn1 N1(C(CC(=C)C)=O)CCOC(C)(CNC(c2cc(Cl)c(Cl)n2C)=O)C1 Cc1ccc2c(C(=O)NC3CCC3CNC(c3cc(C)c(C)o3)=O)c[nH]c2c1 Cc1[nH]nc2sc(C(=O)NCC3CCCN3C(=O)COCC(C)(C)C)cc12 C1(O)(CC#C)CC(C(=O)NCC(C(C)C)NC(C2(N3CCCC3)CCC2)=O)C1 C1(CC)CN(C(=O)CC2CCCC(=O)C2)CC1CNC(=O)CNC(=O)CC(C)C c1(C(N2CCCC(C(C)C)C2)C(=O)NC2CCC2)ccc(C2CC2)cc1F c1(C(N2CC(CC(C)NC(C3CCOC3C3CC3)=O)C2)=O)c[nH]c(=N)nc1C(F)F N1CC(C2CN(C(=O)C=Cc3ccc(OC)cc3)C2)C1.C=CCCC1(NCC)CC1 C(C)(C(=O)N(CC(=O)NCCC12CC(C1)C2)C1CC1)SCCCC Cc1cc(C(=O)C(N2CC(F)(F)CC2CNC(c2n[nH]c(O)n2)=O)=O)ccc1F C1(NC(Cc2cc(C)sc2)=O)C2CC(O)C1N(C(=O)CCCNC(N)=O)C2 c1(C(N(C)CCN2CCN(C(C3CC4CCC34)=O)CC2)=O)ccn2cnnc2c1 C(C(=O)NCCC(=O)O)(C(C)(C)C)n1cc(-c2cccc(C(=O)OC)n2)nn1 C=CC1OCCCC1C(N1CC(COC)CC1CNC(=O)C1=COCC1)=O c1(CC(=O)NC(CNC(=O)CC23CCC(CC2)CC3)CO)ccc([N+](=O)[O-])cc1 N1(C(C(CC(C)C)C)=O)CC=C(C(=O)NC2CCCCCCC2C)CC1 c1(OC)cc2cc(NC(=O)NC(C#N)C(C)O)cnc2cc1OC C1(CC(=O)NCCOC(CNC(C(C)OCC)=O)(C)C)CCOC1(C)C N1(C(COCC(=C)C)=O)CCC(CN(C(=O)C(C)n2cccc2)C)CC1 C1(C(=O)NCCC=C)CCCC1CNC(C1C=C(C)CS1)=O C1(C(NOCC(=O)NCC(c2cccs2)C)=O)CC(O)CN1C c1(C(N2CCC(CNC(CSCC(C)C)=O)C2)=O)c(Cl)nsc1Cl C=C(CNC(=O)C(C1CCN(C(=O)CCOCC2CC2)C1)C)c1ccccc1 c1(OC)ccc(F)c(C(N2CCC(N(C)C(c3ccc(F)c(C)c3)=O)C2)=O)c1F c1(CCN2CC=CC2)ccncc1.C1CCOC1C(=O)NC(=O)CSC c1(CC(N2CC(CNC(C(CC)C)=O)C(C)CC2)=O)nc2ncccn2n1 c1(CN2CC3N(C(c4cnc(Br)s4)=O)C3C2)cccc(Cl)c1Cl C1(C(N2CCC(O)(CCO)CC2)=O)CC(F)(F)CN1C(C1CC(F)(F)C1)=O c1(C2c3nnnn3CCCN2)ccc(C#N)nc1.n1(CC#C)ccnc1COC C(=O)(C1=CCCCO1)N(CC(C)O)CCNC(=O)C(C)(C)C1(C)CC1(F)F C(C(O)CC(=O)N1C(c2cncc(Cl)c2)CCC1C)c1n(C)ncc1 C1(F)(CNC(C2CC(=C)C2)=O)CN(C(c2cc(-c3cnn(C)c3)[nH]n2)=O)C1 CCCCCCC(C)C(=O)NC(CCC(C)C)C(=O)NCC(C)(C)C(C)(F)F Cc1noc(C(N2CC(N(C)C(C3COCC3(C)C)=O)C2)=O)c1C(F)(F)F c1(C(=O)NCCOCCCNC(CCc2cc(C)[nH]n2)=O)n[nH]c2c1NCCC2 CC1(C)CN(C(c2cccc(CO)n2)=O)CC1NC(=O)Cc1ccccn1 C1(C2(O)CCN(C(c3cn4c(n3)C(C)CCC4)=O)CC2)(NC(C2C(=C)C2)=O)CC1 C1(CCNC=O)C2CN(C(=O)CCF)CC12.C1(C(=O)NC)CC1(C(F)F)C1CC1 CCS(=O)(=O)c1ccccc1C(=O)NCCCCC1CN(C(=O)C(C)CSC)C1 c1(OC)cn(CC(=O)N(C)CCN(C(=O)CCC(=O)N(C)C)C)c(C)cc1=O c1(C(CN2CC3C(CNC(C(C=C=C)C)=O)C3C2)=O)c(F)ccc(Cl)c1F C12(CNC(CCCC)=O)CCCCC1CN(C(c1coc(CC)n1)=O)C2 C1(C(=O)NCC2CCC(NC(C(CSC)O)=O)CC2)CCCC(C)CC1 C1(C(N2C(C=C)CC2)=O)CCN(C(=O)Cc2cnccc2C)O1 CC1(C(N2CC(NC(C3CCN(CC(F)(F)F)CC3)=O)C(O)C2)=O)CC(F)(F)C1 c1(C(=O)NCC2(F)CC(NC(C(C(C)O)NC(C)=O)=O)C2)n[nH]c2c1CCC2 N1(C(C(C(CC)C)C)=O)CCCC2(NC(C3(N(C)C)CC3)=O)CC2C1 C(=O)(C(C(=O)NCCCCCNC(=O)CC1CCC(C)(O)CC1)C(C)C)OCC c1(CCC)nnc(CC(N2CC(C(C)NC(=O)CCSc3nccn3C)C2)=O)o1 C1(NC(Cn2ncc(C)c2)=O)CCN(C(C23CC(C2)C(C)O3)=O)CC1F c1(OC(F)F)ccc(CCCCNC2CCN(C3CC3)CC2)cc1 N1(CCCC)CCCC1C(=O)NCC1CC(NC(=O)C=CCOC(C)(C)C)C1 N1(CC)CCCC1C(=O)NCC(CO)NC(c1cnn(C2CCC2)c1)=O CCCC(CCCO)C(=O)N1CCC(NC(=O)C(O)CSC)CC1C C1(NC(CN(C)C(N)=O)=O)CCOC(C(=O)NCC(O)C2CCC2)C1 CC1CC(CNC(c2cn(C(F)F)cn2)=O)CN1C(=O)Cc1cccnc1 c1(N2CCC(C)C(CNC(c3ccc(C(N)=O)[nH]3)=O)C2)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC(CNC(=O)Cc3ccc(F)cc3)C3C2C3)=O)cccc2c1CCO2 c1(OC)cccc(CC(C)NC(c2cnn(C)c2)C2CCCC2)c1O CCCC(C)(CC)C(=O)NCC1CCCN1C(=O)CC1(CSC)CC1 C1(O)(CNC(c2ncc(-c3ccc(F)cc3)o2)C)CC2CC1C2 CCC(C)C(O)C(=O)N1C(C(=O)NCc2cc(O)ccc2F)CC2CC12 CC1(C)CC(NC(c2cncc(-n3cccc3)c2)=O)CN(C(c2cncs2)=O)C1 C(CN=C(NCC1CCCN1C)N(C)CC1(O)CCCOC1)N(CC)CC c1(C(=O)NC2CN(C(Cc3ccc(OC)cc3)=O)C3C2C3)cncc([N+](=O)[O-])c1 n1(CCC(=O)NC(C)CNC(C2CC2(F)F)=O)ncc2ccccc12 N1(C(c2c(C)c[nH]c2CC(N)=O)=O)CC2CC1CN2C(c1cnc[nH]c1=N)=O C12CC3CC(C(C1)C3)CN2.c1(C(=O)OCC)ccnc(C(=O)NC(C)(C)C)c1 Cc1nc2ncnn2c(N2CCC3(CC2)OC(=O)NC3=O)c1C C#CCCCCCC(=O)N1CCN(C(=O)C=Cc2cc(Cl)ccc2Cl)CC1C C1(CNC(CCOc2cccc(C)c2)=O)CCCN(C(=O)CC(C)C2CC2)CC1 c1(SC)ccc(O)c(C(N2CCC(N(C(=O)C(C)P(C)(C)=O)CC3CC3)C2)=O)c1 N1(C(c2c(CC(=O)OC)ccnc2)=O)CCC(C)CC(C)C1.N12CCC(O)(C1)C2 C1(CC)CN(C(=O)C(C)(C)SC)CCN1C(C1CC1c1ccc(OC)cc1)=O n1(CC(=O)NC2CCC(N(C(C3C(C)C3)=O)C)CC2)ccc(O)nc1=O N1(C(C(CC)=CC)=O)CCN(C(=O)C(C)(C)c2csc(C)c2)CC1C(C)C c1(C(N2C(COC)CN(C(C3(O)COC3)=O)CC2)=O)n[nH]c2c1CN(C)CC2 c1(C(=O)NCC(=O)NCC2(O)CN(C(C3C(COC)C3)=O)C2)c(F)cccc1F C1(C(=O)Nc2c(C)cc(NC(=O)CCn3ccnn3)cc2)CN(C)C(=O)CCO1 C#Cc1cnn(CC(=O)NC2(CCCC(=O)NCC(C)(C)N3CCCC3)CCC2)c1 c1(CC(C)C(=O)NCC2CC(NC(c3cc(Cl)c[nH]3)=O)C2)ccc(Cl)cc1 CC(=Cn1ccnn1)C(=O)NC1CCC2CN(C(c3csc(O)n3)=O)CC2C1 C1(CNC(C2(CC=C)CCC2)=O)CC2(CC2)CN1C(=O)Cc1ccc(Cl)cn1 C1(NC(c2c(C)ccs2)=O)CCC(C)(C)CC1CNC(=O)CCc1ccon1 C1(C(N2CCC(C)(O)C2)C(=O)NCCC)CCCCC1CC(F)(F)F C(C)(C)(C(=O)NCc1cc(C(N2CC(CC3CC3)C2)=O)n[nH]1)OC(C)=O C(CC(N)CC(C)(C)C)N.C(CCC)CCC c1(OCC)n[nH]c(=NC(=O)c2ncc(CO)nc2C(F)(F)F)cc1CO C=CC(C)(CC)C(=O)N1CC(NC(=O)C(F)(F)C2CCOCC2)C(SC)C1 Cc1ccn2cc(C(N3CCC(NC(c4ccnn4C)=O)C(F)C3)=O)nc2c1C c1(C(N(C2CCCN(C(C3ON=C(CC)C3)=O)CC2)C)=O)c([N+](=O)[O-])cnn1C C=CC1(NC(=O)C(C)(C2CCC2)NC(c2ccon2)=O)CCCC1 C1(NC(=O)CCc2cnc[nH]2)CC2CCC1N2C(C1CCC2(CCC2)C1)=O c1(C(N2CCCC(N(C(=O)CC(=O)NC3CC3)C)C2)=O)cc([N+](=O)[O-])sn1 C1(CC(=O)N(C)CC2CCN(C(c3ccc(C)o3)=O)C2)(CN(C)C)CCCCC1 CC1CN(C(C2CC2C2CN(C(=O)CC3CCCC(=O)C3)C2)=O)C12CCOCC2 n1(CCCOC)nnnc1C(C)(CSC)NC1CCCC1NC(C)=O C1(CC=C)(C(=O)NC)CCCCN1CC1C(C(=O)OC)C1(C)C N1(C(C=CSC)=O)CC(CNC(=O)C(=Cc2cccs2)C)C(C(F)(F)F)C1 C1(CNC(c2c(CC)nccc2)=O)CCN(C(=O)CCOC(C)C)CC1C C1(C(=O)NCC(C)CNC(C2CC(=C3CCC3)C2)=O)OCC1(C)C C1(NC(c2c(C)onc2C2CC2)=O)CCN(c2ccc(C#N)cn2)CCC1CO c1(C(N(CCNC(C2CC(C(=O)OC)C2)=O)C(C)C)=O)nc(C)ccc1F N1(C(C(C=CC)O)=O)CC(F)CC1C(=O)NCCc1nnc(C)s1 N1(C(C(C2CC2)OC)=O)CC2(CCC2)CC1C(N1CC(C)(OC(C)C)C1)=O C1(F)(CNC(c2n(C)cnc2)=O)CC2CCC(C1)N2C(C1CC2(C1)CC21CC1)=O CC1(C)CC(NC(=O)CC2NC(=O)NC2=O)CN(C(=O)C2=CCC2)C1 C(=O)(C(CC(C)C)C(C)C)NCC1OCCN(C(C2(CSC)CC2)=O)C1 C(=O)(C1=CCC(C)CC1)N1C(C(=O)NCCC2(COC)CCC2)CC(C)C1 C(=O)(NNc1cc(Br)ncn1)c1ccc(C)cn1 C1(C(N2CCN(C(CCCC(=C)C)=O)CC2COC)=O)CC2(CCCCC2)C1 Cc1ccnc(C(=O)NCc2ncoc2CCNC(=O)CC(C)C)n1 S(=O)(=O)(c1cc(C(=O)O)n(C)n1)N1CC(OCC)CC12CCC2 CC1CN(C(=O)C(O)Cc2cnc[nH]2)CC1CNc1cc(O)ncn1 C1(NC(c2cc(C)c(OC)c(C)c2)=O)CCN(C(C2CCC(=O)N2)=O)CC1(C)C N1(C(C(C)(C)n2cnnn2)=O)CC2(CCCC2NC(=O)CN2CCNC(=O)C2)C1 C1(CC(=O)NCC2(OC)CN(C(c3n[nH]c(=N)s3)=O)C2)CC(O)C12CCC2 C(=O)(C(F)C(=O)NCC(C(=O)N1CC(OCC(F)F)C1)N(C)C)OCC C(=O)(C1=CCC(C)CC1)N1C(CNC(c2c(C)c(O)ccc2)=O)CC1 C1(CC)CN(C(=O)CC2CCSC2)CCC1NC(C1CC(O)C1)=O C1(C(N2CCC(O)(c3cn(-c4cccc(Br)c4)nn3)CC2)=O)CC12CCCCC2 c1(C(=O)NCC2N(C(c3cnc(CC)[nH]3)=O)CC2)cnn2ccc(Cl)c(F)c12 CC(=O)n1cc(CNC2CCCC2C(=O)NCC(C)(F)F)c2cccnc12 C(=O)(C(CC(N)=O)NC(=O)C(C)OCC(C)C)NC1(CCC)CCC1 C(=O)(C(C)(C)CC(F)(F)F)NCC1(CNC(C=C(C)C)=O)CCC1 c1(CC)nn[nH]c1C(=O)NC(C1CCCN1C(=O)C(C)SC)(C)C CC1CCN(C(C2(N3CCCCC3)CC2)=O)C1c1cn(CC(F)(F)F)nn1 N1(C(c2ccc(-c3cccc(O)c3)s2)=O)CCCC2CN(CC3(O)CC3)CCC12 CC1=C(C)CC(C(=O)NC2(CNC(c3c(Cl)c(C)nn3C)=O)CCCC2)CC1 c1(C(=O)OCCOCCN(C)C)csc(C(=O)Nc2ccc(Br)o2)n1 C1(C)(CC(=O)N(CCC(C)NC(=O)CCCN(C)C)CCO)CC1(F)F C(C)(C(CC(=O)NCCC1CC1)NC(=O)C(=O)NCC(C)O)OC c1(NC)cnccc1C(=O)NCCO.N12CCCC(C1)c1cn(nn1)CC2 C1(C(N2CCC=C(C)C2)=O)CC2(CC2)CN1C(c1ccoc1)=O N1(C(C=CC)=O)CCC(O)CC1C(N1CC(OC(C)C)C1)=O C=CCCC(CC(C)C)C(=O)N1CC(CN(C)C(c2cocn2)=O)C2(CC2)C1 N1(C(C(CC=C)C)=O)CCC(C)(C)C1CC(=O)NC(c1ncc[nH]1)CC C(C)(N=c1[nH]c2c(c(=NCCC3=CCOCC3)[nH]1)COCC2)C1(S(CC)(=O)=O)CC1 N1(C(C=CC)=O)CCC2(NC(=O)CCCOc3ccc(F)c(F)c3)CC2C1 C12(C(=O)NC(C)C(CO)NC(C3CC4CC4C3)=O)CC3CC(F)(C1)CC(F)(C3)C2 C1(CC(N2C(C(C)C)COCC2)=O)CN(C(=O)Cc2cnoc2)C(C)(C)C1 CC(C)CC(O)CC(=O)N1CC(CC(=O)N(C2CCC(CO)CC2)C)C(C)C1 N1(C(c2ncn(C(C)C)c2)=O)CC2CC2(NC(=O)C(O)Cn2cncn2)C1 C1(NC(c2nccc3[nH]ccc23)=O)COC2(C1)CN(C(C1CCCS1(=O)=O)=O)C2 c1(CC(=O)NC(C)C(CO)NC(C2(C(F)(F)F)CC2)=O)cccc2c1CCC2 N1(C(C(C)NC(=O)OC)=O)CC(N(C)C(c2cc(C(N)=O)co2)=O)C2(CC2)C1 Cc1cc(C(N2CC=C(CNC(=O)CCN3CCCCCC3)CC2)=O)nc(C)n1 N1(CCNC(CC2C(C)CCO2)=O)CCCC(NC(c2ccncc2)=O)C1 CC(CCC(=O)Nc1cccc(SC(C)C(=O)NCc2cccs2)c1)S(C)(=O)=O CCCCC(=O)C(=O)N(C(C)(C(=O)NCCn1ccnn1)C1CC1)C N1(C(C(C)C2CCCOC2)C(=O)NCc2ccco2)CCCOCC12CCCC2 C1(NC(c2ccc(CC)o2)=O)CC2CCC1CN2C(=O)CN(C)C1CC1 C=CCCC(C)(C)C(=O)NCC1(NC(=O)CN(C)S(N)(=O)=O)CCC1 c1(NCC#CC)ncnc(N2CCN(C(c3cc(CCO)on3)=O)CC2)c1C O=C1CCC(C(=O)NCCOC2CCN(C(c3cc(C4CCC4)on3)=O)C2)C1 C(=O)(C(F)C(=O)NC(Cn1cccn1)C(=O)NCC1CCOCC1)OCC N1(C(C(N2C(CC)CCC2)=O)=O)CCCCC(CNC(=O)CCn2ccnn2)C1 N1(C(C)C2CC2)CC(C(=O)NCC=CCSCC(O)CN2CCCC2)CC1=O CC(C(C)(O)Cc1cccc(Br)c1)NC(=O)Nc1cnn(CCO)c1 N1(C(CC(=C)C)C(=O)Nc2coc3c(C)cccc23)CCCC2(CC=CCC2)C1 c1(C(N(CCN(C(Cn2ccc(C)n2)=O)C)C)=O)cc2ncccc2o1 Cc1[nH]nc2c1CC(C(=O)NCC(F)(F)Cn1cc(-c3cc[nH]n3)nn1)CC2 C1(OCC)CCCCC1C(=O)OCCc1nn[nH]n1 C#Cc1ccc(C(=O)NCc2ccc(CF)cc2)o1.C12CC(OC)C(C1)NC2=O CN1CCCC(CC(=O)NCC2CCN(C(C3(c4ccn(C)n4)CC3)=O)CC2)C1 Fc1ccc2nc(CNCCCCc3ccccc3)[nH]c2c1 N1(c2nc(=NCC)s[nH]2)CCC2CCN(CC)CC2C1 N1(C(C(C)CN(C(=O)C=CCO)C)=O)CCOC2COCC2C1 CN1CCN(C(C2CC=CCC2NC(=O)CCN2CCOC2=O)=O)CC1C1CC1 C(=O)(C(O)CC(F)(F)F)NCc1ccc(C(N(C)CC2CC(F)C2)=O)cn1 C1(CNC(C(C)(C)SC)=O)CN(C(c2cnc(NC(C)C)s2)=O)CC1C(F)(F)F c1(SC)ccc(C(=O)NC(C)CCCNC(=O)C(F)(F)CN(C)C)c(Cl)c1 c1(CCC)n[nH]cc1C(=O)N(C1CC(C#N)C1)CC(=O)NC(C)Cc1ccco1 CCC(CC(=O)NCCCCCN(C)C(c1cc(C)n(C2CC2)n1)=O)SC C1(C(=O)NC(CC)CNC(=O)C(C)CF)CCc2ncnc(C)c2C1 c1(NC(c2ncn[nH]2)=O)nc(CCOC2CC2)cc(C)n1.N(CCOC)(CC)C c1(OC)ccc(C(=O)NC2CC(C)(NC(=O)C(C)CS(C)=O)C2)c(F)c1 c1(C(N(CC(C)N)Cc2ccccc2)=O)coc2c(F)c(Cl)ccc12 c1(OCC)cc(C)cc(OC)n1.N12CCCCC1CN2S(=O)(=O)CC.O(C)CC CC(C)C(C)CC(=O)N1CCN(C(c2ccc(N)c(N)c2)=O)C(CCO)C1 CC(F)(F)C(F)C(=O)N1CC(CC(=O)NCC2(C(N)=O)CC2)CC1(C)C CNS(=O)(=O)N1CCC(C(=O)NCCOCCN(C(=O)C(C)N2CCC2)C)CC1 C1(C#N)(C(=O)NCC(C)CNC(c2ccc(CO)s2)=O)CCCOC1 C1(NC(c2sc(C)c(C)c2C)=O)COC2(CCN(C(=O)CN(C)C3CC3)C2)C1 N1(C(c2c(C)cc(C)[nH]2)=O)CC2CCC1CN2C(C1CC1c1cccs1)=O c1(OC)ccc2nc(C(=O)NC34CCC(CC3)N(C(=O)CC(C)CF)C4)cn2n1 C=C(C)c1cccc(NC(=O)C(C2CCOC2)NC(c2cc(CC)nn2C)=O)c1 C12(C(=O)NC(CNC(C(=Cc3ccco3)C)=O)C)CCCCN1CCC2 c1(C(N2C(C)CCC(NC(C3(C(CC)=O)CC3)=O)C2)=O)scc2c1OCCO2 N1(C2CN(C(=O)COC(F)(F)F)C2)CCCN(C(c2cc(Cl)ns2)=O)CC1 C1(CC(=O)NCCCOCCCCCNC(=O)NC(C)(C)C)CC2(CCC2)C1 c1(NC(CC2ON=C(CC)C2)=O)ccc(NC(C2CNC(=O)N2)=O)c(C)c1 N1(CC(=O)NC2CCOCC2NC(=O)Cc2cscn2)CCCNS1(=O)=O N1(C(COC(C)=O)=O)CC2(CC2)CC1C(=O)Nc1sc(C)nc1C C(=O)(CC1=CCCC1)NCC(CC(=O)NCc1cc(C)n(C)n1)OC c1(CC)ncnc(N(CC(C)NC(=O)C=Cc2ccc(OC)cc2)C)c1F C1(CNC(C(C(C)C)SCC)=O)C2CCC(C2)N1C(=O)COc1cccc(C)c1 N(C(=NCCCC(C)(C)O)N(C)CCCN1CCCC1=O)CC(c1cccs1)C CCCCCCC(CC)C(=O)N1CCCCC(CNC(=O)CC2CC3CC3C2)C1 C1(C(=O)NCC2(C(N3CCC3CC3CCC3)=O)CC2)CC2(CCC2)CO1 C1(C(=O)NC(CCCC)C)CC2(CC(NC(=O)C(N)=O)C2)C1 NC1(CNC(=O)C(=O)NCC2(O)CCOCC2)CCN(Cc2ccccc2)CC1 Cc1nn(CC(=O)NCCOCCN(C(=O)CC2(C)CC2)C)c(C)c1[N+](=O)[O-] C1(O)(CNC(C2CC(OC)C2)=O)CCN(C(=O)Cc2cccnc2Br)C1 C(C)(C)(CCC(=O)N1CCOCC(NC(=O)Cn2cccn2)C1)OC CCCC(C(=O)N1CC2CC2C1C(=O)NC(C)Cc1cn[nH]c1)C(C)C N1(C(C2C(C(=O)OC)CC2)=O)CC(C(=O)N(C2(CO)CC2)C)C(C2CC2)C1 c1(N2CC3CN(C(c4cc5ccoc5cn4)=O)C3C2)ncc([N+](=O)[O-])cn1 C(C(C)C(F)C(=O)NCCOCC1CCCC1)NC(CCCC(C)C)=O C12COCC1C(=O)N2.c1(C2(NC(C(C)=C3CCCC3)=O)CC2)cc(C)[nH]n1 C1(O)(CC(=O)NC2(CC=C)CN(C(=O)Cc3cnn(CC)c3)C2)CCCOC1 C1(C(=O)NCCCOCCCNC(CC(=O)NCC)=O)CC(=O)NC(=O)C1 CC(C)(C)C1=NOC(C(N2CC3COCCC3(NC(=O)COCC3CC3)C2)=O)C1 c1(CNCC(=O)NC(=O)NCCC)ccc2c(c1)CCCN2C(C)=O N1(C(C(COC)CC(C)C)=O)CCC2(CCC2NC(=O)CSC(C)C)CC1 c1(C(=O)NCC2CCC(NC(COCCOCC)=O)C2)cnc(C2CC2)nc1O n1(CCC)cccc1C(=O)NC1CCC(CCNC(=O)Cc2n[nH]c(C)n2)C1 c1(C(=O)NCC2N(C(C(C)Cn3ccnc3)=O)CCC2)cccc2c1CCCC2 c1(C(N(C(CNC(CCSC)=O)C)C)=O)ccc2c(c1)N(C)CC2 N1(C(C2CCCC2C)C(=O)NC(C)C)CCN(C2CN(c3ccccc3)C2)CC1 C=CCCCC(=O)NC(CCF)C(=O)NCCC1CCCN1C C1(OCC)CCN(C(=O)C(C)N(C(=O)CCCC2CC2)C)CC1 C(=O)(CC(C)(O)c1ccccc1)NC1CC(CNC(C(C)OCC(C)C)=O)C1 N(C(=NCCCCl)NCc1ncc(CCO)s1)C(C=C)C1CC1 c1(OC)cc(NC2CCCN(C(C3CC4(C3)CC(O)C4)=O)C2)nc(C)n1 CC(=O)CCCC(C)C(=O)N1CC(C2CN(C(C3CCCSC3)=O)CCO2)C1 c1(CC)cc(NC2(c3nnnn3CCC3CC3)CSC(C)C2)cc(F)c1 C(C)(C(C(=O)N1CCOC(C)(C(C)C)C1)C(C)C)NC(c1c(C)nc(CC)o1)=O CC1CCCCN1CCC(=O)NCC1CC(NC(=O)C(C)N2CCCC2)C1 N1(C(CCCCC=C)=O)CC(C)CN(C(=O)CC2(COC)CC2)C(C)C1 C#CC(CNC(c1ncoc1CNC(=O)C(C1(O)CCCC1)F)=O)CC(C)(C)C Cc1ccc(NC(C2CCCN2C(C2CC(=O)N(CC(F)(F)F)C2)=O)=O)c(Cl)c1 CCC(C(=O)N1CCC(C)(CNC(=O)CCCN2CCCCC2)C1)C(C)C CCC(CC)CCC(=O)N1CCCOC(CNC(C2CCCC(=O)N2)=O)C1 C1(NC(CC(C)C)=O)CC2(C1)CC(NC(=O)C(C)(C)Cc1ccccc1)C2 CN1C(=O)CCC1C(=O)NC1(NCC(=O)NCc2ncccn2)CCC1 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NCC(N1CCCCCC1)C Cc1nsc(C(=O)NCC2CCC2C(=O)NCc2ccc(O)nn2)c1N Cc1nc(C)c(CC(N2CC(CNC(=O)CCc3cccc(O)c3)CC2C)=O)s1 C1(NC(c2c(CC)nns2)=O)CN(C(=O)CNS(=O)(=O)C2CC2)CC2(CCC2)C1 c1(C(N2C3C(NC(c4cc(C)sc4C)=O)CC(C3)C2)=O)ccc(S(N)(=O)=O)[nH]1 N1(C(C2CN(C(C)=O)C2)=O)CC2CCC1C(NC(=O)Cn1c(C)c(C)sc1=O)C2 c1(CCC)ccc(C(C)C(=O)Nc2ccc(NC(N)=O)cc2)cc1 Cc1[nH]nc(C(=O)NCC2CCC2NC(C2CC2c2cncs2)=O)c1C C(=O)(C(C)(C)C(C)(F)F)NC1CCN(C(c2ccc(-c3ccc(C)o3)s2)=O)C1 c1(CCC(=O)NC2C3(CC(NC(Cc4nc(C)[nH]n4)=O)C3)C2)nnc(O)nc1O N1(C(C23CC(C)C2C3)=O)CC2CCC(NC(=O)C(=O)NCC(F)F)(C2)C1 N1(C(CCc2cc(C)ncc2)=O)CCC2(CCC(CC(N3CCC3)=O)CC2)CC1 c1(OC)ccc(C(N2C(C(=O)NCC(c3ccccc3)C)CC3CC23)=O)c(Cl)c1 C1(C(C)NC(=O)Cc2cnsc2)CCCN(C(=O)CCC2CCCCCC2)C1 c1(OC)cc(C(N2CCC(C)(CNC(C3(CC4CC4)CC3)=O)C2)=O)cc(F)c1 c1(OC)cc(CC(=O)NCCCCC(C)NC(c2cncs2)=O)ccc1F N1(C(c2occ(C)c2)=O)CC2CCC1C1CN(C(=O)Cc3cncnc3)CC21 N1(C(CCC)=O)CCC2(C1)CN(C(C1CC3CCC1CC3)=O)CC(C)O2 CC(C)CCC(O)C(=O)N1CC(C(=O)NCCCCCCC2CC2)CC(C)C1 Nc1c(C(N2CCCC2C2(NC(C3CC(C(F)F)C3)=O)CC2)=O)ccnc1Br C1(N(C(C(=O)NCCOC(C)C)=O)C)CCCCCC1.C12CCCN1C2=O C(C(CCC)C(=O)N1CC(n2ccnc2)C1)NC(COC1(C#C)COC1)=O C1(CNC(Cc2c(C)noc2)=O)CCC(C)CN1C(c1ccn(C)n1)=O c1(OCC(N2CC(NC(C(CC#C)C)=O)C2)=O)ccc(C)c2c1C(=O)CC2C C1(C(=O)NCC2(C(C)NC(=O)CC3C=CCC3)CC2)CCc2nn[nH]c2C1 N1(CC(=O)N(c2ccccc2C)CC(=O)OC)CCC(F)(F)C(C#N)C1 Cc1ncc(Br)c(N2CCC(C(=O)NCc3cc(C(=O)O)nn3C)CC2)n1 Cc1csc(C(=O)N(C)CC=CC(=O)NC(c2ccn(C)n2)(C)C)c1C N1(C(c2cnn(CC)c2C)=O)CC2(CCC2)CC1C(N1CC2CC2C1)=O C=CC1(C(=O)NC2CCN(C)C2=O)CCN(C(=O)C(C)SC(C)C)C1 Cc1c(-c2nn[nH]n2)cnc2c1N(C(=O)NCC(C1CCOC1)F)CCO2 N(C(=NCCSC)NCC(N1CC(C)OC(C)C1)C)C(COC)CC(C)(C)C Cn1ncc(C(N2CC(CNC(=O)CN3C(=O)CCCC3=O)C2)=O)c1C#N CC1C(NC(=O)COC(F)(F)F)C(C)CCN1C(C12CC=CCN1CCC2)=O C1(NC(=O)NC(CCCC)CC)CCC(C#N)CC1 CN1CCCCC1CC1CN(C(N)=O)C(c2ccccc2)C1 C1(C(F)F)(CNC(C(C2CC2)SC)=O)CCN(C(=O)CSc2ccccc2C)C1 C1(C(N(CCCN(CC)CC)C)=O)CC12CCN(C(=O)CCC1(C#N)CCC1)C2 c1(C(N(CC(C)(C)NC(C(C2CC2)SC)=O)C)=O)c(F)ccc(F)c1F C(=O)(C1CCCc2cccnc21)N1C(CNC(COC)=O)CCC(C)(C)C1 N1(C(CCCC=C)=O)CCC(CC)CC1C(=O)NCC(C)(O)CO N1(C(C(C)=CC2CC2)=O)CC(C)(C)OCC1CNC(c1cncc(F)c1C)=O c1(CC(=O)NC2CC(NC(C3ON=C(C)C3C)=O)CC2O)ccc(C)cc1C N1(C(c2ccnc(F)c2)C(=O)NC(C(=O)OC)C)C2CCCC1CC(O)C2 C12(NC(C(C)C3CC3)=O)CCCCC1CN(C(=O)Cc1cncc(Br)c1)C2 C1(CCC)CN(C(C2CCC(O)C2)=O)CCN1C(=O)C=NOC C12(C(=O)NCC(CC)NC(c3ccc(=NC)[nH]c3)=O)CC3CC1C2C3O C1(C(=O)NCn2c(CC)ncc2)CNC(=O)CN1C(=O)CC(C)N(C)C N(C(=NCc1sccc1C)NC1CC1)C1CCN(C(CC)=O)C1 C1(NC(=O)CC(C(=C)C)OCC)CC2(CCCCO2)C1.C#CC12CN(C1)C2=O Cc1nsc(CC(N2CCCC2C=CC(=O)N(CC(O)C2CCC2)C)=O)c1N c1(C(N2CCC(C)(NC(c3ccc(OC)nc3)=O)CC2)=O)cc(Cl)c(F)cc1O C1(NC(CCOCCCOC)=O)CCC(O)CN(C(c2cnn[nH]2)=O)C1 c1(CC)ncc(C(=O)NCC2CC(O)CN2C(c2ccco2)=O)c(C)n1 CC1(C)CCCOC1CC(=O)NCCC1(NC(c2ccnnc2O)=O)CCC1 C(C1=NOC2CCCCC12)NC(=O)NC12COC(CN=c3nc[nH]s3)(C1)C2 C(=O)(CC(C)C(F)(F)F)NCCCNC(C12C(C(=O)OC)(CCC1)C2)=O c1(C(N2CC(C(C)(C)O)(CNC(=O)CN(C)C)C2)=O)cc(F)ccc1Cl c1(C(N2CCC(C(C)NC(Cc3c(C)non3)=O)C2)=O)cc(S(N)(=O)=O)c(C)s1 CC1(C(=O)NCC2(CC(N3CCOC(C(N)=O)C3)=O)CC2)CCC(O)CC1 C1(NC(Cc2c(C)nc[nH]2)=O)CC2COCC(C1)C2NC(=O)CC(C)C(C)C c1(C(N2CCC3CN(C(C4CCC5(CC5)C4)=O)C3C2)=O)ccn2ccccc12 N1(C(CCCCC#C)=O)CCC=C(C(=O)N2CCC(O)(C#C)C2)C1 C(=O)(CC1CS(=O)(=O)c2ccccc21)OC(CN1C(=O)CC2(CCCCC2)C1=O)=O C1(NC(C(C)=C(CC)C)=O)CN(C(=O)CCn2cccc2)CC2(CCOCC2)C1 C1(F)(C(=O)NC2C(C(=O)NCCC3(COC)CC3)COC2)CC=CCC1 c1(NC(=NCn2c(CC)ncn2)NC2CC2)ccc2c(c1)C(=O)NCC2 N1(C(COCCC=C)=O)CCCC(N(C(=O)C(C)CN(C)CC)CC)CC1 N1(C(c2c(OC(C)C)cccn2)=O)CCC(NC(=O)CCCCC2CC2)C(O)C1 C(O)(C(F)(F)F)C1CC(NC(=O)NC2CCOC2)C1 N1(C(c2n(C)nnc2)=O)C2CCC1C(NC(c1cccc(-n3cccn3)c1)=O)C2 c1(C(=O)NC2CN(C(C(C)N(C(C)=O)C)=O)CC(F)C2)nc2ncccn2n1 c1(NC(=O)CC2CCCN2Cc2c(O)cccc2Cl)ccc2[nH]c(=O)ccc2c1 CC1(CNC(C2CCSC2)=O)COCCN(C(=O)CCc2ncc[nH]2)C1 C(=O)(C(C)C(=O)OC(C)(C)C)NCCCCCNC(C(n1ncc(C)c1)C)=O N1(CC)CC(NC(=O)CC(CNC(=O)CCC2CC2(C)C)OC)C(C)C1 C1(C(=O)NCC2COCCN(C(C(C)=C(C)C)=O)C2)CCc2cnc(C)n2C1 C(=O)(C(C)CC(C)(C)C)N1CCC(C)C1CNC(=O)CCc1ccc(O)nn1 C#CCC(C(=O)NC(c1nc(C)oc1C)C)NC(C1CCC(C)O1)=O Cc1cc(C(=O)NC2CCCC2C(N2CCOCC(O)C2)=O)cnc1F N1(C(C2CCC(=C)CC2)=O)CC2CCCC2C1C(=O)NC1CCOCC1F N1(C(C(c2ccc(Br)nc2)(C)C)=O)CCCC(NC(c2ccc(C#N)o2)=O)C1 C1(NC(C(F)OC)=O)CCN(C(=O)CCC2CC2(F)F)C1(C)C Cc1ccnnc1C(N1CCC(O)(c2cccc(C(F)(F)F)c2)C1)=O c1(OC)ccc(C(=O)NCC2(NC(c3ncncc3F)=O)CCC2)c(O)c1 c1(C(N2C(CNC(C#CC(=O)N(C)C)=O)CC(C)(C)C2)=O)scc2c1OCCO2 N1(C(CCC)=O)CCCC1C(=O)NCC(C)CNC(C1CCCC1O)=O N1(C(CC(=C)C)=O)CCN(C(C2CCN(C(c3ccnnc3S)=O)CC2)=O)CC1 C(=O)(C1c2ccccc2-c2ccccc21)N1CCC(CN(C(CCOC)=O)C)C1 c1(C(=O)NCCOCCCNC(CN(CC(C)C)C)=O)ccn(C(C)(C)C)c1 c1(C(=O)NC2CN(C(C(CCC)OC)=O)CC2C)ccc(C(C)C)nc1F C1(CNC(CSCC=C)=O)CC2(CCN(C(C3CCC4CC4CC3)=O)CC2)C1 c1(C(C)C)ccc(C(=O)OC(c2nc(-c3ccc(F)nc3)no2)C)cc1 C(c1ccc(Br)c(Cl)c1)=CC(=O)NCC(CNC(CC)=O)OC C1(O)(CCNC(c2cc(C3C(C)C3)on2)=O)CCN(C(=O)C(F)(F)CO)CC1 CCCCCC(O)C(=O)N1CCC(N2CCN(c3cc(O)ncn3)CC2)C1 C(C(C)NC(C1(CCF)CCOCC1)=O)(C(C)C)NC(c1cc(C)sc1)=O c1(C(N(CC(C)(C)C)CC(F)(F)F)=O)ccc(N)c2cnccc12 N1(C(=O)Cc2ncccn2)CC2CCN(C(c3ccc(O)c(Cl)c3)=O)C2C1 C1(NC(c2c(C(=O)OC)cccc2)=O)CC(F)(F)C1(C)C.C12(CC1)C(C)NC2=O c1(C(N(C(CCNC(CC2CC(C)C2)=O)C)C)=O)cnc(C2CC2)[nH]1 CCCC(CC)CCC(=O)N(CCNC(c1ccc2c(c1)C(C)CO2)=O)C1CC1 c1(OC(C2C(C)CCCN2C(=O)OC(C)(C)C)=O)ccc2nccnc2n1 c1(OC)ccc(CC(C)C(N2CCN(C(=O)CNC(N)=O)CC2CO)=O)cc1F O=C1CSc2ccc(C(=O)NC3CCC(NC(C4COC4)=O)CC3)cc2N1 N1(C(=O)CC2CC3(COC3)C2)CCCN(C(c2c(O)cccc2Cl)=O)CC1 N1(C(c2c(F)ccc(C)c2)=O)CCS(=O)(=O)C(CCNC(C2CC2C(F)F)=O)C1 C1(CNC(c2n(C)nc(Br)c2)=O)CCCN(C(C2CC23CCC3)=O)CC1 c1(CC(CNC(=O)CC=C(C)C)N(C(C2(CCC)CC2)=O)C)ccccc1Cl Cc1nc(C2CC2)[nH]c1C(=O)N(C(C)CCNC(=O)COCP(C)(C)=O)C Cc1cc(=O)oc(C)c1C(NS(=O)(=O)N(C)C1CCCCC1)=O c1(OC)ccc(C)cc1C(N1CCCC(N(C(=O)C(O)P(C)(C)=O)C)C1)=O N1(C(C(C)C2CC2)=O)CC2CCN(C(=O)CCN3CCCCC3)CC12 CC1(C)COc2c(CCC(=O)NCCCn3cc(CC4CCC4)nn3)cccc21 Cc1cc(C(C)C)nc(=NCC(C)N(C)C(C2CC23CCc2ccccc23)=O)[nH]1 N1(C(C(CCC)C)=O)CCCC(N(C(=O)COC)CC)CC1 Cc1noc2ncc(C(=O)NC3CCC4CN(C(=O)C(C)(C)CF)CC4C3)cc12 c1(C(=O)NCC(CC)NC(c2cscc2F)=O)ccnc(Cl)c1OC c1(C(N(CC(C)CO)C)=O)sccc1CNC(=O)C=CC1CC1 C#Cc1cccc(C(=O)NCC2(C)CC(NC(=O)C3=CCCCC3)C2)c1C C1(C(=O)OC)COC2(CCN(C(=O)NC(c3noc(C4CC4)n3)(C)C)CC2)C1 C1(CC(=O)NC2C(C(N3CC(OC)(CO)C3)=O)C2(C)C)CCC(=O)NC1.C1CC1 Cc1nc(C(=O)NC2(CF)CCN(C(=O)C=Cc3ncco3)C2)ccc1Br c1(C(N(C(CNC(c2cc(C)cc(Cl)c2N)=O)C)C)=O)ccc2nnc(S)n2c1 c1(C(=O)NC2CCN(C(C=C(CCC)CCC)=O)C2)ccccc1S(C)=O Cc1ccc(CC(N2CCSC(C(=O)NCC(O)Cn3cccn3)C2)=O)cc1 C1(CNC(CN(C2CC(C#N)C2)C(c2cc(C3CC3)on2)=O)=O)CCC(F)(F)C1 C1(CN(C(c2ccccc2C2CC2)=O)CC)CCCCN1C(=O)CC1(CO)CC1 c1(C(N2CCC(C3CCCO3)C2)=O)n[nH]c2c1CN(C(c1sccc1F)=O)C2 N1(c2n(CC(CC)(c3ccccc3)c3ccccc3)nnn2)CCC(COC)C1 C1(CCO)(CNCC2(Br)CC2(F)F)CCCO1 CC1(C)C(NC(=O)Cc2cc(O)nc(O)n2)CCN1C(=O)C(O)CC(N)=O N1(C(C(C2CCCCC2)C)=O)CCC(C)(C)C(C(=O)NCc2nncn2C)C1 c1(CN(C(c2csc(Cl)c2)C(=O)NCCC#N)C)cncn1C C12(C(=O)NC(CC=C)CNC(=O)Cc3c(C)nc(C)n3O)C3C4C1C1C2C3C41C N1(C(C(C)OC)=O)CCCC2(CCCN(c3ncc4c(n3)CCC4)C2)C1 Cc1c(C(=O)NC2CCC(C)N(C(=O)C(=O)Nc3ncc[nH]3)C2)cccc1Cl C1(CNC(C2CC(C)OCC2)=O)CN(C(=O)Cc2cccc(C#N)c2)CCN1C C12(CNC(C3ON=C(CC)C3)=O)CCC(C1)N(C(=O)Cc1c(F)cccc1Cl)C2 C1(NC(c2cnc(C(C)O)s2)=O)CC2(C1)CN(C(=O)CC(C)C(C)C)C2 C1(C(=O)NCCc2n(C)ncn2)CCCCN(C(=O)CCOC2CCCC2)C1 Cc1c(C(N2CCC(C3CCCN3CC=Cc3cnn(C)c3C)C2)=O)nn(C)c1N c1(-c2cncc(OC)c2)c(C(=O)Nc2cnc3cc[nH]c3c2)nn2c1CCCC2 C1(CC(=O)NCCC(COC)C)CN(C(=O)CN2CCCCC2C)CC1C c1(COC(C2C(F)(C(=O)OCC)C2)=O)cccc2c1OC(C)(C)C2 N1(C(c2cn(CC)nc2)=O)CCC(C(=O)NC2C3CCCC23)(CF)C1 C12(C(=O)OC)CCC(C1)OC21CN(C(C2CN(S(=O)(=O)c3ccccc3F)C2)=O)C1 Cc1c(C(N2CC(CC(C)NC(=O)Cc3ccc(C(N)=O)cc3)C2)=O)cncc1F C1(C)(CCC(=O)N(CC(O)CNC(C2CCCC2)=O)C)CC1(F)F N1(C(C2C(CC)CCC2)=O)CCC=C(C(=O)N(C2CCN(C)C2)C)C1 N1(C(c2c(C)nc(CNC(C3CC34CCCC4)=O)o2)=O)C2CCC1CC1(C2)N=N1 Cc1cc(C)c(C(N2CC(C(N3CC(C)(C)C3)=O)C(O)C2)=O)c(C)c1 CN1CCOCC1CNCC1CCCOCC1 c1(C(CNC(CSCC=C)=O)NC(=O)CSC2CCOC2=O)ccc(F)cc1F C12(C(=O)NC3CC(C)(NC(c4c(OC)cccc4)=O)C3)CCC(C1)C(C)(C)O2 N1(C(C(C)(CO)NC(C2(CN(C)C)CC2)=O)=O)CCC(CO)C(O)C1 Cc1ccc(C=CC(=O)NCCCC(C)NC(=O)C(C)(C)c2cccnc2)s1 C(=O)(C(C(C)NC(=O)CCOCC(C)(C)C)C(C)C)Nc1cccc(OCC)c1 Cc1cc(=NC(=O)c2cn(CC(F)(F)F)nn2)[nH]n1-c1c(Cl)cc(Cl)cc1Cl C1(OC(F)F)CCN(CCNc2ccccc2OCC(F)(F)F)CC1 C(C(C(C)C(C)C)NC(=O)C=CC(c1ccccc1)=O)NC(CSC(C)C)=O CC1(C(=O)Nc2ccc(-c3cccs3)s2)CCN(C(c2ncccn2)=O)C1 N1(C(C(CC)C#N)=O)CC(C)(C)C(NC(=O)C(C)Cc2ccncc2)C(C)(C)C1 c1(N(CC)CC)ccc(CC(=O)NC2CCN(C(=O)CCC3OCCO3)C2)cc1 C1(CNC(COCCCCC)=O)CN(C(=O)C(=C2CCCCC2)F)CCC1C CC(C)(O)CC(=O)NC1CC(CNC(=O)C(c2ccccc2)O)C(O)C1 N1(C(CC(=C)C)=O)CCC2CCCC12CNC(=O)CCCS(N)(=O)=O N1(C(C(CC)(C)C)=O)CC2(CCCN2C(c2cccc(OC(F)(F)F)c2O)=O)C1 C1(C(=O)NC2C(C(N3CC(Cc4ccoc4)C3)=O)CCC2)(OC)CCSC1 c1(C(=O)NC(CNC(C(CC)NC(N)=O)=O)CO)cc2cc([N+](=O)[O-])ccc2o1 c1(C(=O)NC2CN(C(C3(C)C(C)C3)=O)CC(F)C2)cccc2ccn(C)c12 c1(C(=O)NCCCCC(CO)NC(C2CC(OC)C2)=O)ccc2c(c1)CCCS2 C1(=CC(N2CCC(N(C)Cc3c(C)cc(OC)nc3)C2)=O)CCC(C)(C)CC1 C1(NC(c2c(C)noc2)=O)CCC(CNC(c2cncn2C)=O)CC1 c1(C(C)C)nc(CN(C(c2sccc2Br)C(=O)NC2COC2)C)cs1 C(=O)(N=c1cc(C)[nH][nH]1)C1N(C(c2ccc(NC(C=C)=O)cc2)=O)CC(F)C1 C#CC1CCC(C(=O)NC23CC(NC(=O)CC(C)F)(C2)C3)CC1 C12(C(=O)NC(CC)CNC(=O)CCNC(c3ccoc3)=O)CCCCN1CCC2 c1(C(CNC(=O)Cc2cccs2)NC(=O)CCc2nncs2)cccc(Cl)c1 C1(NC(CCc2cccc(-n3cc(CCN(C)C)nn3)c2)=O)CC2OCCCC12 C1(C(=O)NCCC2(NC(c3cc(C)c(Cl)s3)=O)CCC2)CCCC2(CC2)C1 C12(CNC(c3c(C)nn[nH]3)=O)CCC(CN(C(c3cc(=O)n(C)cn3)=O)C1)C2 C1(OC)CCC2CN(C(=O)CCCCSC)CC12 c1(C(N(CCCNC(C2C(CCC)CCC2)=O)CC)=O)cc(C)c(Cl)cc1F S(=O)(=O)(c1ccc(O)cc1)NC1CN(C(C2C(C)=CCC=C2)=O)CC1O Cn1cc(C=CC(=O)NCC2CCC2C(=O)NC2CCNC2=O)cn1 N1(C(CC2(CC)CCC2)=O)CC(NC(c2cnn(C(C)C)c2C)=O)CC2(CC2)C1 C1(C(N(CCn2cc(Cn3cccn3)nn2)CC)=O)CC2(CCC2O)C1 C#Cc1ccc(C(N2C3CCC(C(=O)OC)C2CC3)C(=O)NC2COC2)c(Cl)c1 N=c1[nH]cc(CCCNC(=O)C(=O)NCC2COCCO2)[nH]1 N1(C(c2cnn(CC)n2)=O)CCCC(N(C(=O)CCC2CCOC2)CCO)C1 C1(O)(CNC(=O)C(F)n2cccn2)CCCN(C(=O)Cc2ccccc2)CC1 c1(C(=O)NC2C(NC(CC(CC)OC)=O)CCC2)ccc(F)c(Cl)c1N C(=O)(C1=CC2(CCOCC2)C1)NC1CC2(N(C(C=COCC)=O)CCCC2)C1 c1(OC)ccc(SCC(N2CCC(C)(NC(=O)CC(C)SC)C2)=O)cc1 c1(C(=O)NCC(C)N(C(C2(CC=C)CCCC2)=O)C)cc(C)ccc1[N+](=O)[O-] C1(CC)(NC(=O)CC#N)CN(C(=O)C(F)CC2CCOC2)C1 c1(C(C(=O)N(CC(COC)C)C)NC(=O)C(C)N(C)C(C)=O)ccnn1C c1(-c2cccc(C#N)n2)ccc2c(C(=O)NCc3ccccc3Br)nsc2c1 C1(C)(C(=O)OC)CC(Nc2sc(Br)cc2F)CN1C(=O)C1CC1 c1(C(=O)NC2C(NC(c3cncs3)=O)COC2)c(Cl)ccc2c[nH]nc12 C1(C(c2ccccc2)C)CN(CC2(C3CCCCO3)CC2)CCO1 Nc1c(C(N2CCC(F)(CNC(=O)C(F)n3ccnc3)C2)=O)cnc2ccnn12 c1(NC2CN(Cc3cccc(C)c3Br)CC2O)[nH]cnc2nc(Br)cc1-2 C1(OCC#C)CCN(C(c2c[nH]nc2CCNC(=O)C(COC)OC)=O)C1 Cc1ccnc2c(C(N3CCC4(C(N5CC6CC6C5)=O)CC4C3)=O)cccc12 C1(NC(C2(COC)CCCO2)=O)CC2CC(C1)N(C(=O)Cc1ccccc1F)C2 C1(O)(C(C(=O)NCC2CC3(CC3)C2)NC(c2c(C)nn[nH]2)=O)CCCCC1 C1(NC(c2ccoc2Cl)=O)CCCC(C(N2CCCC(CO)C2)=O)C1 C1(NC(C2CC23CC3)=O)CCC12CN(C(=O)C=CCCc1ccccc1)C2 C=C1CCCN(C(=O)C(CC)NC(C2CCC2COC)=O)C1 N1(C(c2n(OC)cnc2C)=O)CC(NC(C2CC(C)C2)=O)C(C2CC2)C1 CC(CC(=O)NC1C=CC(C(=O)NC2COC(C(F)F)C2)C1)C(F)F C1(NC(CCC(N)=O)=O)CCOC12CCN(C(C1CCNC(=O)C1)=O)CC2 c1(C(N2CC3C(CNC(c4ccc(Cl)c(Cl)c4)=O)(C3)C2)=O)cccc2cncn12 c1(CNC(C2N(C(C(CC)c3ccccc3)=O)CCC2CC)=O)ccc(C)c(F)c1 c1(C(N(C2CC(NC(C3CCC(=C)CC3)=O)C2)C)=O)cccc2c1C(=O)NC2=O c1(N(c2nc(-c3cccs3)cc(C)n2)C2CC2)cc(F)cc(F)c1F C1(CCOC)CC(c2nnnn2C)(Nc2cnn(CC(F)F)c2C)CCO1 N1(C(c2cc(C)on2)=O)CC(NC(=O)CSCc2ccccc2)CCC(O)C1 c1(C(=O)NC2C3CN(C(c4cc(C)c(F)cc4)=O)C2C3)[nH]c2ccccc2c1Cl CS(C)(=O)=Nc1cnn(CC(=O)NCC2C3CN(C(C4C5C=CSC45)=O)CC23)c1 N1(C(c2nc(CC)[nH]n2)=O)CCC2CCC(C1)N2C(=O)C(c1cncc(F)c1)C S(=O)(=O)(c1cc(C)cnc1NCC(C)Cc1cccs1)NC(n1cccn1)CC CCCCCCC(F)C(=O)NCCC1(NC(=O)CC(CC)C(C)C)CC1 C(C)(C)(CC(=O)N1CCCC(OC2CCOCC2)C1)n1cc(C(CC)CC)nn1 N1(C(C(C=C)CC)=O)C(C(N2CCC2CC(C)C)=O)CC2CCCC12 c1(C(=O)NCC23CC2CN(C(=O)CCN2CCOCC2=O)C3)cc2c(s1)CCC2 C1(NC(Cc2c(C)ncs2)=O)C2CN(C(=O)C(C(C)C)n3cnnc3)CC12 C1(C2CCOCC2)(C(=O)NCCCOCCC(C)C)CC1 N1(C(c2ccc(CC)[nH]2)=O)CC2CCC1CN2C(C1CC(C(F)(F)F)C1)=O C1(CC(=O)N(C(C)CNC(c2cccc(CO)n2)=O)CC)CC12CCOC2 C1(C(=O)NCC2(O)CCCOC2)(COC)C=CCN1C(c1c[nH]c(=N)o1)=O N1(C(CN(CC=C)C(=O)CC2CSC2)=O)CCC(NCCCC)CC1 S(=O)(=O)(c1ccc2c(c1)CC(=O)N2)N(CC(c1cccnc1)N(C)C)CC(F)F CCCC(O)CC(=O)N1CC=CC(NC(c2cccc(SC)c2Cl)=O)C1 C1(NC(c2c(C)nns2)=O)CC2CN(C(=O)CCC(C)(C)F)CC2C1 C(=O)(C1=NOC2(CCC2)C1)N1C(CC(=O)NCCN(C)CCF)CC(O)C1 CCCCCC(F)C(=O)N1CCC(C(=O)NCCc2ccc(C)s2)(CO)C1 C(c1ccc(Cl)cc1F)=CC(=O)NC12CC(CNC(C(CCCC)O)=O)(C1)C2 c1(C(=O)NC2CC(CCNC(=O)CC3CCC(O)C3)C2)ccc2nnn(O)c2c1 CCCC(C(=O)NCc1cc(OC)ns1)NC(=O)CC(C)F CC(C)CC(C)C(=O)NCC1C(C)CCN1C(c1ccc(C2CC2)nc1)=O c1(C(=O)NCCC2N(C(C(C3CCC3)OC)=O)CCCC2)cc(F)c(C)cc1N C(=O)(CN=c1cc[nH]cc1)NCCN(C1CCCC1)C(C1C(C)OCCC1)=O C1(NC(CN(C)C)=O)CCS(=O)(=O)C2(C1)CC(CNC(=O)C(C1CC1)N(C)C)C2 N1(C(C(CC)C#N)=O)CCC(C2CC2)(CNC(c2ccc(OC)s2)=O)C1 N1(C(C=CCN(CC#C)C)=O)CC2(CC2)CC1CNC(=O)CCC1CC1C c1(OC)ncccc1S(=O)(=O)NC1CCC(NC(=O)CCC2CCCC2)C1 C(C(=O)N(CC(C)NC(c1cncc(C(=O)OCCSC)c1)=O)C)(C(C)C)CC N1(C(C2CCN(C)CC2)=O)CC(NC(=O)CSc2cnn(C)c2)CC(F)C1 C1(NC(c2c(C(C)C)cco2)=O)CCCN(C(=O)CCc2nncn2C)CC1 N1(C(C(CC#C)(C)NC(c2n[nH]c(C)c2Cl)=O)=O)C2CCC1CC1(CC1)C2 C1(CNC(C(C2CCC(=O)N2)C)=O)CCN(C(C2CCSCC2)=O)C12CC2 C=C(F)C1(CC(=O)NCc2ncc(CC)[nH]2)CCC1.C1CCC(=O)NC12CCC2 CCC(C)(C)CCNC(C1(CCNC(c2cn(C3CC3)cn2)=O)CC1)=O C1(N(C)C(=O)C2CC2)CCN(C(C2CN(C(C(=O)NCC)=O)C2)=O)CC1 n12cc(nn1)CN1CCCC1C(=O)NCC2C.CC(C)C(O)c1ccco1 C(=O)(C(C)CC(C)(F)F)NCCC1N(C(C(C)SCCCC)=O)CCC1 c1(OC)cccc(O)c1C(=O)NCC1CCN(C(=O)CC2CC(F)C2)C(C)C1 c1(N2CCC(C(N3CCCC(C(=O)OC)CC3)=O)C2)nc(Cl)nc2[nH]c(O)nc12 N1(C(COCCOCC#C)=O)C2CCC1C(NC(=O)CN1CCCC1CO)C2 CC1CCN(C(c2ccn(C)c(=O)c2)=O)CC1C(=O)NOC1CCC1 Cc1onc(C(=O)NC(C)CNC(C2CCCCN2CC(F)F)=O)c1[N+](=O)[O-] C(=O)(CC(C)CC(C)(C)C)NCc1ncc(C(=O)NCC2(CC(C)C)CC2)cn1 C(=O)(CCCC(C)(F)F)N1C(CNC(C(CC)OC)=O)(COC)CCC1 C1(CNC(C2N(C)C(=O)CCC2)=O)CC2CCC1N(C(=O)CSC(C)(C)C)C2 CC1CN(C(C2(C)CCCO2)=O)CC2(CCN(C(=O)Cc3cccc(N)c3)C2)O1 C1(OC)CC2CC(C(=O)NCCCCN(C)C(c3cscc3Cl)=O)CC12 C12(C(=O)NCC(CNC(c3cn(CCC)nc3C)=O)F)CC(C)(C1)OC2(C)C C1(CC(C(CC2CN(C(C)=O)C2)=O)=O)CCCC2(CC2)C1.C12(CCOC1)OC2.NC c1(C(C)NCc2cc(C(C)(F)F)n[nH]2)sc(C(F)(F)F)cc1Br c1(N(C)Cc2nc3ncccn3n2)cc[nH]c(=NCCCCCF)n1 CC1CN(C(=O)CC2CCCNC2=O)CC(C)N1C(C1CC12CCOCC2)=O N1(C(c2c(C)occ2)=O)CCN(C(=O)CCCCNC(N)=O)C(C)C1 C1(=CC(=O)NCC2COCCN2C(C2COCCO2)=O)CN2CCC1CC2 C1(NC(CCS(N)(=O)=O)=O)CN(C(C2CC2(F)F)=O)C2(CCC2)C1 C(C1=CCN(CCCc2ccc(F)cc2)CC1)NC(C1CCCC1)=O c1(CNc2c(C(=O)Nc3ncc(C#N)cn3)nccc2)ccc2nc(O)[nH]c2c1 CCC(CC(F)F)C(=O)NCCOCCNC(c1cc(Br)c(C)cc1C)=O N1(C(C2CC(C(=O)OC)C2)=O)CC2(CCCC2)C1C(=O)NC1CC2(CCCC2)C1 O=C(C1CCCc2cncn21)N1CCC2OCCN(C(c3cocn3)=O)C2C1 C12(C(=O)NC(CNC(C(=Cc3ccccc3)OC)=O)CO)CCC(CC1)C2(C)C C1CCC(O)C(=O)N1.c1(-c2ccc(CCN)o2)ccc(C(F)(F)F)cc1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCN(C(=O)CCc1cc(C)on1)CCC N1(C(=O)CC=Cc2ccc(F)cc2)CC(CNC(C2CC(O)C2)=O)N2CCC1C2 CC1(C)CCC(CC(=O)NCC2(C)CCC(NC(c3ccnnc3O)=O)C2)CC1 C12(CCNC(CCCC)=O)CCC(C1)N(C(=O)CC(C)c1cccnc1)C2 CCCCC(F)(F)C(=O)NCC(CC(C)C)C(=O)N1CC(=O)NC(=O)C1 C1(=O)CCC(=O)NCCCN1.C1(C)(NC(C2C(=C)C2)=O)CN(CC)C1 c1(C(=O)NC2C(C(=O)NCCC(C)CCO)CCC2)cccc2ccoc12 Cc1cc2c(cc1C(=O)NCCCN(C(=O)C(C)S(C)(=O)=O)C)OCO2 c1(C(=O)OC)cc(Cl)cc(S(=O)(=O)NCc2nc(C(=O)O)co2)c1F c1(OC)cc(CNC2CCC(C(=O)NCC(C)(F)F)CC2)cc(F)c1F Cc1nc(O)c(C(=O)N(C)CCNC(=O)C(C)OC2CCCC2)cc1Br N1(C(C)=O)CCCCC12CCN(C(=O)NC1COC(C)C1)CC2 CCCCCCC(C)C(=O)NOCC(=O)NCCCc1nncn1C c1(OCC)ccc(-c2cn(CC(C)NC(c3cnn(C)c3)=O)nn2)cn1 c1(C(=O)NC2C(NC(c3c(COC)ncs3)=O)CCC2)n[nH]c2c1CC(C)(C)C2 c1(C(=O)NC2CCC(NC(C=CC=CCC)=O)C2)ccc2nc[nH]c2c1 C1(OC)CCC2(C(=O)NC3(C(=O)NCCCN4CCCC4)CCC3)CC12 CC1CN(C)CCCN1C(=O)CCC1CCCN(C(=O)Cc2ccc(O)cn2)C1 CC(C)(F)C(C)(F)C(=O)N1CCC2C(C1)CN2C(=O)C=CBr c1(C(N2CCC(O)(C(=O)Nc3c(C)ccnc3Br)C2)=O)c(O)ccc(F)c1F C(=O)(C(S(C)(=O)=O)C1CC1)N1CCC(C(=O)OCC)CC1.c12scnc1CN2 c1(CC(N2CC(N(C(=O)CCN3CCOC3=O)C)C2)=O)cccc(Cl)c1 Cc1ccc(C(=O)NC(CC(F)F)c2ccccc2)cc1-n1cnnn1 C(=O)(C#CC(C)(C)O)NC1CCCC(N(C(=O)Cn2cc(C(F)F)cn2)C)C1 C1(CNC(C2C(C)C2)=O)CC2CCC(C1)N2C(C1(C)CC1(F)Cl)=O N1(C(C(CCC)OCC)=O)CC2CC(C1)N(C(c1cc(C#N)c(N)cc1O)=O)C2 c1(C(=O)NC2(CNC(c3ccnc4[nH]nnc34)=O)CC2)cc2cc[nH]c(=O)c2s1 c1(C(=O)NCC(CC)NC(c2cc(O)nc(Cl)c2)=O)cc2c(C)cccc2[nH]1 N1(C(CC=CC)=O)CCOC(CN(C)C(C2CC3(CC3)CO2)=O)C1 c1(C(=O)OC)nccnc1C(=O)NCc1ccccc1CNC(=O)C=CCF N1(C(c2noc(CC)c2C)=O)CCCC(O)(CNC(=O)Cc2cn(C)nc2C)C1 C1(OC)CC(F)CN(C(=O)C(C2CCCO2)NC(c2cc(CO)[nH]n2)=O)C1 C12(C(N(CC(C)(C)NC(C=C(C)C(C)(C)C)=O)C)=O)CCCCC1NC(=O)C2 N1(C(CC(C)OC)=O)CCC2CCN(C(=O)CCC(=O)c3ccccn3)C2C1 N1(C(c2cncc(COC)c2)=O)CC2CCC1CC2NC(=O)C(C)S(N)(=O)=O N1(C(C(CC)N(C)C)=O)CCC2(CCC(NC(c3ncc(C)cn3)=O)C2)CC1 N1(C(c2cccc(OC)c2N)=O)CCN(C(=O)C(C)C(C)(F)F)CC(CO)C1 c1(C(N2CC(NC(c3c(OC)nccc3)=O)(CO)C2)=O)cc(F)cc(N)c1F c1(C(N2CCCC3(NC(C(CCC)C)=O)C(C2)C3)=O)cc(F)c(F)c(O)c1F CC1COCC(CC(=O)NCC2(F)CN(C(c3cn(C(F)F)cn3)=O)C2)O1 C1(COC)CCC(NC(C2(N(C(=O)CCc3ccc[nH]3)C)CC2)=O)CC1 C#CCC(O)C(=O)N1CC(C2CN(C(=O)CCCCc3cnn[nH]3)CCO2)C1 C1(C2CCCCC2)(NC(c2n(CCSC)nnn2)c2ccsc2C)CC1 CC1(C)CC(CNC(C2CCCC(=O)N2)=O)CN(C(=O)CCc2csc(=N)[nH]2)C1 N1(C(C(C#C)(C)C)=O)CCCC(N(C(=O)C(C)CSc2ccc(Cl)cc2)C)CC1 CCCCCCC(C)C(=O)NCCC1(C(=O)N(CC(O)CO)C)CC1 c1(C(N2CCCN(C3CCCC3O)CC2)C(=O)OC)ccc(F)c(Cl)c1 CC1=C(C(=O)NCCCCCN(C)C(c2cnn(C)c2C(C)C)=O)CC1 C1(NC(CCc2cnc(C)s2)=O)CCCCN(C(c2ccc(CF)cc2)=O)C1 N1(C(C2C(CNC(c3occ4c3CCC4)=O)CCO2)=O)CCCC(F)CC1 C(=O)(C(C)(C)C(C)(F)F)NCC(C(=O)NCCc1ncn(CC)c1)(C)C c1(C(=O)NC2C(C)N(C(=O)C=C(Cl)Cl)CC2)cc2c(nc1O)CCCCC2 C1(C(N(CC#C)OCc2ccccc2)=O)CCc2nnc(O)cc2C1 O=C(CCN=c1[nH]ccs1)N(C1CC1)CC1CCCN1C(c1ccc(O)nc1)=O Cc1cc(C(=O)NC2CCCC2CNC(C2(C)CCCCC2)=O)cc(N)c1O C(=O)(C(CC)C(=O)N1CCC1CNC(c1cn(C(C)(C)C)nc1C)=O)OCC c1(C(N(C2CCCN(C(C3(OC)CCCCC3)=O)C2)CC)=O)cn(C)c(O)n1 C1(NC(N2CCCC2C(N2CCCC2)=O)=O)CCc2cc(Br)ccc2C1O C1(n2ncc(C(=O)NCC(CNC(C(=O)NC(C)C)=O)C)c2)CCS(=O)(=O)C1 C1(NC(N(CC(=O)O)Cc2cccs2)=O)CCOC1 C1(CC=C)(C(=O)N(C)CC2CC2(C)C)CCN(C(=O)CCC=C(C)C)C1 C(C)(C)(C(=O)NCCc1cc(C(=O)NCCC(Cl)Cl)no1)OC(C)=O C1(CN(C(C23CCC(C2)C3)=O)C2CC2)CN(C(C2(c3ccccn3)CC2)=O)CCO1 CC(C)CC(C(=O)NCC(C)OC(F)F)ONC(=O)CCc1csnn1 C1(C)(C(N2CCC(O)(CNC(C3(CCOC)CCCC3)=O)C2)=O)CCN(C)C1=O C#Cc1ccccc1CC(N1CCC(CO)C(NC(C2(CO)CCOC2)=O)C1)=O CC1=NS(=O)(=O)NC=C1C(=O)NCC1(C(N)=O)CN(C(C2CCCSS2)=O)C1 Cc1ncc(C(=O)NCC(C)CN(C(=O)C(C(C)C)N2CCCC2=O)C)c(C)n1 C(N=c1[nH]c(=NCCN(C)C2CC2)c2sccc2[nH]1)C1C(C)COC1 C#Cc1cncc(C(=O)N(CCCN(C)C)CCNC(c2ccnc(S)c2)=O)c1 C1(NC(C(n2cc(Cl)cn2)C)=O)CC2(C1)CC(NC(=O)CC1SC(=N)NC1=O)C2 c1(SC(C)C)ncccc1C(N1CC(CNC(=O)CC2(O)CCCOC2)C1)=O CC(C)(C)CCC(=O)NC(CNC(c1ccc(-c2ccc(Cl)s2)cn1)=O)C1CC1 Cc1ccc2c(c1)C(=O)N(C(C)C(=O)NCC1CC(NC(=O)C(C)C)C1)C2=O c1(C(=O)NN(C)Cc2onc(C(C)OC)n2)ccccc1-c1nc[nH]n1 O=C1CCC(CC(=O)NC2(CC=CC(=O)NC3CC3O)CCC2)N1 C=Cc1cnn(C)c1C(N1CC=C(CNC(=O)C=C2CCSCC2)CC1)=O N(C(=NCCC12CCCC1C2(F)F)NCC1CCCCO1)CCCOCC c1(C(=O)NCC2(C)CCN(C(C3CCN(C)S3(=O)=O)=O)C2)occ2c1CCCC2 c1(OCC)nccc(C(=O)NC2CCC2NC(=O)C(C)OC)c1F C1(CCOC)(NC(=O)C=CI)CCN(C(c2cccc(OC)n2)=O)C1 C1(CNC(C(C)OCCOCC)=O)COCCN(C(c2cn(C)cc2C)=O)C1 C1(C(=O)Nc2scc(S(=O)(=O)NC)c2)Cc2cncn2C(=O)N1 CCC(C)(C)C(O)C(=O)N1CCCC(CN2CCN(C(=O)CC3(C)CC3)CC2)C1 N1(C(C(C)SCCCC)=O)CCCCC12CN(C(=O)Cn1cncc1C)C2 c1(CC=O)ccc(Cl)c(F)c1.c1(C(=O)NCCCN(CC)CC)cncn1C1CC1 C1(CNC(CCCSC)=O)CC2CC1CC2O.C12(CCC1)CC=CC(=O)N2 c1(NC(C2(C#C)CN(C(=O)C(C)c3ccsc3)C2)=O)cc(C#N)ccc1O c1(C(=O)NC(CC)CNC(C2(C)CC(C)=NO2)=O)cnc(N)c(N)c1 CCC(F)C(=O)N(CC(C)CNC(=O)CCSCc1ccccc1)C C(=O)(CC(C)(C)C(=O)NCC1CC2(CCC2)CN1C(=O)Cc1cnsc1)OC c1(CNC(C(CCC)OCC)=O)nnc2n1CCN(C(C1CC1F)=O)C2 c1(CC)cccc(C(=O)NCC(C)=CC(=O)NC(c2cnc(C)s2)C)n1 c1(C(c2nnnn2C2CC(F)(F)C2)NCCCC=C)ccc(Cl)c(C)c1OC C(C1=NOC2CCCCC12)n1cc(CN(C(CCC(C)C)=O)CC2CC2)nn1 c1(C(N2CCC(CC=C)(NC(=O)C(CC)=CC)C2)=O)cc(C)c(Cl)cn1 C1(Nc2c(OC)cccc2)CC12CCN(C(=O)NCc1ncc(Cl)cc1Cl)C2 C1(C)(C(=O)NCC(C)NC(c2cccn(CCN(C)C)c2=O)=O)CC2CCC1C2 N1(C(=O)CN2CC=CC2)CCN(C(C2(CCN(C)C)CC2)=O)C2(CC2)C1 CC1(C)CCC(C)(C(N2CCC(CC(=O)Nc3cccnc3)C2)=O)CC1 c1(C(N2CCC(=CC(N3CC(CCO)C3)=O)CC2)=O)cc(O)nc(O)n1 c1(N2CCC(N(C)Cc3nccc(C)n3)CC2)nnc(C)c(C)c1C#N C1(CNC(c2scc(C)c2Br)=O)CN(C(c2[nH]cnc2C)=O)CCCO1 N(C1COc2ccccc21)C(C1C(CNC(=O)C=Cc2ccncc2)C1)=O N1(C(C(C)OCCC=C)=O)CCC(CO)C(NC(=O)CC2CC2)C1 Cc1cc2ncn(CC(C)Oc3ccc(Cl)cc3Cl)c2cc1C C(CN=C(NC1CCS(=O)(=O)C1)NC1CCCCCC1)OC1CC(OCCC)C1 C1(O)(CNC(Cc2c(C)noc2C)=O)CCN(C(=O)COC(F)F)CC1 CC(CN(C)C)CCC(=O)NC(C(=O)NOCC1CCC1)c1cccnc1 c1(C(=O)NC2CCCCC2CNC(c2ccc(Cl)nn2)=O)cc2c(s1)CCCC2 C1(C(=O)NC2(C)CC=CC2)CN(C(=O)Cc2cccnc2O)CCO1 N1(C(Cn2cc(-c3cccc(NC)c3)nn2)=O)CC=C(c2cc(C)cc(C)c2)CC1 n1(C2CCNC2=O)ccc([N+](=O)[O-])n1.C(=O)(C(F)(F)CC1CC1)NCCCCNC(=O)C N1(C(C(=O)NC2CCC(C(=O)OC)CC2)=O)CC2CCC(N(C)C)C2C1 N1(CCC)CCCC(C(=O)NCC(CCOC)NC(=O)COCC(C)C)C1 C(=O)(CN=c1cc(C)nc(N2CCC(Cc3nc(C)cs3)CC2)[nH]1)N(CC)CC C1(NC(CC2CC(C)(C)C2)=O)CN(C(=O)CCc2cnccn2)C2CC12 C=C1CC2CCCC(C1)N2C(=O)C(C1CCN(C(=O)C(CC)OC)CC1)C Cc1ncnc(C)c1C(=O)NCC1(C)CCCC1NC(c1ccc(F)s1)=O CC(C)CC(C(=O)NCCCC(C)(F)F)NC(=O)C(=O)C(C)C C(CCCCC(=O)N1CCC(C(CC)CC)C1)NC(CCSCCCC)=O CC1CCN(C(=O)CCc2cccc(F)c2Cl)CC1NC(C1CCCS1)=O C(C(CC(C)C)C(=O)Nc1n(C2CCN(C)CC2)ncc1)n1cccn1 O=C(C1Cc2c(Cl)cccc21)NCC12CC1CN(C(c1csc([N+](=O)[O-])c1)=O)C2 C1(NC(C2CCN(C(CC)=O)C2)=O)CC2(C1)CN(C(c1csc(Cl)c1)=O)C2 N1(C(CC2(C=C)CC2)=O)CCC(CCOC)(NC(=O)CCc2cc(C)no2)CC1 CC1CC(NCc2cnc(Cl)n2C)C(=O)N1c1cnn(C)c1 c1(C(=O)NCC2C(NC(C3C(C(=O)OC)CC3)=O)C2)ccc(F)cc1Cl c1(C(=O)NCC(CNC(C(C)(C2CC2)NC(C)=O)=O)F)cc(F)cc(Cl)c1 c1(C(N2CC3C(NC(C#C)=O)C3C2)=O)cccc(C(F)(F)F)c1C(=O)OC Cc1cc(NC(C2(C3CCCN3C(C3CC(O)C(F)C3)=O)CC2)=O)ccc1Cl C1(C#N)(C(=O)NCC(CC=C)NC(C2CC23CC(O)C3)=O)CCS(=O)(=O)CC1 c1(C(=O)NC(C2CCOC2)CNC(CSCCOC)=O)sc(C)nc1CC(C)C C(=O)(CCCCCCCBr)N1C(CC)CN(C(=O)CC#N)CC1 C1(C(=O)NC2CC(C)(NC(=O)COCCCOC)C2)(OC)CCCC(C)C1 c1(C(N2CC(CNC(c3cc(C)sc3C)=O)C(O)C2)=O)cnn2ccc(O)nc12 C(CCCCCC(=O)NCC(CC)(CC)C(N)=O)NC(CCSCCCC)=O C1(NC)CCC(NC(C(=O)C(=O)Cn2nnc(=O)[nH]2)=O)C1.CC(F)F N#Cc1c[nH]ccc1=NC(CNC(C1CC(c2ccccc2)C1)=O)CO C12(C(N(CC(C)C(C)(C)C)C)=O)COCC1CN(C(C1C3(CC3)C13CC3)=O)C2 Cc1cc(C(=O)N(CC(C)CNC(=O)CC(C)c2ccco2)C)c(C)o1 C1(N(CC(C)(C)O)C(C23CC(C(F)(F)F)(C2)C3)=O)CC2CC1CN2 Cc1oc(C(F)(F)F)nc1C(=O)NC(C)(C)CCN(C(=O)CCC1CCOC1)C C(CC(C(=O)NC(C)(CC)C(=O)OC)OC(C)=O)NC(C=CC(CC)=CC)=O CC(CCC(C)(C)C)C(=O)NCC(=O)NCCCC1CC(=O)C1(C)C Cc1noc(C)c1C(C)C(=O)N(C)CCNC(c1cc(Cl)nn1C)=O Cc1cc(C(N2CCC(NC(=O)CC34COC(C(F)(F)F)(C3)C4)C2)=O)nc(C)c1 Cc1ncnc(C)c1CC(=O)N(C)CCOCCCNC(=O)CC1CCOCC1 N1(C(CN(C)CC)=O)CCCC1(C(=O)NCCC(COC)OC)C(C)C C1(C(=O)NC2CC(C(=O)NCCC3CCCC3)C2)(CO)CCOC1 c1(C(N2C(CNC(=O)OC)CC2)=O)ccc2c(c1)COCC2 C(S(=O)(=O)c1ccccc1)c1c(NC(N2CC(C(=O)OC)C(OC)C2)=O)n[nH]c1 N1(C(C(C(C)(C)C)NC(N)=O)=O)CCCCCC(NC(=O)CN2CCSCC2)C1 c1(C(N2CC(C(=O)O)CC(OC)C2)=O)cc(F)c(F)cc1Cl c1(C(N(CCN(C(C23COCC2C3)=O)CC)CC)=O)cc(=O)c(OC)c[nH]1 Cn1cc(CC(C(=O)O)C(c2cnn(Cc3ccccc3)n2)=O)cn1 C(=O)(CCC(O)C(C)(C)C)NC(CNC(CCN1CCC(C)CC1)=O)C1CC1 c1(N2CCCC(NC(Cc3c(C)cccc3)=O)(CO)C2)ncnn2cccc12 CC1CC(NC(=O)CCNc2ccccc2O)CN1c1ncncc1I C1(C(=O)NC2CN(C(C(C)(C)F)=O)CC2O)C2CC(F)(F)CC12 C(CCC(C)C)(C(=O)NCC#CC(F)(F)F)NC(C(CCOC)C)=O c1(C(=O)NCC2CCN(C(C(CCC)CCC)=O)C2)cc2ccnc(Cl)c2[nH]1 c1(C(=O)NCC2(NC(c3nc(COC)sc3)=O)CCCC2)cc(OC)n(C)n1 C1(C(N(C)CC2CC2(C)C)=O)CC1C1CN(C(c2cccn2C)=O)C1 C=CCC(C)C(=O)N1CCC(N(C(=O)CCCn2cccn2)CC2CC2)CC1 C1(NC(c2csc(CNC(C34CC(C)(C3)C4)=O)n2)=O)CCN(C2CCC2)C1=O CCC(C(=O)NC1(C)CC(NC(=O)C(O)CC2CCCCC2)C1)NC(C)=O C1(CCNC(=O)CSC(F)(F)F)CCCN1C(C12CC(c3ccccc3)(C1)C2)=O C1(NCCC(=O)N(CC(C)C)C)CCC(N(C(=O)CN2CC(C)(C)C2)C)CC1 Cc1nc(C(N2CCCC23CCN(C(=O)CC2C=CCC2)C3)=O)c2ccccn12 C1(C(=O)NCCN(C(=O)C(CSC)OC)CC)CCNC(=O)C1 N1(C(CC(CC)O)=O)CCC(O)C(C(=O)Nc2ccc(O)cc2C(N)=O)C1 N1(C(C(OC)OC)=O)CCC2(CCC(NC(=O)Cc3ccc(F)c(Cl)c3)C2)CC1 C=C=CCCC(=O)NC(CSCC)C(N1CCCC1C=C)=O c1(CN2CC(CC(=O)Nc3cnc(OCC)nc3)C2)cccc(S(C)(=O)=O)c1 c1(N2CCC(C(=O)NC)CC2)ncnc(NCCSCc2ncc(C)cn2)c1C c1(-c2cc(C(F)(F)F)cc(C)c2)ccc(C#N)c(I)c1 Cc1cc(O)n2ncc(C(=O)NC3CC(CNC(C4CCN(C)CC4)=O)C3)c2n1 O=C(C(O)C1=CCCCC1)NC1CC(C(N2CCCC2CF)=O)C12CCC2 C1(CNC(=O)Cc2ccns2)COC(C(F)(F)F)CN1C(=O)C=Cc1cn[nH]c1 CC1(C)CCN(CCNC2CC3CC3C2)C1.n12ccc(c1)C(=O)NCC2C CCCCCC(C1CC1)NC(C1CCC1NC(C1(C)C=CCCC1)=O)=O Cc1c(Br)ccc2c1CCN(C(c1ccc3occc3n1)=O)C2 c1(NC(C(=O)NCC2CC2)=O)cc2cccn2c(O)n1.CC12CCN(C1)C2=O c1(OCOC)cc(F)c(-c2cccnc2C(N2CCC(OC)CC2)=O)cc1F c1(C(N2CCC(N(C(=O)CCCCCBr)C)C2)=O)ccc2ccncc2c1 C(=O)(C(C)(C)C(N)=O)N1CC(OCC)C(CNC(c2cccnn2)=O)C1 N1(C(c2c(OC)cnnc2)=O)CCOCC(C(=O)NC2CCCC(CO)C2)C1 C(=O)(C(C)(CC)CO)Nc1[nH]nc(-c2ccc(OCC)cc2)n1 c1(C(N2CCC(COC)CC2)=O)nc2ccccn2c1-c1cc(F)c(O)c(F)c1 Cc1cnc(C(=O)NC2(C)CCN(C(c3cc4c(s3)COCC4)=O)C2)cc1C#N C=C=CC(C)C(=O)NC(CNC(=O)CCOc1ccccc1OC)C1CC1 CC1CC(CNC(=O)C(C)N(C)C(c2cnnn2C)=O)=NO1 C12(C(N3CCN(CCNC(C(C)C4CCC4)=O)CC3)=O)CC3CC(C(=O)N1)C2C3 c1(C(N2CCC(C)N(C(C3COC(C)(C)C3)=O)CC2)=O)n[nH]c2c1CC(C)CC2 N=c1ccc(C(=O)NC23CC2CN(C(C2(C(F)F)CCOCC2)=O)C3)n[nH]1 C(CC(C)C(=O)NCC1CC(O)(CNC(=O)CNC(C)=O)C1)=CCC C1(NC(CC(=C)C)=O)CCCCC12CCN(C(=O)Cc1ccc3c(c1)CCC3)C2 c1(C(=O)NCC2C3CN(C(=O)CC4CSC4)CC23)ccc2cccc(Br)c2n1 C1(CNC(c2cnn(CCC)c2C)=O)(CO)CCN(C(C2CC2C2CCC2)=O)CC1 N1(C(Cc2c(C)ccs2)=O)CC2CCC2(C(=O)NCc2cc(C)sc2C)C1 N1(C(c2c(Br)ncc(C)c2)=O)CCC2CN(C(c3cccc4occc34)=O)CC12 C(=O)(CCN=C(NCC(c1ncc(C)s1)(C)C)NC1CN(C2CC2)CC1C)NC N1(C(C(CCCOC)C)=O)CCN(C(C2(c3ccno3)CCC2)=O)CC(O)C1 C1(CNC(Cc2ccc(C)nc2)=O)(NC(=O)C=C2CCCC2)CCC(F)(F)CC1 N1(C(C2C3N(C(C4C(C#N)CC4)=O)C(CC3)C2)=O)CCCC(O)(C2CC2)C1 CC1C(NC(=O)CCC(=O)N(C)C)CCCN1C(C12CCCN1CCC2)=O c1(COC)cccc(C2(OC)CCN(C3CC(OC)Cn4nnnc43)C2)c1.OC C(C(CNC(=O)CNC1CCC1)CO)NC(=O)COCC1CCCO1 C(=O)(C1=CC2(CCN(C(=O)C(CO)C(F)(F)F)C2)C1)NCC(CN(C)C)(C)O C(C(C)C(=O)NCC(C)(C)CC1CN(C(c2conc2C2CCCC2)=O)C1)OC CCCCCC(O)CC(=O)NCC(C)(CO)NC(c1cc(C#N)cs1)=O c1(CC(=O)NC2C(NC(C(C3CCC3)OCC)=O)COC2)cccc2sccc12 Cc1conc1C(N1CC(O)(C(F)C(=O)NC(CO)C2CC2)C1)=O CC1(C)NC(=O)CC1C(=O)NC1CCN(C(=O)CCc2ccc(Cl)s2)C1(C)C C1(C(N(C(C)CC(=O)NCCCc2nncs2)C)=O)CCCC(C)(C)C1 Cc1ccc(C(C)NC(=O)CC2CN(C(=O)C3=NOCC3)CC2C)cc1 FC1(F)CCC(n2nc(Cc3cccnc3)nc2-c2ccc(Br)cc2)C1 C1(C(=O)NCC(C)NC(c2cnc(OC)c(Cl)c2)=O)CC2(CCCC2)CO1 CC1(C)CCCN(C(c2cccnc2)=O)C1CNC(C1CC12CC2)=O N1(C(c2n(C)ccn2)=O)CCC(C(=O)Nc2nc(F)ccc2Br)C(O)C1 C1(COC(C(C(C)C)n2cnnn2)=O)CC(C)(C)CN1C(=O)OC(C)(C)C N1(C(COC2CCN(C(C(CC)C(C)C)=O)C2)=O)CCCCCCCC1 C1(CC(=O)NC2CC(NC(C(C)SC(C)C)=O)C2)CCCS(=O)(=O)C1 N1(C(CC(=C)I)=O)CC(CNC(=O)CC(C)OC)C(C)C1 C=CC(CC(=O)NC(C)(CNC(c1c(C)coc1C)=O)CO)c1ccccc1 c1(OC)cc(C)c(CONC(C2CC(Cc3ccnc(C)c3)C2)=O)c(C)c1 c1(C(=O)NC2CCCC(NC(CCc3n(C)cnc3)=O)C2)cc2ccncc2s1 Cc1oc(C)c(C(N2CCC(NC(=O)COCc3ccccn3)C2)=O)c1C n1(CC)cc(C(=O)NCC(C)(CO)NC(C23CC(F)(C2)C3)=O)c(C(F)(F)F)n1 CC#CCCCC(=O)N(CCCNC(C1COCCN1C(C)=O)=O)C1CC1 CCC(CC(=O)N(C)CCN(C)Cc1cccc(C(C)C)c1)C1CCC1 c1(COC)nc(NCc2nccn2C)cc(=NC2CC(n3cncn3)C2)[nH]1 C(C1=CCN(C(c2ncc(N(C)C)cn2)=O)CC1)NC(C(CC)NC(C)=O)=O C(=O)(C1=CNC2=NCCC2=C1)N1C(C2CCN(C(=O)Cn3cnnc3O)C2)CCC1 CC1CC(C(=O)NC(C2CCN(C(C3OCCO3)=O)CC2)CO)CC(C)C1 Cc1[nH]nc(C(=O)NCC2C3CC2N(C(C2CC2C(F)(F)F)=O)C3)c1Cl c1(NC(C2(F)CCN(Cc3c(OCC)cccc3Cl)C2)=O)ncnc2occc12 C(=O)(C(O)CCC(F)(F)F)N1CC2(CC(NC(=O)Cn3cnnn3)C2)C1 C1(CC)CC(CC(=O)NCCCCNC(C2CC(F)(F)C2)=O)CCO1 Cc1cccc(Br)c1Oc1ccc(C(N2CCCC2C(=O)NCCF)=O)cc1 CC1c2c(ccc(F)c2Cl)CCCN1C(c1cnc2ccsc2c1)=O c1(NC(CCN(CC=C)C(c2cnc(OC)nc2)=O)=O)cnc2c(c1)CCC2 CC(=O)CCC(=O)N1CCCC1C=CC(=O)NC1CC(N2CCCC2)C1 C1(C(=O)NCCOC2CN(C(CCCC=C)=O)C2)CS(=O)(=O)CC12CCC2 c1(C(c2nnnn2CCC2CC2)NC(CC)C(C)C)cccc(O)c1 c1(N(CCC)CC)ccc(C(N2CC(CCNC(=O)CS(C)(=O)=O)C2)=O)cn1 Cc1c(C(N2CCC(NC(=O)C(C)C3CCCO3)C2(C)C)=O)cnc2nncn12 C1(NC(C(CC=C)C)=O)CC2CN(C(c3ncoc3-c3ccon3)=O)CC12 c1(OC)ccc2c(c1)C(C(=O)N(C)CCn1ccnc1)C(C)N2 CC(CCC(=O)NCc1ccc(CNC(C2(C#N)CCC2)=O)cc1)N(C)C C=CC1(C(=O)NCC(C)(C2CC2)NC(=O)C#CC(=O)N(C)C)CCCCC1 c1(CNC(c2cccnc2)CC)ccccc1SCC(C)C#N CCCC(CNC(c1ncncc1C)=O)C(=O)NC1CC(Cl)(Cl)C1 c1(CCC(=O)NCC2(C(F)(F)F)CC(F)C2)ccc(Br)cc1[N+](=O)[O-] C1(C(C)N)CN(N2CCC(COc3cccc(F)c3)CC2)CCO1 Cc1n[nH]c(C)c1C(c1nnnn1-c1ccccc1)NCC1(CCO)CC1 N(C(=NCCSCC)NCC1(F)CC1)CC(=C)Cl c1(NCCc2ccc(OC)cc2)cc(S(=O)(=O)N(CC(C)C)CC)ccc1C#N C=CC1(C(=O)NCCC2(O)CCOC2)CCN(C(=O)CCc2nccs2)C1 C1(CNC(c2c(C)onc2)=O)C(C)CCN1C(C1COC(C)(C)C1)=O C(=O)(CCS(N)(=O)=O)NC(CCNC(c1nc(C(C)OC)sc1)=O)(C)C c1(CN2CCC(NC(c3cc4cccnn4n3)=O)CC2)c[nH]c2ccc(Br)cc12 Cc1sc(O)nc1C(=O)NCC1(F)CCN(C(C2CCN(C)C2)=O)C1 C1(NC(C=C2CCN(C)C2)=O)CCCC(NC(=O)CN2CC(C)(C)C2)CC1 NC1C(=S)N(C2CCN(S(=O)(=O)CCO)C2)C1 C(=O)(C1=COCCC1)N1CCCC(C)(NC(C(C(C)C)c2ccncc2)=O)C1 C1(NC(c2cc(OC)c(O)cc2)=O)CN(C(c2cc(C)n(C)n2)=O)CC(C)(C)C1 N1(C(C(C)Cc2cnco2)=O)CCC2(CC1)CC2NC(C1CCCN1N=O)=O N1(C(C(CC)=CC)=O)CCC(C)C(N(C)C(c2ncc(OC)cn2)=O)C1 CCCC(O)C(CO)NC(C1CC2CCC1N2C(=O)CCCC1CC1)=O c1(C(N(CC(C)CNC(C2CSCCS2)=O)C)=O)cncc(N)n1 c1(C(N2CCC(=CCNC(C(C)SC)=O)CC2)=O)c(Cl)cc(Cl)nc1N c1(C(N(CCCCNC(=O)C(O)c2ccco2)C)=O)ccccc1Br C1(C(=O)OC)CCCC(n2cc(C3CCN3C(c3cnn(C)c3C)=O)nn2)C1 c1(C(=O)OC)cccc(NNC(=O)NC2CCn3c(C)cnc3C2)c1C C1(CNC(C(c2scc(C)n2)C)=O)CCN(C(C2(C3CCCO3)CC2)=O)C12CCC2 c1(CNC(CSCC2ON=C(C)C2)=O)nc(C)cc(C(F)(F)F)c1C#N Cc1ccn(CC(C)C(=O)NC2CCC(NC(c3ccn(C)n3)=O)C2)n1 C1(C(=O)NCC(CC)NC(c2c[nH]nc2C2CCCO2)=O)CCC(=O)N1 CC1CN(C(C2C3CN(C(C4(C)CCNC4=O)=O)CC23)=O)CC(C)N1C C(=O)(C#CC1CCCCC1)NCC(C(N1CCC(C(C)C#N)CC1)=O)(C)C N1(C(CCC(=O)NCC)=O)CCCC2(CNC(c3cc(C(=O)OC)no3)=O)CC12 C1(C2CCCC2)(C(=O)NCC(C)NC(=O)C(O)CC2CC2)CCNC1=O N(C1CN(C(c2cnn(C(C)(C)C)c2)=O)Cc2ccccc21)C(CC(C)(F)F)=O C12(CCN(C(CCSCCCN)=O)C(C)C)COC(C1)C2 N1(C(c2c(C)nc(C)s2)=O)CC2(CC(NC(c3ccc(Cl)c(C)c3)=O)CO2)C1 C1(NC(CCC=C)=O)CN(C(c2cc(C#N)ccc2Cl)=O)CC1S(C)(=O)=O C(=O)(C(CC1CCC1)NC(C1CC1C(C)(C)C)=O)NCCSC C1(O)(CN(C(=O)CNC(C2CC(c3ccccc3)O2)=O)C)CNC1 C1(CNC(C(=O)NCC)=O)CN(C(=O)Cn2nc(C)c(C)c2C)CC2(CCC2)O1 c1(CC)cc(C(=O)NCC2CCC2C(=O)N(CC(C)(C)CO)C)ncn1 N1(C(CC(=O)NCC#C)=O)CCN(C(=O)C(C(C)(C)C)NC(C)=O)C2CCC12 N1(C(C(CC)=CCCC)=O)CC(C(=O)NCC2(C(C)(C)O)CC2)CC12CCC2 C1(NC(C(C)OC)=O)C2CCC1CN(C(c1ccc3c(c1)OCO3)=O)C2 c1(CC)c(C(=O)NCC(CNC(c2cn(CC(O)CC)nn2)=O)OC)nnn1C N1(C2(C(=O)NC(C3CN(C(=O)Cn4cnnc4)C3)C)CCC2)CCOCC1 C1(C(N2C(C)CC(CNC(=O)CCC3NC(=O)NC3=O)C2)=O)CCCC(=O)N1C N#CC1CN(Cc2ccc(I)c(O)c2)CCN1C(C1CC1c1ccc(F)cc1)=O n1(CC(=O)N(CC(C)O)CCNC(COCC(=C)C)=O)cnc(C(N)=O)n1 C1(C)(CN(C(=O)CCc2cnoc2)C)CCCC1NC(=O)C(O)CCC1CC1 N1(C(CC2N(C(COCCCOC)=O)CC(O)C2)=O)Cc2ccnn2CC1C N1(CC)CCC(C(N2CC3C(C(=O)NCC4CC4)C3C2)=O)CC1 C1(C(=O)NC(CCSC)C(=O)O)CC12CCN(C(C1CC13CCC3)=O)CC2 Cc1cc(S(=O)(=O)O)c(NC(=O)CC2COCCN2C(=O)C(C)C2CC2)cc1Cl CC(C(=O)NCCN(C(c1ccn(C(C)(C)C)n1)=O)C1CC1)S(C)(=O)=O N1(C(C(CC=C)CC)=O)CC(C(=O)NCC(=O)OC)CC(C)(C)C1.C1CC1 c1(C(=O)NCC)ccc2c(F)cc(F)cc2n1.C1(=O)C(C(C)C)O1 N1(C(c2ccnc(OC)c2F)=O)CC2CN(C(=O)CCCN(C)C(C)C)CC2C1 N1(C(C(C2CCN(C(C(C)c3cccs3)=O)CC2)C)=O)CCC(F)(F)C(O)C1 N1(C(C2C(C(=O)OC)C=C2)=O)CCC(C(C)NC(=O)C(C)SC(C)C)CC1 c1(CCN=C(NC(c2cccs2)C)NCCS(C)(=O)=O)cccc2ccccc12 C(=O)(C#CC1CCCO1)N1CC(CNC(c2nncc(CCC)c2)=O)CC1(C)C C#CC1CCC(C(N2CCC(NC(c3[nH]c(C)nc3CC)=O)C(O)C2)=O)CC1 c1(C(N2CCCC(c3cn(CCN(S(C)(=O)=O)C)nn3)C2)=O)occ2c1CCC2 N1(C(C(C)=CCOC)=O)CCCCC(NC(=O)CCc2ccc(OC)cc2)C1 n1(CCOC)cc(C(=O)NCC2CC(NC(C3CCOC3CC)=O)C2)ccc1=O c1(C(=O)NC(CNC(CN(S(CC)(=O)=O)C)=O)C)ccc2c(c1)NC(=O)CCC2 c1(OC)cc(C(N2CC(CNC(=O)C(C)C(F)F)C(C)C2)=O)cc(Cl)c1 C1(C(C)C)CN(C(c2coc(C(N)=O)c2)=O)CC1C(N1CCCC(CCO)C1)=O c1(CC2CN(C(C3CC34CC4CN3C(=O)NCC3)=O)C2)cccc(F)c1 c1(OCCOC(c2ccc(OCCc3nn[nH]n3)cc2)=O)cccc(F)c1F N(C1CN(C(=O)C(O)C2CC2)CCc2ccccc21)C(=O)CC1CCCOC1 C1(NC(c2cccc(CC)n2)=O)CC2CC1CN(C(=O)Cc1cnn(CC)c1)C2 Cc1n[nH]c(C)c1C(C)C(N1CCCC1CCCNC(=O)CCCCF)=O c1(NC(=O)NCCCC2CCC2)ccc2[nH]c3ccccc3c2c1 N(C(=NCCC(=O)N(C)C)NCC1CCCCN1C(=O)NCCF)C(C=C)C c1(C(N2CCC(NC(c3n(C)cc(Br)n3)=O)C2)=O)cc2ncccc2[nH]1 c1(C(N(CCNC(c2cc(C)c(CO)cn2)=O)C)=O)cc([N+](=O)[O-])c(O)cc1N C1(C(=O)NC2C3CCN(C(C(c4cccc(C)c4)=O)=O)C32)CCCC(C)(C)O1 c1(C(=O)NC2(CF)CN(C(c3c(C)scn3)=O)C2)noc(C2CC2)c1C c1(C(=O)NC2CN(C(CCCCSC)=O)CC2C)cc(O)nc2ccccc12 C(C1=CCN(C(C23CC(F)C2C3)=O)CC1)NC(C1(C)CC(C)C1)=O c1(OC)cnc(F)cc1C(=O)NCCC1CCN(C(=O)C(C)(C)C(C)O)C1 C1(C)(C(=O)NCC(C2CCC2)NC(c2c(CC)[nH]cc2)=O)CCCCNC1=O c1(C(=O)OC)ccc2c(c1)CCC2NCCC(N1CCN(C)CC1)=O c1(CC)cc(Cl)ccc1C(=O)NC(C1CCOC1)CNC(c1coc(O)n1)=O N1(C(C(CC=C)(C)C)=O)CC2(C1)OC1(CO)CC2(NC(C2CC3C=CC2C3)=O)C1 C1(C(=O)NC(CNC(C(C)=C(CC)C)=O)C(C)(C)C)CC2(C1)CC21CC1 C1(NC(C2CCSC2)=O)CC2(CCCCN2C(=O)CSc2cccs2)C1 C1(C(=O)N(C)CCOCCOCCOC)(CC)CCC(F)(F)CC1 Cc1ccc(C)c(NC(=O)CC2CCCN(C(C3CC3c3ccoc3)=O)CC2)c1 C1(NC(C=CC=CC)=O)C2CC1N(C(C13CC(c4ccccc4)C1C3)=O)C2 C1(C#N)(CC(=O)NC(CNC(CC(C)c2ccco2)=O)C(C)(C)C)CCCCC1 c1(C(=O)NCC2(F)CC(NC(CC3(C)OCCO3)=O)C2)cnc2sccc2c1 Cc1nc(O)nc(O)c1CC(=O)NCC1CN(CC#Cc2ccccc2)C1 N1(C(CCc2ccc(C)o2)=O)CCC2CC(NC(C3(C(F)F)CC3)=O)CCC2C1 N1(C(c2[nH]cc(CC)n2)=O)CCC(O)(C(C)NC(=O)C=C(C)C)C1 C(=O)(C1=NNC(=O)CC1)NCC(CO)NC(C(C)c1ncco1)=O [N-]=[N+]=NC(CCC(N)=O)C(=O)NC1C=CCN(C(c2cc(C3CCC3)no2)=O)C1 C(C)(CCCCCO)NC(c1c(CNC(c2c(C)nsc2N)=O)n[nH]c1)=O n1(CC#C)cc(NC(=O)C(C)N(C(=O)C(C)OC2CCCC2)C)cn1 C1(C(=O)NCc2c(C)csc2)CN(C(C2CCC(=O)N(C)C2)=O)C(C)(C)C1 CC1CC=CCC1C(N1CCC(CCNC(C2CN(C3CCOCC3)C2)=O)C1)=O N1(C(C(C)C2CCCC2)=O)CCC(NC(c2nnc(O)nc2O)=O)C(CO)CC1 C1(NC(C(COCC)NC(=O)C(C)C#N)=O)CCC(=O)NC1C c1(C(N2CCC(C)(CCNC(C(CC)NC(N)=O)=O)C2)=O)cc(F)c(C)cc1N c1(C(N(CC(CO)(CO)NC(C2CCC(F)(F)C2)=O)C)=O)c(F)ccc(F)c1F C1(C(N(CC(CC)NC(C2(n3cc(Cl)cn3)CC2)=O)C)=O)CC=C(C)CC1 Cc1nc(O)[nH]c1C(=O)NC(CNC(=O)CN(c1cnccn1)C)CO C#CCC(C)(C(=O)NCC1CCCN(C)C1=O)NC(c1coc(CCC)n1)=O N1(C(c2nc(C(C)OC)sc2)=O)CC(CNC(=O)C=Cc2cscn2)C(C)(C)C1 C1(NC(CS(CCCC)(=O)=O)=O)CC2CCC(C1C)N2C(c1ccsn1)=O C(CCCC)(C1=CC=NSC(CC)(C)CC(=O)NCCOCCN(C)C(=O)C1)CC c1(C(=O)NCC(CC)(C)NC(C2CCC2C#N)=O)cc2cccnc2[nH]1 c1(C(=O)NCCOC2CCN(C(C=C(COC)C)=O)C2)cc(C)c(F)cc1F c1(C(=O)OCC)cc2c(Br)c(Nc3ncccc3F)ccc2s1 Cc1nsc(C)c1OCCNC(c1ccncc1)c1nnnn1C1CCOCC1 N1(C(C(C=C)(C)CC)=O)CC2(C=C(C(=O)NC3CC3(C)C)CO2)C1 N1(C(c2c(C)c(Cl)c(Cl)s2)=O)CCCC2(CC(NC(c3ccncn3)=O)C2)C1 C(=O)(C(=O)N=S(C)(C)=O)N1C(CCNC(c2nn(C)c(=O)cc2)=O)CCCC1 CN1CC(C(=O)NCC2(C)CCCN2C(c2cc(Br)no2)=O)NC1=O c1(C(=O)NCCC2ON=C(C)C2)[nH]c2ccc(F)cc2c1Cl c1(CNC(N(CC)CC2(C)CC(F)C2)=O)ccc(N(C)C)cc1 Cc1c[nH]c(C#N)nc1=NCCC1CCCN(C(c2cnn(CC(F)F)c2)=O)C1 c1(C(=O)NCC(CN2CCCC(C)C2)O)cc2cn[nH]c2cc1O c1(C(=O)NC2CC(C)(CNC(CSCC)=O)C2)cccn(C(C)(C)C)c1=O c1(C(N2CC(C(N3CC(N4CC(F)C4)C3)=O)(CC)C2)=O)ccc(C)cc1O N1(C(C=COCC)=O)CCCN(C(c2cnns2)=O)C(C(C)C)C1 c1(C(C(=O)NCc2ccccc2)N(CC#CC)C2CC2)ccccc1Cl C1(F)(NC(C(C)SC)=O)CCCN(C(=O)Cc2cccc(N(S(C)(=O)=O)CCC)c2)C1 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(CCC(C)OC)=O)C(O)C(O)C1 CCC(CC)C(=O)NC1CCN(C(c2cc(OCC(F)F)ccn2)=O)CC1 C1(CNC(C2(C#C)CCCC2)=O)CCCCN(C(=O)C(C)C(F)(F)F)C1 c1(C(=O)NCC=C)ccc(CC(=O)N(C2CCN(C(C3CC3C#N)=O)C2)C)cc1 C1(NC(CC)=O)COC2(C1)CN(C(C1CCCC3(CC3)C1)=O)C2 c1(CCC(=O)NC(C(CO)NC(CN(C)CC)=O)C)nc2ccccc2o1 C(=O)(CCCCC(=O)N(C)C)NC(CC(C)C)CNC(c1cn(C)c(O)n1)=O c1(C(N2CCC(OC)(OC)CC2)C(=O)N(C(=O)C(C)C)CC)ccc2nsnc2c1 c1(C(=O)NC(CNC(C(CC)C2CCOCC2)=O)CC)ccc(Br)cc1N c1(CCC(=O)NCC23CC2CN(C(C2(CS(N)(=O)=O)COC2)=O)C3)ccccc1O Cc1cc(Br)ccc1N(C)CC=CCC(CN1CCOCC1)CC.c1(=O)c(=O)[nH]1 C(CCC(=O)N=c1ccn(C2CC2)[nH]1)NC(CCCCCCC=C)=O CN=c1nc(N2CC3CC2(c2ccccc2)C3)[nH]c(=NCC(C)(C)S(C)(=O)=O)[nH]1 c1(C(=O)NCCCNC(c2c(C)cc[nH]2)=O)cnn(C(C)C)c1Br C1(NC(Cc2ncc(C)o2)=O)CC(F)CN(C(c2ccc(-c3cc[nH]n3)s2)=O)C1 Cc1[nH]ccc1S(=O)(=O)N1CCCC1C=Cc1cccs1 C1(C)(NC(C(CNC(c2c(CC)nns2)=O)OC)=O)CCC(C)=C(C)C1 C(CC(C(=O)N1CCC(CF)C1)NC(=O)COc1cnn(C)c1)=CC N1(CCCN(C(CC(=C)Br)=O)C)CCN(CC)CC1 Cc1csc(=NCC(=O)NC2(CNC(C3CC4COCC4C3)=O)CCOC2)[nH]1 C1(C(=O)NCC(CNC(C2(CO)CC(C)(C)C2)=O)(C)F)CN2CCCN1CC2 CCC(CNC(=O)CCN(C)CC)NC(=O)C(C)c1cccs1 Cc1cnc(C(N2CCCCC2CCCNC(=O)CCN(S(C)(=O)=O)C)=O)cn1 C1(CNC(C2CC(OC)C2)=O)CCCCN(C(C2(C)CCCC2C)=O)C1 C1(C(=O)NC2C(C)CN(C)CC2)C(C2CC2)CCN1C(c1ccccc1)=O N1(C(Cc2c(C)nccc2)=O)CC2CC1CN2C(c1n[nH]c(C)c1F)=O c1(N2CC3CN(CCOC)CC3C2)ccc(S(=O)(=O)NCc2ccsc2)cn1 c1(C(C(=O)NCC(C)N(C(=O)Cn2cncn2)CC)SC)ccccc1 N1(C(C(CC)C2COC2)=O)CCCN(C(c2cnc(Br)s2)=O)CC1C c1(-c2n(C(C)C(F)(F)F)nc(Cn3cccn3)n2)cnc2ccccn12 CCC(CC)CN=C(NCc1ccc(F)cc1)N1CC2C(C1)C2(C)C c1(NC(C2CC(C)(NC(C(CC=C)C)=O)C2)=O)ccc(N(C)C)cc1C c1(C(N2CC(c3cn(Cc4cccnc4)nn3)C2)=O)sccc1Cl C1(C(N2CC(NC(c3sccc3C)=O)C2)=O)(OCC)CCOC1 N1(C(C(COC)NC(C)=O)=O)C(CC(=O)NC2CCOC2)C2CCCC12 C(=O)(C(CCS(C)=O)N(C)C)NC1C(NC(C(F)=C(C)C)=O)CCOC1 C1(CNC(C=CCC)=O)CC2(CCN(C(C3CC3c3nccn3C)=O)CC2)CO1 C1(C(=O)NCC2N(C(CCNC(COC)=O)=O)CC(C)(C)C2)CCC(C)C(C)C1 c1(C(=O)NC2CC(CNC(CN(C)CC)=O)C2)noc2c1CC(C)(C)CC2 C(=O)(CCCCCNC(=O)C1CC1)NCCC1OCC(C)(C)C1 C1(NC(C2CCCN(C)C2)=O)CN(C(=O)CSc2ncccn2)CC(F)(F)C1 CC(C)C(O)C(=O)NCC1CC(NC(c2ccn(C)c2)=O)C1 c1(C(N2CCC(N(C(C(C3CCCC3)OC)=O)CCO)C2)=O)cc(C)nn1C c1(NC(C(c2ccc(F)c(C)c2F)N2CCC(SC)C2)=O)ccc2c(c1)OCO2 CCC(C)C(O)C(=O)NC1CC2CC1N(C(=O)C(c1ccccc1F)(C)OC)C2 c1(C(C(=O)NC(CC)CN(C)C(C2CC(OC)C2)=O)OC)cccnc1 N1(C(C(C)OCC#C)=O)CCC(C(=O)NCCOCCF)C1 C(=O)(C1=C(F)CN(C(=O)CC2CCCC3CC23)CC1)NC1(C)CCCC1 C1(C(C)C)CN(C(c2cccn2C)=O)CCCN1C(c1cc(C2CCC2)n[nH]1)=O C1(C)(CCC(=O)NC2CC(CC)C2)CCCN1C(=O)C(C)C(=O)OC c1(NC(=O)C=CC(=O)NC2(CNC(=O)C(Cl)(Cl)Cl)COC2)cc(F)cc(Cl)c1 c1(SC)ccc(Cl)c(C(N2CCN(C(C3CCCC3(C)C)=O)CC2C2CC2)=O)c1 C(S(C)(=O)=NC(=O)CCOCC1CCCC1)c1cccc(C)n1 C(=O)(C(C)CCNC(=O)CC=C(Cl)Cl)NC(c1cn[nH]c1)C N1(C(c2c(COC)cco2)=O)CCC2CC(C(N3CCC3C(C)C)=O)C2C1 c1(C(N(C2C3CN(C(CC(CC)C(F)F)=O)CC32)C)=O)ccc2oc(O)nc2c1 Cc1ccc(F)c(CN2CCC(C(=O)Nc3cc(N(C)C)cc(Cl)c3)C(F)C2)c1 C1(N(CC(=O)OC)C(c2ccc(C)s2)=O)CCN(C(=O)C(C)Oc2ccccc2)C1 N1(Cc2n(C)ncc2)CC2CC1CN2C(C1CCC(c2ccccc2)O1)=O Cc1[nH]c(C2CCN(C(=O)C3CC3)CC2)cc1C(N1CCC12CCC2)=O C(CN=c1[nH]c2c(c(=NC3CC=C(C)CC3)[nH]1)CCCCC2)N(CCC)C c1(C(=O)NCCCOCCNC(c2c(C)n[nH]c2C)=O)coc2c(F)cccc12 C1(NC(C2(c3ccc(N(C)C)cc3)CC2)=O)CC2CC1N(C(=O)C(O)CF)C2 Cc1cc(C(N2CCCC2C(=O)NCCC(=O)N(C)C2CC2)=O)cc(O)n1 c1(C(N2C(CNC(CN(C)CC)=O)CC2)=O)cnc(N2CCOCC2)s1 c1(C(N2CC(O)CC(NC(C(CC)C#N)=O)C2)=O)cnn2cc(Br)cnc12 c1(C(C(C)NC(=O)CC(C)C2CC2)NC(=O)C(C)(C)C)cccc([N+](=O)[O-])c1 C1(NC(COC(CC)CC)=O)CCN(C(C2(CC(C)C)CC2)=O)CCC1CO C#Cc1cccc(C(c2nnnn2CCCC2CC2)Nc2c(C)cccc2)n1 n1(CC(N2CCC(NC(C3CCC(C)(O)CC3)=O)C2)=O)nnc2ccccc12 N1(C(CCCCSC)=O)CCCCC2(CCN(C(=O)C(C)(C)CS(N)(=O)=O)C2)C1 C(C(=O)N1CC(NC(c2snc(O)c2Cl)=O)C1)(C(C)C)NC(C)=O CCCCCCC(CC)C(=O)NCC1CCCN1C(c1ccc(C)[nH]1)=O c1(N(C)Cc2c(C)nsc2)nc(NCC2CCC(=O)NC2)c2ccsc2n1 N1(C(C=CCCC)=O)C2CCC(C(N3CCCC3CN3CCCC3)=O)C1CC2 N1(C(C=Cc2n(C)ccc2)=O)CC=C(CCNC(=O)CC2CCCS2(=O)=O)CC1 N1(C(CC(=O)NCC#C)=O)CC(C)(C)c2ncc(-c3cc(C)cnc3OC)cc21 C1(N(N2CCCC(O)C2)C)CC(c2nn[nH]n2)N(C=O)C1.C(C)(C)(C)OC=O C1(C(=O)NCC(C)(C)NC(c2ccnc(OC)c2Br)=O)CCCCN(C)C1=O C=CCN=c1[nH]c(C(=O)NC2(CNC(=O)CCC(C)(C)O)CCOCC2)cs1 c1(-c2c(OC)ncc(C)c2)c(C(=O)NCC2COC2)nn2c1CCCC2 CCCS(=O)(=O)CC(=O)N1CC(C(C)NC(c2cnn(C)c2C)=O)C1 N1(C(C2CC(N(C)C)C2)=O)CCCC1C(C)(C)NC(C1(Cc2ccccc2)CC1)=O C(C)(CO)(C(=O)N1CC2CC1C2NC(C1CCCC1c1cnn(C)c1)=O)OC Cc1nc2ccc(C(=O)NCCC(C)N(C(=O)CN(C)C3CC3)C)cc2[nH]1 C1(C)(C(=O)NCC(C)NC(C2CCC(C)CC2)=O)CCOC(C)C1 C(C(=O)N=c1cc2ccccn2[nH]1)(C1(O)CCC1)NC(CCP(C)(C)=O)=O c1(C(N2CCC(NCC3CC3)C2)=O)cccc(S(=O)(=O)N(CCC#N)C2CC2)c1 C1(C(=O)NCCN(C(=O)COc2ccccc2)C2CC2)CC(=O)C12CCC2 N1(C(CCSCCCC)=O)CC(CC(=O)NC(c2cccnc2)C)CC1(C)C C(=O)(CS(=O)(=O)C1CC1)N(CCC(C(C)(C)C)NC(c1c(C)cncn1)=O)C N1(C(C2(CCNC(=O)C3=CCOCC3)CC2)=O)CC2CCC(C1)C(O)C2O C1(C(=O)NC2(C(=O)NCC3CCCCO3)C(C)(C)C2)CCOC(=O)CC1 CC(=O)CCC(=O)NC(c1nocc1C(=O)NC1CCC2CC12)C N1(C(c2c(C)nco2)=O)CC2(CO)CC1(C(=O)NC(c1ccc(F)cc1)C)C2 c1(OC)cc(F)ccc1C(=O)NCCCCN(C)C(C1CC1Cl)=O Cc1nn2ncccc2c1C(=O)N(CC(C)(C)NC(=O)CC1CCC2CC12)C N1(C(Cc2ccc(C#C)cc2)=O)CC2(CCC(C(N3CCC(F)(CO)C3)=O)O2)C1 CON(CCC(=O)N1CC(C)CC(C)C1)C(=O)c1cnnn1C1CC1 CC(C)CC(F)C(=O)NC(C)CNC(c1ccccc1-n1ccnn1)=O C(CC(COC)N1CC(C(c2ccccc2)O)(OC)C1)OC c1(C(=O)NC(C2CCOC2)CNC(CCOCC)=O)cc2cc(Cl)c(Cl)cc2[nH]1 C(=O)(N=c1cc(C(F)(F)F)n(C)[nH]1)NCCC(N1CCN(C)CC1)C c1(OC)nn(C)cc1C(=O)N(C)CC1(O)CN(C(c2ccnn2C)=O)C1 c1(SC)ncc(Cl)c(C(=O)NCC2(F)CCN(C(c3cccnn3)=O)C2)n1 C(=O)(n1c(-c2cccc(C(=O)O)c2)nc2ccccc12)NCc1c(CC)c[nH]n1 C1(C(=O)NCC(F)CO)CCCC12CCN(C(c1ccc(O)c(I)c1)=O)C2 C1(C(N2CCC(C(C#C)C)CC2)=O)CN(C(=O)CC2(COC)CC2)CCC1(C)C C(=O)(C(C)(C)CCC#N)NC1(CNC(c2ccc(C(C)C)nc2)=O)CCOC1 C1(CC)CN(C(=O)C=Cc2cnn(C)c2C)CCC1NC(=O)Cc1csc(Cl)c1 c1(-c2cn(C3CC4N(C(CC(C)C)=O)C(CC4)C3)nn2)c(Cl)cccc1[N+](=O)[O-] C1(C(=O)NCc2nccc(C(N(C3C(C)C3)C)=O)c2)CC2(CC(=O)C2)C1 CC1CCN(C(c2cnc(C#N)s2)=O)CC1CNC(=O)Cc1ccnc(F)c1F C1(NC(c2nc(OC)c(F)cn2)=O)(CNC(=O)C(C)CF)CC2CCC1CC2 Cc1ccc(C(N2CCCC2CNC(c2ccnn2CC(F)F)=O)=O)cc1N c1(CCNCCC=C)[nH]c(=NCCC(C)(C)OC)nc2c1ncn2C(C)C S(=O)(=O)(c1ccc(NCC2CN(C3CC3)C2)c(Br)c1)NCCN(S(C)(=O)=O)C c1(CC)occ(C)c1C(=O)NC1CC(C(N2CC(CC(=O)OC)C2)=O)CC1O N1(C(C(C)(C)OC)=O)CCCC(N2CCC(NC(=O)COC(N3CCCC3)=O)C2)C1 C1(NC(C(CC)C)=O)CN(C(c2csc(NC(C)=O)n2)=O)CC(C)(C)C1 N1(CC(=O)NC2(CCNC(C(F)=CCC)=O)CCC2)C(C)CCC1C c1(CNC(CN(CCC)C(c2ccnc(NC)c2)=O)=O)nc(CN)cc(O)n1 N1(C(COCCC)=O)CC2CC(NC(=O)Cc3cc(Cl)ccc3Cl)CC1C2 c1(OC)ccc(S(C)(=O)=O)cc1C(=O)NC1CCN(C(=O)CCCCl)CC(O)C1 c1(N2CCC(N(CCC)C(C3CCCO3)=O)C2)nc(C)cc(C)c1C(=O)OC C1(CC)C(NC(=O)CCc2cccnc2)CCN1C(c1coc(Cl)c1)=O N1(C(CC(=O)NCC(F)(F)F)=O)CCC(O)(CNC(c2ccc(=O)oc2)=O)C1 Cc1cnn(C)c1C(=O)NCC(CO)NC(=O)CC12COC(C(F)(F)F)(C1)C2 c1(COC)cccc(C(=O)NC2CC(CNC(C3(C)C=CCCC3)=O)C2)n1 c1(CCC(=O)NC2CCN(C(c3cn[nH]c3)=O)C2)ncc(-c2ccccc2)o1 N1(C(C(CC#C)(C)C)=O)CC(NC(=O)CC2CCCOCC2)C(S(C)(=O)=O)C1 Cc1c(NC(C2CC3CSCC(C2)C3)=O)cccc1N=[N+]=[N-] C(=O)(CCCCC(C)(C)C)N1CC(C2(NC(Cc3n(C)ccn3)=O)CC2)C1 N1(CCNC(C(NS(N(C)CC)(=O)=O)=O)=O)CC2C3C=CC(O3)C2C1 c1(C(=O)NC2C(CNC(C(C)OCCCCCC)=O)CC2)nc(Cl)c(CC)[nH]1 N1(C(Cc2cccc(SCC)c2)=O)CCN(C(=O)CC2CC(=O)C2)CC1CCO c1(C(N2C(CNC(c3ccc(CCC)[nH]3)=O)CCC2)=O)cccc(F)c1C(C)C C1(C(=O)NCC(CC)(C)NC(=O)COCCC2CCCC2)CC2(CCC2)C1 c1(CNC(C2CC(F)C2)=O)nc2c(s1)CCN(C(=O)CCCF)C2 CC1(C)CC(C(=O)NCC2CN(CCN)C2)CN1C(c1cc(C(F)F)no1)=O c1(CC2(C(N3CC(NC(C4CCCO4)=O)C3)=O)CC2)ccccc1 c1(OC)cc(C(N2CCOCC2CNC(=O)C=CCF)=O)nc(Br)c1 C(=O)(C(C(C)(C)O)NC(=O)C(=Cc1ccco1)C)N1CCC(CSC)C1 c1(C(=O)NC2(C)CCN(C(c3cnc(C(C)(C)C)o3)=O)C2)cccc2cncn12 N1(C(c2n(C)ncc2-c2cnsc2)=O)C(CN)CC2CCCC12 C#CCC(CC(F)F)C(=O)NCCC1COCCN1C(=O)CCOC Cc1csc2c(NC(N3CC4CCC(CN(C)C)(C4)C3)=O)cccc12 c1(C(=O)NCC2C3CN(C(c4c(C)cccc4)=O)CC32)cccc2c1OCC2C c1(C(N2CCC(N(CCC)C(c3ccn(CC#N)n3)=O)C2)=O)cnn(C)c1Cl c1(CCN(c2cccc(Cl)c2)C(C2CN(C)CCO2)C)ccc(F)cc1Br N1(C(COCCOCC#C)=O)CCCC(F)(NC(c2ccc(OCC)nc2)=O)C1 CCCC(C)CC(=O)N1CC(C)(CCC(=O)NC(CCO)C(F)(F)F)C1 C1(NC(c2c(CC)cccn2)=O)CC2(C1)CC(CNC(c1coc(C)c1)=O)C2 C(=O)(CC(C(F)(F)F)OC)N1CC2(CN(C(C3CCC(CCC)CC3)=O)C2)C1 C#CCC(C(=O)N(CCCOC(C)C)C)NC(c1cc[nH]n1)=O C1(NC(CCN(C(=O)CC(C)F)CC#C)=O)CC(=O)N(CCC)C1 Cc1cc(C)c(C(=O)NCC2CCOC2C(=O)NCC(O)C(C)C)s1 C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(CC)NC(=O)CCNC(=O)C(C)(C)C c1(C(N2CC(C)(NC(=O)CC3CCC(=O)C3)C2)=O)c(Cl)nsc1Cl Cc1c(C(=O)NCCC2=CCN(C(C3CC3F)=O)CC2)[nH]c2c(Cl)cccc12 C1(C(N2C(CCNC(C3(C)CCOC3)=O)CCC2)=O)CC2C=CC1C21CC1 c1(C(C)C)cc(C(N2CCOC(CNC(C3(N(C)C)CC3)=O)C2)=O)cc(Br)c1 N1(C(C(C)N(C(c2ccc(C#N)o2)=O)CC)=O)CC(C)CCCC1C n1(CC(=O)NCC2C3CC2N(C(c2c(F)cccc2F)=O)C3)ncc(O)nc1=O c1(CNC2CCN(C(c3[nH]cc(C(C)(C)C)c3)=O)C2)cccc2c1CCCC2 C(=O)(C(O)CCC(C)C)N1C(C(N2CC(C(CC)C)C2)=O)CCC12CC2 C(CNC(c1cn(C)c(=O)n1C)=O)(CC(F)(F)F)NC(Cc1ncc(CC)[nH]1)=O C(C1(O)CCc2ccccc21)N(C(=NCCC)NCC1OCCC1(C)C)C CCC(F)(F)CC(=O)NCCOC1CCN(C(C23CC(C(C)(C)C)(C2)C3)=O)C1 C(=O)(C(F)(F)C(F)(F)F)N(C)CC1(O)CN(C(c2sccc2F)=O)C1 CC12CCC(O)C(C1)N(C(C1CC(C(F)(F)F)CN1)=O)C2 c12ccc3c(c1)OCC3N(C)CCC(CCOC)C(OCC)CN2 C1(CNC(c2n(C=C)nnc2)=O)CCN(C(=O)C(CSC)OC)CC1C1CC1 N1(C(COCC#C)=O)CC(NC(=O)C(C)(O)CCC)CC2(CCC2)C1 c1(C(N2C(C(N3CCCC(O)C3)=O)CCCC2)=O)cc(F)c(F)c(O)c1F c1(C(N2CCCC2C(=O)O)=O)cccc(N2CCCCC2)c1 CCCCCCCCC(=O)N(CC(C)CNC(c1cnn(C(C)C)c1C)=O)C c12nc(cs1)CC(=O)NC(C)CC1CN(C1)C2=O.c1(CC)ccc(Cl)o1 c1(C(N2CCC(C)(CNC(C(C)(C)SC)=O)C2)=O)ccc(F)cc1O C1(NC(CC=Cc2ccc(C)cc2)=O)CN(C(=O)C(C)C(F)F)CC12CCC2 C(=O)(CS(C)(=O)=O)NC(CC)C(C)NC(=O)CCCN(C)C c1(OC)cc(C(N2CC(NC(C3CC(C4CC4)C3)=O)C2)=O)ccc1Br C1(C(=O)NCC(CC)NC(c2cocn2)=O)COC(C)(C)C1 c1(NCCCCSC)nc(N2CCC(CC#N)C2)nc2scnc12 C1(C(N2C(CCNC(Cc3nc(COC)sc3)=O)CCC2)=O)CCS(=O)(=O)N1 N1(C(CNC(=O)NC)=O)CC(NC(=O)C2=CCCCC2)CC12CCOCC2 C1(C(=O)NCC(CNC(CCc2ccc(C)s2)=O)CO)CCC2(CC1)CC2 N1(C(C(C2CCC2)CC#N)=O)CCCC(C(=O)OC(C)(C)C)C1 c1(C(N(c2nc(C(F)(F)F)n3c2CCCC3)CC)=O)ncnc2sc(C)cc12 CC(C)(CCNC(=O)C=CC1CCCC1)C(=O)NC(C(C)(C)O)C1CC1 C1(C(N2CCCC(CC(C)C)C2)=O)CN(C(C23CCC(C2)OC3C)=O)CCN1C c1(CN)ccc(S(=O)(=O)N2CCOCC2)c(F)c1.C1(C)C(COC)CC1(F)F N1(C(C(C)=CC=C)=O)CCC(C)(C(N2CCC2C=C)=O)CC1 c1(C(=O)NCCC(=O)OCC2CCC(C(C)C)CC2)cc2n(n1)CCC2 N1(C(C2(C)CC2)=O)CC2CCCC1C2CNC(c1cc(C2CC2)nnc1O)=O CCCS(=O)(=O)C(C)C(=O)N1CC(NC(=O)Cc2ccc(C)cc2)CC(F)C1 CC1(C)CCN(C(=O)CCC2CC2)C(C(=O)NCc2nccc(O)n2)C1 c1(NCC(C(=O)OC)=CC(C)C)ccccc1SC(C)C CCCC(C)C(C)NC(=O)CC(C)(C)NC(c1ccncc1F)=O N1(C(c2cncc(OC)n2)=O)CCC2(NC(c3cccc[n+]3[O-])=O)CC2C1 C(=O)(C(C)(O)CC(F)F)N1CCC(CCNC(C(C)(C)N(S(C)(=O)=O)C)=O)CC1 C(=O)(CC(C)C(F)F)N(C1CCN(C(=O)CCc2c(N)cnn2C)CC1)CC#C c1(CC)nnc2n1CCCC2C(=O)N1CCC(NC(=O)COC)C1 c1(CC(N2CCC(N(C(C(C)CC3CC3)=O)C)C2)=O)ccc(O)cn1 NS(=O)(=O)CC(=O)NCc1cn(CCCCNC(C2CCOC2C(F)(F)F)=O)nn1 N1(C(C(CNC(=O)C(C)=CC(C)(C)C)F)=O)CCCC(C)(N(CC)CC)C1 C1(NC(=O)Cn2cccc2)CCCC2CN(C(=O)Cn3cc([N+](=O)[O-])cn3)CC12 C(=O)(C1=CCCOCC1)N(CC(CC)NC(=O)C1=CCN(C)C1)C C1(NC(c2n(C(C)C)ccc2)=O)CN(C(C2(O)COC2)=O)CCC1C(F)(F)F N1(C(C2C(=C)C2)=O)CCOCC(CNC(c2cc(-c3ccc(F)cc3)no2)=O)C1 Cc1cccc(CC(=O)NC2C3CN(C(=O)C=Cc4cccc(O)c4)CC23)c1F C1(C(N(CC(=O)NC2(C)CSC2)C(C)C)=O)CC(=O)CC(=O)C1 c1(CC(=O)NCCCC2(NC(c3ccn(CCF)n3)=O)CC2)cnc(C2CC2)[nH]1 C(C(=O)N(C)CC1CCN(C(c2ncnn2C(C)C)=O)C1)(C(C)C)SC C1(C2(O)CCN(N(Cc3ccccc3)C3CCCC3)CC2)(COC)CC1 c1(OC(CC(c2cccc(C)c2)C)=O)cccc2c1CCCC2 CCCC(C#N)C(=O)NC(C1CN(C(=O)C=CC(C)C)C1)C C1(CNC(c2ccnnc2O)=O)CN(C(c2ccc(F)s2)=O)C2COCC2O1 c1(OC)ccc(N)c(C(=O)NC2CCN(C(c3cnc(C)s3)=O)C2C)c1 c1(CC)ccc(C(=O)NCCC2CN(C(=O)C=NOC)CC2C)cc1F C12(C(=O)NCCC3CN(C(CN4CCC(OC)C4)=O)C3)CC(CO)(CCO1)C2 c1(C(=O)NC2(c3cccc(OC)n3)CCC2)cc(Br)c(C)cc1F c1(NC(C=CCNC(c2c(C)occ2)=O)=O)cccc(C(C)F)c1 C1(OC(C)C(=O)NC2CC2CNC(=O)CC(C)(C)C)CCOCC1 C1(COC)CN(C(c2cc(C)nn2C)C(=O)NCCCSC)C1(C)C CC1(C)CC2(CC(C(=O)NCCC(O)CNC(=O)Cc3ccc4c(c3)CC4)C2)C1 c1(CNC(CC)(C)C(F)(F)F)ccc2c(n1)OCC(=O)N2 c1(CC)ncncc1C(=O)N(C)CC1CN(C(=O)C(C)C2CCCO2)C1 O=NN1CCCC1C(N1CCC(Cn2cc(CC(c3ccccc3)O)nn2)C1)=O C(=O)(C#Cc1ccc(O)cc1)Nc1c(C)nc2ccncc2c1 N1(C(c2ccc(C(N)=O)cn2)=O)CCC2(CC1)CCN(C(=O)CCOC1CC1)C2 N1(C(CS(CCOC)(=O)=O)=O)CCOC2CN(C(=O)Cc3nonc3C)CC12 CCCCC(C)C(=O)NC(C(=O)NCC(C)(C)OC)C1CC1 C1(C)(NC(c2ccn(CC)n2)=O)CCN(C(C2CCC(C(=O)OC)C2)=O)C1 CC1(C)CC(C(=O)NCCc2nnc(O)o2)CN(C(C2C3CCCOC23)=O)C1 c1(C(=O)OCC)ccsc1Cc1ccc(C(=O)C#N)s1.C12(CC1)CC(=O)NC2 C1(CC=C)(C(N2CC(O)(C(N)=O)C2)=O)CCN(C(=O)CC(=O)OCCSC)C1 C(=O)(C1CCCn2nccc21)N1C(CNC(c2c(SC)cccc2)=O)CC(O)C1 Cc1ccc(C(N2CCN(C(=O)CCC(C)N(C)C)CC2C)=O)c([N+](=O)[O-])c1 C1(NC(C(CO)OC)=O)CC2(C1)CC2C(=O)NOCC(=O)NC(C)(C)C C1(=O)C(COC)OCC(C)N(C)C(=O)CC2CC12.C1(OCC)CC(CC)C1 c1(OC)c(Cl)cc([N+](=O)[O-])c(Cl)c1C(N1CCC(C)C1)=O CCC(C)(F)C(=O)NCC1CCCN1C(=O)CN(c1ccccc1)C C(=O)(CCCC(F)(F)C(F)(F)F)NCC1N(C(C2CC=CC2)=O)CC(C)(C)OC1 C1(NC(COCCCC)=O)CN(C(c2ccc(C(F)(F)F)cc2)=O)CC1CC C1(C)(COC(N(CCOC)CCOCc2ccccc2)=O)CC2CC2C1 C1(C(=O)NCCCOCCOCCN)CCCCC(=O)N1.C(=O)(CC(F)(F)F)C(=O)CC c1(OC)c(C(N2CCC(N3CCC3NC(=O)CS(N)(=O)=O)C2)=O)cccc1F C(=O)(CCCC(CC)NC(=O)CC(C)F)NCCOCCC=C c1(C(=O)NC2C(NC(C(CCSC)O)=O)CCC2)ccnc2[nH]c(O)nc12 C1(NC(C(CCC)NC(C2CC(SC)C2)=O)=O)CCn2cncc2C1 C1(C(=O)NC(C2CCCC2)CNC(Cn2c(C)cnc2)=O)CCC(N=[N+]=[N-])CC1 Cc1nc2cc(C(=O)NC3CN(C(=O)C(C)S(N)(=O)=O)CC3N=[N+]=[N-])cnc2[nH]1 N1(CC)C(=O)CCC1CC(=O)NC1CCC1NC(=O)CCCn1ccccc1=O c1(C(N2CCC(C)=C(C)C2)n2cc(C3(COC)CC3)nn2)cc(Cl)cc(Cl)c1Br C1(NC(CC(C=C)CC)=O)COC2(C1)CN(C(=O)CCSC(F)(F)F)C2 CC1CC2(CCN(c3ncnc4[nH]ccc34)CC2)CN1C(C1CC(C)(F)C1)=O Cc1ccnnc1C(=O)NCC(C(C)(C)C)NC(c1ccc(F)o1)=O C1(C(N(OC)Cc2ccc(C)o2)=O)CN(C(c2c(C)noc2N)=O)CC12CC2 Cc1ccc(C(CNC(=O)C(F)=CC2CC2)NC(C2CCCN(C)C2)=O)cc1 C(=O)(C(C)(COC)CC)NCC1(C)CCN(C(c2cnn(CCOC)c2C)=O)C1 C1(C(C)C)CN(C(=O)CC2CC3C=CC2CC3)CCCN1C(=O)C1=COCCO1 C1(C(=O)NCC(CSC)OC)CC2CCCC2N1C(c1ccc(C)[nH]1)=O CC1(NC(=O)CCCC#N)CCN(C(c2cc(C(O)C(F)(F)F)ccn2)=O)CC1 c1(C(=O)NC(CC)CNC(c2cc(C3(C)CC3)n[nH]2)=O)cc(C)cnc1OC c1(C(=O)NCCC2OCCN(C(c3c(C)cc(CO)o3)=O)C2)cncn(C)c1=O C1(C(=O)NC(CCN(C(=O)C(F)C(C)(F)F)C)(C)C)CCC2(CCCC2)C1 Cc1cc(C(=O)NC2CCC(Nc3cc(C4CCCCC4)ncn3)CC2)n(C)n1 c1(C(N2CC(NC(C(C)=CC)=O)C2)=O)cccc(CN2CCCC2=O)c1 C(=O)(C1=NN2CCC(C)N=C2N1)NCC1N(C(C2Cn3c(C)nnc3C2)=O)CC1 n1(CC)ncn(NC(=O)C(F)(CNC(=O)CN(C)C(=O)OC)C(C)C)c1=O N(C(=NCC(C)(C)C#N)NC1CC(c2cccc(Cl)c2)C1)C(C=C)C c1(OC)cnc(C(N2CCCCC(CNC(=O)OC(C)(C)C)C2)=O)c(OC)n1 c1(C(c2n(CC)nnn2)NC2CC(NC(C3CCCO3)C)C2)ccc(Cl)c(F)c1 CC(C(CO)NC(=O)C(=O)OCC(=O)NCC(F)(F)F)NC(=O)CNC(=O)C(C)(C)C c1(C(=O)NCC2(C(N)=O)CN(C(c3cc(C)ns3)=O)C2)ccncc1C(F)(F)F c1(C(=O)NC(CNC(C(CC(C)C)F)=O)(C)CC(C)C)cc2cc(O)ccc2[nH]1 N1(C(C(CC#C)NC(=O)CCCNC(C)=O)=O)CC2C=CC1CC2 C(CCCCC(=O)N1CCCCCC1CCO)NC(=O)C=Cc1cnccn1 C(=O)(C(CC(C)C)C(N)=O)N1CC(CNC(CSCc2c(C)noc2C)=O)(CO)C1 C#CCCCCCC(=O)NC1CCCC(CC(=O)N(CC(F)F)CCO)C1 C(=O)(C1=CC(C)(C)C1)NCCC1(NC(CC(CC)c2ccccc2)=O)CCCC1 CC#CCCC(=O)N(CCCNC(=O)Cc1ccccc1Cl)Cc1ccccc1 Cc1cc(N)c(C(=O)NC(CNC(c2cc3sccc3s2)=O)C2CCC2)cc1F c1(C(CN(C(C)=O)CC2CCS(=O)(=O)C2)SC)ccc(F)c(Cl)c1 N1(C(c2cc(C(C)C)nn2C)=O)CCCC(C(=O)Nc2cccnc2)CC1 CC1CN(C(=O)Cc2ccc(Cl)nc2)CCN1C(=O)CC(C)C1CCCO1 C(=O)(C1=CCCCC1)NC1(CC(=O)NCC(C(N)=O)O)CC1 c1(C(N(C)CC2CCN(C(=O)C=CCOCC(F)(F)F)C2)=O)cc[nH]c(=N)n1 c1(C(C(=O)NCC2CCCO2)N(C2CC23CCC3)C)nc2ccc(Br)cc2s1 N1(C(c2ccc(C)[nH]2)=O)CCC2CC12C(=O)NC(c1ccns1)C Cc1cscc1C(N1CCC1(C)CC(=O)NC1(C(C)C)CCC1)=O c1(C(=O)NC2CC(NC(C(C)S)=O)C(O)C2O)ccc2c(c1)c(I)nn2C Cc1cc(C(=O)NC2CN(C(=O)Cc3nc(C4CC4)cs3)CC2C)nc(C)c1 N1(C(C(=O)Oc2ccccc2)NC(=O)OCC)CCCC(OC(=O)C(C)CF)C1 c1(C(=O)NC2CN(C(c3c(C#C)c[nH]n3)=O)C(C)C2)cc2ccc(Br)cn2c1 c1(CC(=O)N(C(CC)(C)C)Cc2ccc(C)cc2)c(OC)cccc1O C#Cc1cc(C(=O)N(C2CCC(NC(C3(CO)CCC3)=O)C2)C)cc(F)c1 N1(C(C2(COC)C=CCC2)=O)CC2CCC1CN2C(=O)C(C)(C)OC1CCOC1 CC1COC2(C1)CN(C(c1sccc1CNC(=O)C(C)S(N)(=O)=O)=O)C2 c1(CSCC)ccccc1C(=O)NCC1(O)CN(C(=O)CC(C)N(C)C)C1 c1(C(=O)NC2(C(N3CC(C)(CCC=C)C3)=O)CCSC2)cc(Cl)n(C)n1 C12(C(N3CCN(C(C=C(C)C)=O)C(C)CC3)=O)C3CCC(CC13)C2(F)F N1(C(CCCC(=C)C)=O)CCCC(C2CN(c3nc(OC)c(F)c(C)n3)C2)C1 Cc1cc(C(=O)NC2CCCC(NC(=O)C=CCCC(C)C)C2)cc(Br)c1 c1(CN2C(=O)CCN2C(=O)C(=O)NCC(F)(F)CO)ccccc1.CC.OC c1(C(=O)NCC(CO)NC(CC2CCC(C)(C)O2)=O)onc2c1CCCC2 CCCC(C#N)C(=O)NC(c1c(C)cccc1Br)C(=O)NCCOC(F)F c1(CC)ccccc1C(CNC(=O)C(F)CC)NC(c1sc(C)cc1C)=O S(=O)(=O)(c1ccccc1S(=O)(=O)Nc1cccc2c1COCC2)NCC Cc1cc(N2CCC(C3CC3)(CNC(=O)CC(C)C(F)F)C2)n2ncnc2n1 C1(COC)CN(C(=O)C=C2CCN(C)CC2)CCN1C(C)=O N1(C(C2C(C)C2)=O)Cc2ccnn2CC(NC(=O)CC23CCC(CC2)C3(C)C)C1 C(=O)(C(CNC(c1cccnc1C)=O)CC1CCCC1)NCCn1ncc(C)c1 C1(NC(C=CC2(C)CCOCC2)=O)C2CCCN(C(=O)CC3(C)CC3)C2C1(C)C C1(N(C(CSC)=O)C)CN(C(=O)Cc2ccc(-n3cnnc3)cc2)CC1F C1(C(=O)NCCc2c(OC)ccc(F)c2)COC2(CCC2)CO1 C(=O)(C1CNC(=O)c2ccnn21)N1CCCC(CNC(=O)CCC=CBr)C1 C1(CNC(=O)COc2ccsn2)COC(Cn2cc(C(=O)NCC3CC3)nn2)C1 CC(C)(C)CC(O)C(=O)N1CC(CNC(=O)Cc2ccsn2)C(F)(F)C1 Cc1cnc(C#N)c(NC(C23CC(C(=O)Nc4cccc5ccnn45)(C2)C3)=O)c1 C1(C(=O)NCC2CN(C(Cc3n[nH]c(=NC)s3)=O)C2)CCN2CCOCC12 c1(C(=O)NC2C(NC(=O)C3=CCCC3)CCCC2)cc2c(F)c(Cl)ccc2[nH]1 C1(C(C)C)CCC(C(=O)NCCN2CCN(C(=O)C(C)N3CCCC3)CC2)CC1 C(C)(C)(CC=CC(=O)NCCC(=O)NC)NC(C1CC(CC)C1)=O Cc1ncc(Cl)c(C(N2CC(O)(CN(C(=O)C(O)C(C)N(C)C)C)C2)=O)n1 C1(NC(=O)Cc2cccnc2)CCCCC12CCCN(C(c1cnccn1)=O)C2 CCC(C(=O)NC1CC2CC1CN(C(c1ccc(C(N)=O)cc1)=O)C2)C(F)(F)F c1(C(C(=O)NCCCN(C(=O)C(C2CC2)OC)CC)(C)O)ccc(F)cc1 C(=O)(CC(O)CC(C)(C)C)NC1CC(NC(C=CC(=O)OCCCC)=O)C(O)C1 C#CCC(O)C(=O)NC(C)(CNC(c1ccc(CSCCC(N)=O)cc1)=O)CC C1(C(N2CCC(CC=CC)C2)=O)CCCCC1NC(=O)Cn1cc(COC)nn1 C1(CC)COCC1(c1nnnn1C1CCOCC1)NC(C)(C)CNC(=O)OC CCCC(CC)C(=O)N(C(CC)CC(=O)NCc1nc(OC)no1)C S1(=O)(=O)CCN1.c1(C(CC)(C2CCCC2)NCC)nnnn1CC c1(C(=O)OC)ccc(CCNC(N2CCC(C(C3CCCO3)=O)CC2)=O)cc1 c1(C(=O)NC2CC(NC(=O)C(F)CC3CCCC3)C(O)C2)ccc([N+](=O)[O-])s1 CCCC(C(=O)N1CCC2C(C(N3CCC(NC(=O)NC)C3)=O)C2C1)C(C)C c1(CC)ncc(Cl)c(C(=O)NC2(CNC(c3cnc(C)s3)=O)CCOCC2)n1 CCC(C)(CC)C(=O)N1CCC(F)(C(=O)NCCCCOC(C)C)C1 Cc1ccc2c(c1)CC(N(C(C1CCCC3(CNC3)O1)=O)C1CC1)C2 C(=O)(C(=O)C(C)(C)CC)NC(C(=O)NC(C(=O)NCC)(C)C)C(C)C Cn1ncc2c1CC(C(N1CCC(F)(CNC(=O)CCCCCF)C1)=O)CC2 C(=O)(C(C)CC(C)(C)C)N(C(CNC(c1cccc(OC(C)C)c1)=O)C)C N1(C(Cc2[nH]c(=N)sc2)=O)CCC2(CC1)OCCCC2NC(=O)COC(F)(F)F C(c1nccs1)=CC(=O)C1CC1.C1(=O)C(C2CC2)OCC2(CC2)C(C)N1 c1(C(=O)NC2CC(C)N(C(c3cn(C)[nH]c3=N)=O)CC2)c[nH]c2ccccc12 CC1(C)C(C(=O)NC2CC3CC(NC(c4ccc(C#N)cn4)=O)C2C3)CC1(F)F N#Cc1ccc(C(N2CCC(F)(F)C(CNC(=O)Cc3cn[nH]c3)C2)=O)c(O)c1 C1(CNC(CCCC)=O)CC(O)CN1C(=O)C(C)Oc1ccccc1 C1(C(N(CC(C)CNC(C2CCN2)=O)C)=O)CCCN(C(=O)N(C)C)C1 c1(C(N2CC(O)CC(NC(c3cc(F)cc(F)c3)=O)C2)=O)ccc2ncsc2c1 C1(CC=C)(NC(=O)CC(C)(C)O)CCN(C(C2CCC2(F)F)=O)CC1 C(=O)(C(CC(N)=O)NC(c1ccsc1C)=O)NC1CCN(C(C)=O)C1 C1(C(N2CC(CCn3cc(CN(C(C)C)C)nn3)C2)=O)CC(F)(F)C1C C1(CC)CCN(C(=O)C(OC)OC)C1CNC(=O)CCc1cnc(C)s1 N=c1nc2nc3cc3n2[nH]1.N1CCC(C2(O)CNC2)CC1 N1(C(C2C(=C)C2C(=O)OC)=O)CCC2(CC1)CC2CNC(=O)C=CC1CC1 C1(CC(=O)OC)CC(NC(c2ccc(Cl)cn2)C)CCO1 c1(C(=O)NC2C(C)CN(C(C3(C)CC3(C)C)=O)C2)cnc2ccc(Cl)cn2c1=O N1(C(C(C)=CC)=O)CC(C)(C)OCC1CNC(c1cccn1CCC)=O c1(NCC2C=CC(NC(=O)CNC(=O)C(O)c3ccco3)C2)ncccc1O C12(NC(Cc3cc(CC)nn3C)=O)CC3CCC(C1C2)N3C(=O)C(=O)NCC(F)F c1(C(=O)N(CCCNC(C2(Cl)CC23CCC3)=O)C2CC2)cc2c(s1)CCOC2 CCC(C)CCC(=O)N1CCOCC(CNC(=O)CC(C)(C)COC)C1 N1(C(C2C(C)C2C)=O)CC(CNC(=O)C=Cc2cncs2)OC(C)(C)C1 C12(CNC(C(CCSC)NC(=O)Cc3ccccc3F)=O)CC(C)(CCO1)C2 CC(C)(CC(F)F)C(=O)NCCSCc1cn(Cc2ccccn2)nn1 Cc1cc(C(N2CCC(CC3CC3)C2)C(=O)Nc2cnn(C)c2)ncn1 C1(C(=O)OC)CCCS1.C1(C(N(CCCNC)C)=O)CN(C(N)=O)C1 CCCCCCC(=O)NC(C1CCN(C(=O)CC2CCN(OC)CC2)C1)C C1(NC(CC2C(C)(C)OCC2)=O)CC12CCN(C(c1cccc(O)n1)=O)CC2 N1(C(CC2(C(=C)F)CCC2)=O)CC2(CCC2NC(c2cncc(C=C)c2)=O)C1 C=CCC(CNC(c1cc(Cl)cn1C)=O)C(=O)NOCc1ccccc1F N1(C(C(C(C=C)C)C)=O)CCC2(CC1)CC(NC(c1cc(CC)c[nH]1)=O)C2 C12(C(N3CCN(C4CCN(CC)C4)CC3)=O)CCC(F)C1CC2 C1(C(=O)NCCN(C(=O)CCCCC#N)C)CC2CCCCN2C1 N1(C(C2N(C(=O)C3CC3)CC(O)C2)=O)CCCN(C(=O)C2=CCCS2)CC1 CCC(CCc1ccccc1)C(=O)NC(C)CN(C(=O)C(C)CCO)C c1(C(=O)NC2(CNC(C(C3CCC3)OC)=O)CC2)ccnc(CO)c1 N1(C(CCSCCCC)=O)CC2CC(NC(=O)Cc3c(C)nn(C)c3C)CC2C1 N(C1CCCc2n[nH]cc21)C(C1CCC(=O)N(C)C1)=O.C#CCC1C(=O)N1 C1(NC(Cc2c(C)ocn2)=O)CC(N=c2[nH]nc(C(C)C)o2)C1(C)C c1(C2(C(=O)NCCN(C(=O)CCn3ccnc3)CC)CCC2)ccc(Cl)nc1 C1(NC(=O)Cn2ccnn2)CC2CC(NC(C3CC3[N+](=O)[O-])=O)C1C2 O=C(N=c1[nH][nH]c2c1CN(Cc1cc(Br)cs1)C2)c1cc(Cl)cnc1F Cc1nn(C)cc1C(=O)NC1CCN(C(C2CC2c2ccn(C)c2)=O)CC1 c1(OC)c(-c2ccc(C(=O)N(C)C3CC3)c(C)c2F)cc(C)cc1C c1(OC)cc(F)c(C(N2CCC(NC(=O)C(F)=CC3CC3)C2)=O)c(F)c1 C=CCC(C(=O)NC(CC(=O)N(CCC(C)C)C)C1CC1)NC(C)=O C1(C)(C(N2CC(NC(COCC=C)=O)C(SC)C2)=O)CCC12CCC2 c1(NC(c2ccc(CCNC(c3ccc(F)cc3I)=O)cc2)=O)nccc(Br)c1Cl C#Cc1ccc(C(=O)N(CC)CC2CCCCN2C(=O)C(C)S(N)(=O)=O)nc1 C1(C2CC(CC)C2)CCC(c2nc(-c3ccn(C)n3)nn2-c2nccn2C)CC1 c1(N2CC3N(C(c4cc(OC)c(Cl)cc4)=O)C3C2)nc(C)nc2c1CCC2 c1(C(N2CC3CCN(C(C4CCCN4C4CC4)=O)C3C2)=O)cc2cccnn2c1 c1(C(C(=O)N(C2CCN(CCc3n(C)ccn3)C2)CCO)=O)ccc(F)cc1 CC1(C)CC(CNC(c2snc(Cl)c2Cl)=O)N(C(=O)C(O)C(F)F)C1 N1(C(C(C)CF)=O)CC(NC(c2ccc(F)c(Cl)c2)=O)CC1(C)C CC(C(=O)NC1(CNC(=O)CCSC(F)F)CCC(F)(F)CC1)C(F)(F)C(F)F C(=O)(CCCCCSCC)N1CCC(C(=O)NCCN(C(CC)C)C)(C(C)C)C1 C(=O)(C(O)CC(C)(C)C)N(CC(C)O)CCNC(c1n(CC)cnn1)=O c1(C(N2CC(NC(C(C)=C(CC)C)=O)C(C)C2)=O)nc(OC)ncc1C CC1(C(N2CCC(C(C)(O)CNC(=O)CC3CCSC3)CC2)=O)CCNC1=O N1(C(COCC(C)(C)C)=O)CCCCC(NC(c2ccc(Cl)c(Cl)c2)=O)CC1 N1(C(C2CN(C(N(C)C)=O)C2)=O)CCC(C2CCCN(C(=O)C(O)C3CC3)C2)C1 C#CCC(C)(C)C(=O)NCC(C1CCC1)NC(=O)C(F)n1cccn1 c1(CC(=O)NC(C)CNC(C2CC3(C2)CC(C#N)C3)=O)ccc2c(c1)ncn2C C1(CCC)CCC(C(=O)NCC2C=CCN2C(c2nc(C3CC3)oc2C)=O)CC1 c1(C(=O)NC(CNC(c2nc(CCCCC)sc2)=O)(C)C)cnn(CCC)c1C S(=O)(=O)(CCCC1CC1)NC(=O)C(CN1CCCC1)c1ccccc1 C1(NC(CC(C)C2CC2)=O)CCC(F)(CNC(=O)CCc2nnc(C3CC3)o2)C1 C(=O)(C(CC(C)C)n1ccnc1)NCC(N(C(COCC#C)=O)C)C1CC1 c1(N2C(CC)CN(Cc3ccc(Cl)c(Br)c3)CC2)ncc2ccccc2n1 c1(C(=O)NCC(CC=C)NC(=O)C#CC2CCOC2)cnn2cccc(C)c12 N1(C(CCC2(C)CC2)=O)CCCC1CCCNC(=O)Cc1ncsc1Cl N1(C(CC2CCN(C(=O)NCCOC)CC2)=O)CC2COCC2(CO)C1 N1(C(c2cnsn2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)C(C2CCC2)C1 S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1C(C(=O)Nc2c(C)nsc2)C=CC1 C(=O)(CC(O)CC(C)(C)C)N1CCC(CN(C(C2C(CC)C2)=O)C)CC1 c1(OC)cccnc1C(=O)NC(C)C(C)(C)NC(=O)CP(C)(C)=O c1(C(N2CC(NC(C(Cc3ccsc3)NC(C)=O)=O)C2)=O)ccncc1N(C)C O(N=C1CCCCCC1)CC(=O)N(CC(CN(C(c1csc(C)c1C)=O)C)O)C C1(CN(C(COCCC(C)C)=O)C)CCN(C(C2CN(C(N)=O)C2)=O)C1 Cc1ncc(C(N2CCC23CN(C(=O)CCn2cc(Cl)cn2)C3)=O)cc1C#N Cc1ccc(O)cc1CNC(C1N(C(c2ccc(Cl)cn2)=O)CCC1(C)C)=O CC(CC(=O)NCCN(C)C(c1cn(C)nc1-c1ccncc1)=O)C(F)F C1(C(=O)NC2C(NC(CCC(=C)Cl)=O)COC2)CCc2nc(C)sc2C1 N1(C(COCCC=C)=O)CC(C)CN(C(c2ccoc2)=O)C(C)C1 CC1(NC(=O)CSc2ccccc2)CCN(C(=O)CC2CCCNC2)C1 c1(C(N2CCCC(C(C)NC(c3cnc[nH]c3=N)=O)C2)=O)ccc2scnc2c1 C1(N2CC(C3(F)CCCC3)C2)CC2CCC(C1)N2C(=O)CCCn1ccccc1=O c1(CN(CC(N2CCOCC2)=O)CC)cccc(Cl)c1F.C12CCCN(C1)C2=O C1(C(=O)NCC(=O)OCC)CCC(C)(C)N(C(=O)CCCn2ccnc2)C1 C1(CCCC)CCN(N2CCC(c3nc(=N)[nH][nH]3)C2)C1 N1(C(CN(CC)CC)=O)CC2(CNC(=O)Cc3ccc(Cl)cc3)CCC1C2 N1(CC(c2cc(C(=O)O)sc2)=O)CCCC2(CCCCC2)C1 C1(C(=O)NCC2C3CN(C(c4cc(Cl)c[nH]4)=O)CC23)(OC)CCOCC1 N1(C(C(CC)=O)=O)C(C(=O)Nc2nc(C)c(Cl)s2)CC2CC12 C1(NC(c2c(N)snn2)=O)CC2CN(C(=O)CNC(=O)CCCCO)CC12 c1(C(=O)NCC(CCOC)NC(c2sc(=N)[nH]c2C)=O)cc(C)ccc1F c1(C(N(C(CNC(COCCCN(C)C)=O)C)C)=O)ccncc1O CC(C)(C)CCC(=O)N1CC(NC(C2NC(=O)CC2c2ccccc2)=O)C1 c1(C(N2C(CCNC(C(C=C)(C)O)=O)CSCC2)=O)cn2ccnc2cn1 C=CC(C)(C)CC(=O)NC1CCC(CC(=O)NC2C3CCC(C3)C2CO)CC1 CC1(C)CCN(C(=O)CCc2cocn2)C1CNC(c1coc(CO)c1)=O C1(C(=O)NCC(C)(C2CC2)NC(c2coc3c2COC3)=O)CC(S(C)(=O)=O)C1 C(CC(C)(O)C(=O)NC1CCC(C(N2CC(C)CCC2C)=O)C1)N(C)C C1(NCC(=O)NC(C2N(C(CN(C)CCO)=O)CCC2)C)OCCC1C(F)(F)F c1(C(=O)NCC2N(C(C=CCC)=O)CC(C)CC2)cc2cc(OC)ccc2cn1 CN1C(=O)CCC1C(=O)NC1(C2CCCN2C(c2[nH][nH]c(=N)c2Br)=O)CC1 c1(C(=O)NC2(CO)CN(C(c3c(CC)cc(Cl)cc3)=O)C2)cn2ccccc2n1 Cc1cn2c(C(=O)NC3CCCN(C(=O)CS(=O)(=O)C4CC4)C3C)c(C)nc2s1 C1(C)(CNC(c2cc(C)c(C)[nH]2)=O)CN(C(c2cc(O)nn2C)=O)CCO1 C1(C(=O)NCCCn2c(C)nnc2)CCOCCN1C(=O)C1=CCSC1 N1(C(COC2C(C)C2)=O)CCCC2(CCN(c3nc4cc(F)c(F)cc4s3)C2)C1 C1(CCNC(C(CC)F)=O)COCCN1C(c1cc(-c2cccc(C)c2)[nH]n1)=O c1(CC)ccc(C(=O)NCC2(C)CCCN2C(=O)CC(C)(C)F)nc1 N1(C(CC2(C=C)CC2)=O)CCC(C2CC2)C1NC(=O)Cc1cnns1 N1(C(C)=O)CC(NC(c2ccc(C3CC3)cc2)=O)C2CC2C1.CN1CCOCC1 C=C1CCN(C(=O)CCCNC(N)=O)C(C(N(C)C[Si](C)(C)C)=O)C1 C#Cc1ccc(C(N2CCC(CO)(CNC(=O)C#CC(C)C)C2)=O)cc1F S(=O)(=O)(c1ccc(NCC(O)CC(N)=O)c(Cl)c1)NC1(C)CCCOC1 c1(C(N2CCC(NC(CCC(=O)NC)=O)CC2)=O)[nH]c2ccccc2c1Cl C1(NC(C(CC)C(C)O)=O)CCC2CN(C(C3CC3(F)F)=O)CCC2C1 C(N=c1nc2ncn(CC)c2c(NCC(C(C)C)C(C)C)[nH]1)c1c(CC)c[nH]n1 CCCCC(O)C(=O)N1CCC(NC(=O)Cc2ccnn2C2CCOCC2)CC1 n1(CC(N2C(CNC(C(C(C)C)n3cncn3)=O)CCC2)=O)nc(O)ccc1=O C1(NC(c2ccc(CNC(C)=O)s2)=O)CC2(C1)CN(C(C1CCOC1)=O)C2 C1(CCC)CCCN1C(=O)CC1CCN(Cc2ccccc2C)C1.C(=O)O c1(C(=O)NCCNC(=O)CC2(CO)CC2)ccncc1O C(=O)(C#CC1CCCO1)N1C(C)(CNC(c2cc(C)sc2)=O)CCC1 C=CCC(C(=O)NCC1CC(NC(c2cc3c(s2)CCCC3)=O)CCO1)C(C)C C1(CNC(Cc2c(C)ccc(F)c2)=O)CC2CCC1N(C(C1CC(C)(F)C1)=O)C2 C(=O)(C(C)C(C)(C)C)NC(C1(NC(=O)Cc2ccn(C)n2)CCC1)CC c1(NCC2CC(NC(=O)CCc3ccc(Cl)cc3)C2)ncnn2cccc12 c1(CN2CC(NC(c3cccc(C(N)=O)c3)=O)C(O)C2)c(Cl)ccc(F)c1F C1(COC)CC12CCN(C(C1C3CN(C4CC5OCCCC45)CC13)=O)C2 Cc1nc(Cl)nc(N2CC3(COC(CNC(C4CCCCC4)=O)C3)C2)c1F c1(-n2cc(C3CN(C(CC4C(C)C4)=O)C3)nn2)ccc(F)cc1 N1(C(C(C)OC)=O)CCC2(CCC(CNC(c3cccc(Cl)c3C)=O)CC2)CC1 C(=O)(CCC(C)NC(=O)C=C(CC)CC)N(CCCC=C)C C1(N(C(=O)C=C2CCC2)C)CN(C(C2CC2C#N)=O)CC1O Cc1cccc2c1N(C(c1nc(Br)c(C3(C(F)(F)F)CC3)s1)=O)CCN2C1CC1 Cc1cc(Cl)c(CN(C(C)(C)CC)CCCOC(C)(C)C)nn1 c1(CC(=O)N(C2CCN(C(=O)CNC(=O)C(C)(C)C)C2)C)ccc(F)nc1 c1(C(=O)NC(C(C(C)C)NC(=O)CC2C(C)(C)C2(C)C)C)ncc2n1CCCC2 c1(OCC)cccc(CCC(=O)NC(CNC(C2C3CC4C(C3)C24)=O)C(C)C)c1 N1(C(c2cc(OC)ncn2)=O)CC(C2CCCN(C(=O)C(O)CCC(C)C)C2)C1 c1(C(=O)NC2(CNC(=O)CC3CCC3)CCOCC2)cnc2cc(O)ccc2c1 CCCC(CC(=O)NCc1nc(=O)o[nH]1)NC(c1coc(C)n1)=O C=CC1(NC2CNC(=O)OC2O)CCN(C(=O)OC(C)(C)C)C1 N1(C(C2CCN2C(c2nccs2)=O)=O)CC2CCC(C1)O2 N1(C(c2ccc(C(N)=O)s2)=O)CCCCC1C1(NC(c2ccccc2Cl)=O)CC1 c1(OC)cc(F)c(C(=O)NCC(C)N(C(=O)C(F)C2CCOC2)C)c(F)c1 c1(C(=O)NC2C3(CN(C(C(CCC)O)=O)C3)CC2)cc2ccc(Cl)c(F)c2[nH]1 N1(C(C(C=CCCC)O)=O)C(C)CC2CN(C(c3nn(C)cc3Cl)=O)CC12 c1(C(N(CCCNC(=O)C=C(C)Cl)CC)=O)ccc(S(N)(=O)=O)c(OC(C)C)c1 c1(C(=O)NCC(CC)NC(c2c(Cl)cnn2C2CCCC2)=O)cn(C)nc1O C1(OC)CN(C(C2(C)CCCCO2)=O)CC1C(=O)NC(C1CCCCC1)CO c1(C(=O)NC2CC(O)CN(C(c3ccc(CO)cc3)=O)C2)cccc2c1NCC2 c1(NC(CN(C(=O)CN(C)C)CC)=O)cncc(Br)c1C C1(C(N(CC)CC)=O)(NC(c2c[nH]nc2C2CCOC2)=O)CC=CC1 C1(NC(CCC(=O)NCC)=O)CC2CC1N(C(=O)Cc1csc(=N)[nH]1)C2 CS(=O)(=O)C1(C(=O)NC(CNC(c2cccc[n+]2[O-])=O)C2CCC2)CCOCC1 c1(C(=O)NC2CCCC(NC(C3(C)CC3(Cl)Cl)=O)C2)ccc2ccccc2c1O C1(N(C(c2occc2C)=O)CC)CNCCC1(C)C c1(N(C)Cc2c(C)nsc2)nc(N2CC(=O)NC(C(C)C)C2)c2ncccc2n1 CC(C)C(O)C(=O)N1CC(F)CC1CNC(C1C2CCC1CC2)=O N1(C(C(=O)NC(c2c(C)c(Br)ccc2)C2CC2)=O)CCSc2ccccc21 C(c1ccccc1Cl)=C(C(=O)NC(CC)CNC(c1cc(C(C)=O)oc1C)=O)C c1(C(N2CCN(C(CC=C=C)=O)CC(CO)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N2CCC(N(C(c3c(O)cc(C)nn3)=O)C)C2)=O)cccc2c1CCC2 Cc1ncc(F)c(N2CCCCC2)n1.C1(N)CCN(C(=O)CCS(C)(=O)=O)CC1C c1(C(N2CCC(N(C(=O)C3=NOCC3)CCC)C2)=O)ccc2cnoc2c1 N1(C(C(C)=CC)=O)CC2ON=C(CNC(=O)CSS(C)(=O)=O)C2C1 c1(CC(c2n(CC)c(N3CCCC(C)C3)nn2)C)ccc(F)c(F)c1 C(C(O)C(=O)NC1(CO)CN(C(=O)C(F)CC2CCOC2)C1)=CC c1(OCC)sccc1C(=O)NCC(CO)NC(=O)C(C)Cc1ccnn1C N1(C(C(=O)NCC(c2cccc(F)c2)N(C)C)=O)CC2CS(=O)(=O)CC2(C)C1 N1(C(COCC(=C)C)=O)CCC(C(=O)NOCC(O)CO)(C(=O)OC)C1 N1(C(Cc2c(C)nsc2)=O)CCC(NC(c2cn(C)c(C)n2)=O)C(O)C1 N1(CC)C(=O)CCC1CC(N1CCC(O)(CN(C(=O)CC2(C)CCOC2)C)C1)=O Cn1cc(Cl)cc1C(=O)NC(CNC(c1cccnc1O)=O)C1CC1 N#Cc1ncccc1NC(c1ccc(Cl)nc1NC(=O)C=CC1CC1)=O Cc1ccc(CC(N2CCCCC(NC(c3n[nH]c(=N)s3)=O)C2)=O)c(C)c1 C1(NC(CCc2cc(OC)no2)=O)CC2(CCN(C(c3ccc(Br)o3)=O)C2)C1 c1(C(=O)NC(CC(=O)NC(CO)CCF)CC2CC2)cnn2c1CCC2 C(=O)(C1=CC2CCCCC12)N(CCCNC(Cn1nnc(C)n1)=O)C1CC1 CCC(C#N)C(=O)NC1CCCC(CC(=O)N(CC(O)C(C)(C)C)C)C1 c1(NC(N2CC(OC(F)(F)F)(COC)C2)=O)c(C)nsc1C c1(N2CCN(C(C(n3cc(CCC#N)nn3)C)=O)CC2)cncc2nnnn12 c1(C(=O)NCC2C(NC(=O)Cc3cccc(Cl)c3F)C2)ccc2scnc2c1 CCCCCCCCC(=O)N1CC(CNC(=O)COCCC)C2(CC2)C1 c1(OC)cc(F)ccc1NC(C1C=CC(NC(c2cn(C)nn2)=O)C1)=O C12(NC(CC)=O)CN(C(c3c(C)ccc(Br)c3C)=O)CC1CS(=O)(=O)C2 N1(C(c2ccc(C)cc2O)=O)CCCC2(CCN(C(c3c[nH]c(Br)c3)=O)C2)C1 CC1(C)C=C(C(=O)N2CC(F)(F)CC2CCNC(=O)C(F)OC(F)(F)F)C1 C1(C(N(CC)Cc2cnn(C)c2)=O)COC2(C1)CN(C(C1CC3(CC3)C1)=O)C2 c1(C(C(N)=O)N(c2cc(Br)ccc2OC(F)F)C)ccc2ccccc2c1 N1(C(CS(N)(=O)=O)=O)CCCC2CCN(C(=O)COCCF)CC12 c1(C(=O)NCC(=O)NC)ccc(NC(c2cccc(Cl)c2)C)nc1 C1(CNC(CCCC(C)=O)=O)C2CCCC1N(C(=O)CC1CC=CCN1C)C2 C=C(C(=O)NC1CC(n2cc(-c3cc(C#N)ccn3)nn2)C1)C(C)(C)C c1(C(N(CC(=O)NC2CCC(O)CC2)C)=O)ccc(C#N)cc1 N1(C(C(CC)N(C)C)=O)CCC2(CC1)CC(NC(c1cc(Br)n[nH]1)=O)CO2 c1(C(=O)OCC)cc(=NC(C)Cc2ccc3cc(Cl)ccc3c2)[nH]c(Cl)n1 c1(C(C)NC(=O)NC(C#C)CC2CCCO2)ccnn1C C#CCCCC(C)C(=O)NC1CCC12CCN(C(c1cnc(Cl)s1)=O)CC2 c1(C(N2C(C)CC(NC(c3cccn(C)c3=O)=O)C2)=O)cc(F)c2[nH]nnc2c1 C1(NC(c2nc(C)[nH]n2)=O)CN(C(=O)C(C)Sc2ccccn2)CCC1C c1(C(=O)NC(C2CCCN2C(c2nnn(C(C)(C)C)n2)=O)C)ccc(Cl)o1 Cn1cnc(C(=O)NCCC2(C)CC2(F)Cl)cc1=O CC1(C)NC(=O)CCC1C(N1CCCC1CC1(c2cc(Cl)cc(Cl)c2)CC1)=O c1(C(N(CCN(C(C(CC)OC)=O)C)C(C)C)=O)cn2c(n1)CC(C)CC2 c1(C(N2CC(C)(C(=O)NCC3(OCC)CC3)C2)=O)ccn(C)c(=O)c1 c1(N2CCC(CC=C)C2)nc(N2CCC(N(C)C)(CO)CC2)nc2ccccc12 c1(-c2ccc(SC)cc2)c(C(=O)NC(C2CCC2)C2CC2)nn2c1CCCC2 CCCC(C(O)C(=O)N1CC(N(C)CCOCC)C1)NC(=O)CC(=O)OC Cc1cc(C(N2CC(CN(C)C(c3ccnc(C4CC4)c3)=O)C2)=O)nn1C(F)F C1(C2CCCN(c3nc4cccc(Br)c4o3)C2)(NC(C2=NOC(C)C2)=O)CC1 C=CC1(CC(=O)NC(C)CN2CCOCC2)CN(C(C2CCC(CC)CC2)=O)C1 C=CC(C)(CCOC)C(=O)N1CC(CNC(C2CSC2)=O)C(C)C1 N1(C(c2scc(OC)c2)=O)CCCC2(CC(NC(=O)C(C)n3ccnn3)C2)C1 N1(C(CN(CC)CC)=O)CCC2C(NC(c3cc4scnc4[nH]3)=O)CC12 c1(CNC(=O)NC(C2(CN(C)C)CC2)C)cccc2c1C(=O)c1ccccc1C2=O c1(C(CC)NCc2ccnn2C)cc(O)ccc1F C1(OC)C2CCC(C2)C1NC(C1CCC(C(N2CC3CCC3C2)=O)CC1)=O C1(NC(c2ccc(CC)cc2)=O)CCN(C(C2CCN(C)C2)=O)CCC1CO CC(O)(CC(F)(F)F)C(=O)N1CCCC(C)(CNC(c2ncc(C(F)F)s2)=O)C1 C12CCCN(C1)C(=O)Cn1cc(nn1)C2.C1(CC(=O)OC(C)=O)CCCOCC1 c1(C(=O)NC2CN(C(C(C#C)(C)C)=O)CC2C)ccc(F)c(Cl)n1 N1(CC)CCc2nc[nH]c(=NCC(C)c3sc(-c4ccccc4)nc3C)c2CC1 c1(NC(CCC=C)c2nnnn2CCCF)sc2c(c1C=C)COCC2 C(CCC1CC1)(C(=O)NCCCN1CCCC1C)NC(CC(C)c1ccco1)=O c1(CN(CCCC)C(c2ccccc2)=O)cnn2c1NC(C)CC2 c1(C(=O)NC2CC(C)N(C(=O)Cc3csc(=N)[nH]3)C2)cc(C2CC2)cc(F)c1 CCC(CC(C)C)C(=O)N1CCC(C)C1C(=O)NCc1nc(C)ccc1C c1(N(CCN(C(=O)C(=O)Nc2c(C)con2)C)C)cc(Cl)cc(Br)c1OC(F)F c1(CC(CNC(NCCCF)=S)C)ccccc1Cl C1(C(N2C(CNC(c3c(C)csc3Cl)=O)C=CC2)=O)CCn2c(C)nnc2C1 C(=O)(CC(C)CC(F)(F)F)NC1CC2CC(NC(c3c(C)csc3)=O)CC21 c1(C(=O)NCC23CCCCC2N(C(=O)CCF)CC3)cccc2cc(F)ccc12 N1(C(C=CC(CC)C)=O)CC2(C1)OC1(C)CC2(NC(c2nnsc2C)=O)C1 c1(N(C)C)ccc(CN(C(C2(F)CN(C(c3cnn(C)c3Cl)=O)C2)=O)C2CC2)cc1 C1(NC(CCCOCCC)=O)C2CC3C1C3C2C(N1CCC(O)(CC)C1)=O c1(C(N(CC(C)NC(c2ccc(-c3ccon3)cc2)=O)C)=O)cnn2c1OCC2 C(CN=c1[nH]c(=NC(C)CCn2ccnc2)[nH]c2c1CC(C)CC2)N(CC)CC C1(C(N2C(CNC(CCC(C)OCC)=O)CCC2)=O)C2CCCCCCC12 C(=O)(CC(C)(C)CC(=O)N1CCCC1C1CCN(C(c2cnnc(O)c2)=O)C1)OC N1(C(C(CSC)O)=O)C2CCC1CC(F)(CNC(=O)C=Cc1cnn(C)c1)C2 C(C(CC)CC)N(C(C(c1cnn(C)c1)NC(CCC)=O)=O)C1CC1 n1(CCN(C)C(C2CSCCN2)=O)cc(COCC(F)(F)F)nn1 O=C(O)CCCCCCC(=O)N1CCC(c2cncc(Br)c2)C1 C(C1CCCCC1)=C(C(=O)N(CC(C)N(C(CC(C)C)=O)C)C)F C1(c2n(CC(=C)C)nnn2)(NCC2CCOCC2)CCS(=O)(=O)CC1 C1(CC)CCCC(NC(C2CC(F)(F)CN2C(c2cnccc2OC)=O)=O)CC1 C(c1cccc2cccnc12)=CC(=O)NCC(CC)NC(C1CCCN1C=O)=O C(=O)(CC(F)(F)F)N(C1CC1)CC1N(C(C(CC2CCCC2)SC)=O)CCC1 c1(C(=O)NC2C(CNC(C(C(C)(C)C)N(C)C)=O)C2)csc(=NC2CC2)[nH]1 CC(CNC(=O)Cc1cncnc1O)C(F)C(=O)NCCCC(N)=O C1(C2CN(CC(=O)NC)C2)CCCCN1C(=O)C=C1CCC(C)C1 N1(C(C2OCCN(C)C2)=O)CC2CC(C1)C2NC(=O)Cn1nccn1 Cc1cnc2nccc(NC3(CNC(=O)OC(C)(C)C)CCCOC3)c2c1 C1(NC(c2cnn[nH]2)=O)CCCCC1.C12CCCC1NC(=O)C(=O)NC2 CC1(C)CCOC(C(=O)NCCCOCCNC(=O)CSc2cccs2)C1 N1(C(c2c(CC#N)cccc2)=O)CCN(C(C2(C3(O)CCC3)CC2)=O)CC(C)C1 C(C)(C)(CCC(=O)NC1CCCC(NC(c2ccc(C#N)[nH]2)=O)C1)OC n1(CC(CC)C)cc(CCNCC(=O)NCC2C(CO)C2(C)C)nn1 N1(C(=O)NC(c2cccc(C)n2)CC)CCOC2CNCC12 C1(CNC(C(C)OCCCC)=O)CCCC12CCN(C(C1(C#N)CCC1)=O)CC2 N1(C(CC(CCC)(C)O)=O)CCN(C(=O)CC2CCC(=O)NC2)CC12CCC2 C(CC(C(=O)NCCc1cnccc1C)NC(=O)CC1CC(C)(C)CO1)=CC c1(C(N2CCSCC2C)C(=O)NC(C(=O)OC)C)nc(CCCCl)[nH]c1Cl C1(CC(=O)NCC(CC)N(C)C(c2ccc(CO)cn2)=O)CCCS1(=O)=O Cc1nc(C)c(C(=O)NCC2(n3cc(CCC4CCCO4)nn3)CC2)[nH]1 C1(C(=O)OCC)OCCNCC1N(CC(N)=O)C(c1ccc(C)n(C)c1=O)=O c1(NCC2C=CC(C(=O)NCCCCC#C)C2)ncc2c(ccn2C)n1 CC1(NC(=O)Cc2cnsc2)CCN(C(=O)Cc2nc(-c3cccs3)no2)C1 c1(C(C)NC(N2CCC2C(F)(F)F)C2CC2)cn(C)c2cc(F)ccc12 c1(CCC)n[nH]cc1C(=O)N(CC(O)CNC(=O)C(C)n1cccn1)C N1(c2cc(C)nc(-n3nc(C)cc3C)n2)CCC(N)C(C)(C)C1 O=C(CCCn1cncn1)NCCNC(c1cc(Br)sn1)=O N(C(=NCC1CCC1)Nc1cccc(C2SCCS2)c1)CC1(O)CCCC1 c1(OCC(=O)OC)cccc(NC(=O)NC(c2ccccn2)CO)c1 C1(C)(NC(C(n2cc(Cl)cn2)C)=O)CCCN(C(=O)C(N2CCC(C)CC2)=O)C1 N1(CC)CCC2(CC1)CCN(S(=O)(=O)N1CC(N3C(=O)C4=C(CCCC4)C3=O)C1)C2 CC1(C)CC(NC(=O)C(F)C(F)(F)F)CCN(C(C2(C(F)F)CCCCC2)=O)C1 CC(C)C(C(=O)NC1CN(C(C2(OC(N)=O)CC2)=O)CC1C(F)F)NS(C)(=O)=O Cc1ncc(-c2cnccc2-c2nccn2Cc2cnnc(F)c2)cn1 CC1CN(C(C2CC2CF)=O)CC1n1cc(-c2ccncc2F)nn1 C1(CCNC(c2conc2C(F)(F)F)=O)CCCCN1C(C1CCCC12CC2)=O c1(C(=O)NC2(CNC(CCSCCC)=O)CCCC2)cc2ccc(Cl)nc2s1 Cc1ccn2c(=O)c(C(=O)NC3CCCCC3NC(C3CC(O)C3)=O)cnc2c1 CCC(O)C(C)C(=O)NC1(C(=O)NCCC(C)(C)CO)CC(F)(F)C1 c1(C(N2C(C(N(CC)CC3CCCO3)=O)C=CCC2)=O)ccccc1C#N C(=O)(CC(C)C)NCC(=O)NCC1CC(C(=O)NCC(=C)Br)C1 CCC(CN(C)C)C(=O)N1CCC(OCCNC(=O)CC(C)C2CC2)CC1 C(=O)(CCCCC(=O)N1CC2CC1(C(=O)NC1CC1C1CC1C)C2)OC c1(N2CCC(CC(=O)NC(c3cc(N(CC)CC)on3)=O)C2)ncc(C)c(C)n1 c1(CC)ccnc(CNC(=O)C(CO)NC(C2CC23CC3)=O)c1 C1(C(=O)NCCC(CNC(Cc2ccc(C)o2)=O)O)CNC(=O)CC1(C)C C(=O)(C(F)C(F)(F)C(F)(F)F)N(CCCNC(C1CCC(=O)C1)=O)C(C)C Cn1ccc2cccc(C(N3CCC(N4CCCCC4)C3)=O)c12 C1(C(N(C)Cc2ccccc2)=O)C2CCCC1CN(C(c1cnc(Cl)cn1)=O)C2 C1(C(N2CCN(C(C(CC)C)=O)CC2CCOC)=O)Cc2ccncc2N1 C1(CNC(Cc2cc(OC)c(C)cc2)=O)CN(C(=O)C=C(Cl)Cl)CCC1(C)C C1(C(=O)NC(CN(C(c2cnc3sccn23)=O)CC)C)CCc2c[nH]nc2C1 CCC(C)CC(=O)C(=O)NCC1CC1CNC(=O)CS(N)(=O)=O c1(OC)cc(F)c(C(=O)NCC2CN(C(c3cc(C)c(F)c(C)c3)=O)C2)c(Cl)c1 c1(NCC(C=C)C)ncccc1S(=O)(=O)NCc1cccn(C)c1=O c1(C(=O)NC2CC(NC(c3n(C)ncc3[N+](=O)[O-])=O)C2)cnc2c(c1)ncn2C N1(C(C2(CC)CCC2)=O)C2CCC1CN(C(c1ccccc1NC)=O)C2 N1(C(C2(c3c(C#N)cccc3)CC2)=O)CCC2CCC(C1)N2C(=O)C(N)=O CCCCC(O)CC(=O)N1CCC(C)N(C(c2nc(C)ncc2Cl)=O)CC1 CCCCCCC(=O)NCc1cc(C(=O)NC(C(C)C)c2nc[nH]n2)co1 C#Cc1cnc(C(=O)NCCC(C(C)C)NC(=O)C(C2CCCCC2)O)c(C)c1 N(C)(C(=NCCC#N)NCCC(C)C1CC1)C(CCC)C(=O)OC(C)(C)C c1(C(=O)NC(C)Cc2ccncc2)cnc(CNC(=O)CC2CCOC2C)nc1 C(=O)(CCCCCC(C)O)NCC(CO)NC(C(C)(C)SC)=O CC1(C)CCC(N=c2[nH]c(=NCCC34CCCC3C4)c3cc(F)cc(F)c3[nH]2)C1 c1(C(N(C)CC2(CNC(C34CCC(CO3)C4)=O)CC2)=O)ccn2nnnc2c1 C1(C(=O)NCC2(F)CCN(C(C3(CF)CCC3)=O)C2)OCC2CCCC1C2 C=CC(C)(C)C(=O)NCC1CCCN(C(=O)CC23CCCC2C3)C1 Cc1c(O)ccc(C(=O)NC2CCCC(NC(=O)C(O)C3CCCC3)C2)c1C C(C(C(=O)N1CCCC(C#N)C1)C(C)(C)C)NC(C(C)OCCC=C)=O c1(SC)nc(N2CCC(C(=O)Nc3cc(C)no3)C(O)C2)ncc1Br C1(O)(C(=O)NC2CC(OCC(=O)NCC3OCC(C)C3)C2)CCOC1(C)C C1(C(N2CCN(C)CC2CNC(=O)C(=O)NC2CC2)=O)CC2CCC(C1)S2(=O)=O N1(C(C2(C(F)F)CC(=O)C2)=O)C2CCC1CN(C(c1ccn(C(F)F)n1)=O)CC2 N1(C(c2c(CC)c(C)sc2)=O)CC(N=c2[nH]c(Cl)nc3c2COCC3)C(C)(C)C1 c1(NC)c(C(N2CC(CNC(=O)CC3CC3(C)C)C(O)C2)=O)sc2nccnc12 c1(C(=O)NCC2C(NC(=O)CC3(O)CCCCC3)CCC2)ccn2ncccc12 C1(NC(C(CC=C)CC)=O)CCC2(CC1)CN(C(C1CCN(C)CC1)=O)CCO2 c1(NCC)cccc(C(=O)NC(C)(CNC(=O)CN2CCOCC2)C2CCC2)c1 N1(C(CC(n2c(CC)ncc2)C)=O)CCCC1(CNC(=O)C(C)(C)CC)COC c1(OC)cc(Cl)c(Cl)cc1C(N1CCCC1C(C)NC(=O)CC1CCCO1)=O c1(CN(C(C2C(c3cn(CC(C)C)nc3)C2)=O)CCN(C)C)ccc2c(c1)OCO2 C1(NC(CCc2n(C)ncn2)=O)CC2CN(C(=O)C3=CS(=O)CCC3)CC2C1 N1(C(C(C)C(C)(F)F)=O)CC(CNC(C2(O)CCC2)=O)CC12CCOCC2 C(=O)(C(CNC(C1CC1Cl)=O)C(C)(C)C)N(CCC)C N1(C(c2n(CC)ccn2)=O)CCN(C(=O)CC(C)COC)C(CF)C1 c1(C(=O)NC(CCNC(C=CC(=O)OCC)=O)C)nnn(C)c1C(F)(F)F c1(OCC)ccnc(C(N2CC=CC(NC(c3cc(C(N)=O)[nH]n3)=O)C2)=O)c1C C1(NC(CCSC)=O)Cc2ccccc2C1NC(c1ccc(N(C)C)cc1C)=O CC(C)(C)CCC(=O)N1CCCC(NC(c2cnc(C(C)(C)C)s2)=O)C1 Cc1nonc1CNC(=O)C(CC1CCC1)NC(=O)C(C1CC1)C1CC1 C1(OC)CN(C(C2CCS(=O)CC2)=O)CC1NC(c1cnc(C)nc1)=O CC(C)C(C)(CNC(=O)CSc1ccoc1)NC(=O)COC1CCCC1 C1(C)(CNC(CN(C(=O)C(F)C(F)(F)F)CCC)=O)CCC(O)CC1 Cc1ccn2c(C(N3CCC(NC(=O)CC4CCC(=O)N4)C3C)=O)cnc2c1 c1(CCC(N2CC(NC(c3cc(F)c[nH]3)=O)C3C2C3)=O)cccc2ccccc12 Cn1c(-c2ccc(CSC3OCCC4CN(C)CCC34)cc2)nc2ccccc12 c1(C(N(C2CN(C(C3CCN(CCF)CC3)=O)C2)C)=O)ccnnc1O C(N=c1[nH]c(N(C)CC2CN(C)C2)nc2ccccc12)c1c(C)cco1 C1(C)(C(N2CCC(CC(=O)N(C(C(C)SC)C)C3CC3)C2)=O)CCCN(C)C1 Cc1sccc1C(c1ccccc1)NC(N1CCC(CCC(C)C)C1)=O c1(C(N2CCC(C)(CCNC(=O)C(F)F)C2)=O)cccc(C2CC2)c1Cl C1(CC=C)(C(=O)NCc2ccc(C(=O)NCCC(C)CC)s2)CCCC1 C1(C(=O)NCCOC2CN(C(C(C)=C3CC3)=O)C2)NC(=O)CC1C c1(C(=O)NCCC(C)N(C)C(C2CCOC2)=O)cncnc1C(C)(C)C C=C1CC2CC(C1)CC(c1nnnn1CCC1CC1)(NC1(CC(C)C)CCC1)C2 Cc1cc(C(N2CCC(C(=O)N(C)Cc3ncnn3C)CC2C)=O)c(O)nn1 CC(C)(C(=O)NC1CC(C)(NC(C2CC3OC2C2CC32)=O)C1)S(=O)(=O)C1CC1 N1(C(CN(C)C)=O)CC2(NC(=O)CC(C(F)F)c3ccc(F)cc3)CCC1C2 c1(C(N2CCCN(C(=O)CSC3CCS(=O)(=O)C3)CC2)=O)cn2c(n1)CCC2 N1(C(COCCCCC)=O)CCOCC(F)(CNC(=O)Cc2csc(SC)n2)C1 N1(C(C(C2CCN(C(c3ccccn3)=O)C2)C)=O)CC2CCCC2C1 c1(C(=O)NC2CN(CC3CC3)CC2O)ccc2nc(C(F)(F)F)oc2c1 C1(NC(=O)C=Cc2cccs2)CCCC12CN(C(c1occc1Br)=O)C2 CON1CCC(NC(=O)C(C)N(C)C(C2CC3(CC3)CO2)=O)CC1 C#Cc1ccc(C(N2CCC(C(=O)N(C(CC)C3CC3)C)C2C)=O)cc1C C(C(CC(F)(F)F)NC(=O)C(C1CC1)C1CC1)NC(C(C1CCC1)OC)=O c1(C(=O)NC2C(n3cc(COCC)nn3)CCC2)c(Br)c(Cl)nn1C N1(C(CNC(CCNC(C)=O)=O)=O)CCCN(C(c2cncc(F)c2)=O)CC1C N1(C(CCC2(C)CC2)=O)CCC2(C1)CN(C(=O)CCN1CCC(F)C1)C2 c1(-c2ccc(NC(C(N3C(C)CCC(N)C3)=O)=O)cc2)ccc2ccccc2c1 N1(C(C2CCN(CC)C2)=O)CCC(C(=O)NC(C2CSC2)C)CC1C c1(C(=O)NC(CN(C(=O)C(C)(O)c2ccccc2)CC)C)nnn(CC)c1C C(=O)(CCCN=[N+]=[N-])N1CCCC(CN(C)C(C2CC2c2cnc[nH]2)=O)C1 c1(C(=O)NC2C(C)CCN(C(CCCOC)=O)C2)cc2c(s1)COCC2 N1(C(c2c(C)[nH]c(C)c2C)=O)CCC(C)(C)C(NC(c2ncccc2F)=O)C1 c1(C(=O)NCC(CNC(C(C2CCC2)OC)=O)OC)cccc2nn(C)cc12 C1(CN(C(COC(CC)CC)=O)C)CCCC1NC(c1cnoc1C(C)(C)C)=O CC1CCC(C(=O)NCCC(O)CNC(=O)Cc2sccc2Br)CC1 C1(COCC)CCN(C(=NCCC(C)C)NCC23CCC(CC2)OC3)C1 c1(C(=O)NCC23N(C(C(C)OCCOCC)=O)CC(C2)C3)cc2sccc2[nH]1 C(=O)(CC(C)(C)CNC(=O)Cc1cc(CC)on1)NC(c1ccco1)CC S(=O)(=O)(c1ccc(NCc2cc(CO)ccn2)c(Cl)c1)N1CC(COC)OCC1 c1(CC(N2CCC(N(C(=O)Cc3scnc3C)CC)C2)=O)c(C)nc(C)nc1O C=C(C)CC(C(=O)NC1CC1NC(c1ccnn1CCOC)=O)OC n1(CC(=O)NCC(C(C)C)NC(=O)CC(C)n2cccn2)ccc(=O)n(C)c1=O C12(C(=O)NCCCC(C)O)CCC(NC(C3CNC(=O)CC3C)=O)(CC1)C2 c1(C(N2C(CN(C(C=C(COC)C)=O)C3CC3)CCC2)=O)ccc(OC)nc1 c1(C(N2C(CC)CN(C(C3CC3F)=O)CC2)=O)c(OC)cc(Cl)cc1Cl C1(C(=O)NCC(CC)(CC)CC)CC2CC1CN(C(C1(C)CC1C)=O)C2 C1(NC(CC(C=C)C)=O)CC2CCC1N2C(c1cnn(CC2CCCC2)c1)=O C(=O)(C(C)(CN1CCOCC1)CC)NC1CCN(C(C=C(CC)CC)=O)CC1 c1(C(N2C(C=CC(N3CC=C(C)C3)=O)CCC2)=O)ccc(C)cc1C C(=O)(C1=NOC(C)(C)C1)NC1(CC=C)CCN(C(C2(F)CCOC2)=O)C1 C#CCCCC(C)C(=O)NCC1CCN(C(c2cn3c(n2)SCC3)=O)C1 C1(CN)(NC(C2CCC(CNC(=O)CSc3nc[nH]n3)CC2)=O)CCC(C)C1 C(N=c1nc[nH]cc1C#N)C1CCC(N(C(=O)CC2COCC(C)(C)O2)C)CC1 N1(C(c2c(C)c[nH]n2)=O)CCCC2C(NC(C3COCCN3C=O)=O)C(C)(C)C12 C=CCCC(C)C(C(=O)NC1CCN(C)CC1)N1CCC(C(=O)OC)CC1(C)C N1(C(C=C(CCC)C)=O)CC(NC(=O)CNC(=O)CCC)CC(C)C1 C(=O)(CC(C)(C)c1cccs1)NCC(CCOC)NC(c1ncn(C)c1C)=O N1(C(C(=O)NCC)=O)CCN(C(C2CC(C#N)C2)=O)C(COC)C1 Oc1cc(-c2ccc(F)nc2)cnc1NC(c1ccc(Cn2ccnc2)cc1)=O C=Cn1nccc1C(=O)NCCC1(CNC(C2CCOC2=O)=O)CC1 N1(C(CC(C)N(C)C)=O)CCC(N(C(=O)Cc2cscc2Br)C)CC1 n1(CC(N2CC(C)CC(c3ccc(OC)cc3)C2)=O)ncc2ncccc12 CC#CCC(C(=O)NC1CC(=O)N(O)C1)NC(=O)COc1cc(C)on1 C(=O)(C(C)(C)F)NCCCN(C)C(C1CC1(C)C(F)(F)F)=O CCCCC(CC)CC(=O)N1C2CCC1C(CNC(C1CN3CCN1CC3)=O)C2 Cc1nc2sc(C(=O)Nc3ccc4nnc(C(F)(F)F)n4n3)cn2c1Br C1(C(=O)NCC2C(C)CN(C(=O)C(O)C3CC3)C2)CC2(C1)CC(O)C2 CC(C(=O)NCCCC1(NC(C2SCCS2)=O)CC1)C(C)c1ccc(F)cc1 C(=O)(C(C(C)(C)C)NC(=O)C(C)Cn1ccnc1)NCC1CCC(CC)O1 C1(NC(c2coc(CNC(c3cnc(O)o3)=O)n2)=O)CCCCC1F N1(CC)CC(NC(=O)CCOCCCNC(c2n[nH]c(C)n2)=O)CCC1=O c1(C(N2CCC(c3ccon3)C2)=O)cn(C2CCOCC2)nn1 C(CCCC(=O)NCC1CCCN1C(=O)Cc1n[nH]c(=N)s1)SC Cc1cc(CCC(=O)NCC2COC(CNC(c3n[nH]c(=N)s3)=O)C2)on1 c1(OC)cc(C(=O)NCC(C)NC(=O)CC2CCCCC(=O)N2)nc(C)c1 Cc1cc(C)n(CC(=O)N(CC2CCNCC2)CC2CCCOC2C)n1 C1(C(=O)NC2CCC(F)(CNC(c3c(CC)scc3)=O)C2)CCCCC1(C)C Cc1ccc2[nH]c(CN(C(C)CNC(c3ccccc3Cl)=O)C)cc2c1 N1(C(C(C2(O)CCCCC2)CC)=O)CCC(CNC(=O)C(C)(C)N(C)C)C1(C)C c1(NC(COC2CC(NC(C3CC(SC)C3)=O)C2)=O)cc2ccccc2nn1 O=CN1CCCC1C(N1CCC(c2cc(Cn3cccn3)on2)CC1)=O N1(C(C=CCN(C(=O)C(F)C(F)(F)F)C)=O)CCC(C2(O)CC2)CC1 N1(C(=O)NCC(CS(CC)(=O)=O)C)CCC2C(=O)NC(=O)C2C1 C1(N(C(c2scc(OC)c2)=O)C)CCN(C(C2(O)CC(C)(C)C2)=O)CC1C C(CCC(C)C(=O)N1CCC(N(C)C(c2cc(OC)ns2)=O)CC1)OC N1(C(C(CC)(C)O)=O)CC2(C1)CN(C(=O)C(C)OC1CCCC1)CCO2 C1(CCNC(Cc2cnc(C)o2)=O)CCCN(C(=O)C(C)Cc2ccco2)C1 c1(N2CCCC(C(=O)NCC(C3CCCO3)O)C2)ncnc2ccccc12 Cc1oc(C2CC2)cc1C(=O)NCC1CCCC(NC(C2(O)CCCCC2)=O)C1 C1(CNC(CCN(C(C(C)=NOCC#N)=O)CCO)=O)Cc2nccn2C1 CC(C)CC(O)C(=O)NCC(C)(C)OCCNC(=O)COc1c(F)cccc1F C1(CC)CN(C(c2cc(CNC(=O)CC(C)OC)ccn2)=O)CCS1 N1(CCC(=O)NCCC(C)NC(=O)CCCNC(N)=O)CCP(C)(=O)CC1 C(=O)(C(CNC(=O)CSC1CC1)CC1CCCC1)NCC(CC)(C)OC n1(CCC)nccc1C(=O)NCC1(OC)CN(C(=O)CN(S(C)(=O)=O)C)C1 c1(C(=O)NC(C2CCCN2C(c2cnn3c2CCC3)=O)C)cc(=O)cc(Cl)[nH]1 C1(C)(NC(C2(CCC=C)CN(C(=O)C(C)OCOC)C2)=O)CN2CCC1CC2 c1(OC)cc(OC)nc(CN(C)C(=O)NCc2cc(Cl)cnn2)n1 c1(C(=O)NCC(C)NC(=O)COc2ccsn2)ccc2c(c1)N(C)C(=O)C2 N1(C(C(C)OCC)=O)CC2CC(C1)CN(C(c1cnc(OC)s1)=O)C2 C1(C(=O)NCC(c2ccccc2)NC(c2occc2F)=O)(CC)CC1(F)F C1(C(N2CCC(C)N(C(c3cc(CO)[nH]n3)=O)CC2)=O)CCCN(S(N)(=O)=O)C1 CCC(C)(C)C(O)C(=O)N1CC(NC(C2(C#N)CCCO2)=O)C(CO)C1 c1(NC(CCN(C(c2ccc(CC)[nH]2)=O)C)C(C)C)ncnc(Cl)c1[N+](=O)[O-] C(c1ccc(Cl)cc1F)=CC(=O)N(CC(=O)NC1(CCCCNCC)CC1)CC C(=O)(C(F)(F)CO)NCC1(CNC(Cn2cc(C(N)=O)nc2)=O)CC1 C(C(C(C)C(C)C)NC(=O)CN(C)CCO)NC(c1c(CC(C)C)n(C)nc1)=O C1(C(=O)NCc2ncccn2)(NC(CCCNC(N)=O)=O)CC(F)(F)C1 N1(C(CC(C(=C)C)OCC)=O)CCC(C)(C)C(C(=O)N(C)OC)C1 CCCC(CCC)CC(=O)NC(C(=O)NCC(CC)(CC)CC)C1CC1 c1(C(N(C)CC2(CNC(=O)C(C)(C)c3cc[nH]n3)CC2)=O)nnc(S)n1C Cc1c(C(=O)NC2CCC(NC(=O)C(F)(F)c3cncs3)C2)ccc2c1CCC2 c1(CC)ccc(C(=O)NC2(C(N3CCC(C)(O)C3)=O)CC2(C)C)cc1 c1(CNC(C(C)OCC(C)C)=O)ccc(C(=O)NC2C3CCCC23)cn1 CC1CCC(C(=O)NCC23CCCC2CCC3)CN1C(=O)C(F)C(F)(F)F C1(CCCCNC(c2cc(OC)ns2)=O)CCCN(C(=O)C(C)(Cl)Cl)C1 N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCC2CN(Cc3cccnc3)CC12 c1(C(=O)NC2CCCN(C(C3C(C)CCCC3)=O)C2)nc2cccnc2s1 N1(C(C(C2CCC2)OCC)=O)CCC2CN(C(c3cn(C)cc3C)=O)CC2CC1 c1(C(N2CCC(CNC(C(CC=C)C)=O)C23CCC3)=O)cc(S(N)(=O)=O)sc1C C1(CNC(C2(C)ON=C(C)C2)=O)CCCCCN1C(=O)Cc1nc[nH]n1 n1(C2CN(C(CCC)CCC(=O)OCC)C2)c(O)nc2cccnc12 CC1(C(=O)NC2CC(NC(c3cccc(F)c3C3CC3)=O)C2)CCCNS1(=O)=O c1(C(=O)NC(CCCC)CNC(c2csc(C(N)=O)n2)=O)sc2nccn2c1C C(=O)(CCS(C)(=O)=O)N1C(C)(C(=O)NCCC2COCC2O)CCC1 N1(C(CC2(C(=O)OC)CN(Cc3ccnc(Cl)c3)C2)=O)CC2(CNC(=O)OC2)C1 C(C(=O)N(C)OCC)NC(C1CCN(C(C=CC=CCC)=O)C1)=O N1(C(CC(CC2CC2)NC(CCCC(=O)OC)=O)=O)CCc2c(C)cccc21 c1(C(N(CC(O)CNC(c2cnn(C)n2)=O)C)=O)cc(F)ccc1Br c1(C(=O)NC2CN(C(c3ncc(NC)nc3)=O)CC2O)cc2c(Cl)cccc2[nH]1 N1(C(COCC(=C)C)=O)CC(C)CN(C(c2cc3ccccc3s2)=O)C(C)C1 N1(C(C(=O)NC2(CC=C)CN(C(=O)C(C)C3CCC3)C2)C)CCC(O)CC1 C(=O)(NNc1ccc(-c2nn[nH]n2)c([N+](=O)[O-])c1)NCC1C(C)(C)C1(C)C Cc1nc(O)[nH]c1C(=O)N(C)CCOCCNC(c1csc(-c2cn[nH]c2)c1)=O C(=O)(CC(F)(F)C(F)(F)F)NC1CC2(CN(C(CCC(=O)NC)=O)C2)OC1 N1(C(C2(C#N)CC2)=O)CC(NC(c2cnc3ccoc3c2)=O)C(N=[N+]=[N-])C1 C1(CN(C(=O)CN2CCN(C)CC2)C)CN(C(=O)CCCC2CC2)CCO1 n1(CC(=O)NCC2C(NC(C(C)NC(C)=O)=O)CC2)ccc2nc(O)nc(O)c12 C1(C(=O)NCC=C)CN(C(=O)C(C)CSC)CCO1 C(CC(C)(C)C(=O)NC1CCN(c2cnc(F)cn2)C1)NC(C1C(C)C1)=O C1(C(N2CC(O)(C(CNC(C(C)N3CCC3)=O)(C)C)C2)=O)CC2C=CC1O2 CC1(C)CC(C(=O)NOC2CCOC2)(CNCC2(c3nc[nH]n3)CC2)C1 C1(C(=O)NC2C(C(C)C)N(C(c3cc(Cl)cc(Cl)c3)=O)CC2)CC2C(C1)C2(F)F N1(C(c2ccc(C#N)nc2O)=O)CCCC12CCN(C(=O)CC(O)C1CC1)C2 C1(CNC(CNC(=O)NC)=O)COC(C)(C)CN1C(=O)C(O)C(C)(C)C C1(CC(N2C(C(=O)OCC)CC2)=O)CN(C(=O)C(c2ccccc2)F)C(C)(C)C1 c1(C(=O)NCC(CN(C(C2C(OC)CCC2)=O)C)C)ccc2cnccc2c1 Cc1nnc(O)c(C(=O)NC2COCCN(C(=O)C(C)OC3COC3)C2)c1C c1(OC)ccc([N+](=O)[O-])c(CSCC(=O)Nc2ncc(Br)s2)c1 C(=O)(CCCCNC(C1(CNC(c2ccsc2OC)=O)CCCC1)=O)NC N1(C(CNC(C)=O)=O)CCN(C(c2cn(CCO)nc2C)=O)CC2(CC2)C1 C1(C(=O)NC(CC)(CNC(=O)C(C)c2cc[nH]n2)CC)CC=C(C(C)C)CC1 C1(CC)CN(C(=O)CC2(CSC)CC2)CCC1NC(c1nc(C2CC2)oc1C)=O C1(NC(c2c(C)c[nH]n2)=O)CCCC(N(C(=O)C=CC2CCCCC2)C)C1 C1(C(N2CC3C(CNC(Cn4ncc(CC)c4)=O)C3C2)=O)CNC(=O)CC1(C)C c1(CC(=O)NC(COC)CO)c(O)ncnc1O CCCC(C)C(C)N(C(=O)C(O)(c1ccccc1)C1CCCCC1)CCC(N)=O C(=O)(CCCCCCCCCO)N1CC(C(C)NC(CC)=O)OCC1 C(CC(F)F)(C(=O)NCC12CCC(CC1)O2)N(C(=O)CCc1ccccn1)C C1(F)(CNC(C2CCCCC2)=O)CCN(S(=O)(=O)CCc2ccccc2I)C1 c1(NC(=O)Cc2cc[nH]n2)cc(F)ccc1-c1cccc(N2CCC(O)CC2)c1 C1(NC(c2nc(C)sc2C)=O)CC2CCC1(NC(=O)COCc1nccn1C)C2 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)CNS(N)(=O)=O)C2)=O)cc1)NCC(C)C Clc1ccccc1CC1c2n(nnn2)-c2ccc(cc2)O1.C1(OBr)CCCOC1 N1(C(c2[nH]cc(C)c2)=O)CCOCC1CC(N1CCC1c1ccccc1)=O C1(NC(Cc2cn(C)nn2)=O)CCN(C(C2CCC2c2ccc(F)cc2)=O)CC1 N1(C(C(C)SC)=O)CCCC(CCCNC(c2ncsc2C2CC2)=O)C1 C(CC(=O)N=c1ccn(C2CCOC2)[nH]1)NC(C1N(CCC)CCCC1)=O Cc1noc(N)c1C(N1CC(=C(F)CNC(=O)COCC2CCCO2)C1)=O N1(C(c2coc(-c3ccccc3Cl)n2)=O)CCC2(CNC(C3CC3F)=O)CCCC12 C(=O)(C1=CCOCC1)N1C(CNC(c2c(C)cn(C)c2)=O)C=CC1 C(CC(C)C(C)(C)C)(C(=O)NCC1CCCO1)N1CC(N(C)C)C(C)(C)C1 C1(NC(c2n(CC)nnc2)=O)CN(C(=O)COCc2ccnn2C)CC1C1CC1 C1(c2cccc(Cl)c2)(Cn2cc(CCC(CC)O)nn2)CCOCC1 C1(NC(CC2(OC)CCCCC2)=O)CCCN(C(=O)C(C)=C(C)C)CCC1 C1(NC(Cc2cn(C)nc2)=O)CCCCN(C(c2cnc(Cl)c(N)c2)=O)CC1 c1(N2CC(C)(CO)OCCC2)ccc(S(=O)(=O)N2CCC(CC(F)F)C2)cn1 C1(NC(C(CN(C)C)O)=O)CC12CCN(C(c1cncc(OCC(F)F)c1)=O)C2 c1(CC)nc(C)c(C(N2CC(O)CC2C(N2CC=CC2COC)=O)=O)o1 C1(NC(CC2CN(C(c3c(C)n[nH]c3C)CC)C2)=O)CCCCC1C1CCCO1 N1(C(C2ON=C(C)C2)=O)CCC(C)CC1CNC(=O)CNc1ccccc1 C1(C(=O)OC)CCN(Cc2cn(CC(C)N(C)C(c3ccsc3C)=O)nn2)CC1 C=C(C(=O)N(C1CCNCC12CC2)CCNc1ccccc1OC)C(F)(F)F N1(C(CC(CC)C2CC2)=O)CC(CNC(=O)CCC2CCCCO2)C(C)(C)C1 Cc1cccc(NCC(=O)Nc2ccccc2OCCN2CCOCC2)c1 CCC(C)(CNC(=O)COc1ccsn1)C(=O)NCc1ccc(CN(C)C)cc1 C1(CC(=O)NC2(N(C(=O)Cn3ccnn3)C)CC2)CCCC2CC12 N1(C(Cn2ncc(C)c2)=O)CCc2ccccc2C1CNC(C12CC(CO1)C2)=O c1(OC)ncc(C(=O)NC2CCCC2NC(=O)C(C)NC(c2cccs2)=O)nc1C C(CCN(C(=O)CSc1nc[nH]n1)C)(C(C)(C)C)NC(CC(CC)OC)=O C12(CNC(CC=CC)=O)CCC(NC(c3sc(Br)cc3F)=O)(CC1)CO2 CC1CCC=C1C(=O)NC(CNC(=O)CN=S(C)(C)=O)CC(F)(F)F C(=O)(CC=C(Cl)Cl)N1CC(C(C)(C)O)(CC)C1.CCC(C(=O)NCC1CC1)n1cncn1 N1(C(C(C)(C)OC(C)=O)=O)CCCC2(C1)CN(C(=O)CC1CC1(C)C)CCO2 C1(C(=O)NCC2N(C(c3ccc(SC)o3)=O)CCCC2)CCCC12OCCO2 N1(C(c2cccc(CC)n2)=O)CC(C(N2CCOCC2CC(N)=O)=O)C(F)(F)C1 CCCC(CC)CCC(=O)NC1CC(NC(=O)C(C)OC(C)(C)C)C1 C1(C(=O)NCCCCCNC(C2(SC)CC(O)C2)=O)C(Cl)(Cl)C12CC2 N1(C(CCc2c(C)nn(C)c2)=O)CCC(NC(=O)CC2C=CS(=O)(=O)C2)C1(C)C c1(C(=O)NCC2C(N)CCC2)ccccc1NC(c1ccccc1)=O C1(CCC(=O)NCCCN(C(CC2CN(C(C)=O)C2)=O)CCO)CCCC(=O)N1 c1(NC(=O)NC2C=CC(C)(C)CC2)ccccc1S(=O)(=O)C(F)F CC#CCCC(=O)NC1(C)CCN(C(c2c(C)nsc2NC(=O)OC)=O)C1 N1(C(C2CC(=O)N2)=O)CCC2CN(c3ccnc(N4CCCC4)n3)CC2C1 CC1(CNC(=O)CC2CCN2C(c2ncc(F)cc2N)=O)CCCC(=O)N1 c1(CC(N2CCCC(N(C(CC3C(C)=NOC3=O)=O)C)C2)=O)noc(C)c1C#N C(CCCCCCCCCCO)NC(C1CCCN(Cc2n(C)ccn2)C1)=O c1(-c2c(C)c(F)ccc2)cc(C(N2CCN(C3CCC3)CC2)=O)cc2cc[nH]c12 C1(CC(=O)NCCOCCOCCNC(C2(F)CCC2)=O)CC2(CCC2)CCO1 N1(C(CSC(C)C)=O)CCCC(C(=O)NCCNC(C2(C)OCCO2)=O)C1 C(c1ccccc1OS(C)=O)=CC(=O)N(C1CCCN(C(=O)C(C)(C)CCC)C1)C c1(C(=O)NCC(CN(C(=O)CCN2CCNC(=O)C2)C)O)cccc2nn[nH]c12 C1(NC(c2c(C(C)C)noc2)=O)CCCC(NC(=O)C(F)C(C)C)C1 CCCCC(O)C(C)C(=O)NC1CCCCN(C(=O)CSc2cn[nH]c2)C1 CC(C)(C(=O)NCc1ccc(C(=O)NCCC2(C)N=N2)o1)n1cnnn1 Cc1cc(C(N2CCCC2C2CCN(C(C3CCCN3CC(C)C)=O)C2)=O)no1 c1(NCCNC(=O)C=[SH]CC(F)(F)F)cccc(C(=O)NC(N)=O)c1 CCC(C)C(O)CC(=O)N1CCCCC1C(N1CCCC(F)CC1)=O N1(C(C(=O)NCCOC)=O)CC(NC(=O)COCC2CCCCO2)CCC1C N1(C(C2CC(OC)C2)=O)CC(C)(C)C(NC(C2C=CCCC2)=O)C(C)(C)C1 N1(C(C=C(CC)CC)=O)CCC(CCOC)(NC(=O)CN(c2ccncc2)C)C1 C1(C(=O)NC2CCC2NC(C2CC(C(C)C)C2)=O)(CC)CCCC1O c1(C(=O)Nc2c(CSC)csc2)c(C)noc1C(C)(C)NC(=O)C1CC1 C12(CNC(c3[nH]ccc(=N)n3)=O)CCCCC1CN(C(=O)C=Cc1ccco1)C2 c1(C(N2CC=CC(NC(C(C(C)C)n3cnnc3)=O)C2)=O)ccc(Cl)c(C#N)n1 N1(CCCC(=O)NCC(CNC(CCNC(C)=O)=O)(C)O)C(=O)NC(C)(C)C1=O Cc1nc(C(N2CCC3(CC3C(=O)NCCCSCCO)C2)=O)ccc1C#N Cc1cc(C(=O)NCC2CCCC2NC(c2cncc(N)c2)=O)cn(C)c1=O CC1CN(c2ncnc3c2ncn3C(CO)CCCO)CC1N=[N+]=[N-] c1(CCC)nc(C)c(C(=O)NC(CNC(C2CC(=O)N(C)C2)=O)CO)o1 c1(N(CC(C)(C)C)C)nc(N2CCC3(C)C(F)(F)C3(C)C2)c2ncccc2n1 O=C(C1CCc2snnc21)N1CCCCC1C1(CNC(C2CC(O)C2)=O)CC1 N1(C(C(c2ccc(C)o2)C)=O)CCCCC1CCN(C(=O)CCCN(C)C)C N1(C(C(C)CS(C)(=O)=O)=O)CCC(C2(NC(C3(C)CC3Br)=O)CC2)CC1 C(=O)(C(CO)C(F)(F)F)NC(C(=O)N(C)Cc1ncccn1)C(C)(C)C N1(C(c2cc(C)c(C)[nH]2)=O)CC23CCCC2(C1)CN(C(=O)C(CO)C(C)C)C3 C1(C(=O)NC(c2ccc(OC(C)C)cc2)CC#N)CCCCC(C)(C)C1 Cc1cc(C(N2CC(NC(c3cc(C4CC4)[nH]n3)=O)C(F)(F)C2)=O)ccc1F CC1CC(=O)Nc2cccc(C(=O)NC3CCCC(C)CC3)c2O1 n1(CC)cc(C(=O)NCCCN(C)C(c2ccsc2C#N)=O)c(C2CC2)n1 Cc1ncc(Cl)cc1CC(=O)NC(CNC(=O)CC(C)N(C)C)CC(C)C N#Cc1cc(CCN)cc(O)c1.N12CC3(c4ccccc4)CC1(C3)C2=O C(C(COC)C(=O)NCC(C)CC(=O)NC(c1nc(C)cs1)C)OC C1(C(N2CC(CNC(C(C)=C(C)C)=O)C3(C2)CC3)=O)CCC2(CCC2)CC1 c1(OCOC)cc(F)ccc1-c1cnc(Cl)c(C(=O)Nc2nc(C)cnc2C)c1 c1(C(N(C2CCC(NC(=O)CCOCCOC)CC2)C)=O)cccn2cnnc12 N1(C(CCCOCCOCC)=O)CCN(C)C(C(=O)N(CCCCN(C)C)C)C1 C1(CC#C)CCCCN1N1CCOC(c2ccc(C)o2)C1 N1(C(C(C)NC=O)=O)CCN(C(=O)CCn2cncn2)CC1Cc1ccccc1 C1(C(N2CC(C)(C)C(CNC(C3CNC(=O)N3)=O)C2)=O)CC2CCCC(C1)C2 C1(N(C(c2n(CC)cnn2)=O)C)CCN(C(c2cnc(Cl)s2)=O)CC1 c1(CC)ccccc1OCCC(=O)N(C1CCCN(C(=O)C(C)(C)CF)C1)CC c1(N)ccc(C)c(C)c1.C(C(c1nnnn1C)OC(F)(F)F)(C(C)C)OC c1(CNC(c2cccc(Cl)c2)C(=O)OCC)cccc(N)c1C Cc1cc(C(=O)N(C)CC2CCCS2)c(C2CCCCC2)cc1F C1(C(N2CCC(NC(C(=C(C)C3CC3)F)=O)C(CO)C2)=O)CCS(=O)(=O)C(C)C1 c1(OC)ccc(F)c2[nH]c(C(=O)NC3(C)CCN(C(=O)CCNC(N)=O)C3)cc12 N1(C(C2N(C)CCC2)=O)CC2(CC(NC(C3(c4cccnc4)CCC3)=O)CO2)C1 c1(C(N2C(CNC(C3ON=C(C)C3)=O)CC(O)C2)=O)cnn2c(C)ccnc12 C1(OC)(CNC(=O)CC2COCCN2C)CCN(C(c2cnncc2C)=O)CC1 c1(CNCc2ccc(C(N3C(C)CCC3)=O)o2)cn2c(n1)CCC2 C1(C(N(CCC)CCN(C)C)=O)CCC2CCC1N2C(=O)C=CC(F)(F)F n1(CC)cc(C)c(C(N2CCOCC2c2ccccc2F)C(=O)NC2CC2)n1 N1(C(=O)CC2CC3(CCC3)C2)CC2=C(C1)CN(C(c1snnc1C1CC1)=O)C2 c1(SC)ccc(N(c2ccnc(C(N3CC(NCC(=O)OC)C3)=O)n2)C)cc1 N1(C(CC2C(C)(C)C2)=O)CCN(C(=O)CSCC(N2CCCC2)=O)CC(O)C1 CC(C)(C#N)C(=O)NCC(O)CC(=O)NCc1cccc(Cl)n1 CCCC(F)C(=O)NCC(CC(=O)N1CCC(O)(CC)C1)OC N1(C(C2CC(C)(CC)C2)=O)CCC2(CCCCN(C(=O)CCc3cnoc3)C2)C1 C#CCCN=C(NCc1ccoc1C)N1CCN(C(c2ccccc2)CC)CC1 C1(C(N(CCN(C(c2c(OC)cccn2)=O)C(C)C)C)=O)CC2(CCC2)CO1 N1(C(CCNC(C)=O)=O)CCC(O)C(NC(=O)C(C(C)C)NC(N)=O)C1 N1(CC(=O)N(C(C)C(=O)NC(C)C(=O)OC)CCOCC)CCCC1C CC1(C)CC(NC(C23CCCC2CCC3)=O)C(N(C)C)C1.C12(F)CCCN(C1)C2=O CC1CCN(C(c2ccc(F)c(O)c2)=O)C(C)C1NC(c1coc(Br)n1)=O c1(C(N2CCC(C(=O)OC)C2)=O)nc(C)c(C)[nH]c1=O.CCCC1CC(=O)N1 c1(C(=O)OC)cccc(C)c1S(=O)(=O)NC1CC1C(N1CC2CCC1CO2)=O Cc1cccc(NC(=O)CC2CCN(C(=O)Cc3nnc(O)s3)C2)c1C O=C(CCCC(F)(F)F)NC1CCSC12CN(c1nc(Cl)ncc1C1CC1)C2 C1(CNC(c2nc(CCC)sc2)=O)CN(C(c2sncc2C)=O)CC1C C12(C(=O)NC3(C)CCOCC3)CC(CN(C(=O)CC=Cc3ccccc3)C1)C2 C(=O)(CCCCCF)N1CC(O)(CNC(C2N(C(C(CCC)C)=O)CSC2)=O)C1 C1(COC)(NC(=O)CC(C)F)CCCN(C(c2c[nH]c(C(=O)OC)c2)=O)C1 C(=O)(C1=CC(O)C(NC(=O)C#CC2(CC)COC2)C1)N1C(C=C)CC1 c1(-c2c(C(=O)NCC3C(CNC(C(C)=C(C)C)=O)C3)c[nH]c2)ccc(F)cc1 c1(CC2C(=O)N2)cccc(F)c1.C(=O)(C#CC1CC1)NCC(C1CCC1)N.CNC C1(C(=O)NCCC(C)CCNC(=O)C(C)C2CC2)CN(CP(C)(C)=O)C1 C1(C)(C(N(CC(CNC(C2(SC)CCC2)=O)C)C)=O)CCCOC1 CCC(C)CC(=O)N1CC(O)CC1C(=O)NC(C1CCCCC1)C CCC(CC)C(C(=O)NCC1CC1NC(=O)CC1CCCSC1)N1CCOCC1 c1(NC(C=C)CSC)ncccc1S(=O)(=O)NCCS(N)(=O)=O C(N=c1nc(CS(C)(=O)=O)[nH]s1)C1CCCN(C(C)=O)C1 Cc1cc(Cl)c(C(=O)NCCCOCCN(C(=O)CC2OCCC2C)C)s1 c1(C(N(CC(=O)NC(C2CCOC2)C#C)C)=O)ccccc1Br CCC(C)(C)CCCC(=O)NCC1CCCN1C(C1C2Cc3ccccc3C12)=O C1(C(=O)NC(C)Cn2ccnc2)CNC(=O)CN1C(=O)CN1CCSCC1 C=CCCCCCC(=O)N1CC(CNC(=O)CC2CCN(C)CC2)CC1(C)C N1(C(C(COC)(C)C)=O)CCC(NC(c2ccc(S(C)(=O)=O)s2)=O)C(CO)CC1 C1(C(=O)NC(C)CN(C)C(C2(C(C)(F)F)CC2)=O)CC2(CCCC2)CO1 c1(C(=O)NCC(CNC(Cn2c(=N)scc2)=O)O)ccc(F)c2[nH]ccc12 C(=O)(C#CC1CCOCC1)NC1CN(C(C(c2cccc(C)c2)F)=O)CC12CC2 CC(C)CCC(C(=O)NC1CNC(=O)C12CC2)NC(=O)CCC1CCCC1 Cc1cn2cccc(C(N3CC(F)CC3CN(C)C(C3CCS3(=O)=O)=O)=O)c2n1 C#CC1C(C(=O)NCCN(C(=O)CC2CCN(C(C)=O)CC2)C)C1(C)C c1(C(=O)OC)cnc(NCC(N2CCN(C(=O)C=CC(N)=O)CC2)=O)c(Cl)c1 CC1(C)CC(C(=O)NC2(C)CCOC2=O)N(C(C2CCC2(F)F)=O)C1 C1(C)(N(C(=O)C(N)Cc2cccnc2)C)CC2(CCC2)C1 CC1CN(C(=O)Cc2cnc(C3CC3)[nH]2)CCCN1C(=O)C1=NOC(C)C1C C1(NC(CCC(C)C)=O)CCN(C(=O)COCC2CCOCC2)C(C2CC2)C1 c1(C(N(C(C)CN(C(=O)CNS(N)(=O)=O)C)C)=O)cnn2c1CC(C)CC2 C12(NC(c3nc(COC)sc3)=O)CCCC1CN(C(c1nnn3c1CCC3)=O)C2 CON1CCC(C(=O)N(C(C)CN(C)C(c2c[nH]c(=N)nc2C)=O)C)CC1 C(c1cncc(O)c1)=CC(=O)N(CC(C)NC(C1CC12CC(F)(F)C2)=O)C Cn1c(CC(=O)Cc2ccccc2CO)nnc1S.C(C=O)OCCOCCN c1(C(N2CC(OC)C(NC(=O)C3=NNC(=O)CC3)C2)=O)csc2cccnc12 c1(CNC(C2N(C(c3c(C)scn3)=O)CCOC2)=O)ccc(Br)c(F)c1 C1(C)(CNC(CC(C)SC)=O)CCCC1NC(c1ccc(COC(C)=O)cc1)=O c1(C(N2C3CN(C(C(F)=C(C)C)=O)C(C3)C2)=O)cc(-n2cccc2)ccc1Cl c1(C(N2CCN(C(COCCC)=O)C(C)CC2)=O)cccc2c1C(C#N)C2 C(=O)(C(CNC(C1CC(F)C1)=O)C(C)(C)C)NCC(C(CC)C)C c1(SC)nc(C(=O)NCC2(F)CC(NC(=O)CC(C)C3CCCCC3)C2)cs1 c1(C(N2CC(CNC(c3cccc(Cl)c3Br)=O)C2)=O)cn2cc(Cl)ccc2n1 Cc1nc(C(=O)NC(Cc2ccoc2)C(=O)NCCNC(C2CCCC2)=O)cs1 C(C)(C)(C(=O)NCC1(NC(C2CC(O)(CSc3ccccc3)C2)=O)CCC1)OC C1(NC(c2c(C)nccc2)=O)CCOC2(CCN(C(=O)C(C)SC(C)C)CC2)C1 c1(C(=O)NCC2(CCNC(CN(CCC)C)=O)CC2)cccn(O)c1=O C1(C(N2CC3C(NC(C4CC5C(C4)C5(F)F)=O)C3C2)=O)CCn2c(O)nnc2C1 c1(OC)cc(CC(=O)OCC2(c3ccccc3)COCCO2)ccn1 N1(C(=O)C(F)(F)c2cscn2)CCN(c2ccccn2)C(=O)C1 c1(C(N(CC(C)NC(CS(=O)(=O)NC)=O)C)=O)cnc2nccn2c1 Cc1cccc2c1CCN(c1ccc(S(=O)(=O)N(CC(C)CCO)C)cc1F)C2 N1(C(C2N(C(c3cc(C)nn3C)=O)CC=C2)=O)CCOCC(C)(F)C1 C(=O)(C1=CCC(C)CC1)NC(CCCNC(c1c(CC)cccn1)=O)CO c1(C(=O)NCCN(C(C2(C)CC(F)(F)C2)=O)CC)ccc(-c2nnco2)cc1 c1(C(=O)NCC(CNC(C(CC)(C)F)=O)(C)C)cc2n(n1)CC(C)NC2=O C1(C(N(CC(=O)NCc2cnc(C)n2C)CCOC)=O)CCN(C)C1=O c1(C(=O)NC(CC)C(=O)NC2CCOCC2OC)cccc2c[nH]nc12 c1(SC)cccc(C(N2CCC(NC(c3ccc(Br)o3)=O)CC2)=O)c1O c1(SCCNC(C2(C(N(C(C)C)C)=O)CC2)=O)cnc2cc(Cl)ccn2c1=O Cc1cnc(N2CCC(C)S(=O)CC2)c(S(=O)(=O)NCCc2cnco2)c1 c1(C(C)=O)sc2ccccc2c1CS(C)(=O)=O.C12CCCCC1CCC(=O)O2 c1(OCCOC)cccc(-c2nc(C(F)COC)n(C(C)CSC(C)(C)C)n2)c1 C=CCCCCC(=O)NC1CCC1NC(c1ncoc1C(C)C)=O Cc1cc(NC(=O)CC2CC(F)(F)CN2C(=O)CC23CCCC2C3)cnc1Cl C1(CCC(=O)NC)SC(=Nc2ccc(C)cc2)N(CCCc2ccc(C)o2)C1=O c1(OC)cc(C(N2CC3CC3(NCc3cncc(N(C)C)c3)C2)=O)ccc1Br c1(C(=O)NC2COCCN(C(CC(=O)N(C)C)=O)C2)cc2c(F)cccc2[nH]1 CCCCCS(=O)(=O)CC(=O)NCC(C)CN(C)C(C1CCn2cnnc2C1)=O C(CC(C)(C)CC(=O)N1CCC(C)(NC(=O)Cc2c[nH]nc2O)CC1)OC C(=O)(C1=C(Cl)CCCC1)NCCOCCNC(c1ccn(CC)c1C)=O Cc1cncc(C=CC(=O)NC2(CNC(c3occ(C)c3C)=O)CC2)c1 C(C(C)(CNC(=O)C(C)CN(C(=O)CCCn1ccnn1)C)CO)OC C(=O)(CCC(=O)N(C)C)NC(C)CCNC(C1CC(CF)C1)=O c1(CN(C(C2OCCN(C(C)=O)C2)=O)C)ccc(F)c(CO)c1 N1(C(c2cc(C)[nH]c2C)=O)CCN(C(c2cc(Br)c(C)cn2)=O)CC1C#N C1(c2nnnn2C)(NC2(C=C)CCCCC2)CCCCCCCC1 N1(C(c2c(C)coc2)=O)CCC(N(C(=O)C(C)N2CCC2)CC2CC2)CC1 c1(C(=O)NCC(C)NC(C2CC(NC(N)=O)C2)=O)c(OC(F)F)cccc1F N1(C(COCC=C)=O)CCC(C(F)C(=O)N(C)Cc2ccccn2)C1 C12(CCC(C)(C)CC1)C(=O)O2.C1(OC)CN(C(=O)OC(C)(C)C)CC1C(=O)OC N12CCOCC1C(=O)OCC(COC)n1cc(nn1)-c1ncoc1C2.CCOC Cc1ccc(C(N2CC(N(C)C)C(n3ccnn3)C2)C(=O)NC2COC2)cc1C C1(OC)CCC2(C(N3CC(NC(=O)CC4(O)CCCC4)C3)=O)CC12 c1(OC)cccc(NCC2(O)CC3CCC2C3)c1C c1(C(N2CCCC(C(C)NC(c3c(C)nc(C)s3)=O)C2)=O)ccn2cncc2c1 c1(NC(=O)C=C2CCN(C(=O)CCc3ccsc3)CC2)cncc2ccccc12 N1(CC)CCCCC1C(=O)NC(C1CN(C(=O)CCC(C)O)C1)C C1(CC=C)(NC(C2CCCC2CF)=O)CCN(C(=O)CC(C)c2ccco2)C1 C1(C(N2CCCCC(CNC(=O)CCOC3CC3)C2)=O)CC2(C1)CS(=O)(=O)C2 c1(CC(=O)NCC2CCCCC2NC(c2cncc(F)c2)=O)ccc(F)cc1Cl c1(C(N2CCC(CNC(c3scc(OC)c3)=O)C2)=O)sc(F)cc1Cl C=C(C)C1OCCC1CNC(=O)CCC(CC)NC(C1(C#N)CC1)=O c1(C(C(=O)NC(C)(C)C)N(C2CCCCC2)C(C)C)sc(Cl)cc1Br N1(C(Cc2cn(C(C)C)nc2)=O)CCC(CNC(=O)C(F)(F)C(C)O)C12CC2 c1(C(=O)NC2(C)CC(NC(C(CCC)OC)=O)C2)cc2cc(OC)ccc2o1 CC(C)(CC(F)(F)F)C(=O)NCCC1CCCN(C(=O)C(N)=O)C1 c1(C(N(C(C#C)C)CCCC)=O)sccc1CNC(=O)CCC1OCCO1 C12(NC(C(C3CCOC3)OC)=O)CCOC(CNC(c3cncnc3)=O)(C1)C2 c1(CCNC(CCOCCCNC(C2CCC(CC)O2)=O)=O)cccc(O)n1 C1(C(=O)NC2CC(CNC(C=C3CCN(C)C3)=O)C2)CCC2(CCCCC2)C1 O(P(C)(=O)CNC(=O)CCN(C(=O)C(CN(C)C)CC)CCCO)CC c1(C(=O)NCC2C(NC(c3cc(F)ccc3F)=O)CCC2)csc2c1CCCC2 c1(C(=O)NCC(CNC(CC(C)C)=O)(C)O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 c1(CNC(c2c(I)cnn2C)c2n(CC)nnn2)csc(C)c1C N1(C(Cc2cc(C)sc2)=O)CCN(C(c2ncc(F)cc2C)=O)CC1C(C)(C)C c1(C(C)C)cccc(C(=O)NC2CC(F)(CNC(c3nc(=O)n(C)[nH]3)=O)C2)c1F C12(C(N(C)CC3(CNC(=O)CCN4CCCCCC4)CC3)=O)CCC(F)C1CC2 N1(C(CCn2cnc(=N)[nH]2)=O)C(C(=O)NC2CCC(N(C)C)C2)CCC12CC2 N1(C(CC(CNC(c2ccn(C(F)F)n2)=O)OC)=O)CCOC2COCC12 Cc1nc(N(CC(C)C#N)C)cc(NCC2CCN(N(C)C)CC2)n1 C1(CC)CN(C(c2ncc(Cl)cc2Br)=O)CCN1Cc1ccc(C#N)s1 C1(NC(c2cc(CCC)[nH]n2)=O)CC2(C1)CC(C(=O)Nc1ccc(F)cc1O)C2 n1(CCC)ncnc1CCCN(CCCNC(=O)C(C)C1CCCC1)C(C)C CN1CCN(C(C2CC(NC(C3(C)CC=CCC3)=O)C2)=O)CC1=O N1(C(c2c(F)ccc(C)n2)=O)CC2CCN(C(=O)C=Cc3cncc(O)c3)C2C1 C(=O)(C(C(=O)NCC(C)N(C)C(C12CC(C)(CO1)C2)=O)C(C)C)OCC CC(C)CC(C)CC(=O)N1CCOC(CCNC(c2c[nH]cc2C(C)(C)C)=O)C1 CC1CCCN(C(=O)Cc2cncnc2)C1CNC(C1(C)CCC(=O)N1)=O CC1(C)CCC(CO)N(C(C2(NC(C3CCSC3)=O)CCOCC2)=O)C1 c12cc(ncc1C1=COCCC1)C(=O)N2.c1(OC)cc(C(F)(F)F)ccc1I C1(NC(C)C)CCN(C(c2conc2CNC(=O)NC(C)C)=O)CC1 C1(COC)CN(CCC2CCCCC2)C2(CCCCC2)C1 C1(NC(CCc2onc(C)n2)=O)CN(C(c2scc(C)c2C)=O)C(C)(C)C1 c1(C(N2CCC(C3N(C(Cc4scc(C)n4)=O)CC3)CC2)=O)cnn2c1CCCC2 N1(c2ccnc(NC3CC(C)C3)n2)CCCC2CCCCC12 C12(NC(C(C)C3CCCC3)=O)CCCCCC1N(C(=O)C=CC=C(Cl)Cl)CC2 CCC(CCC(=O)N(CC(=O)NCc1cc(C)on1)CC1CC1)OC c1(C(N(C2CCN(C(C3N(CCCC)CCOC3)=O)C2)C)=O)ccc(C)c(Cl)c1 CCCC(CCCO)C(=O)NC1CCN(C(=O)C(n2cc(C)cn2)C)C(C)C1 C1(CN(C)C)COc2ccccc2C1.C(CN=C1NCC(C2CC2)N1)OCC C(=O)(CC(O)C(C)CC)N(CCNC(C(CC)C(C)C)=O)CCOC N1(C(c2c(OCC)ccs2)=O)CCC2(CCN(C(C3CCC(=O)O3)=O)C2)C1 n1(CC)c(CCCN2CCCC(C(C(NNC(=O)OC)=O)F)C2)nc2ccccc12 C1(C(N2C(CCC)CCC2)=O)CCN(C(=O)C2CC3CCCC3C2)O1 C1(C(=O)NCC(C)NC(c2cnc(C(F)F)cn2)=O)CC(=O)N(C)C1 N1(CC(=O)NCC(CCC)NC(=O)CC2C(=O)NN=C2C)CCCNC1=O C1(CCn2cc(C3(COC)CCOC3)nn2)CCN(C(=O)C(C)CC#N)CC1 C1(NC=O)CC2(CCN2C(=O)CC2(C)CCN2C(=O)CNC=O)C1 Cc1ccc(NC(C2(NC(=O)C(C)OC3CCCC3)CCOC2)=O)cc1O C12(CC(=O)N(C3CCCN(C(=O)CCn4ccnn4)CC3)C)CC(C)(CCO1)C2 c1(OC)ccccc1C(C)C(=O)NCC1(C)CC(NC(c2cn(C)cn2)=O)C1 C1(NC(c2cnc(OC)s2)=O)CC(NC(C2(OC)CCC(C)C2)=O)C(O)C1 c1(C(=O)NCC2CCCC(NC(=O)CCc3cnc[nH]3)C2)cc2ccccc2[nH]1 CC(C)C(C(=O)NCC1(C)CCCN1C(=O)Cn1cc(C(C)O)nn1)NC(N)=O C1(NC(=O)CCc2cccs2)CC2CCC1N(c1ncncc1Cl)C2 N1(C(c2c(CCC)occ2)=O)CCCCC(CNC(c2ocnc2C2CC2)=O)C1 N1(c2[nH]c(=NCC3(CC)CCCCC3C)[nH]n2)CC2(CCCCCC2)C1 C1(OC(C)=O)CCN(C(c2cc(CNC(C3CC3C3CC3)=O)cs2)=O)C1 c12cc(I)c(cc1Nc1cnncc1C)C(=O)NC1(CO)CN2C1.CO CC1CCN(C(C2CC2F)=O)CC1NC(c1cccc(-c2nc[nH]n2)c1)=O C(=O)(CC(C)(C)CCOC)NCCN(C(CC(C=C)(C)O)=O)C1CCCCCC1 C(=O)(C(C)C(C)C)NCCC(=C)CNC(C1CCCC(O)C1)=O C1(NC(COCCC=C)=O)CN(C(=O)CNc2nccs2)CC12CCC2 C(=O)(N=c1[nH][nH]c2c1CCCC2)C1C(NCc2ccc(C#N)cc2)C1 C1(OC)CC(F)CN(C(c2ncoc2CNC(=O)CCc2nc[nH]n2)=O)C1 c1(C(C)C)ccc2c(c1)CCN(C(c1cccc(Br)c1Cl)C(=O)NC1CC1)CC2 O=C1CCC(C(=O)N2CCCC2CCCNC(c2nccn3nccc23)=O)=NN1 N1(C(C(CC)(C)O)=O)CC2(CCN(C(C3CC(F)(C(=O)OC)C3)=O)CC2)C1 C(=O)(CCCCN(C)C)NCC(C)(C1CC1)NC(c1nc(OCC)sn1)=O N1(C(C=Cc2cn(C)nn2)=O)CCC2(CCN(C(C3CC(O)C(F)C3)=O)CC2)C1 c1(CNC(CCN(C(C2(CC)CCCC2)=O)C)=O)cccc(Cl)n1 c1(C(C)(C)C)ccc(CC(=O)N(C2CCN(CCO)C2)C(=O)CCc2ccon2)s1 C1(C(N2CCC(O)(C(C)C)C2)=O)CC2(CCN1C(c1ccnn1C)=O)CC2 C(C(C)(C)CC(=O)N1CCC(C)(C(N)=O)C1)NC(C(CSC)C)=O c1(OCC)c(OC)cc(CC(C)NC(=O)NCC(C)C)cc1Cl C(=O)(C(C)(C)c1ccn(C)n1)NCC(CNC(=O)C(C1(O)CCCC1)F)OC n1(CC(=O)NC(CNC(CCc2cc(C)n(C)n2)=O)CO)cccc(N)c1=O c1(C(=O)NCCCNC(C(CC)n2ccnc2)=O)nccc(Cl)c1Cl C(=O)(C1=C(F)CN(C(=O)C#CC2CC(F)(F)C2)CC1)N1CCN(C)CCCC1 N1(C(c2ccno2)=O)CCCC2(CCCCN2C(c2c(Cl)cncc2Cl)=O)C1 C1(OC)CCC12CC(C(=O)NC(C)CCN(C(=O)COc1ccccc1O)C)C2 C1(F)(C(N2CC(N(CCOC)C)C2)=O)CCN(C(C2COCCC2C)=O)C1 C1(NC(c2nn(C)c(Cl)c2)=O)CN(C(=O)C(O)CN2CCCC2)C2CCCC12 C1(C(=O)NC(C=C)(C)C)COC2(C1)CN(C(c1cc(C)[nH]c1C)=O)C2 c1(NC(c2nn(C)cc2SC)c2n(CC)nnn2)cccc(C(=O)NC(C)C)c1 Cc1ccc(N)c(C(=O)NC2(CCNC(c3csc(F)c3)=O)CC2)c1 c1(C(=O)NCCCCC(C)NC(C2CC2(C)C(F)(F)F)=O)ccc2c(c1)OCC2 N1(CC(c2ccccc2)C)CCC(S(=O)(=O)C(C)(C)C)C1 c1(OC)ccc(CC(=O)NCC2CCN(C(C3CN(C(C)=O)C3)=O)C2)cc1F N1(C(c2c(CC)ccs2)=O)CCN(C(=O)CC2CCCCC2)C(C)C1 C1(NCCCC(=O)NCc2ccc(C#N)cc2)CCn2cncc2C1 c1(C(=O)OC)ccc(C(=O)N(C)CC2CN(C(c3ccccn3)=O)C2)cc1C C1(C(C)NC(=O)C(F)Cc2ccccc2)CCCN(C(=O)C(Cl)=CCl)C1 C1(C(=O)NC(CNC(c2ccn(C(C)C)n2)=O)C2CCC2)CN2CCN1CC2C Cc1cccc(NC(=O)CN2CCC(NC(=O)Cc3cccnc3)CC2)c1 C#Cc1ccc(C(=O)NC2CC(C)(NC(=O)C(CC)OCC)C2)o1 Cc1ccc(C2(C(=O)OCCC3CC(C(F)(F)F)C3)CCCC2)cc1 c1(C(=O)NCC2CC(NC(C=Cc3ccc(C)o3)=O)C2)ccc([N+](=O)[O-])c(N)n1 n1(CCC(=O)NC2CC3CCC2N(C(=O)CO)C3)ccc2cc(Cl)ccc12 N=S1(=O)CCC(C(=O)Nc2cnn(Cc3ccccc3)c2)CC1 c1(C(=O)NCC=CCNC(c2cnsc2)=O)cccc2[nH]ncc12 N1(C(c2c(CC)ccc(Cl)c2)=O)CC2CC(NC(=O)COCC3CC3)CC2C1 Cc1cn(C)cc1C(N1CC(O)CC1CNC(c1ccsc1C(F)F)=O)=O N1(C(c2c(C)[nH]cc2)=O)CCCC(C2CCN(C(=O)CC3CCCCC3O)C2)C1 c1(NC(c2c(C)ccnn2)=O)cnc2cnccn12 CC12CCC(C1)N(C)CCOC2.c1(C(=O)NC2CC2)ccccc1C1CCCC1 c1(N2CCC(C(C)NC(=O)C(C)(C)C(F)F)C2)nc(Cl)ncc1[N+](=O)[O-] C1(CNCc2ncn(C)c2)(NC(=O)OC(C)(C)C)CCOCC1 C12(NC(CCCC#C)=O)CCCC1CN(C(=O)Cc1ccc(Br)s1)C2 N1(C(C2C(COC)C2)=O)CCCC12CCN(C(C1(Br)CC1)=O)CC2 C1(C)(OC)CCCN(C(C2CC(O)CN2C(=O)CCC(=O)N(C)C)=O)C1 C1(CNC(CCCOC)=O)(Cn2cc(C(N)=O)nn2)CCCCC1 C1(NC(c2cccc(OC)c2)=O)CN(C2CC2)CC1CNC(C1(OCC)CC1)=O CC1CN(C(c2ncccc2Br)=O)CCC1N(C(=O)CCC(F)F)C C1(NC(C2C=CCC2)=O)COC2CN(C(c3ccc(-c4ccccc4)o3)=O)CC12 N1(C(c2c(OC)ccs2)=O)CCCC(C)(NC(c2ccn(C(F)F)n2)=O)C1 C1(NC(c2n[nH]cc2Cl)=O)COC2(C1)CN(C(C1CCCC3(CC3)C1)=O)C2 c1(CC(=O)NCC(C)(CO)NC(c2ccc(COC)[nH]2)=O)ccnc(C(N)=O)c1 C1(NC(C(C)(C)OCC)=O)CCC(C)(NC(=O)CSc2ccncc2)C1 C(CCC(C)C(=O)NC1CCCC1C(N1CCS(=O)(=O)CC1)=O)OC Cc1cccc2c1OC(C(N1CC3C(NC(C4(O)CCCCCC4)=O)C3C1)=O)C2 CC1(CNC(=O)CC2CCCC2NC(=O)CCCn2ccnn2)CC2(CC2)C1 C1(CNC(CC(C)NC(=O)CN=[N+]=[N-])=O)C(C)(C)C1(C)C c1(CC(=O)NC(CN(C(=O)C(O)CCc2ccccc2)CC)C)cnccc1Cl C(=O)(CCC(=O)NN(C)C)N1C(C(C)C)CN(C(N)=O)CC1 C=CC(C)(CC)C(=O)N1CCC(C(=O)Nc2cnc(O)c(C)c2)O1 CC(CC(=O)NCC1CCN(CCF)C1)C(C)(C)NC(=O)Cc1cc[nH]c1 N#Cc1ccc(C(N2CC(NC(C3CC(C(F)F)C3)=O)CC23CCC3)=O)cc1Cl N1(CC)CCCC1C(=O)NCC1CC(NC(c2scnc2C(F)(F)F)=O)C1 N1(C(c2c(C)snn2)=O)CCC2(CCCN2C(C2CCN(CC(F)(F)F)C2)=O)C1 N1(c2nnc(CC)n2CC2(S(C)=O)CCC2)CCC(S(=O)(=O)CC)CC1 C12(C(=O)NCCOC3CN(C(CC(CC)C)=O)C3)CCC(C(F)F)(CO1)C2 c1(NCC=C)nnc(-c2ccco2)n1CCCC.N12CCCC(C1)COC(=O)C2 C(=O)(CS(F)(F)(F)(F)F)NC1C(C)N(C(=O)CNc2cccnc2)CC1 C1(C(=O)NC2(CCNC(C34CCCC3CCC4)=O)CC2)Cc2ccc(F)cc2O1 C#CCCCCC(=O)NCC1COCC1NC(C1(F)CCN(C)CC1)=O C1(C(N(C(CNC(C=C(CC)C)=O)C2CC2)C)=O)(OCC)CCOCC1 c1(CC(C)C(=O)N(C)CC2CCCN2C(=O)CCc2cc[nH]n2)ccccc1F C1(NCc2c(N(C)C)cccc2)CCN(C(c2cc(F)nc(F)c2)=O)CC1F CC1CCC(NC(=O)Cc2c(F)cncc2Cl)CN1C(=O)CCc1ccnn1C CC1CN(C(c2cccc(F)c2N)=O)CCN1C(C1CCOC(C)(C)C1)=O Cc1ccc(=NCCC(=O)NCC(C)CNC(C2CC(C(F)F)C2)=O)[nH]c1 Brc1cc2n(n1)CCN(Cc1ccc3c[nH]nc3c1)C2 C(=O)(C(O)C(C)(C)CC)NC(CCCCNC(c1nc(CC)oc1)=O)(C)C C#CC1CCCN1C(=O)CC1CCN(C(c2ncsc2NC)=O)CC1 N#Cc1c(F)cc(C(N2CC3CC2C3NC(=O)CC2CCC(=O)N2)=O)cc1F N1(C(CCn2cnc(=N)[nH]2)=O)CCOC(CCNC(c2cccnc2)=O)C1 c1(-c2c(C)onc2)ccc2nc(NC(c3cc4cc(F)ccc4[nH]3)=O)oc2c1 c1(OC)ccccc1CN1CCC(C(=O)NC2(Cc3ccccc3)CC2)(CO)C1 c1(NC(C2C3(CC(NC(C4(C(=O)NC)CC4)=O)C3)C2)=O)cnc(C2CC2)nc1 N1(C(CSC)=O)CC(CNC(=O)C(C)c2cccs2)CC12CCC2.C12(CC1)C(=O)N2 c1(N(CC(=O)OCC2CCCC3(CC3)C2)C)cc(Cl)ccc1Cl C1(OCC)CCC(COC(c2cnn(Cc3ccccc3)c2)=O)CC1 S(=O)(=O)(c1cccc(C(=O)NC2CC2NC(=O)CC#N)c1)N(C(C)C)C C1(C(=O)NCC(C2CC2)N(C(=O)CCCCF)C)(NC(C(CC)C)=O)CCCCC1 c1(C(N2CC(NCC3(O)CC3)C(C3CC3)C2)=O)cc(O)c2cc(F)cc(F)c2n1 Cc1c(C(N2CCC3(CC3C(=O)Nc3cncnc3Cl)C2)=O)cccc1C(F)(F)F C1(C(C(=O)N(C2CCN(C(c3sccc3Cl)=O)C2)CCC)O)CCOCC1 N1(c2snc(C(C)C)n2)CCCC2CCN(C(c3ccc4nc[nH]c4n3)=O)CC12 C1(CNC(C(C=C=C)C)=O)CN(C(=O)COc2nc(O)nc(O)n2)CC12CC2 N1(CC)CCN(C(=O)CC2C3CCCC3N2C(=O)Cc2ccn(C)c2)CC1C N1(CCC)CCC(C(=O)NCC2CCCC2NC(=O)CCN(C)C(C)=O)CC1 C1(CC)CC(O)CN1C(=O)CC1C2CN(C(c3cnc(C)o3)=O)CC12 C1(C(=O)NCC(C)CN(C)C)COC2(C1)CN(C(=O)CCc1ccsc1)C2 C(C(C)CC(=O)N1CCC1CNC(C1C2CCC1(c1cccnc1)C2)=O)OC c1(CN(C(=O)CCNC(C(C)Cc2cn(C)nn2)=O)CC)n[nH]c2ccccc12 N1(C(C(F)OC)=O)CC(NC(c2cc(N)ccc2O)=O)CC12CCOCC2 C1(CNC(C2(C(N(C)C)=O)CC2)=O)CCN(C(=O)C=Cc2ccco2)CC1O CC1CN(C(=O)CCCC2CCCCC2)CCC1CNC(=O)CC1(C)CC1 C=CC(C)(C)CC(=O)N1CCC(NC(=O)C(c2cccc(C)c2)C)C12CC2 N1(C(Cc2nc(C)oc2)=O)CCCC(NC(=O)C(C)C(C)(F)F)C1C c1(C(=O)OC(CCCC#C)C)cccc2cccc(O)c12 c1cc2[nH]c(=NCC3CC4(CCO3)CC4)sc2cn1 C(C(C)(C)CC(=O)N1CCOC(C)C1C)NC(c1c(C)cncn1)=O C1(C#C)(C(N(CC#CC)CC#C)=O)CN(C(c2ccncc2N)=O)C1 N1(C(c2c(CC)nn[nH]2)=O)CCCC(F)(CNC(C2(n3cccn3)CC2)=O)C1 Fc1cc(CCN(C2CC(c3ccccc3)C2)CC(N2CCCCC2)O)ccc1Cl N1(C(CC(CC)OC)=O)CC(CNC(c2scnc2C2CC2)=O)C2(CC2)C1 CC1CC(CCOC(=O)C(C)(C)n2ccc(C(=O)OC(C)(C)C)n2)CCO1 C1(NC(C(C(C)C)F)=O)CCC(C)N(C(=O)CCNC(c2ccncc2)=O)C1 C1(C(=O)OC)COc2ccccc2C1.C(CCCC#N)(C(=O)OC)O c1(C(=O)NC)cccc(C(=O)NCC#CCNC(=O)CC2CCCC(O)C2)n1 N1(C(CC=CC)=O)CCN(C(c2cccc(SCCC)c2)=O)C(C(C)C)C1 N(C(=NCC(C)(O)C1CC1)NCC1CC(=O)N(CC)C1)CC1CCC(CC)O1 N1(C(C2(C(=O)NC)CC2)=O)CC2CC(C(=O)Nc3cccc(F)c3)CC2C1 C(=O)(CC(O)C(C)CC)NCC1(O)CN(C(c2cnc(CC)nc2C)=O)C1 C12(CNC(c3ncsc3Br)=O)CC1CN(C(=O)CC1(C(F)F)CC1)C2 Cn1cc(C(=O)NCC2CC(F)CN(C(=O)COCCF)C2)n(C)c1=O C=C(C)CC(C(=O)N1OC2CCC1CC2)NC(C1CC=CC1)=O CC1(C)CC(CCNC(=O)C(C2CCS(=O)(=O)CC2)F)C(=O)O1 c1(C(=O)NCc2cc(C(=O)NCCCC#C)no2)cc(C)c(F)cn1 c1(C(=O)NCC2COC(NC(=O)C(=O)NCC(F)F)C2)ccc2c(c1)N(C)CC2 Cc1cnc2nc(=NC(=O)CN3CCOC3=O)[nH]n2c1 N1(C(C2CCCCC23CC3)=O)CCN(n2cc(-c3c(C)cn(C)n3)nn2)C(CF)C1 c1(C(N(CC(CNC(c2cnc(C(C)C)[nH]2)=O)O)C)=O)ccc2[nH]ccc2n1 N1(C(C(CC)OCC)=O)CCN(C(=O)Cc2c(F)cccc2F)C(CCO)C1 C(=O)(C(F)C(=O)N1CC(CNC(c2sc(C)cc2C)=O)C1)OCC c1(C(=O)NCC2(NC(C(C)OC)=O)CCCCC2)cnc2ncccc2c1 Cc1ccc(C(F)(F)F)cc1CN(C1CCN(Cc2c(C)nn(C)c2C)CC1)C c1(C(=O)NC(C2CN(C(=O)CC3(C4CC4)CC3)CCO2)C)cccc(CO)c1 C1(NC(C(C)NS(C)(=O)=O)=O)CC2CN(C(c3cccc(C(C)(F)F)c3)=O)CC12 C1(CNC(CC=C)=O)C2CN(C(=O)C(C(C)C)c3ccncc3)CC12 N1(C(C2(C(C)C)CNC(=O)C2)=O)CCCC(CC(=O)NCC2CC2)CC1 C1(CC(N2CCC(NC(C(C(C)C)NS(N)(=O)=O)=O)CC2)=O)CCC(=O)NC1=O C1(N(c2c(OC)nc(Br)cn2)C(c2coc(C)n2)=O)CC2(CCNCC2)C1 N1(C(C(CC)OCC)=O)CCN(C(=O)C(C)(C)CCOC)CC1c1cccnc1 c1(C(=O)NC(C)CCNC(c2coc(C#N)c2)=O)ncnc2c1ncn2C1CC1 c1(C(c2nnnn2CCSCC2CC2)NCC(CO)C2CC2)ccc(Cl)cn1 C1(CNC(Cc2n(C)ccn2)=O)N(C(=O)CC(C)(C)C#N)CCC1(C)C c1(C(N2CCC(C(C)NC(=O)CCn3ccnn3)C2)=O)ncn2cccnc12 C1(C2CCN(C(=O)CCC3OCCO3)C2)(NC(C2CCn3ncnc3C2)=O)CC1 Cc1cc2cc(C(N3CCCC(CN(C(=O)C(C)CO)C)C3)=O)ccc2cn1 C=C(C)CC(C)(C)C(=O)NC1CC(NC(c2c(C)nc3sccn23)=O)C1 c1(C(C(=O)N(CCC)CCNC(c2nocc2C)=O)C)ccc(F)c(Cl)c1 N1(C(C2N(C)CCN(C(c3c(CC)occ3)=O)C2)=O)CCC(F)(F)C(F)C1 N1(CCCCCNC(C(CC)N(C)C)=O)CCN(C(=O)CC2CCN(C)C2)CC1 c1(C(=O)NCC2N(C(C(CC)F)=O)CC2)cnc2sccc2c1 c1(C(=O)NCC2CCN(C(C(C)n3cccn3)=O)C2)cc2c(s1)CCCC2 CC(CC(=O)NC1CC(N(C)C(C2CCCO2)=O)C1)N(C)C CCC(CCC(=O)N(CCNC(=O)C(n1cnc(C#N)n1)C)CC)OC C(=O)(CCCCc1ccc(OC)cc1)NCC(CC)(C)NC(=O)CS(C)(=O)=O C(=O)(CCCCC(C)=O)NCCC1(C(=O)NCC(C(C)C)OC)CC1 C(N=c1[nH]cnc(NCCS(N)(=O)=O)c1C)C1(OCCSC)CCC1 N1(C(c2c(CC)onc2)=O)C2CCC1C(CNC(c1cc(OC)ccc1N)=O)C2 Cc1cc2ccc(C(=O)NCC(O)CN(C)C(C3CC(O)C3)=O)cc2o1 Cc1cc(C)c2nc(N3CCCCC(CNC(C4(C)CCC(=O)N4)=O)C3)sc2c1 C1(CC(=O)N(C2CCN(c3ncc(C(C)(C)O)cn3)C2)CC)CCCNC(=O)C1 c1(CCC(N2CCCN(C(COC(C)(C)C)=O)CC2)=O)cccc2ccccc12 N1(C(C2CC(=O)NCC2)=O)CC2CC1CN2C(c1cc(C2CCC2)n[nH]1)=O CC1CN(C(=O)C(C)(C)CF)CC1NC(C1CCN(CCS(N)(=O)=O)CC1)=O c12ncc(cc1F)-c1cccc(c1)N2.c1(SC)cccc(C(C)OCC(=O)O)c1 c1(C(=O)NC(C(=O)N2C(CC)CC2)CO)ccn2ccccc12 C(=O)(C(O)CC(F)F)N(C1CCCN(C(C2CCC(F)(F)CC2)=O)CC1)C C1(C(=O)NC2C(OCC)CCC2)CCCCCN1C(c1ccsc1)=O N1(CCC)CCCC(C(=O)NC(CNC(=O)CCc2cnc(C)o2)C(C)C)C1 CCC(C)C(C(N)=O)NC(c1csc(CNC(=O)C=CC2CCC2)c1)=O Cc1cc(Br)cc(CNC(C2CC(Cc3c(Cl)cc(Br)c(O)c3Cl)C2)=O)c1O C(=O)(C1=CC2CCCC12)N(CCNC(c1n(CC=C)ccc1)=O)C(C)C C1(C(N(CC(C)NC(C2(C3CCOCC3)CC2)=O)C)=O)COC2(CCC2)CO1 Cc1cnc(C(=O)NC(C)(C)C(=O)N(CC(C)O)C)cn1 c1(C(=O)NC2CN(C(c3c(CC)ncnc3)=O)CC2C)c(F)ccc2c1OCC2 c1(C(=O)NC2(C(=O)NC3C(C)CCC3)CCCCC2)cn(C)c(=O)cn1 C1(CNC(CC(=C)C)=O)CCC(F)(CNC(=O)CCCC2CC2)C1 C(N=c1[nH]c(=NCC2(CO)CC23CCC3)c2sccc2[nH]1)C1C(CCC)C1 c1(OC)cc(C(=O)NC2CCCCC2C(=O)NCc2cnc[nH]2)ccc1C C1(C)(CC(=O)NCc2nc(CCC)oc2)CCN(Cc2ncc[nH]2)C1 c1(CC)c(C(=O)N(C(CNC(=O)C(C)(C)CC#N)C2CC2)C)cccc1C c1(OC)cc(O)c(-c2ccccc2C(N2CCCOCC2C)=O)cc1OC N1(C(C(CC=CC)C)=O)CC(C(=O)N(CC(C)(C)N(C)C)C)CC(C)(C)C1 N1(CCCC(=O)N(C2CCN(C(C3CC3(C)C)=O)CC2)C)C(=O)NC(C)(C)C1=O N1(Cc2cccc(OCCO)c2)CC2(CO)CCC2(CO)C1 N1(CCN=C(NC(COC)C)NCc2cnnn2C)C(=O)NC2(CCCC2)C1=O c1(C(=O)NCCC2OCCN(C(C(CSC)O)=O)C2)ccc(O)cc1C N1(C(C(C=C=C)C)=O)CCN(C(c2ocnc2C2CC2)=O)CC1C(F)F N1(C(c2nncc(OC)c2)=O)CCN(C(c2ccoc2C2CC2)=O)C(C)C1 C1(=O)C(C(C)C)C2CCN(CC2)Cc2ccc(cc2)O1.N1(C(=O)OCC)CCCC1 Cc1nn(C)c(C)c1CNC(=O)C(CO)NC(c1ccc(F)s1)=O c1(C(=O)NCC2(CNC(=O)CCOCC(F)F)CC2(F)F)cnc(O)c(F)c1 CC1(C)CC(=O)C(N(C2CC2)Cc2cn(C(C)(C)C)c(=O)nc2O)C(C)(C)C1 c1(CC(=O)NC2C(NC(c3ccc(CC)cn3)=O)CCC2)cn2cc(C)sc2n1 N1(C(CN2CC(=O)NC2=O)=O)CCOC2CN(C(C3CCCC3(F)F)=O)CC12 CC1(C)CN(C(=O)C=CCN2CCOCC2)CC1CNC(C1SCCCS1)=O c1(C(=O)NC2(CCCNC(C3(CC)CCOC3)=O)CC2)ncnc2cc[nH]c12 c1(N2CCC(NC(=O)CCC(F)(F)F)C(CO)CC2)nc2cccc(Br)c2o1 c1(C(N(CCN(C(C2CN(C(=O)NC)C2)=O)CC)CC)=O)cc(C#N)[nH]c1C c1(OC)ccc(F)c(C(=O)NCC2(O)CC(NC(c3cc(CO)[nH]n3)=O)C2)c1F C(=O)(C(C(C)C)c1ccc(Cl)cc1)NC(CN(C(c1cc(C)sn1)=O)CC)C CC(C(=O)NC(C1CCCCC1)CCO)S(=O)(=O)C1CCOCC1 C1(CC)CN(C(=O)C=Cc2cn[nH]c2)CCC1NC(c1cccc(Cl)n1)=O Cc1ccnc(F)c1-c1cnccc1C(=O)NCc1cc(Cl)cc(Cl)c1 c1(OC)ccc2c(c1)CC(C(=O)NCC1C3CC1N(C(=O)C(C)(C)SC)C3)CC2 N1(C(C2CN(C(CC3(NC(C)=O)CC3)=O)CC2C)=O)CC(C)(C)OCC1C C1(CNC(c2nc(OC)sc2)=O)CCN(C(=O)C=CCO)CC1 Cc1nc2c(F)cccc2cc1C(=O)N(CC(C)NC(=O)C(C)(C)C(C)O)C Cc1ccc(C(N2CC(N(C(=O)CC(C)n3cccn3)C)C2)=O)c(O)c1C N1(C(C2CC(=O)N2)=O)CCC(NC(=O)CC2CCC(F)(F)CC2)C(F)C1 N1(C(C=C2C(C)(C)CCCC2)=O)CCc2ccc(Br)cc2C1C(F)(F)F Cc1cc(-c2cn(C3CC4(NC(c5cccc(F)c5Cl)=O)CC34)nn2)cc(Cl)c1 N1(Cc2ccc(CC(C)C)s2)CCC(C(C(F)(F)F)NC(=O)CO)CC1 C1(CC)CCN(C(=O)CC2OCCC2C)C1CNC(=O)Cc1c[nH]nc1C c1(CC)occc1C(=O)NCC1(F)CC(NC(=O)COCc2ccccc2)C1 C1(O)(C(N2CCN(C(=O)Cc3ccns3)CC2C2CC2)=O)CN2CCC1CC2 c1(SCC(=O)NC(CNC(CC(C)C)=O)CO)cccc(F)c1 S(=O)(=O)(c1ccc(Br)cn1)N1CC(C(=O)NCCC2CC2)C1 c1(OC)c(C)cc(C(N2CCC(CNC(=O)CCCCBr)C(F)(F)C2)=O)cc1C S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(CNC(c2ncc(C)nc2)=O)CC1 CCC(C(C)CN(C)C)NC(C1CCN1C(=O)CC(Cl)Cl)=O C=CC1(C(N2CC(C)(C)C2C2CC2)=O)CCN(C(c2ncsc2C)=O)CC1 CC1(c2nc(C3(c4ccc(Br)cc4)CCCCC3)no2)CCC(C(F)F)CC1 C1(F)(CNC(CCC(=O)NC)=O)CCN(C(=O)C(c2ccccc2)C)CC1 CC(C)C(O)CCN=c1[nH]c(=NCc2cn(C)cn2)[nH]c2c1CSC2 C1(N(C(C2C(=C)C2)=O)C)CCCCN(C(=O)Cc2cncn2C2CC2)C1 c1(C(=O)NC(C)CCCNC(=O)Cc2cn(C)nn2)cc2c(O)ncnc2cn1 N1(C(Cn2c(C)nnn2)=O)CC2CC1CN(C(=O)CCOCCOCCCO)C2 C1(c2nn[nH]n2)(C(N(C2CC(N3CCCNC3=O)C2)C(C)C)=O)CCCC1C CC1CN(C(C2CCC(C3CC3)N2C(=O)CC2CCC(C)(C)C2)=O)CCS1=O Cc1cccc(C(CN)C(=O)NCC(c2cccc(O)c2)O)c1 N1(C(C(C2CCCCC2)OC)=O)CC(O)CC1CNC(C1(CCF)CCC1)=O C1(NC(=O)CC(C2CC2)NC(c2cccc(=S)n2O)=O)CCn2ncnc2C1 c1(C(N2CCC(C)(CNC(C(C)N(C)C)=O)CC2)=O)cc2n(n1)CCCO2 Cc1cc(C(N2CC(CCCCNC(=O)Cc3cnn(CC)c3)C2)=O)n[nH]1.C(C)C N#Cc1ccccc1CN1CCOC2CC12.N12CCCC1CCC2=O N1(C(C2C(=C)C2C(=O)OC)=O)C2CCC1CC(CNC(=O)C(CC)CC=CC)C2 C1(NC(c2c(C)c(Cl)ccn2)=O)COC2CN(C(=O)CCCc3ncco3)CC12 c1(C(=O)NC2C(CNC(C(CCCC)O)=O)CCC2)cc([N+](=O)[O-])oc1C c1(C(=O)NCCN(C(C2(C(C)C)CCCO2)=O)C)csc2nccn12 Cc1ccc2cc(C(=O)N(CCNC(=O)C(N3CCOC3=O)C)C3CC3)cn2c1 C(=O)(CC(C)(C)C(C)(F)F)NC1CN(C(C=Cc2cn(C)nn2)=O)C(C)(C)C1 CC(O)CCCCCC(=O)N1CC(NC(c2cn[nH]c2)=O)CC12CCC2 C(C(C)(C)C1=CCCC1)NC(CC1CCCN(C(C(C(C)C)CN(C)C)=O)CC1)=O c1(N2CCC3(CN(C)C3)C2)nc(=NCP(C)(C)=O)[nH]c2c1CCCC2 C(CC(=O)N1CC(CN=[N+]=[N-])C1)(C1CC1)NC(C(=O)NC(C)C)=O CC(C)(C)CC(=O)NCC1(C(C)(C)C)CCN(C(=O)COC(C)(C)C)C1 N#Cc1ccc(Br)cc1CNC(=O)CN1CCN(Cc2c[nH]ccc2=N)CC1=O C1(O)(C(C)NC(C2CC2C(F)F)=O)CCN(C(=O)CC2(C)CCOCC2)C1 N1(C(C)=O)CCN(C(=O)CCOC(CC2(OCC)CC2)=O)CC(O)C1 O=C(CCCCC1CC1)NCC(O)CCNC(=O)C(c1ccccc1)O C(CC1C(=O)N1)N(C)C.c1(CNC(=O)OC(C)(C)C)ccc(F)nc1 N1(C(C2CC=CC(O)C2)=O)CC2(CO)CC1(C(=O)NCCc1ncccc1F)C2 C1(NC(CSCC=C)=O)CC(F)CN(C(c2ccc(O)c(CC)c2)=O)C1 Cc1ccc(Cl)cc1C(=O)N(C)CC1CCCN1C(c1cc(C(F)F)no1)=O c1(C(C(=O)NCC(Cn2cc(C3(C)CCCO3)nn2)(F)F)O)ccc(F)c(Br)c1 N1(C(=O)Cn2cc(CC(O)C3CC3)nn2)CC(CO)CC1Cc1ccc(F)cc1 C12(C(N3CCC(C(N4CC(C)(CO)C4)=O)(CC)C3)=O)CCCC1C2(F)F CCCS(=O)(=O)CC(=O)NC1(CCNC(C2(O)CCSC2)=O)CCCC1 CC1CN(C(C2CCCN2C=O)=O)CCN(C(=O)C(O)Cc2ccccn2)C1 Cc1cc2[nH]c(C(=O)NCCCN(C(=O)C(F)CC(C)C)C)nc2s1 c1(C(N2CC(C(N3C(CCOC)CCCC3)=O)C2)=O)cccc2ncc(Br)cc12 Cc1scc(C(=O)NCCC2(O)CN(C(c3ccncc3O)=O)C2)c1C c1(C(N(C(C)CNC(C2CCCC(O)C2)=O)CC)=O)cccc(C2CC2)n1 C1(NC(C(C)OCc2ccccn2)=O)CCN(C(=O)Cc2cncn2C)CC1C CCC(CC(=O)NC(C)(C)C=CC(=O)NCC(C)C(F)F)C1CCC1 N1(CC(=C)Br)CCc2ccccc2C1CNC(c1cncc(F)c1)=O c1(C(N(CC(CNC(C(C=C)c2ccccc2)=O)C)C)=O)cc(CC)cnc1O N1(C(CCc2ccc(C)o2)=O)CCC(C)(C)C(NC(C2(C)CCCCC2)=O)C1 C12(NC(=O)OC(C)(C)C)CCN(C(C3(C#N)CC=CC3)=O)CC1C2 c1(OCC)ccc(CC2N(C(CCNC(C3(C)CCNC3=O)=O)=O)CC2)cc1OC c1(C(N2CCN(C(CC(CC)C3CCC3)=O)CC2)=O)cccc2c1OC(C)(C)C2 C1(CC(=O)OC)CC(F)(F)CN1C(c1c(-c2cc(OC)nn2C)cccc1)=O O=C(C1=COCCC1)NC(C(N1CCOC(CO)C1)=O)C1CCCO1 N1(C(CNC(C=CC(CC)C)=O)(C)C)CCN(C(=O)C(C)(C)CO)CC1 N1(C(CCOCCOCC)=O)CCC(C(=O)NC(CO)(CO)CO)C(C)C1 c1(OC)cccc(OC)c1C(=O)NC1CC(NC(C2CSCN2C)=O)C1 c1(C(C2CCOCC2)(C)NC(CCSCC)=O)ccc(C(F)(F)F)cc1 c1(C(=O)NC2C(NC(C(CCCC)C)=O)COC2)ccc2c(c1)OCC2 c1(NCCNC(=NCC)NCCn2cc(Br)nn2)ccc(C)cc1C C(=O)(C(C)CCC(C)(C)C)NCC1(CNC(CC(CC)C(C)C)=O)CCCCC1 N1(C(Cc2c(-c3cccs3)nc(C)s2)=O)CC(NC(=O)C(C)O)CCC(O)C1 Cc1ncccc1C=CC(=O)NCC1(F)CN(C(=O)C(C)(C)O)C1 N1CCS(=O)(=O)CC1.n1(CC)c(C2CCN(C(c3nc(C)cs3)=O)CC2)nnc1O C1(CC(N2CCC(C(C)O)C2)=O)CCN(C(=O)C(C)n2cccc2)CC1 N1(C(C(C(CC)CC)OC)=O)CCOC2CN(C(=O)CCP(C)(C)=O)CC12 N1(C(C2CC3CC2CC3NC(C2(O)CCC2)=O)=O)CC2CCC1C(O)C2O CC1CN(C(c2cc3sccc3[nH]2)=O)C(C)CN1C(c1ccc(=O)n(C)n1)=O C1(C(=O)NCCC(C)(C)NC(C2CC3(CCC3)CO2)=O)CCCCC12CCC2 c1(-c2cc(C(=O)NC3C(NC(CSCC(N)=O)=O)COC3)no2)ccccc1Cl c1(C(=O)NC(c2nocc2C(=O)NC2(C)CSC2)C)nc(=N)cc[nH]1 C1(C(=O)NCc2cccc(C(N3CCC(CC4CC4)C3)=O)n2)CC2CCCC2C1 N1(C(c2scc(C)c2)=O)CC(NC(c2csc(C(C)(C)C)n2)=O)C2(CCC2)C1 c1(C(=O)NC2CC23CC(NC(=O)C(F)Cc2ccccc2)C3)cc2c(s1)CCC2 C12(C(N3CCCC(CCNC(C(C)CF)=O)C3)=O)CC3CC(CC(C3)C1)C2 c1(CNC(CN2CCN(C(CC)CO)CC2)=O)ccc2c(c1)CCC(C)(C)O2 c1(C(=O)NC2C(N(C(CCc3cc(C)on3)=O)C)CCCC2)cncc(Cl)c1C C1(C)(NC(CN(CCOC)C)=O)CCN(C(=O)C(C)(C)O)C1 C1(NC(C=CCC2(NC(C(F)=CCC)=O)CCC2)=O)CCN(CC)C1 N1(C(C(c2ccco2)NC(CCOC)=O)=O)CCCN(C)CCC1 C1(C(=O)NCC23OCC(NC(C(C)(C)OC)=O)(C2)C3)COc2cc(F)ccc2C1 c1(C(=O)OCC)ccccc1NC(C1CC1NS(=O)(=O)CC)=O.C1CC1SC N1(C(=O)OC(C)(C)C)CC2(CCCN2S(=O)(=O)Cc2ccccc2F)C1 c1(CC(=O)NC2(CC(=O)NC(CC#C)CO)CCCC2)ccccc1F Cc1nc(Cl)nc(NC(c2cccc(C(F)(F)F)c2)(C)CO)c1F c1(C(=O)NCc2cccc(OC(c3ccccc3Cl)(C)C)c2)cc(F)ccc1Br C1(CCNC(c2n(CC)ncn2)=O)CCN(c2ncncc2I)CC1 S(=O)(=O)(c1ccc2c(c1)CCN2C(c1csc(Cc2ccccc2)n1)=O)NCC N1(C(C(=O)N(C)C)=O)CCC(C2CCN(C(C3CC4(C3)CC(F)C4)=O)C2)C1 c1(C(=O)NCC(C)N(C(c2cnn(-c3nccs3)c2)=O)CC)[nH]c(C)nc1C c1(C(=O)NC2C(NC(c3nc(CCC)oc3)=O)C2)cncc(-n2cnnn2)c1 C1(C(=O)NC(C(C)(C)C)CNC(C2CC2(F)F)=O)CC2C(C1)C2(F)F N1(C(c2c(CC=C)cccc2)=O)CC2(CNC(C3(C)CCCO3)=O)CC(F)(C1)C2 C(=O)(CCCCCC(C)O)NCC1C(C(=O)NC(c2ccc(F)c(F)c2)C)C1 C(=O)(CCC(CC)NC(=O)C(CN(C)C)CC)N1C(C#C)CC1 C(CC)(C(=O)N1CCCC1C(=O)NCC(C1CCCC1)C)=CC N1(C(C2N(C(C3N(C)CC(C)(C)C3)=O)CC=C2)=O)CC(C2CCCCC2)C1 Cc1sc(Cl)c(C(=O)N(C)CC2CCN(C(c3ccc(C(N)=O)cc3)=O)C2)c1C C1(OC)CC(C(=O)NC2CCC2CC(C)(C)C)N(C(C23CCCC2C3)=O)C1 c1(OC)cc(=O)n(C)cc1C(=O)NC(CO)C(C)NC(=O)C(C)N1CCC1 C1(OC(C)=O)CCC(CN=C(NC2CC2)NC2CC(OCC3CC3)C2)CC1 c1(C(N2CC(CNC(CCC)=O)N(C)CC2)=O)cc2c(C)cccn2n1 C1(CC=C)(NC(=O)CCSCCOC)CCN(C(=O)C=Cc2cnc[nH]2)C1 C1(NC(C2C(C)C2(F)F)=O)CC2C1CCN2C(=O)CN1CCN(C2CC2)C1=O C(=O)(C(C)CCOC)NC1CC(CCC(=O)N(CC)CC2CCOCC2)C1 c1(C(=O)NC23CCC(C2)N(C(=O)C2=CCCSC2)C3)c[nH]c2c(Cl)cccc12 C1(NC(c2cn(CC)nc2C(F)(F)F)=O)CCN(C(=O)Cc2ccco2)CC1C C1(C(=O)NC2CCCN(c3ccnc(Cl)n3)CC2)CC2CC1C1C2C1(F)F C1(CNC(C2CC3(CCC(NC(C)=O)CC3)C2)=O)CCC2(CCC2CCO)O1 CCCCC(CC)CCC(=O)NCCOCCNC(=O)CSCc1cccnc1 S(=O)(=O)(c1cnn(-c2ccccc2)c1F)NC(c1ccc(C(CC)C)cc1)=O c1(CC(N2CC(O)(C(C)NC(=O)C(F)=C3CCCC3)C2)=O)cccc2c1OCC2 CCC(CN(C)C)C(=O)NCC(C(C)(C)C)NC(C1C=CCC1)=O C1(C)(CCNC(C(CCC)N(C)C)=O)CCCN(C(=O)C(CC)OC2CCCC2)C1 C(C(C)C(=O)NCC(C1CC1)N(C(=O)C(C)(C)c1cnsc1)C)SC c1(NC(C2CC(F)CN2Cc2nc3ccccc3[nH]2)=O)ccc2ncnn2c1 C1(C(=O)NCCN2C3CCCC2CC(O)C3)CNc2cccc(Br)c2O1 c1(C(=O)NC(C)(CNC(c2cnc(Cl)s2)=O)C2CCC2)ccnc2cc[nH]c12 C(=O)(C(F)C(C)(C)O)NCCCN(C(C12CCC1C2)=O)CC c1(C(C(N2CCC(CN(C(C3(OC)CC3)=O)C)C2)=O)(C)C)ccccc1F C#CC(CN(C(=O)COC1CC(NC(=O)C=CCO)C1)C)C(C)C Cc1ccc(Cl)c(O)c1C(=O)NCCC1(O)CN(C(C2CC23CC3)=O)C1 N1(C(C2CN(C)C(=O)C2)=O)CC(C)(C)OC2(C1)CN(Cc1ccccc1)C2 c1(C(N(C(CNC(c2ncoc2-c2ccon2)=O)C2CC2)C)=O)ccccc1 N1(C(C2C(C)CCS2)=O)CCC(N(C(=O)CC(F)F)Cc2ccccc2)CC1 C1(C(N2CCC(CC(=O)OCC)C2)=O)CCC(NCc2cccc(F)n2)CC1 c1(C(=O)NCC2(C)OCCN(C(CC(=C)C)=O)C2)ccn2ncc(Br)c2c1 N1(C(C2CN(C)C(=O)N2)=O)CC(N(C)C(c2ccc(=O)oc2)=O)C2(CC2)C1 C1(CCCNC(=O)CCc2ncc[nH]2)CN(C(=O)CCC2CC2(Cl)Cl)CCO1 Nc1ccc(-c2cc(C(=O)NCCCOCCNC(=O)C3=CCCS3)n[nH]2)cc1 S(=O)(=O)(c1ccc2c(c1)CCCC2)NC(C1CCC(CNC2(C#N)CC2)C1)=O N1(C(c2cc(OC)n[nH]2)=O)CCN(C(c2ccsn2)=O)C(c2ccccn2)C1 C(=O)(CCCCC(C)CC)NCC(CC)(CC)NCc1cc(O)nc(C2CC2)n1 C1(C(N(CCCn2cnnc2)C)=O)CCC2CCC1N2C(=O)OC(C)(C)C C1(NC(c2cc[nH]c2)=O)CC(O)CN(C(c2cnc(Cl)c(C3CC3)c2)=O)C1 Cc1c(Cl)cnn1CC(=O)NC1CCOCC1NC(=O)CC1CC2CC2C1 Cc1ncsc1CC(=O)NCC(C(=O)NCCSC(F)F)N(C)C C1(OCC#C)CN(C(=NCC(C)(C)c2ncc(C)cc2Cl)NC(C)CC)C1 N1(C(c2c(OCC)nccc2)=O)CC2CC(C)N(C(=O)CCOC3CC3)C2C1 C1(C2CC2)(CNC(c2cc(C)oc2C)=O)CCN(C(=O)C=Cc2ccncn2)C1 N1(C(C(C)C)=O)CCCCC2(CCN(C(c3cccc(C4CC4)n3)=O)C2)C1 CC1(C)CCc2cc(C#N)c(N3CCSCC3C3CC3)nc21.C12(CC1)C(=O)NC2 C1(NC(c2ccccc2F)=O)CN(C(=O)NC2CCC2)CC1c1ccccc1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(C2N(C)C(=O)CC2)=O)C(F)C1 C(=O)(C1CCCc2ncnn21)NC1C(NC(C2CCN(CCC)CC2)=O)CCC1 N1(C(c2c(C)nc(CNC(CC(CC)C(C)C)=O)o2)=O)CCC2(CNC(=O)O2)C1 C(=O)(CN=c1cc[nH]cc1)NCC1(CNC(Cc2c(C)noc2C)=O)CC1(F)F c1(C(N2CC(NC(CCSCCCC)=O)C3C2C3)=O)cc([N+](=O)[O-])ccc1SC C1(NC(c2c(C)nc(C)o2)=O)CCN(C(=O)CCOC2CC2)CC1C n1(CCNC(CC=CC=C)=O)cc(C(=O)N(C)CC2(O)CN(C)C2)nn1 C1(CNC(C2CCCC(CC)C2)=O)CC2(C1)CN(C(=O)CCc1nncn1C)C2 C1(C)(C(=O)NC(CNC(c2c(C)nn(C)n2)=O)C2CCC2)CCCCCC1 C1(CNC(c2cc(C)on2)=O)(NC(c2cncc(Cl)n2)=O)CCCCC1C C(CCCCCNC(C1CC1(F)Cl)=O)NC(C1(CC=C)CC1)=O Cc1cc(-c2cn(C3CC4(C(=O)N(C)Cc5cocn5)CC34)nn2)cc(C)c1 N1(C(c2scc(C)n2)C(=O)Nc2ccccc2C)CCC(C2(C)CC2)CC1 CC(C(C)C(=O)NCCC1(C)CCOCC1)NC(c1ccn(C)c1)=O C1(NC(c2c(OC)ccnc2)=O)CCN(C(=O)CCCS(N)(=O)=O)CCC1CO c1(C(=O)NC(C)CNC(c2ccsn2)=O)c(Cl)cccc1[N+](=O)[O-] N1(C(c2cc(CC)c(C)s2)=O)CC(NC(=O)CN2CCNC(=O)C2)CCC1C C1(N(C(c2cc(C(C)C)no2)=O)C)CCCCN(C(=O)C(C)CF)C1 CS(=O)(=O)c1cc(Cn2nnnc2N2CCCCC23CCCC3)ccc1F N1(C(c2cn(CCN(C)C)nn2)=O)CC2CCN(C(=O)CCC(CF)CF)CC12 c1(C(=O)OCc2ccc(C(=O)OC)c(OC(F)F)c2)cccc(F)c1C#N CN1CCC(CC(=O)NC(C2CCOC2)CNC(=O)CCSC(N)=O)(C(F)F)C1 C1(=O)C2=C(CCCC2)NCNCC(=C)CCN1.C(=O)(C1=C(C)OCC1)NC(=O)OC N1(C(CC(C)F)=O)CCC(F)(CNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 CCCC(C(=O)NCCCC(C)NC(c1ccc(OC)o1)=O)OCC c1(C(N2CCC(OC)(CNC(=O)C(O)CCN(C)C)C2)=O)n[nH]c2c1CCOC2 c1(C(N2CC(OCC3CCCO3)C(O)C2)C(=O)NC2(C)CC2)ccc(O)cc1 C1(CNC(c2c(C)n(C(C)C)nn2)=O)CC2CCC1N2C(c1cncnc1)=O C1(NC(CCCOCCOC)=O)CCCN(C(=O)Cc2cc(C)sc2C)C1 N1(C(c2n(CC)cc(Cl)c2)=O)CCC(NC(c2ccsc2C#N)=O)CC1C N1(C(CCOCC#C)=O)CCCC(CNC(=O)C(C)NS(=O)(=O)CC)C1C N1(C(C2C(OC)C2)=O)CCCC2(CCN(C(C3CC4(CCOCC4)C3)=O)CC2)C1 C1(C(=O)NCC(CNC(c2c(C)ccc(OC)n2)=O)O)CCCC12OCCO2 C1(C(=O)NCC(C(CC)C)CO)CC(N=[N+]=[N-])CN1C(c1ccn(CC)c1C)=O c1(OC)cc(NC2CC3(C2)CC(NC(=O)CCCCCO)C3)nc(OC)n1 C1(C(=O)NCC2(N(C)C)CC2)CSCN1C(c1ccns1)=O Cc1cn2c(n1)CCC(C(=O)NC(C)CCNC(c1ccc3n[nH]cc3n1)=O)C2 c1(C(=O)N(c2ccnc(OC)n2)C2(C#N)CCNC2)ncnc2[nH]c(C)cc12 Cc1cnsc1C(N1CC(O)(CCNC(=O)Cc2ccccn2)C1)=O N1(C(C2C(CCC)C2)=O)CCC2(CC1)CC2NC(=O)CSc1ccccn1 c1(C(N(CCCNC(c2c(F)ccc(O)c2O)=O)C)=O)cc2c(nc1O)CCC2 CC(CC(=O)N1CC2(CC(NC(=O)CN3CCSCC3)CO2)C1)P(C)(C)=O N1(C(CCN(C)C)=O)CCN(C(=O)C(C)(C)CF)C2(CC2)C1 Cc1c(C(N2CC3C(CNC(=O)Cc4ccon4)C3C2)=O)[nH]c2cc(Cl)ccc12 c1(C(N2CCC(N(C(c3csnn3)=O)CC)C2)=O)nnn(C)c1C c1(CC(C)NC(=O)CC2CCN(C(c3ncoc3C3CC3)=O)C2)cnn(C)c1 N1(C(C=C(CC)C)=O)CC2COCCC2(NC(=O)CSc2cccc[n+]2[O-])C1 n1(CC(C(N2CCC(CN)CC2)=O)C)nnc2ccccc12.CCO C1(C(N(CCNC(=O)Cc2cc[nH]n2)C2CC2)=O)C2Cc3ccccc3C12 C1(C(N2CCC(CNC(CSC(C)C)=O)C2)=O)CC2CSCC(C1)C2(F)F CCC(CC)(C(=O)N1CCC(N2CCC(NC(C3CC3C#N)=O)C2)CC1)OC C1(C(=O)NCCCC(C)NC(=O)CC2COCCO2)(OCC)CCCCCC1 C1(C#N)(CC)CCCO1.c1(CN(CCC)CCOC)ccc(-n2cncn2)nc1 N1(C(CS(CC)=O)=O)CC2CC(O)C1C2NC(c1cc(C)c(Br)o1)=O c1(C(C)NC2N(Cc3cn(CC)nc3)CCC2)nnc2ccccn12 c1(C(=O)NC2C(NC(C(C(C)(C)O)F)=O)CC2)cc2c(cc1O)OCO2 N1(C(CC(C)(C)N(C(=O)CSCC(N)=O)C)=O)CCC(C2CC2)CC1 C1(C(N(C(CNC(C(Cn2ccc(C)n2)C)=O)C)C)=O)CCc2cnnn2C1 c1(C(N(CC(C)NC(c2cc(Cl)c(Cl)[nH]2)=O)C)=O)cnc2c(c1)CCCO2 N1(C(c2ccsc2)=O)CC2CCN(C(=O)CCc3ccccc3)C2C1 N1(C(c2cc(C)ns2)=O)CC2CCN(C(=O)CC(C)F)C2C1 CCCC(CC)CCC(=O)N1CC(NC(c2ccc(OC)c(Cl)c2)=O)C(SC)C1 C1(C)(C(=O)NC(C(N2CC(O)(C(=O)OC)C2)=O)C)CCC(C)C1 N1(C(C2CCN(C(c3cc(COC)sc3)=O)CC2)=O)CC(F)(F)CC1CO CN=c1nc(C(=O)NC2CC(Nc3ncc(C4CC4)cn3)C2)cc(C)[nH]1 Cc1ccc(C(N2CCCC2C(N2CCC(C)CC2)=O)=O)c([N+](=O)[O-])c1 c1(CNC2CC3(CC(NC(Cc4cccc(C)c4)=O)C3)C2)c(Cl)cc(F)cc1Cl c1(CNC(C(=O)NCC2C(C(=O)OC)CCCC2)=O)nc(Cl)ccc1Br C(=O)(C#CC1CCCCO1)N1C(COC)CN(C(=O)Cn2ccnn2)CC1 c1(C(N(CC(C)NC(C(CSC)C)=O)C)=O)cc(O)ccc1F C1(NC(CC2C(NC(CCCOCCC)=O)CCC2)=O)CCC2CC2CC1 Cc1ccc(C(N2CCC(=CCNC(c3c(C)nn(C)c3F)=O)CC2)=O)nc1C N1(C(=O)OC2C(N(C)C)CCC2)CCS(=O)(=O)C(C)(C)C1 c1(C(=O)NC2C(n3cc(C(CC)CC)nn3)CCCC2)ccc(Br)cc1C C(=O)(CC(C)C(F)(F)F)NCCC1(NC(C2N(CC)CCCC2)=O)CCC1 C=CCN=C(NCCSC)N1CCN(Cc2ccc(-c3ccccc3)cc2)CC1 N1(C(C2C(C)(C)OCC2)=O)CC2OCCN(C(=O)Cc3cnns3)C2C1 C=CCCCC(C(=O)NCc1[nH]nnc1C)NC(C1=NNC(=O)C1)=O C1(N(C(c2ncn(C(C)C)n2)=O)C)CCCCN(C(C2(CC#N)COC2)=O)C1 c1(C(=O)NCCCN(C)C(C23CCC2C3)=O)cc2c(Br)cccc2s1 C(CCS(=O)(=O)c1ccc(Cl)cc1)C(=O)NCc1cnc(C(C)C)[nH]1 c1(OC)cc(N)c(F)cc1C(N1CC(CNC(c2ccc(S(C)(=O)=O)o2)=O)C1)=O C1(C(N(CC(C)N(C)C)C(c2c(SCC)cccc2)=O)=O)CCc2n[nH]cc2C1 CC(N=c1[nH]c(=N)[nH]c(=NCCCn2cncn2)[nH]1)c1cccc(F)c1F N1(C(CC)=O)CC(CNC(C2C=CCC2)=O)C(F)(F)C1 Cn1c(C(N2CCC(O)(Cn3cc(C4CCCO4)nn3)C2)=O)cnc1S c1(C(N2C(C)C(NC(c3ccnn3CC(F)F)=O)CC2)=O)ccc(O)c(O)c1 CC1CCCC1(C)NC(c1conc1CNC(C1CCCN1C1CC1)=O)=O c1(OC)c(C(=O)NC2CCN(C(C3CC4COCC4C3)=O)C2C)cccc1C N1(C(c2c(C)cnnc2)=O)CCC(O)(CCNC(C2(C#N)CC(C)C2)=O)CC1 c1(C(=O)NCC(C)NC(C2CCN2C(C)(C)C)=O)csc(CO)n1.C(=O)(C(C)(C)C)N N1(C(CCC(CC)C)=O)CC2(NC(C3CCS(=O)(=O)C(C)C3)=O)CCC1CC2 c1(C(=O)NCC2N(C(C(C)(C)CF)=O)CCC2)cc(S(N)(=O)=O)c(Cl)o1 c1(C(N2CCC(NC(C(CC(C)C)NC(C)=O)=O)C2)=O)csc2cc(C)ccc12 CC1CC(C(=O)N(C2CN(C(=O)CN3CCCCC3=O)C2)C)c2ccccc2N1 C1(C(N2CCCC(C(C)C(=O)NCC3(C4CC4)CCC3)C2)=O)CCOC(=O)CC1 N1(CC(=O)N(C2CCN(C(c3cccc(F)c3)=O)CC2)CC)C(=O)CCCC1=O CC(C)C(CCN(C(=O)C(F)C(C)C)C)NC(c1csc(CO)n1)=O CS(=O)(=O)C1CCCCN(C(C2CC2c2cc(F)c(F)c(F)c2)=O)C1 N(C(=NCC1CCCS1(=O)=O)NCc1ccc(C(C)(C)O)cc1)C(C=C)C C1(C(N2C(C(CC)C)CC2)=O)CN(C(=O)CC2CC=CC2)CCN1C c1(NC(c2ccc(NC(c3nccs3)=O)nc2)=O)ccc(OCF)c([N+](=O)[O-])c1 c1(C(N2CCC(NC(C(CC)OC)=O)C(C)C2)=O)c(N)cc(Cl)cc1F c1(C(C)C)cc(=NCC2CC(C)N(C(c3ccn(C)n3)=O)C2)[nH]cn1 c1(C(=O)NCC2C(NC(C(C)c3ccsc3)=O)C2)cnc2sccc2c1 C(=O)(C(F)(F)C(O)C(C)C)N1CC(O)(CCNC(C(CC=C)CC)=O)C1 c1(CNC(CC(c2ccc(F)cc2)N)=O)cccc(Cl)n1 O=C(CCCc1ncco1)NC1CC(F)(CNC(C2(c3cc[nH]n3)CC2)=O)C1 C1(NC(CN(S(C)(=O)=O)C)=O)CN(C(c2cc(C3CC3)no2)=O)CC1S(C)(=O)=O CC(C)C(CO)C(=O)N1CCC(C(C)NC(=O)C(C)N(C)C)C1 N1(C(C(C)(C)C2CCC2)=O)CCOC2(C1)CN(C(C1CCC(C(=O)OC)C1)=O)C2 CC(CCc1cn[nH]c1)N=c1[nH]c(=NC2CCC2)[nH]c2c1CSC2 N1(C(C2CC(F)(CF)C2)=O)CC(O)CC1CNC(=O)C(F)=CC1CC1 c1(C(=O)NCC2CC3CN(C(C=C(C)C(C)C)=O)CC32)cc2ccsc2c(O)n1 c1(CC)c(C(=O)NC(C2CCCN(C(c3cn(C)[nH]c3=N)=O)C2)C)csc1C O=C(CC1CCOc2ccccc21)NC1COCCN(C(c2ccccc2)=O)C1 C(=O)(CCCCC(=O)N1CCC2CCCC12C(=O)NC(c1ccn(C)n1)C)OC C1(NC(C(C)(C)OCC)=O)CCC2(CC1)CN(C(c1cccnc1)=O)C2 c1(NC2C(F)COC2)nccc(=NCc2cncn2Cc2ccccc2)[nH]1 N1(C(C2(C)CC(C)C2)=O)CC2CC1C2CNC(c1cnc(C(C)(C)C)s1)=O Cc1[nH]c2ccc(Cl)cc2c1C(=O)NCC1COCC1NC(c1cnccn1)=O CCC(COC)C(=O)NCC(C)CC(=O)N1CCCC1C(=O)N(C)C c1(C(=O)NC2CC(OCC(=O)NC3(C(N)=O)CCCC3)C2)nnc(O)nc1O C(=O)(C#CC12CC3CC(CC(C3)C1)C2)NC1C(NC(C2N(C)CC(O)C2)=O)CC1 C1(CNC(c2n(CC)ncn2)=O)CC12CCN(C(=O)CC1CCCOCC1)CC2 CC#CCCCCNC(=O)CCC(C)NC(c1cc(OC)nn1C)=O Cc1cccc2c1CC(C(=O)NC1CC1NC(=O)Cc1ccc(F)cc1F)O2 C1(C(N(C)CC2CCN(C(C(CSC)OC)=O)C2)=O)CCC(N(C)C)CC1 c1(OC)cc(C)ccc1C(N1CCN(C(c2nccnc2Br)=O)CC1)=O C1(CN(C(CCc2onc(CC)n2)=O)C)CCN(C(C2CC(C)C2)=O)CC1 C(=O)(N1CCC(C(=O)NCCC2C=CCC2)O1)c1cn(CC=C)nc1 c1(C(C)NC(=O)NCCNC(=O)CN2CCNC2=N)ccc2nc(O)oc2c1 C1(CCC(=O)Nc2c(C)ncnc2)CCCCN(C(=O)CCCC2CC2)C1 C1(CNC(C(C=CCCC)O)=O)C2CCC(C2)N1C(C1(N(C)C)CCCCC1)=O CC1(C)CC(=O)NCC1C(N1CCC(NC(=O)Cc2cccc(C(F)(F)F)n2)C1)=O c1(C(N(C2C(C)CCN(C(CCCOC(C)C)=O)C2)C)=O)cnn2ccccc12 C1(C(N(C(CNC(CNC(C)=O)=O)C2CC2)C)=O)C=C(C)CS1 c1(C(=O)NC(C)CC2CN(C(=O)CC#N)C2)nccc2ncccc12 c1(CC)cc(C)nc(N(CCCNC(C2CCC(C)C(C)C2)=O)C(C)C)n1 N1(Cc2n(CCC)ncn2)CCCC(NC(c2cscc2C(=O)OC)=O)C1 N1(C(C(C)(C)CCl)=O)CCOC2(COCCN(C(=O)Cc3ccc(O)cn3)C2)C1 c1(SC)cc(C(N2CCC(NC(c3cc(=O)n(C)cn3)=O)C(F)C2)=O)ccc1F c1(OC)cc(C)c(CN2CCC(c3nc[nH]n3)(OC(C)C)CC2)cc1S(C)(=O)=O Cc1nc(CC(=O)NCC(C)(C2CC2)NC(c2n[nH]cc2Cl)=O)n[nH]1 C1(C(=O)NCC2CCN2C(=O)CC=C(C)C)(COC)CCCCO1 Cc1n[nH]c2cc(C(=O)NCC3CCC3NC(C3COCCN3C)=O)ncc12 c1(NC(C2CCN(Cc3ncc[nH]3)CC2O)=O)cccc(Cl)c1[N+](=O)[O-] N1(CC(C)CC2CCC2)CCC(O)C2(CCOCC2)C1 C1(OC)(OC)CCC1CC(=O)N(CCCCNC(=O)C(n1nccc1C)C)C C1(F)(CNC(c2c(CC=C)cccc2)=O)CCCN(C(=O)C(C)(O)CC)C1 C(=O)(C1CCCn2cc(C)nc21)NC(CC)CN(C(=O)C(=O)Nc1ncc[nH]1)C N1(C(CCNC(C)=O)=O)CCC2CCN(C(=O)CCc3nncn3C)CC12 C1(C(N2CC3(C2)SCCC3NC(C2(F)CCCC2)=O)=O)Cc2ccccc2N1 Cc1nn(CC(=O)NC(C)(CNC(C2(CCF)CCC2)=O)CO)cc1Br C1(C(C(=O)NCCOCCNC(C2(c3ccno3)CCC2)=O)O)CCCCC1 Cc1nc(C)n(C(=O)OC2CSCN2C(=O)C(C)(C)C)n1 c1(CC(=O)NC2(CO)CN(C(C(CC(C)C)O)=O)C2)ccccc1S(C)(=O)=O C(c1cccnc1C)=CC(=O)NCCCN(C(=O)CCC1CCCN(C)C1)CC N1(C(C2CCC(N(C(CC(=C=C)C)=O)C)CC2)=O)CC2CCC(OC)C2C1 N1(C(COCCOCCOC)=O)CC(NC(c2snc(Cl)c2Cl)=O)C(O)C1 C1(NC(C2N(CC)CCC2)=O)CN(C(=O)CC(=O)Nc2nccs2)CC2(CC2)C1 c1(CC(=O)NC(C(C)NC(CCC#C)=O)C)ccc(Br)cc1C#N C1(C(N(C(C)CN(C)C(c2ccnc(N(C)C)c2)=O)C)=O)CCc2cncn2C1 Cc1ccc(NC(=O)NC2CC2Cl)cc1OCC(C)(C)C(C)C N1(C(CC=CCC)=O)CCC(F)(F)C(CNC(C2Cc3nnc(C)n3C2)=O)C1 c1(C(N(C(C)(C)C)C(C2CC2Nc2ccno2)=O)=O)nc(Cl)cs1 CC1CN(C(C2CCCCC2C)=O)CCC1NC(C1CCN(C2CC2)CC1)=O c1(OCC)c(C(=O)NCC(C)CNC(c2cnc(OC)c(C)c2)=O)cccc1F C1(C(=O)NC2(COC)CN(C(c3ccc(CC)cn3)=O)C2)CCCCC1C1CC1 CN1CCN(C(C2C(O)CCN2C(=O)CC2CCCSC2)=O)CC1 c1(C(C)OC(C2(C(F)F)CCOC2)=O)cccc(S(=O)(=O)CC(F)(F)F)c1 CCCC(CNC(=O)C(O)CC(C)(C)C)C(=O)NOCC1CCC1 N1(C(c2cnc3[nH]ccc3n2)=O)CCC2CCC(C1)N2C(C1CC12CCC2)=O CN1CCCC(C)(C(=O)N(C)CCOCCC(=O)NCc2cncc(Cl)c2)C1 C(=O)(CCC(C)(C)C(=O)OC)N1CC2(CN(C(C(C=C)O)=O)C2)C1 C1(C(C)C)N(C(c2ccc(CNC(C3COC(=O)N3C)=O)nc2)=O)CC1(C)C CCCCC(C)CCC(=O)N1CC(NC(c2nc(C3CC3)cs2)=O)CC(F)C1 N1(C(c2cc(C#C)c(Cl)cc2)=O)CCCC2(C1)CN(C(=O)C1=CCSC1)C2 N1(C(CCCC)=O)C(C)C2CC1C2NC(=O)CCc1ccc(F)cc1Cl N1(C(C2N(C)C(=O)OC2)=O)CC2=C(C1)CN(C(=O)Cc1cccc(Br)c1)C2 C12(NC(C3C(=C)CC3)=O)CCCC1N(C(c1cnc3ccnn3c1N)=O)CCC2 c1(C(=O)NCC=CCNC(C2C(C(=O)OCC)CC2)=O)cccc2nccn12 Cc1cc(Cl)cc(C)c1C(=O)NCCCCC(C)NC(c1cccc(F)c1O)=O c1(OC)ccc2cc1OC(=O)CC2.C1(NCC)C(C(=O)O)C1(C)C.C(C)(C)(C)O C1(C(=O)NCCCN(C(=O)C=CS(C)=O)CC)CCCOCC1 CC1CN(C(C2CCCN(C)C2)=O)CC(C(=O)NC2(c3cc[nH]n3)CC2)O1 CCN=c1ccc(C(N2CCCC(CN3CCN(C(=O)CC4CC4)CC3)C2)=O)c[nH]1 Cc1cc(F)ccc1CC(N1CCN(C(=O)C(C)N(C)C)CC1C1CCCC1)=O C(CC(=O)NC1CCC(NC(=O)C(C)N2CCC2)CC1)(C1=CCCC1)OCC c1(NC(c2ccnc3c2OCO3)=O)sc2c(c1C(=O)NCCN1CCOCC1)CCC2 N1(C(c2ccc(N(C)C)nc2)=O)CCC(C)(C(=O)Nc2ccc(CO)cc2)CC1 C(=O)(C=C1SCC(=O)N1C)N1C2CC(NC(COC)=O)C1CC2 CC(C(C)C(=O)Nc1cn(C)nc1Cl)NC(c1ccncc1N)=O CC1C(C(=O)NCCC2CCOC2(C)C)CCN1C(C1SCCS1)=O c1(C(=O)NCC2(F)CCC(NC(c3cc(C)sc3)=O)C2)ccc(Cl)nc1O c1(C(=O)NC(CC2CN(C(C(CC=CCC)C)=O)C2)C)cc(=O)c(OC)cn1C c1(CCC(=O)N(C(CCOC(C2(C(=O)NCC)CC2)=O)C)C)cccc(F)c1 C1(NC(c2cnc(C)nc2C2CC2)=O)CC2CCC(C1)N2C(c1cnnc(Cl)c1)=O C(=O)(C(O)C1=CCCCC1)N1CC(NC(c2ccc(C#C)cn2)=O)C(O)C1 CC1(C)CC(C(=O)NCCc2cccnc2)CN1C(=O)Cc1cn[nH]c1 c1(C(=O)NC2(C)CC(NC(CCC(C)N(C)C)=O)C2)[nH]nc([N+](=O)[O-])c1Cl C1(C=O)CC12C1CC3CC(C1)CC2C3.C(=O)(CCOCC)NCCC(CC)C CCCCC(O)C(C)C(=O)N1C2CCCC1CN(C(c1nn(C)cc1C)=O)C2 c1(NCCNC(C)=O)nccc2cc(C)ccc12 c1(CC)ccc(N)c(C(=O)N(C(C)CNC(c2ccc(OC)nc2)=O)C(C)C)c1 C(=O)(C1=CCCOCC1)N1CCC(CCC(=O)NCc2cc(C)sc2)CC1 C1(C)(CC)CCN(c2ccnc(N3CCCC(CN(C)CC)C3)n2)C1 C(CCN=C(NCC(c1ccc(OC(F)F)cc1)C)N1CCSC(C)(C)C1)OCC C1(CC)C(C(=O)NCC2CC[Si](C)(C)C2)CCN1C(C1SCC=C1C)=O C1(CC#N)CCN(N2CCN(c3cc(Cl)cc(Cl)n3)CC2)CC1(F)F N1(Cc2c(C(=O)OC(C)(C)C)cco2)CCOC(CC(N)=O)C1 C1(C(N(CCN(C)C(c2oc(C3CC3)nc2C(F)F)=O)C)=O)CC(=O)NC1(C)C CC1CCCCC1CC(=O)NC1CC(CNC(c2c[nH]nc2C(F)F)=O)C1 c1(C(=O)NCCCN(C(C(COC)OC)=O)CC)cc(-c2nn[nH]n2)ncc1Cl C1(C(=O)NC2(CNC(=O)CC3CC3C(F)(F)F)CC2)CCCC1F c1(C(C=C)(C)O)cn(CC(CNC(=O)CCc2scnc2C)OC)nn1 Cc1cnc(F)c(C(N2CCCC(CO)(NC(C3CCC(C)(O)CC3)=O)C2)=O)c1 Cc1cc(C(C)C)ccc1C(=O)NC1CCN(C(=O)CCn2cccn2)C1 CCCCCCCCOC(C1CN(C(=O)NC2(O)CCCCC2)C1)C C1(C(N(c2cc(O)ncn2)C)=O)CN(C(C2CCC3(CC2)CC3)=O)CC12CC2 C1(C(=O)NCC2C(CC)CCC2)CNC(=O)CN1C(c1cc(C)oc1C)=O C#CCC(CC(=O)NCCS(N)(=O)=O)NC(c1cncc(Cl)c1)=O c12cc(ccc1F)C(=O)N(Cc1ccccc1)c1ccc-2cn1.CC(C)OCC c1(C(n2cc(CNc3ccc(Br)c(O)c3)nn2)C)cc2c(cnn2C)nc1O N1(C(C(=O)NC(C)C)=O)CCC(C(C)C(N2CCC(C(C)(C)C)C2)=O)C1 c1(C(N2C(C(C)(C)C)C(NC(=O)CS(C)(=O)=O)CC2)=O)cnc(O)c(F)c1 n1(CC)ncc2c(C(=O)N(C)C3CC3)cc(C3C(CO)(CO)C3)nc12 C(CCC(N)C(=O)O)NC(C(c1ccc(Cl)cc1)OC)=O N1(Cc2cc(OC)nc(OC)c2)CC(C2CCN(C(=O)CSC3CC3)CC2)CC1 C1(C(=O)NCC(CCNC(c2cnc(CC(C)C)s2)=O)O)OCC2CCCC12 N(C1CCCn2ccnc21)C(=O)C(=CC1CCCC1)C.C(C=O)NCCC C1(CCN(C(=O)CC2CC3(CCC3)C2)C)CCN(C(c2cscn2)=O)CC1 C12(NC(c3c(C)snc3)=O)CC1CN(C(c1noc(-c3cccc(F)c3)n1)=O)C2 c1(C(=O)OC)nc[nH]c(=NCC2(O)CCCN(C(=O)CSC(F)(F)F)C2)c1OC Cc1ccccc1C(=O)NCC1(NC(C2(C(=O)N(C)C(C)C)CC2)=O)CCCC1 CC1CC(CO)CN1C(=O)CCNC(=O)CCc1ccsc1 Cc1nc(C(=O)NCc2csc(C(=O)N(C)CCOCCO)c2)n[nH]1 c1(C(N2CC3C(NC(c4ncc(C)cc4C)=O)(C3)C2)=O)coc2c1CCCC2 N1(C(C(=O)NCc2ccc(SC)o2)=O)CC2(CC(NC(=O)C(C)(C)C)C2)C1 c1(SC)cncc(C(=O)NCCCNC(C2C=CC=CC=C2)=O)c1.C1(S)CCOC1=O C(C1CN(C(=O)CC2CCCC(C)(C)C2)CC1C(=O)NCC(C1CC1)OC)=CC C(C(CNC(c1cnncc1OC)=O)C(F)(F)F)NC(C=CC=CC)=O C#CCC(CC(=O)NC1CN(C(C2CCCC2F)=O)CC1C)c1ccccc1 N1(C(Cc2nc(COC)sc2)=O)CCC(NC(C2CC(=O)NC2(C)C)=O)C(C)C1 C(=O)(CCCCCN(C)C)NCC(CNC(c1cncc(OC)n1)=O)F c1(C(=O)NCCCCCN(C(COCC(=C)C)=O)C2CC2)cncc(C2CC2)c1 c1(C(C)NC(N2CCC2C2CC2)=O)nnnn1CCC(=O)OC(C)(C)C CC(C)CC(C(=O)N(C1(C(=O)NCCCC2CCCCO2)CC1)C)C1CCC1 N1(C(C2N(CC)CCOC2)=O)CCN(C(c2cc(C)c(O)nn2)=O)C2CCC12 c1(OC2CCC(N(CC=C)C(=O)OCC)CC2)ccc2c(c1)OCO2 c1(OC)nccnc1C(=O)NCC1(F)CCC(NC(=O)CC2CCC(C)(C)C2)C1 C1(C(c2nncn2C2CC2)C)CCCCN1C(=O)CCC(N)=O.C(=O)N C1(CNC(=O)C2=C(Cl)CC2)CCCC2(CN(C(c3c[nH]c4ncccc34)=O)C2)O1 C1(C(=O)NCC(CN(C(C2(CC)COC2)=O)C)C)CC(c2ccccc2C)=NO1 C1(NC(Cc2c(C)noc2Cl)=O)CN(C(=O)CC2NC(=O)CNC2=O)C(C)(C)C1 N1(CC(=O)N(C2CCCN(C(c3cc(C)ncn3)=O)C2)C)CCCNS1(=O)=O c1(C(=O)NC2CC(CNC(c3nn(C)c(OC(F)F)c3)=O)C2)ccc(N)c(N)n1 C1(CNC(C2(OC)CCSC2)=O)(NC(=O)C(C)c2ccsc2)CC2CCC1CC2 C1(C)(C(=O)NCC2CC(C)N(C(=O)Cc3ccccn3)C2)COC(=O)OC1 c1(NC(C2CC(C)CN2Cc2cncnc2)=O)ccc(Br)c(Cl)c1 C(=O)(CCCCC(=O)N(CC(O)CNC(=O)Cc1cccc(OC)c1Cl)C)OC C1(C(N(CCC(C)NC(c2c(F)ccc(C)c2)=O)C)=O)CC2(CCOCC2)CO1 Cc1sc(Br)nc1C(N1CC(F)C(F)C1)C(=O)NC1CCCC1 C1(C)(CC)CC(NC(=O)COCC(F)(F)F)CN1C(c1cccc(F)c1OC)=O CCC(C)C(=O)C(=O)N1CCC(C(N2CCC2(C)C(=O)OCC)=O)C1 N1(C(CCC(CC)OC)=O)CCCN(C(c2ccnc(OC)c2Br)=O)C(C)C1 C#Cc1ccc(C(=O)NCc2cc(C)c(C(=O)NC(C3CCCCC3)C)o2)nc1 N1(C(c2c(C)noc2)=O)CCCC(NC(=O)CNC(N2CCCC2)=O)C(F)C1 c1(OC)cncc(-c2ccc(NC(=O)C(N3CCC(N(C)C)CC3)C)cn2)c1 Cc1nc(Cl)nc(N2CCCC2CN(C(=O)C(c2ncccc2F)(F)F)C)c1Cl C1(CCC(=O)N(CCOC)CCNC(C2CC(C)(C)C2)=O)CCCN(C)C1 c1(C(N2C(CCNC(c3nc(C)oc3)=O)COCC2)=O)cc2ccnc(Cl)c2[nH]1 Cc1ccc(C(=O)NCCC2CCCCN2C(C2CCCOCC2)=O)c(O)c1 c1(C(=O)NC2C3CN(C(=O)CCn4ccccc4=O)CC23)ccc2cncn2c1 c1(CCC(=O)C(=O)NCCC(=O)OC(C)C)ccc(Br)cc1.N c1(C(=O)NC(CC(C)NC(C(CC)CO)=O)C)cc([N+](=O)[O-])ccc1SCCO C(=O)(CCCCCCN=[N+]=[N-])NC1C(OC)CN(C(c2cc(C)[nH]n2)=O)C1 Cc1cc(C(N2CC(NC(=O)Cn3cc(C4CC4)cn3)CC2(C)C)=O)c(C)n1C C1(NC(C=C2CCC(C)C2)=O)CN(C(=O)C(c2ccccc2)=O)CC1(C)C c1(OC)c(Cl)cc(C(N2CC(NC(C3(OC(C)C)CCC3)=O)CC(C)C2)=O)nc1Cl CN1CCN(C(=O)C(CCF)NC(=O)C=C2CCCCC2)CC1=O C(=O)(CCCC(F)(F)F)N(CC(C)Oc1ccccn1)C.C1(=O)CO1 C(=O)(CC1=CCCC1)NC1CN(C(CCN(CCC(C)(C)C)C)=O)C1 CC(CC1CCCO1)N=c1cccc(S(=O)(=O)NCCC(F)F)[nH]1 C1(CNC(c2c(C)noc2C)=O)CN(C(C2CNC(=O)O2)=O)CC1(C)C c1(CC)ccc(F)c(C(=O)NCC(CC(C)C)NC(C2(Cl)CC2(C)C)=O)c1F Cc1ccnc(CNC(C23CC2CN(C(c2scnc2C)=O)C3)=O)c1F N1(C(c2ccc(Cl)cc2)=O)CCCC2(C1)CN(C(=O)C(F)(F)C1(O)CCCC1)C2 C1(CC(=O)NC(CNC(C2=CC(C)(C)C2)=O)CO)CC2(C1)CC1(CCC1)C2 c1(NC(C2N(C(C(CC)CN(C)C)=O)C(C)C2)=O)ccc(O)cc1C(=O)OC c1(C(N2CCC(CNC(C(C)CC3CCCC3)=O)C2)=O)cnccc1Br C#Cc1ccc(C2(C(=O)NC3CCC(NC(C4C5CC6C(C5)C46)=O)C3)CC2)cc1 N1(C(c2n(C)cc(Br)c2)=O)CCC(NC(c2ccnn2C(F)F)=O)C(F)C1 C#CCC(CC(F)F)C(=O)N1CCC(C(=O)NCCCC(=O)NC)CC1 C1(CC(=O)NCC2C(CCC)CCC2)CCCN1C(=O)C=CC1(C)COC1 c1(-c2ncn(C)c2)cnccc1C(=O)NCCCNC(=O)Cc1ncc(F)cn1 C1(NC(C(C2CN(C(CCOCCC)=O)C2)O)=O)COCC1C1CC1 C1(C(=O)NCC(F)F)CCC(O)CN1 c1(CC)onc(C)c1C(=O)NCC(C1CCCCC1)NC(C1(C)CC(C)=NO1)=O c1(CCC(N2CC(N(C(=O)CCCF)C)C(C)(C)C2)=O)nc2cccnc2[nH]1 CC1CN(C(c2csc(-c3nc[nH]n3)n2)=O)CC(C)N(C(=O)C2=NNC(=O)C2)C1 c1(C(N(CCNC(Cn2ncc(CC)c2)=O)CC)=O)cc(F)ccc1F c1(C(C(=O)NC(CCCC)CNC(=O)COCC)(C)C)ccc(OC)c(F)c1 C1(CC(C)NC(C(F)=C(C)C)=O)CCN(C(C2(CO)CC2(F)F)=O)CC1 c1(NC(CCCOC)C)ccc(NC(=O)C(O)Cc2ccccc2)cc1F C(=O)(C(C)Cn1cccn1)NCCCN(C(=O)C(C)(C)c1ccccc1)CC N1(C(c2oc(CC)c(C)c2)=O)CC2(CCN2C(C2CC=CCC2C)=O)C1 N1(C(=O)NCc2nnn(C)n2)CCN2CC3(CC3)CC2C1 c1(C(=O)NC(C(C)(C)NC(CCCCOCCC=C)=O)C)cc2c(s1)CCC2 c1(NCC2COCC2c2cn(C)nn2)cc(CC)ccc1C.C12(CC1)CO2.CO C#Cc1cccc(C(c2nnnn2C)NCCn2cc(CC)cn2)c1F [N-]=[N+]=Nc1ccccc1NC(C1COC2(C1)CN(C(c1ccsc1)=O)C2)=O C1(COC)CNC(C(=O)NC2CCOC2c2ccccc2)C1 Cc1scc(C(N2CC(CNC(C3CC3c3cnn(C(C)C)c3)=O)C2)=O)c1C Cc1c(NC2(CO)CCN(C(=O)CCOC3CC3)CC2)ncnc1Cl CCC(C)CCCCC(=O)N(CC(O)CN(C)C(c1ccc(O)c(CO)c1)=O)C c1(CNC(C2CNCCN2c2ncncc2Br)=O)cccc(Cl)c1Cl c1(C2(C(N3CC(NC)(CF)C3)=O)CCC2)c(F)cccc1F Cn1cnn(CCC(=O)NC2COCC2n2cc(CC(O)C3CC3)nn2)c1=O c1(C(=O)OC)sc(C)cc1NC(C1(Sc2ccccc2)CC(C(=O)O)C1)=O N1(C(CN(N(C)CC)C)=O)CCC1(C)CC(=O)NCCCCSC N1(C(C2C(=C)CC2)=O)CCC2(CCCC2NC(=O)C(F)(F)COC)CC1 N1(C(C(c2ccccc2)SCC)=O)CCCC(N(C(=O)CCSCC)CCF)C1 N1(C(CN(CC)CC)=O)CCCC(CC)(NC(c2ccc(-c3cc[nH]n3)s2)=O)C1 C1(CCOC)(NC(C2CC23CC(O)C3)=O)CCN(C(=O)Cn2cccn2)C1 c1(C(=O)NC(CN(C(CN(C(C)C)C)=O)C)C)cc(Br)c2[nH]cnc2c1 C1(NC(c2cc(C)cc(F)c2)=O)CCN(C(=O)CC2CC2)C12CCCC2 c1(CCC(N2CC3C(CNC(CCCC#C)=O)C3C2)=O)cc(C)cc(C)c1 N1(C(CC2CCC(=O)CC2)=O)CCC(C(N2CCCCC2CF)=O)C12CC2 C(c1ccc(Cl)cc1Cl)=CC(N1CC(OC)CC(NC(C=CSC)=O)C1)=O N1(C(c2cc(CCC)n(C)n2)=O)CC(CCNC(=O)C(CC)CC)OC(C)C1 S(=O)(=O)(c1c[nH]ccc1=NCc1cc(Cl)on1)NCCC(C)n1ccnc1 C1(NC(c2ccc(CO)s2)=O)CC(CNC(C2(O)CCCC2)=O)C(O)C1 c1(CCC(=O)NC(CNC(C(C)SCCCC)=O)(C)CO)csc2ccccc12 CC1CN(C(=O)CCC2CCC2)CCCN1C(=O)CCC1CCC(=O)C1 CC1CCC(NC(=O)C(O)CCc2ccccc2)CN1C(=O)C1=CCCOC1 Cc1cc(CNC(C2CN(Cc3ccc(Cl)cc3F)CCO2)=O)cc(C)c1F c1(N2CCC(NC(CC3CCCC(OC)C3)=O)C(F)C2)ncnc(Cl)c1[N+](=O)[O-] c1(-c2ccc(C)o2)nc(C)c(C(=O)NCC2CCC(NC(=O)CNC=O)C2)s1 c1(C(N(CCNC(CN(S(CC)(=O)=O)C)=O)C(C)C)=O)csc(S)n1 C12(C(=O)NCC34CN(C(CSC)=O)C(CC3)CC4)CCOC1CS(=O)(=O)C2 c1(-c2nc(C3(NC(=O)C4CC4)C(C)CN(C)CC3)on2)nnc2c(=O)[nH]ccn12 N(C1c2ccccc2CC1NC(=O)CC(=O)NCC(F)(F)F)C(C(C)SC)=O c1(N(C)Cc2c(C)nco2)nc2cc[nH]c2c(=NCC2CC(=O)NC(C)C2)[nH]1 CCC(C)CCC(=O)NCC1(NC(C2COCC2(C)C)=O)CCC1 C(CCCC(=O)N1CC2CC2(CNC(c2cnn(CC(F)(F)F)n2)=O)C1)OCC C1(CC)CCCC(N=c2[nH]c(=NCC(C)(C)c3cccnc3)c3[nH]ccc3[nH]2)C1 N1(C(CCC=CC)=O)CCN(C(=O)C(C)C2CCCO2)CC1CCO c1(C(=O)NCCC2OCCN(C(C(CC)(F)F)=O)C2)ccnc2c1CCC2 c1(C(=O)NCCN(c2ccccc2Cl)C)ccc(=O)n(CCOCC(F)(F)F)c1 CC1=C(C(=O)NCC(CO)NC(c2cc(C)cnc2C)=O)CCC(C)(C)C1 N1(C(CC2CCC(C)CC2)=O)CCC2(C1)CN(C(=O)CNc1nccs1)CCO2 Cc1conc1C(=O)N(CC(C)O)CCNC(c1snnc1C(C)C)=O c1(C(=O)OCC)cc(=NC2CCCN(C(=O)Oc3ccc(OC)cc3)C2)cc[nH]1 CC1CN(C(c2c(F)cncc2Br)=O)CCCN1C(=O)Cc1cnsc1 C#CC1(C(=O)N(CCCNC(c2cccn2C)=O)CC)CCCC1 N12CCCCCCC1C2=O.CC(C)(O)CC(=O)NCc1nc(CO)n[nH]1 C1(C(=O)NC(CCCCNC(C(C)(C)C)=O)CO)Cc2ccccc2C1(C)C C12CC3(C1)CC1(CC(C1)CN2)C3.C1(C(=O)OC(C)(C)C)CC(CC(N)=O)C1 c1(C(N(CCCNC(C2OCC(C)C2)=O)CC2CC2)=O)ccnc(S)c1 c1(NC(=O)NCCN2CC(C)OCC2)nccc2c1NCCC2 C1(c2onc(-c3cc(OC)n(C)c3)n2)CC2CCC(C1)N2C(=O)C(C)(C)C N1(C(C(Cn2ccnn2)NC(C=Cc2cc(C)no2)=O)=O)CCC(F)C(F)C1 C1(NC(=O)CCCc2ccccc2)CC12CCC(NC(C1CCC1)=O)CC2 C1(C(N2CC(NC(C(C(=O)OC)C)=O)(CO)C2)=O)CCCN1S(=N)(=O)N(C)C C1(COC)CN(C(=O)CC2CC=CCC2)CCN1C(=O)C(C)=C1CCC1 CC(=O)CCCC(C)C(=O)N(C)CC1CCCCN1C(=O)CC1CCC(=O)N1 C=CCCCC(=O)N(C)CCOCCN(C(=O)C(F)(F)CN(C)C)C N1(C(c2ccc(CSC)o2)=O)CCC(C)C(CNC(c2c[nH]c(=N)nc2C(C)CC)=O)C1 N1(C(C(c2cccs2)NC(CCC2N(C)CCC2)=O)=O)CCC(N=[N+]=[N-])C1 C1(OCC(=O)NCCCOc2cocn2)CC(=O)C1 N1(C(C2C(C)C2)=O)CCC(CC(=O)Nc2cncc(-n3cccn3)n2)CC1 C1(NC(c2ccc(C)[nH]2)=O)CCN(CC(=O)NCCSc2ccc(Cl)cc2)CC1O C1(CN(C(=O)C=CCC(C)(C)NC(C2(C)CCC(=O)C2)=O)C)CCCC2CC12 C(N=c1[nH]c(=NC2CCCC2OC(F)(F)F)c2c(F)cccc2[nH]1)c1ccc(Cl)o1 C(=O)(C(N=[N+]=[N-])C(C)C)NC1CC2(C(C(N(CC(CC=C)(F)F)C)=O)C2)C1 Cc1cocc1C(=O)NC1CCC(N(C)C(C23CC(CO2)C3)=O)C1 CC(c1ccccc1)=CC(N1C(C(=O)NC(CO)C2CC2)CCC1C)=O C(=O)(C1=CCC(C)CC1)NC1C(C=C)CN(C(=O)Cc2sccc2Br)C1 c1(C(=O)NCCN(C(C(c2c(C)cccc2)C)=O)C)noc2c1CC(C)CC2 C(=O)(C1=CS(=O)CCC1)N1CC2C(NC(c3c(C)cns3)=O)C2C1 Cc1cc(C(=O)NC2CCCN(C(=O)Cc3cocn3)CC2)c2c(c1)CCC2 N1(C(CC(COCC)NC(CSCC#C)=O)=O)CCCC2(CC2)C1 N1(C(C2C(C)(C)CCN2C(=O)CC2=CCCC2)=O)CC2(CCOCC2)C1 CC=C=CCCN=c1[nH]c(=NCCCCN(C)C2CC2)[nH]c2c1CCC2 N1(C(C2OCCN(C(C(CC#C)O)=O)C2)=O)CCOC2(CC2)C1 N1(C(c2c(C)nc(C(C)OC)s2)=O)CCC2CCC12CNC(=O)CN(C)C(C)=O c1(C(C(=O)NCC(C)C)N(C)Cc2ccc(Cl)cn2)ccccc1CC(F)(F)F n1(C(N2CCC(CNC(=O)CSC3CC3)C2)=O)c(=O)oc2ccccc12 S(=O)(=O)(c1cccnc1N1CCC(n2cc(CO)nn2)CC1)N(CC(C)C)C Cc1cc(F)c(F)cc1NC(c1nnnn1C1CC1)C1CCOC1 CCCC(C)C(CC)(c1nnnn1-c1ccccc1)NCCN1CCCC1=O N1(C(CCC=CCC=C)=O)CCN(CSc2occc2Br)C(CO)C1 N1(C(C(F)OC)=O)CCc2ccccc2C1CNC(c1cncc(Cl)c1Cl)=O CC(O)CC(C)(C)CNC(=O)C(C1CC1)NC(c1cc(Cl)n[nH]1)=O C1(C(N(CC)CC)=O)CN(C(c2c(Cl)cnc(Cl)c2Cl)=O)CC(F)(F)C1 C1(C(=O)NCC(C(=O)NC(c2ccc(CO)o2)C)(C)C)OCC2CCCC12 Cc1cccc(CNC(c2ccc(-c3c(O)cccc3F)nc2)=O)c1Br C(=O)(CCCC(C)(C)NC(c1cn(C2CC2)nn1)=O)NC(C(C)C)CC(=O)O C(=O)(CCCCC(N)=O)NC(CC1(C)CC1)C(N1CCN(C2CCO2)CC1)=O CN1CCCN(C(=O)CCCNC(=O)C(c2ccnn2C)O)CC1=O Cn1nc(CO)cc1C(=O)NN1CC(C(=O)NC2CC(F)(C)C2)C1.[SH](C)(=O)=O C(CNC(=O)CC1CCOC1)(CC(=O)NCCSC(F)(F)F)OC N1(C(c2ncoc2C(F)(F)F)=O)CCC(Oc2ccccc2)C1 C1(CNC(c2c(OC)nsc2)=O)(NC(=O)Cc2cc(C)[nH]n2)CCC(C)(C)CC1 C(=O)(CC(C)(C)C(C)(F)F)N(CCCCCC)CCNC(=O)CC1OCCC1C CC(C(C)(O)C(=O)N1CCC(C)(NC(c2cnc[nH]2)=O)CC1)c1ccccc1 c1(COC)n[nH]c2ccc(C(=O)OC(c3ccc(OC)cc3N(C)C)=O)cc12 c1(C(N2CCC(NC(C3(C)CC=CCO3)=O)CC2)=O)cccc2ncnc(O)c12 C=CC(C)(C)CC(=O)NC1(C)CC(NC(C2CCN(C(C)C)CC2)=O)CS1 C1(NC(CCOC)=O)(CO)CCN(C(C2(c3cccc(C(C)C)c3)CCC2)=O)C1 C1(NC(c2c(C)coc2)=O)CC(C)CN(C(=O)CCc2cccc(Cl)c2)C1 C1(CC)CN(C(=O)CCN2CCCCC2=O)CCN1C(C1CC2COCC2C1)=O c1(NC(C2CCCN(CC(=C)C)C2)C)ccc2c(c1)CCCS2(=O)=O c1(C(=O)NC2C(NC(=O)CC3(O)CCC3)CCC2)cccc(N2CCOCC2)c1 C1(NC(C(C(C)C)c2ccccc2)=O)CCCCN(C(=O)C=Cc2ncco2)C1 CC(C(=O)N1CCC=C(CNC(C23CCCC2C3(F)F)=O)C1)S(N)(=O)=O C1(CNC(c2c(Br)cn(C)n2)=O)CCC2(CCN(C(C3CC3F)=O)CC2)O1 N1(C(C(CCC)(C)C)=O)CC2CCC(C1)C(NC(=O)C(C)Cc1ccccc1)C2 C1(NC(C=CC(C)=O)=O)CCCC12CCN(C(C1CC1C)=O)CC2 CC(CC(F)F)C(=O)NC1CN(C(=O)Cc2csc(=N)[nH]2)CC1F N1(C(c2c(OC)cc(C)s2)=O)CCC2CCN(C(=O)CCCC(C)C)C2C1 C1(NC(C2(CCC)CCOC2)=O)C=CCN(C(C2(Sc3ccccc3)CC2)=O)C1 c1(CC)c(NC(=O)C(=O)NCc2cccc(Sc3ccccn3)c2)cccc1F C12(NC(=O)Cc3c(F)cncc3Cl)CCCC1CN(C(c1cc[nH]n1)=O)C2 c1(C(=O)NCCCCNC(=O)CC2CC23CC3)cc(C)n(C(C)C(=O)OC)n1 C1(C(N2CC=C(CNC(COCC#C)=O)CC2)=O)C2CCC3C(C2)CC13 N1(C(C(C)(C)n2ccnn2)=O)CCC2(CC2NC(=O)Cc2cn3ccsc3n2)C1 C(=O)(C(CC)C(=O)N(C)CCN(C(=O)CCCc1ccc(C)s1)C)OCC c1(C(=O)NCC(CO)NC(=O)CCC2CCCCO2)ccc(F)c2ncccc12 N1(c2c(C(=O)OC)nccn2)CCCC2(NC(=O)Cc3sccc3C)CC2C1 c1(OCC)cc(C(=O)NC2CC3CC(NC(=O)CNC(C)=O)C3C2)ccc1C CCCC(C(=O)N1CCC(C(=O)N(CC(O)COCC)C)(C(C)C)C1)OCC CC(C)CC(C(=O)NCC1(C(N)=O)CN(C(C2(C)CCCN2C)=O)C1)C(N)=O N1(C(COC2CC(NC(C(C)C#N)=O)C2)=O)CC(O)CC1(C)CO c1(OCC)oc(C)nc1C(=O)NC1CCCN(C(=O)CNC2(C)CCC2)C1 N1(C(C2CCC(Nc3nccc(OC)n3)C2)=O)CC(F)(F)CC1C(=O)NC(C)C N1(C(c2cc(CC)ncn2)=O)CC(CNC(=O)CSc2nc[nH]n2)C2(CC2)C1 C1(NCC2CC(C)OCC2)CCN(C(=O)C(C)S(N)(=O)=O)CC1C C1(C(N(CC(C)NC(C23CC2CNC3=O)=O)CC)=O)CCC2(CCC2)C1 N1(C(C(C)NC(CC)=O)=O)CC2(CCN(C(C3CCC(C)O3)=O)C2)C1 Cc1cc(C(=O)NC(CNC(c2ccns2)=O)CC(C)C)nc(O)c1 C1(CC(=O)N(C2C(C)C2C)C2CC2)CC2CC1CN2C(=O)OC(C)(C)C C(=O)(C1=C(C)Oc2ccccc2C1)NCC1CC(NC(CSC)=O)C1(C)C C1(C(=O)NC2CCC(CCNC(C=C(CC)CC)=O)C2)CC2(CCC2=O)C1 O=C(NNc1ccc(Cl)cn1)C1CCCCC(F)(F)C1 c1(C(C(=O)NCC(C)NC(CS(CC)=O)=O)C)c(F)cccc1F C(=O)(C1=CCCCC1C)N1C(C(=O)NCCC(=O)OC)CCC1C(C)C c1(CCC(=O)NCCCCNC(C2C(CC)OCC2)=O)cccc(C#N)c1 c1(CNC2(c3n(CCC)nnn3)CCCC2OC)cccc(Cl)c1Br C(CCCCC(=O)N(CCCNC(C12C=CC(CC1)C2)=O)C1CC1)NC(N)=O C1(NC(Cn2c(CCC)nnc2S)=O)CC2CN(C(C3CC=C(C)CC3)=O)CC12 C1(C(N(CC(C(=O)NCC(C)(C)NC(C)=O)O)C)=O)CCC(C)(C)C1 Cc1c(C(=O)N(C)CC2CCN(C(C3C(F)(F)C34CC4)=O)C2)nn(C)c1Br C1(CCC(=O)N(CC(COCC(C)C)O)C)CCN(C(=O)CC2(O)CCC2)C1 C1(NC(C=CSC)=O)CCOC2(CCN(C(=O)CCc3cn[nH]c3)CC2)C1 N#Cc1cn[nH]c1C(=O)NCC1CC(NC(=O)CCCc2ccncc2)C1 C(=O)(CCC(C)(F)F)N1CCC(C(NOCCC#C)=O)C1C(C)C c1(C(N2CC(CNC(C3(OC)CCC3)=O)C2)=O)[nH]ccc1C N1(C(C2N(C)SCCC2)=O)CCC(CC(=O)NOCC2CC3C=CC2C3)C1(C)C Cn1nccc1-c1nn[nH]c1C(=O)NCC1CC1NC(c1cc(Cl)no1)=O c1(N2C(C(=O)Nc3ncc(C)cc3I)CNCC2)nc(C)nc2ccsc12 C1(NC(c2nc(C(C)C)oc2)=O)CCC2CN(C(=O)C=Cc3cnc[nH]3)CC2C1 c1(C(N(CC(C)N(C(c2c(CC)nns2)=O)C)C)=O)cc(OC)cc(OC)c1 c1(C(N2CC(CCC=C)(C(=O)NCC(F)Cl)C2)=O)ccc(OCCC(C)C)cc1 Cc1nc2c([nH]1)CN(C(=O)C(C)(CO)NC(=O)CCCn1ccnc1)CC2 CC12CNC(=O)N1C(C(N1CCC(CCNC(C3(CO)COC3)=O)C1)=O)CS2 C1(C(=O)NCC2C(CC(=O)NCCC(C)F)C2)CCOC1C Cc1ccc(C(F)(F)F)cc1C(=O)NC1CC1CNC(c1cnc(C(C)C)s1)=O c1(CC(CN(C(C)C(O)Cc2cccs2)CCO)O)ccc(F)cc1O c1(C(c2ccccn2)NCC2(CNC(C)=O)CC2)ccc(F)cc1 N1(C(C(CC=C)C(C)C)=O)CC2CC(C1)CN(C(=O)C(O)CCCCC)C2 CC(C)C(C(=O)NCC1CCN1C(c1cncn1C)=O)n1cnnn1 C1(C(=O)NCC(CN(C(c2ccc(C)o2)=O)C)O)CC12CCC(=O)CC2 C1(NC(c2ccc(CC)[nH]2)=O)CCCCCC1C(=O)N(C1CCOC1)C c12cc(nn1C)CNC2=O.C1(c2ccccc2)(CC(=O)N(C)C)CCCC1 C(=O)(C(O)CC[S+](C)C)Oc1c(C(=O)NCCCN(CC)CC)ccnc1 N1(C(COCC=C)=O)CCC2(CCC2)C(NC(c2ccc3nc(C)cn3c2)=O)C1 C1(NC(C(C)(C)SC)=O)CC(C(=O)NC2(CO)CC(F)(F)C2)CC1O C1(NC(C(CC)N(C)C)=O)C2CC3C1C3C2C(=O)NCC1(O)CCC1 c1(C(=O)NCCC2(C(N3CC(CC)C3)=O)CCC2)occc1CO CCCCC(CNC(c1cc(F)n[nH]1)=O)NC(=O)Cc1csc(-c2nc[nH]n2)n1 C1(OC)CCCC(CC(=O)N(CCCCCNC(C2CC2c2cncs2)=O)C)C1 c1(C(=O)OC)cc(CN2CCCC(NC(c3ccc(N(C)C)cn3)=O)C2)n(C)n1 c1(C(N(C)C(N2CC(C(=O)OC)C(SC)C2)=O)C)cccc(S(N)(=O)=O)c1 c1(CNC(C(=O)NC2OCC(C(=O)OC)C2O)=O)c(C(F)(F)F)cccc1F c1(C(C(=O)NC(CC)C)N(C)CCc2cnn(C)c2)ccc(C(C)(C)O)cc1 C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(=O)C(C)OC2CCCCCC2)C(C)(C)C1 c1(C(=O)N(c2ccc(Cc3ccc(Cl)cc3O)nc2)CO)c(O)cc(O)cc1O C(CN=c1nc(N2CCOC(c3cn(C)cn3)C2)c2c([nH]1)CCOC2)OCCC c1(CNC(=O)NCC(C)(C)OC(=O)CC2CC3CC3C2)cc2ccccc2o1 N1(C(C2CC(C)(F)C2)=O)CCC(C(F)(F)F)C(NC(C2CCOCC2)=O)C1 C(N=c1nc2sccc2c(N2CCC3(CCCC3)C2)[nH]1)C1C(C)CCCC1 C(=O)(C(F)C(=O)NN1C2CN(C(C34CC(C(F)(F)F)(C3)C4)=O)CC21)OC CCC(C)(C(=O)N(C)CC1(NC(c2ccc3cnoc3c2)=O)CC1)C(F)F N1(C(C(c2ccc(Br)s2)OC)=O)CCN(C(=O)CC(F)F)CC1C C1(CC=C)(NC(=O)CN2C(=O)CNC2=O)CCCN(C(=O)CS(=O)CC)C1 C1(CNC(c2n(C(C)C)nnc2)=O)CN(C(=O)CCc2nncs2)CC(C)(C)O1 N1(C(CC2C(COC)C2)=O)CCCC12CCN(C(=O)Cc1cn[nH]c1)C2 CCCC1C(=O)N2CCOC(C2)CCCO1.c1(CC(=O)NCC)ccon1 CCCCC(CC)CC(C(=O)NCCSC)N(C)Cc1occc1C O=C(CCCCCCC(=O)N1CCC1)OCC(C1CC1(Cl)Cl)=O C1(CNC(C2(C)CC(=C)C2)=O)CC(C(C)C)CCN1C(=O)C=Cc1cncn1C N1(CC)CCCC(C(=O)NC2C3CN(C(C4(OC)CCC4)=O)CC23)C1 Cc1cc([N+](=O)[O-])ccc1OC(F)F.C1CCN(C)C(=O)NCCO1 C1(C(=O)NC(C(N2CCC(N(C)CC)C2)=O)CN(C)C)CC2CCCC2C1 C(CC(O)C(=O)N1CCC1CNC(C1(CCC(C)(C)C)CCCCC1)=O)N(C)C CN1N=C(C(=O)N2CCOC(C(=O)NC3CC3c3cnn(C)c3)CC2)CCC1=O Cc1c[nH]cc1C(=O)NC1CCC1C(=O)NCCCc1cnn(C)c1 c1(OC)ccccc1OCCC1CCN(C(=O)C(=O)NC2CC3CCC3C2)C1 c1(C(N2CCN(c3cc(C)cc(Cl)n3)CC2)=O)cc(C)c(C)n(C)c1=O N1(C(C2(C)CC2(F)F)=O)CC2CN(C(c3cncs3)=O)CC2C1 C(=O)(C(C)CCCC(C)C)NC1CCN(C(C2(CC)CCCCO2)=O)CC1(C)C N1(C(C=CCCC)=O)CC(C(=O)NCC23CCC(CC2)O3)C(C)(C)C1 N1(C(C2(OC)CCSC2)=O)CCC(C2(O)CC(NC(C3CCO3)=O)C2)CC1 c1(N2CCCC(C(C)NC(C3CCOC3)=O)C2)ncc2c(n1)CCC2 CCCC(F)C(=O)NC(C1CCN(C(=O)CCc2ccnc(C)n2)CC1)C C1(NC(=O)NCCC)CCC2(CCC2)CC1.N12CCCC(C)(C1)CNC(=O)C2 C(=O)(C(F)C(C)C)N(CC(CNC(C1(CCOCC)CCC1)=O)O)CC Cc1cc(C)c(CC(N2CCCC(CNC(=O)COC3COC3)CC2)=O)c(C)c1 Cc1nc2ccccc2c(C)c1C(=O)NCC(O)CNC(c1cc(O)cs1)=O C1(NC(C2CC(SC)C2)=O)CCN(C(=O)C(C)(C)S(C)(=O)=O)CC(C)(C)C1 c1(-c2nnc(-c3c(CCCCCC)ccs3)o2)c(C)nc2sc(C)nn12 Cc1nc(C(N2CCOC(CCNC(C3CCN(C)C3=O)=O)C2)=O)cc(O)n1 c1(C(N2CCN(C(C3CCn4cnnc4C3)=O)CC2)=O)ccc2scnc2c1 c1(C(=O)NC2C(SC)CN(C(=O)Cc3scnc3C)C2)ccc2[nH]c(=N)[nH]c2c1 C1(NC2(c3n(C(CC)(C)C)nnn3)CCC(C(C)C)C2)CCCC2(C1)CC(O)C2 C1(C(C(=O)N(C)CCO)(C)C)CCN(C(C2CC(=O)CS2)=O)CC1 C(=O)(CCCCCC(C)O)NCC1N(C(c2nc(CC)oc2C)=O)CCC1 c1(C(N2CCC(C(C)NC(COCCOC)=O)C2)=O)cc(COC)oc1C c1(C(=O)OC)cccc(NC(C2COCCN2C(=O)C#CC(=O)O)=O)n1 c1(CC)cc(NC(C2CC3(CC3)CN2C(=O)COC2CCCOC2)=O)ccc1Cl N1(C(C(C)OCC(F)(F)F)=O)CCC2(CC1)CN(C(=O)CCCCCF)CCO2 c1(CNC(=O)CC2CCCN2Cc2cc(Br)cnc2Br)c[nH]c2ccc(F)cc12 S(=O)(=O)(c1cccnc1NCc1cnoc1)N1CCCC(C(=O)NCC)C1 n1(CC)cnc2nc(N3CC4CCC4(C)C3)[nH]c(=NC(C)c3ccnn3C)c12 c1(C(=O)NC(C2(O)CN(C(Cc3c(C)nsc3)=O)C2)C)ccc2sccc2c1 CC1CCc2sc(C(=O)NCCOCCN(C)C(C3(C)CC(F)C3)=O)cc2C1 C1(CC(=O)NCC(C)N(C)C)COCCN1CCNC(=O)CCc1nncs1 C1(C(=O)NC(C)CCN(C)C(C2(CC#N)COC2)=O)CCC(=O)N(C2CC2)C1 N1(C(CC2C(C)(C)C2)=O)CCC(CCCCNC(=O)C=CC=C(Cl)Cl)CC1 CCCCC(C(=O)N1CCCC(F)(C(=O)NC2CC(=O)N(C(C)C)C2)C1)N(C)C N1(C(c2cc(CCCC)nnc2C)=O)CCCN(C(C2CCCO2)=O)C(C)C1 S(=O)(=O)(c1ccccc1F)N1CC2CN(C(c3c(C)nc(F)cc3)=O)CC2C1 C(=O)(C(CC(C)C)N1CCCCC1=O)NC1CN(C(CN(C)CC)=O)C1 CC(CCC(=O)NOCCCCF)NC(=O)Cn1[nH]cnc1=N N1(C(c2c(CCC)nns2)=O)CC(NC(=O)C(C)CO)CC2(CCOCC2)C1 C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NC2CC(O)C(O)C2)CCC(C)C1 c1(C(N(C2CCN(C(C3CCCC(C)C3)=O)C2)CC)=O)cc(C#N)cs1 C1(C)(C(N(CC(CC)NC(=O)CCS(N)(=O)=O)CC)=O)CCCCCCC1 c1(CC(C(=O)OCC)Nc2ncnc(C(=O)OC)c2Br)ccc(F)c(Cl)c1 c1(OC)ccc(CN2CCC(CC(N3CCOC4(CC4)C3)=O)CC2)c(C(F)(F)F)c1 C=CCC(C)(C)CN=c1nc2sccc2c(NC(C)COCC(F)(F)F)[nH]1 c1(C(=O)NCC2C3CN(C(C4(CC#C)CCC4)=O)CC32)cnn2c(=N)[nH]cnc12 C1(CNC(=O)Cc2ccc(Cl)cn2)CC2CCC(C1)N2C(=O)C(O)c1ccsc1 c1(C(=O)NCC(CC(C)C)NC(C(CCC)C)=O)c[nH]c2ccc(F)cc2c1=O c1(C(N2C(C(=O)Nc3ccc(O)c(F)c3)CC3CC32)=O)cccc2c(Br)cccc12 N1(C(CC23CC(C)(OC2)C3)=O)CC2CC(NC(c3occc3Br)=O)CC2C1 C1(CNC(c2n(C)c(O)nc2)=O)CC12CCN(C(=O)C(O)C(F)F)CC2 c1(C(=O)NCC(CNC(C2CCC(F)(F)CO2)=O)OC)c(F)cc(F)cc1F n1(CC(=O)NCC2CC(CNC(C(C)(C)SC)=O)OC2)cc(Cl)c(O)nc1=O c1(C(=O)NC2CN(C(C=C3CCN(C)CC3)=O)C(CO)C2)cnn2c1N(C)CC2 S(=O)(=O)(c1cc(Cl)ccc1Cl)NCCC(=O)NC(C(=O)OC)CSC c1(OC)cc(Br)ccc1CN1CCOC(CNC(c2cc(F)ccc2O)=O)C1 O=CN1CCCC1NC(C(Cc1cn[nH]c1)NC(c1cncc(Cl)c1)=O)=O C#Cc1cc(C(N2CCCC2CN(C(=O)C(CC)SC)CC)=O)cc(Br)c1 CCCCS(=O)(=O)CC(=O)NCCN(CC(C)O)C(c1cnc(C(C)C)nc1)=O N1(C(CCOCCN(C)C)=O)CCCC1CNC(C1C2COCC12)=O C1(C)(NC(c2c(C)cc(C)[nH]2)=O)CCN(C(=O)C(=O)Cc2ccccc2)CC1 Cc1c(C(N2CC(NC(=O)COC3CCC3)CC(O)C2)=O)cccc1F C1(OC)CS(=O)(=O)CC1C(=O)NNC(=O)c1ccncc1C N1(C(C(C)C2CCOC2)=O)CCC2(NC(c3cccc(C4CC4)c3)=O)CCCC12 c1(C(N(CCCN(C(c2cn(C(C)C)nc2)=O)C)C)=O)ccc(F)cc1O N1(C(c2cnc(Cl)s2)=O)CC2CC(N=c3ccnc(C4CCCC4)[nH]3)C2C1 NS(=O)(=O)c1ccc(OCC(N2CCC(c3ccccc3Cl)C2)=O)cc1 c1(C(=O)NCCCCN(C(C2CCC(C)C2)=O)C)ccc2oc(O)nc2c1 C1(N)CCCCN(C(=O)C(N2CCC(C)C2)=O)C1.Cc1nc(CC(C)C)sc1C C1(NC(=O)Cc2cnsc2)CC2CN(C(c3ncc(F)cc3F)=O)CCN2C1=O N1(C(C2(Br)CC2(F)F)=O)CCCC(Oc2ccccc2Br)C1 c1(C(=O)NC2CCN(C(C3(NC(C)=O)CCC3)=O)C2)cnc(O)c2ccccc12 c1(NC(COc2ccc(OC)cc2)C=O)nc(OC(C)C)cc(C)n1.OC c1(OC)ccc(C(=O)NC(C)(C)CN(C(=O)CCS(=O)(=O)N(C)C)C)c(C)c1 Cc1ncccc1C=CC(=O)NC(C)(CNC(C1CCOC1)=O)CO C(=O)(C(O)C(F)(F)F)N1CCCC(NC(C2CC(F)(F)C2(F)F)=O)C1 C12(CC(=O)NC34C(CN(C)C3)C4)CCC1CN(C(C1C=CCS1)=O)C2 C12(CN(C)C(=O)NCc3cscc3Br)CC(F)C1C2 C(CC(F)F)(C(=O)NCC1(C)CCOCC1)N(C)C(C12CC(F)(C1)C2)=O c1(C(=O)NC2(C)CCN(C(c3c(CC)nn[nH]3)=O)C2)cnc2c(F)cccc2c1 C1(CCC)CN(C(=O)CCOC)CC1NC(=O)C(C(C)C)c1cnn(C)c1 C1(C2CC2)(CNC(=O)C=C(Cl)Cl)CCN(C(=O)CCN2CCCS2(=O)=O)C1 c1(C(=O)OC)cc(Br)c(F)cc1N(C1CCNCC12CC2)C(=O)C(OC)OC C1(CNC(c2c(SC)csc2)c2nnnn2C)CC2CS(=O)(=O)CC2C1 c1(CNC(CCSCC)C)nnnn1CC.C(C)(C)(C)OCCO.SCC C1(C(=O)NCCCN(C(=O)CC2CCC(=O)N2)C)CCc2nccn2C1 c1(C(=O)NCC(CC=C)NC(=O)CCCC(=O)NC)cc(F)c(C)cc1Cl CON(CC1CC1)C(=O)C(CCOCCO)NC(=O)CC1CC(C)=NO1 C=CCCC(C)(C)C(=O)NCC(CC(=O)N1CC(CO)(CF)C1)OC c1(OC)cc(C)cc(C(=O)NCC2(NC(=O)C(O)C(C)C)CCCC2)c1O C(=O)(C1Cc2ccccc21)NCCNC(N=c1c(C)cn(-c2ccccc2)[nH]1)=O N1(C(C(C(CC)C)N(C)C)=O)CC2(NC(c3scc(C)c3C)=O)CCCC2(F)C1 N1(C(CSCCOC)=O)CC(CC(C)NC(C2CC2(C)C)=O)C1 C#CCC(C)(CC)C(=O)NCC(CNC(=O)C=CC(=O)OC(C)(C)C)CO CC1C(NC(=O)C2=C(Cl)CCOC2)CC2CCC1N2C(C1CCS(=O)(=O)C1)=O Cc1ccc(CNC(C23CCC2CN(C(=O)CC2CCCN2C)C3)=O)c(O)c1 CC1(C)OCCC1(O)C(=O)NC(C1CCOC1)CNC(C1(O)CCCCCC1)=O C1(C(N2CC(C(C(=O)NCC3(CCC=C)CC3)O)C2)=O)CC(=O)C1(C)C C1(C(=O)NC(C(=O)N2CC(OC(CC)=O)C2)Cc2cn[nH]c2)CCC2(CCC2)C1 CCCC(C)CC(=O)NCCN(CCC)C(N1CCCCCC1)=O C(=O)(C1=CC2(CCOC2)C1)N1CCC(C)(CC(=O)NC2(C)CN(C(N)=O)C2)C1 CCCC(C)(CC)C(=O)N1CC2CCCC2(C(N(C)CP(C)(C)=O)=O)C1 c1(N2CCCC(c3n(C)ccn3)C2)ncnc2c1ccn2C C1(C)(C(=O)NC(C2CCCC2)CNC(c2c(CC)ncs2)=O)CC=CCO1 C1(NC(Cc2cc(OC)c(OC)cc2)=O)CC2CCC(C1)N2C(=O)CN(C)C C1(CNC(c2cnc(C)[nH]2)=O)CN(C(=O)Cn2cc(C(=O)C3CC3)nn2)CCCO1 C1(CNC(=O)CCOCC(F)F)CCCC2CN(C(C3OCCO3)=O)CC12 C1(NC(CC2C(C)CCC2)=O)CCOC(C(=O)NCC2(C)CCCCC2)C1 C12(NC(C(CC)N(C)C)=O)CCC(C1)N(C(C1(NC(C)=O)CCC1)=O)C2 O=C(C1COc2ccc(F)cc21)NCC1(NC(c2ccco2)=O)CCOC1 S(=O)(=O)(c1ccc(N(C)CC2CCSC2)c(F)c1)NCC(CC(C)C)O C1(CC)CN(C(c2cn(C)cn2)=O)CCC1NC(c1ccsc1OC)=O C1(C(C(=O)NCCOC)N(C(C)(C)C)CCOC(=O)C2CC2)CCCC1(C)C C(C)(CCC#N)(c1nnnn1CCCF)NCc1cn(CC)nc1 N1(C(C2(C)CCC2)=O)CCC2(CCCC2NC(=O)CN2CSCCSC2)C1 n1(CCC(=O)NC2C(NC(C3(OC)CCOC3)=O)CC2)c(-c2cccs2)nnc1S C1(c2nnnn2CCCF)(NCCc2ccc(OC)c(F)c2)CCCC(C#N)C1 c1(C(=O)NC2CC(C)N(C(c3cc4ccccn4c3)=O)C2)nc2c(s1)CCCC2 c1(CCC)cc(C(N2CCCC2CCNC(C23CCC2C3)=O)=O)ccn1 N1(CC)CCCN(C(C2(NC(=O)CCC3CCCC3)CCCC2)=O)CC1=O c1(C(=O)NC2CC(NC(c3cccc(C(N)=O)c3)=O)C2)cccc2nc(O)[nH]c12 Cc1nc2c(o1)CCN(C(C1CC1NC(c1ccc(Cl)c(I)c1)=O)=O)C2 C(CCCCC(=O)NCC(C)(CO)NC(c1ccc(C(F)(F)F)c(N)c1)=O)OC N1(C(Cc2cc(C)on2)=O)CCC(C2CCCN(C(C3CC=CCC3)=O)C2)C1 C1(C(=O)OC)COCC2(CCN(C(c3nn(C)c4c3COCC4)=O)C2)O1 c1(CNC(C(=O)NC(c2nc(C)cs2)CC)=O)cc(OC)c(C)c(OC)c1 Cc1noc(Cl)c1CC(=O)NCC(C)CNC(=O)C(c1ccccc1)OC(F)F Cc1cc(C(=O)NC(C)CC(C)NC(=O)C(C)(F)F)cn(C)c1=O N1(C(C(C)Cc2cccc(Cl)c2)=O)CCC(C2(NC(=O)C=CC3CC3)CC2)CC1 C1(CN(C(=O)C(F)CC2CCOCC2)C)CCN(C(=O)C=CC2CCCC2)C1 c1(CNC(C)=O)cccc(C(N2CC(NC(=O)C(C)NC=O)C2)=O)c1 C1(NC(CCC(C)O)=O)Cc2ccccc2N(C(=O)CC2(C)CCCCCC2)C1 C1(C(=O)NCc2cc(Cl)cnn2)CCN(C(c2ncoc2Br)=O)CC1 CCCS(=O)(=O)CC(=O)N1CCCN(C(=O)CN2CCC(C)(O)C2)CCC1 C1(CC(=O)NCC2COC(CNC(=O)CC3(C(F)(F)F)CC3)C2)CC2(CC2)CO1 CN1CCC(CC(=O)NCC(O)C(=O)N(C2(C)CCCC2)C)C1=O N1(c2c(OC)cnc(Cl)n2)CC2(CCCC2NC(C23CCC(C)(C2)OC3)=O)C1 C1(NC(c2c(C)n[nH]c2)=O)CN(CC23CC(CC2Cc2ccccc2)C3)C2CC12 C(C(=O)NCC(C)(C)CCNC(=O)Cc1cccs1)(C(C)(C)C)N(C)C c1(C(N(CC(CC)NC(C2CCCN2C)=O)CC)=O)cc2ccsc2n1C O=C1CCCCC(C(=O)NC2(c3cn(-c4cccnc4)nn3)CCCOC2)N1 C1(NC(C(CN(C)C)O)=O)CCN(C(c2cc(O)nc(O)n2)=O)C12CC2 c1(N2CCC(N3CCN(C(C(CC)C)=O)CC3)CC2)nc(OC)c(F)c(C)n1 C1(NC(Cc2nc(C)[nH]n2)=O)CCN(C)C12CCCN(C(C1CNC(=O)N1)=O)C2 c1(C(C)=O)c[nH]c(C(N2CCCC2C(C)NC(=O)Cc2cnoc2)=O)c1 CCS(=O)(=O)CC(=O)N1CCOC(C(C)NC(=O)CC2CCCC2)C1 CC1CC(O)CN1C(=O)Cc1cccc(CNC(=O)OC(C)(C)C)c1 C12(C(N(CC(C)NC(C3(c4ccnn4C)CC3)=O)C)=O)C=CC(CC1)C2 Cc1cc(C(=O)NCC(C)(F)CNC(c2cnn(C)c(=O)c2)=O)c(C)c(C)c1 N1(C(=O)COC2CCN(C(C3(F)CC=CCC3)=O)C2)CCC2(CC1)CSC2 C12(CN)COCCN1CCN(C(C1(NC(CN(CCC)C)=O)CC1)=O)C2.C(C)(=O)O N1(C(CC(C)(C)OC)=O)CC(NC(c2cc(Cl)c(Cl)n2C)=O)CC1(C)C N1(CC(=O)NC2CCC(NC(C(C(C)C)OC)=O)CC2)C(=O)C(C)C(C)C1=O C1(c2cn(Cc3c(C(=O)OC)con3)nn2)CN(C(=O)CC(=O)N(C)C)CCO1 c1(C(N2CC(CC)C(NC(c3nocc3Cl)=O)CC2)=O)c(C)ccc2nonc12 N1(C(c2n(CC)ncc2)=O)CCC(C)C1C(=O)NCc1nc(C2CC2)cs1 N1(C(c2cnc(C)n2-c2ccccc2)=O)CCC2(CC(NC(=O)C(C)CF)C2)C1 CCC(CC)CC(=O)NCC12CC(CC)(CN1C(C1(C(F)(F)F)CC1)=O)C2 N1(C(c2nnn(C)c2N)=O)CCC2CN(C(c3ccc4c[nH]nc4c3)=O)CC12 CC1CC(NC(=O)C2=CCSC2)CN1C(=O)CC1COC(=O)C1 C(CC(C(=O)NC(C)C(C)(C)CO)NC(=O)Cn1nc(C)cc1C)=CC O=C(O)CCCCOCC(CN1CC(Nc2ccccc2)C1)O C1(C(N2CC(C(C)NC(C(=O)NCC)=O)OCC2)=O)CN2CCN1CC2C C1(CNC(C(C)Sc2n[nH]c(O)n2)=O)CC(C)(C)CN1c1cnc(C#N)cn1 N1(C(CC(C)F)=O)CCN(C(C2OCCCO2)=O)CC1c1cccc(F)c1 C1(C(=O)OC)CCN(C(=O)COCC(C)C)C1CCC(C)C1(n2cnnn2)CC1 N1(CCNC(=O)CCC2OCCO2)CCN(C(c2cscn2)=O)CC12CCC2 C(=O)(C(O)C(F)(F)F)NC1(C(N2CCC(C(C)(C)C)CC2)=O)CC1 C(CC(C)C(=O)N1CCN(C(=O)CNC(C2CSCC(=O)N2)=O)CC1)OC C1(C(N2CC(C(C)NC(C(c3cccc(Cl)c3)CC)=O)C2)=O)CC12CC(C)(C)C2 CSC=CC(=O)NC(C1CCCN1C(c1cn(C)cn1)=O)C C12(C(=O)NC(C)CC(C)(C)O)C(NC(=O)Cc3cccc(C#N)c3)C3CC1C2C3 C1(CNC(C(CC)N(C)C)=O)(OC)CCN(C(C2C(C(=O)NCC)C2(C)C)=O)CC1 N(C(=NCCSC)NC(C)CC1CCCC1)C1C(COC)C1 C12(C(=O)Nc3cc(CC)cc(F)c3)CCN(C(C3(C)CNC(=O)N3)=O)CCC1C2 C(=O)(C(CO)C(C)C)N1C(Cn2cc(CCC(C)=O)nn2)CC1 CSC1=C(C(=O)NC2CC(O)CN(C(c3ccsc3)=O)C2)CCCC1 C(=O)(C(F)C(C)C(F)(F)F)NC12CC(CNC(C3(C=C)CCCCC3)=O)(C1)C2 C1(C(=O)NC2C3CCN(C(C=NOC)=O)C32)Cc2nn(C)cc2C(=O)N1 C12(CCNC(C(C)(C)OC)=O)CCC(C1)N(C(c1cnc(C3CC3)[nH]c1=N)=O)C2 N1(C(C(C(C)(C)C)SC)=O)CC2CCN(Cc3cnc(S)n3CCC(C)C)CC12 C#CCC(C(N)=O)NC(c1nc(Cc2cc(F)ccn2)cs1)=O c1(CC)ccc(C(=O)NCCN(C(=O)Cc2cccc(F)c2Cl)CC)cc1N c1(NC(C=C)=O)ccc(-c2ncccc2C(=O)NC2CCCC2COC)cc1 N1(C(COC(CC)C)=O)CCCN(CCNC(C2CC(C)(C)CO2)=O)CC1 N1(C(C(C)NC(=O)NC)=O)CCOC2(CCN(C(=O)CCc3cnn[nH]3)CC2)C1 C1(CNC(=O)Cc2csc(Cl)n2)CN(C(=O)Cc2cncs2)CC2(CCC2)O1 N1(C(COCCC=C)=O)CCCCCC1C(=O)NC(c1ccc(F)cc1F)C C(CC(C)C)(C(=O)Nc1nnc(Cl)cc1C(=O)OC)NC c1(C(N(C2CN(C(C3(F)C(C)C3)=O)CC23CC3)C)=O)cccc2nc(O)oc12 C(C(=O)N1CCCO1)NC(=O)CCC1(NC(=O)CC2CC3C=CC2C3)CCC1 C1(C(=O)NC2(C#C)CCOC2)CCC(O)CN1C(c1cncs1)=O C1(NC(C23CCCC2CCC3)=O)CCN(CCc2c(C(=O)OC)c[nH]n2)CC1C C1(NC(c2ccc(C)cc2)=O)CC(C)CN(Cc2cccc(C)c2O)C1 c1(C(C(=O)NC(C2CC(NC(=O)CC(C)F)C2)C)(C)C)ccc(F)c(Cl)c1 C(=O)(CS(=O)(=O)C1CCCC1)N(C(C)CCNC(C1(C#N)CCOC1)=O)C N1(C(c2cc(Cl)cc(Br)c2Cl)=O)CC2(CCCN2C(c2cnc(Cl)cc2I)=O)C1 CC1(C)COCCC1C(N1CC(F)(CNC(C23COCC(C2)OC3)=O)C1)=O c1(C(=O)NCCOCCCN(C(CC2C(OC)CC2)=O)C)cc(C2CC2)no1 C1(C(N(CC(C)(C)O)CC)=O)CCC2CCC1N2C(C1CC2(CC2)CO1)=O c1(OCC)ccc(C(=O)NCCOCCNC(C2(C)CC3CC3C2)=O)cc1C CN1CCC(C)(CNC(=O)C(CO)NC(=O)Cc2cnn(C)c2)C1 C(=O)(C(O)CC(C)(C)C)N(CCCNC(c1n(CCC)ccc1)=O)CCO CC(C)CC(CC(=O)N1CCOC(C2CC2)CC1)NC(=O)CSCCN(C)C CCCCCC(C)NC(=O)C(C)N(C(=O)CC1CCN(C)CC1)CC N1(C(C(C=C)O)=O)CCC(C(=O)NOCCOC)CC12CCCC2 N1(C(c2c(C)nn[nH]2)=O)CCC(NC(c2cn3cccnc3n2)=O)C(CO)CC1 N1(C(c2cnc(C)s2)=O)CCC2CN(C(=O)CCN3CCOCC3)CCC12 c1(N(C(CCC(c2cc(C)sc2C)=O)=O)C)cccc2ncccc12 C(C(C(=O)N(CC(F)(F)CC)C)C(C)(C)C)NC(C(CCC)NC(C)=O)=O C1(C(N2CCC2CNC(C2(OCF)CCOCC2)=O)=O)CCC2(CC1)CC2 C1(C(N2CC3(C2)C(=O)N(C)CCN(C)C3=O)=O)CCCC(=O)C1.COC c1(OC)ccc2c(c1)CC(C)N(Cc1cc(C(C)(F)F)ccn1)C2 N1(C(C2N(C(C(C)(C)NC(=O)OC)=O)CCC2)=O)CCCCC(CO)C1 N1(C(Cc2c(C)nccc2)=O)CC2(COC(CNC(c3ccn(C)n3)=O)C2)C1 c1(OCCCc2nnn(C(C)(C)C)n2)ccc(=O)n2c1CCC2 N1(C(CC2CCN(CC(=C)Cl)C2)=O)CCC(C)(C)CC1 c1(C(=O)NC2COCCN(C(C(C)n3cnnn3)=O)C2)cccc2nccn12 CC(C)C(C#N)C(=O)N(C(C)CCNC(c1cn(C(C)(C)C)nn1)=O)C c1(C(=O)NC(CC)CO)ccc(CNC(=O)Cc2cnsc2)o1 N1(C(C(C)=CC)=O)C2CCC1CC(NC(C1CCC1C(F)(F)F)=O)C2 C(=O)(CCCCCSC)NC(CC=C)CNC(=O)CC1CCCC(F)(F)C1 C(=O)(C(C(C)(C)C)NC(=O)CC(C)(C)C)N(CC(C)O)CC N1(C(c2cc(-c3cccs3)[nH]n2)=O)CCOC(c2ccc(Br)cc2)C1 N1(C(CCCC(=O)N(C)C)=O)CC=C(C(C)(C)C(=O)N2CCC(C)(F)C2)C1 C1(NC(c2cc(COC)sc2)=O)C2CCC1N(C(=O)CC(C)CF)C2 c1(CNC(=NC)NCCC(O)C(F)(F)F)cccn2ccnc12 CC1CN(C(=O)CSCc2cccs2)CC(C)C1NC(=O)CC1(O)CCCCC1 c1(CN2CCC3(C(C(=O)NC(CC(=O)OC)C)C3)C2)cccc2[nH]ccc12 C1(CNC(=O)CC2(CO)CC2)CCCCCN1C(=O)C(O)Cc1ccccn1 c1(C(C)C)cc(Cl)ccc1N(C(=O)Cc1cn(CCOC2CCOC2)nn1)CC c1(OC)ccc(C(N2CCC(NC(c3cncnc3C)=O)C2(C)C)=O)cc1C c1(N(C)CCF)ccc(Br)c(S(=O)(=O)NCC2CCCC(CO)C2)n1 c1(OCC)ccc2cc(C(N3CC(O)(CNC(=O)C(C)C(C)(F)F)C3)=O)[nH]c2c1 N1(C(c2ccc(C)o2)=O)CCC2C1CCCN2C(c1cncnc1C)=O CCC(CCC(=O)N1CCC(CO)C(O)C1)NC(=O)CCc1cccnc1 CN1CCC(C)(C(N2CCC(C)(C(=O)NCC3C=CCCC3)C2)=O)C1 C(=O)(C1=CS(=O)CCC1)N1CCC(C(C(C)C)NC(CC)=O)CC1 c1(CC(C(=O)NC(C)CNC(c2ccc(Br)s2)=O)C)cccc(Cl)c1 c1(C(N2CCN(C(C(CCC)CC)=O)CC2CCO)=O)cc(S(N)(=O)=O)c(C)o1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1CC)N(C1CCCCC1)C(CC#C)C CN=S(C)(=O)c1ccc(C(=O)NC2CC(NC(=O)CCC(=O)NC(C)C)C2)cc1 C(=O)(C1=CC2(CN(C(=O)NNC(C3CCCCC3F)=O)C2)OC1)OC CCC(C(=O)NC12CCOC(CNC(=O)CNc3cc(C)oc3C)(C1)C2)C(C)O c1(CC=C)ccccc1C(=O)NC(C(=O)NCCCOCCCO)c1cccs1 C1(C(=O)NCCN(C2CCCCC2)C(c2c(C)coc2)=O)OC(C)(C)OC1(C)C CN=c1nc(N2CCCC(C(=O)N(C)C)C2)[nH]c(=NC(C)CCn2cncn2)[nH]1 C12(NC(c3n(CC)c(O)nc3)=O)CCCC1N(C(c1scnc1COC)=O)CC2 C(=O)(CS(=O)(=O)C1CC1)N(CC(CC)NC(c1cc(F)cc(Cl)c1)=O)CC C(C(C(=O)NC(CO)CCF)NC(=O)CCCC1CC1)SCC C(CC(CC)C(=O)NC1CC(C)(C(=O)NCc2ncccc2C)C1)=CC N1(C(=O)NCCC(O)CC(c2cscn2)=O)CCC(C)(CC(=O)OC(C)(C)C)C1 Cc1ccncc1-c1c[nH]nc1C(=O)Nc1cncc(F)c1 CC1CCC(NC(c2cccc(N)c2)=O)CN1C(=O)C1=CCCCC1 Cc1nc(CC(=O)NC2(CNC(c3ccc(C(N)=O)[nH]3)=O)CC2)cs1 c1(CNC(c2n(CCC)nnn2)c2occc2Br)ccc(C(C)CC)cc1 C=CC(C)(O)CC(=O)NCC(C1CC1)NC(c1ccc(NC(=O)OC)cc1)=O N1(C(Cc2ccc(CC(C)C)cc2)=O)CCC(C)CC1CNC(C1CN(C)C1)=O CC(C)CC(F)(F)C(=O)NC(C)CNC(c1cccc(-c2ccccc2)c1)=O C(=O)(C(C(C)(C)C)SC)N(C1CCC(NC(C2C(=C)CC2)=O)CC1)C C1(C(=O)NC(C)CNC(=O)C(C)(C)C(N)=O)CCC(S(N)(=O)=O)CC1 CC1(CNC(=O)CC2CCOC2)CCCN(C(=O)CCC2CC3CCC2C3)C1 c1(C(=O)NCC(N2CCCC2)C)ncc(N)cc1Cl C1(C)(C(N2C(C(N(CC(O)CF)C)=O)CCC2)=O)CC(F)(F)C1 CCCC(CCC)=CC(=O)NCc1cccc(CN(C(=O)CN(C)C(C)C)C)c1 Cc1cccc(SCC(=O)NCCCC2CCCN2C(c2n[nH]c(C)c2N)=O)c1 N1(C(C2C3CN(C(C(C)CC4CC4)=O)C2C3)=O)CC(=O)NCC1C(N)=O C(=O)(C(F)CCC(C)(C)C)NC1(CO)CN(C(CCC(C)OC)=O)C1 c1(OC)cc2c(cc1C(=O)NC(C)CCNC(c1cnsn1)=O)CCC2 c1(C(=O)NC(CN(C(=O)C(C)CC2CCCC2)CC)C)ncnc(O)c1F Cc1c(Cl)cnc(NC2CC3CCC2N(C(=O)CC2COCCO2)C3)c1C#N N1(N2CC(CC(C)(C)C)C2)CC(C=O)C(CNC(=O)Cn2ncnn2)C1.N(C)C c1(SCCC(=O)N(C2CCN(C(=O)C(C#N)CC)C2)CC)ccc(C)cc1 C(C(=O)N(CCS(C)(=O)=O)C)(C(C)(C)C)NC(CCCCC)=O CCC(CC(=O)N1CCC1(C)CC(N1CCCCC1C(F)F)=O)CC(C)C c1(C(C(=O)NC(CNC(CCOC)=O)C(C)C)O)ccc(Cl)c(F)c1 Cc1c(C(=O)NCC2CC2CC(=O)NCc2cn(C)nn2)noc1C1CC1 N1(C(C2CCC(=C)CC2)=O)CC(NC(c2cc(CCC)nc(O)c2)=O)C2(CC2)C1 c1(CC)cc(C(=O)NC23COC(CNC(C4(C#N)CC4(C)C)=O)(C2)C3)ccn1 C1(CNC(C(CC)SC)=O)(COC)CCCN1C(=O)Cc1cnc(C)[nH]1 C1(C(=O)NCC#CCNC(C(CC(C)C)C)=O)CN(CP(C)(C)=O)C1 CC1=C(F)CN(C(C2C3CCC(C3)N2C(=O)CCc2ncccn2)=O)CC1 C(CNC(C1CC1C(F)F)=O)(CC(F)(F)F)NC(c1c(=N)[nH]cnc1)=O N1(C(C2C(C)(C(F)F)C2)=O)CC2(CCCC2)C1C(=O)NCCC12CC(CCO1)C2 C1(C(=O)NCCN(C(=O)C(=Cc2cccnc2)F)CC)CCC(=O)N(C)C1 C1(C(N2CC(C#C)OCC2)=O)CC2CN(C(=O)CCCOC)CC2C1 CC1(C)CC(C(=O)NCc2c(O)cccc2F)CN(C(C2(C)CC2(F)F)=O)C1 C1(C(=O)NC2CC(NC(C3CC34CC4)=O)C2)CCC=CCC1 C12(OCC)CCC(C(=O)N(CCCCNC(c3occc3Cl)=O)C)(CC1)C2 N1(C(C2CC3(CO)CC2C3)=O)CC(CO)OC2(CC2)C1 N1(C(Cn2ncc(CNC(=O)COC)c2)=O)CC(CC)C2(CCC2)C1 c1(C(=O)NCCC2CC(NC(c3c(C)ncnc3)=O)C2)csc2cncn12 C1(NC(C2CCC(C)C2)=O)(CF)CCN(C(=O)Cn2ccccc2=O)C1 C1(C2CN(C(=O)NC3CCCCC3NS(C)(=O)=O)C2)(NC(C(C(C)C)C)=O)CC1 c1(C(N(CC(CC)NC(=O)Cc2ccc(Cl)cc2Cl)C)=O)ccc(F)c(C)c1 Cc1cc(NC(c2cc3[nH]ccc3s2)=O)ccc1NC(c1ccsc1C)=O Cc1cccc2[nH]cc(C(=O)NC3CCSC34CN(C(=O)COC(F)F)C4)c12 C(CCCCCC(=O)NC1CCCOC1)NC(c1ccc(N)c(F)c1)=O c1(C(N2C3C(NC(c4ccn(C)n4)=O)CC(CC3)C2)=O)ccc2c(c1)COCO2 N1(C(CC2CC(N(C)C)C2)=O)CCCC12CCCN(C(=O)Cn1cnc(=N)[nH]1)C2 C1(CNC(C=C=C(C)C)=O)CC(F)(F)CN1C(=O)C(=O)NCC1CC1 CC1(C(=O)NCCCNC(C2CC2c2cccs2)=O)CCCO1 C=C(C)C(CC(=O)NC1CCCN(C(=O)C(O)C2CCC2)C1)OCC N1(C(CCc2c(C)n[nH]c2C)=O)CC(CNC(=O)Cc2cnnn2C)CCC1C C1(NC(Cc2c(C)nc(SCC)s2)=O)COCCN(C(=O)CC2CCC(=O)O2)C1 C1(C(N2CCC(C(F)F)C2)=O)(COC)C=CCN1C(c1cc(OC)nn1C)=O Cc1cc(Cl)nc(Cl)c1NC(C1CCN(C(=O)C(CO)c2ccccc2)CC1)=O CCC(CCC(=O)NC1CC(CCC(=O)NCCC(C)(C)CO)C1)OC c1(NC(N2CCCC(C)C2CN=c2[nH]nco2)=O)ccc2c(c1)COC2(C)C N1(SCC(=O)NCC2CC(NC(CN(c3cnccn3)C)=O)C2)CCCS1(=O)=O N1(C(C2C(C)CNCC2)=O)CCC(O)CC1C(N1CCOC(C)(C)C1)=O Cc1cc2c(CC(=O)NC3CN(C(=O)OC(C)(C)C)CCO3)csc2s1 N1(C(CCC(=C)Cl)=O)CC2CC1CN(C(c1ccnc3c1CCC3)=O)C2 C1(CN(C)C(C2(c3cc[nH]n3)CC2)=O)CC2CCCC2C1.C1CCCC(=O)N1 C=Cn1nncc1C(=O)NC(C)CCN(C)C(c1ccc(OC(F)(F)F)cc1)=O C1(N(C(CC(CC)C)=O)C)CN(C(=O)CCc2cc(C)cs2)CCC1O C1(C)(C(=O)NCCCCC)CCCN(Cc2c(C)n[nH]c2C)C1 CCCC(C)C(=O)NCC(CC(=O)NCC(C)C(C)O)C1CCC1 N1(C(c2c(C)cn(C)n2)=O)CCCOC(CNC(c2cc(Cl)c[nH]2)=O)C1 c1(C(=O)NCCC2(O)CN(C(C(C)(C)OC(C)C)=O)C2)cn2c(n1)C(C)CCC2 CC1(C)CCC=C(C(=O)N2CCC(NC(=O)C(Cc3ccccc3)C3CC3)C2)C1 c1(CC(=O)NC2C3CCN(C(C=C(C)C(F)F)=O)C32)cnn2c1OCCC2 C(CCCCC(=O)NCC1(OC)CCN(C(=O)C=Cc2cncc(O)c2)C1)OC N1(C(C2ON=C(CC)C2)=O)CCCCC(C(=O)NCCC2(COC)CCC2)C1 C=CC1(C(N2CC(C(C)(C)O)(CNC(=O)CCn3ccc(C)n3)C2)=O)CCC1 N1(C(Cc2ccn(C(C)C)n2)=O)CC2(CCN(C(c3ccnnc3O)=O)CC2)C1 C1(C(N(C)CC2COCCN2C(=O)CC2CCOCC2)=O)CCc2n[nH]cc2C1 N1(C(C23C(NC(c4c(CC)c[nH]c4)=O)C4CC2C3C4)=O)CCc2cccc(C)c21 C1(C(C)(C)C)CCN(C(c2ccco2)=O)C(CNC(c2cc(O)nc(Cl)c2)=O)C1 c1(C(=O)NCC2C(CNC(c3cc(=N)[nH]c(Cl)n3)=O)C2)ccc2nc(O)[nH]c2n1 C1(C(=O)NCCCCNC(C2CCC=CCCC2)=O)CCc2nccn2CC1 c1(C(N2CC(O)(C(=O)NCC3(CC)CCCC3)C2)=O)sccc1C#N N1(C(N(c2ccc(Cl)cc2Cl)C)=O)CCCC12CCCN(CCO)C2=O C1(CNC(c2cccc(F)c2)=O)CC(O)CN1C(=O)COCC1CCC1 C1(CCOC)CN(C(=O)CC(F)F)CCN1C(=O)CCCCCOC N1(C(c2ccc(C)s2)=O)CCN(C)C(C(=O)NC2CCOC(C)(C)C2)C1 C1(CCCC)CCCC1(c1nnnn1C1CCC1)N(C1CC1)CC1CSC1 N1(C(Cc2nnc(C)s2)=O)CCN(C(c2cc(Cl)ccc2C)=O)C(CF)C1 c1(OC)ccc(C(=O)NCC(CO)NC(=O)C(F)(F)C2(O)CCC2)nc1OC N1(C(CSC(CC)CC)=O)CCCC(C2(NC(=O)C(C(C)C)n3cncn3)CC2)C1 N1(C(C(=O)OC)COCCNC(C)=O)CCN(Cc2cn(C3CCC3)nn2)CC1 C(CCCCC(=O)N1CCOC(C)C1)NC(Cc1c(C)occ1)=O C1(C(C(=O)NC2CCC2)N(CC(C)OC)CCOCC)CCC(C)(C)CC1 c1(C(N(CCN(C(=O)CN2OC(C)(C)CC2=O)C)C)=O)cncc(Cl)c1Cl c1(NC(C(C)Oc2ccccc2F)=O)nc2cc(F)c(F)cc2[nH]1 N1(C(C(C=C)C)=O)CCC2(CCN(C(c3ccc(OC)nc3)=O)C2)C1 N1(C(=O)NC2CCCC(C)C2)CCCC(C)(C)C1NC(=O)OC(C)(C)C N1(C(c2c(C)cnnc2)=O)CCCN(C(c2cc(F)c(F)c(F)c2)=O)C(C)C1 c1(CNC(CCC(C)OC)=O)c[nH]c2nc(F)ccc12.C12CCN(C1)C2 S(=O)(=O)(c1ccc(OC(F)(F)F)cc1)C(N1C(C)C(=O)N(C)C(C)C1)=O N1(C(CN(C2CC2)CC)=O)CC(CNC(C2CC(F)(CF)C2)=O)N2CCC1C2 C(N=c1[nH]c(C(=O)NCCOCC)cs1)c1ccc(C#C)s1 C(CC(=O)N1CC(c2cccnc2)C1)(C1CC1)NC(C(SC)SC)=O N1(C(c2ccc(OCCCC)cc2Cl)C(=O)NCC)CCc2c(C)cccc2C1 C1(C(N)=O)CCCC(C(=O)NCCNC(C23CC(C2)C(C(F)(F)F)O3)=O)CC1 c1(CNC(C2CCC(NC(c3ccn(C(C)C)n3)=O)C2)=O)ncccc1Cl c1(C(=O)NC(C(=O)NC(c2ccc(C)cc2)C)C2CCCC2)cccn(C)c1=O CC1CN2CCN1C(C(=O)NC1CN(C(c3ccc4nn[nH]c4n3)=O)CC1C)C2 c1(C(=O)NC2(CN(C)C(C3CC(O)C(F)C3)=O)CC2)cc(Br)cnc1N C=C=CC(C)C(=O)N(CC(=O)NC1C(=O)NCC1O)C CCCCC(CNC(C1OCCO1)=O)NC(c1ncccc1OC(F)F)=O C1(O)(CC(=O)NC)CCCN(CC(c2cc(F)ccc2OC)O)C1 Cc1c(C(=O)N(CC(C)NC(C2CC2c2ccc(F)cn2)=O)C)sc2nccn12 Cc1ccc(F)c(OCC(=O)N(C2CCCN(C(C3CCCCO3)=O)CC2)C)c1 c1(OCC(=O)NCC(CNC(c2onc(CC)n2)=O)C)cc(Cl)ccc1Cl c1(C(=O)NC2(C(N3CCC(C(CC)C)CC3)=O)CC2(C)C)ncc(C)cc1F Cc1ncc(NC(=O)C(C)CNC(=O)C(C)(C)n2ccnn2)cc1C#N c1(C(N2C3(CN(C(C(C)(C)C)=O)C3)CC2)=O)ccc2[nH]nc(I)c2c1 CC1(NC(=O)CCC(=O)N2CCOCC2)CCN(C(=O)C2=CCCCO2)CC1 N1(C(Cc2cc(C(C)C)no2)=O)CC(NC(=O)C(C)CCO)C(F)C1 N1(C(C)C)CCC(NC(=O)CC2CCC(NC(=O)C(C)n3ccnc3)CC2)C1=O c1(C(C(=O)NCC2CCCO2)N(CC(=O)OCC)CC2CC2)cc(C)co1 C1(NC(=O)NCC(O)CC2CCOCC2)CN2CCC1C2 Cc1c(C(=O)NC2CC(NC(=O)C(=C3CCCCC3)F)C2)ccn1C(C)C N1(C(c2c(CC)con2)=O)CCN(C(=O)CCCSC(C)(C)C)CC12CC2 c1(C(C)C(=O)C2C3C(CC2)NCCC2CSCCN2C3=O)ccc(F)cc1F n1(CCOC)ccc(=NC(=O)CC2CC3(CC3)CN2C(C2CC2C(=O)OC)=O)[nH]1 N1(C(c2c(-c3n(C)ccn3)nns2)=O)CCC(CO)(NC(C2CC2(C)C)=O)CC1 N1(C(C(N2CCSCC2)C)=O)CC(NC(=O)Cc2nc(=N)[nH][nH]2)CC12CCOC2 CCC(N=c1[nH]c(=NCCCc2nccs2)c2[nH]ccc2[nH]1)C1CCCCO1 c1(CC)ncoc1CNC(C1CC(F)(CNC(=O)CC(C)F)C1)=O C12(NC(C(C(C)O)NC(N)=O)=O)CCC(CC1)N(C(=O)CNC(=O)C1CC1)C2 CC1CCN(C(=O)CN2CCCCC2)CC1CNC(=O)CCC1CCOCC1 c1(OCC(=O)NC2CCC(CCNC(c3ccc(F)o3)=O)C2)cccnc1 N1(C(COCC#C)=O)CCCC(O)(CNC(c2nc(C3CC3)cs2)=O)C1 C1(F)(CNC(Cn2c(C)nnn2)=O)CCN(C(C2(C)CC=CCC2)=O)C1 C1(CC=C)(NC(C2CC2C(F)(F)F)=O)CCCN(C(c2ccnn2C(C)C)=O)C1 c1(CC)onc(C(N2CCC2CC(=O)Nc2nc(C)co2)=O)c1C c1(OCC(=O)NC2C(CNC(=O)CC3C=CCCC3)CCC2)ccc(F)cc1Cl C1(C(N)=O)CCCN(CCC(=O)NCC2(F)CC(C(=O)NCC3CC34CC4)C2)C1 C(CC(C(C)C)NC(=O)CSCCC(F)(F)F)NC(C1C(C)=C1)=O CC(C(=O)NCCCNC(=O)CNc1ccc(C(F)(F)F)cn1)C(F)F C(C(=O)NC1CN(C(C2(C)CCCO2)=O)C1)(C(C)C)NC(=O)OC C(C(=O)NCC#CCNC(c1ccnnc1O)=O)(C(C)C)c1cnc(C)s1 C(C)(C)(C(=O)N(CCCNC(=O)C(C)N1CCC1)COc1ccccc1)OCC FC1(F)CC2CC1CC2CNc1ccc(CCc2cccc(C(F)(F)F)c2)cc1 C1(O)(CC(=O)NCC(C)CNC(=O)CC2CCCC(=O)C2)CCCN(C)C1 C1(CCNC(CCC)=O)CCN(c2ncc(CSc3ccccc3)cn2)CC1 N(C(=NCC1CCCO1)NCc1ccnn1C)C(c1cnccn1)C C12(C(N3C(C)CCC(NC(c4n(CCC)ncc4)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 c1(-c2nnc(N3C(c4cccc(F)c4)COCC3)n2C)c[nH]c2cc(C)ccc12.CS C1(CN(C(=O)Cn2nnc(C3CC3)n2)CC)CCCN(CCn2cc(N)cn2)C1 C1(C(N(CCCNC(C)=O)C)=O)(NC(=O)CC2CCOC2=O)CC(O)C1 c1(OC)ccc(Cl)cc1C(=O)Nc1ccsc1C(=O)Nc1ccc(C(N)=O)nc1 CCCCCC(=O)NCC(=O)NC(C)(CNC(c1cnoc1C)=O)C1CCC1 C1(CC=C)(NC(=O)C=CC(C)C)CN(C(=O)COCC2CCCOC2)C1 C=CC1CCCN(C(c2coc(CNC(=O)Cc3cnccc3C(N)=O)c2)=O)C1 N1(C(C(CCC)C#N)=O)CCC(C)(C)C(NC(=O)C(C)OC2CCCC2)C1 c1(NC(C(CC)NC(c2ccnn2CC)=O)=O)ccc(C)c(O)c1C N1(C(C(CC2CC2)OC)=O)CCCC(CNC(=O)COC2CC2)CC1 C1(NC(c2c(C)n[nH]c2)=O)CCN(C(=O)CCCc2cnn[nH]2)CC1C Cc1cc(C)c(C#N)c(NCC2CCC(NC(=O)CCc3ncc[nH]3)C2)n1 N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)COc2ccccc2Cl)C(CF)C1 C(C(O)CC(=O)NCc1ncccc1O)NC(=O)CCC1CC1 C1(O)(CNC(CN(CC)CC)=O)CCN(C(C2(C#N)CCC2)=O)C1 C1(C(N(OC)CC2CC2)=O)CC2C=CC1N(C(=O)CCOCCN(C)C)C2 C1(CC(=O)OC)CCCN(N2CCN(C3CCCCC3)CC2)C1 C(=O)(C#CC1CCCCO1)NCC(CNC(C1CC(C#C)(O)C1)=O)C c1(C(N2CC(CNC(=O)CC3CCCOC3)C(C(F)(F)F)C2)=O)cnc2n1CCS2 c1(CC)oc(C)cc1C(=O)NCCN(C(=O)C(C(C)C)n1cc(C)cn1)C c1(C(=O)NCCCCn2cc(C3CC(F)(F)C3)nn2)cc(F)ccc1Cl N1(C(c2nc(C(N(C)CCO)=O)sc2)=O)CCC(Nc2ccc(Cl)cc2)CC1 C1(NC(c2c(CC)ccs2)=O)CCCC1(C)CN(C(=O)C(CO)OC)C Cc1c(C(=O)NC2CCC2NC(=O)C(C)C(C)(F)F)nn2ccccc12 N1(C(C(C(C)C)NC(=O)OC)=O)CCCC(CCNC(c2cn[nH]c2)=O)CC1 S(=O)(=O)(c1ccc(Br)cc1NCC1(CC)CCOC1)NCC1(SCC)CC1 N1(C(CCCC#C)=O)CC2(CC(NC(c3ccc(SCC)cc3)=O)CO2)C1 C(=O)(C1OCCc2c(O)cccc21)NCC(CNC(=O)C=CBr)OC NS(=O)(=O)CC(=O)NCC1CC(F)(CNC(=O)CSC(F)(F)F)C1 C(=O)(CCCCC#Cc1ccccc1)N1CCN(C(C(C=CC)O)=O)CC1CF C1(NC(C2(CC)CCCCC2)=O)CCN(C(C2SCCS2)=O)CC1C(C)C c1(C(N2CCC(CC(=O)NCCn3c(C)ncc3)C2)=O)cc(Cl)c(Cl)cn1 Cn1c(C(=O)NCCC(C)(C)CNC(=O)CCc2cnn[nH]2)cnc1S c1(CC)nc(CC(=O)NCCC(=O)Nc2ccccc2)cs1 N1(C(CCCNC(C)=O)=O)CC2COCC2(C(=O)NC2CC(C)OC2=O)C1 N1(C(c2n(C)nnc2)=O)CCN(C2CCN(C(=O)CNC(C3CCC3)=O)C2)CC1 c1(-c2ncc(C(=O)NCC(CC=C)NC(C)=O)[nH]2)cc(F)ccc1C(F)(F)F c1(C(C)F)ccc(C(=O)N(C)CCN(C)C(c2ncoc2Br)=O)cc1 C(=O)(CCC(C)NC(C12CC1CN(C(C1(O)CCCCC1)=O)C2)=O)OC C1(C(=O)NCCCCCC2CC2)(NC(C)=O)CCCC1C c1(OC)cccc(C(O)CNC2CCC(CC(=O)OC(=O)C3CC3)CC2)c1 c1(C(N2CC(N(C)C(C34CC5CC3C4C5)=O)C(O)C2)=O)cc(F)cc2ccncc12 c1(C(c2n(CCSC)nnn2)NCCC2CC=CCC2)nc(C)n2c1CCCC2 N1(C(C(C)Cc2ccc(CC(C)(C)O)cc2)=O)CC2CC1CN2C(=O)C(C)(C)F C1(C(=O)OC(C(CC)C)C)CC2C=CC1NC2 c1(C(=O)NC(C(C(C)C)NC(c2cnc(C(C)C)s2)=O)C)ccc2nc[nH]c2c1 N1(C(C2CN(CC)C(=O)CC2)=O)CC(CO)C2(C1)CN(C(=O)Cn1cccc1)C2 c1(N2CCC(CCOC)C2)nnc(COC(C)C(C)C)n1CC(C)C C12(NC(Cc3n(C)nc(C(F)(F)F)c3)=O)CCC(CC1n1cc(CO)nn1)C2 C(=O)(C(C)(O)C1CCC1)NCC(Cn1cc(CO)nn1)OC Cc1cc(C(=O)NC2CN(C(C3COCCOC3)=O)CC2C)ccn1 c1(CC)nc(C(=O)NCCCC(C)NC(=O)CC(O)C2CCCC2)cs1 C1(C2CCCOC2)(NC(CC(CNC(C(C)=C2CC2)=O)(C)C)=O)CC1 c1(C2C(C(N(C(C)CCCO)C)=O)C2)cccc(F)c1 C(Cc1ccccc1)(C(=O)NOCC(N)=O)NC(C(CC1CCC1)OC)=O c1(C(N2CC(N(C(Cc3cc(C)no3)=O)C)C2)=O)coc2c1CS(=O)(=O)C2 c1(OC(C(=O)NCC2CCN(C(CCCCC)=O)C2)C)ccccc1C#N Cc1cnc(NCc2c(Cl)cccc2Cl)c(S(=O)(=O)NC2CC3CCC2O3)c1 CCC(C)(F)C(=O)NCC(c1cccc(OC)c1)NC(c1nccnc1C)=O c1(C(C)C)nccc(C(=O)NCC=CCNC(C2CC(C(F)(F)F)CO2)=O)n1 N1(C(C=C(C)C(C)C)=O)CCC2(NC(=O)C(N)=O)CCCCC12 CN=S(C)(=O)c1ccc(C(=O)NCC(C)(C)CNC(c2ccc(O)nc2)=O)cc1 Cc1c(F)cc(C(=O)NCC2(O)CCCN(Cc3ccc(Cl)c(Br)c3)C2)cc1Br c1(C(=O)NC(CC(C)NC(C(C)(C)OCC)=O)C)n[nH]c2c1CCCC2 C1(NC(c2cn(CC=C)nc2)=O)CCN(C(=O)Cc2ccc(C)o2)CCC1CO Cc1cc(C(=O)NCC2(NC(=O)C=Cc3ncc[nH]3)CCCCC2)c(F)cc1N n1(CCOC)cc(C(=O)NC(C)CC(C)NC(c2cc(C)ns2)=O)c(C)n1 c1(C(N2C(CNC(C(C)C#N)=O)CC2)=O)cc(F)cc(S(N)(=O)=O)c1 c1(C(=O)NC2CC(NC(C(CCC)C)=O)C2)c(Br)ccc(F)c1OC C1(NC(c2n(C)c(S)nn2)=O)CCC2CC1CN2C(c1n[nH]cc1F)=O N1(C(c2cccc(NC(C)=O)n2)=O)Cc2cc(Cl)ccc2CC1c1ccccc1 c1(CC)c(C(=O)N(C2CCC(NC(=O)CC3(CSC)CC3)CC2)C)csc1C C1(NC(CCC(=O)NCC)=O)CCN(C(=O)C(F)C(C)(C)O)C12CC2 C12(CC(=O)NC3CC3CNC(=O)COc3cccnc3)CCCC1C2 c1(NC)cncc(C(=O)NC(C(N2CCC(C(C)C#N)CC2)=O)C2CC2)c1 Cc1ccccc1C(=O)NCCC1COCCN1C(=O)CC1COCCN1C c1(C(N2CCOCC(CO)C2)C(=O)NCCC)ccc(F)c(-c2ccccc2)c1 C1(CN(C(Cc2ncc(C)o2)=O)C)CCN(C(=O)CSc2cccc[n+]2[O-])CC1 Cc1nc(C)c(C(=O)NC2CN(C(=O)C=CSCc3ccco3)C3CC23)[nH]1 N1(C(c2ccc(COC)cc2)=O)CC2(C1)CN(C(=O)C(C)SCC)CC2CO CCCCCC(C)C(=O)n1ccnc1C1COCCN1Cc1ccc(F)cc1Cl c1(NC(N(CCC=C)C2CNC2)=O)cn2ccc(-c3cc4sccc4s3)cc2n1 N1(C(CC(C)F)=O)CCN(C(c2cc(F)ccc2Br)=O)C(CCO)C1 Cc1csc2nc(COC(c3ncc(Cl)cc3Cl)=O)cc(=O)n12 N1(C(COCCCCC)=O)CC(NC(=O)CC2CC23CC3)C(n2ccnn2)C1 C1(CNC(c2c(CC)c[nH]n2)=O)CC2(C1)CN(C(C1CCCC(OC)C1)=O)C2 Nc1ncc(C(=O)NCC2(CNC(C3CC(CF)C3)=O)CCC2)cc1C(F)(F)F c1(C(=O)NC(C(=O)NCC(C)(C)N(C)C)CO)ccsc1C#N C12(NC(C3C(CC)OCC3)=O)CCC(CC1)N(C(c1cn(C)nc1C(C)C)=O)C2 N1(C(C=CCC)=O)CCCC(c2n[nH]c(CNC(=O)CC3COCCN3C)n2)C1 c1(OCC(N2CCC(NC(=O)CN3CCS(=O)CC3)C2)=O)cccc([N+](=O)[O-])c1 C=C(C)CC(C(=O)NCCC1(C)CCOCC1)NC(C1CCCO1)=O C1(CCCCCCONC(CC2CCN(C(C)=O)CC2)=O)CCCCC1(F)F C(=O)(C1CCCc2nn[nH]c21)NC1C(CNC(c2ccc(OCC)cc2)=O)CC1 CCCCCC(O)CC(=O)N1CCC(NC(C2CCC(C(C)C)CC2)=O)C(O)C1 c1(C(N(C2CN(C(c3c(C)nc(CCC)o3)=O)C2)C)=O)cnc2ccccc2c1 C1(NC(=O)C2CC2)CCCN(C(=O)CCC#N)CC1.Cn1nnc2c1C(=O)NC2 CCS(=O)CC(=O)NC1CC(CCNC(=O)Cc2ccccc2C)C1 C1(C(C)NC(C(C)OCCC=C)=O)CCN(C(C2CCCC(C(N)=O)C2)=O)CC1 c1(N2CC3C(CNC(Cc4c(C)noc4C)=O)C3C2)c(F)cccc1[N+](=O)[O-] C(CC(C)(C)C)(C(=O)NCCNC(=O)C(C)Cn1ccc(C)n1)OC c1(CNC2CCC(C(=O)Nc3c(C)n(C)nc3)OC2)cc(F)cc([N+](=O)[O-])c1 C1(CN(CC(F)F)C(C2CCC2)=O)OCCC1NC(=O)CCOC1CCOCC1 CC(C)(C)C(CNC(c1c[nH]c(=N)s1)=O)NC(c1cn(C2COCC2F)nn1)=O c1(C(C)C(=O)OCC(=O)NC2CC(=O)C2)ccc(Br)cc1 c1(C(N(C(CC)CO)CCN2CCOCC2)=O)ccnc(OC(F)F)c1 C=C=CC(C)C(=O)N(CCC(=O)Nc1cccc(C(C)F)c1)CC=C C1(C#N)(C(=O)NCC2(COC)N(C(CCOCC#C)=O)CCC2)CCCCCC1 CC1(C)C(CNC(c2cnc(=N)[nH]c2)=O)CCN1C(c1coc(Br)n1)=O CC1CCc2nc(CNC(=O)C(=O)NCC(c3ccccn3)C)sc2C1 N1(C(Cc2cccc(OCC)c2)=O)CCOCC(F)(CNC(=O)C(C)C(C)C)C1 c1(CNC(Cc2c(C)noc2)=O)ccnc(C(=O)N(CCN(C)C)CC2CC2)c1 C1(NC(CSCC=C)=O)CN(C(=O)CC2(C)CCOC2)CC1OC c1(C(=O)NC(C)C(CO)NC(C2(C)CCCO2)=O)ccnc2ccncc12 Cc1ccc2c(c1)C=C(C(=O)NCC(C)N(C)C(c1ccnnc1S)=O)CO2 N1(C(c2cnc(C3CCNCC3)nc2)=O)CC2(CC(C3CC3)=NO2)C1 c1(N(CC=C)C(=O)NCc2ccc(-c3cnc[nH]3)cc2)c(C)cccc1C C(C1=NOC2COCC12)NC(C1C(NC(C(C)N2CCCC2)=O)CC=CC1)=O c1(O)nccnc1N.c1(C(C(=O)OC2C(C(=O)OC)CCC2)O)ccccc1OC c1(CC)ccc(C(N2CCC2CNC(=O)CCc2cc(C)nn2C)=O)c(C)n1 C1(NC(C2(SC)CCC2)=O)COC2(CCCN(C(c3cc(F)ccc3C)=O)C2)C1 N(C(=NCCCN1CCCCC1)NCc1ccccc1)Cc1cnn(CC)n1 N1(C(c2scc(CNC(Cc3cnc(C)s3)=O)c2)=O)CC(CO)OCC1C C1(CNC(C2CCC(F)(F)CC2)=O)CC2(CCC2)CN1C(c1cccc(Cl)n1)=O CC1=CCN(C(=O)C(Cc2ccco2)NC(=O)C(C)N2CCC2)C1 n1(CC(=O)N(c2cccc(C(C)=O)c2)C)c2ccccc2c(=O)c2ccccc12 C1(CC)CCN(C(=O)C=C(C)C2CC2)C(C(N2CCC2CC(C)(C)C)=O)C1 N1(C(C(C)Cc2ccccc2Br)=O)CC2CN(C(c3ccc(O)nc3)=O)CC12 CC1(C)CCC(CNC(C23CCCN2CCC3)=O)N(C(=O)CC2CSCCS2)C1 C1(C(N2CCCC(CCOC)C2)=O)C2CC(CC2F)N1C(=O)C(C)S c1(OC)cc(N2CC(NC(c3cnc(F)c(C)c3)=O)C(O)C2)nc(OC)n1 CC1(C(N2CC(NC(c3nnn(C(C)(C)C)n3)=O)C(F)C2)=O)CCCCNC1=O C(=O)(CC(CNC(C1(CO)CCCC1)=O)C1CCC1)N(c1ccc(Cl)cn1)C N1(C(Cc2c(C)nn(C)c2Cl)=O)CCC2(COC(CNC(=O)C=CC(C)C)C2)C1 C1(NC(C2CS(=O)(=O)C2)=O)CC12CCN(C(c1ccc([N+](=O)[O-])s1)=O)CC2 C1(C(=O)NCCC(C(C)C)OC)CCC2(CC2)N1C(c1cc2n(n1)CCO2)=O C(CC(=O)NN1CCCC1C(=O)Nn1cccn1)C1(C)CCCC1CO CN1CCN(C(=O)CC=C(Cl)Cl)CC1C(=O)NC1(CO)CCOCC1 C(C(C(=O)NCC(O)(C1CC1)C1CC1)C(C)(C)C)NC(C(C(C)C)SC)=O C1(O)(CNC(c2ccc(C3CC3(F)F)cc2)=O)CCN(C(C2CCCC2)=O)CC1 c1(C(N2CCC(N(C(=O)CC3C=CCC3)CC#C)C2)=O)cc(N)ccc1O c1(OC)cccc2c1C(CNC(=O)NCC(C)(C)C(O)C(C)C)CC2 O=C(CCCC(F)(F)CO)NCCC1(C(=O)N(CC(F)F)C2CC2)CC1 c1(C(=O)NC(CNC(C2(C)C(C)C2)=O)C2CC2)ccc(NC(C)(C)C)cc1 CN1CC(NC(c2cn(CCNC(=O)C(=C3CCCCC3)F)cn2)=O)CCC1=O C=CC1(C(=O)NCc2ccoc2C(N2CCC23CN(C)C3)=O)CCOCC1 c1(CNCC2N(C(Cc3cccc(OC)c3)=O)CCOC2)cc(O)ccc1F Cc1nn2c(c1C(=O)NC(C1CCOC1)CNC(=O)CCCCC#N)CCCC2 c1(N2CCC(CCNC(C)=O)C2)nc(C(C)(C)C)ccc1C#N c1(OCC)cccc(Br)c1NC(=O)NC1CCCC1(F)F CCC(CNC(C1CCCCC1NC)=O)(CC)C(=O)Nc1cnn(C)c1 c1(CC(C)C)ccc(C(N2CC(NC(=O)CC3CCCCCC3)C2)=O)cc1 CC(C)CC(CNC(c1nncn1C(C)C)=O)NC(c1scnc1C(F)(F)F)=O c1(NCCOCC(=C)C)cc(Br)ccc1S(=O)(=O)NCC c1(C(N2C(C)CC(NC(C(C)(C)SC)=O)C2)=O)cc2ncccc2cc1Cl c1(C(C=C)NC(c2ccsc2OC)c2nnnn2CCSC)cccc(C)c1 C=C(C)CCC(=O)NCC1(OC)CN(C(c2cnc(C(C)(C)C)nc2)=O)C1 c1(C(=O)NCC2CC(CNC(C=C(COC)C)=O)OC2)cn(C(F)F)c(C)n1 Cc1cc(C(=O)NCCCOCCOCCNC(=O)C(C)(C)C(C)O)cnc1O C1(NC)CC12CC(C(C)NC(=O)NCCCC#CC)C2 C(CC(C)C)(C(N)=O)N(C(C1(NC(C(CCSC)O)=O)CSC1)=O)C C1(C(N(CC(CC)NC(=O)C(=Cc2cnn(C)c2)C)C)=O)CN(S(N)(=O)=O)C1 c1(CC)ccc(C(C)(C)C(=O)NCCC2(CNC(c3ccc(F)s3)=O)CC2)cc1 c1(C(=O)NCC2C(CNC(c3cc(C)nn3C3CCC3)=O)C2)cccc(O)c1Cl C1(NC(c2csc(C)c2C)=O)CC2(CCN(C(c3ncnc4ccsc34)=O)C2)C1 C(=O)(C1CCCc2ccccc21)NCC1CC(NC(C(CN(CC)CC)F)=O)C1 C1(CNC(C2C(OCC)C2C)=O)CCCN1C(c1c[nH]cc1CC)=O c1(C(=O)NC(CNC(CC2(OC)CC2)=O)(C)CO)ccc2c(c1)CCCC2=O n1(CC(=O)NC2CCCC(NC(C3(F)CC3)=O)CC2)cnc2sccc2c1=O C1(c2cn(C(C)C)nn2)(NCc2ncc(-c3ccc(F)nc3)[nH]2)CC(F)(F)C1 N1(C(c2cc(C(CC)CC)no2)=O)CC2CC(C1)C2NC(c1cnsc1)=O C1(C#N)(CNC(C(C)C(F)(F)F)=O)CCN(CC(=O)N2CCC2)CC1 C1(CNC(C=C(C)c2cccs2)=O)CN(C(=O)CC2COCCN2C)CC1(C)C C1(NC(C)C(=O)N(C)CCN(C)C(C2CCCCC2)=O)CCc2cncn2C1 C1(CCN=C(NCc2nnc(C)s2)NCC(C)(C)C)COc2ccccc2O1 C12(C(CNC(=O)C=Cc3nccs3)NC(C)=O)CCC(CC1)C2 c1(C(N(CCNC(CC2CC(CC)OCC2)=O)C)=O)cc(C#N)c2n1CCCC2 CCCCC(CNC(=O)Cn1ncn(C)c1=O)NC(c1scnc1C1CC1)=O C1(C(C)C(=O)NCC2(C(N)=O)CC2)CCN(C(c2cnn(CCF)c2)=O)C1 N1(C(CCC=CC)=O)CCC(CO)C(NC(=O)CCc2cccc(C)c2)C1 N1(C(C2CCCN(C(C3C(CCOC)C3)=O)C2)=O)CCCC(C(N)=O)CC1 C1(NC(=O)COC2CCCC2)(CNC(=O)C(F)(F)c2ccccc2)CCOC1 C=C(C)C(CC(=O)NCC(C)(C(C)C)NC(=O)Cc1ccc(Cl)cc1)OCC C(c1nc(C)c(C)[nH]1)=CC(N1CCC(OCCNC(C(CCOC)C)=O)C1)=O C(=O)(C(C)(O)C(C)C)NC1CN(C(C2CC(C(=O)OC)C2)=O)C(C)C1 CCC(CC)C(C)C(=O)NC(C)(C)CNC(c1c[nH]nc1-c1cccnc1)=O C1(C)(C(=O)NC(c2cn(C3CC(CSCCO)C3)nn2)C)COCCO1 C1(CN(C(Cc2cc(C)ns2)=O)C)CCCCN1C(=O)C(C)CC1CCCCC1 c1(NC(=O)CCc2ccc3c(c2)OCO3)cc(OC(F)(F)F)nc2ccccc12 Cn1ncc(C(=O)NC(CNC(c2ccc(F)c(Cl)c2N)=O)CO)c1S(C)(=O)=O c1(C(=O)NC2CN(C(c3cccc(CC)c3F)=O)C2)cc2sc(N(C)C)nc2s1 CCC(C#N)C(=O)NC(C)CCNC(c1coc(-c2cccnc2)n1)=O CC1CCN(C(=O)CC2CCN(C)C2=O)CC1NC(C1CC(NS(C)(=O)=O)C1)=O c1(C(N2CCC(CCNC(CC(C=C)(C)O)=O)CC2)=O)ccc2ncc(C)n2c1 C(=O)(C1=CC(C)(C)C1)NCC(CC)NC(c1cnoc1-c1ccccc1)=O C1(C(N(CC(C)(C)CNC(c2ccc(C(F)(F)F)s2)=O)CC)=O)NC(=O)OC1C C1(NC(C23C(C)OC(C)(C2)C3)=O)CCCC2CN(C(=O)CC3CCC(=O)N3)CC12 c1(NC(C2C(C(=O)OC)C2)=O)ccc(F)c(C(=O)Nc2ccc(Br)cc2O)c1 C(C(C)(CC)C(C)O)NC(CC1(NC(C=C(CCC)CCC)=O)CCCCC1)=O c1(C(=O)NCC2N(C(c3cc(C4(C)COC4)no3)=O)CCC2)cnc(F)c(F)c1 c1(C(=O)NC(C2OCCN(C(c3c(CC)ccs3)=O)C2)C)cc(F)cc(C)c1N C1(NC(C=CCN(CC)CC)=O)CCC(CNC(=O)C(C)(C)c2cnsc2)CC1 CC1CN(C(c2ccc(Cl)nc2O)=O)CCCN1C(=O)CCc1cc[nH]n1 c1(C(=O)NCCCN(C(C)C)C(c2ns[nH]c2=O)=O)cc2c(F)ccc(F)c2s1 N1(C(c2nccc(C)c2)=O)C(CNC(=O)Cc2cnc(C)[nH]2)CC2CCCC12 C1(CNC(CCC(C)(C)F)=O)CCN(C(c2cn(CCO)nn2)=O)CC1(F)F c1(C(=O)NC(CC=C)C(=O)NCC2(F)CC(CO)C2)cc(C)c(F)cn1 C1(C(=O)NCCn2c(C)nc(C)n2)CCN(C(=O)C(C)N=[N+]=[N-])O1 c1(C(=O)OCC)ncc(OC)cc1Cl.C12CC(F)CN(C1)C(=O)CC1(C)CN(C1)C2 C(=O)(C(C)C(F)(F)C(F)F)N1CC(SC)C(NC(=O)CC(C)CN(C)C)C1 CC(O)CCCCCC(=O)NC1CN(C(=O)CSCC(N)=O)CC1CC1CC1 C1(NCCc2ccc(C)cc2)CCCN(Cc2ccccc2)C1=O N1(C(c2cc(C)no2)=O)CCOCC1CNC(c1ccc(-c2ccco2)nc1)=O c1(CNc2cc(NC(C3CC4CCCN4C3)=O)ncn2)ccc(Br)c([N+](=O)[O-])c1 N1(C(C2(CC(=O)OC)CC2)=O)CCC(NC(=O)CC2CCCNC(=O)C2)C(O)C1 C(C(C)(F)C(C)(C)F)NC(C(C)(CO)NC(CC1CC(N(C)C)C1)=O)=O c1(CC(N2CC(OCCNC(CC3CCN(C)C3)=O)C2)=O)sc(O)nc1O c1(C(=O)NCC2CCC(NC(c3nc(C)n(C)c3)=O)C2)nccc2ccncc12 S(=O)(=O)(c1c[nH]ccc1=NC1Cc2cscc2C1)N(CC(C)(C)CO)C CCC(CC)C(=O)NCC(=O)NC(C)C(C)(C)NC(=O)Cc1ccoc1C c1(NC(C(C)Cc2ccc(Br)cc2)=O)cc2cccc(Br)c2n1C CC1CC(C(=O)NC2CN(C(c3cncc(C(F)F)c3)=O)C2)CCO1 c1(C(=O)OC(C(C)SC)C)cnn2ccc(OC)cc12 CC1(NC(C2CC(O)CCN2C(=O)CC2CCOCC2)=O)CCCC1(F)F CC(O)C(C)C(=O)N(C1CC1)CC1CCCN1C(c1ccccn1)=O C1(NC(c2c(CC)n[nH]c2)=O)C2CC1CN(C(=O)CNC(c1ccco1)=O)C2 C1(NC(C2(C(=O)NC)CC2)=O)CCC(O)CN(C(c2cccc(=S)n2O)=O)C1 Cc1ccc(C=CC(N2CC(NC(=O)CC3CCCCN3C)C3(CC3)C2)=O)cc1 c1(OCC)ccc(F)cc1NC(C1CC12CN(Cc1c[nH]ccc1=N)C2)=O n1(CC)nc(C(=O)NCCCCNC(=O)C(F)(F)c2ccc(Cl)s2)ccc1=O C=CCCC(CC(C)C)C(=O)NC1(NC(=O)CCCCC(CC)CC)CCC1 C(=O)(CCCCC#N)N(CCCN(C(=O)CCN1CCCCC1)C)C C(CCCCC(=O)NC1CCCC(NC(c2c(OC)nsc2OC)=O)C1)OC c1(OCC)cc(C(N2CCC(NC(=O)C(C(C)C)OC)C2)=O)cc(Cl)c1OCC N1(C(C2(C#N)CCC2)=O)CCC2(CO)CN(C(=O)Cc3ccccc3F)CC2C1 C=C(Cl)CC(C(=O)NCCC#CCO)NC(=O)CN1CC2CC2C1 CC(C)CC(C)C(=O)NCC(C(C)(C)C)NC(C1CCCCN1C)=O C1(NC(c2n(CC)ncc2Cl)=O)CC2CC(C1)N(C(=O)C(F)C(C)(C)O)C2 N1(C(C=COC(=O)CCC(C)CC)=O)CC(OCC)CC2(CCOCC2)C1 C1(N(C(c2cnc(C3CCOC3)s2)=O)CC)CCN(C(c2cncnc2)=O)C1 N1(C(C(CC)(C)C)=O)CC(C2CC2C(N2CCC(N(C)CCO)CC2)=O)C1 C1(C2CC2)(CNC(C2CN3CCN2CC3)=O)CCN(C(=O)CCc2cc[nH]n2)C1 N1(C(c2nncn2C)C)CC(NC(c2ccoc2C2CC2)=O)CC2(CCOCC2)C1 n1(C(C)C)cncc1CN(C(=O)C(F)C1CCOC1)C C(=O)(C1CCCn2cncc21)NC1(C2CCN(C(CCC(=C)Cl)=O)C2)CC1 N1(C(CC(CC2CC2)NC(C(COC)(C)C)=O)=O)CC(C(N)=O)C2(CC2)C1 C(N=c1[nH]c(C2CC2)nc(C)c1C)C1(OC)CCC(C)C1 c1(C(=O)NCCN(C(C2C(CC)OCCC2)=O)C)c(S(C)(=O)=O)cnn1C C1(C(=O)NCCCC=C)CCC2(CC2)N1C(C1CC(C(C)C)C1)=O c1(OCC(N2CCC(NC(C(C(C)C)N(C)C)=O)C2)=O)ccc(S(N)(=O)=O)cc1 C1(C2(NC(c3cc(C)no3)=O)CC2)CCCCN1C(=O)CCC1CCC(=O)NC1 N1(CC(=O)Nc2cccc(OC3CCCC3)c2)CC=CCC12CCOCC2 c1(C(c2n(CCC)nnn2)NCC2(C)CC2(C)C)cnc(OC)nc1 C12(NC(C(C)c3cccs3)=O)CCCC1N(C(C1CSCN1C)=O)CC2 Cc1ccnc(C(=O)NC(C2CCCC2)CNC(=O)CC2CC2(C)C)c1 C1(C(=O)NCC2N(C(CCS(C)(=O)=O)=O)CC2)CC12C1CC3CC(C1)CC2C3 Nc1cnc(C(=O)NCc2ccc(CNC(C3CC3c3ccoc3)=O)cc2)cn1 c1(C2C(C(=O)NC3CN(C(CC(=C=C)C)=O)CC3C)C2)ccc([N+](=O)[O-])cc1 C1(C(=O)NCC2C=CC(NC(C3CN(C)C(=O)N3)=O)C2)CC2(C1)CC2(F)F Cc1[nH]nc2ccc(C(=O)NC3CCCCN(C(=O)C4=NOCC4)C3)c(Cl)c12 C12(CNC(c3ccn(CCOC)n3)=O)CC1CN(C(=O)Cc1ccc(C)cn1)C2 C1(=CCNC(=O)CC2CC3CCC2O3)CCN(C(=O)Cc2cnccn2)CC1 C(=O)(CCCC(C)(C)NC(C1CC1(F)Cl)=O)N(CC(C)N(C(C)=O)C)C Cn1cc(CN2CC3CN(C(C4CCSCC4)=O)CC23)c2cc(Br)ccc12 c1(C(=O)NCC2CCCC(NC(CC=C)=O)C2)cccc2c1CCN2 c1(C(C)(C)C)ccc(N=c2nc(-c3ccccc3)nc(C(N)=O)[nH]2)c(Cl)c1 C1(CNC(CCSCCC)=O)CN(C(=O)C(=Cc2cccnc2)C)CC(C)(C)O1 C1(N(C(c2cnc(SC)s2)=O)CC)CCCN(C(=O)Cc2cccc(C)c2)CC1 c1(NC(C2N(C(c3cc(C)sc3C)=O)CC(=O)NC2)=O)ccc(C#N)cc1O N1(C(C(CC)OC)=O)CCOCC(C)(CNC(=O)C=CC2CCCC2)C1 C1(OCCC)CCN(C(C2CCCN2C)=O)CC1 c1(C(=O)NC2C(N(C)C(c3ccoc3)=O)CCCC2)ccc(F)c2c1CCC2 c1(CC)nnc(C)cc1C(=O)NC(CNC(C1(F)CCS(=O)(=O)C1)=O)C1CCC1 C1(NC(C(=CC2CCCC2)C)=O)COC2(CCN(C(C3(C)CCSCC3)=O)C2)C1 C1(NC(c2cnnn2C2CC2)=O)C2CC3C(C2)C13C(=O)NCCc1ncc[nH]1 C12(CC)CN(C(=O)NC3C(C)OC(C)C3C)C(CO)(C1)C2 C1(NC(CN(C(=O)C(CC(C)C)OC)CC)=O)CC(C)(OC)C1(C)C C(=O)(CCCC(=O)NOC(C)(C)C)N(CCNC(C(CC)C(C)(C)CC)=O)CC c1(-c2scc(C(=O)NC(C)CN(C)C(C34CCC3C4)=O)n2)ncccc1Cl Nc1cnc(C(N2CCCC2C=CC(=O)NCCC2CCCOC2)=O)cn1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(c2cc(C)c(N)cn2)=O)C2COCC12 CC1CN(C(c2ccc(CNC(c3ccc(C(F)F)o3)=O)cn2)=O)C(C)C1C c1(C(N2C(C)CC(NC(=O)Cc3cnn(C)c3)CC2)=O)csc2c(O)ccnc12 C1(CC)CC(C)N(C(=O)CNC(=O)CNC(=O)C(O)Cn2cncn2)C1 N1(C(c2ccc(SC)cc2)=O)CC(NC(=O)CNC(C)=O)CC(F)C1 Cc1nc(NC(C2CCCN(C(c3cccc(O)c3)=O)CC2)=O)cnc1Cl c1(C(=O)NC2C(CC(N3CC(C#CC)C3)=O)C(O)C2)ccn(C)c(=O)c1 N1(C(C2CCN(C(C)=O)C2)=O)CC2(CCN(C(=O)CC3CCCC34CC4)C2)C1 c1(OC)ccc(NNC(=O)Nc2nc3c(F)cc(F)cc3s2)nc1.C1C(=O)NNC1=O N1(C(c2n(C(C)C)cnc2)=O)CCC(CCN(C(=O)CCC2CC2)C)CC1 C1(CNC(C2(C#C)CC2)=O)C(C)CCCN1C(=O)CC1(O)CCCCC1 N1(C(C(CCC(C)C)F)=O)CC(C2CCN(C(C3CC4(CCO3)CC4)=O)CC2)C1 c1(OCC(=O)N(CC(C)N(C)C(c2cc(=O)cc[nH]2)=O)C)ccccc1O C(=O)(CCCCCO)NCC(C)N(C(=O)C(O)CCc1ccccc1)C c1(C(=O)NC(CNC(c2c(C)csc2)=O)C(C)(C)C)cc2n(n1)CCNC2=O C1(CCN(C)C(c2cc(Cl)n[nH]2)=O)CCN(C(C2CCCO2)=O)CC1 c1(C(N(CCCCNC(C2CC2(C)C)=O)C)=O)cc2c(F)ccc(Br)c2[nH]1 C(=O)(CC(CC)CCCC)N1CCC(NC(C=C)=O)C(CO)CC1 C12(C(N(CCC(C)NC(C3CCOC3C)=O)C)=O)CCN(CC1)S(=O)(=O)C2 N1(C(Cc2cc(=N)[nH]cc2)=O)CCC2C(C1)CN2C(c1c[nH]cc(Br)c1=O)=O N1(C(c2cc(OCC)ncc2)=O)CCC(NC(c2nnccc2C)=O)C(CO)C1 c1(NC(=O)CCC2CC(C(F)F)C2)nnc(C2CC2)s1 N1(C(C(CC)(CNC(C2CC2Cl)=O)CC)=O)CCOCC2(CCC2)C1 C(c1nc(C)cs1)=CC(=O)N(C1CCN(C(C2OCCC2C(C)C)=O)C1)CCC Cc1ccc(C(=O)NC(C)C(C)(C)C(=O)NCc2cn(C3CC3)cn2)c(F)c1 N1(C(C2(C)CC2)=O)CCC(Nc2ccc(C)cc2)C(F)C1.C1(C(=O)N)CC1(Cl)Cl c1(-c2nc(-c3ccc(Cl)cn3)n[nH]2)cc(F)ccc1Cl.FC(F)(F)OCCC1CC1 C1(C(=O)NC(CCCC)C)CC2(CC(NC(C3CCC3)=O)C2)C1 C1(NC(C(C(=O)OCC)=O)c2ccccc2)CC2CCCCN2C1=O c1(NC)cncc(C(=O)NCC2CN(C(=O)CCc3nc(C)no3)CC2C)c1 c1(SC)ccc(C(=O)NCC(C2CC2)NC(c2ccc(C(F)(F)F)nn2)=O)cc1 CCCCC(CNOCC(F)F)CC c1(CCC)ccccc1C(=O)NC(C)CNC(=O)COc1ccccc1C N1(C(C(C)NC(CC)=O)=O)CC2CN(C(c3cc(CC)c(=O)n(C)c3)=O)CCC12 c1(C(N(CCC)CCNC(=O)C=CS(C)=O)=O)cccc(O)c1C CC1CNC(=O)CN1C(C1CCCCN1C(C1COCCO1)=O)=O c1(C(N(CCNC(c2nc(C)oc2OC)=O)CC)=O)[nH]nc2c(=O)n(C)cnc12 C1(CCC(=O)NC2(COC)COC2)CCC(NC(=O)C(F)=CC2CC2)C1 C1(NC(=O)C(O)Cc2ccc(F)cc2)CCC2CC1CN2c1ccncn1 C(=O)(C(C)S(N)(=O)=O)N1CC(CCNC(C2N(C(=O)OCC)CSC2)=O)C1 C1(C(=O)NC(CNC(c2c(C)ncn2O)=O)C)C2CCC1(C)C2(C)C Cc1cnc(C(=O)NCC2COCCN2C(c2cc(C)c(Br)s2)=O)cn1 CC1=C(C(=O)N2CCCC2CCNC(c2ccc(C)s2)=O)CCO1 CCC(C)(C)CC(C(=O)NCCOC)N1CCS(=O)(=O)C(C)C1c1ccccc1 c1(COC)cc(C(N2CCC(C)C2CNC(c2cc(CO)c(C)o2)=O)=O)c(C)o1 O=C(CC1=CCN(C(=O)Cn2cccc2)CC1)NC1CCC2(CCC2)C1 C#Cc1cccc(CC(=O)N(CCC(C)NC(=O)CC2CC(F)C2)C)c1 Cc1n[nH]c(C)c1CC(C)C(=O)NCC1CC1NC(=O)C=C(Cl)Cl Cc1cc(C)c(C(=O)NC(Cn2cc(C3CCN(C)CC3)nn2)C(C)(C)C)c(O)n1 c1(C(N2CC(CN(C(CCSCC)=O)C)OCC2)=O)ccc2n[nH]c(C)c2c1Cl C=CCCN=C(NCCc1ncn(C)n1)N1CCC(CCC)C1 Cc1nscc1CNC(=O)C(Cc1ccco1)NC(C1CC(=C2CC2)C1)=O c1(C(=O)NC2C(OC)CN(C(=O)CCn3ccnn3)C2)cc(C)c(C#N)cn1 c1(C(=O)NC(C)(C)CNC(C2CC2(C)Br)=O)ccc(O)nc1 N#Cc1ncc(C(=O)NC2CCC2NC(c2cc(-n3cccn3)ccn2)=O)s1 Cc1cc(C)c(C(N2CC(O)CC2CNC(c2nn(C)cc2Cl)=O)=O)cn1 N1(C(C=Cc2cc(N(C3CCCCC3Cl)C)ns2)=O)CCC(CN=[N+]=[N-])C(C)C1 N1(C(CC=C)=O)CC(OC)CC1CNC(c1sc(C)nc1-c1ccc(C)cc1)=O C=C(C)CCCC(=O)N1CCC(NC(=O)C(C)NC(=O)CC(C)(C)C)C(F)C1 c1(C(=O)OC)cccc(CN2CCSCC2C(=O)Nc2cncnc2Br)n1 c1(C2(Nc3nc(C(=O)OCC)n(C)c3)CCCC2)ccc(F)cc1F Cc1ccc(NC(c2occc2CNC(=O)C(C2CCCCC2)C)=O)cc1C C(C(C)(O)CCCO)N(C(c1ccc(CC)o1)=O)CC c1(C(N(CCNC(C(C(C)C)NC(=O)OC)=O)C)=O)ccc2c(c1)COC2(C)C C1(C(=O)NC(C#C)C)C2CN(C(=O)CCCn3ccnn3)CC12 CN1CC(NC(C2CN(C(=O)CCc3ccccc3)CCN2C)=O)CCC1=O C(=O)(CS(=O)(=O)CC(=O)N1CC(F)(CNC(=O)CCc2cn(C)nn2)C1)OC N1(C(C2C(C)(C)CCO2)=O)CCC2(CC1)CC(NC(C1(F)CCC1)=O)CO2 C1(NC(C=C(C)C(F)F)=O)CN(C(=O)CCCc2ccc(O)cc2)CC1C C1(NC(c2nsnc2O)=O)CCCC(NC(c2nn[nH]c2C(F)(F)F)=O)C1 C1(NC(C(F)=CC)=O)CCCCC1NC(=O)CSc1ccc(OC)cc1 C1(C)(CNC(C(F)(F)C2(OC)CCC2)=O)CCCN(C(=O)Cc2cncs2)C1 C(=O)(C(O)CCS(C)=O)N(C)CC1(O)CCN(C(Cc2ccc(C)cc2)=O)CC1 c1(C(=O)NC(C(C)C)CNC(=O)C=Cc2ccco2)ccc(S(N)(=O)=O)c(F)c1 C(CCO)(C(F)(F)F)NC(C1C(CC)CCN1C(=O)CC1(COC)CC1)=O N1(C(c2cnc(SC)s2)=O)CCOCC(F)(CNC(C2CCCOCC2)=O)C1 N1(S(CCC)(=O)=O)CCCC(C(=O)N(CCNC(=O)CN(C)CCO)C(C)C)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NC1CC(CNC(CCc2c(C)n(C)nc2)=O)C1 c1(C(=O)NC(CC)CNC(C2CCN(CCO)C(=O)C2)=O)cc(F)c(Cl)cc1Cl CCC(CCCC(=O)N1CCC1C1CCC1)NC(c1csc(C)n1)=O N1(C(C2(Br)C(C)(C)C2)=O)CCC2(CCCN(C(C3CC(C)(C)C3)=O)C2)C1 C1(CC)(NC(=O)CSCc2ccncc2)CCCN(C(C2(C#N)CC2(C)C)=O)C1 C1(C(=O)Nc2ccc(O)cc2)(NC(C2CC(OCC)C2)=O)CCCC1C N1(C(C(C)NC(C)=O)=O)CC2(CCOCC2)CC1CNC(c1c(C)ncn1O)=O N1(C(Cn2c(C)ccc2C)=O)CCC=C(C(=O)N2CCCC(CC(C)C)C2)C1 c1(OC)ccc(CC(C)(CO)NC(=O)C(c2cccc(Br)c2)(C)C)cc1Br CCCCS(=O)(=O)CC(=O)NCCN(C(c1csc(COC)c1)=O)CCC1CC1 C(=O)(C(C)C(O)C(C)C)NC12CC(NC(COc3c(C)ccc(C)c3)=O)(C1)C2 C=CC(C)(O)CC(=O)NC1CCCC(CNC(=O)C=Cc2cncs2)C1 C1(C)(C(=O)NC2CN(C(C(C)Cc3ccc(F)cc3)=O)C2)COCC1(F)F C1(C(=O)NC2CCCC2C(N)=O)(CC)CCN(C(=O)CC23CCCC2C3)CC1 N#CC1(CNC(=O)C(O)CCCNC(=O)C(C2CC2)C2CC2)CCCCC1 N1(C(C(CC)OC)=O)CC(NC(c2ccc(NC=O)cc2)=O)C2(CC2)C1 c1(CC(=O)NCC2(OC)CCC2)ccc(CNC(=O)C(C)Cc2cnc[nH]2)cc1 c1(C(C)NC(c2ccnn2C2CCCC2)=O)cc(F)cc(F)c1 C(=O)(C1CCCc2nc[nH]c21)N1CCCCC(CNC(=O)CC2COC(=O)C2)C1 c1(C(N(C2CCCC(NC(=O)CCCCC#N)C2)C)=O)ccc2nccn2n1 N1(C(c2ccc(C#N)[nH]2)=O)CCC2CC1CN(C(=O)Cc1cc(F)cc(F)c1)C2 C1(N(C(C)=O)CCSc2ccc(F)cc2)CCN(C(C(=O)NC)C2(C)CC2)CC1 c1(C(=O)NC2CC(NC(c3c(C)cn(C)c3)=O)C2)ccc2c(c1)CCC(C)N2 Cc1sc(O)nc1C(=O)N(CCCNC(C1CCC(=O)NC1)=O)C(C)C C1(NC(c2cn(C=C)nc2)c2nnnn2CC(=C)C)CCCCN(C)C1=O c1(C(N2C(CNC(CN(CCC)C)=O)CC(O)C2)=O)cc2c(s1)CCS(=O)(=O)C2 CCC(C(=O)NCCCCCCN(C(=O)CCCCOC(C)C)C)C(C)O c1(CC)n[nH]cc1C(=O)NCc1cn(C(C)C(=O)NCC2CNC(=O)O2)nn1 N#Cc1cn[nH]c1C(=O)NCCNC(c1ncsc1-c1ccccc1)=O c1(NC2CC(F)(CNC(C3CCCCC3)=O)C2)ncc2cccnc2n1 C#CCC(C)(CNC(=O)C(CNC(=O)C(C)CC1CCCC1)N(C)C)CO c1(CC(C2(C)CCOC2)NC(CC)(C)c2nn[nH]n2)ccc(F)cc1 c1(C2C(C(=O)NCCN(C(=O)CC3(C)CCCO3)CC)C2)ccc(Cl)cc1F c1(C(N2CCCC(CNC(C(C3CC3)OC)=O)CC2)=O)ccc2[nH]ccc2c1 N1(C(C2C(CC)CCO2)=O)CC(C(=O)Nc2cnc(C)nc2C)C(C)(C)C1 CC(C)(C)C(C#N)C(=O)N1CCOC(CNC(c2cc3cscc3s2)=O)C1 C1(C(=O)NCC2CCN(C(c3ccc(C)[nH]3)=O)C2)CCCN(C)C1 C1(NC(CC(C)C(F)F)=O)CN(C(C2CCS(=O)CC2)=O)C2(CCCC2)C1 c1(OC)cc(OC)[nH]c(=NCCC(C)NC(=O)CSCc2ccccn2)n1 C1(C(=O)NCc2c(C(=O)NC(CC#C)C(=O)NC)scc2)CC2(CCC2=O)C1 Cc1cnc(C)c(NC(C2CCN(C(=O)CSCC(N)=O)C23CC3)=O)c1 N(C1CC2(CN(C(=O)C(O)CSC)C2)n2ccnc21)C(C1(C=C)CCOCC1)=O S(=O)(=O)(c1ccc(Cl)nc1)NC1CCC(NCc2c(C)c(Cl)ncc2)C1 Cc1nnc(CN(CCF)C(c2coc(C3CCCCC3)n2)=O)s1 C1(CC)CC(C(=O)NCC2CN(C(c3ccc(Br)o3)=O)C2)CC(=O)N1 CC(CS(C)(=O)=O)C(=O)NC1CC1NC(c1ccc2nccn2c1)=O CCN=c1[nH]c(C)c(C(=O)NC2CCN(C(=O)CCc3nc[nH]n3)CC2(C)C)s1 C(=O)(C1=NOC(C)C1C)NCCC(=C)CNC(C1Cc2ccccc2O1)=O C12(NC(Cc3cc(C)[nH]n3)=O)CC1CN(C(C1CCS(=O)(=O)C1)=O)C2 Cc1cc(C(=O)N(CC(C)NC(=O)CC(C)(C)C2CC2)C)c(F)c(Br)c1 N1(C(CC(=C=C)C)=O)CCC(NC(c2cccc(P(C)(C)=O)c2)=O)C2(CCC2)C1 c1(C(=O)NC2CC3(CN(C(C(CC=C)CC)=O)C3)C2)cc2cc(Cl)cc(C)c2[nH]1 C1(CNC(C(CC#C)O)=O)CN(C(=O)Cc2c(C)noc2C)CCC12CCC2 C12CCCCN1C(=O)CCC1CCN(C1)C(=O)C2.c1(COC)ccon1 Cc1ncc(C=CC(=O)NC2CC2CNC(c2cnc(N(C)C)o2)=O)s1 C12(CNC(=O)CC(O)C3CC3)CCC(C1)N(C(c1cncs1)=O)C2 c1(C(=O)NC(C(C)(C)NC(C(C)=C2CC2)=O)C)ccc(N)c(OCCO)c1 C12(C(=O)NC(CCNC(C(C)=C(CC)C)=O)C)CCCC(CO1)C2 CC(C)CC(C(=O)N(C)CC1CCCN1C(c1cc(C(F)F)on1)=O)C(N)=O O(N1CCC(NC(=O)CCN(C(c2ccc(C)cc2)=O)C2CC2)CC1)CC c1(C(N2CCCC(F)(CNC(C3CC4CCC3O4)=O)C2)=O)cc(F)c(Cl)cc1Cl Cc1cc(Br)c([N+](=O)[O-])cc1C(N1CC(NC(c2[nH]ccc2C)=O)C(F)C1)=O c1(CC)nccc(=NCC2(O)CN(C(C3CC34CCSCC4)=O)C2)[nH]1 Cc1cc(C(N2CCC(CC(C)NC(=O)C3=CCCSC3)CC2)=O)cc(C)c1O c1(C(=O)NCCC(=O)NC(CN(C(CC(C)C)=O)CC)C)cc(C(C)(C)C)c[nH]1 c1(C(N(C2CC(NC(c3cc(C)ncc3)=O)C2)C)=O)ccc(F)cc1Cl CC1(C)CC(CCNC(C2CCOC2CNC(C2(C)CCC(=O)C2)=O)=O)CO1 C(CCC(=O)NC1(C(N)=O)CC(O)C1)N(C(C(C)=C(CC)C)=O)C c1(OC)ccc(Br)c(C(=O)NC2CCC(NCc3cnc(C(C)(C)C)nc3)C2)c1 c1(C(N2CCC(NC(C3CCN(C(C)=O)C3)=O)C23CC3)=O)ccnc2[nH]nnc12 C#Cc1ccc(F)cc1C(N1CCOC(CNC(c2cnc(F)c(F)c2)=O)C1)=O N1(C(C2ON=C(C(C)C)C2)=O)CC2CCN(C(c3cnc(Cl)s3)=O)C2C1 C(=O)(C(C)(C)CCCO)NC(C)CN(C(c1c(C)nc(C2CC2)o1)=O)C C1(CNC(CC(C(C)C)O)=O)CC2CCC(C1)N2C(C1CC(C)(C)C1)=O c1(C(NS(=O)(=O)N(C)C2CCS(=O)(=O)C2)C)cc(Br)c2c(c1)CCO2 c1(CN(C(C(=O)NC2CCN(C(CC)C)CC2)=O)C)cc(OC)c(OC)cc1C C1(CC(NOCC(=O)NC(C2OCCOC2C)C)=O)CC(O)C1(C)C Cc1[nH]c(=N)ccc1S(=O)(=O)NOCc1ccc(C#N)cc1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC2(CNC(=O)CCC=C(C)C)C1 c1(C2C(C(=O)NC3(C)CN(C(CNC(CC)=O)=O)C3)CCO2)cccc(F)c1 C1(C(=O)NC(C(C)NC(=O)CC2OCCCO2)C)C2CCC1(c1ccco1)C2 N1(C(CNC(C(CC)C)=O)=O)C(CC(=O)N(CCN=[N+]=[N-])C)C2CCCC12 C1(NC(C(C)N(C(C)=O)C)=O)(CNC(c2ocnc2C)=O)CCOC1 C#CCCC(C(=O)NCC1CC12CCC2)NC(=O)C(CC)NC(N)=O N1(C(c2ccsc2Cl)=O)CCC2CCN(C(C3CCn4ccnc4C3)=O)CC2C1 c1(C(=O)NCC(CC=C)NC(=O)C(C(C)(C)C)SC)ccc(OC)c2cn[nH]c12 c1(CCC(=O)NCCC(C)NC(=O)C2=CCSC2)ccccc1N c1(C(=O)NCCNC(c2n(CC)ccn2)=O)ccc2c(c1)SCCN2 CC1CC1C1CC1C(=O)CC(=O)C(=O)NCC(C)(C)C1CCC1.c1(S)cnn(C)c1 c1(C(N2CCCC(NC(C3CCCC(=O)C3)=O)CC2)=O)ccc2nc(Cl)nn2c1 C1(C(=O)NCCN(CC(C)O)C(c2ccncc2)=O)CCc2nc(=N)[nH]cc2C1 C=CCC(C)(C)CC(=O)NC(C1CCN(C(=O)C(C)Cc2cnco2)C1)(C)C C1(C(=O)OC)CCN(C(C2CCOC(C)C2)C(=O)NCCC2CC2)CC1C C12(C(=O)Nc3cc(Br)cnc3OC(F)F)CCCCC1CS(=O)(=O)C2 N1(CC(=O)NCC2(F)CN(C(=O)C(O)CF)C2)CCCCCC1 C(c1cccc(F)c1Cl)=CC(=O)NC1(C)CN(C(CC(CC)(C)C)=O)C1 N1(C(c2ccc(CC)c(CC)c2)=O)CC2CC(C(=O)OC)(C1)C2O C1(NC(C(F)=CCC)=O)CCCCC12CCCN(C(c1cnc(N)c(N)c1)=O)C2 CC(C)CC(O)CC(=O)NC(C1CCCN(C(=O)C=Cc2nccs2)C1)C N1(C(C(=O)NC2CC(=O)NC2)=O)CCC(c2ccccc2)(C(F)(F)F)CC1 C1(C(=O)NCCC2N(C(CN(C)S(N)(=O)=O)=O)CCOC2)CCCCC12CCC2 C12(NC(=O)NC3CC34CCOCC4)CC(CO)(C1)OC21CCNCC1 C1(C(=O)NCc2cccnn2)CCCCCCN1C(C1CC2C(C1)C2(F)F)=O N1(C(C2(c3ccc(C)nc3)CC2)=O)CC(N(C)C(c2n[nH]cc2C)=O)C2(CC2)C1 CCC(CC)(CO)C(=O)NC(C)C(CO)NC(c1c(OC)ccnc1F)=O CC(C)CC(C(=O)NC(C)CCN(C)C(c1ccc(C#N)cc1)=O)C(C)C C1(C)(NC(C(Cc2cn[nH]c2)NC(CCSCCCC)=O)=O)CCOC1=O C1(C(=O)OC(C)(C)C)CCC2(CC2)CN1C(=O)N(c1ccc(Cl)c(F)c1)CCO c1(C(=O)NCCOCCN(C(c2cc(CC)on2)=O)C)cnn(C)c1Br CCC(CC)(CCNC(c1cnn(C(C)C)c1)=O)NC(=O)CC1COC(C)(C)C1 CCC(C)(CNC(C1CC2(C1)CC21CC1)=O)C(=O)NC1CCN(C(N)=O)C1 c1(C(=O)OC)cc(OC(c2ccccc2)C2COC2)cc(C(=O)OC)c1 N1(N(C(CN(CCOCCNC(CNCCC=C)=O)C)=O)C)CCCC1.CC#N CCCC(C(=O)OC)C(=O)NN=c1[nH]ccnc1OC c1(C(=O)NCCC(=O)NCC(n2ccnn2)C)nc(=N)cc[nH]1 C1(F)(C(=O)NCCCNC(CSC(C)(C)C)=O)C2CCCCC12 C1(CNC(c2nc(COC)sc2)=O)CC(C(F)(F)F)CN1C(c1cn(C)nn1)=O c1(C(N2CCCC2c2ccccc2)C(=O)NCC)ccoc1C c1(C(=O)NCCCCCNC(C(CC)C(=O)OC)=O)cc2cccnc2nc1C C1(NC(C2(CC(C)C)CCCC2)=O)CCN(C(C23CC(C)(C2)C3)=O)CC1(C)C CC1=CCN(C(C2CC(N(C(=O)Cc3cc(C)nn3C)C)C2)=O)CC1 c1(OC)cncnc1N1CCSCC1C(=O)NC(c1cccc(F)c1)C C#CCC(C)(C)C(=O)N(C)CC1(CNC(c2cccc(C)c2N)=O)CC1 C1(NC(c2c(CC)nns2)=O)C2CC3C(C2)C13C(=O)N(C)CC1COCCO1 Cc1cnnc(O)c1C(N1CCCC(N(C(=O)C(N2CCN(C)CC2)C)C)C1)=O N1(C(CC(C)c2ccco2)=O)CCCC1(C)C(=O)NCCN(CC(F)(F)F)C1CC1 c1(CNc2nc(-c3c(F)ncc(OCC)c3)sc2)ccc(C)c(C#N)c1 CC1CCC(NC(c2cc(-c3ccccc3)nn2-c2ccc(F)cc2)=O)CC1 c1(C(=O)NC2CCC(N(C(=O)C(=O)NCC3CC3)C)C2)n[nH]c2c1COCC2 N1(C(CC(=O)NCC#C)=O)C2CCC1C(F)C(NC(=O)Cn1ccnn1)C2 C(C1CCCCCC1)=CC(N1CC(NC(C2CC(OC)(OC)C2)=O)C(C)C1)=O c1(CC)cc(C(=O)NC2CCC(NC(C3(O)CCOC3)=O)C2)ccc1Br Cc1cc(C(N2CCCCC(CNC(=O)C(C)NC(N)=O)C2)=O)c(O)c(C)c1 N1(C(C2CCN(C(COCC(=O)OC)=O)C2)=O)CCCCC1CC(N)=O N1(C(CCCCCOC)=O)CCC(NC(c2cnc(C(C)C)s2)=O)C12CCC2 CCCCC(O)CNC(c1c(CNC(C2CC2OC(C)(C)C)=O)nnn1C)=O C12(C(=O)NC(CCCC)(CC)c3nn[nH]n3)CCCN1S(=O)(=O)CC2 N1(NC(=O)NC2CC(C(=O)OC)(CO)C2)CCOC(c2cnn(C)c2)C1 Cc1ncccc1CCNC(C1C=CCN1C(=O)CCl)=O C1(C(N2C(C)CSCC2)=O)CN(c2nnnn2-c2cc(O)c(F)cn2)CC1(F)F N1(C(CCSCCCC)=O)CC2CC(C1)C2NC(c1cccc(OC)c1F)=O C1(C(C)C)(C(=O)NCCCc2cc(O)n[nH]2)CCCN1C(C1CCCCO1)=O Cc1ccnc(O)c1C(=O)NCCN(C(=O)Cc1cn[nH]c1)C N1(C(CC2(N(C)C)COC2)=O)CCN(C(C2(C)CC2(F)F)=O)CC12CC2 N1(C(CC2CC(C)C2)=O)CCCC(C)(NC(=O)CCOc2cccnc2)C1 C(C1c2ccsc2CCN1C(C1CCCC1(C)C)=O)NC(C1(SC)CC1)=O c1(CCC(=O)NC2CC2CNC(C2(CCF)CC2)=O)ccccc1F Cc1cc(Cl)ccc1C(=O)NC1CC(CNC(c2cncnc2C(C)C)=O)C1 CC(C)S(=O)(=O)CC(=O)NCC1CCCC1NC(c1c[nH]c(C#N)c1)=O c1(C(=O)NC(C)CN(C)C(C2CC3(CCOC3)C2)=O)cc2ccc(Cl)c(F)c2o1 CC1CN(C(=O)C(F)C2CCOC2)CC1n1cc(C(NS(N)(=O)=O)(C)C)nn1 N1(C(c2c(C)n[nH]c2C)=O)CCC2(CC1)CC(CNC(=O)C1=CCCC1C)C2 c1(NCc2ccc(OC)nc2)nc(N2CC3CC3(CO)C2)nc2c1cnn2C CCC(CC(=O)NCC(=O)N(C)O)N(C)C(C1CC1c1ccccc1)=O COn1cnc(C)c1C(=O)NCC(C)(C)OCCNC(c1cncn1C)=O C1(C(=O)NC(C)CNC(=O)CC23CC(C2)C3)CCOC2(CCCC2)C1 C1(NC(CC=CC)=O)CC(CN(C(C2CCOC2)CO)C(=O)CO)C2CC12 c1(OC)ccccc1NC(=O)C(=O)N(C(C)CS(C)(=O)=O)C1CC1 C=CCC(CC(=O)Nc1cccc(O)c1F)NC(=O)COCC(C)(C)O c1(Nc2cc(Cl)cc(Br)c2)cnc2c(Cl)ccnn12 c1(NC2CN(CCC)C(=O)C2)[nH]c(=NCC(C)(CC)NC(C)=O)nc2sccc12 C(C)(CCC(=O)NCC1CCCCN1C(c1cc(C2CC2)ncn1)=O)OC N1(C(CNC(C)=O)=O)CCCC2(CNC(=O)Cc3ccnc(O)c3)CCCCC12 C1(OC)CCC2(C(N3CC(CNC(=O)Cc4ccnc(OC)c4)C(C)C3)=O)CC12 N1(C(C(CC)(F)F)=O)CC2CCCCC2(CNC(=O)CCCOC(C)C)C1 N1(C(c2c(SC)cccn2)=O)CC2ON=C(CNC(C3(C4CC4)CC3)=O)C2C1 N1(C(C2CCC(NCc3c(C)csc3)CC2)=O)CCC2(CCOC2)C1 Cc1c(CC(=O)NCC(O)CN(C)C(C2(C(F)(F)F)CC=CC2)=O)cnn1C C1(CNC(CCCCC#C)=O)CC12CCN(C(=O)C=Cc1ccc(C)s1)CC2 c1(C(N2C(C)CC(NC(=O)CCC(C)CN(C)C)C2)=O)c(O)nnc2c1CCC2 C1(C2CCOCC2)(NC(CN(C(=O)C#CC(C)(C)C)C)=O)CC1 N1(C(CNS(C)(=O)=O)=O)CC=C(CNC(C2CCCCC2F)=O)CC1 CCC(C)C(C(=O)N1CC(CO)(NC(c2sc(OC)nc2C)=O)C1)NS(C)(=O)=O c1(C(=O)NC(C(N2CC(CC)(OC)C2)=O)Cc2cn[nH]c2)ccc(C2CC2)cc1 C#CC1CN(N2CCCC(Oc3ccccc3C)C2)C1 Cc1nc(N)cnc1C(=O)NC1(C)CCC(NC(=O)CC2CCCCC2)CC1 CC(O)CC(CCC(=O)NOCCOCC1CCCC1)c1ccccc1 N1(C(C2N(CC)CCOC2)=O)CCCC2(CCN(C(c3csnc3Cl)=O)C2)C1 C1(C(=O)NCC(CC)(C)CC)CCN(C(=O)CCN(C)C)O1 N1(C(=O)NCCCOC)CCOC2(CCN(C(c3cc(C)nc(C)c3)=O)C2)C1 c1(C(=O)NC2C(NC(=O)CC(C(F)F)N3CCOCC3)C2)ccc2occc2c1 N1(C(C)=O)CCOC(C(N2CCCC2C2(NC(C3CC(Cl)(Cl)C3)=O)CC2)=O)C1 C(=O)(C1=CC2CCCCC12)NC(CCNC(C12CC(CSC)(OC1)C2)=O)C c1(C(N2CC(CNC(CC(C)c3ccncc3)=O)C2)=O)[nH]nc2c1CCC2(C)C C1(C(N(CC(=O)NCCOC(=O)OCC)C)=O)(C(=O)O)CC2CC2C1 c1(CC(=O)NC2(c3cn(CC=C)nn3)CC(F)(F)C2)cc(C)c(Cl)c(F)c1 N1(C(c2c(C)nco2)=O)CCCC(C)C1CNC(=O)Cc1ccc(Br)nc1 c1(CC(=O)NCC(CC=C)N(C(=O)CC2(O)CCC2)CC)ccc(C)c(C)c1 N1(C(C2C(OC)CCC2)=O)CC(C(=O)NCC(O)CC(F)(F)F)CC(C)(C)C1 Cc1cc(F)c(N)cc1C(=O)NC(C)CCCNC(c1occ2c1CCOC2)=O N1(C(CCC(CC)C)=O)C2CCC1CC(C(=O)NC1CCN3CCC1C3)C2 N1(C(C(C)c2cccs2)=O)CC2(CCC(CNC(=O)C(Cl)(Cl)Cl)O2)C1 C1(CCCC)CCC(C(=O)NC2CCCC2CNC(=O)C(C)(F)F)CC1 C1(O)(CNC(=O)C=Cc2cncs2)CCN(C(C23CCCC2C3(F)F)=O)CC1 C1(N(C)C(=O)NCc2ccc(Br)cc2F)CC2CCC(C1)N2C c1(C(=O)OCCCOC2(CC#C)CCC2)nn(C(C)(C)C)cc1[N+](=O)[O-] c1(CC)conc1C(=O)N(CC(CC)NC(=O)CN(C)C(N)=O)C C1(NC(=O)CC2(NC(=O)NCCCl)CCCC2)CCCC2(C1)N=N2 c1(C(=O)NCC2C(CNC(c3cnc(OC)s3)=O)C2)cn(C)nc1Br c1(C(=O)NCCCN(C2CCCC2)C)ccc(C(N)=O)cn1.C1(C)(C=O)CCCO1 c1(CC(N2CCC(C(CNC(C(C)C#N)=O)C3CC3)CC2)=O)cccc(F)c1F N1(C(Cc2ccc(OC)cn2)=O)CC(N(C(=O)CC2CCOC2=O)C)C(C)(C)C1 N1(S(c2n(C)ccn2)(=O)=O)CCc2sccc2C1c1cccs1 N1(C(c2cccnc2F)=O)CC2CCC(C1)C2NCc1ccc(Cl)c(F)c1 C1(N=[N+]=[N-])(C(N2CCC(=CCC)C2)=O)CCN(C(=O)C2=NOCC2)C1 c1(OC)ccnc(C(=O)NCC(n2cc(C(C)(C)CC3CC3)nn2)C)c1C CS(=O)(=O)c1coc(C(=O)NC2CCCC2NC(C2CCC(N=[N+]=[N-])CC2)=O)c1 CCC(CC)CC(F)C(=O)NCCSCC(N1CCC1C(=O)NC)=O C(=O)(CC(C(F)(F)F)NC(C1CC2C=CC1O2)=O)N(C)CCc1cc[nH]n1 C1(CC(=O)NCC(CO)NC(C(C)=C2CC2)=O)CCN(C)C1=O S(=O)(=O)(CCC(=O)N1CCCC1C(C)(C)NC(=O)Cc1ccn(C(C)C)n1)NC C#CC1(C(=O)NC2CCCC2CC(=O)N(CC(C)CO)C)CC(=O)C1 c1(C(C)C)cccc(NC(=O)Cn2cc(-c3nccn3C(F)F)nn2)c1 C(=O)(C(C(C)C)C(C)C)NC(c1cnn(C)c1)C(=O)NC(c1c(C)ncs1)C CCCC(C)C(=O)N1CCCCC1CN(C)Cc1ccsc1 C1(C(=O)NCC(CN(C(CCC(=O)OCC)=O)C)C)CC2(C1)NC(=O)NC2=O C(=O)(C1=CCc2ccccc21)N1CCC(C(C)(C)NC(C(CCCC)F)=O)C1 O=C(CCN1C(=O)CSc2ccccc21)NC1CC(C(F)(F)F)NC1=O c1(OC)cc(C(N2CCC(O)(CNC(c3ccc[n+]([O-])c3)=O)C2)=O)cc(O)c1O C(=O)(CCCS(N)(=O)=O)N1C(C2(NC(CCOCC(C)C)=O)CC2)CCC1 C1(CCOC)(NC(C2CC2C(=O)OC)=O)CCN(C(C2CC=CCC2)=O)C1 c1(C(COCC2(C(C)NC(=O)N(C)C)CC2)(C)C)ccc(Br)nc1 c1(C(N2CC3CN(Cc4nc(C)nn4C)CC3C2)=O)cccc2cccnc12 c1(CC(=O)NCC2(C)N(C(C3C(COC)CC3)=O)CCC2)ccc(O)c(F)c1 c1(C(=O)NC(c2cccnc2)C(=O)NC(CC(C)O)C)cnc(O)c(F)c1 C(CN=c1cc(C)c(S(=O)(=O)N(CC(C)C(F)(F)F)C)c[nH]1)c1ncc(C)nc1 N1(C(C(CC)C(C)O)=O)CCC(CNC(=O)CCc2cn(C)nn2)C(F)(F)CC1 c1(OC)ccc(Br)c(F)c1CN1C(C(=O)NC(C#N)C(N)=O)CCC1C C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC(NC(=O)CCC2CCOC2)C(F)C1 C(=O)(CC(O)CC(C)(C)C)NCCC1(C(N(C(C)C)CCN(C)C)=O)CC1 N1(CC(N2C(CCNC(Cn3c(C)cnc3)=O)CCC2)=O)CCC(O)CC1 CC1(C(=O)NC2CCCN(C(=O)CCc3cccc(O)n3)C2)CCCCO1 C1(CNC(=O)C(=O)N2CC(Cc3cccnc3)C2)CCCCC1O C1(C)(CNC(C(=O)N(C)C)=O)CCCN(C(c2ccc(N)c(O)c2)=O)C1 N1(C(CCc2ccc(C)s2)=O)C2CCCC1CN(C(c1ccnn1C)=O)CC2 c1(CC)nn(C)c(C(=O)NC2CCC(CCNC(=O)CC3OCCO3)C2)c1Cl S(=O)(=O)(c1cnc(NCCCCN(C)C)c(Cl)c1)NC(C)CC1CCOC1 CCC(C)(C)C(O)C(=O)N1CCC(C(C)C(=O)NCc2ccc(C)o2)CC1 c1(CC(=O)NCC(C)NC(c2ncccc2N)=O)ccc(F)cc1C(F)(F)F c1(OC)cccc(NC(=O)C(C2CN(C(=O)OC(C)(C)C)C2)NCCC(C)C)c1 C(=O)(C(C)(C)CS(N)(=O)=O)NC(CC(C)NC(C(C(C)C)C#N)=O)C C1(CC=C)(C(=O)NCC2COCCO2)CCN(C(=O)Cc2csc(CC)n2)C1 C1(COC)(CNC(C2CC2(C)C)=O)CCN(C(=O)CN2CC3CC3C2)CC1 C1(C(=O)NOCC2CCCCC2)(CC=C)CCCN1C(c1cnncc1C)=O CC(C)CCCCCCC(=O)NC1CN(C(=O)C(C)NS(C)(=O)=O)C(C)(C)C1 N1(C(C2(OCC)CCCC2)=O)CC2(CCC2NC(=O)C=CCO)C1 c1(N2CC=CC2)nc(=NCc2csc3ccccc23)[nH]c2c1SCC2 C1(CCCC)CN(C(=O)CNS(N)(=O)=O)CCN1C(=O)Cc1cc[nH]n1 C1(NC(C(C2CCCC2)OC)=O)CCCC1NC(=O)CC1CCC1 CC(CC(=O)NCC1CCN(C(C2(CCN(C)C3CC3)CCC2)=O)C1)P(C)(C)=O c1(CC)ccc2ncoc2c1.c12ccncc1OCCN(C)CCOCC(=O)N2C C1(C(=O)NCC2CC(NC(=O)CC(C)N3CCCC3=O)C2)(OC)CCOCC1 C(c1c(C)noc1C)=CC(=O)NCC1N(C(c2c(C)cc(C)o2)=O)CCC1 N1(C(C(Cc2cn(C)nc2)O)=O)CC(O)(C2CCN(C(=O)C(O)C(F)F)CC2)C1 c1(CC)sc(=N)[nH]c1C(=O)NCC(C)CNC(=O)CCc1nccs1 N1(C(CN(C(c2n(CC)c(C)nc2)=O)C)=O)CCCC(OC)C1C c1(C(=O)NC2C(CC)CN(C(=O)C=C3CCC3)CC2)cnc2c(c1)CCOC2 c1(-c2cccc(C)n2)ccc2cc(C(=O)NC3CCNC3=O)oc2c1 C(=O)(C(C)CCC(C)(C)C)NCC1(CNC(C(C)OC)=O)CCOCC1 CC#CCC(C(=O)N1CC(C2C=NNC2=O)C1)CCCc1sc(C)cc1C c1(C(=O)NC2CC(NC(C(CCOC)OC)=O)C2)cc2nc(=O)ccn2[nH]1 N1(C(c2c(CC)ccs2)=O)CC2(CCC(NC(=O)CCCn3ccnc3)CC2)C1 C1(CNC(C(CCSC)O)=O)CCC2(CN(C(=O)CN(c3ccccc3)C)C2)O1 c1(N2CCCC(C)(NC(C3C(C(=O)OC)C3)=O)C2)ncnc2c1oc1ccccc21 N1(C(C2C(C)(C)CN(C(C3C=CCS3)=O)C2)=O)Cc2cncnc2C1 c1(-c2nc(CC(CC)C)nn2CCc2ccccc2OC)cnn2c1CCCC2 C1(C)(CC)CC(C(=O)NCCN(C(=O)C=CC(C)(C)C)CC2CC2)C1 c1(OCC)nc(Br)cnc1NC(c1cc(-c2c(F)cccc2F)cnc1Cl)=O CC(C)C(Cc1ccccc1)C(=O)Nc1ccnn1-c1cccnc1 C12(C(=O)NCCC3N(C(c4sccc4F)=O)CCSC3)CCCC1C2(F)F c1(CC)cc(=NCCCCC(C)NC(C2CC3(CCOCC3)CO2)=O)[nH]cn1 C(=O)(CN=S(C)(C)=O)N(C)CC1N(C(c2cnn(C(CC)C)c2C)=O)CCC1 c1(C(=O)NC2C(NC(C3(C=C)CCC3)=O)C2)ccc(OC)cc1OCCC c1(CC)[nH]c(C(=O)N(C)CC2CCN(C(c3ccnc(O)c3)=O)C2)nc1Cl C1(NC(c2cccc(NC(C)=O)c2)=O)CC2CC1N(C(C1(CF)CC1)=O)C2 N1(C(c2c(CC)noc2)=O)CCC2CN(C(=O)CC3SC(=N)NC3=O)CC2C1 c1(-c2nnc(CC3(CC(COC)(C)C)CCC3)s2)ccc(Cl)cc1 c1(OC)ccc2[nH]c(=NCC3CCN(C(=O)CC4CC(O)C45CCC5)C3)sc2n1 CC1(C(=O)Nc2cnn[nH]2)CCCN(CCNCc2ccccc2C(F)(F)F)C1 CCC(F)(F)CC(=O)NCC1(C(=O)NC2CCC(COC)C2)CC12CCC2 CCC(C(N)=O)NC(=O)C=CCC1(NC(C2CC(=O)C2)=O)CCC1 Cc1[nH]nc(C(N2CCCC2CNC(C2(F)CCOCC2)=O)=O)c1N C1(NC(c2ccc(C(C)C)s2)=O)CCC2CN(c3ccncn3)CCC2C1 c1(-c2cc(O)c(F)cc2)n[nH]c(=NCCCF)s1 C1(C(C)NC(c2cc(C)ns2)=O)CN(C(=O)Cc2cnccc2C)CCO1 c1(NC(C(=O)NCC=Cc2cncc(OC)c2)=O)c(Cl)cc(Br)cc1Cl C1(N(C(CCc2onc(CCC)n2)=O)C)CN(C(=O)CC(C)(C)OC)CCC1C C1(NC(Cc2c(C)nc(S)s2)=O)CC2CCC1N2C(c1ccc(C(F)(F)F)o1)=O C1(C(=O)NCCCCOCC)CCC(=O)N1Cc1ccccc1 CCC1=NOC(CC(=O)NC2(CCNC(=O)C(c3ccccc3)C)CCCC2)C1 C1(C)(NC(C)=O)CCN(C(=O)CN(C(=O)CC2C(C)(C)C2(C)C)C2CC2)C1 CC1CC(CNC(=O)CCCC2CC2)CCN1C(C1CCC2(CCC2)C1)=O C1(C)(C(=O)NC2(c3cccc(C)c3)CC2)CCCN(CCc2ccccn2)C1 Cc1cc(C(=O)NC(CNC(c2cnc(C(C)C)s2)=O)C(C)C)no1 c1(N2CCC(N(C)C)(CC)C2)nc(=NCCC2=CCCCCC2)[nH]c2c1SCC2 S(=O)(=O)(c1cnc2c(Br)csc2c1)NCCS(N)(=O)=O N1(C(C(C)CC(F)F)=O)CC2CCC(N(C)C(C3CCC4(CC4)C3)=O)C2C1 c1(C(N2CCC(CCN(CCC(C)C)C)CC2)=O)cc2sccc2[nH]1 C(C(C)(CC(=O)NCC(C1CCC1)NC(=O)C(C)(C)O)C(F)(F)F)N(C)C n1(CC)nncc1CNC(=O)NC(C)C1CC1 C(CC(=O)N(C)CCN(C)C(C1CC2(C1)CC(O)C2)=O)(C(N)=O)NC(C)=O c1(CC(=O)NC2(CN(C(=O)CSCC3CCCCO3)C)CC2)ccc(Cl)s1 C12CCCC3CN(CC13)C2.N1(C(C2C(CC)C2)=O)CCCC1C(=O)Nc1cnsn1 c1(C(N2CC(OC)CC(NC(CSCC)=O)C2)=O)cc(F)c(F)cc1Cl C12(NC(c3cncs3)=O)CCCC1N(C(c1nnc3ccccn13)=O)CC2 c1(-c2scc(C)n2)nc(-c2cncc(-c3ccco3)c2)n(C2CCCC2(C)C)n1 Cc1ccccc1COC(C)C(=O)NC1CC(NC(c2cnnn2C)=O)C1 c1(C(=O)NCC(CNC(c2c(C)snn2)=O)C)c(C(F)(F)F)ncn1O c1(OC)cc(C(N2CC(Cn3ccnn3)C2)=O)c(F)c(F)c1F C(C(C)(C)CCNC(=O)CC12CCCC1C2)NC(CCCn1ncc(C)c1)=O c1(CONC(=O)NCC2CC2(Cl)Cl)cccc(Cl)c1 N1(C(C(=O)N(CC(=C)C)CC)C)CCC(C(=O)NCCC2CC(C)(C)CO2)CC1 C1(C(=O)NC(C)(CNC(=O)CCCc2ccsc2)C2CC2)CC12CCOCC2 c1(-c2ccc(C(=O)Nc3cc(OC)ncc3C)cc2F)ncnc2[nH]cc(C)c12 N1(C(CC)=O)CCCCC1C(=O)NC1CN(C(=O)C(N)=O)C1 C1(NC(c2c(C)nn(C)c2)=O)CN(c2cc(C(N)=O)nc(Cl)n2)C2CCCCC12 c1(C(=O)NC(CC=C)CNC(c2cc(-c3ccns3)on2)=O)cncc(C)n1 CS(=N)(=O)C1CN(C(C2(NC(C3CC4(CCC4O)C3)=O)CCSC2)=O)C1 c1(OC)ccc(C(c2nnnn2CC(F)F)NC2CC3CC3C2)cc1F N1(Cc2c(Br)cn(C)n2)CC2(CCN2C(c2ccc(C(=O)O)c(Br)c2)=O)C1 c1(OC)ccccc1Sc1ccc(C(N2CC(N(C(=O)C(C)SC)C)C2)=O)cc1 c1(CC(=O)NCCCCCCN(C(COC(C)C)=O)C)ccc(Cl)c(Cl)c1 N1(C(C(CN(C)C)O)=O)CCCC(N(C(=O)CCCNS(C)(=O)=O)C)C1 C(=O)(C(C)(O)C(F)(F)F)N1C(CNC(CC(C=C)(C)C)=O)CN(C)CC1 C1(C)(CC(=O)NC2C(CNC(CC(C)(C)O)=O)COC2)CCS(=O)(=O)N1 c1(SC)ccc2c(c1)CN(C(c1sc(CNC(=O)OC(C)(C)C)cc1C)=O)C2 CCCCCC(O)C(=O)NCC1CCN(C(c2sccc2Br)=O)C1 C1(C(N2C(CN(C(=O)Cc3cnc(C4CC4)[nH]3)C)CCC2)=O)CCCCNC1=O c1(C(=O)NCCCNC(C(=O)NCCNC(C)=O)=O)cn(C)c(=O)cc1C c1(C(C)(C)C(=O)NCC2CCN2C(=O)CC2(O)CCOC2)cccnc1F c1(C(N2CCC(N)C(C)(C)C2)C(=O)NC)ccc2c(c1)nnn2C C1(NC(c2ccc(N(C)C)c(F)c2)=O)CN(C(C2CCOC2)=O)C2(CCCC2)C1 C(C(=O)N(C1CN(C(C2CC2C(F)(F)F)=O)C1)CC)(C(C)C)OCC C(CO)(C(O)C1CCCC1)N(C(C(=O)O)C1CCCC1)CCO c1(C(N2CC(N(C)C(C34CCC(F)(CC3)C4)=O)C2)=O)cc2c(nc1O)CCSC2 C1(NC(c2c(C)c[nH]n2)=O)CC(O)CN(C(c2cc(Cl)cnc2O)=O)C1 N1(C(CCC2C(C)C2)=O)CCC(C)(CNC(=O)CCCc2ccsc2)CC1 N1(Cc2cnn(CCC)c2C)CCOCC(NC(c2ccnc(Br)c2)=O)C1 N1(C(c2c(C)cnnc2O)=O)CCN(C(=O)Cc2cscn2)CC(C)(F)C1 C1(N(C(CSCC#C)=O)C)CCCCC1NC(=O)CC1CC(=O)NC1=O C1(NC(C2CCN(C(c3cc(C)sc3)=O)C2C(C)C)=O)CC(C2CCCC2)C1 c1(C(=O)NCC2N(C(C3CCOC3)=O)CCN(C)C2)n[nH]c2c1CCSC2 Cc1ncnc(C)c1C(=O)NCC1(C)CCCN1C(C1C=CC=CC=C1)=O C1(C(N(CC(C)(C)NC(c2nn[nH]c2Cl)=O)C)=O)CCOC(C2CC2)C1 c1(C(=O)NCC(C)N(C(C(C)C2CCOC2)=O)C)ccc(C(F)(F)F)c(F)c1 C(c1cccs1)=C(C)C(=O)NCC1(NC(=O)COc2ccon2)CCOC1 N1(C(CC(CN(C)C)O)=O)CCC(CNC(=O)CCCCN(C)C)C12CCC2 CC(C)C(C(C)NC(c1ccncc1)=O)NC(=O)C=C1CCOCC1 C(=O)(CC(C)CN=c1[nH]c(N2CCC(OC(C)(C)C)C2)nc(=N)[nH]1)NC c1(C(C)NC(C2CC3(CC(NC(CCC)=O)C3)C2)=O)ccc(Cl)c(C)c1Cl C1(C=O)CCCC(O)C1.C1(C(=O)OC)CCCC1C(=O)NCC1CC(F)(CO)C1 C(=O)(C(Cn1cccn1)NC(C1(SC)CC(=O)C1)=O)N(CCCC)C c1(CCC)ccc(C(=O)NCC2CCN2C(=O)CSC(F)(F)F)cc1S(N)(=O)=O c1(C(=O)NCC(CNC(C2CC3CC3C2)=O)F)csc(C(c2ccccc2)=O)n1 Cc1c(C(=O)NC(C)Cn2cc(CC(O)C(C)C)nn2)cncc1Br c1(N2CCCC(NC(C(COC)(C)C)=O)C2C)nc2ccc(Br)cc2s1 Cc1cnc(C(=O)NCC2CCC(NC(C3(CF)CC3)=O)C2)cc1C#N c1(C(C)C)ccccc1CC(=O)NCC1CC1NC(c1c(Br)nnn1C)=O C1(C(=O)OC)CN(Cc2ccc(F)c(C)c2Cl)CCC12CCC2 c1(C(=O)OC)cc(OC)cc(Oc2ccccc2)c1.c12ccnc(c1F)NC2=O c1(C(N2CC(NC(C3C(F)(F)C34CC4)=O)C2)=O)ccc2c(c1)S(=O)(=O)NC=N2 c1(NC(C)C(C2CCCCC2)NC(C2CCOC2)=O)ncccc1[N+](=O)[O-] N1(C(C2C(CCOC)C2)=O)CCC2CC1CN2C(c1cccc(C(N)=O)n1)=O C1(NC(C(F)=CCC)=O)CC(O)CN(C(c2scc(C)c2OC)=O)C1 N1(C(C2CCC(C)O2)=O)CCC2(CCOCC2)C(NC(c2nn[nH]c2Cl)=O)C1 N1(C(c2n(CC=C)ccn2)=O)CCN(C(C2CCCOC2C)=O)C(C)C1 C=CC(C)(CC)C(=O)NCCCOCCC(=O)NCc1cc(O)ccc1F Cc1ccc2c(c1)CCC(C(=O)NCCCC(C)NC(=O)Cc1ncc(C)s1)O2 c1(OCC)cccc(F)c1CN1CCCC1C(=O)Nc1cccnc1C C1(C(=O)NCCCNC(c2c(C)oc(C(C)(C)C)c2)=O)CC2(CCOCC2)CO1 C(N=c1cc(NC2CC3CC3C2)nc(C(F)(F)F)[nH]1)c1c(C)nn(C)c1N(C)C c1(C(N(C)Cc2ccc(CNC(CC(C)F)=O)cc2)=O)c(F)ccc(F)c1N C1(NC(C2(C)C(C)C2)=O)CC(CNC(=O)C(F)(F)C=Cc2ccccc2)CC1O C12(C(=O)NC3CCCC(C#C)C3)CCC(CC1)N(C(C1CC(SC)C1)=O)C2 C1(C(=O)NCC2(O)CCCOC2)CCN(C(=O)C2CCC23CCC3)O1 c1(CCC)[nH]ccc1C(N1CC(F)(CNC(=O)C(c2ccccc2)C2CC2)C1)=O Cc1cc(=N)[nH]c(C)c1NC(=O)NC1CC(N(C)C(=O)C2CC2)C1 N1(C(C2(C)ON=C(C)C2)=O)CC2CC(NC(=O)CCN(C)CCO)CC2C1 c1(OC)ccnc(C(=O)NC2CC(F)(CNC(C3(C(C)C)CCC3)=O)C2)c1F CC1CC(=O)NC1CNC(C)(C)CNC1CNC(=O)N1.C1(=O)CN1 N1(C(=O)CC(F)(F)F)CC2(C1)CN(C(C1(O)CCOC1)=O)CC2CO c1(C(=O)NC2CCCC(NC(c3ccc(NC)cc3)=O)C2)c(C)ncnc1O CC1(C)CC(C(N2CCCCNC(=O)C2)=O)CCN1C(=O)C=Cc1nccs1 c1(C(=O)OC)cc(CC(N2CCC(COC(=O)Nn3cncn3)C2)=O)on1 S(=O)(=O)(c1ccc(C#N)c(C(F)(F)F)c1)NCCS(CCOC)(=O)=O C1(C(=O)NCCC2(OC)CN(C(C3(N(C)C)CC3)=O)C2)CCC2(CCC2)CO1 N1(Cc2cc(OC)cc(OC)c2)CC2(CCN(C(=O)C=CC(C)C)CC2)C1 c1(OCC(=O)Nc2cccc(OCCCC)c2F)c(F)cc(COC)cc1Cl C1(C(=O)NCC2(NC(C(c3cncn3C)N(C)C)=O)CCOC2)CC2CCC1CC2 N1(C(c2c(OC)nccc2C)=O)CCCC2CN(C(=O)Cn3cncn3)CC12 Cc1cc(NC(c2c(C(F)F)cccc2Cl)=O)cc(C)c1 C#Cc1cn(C)nc1C(=O)NC1CCCCCC1NC(=O)CCS(N)(=O)=O N1(C(c2c(C)scn2)=O)CC2(C1)CN(C(c1c(C)noc1C)=O)CCO2 N1(C(c2n(CC)cnn2)=O)CCC(CNC(C23CC(c4cccs4)(C2)C3)=O)CC1 c1(CCC(N2CC(F)(CNC(C(C)OCC(C)C)=O)C2)=O)cccc(O)c1 C1(C(N)=O)(CNC(C2CCC2C(N)=O)=O)CN(C(C2CCC(=O)N2)=O)C1 c1(C(N2CC3C(NC(C4CN(CCC)C(=O)C4)=O)C3C2)=O)cc(C)c(C)c(F)c1 N1(C(C2(CNC(C3C(C)CCC3)=O)CC=CC2)=O)CCC(C)(C)C1 C1(NC(CC(c2c(C)n[nH]c2C)C)=O)CN(C(c2csnn2)=O)CCC12CCC2 c1(N(C)C)cnc(C(c2nnnn2CCCF)Nc2cc(C3CC3)sn2)cn1 C(CN=c1[nH]c(=NCC2CCCC(C)O2)[nH]c2c1SCC2)OCCC=C CC(C(=O)N1CCOC(CNC(C2(c3nccs3)CC2)=O)C1)S(N)(=O)=O N1(C(Cc2n[nH]c(=N)s2)=O)CCC2(CCC2)C(NC(c2csc(S)n2)=O)C1 N1(C(CSC(C)C)=O)CC2(CCNC(=O)CCc3cccnc3F)CCC1C2 Cc1cc2cc(C(C)NC(c3nc(Cl)nc(C)c3CO)=O)oc2cc1C c1(C(=O)NCCCCCCNC(CC2(C)CCCCC2)=O)cccc(F)c1N C(c1c(F)cccc1F)=CC(=O)NCC(C(C)C)NC(c1coc2c1CSC2)=O c1(C(N(CC(CNC(C2(C)CCN(C)C2=O)=O)O)C)=O)cnc2sccn2c1=O c1(C(=O)NCCN(C(=O)CC(C)C2CCCC2)CC)ccc2c(n1)CCCC2 C1(NC(c2c(OC)n[nH]c2)=O)C(C)CN(C(c2[nH]c(O)nc2C)=O)CC1C c1(N2CCC(C)(NC(CCC3C(C)=NOC3=O)=O)C2)cc(C)c(C#N)c(C)n1 Cc1cc(N(C)C)ncc1S(=O)(=O)N1CCC(O)(NC2CCC3(CC3)C2)CC1 C=C1CCC(C(=O)NC(CCN(C)C(C2COCC2C(F)(F)F)=O)C(C)C)CC1 C1(C#N)(C(=O)NC(C2CCN(C(c3ccc(CC)[nH]3)=O)C2)(C)C)CC12CCC2 c1(N2CCC(C)C2CNC(=O)CC2(C)CC2(F)Cl)ncc2c(n1)COC2 CC(C)CCCCCC(=O)N1CCOC(CCCNC(=O)C=CC(=O)OC(C)C)C1 C1(C(N(CCCN=[N+]=[N-])CC)=O)CCN(C(=O)C2CCOCC2(C)C)O1 C(=O)(C(CNC(C1COCC1C(N)=O)=O)OC)NCC(CC1CC1)OC C1(c2cccs2)(C(N(CC(O)CNC(=O)Cc2cncn2C)C)=O)CCCCC1 C12(CC(=O)NCC(C)Cc3cn[nH]c3)CCC1CN(C(c1ncccc1F)=O)C2 C1(NC(c2coc(Cl)c2)=O)(CO)CCCN(C(C2(c3ccccc3)CC2)=O)C1 N1(C2CN(C(CC3(C)CC3(Cl)Cl)=O)C2)CCN(C(c2ncc[nH]c2=O)=O)CC1 CCC(CC)CC(C(=O)NCC)N1CCOCC1c1ccc(C)o1 N1(C(C=C(C)C(F)F)=O)CCCCC(NC(=O)CC2OCCCC2(C)C)C1 N1(C(CC2CCC(OC)CC2)=O)CCC2C1CCCN2C(=O)Cc1ccn(C)n1 c1(NC(CCNC(C2(C=C)CCC2)=O)=O)cnc2[nH]ncc2c1 N1(C(CCC(C)C)=O)CCC2CN(C(C3(C(F)F)CCOCC3)=O)CCC12 C1(F)(CNC(CCC(C)OCC)=O)CCC(CNC(=O)Cc2cnn(C)c2)CC1 c1(C(=O)NC(CCNC(CCC=CC)=O)(C)C)nc(S(N)(=O)=O)c2ccccn12 CC(C)(C)CCCCCC(=O)N1CCC(CNC(c2c(O)cccc2F)=O)C1 C1(c2cn(CCC3CN(C(c4cnn[nH]4)=O)C3)nn2)(C(=O)OC)CCCCC1 CN1CCCC(CC(N2CCOCC2CNC(C2(C)CCSCC2)=O)=O)C1 C=C=CCCC(=O)N(CCNC(C1CCCC1C)=O)CC Cc1ccc(=N)[nH]c1C(=O)NC1(CNC(=O)CC2CCCN2C(C)C)CC1 N1(CCC)CC(C(=O)NCCN(C(=O)CCN2CCOCC2=O)C)CC1=O Cc1cccc(C(=O)NCCCCCCN(C)C(c2ncn(C(C)C)n2)=O)c1N O=C1CC(C(N2CCCOC(CCNC(=O)C=CC=C(Cl)Cl)C2)=O)CC(=O)N1 c1(N2CCC(C(CC)C)CC2)ccc(Br)c(S(=O)(=O)NCC2(OC)CCC2)n1 c1(C(=O)NC(CCNC(Cn2cc(C)c(C(F)(F)F)n2)=O)C)ccnc(C)c1N c1(N2CCC(C(=O)NC3CCOCC3)C2)ccc(NCC2CCNC2)cc1 S(=O)(=O)(c1ccc(Br)cc1F)Nc1c(C(C)OC)cc(F)cc1 N1(C(CCCC#CC)=O)C2CCC1CC(N(C)C(C13CCC(OC)C1C3)=O)C2 CCC1CN(C(C)C(=O)Nc2ccc3nsnc3c2)Cc2ccccc21 N1(C(C(CNc2ccc(OC)cc2)O)=O)CC2(C1)CN(C)CCO2 N1(C(C=CC)=O)CCC2(CC1)CC2C(=O)NCCOC O=C1CC(C(=O)NC2CCN(C(=O)C(O)C3CCC3)CC2)Cc2ccccc21 CC(C)CC(C)(O)C(=O)N1CCN(C)C(C(N2CCC2c2ccccc2)=O)C1 N1(C(CC(C)OC)=O)CCC(C)(C)C(NC(c2ccc(C)cc2Cl)=O)C1 N1(C(c2c(OC)nccn2)=O)C2CCC(C2)C1CC(=O)NC(c1ccsc1)C N1(C(C2CC(CC(=O)NC(CC#C)C(=O)NC)C2)=O)CCC(O)CC12CC2 CC1CCCC=C1C(=O)NC(C)(C)CCNC(=O)CCC1(C)CC1(F)F C1(CNC(CCCN(C(C)C)C)=O)CCN(C(c2cc(C3CC3)ns2)=O)CC1C Cc1ccc(C(=O)NCC2C=CCN2C(C2CC2C2CCC2)=O)cc1Cl C1(C(=O)NC23CN(C(c4cc(C)[nH]n4)=O)C(C2)C3)CCCCC1C1CC1 c1(CNCC(C)Oc2ccccc2F)cnc(F)c(Cl)c1 C(=O)(C(C(C)NC(c1cncc(OC)n1)=O)C(C)C)NC(CCCC)CCC C(CC(C(=O)N1CC(O)(C#N)C1)NC(=O)C(c1ccccc1)C)SC CC(O)C(C(=O)N(CCCNC(C1CSC1)=O)C)NC(c1ccoc1)=O c1(OC)cc(C(=O)NCC2(C)CCCC(F)(F)C2)cc2ccccc12 c1(OC)ccc(C(=O)NC2COCC2NC(c2ccccc2)=O)c(C)c1 c1(CC)c(C(=O)NCC(C2(O)CCN(C(=O)CN(C)C(N)=O)C2)C)csc1C C(C(=O)NC(C)C(CO)NC(=O)C(O)CN(C)C)(C(C)C)NC(CCC)=O C(C)(CCC(=O)N1CCC(NC(=O)CCCF)C1)OCC C(=O)(CC(F)(F)F)NCC(N1C(CNC(=O)C=Cc2ncc[nH]2)CC1)=O C1(NC(CN(C(=O)COC2CCC2)CC)=O)CCC(C2CC2)C1 N1(CC(N2CCC(CN(C(=O)CSC(F)F)C)C2)=O)CCCC(C(N)=O)C1 c1(C(C)C)c(Cl)ncnc1NNC(=O)C1(c2ccc(Cl)cc2Cl)CC1 C#CCC(C)(C)NC(=O)CC1CCCC1NC(=O)C(CC)N(CC)CC CC(CC(=O)NCC1CC(NC(c2cnc3c[nH]nc3c2)=O)C1(C)C)P(C)(C)=O N1(C(C2C(C)(NC(c3cnc(C4CC4)nc3)=O)CCCC2)=O)CCC2CCC(C2)C1 c1(OCC2(C(N3CC(OC4CC4)C3)=O)CC2)nnn(C2CC2)c1C(F)F.CC(C)OCC.C CC1OC2(C(N3CC(F)(CNC(=O)CCCC4CC4)C3)=O)CC1C2 c1(CC)ccc(C(=O)NC2CCC(F)(CNC(=O)C(C)OCCOC)C2)cc1 CN(C1CCCc2c1cnn2C)C(=O)NC(CC(F)F)C(=O)O c1(C(=O)NCCCc2c(C)cccc2)c(C)ccc2ncccc12 Cc1nccnc1C(=O)NC(Cc1cnc[nH]1)C(=O)NCC1CCCCO1 N1(C(C=C(C)C(F)F)=O)CCCC(NC(=O)C(C)Cc2c(C)noc2C)C1C CCCCC(C)C(=O)NC1(C)CCN(C(C2CC3(CC3)C2)=O)CC1 c1(C(=O)NC(CN(C(c2c(CC)nco2)=O)C)CC)cnn(C)c(=O)c1 c1(C(N(C2CCCN(C(c3cn(CC)nc3C)=O)C2)C)=O)cc(Cl)c(O)cc1C c1(CC(=O)N(C2CC2)CCOC)ccc(F)c(Cl)c1.C1(C=O)CC2CCCC2C1 C(=O)(CC(F)(F)F)NC(CCNC(C(C1CCC(=O)N1C)C)=O)(C)C c1(C(N2CC3(CCN(C(C(COC)O)=O)C3)C2)=O)cnn2c(Br)cccc12 c1(CC(=O)NC2C=CCN(C(=O)C=C(Cl)Cl)C2)ccc(Cl)cc1 n1(CC)cnc2c(NCCc3cc(C)oc3C)[nH]c(=NCCn3cnnc3)nc12 C(=O)(C1=CC2(CCN(C(c3cn[nH]c3)=O)C2)C1)NC1C(C)(C)C(=O)NC1 c1(C(=O)NCC(CNC(c2c(OC)nccc2)=O)O)cnc(C)c(N)c1 C1(NC(C(CC=C)NC(c2cc(C)[nH]n2)=O)=O)CCCC(O)CC1 c1(C(=O)NC(c2ncc(Br)cn2)CCC)ccc2c(C)cc(Cl)nc2c1 C1(C#N)(C(N2CCC(O)(CN(C(CCOC(C)C)=O)C)C2)=O)CC2CC2C1 Cn1ncc(C(N2CCCCC2C(=O)NCC2CCCSC2)=O)c1C#N C1(NC(C(CC=C)OC)=O)CCCCCN(C(=O)C(O)CCCCC)C1 N1(c2cc(OCC)ncn2)CCC(O)(C2(NC(=O)COC)CC2)CC1 O=C(C1=C(Cl)CCC1)N1CC2CC1CN2.C1(N2CC(C(=O)N)C2)CCCCC1 c1(C(=O)NCCCCCCNC(c2ncsc2C2CC2)=O)ccc2ccnn2c1 C1(NC(C(c2cc(C)oc2C)C)=O)CN(C(c2cnns2)=O)CC12CCOCC2 c1(C(N2CCC(NC(C3C(OCC)C3)=O)C2(C)C)=O)cccn2ccnc12 N1(C(CN(S(CC)(=O)=O)C)=O)CC(NC(c2cnn(CCO)c2)=O)C(C2CC2)C1 c1(C(N(C2C3CN(C(=O)CCc4nc(O)n[nH]4)CC23)C)=O)ccc2ncnn2c1 N1(C(C=CC=CC)=O)CCC(C(C)C(N2CCC(c3ncco3)C2)=O)C1 N1(C(CNS(CC)(=O)=O)=O)CC2(CCC2)CC1CNC(=O)CCCCNC(N)=O C1(C(C)C)CC(O)CN1C1c2cnn(c2)NC1=O.C1(CC2CCC2)CCOCC1 N1(C(CCN(C(C(=C)F)=O)C)=O)CCN(C)C(=O)C1C c1(NC(=O)OC(C)(C)C)nccc(NC(c2cnn(-c3cccnc3)c2)=O)c1Br C1(NC(=O)Cn2ncnn2)COCCN(C(=O)Cc2ccncn2)C1 c1(CC)ncc(C(N2CC(NC(=O)CCC(C)O)CC2C)=O)c(C)n1 C1(F)(CNC(C(c2n(C)cnc2)O)=O)CCC(CNC(=O)CC2(C)CCCC2)C1 C=C=CC(C)C(=O)N(C)CC1CCN(C(=O)COCc2ccncc2)C1 C(=O)(CC(CCN)CC(=O)N(S(C)(=O)=O)C)NCCCOC C(=O)(C1=CCCC1(C)C)N1CCC(C(C)(C)NC(COc2cc(C)on2)=O)CC1 CCCC(O)C(=O)N(C)CCN1CCN(C(=O)CSCC#N)CC1 C(=O)(C(C)(C)C(F)F)NCCCN(C(C1C(C=C)OCC1)=O)C(C)C CC(C)CC(C)(C)NC(C1CCC1CNC(=O)CC1OCCC1(C)C)=O C(=O)(C(C)(C)C(F)F)NC(C)C(C)C(=O)N(C)Cc1ccco1 C(=O)(C1CCCc2ccnn21)NCC1CC(NC(C2CN(CCC)C(=O)C2)=O)C1 C1(N(C)C)CCC(C(=O)NCC=C2CCN(C(=O)C(=O)N(C)C)CC2)CC1 C=C(Cl)CCC(=O)N(C)CC1CN(C(c2cnc(COC)s2)=O)CCO1 C1(NC(CCN(C(C2C(C)CC2)=O)CCO)=O)CCN2CCCC12 CC1CCn2c(C(N3CCCC(NC(=O)CC(C)C4CCCC4)C3)=O)cnc2C1 C(C(CC)N=c1[nH]c(=NC(C)COCC)[nH]c2c1SCC2)N(CC(=C)C)C CC1CCCN(C(=O)C=CCC2(CNC(=O)OC(C)(C)C)CCC2)C1 CC1CN(C(=O)C(C)(C)c2cncs2)CC1NC(c1cnco1)=O C1(C(=O)NC2CCC(CC)CC2)COCCN(NCc2cccc(F)c2Cl)C1 C1(C(=O)NCCc2nc(C)oc2C)CC(C)(C)CN1C(=O)C(C)Cn1ccnc1 N1(C(CCC2CC(OC)C2)=O)CC(CNC(c2ns[nH]c2=O)=O)OC(C)(C)C1 c1(CC(C(=O)NC2C(NC(c3cncc(C)c3)=O)CCC2)C)ccc(F)cc1F n1(CC)ncc2cc(C(=O)NCC(C)NC(c3cnsn3)=O)cnc12 C1(C(N2CCCC(NC(C(CC=C)(C)C)=O)C2C)=O)CCc2cnc(C)n2C1 c1(C(=O)N=c2[nH][nH]cc2-c2nn[nH]n2)cc2c(s1)CCCCCC2.c1ccccc1 C(=O)(C(F)(F)CC(C)C)NCCC1(C)CCN(C(C(CCOC)C)=O)C1 c1(C(=O)NC2C(CNC(=O)C=Cc3cccs3)C2)cc([N+](=O)[O-])ccc1OC(F)F c1(C(=O)NC2(C)CCN(CCC3COCCOC3)C2)ccc(F)c(F)c1 c1(N2C(C)(CNC(C3C(C)OC(C)C3)=O)CCC2)ncnc2sccc12 CCC(C)(CN=c1nc2c(cnn2C)c(NCC2(CO)CC(F)(F)C2)[nH]1)C(N)=O C(N=c1[nH]c2c(C(=O)OC)cccc2o1)C1CN(C(C2(CCCC)CC2)=O)CC1C c1(CC(=O)NC(CN(C(=O)CCCc2nc(C)cs2)CC)C)ncn(C)c1C Cc1cc(C)c(C(=O)NCCC(C)(C)NC(=O)CC2CC2(C)C)c(C)c1Br c1(CNC(=O)CC2CN(C(=O)NC3(CC)CCC3)C2)cc(O)ccc1C CC1CN(C(=O)C(C)(C)N2CCOCC2)CCC1NC(c1csc([N+](=O)[O-])c1)=O C#Cc1ccc(F)cc1C(N1CC(NC(c2c(F)cc(Cl)cc2F)=O)C(C)C1)=O N1(C(CCCOCCC)=O)CC(NC(=O)C(C(C)C)NC(=O)OCC)C(C)C1 c1(C(N2CC(CNC(C3CC(CF)C3)=O)C2)=O)ccnnc1 c1(C(=O)NCC2CN(C(CP(C)(C)=O)=O)C2)ccc(Br)c(F)c1N c1(C(=O)NCC(c2ccccc2)C(C)C)c(C)oc(C)c1C.C#CC(C)(C)C(=O)N C1(CC#C)(C(=O)NC2CC(NC(=O)CCc3cc(C)no3)C2)CCOC1 C1(OC)C=CCN(C(=O)CC(C)CNC(C2CC2Cc2ccccc2)=O)C1 c1(C(N(C)CC2CCCC(NC(c3c(C)nccn3)=O)C2)=O)cc[nH]c(=N)c1Cl O=C1NCc2c1ccnc2C(N1CCCNCC1)=O N1(C(Cc2scc(C)c2)=O)CCC(F)(C(=O)NC(c2ncn(C)n2)C)CC1 c1(C(N(CC(CN(C(c2cnc(C(C)C)s2)=O)C)O)C)=O)ccc(F)nc1 c1(CCN(C(=O)C(C2CC2)N(C)C(c2ccsc2Cl)=O)C)ccncc1 C1(NC(c2cn(CCCOC)nc2)=O)CCCN(C(c2nc(C)oc2C)=O)CC1 C1(C(=O)NCC(CCNC(CCC(=C)C)=O)(C)C)CC2CCC(C1)N2C(C)C N1(CC=CC(=O)NC2CC(C(C)NC(C=CC(C)C)=O)C2)CCOCC1 N1(C(c2ccc[nH]2)=O)CCC(NC(C23CCC(CO2)C3)=O)C(CO)C1 C(CCCC(CO)NC(=O)Cc1coc(C)n1)NC(C1CN(CCC)C(=O)C1)=O C1(NC(CN(C)C)=O)CN(C(C2CNC(=O)N2)=O)CC1F C1(C(=O)NCC(C(=O)NC(C)CCC(C)C)OC)CC(C)(C)CO1 N1(C(Cc2ccc(C)nc2)=O)CCCC(O)(CNC(=O)C2=CCCCC2)CC1 C=CC(C)(O)CC(=O)N(CC(C)(C)CNC(C1CCC(C)O1)=O)CC N1(CC(=O)Nc2cc(C)no2)CCC2(COCC3C(F)(F)C34CCC4)CCCC12 C(C(CC(C)C)NC(c1[nH]nnc1C)=O)NC(c1cnc(C)s1)=O C(CC(C)(C)C(=O)N1CC(NC(c2ncncc2Br)=O)C2(CC2)C1)OC n1(CC)cnc(C(N2CC(C)(NC(c3ccn(CC(F)(F)F)n3)=O)C2)=O)c1 C1(CC(=O)NCC(C(C)O)C)CC(C)N(C(c2cccc[n+]2[O-])=O)C1 Cc1nc(C)n(CC(=O)N(CC(O)CNC(c2nnc(S)n2C)=O)C)n1 CC(C)CC(CC(=O)NCCC1CCC(C)(C)O1)NC(c1cc[nH]n1)=O N1(C(Cn2c(N)cc(C)n2)=O)CCN(C(=O)CN2CCC2)C(C2CCCC2)C1 C1(N(C(CCCN(C(C)=O)C)=O)C)CC(C)N(C(=O)CN(C(=O)C(C)C)C)C1 C(C#CC1CCCCO1)NC(C(c1ccc(C)s1)C)=O c1(NC(c2nc(-c3ccc(-c4cn(C)nc4)cc3)sc2)=O)ncc2sccc2n1 C(=O)(C(F)(CNC(c1sc(F)cc1C)=O)C(C)C)NCC(C#C)OC C1(C)(NC(C2CCC(C(C)=O)O2)=O)CCCN(C(C2(c3oncc3C)CC2)=O)C1 c1(C(=O)NC2CN(Cc3nnc(CC)s3)C(C)CC2)cc2c(cnn2C)nc1O CC1CN(C(c2sccc2CC#N)=O)CC1NC(=O)CN1CCCNC1=O C(=O)(C(CC(C)C)C(C)C)N1CC(C(=O)NC(COC(C)=O)CO)C(C)(C)CC1 NC(=O)CCCC(=O)NC1CC(CNC(=O)CSCc2ncc[nH]2)C1 C(CC(C)C(=O)N(C(C)C(N1CCOC2CC12)=O)C1CC1)=CC C1(C(N(C2CCC(NC(C3CC(=O)C3(C)C)=O)CC2)C)=O)CCCCN1N=O c1(C(=O)NCCOC2CCN(C(=O)CN3CCC(O)CC3)C2)cc[nH]c2nccc1-2 N1(CC(=O)NCCc2nnc(C)s2)CC2(CS(N)(=O)=O)CC1CO2 c1(C(=O)NCCCCNC(c2nccc(OC)c2)=O)ccc(Cl)cc1OC c1(OC)ccc(C(F)F)cc1C(=O)NC1CN(C(=O)C(C)(F)F)C2CC12 N1(C(C(C=CC)O)=O)CCC(CNC(c2c(C)cccc2OC)=O)C(F)(F)CC1 C1(NC(=O)CCc2nc(Cc3ccccc3)no2)CCOCC12CCCC2 Cc1csc2c(C(N3CCC4(CCC4NC(=O)C(C)C(C)O)CC3)=O)ncnc12 c1(CC)cnc2ccccc2c1C(=O)NC1CCCC(NC(c2cocn2)=O)C1 C1(C(=O)NCCCC(C)(C)NC(=O)Cc2ccnc(Cl)c2F)CCCC12CCC2 c1(NC(C2CCC(NS(=O)(=O)CCCCCl)C2)=O)cc(Cl)ncc1F C(=O)(CCCCCCNC(=O)C1=CCCCCC1)NC(CCC)CC c1(C(N2CC3C(NC(CS(CC)=O)=O)(C3)C2)=O)c(C)nn(C)c1Br c1(CN(C(c2c(CC)noc2)=O)C)ccccc1CNC(=O)C(C(C)O)N(C)C C1(NC(N2CCC(N3CCCOCC3)CC2)=O)CCOC(C(F)(F)F)C1 Cc1[nH]nc(C(N2CCC(C(=O)N(C3CC3)CC3(O)CCC3)C2C)=O)c1C CCC(C)C(O)C(=O)NCCC(C)(C)CNC(C1CNC(=O)C1)=O c1(OC)cccc(F)c1C(=O)NC1CN(CCn2cccn2)CCC1C N1(C(c2c(Br)cn(C)n2)=O)CCCC(C(N2CC3CC2CN3)=O)CC1 C1(C(=O)NCC2(CN(C(C(C)OCCC=C)=O)C)CC2)COc2ccccc2C1 C1(CCC(=O)NC(c2nc[nH]n2)CC)(NC(=O)CC2CCOCC2)CCCC1 c1(N2CCC(C#N)CC2)nc2c(c(=NCCc3cccn4ccnc34)[nH]1)CSC2 c1(C(=O)NCC2CCN(C(C(CC)(C)CO)=O)CC2)ccc(N)c(F)c1F N1(C(C2(C=C)CC2)=O)CC2C(N(C)C(c3cnc(C(F)(F)F)s3)=O)C2C1 CC1(C(N2CCCC(C)(F)C2)=O)Oc2ccccc2NC1=O C(c1cn(C)nn1)=CC(=O)NC(C1CN(C(=O)CC2CN(C)C2)CCO1)C Cc1cc(C(=O)N(C(C)CN(C(=O)C(C)Oc2ccccn2)C)C)cs1 Cc1ccnc(F)c1C(=O)NCCC(C)CO.C12(CCC1)CC(=O)N2 c1(OCC)cc(C(=O)NC2CC(CNC(c3ccc(CCOC)o3)=O)C2)on1 c1(C(N(CC(C)O)CCNC(C(CSC)O)=O)=O)cccc(CO)c1 N1(C(C(C)OC(C)=O)=O)CCC2CN(C(c3cc(C)no3)=O)CC12 CCC(CC)(C(=O)NC1CC1C(=O)Nc1cccnc1C(C)C)C(=O)O C1(C)(CC)CC(OC)CN1C(=O)CS(=O)(=O)Cc1ccc(Cl)s1 CC(C)CCC(O)C(=O)NC(C)CCCCNC(c1cccc2[nH]ncc12)=O C1(CC=C)(NC(=O)CCC=CC(C)C)CCN(C(c2nccn2CCOC)=O)C1 C1(C(=O)NCCCNC(C(C)(C2CC2)OC)=O)Cc2cc(Cl)ccc2O1 C=CCCCCCC(=O)N1CC(CC(=O)Nc2cc(C)c(O)c(C)c2)CC1C N1(C(CC(=C)C)=O)CC(C)N(C(c2c(F)ccc(F)c2OC)=O)CC1C N1(C(C(CC#C)C)=O)CC2CCCC(C1)N2C(c1nn(C)c(Cl)c1C(F)(F)F)=O N1(C(c2c(C)ccs2)=O)CCC(C2CC2)(NC(=O)C(C)OC2CCCC2)C1 C1(C(N(CCS(N)(=O)=O)C)=O)CCN(C(=O)CN(C2CCCC2)C)C(C)(C)C1 c1(OC)ccc(C)nc1C(=O)NC1CCC12CN(C(c1ccc(F)cc1O)=O)C2 CCCC(C(=O)NC)NC(=O)C(c1cccs1)NC(c1cccn1C)=O C(=O)(CC(C)C(F)(F)F)NC1CCCC(C(N2CCC(C)(COC)C2)=O)C1 C(C)(C)(CC(c1nnnn1-c1ccc(OC)cc1)NC1CC(C)C1)OC c1(OC)ccncc1C(N1CC(OC)C(C(=O)N(C)Cc2cc(=O)cc[nH]2)C1)=O N1(C(C=CCCC)=O)CC(NC(=O)CCC2CCC(=O)C2)C(n2cccn2)C1 CC(C)(C)C#CC(=O)NC1CCC(NC(c2cc3occc3[nH]2)=O)C1 c1(NC(N(C)Cc2cocn2)=O)cnc(F)cc1CO Cc1nc2ccccc2n1CCC(=O)N1CCC1C(=O)NC(c1cnn(C)c1)C CC(C)C1=NOC(C)(C(=O)NCC23CC2CN(C(=O)C(c2ccccc2)=O)C3)C1 c1(C(N2CC(CC)N(C(=O)CCc3cccs3)CC2)=O)cccc2nc[nH]c12 c1(OC)ccc(S(=O)(=O)CCN2CCC(c3ncc[nH]3)CC2)cc1 C1(C#N)(N)CC12CCOCC2.C1(C)(C2CC2)C(=O)NCCN1C(C)(C)C.CO C1(CNC(=O)NCCS(=O)(=O)C2CC2)CC12CCS(=O)(=O)CC2 N1(C(CSCC(C)C)=O)CC2CC1CN2C(c1ccnc(C(C)(C)O)c1)=O C(CCC1CC1)(C(=O)NOCCF)NC(c1n(C)c(S)nn1)=O C(C(C)C(=O)NCC1CC1CNC(=O)C(F)(F)c1csc(=N)[nH]1)SC c1(C(N2CCC(CNC(C3(C)CC(C)(C)C3)=O)C2)=O)ccn(CCO)c(=O)c1 c1(C(=O)NC(CCN(C(c2c(C)c[nH]n2)=O)C)C)cc2ccc(Cl)cc2s1 N1(C(C(C)NC(CC)(C)C)=O)CCC(F)(CNC(=O)Cc2ccon2)C1 c1(N(S(=O)(=O)CC2Cc3nnsc3S2)C)cc(=O)oc2c(C)cc(C)cc12 N1(c2cc(NCCc3[nH]cnc3C)nc(C)n2)CCC2(CCC2)S(=O)(=O)CC1 C1(NC(C=CC)=O)CCOC12CCN(C(=O)C(C(C)C)c1cnc(C)s1)CC2 Cn1ccc(S(=O)(=O)N2CCN(C(c3cc(C#N)c[nH]3)=O)CC2CC#N)n1 NC(=O)CC(O)C(=O)NC(CCOCCO)C(=O)NCCc1ccsc1 c1(C(c2nnnn2CC2CCCO2)NC2(CC=C)CCC2)nc(C)cn1C c1(C(=O)NCCC2C(C)CN(C(=O)CCNC(N)=O)C2)cccc(F)c1C#N S(=O)(=O)(c1ccc(NC(c2ccns2)C)c(C#N)c1)NC(COC)C1CC1 c1(C(N2C(C)CC(NC(c3cc(C4CC4)ccn3)=O)C2)=O)cccc2nccn12 C12(CNC(=O)CC3CCSC3)CCC(NC(c3ccnnc3O)=O)(CO1)C2 c1(C(N2CC(C(=O)NCCc3conc3Br)C2)=O)ccncc1Cl C1(N(C(Cn2c(C(C)C)nnn2)=O)CC2CC2)CCCN(C(C2CC2CF)=O)C1 c1(SC)nn(C)cc1C(N1CC=CC1CNC(=O)CCC1CCCCC1)=O c1(C(=O)NC(CCCC)CNC(C2CC2(F)C(=O)OC)=O)cc(C)ccc1Cl Cc1cc(=O)oc(C)c1C(N1CCC(N(C)C(c2cnn(CC3CC3)c2)=O)C1)=O CC(C)(C)C(CNC(=O)Cc1ccoc1)C(=O)NCC1(CCO)CCC1 CC(=O)CCN=C(NCC(N1CCCC1)C)N1CCC(c2cccnc2)C1 C1(C(=O)NC2C3(CCN(C(CC4(C#N)CC4)=O)CC3)C2)CCC2(CC1)CC2(F)F C#Cc1ccc(CCC(=O)NC2CCCNC2)cc1 N1(C(Cc2cnc(C)s2)=O)CC(C(=O)Nc2cccc(-n3cccn3)n2)CC(F)C1 c1(C(N2C3CN(C(=O)C(F)(F)Cl)CC32)=O)c(F)ccc([N+](=O)[O-])c1F N#Cc1ccc(CNCC(S(C)(=O)=O)c2ccccc2)s1 Cc1nc(NC(=O)C(N2CCC(C)CC2)C)c(Cc2cccnc2)s1 c1(C(=O)NCC2(F)CCN(C(C3(F)CCCCC3)=O)C2)ccc2c(c1)CCC2 CCN=c1[nH]c(C)c(C(=O)N(C2CCCN(C(=O)C(C3CC3)OCC)CC2)C)s1 C1(CC=C)(C(=O)NCC(C(=O)OC)OC)CCCN1C(c1cc(CC)n(C)n1)=O N1(C(Cc2n(C)ncc2)=O)CC(CNC(C2(CF)CC2(F)F)=O)CC(C)(C)C1 N1(C(c2c(CC)n(C)cc2)=O)C2CCC1C(C(=O)Nc1cnc(OC)c(C)c1)C2 C(=O)(CC(C1CC1)NC(C)=O)NC(C(=O)NCCC=CCCC)C N1(C(CC(=O)OCC)=O)CCC(C)(NC(=O)C(C(C)C)OC)C1 CCC(F)C(=O)N(C1CN(C(=O)C(C)N(CC(F)(F)F)C)C1)C c1(NC(c2cc(Br)ccn2)c2n(CC(=C)C)nnn2)cccc(SC)c1 CCCCCCCC(=O)N1CCN(C(=O)Cc2ccc(S(C)=O)cc2)C2CC12 c1(C(N2CCCC(NC(c3nccc(C)c3)=O)CC2)=O)cc2nc(C)ccc2o1 C12(CC3CC1CC3)c1nnnn1C(c1ccccc1)C(=O)N2.C(CCF)OCC N1(C(c2ccc(CCC)s2)=O)CCC12CN(C(=O)C=Cc1ccncn1)C2 C(CC(C)C(=O)NCC(C1CC1)N(C)C(c1ccc(N(C)C)nn1)=O)=CC C1(CNC(COCCOCC)=O)CC2CCC(C1)N2C(=O)CCc1ccc(C)s1 c1(C(C(N2CCC(C(C)(C)NC(=O)Cc3ccco3)C2)=O)=O)ccc(O)cc1 C1(CCC)CCCC1C(=O)NCCCN(C(=O)CCN1CCCC1=O)C N1(C(C2(C=C)CC2)=O)CC(NC(C2(C(C)(F)F)CC2)=O)C(C2CC2)C1 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C)CN(C(=O)CCSc1nnnn1C)C CC1CCn2cc(C(N3CCC(C4CCCN4C(C4CCOC4)=O)C3)=O)nc2C1 C(=O)(C1CCc2cccnc21)NCC(CN(C(CCC(=O)OCC)=O)C)(C)C C(=O)(CCC(F)(F)C(F)F)N1CC(NC(COC(C)C)=O)C2C1CCC2 CC(C)CCC(O)C(=O)NC1(C(=O)NOCC2CCCO2)CCOCC1 N1(C(CC)=O)CC(CNC(=O)CSc2nc3ccccc3[nH]2)N2CCC1C2 C1(CNC(c2cnc(C(C)=O)s2)=O)CCCN(C(=O)C(Cl)=CCl)C1 C(=O)(C(c1ccoc1)NC(C1CC1Cl)=O)N(CC(C)O)CC(F)F CC1CC2(CCC2)CN1C(c1noc2c1CCC2)C(=O)NCCCNC(N)=O C(=O)(CCCCC1CC1)N1CC(=C(CNC(=O)C(C2(O)CCCC2)F)F)C1 Cc1c(C(N2CCN(C(=O)C(C)C(C)C)CC2C)=O)ccc2cncn12 c1(C(N2CCC(C)(CC(=O)NC(C#C)C(C)(C)C)C2)=O)nccc(C)c1N N1(C(Cc2cnc(C)o2)=O)CCCN(C(=O)Cc2cn3c(C)csc3n2)CC1C c1(N)ccc(C(=O)N(C)C)cc1.c1(C(c2nnnn2CC)CCCC)csc(Br)n1 CC(CC(=O)N1CC(NC(c2cnc(O)s2)=O)C(F)C1)C(F)F C1(CNC(N(C(C2(C)CC2)C)C)=O)CC12CCCC2 C1(NC(C23N(C(=O)CC45CCCC4C5)CC(C)(C2)C3)=O)CCn2nnnc2C1 Cc1cc(N2CCC(N(C)C(c3cc(C(F)(F)F)cc(Br)c3)=O)C2)nc(C)n1 C(=O)(C#CC1CCOCC1)N1CC(CCCNC(CSCC(C)C)=O)OCC1 c1(C(=O)NC2CC(C)N(C(=O)C(=O)NC(C)(C)C)CC2)cnc2c(c1)CCCO2 c1(C(N2CCN(C(Cc3onc(C)n3)=O)CC2CO)=O)c[nH]c2cc(Cl)ccc12 Cc1nccc(C(=O)NC(c2ccccc2)CC(C2(CC3CC3)CC2)=O)n1 C(=O)(C(C)(C(C)C)N(C)C)NC1C(OC)CN(C(C2(CSC)CCCCC2)=O)C1 CC1(C)CN(C(C2CCN(C(=O)C(C)(C)n3cccn3)CC2O)=O)CC(=O)N1 C(=O)(CCC(=O)NN(C)C)NCC(CN(C(c1c(C)cc(O)c(Cl)c1)=O)C)(C)C CN1CC(C(=O)NC2CCCC2NC(=O)CC2(C(F)(F)F)CC2)CCC1=O C1(N(C)Cc2ccccc2NC(=O)NCc2ccccc2)CCCCC1(C)O CCCC(C(=O)NC1CCCCC1NC(c1ncn2ccccc12)=O)S(N)(=O)=O C(=O)(C(C)(F)C(=O)N1CCC(F)(C(=O)NC(CO)CC(F)(F)F)CC1)OC S(=O)(=O)(c1cccc(=NC(C)c2cccn2C(C)C)[nH]1)NCCCNC(=O)NC n1(CC(=O)NCCC2CC(NC(C(CC=C)NC(C)=O)=O)C2)cnc([N+](=O)[O-])c1 C=CCCCC(C)(C)C(=O)NC1CCC(F)(CNC(c2cnco2)=O)C1 C1(CNC(c2c(C)cnnc2)=O)CN(C(=O)CC2CC2(C)C)CC2(CCC2)O1 C(C1CN(C(c2cccn2C(C)C)=O)Cc2ccccc21)NC(CC)=O N1(C(C(CC)N(C)C)=O)C2CCC1C(F)C(NC(c1cn3ccsc3n1)=O)C2 Cc1ccccc1C(N1CCCCC1c1n[nH]cc1C(=O)N(CCN=[N+]=[N-])C)=O N1(CCC)CCCC(C(=O)NC(C2CN(C(C3CCCN3C)=O)CCO2)C)C1 C1(C(=O)NC2CCCN(Cc3cccc(Cl)c3Cl)CC2)CCCCC1C1CC1 c1(C(=O)NC(c2c(SC)cccc2)CO)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] c1(C(C(=O)N(CCNC(C2C(OCC)C2)=O)C)=O)c(C)nn(C)c1C C(C(CCO)CC(C)C)NC(CC(C)OC)c1nnnn1C1(C)CC1 c1(C(N(C)CC2(CNC(=O)CC3CCOC3)CC2)=O)c(F)ccc(F)c1Cl Cc1c(Br)ccc(C(=O)NC2C=CC(C(=O)NCc3ccc(Cl)c(Cl)c3)C2)c1F N1(C(C2CCC(OC)CC2)=O)CC(C2CC2)(CO)C1.N12CCC(C1)OCC2=O n1(C(C)C2CC2)cc(CC(N2CCC(N(C(=O)CCCF)CCO)C2)=O)cn1 C1(CN(C(C(=O)N(C)C)=O)C)CCCN(C(c2ccc(C3(O)COC3)cc2)=O)C1 N1(C(c2ccn(C)c2C2CC2)=O)CCC2(CCCC2NC(=O)C2=CCCCC2)C1 N1(C(C2OCCN(C(C)C)C2)=O)CCN(C(=O)CCCN2CCCC2)CC1C c1(C(=O)NCCCCCCNC(C(C)N(C)C)=O)c[nH]c2ncccc12 c1(OCCC(=O)N(CC)CC)ccc(F)cc1Cl.C1(=O)CC2(CC2)N1 C1(CC(=O)NCC(CN(C(c2c(SC)ccs2)=O)C)C)CCOC1(C)C c1(C(=O)NCC2C(CNC(CSCCCC)=O)C2)cnc(C2CC2)cn1 N1(C(C2N(C(C(C)NC(CC)(C)C)=O)CCCC2)=O)CCC2CC1C(=O)N2C N1(C(c2c(C)onc2)=O)CCC2(CC1)CN(C(C1(N3CCCC3)CCC1)=O)C2 C(=O)(CC1OCc2ncccc21)NC1CC(NC(c2c[nH]cc(C)c2=O)=O)C1 C1(CNC(Cn2cc(C(=O)OC)nc2)=O)C(C)CCCN1C(C1(F)CCCC1)=O C1(O)(CNC(C2C3CCCC23)=O)CCN(C(c2ccc(C(F)F)cc2)=O)CC1 Cc1ccc(F)cc1C(F)(F)C(=O)NCCCN(C)C(c1cc(Cl)n(C)n1)=O C(=O)(C1=CCCOCC1)N1CC(C2CC2)(C(N(C(C#C)C2CCC2)C)=O)C1 c1(OC)cc(C(=O)N(C2CCN(C(=O)Cc3csc(Cl)c3)C2)C)nn1C c1(C(=O)NCCC2CC(NC(CN(c3ccccc3)CC)=O)C2)cc(C)c[nH]1 C1(CCCNC(c2cnc(CC)[nH]2)=O)CN(C(c2ccon2)=O)CCO1 c1(C(=O)NC2(COC)CN(C(C3COCCC3C)=O)C2)nn(C)cc1S(C)(=O)=O Cc1cc(-n2cncn2)ccc1C(N1CCC2CCC12CNC(C1CSC1)=O)=O CCC(C)(COC)C(=O)NCc1ccc(C(=O)NC2(C)CC(F)C2)o1 C(=O)(C(COC)CC(C)C)N1C(CC(=O)NC(CC)C(C)CN(C)C)CC1 C12(C(N3C(C)(C(C)C)CC3)=O)CC1CN(C(C1CSC1)=O)C2 N1(C(C2CC(CC)C2)=O)CCCC1CNC(=O)Cn1cnc(C(N)=O)n1 c1(CC)nnsc1C(=O)NCC1CC(F)(CNC(=O)C(C#N)C2CC2)C1 c1(C(=O)NCCSC)ccc(C)c(NC(=O)OCC)c1.C=CCC1C(=O)N1 C1(c2n(C)nnn2)(Nc2cccc(CC(F)F)c2)COC(C(C)(C)C)C1 N1(C(CC=C)=O)CC(NC(=O)C(C)CS(C)(=O)=O)CC12CCOCC2 CC1CCC(C)N(C(=O)CCCCN(C(=O)CC23CCCC2C3)C)C1 CC1CCN(C(=O)C(C)(C)O)CC1NC(c1ncc(Cl)n1C)=O C=CCC(CC)C(=O)N(CCCCC(=O)NC1CCCCNC1=O)C c1(C(=O)OC)ccc(C(=O)NCC(C)CNC(c2cn(C)nc2Cl)=O)c(C#N)c1 c1(NC(=O)CC2CN(C(c3snnc3-c3ccccc3)=O)C2)ccc(I)cc1I c1(C(N2CCN(C(Cc3cn(C)nc3)=O)CC2C2CC2)=O)cnn2c(Cl)cccc12 C1(C(N(C2CC(O)C2)C)=O)CC1C1CN(C(c2ccnn2C)=O)C1 N1(C(c2cnn(CCC)c2Cl)=O)CC2CCN(C(=O)CCOC(C)C)CC12 C1(OC)CCCC(CN2CC(O)(CNC(=O)C(C)Oc3ccc(Cl)cc3)C2)C1 C1(C(=O)OC)CCC1(C)C(N1CC(C)(NC(=O)CCC=CC(C)C)C1)=O N1(C(c2cc(COC)no2)=O)CCCC2CN(C(=O)CC3=CCCC3)CCCC12 c1(OC)ccc(CCC(=O)OC(C)C(=O)Nc2cc(Br)ccc2OC)cc1O N1(C(C(C(C)C)SC)=O)C(C(=O)NOCc2cccc(C)n2)CCC12CC2 N1(C(C23CC(C)C2C3)=O)CC2(CCCN(C(=O)CCC(N)=O)C2)C1 C(=O)(C#CC1(C)CC1)NCCCN(C(c1cccc(Cl)c1)CC)C c1(OC)cccc(C2=NOC(C(=O)NCC=CCNC(=O)C(C(C)O)SC)C2)c1 C(=O)(C(C)C(C)NC(=O)C(C1CCCCC1)O)NC1(c2nc(C)sc2)CC1 N1(C(C=CC=CCC)=O)CCC(CNC(c2cc(N(C)C)ccc2F)=O)C(C)C1 C1(CNC(=O)NC(CCCC)CO)CC2CCCCC12 c1(C(N2CCC(N(C(C3CC(C)=NO3)=O)CC)CC2)=O)ccc2c(c1)NC(=O)C2 N(C(=NCCC1CCCCC1)NCCN1CCOCC1)C1C(N)CCCCC1 C#Cc1cccc(C(=O)NC23CC2CN(C(C2CC4(CCC4)C2)=O)C3)c1Cl C(C(C)C(C)C(=O)N1CCC(OCCNC(c2cccnc2)=O)CC1)OC CC(C)(C)CCC(=O)N1CCOC(CCCNC(=O)C=Cc2cocn2)C1 C#CCCC(O)C(=O)NCC1(CNC(=O)C(C)(C)C2CC2)CC1(F)F C(C(C)CN=c1[nH]c(=NC(C)CCc2cccn2C)[nH]c2cccnc12)OC c1(-c2ccc(C)o2)nc(C=Cc2ccc(SCC(=O)NC(C)C)cc2)n(C(C)C)n1 C1(NC(COCC#C)=O)CCN(C(c2ccc(C(C)C)cc2)=O)CC1CC Cc1nn(CCO)c(C)c1C(N1CCC(C)(NC(=O)C(C)N=[N+]=[N-])C1)=O N1(C(CSCCC)=O)CCC(CNC(C2(c3ccccc3)CC2(C)C)=O)CC1 N1(C(C2C(NC(c3c(C)ccc(Cl)c3)=O)C2)=O)Cc2cc(Br)cnc2C1 c1(C(N2CCC(NC(c3oc(C)c(Br)c3)=O)C2)=O)ncc(Cl)cc1F N1(C(Cc2cn(CC)nn2)=O)CCC2CC1CN2C(=O)Cc1cccc2c1OCO2 Cc1c(C(=O)NC(C)CC2CN(C(C3C4CCCC34)=O)C2)oc2c(Cl)cccc12 N1(CC)CCC(NC(=O)C(C)(C)CCNC(c2cnc[nH]c2=N)=O)C(C)C1 c1(C(C)(C)C)conc1C(=O)NC(CNC(=O)C(C)(O)C1CCOC1)C1CC1 C(=O)(C(O)CCS(C)=O)N1CC2C(CNC(c3c(OC)ncnc3OC)=O)C2C1 O=C(C#CC1CCCCC1)NCC1N(C(C2CCCOC2)=O)CCCC1(C)C N1(C(c2n(CC)ccn2)=O)CCOCC(NC(C2CCCCN2CC(F)F)=O)C1 c1(C(=O)NCC2(C)CCCN2C(c2cnc[nH]2)=O)ncc(Br)cc1N C(=O)(CS(=O)(=O)C1CC1)NC1CCCC(N(C(Cc2c(C)n[nH]c2C)=O)C)C1 C(C)(CCC(F)(F)F)NC(C(CSC)(C)NC(C1CC12CCCCC2)=O)=O c1(OC)nc(C)ncc1C(=O)NCCC(O)CNC(=O)Cc1cncnc1 C=CC12CCN(C1)C(=O)CONC2=O.C1(COC)CCCN1NCC N1(C(CCC(C)SC)=O)CCC(NC(C2(F)CCCCC2)=O)C12CCC2 C(CC(C(C)C)NC(c1cc(C)no1)=O)NC(C(CC)n1cccn1)=O C1(N(C)C(=O)OC(C)(C)C)CC2CC(NC(=O)NNC(=O)C3CCCCO3)C2C1 C1(NC(C=CC=CC)=O)CN(C(=O)CC2(OC(C)=O)CCCCC2)C2(CCC2)C1 C1(CNC(C2C(NC(CC3C(C)=NNC3=O)=O)CC2)=O)CCC(C)(C)CC1 c1(OC)cc(CC(C)NC(C2CCC(N)C2N)=O)ccc1O c1(C(=O)NCCCC2N(C(CCC=C(C)C)=O)CCC2)ccnc(C2CCC2)c1 CC(O)CCCc1cn(CCCN(C)C(c2ccc(C(N)=O)[nH]2)=O)nn1 C1(C(=O)NC2CC(F)(CNC(C=C(C)Cl)=O)C2)CCn2c(C)nnc2C1 C(C(C(=O)NCc1cc(C)co1)C(C)(C)C)NC(C(COC(C)=O)C)=O c1(C(N(CCCNC(c2cn(C(F)F)cn2)=O)C(C)C)=O)nc(=O)n(C)[nH]1 C1(NC=O)COCCN(C(=O)C=CBr)C1.c1(-n2cccn2)ccc(O)cc1 N1(C(c2cnc(SC)nc2)=O)CC(NCc2ccc(Br)nc2)C2(CC2)C1 c1(N2CCN(CCNC(C(CC)O)=O)CC2)nc2ncc(Cl)cc2o1 C#CC1CCN(C(C2(C(C)C)CCN(C(=O)CC3OCCO3)C2)=O)C1 c1(CCC=CC(=O)NCC2CN(C(C3CN(C4CCOC4)C3)=O)C2)ccccc1 N1(C(C2CN(CC)C(=O)C2)=O)CC(NC(=O)CCOCC(C)C)C2(CC2)C1 c1(C2C(C(N(C3CC(NC(=O)C(F)=C4CCCC4)C3)C)=O)CC2)nc(S)n[nH]1 Cn1nc2c(c1C(=O)N=c1[nH]onc1C1CC1)CN(S(=O)(=O)C1CC1)CC2 CCC(C)CCCC(=O)NCCC1CSCCN1C(c1cc(SC)n(C)n1)=O c1(CC(N2CC(CNC(C(c3c(C)cncc3)C)=O)C2)=O)cccc2cn[nH]c12 C(=O)(CCC(=O)NN(C)C)N1CC(CC)N(C(c2cc3c[nH]cnc-3n2)=O)CC1 C1(C)(C(=O)OC)CCCN(c2nn(Cc3ccc(Cl)cc3)cc2I)C1 Brc1ccc2nc(C3CCN3Cc3ccsc3-c3cc4ccccc4[nH]3)[nH]c2c1 CC(C)(CS(N)(=O)=O)NC(=O)NC1CC(C)(NC(=O)Nc2ccccc2)C1 C1(CCC)CCCC1C(=O)NCCCOCCNC(=O)C=CC(F)(F)F c1(C(=O)NCCOC2CN(C(C(C)C3CCCO3)=O)C2)cccc2sccc12 c1(C(C(=O)OC)N(C)C(c2c(Cl)n[nH]c2C2CC2)=O)ccc(Br)cn1 c12cc(C(F)(F)F)ccc1OC1(CC1)CN2.c1(C(=O)OCC)cn(CN)nn1 C(CCC(=O)NCc1ccoc1C)(C(C)C)NC(CCC#C)=O c1(CC)nc(Cl)nc(N2CCC(C)(NC(=O)CCC(C)N(C)C)C2)c1C#N N1(C(C(=O)Nc2ccc3c(c2)COC3=O)=O)CCc2cc(Br)cc(Cl)c2C1 CC1(CCC(=O)NC23CC(F)(C2)C3)CCCN1C(=O)C=CC(=O)NC1CC1 N1(CC(=O)NC2(CCNC(C34CCC(CC3)C4)=O)CC2)CC(=O)NC1=O N1(c2n(CC)ncc2)CCCC(NC(=O)N(C)CC2(F)CCOC2)C1=O c1(C(N2C(C)C(NC(c3cn(C4CCC4)cn3)=O)CC2)=O)ccc2c(c1)CC2 C1(C(c2n(C(C)C)nnn2)NCc2ccccc2C(F)(F)F)(CO)CCOCC1 C=CCC(CC(C)C)C(=O)NC1CN(C(c2ncncc2Cl)=O)CC2(CCC2)C1 C1(CC(=O)N(C2CSC2)C)CCCC12CN(C(=O)CCc1cccnc1)C2 c1(C(F)F)cc(N2CCC(CNc3cccc(Oc4ccccc4)c3)C2)ncn1 C1(C(=O)NC2CCCN(C(C3(C(C)C)CNC(=O)C3)=O)C2)CCC(C#N)CC1 c1(C(=O)NCC2CN(C(=O)CC3CCCOCC3)C2)cc(F)cc2nc(S)[nH]c12 C1(N(C)C(c2ccnn2C2CC2)=O)CCCCN(C(=O)C=Cc2ccncc2)C1 N1(C(C2CN(C(C)=O)C2)=O)CCC(N(C)C(c2ccc(N)cc2F)=O)C(C)C1 C(C)(C(C)NC(=O)NCC1(O)COC1)(C1CC1)OC n1(CCSC)nnnc1C(c1ccccn1)NCC1(c2ccccc2)CC1(C)C C(=O)(C(F)(CC)C(=O)OC)NC(CC)CN(C)C(c1ccc(C2(C)CC2)cc1)=O C(=O)(C(CCOCCO)NC(c1ccc(O)nn1)=O)NCc1cc(CC)no1 N1(C(C2CC(=O)NC2)=O)CCCC2C1CCN2C(c1cnnc(C2CC2)c1)=O c1(-c2cn(C3CC(C(N(CC(C)OC)CC)=O)C3)nn2)c[nH]c2ccccc12 C1(C(=O)N(CCC(C)NC(C2(C)CCCS2)=O)C)(OC)CCCOC1 c1(C(=O)NCC(N2CCC(C(C)NCCN(C)C)CC2)=O)ccc(O)c(N)n1 c1(C(N(CCNC(C2CCC(=O)N2)=O)CC)=O)cc(C)n(-c2ccon2)c1C c1(C(C)C)ccc(NC(=O)C(N2CCN(CCN)CC2)C)cc1 N(C(=NCCCC(C)(C)O)NC1CC1c1c(Cl)cccc1Cl)CC(C)(C)C C(=O)(C1CC(O)c2ccccc21)NCC1C(CNC(c2cn[nH]c2)=O)C1 N1(C(C2CC(CC)OCC2)=O)CCN(C(c2ccc(Cl)c(O)c2)=O)C2(CC2)C1 CCC(CC)C(C)NC(=O)CC1(NC(=O)CCc2cccs2)CC1 N1(C(CC2OCC(C)(C)C2)=O)CC2(CC2)CC1C(=O)NC1CNC(=O)C1(C)C C(=O)(C(C)(C)CC(C)(C)C)NC1C(NC(c2nn(C)c(=O)cc2)=O)CCCC1 C1(NC(C(=O)O)C2(c3ccc(Cl)nc3)CC2)CC(C(=O)O)CC(C(F)(F)F)C1 C1(NC(CSCCCC)=O)COC2(CCN(C(c3cc4nc[nH]c4cn3)=O)C2)C1 C(C(=O)N1CC2C(NC(=O)CCn3ccc(C)n3)C2C1)(C(C)C)NC(C)=O C#CCCC(=O)NCC1CC(CNC(=O)CN2CCCC2CO)C1 C(=O)(CS(=O)(=O)N1CCOCC1)NC(CNC(=O)Cn1ncnn1)C1CCC1 C1(N(CC(CC)C)C)CCCN(C(C2CC(F)(F)C2)C(=O)NC2(C)CC2)C1 C(=O)(C(C)CC(C)C(C)=O)NC(C(=O)N(C)Cc1scc(C)c1)CCF N1(C(C(CC)COC)=O)CCN(C(=O)CCc2ccc(Br)cn2)CC1C C12(C(=O)NC3CC(C(C(=O)NCCN4CCC(OC)C4)F)C3)CC1CNC2=O CC#CCC(C(=O)NC(C)CCc1cn[nH]c1)NC(c1cnco1)=O c1(C(C(=O)NCCCOC)N(C)Cc2nn(C)cc2Cl)csc2cc(Cl)ccc12 C(=O)(CC(C)(C)CC(=O)NC(C1CCOC1)CNC(c1cccc(=O)o1)=O)OC C(=O)(C(CC(C)C)NC(=O)C(C)(C)C)NCCc1cn(CCC(=O)OC)nn1 CC1(C)C(CNC(=O)C(O)C2CC2)CCN1C(c1nnc(C(F)(F)F)s1)=O C1(C(N2CCC(F)(CNC(CNS(CC)(=O)=O)=O)C2)=O)CC2(CCC2)CCO1 C1(C(=O)NCc2c(C)ccc(F)c2)CCN(C(c2cc(C)n(C)n2)=O)C12CCC2 C(N=C(NCc1cccs1)N1C(CO)CC2COCC12)c1occc1 C1(C(=O)Nc2ccc(OC3CCNC3)cc2)CC2CC(N)C2C1 C1(NC(C(=O)NCCCCCC)=O)CCN(C(=O)NC2CCCN(CC)C2)CC1 CC(CC(=O)NCC1CN(C(c2ccccc2)=O)CC12CCC2)C(C)(C)C C1(CNC(CC(CC)C)=O)CN(C(=O)CCn2ccnn2)CCC12CCOCC2 C(C(C)(C)CNC(C1CCOC1=O)=O)N(C(=O)CCc1cnn(C)c1)C C=CC1(C(=O)NCCOC(C2CCC2)=O)CCN(C(=O)CC2C=NN(C)C2=O)C1 c1(NC(=O)NC(C)CC#N)ccccc1 CC1CCCN1C(c1cn(CCNC(C2CC2C2CC2)=O)nn1)=O C(=O)(CCC(=O)NC1CCC(CNC(=O)CSc2nnnn2C2CC2)C1)OCC C(=O)(C(CO)C(C)(C)C)N1CCC(C(=O)NCCc2onc(C)n2)C12CC2 C(C(F)C(=O)N1CCC(C(C)(C)NC(=O)CC2CCC(=O)O2)C1)N(CC)CC N1(C(C2C(=C)CC2)=O)CCCCC1c1cn(CC2CCCOC2)nn1 C=Cn1nccc1C(=O)NCC(O)CNC(c1cnn(C)c1Br)=O CC(C(=O)OCc1c[nH]ccc1=N)C(=O)N1CCOCC1.C1C(=O)O1 N1(C(C2C(CCC)C2)=O)CC2(CCN2C(=O)COc2cc(F)ccc2F)C1 c1(CNC(C(c2cnn(C)c2)NC(C(C)N(C(C)=O)C)=O)=O)cc(C)c(C)o1 c1(C(=O)NCC2(C(N)=O)CN(C(C3(OC)CCC3)=O)C2)cccn(C(C)C)c1=O C1(NC(C2C(C)CN2C(=O)CSc2nc[nH]n2)=O)CC(C)(C)OC1=O Cc1cnn(C(C)C(=O)NC2CC(C(C)NC(c3occc3C)=O)C2)c1 c1(CN(C)C(c2n[nH]cc2CNC(c2ncn(C)n2)=O)=O)nccn1C C1(CCNC(c2cc(CO)[nH]n2)=O)CCCCN1C(=O)CCF c1(CCN(CC)CC)nc(-c2ccco2)nn1-c1ccc(OC)cc1 C(C)(CCC(=O)NC12CC(C1)N(C(=O)C(C)c1ccco1)C2)c1cc(C)no1 CC1CS(=O)CCN1C(=O)CC1CCCN1C(=O)CN1CCCCC1C N1(C(C2CC(C)(C)OCC2)=O)CCC12CCCOC2 c1(-c2ncc(CN3C(CCO)CCCC3)s2)cccc(Cl)c1 C1(NC(c2cc(CC)oc2C)=O)CN(C(c2sccc2C(F)F)=O)CCC1C C(=O)(C1CCCc2sccc21)NCC1(F)CCCN(C(Cc2n(C)ccn2)=O)C1 N1(C(c2cc(C#N)on2)=O)CCCC(NC(c2ccc(N3CCC3)nc2)=O)CC1 C1(CNC(c2ccc(C#C)o2)=O)CN(C(C2(O)CCC2)=O)CCC1C N1(C(C(C)OCCC=C)=O)C2CCC1CN(C(=O)CC(=O)OCC)CC2 N1(C(C2CC(C#C)(O)C2)=O)CCC2CC(CNC(=O)C3=COCCO3)CCC2C1 N1(C(C=C(CC)CC)=O)C(CNC(=O)CCNC(C)=O)CC2COCC12 c1(C(N2CCC(N(C(C(c3ccccc3)SC)=O)C)C2)=O)ccc(C#N)o1 O(NC(=O)CNC(=O)C(CNC(C1(CCOC)CCCC1)=O)N(C)C)CCOC C1(C(N(C2CC(CC3CCCN3C(=O)C(=O)N(C)C)C2)C)=O)CCCCCC1 c1(C(=O)NCC(=C)CCNC(=O)CC2CC(F)C2)cnc(O)n(C)c1=O C1(C(C(=O)NCC(C)C)(C)C)CCCCN1C(C)=O.c1(C(=O)OCC)ccccc1 c1(OCC)c(OC)cc(C(=O)NC(CNC(C23CCC2C3)=O)CC(C)C)cc1Cl C1(CNC(c2coc(C(F)F)n2)=O)CC2CCCC(C1)N2C(=O)C(F)C1CCC1 N1(C(C2N(C(N)=O)CC(O)C2)=O)CCC2(C1)CN(C(c1cc(CO)ccn1)=O)C2 C1(CN(c2ccccn2)C)CCN(S(=O)(=O)CCOC(F)F)C1 N1(C(C(C)C2CCC2)=O)CC2(CCC2)CC1CNC(c1coc(Br)n1)=O C#CC12CCC(C(=O)N(CC(C)NC(C3CCC(COC)CC3)=O)C)(CC1)CC2 CC1OCCC1C(N1CCC1CN(C(=O)CCC1CCC(=O)C1)C1CC1)=O N1(C(CC2C(C)C2)=O)CC2CCC(C1)C(NC(C1CCOCC1(C)C)=O)C2 C#Cc1ccccc1CC(=O)NC1CCC(C(=O)NCC(c2ccncc2)C)C1 N1(C(c2cc(C)ccn2)C(=O)NCC=C)CC(C)OCC1C N1(CC)CCN(CC(N2CC(NC(=O)C(F)=C3CCC3)C2)=O)CC1 C1(C(N(CC(C)N(C(C)=O)C)C)=O)(NC(c2cc(O)ncn2)=O)CCN(C)C1 C1(C(N2CCC3CN(C(COC(C)=O)=O)CC32)=O)CCc2cc(Br)ccc2O1 c1(C(=O)NCC(CC=C)NC(c2ccc(CO)s2)=O)ccc(O)c(F)c1F C(C)(C)(C(=O)N(CCCCCNC(C1(C(F)F)CCCC1)=O)C)NC(=O)OC c1(-c2cc(OC(C)C3CC3)ncc2)ccc(S(=O)(=O)NCc2nccs2)cc1 C(=O)(CCC(=O)NN(C)C)NC(C(=O)N(CCC1CN(C)C1)C)CCC1CC1 c1(C(=O)NCC=CC(=O)NCC(C)OCC=C)ncncc1N c1(NCC2(NC(C(C=C)O)=O)CCCCC2C)ccnc2ncnn12 c1(C(=O)NC2CCC(CNC(C(C)SC)=O)CC2)cn2cccc(Br)c2n1 CCC(CC)(CC)C(=O)NC1CCC(NC(c2cc3ncccn3n2)=O)C1 S(=O)(=O)(c1cn(C)cn1)NCC(N1C(CNC(C(C(C)C)NC=O)=O)CC1)=O c1(C(=O)NC(CNC(C(C)(CO)OC)=O)CC(C)C)ccc(F)c(Cl)c1 CCC(COC)C(=O)NCCCN(CCCCNC(C1CC1CC)=O)C CC1CN(C(c2cncc(NC3CCC3)c2)=O)CC1NC(=O)CCC#N c1(OC(C(=O)NC(C)CC2CN(C(c3ncc[nH]3)=O)C2)C)ccccc1Cl c1(C(=O)NCC2(F)CN(C(CC3CC(CC)OCC3)=O)C2)cc2sc(C)cc2s1 C1(C(=O)NC2C(OC)CN(C(=O)CCN3C(=O)CCC3=O)C2)CC2(CC(=O)C2)C1 C(CCCCCCCC(=O)O)ONC(C(N1CCN(C2=NCCS2)CC1)(C)C)=O N1(C(c2c(C)nc(COC)s2)=O)CC(NC(c2cnc(Cl)n2C)=O)CC(C)C1 N1(C(C(CCC)(C)O)=O)CCC2(CC1)CN(C(c1ccc(OC)nc1C)=O)C2 N1(C(COCCC=C)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1C1CC1 C(=O)(C(C)(C)CCCF)N1CC(OCC)(CNC(=O)Cc2cccc(F)c2)C1 C(=O)(C(C)CS(C)=O)N(CCNC(c1n[nH]c(C)c1Br)=O)C(C)C c1(C(=O)NC(C2OCCN(C(C3(COC)C=CCC3)=O)C2)C)cc(O)cc(Cl)c1 N1(C(CCCN(C(=O)COCCCF)C)=O)C2COCC1C2 N1(C(=O)Nc2c(OC(C)(C)C)cccn2)CCCC2(CC(O)C2)C1 N1(C(=O)Cc2cscn2)CCCC(F)(C(=O)NC(CC2CC2)CO)C1 C1(CC(C)NC(CSC)=O)CC2CCC(C1)N2C(c1cn(C2CCOC2)nc1C)=O C1(C(=O)NCc2c(=O)ccn(C)n2)CC2CN(C(=O)OC(C)(C)C)CC1O2 Cn1nc(C(=O)NCC2CCCC2NC(=O)CCC2CCC(=O)NC2)cc1C#N c1(C(N(C(CCNC(CCC#CC)=O)C)C)=O)cnc2ccc(C)cn2c1=O c1(C(=O)NC(C)Cn2cc(C3(C)CCCO3)nn2)c(F)cccc1Br C1(C(=O)NC(CNC(=O)Cn2ncc(O)nc2=O)CO)CC2CSCC(C1)C2 c1(C(N2CC(C(C)NC(C3CCC3)=O)C2)=O)ncn(C(C)(C)C)n1 Cn1cnc2c(C(N3CC(CNC(=O)C(C)(C)O)C3)=O)cccc12 Cc1cc(C(=O)NC2CN(C(C3CCCC3(C)C)=O)CC2O)cc(C)c1Cl CC12CCC(C(=O)NC3(CC(N4CC(CO)CC4CO)=O)CCC3)(CO1)C2 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC(C1N(C(CC(C)OC)=O)CCC1)C CC1CC(=O)NC1C(=O)NCCCCn1cc(CN(c2ccccc2)C)nn1 N(C(=NCc1ccc(CC)cc1)NCC1COCCOC1)C(C=C)C C1(OC)CCC(CNC(c2cn(Cc3ncccn3)nn2)=O)CC1 N1(C(C(CC)NC(C)=O)=O)CCC(F)(F)C(CNC(=O)CCCNC(N)=O)C1 c1(C(=O)NCC2(O)CCCN(C(C3C(=C)C3)=O)C2)c(F)cc(Cl)cc1Br CC1CN(C(C2(NC(=O)OC(C)(C)C)CC2)=O)CCC1NC(=O)CP(C)(C)=O C1(Cn2cc(CCOC)nn2)C(C2CC2)CCN1C(=O)Sc1ccccc1 CCC(CO)CN=c1[nH]c(=NC(C)CCSCc2ccccc2)c2ccccc2[nH]1 c1(OC)ccccc1C(c1ccccc1)NC(=O)N(C1CCN(O)C1=O)C(C)C N1(C(C2CCN(CC(C)C)C2)=O)CCC(F)C(NC(=O)CCCN(C)C(C)C)C1 CCCCCCCN(C1CCCCC1)C(c1cc(C)on1)=O c1(OC)cc(Cl)c(Cl)cc1C(c1nnnn1C(C)C(=O)OC)NC1(COC)CC1 c1(OC)cc(C(=O)NCCN2CCCOCC2)ccn1 c1(-n2cc(CN3C(C(=O)NCC)COCC3)nn2)cc(Br)cc(C)c1F CCN=c1[nH]c(C(=O)NCC2(F)CCN(C(=O)CN3CC(CC)C3)C2)cs1 CS(=O)(=O)c1ccc(C(=O)NC(CC2CCC2)CO)s1 c1(C(=O)NCC2CN(C(C(CCCC#C)C)=O)CC2O)ccc2c(c1)NC(=O)C2 N1(C(C(C)N2C(=O)C2)=O)CCC(CO)CC1C.C(=O)(CC(F)(F)F)OC Cc1[nH]cc(C(N2CCC(F)C(NC(c3c[nH]ccc3=N)=O)C2)=O)c(=O)c1Cl C(N=c1[nH]c(=N)[nH]c(=NCc2cc(-c3ccccc3)on2)[nH]1)C1CCN(CC)C1 c1(C(=O)NC2C(NC(C3CC(C)(C)C3)=O)CC2)cc2ccc(F)cc2[nH]1 C1(C#N)(C(N2CCC(c3c(CNC(CSC)=O)c[nH]n3)C2)=O)CCCOC1 CC1CCOC1CC(=O)NC1CCCC1CC(=O)N(C1CCOC1C)C1CC1 C12(COC)CC(CN1C(c1cccnc1)CO)C2 C1(C(C(=O)NCCN(C(C(C(C)C)SCC)=O)C(C)C)O)CCS(=O)(=O)CC1 C1(C2CCOCC2)(C(=O)NCCN(C(=O)COCc2ccccc2)CC)CC1 CC1(C)C(C(=O)NCCOCCOCCNC(=O)C(O)C2CCC2)CC1(F)F CCCCC(CC)CC(=O)NCC1(F)CCN(C(c2c(C(C)C)n[nH]c2C)=O)C1 N1(C(C2CCN(C(COC)=O)C2C)=O)CCC2(CC1)CSC2 c1(CN(C)C)cc(C(=O)N(CCCNC(=O)C(C)(F)c2ccccc2)C)ccn1 N1(C(CC2(C=C)CN(C(=O)OC(C)(C)C)C2)=O)CCOCC(O)C1 C=CCC(CC(C)C)C(=O)NCC(C)NC(C1(CC)CCCCO1)=O N1(C(C(CC)N2CCCC2=O)=O)CCC(C)(NC(c2cc(C3CC3)ncn2)=O)C1 C(=O)(CCCCC(=O)NCC1(O)CCN(C(C2CC(O)CN2C)=O)CC1)NC C=C(C)CC(C(=O)N1CC2CC1CC2O)NC(c1ccsc1Cl)=O C1(C(=O)OCc2c(C(=O)OC)[nH]nc2Br)C(C)CN(C(=O)OC(C)(C)C)CC1C C(=O)(CC(C(F)(F)F)NC(C1(C)CC(C)=NO1)=O)N(C(CC)C)C c1(C(=O)NC2CC(NC(C(C3CCCC3)OC)=O)C2)ccc2sc(O)nc2c1 c1(C(=O)NCC(C2CCN(C(C3CC3[N+](=O)[O-])=O)CC2)(C)O)cc(F)ccc1F C(=O)(C(S(C)(=O)=O)C1CC1)N.Cc1nc(C)n(CC2(CN)CC2)n1 N1(C(CS(CCC)(=O)=O)=O)CCN(C(c2cccc3oncc23)=O)C2COCC12 O=C1CCC(C(=O)NCCc2n[nH]cc2C(=O)NCC2(O)CCOC2)N1 C1(NC(C2CCS(=O)(=O)CC2)=O)CC2(C1)CC(CNC(C1CC3CCC1O3)=O)C2 C12(C(N(C3CN(C(Cc4c(C)ccs4)=O)CC3F)C)=O)CC3CC1(CO)CC3C2 c1(C(N(C(C(N2CCCC(OC)C2)=O)(C)C2CC2)C)=O)cc(=O)n(C)cn1 CC(C)C(CCN(C)C(C1CCOC1C)=O)NC(=O)CCc1cnn[nH]1 C1(NC(c2c(C)coc2)=O)CCC(C)(C)CC1CNC(c1ccnn1CCF)=O CCC(CN(C)C)C(=O)N(CC(=O)NC(c1ccn(C)n1)C)C S(=O)(=O)(c1cccc2c(C)ccnc12)N1c2ccc(OC)cc2CC(N)C1 c1(C(=O)NC(c2ccoc2)C)cc(CNC(=O)CSc2nc[nH]n2)[nH]n1 c1(N2CCCCC(CNC(C3N(CC)C(=O)CC3)=O)C2)nc(C)nc(C)c1C C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C)CNC(=O)C(F)Oc1ccc(Cl)c(F)c1)C c12cc(c(Br)cn1)CC(=O)O2.c1(OC)cccc(CCCCO)c1 C1(NC(=O)C(Cn2ccnn2)NC(=O)Cn2cc(CO)nn2)CCC(O)C1O Cc1ccnnc1C(=O)N(CCNC(=O)C(C1CC1)SNCc1ccccc1Cl)C C1(C(=O)NCCN(CCCC)C)OCCC1NC(C1CCC1C)=O C1(C(=O)NC2CCC(NC(c3cn(CCN(C)C)nn3)=O)C2)CC(S(C)(=O)=O)C1 CC1CC(NC(=O)Cc2cccnc2F)CCN1C(c1cc2sccc2[nH]1)=O C1(C(N2CC(CN(C)C(c3csc(-c4cccs4)n3)=O)C2)=O)CCCC1C1CC1 CC1Oc2c(C(=O)NOCC(C)(C)C3CC3)cccc2C1C N1(C(CCC(C)(C)C)=O)CC(NC(=O)CC2CC(F)(F)C2)C2(CCC2)C1 C(=O)(C(C)(C)CCC#N)N1CCCC(C(N2CCC(COCC)C2)=O)C1 C(=O)(CCCCCN(C)C(c1cocc1C)=O)N(CC#C)CC1CCCO1 c1(NC(CC2OCCN(C(C3C(C)C3)=O)C2)=O)nnc2n1CCCCC2 N1(C(C=CC=CC)=O)CC2CCC(C1)N(C(c1cn(C)nc1Cl)=O)C2 N1(C(CC(C=C)C)=O)CCN2CCN(C(=O)Cc3ccc(F)cc3Cl)CC2C1 c1(C(N(CCOCCCNC(c2c(C)nsc2)=O)C)=O)cnc2ccccn12 C12(C(=O)NCC3N(C(c4nn(C)c(C#N)c4)=O)CC3)CC3CC(C(=O)N1)C2C3 N1(C(C2C3(CCN(C(C(CC)(C)CC)=O)C3)C2)=O)CCC2(CCN(C)C2)C1 C(=O)(C1CCCn2cncc21)N1CCCC(O)(CNC(C2CCC(=C)CC2)=O)C1 Cc1nn(C2CC2)c(C)c1-c1ccc(C(=O)C(C)C)cc1 N1(C(C(N2CCNC2=O)C)=O)CCN(C(=O)C(C)(F)F)C(c2cccc(Cl)c2)C1 c1(C(=O)OCC)coc(CN(CC(C2CCCO2)O)C)n1 C1(CNC(c2c(CC)n[nH]c2)=O)(CO)CCN(C(=O)CC2CCC(=O)O2)CC1 N1(C(CC(C)(C)O)=O)CCc2c(C(N3CCNC(=O)C3)=O)cccc2C1 C12(NC(CCCCC=C)=O)CCCC1CN(C(=O)CCC1CCOC1)C2 c1(N2CCCC(C(F)(F)F)C2)ccc(NC(C2(CSC)CC2)=O)c2ccccc12 C1(CNC(CCCCC)=O)CCN(C(C2COC(=O)N2C)=O)CC1C C1(C2CC2)(NC(C2CSCN2C(=O)C#CC2CC2)=O)CCOC1 CN1CC(NC(C2CC(N(C)C(c3ccc(C4CC4)o3)=O)C2)=O)CC1(C)C N1(C(c2ccc(C)s2)=O)CCOCC1CCNC(C1CCN1C)=O C1(C(N2CC(CNC(c3c(CC)onc3)=O)C(C)C2)=O)CCc2nc(C)cn2C1 c1(C(N2CCN(C(C=CC)=O)C(CCO)C2)=O)ccc2c(O)ncnc2c1 N#Cc1c[nH]ccc1=NCC1(O)CCN(C(C2CCCC23CCC3)=O)C1 O=C(C#CC1CC1)NCC1(CNC(c2cc(CC3CC3)on2)=O)CC1(F)F C1(C(=O)NCC(C(C)(C)C)NC(Cn2c(C(C)C)ncc2)=O)CCCC2(CC2)C1 C(S(=O)c1ccccc1)c1onc(CCS(N)(=O)=O)n1 C(=O)(C(=O)N=c1[nH]n(CCCC#N)cc1C)N1CCC(N(CCC)C)CC1.O N1(c2c(OCC)cc(O)cc2)CCC2(CC1)CC2(C)C(=O)NCCCOC CC1CC(NC2CC2C2CC2c2nncn2C)CC(C)(C)C1 c1(C(=O)NC2CC(N(C)C(c3cc[nH]c3C3CCCC3)=O)C2)cc(F)cnc1O N1(C(C(C2CC2)OC)=O)CCC12CN(C(=O)COC1CCC1)C2 C1(CC(=O)NCC2CCCCC23CC3)COCCN(C(c2cc(CO)[nH]n2)=O)C1 C12(NC(=O)Cn3cncn3)COCCC1CN(C(=O)C1=CCS(=O)(=O)C1)C2 N1(C(C(C=C)(F)F)=O)CCCC2(C1)CN(C(=O)CCc1cncnc1)CCO2 c1(CN2CC3C(C(=O)Nc4c(C)cccc4Br)C3C2)cc2ccccc2o1 C#CC1(O)CC(C(=O)NCC2CCCN2C(=O)Cc2sc(SC3CC3)nc2C)C1 CC1(C)C(NC(c2ncc(CO)s2)=O)CC1CC(=O)NCCn1cccnc1=O c1(NC(c2ccsc2Cl)=O)ccc(C2(Nc3ncncc3F)CCC2)cc1 C1(n2cc(C(C(C)C)(C)C)nn2)CN(C(=O)CNC(=O)NC2CC2)CC1C C1(C(N(C)CCO)=O)CC2OCCC2N(C(c2ccc[nH]2)=O)C1 CCC(CC1CCCC1)C(=O)NC1CCCC1NC(c1c(C)nsc1N)=O C1(CNC(c2c(CC)non2)=O)CC(F)CN1C(=O)C(C)CC1CCCCC1 CC(C)(C)CC(=O)N1CCCCC1CCNc1cc(-c2cccc(Cl)c2)ncn1 C1(CC)CCCN(CC(=O)NC23COC(CNC4CC4c4ccccc4)(C2)C3)C1 C1(CNC(c2c(C)cco2)=O)CN(C(=O)C(O)CC(F)F)C2(CCC2)C1 Cc1cccc(F)c1C(=O)NCC1(O)CCN(C(c2coc(CO)c2)=O)C1 C1(C2(O)CCOC2)(C(=O)Nc2c(CC)ncc(C)c2)CC1 c1(C(C)C)cc(C(=O)N(CCC(=O)NC2C3COCC23)CCO)n(C)n1 c1(N(C(c2ccco2)C)CC2CC2CN)ccc(C(=O)O)cn1 N1(C(C=CC)=O)CC2COCC(C1)N2C(c1[nH]cnc1C(=O)O)=O c1(C(N(CCOCCNC(CSCCC)=O)C)=O)cc(C(C)=O)cn1C C1(NC(C(Cc2ccoc2)NC(C2CCC(C)(C)C2)=O)=O)CC2CC3C(C2)C13 N1(C(C2OCCN(C)C2)=O)C2CCC1CC(O)(CNC(=O)Cc1ccsn1)C2 N1(C(c2nc(C)oc2)=O)CCSCC1C(=O)Nc1ccc(-c2ccsc2)nc1 N1(C(c2nccc(C)c2)=O)CCCC(C(=O)NCCc2cc(C)n(C)n2)CC1 C(=O)(CC(C)C(C)(C)CC)NCCC1CN(C(C=CCCC=C(C)C)=O)C1 Cc1ncc(C(N2CCC(O)(CNC(=O)C(CO)N(C)C)C2)=O)cn1 N1(C(C2C(=C)C2)=O)CC(NC(=O)COc2ccc(Cl)c(C(F)(F)F)c2)C(C)(C)C1 Cc1cccc2nc[nH]c(=NCC(C)CNC(=O)C3=C(Cl)CC3)c12 c1(CN(C(c2ccnc(C)c2)C(=O)NC(CC)C)C)cn2cc(C)ccc2n1 c1(OCC(=O)NCC2N(C(C3N(CCOC)CCC3)=O)CC2)ccc(Cl)cc1 c1(NC(N2C(COC)CCOCC2)=O)cccc(C#Cc2ccccn2)c1 n1(CCC)nnnc1C(c1cc(OCC2CCCC2)ns1)NCCCOC(C)C N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CC2(C1)SCCC2NC(c1csnc1Cl)=O c1(C(N(CCC)CCNC(=O)CCC(C)C)=O)ncnc2c1c(Br)cn2C Cn1ncc([N+](=O)[O-])c1C(N1CCN(C(=O)C=CCF)C(C2CCC2)C1)=O c1(CC)ccc(F)c(C(N2CCN(C(=O)C(F)C(C)(F)F)CC2C)=O)c1 C1(NC(CC2C(C)CCO2)=O)CCN(C(=O)COCCN(C)C)CCC1CO N1(C(CC2C(NC(C3C(C)CC3)=O)CCC2)=O)CC(F)CC1CO C1(CC(N2CC(C)(CF)C2)=O)C2CCCC2N1C(=O)CCc1cnccn1 N1(C(C2CNC(=O)N2)=O)CC2(CCN(C(c3cnccc3Br)=O)C2)C1 C1(C(=O)Nc2ccc(COC)cc2)(CC)CCCN(C(=O)COCCF)C1 CC1CCC(NC(c2cscc2Cl)=O)CN1C(C1NC(=O)OC1C)=O N1C2CCC(C(=O)N3C(C)C3)C1CC2.C(C(=O)C)SCC=C.CC(C)C.NCPBr N1(C(CC2CNC(=O)O2)=O)CC2(CCCC2)C1C(=O)NC1CCC([N+](=O)[O-])CC1 n1(CC)nc(C)cc1C(=O)NC1CCCCC1C(=O)NC1(CCO)CCCCC1 C=C1CCC(CNC(=O)CCN(CCOC)C(c2cnn(C(C)C)n2)=O)CC1 c1(C(N(CC(N)=O)CC)=O)ccc(SCc2conc2C2CCCO2)cc1 N#Cc1cncc(CNC(=O)CCC2CCCN2C(C2CCC(O)C2)=O)c1 c1(CNC(N(C23CC4CC(CC(C4)C2)C3)C)=O)ccc2c(c1)COC(=O)N2 C1(CCNC(c2cc(C)[nH]n2)=O)CCN(C(C2C=CC=CC=C2)=O)CC1 C1(C(=O)NCC2(O)CCCN(C(c3ccc(O)cn3)=O)C2)CC2COCC(C1)C2 N1(C(c2nc(C)[nH]n2)C)CC2C(NC(=O)CCCc3ccc(C)s3)C2C1 C1(C(=O)NC(C2CCCC2)C#C)CCCCC1NC(=O)C=C(C)c1ccco1 c1(C(=O)NC2C(C)N(C(=O)C3=COCC3)CC2)cc(Cl)ccc1-n1ccnc1 N1(C(c2c(OC)ncnc2)=O)CC2CN(C(c3cc4sccc4s3)=O)CC2C1 N1(C(C(C(C)OC)N(C)C)=O)CC2(C1)OCCCC2NC(=O)CCc1cn[nH]c1 Cc1ccc(C#N)cc1C(=O)NC1CCCC1NC(=O)C(C(C)C)NC=O N1(S(=O)(=O)c2cn[nH]c2)CCC2CN(c3ncnn4cc(Br)cc34)CC2C1 c1(CNC(c2cccnn2)=O)ccc(CNC(=O)C(O)CN2CCOCC2)cc1 C1(C(=O)NC2C(C)CN(C(=O)C(C)O)C2)CNC(=O)CC1(C)C C1(NC(=O)CCc2cc[nH]n2)CCN(C(C2CC3C=CC2C3)=O)CC12CCC2 c1(OC)ccc(C(=O)NC2CCCC(NC(=O)CN3CCC3C)CC2)cc1SC N1(C(CN(c2c3c(nn2C)CCC3)C)=O)CC(NC(OC(F)(F)F)=O)CC(C)(C)C1 c1(C(=O)NCCC(=C)CNC(C2(C(=O)OC)CC=CC2)=O)ncncc1C Cc1ccc(F)cc1C(F)(F)C(=O)NC(CNC(c1c(Cl)cncc1Cl)=O)CO C(=O)(C(C(=O)NCC1CC(C(=O)Nc2ccccc2C(C)C)CO1)OC)OC N1(C(C(C)c2ncco2)=O)CCCC(F)(CNC(c2cc(O)ncn2)=O)C1 CC(CC(=O)N1CCC2(CC(C(N3CCC4(C=CCO4)C3)=O)C2)C1)CC(C)(C)C c1(C(=O)NC2CC3N(C(c4c(CC)cno4)=O)C(CC3)C2)c(F)cccc1[N+](=O)[O-] C1(C(=O)NCC(C(C)C)(C)NC(=O)C(Cl)=CCl)CC12CCOc1ccc(F)cc12 N1(C(C(CC)OC)=O)CC(NC(c2c[nH]c(Br)c2)=O)CC12CCCCCC2 CCS(=O)CC(=O)NC1CN(C(=O)C=Cc2nc(C)cs2)CC1SC c1(C(=O)NCC2CCC(C)N(C(c3cnccc3Cl)=O)C2)cccc(N=[N+]=[N-])c1 C(=O)(C(F)C(C)C(F)(F)F)N(CCCCCNC(c1ccnc(OC)c1F)=O)C c1(NC(N(C)CC)=O)ccc(S(=O)(=O)N2CCCC(COC)C2)cc1 CCC(C)(C#N)C(=O)NC(C)(C)CC(=O)NCC1CC(=O)N(CC)C1 C1(C)(CNCC(C)C)CS(=O)(=O)CCO1 C12(c3n(C)ncc3)CCC(C1)C2C(N1CCC(NC(C23CC(CO)(C2)C3)=O)C1)=O N1(C(C(C)(F)F)=O)CCC2(CCCC2NC(=O)CC2CC=CCC2)CC1 CC(CCNC(=O)COc1ccc(F)cn1)CCNC(=O)Cc1cnccc1Cl c1(CN(CCC)CCNC(C2CC2(F)F)=O)nnn(C(C)C)n1 CC1CN(CCF)CCN1CC(=O)Nc1coc(Br)c1 CC(C)CC(C)C(=O)NCC(CC(F)(F)F)NC(=O)CC1CCC(C)(C)O1 c1(C(N(CC(CNC(CN(C)CC)=O)C)C)=O)ccccc1 c1(CC)nonc1C(=O)NC1CCC(CNC(=O)C(CC)Oc2ccccc2)C1 N1(C(CS(CCOC)(=O)=O)=O)CC2CC(C1)CN(C(C1CCC3CC3CC1)=O)C2 c1(C(=O)NCC2CCN(C(C(CC)OCC)=O)C2)cccc[n+]1[O-] C1(c2n(CC)nnn2)(NCCCOCC)CCC2CCCC2C1 Cc1nc2cncc(C(=O)NCCCCNC(=O)C(C)OCC3CCCO3)c2[nH]1 c1(CC(=O)NCC(N2CCOC(CNC(C3CCCC3)=O)C2)=O)ccccc1Br C1(CNC(c2c(C#C)c[nH]n2)=O)CN(C)CCN1C(=O)Cn1ccc(C(F)F)n1 c1(C(=O)NCC(CNC(CC(COC)(C)C)=O)O)nc2c(s1)CCCC2 C1(C(N2CC3CCN(C(c4cnsn4)=O)CC3C2)=O)CC(c2ccncc2)=NO1 CC(C)CC(O)C(=O)N1CCN(C(=O)COC2CCCCC2)C(c2cn[nH]c2)C1 N1(C(=O)CC2(O)CCCC2)CC2CC(C1)C2N=c1[nH]c(C(F)(F)F)nc2[nH]ccc12 c1(CC(=O)NC2CCN(C(C3CCC34CCC4)=O)CC2O)ccnc(Cl)c1F CC(CC(=O)N(C(C)CCNC(=O)C1CC1)C)C1CC1 C12(C(=O)NC(C(=O)OC)C(C)C)CCC(CN(C(C3CNC(=O)N3)=O)C1)C2 N1(C(C2(CC#C)CCOC2)=O)CC(NC(c2cn(C)cc2C)=O)C(O)C1 N1(C(c2ccc(CCCC)cc2)=O)CC(CNC(C2(COC)CC2)=O)C2(CC2)C1 c1(C(=O)NC(CNC(C2(CC)CCOC2)=O)CC)sc2ccc(C#N)cc2c1C c1(-n2cc(C3(F)CCN(C(CCN=[N+]=[N-])=O)C3)nn2)c(Cl)cccc1Cl N1(C(C#CC(C)C)=O)CCC2CCCC12C(=O)NCc1nnn(C)n1 Cc1c(CN2CCCC2(C)C(=O)NC(c2ccccn2)CO)cncc1Br c1(C(N2CCC(C(C)NC(=O)Cn3cccn3)C2)=O)cc2ccccc2cc1O N1(C(C(C2CCOCC2)OC)=O)CCCC(NC(c2cnnc(O)c2)=O)C1 CCC(O)C(F)(F)C(=O)NCC12CC(CO1)N(C(c1ncc(Cl)cc1Cl)=O)C2 C1(C(=O)NCc2ncn(C)c2)CCC(NCc2cccnc2F)CC1 C12(CCCN(C(=O)COC(C)=O)C1)C(=O)NC2.C(C)(C(C)C)OCC N1(C(CC2CNC(=O)O2)=O)C2CCC1CC(NC(C1CCOC(=O)CC1)=O)C2 c1(C(N2C(COC)CN(C(=O)C3=CCC3)CC2)=O)ccc(Br)c(Cl)c1F C1(C(N2CCSCC2)=O)CCC(n2cc(-c3cscn3)nn2)CC1 N1(S(=O)(=O)CC23CCCC2C3(F)F)CC2(CCCCC2)C1 N1(C(COCCCCCC)=O)CCC2(CC1)CC2NC(=O)C(C)CC(F)(F)F CC(CCCC(=O)N1CCCCC1c1n[nH]cc1CO)c1ccccc1 c1(-n2c(CNCCC(=C)CO)nnn2)cc(C)ccc1OCCCC C1(CC)CN(C(=O)Cc2cc(COC)on2)CCN1C(C1CC(C(C)C)=NO1)=O C(CN=c1[nH]c(Cl)ncc1C(F)(F)F)C1N(C(C(CC)C)=O)CCCC1 C1(C)(C(=O)NCC2(C(C)NC(c3cc(O)n(C)n3)=O)CC2)CCCC1(F)F c1(C(=O)NC(C(CO)NC(C(CC)(C)O)=O)C)cnc(OC)cc1C(F)F Cc1ccc(C(=O)NC(C)CC(C)NC(=O)CCCC(N)=O)cc1S(C)(=O)=O C1(NC(C(=Cc2ccco2)C)=O)CCCC(CN(C)C(C2CC(C)(O)C2)=O)C1 C1(NC(c2c(C)c[nH]n2)=O)CC2CC1CN(C(C1CCC(C)CC1)=O)C2 C1(CNC(C2(c3ccccc3)CC2)=O)(NC(C2CC3(CCC3)C2)=O)CC(F)(F)C1 C1(C(C)(C)NC(C(C)N2CCCC2)=O)CCCN1C(C1CCN1C)=O C(C(C)CC(C)C)N1CC(CC=C)(NC(C2CCCN2C2CC2)=O)C1 C1(NC(c2cccc3c2CCC3)=O)CCC12CCN(C(C1CCSCC1)=O)CC2 N1(C(C(CN(C)C)O)=O)CCC(C)(C)C1CC(N1CCCC1CN=[N+]=[N-])=O c1(CN2CCCC(N(C(=O)CCC3CCC3)C)C2)cccc(F)c1F N1(C(c2csc3ncnc(O)c23)=O)C2CCC1c1cc([N+](=O)[O-])cnc1C2 C(C(C)(C)C(=O)NC(C1CCN(C(=O)CCCNC(C)=O)CC1)C(C)C)OC C(=O)(C(=O)C(F)(F)F)NCC(c1cccc(Cl)c1F)(C)C c1(CC)cccc(C(N2CCC(C(C)CNC(=O)CC(F)(F)CC)CC2)=O)c1N c1(CCC(=O)NCC2CCCN2C(=O)C(F)n2ccnc2)cccc(F)c1 CCC1=NOC(C(=O)N(C(CNC(C2(C3CCC3)CC2)=O)C2CC2)C)C1 n1(CCC)ccc(CNC(c2ccnn2C)c2nnnn2C(C)C)c1 Cc1cc2[nH]c(C(=O)NC3CN(C(=O)CC4CCCC5(CCC5)O4)C3)cc2s1 N1(C(C2(C)C(C)OC(C)(C)O2)=O)CC23CCCCC2(C1)CN(C(=O)CCCF)C3 CC(C)CC(F)C(=O)N(CC(O)CN(C)C(c1cnc(O)c(Br)c1)=O)C C1(C(N2CC3(CN(C(C4OCC(C)(C)OC4)=O)C3)C2)=O)COc2ccccc2O1 c1(C(=O)NC(CC)CN(C(=O)CC2CC(C(F)F)C2)C)cc2scc(C)c2[nH]1 N1(C(c2c(OCC)cccn2)=O)CCC(NC(=O)CN2CC(=O)NC2=O)C(F)C1 N1(C(C(C2CCCC2)NC(C2=C(C)OCCS2)=O)=O)CCC2CN(C)CC2C1 C1(NC(c2c(C)coc2)=O)CCN(C(c2ccc(CN=[N+]=[N-])cc2)=O)C(C)C1 c1(CC)nc2sc(C)cn2c1C(=O)N(CC(C)NC(=O)C(CC)n1ccnc1)C c1(Cn2cc(CCC(CC)O)nn2)ccc(C(=O)N(C)CC2CCCOC2)nc1 C=CC(F)(F)C(=O)NCC(CCCC)NC(c1cnc(C(C)C)o1)=O C1(C(=O)NC(CC)CNC(=O)C(C2CCCCCC2)F)CC(=O)C12CCCC2 N1(C(c2c(C)nn(C)c2C)=O)CCC(O)C2CCCCC12 N1(C(C2(CC)CC2)=O)CC2CCC1CC2NC(C1(C2CCC2)CCC1)=O C1(CNC(C(CC)O)=O)N(C(=O)CCc2nncn2C)CCC1(C)C C(c1cncc(O)c1)=CC(=O)NCCN(C(CN1CCC(C)C1)=O)C(C)C CC(CC(N)=O)C(=O)NC1CC(C)CN(C(=O)Cc2csc(Cl)c2)C1 c1(CC(N2CCC(N(C(C3C(F)(F)C34CC4)=O)CC)C2)=O)cn2ccccc2n1 N1(C(CCC(CCC)CC)=O)CC=C(C(C)(C)C(=O)NC(c2ccccn2)C)C1 c1(C(=O)NC2C3(CC(NC(=O)CCc4cccs4)C3)C2)ncn2c1CCC2 O(NC(=O)CC1CCC(NC(C2CCSCC2)=O)C1)CCCCC C(=O)(C1=C(C#N)CCC1)NCC1C(NC(c2c(C)n(C)nn2)=O)C1 CCCCCCC(C)CC(=O)OCC(C)(C)C.C12(F)CCCN(C1)CCONC2=O CC#CCCC(=O)NC1(CF)CCN(C(=O)C(C)OCCN(C)C)C1 CC1CCc2[nH]nc(C(=O)NC(C)C(=O)N3CC(Cc4ccoc4)C3)c2C1 C(=O)(CCCCCC(C)(C)C)N1CCCC(CN(C(c2c(C)ccnn2)=O)C)C1 CC(C)C(C)(C)C(=O)N1CCC(CNC(=O)C(c2ccc(Cl)cc2)C)C1 C(=O)(CC(C)(C(F)F)N(C)C)NC(C)CC(C)NC(=O)CC(C)(C)C c1(C(=O)NC2CCOCC2NC(C2CSC2)=O)cc(F)c(Cl)cc1Cl C1(CNC(C2C(NC(CCSC)=O)CCO2)=O)CCC(=O)NC1 N1(C(CCc2ccc(C)s2)=O)CC(CNC(=O)C(F)C2CCC2)CC12CCC2 N1(C(C(CCC)N(C)C)=O)CCC2(C1)CN(C(=O)CC1CC(F)(F)C1(F)F)C2 Cc1nn(C(C)C)cc1C(=O)NC1(C)CN(C(=O)CC2CCCO2)C1 N1(C(C(C)n2ccnn2)=O)CC(C2CC2)(C(=O)NCCCS(C)=O)C1 c1(C(=O)NC(C(=O)N(CCC#C)CCO)CCN(C)C)cccc2[nH]ncc12 c1(C(N(C(CC)CC(=O)NC(c2cccnc2)CC)C)=O)cc([N+](=O)[O-])c[nH]1 C(C)(C)(CCCC(=O)NC1CC(CF)C1)NC(C(N1CC(C)C1)C)=O C#CCCCCCC(=O)NCC(C1CCC1)NC(c1cccc(C(N)=O)c1F)=O c1(SC(C)C)n[nH]c2ccc(C(=O)NC3CCN(C(=O)OC(C)(C)C)CC3)cc12 C1(C(=O)NC(C(N2CCC(C)C2)=O)(C)C)CC2OC1C1CC21 C#CCCCCCCC(=O)NCCC1=CCN(C(C2CCNC(=O)C2)=O)CC1 C(c1cc(Br)cs1)=CC(=O)NC(C(C)NC(=O)C=Cc1ncc[nH]1)CO CC1OC2CCC1(C(=O)NCC1CC(C(=O)NCCCC3CCC3)=NO1)C2 C1(N(C(c2c(C)nsc2C)=O)C)CCCN(C(=O)Cc2cccnc2)CC1 C1(CNC(c2cn(C)nc2C(F)F)=O)CCN(C(=O)CCc2ncc[nH]2)C12CC2 c1(C(=O)NC(C2(O)CCN(C(C(COC)(F)F)=O)C2)C)ccnc2c1ccn2C N1(C(C2CCN(CCC#C)CC2)=O)CCCC(NC(=O)C=NOC)C(F)C1 N1(C(CC2C(CN)C2)=O)CCC(C)(NC(=O)Cn2cncn2)C1 N1(C(C2CC(C#N)C2)=O)CC2CCCN(C(c3ncc[nH]c3=O)=O)C2C1 C1(C)(C(=O)NC2CC(CCC(=O)N(CC(C)(C)O)CC(N)=O)C2)CCCS1 CCC(CC(=O)NCC(c1ccccc1)NC(c1nc(O)c(C)s1)=O)CC(C)C c1(OC)cc(F)ccc1CCNC(=O)Nc1c[nH]nc1-c1cnccn1 N1(C(c2cnc(C)nc2)=O)C2CCC1CC(NC(C1CC3(CC3)C1)=O)C2 c1(-n2c(C(C(CC)C)OC)nc(-c3cncnc3)n2)ccc(Br)c(C)c1 c1(C(=O)NCCCNC(C(C)N(CC(F)(F)F)C)=O)cnc(OC2CCC2)cn1 C1(CC)CC(C)CN(C(c2cn(C)c(-c3ccccn3)n2)=O)C1 CCN=c1[nH]cc(C(=O)NCCCCC(C)NC(=O)Cn2cc(C(C)O)nn2)s1 CCCCC(CNC(c1cnsn1)=O)NC(=O)CC1CCOC1 N1(C(CN(C(CCCCSC)=O)C2CCC2)=O)CCN(C)C(C(C)C)C1 N1(C(C2C(C)=C2)=O)CCC(C)C1CNC(=O)C(CN(C)C)c1ccccc1 C=CCC(C(=O)NC(c1cccc(Cl)c1)CNC(C1(CC)COC1)=O)NC(C)=O c1(-c2nnc(CC(C)(C)C)o2)nc(=NC(=O)CC2CCS(=O)(=O)C2)s[nH]1 C(=O)(C1=CCCN(C(=O)CCc2nccn2C)C1)NC(CCCOC)C c1(NC(C(c2sc(Cl)cc2Br)N(CC(F)(F)CC)CC)=O)ccc(F)cc1 C1(C(=O)NCC(C)NC(c2ccc(C(N)=O)[nH]2)=O)CN(C)CC1C(F)(F)F N1(Cc2c(C)cccc2O)CC2CN(c3nccc(-c4cccnc4)n3)CC2C1 N1(C(C)=O)CCN(CC(=O)Nc2nc(C(C)C)cs2)CC1.C12CCCN1C2=O c1(C(=O)NC2C3CCN(C(C(C)N(C(C)=O)C)=O)C3C2)cc(F)c(C)cc1Cl CC(CCC(=O)N1CCCCCC1)n1cc(CCN(C)S(N)(=O)=O)nn1 N1(C(C=C(C)Cl)=O)CCC(NC(c2ccnnc2S)=O)C1C1CC1 N1(C(c2cnc(COC)s2)=O)CCC(CNC(=O)CN2CCCC2=O)C1(C)C N1(C(C2CC(SC)C2)=O)CC(C)CCC1CNC(c1cc(Br)c(C)o1)=O C#CCC(C(=O)N1CC(C(=O)N(c2ccccc2O)CC)C(CC)C1)C1CC1 CCCCCCCCC(C)CC(=O)NCC1CC(NC(=O)CCC(C)CC)CC1 C1(CNC(Cc2nnc(C)s2)=O)CC(F)CN1C(=O)C(c1ccccc1)C C(C)(CO)(C(=O)N1CCC(NC(=O)CNS(=O)(=O)N(C)C)CC1)OC C=CCC(C)(CC=C)NC(=O)CCC1CCCN(C(=O)CCCOCCC)C1 c1(OCC(C2CCCO2)C)ccnc(C(C)(C)CNc2cc(O)n(C)n2)c1 c1(CCC(=O)NCC2(C3CCCCN3C(C3CC=CC3)=O)CC2)cccnc1F c1(CNC(=O)Cc2ccsn2)nc(CNC(=O)CN2CCCCC2=O)cc(O)n1 N1(CC(=O)N(C(CN(c2nnnn2C(C)C)C(=O)OC)C)C)C(=O)CCC1=O C1(C(N2CC(NC(C3C4(CC(C)(C)C4)C3)=O)C2)=O)CS(=O)(=O)CC12CC2 C(=O)(C#CC1CCCO1)Nc1cccc(CNC(Cc2ccc(OC)nc2)=O)c1 C(=O)(CC(O)CNC(N1CCCC1)=O)Nc1c(C(=O)OC)occ1 CP(C)(=O)c1ccc(C(N2CCC(c3nc4c([nH]3)COCC4)CC2)=O)cc1 N1(C(C2C(C)C2)=O)CCC(NC(=O)CCCN(C)C)C12CCC2 C(=O)(CCC(F)F)NC(CC=C)CNC(=O)C(C)Sc1nncn1C Cc1ccc(F)c(NC(=O)C(=O)N(C(C)C(N)=O)C2CC2)c1 N1(C(c2csc(Cl)c2)=O)CCC(NC(C23CC(CO2)C3)=O)C12CCC2 C1(NC(c2cscn2)=O)CN(C(c2cc(Cl)cnc2O)=O)CC12CCCC2 C12(NC(COCCC)=O)CCC(CC1)N(C(c1cncc(F)c1Cl)=O)C2 n1(CC(=O)NCC(N(C(C2CC(SC)C2)=O)C)C2CC2)cnc(C#N)n1 N1(C(c2cc(OC)nc(C)c2)=O)CCC(NC(c2cc(C)oc2C)=O)C(C)(C)C1 c1(-n2cc(CC(COC)O)nn2)cccc(NC(=O)C(CC)OCCOC)c1 C1(N(C(c2cc(C3CC3)ccn2)=O)CC)CCCN(C(=O)CCC2OCCO2)C1 c1(N(C)C)ccc(CNC2CC2C(=O)NC2C3CNC2C3)cc1 c1(C(N2C(C)(CNC(=O)CCC3CC3(F)F)CCC2)=O)ccc2c(c1)CCCS2 c1(C(=O)NC(C2OCCN(C(C(C)=C(C)C)=O)C2)C)cc(C)cc(C)c1C Cc1cc(C(=O)NC(CNC(c2ccc(-c3ncc[nH]3)nc2)=O)CO)ncc1F c1(C(=O)NC(CN(C(=O)CC2CC(F)C2)CC)C)cccc(-n2cccc2)c1 n1(CC(=O)N(C(C)C)C(C2CCC2)C)cc(CN(C)C)nn1 N1(C(C(C)N(C)C)=O)CC(C2CC2)(C(N2CCC(N(C)C)C(C)C2)=O)C1 c1(C(=O)NC23C(CN(C(c4c(C)cnnc4)=O)C2)CC3)ccc2[nH]nc(O)c2c1 C1(NC(C(C)n2cncn2)=O)CCN(C(=O)CSCCc2ccccc2)C1C Cc1[nH]nc(C(=O)NCC23CCCC2N(C(c2cncn2C)=O)CC3)c1[N+](=O)[O-] c1(C(C(=O)NC2CCOC2)N(C)Cc2cn[nH]c2)cn(C)nn1 Cc1nc(=NC2CCC3CN(C(c4cc(CN(C)C)c[nH]4)=O)CC23)s[nH]1 C12(c3n(C)ncc3)CCCCC1CN(CC1(c3cc4nn[nH]c4cc3F)CC1)C2 c1(C(=O)NC(C2CCOC2)CNC(C=CCC)=O)cc2oc(C)c(C)c2[nH]1 C(=O)(CCS(C)(=O)=O)N1CCC(C(=O)NC(CC=C)CC)(CC)C1 C1(NC(C(CCN(C)C)O)=O)CC2CC(NC(=O)CCOCC3CCCO3)CC12 CCCN=C(NCC1(S(C)(=O)=O)CC1)N1CCC(CC2CCCC2)C1 C1(NC(c2ccc(C(=O)O)o2)=O)C2CCC1CN(C(c1cc(Br)ncc1F)=O)C2 N1(C(c2cc(CC)on2)=O)CCCC2CCN(C(C3(c4cccs4)CC3)=O)CC12 C1(CC(=O)NC(CC)CNC(=O)CCc2ccccc2C)CN2CCN1CC2 Cc1cccc(-n2cc(-c3ccnc(Br)c3)nn2)c1 C1(NC(CC2(OC)CCOCC2)=O)C2CCN(C(=O)C(F)=CCCF)CCC12 c1(NC(CC2N(c3ncc(OC)cn3)CCOC2)=O)cc(Br)cc2cc[nH]c12 N1(C(C(C)C#N)=O)CCCCC1CNC(C1CC(OC(F)(F)F)C1)=O N1(C(C2C(CC)C2)=O)CCCC1C(C)(C)C(=O)NCCC(=O)NC(N)=O N1(C(CC=CC)=O)CCC(NC(c2nnn(-c3ccccc3)c2C)=O)CC1 c12c(C)nn(c1C)CCC(=O)NOCC(=O)Nc1cn-2nn1.N(C)(C(C)C)CC N1(CC(=O)N(CC(N2CC(CN)C2)=O)Cc2ccccc2F)CCC(C)CC1.CC c1(SCC(=O)NCC2C(NC(C(C)OCOC)=O)CCC2)ccsc1[N+](=O)[O-] c1(C(N2CCC(CCNC(c3cc(C)nn3C)=O)CC2)=O)ccc2cnnn2c1 c1(OC)ccc(C)c(C(=O)N(CC(C)O)CCNC(=O)CCc2cnccn2)n1 c1(C(N2CC3CC(C2)N(C(c2cscc2C(F)F)=O)C3)=O)ccc2n[nH]cc2n1 N1(C(c2ccn(CC(F)F)n2)=O)CC(N=c2[nH]c3ncc(Cl)cc3s2)C1 C1(NC(c2c(CCC)nco2)=O)CN(C(=O)CS(=O)CC)CCC12CCOCC2 C(=O)(C(F)(F)C(O)C(C)C)NCC(CC)NC(=O)Cc1cc(O)nnc1O C1(NC(C(C)CCO)=O)CCC2CN(C(c3ccc(C4CC4)s3)=O)CC2C1 C1(C)(CNC(C2(CC(C)C)CCCC2)=O)CCN(C(c2c[nH]nc2C2CC2)=O)C1 C(=O)(C(O)CCN(C)C)N(C(C)CNC(C1CCCC1C)=O)C c1(C(=O)OC)cccc2c1CCC2NC(=O)C(=O)NCCSCc1cccnc1 C(C1c2ccsc2CCN1C(=O)C=CCO)NC(C(CN(C)C)(C)C)=O c1(OC)ccc(C(=O)NC2CC2NC(=O)CC(C)c2ccco2)cc1O C1(CNC(c2ccc(CCC)[nH]2)=O)C(C)CCN1C(c1coc(Cl)n1)=O c1(C(=O)NC2CN(C(c3cncc(N)n3)=O)CC2CO)cccc2c1CCCC2 c1(CCC(=O)NCCC(=C)CNC(=O)C#CC2CCCC2)n[nH]c2c1CCCC2 c1(CC(=O)NCC(C)NC(C2(COC)CCCO2)=O)cccc(SC)c1 Cc1nc2cc(NC(C3(C)CCN3C(C3CCCN(C)C3)=O)=O)ccc2o1 N1(C(CC(C)F)=O)CCCC(C2CN(C(c3conc3C(C)(C)C)=O)C2)C1 c1(C(C(=O)NCCC2(OC)CN(C(C3(F)CC=CC3)=O)C2)C)ccccc1C CCCC(CNC(c1cnncc1OC)=O)C(=O)N1CC=C(CO)CC1 CC#CCC(C(=O)NCCN1CCOCC1)NC(c1ncc[nH]1)=O CC(C)(C(=O)N1CCCCO1)C1CCN(C(c2cccc(=O)o2)=O)C1 n1(CCOC)ccc(=NC(=O)C2CCCN2C(=O)CC2OCCC2(C)C)[nH]1 n1(CC)nc(C)c(C(=O)NCC(Cc2ccccc2)NC(=O)C(C)C#N)c1C N1(C(=O)Nc2cncc(C)c2)CCCS(=O)(=O)CC1c1cnn(C)c1 C12(C(N)=O)CCCC1(C(=O)NC1CCC(CNC(c3ccoc3Cl)=O)CC1)C2 C=C(C)CC(C(=O)NOCCCN(C)C1CC1)NC(=O)CCC1OCCO1 C1(C)(NC(COCCCC)=O)CCN(C(c2ccc(C(N)=O)nc2)=O)CC1 c1(C(N2CCC(NC(Cn3nnc(C)n3)=O)C(C)C2)=O)n[nH]c2ccc(Cl)cc12 CC(C)(C(=O)NCS(=O)(=O)CCC1CCCC1)C(F)(F)F C1(C)(C(=O)NCCN(C(=O)C=NOC)CCOC)CC(OC)CN1C c1(C(=O)NCC2(NC(C(C)CCN(C)C)=O)CCCC2)cc(F)c(N)cc1F c1(C(=O)NCCC(CNC(C(C(CC)O)C)=O)(C)C)c[nH]c2nccc-2c1 Cc1sc(O)nc1C(=O)NC(C)CNC(C1CCC(O)(c2ccc(Br)cc2)C1)=O c1(OC)ccc(CCCC(=O)Nc2ccccc2SC(C)(C)C)c(Br)c1 N1(C(c2sc(C)c(O)n2)=O)CC2(C1)C(NC(=O)C(C)CN(C)C)CCS2(=O)=O c1(OCC)ccc(C)cc1C(=O)NCC(C)CNC(=O)Cc1ncccc1C N1(C(CCC#N)=O)C2CCC(C2)C1CNC(=O)CSC1CC1 CC(C)CC(C(=O)NC1C2CN(C(C3CCCN3C3CC3)=O)CC12)N(C)C c1(NC(C(C)=CC)=O)cccc(C(=O)NC2(C(F)F)CC(C(=O)OCC)C2)c1 c1(CN2C(CNC(c3ccc(C)cc3)=O)CC2)cccc(F)c1I N1(C(C(CC)(C)CNC(c2cn(C)c(=O)cn2)=O)=O)CCC(C)C(F)(F)C1 c1(C(N2CCN(C(C(CC)(C)O)=O)C3C2C3)=O)cc(Br)c(O)cc1O N1(C(COCC=C)=O)CC(CO)(CNC(=O)CSCc2cccnc2)C1 C1(C(=O)NCC2C(C)CCN2C(=O)C2=CCCCO2)CC2(CCOCC2)CO1 c1(C(N2CC(C)C(C(N3CC(c4ncc[nH]4)C3)=O)C2)=O)cccc(O)c1F CCC(CC)C(C)(F)CN(CC(C(C)(C)C)ON)C=O Cc1cc(S(=O)(=O)NC(C2CCOCC2)CCO)n(C(C)C)n1 c1(CC(=O)N(C)CCNC(C2(c3cccs3)CC2)=O)ccc([N+](=O)[O-])cc1F CC(C(=O)NCC1CCC1C(=O)NCCCc1ccccc1)C(F)(F)F N1(C(C)C)CCOC(C(=O)NC2CC23CC(NC(=O)COCCF)C3)C1 C(=O)(CCCCCCNC(c1cn[nH]c1)=O)N1C(COCC#C)CCCC1 C1(C)(CC)CC(NC(=O)COC(C)(C)CC)CN1C(=O)COc1ccc(C)cc1 c1(C(=O)NCCN(C(c2cc(CC)c(CC)o2)=O)C)cc(C)c(F)cc1Br C(=O)(CC(O)CC(C)(C)C)N1CCCC(N(C(=O)C=Cc2ncco2)C)C1 Cc1cc(C(N2CCC(CNC(=O)C3=CCCC3)CC2)=O)c2n[nH]cc2c1 c1(C(=O)NCCCC2N(C(CCCC#C)=O)CCCC2)cc2c(s1)CCC2=O C1(NC(CC(C)C)=O)CC(F)CN(C(c2cnn(C(C)(C)C)c2N)=O)C1 Cc1nc2ccc(C(=O)NC3CC4CC(C3)N(C(=O)C(N)=O)C4)cc2nc1C CC(C)CC(O)C(=O)NC1C=CCC(C(=O)N(CC(c2nn[nH]n2)C)C)C1 N1(C(c2c(C)n(C)nn2)=O)CCC2CN(C(c3cc(O)cc(Cl)c3Cl)=O)CCC12 C1(NC(C2(CC)CCC2)=O)(CF)CCN(C(=O)C(C)COC(C)=O)C1 C1(C)(C(=O)NCC(C)CNC(=O)C(C)n2ccnc2)CC1(Cl)Cl C1(C(=O)NC2(C(C)O)CC2)CC2C=CC1N(C(c1c[nH]c(C#N)c1)=O)C2 c1(NC(C(C(C)C)F)=O)ccc(OCc2cc[nH]n2)cc1C(F)(F)F C1(NC(c2c(C)nc(-c3ccccc3)s2)=O)CCN(C(=O)C(C)O)CC12CCC2 O=C(C1=CCCSC1)NC1CC2CC(NC(=O)CC3CC=CC3)C2C1 c1(C(C)=O)ccsc1NC(C1CCN(C(=O)Cc2cccnc2)C1)=O CCCC(C(=O)NC1CC(F)(CNC(C2(O)CC2(C)C)=O)C1)OC Cc1cccnc1CCC(=O)NC(C)(CNC(=O)CC(=O)OC(C)(C)C)C1CC1 c1(OC)cc(C(N2CCC(NC(=O)CCc3nc[nH]n3)C2)=O)c(N)c(Br)c1 N1(C(CC(=C)C)=O)CCC2(CC1)CC(CNC(=O)CSc1cnn(C)c1)C2 N1(C(=O)CCC(F)F)CC23CCCCC2(C1)CN(C(=O)CCC1CCCO1)C3 O=NN1CCCCC1C(N1CC2CCC2(CNC(=O)CCC2CCC2)C1)=O CC(=O)CCCCC(=O)N1CCOCC1CNC(=O)C=Cc1ncc(C)[nH]1 c1(C(=O)NC2CCN(C(c3c(C)cc[nH]3)=O)C2(C)C)ccc2c(n1)CCC2 C(=O)(C1=C(Cl)CCOC1)NC1C(C)CN(CC(O)CCc2ccccc2)C1 c1(CC(=O)NC(C2CCCCC2)CNC(CC(CC)C)=O)cccc(F)c1NC C(=O)(C(CC)CC(F)F)NC(CC)CN(C(=O)Cn1ncc(O)nc1=O)C C=CCCC(C)(C)C(=O)NC1CC1NC(C1CCOCC1)=O.C12CCN1C2=O c1(C(=O)NC2CCN(C(C(C)(CO)OC)=O)C2)oc2c(C)ccc(C)c2c1C C#CC(CNC(=O)CC(CC)NC(C1(C(N)=O)CC1)=O)C(C)C C1(CC)CN(C(=O)C(Cc2ccoc2)NC(c2cnncc2NC)=O)CC1O CC(N=c1[nH]c(N2CC(F)(F)C(F)(F)C2)nc2c1CCC2)c1ccc(Cl)c(Cl)c1 CC1(C)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)C1C(N1CCC2(CCC2)C1)=O N1(C(C(=O)NC(c2cn(CO)nc2)C)=O)CC(CNC(=O)OC(C)(C)C)C(C)C1 O=c1c2cc(Br)sc2nc(Cl)n1C1CCN(Cc2ccoc2)CC1 C1(C(=O)NC(C)C(C)C(=O)N2CCOCC2C(F)F)CCC(C#N)CC1 C1(CC)(NC(=O)C=CC2CCCN2C)CCCN(C(=O)CC2CC2)C1 C(=O)(CC(C(F)F)NC(C1(C)CC2C=CC1C2)=O)NCc1cn(CC=C)nn1 c1(C(N(C2C3CN(C(C(CC)(C)F)=O)CC32)C)=O)cnc2ccccc2n1 N1(C(c2nc(C(C)C)sc2)=O)CC(NC(C2C(C)C2C)=O)CC2(CCOCC2)C1 N1(C(C(C)OCC)=O)CCN(CC2CN(C(=O)C(c3cccc(C)c3)C)C2)CC1 N1(C(CCC(=O)NC)=O)CC2CCC1CN2C(=O)Cc1cc(C)sc1C C=CC1(C(N(CCSC=C)CC)=O)CCN(C(=O)Cn2nc(C)cc2C)C1 C1(NC(c2ccoc2)=O)CC2CCC1CC2NC(C1Cc2nnsc2S1)=O N1(C(c2sc3cccc(OC)c3c2)=O)CC2COCCC2(NC(=O)C(C)C)C1 Cc1c(F)ccc(C(=O)NCCC(C)NC(=O)Cc2c(F)cccc2F)c1C#N c1(CC(=O)NC(CNC(c2nncc(OC)c2)=O)C2CCC2)ccc(C)c(F)c1 c1(CCC(N2CC(CC)N(C(=O)C(C)C(F)F)CC2)=O)c[nH]c2cccc(C)c12 S(=O)(=O)(c1cc(Br)ccc1Br)N1CC(CC#N)N(c2ncnc3c(Br)csc23)CC1 C12(NC(CN(CCOC)C)=O)CCCC1N(C(c1cc(C)c(Cl)cc1F)=O)CC2 C1(NC(=O)Cc2csc(Br)c2)CCCN(C(C23CC(O)C2C3)=O)C1 c1(NC(C2N(Cc3ccnc(OC)c3F)CC(F)C2)=O)c(Cl)cc(Br)cc1Br C1(C(=O)NCc2n(C)nnc2)CN(C(=O)COc2ccon2)CC(C)(C)C1 N1(Cc2cc(C)cc(F)c2)CC(C(N2CC3CC2CN3C)=O)CC(F)(F)C1 c1(NC(N(C(C)C)CC2CCCC2C)=O)cnn(C(C)(C)C)c1 CCC(C(=O)NCCN(C(=O)CCCSC1CC1)C(C)C)NC(C)=O C=CCC(C(=O)NCC(C)(Cn1cccn1)NC(=O)CN(C1CC1)CC)C(C)C C1(C(C)C(=O)NC(C2CCCC2)CNC(C2(Oc3ccsn3)CC2)=O)CCC(=O)N1 c1(-c2cc(CC)c(O)cc2)cc(S(=O)(=O)NCC(=O)NCC(F)F)ccc1OC C1(C(=O)NCC(CC)NC(c2cnc(=N)[nH]c2)=O)CC2CCC1C2 C1(CNC(C2C(C#N)C2)=O)CC12CCN(C(c1ccon1)=O)CC2 C1(NC(c2c(C)cc[nH]2)=O)C2CC1CN(C(C1(Cc3cccnc3)CC1)=O)C2 CC1(C)COCC(CC(=O)NCC(c2ccccc2)NC(C2CNC(=O)N2)=O)O1 c1(CC)nc(C)c(CC(=O)NCC(O)CCNC(=O)C(F)CC2CC2)c(C)n1 O=C(C1CCCc2nn[nH]c21)NC1CCN(C(=O)CCn2cncn2)CC(O)C1 O=C1NCC(C(=O)NCC2(O)CC(CNC(C3(c4nccs4)CC3)=O)C2)O1 C1(CCn2cc(C(N3CCSCC3)C)nn2)CCN(C(C2CC2C(=O)O)=O)CC1 CC1CCN(C(C23CCCN(CCC2)C3)=O)CCN1C(=O)CCC(C)N(C)C C(=O)(C(C(C)CC)OC)NC1(C(F)F)CCN(C(C2(OCC)CCCC2)=O)C1 c1(C(C(=O)NCCC#N)N(CC(Cl)Cl)C)nc2c(s1)CC(C)(C)CC2 CCC(CC(=O)NC(C)CC1CN(C(=O)C(c2ccccc2)N(C)C)C1)C(C)C c1(C(=O)NC2CC(NC(c3nc(C(C)OC)sc3)=O)C2)cc(=O)c(C)c[nH]1 N1(CC2CC(C(C)C)OCC2)CC2CN(C(=O)CCCC3CC3)CC2C1 C(=O)(C1=CC2CCCCC12)NCC(N(C(CCC=C(C)C)=O)C)C1CC1 CC1CC(CCNC(c2ccns2)=O)CN1C(=O)OC(C)(C)C c1(C(N2CCCC(c3ccccc3)C2)=O)cc2c(-c3ccoc3)cncc2s1 C(=O)(CN=S(C)(C)=O)N1CCCC(N(C(CCC(C)N(C)C)=O)C)C1 N1(C(C2CCSC2)=O)CCCC(c2cn(CC(=O)C3CCC3)nn2)(C(=O)O)C1 C(=O)(C(F)(F)CC(C)C)N1CC(N(C(CCC(=O)NCCC)=O)C)C(O)C1 C1(CNC(CC2CC(CC)C2)=O)CCCCC1N=c1ncnc2[nH][nH]c(C)c1-2 C(C)(C)(CC(=O)NCC12CC1CN(C(c1cc(C)nn1C(C)(C)C)=O)C2)OC C1(C)CN(C(C)C)CCC1C(F)(F)F.C1(n2cc(CC)nn2)C2CC3C(C2)C13 c1(-c2cn(C)nc2)ccnc(N2CCC(C(=O)Nc3ccc(F)cc3)CC2)n1 CC(C)C(F)(CNC(=O)C=CCF)C(=O)NCC1(CO)CCN(C)C1 c1(NC(c2c(C)cncc2C)c2n(CCOC)nnn2)cc(C)cc(O)c1 C12(NC(CC=C)=O)CCCCC1CN(C(c1cccc(NC(C)=O)n1)=O)C2 CCC(C)(COC)C(=O)NC1CC2(C1)CC(CNC(C1CC(OC)C1)=O)C2 N1(C(C2C3(CC(NC(Cn4cnc(C#N)n4)=O)C3)C2)=O)CCc2nocc2C1 C(=O)(C(C)CC(C)(C)C)NCC1(C(N2CCCCCC2CC)=O)CC(=C)C1 C1(n2c(-c3ccc(CCC)s3)nc(C(C)O)n2)CCCS(=O)(=O)C1 C1(NC(C2(c3onc(C4(N=[N+]=[N-])CC4)n3)CC(F)(F)C2)=O)CC(CO)C(O)C1 C(=O)(C1CCN(C)c2ccccc21)N1CCN(C2C(C)CN(C)C2)CC1 C(=O)(CC(C(F)(F)F)N1CCOCC1)NCC(C)(CO)NC(=O)C1=CCCCC1 CC(C)(C)C(CNC(C1CCN(CCO)C(=O)C1)=O)C(=O)NC1CC1 c1(-c2nc(CCCCC)nn2Cc2ccccc2)ccc(S(=O)(=O)C(C)C)cc1 Cn1nc(C(F)F)c2cc(C(N3CCC(O)(c4cccc(F)c4)C3)=O)sc12 C(=O)(C(C)C1=CCCC1)NCC(N1CCN(C(c2ccc(C)nc2)=O)CC1)C n1(CCCC)ccc(=NC(=O)CC(C(F)(F)F)NC(C2(C)CC(=O)N(C)C2)=O)[nH]1 Clc1ccccc1C(c1nnnn1Cc1ccccc1)NCC1CC2CCC1C2 C1(C(C2CCC2)NC(c2n(CC)nnn2)c2ccncc2)CC2(CCC2)C1 c1(C(=O)NC2CC(C)(NC(C3CCS(=O)(=O)N3)=O)C2)c(C(F)(F)F)cccc1O Cc1nsc(CNC(c2cnn(C)c2)Cn2ccnc2C)n1 N1(C(=O)C(c2ccccc2)NCc2cc(O)ncc2F)CCC2CCC(O)C1C2 CCCC(O)(CCC)CC(=O)N1CCN(C(=O)CC(O)C2CCCC2)CC1CF Cc1ccc(C)c(CC(=O)NC2C=CCN(C(c3nc(C)n(C)c3C)=O)C2)c1 Cc1c(Cl)cnn1CC(=O)NCC(CNC(=O)CC1CCCOC1)CO N1(CC=C(C)C)CCN(Cc2ccncc2)C(=O)C12CCCCC2 C1(C(=O)OCCC(C)(C)C)(COC)C=CCC1 c1(CC)nc(N2CCCC2CNC(c2nn(C)cc2Br)=O)cc(C)n1 c1(Cc2ccc(CCN(C)C)cc2)nc(=NC(=O)N2CCN(OC)CC2)s[nH]1 O(NC(=O)CC(C)C(C)(C)NC(=O)CC1(O)CCOCC1)CCOC c1(C(N(CC(CNC(c2c(COC)cc[nH]2)=O)O)C)=O)ccc(CO)cn1 C1(C(=O)NCC(CCCC)NC(c2cnn(C3CCC3)c2)=O)CC(=O)NC1(C)C C1(C(=O)NC(CCOC)CNC(C2CC2C)=O)C(C)(C)C1(C)C N1(C(CC=CCC)=O)CC(NC(c2oc(C3CC3)nc2C)=O)CC1(C)C C1(CNC(c2cc(C)c(O)nc2)=O)CN(C(=O)Cc2ccon2)C2(CCC2)C1 N1(C(C(C(C)N)N2CCOCC2)=O)CCCN(CC2(C(=O)N(C)C)CC2)CC1 c1(C(N2CC(NC(C3C(C)(C)CC3)=O)C2)=O)cc(C(F)F)ccc1F CC(O)C(F)(F)C(=O)NCC1C2CN(C(c3cccc(N)c3N(C)C)=O)CC12 c1(C(=O)NCCC2N(C(C(CC)SC)=O)CCOC2)cccc2c1CCOC2 C1(CC(=O)N(C)CCOCCNC(=O)CN(C)C(c2ccsc2)=O)CCCC1O C1(NC(C(C(CC)O)C)=O)CC2(CCCCN2C(=O)CN(CC(C)(C)C)C)C1 C1(CC(=O)NC2(C(=O)NOCCCCF)CC(CO)C2)CCCC2CC12 C1(C(=O)NCCOCC(=O)NCC(F)CO)CC=CCC1 C1(C(=O)NCC(C)CC2CC2)(NC(=O)CCc2nccn2C)CCC(C)(C)C1 C=CCC(C)C(=O)N1CCCCC1CN(C(=O)CC1(COC)CCC1)C Cc1c(SC2(C(N3CC(NC(=O)CN(C)C)C(C)C3)=O)CC2)oc2ccccc12 c1(N(C)C)ccc(C(=O)NCC2(C)CCN(C(C3CCOCC3)=O)C2)nn1 C1(CNC(CC(C)c2ccco2)=O)CC(NC(=O)C=CC(C)(C)C)CCO1 c1(OC)cncnc1C(=O)NC(C(N)=O)C(C)O c1(NC(=O)C(=O)N(C)CCOCC)cccc(C(=O)NC2(C)C(NC)CCC2)c1 C1(NC(CC2(OCC)CC2)=O)CCSC12CN(C(C1CC(CC(F)F)C1)=O)C2 C12(CNC(C=CC=CC)=O)CC1CN(C(=O)C(C)Oc1ccccc1F)C2 C1(C)(C(=O)NC(C2N(C(c3cc(Br)cs3)=O)CCC2)C)CCC(F)(F)CC1 C1(C(=O)NC(C(=O)N(CC)CC)C)C=CC(NC(=O)CC2CCCCC2)C1 C1(C(=O)NCCC=CC=C)CCC(O)CN1C(C1CC=CC1)=O c1(C(=O)NCCN(C(=O)CN2CC3C=CC2C3)C)noc2c1CC(C)(C)CC2 N1(C(C(N(C(c2cnc(OC)s2)=O)C)C2CC2)=O)CCc2nc(O)[nH]c2C1 c1(C(C(=O)NC(CNC(c2nccc(C)c2)=O)CC(C)C)C)ccc(F)cc1F C1(C(N2CCC(O)(C(C)NC(c3cscc3Cl)=O)C2)=O)CCOC(C)(C)C1 CC1=C(C(=O)NC(CCC2CC2)C(=O)NCC2(O)CCN(C)C2)CC1 C1(F)(C(=O)OC)COCCN(C(=O)NCc2cc(COC(C)(C)C)n(C)c2)C1 C1(CNC(C(CC)=CC)=O)CCN(C(=O)CC2CC2C(F)(F)F)CC1O C1(C(=O)NCc2cc(C(=O)NCC(C)(CO)OC)on2)CCCC(=O)CC1 C#Cc1cnc(C(=O)NCC(C)CN(C)C(c2c(OC)cccc2F)=O)c(C)c1 C#Cc1cn(C)nc1C(=O)N(C(C)CN(C)C(c1scnc1COC)=O)C C(=O)(C1CCCc2sccc21)NCC1N(C(C2(CC#C)CCC2)=O)CC1 Cc1c(C(N2CCCC2C(C)(C)C(=O)NC(c2ccn(C)n2)C)=O)cccc1O CC1CCN(C(=O)C(C)C2(O)CCC2)CC1NC(=O)C=Cc1ncc[nH]1 c1(C(N2C(C(=O)NCCC=CCCC)(CC)CCC2)=O)ccc([N+](=O)[O-])[nH]1 CC1(C(N2CCC(NC(C3CCCCC(=O)N3)=O)C2)=O)CCC2CC2C1 C1(NC(C(c2n(C)ccc2)=O)=O)CC2CCCC(C1)N2C(c1cnc(O)[nH]1)=O c1(C(=O)NC2C3CN(Cc4c(C)nc(C)o4)CC32)c(F)ccc(F)c1Cl C1(NC(CCC(=O)NC)=O)CC2CC1N(C(c1cccc(Br)c1Cl)=O)C2 Cc1cc(C)c(C(=O)NC2(CN(C)C(c3cc(C(F)(F)F)n[nH]3)=O)CC2)n1C c1(CC(C(=O)NC(c2ccsc2Br)C(=O)OC)OC)ccc(F)cc1 N1(CC2ON=C(C(C)C)C2)CCN(S(C)(=O)=O)CCC1C C1(C(N2C(CC(=O)NCC(C)(C3CC3)OC)CC2)=O)(CO)CCOCC1 N1(C(c2c(C)noc2C)=O)CC2CCCCC2(NC(=O)CCCCN(C)C)C1 C1(NC(C2CCOCC2)=O)COC2(CCN(C(c3cncc(Br)c3)=O)CC2)C1 C1(CC)CN(C(c2scc(C)c2-c2ccc(OC(F)(F)F)cc2)=O)CCCO1 C1(NC(=O)CCC2CCC2)CCN(C(C2CC2F)=O)C12CCC2 C1(C(N2CC(C)C(NC(C3(S(C)(=O)=O)CCCC3)=O)C2)=O)CCCC2CCCN12 Cc1ncc(NC(=O)CC=CCNC(=O)C(O)CC2CCCC2)cc1Cl N1(C(c2cc(CC)[nH]n2)=O)CC2CN(C(=O)CC3C=NN(C)C3=O)CC2C1 C1(C2CCCCO2)(C(=O)NC2C(CNC(c3ccsn3)=O)COC2)CCOCC1 c1(OC)ccc(Cl)c(C(=O)NCCN(C(=O)Cc2cncn2C2CC2)C)c1 C1(NC(CCC(=O)NC)=O)CCN(C(c2ocnc2C(C)C)=O)CC1(C)C CC(C)C(O)CC(=O)N(C1CCCN(C(=O)C(C)CN2CCOCC2)C1)CCO N1(C(CN(CC)CC)=O)CCCN(C(=O)COC2CCOCC2)CC1CO N1(C(CSCCC)=O)CCC(NC(=O)C=Cc2cnc[nH]2)CC1c1ccccc1 c1(C(N2CCC(CC=C)(NC(=O)C(CCC)N(C)C)C2)=O)c(N)ccc(C)c1F c1(OC)c(C(=O)NCC(C)(C(C)C)NC(c2cn(C)cn2)=O)oc2ccccc12 Cc1coc(C(=O)NC(C(C)NC(=O)CC(C2CCC2)C2CCC2)C(C)C)c1C N1(C(C(c2n(C)cnc2)O)=O)CC2CCOC2(CNC(c2ccco2)=O)C1 CCCC(CNC(c1coc(CC2CC2)n1)=O)NC(=O)CCCc1ncco1 C#CCC(C(=O)N1CC(CNC(=O)CCn2cc(Cl)cn2)(OC)C1)C1CC1 C1(C(C)(C)O)CCN(C(C2CCCN2C(c2coc(C(=O)OCCO)c2)=O)=O)C1 Cc1cnc(C(=O)NCC2CCCCN2C(C23CCCC2(C(N)=O)C3)=O)nc1 C(=O)(C(F)C(C)(F)F)NCc1ccc(C(=O)NC(c2cccc(O)c2)C)cn1 CC(C)S(=O)(=O)C(C)C(=O)NCC1C(C2CC2)CCN1C(C1CN(C)C1)=O CC1OCC2(CCN(C(c3ccc(Cl)cc3O)=O)CC2)C1NC(C1CCCO1)=O c1(OC)c(C(N2CC(N(C(=O)C(C)OC)C)C2)=O)cccc1[N+](=O)[O-] N1(C(C(F)OC)=O)CC(CNC(=O)Cn2nccn2)C(O)C1 C(=O)(CC(=O)NCC(O)CCC1CC1)N.C1(CCC#C)(CN)CCC1 CCCC(C)(O)CC(=O)N1CCN(C(C2(S(C)(=O)=O)CC(O)C2)=O)CC12CC2 CCCC(CCCNC(=O)C(C)(C)n1cnnn1)NC(c1nc(CC)c[nH]1)=O c1(OC)ccc(Cl)c(C(=O)NCCC(C)(C)NC(=O)CCCC2CC2)c1N FC1(F)CC12CCS(=O)(=NC(=O)C1CCCN1CCN1CCOCC1)C2 C1(CNC(C=Cc2ccc(C)o2)=O)CC2(CC2)CN1C(C1CC2CC1C1CC21)=O c1(C(=O)OC)cccc(C(=O)Nc2cccc(NC(C3CC3(F)F)=O)c2)c1O Cc1ccc(N2CCCC2)c(CO)c1.C12CC(C1)NC(=O)C2.C(C)(C)(C)O C#CCC(C(=O)NCC(C)(C)CO)NC(C1CN(CC)CCO1)=O CC1(C)CN(C(C2COCCN(CCCCF)C2)=O)CCN1CCn1cnnc1O c1(N(CCC)CCNC(=O)C=C2CCSCC2)nc(Cl)nc(CC)c1C#N C12(C(=O)NCC(CC)(CC)NC(=O)C#CC3CCC3)CCC(CC1)CO2 c1(C(N2CCC(C(=O)OCC)(CCCC)CC2)C(=O)N)cc(F)c(Cl)cc1Cl C1(NC(C23CC(NC(c4c(Cl)cc(C#N)s4)=O)(C2)C3)=O)CCOC2(CCC2)C1 c1(C(=O)NCCN(C(C(CC)C2CCOCC2)=O)C)nn(C)cc1Cl N1(C(C(C(CC)C)N)=O)CCOCC(CNC(C2CCc3ccoc3C2)=O)C1 c1(N(C)CCOC2CCC2)nnc(C2CC2)n1Cc1cncc(F)c1 c1(C(N2C(CNC(C(C(C)(C)O)F)=O)CCCC2)=O)nnc2ccccn12 c1(C(C(=O)NC2(CO)CN(C(C(C)OCC#C)=O)C2)O)ccccc1Cl CN1CCCC2C1CCN2C(=O)Cc1csc(-c2ccsc2)n1 Cc1c(C(=O)O)c[nH]c1C(=O)NCc1ccnc(OC(C)C)c1 c1(CC(=O)NCC(C)CNC(c2cnc(CC3CC3)s2)=O)cnn2ccccc12 C1(C)(NC(C2N(C(CCCOCC)=O)CC2)=O)CCC(C)(C)C1 c1(NC(CC)CS(C)(=O)=O)nc(C)cc(=NC2CC(N3CCCC3)C2)[nH]1 c1(C(=O)NC2(C)CCN(C(CN(C)C3CC3)=O)C2)cc2c(Cl)nccc2s1 Cc1cc(CCC(=O)NC2CCC(NC(C3CCC(C(N)=O)O3)=O)CC2)nn1C c1(C(C(N2CCC(N(C(C(C)C3CC3)=O)CCO)C2)=O)(C)C)cccc(C#N)c1 C1(C(=O)NC(C#C)CC)(CC)CN(C(c2nccn2C)=O)C1 C=CCC(C)(C)CNC(C12CCC1C2)=O C(=O)(C1CCCn2cnnc21)NC1C(C)CN(C(=O)C(F)=CC2CC2)CC1 Cc1cccc2c(C(=O)NC3CCN(C(C4C5CNC(=O)C45)=O)C3)coc12 Cc1ccc(-c2noc(C(N3CCC(CNC(=O)CNC4CCC4)C3)C)n2)cc1 Cc1cc(C2CC2)ccc1C(=O)OCCOC(=O)Nc1ccccc1 c1(-c2ccc(C(C)C)cc2)n[nH]c2c1CN(C(=O)C(C)(C)CC1CC1)C2 n1(CCCC2CCN(C(=O)NCCF)CC2)cnc2c1CCCC2 N1(C(C)C)CCCCC1CN1CCOCC1.c12ccc(cc1)NC(=O)C(=O)NC2 n1(CCC2CN(C(C3(Br)CC3)=O)C2)cc(C2C3COCC23)nn1 C1(CNC(c2n[nH]cc2Cl)=O)(CO)CCCN(C(=O)C(=CC2CCCCC2)F)C1 C1(NC(CC(CC)SC)=O)CN(C(=O)COC2CC2)CC12CCOCC2 C12(C(N3CCC(SC)C3)=O)COCC1CN(C(c1cccnc1C)=O)C2 c1(C(N2CC(CNC(=O)CC3CCOC3)C(O)C2)=O)ncc(Br)cc1F N1(C(c2c(Cl)cc(C)c(N)c2)=O)CCC2CCN(C(=O)C(C)NC(N)=O)CC2C1 Cc1nc2c([nH]1)C(C(=O)NCCCCNC(=O)CCc1ccc(C)o1)CCC2 N1(C(C2C3C=CC(CC3)C2C(F)F)=O)Cc2cc(Br)ccc2CC1C(F)(F)F N1(C(CCC(CC)NC(c2cnc(O)c(C)c2)=O)=O)CC2CN(C)CC2C1 C1(C(N2CCCC(CN(C(=O)CSC3CC3)CC3CC3)C2)=O)CCCOCC1 C(CCCCC(=O)NOCC(=O)OC)OC(C(CCC)O)=O C(CCC(O)C(=O)NCC1CNC(=O)C1)NC(CC=CC=C)=O N1(C(c2occ(C)c2)=O)CC(CNC(=O)CC2OCCCO2)CC(C)C1 c1(C(=O)OC)ccc2c(c1)CN(C(c1sc(C)cc1Br)=O)CCO2 c1(CC(=O)NCC(CO)NC(CS(CC)(=O)=O)=O)cn2cccc(C)c2n1 C1(C(=O)NCC2(C(=O)NCC3CC3c3nn[nH]n3)CC2)(OC)CCCC1 CC1(C)CCC(CC(N2CC(O)(CNC(C3CCCC(F)C3)=O)C2)=O)C1 C1(F)(CNC(c2c(CC)cc(Cl)cc2)=O)COCCN(C(=O)C2=NOCC2)C1 C1(NC(C)=O)CCN(C(=O)CC2CC3CC3C2)C1C.C12(CC1)C(=O)N2 N1(C(c2c(C)n[nH]c2)=O)CC2CCC1C2NC(=O)C=Cc1ccc(O)cc1 C1(C(C)(F)F)CCCCN1C(C1CCCN1C(c1ccccc1)=O)=O n1(CC)nc(C(=O)N(CC(C)NC(=O)CC(C)=C(C)C)C)c(Br)n1 c1(C(=O)NC23C(CN(C(c4c(C)occ4)=O)C2)CCC3)cc2ccsc2c(O)n1 c1(C(=O)NC2CCN(C(CS(=O)(=O)NC)=O)C2)csc(S(C)(=O)=O)c1 c1(CNC(CN(C(=O)COCC2CC2)CC)=O)cnccc1CO C(=O)(CCC(C)(F)F)NCC(C)N(C)C(c1coc(Cn2cccn2)c1)=O CCCC(C(=O)NCCCF)N(C1CC1)CC C(CC(=O)NCc1cccnc1C)(CC(C)C)NC(C(CC=CC)CC)=O c1(-c2onc(-c3cccc(C4(S(C)(=O)=O)CC4)c3)n2)cc2cn[nH]c2cn1 n1(C(C)CC(=O)N2CC(CNC(c3ccc(F)o3)=O)C2)cnc2ccccc12 CCC(C)C(O)C(=O)NCC(C1CCN(C(=O)C(O)CN2CCOCC2)CC1)O N1(C(C=CCC)=O)CCCC(C(=O)N(C)Cc2ncn(C)n2)C1C C(=O)(C(F)(F)C(F)F)N1CCC(N(C(C(C)OC)=O)Cc2ccncc2)CC1 c1(C(N2C(C)CC(NC(=O)CC(F)(F)F)C2)=O)ccc2c(O)nccc2n1 C1(NC(CN(C(C2(CCCC)CCC2)=O)C2CC2)=O)CSCC1C N1(C2CCN(C(c3c(C)nns3)=O)C2)CCC(NC(=O)CCc2cscn2)CC1 c1(SC2CCN(c3c(C(C)=O)cnc(Cl)n3)C2)noc2c1CCCC2 C1(C)(C(=O)NCC2C(NC(CCCNC(C)=O)=O)C2)CC(C2CC2)=NO1 CC1C(NC(C2CC3CCC2C3)=O)CCN1C(=O)C1CC1 c1(C(N(C(C)C)CCNC(=O)C(O)C2CC2)=O)cc2sc(Cl)cc2[nH]1 C1(NC(C(CC)NC(C)=O)=O)CCC2CCN(C(=O)C(C)(C)C3CCC3)C1C2 c1(C(N2C(C)(C)C(NC(=O)COCCO)CC2)=O)cc(F)cc2ccncc12 c1(SCCNCC(C2CCCC2)OCC)ccc(C#N)cc1 C1(NC(CCN(C(C)=O)C)=O)(CF)CCN(C(=O)CC2(C)CCOC2)C1 C(CCCCNC(=O)CC1CC1(C)C)N(C(C1CCC1)=O)CC C12(NC(COCC)=O)CCCC1CN(C(c1cc(-n3cccn3)ccn1)=O)C2 N1(C(=O)CC2CC23CC3)CCCC(CCCCNC(=O)Cc2ccncc2Cl)C1 c1(C(=O)NCC(CN(C(=O)C2=CCCOCC2)C)O)nc2cc(O)ccc2[nH]1 Cc1ncc(C(=O)N(C(C)C(=O)NCC23CCC(CC2)O3)C2CC2)c(=N)[nH]1 C1(NC(C2SCCS2)=O)CCCCCN(C(C2CC(C3CC3)=NO2)=O)C1 C=CCCCCCCCC(=O)NC1CN(C(C23CCCCN2CCC3)=O)CC1C C1(O)(CN(C(C2C(=C)CC2)=O)C)CN(C(=O)CCOC2CCC2)C1 C(=O)(CCCC(=O)N(C1CCN(C(c2ccncc2F)=O)C1)CCO)NCCC C1(C(N(CC(=O)NC2(CCOCC)CC2)CC#C)=O)CCOC1C C12(NC(CC(CCCC)O)=O)CC3CCC(C1C2)N3C(c1ccc(=N)[nH]c1)=O c1(CC(=O)NC2CC3(C2)CC(C(=O)Nc2ncco2)C3)ccc(Cl)cc1F C1(C(=O)Nc2cccnc2)CCCC1(C)C.C12CC(C1)CNC(C)C=CC(=O)N2 c1(NC(COCC(=O)NCC(CC)CCO)=O)ccc(F)c(F)c1 CC1(C(N2CCCC(CCNC(c3ncc[nH]c3=O)=O)C2)=O)CC2CCC(C1)S2 CC1Oc2ccccc2OC1C(=O)NCCCN(C)C(c1cnc(O)s1)=O CCCCC(C)(CO)NC(C1(N(C)C(c2ccc(O)c(F)c2)=O)CC1)=O c1(C(N2CCCC(C)(CNC(CC)=O)C2)=O)cc(F)c2nc(C)cn2c1 c1(NC(C2CCN(C(=O)CCCc3ccc(F)cc3)C2)=O)ccc(O)c(F)c1F c1(N2CCCN(C(c3c(Br)ccc(C)c3)C3CC3)CC2)ncnc2n[nH]cc12 c1(NCC(CNC(CCC(C)SC)=O)C)ncnc(O)c1Br CC(C)CCC(O)C(=O)NCCC(C)CCNC(c1cc(N)cc(F)c1)=O C(=O)(CS(=O)CCC(F)(F)F)NC1CC(C)(CNC(COC(C)C)=O)C1 N1(C(c2scc(COC)c2)=O)CC(NC(C2(c3cccs3)CC2)=O)CCC1C C(=O)(CCCC(F)(F)F)NC(C)CCCCNC(=O)CN(C1CCSC1)C N1(C(C2N(C(c3n(C)ccn3)=O)CC(F)C2)=O)CCOC2(CC2)C1 C(=O)(CCC(C)(C)C#N)NCCCN(C)CC=Cc1cccnc1 O=C1CC2C(C(=O)NC3(C(=O)NCCOC4CCC4)CC(O)C3)C2C1 C(=O)(C1=NNC(=O)C1)N1CC(CN(C)C(c2cc(Cl)cc(Br)c2)=O)C1 C(=O)(CCCC(=O)NC1CC1NC(c1scc(C)c1C)=O)N(CC)CC C1(C(=O)NCCN(C(=O)CN(C)C)C(C)C)CC12CCC(C)(C)CC2 C=C1CCN(C(C2C3CCC(C3)CN2C(=O)C(F)(F)F)=O)C(C(=O)OC)C1 N1(C(c2n(C)cnc2)=O)CCN(C(C2CC2CF)=O)CC1c1cc(F)ccc1F c1(C(=O)NN(C(=O)CCCOCC)CC(C)SC)cnn(-c2ccccc2)c1C c1(C(N2CCC(NC(c3c(C)onc3)=O)CC2C)=O)ccc2c(c1)CCN2C N1(C(C(C2(C)CC2)NC(CCn2ccc(C)n2)=O)=O)CCC2CN(C)CC12 C1(OC)CC2(C1)CC(C(=O)NC1CN(C(=O)C(C)SC)CC1c1cnn(C)c1)C2 c1(CCC(=O)NCC(CC)NC(c2cc(C)c[nH]2)=O)ccc(Cl)cc1 C1(Cl)(C(=O)NC2CC(OC)CN(C(C)=O)C2)CC12CCOCC2 c1(C(C)C)cccc(NC(c2cncnc2)c2nnnn2CC2CCCO2)c1 N1(C(c2occ(C)c2)=O)C2CCC1C(CO)N(C(c1cccc(N)c1)=O)C2 c1(CNC(C2CCN(C(c3ccc(F)s3)=O)CC2O)=O)cc(F)cc(Br)c1 CCCC(CCCNC(C12CCOC1CCOC2)=O)NC(c1cnc(CC)s1)=O C1(CCC)CCN(C(=O)C(C2CCCC2)NC(=O)CCn2cnc(=N)[nH]2)C1 c1(CC)nnc(C=CC(N2CC(CCNC(=O)CC3CCC3)C(C)C2)=O)o1 C12(C(=O)OCc3cccnc3F)CCCCCC1CNC2 CN1CC=C(CC(=O)N2CCC(NC(=O)CSS(C)(=O)=O)C(C)(C)C2)CC1 c1(CC(=O)NCC(C)N(C)C(c2cnc(C3CC3)o2)=O)ccc(Br)c(F)c1 N1(C(C(C=C)OC)=O)C2COCC1CC(NC(=O)C(CC)c1ccccc1)C2 c1(C(=O)NC(C)C=CC(=O)NCCC(C)(C)F)ccc(Cl)cn1 Cc1cc2cc(C(N3CC(C)N(C(C4CCC(=O)N4)=O)CC3C)=O)[nH]c2cc1Cl c1(C(=O)NC(CN(C(C(C)NC(CC)=O)=O)C)C)c[nH]cc(F)c1=O c1(C(=O)NCCCC(=O)NC2CN(C(CC)=O)CC2C)ccc2c(c1)CCC2 CS(=O)(=O)C1CN(C(=O)CC2(CO)CC2)CC1NC(=O)CC1CCCCCO1 C1(C2(O)CN(C(=O)CCC3CCCC3)C2)(CNC(=O)CN2CCCS2(=O)=O)CC1 C1(CNC(C(=O)N(CCCCO)CC)=O)CCN(C)C1 c1(C(N2CCC(NC(CC3CC(OCC#C)C3)=O)CC2)=O)ncc(C#C)cc1C c1(C(=O)Nc2cnn(-c3ccncc3)c2)ccc2c(c1)CNC2=O C(CC(=O)Nn1ccnn1)N(C(c1c(CC)cns1)=O)C c1(N2CC(NC(CCN(CC)CC)=O)CC(C)(C)C2)c(C#N)cccc1[N+](=O)[O-] N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)Cn2ncnn2)CC1C1CCCC1 O=C1CN(C(c2c[nH]ccc2=O)=O)C2CCN(C(=O)Cc3cnc[nH]3)CC2N1 CC(C)C(C)(CNC(C1(C)CC=CCC1)=O)NC(=O)COC1(C)CCOCC1 Cc1cc(C(=O)N(CCCN(C(=O)C(n2nc(C)cc2C)C)C)C)cc(N)c1 C12(CNC(C3COC(CNC(c4cocn4)=O)C3)=O)CCCC1C2 C12(C(=O)NC3CN(C(CS(CC)=O)=O)C(C)C3)OCCCC1C2(F)F Nc1ccc(C(=O)NCC2(CNC(c3cc4scnc4[nH]3)=O)CCCC2)cc1F C1(C2CC2)(C(=O)NCCC2N(C(C3N(CCC(C)C)CCC3)=O)CCC2)CCC1 c1(OC)ccc(C=CC(=O)NC2(C)CN(C(c3cccc(CSC)c3)=O)C2)cc1 N1(C(C(c2nc(C)sc2)=O)=O)CCC2CN(C(c3ccn4nccc4n3)=O)C2C1 c1(C(=O)NCCN(C(=O)CC(C)(F)F)C(C)C)c[nH]c2cc(Cl)ccc12 C(CCCCC(=O)NC1CC2(C1)CC(NC(=O)C(C1CCCC1)OC)C2)OCC CCCC(C)CC(=O)NCCN1CCCN(C(C2(N(C)C)CCCC2)=O)CC1 C1(CNC(C(C2CC2)OC)=O)CC2(CC2)CN1C(=O)Cc1cnc(C)[nH]1 C1(N(C(=O)CCCNC=O)C)CN(C(=O)CC2CCOC2)CC1O.c1ccccc1 C(CC1=CCN(C)CC1)C(=O)NC(c1ccc(CC(F)(F)F)cc1)C CN1C(=O)CCC1C(N1CCC(F)(C(N2CCC(CF)(CO)C2)=O)C1)=O C(=O)(CCC1=NNC(=O)CC1)N1CCC(C2CC2)(NC(c2cnc(OC)s2)=O)C1 C1(C(=O)Nc2ccc(-c3scc(C)n3)cc2C)CC12CCN(S(=O)(=O)CCl)CC2 CC1CN(C(=O)C(C)(C)C2CCC2)CC1NC(C1CCCN1c1ncccn1)=O N1(C(=O)CCc2cn[nH]c2)Cc2[nH]nc(C(=O)NC(c3nc[nH]n3)CO)c2C1 N1(C(CCC(=C)C)=O)CCC2(NC(=O)C3=NOC(C(C)(C)C)C3)CCCC12 N1(C(C2C=CC(NC(CCCNC(C)=O)=O)C2)=O)CCC(O)C(C)C1 Cc1c(NC(C2C3CN(C(c4c(Cl)cccc4Cl)=O)CC23)=O)ccc(C#N)c1Cl c1(NC(C2CCCN(CC(c3ccccc3)SC)C2)=O)cccc(S(N)(=O)=O)c1 C1(C(=O)NC(C)CCNC(C2CC=CCC2)=O)CCS(=O)(=O)C(C)C1 Cc1cc(=NC2CC2C2CCCC2)[nH]c(NC2CCN(CC(N)=O)CC2)n1 C1(CC)CN(C(=O)C(C)(C)COC)CCN1C(=O)C(CCOC)c1ccc(Cl)cc1 C1(NC(C2C(C)(C)C2)=O)C2CC3C(C2)C13C(=O)N1CC(O)CO1 N1(C(C(CC(C)C)F)=O)Cc2nccn2CC(NC(C2CC2(F)F)=O)C1 c1(C(=O)NC2(CN(C(C(C(C)O)(F)F)=O)C)CC2)ccc2oc(O)nc2n1 CCCC(C)(CC)C(=O)NC1CCC2CCN(C(c3cc(C)nc(O)c3)=O)C12 C1(C(=O)NCC2(C(C)(C)C)CCN(C(c3cncs3)=O)C2)CCC2(CCC2)C1 c1(C(N2CCC(O)(C(C)NC(=O)Cn3ccnn3)C2)=O)ccc(N)cc1O C1(CC)CCN(C(c2ccn(C)c2)=O)C(C(=O)Nc2cccc(CO)c2C)C1 N1(C(c2c(C)onc2-c2ccccc2F)=O)CC2(CCN2C(C2CC2F)=O)C1 CN1CC(C)(C(=O)NC2CC(CNC(C3C=CCCC3)=O)C2)CCC1=O n1(CC(N2CCN(C(C(CCC)C#N)=O)CC2C)=O)ccc2ccc(F)cc12 C1(O)(CNC(=O)CCC2(C)CC2)CCCN(C(=O)CC2CCCCC23CC3)C1.C1(C)CC1 N1(C(c2ccc(SC)o2)=O)CC(C(=O)NCC2(SC3CC3)CCC2)C(F)(F)C1 CCC(CC)(CO)C(=O)NC1CN(C(=O)CCc2cccc(F)c2F)CC1F N1(C(C(C)OC(C)(C)C)=O)CC2(CNC(C3CC3C(F)F)=O)CC1CO2 CCCCC(O)CC(=O)NC1CC(C(F)C(N2CCOCC(C)(C)C2)=O)C1 c1(C(N2CCOCC(NC(c3ncn(C(C)C)n3)=O)C2)=O)ccc(S(N)(=O)=O)s1 C12(NC(CN(C)CC)=O)CC3CCC(C1C2)N3C(C1CCc2nnnn2C1)=O c1(C(N2CCC(N(C)C)(C(N)=O)CC2)=O)cc2nc(O)[nH]c2cc1N C1(C(N(C(c2ccc(F)cc2)c2ncc(C)s2)C2CC2)=O)CC2CC1CO2 c1ccc(S(N)(=O)=O)[nH]1.C=CCC(CC)C(=O)N(CCCCN(C(=O)CC)C)C C(=O)(N=c1[nH][nH]cc1I)C1C(O)CCN(C(C2=CC(C)=CC=CC=C2)=O)C1 C1(C(=O)Nc2c(C(=O)OCC)sc(Br)c2)CN(C(C23CC(C2)C3)=O)CC(F)(F)C1 C(=O)(CCCCCF)N1CCCC(N(CCC(=O)NCC2ON=C(CC)C2)C)C1 c12cc(sn1)C(=O)NCC(=O)N2.C1(SCC)C=CCOC1 C(=O)(C(F)(F)C(F)F)N(CC)CC1CCN(C(=O)CC2CCCS2(=O)=O)C1 C(C(O)CC(=O)N1CCOC(CNC(=O)CCCC2CCCCC2)C1)N(C)C c1(NC(CC(CNC(=O)C(C)(C)C#N)OC)=O)ccc2ccncc2c1 c1(CCC(N2CCOCC(CNC(c3cc[nH]n3)=O)C2)=O)nc2cnccc2[nH]1 N1(C(CCC(C)O)=O)CC2CN(C(=O)CN3CCOCC3)CC2C1 C1(OC)CCC2CN(C(C3CCCCCN3C(C34COCC3C4)=O)=O)CC12 C1(C(=O)NCC(CC)Oc2ccccc2F)CCN(C(=O)CN(C)C)CC1 C1(NC(CCn2ccc(C)n2)=O)CCCCN(C(c2cnn(C)c2F)=O)C1 C(C(C)CC(=O)NCC(c1ccc(C(C)(C)C)cc1)(C)C)OC C1(NC(CN(C)CCO)=O)CCCN(C(c2nn(C)cc2Br)=O)C1.C(C)(C)(C)O c1(OC)ccc(C=NC(=O)C(=O)NCc2cnc(C)n2C)cc1F Cc1cc(C(=O)Nc2ccc(Br)cc2I)cc2c1CCC2 c1(C(=O)NC2CCN(C(CCOCC#C)=O)C(C)C2)cc([N+](=O)[O-])ccc1SC N1(C(c2[nH]cc(C)c2)=O)CCC(O)(CCNC(c2ccn(C(F)F)n2)=O)CC1 c1(C(=O)NCC2(F)CN(C(Cc3c(F)ccc(C)c3)=O)C2)cc([N+](=O)[O-])cn1C N1(C(C2C(C#C)C2(C)C)=O)CCCC2(C1)CN(C(c1coc(CO)c1)=O)C2 c1(SC)cccc(CC(=O)NC2CN(C(c3ccc(C4CC4)s3)=O)CC2F)c1 C1(OC)(CNC(=O)CCC(C)N(C)C)CCN(C(=O)CC2CCOC2(C)C)CC1 C1(C(C)C)CN(C(=O)CCCC(F)F)CCC1NC(c1cn(C)nn1)=O N1(C(CNC(CN(C)C)=O)=O)CC(O)(CNC(=O)CC2(C)CC2)C1 C12(NC(=O)CNC(=O)C(O)c3ccsc3)CC(CNC(c3cnco3)=O)(C1)C2 C1(C(=O)NC(CCC)C)(NC(=O)C(CO)C(F)(F)F)CCc2cc(Br)ccc2C1 N1(C(C2(CC#C)CC2)=O)CCCC(C2CCN(C(C3C=CCC3)=O)CC2)CC1 C1(NC(c2c(O)cccc2F)=O)CN(C(=O)C=CC2CCCO2)CC12CCC2 C(CC(=O)NC1CC1NC(=O)CC1CCSCC1)(C(F)(F)F)OC c1(NC(c2cc3cccc(OC)c3o2)c2nnnn2C)ncc(C)cc1[N+](=O)[O-] c1(C(=O)NC2CC(NC(Cn3c(C)c(Cl)cn3)=O)C2)ccc2ccnc(Cl)c2n1 C1(O)(CNC(c2nc(OCC)sn2)=O)CCN(C(=O)CNC(C2CCC2)=O)C1 N1(CCNC(C=C(C)C(C)(C)C)=O)CCCN(C(C2CCCCN2C)=O)CC1 C1(C(N(C)CC2CCCN2C(c2nnsc2N)=O)=O)COCCN1C c1(C(=O)OC)cccc2sc(C(=O)NCC(C)(C)NC(C3C4CCCC34)=O)cc12 c1(C2N(C(=O)CC3(OCC(F)(F)F)CCC3)CC2)cc(Br)ccc1O c1(C(N2CC(NC(C(C)CC3CCCC3)=O)C(F)CC2)=O)cc2c(ncn2C)s1 c1(CN2C(CC)CN(C(c3sccc3Cl)=O)CC2)cccc2cn[nH]c12 c1(C(=O)NC2CC(F)(CNC(C(C(C)(C)C)SC)=O)C2)ccc2nc(C)[nH]c2c1 S(=O)(=O)(c1cnc(NCCC(C2CCOCC2)O)c(Cl)c1)N(C)CC1CC1(C)C c1(OC)n[nH]c(C(=O)NC2CC(CNC(C3(C)CCCS3)=O)C2)c1Cl N1(C(c2c(C(C)C)cccc2)=O)CCn2ncc(CNC(=O)CCC(C)O)c2C1 C=CCCC(C(=O)NC1CCS(=O)CC1)NC(=O)CNC(C1CC1C)=O c1(C(N(C(CN(C(CCCCOC)=O)C)C)C)=O)nccc2ccn(C)c12 C1(NC(CN(CC)CC)=O)(CNC(=O)CSC2CCS(=O)(=O)C2)CCCCC1C CC1(C)CN(C(=O)CCC2CC2)CC(C)(C)C1NC(C1CC12CCSCC2)=O CCC(F)(F)C(C)(C)C(=O)NCCN(CC(C)O)C(c1ncoc1C1CC1)=O C(=O)(N=c1cc(C)n(CCO)[nH]1)C1C(CC)CCN1C(=O)CCC1(C#N)CCC1 c1(CCC(=O)NCC2CCN(C(C(CC)(C)O)=O)C2)ccc(Br)c(C)c1 C1(CCC)CN(C(C2C(C)(C)OC2(C)C)=O)CCN1C(C1CCN(C)C1C)=O C(=O)(C1CCCc2ncnn21)N1CCC2(CCN(C(=O)CC3CC=CC3)C2)C1 c1(C2(OC)CC2)ccccc1OC.n12nccc1CNC(=O)C1CCCC21 c1(CC(=O)NC2(C)CCCN(C(c3n[nH]cc3F)=O)C2)ccc(S(C)(=O)=O)cc1 C(CC(F)F)(C(=O)NOC(CO)C(C)C)N(C(c1nc(C)sc1)=O)C C1(NC(C(CSC)C)=O)CCN(C(=O)C(C(C)(C)C)NC(N)=O)C(C)C1 N1(CCOC)Cc2ccccc2C(NC(c2c(Cl)nc3sc(C)cn23)=O)C1 Cc1ccncc1C(C)Nc1nc(Cl)c(C(F)F)s1 N1(C(CCNC(C)=O)=O)CC2CCC1CN2C(c1ccc(Cn2ccnc2)o1)=O C(=O)(CC(C(F)(F)F)NC(=O)CCNC(=O)COC)Nc1n(CC)nc(C)c1 C1(F)(CNC(C2(COC(C)C)CC2)=O)CCC(NC(=O)C=C(Cl)Cl)C1 CCC(O)C(C)C(=O)NCC(C1CCCCN1C(c1ccoc1C1CC1)=O)(C)C C(C(C(=O)N1CC(CNC(=O)CCC2CC2C)C1)OC)OC C1(CC)CN(C(=O)CSC)CCN1C(C12CCC(NC(C)=O)C1C2)=O N1(c2ccc(C)c(Cl)c2)N=C(C(=O)N2CCCC2(C)CN)CC1=O N1(C(C(C=C)(F)F)=O)CC2CCN(C(c3cccc(CC(C)C)c3)=O)CC2C1 C#CCCCC(=O)NCCC1COCCN1C(c1cc(C(N)=O)no1)=O C=CCCCC(C(=O)N1CC2CC(O)CC2C1)NC(c1ccoc1)=O C(CC(C)CC)(C(=O)NC1(C#C)CC(F)(F)C1)NC(C(CC#C)C1CC1)=O c1(C(N2CC(C)N(C(C3(C)CC3)=O)CC2)=O)nc2ccc(Br)cn2c1N c1(CN2C(C(=O)NCCC(F)=C(F)F)CCCC2)c(O)ccc(F)c1Br C1(CN(C(=O)COc2cccnc2)CC)CCN(C(C2(C)CCC(C)C2)=O)CC1 C1(CNC(=O)COCCF)CCC(C(=O)NCC2CN3CCC2C3)CC1 N1(C(CSc2cccc(OC)c2)=O)CCC(C(F)(F)F)C(NC(=O)C(C)(F)F)C1 C(c1ccc2c(c1)CCO2)=CC(=O)NCC1CCN(C(=O)CCN2CCCC2)C1 c1(OCC)ccc(Cl)c(C(=O)NCCCCNC(c2ccn(C(C)(C)C)n2)=O)n1 Cc1noc(Cl)c1CCC(=O)NCCC1(O)CCN(C(=O)CC2C=CCC2)C1 C(=O)(C(C)(C)CN(C)C)NCC(CC=C)NC(C1CC(C)CCO1)=O C(=O)(C1CCCc2ccnn21)NCC(=C)CCNC(c1cnoc1C)=O Cc1cc(Br)cc(F)c1C(N1CC(F)(C(N2CCN3C(=O)CCC3C2)=O)C1)=O Cc1cc(C(=O)NC(CO)C(C)NC(=O)C(C)(C)Cc2cnn[nH]2)cn(C)c1=O N1(C(C(C)=C(CC)C)=O)CC(C)(OCC(=O)NCC2(Cl)CC2(F)F)C1 Cc1[nH]nc2ncc(C(N3CCC4C(C3)CN4C(=O)CCCOC(C)C)=O)cc12 C(C(=O)NCCC(O)CNC(c1csc(-c2ccccc2)c1)=O)(C(C)C)OCC n1(CC)nncc1C(=O)NC1CC(CNC(C2CCCC2O)=O)C1 C1(C(N(C2CN(C(C(COC)OC)=O)C2)C)=O)Cc2ccccc2N1 Nc1c(C(=O)NCC2CC2NC(C2CC3CCC2O3)=O)cccc1Br N1(C(c2cc(F)cc(Cl)c2)=O)CCCC2(CCN(C(c3cc(F)cs3)=O)C2)C1 c1(C(N2CCCC(NC(CC(CC)OCC)=O)C2)=O)cc(C)n(CC)c1C C1(NC(CC=CC)=O)CC(O)CN(C(c2cnn[nH]2)=O)C1 C1(C(N2CC3C(NC(c4c(CC)nco4)=O)C3C2)=O)CCc2cnnn2C1 c1(C(=O)NC(CCCC)CNC(=O)C(C)COC)cc(C(N)=O)cc(F)c1 c1(C(N(C2CCN(C(CCC#CC)=O)CC2)CCO)=O)ccc(Br)c(F)c1C C1(NC(C2(OCC)CCCCCC2)=O)CN(C(=O)C(C)C2CC2)CC2(CC2)C1 c1(NC(C2OCCN(C(c3scc(C)c3C)=O)C2)=O)ncc2cc(Br)ccc2n1 CC1COC2(C1)CN(C(C1CN(C(=O)OC(C)(C)C)CCC1(C)C)=O)C2 N1(c2cccc(C)c2)CCN(C(=O)N(c2cc(C(N)=O)ccc2C)C2CC2)CC1=O CN1CC(NC(=O)CCC2CCN(C(c3ccn(C)n3)=O)C2)C(=O)N1 c1(C(N2CC(CCNC(c3cc(C)cc(N)c3)=O)(OC)C2)=O)c(C)cccc1C C(CC(C(=O)NCCN(C)C(C1C(C)(C)C1(F)F)=O)NC(N)=O)SC c1(C(N2CC(CC(C(=O)NCC(C)N(CC)CC)F)C2)=O)cnn(C)c1C C1(CNC(c2ncccc2Br)=O)CCCCCN1C(=O)C=CC1CCCO1 C1(CCNC(Cc2c(C)nc[nH]2)=O)CCCN(C(=O)COC2CCCCC2C)C1 C(CN=c1[nH]cc(C(C)=O)cc1C)N(C(=O)C=Cc1cccc(F)c1)CC CC1CN(C(c2ccccn2)=O)CC(C)CN1c1cccc(F)c1C#N C1(NC(CCc2cnc(C)s2)=O)CCN(C(=O)Cc2ccon2)CC1C(C)C N1(C(c2cn(CC)nc2)=O)CCC(C(C(C)C)NC(c2ccc(=N)[nH]c2)=O)CC1 CCCC(CC(C)C)C(=O)NCC1(C(=O)NC2(C)CCSC2)CC2(CC2)C1 Cc1ccc(C(=O)Nc2ncc(C(F)(F)F)cc2O)c(C)n1 N1(C(CN(C2CCCC2)C)=O)CCCC1(C)CNC(=O)CP(C)(C)=O N1(CC(=C)C)C(=S)NC(c2nn(C)cc2Br)C2=C1C(c1ccccc1Br)NC2=O c1(OC)ccc(C(=O)N(CC(C)(C)CNC(=O)C(C)NC(=O)C2CC2)C)cc1 N(C1C(=O)Nc2c(Cl)cccc21)c1nccc(=NCc2nnc(CC)s2)[nH]1 c1(C(=O)NC2CN(C(C(C(C)C)NC(C)=O)=O)CC2O)cn(C)c(=O)cn1 C(C)(C(CC(=O)NC1(c2cc[nH]n2)CC1)NC(c1cc(=O)cc(C)[nH]1)=O)OC c1(C(=O)NCCNC(C(c2c(C)nc(C)[nH]2)N)=O)ccc2nc(O)[nH]c2n1 N#Cc1ccnc(N2CCC(NC(=O)CCc3ccc(Br)cc3)C(O)C2)n1 CCC(CC)C(C)C(=O)NC1CCCC1C(N1CCC(CO)C(C)(C)C1)=O c1(C(N2CC(NC(C3(F)CCCC=C3F)=O)C3(CC3)C2)=O)ccc(F)cc1Cl C1(NC(=O)CCSc2ccc(F)c(F)c2)CCN(C(=O)CCC(F)F)C12CC2 C(=O)(C(C)(C)NC(=O)C(F)CC1CCOC1)N(CCCCC)CCN(C)C c1(C(C)=O)cn(CC(N2CCCC2CCC2CC2)=O)nn1.c1(CC(=O)N)oncc1C CC(C)C(C(=O)NC1CC(NC(=O)CCc2ccccn2)C1)N(C)C Cc1ccc(C=CC(=O)N(C)CC2(NC(=O)CC3CSCCO3)CC2)s1 CC(C)(C#N)CCCC(=O)N1CCC(CNC(=O)C2=NNC(=O)C2)C12CC2 C1(C(N2CC(F)(F)C2)=O)(CC)CN(C(c2cccnn2)=O)C1 C(=O)(CC1=CCCCC1)N1CC(CC(N2CCC(CC)OCC2)=O)CC1(C)C C1(NC(c2cncc(Cl)c2)=O)CCC12CN(C(c1cncc(C3CC3)c1)=O)C2 C(CC(C(=O)N1CC(CC(F)F)C1)NC(C1CCC1N(C)C)=O)OC CC(C)C1=NOC(C(=O)NCCC(O)C(=O)NC2CCCC2(C)CO)C1 CC1(NC(=O)CCC2CCCCO2)CCCC(F)(F)C1O C1(NC(Cc2c(F)ccc(C)c2)=O)CN(C(c2nocc2Cl)=O)CC1S(C)(=O)=O C=CC1(CC(N2CCC(C)CC2CNC(C2(F)CCOC2)=O)=O)CCOCC1 c1(OC)ccc(C(=O)NC2(C3CCCCN3C(C3CC(C)C3)=O)CC2)cn1 c1(C(N2CC(C(C)C)N(C)CC2)C(=O)NCC2CC2)cc(Br)cc(Cl)c1F C(=O)(C(O)CC(C)(C)C)NCCc1c(CNC(COC(CC)CC)=O)nco1 c1(CC(=O)NC(CN(C(C2CC2CF)=O)CC)C)ccc(-n2cnnc2)cc1 c1(C(=O)NC(C(C)C)CCOC(F)(F)F)ccc2c(c1)C(C)(C)CN2 C(=O)(CCCCCBr)NCc1nccc(C(=O)NCC(=O)NCCO)c1 C#Cc1ccccc1CC(=O)NC1(CCOC)CCN(C(=O)C(C)C2CC2)CC1 C1(C(N2C(C)CC(NC(c3occc3Br)=O)C2)=O)CCc2c[nH]nc2C1 N1(C(C(C)OC)=O)CCN(C2CCCN(C(c3csc(C(F)(F)F)n3)=O)C2)CC1 Cn1cnc2cnc(N(CCNC(c3ocnc3-c3ccccc3)=O)C3CC3)nc12 C=CC1CN2CC1NC(=O)CCCC2=O.C(=O)(CS(=O)(=O)NCC)N(C1CC1)CC c1(C(N2CC(SC)C(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)c(N)cccc1Cl N1(C(C(CCCC)F)=O)CCC2CCC(NC(c3cc[nH]n3)=O)C1C2 c1(C(=O)NC2CCC(NC(=O)CCCC3CCOCC3)C2)ccccc1Br c1(C(N2C3C(C(=O)OC)C(C3)C2)=O)cc(NC(=O)C(F)C(C)(F)F)cc(C)c1 C1(NC(c2cccc(C(N(C(C)SC)CC)=O)c2)C(=O)NC)CCC2(CC1)CC2 C12(C)CCN1C2=O.C1(CN(C)C(=O)OC(C)(C)C)CCN(C(=O)C=C2CCC2)C1 C1(CC(=O)NCC2CCC(C)CN2C(C2CCCC2)=O)(OC)CCC(C)(C)CC1 C1(CC=C)(NC(c2cc(C3CC3)on2)=O)CN(C(c2coc(C)n2)=O)C1 C1(NC(C(c2cn(CC)nc2)=O)=O)CCCCC1CNC(=O)C(C)C c1(C(C)C)cc(C(=O)NC2CCOCC2SC(=O)O)c(C(C)C)o1.C12CCN1C(=O)C2.C.N C1(C(=O)NCC(C)(C2CC2)NC(c2c(CC)cno2)=O)Cc2nccn2C1 Cc1cnn(CC(=O)NOCC(=O)NCCCC2CCCCC2)c1 Cc1c(C(=O)NC(C)CNC(c2coc(C#N)c2)=O)c(C)n(C)c1Br c1(N2CCC(c3ccc(C)cc3)CC2)ncnc2c1ncn2CCC1(CSC)CC1 Cc1ccc(CCC(=O)NC2CC(C)N(C(c3ccc(=O)n(C)c3)=O)C2)cc1Cl N1(C(COC(CC)C)=O)CCCN(C(=O)C=Cc2ccsc2C(F)(F)F)C(C)C1 c1(C(=O)NCC2N(C(CC3(C)CCCC3)=O)CCC2)cccc(NS(C)(=O)=O)n1 N1(C(CC(CC)OC)=O)CC2CN(C(c3cc(C)cc(C)n3)=O)CC2C1 Clc1nc(Nc2cnn(C3CC3(F)F)c2)c2[nH]ccc2n1 C1(C(=O)O)CC2(CCSCC2)CN1C(=O)Cc1csc(-c2ccco2)n1 C(CCCCC(=O)N1CCC(C)(CC(=O)NCCC2(CO)CC2)C1)N(C)C C1(CCC)CN(C(c2cc(COC)ccc2Cl)=O)CCN1C(=O)CC(C)(C)F Cc1cc(C(=O)C(=O)NCC2CC2NC(c2cccnc2C(F)F)=O)ccc1F c1(C(=O)NC2CCCN(C(c3cncc(C)n3)=O)C2)sc(Br)c(C)c1C CC1(C)CCC(C(=O)NC2CC3(C2)CC3NC(=O)CCn2cnccc2=O)CO1 C1(F)(CNC(c2c(C)ncnc2)=O)CCCN(C(c2ccc(C3CC3)cn2)=O)C1 c1(C(=O)NCCC(C)NC(c2cc(C)cc(Cl)c2)=O)ccc(F)c(Cl)c1N C1(NC(C2CCC3(CC3)C2)=O)CCN(C(=O)CCCCc2cnc[nH]2)CC1O c1(OC)ncc(C(=O)NC(CNC(=O)CCSC(F)(F)F)C(C)C)cc1C c1(C(=O)NC2C(OC)CN(C(=O)CC(O)C(C)C)C2)nc2ccccc2s1 N1(C(CN(C)CC)=O)CCCN(C(c2ccc(C(C)C)c(C)c2)=O)CC1C(C)C CCC(C)(C)C(O)C(=O)N1CCC(N(CCO)C(=O)OCCl)C1.C(C)(C)C c1(NCC2(O)CN(C(C(C)(C)NC(C)=O)=O)C2)nc(C)nc2c1cnn2C C(=O)(CC(O)C(C)C)NC(CCC(=O)N1CC(O)(CC=C)C1)C c1(C(=O)OCC(=O)Nc2c(OC)cc(NC(C)=O)cc2)ccc2c(c1)CN(C)C2=O c1(OC)ccnc(CNC(C2(C)CC(NC(=O)CC3C=NN(C)C3=O)C2)=O)c1 CC(CN1CCOCC1)C(=O)NCC1(F)CC(NC(C2(c3cc[nH]n3)CC2)=O)C1 N1(C(C(CC=C)C)=O)C2CCCC1CN(C(C1(F)CCOCC1)=O)C2 CS(=O)(=O)CCCC(=O)NC1(CF)CCN(C(=O)CCC2CCOCC2)C1 CC1(c2nn[nH]n2)CCN(C(c2cnc(OCF)cn2)=O)C1 c1(C(=O)NC2C(NC(CCCCC)=O)COC2)cc([N+](=O)[O-])c(C)c([N+](=O)[O-])c1 O=C1CCCC(NC(=O)c2ccc(C(=O)NC3CCN(CCC(=O)O)C3)cc2)CC1 c1(SCC(N2CC(NC(=O)Cc3cccnc3)(CO)C2)=O)ccc(F)cc1 c1(N2CCC3(CC(NC(c4ccc[nH]4)=O)C3)C2)c(F)cc([N+](=O)[O-])cc1F c1(COCC)nc(N2CCC(CC(=O)NCC3(C)COC3)C2)cc(C)n1 c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)CC(C)(C)C2)cc2c(nn1)CCCO2 Cn1nnc2cc(C(N3CC(NC(=O)COCC4CC4)C4(CC4)C3)=O)sc12 Cn1ccc(C(=O)NCC(CNC(c2ncccc2C(F)F)=O)CO)cc1=O N1(C(Cc2c(CC)cccc2)=O)CCN(C(c2ccc(C)cc2)=O)C(CCO)C1 c1(C(=O)NCC(CC(C)C)NC(=O)C(Cl)=CCl)ccc2nnc(O)n2c1 CCC1=NOC(CNC(C2CC(NC(c3coc(CO)c3)=O)C(O)C2)=O)C1 C(C(C)(C(=O)N1CC=CC(O)C1)NC(c1ncsc1C)=O)SC CCCCCC(F)C(=O)NC(C1(O)CCCCC1)CNC(C1C=CCC1)=O c1(C(=O)NCCC2CN(C(CCC(=O)NC)=O)CC2C)cnc2c(c1)COCC2 C1(NC(C2CC2(F)F)=O)CCCCN(C(=O)Cc2csc(Cl)n2)C1 N1(C(=O)NCC2(CCO)CC2)CC2CCCCN2c2ccccc21 C(C(C(=O)NC1CC(F)(F)C1)N1CCC(C(O)CO)CC1)(C1CC1)OCC CC1(C)CCC(N=c2cccc(S(=O)(=O)NCCC3CCCCC3O)[nH]2)C1 C1(CNC(c2ncc(C(=O)OC)nc2)=O)CCCCN(C(=O)CC(C)(C)C)C1 N1(C(C(CC)OCC)=O)CCN(C(c2cccc3c2COC3)=O)C2COCC12 C1(C#C)(C(NOCCCC#C)=O)CCN(C(C2CC(C3CC3)=NO2)=O)C1 n1(CC(N2CC(NC(C3(n4cncn4)CC3)=O)C3CC23)=O)cnc([N+](=O)[O-])c1 c1(C(N(c2ncc(OC)cn2)C2CC(N)C2)=O)ccc(F)c(C)n1 C1(C(=O)NCC(CC(C)C)NC(CNC(CC)=O)=O)CCC(F)(F)CO1 c1(N2C(C(C)(C)NC(C(C)n3ccnc3)=O)CCC2)nc(Cl)nc2[nH]cnc12 c1(C(N2CC(N(C(c3c(OC)csc3)=O)CCO)C2)=O)ccc2c(c1)CN(C)CC2 N1(C(C(C2CC2)NC(C2CC(O)C(F)C2)=O)=O)Cc2cncnc2C1 C1(NC(Cc2cccc(OC)c2)=O)CCN(C(C2OCCO2)=O)C(C)C1 C1(CCNC(CCOC(C)C)=O)CSCCN1C(=O)Cc1coc(C(F)F)n1 c1(COCC)nc(Cl)cc(=NC2CC(CNC(C3CC3F)=O)C2)[nH]1 N1(C(C(CC)OC)=O)CCC2(CCN(C(c3cc4cccc(Cl)c4s3)=O)C2)C1 c1(C(=O)NCC(CNC(Cn2c(C)cnc2)=O)O)cc(O)cnc1N C1(CNC(Cc2ccc(C)s2)=O)CCC2CN(C(C3CC3C#N)=O)CC12 c1(C(N2CC(N(C(C(COC)(C)OC)=O)C)C2)=O)cnc2c(C)cccc2c1 C#CC1(O)CCN(C(=O)CNC(=O)CCCCOCC)CC1 C=CCC(C)(C)CC(=O)NCC1CCCC1NC(=O)Cc1cccc(F)c1O c1(-c2cc(C)c(OC)c(C)c2)ccc2c(CC(N3CCC(C)(O)C3)=O)n[nH]c2c1 Cc1cc(CNC(=O)NC2CN(C)CCN2C)c(N(C)C)nn1 CS(=O)C=CC(=O)NCCN(C1CCCCCC1)C(c1ccc(C2CCC2)nc1)=O c1(CC(N2CCCC(N(C(=O)C(F)C(F)(F)F)CC)CC2)=O)ccc2c(c1)CCO2 N#CC1(C(=O)NC(CNC(=O)C(C2CCOCC2)F)CO)CCCCCC1 C(=O)(C(CCC1CCC1)NC(c1nonc1N)=O)N(C)Cc1ccsc1 Cc1sc2ncc(C(=O)NC3CCCCC3n3cccn3)n2c1C Cc1cc(C)n(C(C)C(=O)NC(C)CCCCNC(c2cc(C(C)C)[nH]n2)=O)n1 O=C(CCN(C1CCC1)Cc1ccccc1)N=c1nc(-c2cccnc2Cl)[nH]s1 N1(C(COCCCC)=O)CCN(C(C2(C)CC(C)=NO2)=O)CC1C c1(C(N2CCCC(NC(c3c(C)ncc(N)c3)=O)C2)=O)cc(S(N)(=O)=O)co1 C#CC1(NC(C2CCCC2NC(=O)C=Cc2nccs2)=O)CCC(C)(C)C1 c1(C(C)C)cnc(O)c(C(=O)NC(C)(CNC(=O)CCC=CBr)C2CC2)c1 N1(C(c2c(C(C)C)occ2)=O)CC2(CC(NC(c3cnncc3O)=O)C2)C1 c1(C(N2CCCN(C(c3cc(C)ns3)=O)CC2C)=O)cc2cc(O)ccc2[nH]1 c1(NC(C(CO)NC(c2cc(C)cc(O)n2)=O)=O)cccc(C#N)c1C N1(C(c2c(C(C)C)ncs2)=O)CC(NC(C2CC(C)(C)C2)=O)C(C2CC2)C1 Cc1ccc(C(=O)NCC(C2(O)CCN(C(=O)Cc3nncn3C)C2)C)nc1O C1(C)(C(N2CC=CC(NC(c3cc(C)oc3)=O)C2)=O)CCCCC1(F)F c1(C(N2C(C)(C(N(C3CCN(C)C3)CC)=O)CC2)=O)ccc(CO)cn1 c1(OC)cnc(F)c(C(=O)NC2CCCCC2CNC(=O)CCC(=O)N(C)C)c1 C1(NC(=O)Nc2cccc(C)c2CO)CCCC2(CN(C(=O)OC(C)(C)C)C2)O1 c1(C2C(=O)NCC(C)N2CC(=O)NCCC)cc(OC)c(F)c(F)c1.C(=O)OC c1(C(N(CC(N)=O)CC=CC=C(C)C)=O)cccc(-c2nccs2)c1 N1(CC(C)O)CCCN(C(C2CCC(NC(=O)C(C#N)C3CC3)CC2)=O)CC1 C1(NC(C(C(CC)C)O)=O)CC2CCC1CN2C(c1cc2c([nH]1)CCCC2)=O CCCCCC(F)C(=O)N1CC(OC)C(C(=O)NCCCc2cccs2)C1 C1(NC(c2nnc(C)s2)=O)CC(CNC(=O)Cc2cc[nH]c2)C12CCC2 N1(C(c2c(CC)onc2)=O)CCN(C(C)CNC(=O)C(C)(COC)OC)CC1 CC(CC(=O)N1CCC(C(C)(C)NC(=O)Cn2cccc2)C1)C(F)F Cc1ccncc1N(C(=O)C(C)CNC(=O)COC1CCCC1)C c1(C(C(=O)NC(CNC(C(c2cncnc2)C)=O)C2CC2)(C)C)ccccc1F c1(COCCCC(=O)N(C2C3CN(C(=O)C(C)(C)O)CC23)C)ccc(F)cc1 N12CC3(C1)CN(C(C)(C)C)CC3c1ccccc12.c1c(F)c(Br)c(F)c(Br)c1F.c1(C(C)CCCC)ccccc1 CCCN=C(NCc1nc(COCC)no1)NCC(C(F)(F)F)N1CCOCC1 c1(OC)cc(C)c(S(N)(=O)=O)cc1C(=O)NC(C)C(C)(Cl)CC c1(C(N(CC(CNC(C(F)OC)=O)C)C)=O)ccc(C(N)=O)c(Cl)c1 N1(C(C2(NC(c3ncn(C)n3)=O)C(C)CCC2)=O)CC=C(CO)CC1 C(CN=C(NCCc1cccs1)N1CCC(n2cc(Cl)cn2)C1)N1C(=O)NCC1 C1(O)(CNC(c2c(CC)cco2)=O)CCCN(C(c2ccncc2C(F)F)=O)C1 c1(C(N(C)CC2N(c3nnc(C)s3)CCC2)=O)nn(C)c(Cl)c1Cl c1(OC(CNC(CCC(=O)NC)=O)=O)ccc(C(F)(F)F)cc1Cl c1(NC(c2c[nH]c(=NC)o2)=O)cc(CC(N2CCC2)=O)ccc1C.CCC=CC CC1CCC(C(=O)NCc2cccc(C#N)n2)N(C(c2csnn2)=O)C1 c1(CC(=O)NC2(C)CN(C(c3cc(CC)no3)=O)C2)ccc2nsnc2c1 C1(C)(NC(c2ncn(C)n2)=O)CCN(C(c2cc(C(F)(F)F)ccc2Cl)=O)CC1 N1(C(C(CCN(C)C)NC(CCOC)=O)=O)CC2C3CCC(C3)C2C1 CC=C=CCCN=C(NCc1csc(C(F)(F)F)c1)NC1CC1C N1(C(c2ccc(F)s2)=O)CCOC2(C1)C1CC3CC(C1)CC2C3 C1(NC(C=CCN(C)CC)=O)C2CC(NC(=O)C(c3c(C)noc3C)C)CC12 C1(CNC(C(CCC=C)(F)F)=O)CCCC2CN(C(C3CCC(C)O3)=O)CC12 CCC(F)(F)CC(=O)N1CC(C(=O)NC(C)(COC)CCO)(COC)C1 C(CC(=O)N(CC)CC)(C(F)(F)F)NC(C(N1CCC(C(C)C)(CC)C1)CC)=O O=C1CC(C(=O)N2CCC(NC(=O)CSc3ccc(O)cc3)C2)=NN1 c1(C(=O)NCC2(C)CCCN(C(C3(C#N)CC=CC3)=O)C2)nnn2ccccc12 C=CCCCCCC(=O)NCCCCC1(NC(=O)C(F)CCC)CC1 c1(OC)cc(OC)c2cc(NC(c3ccc(C)c(CN)c3)=O)ccc2c1 C1(CNC(CCC(=O)OC)=O)CN(C)CCN1C(C1CCN(C)C1C)=O N1(C(CC2(C=C)CC2)=O)CC(NC(c2c(CC)cccc2F)=O)CC(C)C1 O(NC(=O)CCC(C)NC(C12CCN(CC1)CC2)=O)C(C(=O)OC)(C)C Fc1ccc2c(c1)OCCC2NCC1CCCC2(CNC2)O1 C1(C(N(CCCN(C(C2CN(CC)C(=O)C2)=O)C)C)=O)CCN(C)C(C)C1 C(=O)(C(CCC)OC)N(CCC(=O)NC(c1nc(CC)[nH]n1)C)CCO c1(CN(C(=O)NCCCOC2CC(NC(C)=O)C2)C(C)C)ccccc1 c1(C(=O)NCCC2CC(NC(CCCSC)=O)C2)cccc(N2CCOCC2)n1 C(CCCC(=O)N1CC(c2ccc(Cl)cn2)C1)N(C(C)=O)C N1(C(C=C(C)Cl)=O)CC2CC3CC2C1C3NC(=O)C=Cc1cccc(Cl)c1Cl c1(-c2cc(CC(=O)Nc3c(OCC)cnnc3)ncc2)cnc(F)cc1C C1(C(N(CCN(C(C2CC(C(F)(F)F)(OC)C2)=O)C)C)=O)COC2(CCC2)C1 c1(C(=O)NC(C2(O)CN(C(c3cnn(CC)n3)=O)C2)C)ccc(OC)nc1 c1(C(=O)NCC23CCC(CC2NC(C24CC(F)(C2)C4)=O)C3)cc2cc[nH]c2cn1 c1(-c2n(CC)c(N3CCOC(C(C)(C)O)C3)nn2)nc2c(Cl)ccnc2[nH]1 C(=O)(C(CC(C)C)NC(=O)CCC1CCCO1)NC(C(=O)NCCC)(C)C CC1CN(c2ccnc(N3CC4(CCOC4=O)C3)n2)C(C)(C)CO1 c1(C(=O)OCC)c[nH]c(=NCC2(C)CCN(C(=O)C(C(C)C)N(C)C)C2)s1 Nc1ncc(C(=O)NC2CCN(C(=O)Cc3csnn3)C2)cc1CO N1(C(C(C)(C)OCC)=O)CCC(NC(=O)CCOc2ccccc2C)C(C)C1 C1(CCN(C(=O)C(C2CC2)N(C)C)C)CCN(C(=O)CCC2(C)N=N2)CC1 c1(OCCC(=O)Nc2ccc(NCC)cc2)cc(C)ccc1OC C(=O)(C(O)C(F)(F)F)N1C(CNC(C2CCC(CCC)CC2)=O)CC(COC)C1 C(N=c1[nH]nc(C(F)F)o1)C1CN(C(C=CCC)=O)CC1C(F)(F)F Cc1cc(C(N2CCC(CC(=O)NC(C3CCCC3)C)C2)=O)cc(C)c1F N1(S(CC(=O)OCC)(=O)=O)CCCN(C(c2cc3ncccn3n2)=O)C(C)C1 C(C)(N=c1ccnc(NCc2csc(-c3ccccc3)n2)[nH]1)c1c(CC)nns1 c1(SC(C(C)C)C(C)NC(=O)Cc2cnccc2Cl)ccc2ccccc2c1 c1(CC(C(=O)NC(C)(C)CNC(=O)CC(C)F)OC)ccc(F)cc1 N1(C(CCC#C)=O)CC2CC(NC(=O)CSCc3ncc[nH]3)CC2C1 c1(CC(=O)NCCN(CCOC)C(C23CC(C)(C2)C3)=O)ccccc1F C1(C(N(C2CCS(=O)(=O)C2)CC)=O)CCCCN1CC(=O)NC1CC2C=CC1C2 c1(CC(=O)NCC(C2CCOCC2)(C)OC)nc(C)sc1Cl Nc1cc(C(=O)NC2C3CN(C(C4(Oc5ccccc5)CC4)=O)CC23)ccc1F C1(NC(C23OCC(COC)(C2)C3)=O)COC2(C1)CN(C(=O)C(C)CC1CCC1)C2 CCC(C)(O)C(=O)NC(C)(C)CCC1CCCCN1C(=O)CS(=O)(=O)NC S(=O)(=O)(c1cnnc(C)c1)NC(CCC(=O)OCC)C n1(CC)nc(C(=O)NCCC2CCCN(C(c3ccncc3)=O)C2)c(Br)n1 C1(C(N(C2CC2)Cc2ccc(OC)cc2)=O)Cc2ncccc2N1CC(C)(C)O c1(NC(c2nc(C)n(C)c2C)c2n(CC)nnn2)nc2cnccc2[nH]1 N1(C(CSc2c(C)n[nH]c2C)=O)C2CCC1CN(C(=O)C(C)C(C)C)CC2 N1(c2ncc(C)cn2)CCC(O)C(C(=O)NC2CCN(c3ncccn3)CC2)C1 C1(NC(Cc2cccc(C)c2)=O)CC(O)CN(C(c2cnccc2C)=O)C1 C(=O)(C1=CCCCC1C)NCCC1CC(C(=O)NC(C(=O)OC)(C)C2CC2)C1 N1(C(CCOC2CN(C(c3c(C)cc(F)cn3)=O)C2)=O)CCC(O)C(C)(C)C1 C1(COC)(NC(=O)Cc2cn(C)nn2)CCN(C(=O)CC(C)(C)O)C1 c1(CN(C(C)CNC(=O)Cn2cnnn2)C)cn(C)nn1 c1(CN(C(=O)CCC2(C)CC2)C)cccc(CNC(=O)C(C)(C)c2cnco2)c1 C(=O)(C(C)(O)CC(C)C)NC(CNC(c1cc(C)c(O)cc1)=O)C c1(C(=O)NCCC(C)N(C)C(c2cscc2Cl)=O)cccc2oc(C(N)=O)nc12 Nc1ccc(C(N2CCC(NC(C3CC4CC3C4)=O)CC2)=O)cc1Cl n1(CC)nnc(C)c1C(N1CCC(OCCCNC(=O)C(C)(C)CF)CC1)=O N1(C(c2c(C)ocn2)=O)CCC(C(=O)NOCCOCCF)CC1(C)C c1(C(N2C(C)C(NC(C3(C)CC=CC3)=O)CCC2)=O)cccn2c(CO)nnc12 Cc1nn(C)c(C)c1C(=O)NC1CC(C)CN(C(c2cccn(C)c2=O)=O)C1 C1(F)(CN(OCC)C=O)CCCN(C(c2ccc(C(C)=O)o2)=O)C1 c1(C(=O)NCC2CC(OC)CN2C(c2cc(C)cc(F)c2)=O)c(C)cncc1F c1(N2CC(COC)OCC2)cc(C)c(S(=O)(=O)NCC(Cl)(Cl)Cl)cn1 c1(OC)ccc2nc(N3CCCC(N4CCOCC4)C3)sc2c1 Cc1nc(F)ccc1-c1cn(CC(=O)N(CC2CCC2)CC2CC2)nn1 c1(NC(c2cccc(CC)c2)c2n(CCS)nnn2)ccc(C)c(F)c1F.CCNC c1(NC(c2cc(CNC(COCC(=C)C)=O)no2)=O)cccc2ccoc12 C(C(CNC(c1cc(Cl)cn1C)=O)C(F)(F)F)NC(C(C=C)O)=O C(=O)(CCC(F)(F)F)NC(C1CCCN1C(c1ccc(C2CC2)cc1)=O)C C(=O)(CCCCCC#N)NCC(C(C)(C)C)NC(c1c(C)nn(CCC)c1C)=O Cc1cc(Br)sc1N(N1C(C(NNC(=O)C2CC2)=O)CC1)C(C)(C)C.C=O c1(CC)conc1CC(N1CC(C(C(=O)N(CC(F)Cl)C)OC)C1)=O c1(C(N(C2CC(NC(=O)Cc3ccoc3)C2)C)=O)cnc(O)cc1C(F)(F)F CON=CC(=O)NCC(C)(Cn1cccn1)NC(c1ccsc1Br)=O C1(CC(=O)NCC(CN(C(=O)CN2CCC(C)(C)C2)C)(C)C)CC2CCC1C2 C(=O)(C(C)(F)C(F)(F)F)NCCCc1cn(-c2scc(C(=O)OCC)n2)nn1 c1(C(N2CC(CCNC(C=CCCC)=O)C(C)C2)=O)ccc2c(n1)OCC(=O)N2 c1(N2CC(CNC(C(CC#C)(C)C)=O)N(C)CC2)nc(C)nc2c(C)csc12 c1(C(C)=O)cccc(OC(C)C(=O)N(CCCCCNC(=O)C(=O)N(C)C)C)c1 CC1(CNC(=O)CC2CCCCC2O)CCCC1NC(=O)Cc1ccno1 c1(CCC(=O)NCCC2CCN(C(=O)C3=CCSC3)C2)ccc(Cl)cc1F c1(C(N2CCCC2CCNC(C23COCC2C3)=O)=O)cnn2c1S(=O)(=O)NCC2 CCC(C)C(C)(O)CNC(=O)CCN(C(c1c[nH]c(C)c1)=O)CC1CC1 c1(C(=O)NCCN2C3(CC3)C2=O)noc(C2(C)CC2(F)F)n1.C(C)=O.CCS C1(CNC(CC(=C)C)=O)C(C)CCCN1C(=O)COCC=C c1(CNC2(c3nnnn3CCCOC)CC(COC)C2)c(F)cc(Cl)cc1F N1(C(c2cc(C(C)=O)sc2)=O)C2CCC1CN(C(c1cc3n(n1)CCCC3)=O)C2 C(=O)(CC(N=c1ccc(Br)c(S(=O)(=O)NCc2ocnc2C)[nH]1)C1CC1)NC C(=O)(C1=NN(C(C)C)C(=O)CC1)N1CC(O)(CN(C(C(CC)F)=O)C)C1 c1(C(=O)NC2(CF)CCN(C(c3n(CC=C)ccc3)=O)C2)cn(C)ccc1=O Cc1cccc(C(=O)NC(c2cn(C)nn2)C(N2CCOC(C3CC3)CC2)=O)c1C C1(C(N2CC3(CN(C(CC4CCC(=O)C4)=O)C3)C2)=O)CCC2C(C1)C2(F)F Cc1cccn2ncc(C(=O)NC3CC(NC(=O)CC4CC5CC5C4)C3)c12 Cc1sc(C)c(C(=O)NCCN(C)C(C23CC(CCO2)C3)=O)c1Br c1(SC)cc(C(=O)N=c2ccn(C)[nH]2)c2cc[nH]c2c1.c1ncc2c(n1)NC(=O)C2 N1(C(c2ccc(F)cc2Cl)C(=O)NCC(F)F)CCCCC12CCC2 N1(C(CC2(N(C)C)COC2)=O)C2CCC1CN(C(C1CCS(=O)(=O)N1)=O)C2 Cc1ncccc1CCC(=O)NC1CN(C(c2cccs2)=O)CC1O c1(C(N(C(C)C(=O)NC(C2(CO)CC2)C)CC)=O)ncccc1F C1(C)(C(=O)NCCN(CC(C)O)C(c2cnnn2C)=O)CCCN(C)C1 C1(OC)CC(NC(=O)C(C)CC2CC2)CN(C(=O)CC23CCCN2CCC3)C1 c1(C(C)C)ccc(C(N2CCC(OCCNC(C3(C)CCCO3)=O)C2)=O)c(F)c1 Cc1ccc(C(N2CC(NC(=O)COCC3CCC3)CC(F)C2)=O)c(F)c1F c1(C(C)NC2CCN(c3ccc(Cl)nc3)C2)[nH][nH]c(=N)c1-c1ccccc1 Cc1cnc(C(N2CC(CC(C)NC(=O)CC(O)C(C)C)C2)=O)cc1C#N N1(C(COC(C)(C)C(F)(F)F)=O)CC(F)(F)CC1CNC(C1CC1(C)C)=O N1(C(C2C(CCC)CN(C(=O)CC3(C)OCCO3)C2)=O)CCC2(CCCC2)CC1 N1(C(C(C)N(C(c2c(C)oc(Cl)n2)=O)C)=O)CC(CO)CC(C)C1 c1(C(C)=O)ncnc2c1ccn2CC(=O)NC1(C)CN(C(=O)C(C)C(C)O)C1 C1(C(=O)NC2(CNC(=O)CCCc3cccnc3)CCOC2)OC2CCC1CC2 C(=O)(CCCCCC#N)NC(C(C)NC(CCC(=C)Br)=O)(C)C Cc1ccc(Br)c(CCC(=O)OC(C)(C)C)c1.C12(CF)CCN(C1)C(=O)NC2 c1(C(C(N2C(C(C)NC(C)=O)CCC2)=O)C)ccc(N(C)C)cc1 c1(CC(=O)NCC2(NC(C3C(C#C)C3)=O)CCOCC2)cccc2nonc12 C(C(CC)(CC)C(=O)NC1CC(O)C(O)C1)NC(c1ncc(CC)cn1)=O c1(C(N2CC(C)C(CNC(=O)CCc3ccncn3)C2)=O)c(F)ccnc1F C1(N(C(=O)Cc2ccon2)C)CCCC(N(C)C(c2ccsn2)=O)C1 C(=O)(CC(C)C(C)(C)NC(=O)CCc1cnn(C)c1)NCC(C)S(N)(=O)=O c1(NC(c2n(CC)c(O)nc2)=O)ccnc(N2CCOCC2)c1I C(C(C)C(F)C(=O)NC1(CCOC)CCCC1)NC(COCCCOC)=O c1(C(N2CCC(N(C(CN(CCC#C)C)=O)CCC)C2)=O)ccc(C)cc1 C1(CNC(CN(CC)CC)=O)C(C2CC2)CCN1C(c1ncnc2sccc12)=O c1(CC(N2CCC(NC(=O)C(Cl)(Cl)Cl)C2)=O)ccccn1 N1(C(C2CCN(C)C2=O)=O)CCC(O)C(NC(C2(CC3CCC3)CC2)=O)C1 C(=O)(C(C(=O)OCC)C(C)C)NCC(C)N(C(CC(C=C)(C)C)=O)C O=C1CCC(CNC(=O)CN(C2CCC2)C(c2ccn(C3CC3)n2)=O)N1 N1(C(c2c(OC)c(C(F)F)ccc2)=O)CCCC12CCN(C(=O)COC(F)F)C2 N1(C(c2n[nH]c(CC)c2C)=O)CC2(C)CC1(C(N1CC(C)CCC1C)=O)C2 C1(C(=O)NCCCN(C(c2ccc(CO)nc2)=O)CC)CC2CCCC2C1 C1(C(C(=O)N(CCC(N)=O)CC)(C)C)CCCN(C(=O)CC(C)C)C1 c1(C(=O)NCC2C(NC(C(C)Cc3ccco3)=O)C2)cccc2c1CNC2=O Cc1cccc2cc(C(N3CCC4CN(C(C5CSCCS5)=O)CC34)=O)oc12 c1(NCC2C(NC(CCC(C)SC)=O)CCC(C)(C)C2)cccc(F)c1[N+](=O)[O-] Cc1cc(C(=O)NCC(C)(F)CNC(C2CCCCO2)=O)c(Cl)cn1 c1(C(N2CC(CN(C(C(C)SC)=O)C3CC3)C2)=O)cc(C)nn1-c1ccccn1 N1(C(=O)CC2CC(NC(C3CCC(F)C3)=O)C2)CCc2cc(O)ccc2C1 C1(C(N(C)CC2CCN(C(c3cccc(C)c3Cl)=O)C2)=O)CC2(CCCCO2)C1 N1(C(c2cc(C)on2)=O)CC(NC(c2ccc(OCCC(C)C)cc2)=O)C(O)C1 C12(NC(c3n(CC)nc(C)c3)=O)CCCN(C(=O)Cn3cnnc3)CC1C2 c1(OC)cc(C(=O)NCC2CC3CC3N2C(c2ccnn2C2CC2)=O)cc(F)n1 C(=O)(CCCC(F)(F)CO)NC(CCCCNC(C=CC(C)(C)C)=O)CO O=C1CC(C(=O)NCCC2CN(C(=O)CC3CCCS3(=O)=O)C2)c2ccccc21 CCS(=O)CC(=O)NCCc1ocnc1CNC(=O)C=CS(C)=O C1(NC(c2c(SC)scc2)=O)CCOC2(CCN(C(=O)CSC(C)C)CC2)C1 c1(C(N2CC(F)(CNC(C3C(C)(C)CC3)=O)C2)=O)ncn2cc(Br)sc12 c1(C(=O)NC(C(C)NC(C(COCC)(C)C)=O)C)ccc(OC)c(F)c1 C(=O)(CC(c1cccs1)C1CC1)NC(C1CN(C(C2(n3ccnn3)CC2)=O)C1)C c1(C(N2CC(N(C(=O)Cc3cc[nH]n3)C)C(F)C2)=O)cnc2c(c1)N(C)CCO2 C1(O)(CCNC(C2(Cl)C(C)(C)C2)=O)CCCN(C(=O)Cc2ccsc2)C1 c1(NC(C2(C)N(C(c3n(C=C)nnc3)=O)CC(O)C2)=O)cnc2[nH]cnc2c1 n1(CC(=O)NC2CCN(C(C3CCCOC3)=O)C2)cnc(Br)c1Br C1(C(N(CCC=C)C2CC2)=O)(SC)CN(C(=O)C(C2CCCCC2)O)C1 N1(C(C(C=C)O)=O)CCN(C(CN2CCN(C(=O)NC)CC2)=O)CC1.C1(=O)CCN1 C(=O)(CCCS(C)(=O)=O)N1C(CNC(C2N(CCC)CCCC2)=O)CC(CC)C1 C1(CNC(C2C3COCC23)=O)CCCCN1C(C1(F)CCCC1)=O N1(C(C2C(CCOC)C2)=O)CC(CNC(c2cc(Cl)c(C)cn2)=O)C2(CC2)C1 C1(CCNC(c2c(C)[nH]cc2)=O)CC(F)(F)CN1C(=O)CNc1cccc(F)c1 C1(NC(N)=NC2CCCC(F)C2)CCCCC1C(N)=O.c1(OC)nscc1C N#Cc1ncc(Br)cc1NC(C1CCCN(Cc2c(O)cccc2Br)CC1)=O C1(OCC)CC2CCC(C1)N2C(=O)CC(=O)NC(c1cn(C(C)C2CC2)nc1)=O C#Cc1ccc(C(=O)N(CCCNC(c2nn(C)cc2C)=O)CC)c(F)c1 C(=O)(C(C(C)CC)NC(=O)CN1CC2CCC1C2)N(C(C#C)C1CCC1)C Cn1nnc2c1CCN(C(c1cc(CO)on1)=O)C2.C12(CCC1)CCNC2=O Cc1nn(Cc2ccccc2Cl)c(=O)n1C1CCCC1 CC1CN2CCN1C(C(N1C3CCC1C(CNC(=O)C(CO)NC(N)=O)C3)=O)C2 N1(C(C2CC2F)=O)CC2CCCC(C1)N2C1CCc2c(Cl)cccc21 CCC(C)CCC(O)CC(=O)N1CCC(NC(C2CCSCC2)=O)C1 c1(C(=O)NC2CN(C(C3(CC=C)CCC3)=O)CC(F)C2)cc2nc[nH]c2cc1F C1(NC(C(C)N(C(C)=O)C)=O)CC12CCN(C(=O)COCC(F)(F)F)C2 C(CCN=C(NCCC1CCC1C(F)(F)F)NC1CCS(=O)(=O)C1)OCC c1(CC)nccnc1C(=O)N(C)CCOCCN(C(=O)C=Cc1ccncn1)C c1(C(=O)NCCC2N(C(C3NC(=O)OCC3)=O)CCC2)cn2ccnc2cn1 Cc1cc(-c2ncc[nH]2)ccc1NC(c1cnc(C2CCOCC2)o1)=O c1(SCC(=O)NCC2CC(NC(C3CC(=C)C3)=O)C2)ccccc1[N+](=O)[O-] C1(CCCNC(C2CCOCC2)=O)CCCN1C(=O)C(=C1CCCCC1)F C(=O)(CC(C)C(C)C)N1C(CN(C(c2nn(CC)c(C)c2)=O)C)CCC1 C1(C(N2C(CN(C(CC(C)OC)=O)C)CCCC2)=O)CCc2ncccc2C1 C1(CC(=O)NCC(CNC(CC=CC)=O)O)CCCCN1C N1(C(CC2(CC)CCC2)=O)CC=C(C(=O)N(CCC(O)CO)C)C1 C1(NC(CCOCCOC)=O)CC(NC(c2oc(C)cc2C)=O)CC1O C1(C(C)NC(=O)Cc2cnc[nH]2)CCN(C(C2(C3CCCCO3)CC2)=O)C1 C=C(F)C1(CC(=O)NC(C)C=CC(=O)NCC2CCCN2C(C)C)CCC1 c1(C(N2C(CNC(c3n(CC)c(O)nc3)=O)CCC2)=O)cnc2c(C)cnn2c1 N1(C(C(=O)NC)C(C2CCC2)OC)CCOC2(CCN(C)CC2)C1 C1(CC(C)(C)C)CN(C(=O)C(=O)NCC2CCCN2c2ccccc2)CCO1 c1(C(=O)NCCCCNC(CCc2ncc(C)[nH]2)=O)cn(C)nc1O N1(C(CC2CNC(=O)O2)=O)CCN(c2cc(C3CC3)no2)CC1 C=C(Cl)CCC(=O)NC(C(=O)O)C(=O)OCC C(=O)(C(O)CC1CC1)N(C(CNC(C=CCOC)=O)C)CC N1(C(C(C(C)(C)O)F)=O)CCC2(C1)CN(C(c1ccnc(-n3ccnc3)c1)=O)C2 Fc1ccc(Cn2ccnc2-c2cscc2-c2cc3ncccc3[nH]2)c(F)c1F N1(C(c2c(CCC)nns2)=O)CCC(C)C1CNC(=O)CC1CSCCS1 C(=O)(C(=O)C(C)(C)C)NCC(C(N1CCC(CCOC)C1)=O)C CCCC1C(N2CC=CC(C(=O)OC(C)(C)C)C2)C(=O)N1.NC CC1C(C)N(C(=O)CNc2nccs2)CCN1C(c1cc2cscc2s1)=O C1(C(C)NC(COC(CC)(C)C)=O)CCN(C(c2ccn(C(C)C)n2)=O)C1 CC1=NN(C)C(=O)C1CC(=O)NCCC1CC(NC(C2CCSCC2)=O)C1 C1(CNC(c2c(C(=O)NC(c3ccccc3)C)cccc2)=O)CCC2(CC2)CO1 c1(C(C(=O)NCC(CO)NC(C=CC=CCCCCC)=O)C)ccc(F)cc1F C1(C(N2C(c3cn(CC(CC)C)nn3)COCC2)=O)CC2(CCC2=O)C1 c1(CC)cc(C(=O)NC2CC2CNC(c2nn(C)cc2SC)=O)c(C)o1 CC1CCCC1(C(=O)NONCCCO)NC(c1cccc(CCCF)c1)=O CC(C)CC(O)C(=O)N1CC(CC(C)NC(c2ccc(F)c(F)c2)=O)C1 C(C(CC(=O)NCCCCCF)NC(=O)COCC1CCC1)OC C1(CNC(COCCCC#C)=O)CCCCC1NC(=O)CCC1CCC1 C1(NC(C(C)NS(C)(=O)=O)=O)CCN(CC(c2ccc(F)cc2)O)CC1 C1(c2n(C)ncc2)C(=O)NCCN1C(C1CCC2(CC1)CC2)=O C(=O)(C(C)CC(=O)NC1CC2CC(NC(c3cc(Cl)cs3)=O)CC12)OC C1(NC(c2c(CC)csc2)=O)CCSC12CN(C(c1ccc(N(C)C)cn1)=O)C2 c1(C(=O)NC(CC)(CNC(C2(S(C)(=O)=O)CC2)=O)CC)coc2cc(C)ccc12 c1(CC(=O)NCCCN(C)C(C2CC2F)=O)csc2cc(Cl)ccc12 c1(C(=O)NC(C)C(C)NC(=O)C(C)OC2CC2)cccnc1Sc1ccccc1 N1(c2nc(C)nc(C)c2F)CCC2(CCCC2NC(=O)C(O)C(C)(C)C)CC1 C1(C(=O)NCC2CC(NC(c3ccc(C)o3)=O)CC2O)CC12CC(C)(C)C2 C1(OCC)CN(C(C2CCC(NC(=O)CC3CCCO3)C2)=O)CC12CC2 c1(C(=O)OCC)cc(CN2CCC(CO)(COC)CC2)ccc1O.c1ccccc1 c1(C(=O)NC2(CN(C)C(C3CC3C(F)F)=O)CC2)cnc2nccn2c1 N1(C(c2ccn(C)n2)=O)CC(NC(c2ccc(-c3ccccc3)s2)=O)C(F)(F)C1 N1(C(C2C=C(C)CS2)=O)CC2CCC2(CNC(=O)CC2(C)CCCCC2)C1 C12(CCCCCC1)CN(C)C1CC(OC)CN(C1)C(=O)O2.C(C)(C)(C)OCCO Cc1c[nH]cc(C(=O)NCC(C)(CNC(=O)C(C)(O)CCN(C)C)OC)c1=O C1(C(N2CCC(=CCNC(c3c(OC)n[nH]c3)=O)CC2)=O)CCc2nncn2C1 c1(NCCOC)cc(C(N2CCC(C(C)NC(=O)Cc3ccsc3)C2)=O)ccn1 C1(CNC(C2(COCC)CCC2)=O)(CNC(c2cncc(Cl)c2)=O)CC12CCC2 N1(C(c2cc(C)cc(Br)c2)=O)CCCCC1C1=NCCN1C O=C(C1=NOCC1)N1CC=CC1Cn1cc(CC2(CO)CCCC2)nn1 c1(C(C)NC(c2c(CNC(c3c(CC)c[nH]c3)=O)cc[nH]2)=O)cccc(O)c1 CC1=C(C(=O)N2CCC3(CC3C(=O)NC(C)CCF)C2)SCCO1 Cn1nc(C(=O)NC2CCC2NC(C2(c3ccccc3)CCCO2)=O)ccc1=O N1(C(C2C(C)OCC2)=O)CC2CC3CC2C1C3NC(c1nccn2nccc12)=O C12(CC(=O)NCCC(CNC(c3cnc(O)c(F)c3)=O)OC)CCC(CC1)CC2 Cc1noc(CC(=O)NC(C(=O)NCCN(C2CCCC2)C)c2cccs2)n1 Cc1n[nH]c(C)c1CC(=O)NC(C1CCCCC1)CNC(C1CC2CC1C2)=O Cc1cccnc1C=CC(N1CC(CNC(=O)Cc2ccccc2)C(O)C1)=O c1(OC)cc(Cl)c(S(=O)(=O)N2CCOC(C)(CCO)C2)cc1Cl C1(CC(=O)N(CC(C)(C)C)CCC)C2CCCC2N1C(=O)CCP(C)(C)=O C1(c2ccccc2)(CNC(CCCOC)=O)CCN(C(c2cnco2)=O)C1 C(=O)(CCCCCCCCCO)NC(C)(CNC(c1cc(CO)[nH]n1)=O)CO N1(C(c2nccc(OC)c2OC)=O)CCC(O)(C2CCN(C(C3CC3C)=O)CC2)C1 N1(C(CCC#CC)=O)CCC(C(N2CC(N3CC(F)C3)C2)=O)CC1CC N1(C(C2C(C)C2)=O)CC2CCC1C(NC(=O)CC(=O)OC1(C)CCCCC1)C2 c1(CC)ccc(C(=O)NCCCCC(C)NC(c2cccs2)=O)cc1OC CC(CC(F)(F)F)C(=O)N1CCC2CC12C(=O)N(C1CC(O)C1)C C1(C(=O)OC)C(C(=O)N(CC(C)CNC(=O)C(O)CC2CC2)C)C1(C)C c1(C(=O)NCC2N(C(C3(OC)CCCC3)=O)CCC2)occ(C)c1C c1(CC(=O)NC(C2CCCN2C(=O)Cc2ccsn2)C)cccc2ccoc12 CCC(C)C(C)N=c1nc2sccc2c(NCc2c(F)cccc2Cl)[nH]1 Cc1ccc(C=CC(=O)NC(C2CCCC2)CNC(c2ccc(C)o2)=O)cc1 c1(C(=O)NC(CN(C(C(C)CN(C)C)=O)C)C)cc2c(Cl)c(F)ccc2[nH]1 C(C1(C)CCOCC1)=CC(=O)NCCCN(C(C1(COC)COC1)=O)C c1(C(=O)NC2CCCCC2(F)F)ccc2c(c1)CN(C(c1nc[nH]n1)=O)CC2 C1(NC(c2ccc(OC)nn2)=O)CCSC12CN(C(C1(F)CCS(=O)(=O)C1)=O)C2 N(C(=NCC1CCCO1)NCC(C)(C)OC)CC1(CC)COC1 N1(C(CCc2scc(C)n2)=O)CC2CC(NC(=O)CC(C)(C)C)CC(C2)C1 C(=O)NNC(=O)C(N)=O.c12cccc(Cl)c1n1cc(nn1)c2=O.CO C#Cc1cccc(CC(N2CCC3(NC(c4cc[nH]c(=N)c4)=O)CC3C2)=O)c1 C(C(F)(C(=O)NCC(C1CC1)OC)C(C)C)NC(Cc1c(CC)con1)=O C(=O)(CCCCC(=O)N1CC=CC(NC(c2c(COC)cnn2C)=O)C1)NC C(C(CC(C)C)C(=O)NCCOc1cccc(Cl)c1)OC.c12ocnc1C(=O)N2 Cn1cc(C(=O)OCCOCCCSc2cscn2)nn1 c1(NC(c2c(CC)n[nH]c2)c2nnnn2C2CCOCC2)nc(C)ccc1C c1(C(=O)NCC(C)CNC(c2c(F)ccc(N)c2F)=O)cc2c(cn1)COCC2 c1(C(=O)OC)ccc(CN2C(C(=O)Nc3c(C(=O)OC)cnn3C)CC2)c(F)c1 C1(C(N2CC(CNC(c3n(CCOC)ncc3)=O)(COC)C2)=O)C(C#N)C1(C)C O=S(=O)(CCN=c1[nH]c2ccccc2s1)N1CCC(C(F)(F)F)CC1 C(=O)(C#CC1(C)COC1)N1CCOCC(CNC(C2(CC)CCNC2=O)=O)C1 C#CC1CN(C(=O)CC2(CC)CCOCC2)CCN1C(c1c[nH]c(=N)o1)=O C1(O)(C(C)NC(COCC(=O)OC)=O)CCN(C(c2cnc(Cl)s2)=O)C1 C1(C(=O)NCC(C(C)C)O)C(O)CCN1S(=O)(=O)CCCl c1(C(N(CC(CNC(CCCCOC)=O)C)C)=O)c(N)ccc(F)c1C CCC1(C)COC(=O)CCNC1=O.C1CCCC12CC2 Cc1cnc2c(C(=O)NC3CC(NCc4ccc(C#N)nc4)C3)cnn2c1 C(CCN(C)C(C1(CC(F)F)CC1)=O)(C(C)C)NC(CCC=CC(C)C)=O C1(C(N2CCC(NC(CC(C(C)C)O)=O)(CF)C2)=O)CC2(C1)CC1(CCC1)C2 C1(O)(CN(C)C(c2ccns2)=O)CN(C(=O)CSC(F)(F)F)C1 c1(OC)cc(C)c(C(=O)NC(c2cc(F)ccc2OC)c2ccccn2)c(C)c1 c1(OC)cn(C)c(C(N2CC=CC(NC(c3[nH]c(C)c(C)c3C)=O)C2)=O)cc1=O CC#CCCC(=O)N(CC(C)CNC(=O)C(c1ccc(Br)cc1)CC)C S(=O)(=O)(c1ccc(N2CC=CC(O)C2)nc1)NC(c1cccc(F)c1F)C C(CC(=O)NCCC(C)OC)(C(C)(C)C)NC(C=CC)=O CC1(C)CC1(C)C(=O)NC(c1ccccc1)CNC(C12CC(F)(C1)C2)=O c1(C(=O)NCC2CC(CNC(C3COC3)=O)CO2)cn2cccnc2n1 N1(CC)CCN(CC(=O)N(CCCCN(C)C(C2CCCC(=O)O2)=O)C)CC1 c1(C(N2CCC2CC2CC2c2ccc(Br)s2)=O)ccccn1 C1(S(C)(=O)=O)(C(=O)NCC(CCNC(CCC=CCC=C)=O)O)CCOCC1 C(=O)(C1CCCc2scnc21)N1CC2C(CNC(c3ccncn3)=O)(C2)C1 c1(OCCCC(C)C)ccccc1C(N1CCCC(n2ccnc2)C1)=O Cc1c(C(=O)N(C2(C(=O)NCC3CN4CCC3C4)CCC2)C2CC2)cccc1F c1(C(=O)NC2CC(CNC(c3c(C)[nH]cc3)=O)C2)csc(S(N)(=O)=O)c1 c1(OC)ncc(C(=O)NC2CCCN(C(=O)CCc3cc(C)[nH]n3)C2C)nc1C C1(CNC(c2cncc(SC)c2)=O)C(O)C(O)CN1C(=O)C(F)CC1CC1 C1(C)(CCS(C)(=O)=O)c2n(nnn2)N1.C1(CCOC)CCN(C2CC2)C1=O N1(C(C2(C)C(C)OCC2)=O)Cc2[nH]nc(C(=O)NCCCOC3CCCC3)c2C1 N12CCC(C(C(=O)O)C1)C2=O.c1(COCC)ccn(-c2ccccc2)n1 C1(NC(CN(C(C(C)OCC=C)=O)CC2CC2)=O)CCOC(C)C1 c1(OC)cnccc1CNC(C1(NC(=O)CCc2cc(C)[nH]n2)CCSC1)=O c1(C(=O)NC(C)CN(C)C(C2C3CNC(=O)C23)=O)ncc(C(F)(F)F)cc1O N1(C(C(C)=CC2CC2)=O)CCN(C(c2ccn(C)n2)=O)C2CCCCC12 C1(C(=O)NC(c2ccccn2)C)(NC(c2cc[nH]n2)=O)CC1(C)C C1(O)(C(=O)NCC(CCNC(=O)CC(C)N(C)C)OC)CCOC1(C)C N1(C(c2n(CC)ccn2)=O)CCOC2CCN(C(c3cc(C#N)c[nH]3)=O)CC12 c1(C(=O)NC2CCC(NC(C3CCC(=O)NC3)=O)C2)cc(Br)cc(Cl)c1F C1(NC(c2cc(C)nnc2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 Cn1cc(C(C(=O)OC(C)(C)C)N(C2CCOCC2)C)c2ccccc12 c1(C(=O)NCC(C)(C2CC2)NC(C2CC(C3CC3)=NO2)=O)ccc(N)c(N)c1 C(=O)(CC1CNc2ccccc21)N(CC(CN(C(=O)CC1COCCO1)C)O)C n1(CCC(=O)NC(CC)CNC(C2CCNC(=O)C2)=O)ncc2ccccc12 N1(C(COCC)=O)CCC(C(=O)N(CC(C)C)CCO)CC1 Cn1ccn2ncc(C(N3CC(NC(=O)CN4CCCC4CO)CC3(C)C)=O)c12 C(CCCCC(=O)NC(C)CN1CCN(C(=O)C(C)C2(O)CCC2)CC1)OC c1(C(N(C2CN(C(c3cc(CCCCC)[nH]n3)=O)C2)C)=O)n[nH]c2c1COCC2 c1(C(N(C2CCN(C(C(=O)NCC)=O)C2)C)=O)sc(S(N)(=O)=O)c(C)c1Cl c1(C(=O)NCCNC(C2(C)CCCC2O)=O)cc2c(s1)CCCC2 c1(CC(=O)NC2CCN(C(c3ncc(C)cn3)=O)CC2O)c(C)cc(C)nc1O C1(NC(c2nn(C)nc2C(F)(F)F)=O)CC2CCC(C1F)N2C(=O)C(Cl)=CCl C(=O)(CCC(C)(C)C(=O)NC1CCC1NC(c1ccc(C(C)(F)F)cc1)=O)OC C1(C(=O)NCC23CC(NC(Cn4ncc(C)c4)=O)(C2)C3)CCC2CCC1O2 C1(CC(C)NC(=O)C2=CCCC2)CCN(C(=O)CCn2ccnn2)CC1 N1(C(C(C=C(CCC)C)O)=O)CCC(OC(=O)Nc2cccc(Cl)c2)CC1 Cc1cc(C(N2CCOC(CNC(c3cnn(C(C)C)c3)=O)C2)=O)ccc1Br Nc1c(C(=O)NCC(O)CNC(=O)C=Cc2cscn2)sc2ncccc12 Cc1cc(C2CC2)ccc1C(=O)NC1CC(NC(C2CCNC2=O)=O)C1 c1(C(N2CCCC(NC(C(C(C)O)NC(C)=O)=O)CC2)=O)cc(C#N)cc(C)n1 Cn1cc(C(=O)NCCCNC(=O)CC2(N(C)C)COC2)ccc1=O N1(C(C2N(C=O)CCC2)=O)CCCC2CN(C(=O)C(F)(F)c3cscn3)CC12 C(=O)(C(F)CC(C)(C)NC(=O)CN1CCNC(=O)C1)NCC1CN(CC)C(=O)O1 C(=O)(CCSc1ccco1)N(CCN(C)C)CC1COC1 CC(C)C(O)C(=O)NC(C)(C)CNC(c1ccnc(OCCO)c1)=O c1(CNC(C2CC3(CC(NC(C(=O)NC)=O)C3)C2)=O)ccc(S(C)(=O)=O)cc1C n1(CC(=O)OCC)c(NC(=O)Cc2ccc(N=[N+]=[N-])cc2)nc2ccccc12 C1(NC(C(C)(C)c2ccsc2)=O)CCN(C(=O)C=C(Cl)Cl)C1c1cn[nH]c1 C1(CC)CN(C(=O)Cn2nc(C)n(C)c2=O)CCC1NC(=O)CCc1cnc[nH]1 c1(NC(C2(C(=O)OC)CC2)=O)cccc(OC2CC2)c1.c12ccc(cc1)[nH]c2=O CC1CC(C(=O)NCCC(O)CNC(c2cscc2C(F)F)=O)=NO1 C1(C(=O)NC(C#C)CCC)(CC)CCCN1C(c1nonc1CC)=O CC(C(=O)N1CCC(C(=O)NC2CCC3(CCC3)C2)C1)C(C)(C)C CC1COc2ccc(C(N3CCCC3c3nncn3C)=O)cc21 c1(NC(C(C2CCCN(C(=O)CCC(=O)C3CC3)C2)C)=O)cccc(F)c1 C(C(=O)NCc1c[nH]nc1C(=O)NC1CC(C)CCC1O)(C(C)(C)C)SC Cc1cnccc1C(C)C(=O)N(CC(C)NC(=O)COC1(C)CCCC1)CCO C12(C(N3CCC(C(C)NC(CCC(=C)Cl)=O)C3)=O)CCCC1CC(=O)CC2 Cn1c(C(=O)NCC2CC2C(=O)Nc2cccc(CON)c2)cc2ccccc12 C1(NC(=O)Cc2ccc(F)nc2)CC2CCC1N2C(=O)CC1CCOC1 C=CC1(C(=O)N(CC)OCC)CCN(C(c2cncnc2)=O)C1 c1(C(C)C)c[nH]nc1C(=O)N(C1CCC(NC(=O)CC(=O)N(C)C)C1)C c1(Nc2cc(=O)n(C3CC3c3ccccc3)cn2)cccc2ccnn12 C#CCC(C)(CC)C(=O)NC1CN(C(=O)CCCCC)CC1n1ccnn1 N1(C(CSC(C)C)=O)CC(CNC(=O)C(F)(F)C(C)O)OC2(CCC2)C1 c1(OCC)ccnc(NCC2CCN(C(=O)CCOC3CCOCC3)C2)n1 C1(N(C(C(COC)(C)C)=O)C)CC2CCC(C1)N2C(c1cncc(SC)c1)=O c1(C(=O)NC2C(CNC(C(C)n3ccnc3)=O)CC2)coc2c1C(=O)NCCC2 CC(C)(CC#N)C(=O)Nc1cccc(NC(C2CC3CCC2C3)=O)c1 c1(OCCC)ccc(NC(=O)Nc2ccc(-n3cncn3)cc2)c(C)n1 c1(NC(N2CCOC(CSc3cn(CCCCF)nn3)C2)=O)cc(Cl)c(Cl)[nH]1 c1(C(=O)NC(C2CCCN2C(=O)C(C)(C)F)C)ccc2nc(O)n(C3CC3)c2c1 C(=O)(CCC(=O)NC(CC1CCOCC1)C(=O)NCC(C1CCC1)OC)NC N1(CCC)CCCC1C(=O)NC(C)(C)C(=O)NC1CCCC1CN(C)C C1(C)(CNC(C(COC)OCCc2cc(C(=O)NN(C)C)no2)=O)CCC(=O)N1 CCCC(CCC)CCCC(=O)N1CCN(C(=O)CC(C)SC)CC1CCCC c1(C(=O)NCCC2(NC(C3C(CC)OCC3)=O)CCC2)ccc2oc(C)nc2c1 c1(N(CC(=O)NOCC(O)C2CC2)C)nccc(Br)c1C.C12CCN(CC1)C2=O C1(CC(N(CC(C2CCC2)OC)CC)=O)CC(NC(C2CC(C)(C)C2)=O)C1(C)C N1(C(c2c(C)cc(F)nc2)=O)CCc2[nH]nc(-c3cc(F)c(F)c(F)c3F)c2C1 Cc1c(C(=O)NC2CC(NC(=O)CCCc3ncco3)CC2O)ccn1C C1(CNC(C(C)(C)C2CCC2)=O)CN(C(=O)CCCn2cccn2)C2(CCC2)C1 C1(OCC)CC2(C1)CC2C(=O)NC(CN(C)C(c1ccnn1C)=O)CC CC1CN(C(c2ccnn2C)=O)C(C)CN1C(C1COCC1C(N)=O)=O c1(C(=O)NCC(C)N(C)C(C2CCCSC2)=O)conc1C1CCC1 S(=O)(=O)(c1ccccc1)NC(C)C(=O)NC1CCCN(CCCc2nn[nH]n2)C1 c1(OCC)ccc(C)cc1NC(=O)C=CCC1(NC(C2(C)OCCO2)=O)CCC1 Nc1cc(C(=O)NCCC2(O)CN(C(C3CC3C(F)F)=O)C2)ccc1F N1(C(c2c(CC)noc2)=O)CC(C)(C)OCC1CNC(C1CCC(C)(C)CO1)=O CC(C)S(=O)(=O)CC(=O)NC(C)CNCc1ccc([N+](=O)[O-])cc1 c1(C(N2CCC(C)(C(=O)Nc3nccc(C)c3Br)C2)=O)cc(C)c(CN)c(C)c1 CC(C)(C)C(O)C(=O)NCCCn1cc(C(O)C(C)(C)C)nn1 C(C(C(=O)NOCCCC1CC1)C(C)(C)C)NC(C1OCCN(C)C1)=O c1(C(=O)NC2CCN(C(c3cccc(C(F)F)c3)=O)CC2)ccc(F)c(F)c1F C1(C(N(CCCN(C)C(C2(F)CCOC2)=O)C)=O)CCc2ncsc2C1 Cn1cc(Br)c(C(=O)NCC2CCCC2NC(=O)CCc2nc[nH]n2)n1 CCC(CC(=O)N1CCCC1CNC(=O)Cc1ccc(Cl)cn1)c1ccccc1 N1(C(C2(C)CC(F)C2)=O)CC(C(=O)NCCCS(N)(=O)=O)C2(CC2)C1 C1(C(N2CC(N(C(CN3CC(C(=O)OC)C3)=O)C)C2)=O)CCC(N=[N+]=[N-])C1 c1(C(=O)NCCC2(O)CN(C(CC=CC)=O)C2)cc2c(Br)cccc2c(=O)o1 N1(Cc2ccc(C)nc2)CCCN(Cc2cnc(N(C)C)nc2)CC1 c1(C(=O)CC2C(C(N(OCC(=O)OC)C)=O)CCC2)ccc(C#N)cc1 c1(OC)cccc2ncnc(N3CCC(CNC(c4cnn(C)n4)=O)C34CC4)c12 c1(C(=O)NCC(CNC(=O)Cc2nnc(O)s2)O)cc(=O)cc[nH]1 C1(OC)CCC2(CCN(C(=O)CC(C)CNC(=O)COC3CC3)C2)C1 C1(C(N(CCCCNC(C2CCCCN2C)=O)C)=O)CC12CC(F)(F)C2 C1(C(CC(C)C)NCC(C(F)F)n2cccn2)CCCCCC1 c1(C(N2CCC(C)(CNC(C(C)C3CCC3)=O)C2)=O)ccc2oncc2c1 C(CC)(CC)(CCNC(=O)C(C)(C)CC)NC(c1cccc(CC)n1)=O N1(Cc2ccc(OC)c(I)c2)CC(C(=O)NCC2CCOC2)CC(F)(F)C1 c1(NC(C)=O)cccc(C(=O)N(C(=O)C(C)C)CCC#N)c1.C12CCC1CN2 CCCC(CCCO)C(=O)N1CCC(C)(NC(c2cccc(S(C)=O)c2)=O)C1 C(=O)(C(CCCOC)NC(=O)C(C)O)NC1(CC=C)CCCCC1 c1(C(N2CC(NC(C(CCC#C)O)=O)C2)=O)coc(S(=O)(=O)N(C)C)c1 C1(NC(C(C)CC2CCCC2)=O)C=CCC(C(=O)NCC(C)(O)CCO)C1 C(c1cnn(C)c1)=CC(=O)NC(C1(O)CN(C(=O)CSc2nc[nH]n2)C1)C C(=O)(CC(C)CC(C)(C)C)N(C1(C)CC1)CCNC(C(=O)OC)CCC(=O)N(C)C c1(OC)ccc(C(=O)N(C)CCNC(=O)CCCOc2cccc(Br)c2)nn1 c1(C(N(C2CC(NC(=O)C(O)C3CC3)C2)C)=O)cccc2c(Cl)c(Cl)sc12 C#CCC(C)(C(=O)NC1CCCC1C(N)=O)NC(C1COCCN1CC)=O c1(OCCOC)cccc(C(=O)NC(CNC(c2nccnc2Cl)=O)C2CC2)c1 CCCC(CC(=O)NCc1cc(Cl)no1)NC(=O)CCc1ccc(C)o1 N#CCS(=O)c1ccc(C(=O)NC(CNC(=O)C2CC2)CC(F)(F)F)cc1 c1(C(N2CC(NC(C(C)NS(C)(=O)=O)=O)C3(C2)CC3)=O)cn2cccc(Cl)c2n1 c1(NC(CC2(COC)CC2)=O)ccc2c(C)[nH]nc2c1 c1(NC(C(=O)N(C(CC=C)=O)C2(c3ccc(F)cc3)CC2)=O)ccc(OC)cc1 c1(CC)nc(C(=O)NCCC(C)N(C(=O)CCF)C)c2ccccn12 N1(C(c2c(OC)c(F)ccc2F)=O)CC2CCCN(C(=O)COC(C)=O)C2C1 C1(CC)C(C(=O)NC(C)CS(C)(=O)=O)CCCN1C(c1ccc(CO)o1)=O C1(C(=O)NC(CN(C)C(c2ccc(C(C)(C)C)[nH]2)=O)(C)C)CCCOC1 N1(C(c2noc(C)c2C#N)=O)CCC(CN)CC1C(F)(F)F C1(OC)C(OC)CN(C(=O)CO)C1CNC(c1ccc(F)c(C(F)F)c1)=O C1CCc2ccccc2C1.c1(OC)cc(NC(=O)CC2CCCN2C=O)ccc1F CCCC(CCC)=CC(=O)NCCC1(O)CN(C(=O)Cc2cnns2)C1 c1(N2CCN(C(=O)OC(C)(C)C)CC2)ncnc2sc([N+](=O)[O-])cc12 c1(C(=O)NCCN(C(=O)C(c2ccc(C3CC3)cc2)O)C)ccc(P(C)(C)=O)nc1 c1(C(=O)Nc2c(OCC#C)nccc2)cc(C)c2sccc2c1 Cc1cccnc1C(=O)NC1CCCN(C(C23CC(CN2C2CC2)C3)=O)C1 Cc1nc(C2CC2)nc(O)c1C(=O)N(CC(C)(C)NC(C1(C)CCCS1)=O)C C1(C)(C(=O)NC2(CC=C)CN(C(=O)Cc3cc(Cl)cs3)C2)CC(C)OC(C)C1 C(=O)(C(C)P(C)(C)=O)OCC1(CC)CCOCC1 c1(CNC(C2(CCC=C)CCC2)=O)nc(C(=O)NC2(C)CCOCC2)c(C)o1 Cc1cc(C(=O)NC2CC(CNC(=O)C(c3ccc(Cl)s3)C)C(O)C2)ncn1 C(=O)(CC(C)(C)C#N)N1C(CNC(=O)CCC2C(=O)ON=C2C)CC(COC)C1 Cc1ccc(F)cc1CN(C(=O)C(c1ccc(O)nc1)(C)C)C CC1CCCCC1C(N1CCCC1CN(C)C(c1csc(Cl)c1Cl)=O)=O N1(C(C2CC(C)(C(N)=O)C2)=O)CCC2CN(C(C3CC34CCOCC4)=O)C2C1 Cc1ccc(F)c(N)c1C(=O)NC1CCC(NC(C2(Br)CC2(C)C)=O)CC1 N1(C(C2CC(C)C2)=O)CCC(NC(=O)C(F)OC(F)(F)F)CC1.N12CC(C1)C2=O C=C(Cl)CCC(=O)N(C1CC(NC(=O)CC(C)n2ccnc2)C1)C n1(CC(COC)O)cc(C#CCNC(=O)CC(C)(C)C#N)nn1 CCC(CC(=O)NCC12CC1CN(C(=O)C(C)(C)C(C)C)C2)CC(C)C n1(CCC)cc(C(=O)NCC(F)CNC(c2cncc(C(C)C)c2)=O)c(C)n1 Cc1ccc(C(N2CC(NC(c3nc(Cl)sc3C)=O)C(C)C2)=O)cc1F O=C(C#CC1CCOC1)NC1CCC2CN(C(c3ccc(O)cn3)=O)CC12 C(=O)(C1CCCn2nccc21)NC(CC)CNC(=O)C(C)Cc1cnc[nH]1 N1(C(c2c(CNC(C=C(CC)CC)=O)cnn2C)=O)C2C=CC(C2)C1CO C1(NC(C(c2cccc(O)c2)C)=O)CCC2CCN(C(=O)C3=NNC(=O)CC3)C12 c1(C(N2CCC(N(C(C=CCC)=O)C)C(C)C2)=O)cccc2c1CCC2 Cc1ccc(I)c(C(=O)NC2CCCN(C(c3ccnc(F)c3C)=O)C2)c1 c1(C(=O)NC(CC)CNC(=O)C(C)(C)C2CCCCO2)cccn2cnnc12 c1(C(N2C(C(C)NC(C(C)OCCCC)=O)CCC2)=O)ncncc1Br CC1(CNC(c2cnn(CC(F)F)c2)=O)COCCN(C(=O)C=CC(F)(F)F)C1 c1(C(=O)NCC(C)CNC(C23CCCC2C3(F)F)=O)cnc2c(F)cccn12 N1(C(C=C(CC)C)=O)CC2CCN(C(=O)C=CCOC)CC2C1 C1(C)(NC(C(C=C=C)C)=O)CCCCC1C(N1CCCC(OC2CC2)C1)=O N#Cc1c[nH]ccc1=NC1CCCCC1NC(=O)C(F)(F)C(F)F Cc1cc(Br)c2oc(C(=O)NCC3CN(C(C4(N(C)C)CC4)=O)C3)cc2c1 C1(CNC(C(n2ccc(Br)n2)C)=O)CC(O)CN1C(C1CCC(=O)NC1)=O N1(C(c2cc(CC)no2)=O)CC=CCC1C(=O)NC(CC)C(C)(F)F c1(C(=O)NC(CC(C)C)(C)CNC(=O)C(C)P(C)(C)=O)ccc2c(c1)CCCC2 c1(CC(=O)NCc2cn(CC(=O)Nc3c(C)nccc3)nn2)ccc(Cl)cc1Cl CC(CCCCNC(C1CC1(C)C(F)F)=O)NC(=O)C=CCOCC(F)(F)F C1(C(N2CC(CCC(=O)N(C3CCN(CC)C3)C)C2)=O)CCC(C)CC1 c1(C(=O)NC2CCN(C(C(CC=CCC)C)=O)C2CC)ccn2c(C)cnc2c1 C1(CCN(C)C)(CC)CCC1.C1(C(=O)OC)(N(CC(N)=O)C(C)C)CC1 Cc1nn(C)c(Cl)c1C(N1CC2C(CNC(=O)CC3CCC(C4CC4)O3)C2C1)=O C1(CNC(C(C=C)(F)F)=O)CN(C(=O)C(c2ccc(C)cc2)=O)CCC1(F)F C1(NC(CC(C)(C)OC)=O)COC2CN(C(=O)CC3CC4(CCC4)C3)CC12 CON(CCC(=O)N1CC(OC)CC1CF)C(=O)CSC C1(NC(c2c(OC)ccc(C)c2)=O)CCC2CN(c3snc(C)c3C#N)CC2C1 CC(C)CCCOCC(=O)NCCC(C)NC(c1ncoc1C(F)(F)F)=O Cc1cc(=NC2CCCC(NC(=O)CCc3cccnc3)C2)c(C#N)c[nH]1 C1(NC(CCC=C=C)=O)CCN(C(=O)CCOc2cc(Cl)ccc2Cl)C(C)C1 C1(NC(C2N(Cc3ccnc(OC)c3F)CC2)=O)CCc2n[nH]cc2C1 C12(C(=O)NCC3N(C(C4C5CC6C(C5)C46)=O)CCCC3)CCCCCC1OCC2 C(=O)(C(N=[N+]=[N-])C(C)C)NC12CC(C(=O)NCCc3c(C)ccnc3)(C1)C2 N1(C(C(C(C)C)C)=O)C2CC=C(C(=O)NCc3cc(O)cc(F)c3)C1CC2 C#Cc1cnc(C(N2CCC(CC)C2CNC(=O)C(C)NC=O)=O)c(C)c1 c1(CNC(N2CCOC(Cn3cnnn3)C2)=O)cc2cc(Br)ccc2o1 C(=O)(CS(=O)(=O)CC(C)C)N1CCN(C(C(C)OCOC)=O)C(CC2CC2)C1 Cc1c(C(=O)NC2(C#N)CCN(Cc3ccc(F)c(F)c3)C2)ccc(F)c1F C(=O)(CCCS(N)(=O)=O)NC1(C)CCN(C(c2ccc(C(=O)NC)c(F)c2)=O)C1 c1(C(=O)NCC(C)N(C(C2C(CC)OCC2)=O)C)cc2n(n1)CCOC2 N1(C(C(CO)N(C)C)=O)CCC(F)(F)C(CNC(=O)Cn2cc([N+](=O)[O-])cn2)C1 C(C(CC1CCCC1)C(=O)NCC1(F)CCOCC1)NC(C1(NC(N)=O)CC1)=O C1(C(=O)NCCC(C)N(C(CCOCC(C)C)=O)C)CCCC1c1cnn(C)c1 C(=O)(C(CC(C)(C)C)NC(c1cn(C(C)C)cn1)=O)N1CC(C(C)OC)C1 N1(C(C(C2CCOC2)OC)=O)CCN(C(=O)C2=CCCC2)CC(C)C1 c1(C(N2C(CCC)CN(C(c3nnn(C)c3C)=O)CC2)=O)cnc2c(c1)COC2 CC1CC(C(=O)N(CCCN(C(=O)Cn2nnc(=O)[nH]2)C)C)CO1 C1(NC(CCC(=O)NC)=O)CN(C(=O)CCc2scnc2C)C(C)(C)C1 C(=O)(C(C(C)C)C(C)C)NCC1CCN(C(COCc2cc(C)no2)=O)C1 c1(N2C(C(C3CN(C(C)C)C(=O)CC3)=O)CCC2)nc(O)c2c(ncn2C)n1 C(=O)(C(C)(C)CCCNC(=O)CC#N)N1CC(C)SC(C)C1 c1(C(N2CCCC(CC(=O)Nc3c(Cl)ccnc3Br)C2)=O)ncc(F)cc1F c1(C(=O)NC(CNC(C(CO)N(C)C)=O)C2CC2)nccc2ncccc12 c1(C(N2CC(CNC(C3C(CCC)CCC3)=O)(OC)C2)=O)c(C)cc(=O)oc1C CCC(CC(=O)NCC=CCNC(=O)Cc1csc(C(C)C)n1)C(F)F C1(C(=O)NC2CN(C(CS(=O)(=O)NCC)=O)CC2F)CCn2c(C)cnc2C1 c1(OC)ccc2[nH]cc(CC(=O)NCC(O)CNC(C3C(C)C3C)=O)c2c1 C1(NC(c2cc(C)cc(Cl)c2)=O)CC2CC1CN(C(C1CC(C)CCO1)=O)C2 N1(N2C(CC(=O)CC)CCC2)CCCC1(C)C(C)(C)C.C(=O)O N1(CC2(NC(C(C)=CC3CC3)=O)CC2)CCN(C)CC1.C12CC1NC2=O C(=O)(CCCCCCCC1CC1)N1C(C)CN(C(C2COC(=O)N2C)=O)CCC1 c1(SC)ccccc1C(N1CCN(C2CCC(NC(=O)C3=CCC3)CC2)CC1)=O Cn1ncc2c1CCC(C(=O)NC1(C)CCCN(C(C3(C4CCC4)CC3)=O)C1)C2 N(S(=O)(=O)N(C)C)CC(=O)NC(CC)CNC(C1CC1CCOC)=O C(C)(CC(=O)NCC12CC(NC(=O)CCCn3ccnn3)(C1)C2)SC Cc1ncc2n1CC(C(=O)NCCN1CCN(C(=O)C(C)(C)C#N)CC1)CC2 c1(NC2(c3ccccc3)CN(C(C(C)OC)=O)C2)cnc(F)cn1 C1(CNC(=O)CCC2CCCCC2)CN(C(=O)C(O)CC2CCOCC2)CCO1 c1(SCc2n(CC)nc(C)c2)cccc(CC(=O)NCC2CC2CNC(C)=O)c1C c1(C(=O)NCCNC(C2(C)CC(=C)C2)=O)c[nH]c2c(C)cc(F)cc2c1=O Cc1nn(C)c(C)c1NC(=O)C(C)N(C)CC1CCCN1C(=O)C(C)C(C)C C1(CC)CN(C(=O)CC2CC2CNC(C2COC(=O)N2C)=O)CCS1 c1(C(=O)OCC)nc(C)c(NC(=O)NCc2nc(C)n(C)n2)cc1C c1(N(C(Cc2cc(C)on2)=O)CC2CCCO2)cnc(F)nc1 c1(C(=O)NCC(C(=O)N(C(C(=O)OC)C)C2CC2)OC)ccc(C)c(F)c1 c1(NC(N2CCCC(C(=O)Nc3ccc(Br)cc3)CC2)=O)nc2cc(Cl)ccn2n1 C1(C(=O)OC2CCC(C(N)=O)CC2)C2CCC(O2)C1C(F)(F)F c1(OC(F)(F)F)ccccc1C(n1cc(C2CCCN2C(=O)C(Br)Br)nn1)(C)C c1(C(=O)NCC2CCN(C(C3CCCCC3)=O)CC2)ccc2c(c1)CCNC2=O C(C(COC(=O)C(=O)N(C)C)C(C)C)OC.N12CCCC1CCC2 c1(CC(C)(C)CO)nc(-c2cccc(-n3cccc3)c2)n(CCOC)n1.C1(C)CCC1 Cc1cc(Br)cc(C(=O)NCC(C)CN(C(=O)CC2CCC23CCC3)C)c1C Cc1c(C(=O)N(C)CCNC(=O)C(C)CF)cnn1C1CCC1 C12(C(=O)NCC3C(C)CCN3C(=O)CN3CCC3C)CCC(F)(CC1)CC2 C(C)(CC(C)N=c1[nH]nc(C2CC2)s1)NC(c1c(CC)nccn1)=O c1(CCC(=O)NCCCc2cn(C(C(=O)OC)C)nn2)ccc(F)nc1 CCC(CC)(CC)C(=O)N(CCCC(=O)NC(c1ccco1)CO)C C(C)(C)(CCCC(=O)NC(C(C)C)C1CCC1)NC(c1c(C)cc(CC)o1)=O c1(NC(c2cc(OC)ns2)C)cc(N2CCOCC2)nc(C)n1 N1(C(c2c(C)nsc2)=O)CCC(C2CCN(C(c3cc(N)ccc3Cl)=O)CC2)C1 c1(C(=O)NCC2CN(C(C(C)(C(C)C)NC(C)=O)=O)CC2C)cc(C)nc(C)c1O C(=O)(C(C)C(O)C(C)C)NC(c1ccc(CNC(C2(C(=O)NC)CC2)=O)cc1)C C(=O)(C(C(C)(C)C)OC)NCC(=C)CCNC(C1(c2ccno2)CCC1)=O CCC(C)(CNC(=O)C(C(C)(C)C)OC)C(=O)N1CCC(O)C1 N1(C(C(Cc2cnc[nH]2)NC(c2cc(C)[nH]n2)=O)=O)CCSC(C)C1 C1(C(N2CCCCC2CNC(C23CC4CC2C3C4)=O)=O)CCc2nncn2C1 c1(N2CCC(COC)(NC(c3ccsn3)=O)CC2)ncc2c(n1)COC2 N1(C(=O)OC(C)(C)C)CCC1CC(=O)C(CN(C1CN(CC2CC2)C1)CC1CC1)=O C(C(=O)N(C)CC1CCCCN1C(C1C2CC3C(C2=O)C13)=O)(C(C)(C)C)SC Cc1nscc1CC(=O)NCCOCC(=O)NC(C1CCCC1)C C1(C(N2CCC(OCCNC(CCCC)=O)C2)=O)CCC(=O)CC1(C)C c1(OCCC(=O)NC(CNC(C(CC)=CCCC)=O)C2CCC2)ccccc1O c1(C(=O)NCC(CN(C(C(C)OCC)=O)C)C)c(C)cc(OC)cc1F c1(C(=O)OCC)ccc(C2CC(NCc3cn(C)nc3I)C2)cc1 N1(Cc2c(C(C)C)cnn2C)CCC2(C)CNCC12 c1(C(N2C(C)(C)C(CNC(=O)CC3CC=CCC3)CC2)=O)ccc2cnoc2c1 c1(SC)cc(C(=O)NCC2CN(C(=O)CC3NC(=O)NC3=O)CC2O)ccc1F N1(C(c2c(C)nn(C)c2)=O)CC2CC(N=c3nc(-c4ccccc4)[nH]s3)C2C1 Cc1cnc[nH]c1=NCC1CCCC(NC(=O)C(C(C)C)OCC(C)C)C1 C1(NC(C2(C(CC)=O)CC2)=O)CCN(C(C2CC3CC(OC)C3C2)=O)C(C)C1 CN1CCCC1(C)C(N1CCCC1CNC(c1ncc(Br)cn1)=O)=O C12(CNC(CNC(=O)OC)=O)CCC1CN(C(=O)CCCN1CCCCC1)C2 c1(CC(=O)NC2CCc3nccn3C2)cccc2cccnc12 Cc1cccc(CC(=O)NCC(O)CCNC(=O)CN(C2CCCC2O)C)c1 c1(OCC(=O)NCC(C(C)C)NC(C2C(=C)CC2)=O)ccc2c(c1)CCC2 c1(C(C)C(=O)NCC2CCCN(c3cc(O)ncn3)CC2)cccc([N+](=O)[O-])c1 C1(NC(C2CCC(C)(C)C2)=O)CCN(C(c2cnc(N3CCCC3)s2)=O)CC1O CCC(COC)(CC)C(=O)N1CCCC(C(=O)NC2COC(C(F)F)C2)C1 N1(C(CC=CC=C)=O)CCOC2(CCN(C(C3CCCC4CCCN34)=O)C2)C1 n1(CC)ccc(C(=O)NC2CN(C(C3(C(N)=O)CC3)=O)CC2C)c1C CC(C)CC(C)CC(=O)NC1CCCC1C(=O)NCC(O)CC1CCCC1 N1(C(C2(O)CCCC(C)CC2)=O)CC2(CCC(NC(C3CSCCS3)=O)CC2)C1 c1(C(CNC(=O)NCC(=O)Nc2cccc(C)c2)C)ccc(F)c(Br)c1 c1(CNC2CCC(C(N(CC#N)CC#N)=O)CC2)cc(Br)cc(F)c1F N(C1CCOc2cc(Cl)ccc21)C(CCCOC)C(=O)OC C1(CN(C)C(C2C(COC)C2)=O)CCCN1C(=O)C=CCOCCO Cc1nc2cc(C(N3CCN(C(C4CC(O)C4)=O)C(CO)C3)=O)cnc2s1 c1(CN(C(=O)CN2CCC(NC(c3cnoc3)=O)C2)C)cccc(F)c1 c1(C(N2C(C(=O)NC3CC(C)OC3=O)CCC2)=O)cc2ccccc2o1 C1(NC(c2c(C)cc(CNC(C(C=C)CC)=O)o2)=O)CCOCC1(C)C CC#CCCCC(=O)NC1CCOC(CNC(c2ccncc2N(C)C)=O)C1 c1(C(=O)N(C(C(=O)O)C(O)Cc2ccccc2)CCO)coc2cccc(O)c12 CC(C)(C)CC(O)C(=O)NCC1CC(F)CN1C(c1ccc(OC(F)F)cn1)=O c1(C(=O)NCC(C)NC(=O)C(C)OC2CCCCC2)ncc(C#N)cc1Cl c1(CNC(C(C)NC2C(OC)(OC)CC2)=O)ccc2c(c1)CC2 c1(CCC(N2CCC(C)C(NC(c3cc(F)cs3)=O)C2)=O)nc2ccccc2s1 C1(C(=O)Nc2cnc(C)nc2C)(OC)CCN(C2CCNCC2)CC1 N1(C(CCOC)=O)CCOC(N(C2CN(C(C(C)OCCOC)=O)C2)C)C1 Cn1nc(C(=O)NCCC2(C)CCCN(C(=O)NCCCN=[N+]=[N-])C2)c(Cl)c1Cl N1(C(C=C2CCC(C)C2)=O)C2CCC1CN(C(=O)CNS(=O)(=O)C1CC1)C2 C(C(=O)Nc1ccccc1)(C(=O)O)OC.c12ccccc1NC(=O)C2(F)F c1(C2C(C(N3CCCC(N(C)C(c4cocn4)=O)C3)=O)C2)ccc([N+](=O)[O-])cc1 c1(C(N2CC(NC(CCC=CCC=C)=O)C(F)C2)=O)nc2cncnc2[nH]c1=O N1(C(CCOC)=O)CCN(C(c2cccc(Cn3ccnn3)c2)=O)C2CCCCC12 N1(C(CC2CC(=O)C2)=O)C(C(N2CCC(O)C(C)(O)C2)=O)C2CC(O)C1C2 C1(CC(=O)NCC2CC2NC(=O)CNc2nccs2)CCC(O)CC1 N1(C(c2nccc(C)c2)=O)CC(NC(=O)CN2CCOCC2)CC(F)(F)C1 N1(CCCNC(=O)CSC(F)(F)F)CCN(C(C23CCCCC2C3)=O)CC1 C(=O)(C(C)CC(F)F)NC1C(OC)CN(C(=O)CCc2ccncn2)C1 N1(C(=O)Cn2ccnn2)CCCC(N=c2[nH]nc(C3CC3)o2)CC1 c1(C(=O)NC(C(C)NC(c2c(CC)onc2)=O)CO)ccc(=O)n(C2CC2)c1 N1(Cc2ccc(OC)c(O)c2Br)CCN(C(c2cccnc2)=O)C2(CC2)C1 C1(C(N2C(C)C(NC(C3CC(=O)NC3(C)C)=O)CC2)=O)CN(C)CCN(C)C1 C1(C)(C(N2CC(CCNC(c3nccn3C)=O)(OC)C2)=O)CCCC1CC c1(N)ccc(OCC(N2CC(CNCC)C2)=O)cc1.C1(S)CCOC1=O.CC c1(NC(CC)C(=O)NCCN(C)C(c2cc(C(C)(C)O)on2)=O)ccccc1C c1(C(=O)NCC(CC)NC(=O)C(O)C2CCC2)cc(COC)[nH]n1 C=C1CC2CCC(C1)N2C(=O)C(CNC(C1(c2ccno2)CC1)=O)CC c1(C(C(=O)NC2CCOCC2)N(CC)CC2CCC2)cccc(C2CC2)c1F N1(C(COCCOC)=O)CCC(C2CN(C(=O)CC3CCOCC3OC)C2)CC1 CCCCS(=O)(=O)CC(=O)NCC1CC2CCC(C1)N2C(=O)C=CC1CCCO1 Cc1ccc(O)c(C(=O)NC2(C)CC3CCC2C3)c1.c12cncc(c1)CNC2=O c1(C(=O)NCCCCN(C)C)ccc2c(n1)CCC(C)(C)C2 C#CC(C(C)OC)NC(c1coc(CNC(C2(SC)CC2)=O)n1)=O C1(C(=O)NCCN(CC(C)O)C(C2CCCC2OC)=O)(OC)CCC(C)(C)CC1 N1(C(c2cc(C)no2)=O)CCC(NC(c2cnc(Cl)c(N)c2)=O)C(CO)C1 C(=O)(CS(=O)(=O)Cc1cccs1)N1CCC(CC=C)(NC(c2cnn(C)n2)=O)C1 C(=O)(CC(C)C(F)(F)F)NC1CCCN(C(c2n(C=C)ncc2)=O)CC1 c1(C(N(CC=CC(=O)N(C(C#C)C2CCC2)C)C)=O)ccc([N+](=O)[O-])o1 CC1CC(CNC(=O)C=C2CCC2)CN1C(c1ncncc1Cl)=O c1(CN2CC(N3C(CC)C(=O)NCC3)C2)ccc(F)cc1C#N c1(C(C)NC(=O)C(CN(C)C)NC(=O)COCCCN(C)C)ncn(C)n1 c1(CC(=O)NCC(C2CC2)NC(CCc2cc(C)on2)=O)ccc2nsnc2c1 C12(CNC(=O)CC3COCCN(C(=O)C4CC4)C3)CCC(CO)(CC1)CO2 c1(C(N2CC(C3(NC(c4ccc(C)cn4)=O)CC3)C2)=O)cc(Cl)cc2c1OCC2 c1(C(N(C2CCN(C(C3CC(F)C3)=O)C2)CC)=O)cccc(C(N)=O)c1 Cc1c(C(=O)NCCCCCCNC(=O)C(C)(C)CF)cc(C(F)(F)F)cc1N N1(C(c2ccc(OC)cc2F)=O)CCCC2(CCCN2C(c2cc(C)ns2)=O)C1 CCC(C)CC(C)C(=O)NCC1CC2(CO1)CN(C(=O)COC1CCCOC1)C2 N1(C(C(c2ccccc2)C)=O)CCC2(CC1)CN(C(=O)CC(C)F)CC2CO N1(Cc2cc(OC)cc(=O)o2)CCCC2(CC1)CNC(=O)C2 c1(C(=O)NCC2CCN(C(c3cc(C)[nH]n3)=O)C2)cc2c(C)c(Cl)ccc2[nH]1 C1(C(=O)NCC2(F)CN(C(c3c(O)cccc3Cl)=O)C2)CCCCC1C1CC1 N1(C(C(C)=CC)=O)CC2CCCC(CNC(c3cc(Cl)c(F)cc3F)=O)(C2)C1 C(=O)(N=c1cc(C)n(C2CC2)[nH]1)c1c(C)cccn1.c12ocnc1CNC2 C1(C(N2CCC(C)(NC(=O)CCc3cn[nH]c3)C2)=O)CC(C2CCC2)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CC2CC2(CNC(=O)Cn2ncnn2)C1 Cc1ccc(O)c(C(=O)NC2CC(NC(c3cnc(C(N)=O)s3)=O)C2)c1 N1(C(C2CC(CCC)OCC2)=O)CC2(CC(CNC(=O)Cc3ccoc3C)C2)C1 CCC(CCN=c1[nH]c2c(c(=NCC3(C(=O)NC)CCC3)[nH]1)CCCC2)OC c1(C(=O)NCCCNC(C2CC2OCc2ccccc2)=O)ccnc2c1CCC2 C(=O)(CP(=O)(C(C)C)C(C)C)N1C(CNc2cccc(C)n2)CCC1 CCC(CO)(C(=O)NCC1COCCN(C(c2cc(CCO)on2)=O)C1)OC C(=O)(C1CCCc2nn[nH]c21)NC1CC(C)(NC(C(CC)C)=O)C1 N1(C(c2cccc(C(=O)OC)c2)=O)CCn2cccc2C1C c1(CC(=O)N(CC=CC(=O)NC(c2ccccn2)C)C)cnnn1C c1(C(N2CC(C(=O)NC(COCC)C)C2)=O)cccc(-c2ccc(O)nc2)c1 C(=O)(C(O)CN1CCOCC1)NC1CN(C(C2C(C)C2C)=O)C1 C1(S(C)(=O)=O)(C(N(C2CCC(C(c3ccccc3)=O)CC2)C)=O)CNC1 c1(C(=O)NC(C)CCN(C)C(c2cc(CO)[nH]n2)=O)cc(C2CC2)ccc1Cl c1(CNC2(c3n(Cc4nnn(C)n4)nnn3)CCC2CC#N)ccc(Cl)c(Br)c1 c1(C(N2CCC(CNC(C=CC(=O)N(C)C)=O)C2(C)C)=O)cc(N)c(Cl)c(O)c1 C1(CNC(C2CCO2)=O)CCC(C(=O)NCC2CC(N(C)C)C2)O1 C1(CNC(COCC(C)(C)C)=O)CCC2CN(C(c3ncc(F)cc3F)=O)CC12 C(=O)(C(CNC(c1ccc[n+]([O-])c1)=O)CCC)NCC=CCCC C(=O)(CC(C)(C)C=C)NCC1(C(N2C(C=C)CC2)=O)CC12CCC2 N1(C(CCOCCOC)=O)CCCCC(CNC(=O)C2=COCC2)C1 C(=O)(C(C)S(N)(=O)=O)NCCOC.C1(CC)CCN(C(C2CC3(CSC3)C2)=O)CC1 Cc1ccc(S(=O)(=O)CCC(=O)N2CCC(C)(NC(=O)Cc3cncs3)C2)cc1 c1(NC)cc(Cl)ccc1C(N1CC(CNC(c2cc(F)n[nH]2)=O)C(C)(C)C1)=O C1(NC(CC(C)c2ccco2)=O)(CO)CCCN(c2ccc(C#N)nc2)C1 c1(CNC(=O)OC(C)(C)C)cc(F)ccc1O.C1CCCNC(=O)N(C)CC(=O)N1 CCC(C(=O)NC(C(=O)NC(C)CC(F)(F)F)c1cccs1)C(C)(C)CC CCC(C)(C)C(C)CC(=O)NCc1c[nH]nc1-c1ccc(OC)c(OC)c1 C(=O)(CS(=O)(=O)C1CCCC1)NCC(CNC(C(c1n(C)ccc1)=O)=O)(C)O c1(C(CC)NC(=O)C(=O)NC2CC(C3CC3)C2)ccc(Br)cc1 C12(CNC(C(c3cccc(O)c3)C)=O)CC(CN1C(=O)Cc1ccc(O)nc1)C2 N1(C(C2CC23CCOCC3)C(=O)NCC)CCCC(O)(C2CC2)C1 C1(C(N2CC(F)(CNC(c3c(C)cncc3)=O)C2)=O)CCc2ccccc2C1 C12(NC(COCCC#C)=O)CCCN(C(=O)Cc3cc(F)c(F)cc3F)CC1C2 c1(OCCC)nc(C)ccc1C(N1CCC12CN(C(=O)Cc1ccsc1)C2)=O C1(C)(CC(=O)NCCC(C)NC(CC2(COC)CC2)=O)CCCO1 c1(C(C)C)cc(C(=O)Nc2nc(C(=O)NC(c3cnccn3)C)cs2)n[nH]1 c1(CC(N2CCC3C(NC(C4N(CC)CCOC4)=O)C32)=O)cccc(C#N)c1 c1(C(=O)NC(CCCNC(c2c(OCC)n[nH]c2)=O)C)cc(C(C)(C)C)[nH]c1C n1(CC)nc(C(=O)NCCC2CCC(NC(=O)CCCF)C2)cc1C C1(C(=O)NCC=C2CCN(C(=O)CCc3ccsc3Cl)CC2)CC2C=CC1CC2 C1(Cn2cc(-c3nc(C(=O)OC)cc(OC)n3)nn2)CCCC2(CCOC2)O1 c1(C(=O)NCC2(CN(C(C=C(C)C)=O)C)CC2)c(C(C)C)n[nH]c1C C1(CC(=O)NC2C(C)(C(F)F)C2)CCCCC1NC(=O)C(O)CN(C)C N1(C(C(C2CC2)OCC)=O)CC2CCCC2(NC(c2nccn2CC)=O)C1 c1(C(NOC(CCC)C(=O)N2CCC(O)CC2)=O)cc(Cl)ccc1OC c1(CCC(=O)NCC(C)NC(c2ccc(N(C)C)cc2)=O)ccc(F)cc1Cl CC1(NC(=O)CCNC(c2ccccc2)=O)CCN(C(C2CC2(C)Br)=O)CC1 n1(CCS(=O)(=O)NC(C)(C)C)c(N2CCC3CC3C2)nnc1-c1ccccc1 c1(NC(CC)=O)ccccc1C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CO C1(NC(c2ccsc2)=O)CC(F)CN(C(C2CCOC2=O)=O)C1 c1(C(=O)NC2C(NC(C(C(=O)OC(C)(C)C)C3CC3)=O)C2)cc(Cl)nnc1O CC1(C(=O)NCc2cc(O)nc(CNC(C3CCOC3)=O)n2)CCCC1(F)F N1(CC)CCCC(C(=O)NC2CC(NC(=O)C(c3ccc(C)cc3)=O)C2)C1 Cc1c(Cl)cnn1CC(=O)NC1CC(F)(CNC(=O)C(C)OC2CCCCC2)C1 c1(CNC(=NC)NCC(O)(COC)COC)c(N2CCOCC2)ncnc1Cl c1(C(N(C2CCC(NC(=O)CCC(C)(C)C)CC2)C)=O)ccc2nccn2c1 N1(C(CS(CCC)(=O)=O)=O)CC2CN(C(C34CC3CNC4=O)=O)CC(C1)O2 c1(C(=O)NCCCC(C)NC(=O)Cc2cc(Cl)cs2)nc[nH]c2nccc1-2 c1(OC)cc(C(N2CCOC(CN(C(=O)C#CC3CC3)C)C2)=O)nnc1C1CC1 C12(C(N(C3CCCCC3)CCNC(C=CSC)=O)=O)CCC(C(F)F)(CC1)CC2 CC(C)(CNC(C1CCC12CCC2)=O)CCNC(=O)COc1ccccc1 N1(C(C(CC)n2cncn2)=O)C(C(=O)NCCn2cnnc2C)CCC1C1CC1 C1(NC)CC(CNc2nccc(-c3ccccc3F)n2)C1(C)C c1(OC)ccnc(C(=O)NC2CCCC(NC(=O)C=C3CCC3)C2)c1N C1(C(N2CCC(C)(CNC(c3ccnnc3O)=O)C2)=O)CC2(C1)OCCO2 N1(C(CCOCC#C)=O)CCN(C(c2cc(C)nn2CCC)=O)CC1CC(F)F C1(CNC(C(F)=CCC)=O)CN(C(c2ccsc2SCC)=O)CC1(F)F C1(C(=O)OC)CCN(C(=O)C(CNC(C2(C(N)=O)CC2)=O)CC2CC2)C1C c1(C(N(CC(C)NC(c2coc(Br)n2)=O)C)=O)c(F)c(N)cc(Cl)c1F C1(C(N2C(C)CCSCC2)=O)C2CC(O)C(C2)N1C(=O)CCC(=O)C1CCCC1 c1(CSC(C)C(=O)NCC(C2CC2)N(C)C(c2ccc[nH]2)=O)ccccn1 C(=O)(C1=CC2(CCOC2)C1)NC1(C)CC(NC(c2n[nH]c3c2CCC3)=O)C1 C1(CNC(c2scc(C)c2)=O)CC2(CCC2)CN1C(c1ccn(CC#N)n1)=O c1(CC(=O)NC(CN(C(=O)CSC2CCCO2)C)(C)C)cc2cc(Cl)ccc2[nH]1 C1(C2CNC2)(NCC(O)CN(C(=O)CN(C)CCNCCNC(C)=O)C)CC1 Cc1cc(C#N)cc(C(=O)NCC(O)CNC(c2nc(C(F)(F)F)cs2)=O)n1 N1(C(c2csc(Cl)c2)=O)CCN(C(C23CC(CC(F)(F)F)(C2)C3)=O)CC1 c1(C(=O)NCCNC(c2cc(C(N)=O)[nH]c2)=O)ncnc2cc[nH]c12 O=C1CC(CC(=O)NC2(C(F)(F)F)CC3(CCC3)C2)c2ccccc2N1 N1(C(C(C=C)OC)=O)CC2CN(C(=O)C)CCC12.N(CC)CC C(CCCCC(=O)N1CCN(C(=O)CSCc2ccc(F)cc2)CC1C)=CC N1(C(c2[nH]c3nc(C)sc3c2)=O)CCN(C(=O)CN2CCCCC2)C2(CCC2)C1 C1(NC(C(c2cnccn2)C)=O)CCCN(C(c2c(Cl)csc2Cl)=O)CC1 C1(NC(=O)COC(F)(F)F)CN(C(=O)CC2CCCCC2O)CC1CC1CC1 c1(C2CN(C(C(C)N(C(C3N(CC)CC3)=O)C)=O)C2)nc(=O)o[nH]1 C1(NC(c2cc(CNC(C(C)=NOCC#N)=O)no2)=O)CCCC(O)C1O CC1OCCC1(C)NC(=O)NCC1(CO)CC(C)(C)C1.c12ncccc1NC2=O CCC(CCC(=O)Nc1cccc(Cl)c1)NC(c1cc(C#N)cs1)=O C=CC(C)C(C)C(=O)NCC1(O)CCN(C(c2cn(C)nc2O)=O)CC1 CC(C)C(CNC(N1CCOCC1)=O)CO N1(c2n(CC(=O)NC)nnn2)CCOCC2(C1)CC2(F)F N1(C(Cn2cc(-c3ccn(C)c(=O)c3)nn2)=O)CCc2sc(C(F)(F)F)cc2C1 CCC(CCOC)C(=O)N1CCCCC1CNC(=O)CC1CC=CCC1 c1(C(C(=O)NCC(c2cccc(CO)n2)N2CCCC2)(F)F)cc(F)ccc1F c1(CN(C(C2C(C(=O)NCC#C)C2)=O)CC)ccc(Br)c(Cl)c1 CC(C)C(C)(O)C(=O)NCC1CCN(C(=O)Cn2nccn2)CC1O C1(C)(NC(C(c2cnn(C)c2)NC)=O)CC1(C)C CCC(C)(C(=O)N1CCC(CC(=O)NC)C1)OC(=O)CCc1cncnc1C C(=O)(C1CCc2nccn21)NC1CC(NC(c2[nH]n(C)c(=O)n2)=O)C1 C(=O)(CCCC(C)(C)NC(C1CCCCCN1C)=O)N(CC)Cc1cncn1C c1(NC(CC)CC(F)(F)F)[nH]c(=NC2CCCN(C)CC2)nc2c1ncn2CC CCC(C)(C)C(C)CC(=O)N(C1CCCCC1)CSC1CC(=O)N(C(C)(C)C)C1 C1(CCC)(NC(c2ccc(F)cc2)=O)CCCN(C(c2ncncc2C#N)=O)C1 c12ccc(cn1)c(=O)n2C(C)C.C1(C)(NC(C)=O)CC(NC(=O)CC2C=CCC2)C1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC(C)(NC(c2cccc(CCO)c2)=O)C1 N1(C(C)=O)CC2CC2(C(=O)N(CCCCN(C)C(C2CCN2C)=O)C)C1 CC1(C)CC(NC(C2CCCO2)=O)CN(C(=O)Cc2csc3nccn23)C1 C(C(C(C)C(C)C)NC(c1cnn(C(F)F)c1)=O)NC(c1ccc(C(C)=O)[nH]1)=O N1(C(C=C(C)C)=O)C2CCC(C2)C1C(N1CCOCC1C(C)(C)C)=O C1(NC(C2C(NC(CCc3n(C)ncc3)=O)COCC2)=O)CCOC12CCCC2 N1(C(c2cccc(N(C)C)c2)=O)CC(C(=O)Nc2cnncc2Br)CC(F)C1 CCC(CN(C)C)CC(=O)NC1C2CN(C(c3cnc(OCC4CC4)cn3)=O)CC12 c1(NCCc2ncn(C)n2)nc2ccccc2nc1N(CC1(C)CC1)CC1CC1 N1(C(C(C)C(C)O)=O)CCCC(O)(CCNC(=O)CCc2cocn2)C1 c1(NC(C2CC2C(=O)NC(c2ccc(Cl)cc2)CO)=O)cnn2cccnc12 C1(C2CC2)(CNC(C(CC)F)=O)CCN(C(=O)CC(=O)NC)C1 N1(C(C2C(C)(C(F)F)C2)=O)CCCCCC1CNC(=O)Cc1ccccc1 c1(OCC)ccc(CC(N2CCC(CNC(=O)C(C(C)C)SC)(OC)C2)=O)cn1 CC1Cc2cccc(NC(=O)C(N3CCCC(N)CC3)=O)c2C(=O)O1 c1(NC(CN(C)C(C2CC3CC3C2)=O)=O)cccc(F)c1F C(=O)(C(F)C(C)CNC(=O)CN1CCCC1)N1CCC(C(C)C)(CO)C1 c1(C(N(C2CN(C(c3nc(C)nn3C)=O)CC2O)C)=O)nn(C)c2ccccc12 N1(C(c2[nH]c(C)c(C(C)=O)c2C)=O)CC2(CCCC2NC(=O)CCCN(C)C)C1 N1(C(C2C(CC)CN(C(c3cnccc3C)=O)C2)=O)CCCC(CO)CC1 Cc1c[nH]c(C(=O)NC2CN(C(C3CCC(CO)CC3)=O)CC2C)c1C Cc1c(NC(=O)C(O)CNC(C2(F)CCOC2)=O)cccc1F C1(NC(c2ccn(CC)n2)=O)CCCCCN(C(=O)CN2CCP(C)(=O)CC2)C1 N1(C(C(C=CC)O)=O)CC2(C)CN(C(=O)Cn3cc(C4CC4)cn3)CC2(C)C1 c1(C(=O)NCC(F)F)cc2ccc(-c3cc(O)cc(Cl)c3)nc2[nH]1 C1(C(=O)NC(CN(C(=O)CNS(=O)(=O)N(C)C)CC)C)CC(O)CN1C(N)=O C1(CC(C)(C)CNC(=O)OC(C)(C)C)CCn2c(cnc2-c2ccccc2)C1 c1(C(N2C(CN(C)C(C3C(C(F)F)C3(C)C)=O)CCCC2)=O)cc(=O)n(C)cn1 Cc1cccnc1-n1cc(C2C(C)CCN2C(=O)COc2nc(C)c(C)s2)nn1 CC(CC=Cc1ccccc1)C(=O)NCCNC(c1nscc1Br)=O c1(SC(C)C(=O)NC(C)CN(C(=O)CSC(F)(F)F)C)nnnn1C1CC1 C12(C(C)(C)C)CC(C(=O)NCCCN(CCO)Cc3ccccn3)(C1)C2 c1(-c2cn(C)nc2)ccc2ccnc(Nc3c(F)cc([N+](=O)[O-])cc3F)c2c1 C1(C(C)C(=O)NC2CC2C2CCC2)CCN(C(C2(F)CCCC2)=O)CC1 c1(C(=O)NCC2CC(CC(=O)OC)C2)cc(SCCc2cccs2)nn1C c1(C(C)C)nc(C2C(OC(C3N(C(C)=O)CC34CC4)=O)C2)no1.C(C)(C)(C)S c1(C(=O)NC2CC3(CN(C(C(C)NS(C)(=O)=O)=O)C3)C2)cc2c(nn1)CCOC2 N1(C(c2cccc(OC)n2)=O)CC12CCN(C(=O)CC(C)(C)C)C2 C1(C(=O)NC2(CNC(C(=Cc3cccs3)C)=O)CCC2)CN2CCCC1CC2 CC1(C(=O)NC2CCC(NC(=O)C(C#N)=CC3CC3)CC2)CCCOC1 N1(C(c2cc(C)[nH]c2C)=O)CC2CCCC1CN(C(C1CCCCC1)=O)C2 C(C(C)(O)CNC(c1cc(CC(=O)OC2(C(=O)N(C)C)CCC2)on1)=O)N(C)C O=S(=O)(c1ccc(NCC=CCl)cc1Cl)NCC1CCn2ccnc2C1 c1(CNC(=O)Cn2ncccc2=O)nnc2n1CCS2 Cc1nc[nH]c1CC(=O)NC(C)CNC(=O)C(C)CSc1ccccc1 C(CC(C)C(F)(F)F)NC(C(CCOC)NC(c1ncc(CC)cn1)=O)=O c1(C(=O)NC(C(C)C)(C)CNC(C2CCCC(=O)O2)=O)cncc2nc[nH]c12 C1(CC=C)(NC(c2nocc2Cl)=O)CCN(C(=O)C(C)=CCO)C1 C1(OC)COc2cc(C(=O)OC(C)Cc3cccc(S(C)=O)c3)nn2C1 C(CN=C(NCCNC1CCSC1)NS(C)(=O)=O)NC(=O)OC(C)(C)C C1(C(=O)NC(CNC(C2(N(C)C)CC2)=O)C(C)C)(OC)CCCCC1.CCS CC(C)CC(CNC(=O)CC1(O)CCCCC1)C(=O)NCC1CC1Cl C1(C(N2C(C)CC(NC(c3cnn(C)c3N)=O)C2)=O)Cc2ccccc2CO1 c1(C(=O)NC2CCC(NC(c3cn(C)nc3)=O)CC2)ccc2cccnc2c1O C1(C2N(C(Cc3c(C)con3)=O)CCC2)CCN(C(C2(C)CCCCO2)=O)CC1 C1(n2cc(C(CCC)=O)nn2)CCCCC1N(C(=O)CCC1CCC(=O)C1)CC N1(C(c2ccn(CC)n2)=O)CC(C)(C)OCC1CNC(=O)CN1CC(=O)NC1=O c1(C(N2CC(CNC(C34C(C)OC(CO)(C3)C4)=O)C2)=O)cc2c(Cl)cccc2s1 CN1CCN(c2cc(NCC3CC4CCCCC34)ncn2)C2CC12 N1(C(c2c(C)n(C)cc2)=O)CCN(C(C2CCCSC2)=O)C(C)C1 c1(OC)cccc(C(CF)NC(=O)NCCSCC(=O)OC)c1 N(C(=NCCCCCCC(C)C)NC1CCCCC1)C1CC(OCCOC)C1 Cc1scnc1C(=O)NCC1(C(=O)N(C2CC2C2CC2)C)CC1 Cc1nc2c(C#N)cnn2c(C)c1CC(=O)NCC(C)(O)CNC(=O)COCCF C12(CC(N3CC(N4CCN(C(CN5CC(C)C5)=O)CC4)C3)=O)CCCN1CCC2 c1(OC)ccc2oc(-c3cccc(C(=O)OCCF)c3)cc(=O)c2c1 c1(OCC(=O)N(CC(C)NC(c2c(C(C)C)cco2)=O)C2CC2)ccc(Cl)c(F)c1 C1(CCNC(=O)CC2CCCC2)CN(C(=O)CC2CCCC3(CC3)C2)CCCO1 C#Cc1ccc(C(=O)N(CC(O)CN(C)C(c2nnc(S)n2C)=O)C)o1 N1(C(c2cc(C)sn2)=O)CC(C)(C)OCC1CNC(=O)COC1CCCC1 C(COC)(CC(=O)NC(C)(C)CCOC)N(C(=O)C(C)(C)C)C c1(C(N2CCC(C(C(=O)NCCc3ccc(C)cc3)F)C2)=O)nc(C)ccc1O CC(C)CC(C)C(C(=O)NCC1CC1)N1CCCCC1c1nc[nH]n1 CCC(C(=O)NCCCOCCNC(=O)C(F)(F)CC1CC1)C(C)O c1(C(N2C3CCC(NC(=O)Cc4ccco4)(CC3)C2)=O)cc2nccn2c(O)n1 c1(OCCC)ccc(C(=O)NC(C2CCCC2)CNC(=O)COCCC)cc1 Cc1nncn1NC(=O)CC(C(C)(C)C)NC(c1nnc(S)n1C)=O CC1CN(C(c2nccs2)=O)CC1NC(=O)C(F)=C1CCCC1 c1(CN2C(CNC(C3CN(C(C)C)C3)=O)CC2)ncccn1 C#CCC(C)(C(=O)NCc1ccc(Cl)o1)NC(c1nnn(C)c1N)=O c1(C(N(C(C)CNC(c2nocc2C)=O)CC)=O)nc(OC)ccc1Cl Cc1ccc(F)c(S(=O)(=O)N2CCc3[nH]nc(C(N4CCCC4CO)=O)c3C2)c1 CC1CCc2nc(C(N3CCC3CNC(=O)CN3CCCC3C)=O)cn2C1 c1(C(=O)NCCN(C(=O)C=Cc2cnn(-c3ccccc3)c2)C)nc(=N)cc[nH]1 C(=O)(C1=CCC2CCC1N2C(=O)CCc1ccc[nH]1)NCC1CCCN(C)C1=O CC(C(=O)NCC1CN(C(C2(F)CC3(CCC3)C2)=O)CCCO1)S(N)(=O)=O CC1=CCN(C(c2cccnc2CNC(=O)CSc2cn[nH]c2)=O)CC1 N1(C(C(C)N(C)C)=O)CCN(CC(C)NC(c2ccc(COC)o2)=O)CC1 C1(CNC(CCc2scc(C)n2)=O)CC(C)N(c2nnc(CC(C)C)s2)C1 CC1(C)C(NC(=O)CSc2csnn2)CCN1C(C1CCC1)=O c1(OC)ccc(Cl)c2sc(NC(=O)NCc3ccn4ncnc4c3)nc12 S(=O)(=O)(c1ccc(C(=O)NC2CCN(C(=O)COCCF)C(C)C2C)o1)NC N1(C(C(CC=C)NC(=O)Cc2cncnc2O)=O)CCN(C)C(C)C1 CC(C)CCC(=O)NCC(=O)NCC(C)(O)CNC(=O)C=Cc1cocn1 c1(C(N(C(C)CNC(=O)CN2CCSCC2)CC)=O)cn(C(C)C)nn1 N1(C(C(C=CC)O)=O)CC(C)C(C)(CNC(c2cnn(-c3ccccc3)n2)=O)C1 C(=O)(C1SCCc2ccccc21)NC(C)(C)CCNC(C1CC2(CC2)CO1)=O N1(C(C#CC)=O)CC(NC(c2c(O)cccc2O)=O)CC(F)C1 Cc1sc(N)c(C(N2CC(NC(=O)C(F)CC3CCC3)C3(CC3)C2)=O)c1C C1(C(=O)NC(CCNC(C(CC)(C)C(N)=O)=O)(C)C)Cc2ccc(F)cc2O1 C1(CNC(c2cc(C)oc2C)=O)CC(C)CN(C(C2CCCCCN2C)=O)C1 c1(OC(C(=O)NCCN(C(C(F)=CCC)=O)CC)C)ccc(F)cc1 n1(CCOC)ncc(C(=O)NC2CCCCC2CNC(c2sc(F)cc2Cl)=O)c1C C12(COC)CC(CNC(c3ccc(F)c(F)c3)=O)(CN1C(C1CCC(F)C1)=O)C2 n1(CC(=O)N(CC(C)NC(C2CC2(C)C(F)F)=O)C)cnnc1O Cc1cc(O)ccc1-c1cn(C2CN(C3CCC(=O)N3C)C2)nn1 c1(C(=O)NC(c2ccccc2)C(C)NC(C(F)=CCC)=O)cn(C)c(=O)n1C c1(C(=O)NCC2CN(C(Cc3n[nH]c(=NC)s3)=O)C3C2C3)cnc2cc[nH]c2c1 CCC(CC(=O)NC(C)(C)C(=O)NC1(C(=O)NC)CC1)C(F)F N1(C(C2(C)N(C(c3n(C)cnc3)=O)CC=C2)=O)CC(S(C)(=N)=O)C1 C=C1CCC(C(=O)NC2(c3cccc(F)c3)CCN(C(C3COC3)=O)C2)CC1 C1(NC(C2(COC)CC(=C)C2)=O)CC(C(=O)NCCc2cc(C)no2)=CC1O Cc1ncccc1C(=O)NCCCCN(C)C(C1CCC(O)C1)=O c1(C(N(C(CNC(C(CC=C)(C)C)=O)C)C)=O)cnc(O)n(C)c1=O c1(N(C)Cc2n(C(C)C)cnn2)nc2ccccc2nc1N1CC2CC1C2 CCCCCCC(C)C(=O)N(CCC(N1CCC2C(C(N)=O)C2C1)=O)C1CC1 Cc1cnc(C(=O)NCCC(C)(C)C(=O)NC2CCCCCC2)cc1C Cc1ncnc2c1CC(C(=O)NC(C1CN(C(C3CCS(=O)(=O)N3)=O)C1)C)CC2 C1(CN(CC(C)O)CC)CNCC(F)C1 c1(OC)ccc(NC(c2ccc(NC(=O)C(C)N(C)C)nc2)=O)cc1-n1cnnn1 C(=O)(CCCCCS(N)(=O)=O)N1CCN(C(c2[nH]n(C)c(=O)n2)=O)C(C(F)F)C1 Cc1ccc(C=CC(N2CCCC2CN(C(=O)C(C)CC2CCC2)C)=O)cn1 CC(C)(C)C(CO)C(=O)NCC1(C(N2CCC3(CCC3)CC2)=O)CCC1 C(=O)(CCCC(=O)N1CCCCC1CCNC(C1C2CCN1CC2)=O)OC N1(C(C2CC(CC)C(=O)CC2)=O)CC(C)CN(C(=O)C(F)=C2CCCC2)C(C)C1 c1(CNC2CCC(C(=O)Nc3c(OC)nc(C)cc3)C2)c(F)ccc2occc12 c1(C(N2CC(N(C)C(c3cn(-c4ccccc4)nn3)=O)C2)=O)cnccc1Cl C1(N(c2nc(C)cc(C)n2)C(C(C)NC(C=C)=O)=O)CCNCCC1C c1(C(=O)OC)cc2c(Nc3ccc(C)cc3OCC(F)(F)F)ncnc2n1C c1(OC)ccc(CC(N2CC3(CCN3C(c3ccc(O)c(F)c3)=O)C2)=O)cc1C C(=O)(CC(CC(=O)O)C(F)F)NCc1cc(C)nc(C2CCCCC2)n1 C1(C(=O)NC2CC(NC(C(CN(C)C)N(C)C)=O)C2)COC2(CCC2)C1 CC(C)C(F)(F)CC(=O)NCCOCCCNC(c1csnn1)=O c1(CN2CCC(NCC(CN=[N+]=[N-])O)CC2)csc2ccc(Br)cc12 O=C1OC2C(NCCc3nnc(-c4ccccc4)o3)C3CC1C2O3 C1(C(=O)NCCCCN(C)C(C2CC(O)(C(F)(F)F)C2)=O)CCC2(CCC2)C1 c1(C(=O)NC2C(C)CN(C(=O)CN3CC(=O)NC3=O)C2)cc([N+](=O)[O-])cnc1N C1(CCNC(Cc2cc(C)sc2)=O)CSCCN1C(=O)CC1CC(C2CC2)C1 Cc1cc(O)c(C(=O)NCC2CCCN(C(=O)COc3ccccc3)CC2)nn1 c1(OC)cnc(F)c(C(=O)N(CC(C)(C)NC(=O)Cc2cnccc2C)C)c1 c1(C(=O)NCC(C)N(C)C(C2C3CC4C(C3=O)C24)=O)ccc2c(c1)CC(=O)N2 Cc1ccc(C(=O)NCC2CCCCC2NC(=O)C2=CCSC2)cc1N C(=O)(C#CC1(C(F)(F)F)CC1)NC(C)CCCCNC(=O)C=Cc1ccccc1 CC(CN=c1[nH]c(N2CCC(CF)C2)nc2c1COC2)c1cccc(F)c1 C1(COC)(CNCc2ccc(CN(C)C)cc2)CC(F)(F)C1 c1(CC2N(C(=O)NCCn3ccnn3)CCCC2)cccc(Cl)c1Cl N1(C(C(C)NC(CC)(C)C)=O)CC2(CC(NC(=O)C3=C(Cl)CC3)CO2)C1 CC1CC(C(N)=O)CN(C(=O)CCC(c2cc(F)ccc2F)=O)C1 c1(COC)ccccc1CNC(=O)NC(CC(=O)OC(C)(C)C)c1ccccc1 Cc1cc(C(=O)NCC(C)(O)CNC(C2COCCO2)=O)c(N)c(Cl)c1 CC(c1ccccc1)=CC(N1CCC(O)C(NC(C2CCC(C)(C)C2)=O)C1)=O CCCCCC(O)CC(=O)N1CCCN(C(=O)COc2ccc(Cl)cc2)CC1C Oc1cc(C(F)(F)F)ccc1SCCN1CCS(=O)(=O)CC1 c1(C(C(C)C)SC)ccc(-c2nnnn2CCCC2CC2C)cc1 C1(NC(c2cn(C)nn2)=O)(CNC(C2CCC2C(N)=O)=O)CN(CC)C1 Cc1cc(C(N)=O)cc(C(=O)NC2CCOCC2NC(=O)CC2CCOC2=O)c1 CCCC(CC(=O)NCC1(CO)CC2CC2C1)NC(=O)C(C)(COC)OC C1(OC)CC(CNC(=O)CCOc2cccnc2)N(C(=O)C=C2CCC(C)C2)C1 N1(C(CC2N(C(CC(CC)O)=O)CCOC2)=O)CCc2cc(C(=O)O)ccc2C1 C1(F)(CNC(c2nn(C)c(Cl)c2)=O)CCCN(C(=O)C2=CCCCO2)CC1 Cc1ccc(C(=O)CCC(N2CCC(NC(=O)CC3CCOC3)CC2)=O)cc1 C(CC(C(=O)Nc1ccc(C2CC2)nc1)NC(=O)COCC(F)F)=CC C=CC1OCCC1NC(N1CCC(C)(c2cccc(F)c2)C1)=O c1(-n2c(C(=O)NCC3C(NC(=O)COC4CCOC4)C3)cnn2)ccccc1Cl C1(NC(C=CC(N)=O)=O)CCCOC12CCN(C(c1cc(F)cnc1Cl)=O)CC2 c1(C(N(C)CC2CCN(C(=O)OC(C)(C)C)C2)=O)ccccc1S(=O)(=O)C(F)F c1(C(=O)NC2CCCC(NC(Cc3cc(C)[nH]n3)=O)C2)cc2sc(Cl)cc2s1 C1(NC(c2cc(Br)co2)=O)CN(C(C2CC2C(F)F)=O)CC1C(F)F C1(C(N(CC(C)NC(c2ccco2)=O)CC)=O)CC(C(C)=O)C1(C)C C(=O)(C(C)C(O)CC(C)C)NCC1(F)CN(C(c2ccc(C)nc2)=O)C1 CCCCCC(CC)C(=O)NC1CN(C(c2ccnn2CC)=O)CC2CC12 c1(C(N(CCNC(C(C)C2CCOC2)=O)C)=O)cc(Cl)cc(Cl)c1N C1(C(N2CC(C(C)NC(CC(=O)NCC)=O)OCC2)=O)(CF)CC2(CCC2)C1 C1(C(=O)NC(CN(C)C)C(N2CC(F)(C3CC3)C2)=O)CC(=O)C12CCC2 C1(C(=O)OC)Cc2ccccc2CN1CC1Cc2ccc(-c3nn[nH]n3)cc2O1 C1(NC(Cc2nc(C)c(C)s2)=O)CN(C(C2CC23CCCC3)=O)CC12CC2 C1(NC(c2cc(C)sc2)=O)CCN(C(=O)CNC(c2ccco2)=O)C(C2CC2)C1 N1(C(CCC(=C)Br)=O)CC2CCC2(CCNC(=O)CCn2cnccc2=O)C1 c1(CC)ccc2[nH]ccc2c1.N12CCCC(COC)(C1)NC(=O)C1(COC1)C2=O c1(CCC(N2C(C(C)NC(=O)C=CC=C(Cl)Cl)CCC2)=O)c(C)n[nH]c1C C1(C(C)NC(C2N(C(Cc3cc(C)no3)=O)CC2)=O)CC2(CCC2)C1 c1(OC)ccnc(NC2CN(C(=O)Cn3cncc3C)CC2C)n1 c1(C(C(=O)NCC(CNC(COCC(C)C)=O)F)N(C)C)cc(F)c(F)c(F)c1 N(C(=NCC1CC2(CCOCC2)C1)N1CCC(NS(C)(=O)=O)C1)C(C)C C(=O)(CC(C(F)(F)F)n1cccn1)N.Cc1cccnc1C(=O)NCCNC1(C)CC1 N1(CC)N=C(C(=O)N2CCC(C)N(C(=O)C3=C(C)OCC3)CC2)CCC1=O c1(C(=O)NCC(C2CC2)NC(C(C=C)OC)=O)ccc2cnnn2c1 c1(CNC(NC(COC)C)=NCC2(C(F)(F)F)CCOCC2)ccc(C)c(C)c1 C(C(C)(CO)OC)NC(C(C1CC1)NC(C(F)=CCC)=O)=O N1(C(C(CC)(C)O)=O)CCC2(CCOCC2)C(CNC(c2ncccc2Cl)=O)C1 C1(C(=O)NCC2C(NC(c3nc(N(C)C)oc3)=O)CCC2)CCC2(CCC2)CC1 c1(NC(C2(F)CN(Cc3c(C)ncs3)C2)=O)c(C#N)cnc2c(C#N)cnn12 n1(CC(=O)NC(c2cn(C)nn2)C(=O)NCC(C)CO)cccnc1=O N1(C(CC(=C=C)C)=O)CCCCC2(CCN(C(C3(COC)CCC3)=O)C2)C1 N1(C(c2c(C)cn(C(C)C)c2)=O)CC2CN(C(=O)CCC=CC(C)C)CC2C1 c1(OC)csc(C(=O)NCC(F)CNC(=O)C(C)(C)c2ccccc2)c1OC C1(C(C)NC(CCSCCC)=O)CCCN1C(c1ccc[nH]1)=O N1(C(CC)=O)CCN(C(c2sc(Br)c(C)c2C)=O)CC1CC1CC1 C=C(C)CCCC(=O)N1CCCC(CCC)(NC(c2cncc(OC)c2)=O)C1 CCC(CC)C(=O)N1CC2CC2C1C(=O)NCCC(C)N1CCCC1 CCN=C(NCCCc1snnc1C)NCc1cnnn1-c1ccccc1 CC1CN(C(=O)CCOc2ccccc2)CC1NC(C1CC12CCOC2)=O C1(NC(c2c(C)nsc2N)=O)CC2(CCC(NC(=O)OC(C)(C)C)CC2)C1 CC(CCCCNC(C1CC1C#N)=O)NC(=O)CC1(C)CC(F)(F)C1 c1(C(C(F)(F)F)OC(C=C2CCN(C)CC2)=O)c(F)cccc1F c1(C(CC(=O)N(CC(CC)NC(=O)C(F)(F)CO)C)C)ccc(F)cc1 CSC=CC(=O)NCC1(NC(c2scnc2C(F)(F)F)=O)CCC1 c1(OC)cnc(Cl)c(C(=O)NCCN(C(=O)C(C)n2cccc2)C2CC2)c1 c1(CN(C(C(N2C(CC)CC2)=O)=O)Cc2ccccc2F)nn(C)cc1N C(=O)(CCN(OC)C(=O)C1CCCC(CC)CC1)NCC1C(CCC)C1 C1(C)(c2nc(CC)[nH]n2)CCN(C(c2cnn(C)c2)C(=O)NCCCC2CC2)C1 c1(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(CCC)O)C)cccc(Cl)c1 c1(CCNC(C(C2CCN(C(C3CS(=O)(=O)C3)=O)C2)C)=O)cnn(C)c1 C1(NC(CC2CCCN(C(c3c(C)csc3)=O)C2)=O)COC2(CCC2)C1 C=C(C)CC(=O)NCCOCCCN(C)C(c1csc(CC(F)(F)F)n1)=O C1(NC(Cc2nc(C)sc2)=O)CC2CC(C1)N(C(c1cnn(CCO)c1C)=O)C2 N1(C(c2n(CC#C)ccc2)=O)CCC(C(C)NC(c2cn(C)[nH]c2=N)=O)CC1 N1(C(C(C)OCC2CCCCO2)=O)CCC2(CC1)CCN(C(C1CC1C#N)=O)CC2 C1(NC(CCc2cncc(OC)c2)=O)CC(O)CN(C(=O)Cc2cnoc2)C1 c1(OC)ccnc(O)c1C(=O)NCC1(NC(C2CCNC2=O)=O)CCOC1 c1(C(=O)NC2CC2NC(C2C=CCS2)=O)ccc(F)c(Cl)c1F c1(C(=O)NCC(Cn2cc(C(C(C)(C)C)O)nn2)(F)F)nc(=N)cc[nH]1 N#CC1CCN(C(c2nc[nH]n2)=O)C(C2CC2)C1 C12(NC(C(C)N3CCCC3)=O)CCCC(NC(=O)CSS(C)(=O)=O)(C1)C2 c1(OC)cc(S(=O)(=O)NCC2CC23CC3)c(Cl)cc1-c1csc(=N)[nH]1 C(C)(C)(CC(F)C(=O)NC1(CF)CC1)NC(C(N1CC(C)C1)C)=O n1(CC=C)cccc1C(=O)NCC=CCNC(=O)C(C)Cc1ccco1 CN1CC=C(CC(=O)N2CCC(F)CC2C(=O)NCCCSC(F)F)CC1 c1(C(=O)OC)c(C)nn2ccc(NC(=O)NC3CCC(F)(F)CC3)nc12 c1(C(N2CCN(C(c3ccc(C)o3)=O)C(C#N)C2)=O)c(F)ccc2[nH]ccc12 C1(c2ncc(C(=O)OC)[nH]2)CCCN(N2CCC3C(CNC(=O)C3)C2)C1 N1(C(c2c(COC)cc[nH]2)=O)CCOC(CCCNC(C2CCC(F)(F)C2)=O)C1 c1(-c2nc(CC(CC)CC)n(C3(OC)CCOCC3)n2)cccc(S(C)(=O)=O)c1 c1(CNC(C2SCCN(C(c3ccc(OC)s3)=O)C2)=O)cccc(O)c1F C1(NC(c2c(CC)cc[nH]2)=O)CC2CN(C(c3cnc(CC4CC4)s3)=O)CC2C1 N(S(=O)(=O)N1CCC(n2c(CC)nc3cc(OC)ccc23)C1)(CCCC)CC N1(C(C2(F)CCN(Cc3cc(F)cc(Cl)c3)C2)=O)CCc2cccc(Cl)c2C1 C1(CC)C(NC(=O)C(C)CNC(C)=O)CCN1C(c1ccc(NC(C)C)cn1)=O N1(C(C=C(C)C)=O)CC2CCN(C(c3ccc(C)c(CO)c3)=O)C2C1C C1(NC(CC(C(=O)OC)C)=O)CCC2(CC1)CC(NC(=O)Cc1csc(C)n1)C2 c1(C(=O)NC(C(=O)NC(C2CCOC2)C#C)c2cccs2)coc(C)c1 C1(NCc2n(C)ccc2)CCC(CC(=O)NCc2cccnc2F)CC1 C(=O)(C(C)(C)CCC#N)NCC1CCC(C(N(C)CC2CC(=C)C2)=O)O1 N1(C(CCSC)=O)CCC(CNC(c2oc(-c3cnn(C)c3)nc2C)=O)CC1C N1(C(CC2(C)CCCC2)=O)CCC2(CC1)CC2NC(c1cc(C#N)c[nH]1)=O N1(C(=O)CC(F)(F)Cl)CCN(C(C2CC(O)C2)=O)CC12CC2 C1(C(N2C(C)C(NC(c3ccc(F)c(O)c3)=O)CC2)=O)CC(C)(C)SC(C)(C)C1 CN1N=CC(CC(=O)NC2CCCC2C(=O)NCC2CCC3(CC3)C2)C1=O c1(CC)nccn1C(C)CC(=O)N1CCC(C(C)NC(C2CC3(CC3)C2)=O)C1 C(CC(C)(C)C(=O)N1CCOCC(NC(C2CC2C(F)(F)F)=O)C1)SC c1(C(N2CCC(N(C(C(CC)C)=O)CC3CC3)C2)=O)cc(CC)cc2c1OCC2 Cc1csc(CCNC(=O)C(CC2CC2)NC(c2cc(Cl)c[nH]2)=O)n1 c1(NCc2ncc(OC)nc2)cc(=NC2CCCc3occc32)[nH]c(C(C)C)n1 O(C=C(C#N)C(=O)N1CC(CNC(=O)C(c2ccc(Cl)c(F)c2)O)C1)CC N1(C(CCC(=O)NC)=O)CCC2(CCC2NC(c2cn3cc(C)sc3n2)=O)CC1 C(=O)(C(C)(CO)NC(=O)CC1(C)CC1)NC(c1nc(C)[nH]n1)C C(=O)(C(C)(C)CC(C)(C)C)N(C(=O)CCC(=O)N(CCC)C)C.CNO C(=O)(C1=CCCSC1)N(CC(C)O)CCNC(c1n(CC#C)ccc1)=O CC(C)S(=O)(=O)C(C)C(=O)N(C1C2CN(C(=O)C=C3CCSCC3)CC12)C CC1CCN(C(=O)CCc2ccc(F)nc2)CCN1C(C1(C2CCCO2)CC1)=O C(=O)(CCC(=O)NC(C)(C)CC=CC(=O)NC1(CC)CCOC1)NCCC CCCCC(O)CC(=O)N1CCCC1(C)CNC(c1cn(C(F)F)c(C)n1)=O N1(C(C2CC(CC)OCC2)=O)CC2(C1)CN(C(C1CC1c1ccccc1)=O)C2 N12CC=C(c3cncnc3C1=O)CC2.c1(COC(C)=O)cc(Br)ccc1C#N C1(C(F)F)(NC(C(C2CCCC2)OCC)=O)CCCN(C(=O)OC(C)(C)C)C1 C1(F)(CNC(c2ccc(Cl)cc2C(F)F)=O)CCCN(C(C2CCCC2)=O)C1 c1(OC)cccc(=Nc2cccc(C(N3CC4(C)CC3CCO4)=O)c2)[nH]1 N1(C(c2c(C)noc2)C(=O)Nc2ccc(F)cc2)CCC2(CC1)CC(C1CC1)=NO2 N1(C(C(C)OCCOC)=O)CC2CC1CN2C(c1sc(Cl)c(Cl)c1OC)=O N1(C(CCCSC)=O)CCN(C(C2(c3cccc(C)c3)CCC2)=O)CC1 C(=O)(C(C)C(C)NC(=O)CC1CC(=O)C1)NC1(c2nc(C)on2)CC1 c1(C(=O)NC2C3(CN(C(c4cccc(N)c4O)=O)C3)CC2)cc2ccccc2s1 c1(C(=O)NCC2C(NC(c3cc(CC)nn3C)=O)CC2)cc2cc(F)ccc2o1 N(C1CCOc2cc(F)ccc21)C(N1CC(C2C(NC(=O)OC(C)(C)C)C2)C1)=O c1(C(C)NC(CN(C(=O)CSCCC#N)CC=C)=O)cn(C)cn1 c1(CCNC(=O)NC2CC(C)OCC2)cc2ccccc2o1 C(CCC(C)C(=O)NCC1(F)CN(C(c2cc(O)cc(Cl)c2)=O)C1)OC C1(C(N(CC(CN(C(CCC=C=C)=O)C)O)C)=O)COCCC1(F)F Cc1cc(O)nc(C)c1C(N1CC(NC(=O)CSCC(F)F)CC(F)(F)C1)=O c1(C(=O)NC(CC)CNC(=O)CN(C)CCO)ncnc2c1OCCO2 C1(c2cccc(F)c2)(C(=O)NCC2C(NC(=O)C=CCO)CCC2)CCCCC1 n1(CC)cc(Cl)c(C(=O)NCCCCC(C)NC(=O)CC(C)c2cnn(C)c2)n1 C1(CNC(C2(C=C)CCC2)=O)CCC2(CN(C(c3cc(C)c(Cl)cc3C)=O)C2)O1 CC(CC1CC1)C(=O)NCC1CCN1C(C1CCC(C(=O)OC(C)(C)C)O1)=O c1(OC)ccc(CO)cc1C(=O)NC1CS(=O)(=O)CC1NC(c1occc1C)=O N(C(=NCC1CC(F)(C(=O)OC)C1)N(C)Cc1ccc(C)cc1)C(C=C)C CCC(C)C1C(=O)N1C.C1(NC(c2cnc(C)o2)=O)CCN(OCC)CC1 c1(N2CC3CN(C(c4cc(Cl)cc(Cl)c4Cl)=O)CC32)ncnc2sc(Br)cc12 C1(c2c(C(=O)NC3(CC#C)CC3)c[nH]n2)CCCCN1C(=O)CC(C)N(C)C N1(c2n(C)nnn2)CCC2(CC2CO)C1 C1(F)(CNC(=O)CCCn2cncn2)CCN(C(=O)CS(=O)(=O)NC2CC2)CC1 N1(C(c2c(C)nc(C)o2)=O)CC2CCC(C1)N(C(c1ccc(F)c(CO)c1)=O)C2 c1(C(=O)NC2CN(C(Cc3cnc(C)s3)=O)C(C)(C)C2)ccc2c(n1)NCC2 N1(C(c2cnn(C)c2N)=O)C(C(=O)NCc2ncsn2)CC2CCCC12 N1(C(C(C(C)CC)N(C(C(C)OCC#C)=O)C)=O)CCC(N(C)OC)CC1 CC(C)CCC(O)C(=O)NC(CC(=O)NC(C)C(C)(C)C)C(F)F c1(C(C)C)ncc(C(N2CCN(C3CCCC3NC(C3CCO3)=O)CC2)=O)cn1 C1(CC=C)CCCCC1N=c1[nH]c(=NCc2cccc(F)c2Cl)[nH]c2c1CCC2 Cc1nc(C(F)(F)F)ccc1C(=O)NC1CCCCC1NC(=O)CS(C)(=O)=O N1(C(C(COCC)n2cc(CCOC)nn2)=O)CCCC(OC2CCOC2)C1 C1(NC(C(C2CCCC2)OC)=O)C2CC(NC(C3COCC3(C)C)=O)CC12 N1(C(C(C)OCC#C)=O)CCCC(CC(=O)NCc2cc(C)cc(C)n2)CC1 CC1CCN(C(C2CCC(C)CC2)=O)CC1NC(C1COC(C)(C)C1)=O CC(CCCCCO)NC(C1CC2CCC1(CO)C2)=O.c12ccccc1C(=O)N2 CC(O)C(C)C(=O)N(C)CCC1CCCCN1C(c1csnc1Br)=O c1(C2N(C(=O)NCc3c(F)ccc(CC)c3)CCS2)c(C)cc(C)cc1C N1(C(C(C)N(C(c2cn(CC=C)nc2)=O)C)=O)CCC2(CCOC2)C1 N1(C(C2(CC=C)CC2)=O)CCC(NC(C2CCCCC23CC3)=O)C12CC2 c1(C(=O)NCC2CN(C(c3c(CC)ccs3)=O)C(C)C2)cnn2cnnc2c1 c1(N(c2cc(C)ccc2N2CCC3CCNCC3C2)C)cnn2c1OCC(C)(C)C2 c1(CNC(CN2C(C)CCC2)=O)ncccc1C(=O)NCC1(O)CCSCC1 c1(CC(N2CC(NC(=O)C(F)=CC3CC3)C3C2C3)=O)ccc2c(c1)OCCCO2 N1(C(C)=O)CC(C(=O)NC(=O)CSCc2ccc(F)cc2)CC12CCOC2 C1(N(C(=O)CCCN2CCOC2=O)CC)CCN(C(=O)CC2CCOC2=O)CC1 C1(=CC(=O)NC(CCOC)CNC(=O)Cn2nc(C)cc2C)CCC(C)(C)CC1 C(=O)(CCCCC(N)=O)N1CC(CCNC(C(C(COC)C)C)=O)(OC)C1 O=C(C1=CC2CCCC12)N1CC2(C1)CN(C(C1(CCF)CCOCC1)=O)C2 c1(C(=O)NC(CNC(c2c(C)coc2C)=O)(C)C2CCC2)ccc(S(C)=O)cc1 C(=O)(C1CCCc2ncnn21)NCC(CNC(c1c(OC)cc(Cl)cc1)=O)F c1(C2C(C(=O)NC3(C)CN(C(c4cnc(CSC)s4)=O)C3)C2)ccc(F)c(F)c1 C1(COC)(NC(c2cscc2C(F)(F)F)=O)CCCN(C(=O)C(F)(F)C(F)F)C1 N1(C(C=CCCC)=O)CCCCCC1CNC(c1cc(OC(F)F)ccc1C)=O C1(NC(Cc2ccc(C)s2)=O)CC(C(=O)N2C(CO)CC2C)=CC1O CC1CN(C(C2(CO)CCC2)=O)CC(C)N(C(c2cnc(C3CC3)nc2)=O)C1 c1(C(N2CCC(C(CNC(CC(C)(F)F)=O)(C)O)C2)=O)cc(C(N)=O)ccc1F C1(COC)(NC(C2CC2(Cl)Cl)=O)CCCN(C(c2ccc(NC3CC3)cc2)=O)C1 c1(C(=O)NCCCC2CCN(C(CC(CC)C)=O)CC2)cc2ccccn2n1 N1(C(c2ncc(NC)nc2)=O)CCC2CN(C(c3cn[nH]c3)=O)CC2CC1 c1(CC(=O)N(CCCNC(=O)CNC(c2ccsc2)=O)CC)ccoc1C c1(C(N2CC3C(CNC(CC=CCC)=O)(C3)C2)=O)ccc2c(c1)CCC2(C)C N1(C(CC(C(C)C)O)=O)CC2CC(NC(=O)CC3CC(F)(F)C3)CC1C2 C(C(=O)NC1CC(CO)C1)(C1=CCC2CC2C1)NC(=O)OC(C)(C)C Cc1ccc(Cn2nc(-c3cccs3)nc2CC(F)(F)F)cc1 c1(C(c2n(CCCSCC)nnn2)NCCn2cnnc2)cnn(C)c1C(C)C C(C1=NOC2(CCC2)C1)NC(C(CCCC)NC(=O)CCc1cscn1)=O C1(F)(C(N2C(C(=O)OC)CC2)=O)CCN(C(=O)C=CCO)CC1 Cc1c(C(N2CCCC2C(C)NC(=O)C2=C(Cl)CC2)=O)n[nH]c1C1CC1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CSc2ccc(Cl)nc2)C(C2CCC2)C1 Cc1nc(C(F)(F)F)ccc1C(N1CCC(=CC(=O)Nc2ncc(F)s2)CC1)=O c1(C(=O)NC2C(CNC(C3(C)C=CCCC3)=O)COC2)cc(O)cc(=O)o1 CCC(CC(=O)N1CC(CC(=O)N(CC#CC)CC)C(C)C1)SC C#CCCC(O)C(=O)NC(c1ccccc1CC)CNC(c1ccccc1F)=O N1(C(CSC(C)C)=O)CC(CNC(=O)CCCNC(=O)C(C)(C)C)CCC1C C1(NC(C(CCNC(C(C(CC)O)C)=O)OC)=O)CCc2nncn2C1 c1(CNC(C2CCC(C(C)(C)C)CN2)=O)cccc(Br)c1O N1(C(CCC2(C)CC2)=O)CC(CNC(=O)Cc2ccc(Cl)nc2)C2(CC2)C1 c1(OC)ccc(NNC(=O)Cc2cccs2)cc1 C1(OC)CN(C(=O)C(C2CCC2)NC(=O)CC2CC2(C)C)C1 n1(CC)ncc2c(N3CC(C)CN(C(c4ncn(C)n4)=O)CC3C)ncnc12 N1(C(C(F)=C(C)C)=O)CCc2sccc2C1CNC(=O)CCOCC1CCCO1 c1(CC(N2C(CC(=O)OCC)CCC2)=O)cc(N)ccn1 C(=O)(CC1NC(=O)c2ccccc21)NC1CN(C(CCCC(C)=O)=O)CC1C N1(C(C(C2CCCN(C(Cc3c(C)cccc3)=O)C2)(C)C)=O)CC2CCOC2C1 C1(CCOC)CN(C(=O)C(C2CC2)OC)CCN1C(c1cc(Br)co1)=O C(CCCCC(=O)NC(=O)COCCOCCNC(C1C(CC)C1)=O)SCC c1(CC(=O)NCC2C(NC(c3nc(OCC)oc3)=O)COC2)cc(F)ccc1F c1(OC)ccc2nc(C)nc(N3CCCC3C(=O)NCC3CCCO3)c2c1 CN1CCCC(C(C)(C)C(N2CCC(CO)(NC(=O)CS(=O)(=O)N(C)C)C2)=O)C1 C1(C(=O)NCc2ccncn2)(CC)CCN(C(C2CN3CCC2C3)=O)C1 CC1CN(C)CCC1NC(C1CNC(=O)CN1C(c1ccc(CC#N)cc1)=O)=O c1(NC(=O)NCC2N(C(=O)NC3C(C)CCCC3)CC2)nc2ccc(Cl)nn2n1 CN1CCC(C(=O)NCC(C)(CO)NC(c2cnc(Cl)s2)=O)c2ccccc21 C1(C#N)(C(=O)NCCC2(OC)CN(C(C(CC#C)(C)C)=O)C2)CCN(C)CC1 C(=O)(C(F)C(C)CC(C)(C)C)N(C)CC1CCN(C(CCCCOC)=O)C1 N(C(=NCCc1ccco1)NCC1CC1)CC1(OCC)CCOC1 c1(C(=O)OC)[nH][nH]c(=NC(=O)N2CCN(CCO)C(=O)C2)c1C1CC1 C1(CNC(C2CC2C(=O)OC)=O)CCCN(C(c2nccc(COC)c2)=O)CC1 N1(C(C2N(C(CC)=O)CCCC2)=O)CCN(C(C2CC(N(C)C)C2)=O)CC1CO c12cc(ccn1)SC1C(CCCC1)N2C(NC)=O.C1(C2(c3nonc3C)CC2)CC12CC(O)C2 c1(C(N2CC(N(C(c3c(C)ccnc3)=O)C)C3(C2)CC3)=O)cc(O)cc(N)c1Cl c1(C(N2CCCC(C)(CNC(CC3CC(OC)C3)=O)C2)=O)ccc(S(C)(=O)=O)[nH]1 C1(NC(c2c(C)[nH]cc2)=O)CN(C(c2ocnc2C2CC2)=O)CC1C1CC1 N1(C(C2CN(Cc3ccc(C)s3)CC(F)C2)=O)CCc2nc[nH]c2C1 c1(-c2c(C(=O)NCc3cnc(C(C)(C)C)s3)n[nH]c2)cc([N+](=O)[O-])ccc1C#N c1(C(N2CC(NC(=O)C(F)=CCCF)CC(C)(C)C2)=O)ccc([N+](=O)[O-])c(N)n1 c1(C(=O)NCC2=NN(C)C(=O)C2)cnc2[nH]cc(C3=COCC3)c2c1 c1(C=O)cc(F)ccc1F.N12CC(C(C)(C)C1)C(C)n1cc(nn1)C1CCN21 C1(NC(CSCC)=O)CC2CCC1(NC(c1nc(C)sc1C)=O)C2 OC1COC2(CCN(Cc3ccncc3Cl)CC2)CC1O CN1C2CCC1CC(C(=O)NC1C=CCN(C(=O)Cc3cccnc3N)C1)C2 C1(C(=O)NCc2cnccn2)(CNC(C2C(C)C2C)=O)CC12CCC2 C(=O)(N=c1nc2ccc(Cl)cn2[nH]1)NCC(c1ccccc1)C c1(CC(N2CC(CC(=O)NCc3cccnc3F)OCC2)=O)cc(Br)ccc1Br c1(NCCOCC)cc(NC(c2cccs2)=O)nc(C(F)(F)F)n1 c1(NC(c2nc(NC(c3scc(C)n3)=O)sc2)=O)cnc(C)c(F)c1 CC1(C)CC(CNC(=O)C(F)C2CC2)N(C(=O)CCc2ccccn2)C1 c1(CC)cccc(OCC(=O)NCCC2CN(C(c3ncsc3C)=O)CCO2)c1 C1(NC(CCC2C(C)C2)=O)CCCC1NC(=O)C(F)F C(CCCCCNC(=O)Cn1cc(Br)cn1)N(C)C(c1ncn(C)n1)=O CCC(C)C(C)(O)CNC(C1(CNC(c2nocc2Cl)=O)CC(C)(C)C1)=O c1(NC(COC2(C)CN(C(C3CCC(C)CC3)=O)C2)=O)cccc(Cl)c1Cl N1(C(c2cnc(CC)[nH]2)=O)CCC(C)(CNC(=O)CCC2CCCCO2)C1 Cc1ccc(C)c(OCC(N2CCC(NC(C3CC=CCO3)=O)CC2C)=O)c1 c1(C(N2CC(C(C)NC(=O)CC3CCOC3)OCC2)=O)cc(C#N)ccc1N C1(CC)CC(CNC(c2ccns2)=O)N(C(C2CCCN(S(C)(=O)=O)C2)=O)C1 N1(NC2CCC2)Cc2[nH]nc(C(=O)NOCC(=O)C(C3C4CC(=O)CC43)=O)c2C1 N1(CCC)CCC(N=c2[nH]c(=NCCCSCC)[nH]c3c2CCCCCC3)CC1 C(=O)(C#CC1CCCC1)N(C)CC1N(C(C(C)C(F)F)=O)CCC1 N1(CCCCCOC(N(S(CC=C)(=O)=O)C2CC2)=O)CCN(CC)CC1 C(=O)(C1OCCc2ccccc21)NC(C(C)C)CCNC(=O)CC=C(Cl)Cl CCC(C#N)(CC)C(=O)N1CCCCC(CNC(=O)Cc2ccccc2OC)C1 CC(C)C(C#N)C(=O)N1CCCC(C(=O)NCC2CN3CCC2C3)CC1 C1(NC(CC2CC(OC)C2)=O)CC2CCCC(C1)N2C(C1(OC)CCC1)=O CCCC(C(N)=O)NC(C1CCCN1C(c1cc(C)oc1C)=O)=O C1(C)(C(=O)NCC2N(C(CC(C)C3CC3)=O)CCC2)CCCNC1=O C1(NC(=O)COCC2CCCCO2)CN(C(=O)CCC2CC2)C2(CCCCC2)C1 N1(C(c2sccc2Cl)=O)CCN(C(=O)CC2OCCO2)C(C2CC2)C1 C1(OC)CCCCN(CC(N2CCC(C(C)N(C)CCO)CC2)=O)C1=O C1(C(C)NC(C2C(CC)CCC2)=O)CN(C(c2cnc(SC)[nH]2)=O)CCO1 C1(C(=O)NC)CC2(CC2)CN1c1nccc(Oc2ccccc2)n1 c1(C(C(N2CCC(CCOC)(NC(C=CCC)=O)C2)=O)C)ccc(OC)c(F)c1 C12(C(=O)NCCN(C(COCc3n(C)ncn3)=O)C3CC3)CC=CCN1CCC2 [N-]=[N+]=NC1CN(C(c2csnn2)=O)CC1NC(c1ccc(Cl)nc1O)=O N1(C(C2(CC=C)CCCC2)=O)CCCCC1C(C)NC(c1cn(C)nc1C)=O CC1CCOC1C(=O)N(CC(C)CNC(=O)CC(=O)N(C)C)C c1(N2C(C)CC(CNC(c3cn(C(C)(C)C)nn3)=O)C2)ncnc2c1CCO2 N1(C(C(=O)N(C2CCCC2)C(C)CN2CCOCC2)=O)CC(F)(F)C1C1CC1 C#CCC(C)(CC)C(=O)NCCCC(=O)NC1CC2C=CC1C2 N1(C(C2(COC)CN(C(=O)C(N=[N+]=[N-])C(C)C)C2)=O)CC=CC12CCCC2 c1(OC)cccc(C(=O)NC2CCN(C(C3COCCO3)=O)CC2CO)c1OC CCC(CC)(CC)NC(=O)CC1CCCC(NC(=O)COCCF)C1 C1(CN(C(c2cccc(C)n2)=O)CC)CCCCN1C(c1ccc(CSC)o1)=O C1(NC(=O)C(F)OC(F)(F)F)CCCC12CN(C(c1cccs1)=O)C2 c1(C(N2C(c3nc(C)[nH]n3)COCC2)C(=O)NC2CCCC2)ncc(F)cc1Cl c1(C(N(C)C)=O)cncc(C(N2CC=CC(NC(=O)CC3CCCOC3)C2)=O)c1 c1(COCC)ccnc(C(=O)NCCCSCCO)c1.C1C(C)C(=O)N1 c1(CC(N2C(C)CC(NC(=O)C=Cc3cnc[nH]3)C2)=O)ccc2oc(O)nc2c1 n1(CC)nc(C)c([N+](=O)[O-])c1NCCC(C)(C)NC(=O)COCc1cc(C)on1 CCS(=O)(=O)c1ccc(CCCN2CCCC(C)(C)C2C=Cc2cccs2)cc1 C#CC(CC(C)C)NC(C1CCC1NC(C1(C)CCNC1=O)=O)=O C1(OC)CN(C(=O)COc2ccccc2F)CC1NC(c1ccoc1)=O c1(C(N2CC(CC)(NC(c3ccon3)=O)C2)=O)nccc2cc[nH]c12 CC(C)CCC(O)C(=O)N1CCC(C(=O)NCCCC(C)O)C(C)C1 C1(NC(=O)NC2CC3CCCC3C2)CC2C(O)C(O)CC12 C#CC(C)(C)C(=O)NCC(c1ccc(F)cc1)NC(=O)C(F)CC1CCC1 N1(C(c2n(C)ncc2)=O)CCCCCCC1C(=O)NCC1CC(O)C12CCC2 C1(C)(NC(=O)C(=O)Nc2ccc(F)cn2)CC2CCC1C2.C12(CC)CN(C1)C2 N1(C(C2CCC(NC(=O)CNC(C)=O)C2)=O)CCC(OCCOCC)C1 c1(C(=O)NCC2CN(C(C(C(C)(C)C)SC)=O)C(C)C2)nsc2ccccc12 n1(C(C(=O)NCC2(CNC(CCCC#C)=O)CC2)C)c(C)cc(O)cc1=O c1(C(C(N)=O)NC(COC(C2C(C(=O)OC)C2)=O)=O)ccc(Cl)cc1 n1(CCC)ncc(C(C(=O)NCCSC)N(C2CCC2C)C)c1C c1(NC(CC(C)NC(C23CC(C)(C2)OC3C)=O)C)ncc2c(n1)COC2 c1(C(=O)NC2CSC2)n[nH]c2c1CN(C(C1CSC1)=O)C2 Cc1cc(C(=O)NCC(=O)NCC(N2CCC=C(Cl)C2)=O)ncn1 c1(C(=O)NC(CC=C)C(=O)NC(c2cccnc2)CO)cc(F)ccc1F c1(NC(=O)NCC2C3CCOCC23)ccc(O)cc1F n1(C(C(=O)N(C(C)C(=O)O)CCC)C)cc(CCC(O)c2cccs2)nn1 n1(C(CC)C)nccc1NC(=O)NCCCSC C(=O)(CC(C)(C)C#N)NCCn1cc(C2CCCCC2Oc2cn(C)nc2)nn1 Cc1ccn(CC(=O)NCCC(C)N(C(=O)CCSC2CCCC2)C)n1 Cc1ccc2c(C(N3CC(CCNC(=O)CCC4CCCCO4)C3)=O)n[nH]c2c1 N1(C(C2N(CC)CC2)=O)CCC2(CCC2NC(C23CC(C)(C2)C3)=O)CC1 CC1C(C(=O)NCCCSCCO)CCCN1C(c1cncn1C)=O CC#CCC(C(=O)NCC(N1CCOCC1)C)NC(c1cnn(C(F)F)c1)=O c1(CN2CCC(OCCOC)C2)cccc2c1oc1ccccc21 c1(C(=O)NC(C(C)NC(c2ccc(OC)cc2)=O)C(C)C)ccnc2ccsc12 C1(C(=O)NCC(CNC(C2(OC(C)=O)CC2)=O)(C)O)CC(C)(C)CCO1 n1(CC=C)cc(CNC(C2OCCC2NC(C2CCSCC2)=O)=O)nn1 C1(CNC(C(CC)n2cncn2)=O)CCCCN(C(c2cc(C)c(C)s2)=O)C1 c1(C(=O)OC)ncc[nH]c1=NCC1C(C)CCCN1C(C1CCS(=O)(=O)N1)=O CCC(C)CCCCC(=O)NCC(C(C)(C)C)NC(=O)C(C)Cc1ccco1 C(=O)(CCCC(=O)N1CCC(C(N2CC(OC(=N)O)C2)=O)C1C(C)C)OC S(=O)(=O)(c1ccc(NCC2(CO)CCOC2)c(Br)c1)NCC1(C)CCCCCC1 C(CC(=O)N(C1(CO)CC1)C)(C(C)OC)NC(c1nn(CC)c(C)c1)=O c1(CC(N2CC(C)C(NC(C(C)C)=O)C(C)C2)=O)nn(C)c2ccccc12 C1(C(C(N2CCNCC2)C)=O)CCCN(c2ccc(Br)cc2)C1=O C1(C(N2CCC(C(F)F)(CNC(C(=O)NC(C)C)=O)C2)=O)CC2(C1)CC(F)(F)C2 C(C(=O)N1CCN(CCCCCNC(=O)CN(C)C)CC1)(C(C)C)N(CC)CC c1(CC(=O)NC2(C)CCN(C(C3N(C)CCC3)=O)C2)ccc(S(=O)(=O)N(C)C)s1 N1(C(COCCOC)=O)CCC2(NC(c3cccc(C(N)=O)c3C)=O)CCCC12 c1(CC)ccc(C(N2CCCC(C(N3CC(OC(C)=O)C3)=O)CC2)=O)cc1[N+](=O)[O-] C1(C#CC(=O)NC2CCC(C(=O)NCCCC(C)CO)C2)(CC)COC1 C1(OC)CC(CNC(=O)CC(C)(C)C2CC2)N(C(C2CC2CC(C)(C)C)=O)C1 c1(OCCC(=O)NCC(C2CCOC2)NC(C=COCC)=O)cccc(Cl)c1 c1(C(N(CCNC(C(C(C)C)CC2CCCC2)=O)C)=O)cn2c(n1)CCCC2 Cc1[nH]c(C)c(C(N2CC(NC(=O)Cc3ccc(Cl)nc3)C3CC23)=O)c1C N1(C(c2n(CC=C)ccc2)=O)CCC(C(C)C)CC1CNC(=O)C(O)CC(F)F C1(CC)CCN(C(=O)CCC2CCN(C(c3sccc3Cl)=O)C2)C1 S(=O)(=O)(c1ccc(Br)cc1Br)NC(C1CN(C(C2(C(=O)OCC)CC2)=O)CCO1)=O N1(Cc2c(Cl)ccc(OC)c2)CC2CN(C(=O)CCOC(=O)C(C)C)CC2C1 N1(C(C(C(C)C)C)=O)CC(C)(C)OCC1CNC(=O)C1=CCCC1 c1(C(N(C2CCCC(NC(=O)CC3CCCC3)C2)C)=O)csc2ccccc12 Cc1c2ccc(C(=O)NCCCn3cc(COc4ccccc4)nn3)cc2nn1C c1(CCC(=O)Nc2ccccc2COc2ccccc2)n[nH]c2c1CCCC2 N1(C(C(CCNC(C(C)SC(C)C)=O)O)=O)CCN(C)CC1CCO N1(C(c2n[nH]c(C)c2Br)=O)CC2CC1CCN2C(C1C2CC3C(C2)C13)=O c1(C(N2C3CN(C(CCCOC)=O)C(C3)C2)=O)cc2cc(Cl)cc(Cl)c2[nH]1 N1(CCC)CCC(O)(C(=O)Nc2ccc(NC)cc2)CC1 N1(C(CCN(CC)CC)=O)CC2CC(CNC(c3cncc(Cl)c3Cl)=O)C2C1 O=C1CN(C(C2CCC(C3CC3)O2)=O)C(C(=O)NCC2CCCO2)CN1 N1(C(C(CCC#C)NC(c2ccccn2)=O)=O)CCc2ncn(C)c2C1 N1(C(C2CCN(C)C2=O)=O)CCC(F)C(NC(c2ncoc2-c2ccco2)=O)C1 C1(CNC(C2C3CC4C(C3)C24)=O)CN(C(=O)CC(O)C2CCCC2)CCC1(F)F C1(C(C)O)CCC(NC(C2CCN2C(=O)CCc2ccncc2)=O)CC1 c1(NC2CC3CN(C(C(c4cccnc4)C)=O)C(C2)C3)ncc2ncn(C)c2n1 Cc1cnccc1NC(=O)CN1CCN(S(=O)(=O)C(C)C)CC1 C(CCCC(=O)NC(CNC(c1cc(C)c(SC)s1)=O)C1CC1)SC C1(Cc2c(Br)cccc2)CN(N2CC(C3CCCCC3)C2)C1 c1(C(=O)NCC(CO)NC(C(CCC)(C)C)=O)c[nH]c2cc(Cl)c(OC)cc12 N1(C(c2c(C)nc(C)o2)=O)CCC2(CC2)CC1C(N1CCC(F)(F)C(F)C1)=O N1(C(CC2CCC(C)CO2)=O)CCCC2(C1)CN(C(=O)C(C)C(C)C)C2 C1(CC(=O)NCC2CC(NC(C3(C(C)C)CC3)=O)C2(C)C)CN2CCC1CC2 C1(CNC(Cc2cc(OC)no2)=O)COCCN(C(C2CCCS(=O)(=O)C2)=O)C1 C12(C(N(CCCNC(C3(C)CC=C(C)CC3)=O)CC)=O)CCCC1CC(=O)C2 C1(Cn2cc(CCCC(C)=O)nn2)CC12CCN(C(=O)COC1CCCC1)CC2 C(=O)(C(O)CCCNC(C1CC(=O)OC1(C)C)=O)N(CCCOC)CCO C(C(F)(F)CC(=O)Nc1cccc(CCF)c1)N(C)C C1(F)(CNC(C(C)NC(C)=O)=O)CCN(C(=O)Cc2ccc(Br)cc2)C1 c1(CCC)nc(C)c(C(=O)NC2(C)CCN(C(c3cncc(C)n3)=O)C2)s1 N1(C(C(C(=C)C)(C)C)=O)CCC2(CCCC2NC(=O)C=C2CC2)CC1 C=C(C)CC(C(=O)NC1CCNC1=O)NC(=O)CCC1CCCN1C C1(C(=O)NCC2C3CCCCC23)CN(C(=O)Cc2ccc[nH]2)C2(CCC2)C1 N1(C(c2n(C)ccc2)=O)CC(CNC(c2cc3scc(Cl)c3[nH]2)=O)CC12CCC2 N1(C(CN2C(CO)CCC(C)C2)=O)CCC2(CC1)COCC(CO)O2 c1(C(=O)NCCN(C)C(C2OCCO2)=O)cc2nc[nH]c2cc1[N+](=O)[O-] c1(C(=O)NC2CCN(Cc3ccc(=O)n(C4CC4)c3)C2)cccn2c(O)nnc12 Cc1ccncc1-c1cn(CC(N2CC(C(F)(F)F)C(C(F)(F)F)C2)=O)nn1 N1(C(c2cc(SC)oc2)=O)CC2(C)CC1(C(=O)NC(C)(C)C(C)O)C2 CC1(C)C(C(=O)NC2CC(C(=O)NC3CCS(=O)CC3)CC2O)CC1(F)F C(CCCC(=O)NC1(C2CCCN2C(=O)CO)CC1)OCCC=C C(=O)(CCN=c1[nH]ccs1)N1C(CNC(c2cc(C3CC3)[nH]n2)=O)CC(OC)C1 c1(N2CCC(NC(c3ccn(C(CC)CC)n3)=O)C2)ncnc(Cl)c1C(C)=O n1(CC(=C)C)nc(-c2cncnc2)nc1Cn1nnc(C(C)(C)C)n1 C=CCC(CC)C(=O)NCC(O)C(N1CCCC(CCC)CC1)=O c1(C(=O)NC2CCCCN(C(CC(C)F)=O)C2)cnn2cccc(Cl)c12 Cc1cc(OCCC(=O)NC2CN(C(=O)COC3CC(C)CO3)C2)ccc1Br CN1CCN(C(=O)COC2CC=CC2)CC1C(=O)N(C)Cc1cccnn1 N1(C(C2C(C)(C)C2)=O)CCCC(C)(C)C1CNC(c1sccc1CC#N)=O c1(C2N3CCCC(C)(C3)NC2=O)cnc2ccnn2c1.CCC(C)(C)OC.C(C)(C)N N1(C(CNS(NC)(=O)=O)=O)CC(NC(c2ccsc2)=O)CC12CCCC2 C1(C(N2CCN(C(C(CC)n3cncn3)=O)CC2CF)=O)CC2(C1)CC1(CC1)C2 c1(NC(C2C3CN(C(C(N4CCCC4=O)C)=O)CC32)=O)cc(O)ccc1F N1(C(C2CC(C(=O)OCC)C2)=O)CCCC2(CCC2)C1C N1(C(C2C(C)CC(=O)N2)=O)CCN(C(=O)CCOCC(F)F)C2(CCC2)C1 c1(CC)nc(C)c(C(N2CCC(NC(=O)C(C3CCCO3)C3CC3)C2)=O)o1 n1(CCNC(C2(C(C)C)COC2)=O)cc(C(=O)NC(CO)CCO)nn1 C1(NC(=O)NC2CC3OC2C2CC32)CCC(=O)N(CC(F)(F)F)C1 CCCC(C(c1nnnn1CCC1(C)CC1)NCC1(COC)CCC1)OC N1(C(C(CN(C)C)NC(Cc2c(C)cccn2)=O)=O)CCC(C)(O)C(O)C1 c1(OC)cc(C(=O)NC2CCCCC2C(=O)Nc2nnc(C3CC3)o2)cc(O)c1O C1(C)(CC)CC(NC(=O)CCSC(C)C)CN1C(=O)CCN(C)CC C(=O)(C1CCCc2ccnn21)NCC(CNC(=O)C(C)(C)OC)OC c1(OC)ccc(C(=O)NC2C3CC2N(C(C2CC(C)=NO2)=O)C3)c(F)c1F C(=O)(CCCCCC(C)(C)C)NC(CCNC(C(C)C(F)F)=O)Cc1ccccc1 c1(C(=O)NC2C(C(C)C)N(C(c3cc(C(F)F)[nH]n3)=O)CC2)cn2ccsc2n1 Cc1[nH]cc(C(=O)NCC(C)CNC(=O)C(C)(C)C(C)O)c(=O)c1Br C1(NC(c2c(C)nn(C3CC3)c2)=O)CCC2CCN(C(C3CC3F)=O)C12 Cc1cncc(C(=O)NC2CCC2CNC(c2sccc2C(F)F)=O)n1 c1(C(=O)NCC(C2CCC2)NC(CC(C)C)=O)cccc2nsnc12 CC1CN(C(c2ccc3nonc3c2)=O)CC(C)C1NC(c1nncs1)=O c1(CNC(CCSC(C)C)=O)cn(C2CN(C(C3CC(=C(C)C)C3)=O)C2)nn1 C1(C(N2CCC(CC#C)C2)=O)CC(NC(=O)COCCCCC)C(O)C1 N1(C(c2c(C)oc(C(C)C)c2)=O)CC2CCC1C1CN(c3ncc(O)cn3)CC21 C(C(C)(C)CCC#N)(c1nnnn1C(C)C(=O)OC)NC(CC=C)CC C1(C(=O)NC(CC)CNC(=O)C=CSC)(Cc2ccc(F)cc2)CCCCC1 N1(C(c2cc(C)[nH]c2)=O)C2CCC1C(C)C(NC(c1occc1Br)=O)C2 c1(OC)c(C(N2CCCC(CN(C)C(C3(CCF)CC3)=O)C2)=O)cnn1C CCCCN=C(NCc1cn(C)nc1CC)NCC1CCC(C)(C)O1 C=Cn1nccc1C(=O)NC1C=CCC(C(=O)NC(C2CCCC2)CC)C1 N1(C(c2cc(C)[nH]c2C)=O)CC(C)N(C(c2cc3c(ncn3C)[nH]2)=O)CC1C N1(C(C(CC(C)C)ONC(c2ccc(F)s2)=O)=O)CCC2CN(C)CC12 N1(C(c2c(COC)cco2)=O)CC(NC(=O)CCC2CCC(=O)N2)CC(F)C1 CCCC#CC(C)(C)NC(C1CC(C(=O)NCC2(C)CCC(=O)NC2)C1)=O C1(C(=O)NCc2ncc(C)o2)CNC(=O)CN1C(=O)C=CC(C)C C1(C)(C(=O)NCC#CCNC(COCc2ccc(C)cc2)=O)CC(C)OC(C)C1 c1(OCCC)cc[nH]c(=NCCCC(C)NC(=O)Cc2ccsc2)n1 c1(SC(C2(C)CCCS2)=O)ccc(Cc2nc(C)on2)cc1 N1(C(C(C)(C2CC2)OC)=O)CC2CCC1C(CNC(=O)C=C(C)C(C)C)C2 c1(C(N(C(C)C)CCN(C)C(=O)C2CC2)=O)csc(CS(C)=O)n1 S(=O)(=O)(C1CCN(C(=O)Nc2ccco2)C1)NC(CN(C(C)C)C)C C12(CC(=O)NCC(CNC(Cn3ccc(C)n3)=O)C)COC(C)(C1)C2 c1(CC)cc(C(=O)NC2CCC(NC(=O)C(C)(C)n3cnnn3)CC2)cc(O)n1 CCC(C)(CNC(=O)CCCCNC(=O)CCCc1ncco1)C(C)O C(=O)(C1=CC2CCCCCC12)NCC1(CNC(c2c(C)cc[nH]c2=N)=O)CCC1 C1(C(N(CC(O)CF)C)=O)C2CC(O)C(C2)N1C(=O)CC(C)(C)C C(=O)(CCCCC(N)=O)NCC1C(C)CN(C(C2(F)CC2c2ccccc2)=O)C1 CCCCCC(C)C(=O)NC1CC(C)CN(C(c2cccn2C)=O)C1 c1(C(=O)NC2(CO)CCCN(C(c3n[nH]c(O)n3)=O)C2)nc(Br)n2c1CCC2 C(=O)(N=c1cc[nH]c(C)c1F)C1CC(NC(C=Cc2ccc(C)cc2)=O)C1 C(=O)(CCC(C)(C)C#N)N1CCC(CCOC)CC1C C1(CCC)CN(C(c2ccc(C(C)C)o2)=O)CC1C(N1CC2(CCC2)C1)=O C1(CC(=O)NC2(CNC(C(CC=C)C)=O)CCOCC2)CCOC(C)(C)C1 c1(COC)cc(C(=O)NCCC(CNC(=O)CC(C)NC(N)=O)OC)no1 CC1(C)OCC(C(=O)NCC2(C)CCN(C(=O)CCSC(F)(F)F)C2)O1 c1(-c2ccc(COC)s2)cn2cc(C(=O)NCc3ccno3)ccc2n1 C(=O)(C(O)CCCCC)NCC(CC=C)C(=O)N1CCOC(C(=O)NC)C1 C(=O)(C#CC1CCOCC1)N1CC(C2CN(C(=O)Cc3ncccc3F)C2)C1 C1(CC(=O)N(C(C)CNC(c2sccc2Br)=O)CC)CCCN(C)C1 N1(C(c2c(NC)ccc(F)c2)=O)CCC2(CCC2NC(C2(F)CCCC2)=O)CC1 c1(C(N2CCC(F)(CNC(=O)CC3=CCCC3)C2)=O)cc2c(O)cccc2[nH]1 C1(C)(CC(=O)N(CC)CC)CN(C(c2cc(C)[nH]n2)=O)C1 S(=O)(=O)(c1cn(C)c2c(Br)cccc12)N(c1ccc(Br)c(C(F)(F)F)c1)C N1(C(c2cc(C)c(O)nn2)=O)CCN(C(c2cccc(CO)c2)=O)C2CCC12 C1(C(N2CC(C#C)(N(C)C)C2)=O)CN(C(=O)CNC(c2cc[nH]n2)=O)CC12CC2 C(=O)(C(CC(C)C)N(C)C)N1C(C(N(C)Cc2onc(C)n2)=O)C(C)CC1 C(=O)(CCC(C)(C)F)N1C(CO)CC(NC(c2c(C)n(C)cn2)=O)C1 N1(C(c2cn(CC(=O)OC)nc2)=O)CC(NC(=O)Cc2ccc(O)cc2)C(C)C1 c1(NC(c2ccc(C3CC3)c(C)c2)c2n(CC=C)nnn2)ccc2c(c1)COC2 c1(C(=O)NC(CNC(=O)C(O)C2CCC2)C2(CO)CC2)ccc2c(c1)C(=O)OC2 CCC(CC(C)CO)NC(c1n[nH]cc1CNC(c1ccc(OC)nc1)=O)=O c1(C(N2C(COC)CN(C(=O)Cc3cncs3)CC2)=O)cnc2sccc2c1 C#CCC(C)(C)C(=O)NC1C=CCC(C(=O)NCc2cc(C)[nH]n2)C1 C1(C2CCCO2)(C(=O)NCC(CNC(c2c(C)snc2)=O)(C)O)CCOCC1 Cc1cc(CC(=O)NC2CN(C(c3cnn(C)c3)=O)CCC2C)cc(F)c1 CCCCCC(O)C(=O)NC(C(=O)NCCc1cnco1)C1CCC1 c1(C(C(=O)NCC23CC(NC(C(C)=CC4CC4)=O)(C2)C3)O)cc(F)c(F)cc1F N1(C(c2ccc3ccoc3c2)=O)CCC2CCC(C1)N2C(c1snc(O)c1Cl)=O CCC(C)CC(=O)NC(Cn1cccn1)C(=O)N1CC=CC1CN(C)C Cc1nc(N(CCCOCCCO)C)cc(NCCCC2CCC2)n1 N1(C(C(CCO)N(C)C)=O)CCC2C(CCN2C(c2ccnn3ccnc23)=O)C1 N1(c2nccc(SC)n2)CCC2(CC(NC(c3cc(-c4cccs4)on3)=O)C2)C1 N1(C(CCC(=C)C)=O)CC(C)CCC1CNC(c1ccn(C(C)C)c(=O)c1)=O N1(C(c2c(C)n(C(C)C)nc2)=O)CCCN(C(=O)C(C)Oc2ccccc2)CC1 c1(C(N(CC(CC)NC(=O)C(O)CN2CCCC2)C)=O)cccc2nonc12 C(CCN=C(NCc1ccc(Cl)nc1)NCC1CC2CCC1O2)OCC N(C(=NC(C)C)N1CCC(O)C(C2CCCC2)C1)Cc1ccc(C)c(Br)c1 C1(COC)(CO)CCN(C(c2cc(C3CCC3)on2)C(=O)NC2(C)CC2)C1 C1(C(=O)NCCOCCN(C(=O)CS(C)(=O)=O)C)CC(O)C(O)C1 C(c1c(Cl)cccc1Cl)=C(C)C(N1CCC(F)(CNC(C2(C)CCCS2)=O)C1)=O N1(C(c2ccn(C)c(=O)c2)=O)CCC2CN(C(C3(C4CCC4)CC3)=O)CC2CC1 N1(C(COCCCC(C)C)=O)CC(C)(C)OCC1CNC(C1CC1C)=O c1(C(=O)OCC)c(-c2ccc(C(C)CC)cc2)cnn1C C(=O)(C(CNC(c1n[nH]c2c1COC2)=O)C(C)(C)C)NC(C#C)C1CC1 C1(CNC(c2cc(O)ncc2F)=O)CCN(C(=O)C=C2CCC2)C12CC2 c1(C(=O)NCC2CCN(C(C(n3cc(Cl)cn3)C)=O)C2)cc[nH]c(=N)c1Cl N1(Cc2cncc(C)n2)CCC(F)(F)C(C(N2CC(O)CC2CO)=O)C1 c1(NC(c2c(CNC(c3ncc(CC)cn3)=O)ccs2)=O)ccc(Cl)cc1C c1(CNC(CC(C(C)C)OCC)=O)nc2c(s1)CN(C(=O)C(O)CC)CC2 N1(C(c2cccc(C)c2F)=O)CCc2sc(CNC(C3CCCN3C)=O)nc2C1 c1(CN=C(NC2C(C)C2)NCc2ncc(Cl)s2)cccc([N+](=O)[O-])c1C Cc1cccn2cc(C(=O)NC(CNC(=O)CCCn3cccn3)C3CC3)nc12 CC(C)CC(O)C(=O)NC1CCC(N(C)C(c2cc(Cl)c(Cl)[nH]2)=O)CC1 c1(C(C)=O)cc(C(=O)NCC=CCNC(=O)CCCOc2ccccc2)co1 N1(C(c2cn(C)[nH]c2=N)=O)CCC(CNC(c2ccc(F)cn2)=O)C12CCC2 C1(F)(NC(=O)NC)CC(C(=O)NC2CC2)C1.C(=O)(C(=O)NC1CC1CF)N N1(C(CC2CC(=O)NCC2)=O)CC2(CCC(NC(=O)CCc3ncc[nH]3)CC2)C1 c1(OC)ccc2cnc(Nc3cc(-c4cnn(CC(C)(F)F)c4)ccn3)nc2c1 C1(OCCC)CCCN(c2nnc(C3CCOC3)n2Cc2csc(CC)n2)C1 C(=O)(C1=CC(C)(C)C1)NC1C(CC(N2CC=CC(OC)C2)=O)C(O)C1 C1(C(=O)NC2CN(C(c3cc(C4CCC4)[nH]n3)=O)CC2C)(OC)CCCSC1 N1(C(CCC2(NC(c3nccc(OC)c3)=O)CCCC2)=O)CCCC(CO)CC1 C(=O)(CCN(OC)C(=O)C1(C)CC1)NC(C=C)COC Cc1ccn(C(C)C(=O)N(C(c2ccccc2)CNC(C2(C)CC2)=O)C)n1 C1(N(C(=O)C(C)OC(C)(C)C)CC(=O)NCCOC)CCC2(CCC2)C1 C1(C(C)(O)CNCc2ccncc2F)CCN(C(=O)OC(C)(C)C)CC1 C#Cc1ccc(C(=O)NCCCCC(CO)NC(=O)C(C)OCC)nc1 C1(Nc2nccc(CC(=O)OC)n2)CS(=O)(=O)CC1NC(c1c(C)coc1C)=O C(C(C)C(C)(C)C)NC(C1CC(NC(C(c2cc(OC)no2)N(C)CC)=O)C1)=O C1(C)(COC)CCN(C(=NCC2CCOC2)NCc2cccc(OC)n2)C1 C(=O)(CCP(C)(C)=O)NCC(CNC(c1snnc1C1CC1)=O)OC C(CC(C)C)(C(=O)NCCC(C)NC(c1cc(C)c(CO)cn1)=O)OC C(=O)(C1=NOC2COCC12)N1C2CCC(CNC(C3C(=O)NCCC3)=O)(CC2)C1 c1(C(=O)NC2C(NC(C(c3cccs3)SC)=O)C2)nn(C)c2c1CCCC2 c1(C(=O)NC2C(n3cc(-c4ccc(C(=O)OC)s4)nn3)COC2)cc(Cl)c(Br)s1 C#Cc1cn(C)nc1C(=O)NC1CCC(C)(CNC(c2ccnc(Cl)c2O)=O)C1 C1(C(=O)NC2CCC(NC(c3cc(C)c(C)o3)=O)C2)CC2(CCCCC2)S1(=O)=O C(=O)(C(O)CCCNC(C1CCCCC(=O)N1)=O)N(CCNC(C)=O)C C1(CNC(c2cc(CC)[nH]n2)=O)CCCCCN1C(=O)Cc1cc(C)cc(F)c1 C1(C(=O)NC2CC(C#N)(OC)C2)CCN(C(=O)CC(O)C2CCCC2)C(C)C1 c1(NC(C2CN(Cc3c(C)cccc3O)CC(F)C2)=O)cccn2cncc12 CCS(=O)CC(=O)NCC(C1CCN(C(c2ccnn2CC(F)(F)F)=O)CC1)C CN1CCC(CC(N2CC(NC=O)C(NC(=O)CC3CC3)C2)=O)CC1 Cc1ccsc1CN.C1(C(N2C3C(C3)C(=O)N2)=O)CCCN1Cc1ccccc1 c1(OC)c(C)cc(C(N2CCCC2C2CCCCN2C(=O)C(Cl)=CCl)=O)cc1C n1(CCOCC=C)c(N2CCC(C(=O)NC)C2)nnc1-c1sc(C2CC2)nc1C C1(N(C(=O)C(O)C(F)F)C)CC2CCC(C1)N2C(c1ccc[nH]1)=O N1(c2cc(N(C)Cc3ncc(Br)s3)nc(C(F)(F)F)n2)CCn2cnnc2C1 C1(CNC(CCC=C(C)C)=O)C(C)CCCN1C(c1ccn(CCO)c(=O)c1)=O c1(C(=O)NC23CCCC2N(C(C2SCCS2)=O)CC3)coc2c1C(=O)NCCC2 C(C(C)CC(=O)NCc1cn(C2CC2)cn1)NC(c1c(CC)ncs1)=O c1(CC)ncc(C(=O)NC2CN(c3ccc(=O)n(C)n3)C2)c(C)n1 CN1CCN(C(C2CCCCNC2=O)=O)CC1C(=O)NC1(CN(C)C)CCCCC1 CC1(C)CCC(CCNC(N2CCC(NC(c3ccc(Cl)cc3)=O)CC2)=O)O1 c1(OCC)c(C(=O)NC2CCOC(CNC(=O)Cc3cnns3)C2)cccc1F C1(NC(c2cc3ccc(O)nc3s2)=O)CN(C(=O)CC=C(Cl)Cl)C2(CCOC2)C1 c1(CC)ccc(C)c(F)c1F.n12nnnc1C(CCC1CCCOC1)NC21CC1 C(=O)(CCCC(=O)NC1CN(C(C2CC(O)CN2C(N)=O)=O)CC1O)NCC CCC(CCC(=O)NC1CCCC1CN=[N+]=[N-])NC(C1(C#N)CC1(C)C)=O c1(C(N2CC(NC(CCCOC(C)C)=O)C(F)CC2)=O)cc2n(n1)CCCN2 C=CCCC(C)(C)C(=O)N(C(C)C(=O)NCC1(CO)CCOC1)C1CC1 C1(C(N2CCN(C(C3CCC(F)(F)C3)=O)C(C3CC3)C2)=O)CCC2(CCC2)CC1 C(=O)(C1=NOC(CNC(C2(O)CCCCC2)=O)C1)N1C(C)(CCO)CC1 C12(C(=O)NCCSC(C)CO)CC(NC(c3ccnnc3)=O)(C1)C2 C1(N(c2ccc(C)c(O)c2)C(c2ccc(O)nn2)=O)CCCC12CCNCC2 C1(C(=O)NC2CC3(CC(NC(C(CC)OC)=O)C3)C2)CC2C=CCC(C1)C2 C#CC(CO)(CO)NC(=O)C(C1CN(C(=O)CC2COCC(C)O2)C1)SC c1(C(=O)NC2(C)CCC(NC(C3(O)CC3)=O)CC2)cc2cccc([N+](=O)[O-])c2[nH]1 N12CCC3(CC3C1)C2=O.c1(N2CCN(CC(=O)NC)CC2)cc(C)ccc1F CC1CCCN(C(=O)CC2(NC(=O)C=CC3CC3)CCCCC2)C1C N1(C(=O)NC(c2ccncc2)CC)CCc2c(C)cc(C)cc2C1 CC1(C)CC(c2ccccc2)N(CC2=C(C(F)F)CC[SH]2C=O)C1.C1(Br)CC1 CC1(C)CCN(C(C2CC(=O)C23CCCC3)=O)CC1.C(C)(C)(C)O N1(C(C(CC(C)C)OC)=O)CCC(NC(=O)CCC(C)(F)F)C12CCC2 c1(CC(=O)NC(c2ccco2)CC)c(C)nn(C(F)F)c1C Cc1nnc2n1CCCC2C(=O)NCCCNC(C1CC(C2CC2)=NO1)=O N1(C(C(CC(CC)C)NC(=O)C=Cc2ccccc2)=O)CCC2CN(C)CC2C1 C1(CNC(=O)CC2CCSC2)(NC(c2ccc(F)s2)=O)CCC(F)(F)CC1 C1(C(=O)NCC2(F)CN(C(C3C(C(C)(F)F)C3)=O)C2)CCCC2CCCN12 C1(CC(=O)OCC)CCN(N2CCC(C(c3cccs3)=O)CC2)CC1 N1(C(C2CCC(=C)CC2)=O)CC(NC(=O)Cn2nc(C)c(Cl)c2C)CC(C)(C)C1 C1(CNC(c2scc(C(C)=O)c2)=O)(NC(=O)C(O)Cc2cnc[nH]2)CCCCC1 c1(C(N2CCCC(C)(O)C2)=O)cc(O)nc2c1CN(C(C1C=CCS1)=O)CC2 O=C1NC(=O)C(CC(N2CC3CC2C3CNC(=O)C(F)n2cccn2)=O)N1 CC1(N)CCC(CNc2ccc(Cl)cc2)CC1.c12ccoc1C(=O)NC2 N1(CC(=O)N(CCC)C(C2CC(=C3CCC3)C2)=O)CC=CCC12CCCCC2 N1(C(=O)NCC2(n3cnnn3)CCOCC2)CCc2cc(O)nnc2C1 c1(CC(=O)NCC=C)ccc2n[nH]cc2c1.N12CCC(CC1)C2 C(=O)(C(C)CC(F)(F)F)N1CCC(C(=O)NC2CC3CCC2C3)(COC)C1 C1(C(=O)OC)CC(n2cc(-c3cncc(F)c3)nn2)CN1Cn1cccc1C=O CC1CCN(C(=O)Cc2cc(C3CC3)no2)CC1N(C(=O)CCc1nccs1)C C(=O)(C(C)P(C)(C)=O)NCCC(C)N(C)C(c1ccc(CCN(C)C)cc1)=O C1(NC(C(N2C(Cn3c(=O)cc(C)nc3)CCC2)=O)=O)CCC2(CCNCC2)O1 c1(OC(CC(COC)C)=O)ccc2nc(Br)sc2c1 C(=O)(C(CO)C(C)(C)C)NCCC(CCNC(c1nc(C)oc1)=O)C C1(NC(c2ccc(CC)[nH]2)=O)CCCCCN(C(C)=O)C1 c1(CCC(=O)NC(C(C)NC(c2ccc(C(C)=O)o2)=O)C)nnc(S)nc1O N1(C(CNC=O)=O)CC2(CNC(c3c(C)csc3Cl)=O)CC1C2.C=CCO C=C=C(C)CC(=O)NC(C)C(C(C)C)NC(c1ccnc(C)c1)=O Cc1cc(F)cnc1C(=O)NC(C1CCCC1)CNC(=O)CN1CCCCC1=O c1(C(=O)NCC2(C)CCCN(C(C3(C(F)F)CCC3)=O)C2)cc(Cl)c(O)c(Cl)c1 N1(C(C2N(C(c3cc(C)sc3N)=O)CC2)=O)Cc2nncn2C(C)C1 C1(CCNC(C=CC)=O)(NC(=O)CC2CC(C)=NO2)CCCC1 Cc1ccc(C(CN(C(=O)CCNC(N)=O)C)NC(C2CC2C)=O)cc1 C(CC)(CC(=O)NCc1cnc(C)n1CC)NC(CCC#C)=O c1(C(N2CCN(C(CC3CC(=C)C3)=O)CC2CC)=O)ncn2ccccc12 C1(CC=C)(NC(N2CCCC2C2CCOC(C)C2)=O)CCCCC1 c1(C(C)C)cc(C(=O)NCCC2(O)CN(C(=O)C(C#N)C3CC3)C2)c(C2CC2)o1 N1(C(c2[nH]nc(OC)c2Cl)=O)CC(NC(c2cnc(O)c(OC)c2)=O)CC(O)C1 c1(OC)ccc(F)c(NC2CC(C)N(C(=O)OC(C)(C)C)C2)c1 C1(NC(C(C)(C)C)=O)CN(Cc2ccccc2C(C)(C)C)CC1(F)F C1(C)(CC)CCCC1NC(C1C2CCN(C(=O)Cn3cccc3)CC12)=O C1(C(C)C)CN(C(c2ccoc2)=O)CCCN1C(c1cccc(SC(F)(F)F)c1)=O C1(C(=O)NCCOC2CCCN(C(=O)C=C3CCC3)C2)CC2(CCC2O)C1 C1(CNC(C(CC)=CC)=O)COC(C(F)(F)F)CN1C(c1cocc1C)=O c1(NC(C(C)C)CNC(=O)C(C)N2CCC2)nc(C#N)c(Cl)s1 O=C(C1=COCCC1)NC1(CNC(=O)C(C2CC2)C2CC2)CC2CCC1C2 C(=O)(C(C#N)C(C)C)NCC1(NC(C(CC)O)=O)CC(C)(C)C1 c1(CC(N2CCCCC(N(C)C(C3CCC3(C)C)=O)C2)=O)csc2ccccc12 N1(C(c2c(F)cc(OC)nc2)=O)CCCCCC(NC(=O)CC2(C)OCCO2)C1 c1(SCC(N2C3CCC2CC3)=O)cccc(C(=O)NOCc2nc[nH]n2)n1 N1(C(C2CCC(C)O2)=O)CC2CCC1CN2C(=O)CNC=O N1(CC(=O)N(CC(C)NC(C(C=C=C)C)=O)CC)C(=O)c2cccnc2C1=O N1(C(c2cc(OC)no2)=O)CC(CNC(c2cc(C3CC3)no2)=O)C(C)C1 C1(CC(=O)NC2(C#C)CC2)CCCN1C(c1ncccn1)=O CCCCCC(C)CC(=O)NCc1ocnc1-c1cn(-c2ccc(C)c(F)c2)nn1 c1(-c2c(NCc3c(OC)c(Cl)sc3)cccc2)ccc(CN2CCCC2)cc1F Cc1cnn2ccc(C(N3CC(O)(CNC(C4(C#N)CCSCC4)=O)C3)=O)nc12 C1(NC(c2c(C)ncc(Cl)c2)=O)COC2(C1)CN(C(=O)Cn1ncnn1)C2 Cn1cc2ccc(C(=O)NCC3(F)CC(NC(=O)C=CC4CCCC4)C3)cc2n1 C(=O)(C(CN(C)C)CC)NC(C(=O)NCC(CCC)O)C1CC1 N1(C(CC(C)(C)OC)=O)CCC(NC(c2cnc3n2CCCC3)=O)C(C)(C)C1 C12(CNC(C3N(C)CCC3)=O)CCCCC1N(c1ccc(S(C)(=O)=O)cn1)CC2 N1(C(C(CCCNC(=O)CCC2CC2)O)=O)CCC(O)(C2CC2)CC1 C#Cc1cn(C)nc1C(N1CCN(C(=O)C(C)(C)C)CC1c1nccn1C)=O C1(C(=O)NCC2C3CN(C(C(C4CCOC4)OC)=O)CC32)CCCCC12CCC2 C#CCC(C)C(=O)NCC1CCCN(CC2CCC2)C1 N1(C(c2cc3cccc(Cl)c3[nH]2)=O)CCCC(C2CN(Cc3ncc[nH]3)C2)C1 c1(C(=O)NC(C(=O)OC)C2CCOC2)cccc(C2(N)CC2)c1 CCC(O)C(C)C(=O)NCC1(C(C)(C)C)CCN(C(=O)CC(C)(C)C)C1 N1(C(C(C)N(C(C)=O)C)=O)CCCCC1c1n[nH]cc1NC(n1cc(CO)nn1)C Cn1c([N+](=O)[O-])cnc1C(=O)NCC1CN(C(=O)C(C)(C)c2ccno2)CCO1 C(CC(C)C(=O)NCC=CCC(=O)NCC1(C)CCCC1)OC N1(C(C(c2ccccc2)N(C)C)=O)CC(C2CN(C(c3cccc(=O)o3)=O)C2)C1 C(CN=c1[nH]c2c(c(=NCCF)[nH]1)SCC2)N1C(CC)CCC1 c1(C(=O)NC(C)CC2CN(C(c3nccnc3N)=O)C2)ccc(F)cc1Cl C(C)(CCI)(c1nnnn1C1CCCCC1)NCC=CCSC c1(C(=O)NCC(CC(C)C)NC(=O)C(C)C(F)(F)F)ccc(C(C)C)nc1O N1(C(C2(NC(C)=O)CCCC2)=O)C2CCC1CN(C(=O)CN(C)C(C)C)CC2 C(=O)(C1=CCC(NC(=O)CCS(C)(=O)=O)C1)NCC1C(C)C1C C1(C(C)(C)C)CCCN1C(=O)Cc1nc[nH]n1.c12cnn(c1)CC(=O)N2 CC1(C)COC(C(=O)NC2CC(C)(NC(=O)CCOCC(F)(F)F)C2)C1 c1(C(C)C)cc(C(=O)NC(CN(C)C(C2CCOC2)=O)Cc2ccccc2)n[nH]1 C1(CC(F)F)C(=O)Nc2sccc2C(=O)N1C.C1(CO)(CO)CCN(C)C1 N1(C(Cc2cn(CC)nn2)=O)CCCCC1CCNC(C1(C)CNC(=O)C1)=O C1(NC(c2c(CCC)n[nH]c2)=O)CCC(C2CC2)C1.C12CCC(CC1)C(=O)NC2 Cn1cnc(C#N)c1C(N1CC2CC1C2CNC(=O)CC1CC(C)(C)CO1)=O c1(CN2CCCC(C(=O)NCC3CCC4CCC34)CC2)cn2c(n1)CCCC2 C(C(C(=O)N1CC(C#N)C1)C(C)(C)C)NC(c1c(C)cncc1C)=O N1(C(CN(C(C)=O)C)=O)Cc2ccccc2C(NC(=O)Cc2cnoc2)C1 N1(C(C=CCN(C)CC)=O)CC2CCN(C(c3ccc(Br)c(Cl)c3)=O)C2C1 c1(CC)csc(NC(=O)NC2CC(NC(=O)OCc3ccccc3)C2)n1 c1(C(=O)NC(C)Cn2cc(CC3CCOC3)nn2)ccc2c(c1)OC(C)(C)OC2 CC1CN(C(=O)C(F)(F)c2cnnn2C)CC1NC(c1nc(C(F)(F)F)cs1)=O C1(C(N(CCCO)C)=O)C2CC3C(C2NC(=O)CC2CCC2)C13 CCCC(CNC(=O)CC(C)SC)C(=O)NC1CCCCC1CO CCC(C)(C#N)C(=O)N(CCCNC(=O)CCN1CCCCC1=O)C1CC1 CC1(C)CN(C2(c3ccccc3)CCC2)CC1NC(=O)NC1CC1OC(C)(C)C C(=O)(C1Cc2ccccc21)NCCCN(C(CC(CC)OC)=O)CCO C1(CNC(CSC)=O)CC2(C1)CN(C(=O)CC1CCCC(F)(F)C1)C2 C1(C(N(CCNC(=O)Cc2ccco2)CC)=O)CC(=O)N(C)C1c1ccccc1 c1(CC(=O)OC)ccc2c(CC(N3CCCC(C)C3CCO)=O)n[nH]c2c1 c1(CS(N2CC(C(c3ccc(F)cc3)=O)OCC2)(=O)=O)ccc(F)cc1F C1(CNC(c2c(SC)scc2)=O)CCN(C(=O)C(C)n2cncn2)CC1C C(C1CCC(C)CC1)=C(C)C(=O)N(CC(C)NC(c1cc(Br)ccc1C)=O)C c1(N(C)C)cnccc1C(N1CCC(NC(c2cnns2)=O)C1C1CC1)=O N1(CC(C)NC(=O)C=CC2CCC2)CCN(C(=O)CCC2CCC(C)O2)CC1 N1(CC(=O)N(c2cccc(F)c2Cl)C)CC2COCC2(CO)C1 CC(c1ccsc1)=CC(N1CCCC1CNC(=O)CC(O)C1CCCC1)=O N1(C(C2(C(C)(F)F)CC2)=O)CC2CC(NC(=O)Cc3cnccn3)C2C1 C1(O)(CNC(C2C=CCN(C(CN(C)CC)=O)C2)=O)CCC(C)(C)C1 C1(C(=O)NCC2CN(C(CC3N(C(C)C)CCC3)=O)C2)CCn2nccc2C1 N#Cc1ccccc1C(N1CCCOC(CNC(=O)CC(F)F)C1)=O C12(C(=O)NCC(CO)NC(=O)C(F)(F)c3ccccn3)C3CCC(CC13)C2(F)F c1(C(=O)NCC(=C)CCNC(=O)C2=CSCS2)nc(C2CC2)ncc1Cl CC1=C(C(=O)N2CC3C(CC(=O)N(C(C)CC(C)C)C)C3C2)CCCO1 CC(C)P(=O)(CC(=O)N1CCC(O)(CNC(c2coc3c2COC3)=O)C1)C(C)C C1(C(=O)NC(C(N2CC(C)(C(N)=O)C2)=O)(C)C)CCCCC1F C1(NC(c2c(C)csc2)=O)CN(Cc2c(Br)cnn2C)CC1F C1(F)(C(=O)NC2CN(C(c3c(C(C)C)ncs3)=O)CC2C)CCC(=O)CC1 N1(C(C2C(C)(NC(=O)CCC(N)=O)CCCC2)=O)C2CCC1CC(O)C2 N1(C(C(C(C)CNC(=O)CCc2cnn[nH]2)F)=O)Cc2cnn(C)c2C1 Cc1cc(C(=O)NC(C)CCNC(c2ccc(OC(F)F)cc2)=O)c(N)cc1F C=CCCCC(=O)N1CCCC(C(C)(C)C(=O)NCCC2(CSC)CC2)C1 C1(CNC(c2cc(C)oc2)=O)CN(C(C2(P(C)(C)=O)CC2)=O)CC1(C)C C1(O)(CCNC(C2CC(=C)C2)=O)CCCN(C(=O)C(C)C(C)(F)F)C1 N1(C(C(=O)NC)CCCC2CCCO2)CCc2c(F)ccc(C(=O)OC)c2C1 N1(C(CCc2c(C)cncc2)=O)CCCC12CCN(C(C1CCN(C)C1)=O)C2 C(CC(N)C(=O)NC1CCC(c2nn[nH]n2)C1)OC C1(NC(CNC(=O)OC)=O)CCC2CN(C(=O)C3=CCCCCC3)CC2C1 N1(C(C2C(C)CC(=O)N2)=O)CCCC2(C1)CN(C(=O)CSC(F)F)C2 Cc1c(C(=O)NCC2CC(C)N(C(=O)CC3CCS(=O)(=O)C3)C2)sc2cncn12 c1(C(=O)NC2CC(CNC(C3N=C(C)SC3)=O)C2)c(C)nn2ccccc12 C#Cc1cn(C)nc1C(=O)NC1CC(CNC(=O)CN2CCC(O)CC2)C1 C#Cc1ccc(C(=O)NC(C2CC=CCC2)C(N2CC(OC)CC(C)C2)=O)cc1 CN1CC2C(C(=O)NC(CNC(c3cnn(CCC(F)(F)F)c3)=O)CO)C2C1 c1(OC)cccc(C)c1C(N1CC(NC(c2scnc2Cl)=O)CC(O)C1)=O c1(CN2CC(C(=O)NCCOc3c(C)cccc3)SCC2)cccc(C#N)c1 c1(C(=O)NCC2(NC(C(C)NC(N)=O)=O)CCCCC2)ccc2nccn2n1 c1(C(=O)NCC2(F)CC(CNC(C=CC)=O)C2)ccc2oc(=N)[nH]c2c1 C1(C)(CC)C=C(C(=O)N2CC(O)(CN(C)C(c3ncc(N)cc3Cl)=O)C2)C1 c1(CCNC(=O)CCC2CCN(C(=O)Cn3cnnc3)C2)ccncc1F O=C1NCCc2c(C(=O)NC3CCCC(CNC(C4(O)CCC4)=O)C3)cncc21 C12(NC(c3ccc(OCCF)cc3)=O)CCCC1N(C(C1CC(O)C1)=O)CC2 C(=O)(C#CC1(C)CCCO1)N1CCCC(CNC(C(C(C)C)NC=O)=O)(CO)C1 C=CCC(CNC(C1(CSC)CCC1)=O)C(=O)NCC(O)C(C)C c1(C(=O)NC2CC(CCNC(COC(CC)(C)C)=O)C2)cc2ncccn2n1 N1(C(C=CC(C)(C)SC)=O)CC(C(N2CCCC2C(O)CO)=O)CC(C)(C)C1 c1(-c2nnc(C)o2)ccc(C2CC2)cc1.C12CCCN(C1)c1nc(no1)NC2 C(CCC(C(=O)NCC(F)F)N(C1CC1)Cc1n(CC)ccn1)OCC C12CCCN1C(=S)NCC2.c1(OCC#C)ccccc1 C1(NC(COCCC=C)=O)C=CCN(C(C23COC(COCC)(C2)C3)=O)C1 CS(=O)c1nc(NC2CCCCN2CCNC(=O)OC(C)(C)C)ncc1C#N C1(O)(C(C)NC(=O)COCC2CCOC2)CN(C(c2ncnn2C)=O)C1 N(C1CCCn2ncnc21)C(C(CC1CCC1)NC(C1N(CC)CCC1)=O)=O CCCCC(CC)CC(=O)NCC1CC2CC2N1C(C1CCCCN1C)=O Cc1cc(C(N2CC(C)(NC(=O)CC(O)C3CCCC3)C2)=O)ns1 C1(CNC(c2ccn(CCF)n2)=O)(NC(C2CC3(CSC3)C2)=O)CCCCC1 C1(C(=O)NCC(C)(O)CNC(=O)Cn2nnc(=O)[nH]2)(C2CC2)CCC(F)(F)CC1 C1(NC(c2ccc(C)c(I)c2)c2nnnn2C2CC2)CC(F)(F)CCC1(C)C c1(OCC=C)cccnc1C(=O)NCCN(C(=O)CSc1nncs1)C1CC1 C(c1cc(F)cc(F)c1)=CC(=O)NC(CC1CN(C(C(CSC)(C)C)=O)C1)C c1(C(=O)NC2CC(C)(CNC(c3cccc(C(C)C)n3)=O)C2)cccn(C)c1=O c1(C(=O)Nc2cncc(-c3ccc(OCC)cc3)c2)ccc(C(C)C)c(F)c1 Nc1ccc(F)cc1C(=O)NC(C1CCOC1)CNC(=O)C1=C(Cl)CC1 C1(C(=O)NC(C2CCOCC2)C#C)CC(C)CN(C(=O)CSCC(N)=O)C1 c1(CC(C)(C)O)ccc(NC(=O)Cc2csc(Cl)c2)cc1 N1(C(c2cc(SC)oc2)=O)CC(C)OC2(CCN(Cc3nc(C(C)C)cs3)C2)C1 C(=O)(C(C)(C)C(C)(F)F)NCCCN(C(C1CCC(C(=O)OC)CC1)=O)C(C)C C1(C(N)=O)COCCC1NC(=O)C(C1(O)CN(C(=O)CNc2ccccn2)C1)F C(C(C)CC(=O)N(CCC(C)(C)O)CCO)NC(CN1CCC(C)C1)=O Cc1nccc(C(N2CC=CC(NC(c3nc(C4CC4)cs3)=O)C2)=O)c1N C1(C2CC2)(C(=O)NCCn2ccc(C)n2)CN(C(=O)C(C)C#N)C1 CC(C)(C)CCC(F)C(=O)N1CCCN(C(=O)C(O)C(F)(F)F)C(CO)C1 C(=O)(C(C)(C)C(C)(C)C)NCC(C(=O)NCCC1OCCC1(C)C)N(C)C N1(C(c2cc(C)nn2C)=O)CC(CNC(C2(C(F)F)CC(=O)C2)=O)OC(C)(C)C1 C1(NC(=O)CN2CCCCCC2)CCCCN(C(=O)C=Cc2ccccc2)CC1 C12(CCOC1)C(=O)N2C.c1(C(C)(C)SC)cn(C2CC(C(=O)O)C2)nn1 c1(OC)nc(=NC(C)c2ccc(F)nc2)cc[nH]1 Cc1cc(C(=O)NCCOCCNC(=O)C2=CCCC2)nn1C1CCCCC1 C1(NC(C(CC=C)CC)=O)CC2CCC1CN(C(C1CCO1)=O)C2 CCCCC1CNC(=O)C2(CC2)CN1.C(=O)(C(Cc1ccccc1C)CC)OC CC1CCC1C(=O)N(C1(CC(=O)N(C)CC2CC2(F)F)CC1)C N1(CC)CCCc2cc(CNC(=NCC3CCOCC3)NC3CC3C)ccc21 n1(C(C)C)nc(Br)cc1C(c1nnnn1CCC1CC1)NCC1(C)CC(C)=NO1 C12(CN(C(=O)Cc3nccn3C)C)CCC(CC1)N2C(=O)CCOCC(F)F CC1CN(C(C2CCCN2C)=O)CCC1NC(c1cccc(C(N)=O)c1)=O C(=O)(C1=CCCS1)NC(c1ccccc1)C(C)NC(C1(CCC=C)CC1)=O CC1(C)CC(C(=O)NC2CCC23CN(C(=O)CC2(N4CCCC4)CC2)C3)=NO1 c1(N(C)Cc2ncn(C)n2)nc(=NCC2COCCN2C)[nH]c2c1SCC2 C1(CNC(CCC=C)=O)CC2(CCN(C(c3c(SC)nc(O)nc3C)=O)C2)CO1 C12(CNC(C(N)=O)=O)CCCC1N(C(c1ccc(Br)c(O)n1)=O)CCC2 c1(C(N2C(CCNC(C(=O)NCC)=O)CCC2)=O)cc(F)cc(N)c1N c1(C(=O)NCC2C(NC(C(=Cc3cnc[nH]3)C)=O)C2)cc2ccncc2[nH]1 c1(C(C(=O)NCC2CCC(F)(CN)C2)NC(=O)OCC)c(C)cccc1Br c1(C(=O)NCCCC(C)NC(CC=C)=O)ccc(OC(F)F)c(OC)c1 N1(C(c2c(C)c[nH]n2)=O)CCC2(CC1)CC2NC(C1CCC(N(C)C)CC1)=O C1(NC(Cc2c(C)cco2)=O)CCN(C(=O)CC2CCCC23CC3)CC(C)(C)C1 N1(C(Cc2c(C)cco2)=O)CCCC(NC(=O)CC(=O)NCC(F)(F)F)C1 C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1(F)CC(NC(c2c(CCC)n[nH]c2)=O)C1 c1(NCC(C)N(C(C(C(CC)C)Nc2ccccc2)=O)C)nc2ccccc2s1 c1(N2CCC(C(CO)O)CC2)[nH]c(=NC2CCCc3[nH]ccc32)nc2scnc12 Cc1[nH]c2ccccc2c1CC(=O)NC1CC(NCc2cn3cccnc3n2)C1 CC(C)(CNC(=O)CC1CC(O)C1(C)C)CC(=O)NCC1CC(CF)C1 Cc1noc(C)c1C(N1CCC(NC(C2(C3NC(=O)NC3=O)CC2)=O)C1C)=O Cc1nc[nH]c1CC(N1CCCC1CNC(=O)Cc1ccnn1C)=O N1(C(c2cc(C(=O)OC)no2)=O)CCC(O)(Cc2nc(C)cs2)C1 N1(C(C23N(C(C4COCCO4)=O)CC(C)(C2)C3)=O)C2CCC1CC(CO)C2 C(=O)(C1c2c[nH]nc2CCC1C)NC(C1CN(C(C(C)=C(C)C)=O)C1)C C(=O)(C1CCCc2c1ncn2C)N(C)CC1CC(C(=O)OC)C1(C)C C(=O)(C1CCCc2ccccc21)CN1C(CNC(CCNC(=O)C=CCl)=O)CC1 C1(CO)CC2CC(C1)N(CCc1cn(CCCCCCO)nn1)C2 N1(C(C)=O)CC=CC(NC(C2(N(C(=O)CSCC(F)F)C3CC3)CCC2)=O)C1 C(=O)(C1CCCn2cnnc21)N1CC2(N(C(CCc3c(C)noc3)=O)CC2)C1 CCC(CC)(CC)C(=O)NCCC1CCCN1C(c1nc(Cl)c(Cl)s1)=O N1(C(C2CC(C)(CC)C2)=O)CCC(C)C(CNC(c2coc(C(C)C)n2)=O)C1 C(=O)(C(F)C(F)(F)F)NCc1ccc(CN(C(c2ncn(C(C)C)c2)=O)C)cc1 N1(C(C(C(C)(C)C)SC)=O)CCc2[nH]nc(O)c2CC1 c1(C(=O)NCC2CC(C)N(C(C3CCC(=O)N3C)=O)C2)sccc1S(C)(=O)=O C(=O)(C1CCc2nccn21)NCC=CCNC(c1cc(Cl)ns1)=O Cc1ccc(C(N)=O)cc1C(N1CCC2CCC12CNC(=O)CCOC1CC1)=O Cc1n[nH]c2cnc(C(N3CCCC34CCN(C(C3COC3)=O)C4)=O)cc12 C1(C2CN(C(=O)CS(N)(=O)=O)C2)(NC(CN(C)C(=O)C2CC2)=O)CC1 c1(CC(c2nccs2)N(C(=O)C(=O)NC2CCOCC2)C)c[nH]c2ccccc12 N1(c2nc(N3CCC(F)C3)cc(C)n2)CCc2cccc(CO)c2C1 C1(C(=O)NCC(CC)(C)CO)CCCCCN1C(=O)CCN(C)C C(=O)(CCCCC(N)=O)NC1CC(CCNC(CC2(C=C)CCC2)=O)C1 c1(NC(=O)NC(C)CCN2CCOC2=O)cc(-c2ccccn2)n[nH]1 C1(C(N2CCC(CC=C)(NC(C3CC3C)=O)C2)=O)CCC2CC(C)CN2C1 c1(OCC)ccc(-c2nc(C3CN(C)CCO3)nn2-c2ccc(Cl)cc2)cn1 N1(C(CNCC)=O)CC2CC=CCC12.CN(C)S(=O)(=O)NC(=O)CCN1CCCC1 C1(C(N(C)Cc2ncco2)=O)CN(C(C2CC2Cl)=O)CCO1 C1(NC(Cc2c(C)ccnc2)=O)(CNC(C2CCCCS2)=O)CCCCCC1 C1(NC(C2N(N=O)CCC2)=O)CC2CC1N(C(=O)COc1ccc(F)nc1)C2 N1(C(c2cnc(C)s2)=O)CC2CN(C(c3cccc4nc(C)nn34)=O)CC2(C)C1 c1(C(N2CC(C)(NC(C3CCC(CC)C3)=O)C2)=O)ccc2oncc2c1 N1(C(CC(C=C)(C)C)=O)CC2(C=C(C(=O)NC(C)C(C)SC)CO2)C1 N1(C(CCCNS(C)(=O)=O)=O)CC(C2CN(C(c3cnc4sccc4c3)=O)C2)C1 c1(C(N(C(C)CNC(C2CCC(F)(F)CC2)=O)CC)=O)ccc(C)nc1O c1(OC)cc2ccccc2cc1C(=O)OCc1cc(Br)ccc1Cl C1(F)(C(=O)NC(C2CCCC2)CNC(C2(CC(C)C)CCC2)=O)CC=CCC1 C1(NC(C=CC(C)=O)=O)CN(C(=O)CCc2nnc(S)nc2O)CCC1F N1(C(C2C(NC(C3C(C)(C)OCC3)=O)CCCC2)=O)CCN2CC(F)CC2C1 c1(C(N2CC(CNC(C(C)=C(CC)C)=O)OCC2)=O)cccc(C#N)c1Br CC1=CCN(C(C2CC(C)N2C(=O)C=Cc2cscn2)=O)CC1 N1(CC)CC(C(=O)Nc2cc(-c3ccc(C(=O)OC)cc3)[nH]n2)CC1=O C12(NC(c3ncoc3C3CC3)=O)CCCC1N(C(=O)CNc1cccnc1)CC2 N1(C(CCCOCC)=O)CC2(COC(CNC(c3cn(C)nc3CC)=O)C2)C1 N1(C(CN(C(C(C)OCC#C)=O)C2CC2)=O)CC2(CCCO2)C1 c1(CCC)ncoc1C(=O)NC1CCCC1Cn1cc(-c2csc(C3CC3)n2)nn1 Cc1nn(CC(=O)N(CCCn2cc(-c3cccc(F)c3C)nn2)C)c(C)c1C C#CCC(C(=O)N1CCC(C)(NC(=O)C(C)CCC)C1)C1CC1 C1(NC(C(Br)=C(C)C)=O)CCCN(C(c2cnc[nH]2)=O)CC1F c1(CNC(C2CCN(C(=O)CC34CCC(CC3)OC4)C2)=O)cccn2nccc12 c1(C(N2CCC(CNC(C=CCOC)=O)C2)=O)cnc(C(=O)OC(C)(C)C)c(C)n1 c1(C(=O)OCC)cccnc1NC1CC(C)N(C(=O)COCC2CCOC2)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)C2CC=C(C(=O)N(CC(C)O)CCF)C1CC2 C(=O)(CCC(=O)c1cccc(N)c1)NC(C)(C)CNC(C1(CCF)CC1)=O C1(CC)(CNc2cc(N3CCCC(NC(C)=O)C3)ncn2)CCC(=O)N1 c1(C(N(CCC(C)NC(C2N(CC)CCCC2)=O)C)=O)nc(C)[nH]c2nccc1-2 c1(C(=O)NCC(CC=C)NC(c2csc(-c3ncc[nH]3)n2)=O)cnc(N)cn1 C(C(C)(Cn1cccn1)N=c1[nH]nc(C#N)s1)NC(c1c(C)nn(CCO)c1)=O C1(CC=C)(C(=O)N(C(CSC)CC)C)CCN(C(C2CCC=CCC2)=O)C1 C12(CN=C(NC(CC=C)C)NC(c3cccs3)C)CCC(CC1)OC2 c1(C(N2CC(C)C(NC(=O)C(C3CC3)C3CC3)C2)=O)ccc2nccn2c1 N1(C(CCC(=O)OCC)=O)C2CCC1CN(C(=O)CC13CCCC1C3)CC2 CCC(CC)(CC)NC(=O)CC1CCCCC1NC(=O)CCCn1cccc1 c1(CN2CCC(NC(C(C)O)=O)C2)cccc(Cl)c1F C(=O)(C(CC(=C)C)NC(C1CCCOCC1)=O)NCC(C=C)(C)C C1(C)(CC)C=C(C(=O)NC(C2CCCCC2)CNC(c2sc(F)cc2C)=O)C1 c1(CN(CCC)CCC)cnn(C(C(c2csc(CC)n2)=O)=O)c1C(=O)OC.C(C)CN.OC C1(N(C(C2(CCOC)CCC2)=O)C)CCN(C(=O)C(n2cnc(C#N)n2)C)CC1 C1(CCC)(NC(=O)C=Cc2ccc(C)s2)CCCN(C(c2ccc(N)cn2)=O)C1 C(CCCC(=O)NC(C1(C(=O)NCCc2ncccc2C)CC1)C)NC(C)=O Cc1noc(C)c1CC(=O)NC(CCC1CC1)C(=O)NC1CN(C2CCC2)C1 C(=O)(C#CC1CCCC1)NCCC(=O)OCC(=O)N(C(C)C1CC1)C c1(C(N2CC3CC3(C(=O)Nc3nc4sccc4s3)C2)=O)cc(O)nc(Cl)c1 C(=O)(C1=CCC(C)CC1)N1CC(Nc2cc(C(F)(F)F)ccc2F)C(C)C1.CC=O C1(CNC(C2C(=C)CC2)=O)CC2COCC2N1C(c1noc2c1COCC2)=O c1(C(C(=O)NCC(=O)NCCc2c(C(=O)OC)nco2)OC)ccc(CO)cn1 c1(C(N2C(C(N(CCCC)CCO)=O)CC(C)C2)=O)cccc2sccc12 n1(CC)ncc(C(N2CCC(C)(NC(=O)C=C(C)C3CC3)C2)=O)c1C(F)(F)F Nc1cc(F)cnc1C(=O)NCCC1(O)CCN(C(C2CCCCNC2=O)=O)C1 C1(C(C)NC(C(=O)NCC)=O)CCN(C(c2csc(CC(F)(F)F)n2)=O)C1 C1(NC(COc2c(C)cccc2)=O)CCN(C(C2C3CC4C(C3)C24)=O)C1(C)C N1(C(C(C=CCCC)O)=O)CCN(C)CC1CNC(c1c[nH]c(=N)o1)=O C(C(CC(F)(F)F)NC(C1(O)CCSC1)=O)NC(COC(CC)CC)=O c1(C(=O)NCC2(NC(C3C4CC5C(C4)C35)=O)CCCC2)cnc(S)nc1 C1(NC(C(C2CN(C(C3C(OC)CC3)=O)C2)O)=O)CC(C)CC(C)(C)C1 C1(CCC(=O)NC2CN(C(C)=O)C2)CCN(C(=O)Cc2ccn(C)c2)C(C)C1 O=C1NCCN2CCN(CC3CCCCC3(F)F)CC12 CC1CC(C)(CNC(C2CN(CC(c3nccs3)C)C2)=O)C1 C1(C(N(CCOCCC(=O)NC(CC)C(=O)OC)C)=O)CCC(C)=C(C)C1 c1ccsc1C(=O)CC.c1(C(N(CCOCCN)C)=O)conc1C(C)C C1(NC(C(OC)OC)=O)CN(C(=O)Cc2cc(Br)cs2)C2(CCCC2)C1 Cc1cc(C)c(C(=O)NCC2CC3CCC2N(C(=O)C(O)C(C)C)C3)cc1C C1(C(=O)OC)CCCCC(NC(=O)NC2CCC(OC)(OC)CC2)C1 c1(C(N2CCC(C)(CC(N3CCC(O)(C(N)=O)CC3)=O)C2)=O)cc(F)ccc1F c1(C(=O)NCC2N(C(CC3ON=C(C)C3)=O)CCC2C)n[nH]c2c1CCCCC2 Cn1nccc1COCC(N1CCCC1CCNC(=O)CCn1cc(Cl)cn1)=O c1(CC)ccc2c(c1)CCC2.CCC1C(O)C(=O)N1 N1(C(c2cc(OC)ncc2)=O)CC2CCN(C(=O)C(C)(C)O)C2C1 c1(CN(C(C2CCC(CNC(C)=O)CC2)=O)C(C)C)ccc(C)c(C)c1Cl C(=O)(C(O)C1CCCC1)N(CC(C)NC(=O)COC(F)F)CC C1(N(C(=O)Cc2cnoc2)CC#C)CCN(C(=O)C=Cc2cnc[nH]2)CC1 N1(C(C(C=C=C)C)=O)CCC2(CCN(C(=O)CCOCC)C2)C1 C(=O)(C#CC1CCCCO1)NCCCN(C(CCS(=O)(=O)NC)=O)CCO c1(CC)nn(C)c(Cl)c1C(=O)NC1C2CN(C(=O)CCC3CCOCC3)CC12 C(=O)(CCC(C)(C)F)N(C)CC1CN(C(C2CC2(C)C(F)F)=O)C1 C1(O)(C(=O)NC(=O)CCC2CCN(C(c3cc(C)sn3)=O)C2)CCC(C)(C)CC1 c1(C(=O)NC(CC)C(=O)NC)cc2c(N)nccc2o1 c1(OC)cccc(C(=O)NCCOCCOCCNC(C2CNC(=O)N2)=O)c1 N#CC1(C(=O)NCCNC(C23CCC(C(F)F)(CC2)C3)=O)CCSCC1 c1(NC(N2CC(C)(C(F)(F)F)OCC2)=O)cn2cc[nH]c(=O)c2n1 C(C(C)(C(C)C)NC(c1cc(C2CCOC2)[nH]n1)=O)NC(C=CC=CC)=O c1(NC(C2CCN(Cc3ccc(C)cc3)CC2)=O)ccc([N+](=O)[O-])cn1 c1(C(=O)NC2(CF)CCN(C(CCC)=O)C2)ccc(P(C)(C)=O)s1 c1(C(=O)NCCN(C(=O)C(C)Cc2ccccc2Cl)C(C)C)cc(C#N)no1 C1(c2cn(CC3CN(C(=O)CN(C)C(C)C)C3)nn2)(OC)CCOC1 C1(CNC(C2(C)CC(C)C2)=O)CN(C(=O)C2=CCSC2)CCCO1 c1(OC)ccc(C(=O)NCC(CC(C)C)NC(c2nncs2)=O)c(O)c1 C1(COC)(CNC(=O)C=Cc2cscn2)CCN(C(c2ccon2)=O)C1 c1(C(=O)NC2CC(C(C)(C)O)C2)cccnc1CNC(=O)C(C1CC1)C1CC1 CC12CCC(C(=O)NC3COCC3NC(=O)Cn3cnc(=N)[nH]3)(CO1)C2 N1(C(C2C(C(C)O)C2)=O)CCCC(NC(=O)Cc2cccs2)C1C C1(C(N2CC(NC(C3(CC)CC3)=O)C(OC)C2)=O)CN2CCN1C(C)C2 c1(C(=O)NCCOC2CCN(C(c3cn(C)c(O)n3)=O)C2)ccc(F)c(F)c1F Cc1cc(I)ccc1CNC(=O)C(N1CCCC1c1sccc1Cl)=O CC(C)CCCC(C)CNC(=O)CC1CCN1C(=O)CC(C)OC c1(OCC)ccc(NC(=O)N(C(CO)CO)Cc2ccccn2)cc1C#N c1(NC2(c3nnnn3C3(C)CC3)C(C)OCC2)ccc2[nH]ncc2c1 c1(C(N(CCCCNC(c2n[nH]c(C)c2Cl)=O)C)=O)c[nH]c2c(Cl)cccc12 c1(C(=O)NC(CCNC(c2c(C)[nH]nc2C(F)(F)Cl)=O)C)nnn2c1CCC2 N(C(=NCc1cccc(N(CC(F)(F)F)C)c1)NC1CSC(C)C1)C(C=C)C N1(C(CC(C=C)C)=O)CC(C(=O)N(CC(F)F)CCC)CC(C)(C)C1 C(=O)(C(C)(CNC(C1CCCC1F)=O)CC)N1C(C)(C(=O)NC)CC1 C(C(CC1CC1)C(=O)N(CC(C(=O)Nc1nnnn1C)c1ccccc1)C)SC N1(C(CN(C(=O)OCC)C)=O)CCC(C)(C)C1CC(=O)N(CC(C)(CO)CO)C C1(C(N(CCOC)CC)=O)C2CCC(C2)N1C(c1n[nH]c(C)n1)=O N1(C(C(C)n2ccnn2)=O)CCCC(N(C)C(c2cc(C(C)(C)C)c[nH]2)=O)C1 N1(C(CNC(CCNC(C)=O)=O)=O)CCCC(O)(CNC(C2(C)CC2(C)C)=O)C1 O=C(CC=C(Cl)Cl)NCC1(C(=O)NCC(O)C2CCC2)CC1 C1(C(N2CC(F)(CC)C2)=O)CC(F)(F)CN1C(=O)Cc1ccn(C)n1 c1(CN2CC(C(=O)Nc3nc(O)cc(OC)n3)OCC2)c(Cl)ccc(F)c1F N1(C(C2CC(=C)C2)=O)CCCCC1CCNC.C(CCC=CC(=O)O)=CC=CC=CC=C C1(F)(C(=O)NCC2(CO)CC(C)(C)C2)CCCN(C(=O)CCC2CCCO2)C1 C(C(C)(CNC(=O)CCCC1(NC(=O)CN2CC(C)(C)C2)CCC1)CO)OC c1(-c2cc(C)sn2)nc(-c2cccc(Cl)n2)nn1-c1ccn(C)n1 c1(-c2ncc(C(=O)Nc3nccc(OCCOC)n3)nc2)ccc2cncn2c1 C(=O)(CCC(C)(C)F)NC1C(CNC(c2ccc(OCCCC)nc2)=O)C1 Cc1ccc(C(N2CC3(CNC(=O)C(C)(C)C4CC4)CCC2CC3)=O)c(Cl)c1Cl Cc1cc(CNC(=O)C(=O)N(C)Cc2sccc2Cl)n(C)n1 N1(C(C(C)(C)C)=O)CCCC1C1CCCCN1C(=O)CCc1cccnc1 Cc1ccc(-c2nc(C(=O)NC(C)CN3CCOCC3)cs2)c(C)c1 c1(N(C)CC2CCCC2)nnc(C2CCCC2)n1CSc1cncc(Br)c1 c1(CC(N2CC(CCO)(CNC(=O)Cc3cscn3)C2)=O)nnc(O)nc1O.C1CC1 C1(C(=O)NCC(C)O)CC2(C1)CN(C(=O)CC(=O)N(C)C)C2 N1(C(CCc2c(C)noc2)=O)CCCC(C)(NC(=O)C(C)Cc2cnco2)C1 N1(CCOC)CC(C(=O)NCC2CC3CC3N2C(=O)CCSC(C)C)CCC1=O Cc1cc(C)c2c(c1)C(N(C)C(c1ccc(C(F)(F)Br)nc1)=O)CCO2 c1(C(CF)NC(=O)NC2CC=CC2)ccc(F)cc1 c1(OC)cc(C(=O)NC23CC(CNC(C45CC4COC5(C)C)=O)(C2)C3)c(F)cn1 C12(C(=O)NC3CC=CCC3C(N3CCC(CO)C(O)C3)=O)CCCC1CCC2 C(=O)(CCCS(N)(=O)=O)NC1CC(C)(C)N(C(C2CNC(=O)C(C)(C)C2)=O)C1 C1(OC)CC2CCC1CC2C(=O)NCC1CC(CNC(=O)C(C)(C)C2CC2)CO1 C(=O)(C1=CCC(F)(F)CC1)N(C(C)C(c1ccc2c(c1)OCO2)=O)C c1(C(=O)NCC2C(NC(C(C)OCC)=O)CC2)cnc(Br)s1 N1(C(C2CN(C)C2)=O)CC(NC(C2CC3C(C2)C3(F)F)=O)CC(F)(F)C1 c1(SC)ncc(N)c(C(=O)NC2CN(C(=O)CC3C(=O)NN=C3C)C2)n1 O=C(C1Cc2c(Cl)cccc21)NC1(CCO)CN(C(c2ccncc2)=O)C1 N1(CC(N2CC3CCC2(CNC(C2(O)CCC2)=O)C3)=O)Cc2ccccc2C1=O C(=O)(CC(C)CC(F)(F)F)N(CC(C)NC(c1ccnc(C)n1)=O)CC c1(CC)ccc(F)cc1NC(=O)CC(C)(C)NC(=O)CN(C1CCC1)C C1(NC(CC=C)=O)CC2CCC1N2C(=O)Cc1ccn(CC(F)(F)F)n1 C1(NC(c2nccc(C)c2)=O)CCN(C(c2ccc(C)nc2N)=O)CC1C c1(OC)ccc(C(C)NC(C2CCN2C(=O)CC2CCCCO2)=O)cc1 C#CC1C(C(=O)NC(C2CCCCC2)CNC(C2CC23CC3)=O)C1(C)C c1(OCC(C)NC(C2(CN(C(CSSC)=O)C)CC2)=O)ccccc1 N1(C(C=C(CC)CC)=O)CCN(CCN(c2ccoc2C)CC)C2CS(=O)(=O)CC12 CC1CCC(NC(=O)CC(C2CCC2)C2CCC2)CN1C(C1(O)CCC1)=O C#CC#CC(C)(C)NC(C1CN(C(C2CCC(OC)C2)=O)CC1CC)=O C1(N(C(C)C)CC)CC2(C1)CC2CC(=O)O.N12CCCC1c1cn(nn1)CC2=O N#CC1(C(=O)NCC2CC(NC(=O)C(O)Cc3ccccc3)C2)CCC1 CC1=NOC(CC(=O)NCc2ccsc2C(=O)NOCC2CCCO2)C1 C1(C#N)(C(=O)NCCN(CCCN(C)C)C(C2(C)CCNC2=O)=O)CC1(C)C C1(COC)CN(C(=O)C(F)C2CC(NC(=O)C=CC3CCCCC3)C2)C1(C)C N1(C(C(c2cccs2)NC(c2nc(CC)sc2)=O)=O)CCCC(C)C1CO C=CCC(CNC(c1cc(C(C)C)on1)=O)C(=O)NC1CCCCC12CC2 C=Cn1nccc1C(=O)NCC(C)(C1CCC1)NC(=O)C(C)Cc1cnn(C)c1 c1(N2C(CC)CCC2)cc(C(=O)OC)ncn1.C12CC1C(=O)N(C)C2(C)C N1(C(c2cc(SC)cc(Cl)c2)=O)CC2CCC(C1)C(NC(=O)C1=CCCC1)C2 c1(NC(N(C2CCN(C)C2=O)C)=O)ccc2nccn2c1 C12(CNC(C3CN(C(C)=O)C3)=O)CN(C(C3COCCO3)=O)CC1CS(=O)(=O)C2 CC1(C)CCOC(CC(=O)NCC#CCNC(c2ccncc2Br)=O)C1 c1(CN2CCC(CNC(c3cc(C(C)(C)C)ncc3)=O)C2)cc(O)ccc1Cl C(=O)(CCCC(C)(C)NC(c1ccc(F)cc1F)=O)NCC(C(C)(C)C)OC C(CC(C(=O)N1CCOC(CCF)C1)NC(=O)CC1(CS(C)(=O)=O)CC1)SC CC(C)CC(O)CC(=O)NC1CCCN(C(=O)COc2ccccc2C(N)=O)C1 C1(C(N(CC(C)N(C)C(c2ccc(CN=[N+]=[N-])o2)=O)C)=O)CCCCN1C1CC1 C(=O)(C(C(C)C)C(C)C)NC1C(C(N(CC(C)(C)C)CCC#C)=O)CCCC1 CC(C)CCCCCC(=O)N1C2CCC1CC(CNC(c1cnn(C)c1F)=O)C2 c1(C(C(N2CCCC2=O)C)=O)ccccc1NC(=O)NNC(=O)C1COCCO1 c1(OC)ccnc(C(C(=O)NC2(C)CC2)N(C)Cc2cnn(C)c2)n1 C(CC(=O)N1CCC(COC(C)=O)C1)(C(F)(F)F)NC(C(COC)OC)=O Cc1nc(C)c(C(N2CC(NC(=O)Cc3ccc(C(C)C)cc3)C(F)C2)=O)s1 n1(CC(N2CC(OC)C(NC(C3CC(SC)C3)=O)C2)=O)nc(C)c(C)c1C c1(CN2C(C(=O)Nc3nc(C)nc(Cl)c3)CC(C)C2)ccc(C)c(C#N)c1 N1(C(CC2(NC(C)=O)CCC2)=O)CC2=C(C1)CN(C(=O)CCC1(C)CC1(F)F)C2 N1(C(CC2N(CC)CCOC2)=O)CC=C(CCNC(C2CCSC(C)C2)=O)CC1 CCC(C)(CN=c1nc(N(C)Cc2ccnc(C(F)F)c2)c2sccc2[nH]1)OC N1(C(C2CCN(S(C)(=O)=O)CC2)=O)CC2(CCN(C(=O)CC3COCCO3)C2)C1 C(=O)(C1CCOc2ccccc21)NCC1(NC(C23COC(C2)C3)=O)CC1 CC(C)CCC(=O)NCc1cc[nH]c1C(=O)NCC(CN(C)C)CO c1(C(N2CC(NC(C3(O)CCSC3)=O)C(C(F)F)C2)=O)nccc2cc[nH]c12 N1(C(C(C=C)c2ccccc2)=O)CCC(CO)(Nc2ncnc(C(C)C)n2)CC1 C(=O)(C(C)CC(C)(F)F)NCCCCC(C)NC(=O)C(C)(C)CF c1(C(=O)NCC(CO)NC(CC(CN(C)C)O)=O)cc(Cl)ccc1O N1(C(=O)Cn2cnnn2)CCC(C2CC2)(NC(C23CC(F)(C2)C3)=O)C1 N1(C(=O)Nc2scc(CCC)n2)CC2CC1C2c1cn[nH]c1 N1(C(COCCC=C)=O)CCn2ncc(CNC(=O)C=C(C)C(C)C)c2C1 c1(CCCCCC)nc(-c2cc(=O)cc[nH]2)n(-c2ccc(-c3ccco3)cc2)n1 N1(C(C(n2c(C)ncc2)C)=O)CCCC(F)(C(N2CCCC2CCO)=O)C1 c1(C(N(CC(C)NC(C2(C(C)(F)F)COC2)=O)C)=O)cc2cc(Cl)c(Cl)cc2[nH]1 C#CC1CCN(C(C2(CNC(c3cc(OC)n[nH]3)=O)CCOCC2)=O)C1 N1(C(C(C(CC)C)O)=O)CC2(CCOCC2C(=O)N(OC(F)(F)F)C)C1 c1(C(=O)NCCNC(c2c(CC)scc2)=O)cnc(C)cc1C CCC(F)(F)C(C)(C)CN1CCCC1Cc1ccc(C#N)cc1 c1(C(=O)NC(C)CCNC(C2(C)COC(C)(C)OC2)=O)cc(F)c2c(c1)CCC2 C1(CC=C)(NC(=O)C(COC(C)C)N(C)C)CCN(C(=O)Cc2ccccn2)C1 C1(NC(c2cnc(C)[nH]2)=O)COC2(CCN(C(C3(F)CCCC3)=O)C2)C1 c1(C(=O)NCC(N(C(C(C)CO)=O)C)C2CC2)cn(C)nc1C1CC1 CC1CCCN(C(=O)CN(C)Cc2ncoc2C2CN(C(=O)C(C)CO)C2)C1 c1(OC)cncc(Br)c1C(=O)NCCN(C(=O)CCCOC(C)C)C c1(OC)c(C)c(NC(=O)C(C)NC(=O)C(C)(C)C)c(C(C)=O)c(C)c1C CON1CCC(CC(=O)NCC2(CNC(=O)C(F)CC3CCOCC3)CC2)CC1 CCC(CC(=O)NCC1CCCC1C(=O)NC1CCC(C)CC1)C1CCC1 Fc1cnc(Br)c(CNc2ncc(-c3ccnnc3)s2)c1 c1(C(C)C)cccc(CN=C(NCC(=O)N(C)C)NCC2CCC2)c1 Cn1cccc1C(=O)NC1(C2CCCN2C(=O)CCC2(C)N=N2)CC1 CCC(CC(=O)N1CC(CC(=O)N(C)CC2CCCC2(C)C)C(C)C1)C(C)C C1(CNC(C2(CC#C)CCCO2)=O)CN(C(c2nc(C(C)(C)C)no2)=O)CC1C S(=O)(=O)(c1ccc(C(F)(F)F)cc1)CCN1C(CNC(CC(C)C)=O)CCCC1 c1(N(C)CCNC2CCC2(C)C)cc(=NCC(C)(C)C2CCC2)[nH]cn1 CC(CC(F)F)C(=O)NCC1CCN(C(c2cnc(-c3cnccn3)s2)=O)C1 C1(NC(CC2CC(=O)NCC2)=O)CC2CC1N(C(=O)C=C1CCCCC1)C2 c1(C(=O)NCC(CC=C)NC(c2ccn(CCO)c2C)=O)cccc2nncn12 Cc1[nH]nc2cc(Nc3cc(=NCC4(C)CCS(=O)(=O)CC4)[nH]cn3)ccc12 C1(NC(=O)C(O)CC(F)F)CC2(CCN(C(=O)C(F)=CC3CC3)C2)C1 C1(C(N2C(C)CN(C(C3CC(C4CC4)C3)=O)CC2)=O)CN=C2N=CNN2C1 Cc1ncc(N)cc1C(N1CCN(C(=O)C(c2ccc(F)cc2F)(F)F)CC1)=O c1(CCC(=O)N(C)CCNC(=O)C(C)(C)c2ccccn2)ccccc1Br Cc1ccncc1CNC(c1ccc(CNC(=O)C(C)C2CCOC2)nc1)=O c1(CSCCC(=O)NC2CCN2)cccc(C(F)(F)F)c1 n1(CC=C)c(C(=O)N(CC)CC)cc2ccccc12.O C1(NC(c2ccc3oc(O)nc3n2)=O)CCCC12CCN(C(c1cnsn1)=O)C2 CN=c1ccc(Br)c(C(N2CCC(F)CC2)=O)[nH]1 C1(C(=O)NC2(CC)CN(C(c3c(CC)nccc3)=O)C2)CC2CCCCN2C1 CC(CC(=O)N(C)Cc1nc(=O)o[nH]1)C(C)(C)NC(=O)C(C)N1CCCC1 C(=O)(C(C)(C)CS(N)(=O)=O)NCC1CC(NC(c2c(C)nc(C3CC3)cc2)=O)C1 CCC(N=c1[nH]c(=NCCC(C)N(C)C)c2ncccc2[nH]1)C(C)C Cc1ccc2nc(C(=O)NC3(C)CCN(C(C4CCCC45CC5)=O)C3)cn2c1 c1(C(=O)NC(CC=C)CNC(=O)Cc2ccc(C)nc2)ccc(Cl)c(OC)c1F CC1(C)CNC(=O)C2CC(C2)CC(CC)C2C(C1)CN2C(c1sccc1F)=O CC1CCN(CCC(=O)NCC2CN(C(=O)C(C)Cc3ccc(F)cc3)C2)CC1 CC1CN(C(=O)C(C)NC(C2(O)CCOCC2)=O)CC(=O)N1 c1(CC=C)nc(C2CCCCC2)nn1-c1ccn(CC)n1 N1(C(c2cc(C)cc(F)c2)=O)CCC2CC1CN2C(c1cc(C#N)cc(C)n1)=O N1(C(c2ccc(CC)[nH]2)=O)CCC(C)C1CNC(=O)C=C1CCCC1 C(=O)(CS(=O)(=O)CCO)NC(C1(O)CCN(C(=O)CC2CCC(F)(F)CC2)C1)(C)C C#CCC(CC#C)C(=O)NCCOCCNC(=O)C(C)(C)C1CC1 C(=O)(C1=C(C)CCC1)NC1CN(C(CCNC(C)=O)=O)CC1Cc1ccccc1 O=C(C1CCCc2nc[nH]c21)NCCO.C1CCC(=O)N1 CCC(C)C(C(=O)OC1CCCN(Cn2nc(C3CC3)n(C)c2=O)C1)N(C)C c1(C(=O)NC2CC3CN(C(CC=C(C)C)=O)C2C3)ccc(S(N)(=O)=O)c(C)c1 c1(SC)ccc(N)cc1C(=O)NCC(O)CN(C(=O)C(CC1CCCC1)OC)C C(C(=O)NC(C)(CNC(=O)CNS(C)(=O)=O)C1CC1)(C(C)C)n1cc(C)nc1 CC1CN(C(=O)Cc2ccco2)CC1NC(=O)CCc1ccc(O)nc1 C1(COC)(NC(C2CSCCS2)=O)CCCN(C(c2ccc(C3CC3)cc2)=O)C1 CC1(C)CC(C(=O)N2CC(CO)(NC(=O)CCC(=O)N3CCC(O)CC3)C2)=NO1 Cc1nc(C2CCC2)oc1C(=O)NC(C)CC(C)NC(C1(CO)CCCCO1)=O c1(C(=O)NCC(CC)NC(=O)CC(O)CN(C)C)cc(N(C)C)ccc1N c1(C(C(=O)NCCOC)N(C)CCc2ccccc2)cnc(C)c(C)c1 N1(C(C(C)C(F)F)=O)CC2CCC1C1CN(C(=O)C=CS(C)=O)CC21 C(=O)(C(CCCOC)NC(=O)Cc1cn(C)nc1C)N1CC(CC)SCC1 O=C(CS(=O)(=O)c1ccc(-c2ccnnc2)cc1)NCCOC1CCNCC1 N1(CC(=O)N(C2CCCCC2)C(C)C)CC(=O)CC(C)C1 c1(C(C(=O)NC)N(C2CCN(CC)CC2)C)ccc(C#N)c(F)c1 C(=O)(CC(C(F)F)n1ccnc1)NC1(CNC(C=CCCC)=O)CCOC1 c1(N2CC(F)CC(C(=O)Nc3ccnc(Cl)c3I)C2)ncnc2[nH]cc(I)c12 c1(CNCc2cccc(C(=O)NCCC)c2)ccccc1S(=O)(=O)F Cc1cn2c(CCC(=O)NC3CN(C(=O)C(C)C#N)CCC3O)csc2n1 Cc1ccc(-c2nc(C(C)O)nn2CC(C)(C)CO)cc1OC(C)C C(=O)(C(C)N=c1cc[nH]cc1)NC(C(C)NC(CC1CC(CC)C1)=O)CO c1(C(N2CCC(NC(C(C)Cc3cnn(C)c3)=O)C2C)=O)ccc2n[nH]cc2c1 C1(NC(c2cn(CC)nn2)=O)CCC(C(N2CCC2CF)=O)CC1 c1(C(N2CC(C)N(C(c3ccc(Br)o3)=O)CC2)=O)coc2c(F)cc(F)cc12 C1(NC(CC=C(C)C)=O)CCN(C(=O)CCc2cccc(C)c2)CC1F C=C(C)CC(C(=O)NCC(C)N(C)C)NC(c1nn(C)cc1Cl)=O C1(N(C(=O)C2CC2)CC)CCN(C(=O)OC(C)(C)C)C1C(F)(F)F C(=O)(CCCC(=O)N1CCCC1C(C)(C)NC(C1CC12CCOC2)=O)NC c1(NCC2CCC(C#N)CC2)cc(Cl)c(C#N)c(Cl)c1 C=Cc1ccc(C(=O)NC(C)(C)CC=CC(=O)NC2(C)CCC(O)CC2)cc1 C(c1cscn1)=CC(=O)NCCN(CC(C)O)C(=O)CC1CCCN1C CCN=c1ccc(C(N2CCC(NC(C3CC(=O)N3)=O)C(F)C2)=O)c[nH]1 c1(CC(=O)NC2C(NC(C=CCC)=O)CC2)nocc1C c1(C(=O)NC2C(OC)CN(C(CCCCC=C)=O)C2)ccc2c(c1O)CCCC2 CC(CCC(C)(C)C)C(=O)N1CCC2(C(=O)NCC3(CN=[N+]=[N-])CC3)CCCC12 C(=O)(CC(C)CC(F)(F)F)N1CCC(C)C(NC(c2cc(C)nc(Cl)c2)=O)C1C n1(CC)cc(C#N)c(=NC(=O)C2CC(NCc3c(C)[nH]c4ccccc4c3=O)C2)[nH]1 C(=O)(CC1CCc2ccccc21)N1CC(COC)(CNC(C2(F)CCC2)=O)C1 N1(C(C=COCC)=O)CC(NC(=O)C(N2C(=O)CCC2=O)C)CC(C)C1 C#CC1(NC(C2(F)CCN(C(=O)CNC(=O)C(C)CC)C2)=O)CCCOC1 n1(CC)c(C)cc(C(=O)NCC(C2CCC2)NC(c2ccc(C)cn2)=O)c1C N1(c2ccnc(N(CCCC(=O)NC)C)n2)CCS(=O)(=O)CC(C)C1 c1(C(N(CCCCNC(Cn2ncc(C)c2)=O)C)=O)cccc2c1SCCC2 Cc1ncnc(N2CCC(NC(c3ccon3)=O)C(C)(C)C2)c1C#N CCC(C(=O)NCC1(C)CCN(C(c2sccc2Br)=O)C1)C(F)(F)F c1(C(=O)NC2(CC)CCN(C(C(C=C)(C)C)=O)CC2)cc2c(nc1O)CCSC2 c1(N(C2CC3CNC2C3)C(CN2C(C)CCC2)=O)cccc(F)c1Cl Cc1c(C(=O)NC2CCN(Cc3cc[nH]c3)CC2(C)C)ccc(F)c1[N+](=O)[O-] CCCC(F)C(=O)NC1(C)CCN(C(=O)Cc2ccccc2)C1 C(=O)(C1CCCn2cnnc21)NCCN(C(=O)C(C(C)CC)OC)CCC c1(C(N(CCCNC(C2CC(F)(F)C2)=O)CCO)=O)[nH]nc2ncccc12 C(=O)(C(C)(C)CC(F)(F)F)NC1C(NC(c2nnn(C)n2)=O)CS(=O)(=O)C1 C=C(C)CC(C)C(=O)N(C1CCN(C(c2cc(CO)oc2C)=O)CC1)CCC C1(C(N2CCC(NC(c3c(C)ccnc3C)=O)C(F)C2)=O)CC2(COC(=O)N2)C1 CCC1=NOC(C(=O)N(C)CC2COCCN2C(=O)CNC(=O)OC)C1 N1(CCC(C)C)CCCCC1C(=O)NCCNC(=O)Cc1cccnc1F N1(CCCOC)CC(COC(=O)Cc2ccc(OCCC3CC3)cc2)CC1=O C1(F)(C(=O)NCc2nn(C)c(=O)o2)CCCN(C(=O)C(C2CCCCC2)F)C1 c1(CC(=O)NC2CCCC2NC(c2ccncc2C2CC2)=O)ccc(F)cc1F c1(CCC(=O)NCC(CN(C)C(c2cnn(C)c2F)=O)O)ccc(O)cc1 N1(C(CCC)=O)CCC(CN(C(=O)COc2ccc(Br)cc2)C)CC1 N1(C(=O)Nc2c(C)ccc(Br)c2)CCN(C(=O)CN(C)C)C2(CC2)C1 N1(C(C(C(C)(C)C)SC)=O)CC2(CC(NC(=O)C=Cc3cnccc3C)CO2)C1 C1(C(N2CC3C(CNC(Cc4cc(C)sc4C)=O)(C3)C2)=O)CC(C2CC2)=NO1 C1(C(N2CC3(CC(NC(C(F)=CCC)=O)C3)C2)=O)(OC)CCC(C)(C)CC1 N1(C(C2(NC(=O)C(F)C3CCCC3)CCSC2)=O)CCOC2CCC12 C1(C(=O)NC2CCN(C(C(CC=C)C)=O)C2C)CNC(=O)CC1(C)C C=CCCCC(=O)N1CC2C(CNC(c3ccccc3NS(=O)(=O)CC)=O)C2C1 C(=O)(C1=CCCOCC1)NC(CNC(C1N(C(C)(C)C)CC1)=O)C1CC1 CC1(C(=O)N2CC(NC(C34CC(F)(C3)C4)=O)C(O)C2)CCCc2ccccc21 Cc1ccc(COC2CCN(C(=O)C(O)CCCN3CCCC3)CC2)c(C)c1 C(=O)(CCCCCCCC(=O)NC(C)C(C)NC(=O)CC1=CCOCC1)OC C(CCCCCCCO)=CC(N1CCN(C(CC(C=C)C)=O)CC1C(C)C)=O C=CCN=C(NCC1(C2CCOCC2)CCC1)N1CCC(Oc2ccncc2)C1 c1(OC)cnc(F)cc1-c1nc(CCCN(C)C)nn1CC1CCCO1 c1(C(=O)NCCCN(c2nc(C)c(C#N)cc2)C)ccc2c(c1)C(=O)NCC2 c1(CC(=O)N(C(C)C)CCN(C)C(c2ccoc2Cl)=O)cccnc1Cl C(=O)(C(C)(C)CCCF)N1CC(CCNC(c2nc(OCC)oc2)=O)C(C)C1 N1(C(CN(C(CN2CCC(C)CC2)=O)C)=O)CCC(N=[N+]=[N-])CC1 CC(C)C(C)C(C)CC(=O)NCCCc1cn(CC2CC3(CCC3O)C2)nn1 N1(C(c2csc(-c3ccccc3Br)n2)=O)CCN(C(C2CC2F)=O)C2CC12 C1(CC)CN(C(=O)CC(C)(C)CC)CCN1C(c1cccn1CC)=O N1(C(Cc2cccc(C)c2Cl)=O)C2CCC1CN(C(c1scnc1C)=O)C2 CC(C(=O)N1CCSCC1CCNC(=O)CC(C)n1ccnc1)C(C)S(C)(=O)=O CCS(=O)(=O)CC(=O)NCC(O)CNC(c1cc(-c2ccc(OC)cc2)[nH]n1)=O c1(C(=O)NC(CC2CN(C(CCCN(C(=O)OCC)C)=O)C2)C)cn(C)c(O)n1 C(=O)(C(C(C)NC(=O)CC1CCOC1)C(C)C)NCCc1nc(C)oc1C Cc1cc(N2CCC(C(N3CCC(c4cnc(N(C)C)nc4C)C3)=O)C2)ccc1Br c1(N(CCNC(C2CC3CC3C2)=O)CC)ncc2c(ncn2C)n1 c1(CNC(c2ccc3nnn(C)c3c2)=O)nc2ccc3ccccc3c2[nH]1 C1(F)(CNC(Cn2cc(-c3cn(C(C)C)nc3)nn2)=O)CCC(C(=O)O)C1 O=S(=O)(c1cccnc1NCC1(C2CCCO2)CCC1)N1CCCCC1CCO c1(C(N2CC(NC(C3CC4(CCC4)C3)=O)(CF)C2)=O)cccnc1S Cc1cc(C(=O)NCc2cn(CC(=O)NC3CC(O)C(F)C3)nn2)c(C)o1 C1(NC(Cn2c(C)ccn2)=O)(CNC(=O)C=C2CCN(C)CC2)CCCCC1 C1(NC(C2(CC=C)CCCN2C(=O)C=CC(F)F)=O)CCC(C#N)CC1 c1(CN2CCN(c3cncc(OC)n3)CC2)ccc(CC#N)c(F)c1 N1(C(C2(OC)CCC2)=O)C2CCC1C(CNC(c1cccc(C(F)(F)F)n1)=O)C2 c1(C(N(CCNC(COC(CC)C)=O)CC)=O)cnc(O)c(C)c1 N1(C(C(=O)NCCOCC)C)CC2CC(NC(c3cc4ccsc4s3)=O)CC1C2 c1(NC(=O)NCCc2cncc(OC)c2)ccc(F)cc1OCCC(C)C N1(C(C(CC)n2cncn2)=O)C2CCC1CC(NC(C1CCC1)=O)C2 c1(NC(CC2(Nc3ncc(C)c(C)n3)CCC2)=O)ccc(C#N)cc1F c1(C(=O)NCC(CCNC(C2C(CC)C2)=O)(C)C)cncc(OC)c1C c1(NC(c2c(OCC)oc(C)n2)=O)cc(C)ccc1OC.C12CC(F)CN1C2=O C=C(C)C(O)CC(=O)NC1(C)CCC(NC(c2cncs2)=O)CC1 c1(CC(C(=O)N(CCN(C(=O)CCCN(C)C)C(C)C)C)C)cccc(Cl)c1 c1(C(=O)NC2CCCC2NC(C2(O)CC2)=O)ccncc1O N1(C(C2(C=C)CCC2)=O)CCCC(N(CCO)C(c2ccoc2Cl)=O)C1 C1(C(=O)NC(Cc2c(C)n[nH]c2C)C)CN(C)CCN1C(=O)CCc1cn[nH]c1 CC(CC(=O)NCC1CC(F)CN1C(c1cnc(C(F)(F)F)nc1)=O)P(C)(C)=O CCC(C)(C)C(O)C(=O)N1CCCC1C1CCN(C(=O)Cc2cnsc2)C1 N1(C(CC2CCN(C(CCCOCC)=O)C2)=O)CCC(O)CC1C1CC1 C1(NC(c2c(C)cc[nH]2)=O)C2CCC(C2)C1C(=O)NC1(CCO)CCOC1 C1(C(N(CC(C)OC)CC)=O)(NC(c2ccc(C(F)F)o2)=O)CCSC1 c1(CNC(c2c(OC)n(-c3ccccc3)nc2)=O)cc(Cl)c2ccncc2n1 C1(CN(C2CCC2O)C)CC12CCOCC2 c1(C(=O)NCCCCC(C)NC(=O)Cc2cc[nH]c2)ccccc1N=[N+]=[N-] N#CC1(CNC(=O)CCC2(NC(=O)Cn3cc(Cl)cn3)CCCC2)CCCC1 Cc1ccc(F)c(C(N2C(C(=O)NC3COCC3CO)CC3CC23)=O)n1 N1(C(C=C(CCC)C)=O)CCN(C(=O)COCC(C)C)C2COCC12 c1(CC(=O)NC2CCC(C)(NC(C(CCC)OCC)=O)C2)ccc2nsnc2c1 N(C1c2cc(C)ccc2CC1C)C(CC(C)(C(F)(F)F)N(C)C)=O C1(NC(C2C(OC)CCC2)=O)CC2CC1CN(C(c1cc(O)cnc1Cl)=O)C2 C(=O)(C1CCc2ccccc21)N1CC(C)(C)C(C(=O)NCCC(=O)NO)C1 c1(C(=O)NCC(CC=C)NC(c2cnn[nH]2)=O)ccc2nn(C)cc2c1 N1(C(C2(CC#C)CCCO2)=O)CCC(NC(=O)Cc2cccc(OC)c2)C(O)C1 C(C(C)CC(=O)NC1C2CC1N(C(=O)C(n1nnnc1C(C)(C)C)C)C2)OC O=C(CC1=CCOCC1)NCC1(F)CCCN(C(c2ccc(C(F)F)o2)=O)C1 Cc1ccc(-c2cc(C(=O)NC(c3nc(C4CC4)n[nH]3)C)n(C)n2)cc1 C1(NC(C2CN(C(CCCCCN(C)C)=O)C(C)(C)C2)=O)CCOC2(CCC2)C1 CN1CCC(C(N2CCCC(N(C(=O)CCN(C)CCO)CCF)C2)=O)CC1 c1(N2CC(C)C(NC(C3CC4(C3)CC4(F)F)=O)CC2)nc2c(cc1Cl)C(=O)OC2 c1(C(=O)NC2CCC2CNC(C2CCS(=O)(=O)N2)=O)cc(Cl)ncc1O c1(OCC)ccc(S(=O)(=O)NCCCC2COCCO2)cc1CC N1(C(Cc2nnn(C(C)(C)C)n2)=O)CCCC(NC(=O)CC2CC23CC3)CC1 C(CCCCC(=O)NC(C1(O)CCCCC1)C(N1CCN(CC)C(C)C1)=O)=CC C12(NCc3ccc(C#C)cc3)CCC(C(=O)NCc3cncs3)(CC1)CC2 c1(C(=O)NCCCN(C)C(c2cccn2C2CCCC2)=O)ccc(N)cn1 C1(NC(C(C)(C2CC2)OC)=O)CCCCCC1NC(C1CCC(=O)O1)=O N1(C(C2CC(NC(C3C=C(C)CS3)=O)C(O)C2)=O)CCCC(N=[N+]=[N-])C1 c1(C(=O)NC2CCN(C(C(CCCC)CC)=O)C2C)ccc(C)cc1[N+](=O)[O-] c1(C(=O)OC)cc(C(=O)Nc2cn[nH]c2)c[nH]1 N1(C(Cc2cnc(C)[nH]2)=O)CC(NC(c2cncc(CO)c2)=O)CC1(C)C O=C(CC(O)C1CCCC1)NCC1(CNC(c2coc(Cl)n2)=O)CC1(F)F c1(C(N2CC(C(=O)Nc3cnc(C)c(Cl)c3)SCC2)=O)c(C)ccc(C)c1O Cc1oc(-c2ccco2)nc1CC(N1CCC(N(C)C(C2OCCC2C)=O)C1)=O Cc1ccc2oc(C(=O)NC(C)(C)CNC(c3cncn3C(C)C)=O)cc2c1 N1(C(Cc2cc(C)[nH]n2)=O)CC(CC(=O)NCc2csc(C)c2)CC1C N1(C(c2ccnc(NC3CCN(C)C3=O)c2)=O)CCC(O)CC(C)(C)C1 c1(CC)ccccc1C(N1CC=CC1CNC(c1conc1COC)=O)=O.C1CC1 C(=O)(C(CC)C(=O)NC1CN(C(=O)Cc2cnoc2)C(C)(C)C1)OCC C1(NC(CN(C(COCC#C)=O)C(C)C)=O)CCCCC1CCC=C N1(C(c2c(N)csn2)=O)CCC(C(=O)CCO)C(F)(F)CC1 c1(N(CCOc2cc(C)cc(C)c2)C)nccc(=NC2CCCC2C#N)[nH]1 c1(C(C2(CCCNC(CSCC#C)=O)CC2)=O)ccncc1NCC1CC1 C(=O)(C1=CCc2ccccc21)NCCC1(CNC(C2CC(=C)C2)=O)CC1 CC1(CNC(C2CC2(Cl)Cl)=O)CCN(C(=O)C=Cc2cncc(F)c2)CC1 C1(C(C)NC(C2CCC2)=O)COCCN(C(=O)C(C)(C)N(C)C)C1 C12=NC=CC(=NCCN1)N2.c1(OCC)ccc(-c2csc(=NC)[nH]2)c(F)c1F c1(-c2ccc(C)cc2)csc(=NCC(C)N2CCN(C(C)=O)CC2)[nH]1 c1(CNC(=NCCC)NC2CCOC(C)C2)cc(F)c(OC(F)F)c(F)c1 c1(C(=O)NCCC(C)(C)NC(CSCCC)=O)ccnc(S)c1 C1(NC(c2cc(CSCC)on2)=O)CN(CC(c2cc(C(C)C)[nH]n2)=O)CC1C N1(C(C2CC(C)C2)=O)CCN(CCO)C(C)(C)C1 Cc1nc(C#N)c(NCCC(N2CCC(C)C(NC(=O)COC(F)(F)F)C2)=O)o1 CC1(C)CCN(C(c2cnccn2)=O)C(C(=O)NCC2COC(=O)C2)C1 N1(C(CC2N(C)CC=CC2)=O)CC2CC1CN2C(C1CNC(=O)O1)=O C(CCC(C(=O)NCCCNC(C)=O)NC(=O)CC1NC(=O)NC1=O)OC c1(C(N2CCC(C(=O)NC3CC(C)C3)C2)=O)csc2ccccc12 CCC(C#N)C(=O)N1CCCC(C(C)(C)C(=O)NCC(N2CCCCC2)C)C1 N1(CC)CC(CNC(=O)CCC2CCCN2C(c2ccc(C)n2C)=O)OC1=O CCC(C)C(=O)C(=O)N(CCCNC(C1(C(F)F)CCCO1)=O)CC CCCCC(O)C(=O)NC1CC2CC(NC(=O)COc3ccc(F)c(Cl)c3)C1C2 C1(C)(NC(C(CC(F)F)N(C(c2cnc(CC)s2)=O)C)=O)CCCCC1(C)C Cc1nc(=N)[nH]cc1C(=O)NC1CCC(CNC(C2CC(n3cccn3)C2)=O)C1 c1(Cn2c(C)ncc2)ccc(NC(=O)C(=O)NC(C)Cc2ccc(Cl)cc2)cc1 O=C(C1CCCc2n[nH]cc21)N1CCC2(CC1)CN(C(C1CCO1)=O)C2 Cc1cc(N2CCCC(OC(=O)N(C)C)C2)nc(N2CCOC(C)CC2)n1 C(=O)(C1=CCCOCC1)N(CCNC(=O)Cc1ccc(F)cn1)CC1CC1 C=C(Cl)CCC(=O)NCc1ocnc1Cn1cc(Cn2ccnc2C)nn1 C(=O)(CCCC(=O)NOC(C)(C)C)N(CCCCNC(c1c(C)sc(O)n1)=O)C c1(CC(N2CC=C(CNC(C3(C)CC3(Cl)Cl)=O)CC2)=O)ccc2nn[nH]c2c1 N1(C(c2c(C)c[nH]c2)=O)CCC(N(C)C(C2C3CCCC23)=O)CC1 c1(C(=O)NCC(=C2CN(C(C3CCC(C(=O)OC)O3)=O)C2)F)cc(=O)cc[nH]1 N1(C(c2cnc(C)nc2)=O)CCC2(CC2C(=O)Nc2ccnc(C(F)(F)F)c2)C1 N#Cc1cc(Br)cnc1NCC1CCCCN1C(c1cnc(CC2CC2)s1)=O CC1CN(C(=O)CC2CC(C)(C)NC2=O)CC(C(=O)O)O1 N1(C(CC(C(=C)C)OCC)=O)CC2(CCN(C(=O)CN3CCC(O)CC3)C2)C1 N1(C(C(C)Cc2cnc[nH]2)=O)CCN(C(=O)C(C)(C)C2CC2)CC12CC2 C12(CC(=O)NC(C3CCN(C(CC=C(C)C)=O)C3)C)CCC(CC1)C2 CC(C)(CCCNC(C1CCSC1)=O)C(=O)NC1CCOC1C1CC1 C1(C(N2CC(C=C)C(NC(=O)Cc3ccoc3)C2)=O)CC(C2CCCC2)C1 Cc1cc(C(N2CCC(CNC(=O)CC3(N(C)C)COC3)C2(C)C)=O)cc(C)c1 C1(CNC(CCCCOC)=O)CC12CCN(C(c1ccnnc1O)=O)CC2 c1(C(C(C(=O)N(C2(C)CC2)C2CC2)N(C(CC#C)C)C)C2CC2)ccc(Br)cc1 N1(C(CCn2ncc(C)c2)=O)CCN(C)C(C(=O)N(C(C)CO)C)C1 Cc1nc2c(o1)CCN(Cc1cc(C)c(C)c(C)c1)C2 N1(C(C)C)CCCC(C(=O)NCC2CCN(C(c3cc(C(F)F)no3)=O)C2)C1 C(C(N=c1nc[nH]n2cccc12)C(C)C)NC(CC1(C=C)CCOCC1)=O C(CCCCC(=O)NCC1(C)CCN(C(=O)CN2CCC(C)C2)CC1)OCC C1(CNC(=O)NC2CC(=O)N(C3CCCC3)C2)CNCCC12CCOC2 C(CN=C(NC1CCC1)N1CCC(CC2CCOC2)CC1)c1cnsc1 C12(CNC(C(C3CC3)OC)=O)COC(NC(=O)CSc3n[nH]c(C)n3)(C1)C2 c1(OCCC)ccc(NC(=O)C(CC2CCC2)NC(=O)CC23CCCC2C3)cc1 c1(C(C)(F)F)cc(C(=O)NCCCNC(C2CSCCS2)=O)ccn1 c1(CCOC)nc(-c2ccc(-n3nc(C)cc3C)nc2)nn1Cc1ccccn1 N1(C(CCC2(NC(=O)Cc3nocc3C(=O)O)CCCC2)=O)CCC(F)CC1 C1(c2n(CC=C)nc(CCC3CCCN3C)n2)CCCCN(C)C1 C1(OCCNC(c2ccnn2CCF)=O)CCN(C(=O)CCCc2cnn[nH]2)C1 C(=O)(C(O)C(C)(C)C)NCCN(C(=O)CC1CC1)C(C)C c1(C(=O)NC(CN(C(C(CC)C)=O)C)C)ccc(OC)c(N)n1 C(C1=CCCN(C(=O)C(C)(C2CC2)OC)C1)NC(CC=CCCCCC)=O N1(C(CCCCCSC)=O)CCC2C(C1)CN2C(=O)C(F)CC1CCOC1 N1(C(=O)NC2C(CC)(CC)C(OC)C2C)CCC(CO)CC1C c1(-n2c(CC(=O)OCC(c3c(C)noc3)=O)nnc2C)ccc(S(N)(=O)=O)cc1 N1(C(=O)NC2CCCCC2n2cccc2)CCC(CO)C12CCOCC2 N1(C(c2cncc(C)c2Cl)=O)CC2CC(NC(c3ccoc3)=O)CC(C2)C1 c1(C(=O)NCCN(C(C2CN3CCC2C3)=O)CC)ccc(C)c(S(N)(=O)=O)c1 CC(C)(C)C#CC(=O)NCC1CCN1C(c1cn(C2CCOC2)nn1)=O C(CCCCCCC(=O)NC1CN(C(c2ccc(C)c(C)c2)=O)CC1OC)SC Cc1ccc(CN2CCC(CCC(=O)Nc3cnnc(O)c3)CC2)cc1F N1(C(C(CC)c2ccccc2)=O)CCCCCC1.C(=O)(COC(C)C)NCC N1(C(C23CC(COC)(OC2)C3)=O)CCCC(NC(C2CCC(F)(F)CC2)=O)CC1 C(CCC(C)NC(C1COC(=O)O1)=O)NC(COCCOCC#C)=O N1(C(COCC=C)=O)CCN(C(=O)Cc2coc(C(F)F)n2)CC1C1CCCC1 C1(C(C)N)CN(C(=O)C(N2CCCC2c2cccc(Cl)c2)=O)CCO1 CC1(C)C(NC(C2CC(O)C2)=O)CCN1C(C1CCCN1S(C)(=O)=O)=O C(=O)(CCCc1nc(C)no1)N(CC(CC)NC(C1CC(CC(=O)OC)C1)=O)CC CCC(C)(F)C(=O)NC1CC(N(C)C(c2ccc(OCC(N)=O)cc2)=O)C1 c1(C(N(C2CCN(Cc3ccccc3)CC2)CC(CC)O)=O)ccc(F)cc1OC C1(C2(O)CCOCC2)(CNC(C(C(C)O)N(C)C)=O)CC1 N1(C(CSCC#C)=O)CC2(CCCCN(C(c3oc4ccccc4c3C)=O)C2)C1 c1(C(=O)OC)ccc(CCC(=O)NC2CC(CNC(c3ccn(C4CC4)n3)=O)C2)[nH]1 C1(NC(C(CC)=CC)=O)CC(F)CN(C(c2ccc(-c3cscn3)cc2)=O)C1 N1(C(C(CC=C)OC)=O)CCCC(O)(CCNC(=O)C(C)CSC)C1 c1(N(N(C)C)C)ccc(NC=O)cc1.C(C(O)CCNC(=O)CO)NC(=O)CC C1(=O)C2=CCC(C2)O1.C(=O)(CC(C)(O)c1ccccc1)NCC(=O)OC(C)(C)C N1(C(CC(=C=C)C)=O)CC2CCCC(N(C(=O)CN(C(=O)C3CC3)CC)C)C2C1 c1(-c2cn(CC(=O)NCc3c(C)nc(C(C)C)cc3)nn2)ccc2[nH]ncc2c1 c1(NC)nc(C)cc(=NCC2CN(C(=O)C(C)(C)O)CC23COC3)[nH]1 C(=O)(CC1=CCOCC1)NC(c1ccccc1Br)C(=O)NCC(CC)n1cccn1 Cc1cncc(CCC(N2CCCC2C2(O)CN(C(=O)COC3CCC3)C2)=O)c1 C=CC(CC)CC(=O)NC1CC2(C1)CC(NC(C1C(C(C)=O)C1(C)C)=O)C2 Cc1cc(C(=O)N(C)CC2CCN(C(=O)CC3CCCC(O)C3)CC2)[nH]c1C CO[Si](CCCN(C)CC1CCOC(CN)C1)(OC)OC C1(C)(CNC(C(CC(C)C)C)=O)CC(F)(F)CN1C(=O)CCC1CCC1 c1(SC)ccc(C(=O)NCC2(O)CCN(C(=O)CC3C=NN(C)C3=O)C2)cc1 C(=O)(C(O)CCCNC(=O)CC1C=CCC1)NCC(CC)C#N N1(C(C2CC(C)(C)OCC2)=O)CCC2(CC1)CC2C(N1CC(CS(C)=O)C1)=O C12(C(=O)NC(C3N(C(C(CC#C)O)=O)CCC3)C)CCN(CC1)CC2 N1(C(c2cc(C(C)=O)sc2)=O)CCC2(CCC(NC(=O)C(O)C(F)F)CC2)C1 C12(NC(C(C3CC3)OCC)=O)COC(C1)C(NC(=O)Cc1cc(Cl)cnc1C)C2 C(=O)(C#CC1CCOC1)NC(CC=C)CC(F)F.C12CCCN1C2=O c1(C(=O)NCC2N(C(CC3ON=C(CC)C3)=O)CC(O)C2)cc2c(C)cccc2o1 C1(NC(c2n(CC)nnc2)=O)CN(C(=O)C=CC=C(C)C)C(C)(COC)C1 C1(C(N2CCC(O)(CNC(c3ncc(C(F)F)s3)=O)C2)=O)CCCC2(CCC2)C1 c1(CC)ccc(C(=O)NCC2(O)CC(C(=O)OC)C2)c(F)c1F.n12cc(nn1)C2 c1(CC(N2C(C)(CNC(c3ncc(OC)nc3)=O)CC2)=O)c[nH]c2ccccc12 C=CC1(CC(=O)NC2CCC2N(C)C)CN(C(C23CSCC2C3)=O)C1 CC1CCCC(C(N2CCC(OCCNC(C3(O)CC3)=O)CC2)=O)CC1 c1(C(N2CCC(CCNC(Cn3c(=N)[nH]nc3)=O)C2)=O)ccc(O)nn1 C1(NC(C2CC(C(C)C)C2)=O)C2CCC1N(C(c1ccc(=O)n(C)c1)=O)C2 c1(C(N(C2CCN(C(COCCC=C)=O)C2)C)=O)cc(C)c(CC)nc1O C(=O)(C(O)CC(N)=O)NC1CC(C)(NC(c2ccc(CCNC(C)=O)cc2)=O)C1 N1(C(C2ON=C(CC)C2)=O)CCC(C)C(NC(=O)Cc2ccc(CO)c(C)c2)C1 N1(C(c2cnc(OC)nc2C)=O)CCC2CN(C(C3CC(SC)C3)=O)CCC12 CCCCCCC(=O)N1CCN(C(C23CC2COC3(C)C)=O)C(C2CC2)C1 c1(NC(C2(CC)CCCO2)=O)cccc(NC(c2cc(F)n(C)n2)=O)c1 Cc1ccn2ncc(C(=O)NCC34CC3CN(C(=O)C(F)(F)CO)C4)c2c1 c1(OCC(=O)NC2CC(OC)CN(C(C(CSC)C)=O)C2)cccc([N+](=O)[O-])c1 c1(C(N(CCC(C)NC(CN2CC(C)C2)=O)C)=O)cnnn1C1CC1 c1(C(=O)NC(C(C)(C)C)CNC(=O)Cn2cccc2)cc2ccsc2s1 c1(C(N2CC(NC(C(C)P(C)(C)=O)=O)C(O)C2)=O)ccc2c(c1)CCN2C C12(CNC(C3(C)CCCCO3)=O)CCCCC1N(c1ncccn1)CC2 S(=O)(=O)(c1cc(C)ccc1C)NCC(=O)NCCN(C(CC1C(OC)CC1)=O)C C1(NCCOCC#C)N(C(=O)C(C)OCC=C)CCCC1(C)C c1(C(N(CC(C)NC(c2nc(OC)ccc2Cl)=O)CC)=O)nccc2[nH]ccc12 N1(C(CCC(C)C)=O)CC(C(N2CC3CC2CC3CF)=O)CCC1(C)C C1(NCC(CC)CC)CNCC12CC2 CC(C)CC(O)C(=O)N1CC(C)(NC(C2CC2C2CCC2)=O)C1 Cc1nc2ccc(C(=O)NC(C)(C)CNC(=O)CC3CCNC(=O)C3)cn2n1 C1(F)(C(N2CCC(CN(C(c3c(CC)cncc3)=O)C)C2)=O)CCC(C)CC1 c1(C(N2CC3CCN(C(=O)C4=CCS(=O)(=O)C4)C3C2)=O)cccc2c1CCO2 C(=O)(C(C)C(C)C(C)(C)C)NCCC1CN(C(CCc2c(C)n(C)nc2)=O)C1 O=C1CCC(CC(N2CC(F)(CNC(=O)CN(C3CCCC3)C)C2)=O)CN1 c1(SC)ccc(CN2CCCC(C(=O)NC3CONC3=O)C2)cn1 C(=O)(CCCN=[N+]=[N-])NCC1(C(N(C(C2(C)CC2)C)C)=O)CCC1 c1(C(N2CC(NC(c3c(C)ccc(Cl)c3)=O)C(O)C2)=O)ccnc2c1CC(=O)N2 N1(C(c2n(C)c(S)nn2)=O)CC(CNC(c2ccc(Cl)o2)=O)C2(CCOCC2)C1 c1(C(N(C2CCCC(NC(C(C)=C3CC3)=O)C2)C)=O)ccc2sccc2c1 c1(C(N(C2CCN(C(c3nn(CC)c(O)c3)=O)C2)C)=O)cc(Cl)c(OC)cc1Cl C1(CCC)CN(C(=O)C2=CCCC2)CCN1C(=O)Cc1csc(S)n1 N#CCCCCC(=O)NCC1CCC(NC(=O)C(F)=CC2CC2)C1 c1(OC)cc(C(=O)NC2CCN(C(=O)CC3CC3C)CC2)c(C)c(Br)c1 C(C1CCN(C(C2CCSC2)=O)CC1)=CC(=O)N(CC(C)O)CC(C)O CCC(C)CCCC(=O)N1CC2(CCCC2)C1C(=O)NCC12CCC(CO1)C2 N1(C(C(C)(C)OC)=O)CCC(NC(=O)C(c2cnn(C)c2)C)C(CO)CC1 N1(C(CNC(=O)OCC)=O)CC(C)(CNC(C2CCC2)=O)CC1(C)C Cc1cc(C(c2nnnn2CC(F)F)NCc2cc(Cl)cc(Cl)c2)cc(C)c1Cl c1(CNC(C)=O)ccc(C(=O)NCC2CCN2C(=O)CN(C)C(=O)C2CC2)o1 C1(C2(O)CCOCC2)(C(=O)NCC2C(CNC(c3cnccc3Cl)=O)C2)CC1 Cc1ccc(C(=O)N(C)CC2(O)CCCN(C(C3CCC(F)CC3)=O)C2)cc1Cl c1(CC)ccc(N)c(C(=O)N(CC(CO)(CO)NC(=O)CN2CC(C)C2)C)c1 c1(CNC(CC2CCC(C)C2)=O)ccc(CCNC(=O)C(C)(C)CC2CC2)cc1 Fc1cc(N2C(=O)NC(Cc3ccccc3)C2=O)cc(F)c1F.C1CC1 C1(C(N(CCNC(COC)=O)C2CC2)=O)CCN(Cc2cccnc2)CC1 C1(NC(CN(C2CC2)CC)=O)CCN(C(=O)C(C)(F)F)CC1 Cc1cnc(C)c(NC(=O)C(=O)Nc2ccccc2N(C)Cc2ccncc2)c1 CCC(C)C(O)CC(=O)N1CCC(CC)(NC(c2cc(Cl)n(C)n2)=O)CC1 C1(C(=O)NCCCCNC(c2cc(C)nnc2)=O)CCC(S(N)(=O)=O)CC1 Cc1cc(C(=O)Nc2cc(Br)nn2-c2ccccc2)nn1-c1cccc(Br)c1 C1(C(N2C(C)(COC)CC2)=O)Cc2ccc(Br)cc2C(=O)O1 N1(C(C#CC2(C)COC2)=O)CC(C2CCCN(C(C3C4CCCOC34)=O)C2)C1 N1(C(c2c(C)ccs2)=O)CCC(CO)C(NC(c2oc(CO)cc2C)=O)C1 N1(c2snc(SC)n2)CC2CCC(NC(c3c(C)noc3C)=O)CC2C1 CC(C(=O)N(C)CCN(C)C(c1cc2n(c1)CCSC2)=O)C(F)(F)C(F)F CC1(C2CCCN(Cc3cccc(-c4ncccc4C(=O)O)c3)C2)COC(=O)N1 c1(COC)cccc(C(c2ccccc2Cc2nn[nH]n2)O)c1 C(=O)(C1=CC2(CCOC2)C1)NCC(C1CC1)NC(=O)COc1cccnc1 CCCC(C(=O)OC)C(=O)NCC1CCC1NC(C1(Cc2cccnc2)CC1)=O c1(C(=O)NC(C2CCCCC2)CNC(=O)CCc2ccc[nH]2)nccc(Cl)c1F Cc1noc(C)c1CNC(=O)CC1CCN(C(=O)CSc2ccccc2)C1 c1(OC)ccccc1C(=O)NC1CC(NC(=O)Cc2c(C)noc2Cl)C(O)C1 N1(C(CCOCC)=O)CCCC1C(=O)NC1CSCSC1 N1(C(CC(C=C)C)=O)CCC(C2CC2)(CNC(=O)Cc2cccc(Cl)c2F)C1 C12(CC(=O)NC(CN(C(C(C)SCc3ccccc3)=O)C)C)COC(CF)(C1)C2 C(=O)(C1=CCC(C)CC1)N1CCC(C(C(N2CCCC(CC)CC2)=O)(C)C)C1 C1(C(N2CCC(C(C#C)C)CC2)=O)CCN(C(C2C=CC=CC=C2)=O)C1(C)C c1(C(C(N2CCCC(NC(c3c(CC)occ3)=O)C2)=O)=O)cc(F)cc(Cl)c1 c1(CC(=O)OCC(CCC(c2ccccc2)NC(C)=O)=O)cn2ccsc2n1 Cc1oc(C(C)(C)C)cc1C(N1CC(CNC(=O)Cc2nnc(O)s2)C2CC12)=O C12(C(=O)NCCN(CCO)CC)CCC(NC(c3cnc(Cl)cn3)=O)(CC1)C2 CCC(O)C(=O)NC(C(=O)NCCCc1nncn1C)c1ccco1 C1(NC(COc2cccc(CC)c2)=O)CN(C(=O)Cc2csnn2)CC(F)(F)C1 C1(CS(N)(=O)=O)CCCN1Cc1ccc(-c2ccccn2)o1 N1(C(CCOCC#C)=O)CCCC1C1CCCN1C(c1cnc(COC)cn1)=O N1(C(CSCC(=O)OC)=O)CCC2CCCC12CNC(c1cnc(S)[nH]1)=O N1(Cc2cn(C)nn2)CCOCC1C(N1CCC(C(=O)N(C)C)CC1)=O c1(OC)ncc(Cl)c(C(N2CCC(NC(C3CCCC3(C)C)=O)CC2)=O)c1Cl CC1CCN(C(c2cc(CO)[nH]n2)=O)CC1CC(=O)NCCCc1ncn(C)n1 c1(CC(C(=O)NCCC(C)N(C(C=C2CCC(C)C2)=O)C)=O)cccc(Cl)c1 C1(COC)(NC(C2CNC(=O)C2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1 S(=O)(=O)(c1cnc(NC2CC2F)c(Cl)c1)N1CCC(CC(N)=O)CC1 O=C(CC1NC(=O)c2ccccc21)NCC#CCNC(c1cnc(Cl)s1)=O C1(NC(C(C)Oc2ccccn2)=O)CC2CN(Cc3cc4n(n3)CCSC4)CC2C1 Cc1nccc(C(=O)NCC(C)(C)OCC(=O)NCC2CCCS2)c1C C1(NC(C(=O)NC(C)C)=O)CCC(C)N(C(=O)CC2CCC(C)(C)CO2)C1 c1(C(C)NC(C2CC2c2c(F)cccc2F)=O)c(F)ccc(Cl)c1F c1(C(=O)NCCN(CCC)C(C2CCCC2C)=O)cnc2cccnn12 Cc1nc(C)c(C(N2CCC(CO)(NC(=O)CCC3(O)CCC3)CC2)=O)nc1C C(CC(CO)C(C)C)NC(CC=CCCCCC)=O.C12CCCC1C(=O)NC2 Cc1nc2c([nH]1)C(C(=O)NC1CCCC1NC(=O)CN(C)CCO)CCC2 C1(NC(C2CCOC2)=O)CCN(C(=O)C2=CCCC2)CC12CCC2 N1(C(C=Cc2ccc(C3C(C)C3)o2)=O)CC2CC(C1)C2NC(=O)C(O)C(C)C c1(C(N2CC(CNC(CSCC)=O)C2)=O)cc2ccccn2c1 N1(C(CNC(CNC(C)=O)=O)=O)C2CCC1CN(C(=O)Cc1ccsc1Cl)C2 C1(NC(c2c(C)ccnc2)=O)CCCCN(Cc2nc(C(C)(C)C)n[nH]2)C1 C1(CNC(c2cccc(C)c2)=O)CCCC2CN(C(=O)CC3CCCO3)CC12 N1(CCCOCCNC(Cn2c(C)ccc2C)=O)CCN(C)C(=O)C1C c1(C(=O)NC2(CCCNC(C(C=C=C)C)=O)CC2)cccc(CC)c1F N1(C(C(CC2CN(C(c3c(CC)nns3)=O)C2)F)=O)CC2(C1)CC(C)(F)C2 N1(C(CC2CCC(C)C(=O)N2)=O)CC2=C(C1)CN(C(c1[nH]nc3ncccc13)=O)C2 N1(C(c2nc(C)sc2)=O)CC2CC2(C(N2CCOCC2C2CC2)=O)C1 C1(NC(c2cnn(-c3ccccc3)c2Cl)=O)CCCN(C(=O)Cc2cncs2)C1 N1(C(C(CCF)NC(c2ccc(O)nc2)=O)=O)CC2CCC1C(O)C2O c1(C(=O)OCC)ccc(S(C)(=O)=O)cc1[N+](=O)[O-].C1CCC(=O)N1C(C)(C)C N1(C(c2scc(OC)c2OC)=O)CC2COCCC2(NC(c2cnc(Cl)s2)=O)C1 C1(NC(C(C#C)(C)C)=O)CCC2CN(C(=O)CC(O)c3ccccc3)CC2C1 C1(NC(C(C(CC)C)C)=O)CCC2CN(C(=O)Cc3ccc(F)c(F)c3)CC2C1 c1(CN2CC(CC(=O)Nc3c(CC)c(Br)ccc3)C2)c(O)cc(Br)cc1F C(=O)(C(C)C(C)(C)C)NCC(CCNC(CCCN(C(C)C)C)=O)O C1(NC(C(CC)N(C)C)=O)CC2(CCN(C(C3CCOC3)=O)C2)C1 C(=O)(CC(CC)CCCC)NCCC(CNC(C1(C)CC(=C)C1)=O)OC Cc1cc(F)c(C(=O)NCC2CN(C(c3cocn3)=O)CC(C)(C)O2)c(F)c1 CC1(CNC(=O)CC(C)C2CC2)CCCN(Cc2cccc(O)c2Cl)C1 C1(CC(=O)NCCN(C(=O)CC2(C(F)(F)F)CCC2)CC)CCC(=O)C1 c1(CN2C(C(=O)Nc3cncc(O)c3)CC(C)C2)ccc(Br)cc1C(=O)O c1(OC)cccc(Br)c1C(N1C2CCC(C2)C1C(N1CCOC(=O)C1)=O)=O C1(C(N(CC(COCC)O)C)=O)CCCC(NC(c2cccnn2)=O)C1 C1(NC(c2csc(Br)c2)=O)CC(=O)N(C2CN(CC(O)Cn3cccn3)C2)C1 CC(C)(C#N)CCCC(=O)NCCCC(O)C(=O)NCc1cc(C2CC2)on1 C1(CCNC(CC=CC)=O)CN(C(=O)C(O)CCC)CCS1(=O)=O c1(C(N2CC(CC=C)(OC)C2)=O)cnc(F)c(F)c1.c12oc(C)nc1CNC2=O Cc1ccc(C)c(C(=O)NC2CCOCC2C(=O)NCc2c[nH]nc2C)n1 CCC(C(=O)NCC1C(C)CCN1C(c1cc(O)nc(O)c1)=O)C(C)O C(CC(F)F)(C(=O)N(CCCCN(C)C)C)N(C(CC(CC)C1CCC1)=O)C Cn1nc(C(N2CCNC(=O)C2)C(=O)NCCNC(=O)CC2CCOC2)cc1I N1(C(C2CC23CCCCC3)=O)CCCC12CCN(C(C1CC(CF)C1)=O)C2 C1(CC(=O)NC2CC2NC(c2ccc([N+](=O)[O-])cc2)=O)CCC2(CCC2)CO1 n1(CCC)[nH]c(=NC(=O)C(F)(F)C(F)Cl)cc1C c1(C(N2CC(CN(C(c3n[nH]c(C)c3C)=O)C)OCC2)=O)cc2cnccc2[nH]1 c1(OC)c(C(N2CCN(C(=O)CC(c3c(C)noc3C)C)CC2)=O)c(C)nn1C C1(CNC(c2cc(C)ncn2)=O)CN(C(=O)CCc2cscn2)CCC12CCC2 C(=O)(C1=C(Cl)CCC(C)C1)NC1C2C(CNC(C(=O)N(C)C)=O)C3C(C2)C13 CCCC(C)CCCC(=O)N(CCCNC(c1c[nH]c(=N)cc1C)=O)CC CC(C(=O)NCC(C1CC1)NC(c1cnc(-c2ccccc2)[nH]1)=O)C(C)(F)F c1(C(=O)NCC23C(NC(c4c(C)nn[nH]4)=O)CC(CC2)C3)ccn2c1CCCC2 CC(C)(C)C1=CCC(C(=O)OCCCOCC(O)C(C)(C)C)CC1 c1(-c2cccc(CNC(C3(c4ccc(F)cc4)CC3)=O)n2)ccc2c(c1)NCCO2 C1(NC(CC=CC=C)=O)CC(=O)N(C2CN(C(=O)CCc3cnccn3)C2)C1 N1(C(=O)COCCO)CC2OCCN(C(C3(c4c(Cl)cccc4Cl)CC3)=O)C2C1 c1(C(=O)NC(CNC(C(C(CC)O)C)=O)(C)C2CC2)ccc(C)c(C)c1Cl c1(CC)cc(C)c(C(=O)NC2(CNC(c3cc(C)co3)=O)CCOC2)o1 c1(NC(N)=O)ccc(Cl)c(C(=O)NC2CCC23CN(C(=O)C2=CCCCO2)C3)c1 N1(C(C2CC(C)SCC2)=O)CCC2(CCCN2C(=O)CNC=O)C1 CC(CC(=O)NC1(C2CCC2)CC1)C(C)(C)NC(=O)C(C)CC1CCCC1 N1(C(c2ccn(C3CC3)c2)C(=O)NCC)CCC(NC(c2csc(C)n2)=O)CC1 c1(C(N2CCCC2CF)C(=O)NCC2CCOCC2)ccccc1Cl N1(C(C(CC)C2CCOCC2)=O)CCCC(C2CCN(C(=O)COC3CC3)C2)C1 c1(C(=O)NCC2CC(NC(Cc3n[nH]c(=N)s3)=O)C2)cc(O)nc2ncccc12 c1(C(=O)NC2C(CNC(c3cc(COC)on3)=O)C2)nc(C)sc1C c1(C(=O)NCC2CN(C(CC(=O)NC3CC3)=O)CC2O)cnn2ncccc12 C1(NC(=O)OC(C)(C)C)CC(NCc2oc(C(=O)O)cc2C)C1(C)C C1(C)(C(=O)NC(COC)CCO)CN(C(=O)C(C)NC=O)C(C)(C)C1 c1(OC)cc(C(C)NC(C2CCCNC2)=O)cc(OC)c1OC c1(CC(=O)N(CC(C)O)CCNC(C2C(OC)COC2)=O)c(C)ncnc1C CCCC(CCNC(C1CCN(C(=O)C(CC)OC)C1)=O)C1CC1 CCCC(C)CC(=O)N1CCC(N2CC(C)(CNC(C3CCSC3)=O)C2=O)CC1 C#CC1(OCC(=O)NCC(C)N)COC1.C1(=O)CCOCC1.C1CO1.OC c1(C(=O)NCC2N(C(c3cnn(C(C)C)c3N)=O)CCCC2)ncc(F)cc1F N1(C(c2c(C)nc(OC)s2)=O)CC2CN(C(c3cc(C)n(C)n3)=O)CCC12 N1(C(C=C(C)C(C)(C)C)=O)Cc2[nH]nc(C(N3CCC(C)(F)C3)=O)c2C1 Cc1cc(Cl)ccc1N(C(C)C(=O)O)C(N1CCN(c2nccn2C)CC1)=O C12(C(N3CC(CNC(c4ccnc(OC)n4)=O)C3)=O)CCC(C)(C(=O)O1)C2(C)C CCC(C)(COC)C(=O)NCC1CCN1C(=O)CC=CCc1ccccc1 CC1CN(C(C2CC3(C2)CC(F)C3)=O)CCC1CNC(=O)C(C)(C)C#N C1(NC(C(c2cncn2C)N(C)C)=O)CCN(C(c2n[nH]c3c2COC3)=O)C1(C)C CCC(C(=O)N(C(C)CNC(c1cnc(O)c(F)c1)=O)C)C(C)(C)CC c1(NC(=O)NC2(c3cccc(F)c3)CC2)cccc(F)c1Br N1(C(C(C)NC(c2cscc2Cl)=O)=O)CCC(C2CCC2)CC1 N1(C(=O)NCC(c2ccc(OC)c(OC)c2)C)CCC2(CC1)CN(C)C2 c1(C(=O)NC(C)C(C)(C)NC(=O)C(CO)N(C)C)c(Cl)nn(C)c1Cl C1(NC(=O)CSC(F)F)(CO)CN(C(=O)C=CC2CCCO2)C1 c1(CN(C(CC)Cc2ccc(C(F)(F)F)cc2)CC)ccccc1-c1ccccc1 c1(NC(CNS(CC(C(C)C)N(C)C)(=O)=O)=O)nc(Cl)c(=O)n(C)c1N N1(C(CCCCC(=O)NC)=O)CC(C2CCCN(C(C3CCNC(=O)C3)=O)C2)C1 C12(CCCCC1C)C(=O)N2.C1(C(=O)OC)(NCC(C)COC)CCC1 c1(C(C(=O)NC(CCC)C(=O)NC)NC(=O)CC2CC(=O)C2)ccc(Cl)cc1Cl c1(N(C(C)C)C)nnc(-c2ccccc2Cl)n1CCCN1CCOCC1 CN1CCCC2CN(C(=O)C(=O)NCC(=C3CCCC3)F)CCC12 N1(C(CCOC(C)=O)=O)CCC(O)(CN(C(C2CC2c2ccccc2Cl)=O)CC(C)C)C1 CC1(C)C(CNC(C2CC2C2CC2)=O)CCN1C(=O)CCN1CCCCC1=O O=C(C1=NOC2(CCOC2)C1)NC1CC(C2CCN(C(C3SCCS3)=O)C2)C1 c1(C(=O)NC(CN(CCCC)C)C)cc(NC(=O)COC)ccc1OC N1(C(C2CCC(N(C)C)CC2)=O)CC(C(=O)OCC)CC(CC)C1 C1(NC(N2CCCC(C(C)N)C2)=O)CCc2nnsc2C1 N12CCC(CC1)C2=O.c1(SCCNC(C2C(Cl)(C(=O)OC)C2)=O)ccc(Cl)nc1 c1(C(N2CCC(NC(CCCc3nc(C)sc3)=O)C2C)=O)ccc([N+](=O)[O-])cc1 C1(C)(CC)CCC(N=c2[nH]c(N3CCNC(=O)CC3)nc3c2CCC3)CC1 c1(OC)cc(C)c(C(=O)NC2CCC2NC(c2ccoc2C)=O)cc1OC CC1=C(C)CC(C(=O)NC(C)CCCNC(=O)CCCn2ccnc2C)CC1 c1(C(C)(C)C)ccccc1C(=O)NC1CCCN(C(=O)Cc2coc(C(F)F)n2)C1 C(=O)(C#CC1(C)CCCO1)NCC(CC)NC(=O)Cc1ccc2scc(C)c2c1 C1(C(N2CC(CN(C)C(C34CCC(C3)OC4)=O)C2)=O)CCCC2CC12 c1(C(N(CCN(C(c2cc(C(=O)OC)sc2)=O)C)C)=O)c(C)c[nH]c1CC(N)=O c1(C(=O)NC2CCN(C(C(C)(C)OCC)=O)CC2CC)cccc2nn[nH]c12 c1(C(N(CC(=O)NC(c2n(C)ncc2)C)C2CCC2)=O)ccc([N+](=O)[O-])[nH]1 N1(C(C2(CCC)CC2)=O)CC2(CCC(CNC(=O)CCc3ccccc3)O2)C1 Cc1cccc2oc(=NCCCNC(=O)C(CCN(C)C)N(C)C)[nH]c12 c1(OC)ncc(Cl)c(C(=O)NCC(O)CN(C)C(c2ccnnc2)=O)c1Cl c1(OC)cc(C)c(C(N2CCC(CNC(=O)CCCC#N)(OC)CC2)=O)cc1Cl N1(C(C(CC)C2CCC(=O)N2)=O)CC2(CCN(C(=O)C3=NOCC3)CC2)C1 C(=O)(CP(=O)(C(C)C)C(C)C)N(CC(CC)NC(=O)CCNC(=O)CO)C C(C(CNC(=O)Cc1ccsn1)CO)NC(C1CC(SC)C1)=O N1(C(C(CC=C)CC)=O)CCCC2(CCCN2C(=O)COCC(C)(C)C)C1 C(=O)(CP(C)(C)=O)N1C(C(=O)NC(c2ccc(NC(C3CCCC3)=O)s2)C#C)CC1 N1(C(C(CC#C)C)=O)CCC2(CC1)CC(NC(c1nn(CC)cc1[N+](=O)[O-])=O)C2 CN1CCC(c2cn(CC3CCCN(C(=O)CSc4nccn4C)C3)nn2)CC1 c1(CNC(c2occ(C)c2)=O)cccc(C(N2CCCC(OC(C)C)C2)=O)n1 C1(CC#C)(C(=O)NCCC2(O)CCC2)CCC1.C12(CCC1)C(=O)N2 c1(-c2ccc(C#N)s2)ccn2ncc(C(=O)Nc3cc(Cl)ncc3F)c2c1 N1(C(CCC)=O)CC2(C1)CN(C(=O)C#CC1CCOC1)CCO2 CCC(C)S(=O)(=O)Cc1nnc(N2CCC(c3nc[nH]n3)CC2)n1CC1CC1 C1(NC(c2ccc(C)[nH]2)=O)CCCC12CN(C(C1CC3C(C1)C3(F)F)=O)C2 c1(CN(C)CC2(O)CCCN(C(C3CCCOC3)=O)C2)nc2ccccc2o1 C(CCC)(C(O)C(=O)N1CCCC1CNC(C)=O)NC(C(C=C)O)=O C1(C(C)NC(c2cc(C3CCOCC3)on2)=O)CN(C(=O)C#CC2CC2)CCO1 C1(C)(OC)CN(CC(=O)NCCC2(C(=O)NC(c3nccn3C)C)CCC2)C1 c1(C(N2C(C)CCC(CNC(C=CC)=O)C2)=O)cc2cncn2c(O)n1 Cc1cc2[nH]c(=O)c(C(N3CCC(CNC(c4n[nH]c(C)c4C)=O)C3)=O)cn2n1 CC1CN(C(=O)C#CC(C)(C)O)CCN1C(C1CCOC(C)(C)C1)=O c1(OC)ccc(C(N2CCC(CS(N)(=O)=O)C2)C(=O)NCC2CC2)c([N+](=O)[O-])c1 c1(CCSC)cn(CC(F)CCNC(=O)C(C)(C)Cl)nn1 Cc1cn2cc(C(=O)NCC3CCN(C(=O)Cc4cn[nH]c4)CC3C)sc2n1 C1(NC(COCCC=C)=O)CCN(C(c2sccc2C2CC2)=O)CCC1CO CCC(C(=O)N1CCCOC(CCNC(c2cccc(CO)c2)=O)C1)C(C)(F)F C1(C(C)C)C(NC(=O)C=CC2CCCCC2)CCN1C(C1CC12CC(O)C2)=O c1(C(=O)NCC2CCN2C(=O)C(O)C2CCC2)occ2c1CCCC2 C(=O)(CCCCC(C)(C)C)NC1C=CCC(C(N(C2CC2c2ccco2)C)=O)C1 C1(C(N(c2ncccn2)CCCC)=O)CC(F)(F)C12CCC2 C=CCCC(=O)NC.c1(CCC(=O)NCC)nc(-c2nc[nH]n2)no1.C12(CC1)C(C)C2 c1(C(C)=O)ccc(C(N2CCC(C)C(NC(=O)C(O)C3CC3)C2)=O)c(F)c1 Cc1ccc2nc(C(=O)NCC(CO)NC(c3c(C)cncc3C)=O)cn2c1 c1(CC)nc(N2CCN(C(=O)CC3CCCS3(=O)=O)CC2)cc(C#N)n1 c1(NC(C2CCN(C(c3n(C)ncc3)=O)CC2O)=O)cccc2c1CNC2=O C1(NC(CS(C)(=O)=O)=O)COC2CN(C(=O)CCCCc3ccccc3)CC12 N1(C(c2ccc(OC)c(OC)c2Br)=O)CCCC2(C1)CN(C(=O)C(C)S)CCO2 N1(C(C2C(C)(CC)C2)=O)CCCC(C)(C)C1CNC(C1CNC(=O)N1)=O n1(CC(N2CCCC(NC(CC(C)OC)=O)C2)=O)ncc(C#N)c1Br N1(CC(C)NC(=O)CN2C(=O)C(=O)N(C)C2=O)CCC2(CCN(CC3CC3)C2)C1 C1(C(=O)NCCC2(C(=O)NC(c3cncs3)C)CC2)CCCN1C1CC1 N1(c2ccnc(N3CC(C)C(O)C(C)C3)n2)CCc2c(CO)nn(C)c2C1 C(=O)(C1=CCSC1)N1C(CNC(C2CCC(C)C2)=O)CCC1 N1(C(C2N(C(C)=O)CSC2)=O)CC(NC(c2ccc(C)cc2F)=O)C(F)(F)C1 CC1CN(C(c2cccnc2)=O)CC1NC(=O)CNC(C1CC1(C)C)=O C(C(C)(CC(C)C)NC(=O)C=CC1CCCN1C)NC(CCN(C(C)=O)C)=O CC#CCCC(=O)NC(C1(O)CCN(C(c2oc(C)nc2C(F)(F)F)=O)C1)C C1(CCNC2CCC(CC(=O)NC(C3(O)COC3)=O)C2)CC2CCC1O2 C1(C(N2CCC(NC(c3cnc(C)o3)=O)C2)=O)CC(=O)N(CC(F)(F)F)C1 Cc1c(Cl)nc[nH]c1=NCC1CC(c2cc[nH]n2)C1.N1(C2C(=O)N2)CCCCC1 N1(C(C(C(C)C)SC)=O)CCC(C2CN(C(=O)COCC(C)(C)C)C2)C1 c1(COC)ccccc1SC(C)C(=O)NC(=O)OCC(C1CCCO1)=O c1(C(=O)OC)cnn(C2CCN(Cc3cccc(-c4ccnn4C)c3)CC2)c1C C1(NC(CSCC)=O)CCCCC12CCN(C(c1cc3nnn(C)c3s1)=O)CC2 C1(CNC(C=COCC)=O)CCN(C(c2ccc(C(N)=O)nc2)=O)C1(C)C C1(C(=O)NCC2C(NC(=O)Cc3cocn3)C2)CCCN(c2ccc(Cl)nn2)C1 N1(C(Cc2c(C(C)C)con2)=O)CC2CC(NC(c3n[nH]c(O)n3)=O)C2C1 Cc1cnc(S(C)(=O)=O)nc1N(C1CC1)Cc1ccc2c(c1)CNC2 c1(C(=O)NC(CN(C(=O)CC2CCCS2(=O)=O)CC)C)cc(C(N)=O)ccc1F N1(C(CCNC(C)=O)=O)CCC(C=CC(=O)NC(C)C(C)n2cncn2)CC1 N1(C(Cc2cc(C)c(O)cc2)=O)C2CCC1C(C)C(NC(c1ncn(C)n1)=O)C2 c1(C(N2CCCN(C(C3C(CC)CCO3)=O)CC2)=O)csc2c1CCCC2 C1(CC(=O)NCCCOCCC(N2CCC(=C)C2)=O)CCC(C)(C)C1 C1(NC(c2ccccc2)=O)CCN(C(c2cnnc(O)c2)=O)C12CCCC2 C1(C(C)C)CC(O)CN1C(C1COCCC1NC(=O)C(C)(C)C1CCC1)=O c1(C(=O)NC2(C)CC(NC(=O)CO)C2)ccc(F)c(C(F)(F)F)c1F C1(N(C)CC2CC2)CCCN(C(=O)CC2C3CN(C(C4(C5CC5)CC4)=O)CC23)C1 CC1CC(=O)NC(C(=O)NCC2(O)CN(C(=O)CNC(c3ccccn3)=O)C2)C1 c1(NC(CNS(C)(=O)=O)=O)ccc(C(F)(F)F)cc1F.C(N)(=O)N CC1CN(C(=O)CCSCC(N)=O)CCC1NC(C1CCCCS1)=O CC1(C)CNC(=O)c2cc(C(N3CCOc4c(Cl)cc(Br)cc4C3)=O)ccc2O1 C1(NC(CCC=CC(C)C)=O)CCN(C(=O)CSc2nc[nH]n2)CC1O C1(OC)CCCC1C(=O)NCC1CCN1C(=O)C(=O)C1CCCC1 C(C(F)C(=O)NC(C)(C)CCNC(c1cnn[nH]1)=O)N(CC)CC C1(CC(=O)NC(CNC(COCCCCOC)=O)CO)CC2CCC1C2 C(CCCCNC(=O)C(CC1CC1)NC(=O)C(N1CCOC1=O)C)SC C(C)(C(=O)N1CCC(NC(=O)CCc2cccs2)C(CO)C1)(C(C)C)OC C(=O)(CS(C)(=O)=O)NC(c1ccco1)C.C1(=O)CO1 Cc1cc(=O)oc(C)c1C(=O)NC1CN(C(=O)Cn2nccn2)CC1S(C)(=O)=O C#CCC(O)C(=O)NCC1COCC1NC(=O)CC1CC(=C)C1 C1(SCC)C(NC(C2(C)CC2C(=O)OC)=O)CCN1C(=O)C1=COCC1 N1(C(C2(C)CC2F)=O)CC2(CCN(C(c3ccc4c(N)nccc4c3)=O)CC2)C1 N1(C(C(CC2CCC2)OC)=O)CCCC(C)(CNC(=O)CN(C(=O)C(C)C)C)C1 C(=O)(C(C(C)C)c1ccc(Cl)cc1)NCC1CCN(C(CC=C)=O)C1 C1(OCC)(CNC(CC2CN(C(C3C4CCCC34)=O)C(C)C2)=O)CCCCCC1 CCC1=NOC(C(=O)NC2(C(=O)OC)CN(C(=O)C(C)NC(=O)C(C)(C)C)C2)C1 c1(CNC(c2cc(F)ncc2NCc2cc(O)cc(F)c2)=O)cc(Cl)cc(Br)c1 C=CCCCCCC(=O)NCC1CCN(C(c2cc(SC)c(Cl)cc2Cl)=O)C1 c1(OC)ccc(NC(C23CC2CN(C(c2cccc(C)c2)=O)C3)=O)c(C)n1 C=CC1(C(=O)NCc2ncc(CC)o2)CCN(C(=O)CCc2nccs2)C1 c1(N2CCC(NCC3N(Cc4nnc(C)s4)CCC3)C2)ccc([N+](=O)[O-])cn1 c1(C(=O)NC(c2nc(C)no2)CC)cccc2nc(O)n(C)c12 N1(C(C(C(C)C)=O)=O)CCCC(C2(NC(=O)C=C3CCN(C)CC3)CC2)C1 N1(C(C2CC(NC(C3CCCO3)=O)C2)=O)CCC(Oc2ccccc2Cl)CC1 c1(OC)cccc(CSc2nc(Cc3cnn(C)c3)nn2-c2ccnnc2)c1 c1(CC)ccc(C(=O)NC2CC(NC(C3(OC)CS(=O)(=O)C3)=O)C2)cc1F n1(CCC)ccc(C(C(=O)NCCC2CC2)N(CCC(C)OC)CC)c1 N=c1[nH]c(N2CCCC(N3CCCC3=O)CC2)nc2c(Br)c[nH]c12 N1(C(C2CCC3(CCC3)CC2)=O)CC2CCCC(C1)N2C(C1CCCC(F)C1)=O c1(C(=O)NCCC(=C)CNC(C2(SC)CCC2)=O)cc(F)ccc1N c1(N2C(C3(NC(=O)C=Cc4cocn4)CC3)CCC2)ncnc2[nH]cnc12 c1(CN2C(C(N(CCC(=O)OC)C3CC3)=O)C=CC2)ccc(C(F)(F)F)cc1Br CCCCCCC(CC(c1ccccc1)=O)CC.N12CC(F)(C3(CCC3)C1)C2=O c1(C(=O)NCCN(CC(=O)N(C)Cc2ccc(O)cc2)CC)ccc(O)cc1 Cc1nn(C)c(Cl)c1C(=O)NCC(O)CNC(c1coc(=O)[nH]1)=O C1(N(C(CCC=CC)=O)C)CCN(C(C2CCCCN2C(=O)CC(C)C)=O)CC1 c1(C(N2CCC(CNC(C3(CF)CC3)=O)C2)=O)cc(O)nc(O)c1 N1(C(C(CCC)CNC(=O)CCN=[N+]=[N-])=O)CCOC(C)(C)CC1 C1(CNC(c2cnc(Cl)[nH]2)=O)CC(O)CN1C(=O)Cc1cscn1 Cc1c(C(=O)NC2CC2NC(=O)CCC(F)(F)F)cccc1F C1(NC(c2ccc(OCC)nc2)=O)CC2CC(NC(=O)C(C)C)C2C1 c1(C2C(C(=O)NC3CC(CNC(=O)CCF)C3)C2)cccc(Cl)c1 C1(C(N2CC=CC(NC(c3c(C(C)C)nns3)=O)C2)=O)C(C)OC(C)C1C CC1(C)COCCC1CC(N1CCCC(NC(=O)CN2CC3C=CC2C3)CC1)=O c1(C(=O)NC(C2CCN(C(c3cc(C(=O)OC)on3)=O)C2)C)ccccc1O c1(C(=O)NCCC2(NC(CN(C)C)=O)CCCC2)ccnc2c1CCC2 c1(CNC(C2C(C)N(C(=O)CCCCC3CC3)CC2)=O)cccc(C#N)n1 C=CCCCC(C)(C)C(=O)N1CCC1C(N1CCC(C)(F)CC1)=O C(=O)(C(F)(F)C(O)C1CC1)NCC1(CNC(CCC(C)SC)=O)CCOCC1 C1(CC)C(C(=O)NCC(C)(C)C#N)CCN1C(=O)C=NOC c1(OC)ccc(CCNC(C2CC2NC(=O)COC(F)F)=O)c(F)c1 c1(C(C)C(=O)NC(C)CC(C)NC(=O)C#CC2CC2)ccc(F)c(F)c1 N1(C(C2CCC(CC)O2)=O)CC(CO)C2(C1)CN(C(C1CN(C)C(=O)N1)=O)C2 C1(C(=O)NC2C(C)N(C(=O)CCCC(F)(F)F)CC2)CC2(CCCC2)CO1 Cc1cc(C(N2C(CNC(c3nnc(O)nc3O)=O)CC3CC23)=O)cnc1C c1(CO)nc(N2CCc3cc(C(F)(F)F)ccc3C2)c2c(F)cccc2n1 CCCCC(O)C(C)C(=O)NCCC1COCCN1C(=O)C(C)=Cn1ccnn1 c1(Cc2scc(C(=O)NCC(N3CCC(C)(C#N)C3)=O)n2)c(F)ccc(Cl)c1F N1(C(c2ccc(F)cc2I)C(=O)NCc2ccccc2)CCc2cnccc2C1 c1(C(=O)NC2C(CC)CN(C(=O)C3=C(C)OCC3)CC2)ccc2c(n1)OCCO2 C1(NC(CCOc2c(C)cccc2)=O)CCN(C(C2(CF)CCC2)=O)CC1C C(=O)(C1=CCOCC1)NC(CN(C(C(C)SCC)=O)CC)C c1(C(N2CC(CC(CNC(C=C(CC)C)=O)(C)C)C2)=O)cc2cccc(O)c2[nH]1 c1(N2C(C)CC(NC(c3nc(C(C)C)oc3)=O)C2)ccc(F)cc1[N+](=O)[O-] C1(CC(=O)N(CCCCC)C)CN(C(=O)COCCCN(C)C)CC1C c1(SCC(=O)NC2C(CNC(c3cc(OC)ncc3)=O)C2)csc2ccc(C)cc12 N1(C(C2(C#C)CC2)=O)CCC(NC(=O)Cc2cncs2)C(C(C)C)C1 N1(C(C2ON=C(C(C)C)C2)=O)CCC2(CCN(C(=O)C(C)CCN(C)C)C2)C1 N1(C(CC2C(C)(C)OCC2)=O)CCC2(CC2C(N2CCC(c3cnco3)C2)=O)C1 Cc1ccc(O)cc1NC(C1OCCC1NC(C1CC12CCCC2)=O)=O C1(CS(C)(=O)=O)CCCN(C(=NCCN2CCC2)NC(C)C2=CCCCC2)C1 C1(NC(c2c(C)noc2C)=O)CN(C(=O)C=Cc2ccc(Cl)cc2)CCC1F c1(-c2ccc(CNC(c3ccc(OCC)nn3)=O)cn2)ccc([N+](=O)[O-])c(C)c1 C1(C(C)C)CN(C(=O)CC2CSC2)CCN1C(=O)CC1CCC(=O)N1 c1(C2C(C(=O)NCc3c(OCOC)cncc3)C2)c(O)cccc1F C1(CNC(CCC#C)=O)CCN(C(c2c(SC)cccc2F)=O)CC1CO N1(CCC)CC(N=c2[nH]c(=NCCCNC(C3CCC3)=O)[nH]c3ncn(CC)c23)C1 C(C)(C(C(=O)N1CCC2CC12)NC(=O)C=CC1CCOCC1)OC C1(C(N2CC(CNC(c3cnc(Cl)nc3)=O)OCC2)=O)CCC2(CC1)CC2 c1(C(N2CCC(NC(c3cc(COC)sc3)=O)C2C)=O)cccn2nccc12 CC(C)(CO)C(=O)N1CCC1C(=O)NCCN1C(=O)CCC1=O c1(CNC(N2CCC(N(C)Cc3cccc(Br)c3)CC2)=O)cn2ccccc2n1 N1(C(c2c(NC)nccc2)=O)CC2CC(C1)N(C(c1cc(O)nc(Cl)c1)=O)C2 C1(CC(=O)NC(CC=C)CNC(C2CCS(=O)(=O)N2)=O)CC(=O)NC(=O)C1 c1(C(=O)NC2CC(CNC(c3ccc(F)s3)=O)C2)cc2nc(F)ccc2o1 CN1CCN(S(=O)(=O)N2CCCC(NC(C3CCC3)=O)C2)CC1 c1(C(=O)NC2CN(C(c3ccc(C#C)o3)=O)CC2F)csc([N+](=O)[O-])c1 C(=O)(C(C)CC(F)(F)F)NCC(C(=O)NCCCSCC)CC1CC1 C1(C)(NC(CCN(C(C(C=C)OC)=O)C(C)C)=O)CCC(C)(C)C1 N1(C(Cc2ccc(C)o2)=O)CCCC(C(=O)N(C(C)CC(C)C)C)C1C n1(CC)cnc2nc(N3CCC(C)(CC)C3)[nH]c(=NC(C)c3ccc(Br)cc3)c12 C=CC1CN(C(=O)C(F)(F)c2ccsc2Cl)CC1NC(=O)C(C)CC C12(C(=O)NC3CC(CNC(C(C(C)C)OC)=O)CC3O)CC3CC1C2C3O c1(CC)cccc(F)c1C(=O)NC1CN(C(c2sc(C3CC3)nc2C)=O)CC1C C1(C(=O)NC(c2ccccc2)CC2CC2)CC2CC2N1C(c1sccc1Cl)=O C1(CNC(C2C(C(C)C)C2)=O)CCC(NC(=O)CSc2ccccc2)CC1 Cc1c(C(=O)NCCCCCCO)[nH]ccc1=O.c12ccc([nH]1)CC(=O)NOC2 N1(C(CC)=O)CCCC(C(=O)NCC2(F)CC(CNC(C3CCCN3C)=O)C2)C1 C=C1CC(C(=O)Nc2cnoc2)N(C(=O)C(c2ccccc2)O)C1 c1(CCC(=O)NCC(CO)NC(c2cc(C)[nH]c2C)=O)csc2ccccc12 CC(C(=O)NC1CC(C)(NC(C2CC2c2ccc(F)c(F)c2)=O)C1)S(N)(=O)=O C(=O)(C(O)CC(C)(C)C)N1CCCC(N(C)C(c2cccc(Cl)c2C(F)F)=O)C1 C(C)(C(=O)N1CCC1C(=O)NCc1cccc(F)c1C)(C(C)C)OC c1(C(=O)OC)cc(C(N2CCC2CNC(c2coc(C)c2)=O)=O)c(F)cn1 C(C)(CCCCNC(c1ccc(C(F)F)s1)=O)NC(CCc1scc(C)n1)=O c1(C(N2C3CC(NC(C(C)=C(C)C)=O)(C3)C2)=O)cc(N(C)C)nc2ccccc12 C1(C(=O)NCCC2N(c3nnc(CCC)s3)CCCC2)COc2ccccc2O1 C(C(C)(C)C1=CCOCC1)NC(NCc1nc(CC(=O)OC)sc1)=N C(=O)(C1=CCCOCC1)NC1CCC(C)(NC(=O)CC2CCC(F)(F)CC2)CC1 c1(SC)sccc1C(N1CCCC1C(C)(C)NC(C1(C)CC(F)C1)=O)=O C1(C(=O)NCCC(C)(C)NC(c2cccnc2O)=O)CC2(C1)CC(F)(F)C2 c1(C(=O)NCCC2CC(OC)CN2C(=O)CCCC2CCC2)cc(C)nc(O)n1 Cc1nc2nccc(C(C)NCc3cn(C)nc3C)n2n1 C(=O)(C(C)(O)C(F)(F)F)NCC(CC(=O)N(CC=C)CCO)O Cc1cc2c(cc1Cl)C(N)CO2.N1(c2cc3cc(n2)OC3)CCc2cccc(Cl)c2C1 C=CCC(C(=O)NC(C)CCCCNC(C1CN(C(C)=O)C1)=O)N(C)C C=C1CCC(C(=O)NCC(=O)NCC(F)(F)F)CC1 N1(C(C(CC)COC)=O)CC2(CCC2NC(c2cc(C)n(C3CC3)n2)=O)C1 C1(C)(NC(C2N(CCC)CCC2)=O)CCN(C(C)CN2CCC(O)CC2)C1 c1(C(N2C(CNC(c3n(CC)ccc3)=O)CC2)=O)cncc(OCC(F)F)c1 c1(C(N=c2cnn(C)[nH]2)=O)cc(-c2ccc(C3(C#N)CC3)cc2)cn2ccnc12 c1(CNC(C(C=CC)O)=O)ccccc1CN(C(=O)C(C)OCCF)C C1(CN(C)C(c2cccc(C(C)(F)F)c2)=O)CN(C(C2CCOC2)=O)CC12CC2 C=CC(CC)CC(=O)NCC(c1cccc(C)c1)NC(c1ccoc1C)=O c1(C(N2CC(OC)(CNC(C3CCC34CCC4)=O)C2)=O)ccc(F)cc1Cl c1(NC(=O)C=C2CCN(C(c3ccns3)=O)CC2)cccnc1[N+](=O)[O-] c1(C(N(C2CCN(C(C3CCCN3CC(F)(F)F)=O)C2)C)=O)cc(C(N)=O)cn1C c1(C(=O)NCCC2(O)CCCN(C(c3cnco3)=O)C2)ccc2nccnc2c1 N1(c2ncc(C#N)cc2Cl)Cc2ccccc2C(CNC(=O)C2=CCSC2)C1 c1(C(C(=O)NCCC2(NC(C3C(C(=O)OC)CC3)=O)CC2)O)ccccc1F N1(C(C=C(CCC)C)=O)CCCC1C1CCCN1C(=O)C=Cc1c(C)coc1C c1(C(=O)NCC(CC)NC(=O)CN(C2CCCC2)C)cnc2cnc(Cl)cc2c1 S(=O)(=O)(c1cc(Cl)ccc1F)Nc1ccc2c(c1)CN(C(c1c(C)nco1)=O)C2 c1(C(N(CC(CN(C(=O)Cc2ccon2)C)O)C)=O)nnn2c1COCC2 N1(C(CCOCC#C)=O)CCCN(C(c2ccc(OC(F)F)cc2)=O)C(C)C1 N1(CCNC(=O)NCc2n(CC)nnc2C)CCc2sccc2C1 Cc1nc(-c2ccccn2)ncc1C(N1CCC(N(C(=O)C2=NOCC2)C)C1)=O N1(C(C2(CO)CC2)=O)CCC2(NC(=O)C=CCN3CCCC3)CCCC12 C1(N(C(=O)C=CBr)C)CCN(C(C2CCCN2C(=O)C(C)(C)C)=O)C1 N1(C(CC(=C)C)=O)CCCCC1CN(C)C(C1(CSC)CC1)=O Cc1nc2c(s1)CN(C(C1CCC(NC(c3cnccc3C#N)=O)CC1)=O)C2 C(=O)(C1=CCC(C(F)(F)F)OC1)N1CC(CNC(CN(C)CC)=O)N(C)CC1 c1(C(C)NCCc2ccc(Cl)c(C(F)(F)F)c2)cccc(O)c1Cl C1(NC(COCCC=C)=O)CC(NC(c2cnc(CC)s2)=O)C12CCC2 n1(CC)cc(C(=O)NCC(CNC(C2(CF)CC(F)(F)C2)=O)CO)c(C)n1 Cc1cc(=O)n(C)cc1NC(c1cccc(-c2cn(CC3CCC3)nn2)c1)=O C1(NC(c2cnn(CC)n2)=O)CCCCC1NC(C1CCCN1C(=O)C1CC1)=O CCC(CC(=O)NCC1(F)CN(C(C2Cc3ccccc3O2)=O)C1)C(C)(C)C c1(Cn2cc(C3(O)CN(C(C4(C)CC4(Cl)Cl)=O)C3)nn2)ccccc1[N+](=O)[O-] c1(C(=O)NC(C)=O)n[nH]c(C(C)C)c1Br.C1(=O)CCC(=O)NCCC2(CC2)N1 C(CC(=O)NCCOC1CCOC1)(C(F)F)NC(C1CC(N(C)C)C1)=O CC1CN(C(=O)Cc2ccc(Cl)s2)CC1NC(=O)CCc1cnc(C2(C)CC2)o1 c1(C(N2CC(CO)CC(F)C2)C(=O)NC(C)C)ccc(Br)cc1Cl C=C1CC2(C1)CC(C(=O)NC1CC(C)(NC(C3CC3(F)F)=O)C1)C2 N1(C(c2ccc(C(C)=O)o2)=O)CCOCC1C(=O)N(C)Cc1cnn[nH]1 N1(C(c2ccn(C)c2)=O)CC(O)CC1CC(=O)NCCOCC1CCC1 C1(CCNCC2(Cl)C(F)(F)C2)CSc2ccccc2O1 c1(C(=O)NCC2(NC(c3ccn(CCC)n3)=O)CC2)ccc(C(=O)OC)c(F)c1 Cc1cc(C(F)(F)F)c2cc(O)ccc2n1.C(=O)(CN)NCCN(S(C)(=O)=O)C Cc1cc(F)ccc1C(O)C(=O)NCC1(N2CCN(C)CC2)CCCCC1 N1(C(c2ccc(OCC=C)cc2)C(=O)NCC=C)CCC(OC)C12CCC2 C(=O)(C(C1=C(C)CCCC1(C)C)N1CCC2(CC(O)C2)C1)NCC(CC)(C)OC C(=O)(C(CCCO)c1ccccc1)N1CC(COCCOCCOC)OCC1 c1(C(C)=O)cncc(C(N2CCCC2CCCNC(C2C=C2C)=O)=O)c1 CC1CCN(C(c2[nH]ccc2CN(C)C)=O)C(C)C1NC(=O)C=C1CCCCC1 c1(CC(=O)N(CCN(C(C(C)SCC)=O)C)C)ccccc1OC(F)(F)F CCCCC(O)CC(=O)NC(C)(C)CCC(=O)N(C(C)CC(N)=O)C N1(C(c2cc(C)ncc2C)=O)CCC2OCCN(C(c3nn(C)cc3Cl)=O)C2C1 O=C1COc2ncc(C(=O)NC3CCN(C(=O)CC4C=CCC4)CC3F)cc2N1 C1(CC(=O)NC(CNC(c2nc(C)c(C)s2)=O)(C)C2CCC2)CCC(=O)NC1=O C1(OC)CCC(C(=O)NCC2CC2CNC(=O)C=Cc2cnc[nH]2)CC1 C(=O)(CP(=O)(C(C)C)C(C)C)NCCOCCNC(c1c(C)cc(C)cc1O)=O c1(N2CCC(C(C)NC(C=NOC)=O)C2)nc(C)nc2scc(CC(C)C)c12 C(=O)(CN=S(C)(C)=O)N1CCCC(C(C)NC(c2ccncc2F)=O)C1 C1(C(=O)NCC(C)CN(C)C(c2cc(N)cnc2Cl)=O)CCCC12CCC2 N1(C(c2cc(C)n(CC)c2C)=O)CCC2CN(C(c3ccc(Cl)o3)=O)CCC12 C1(O)(CNC(C(CCOCC)NC(c2cn(C3CC3)cn2)=O)=O)CCC(C)(C)C1 c1(C(=O)NC(CNC(C(CC)(C)CO)=O)(C)C)cncc2c1CCNC2=O c1(-c2cnc(C(F)(F)F)o2)cccc(CN2CCSCC2)c1 c1(CCC(=O)N(CC(CC)NC(c2n[nH]cc2F)=O)C)cc(F)c(F)c(F)c1 N1(C(C2(COC)CC2(F)F)=O)CCC(O)(C(C)NC(c2cnc[nH]2)=O)CC1 N1(C(C(C=C)C)=O)CCC2(CCC2NC(c2ccc(OC)nc2)=O)CC1 C(=O)(CCCC(=O)N(C)C)NC1CC(F)(CNC(Cc2c(CC)cccc2)=O)C1 C1(NC(CCCC=C)=O)CN(C(=O)C(O)C(C)C)CC1(C)C N1(C(Cc2cccc(C)c2)=O)Cc2ccc(NC(c3cncs3)=O)cc2C1 C(C(F)C(=O)NCC1CC(C(=O)NC2CC(C(=O)NC(C)(C)C)C2)C1)OCC Cn1ncc([N+](=O)[O-])c1C(=O)NCCC(C)(C)NC(c1n[nH]cc1Br)=O c1(N2CC(c3onc(-c4c(OC)ccc(C)n4)n3)C2)c(O)nc(=O)n(C)c1N CC1(C)C(C(=O)NCCOC2CCN(C(c3cc(C4CC4)ncn3)=O)C2)C1C#N c1(C(N2C(C(=O)Nc3n(C)ncc3I)COCC2)=O)ccc2c(c1)CC2 C12(C(=O)OC)CC1CCCN2C(=O)C(n1cc(-c2cc(C)cnc2Cl)nn1)C CN1CC(c2nnnn2Cc2ccccc2)(NC(C)(C)CCCF)CCC1=O C=O.CS(=O)CCNC(=O)CCC1CCCC1 c1(C(=O)NC(C2CN(C(=O)C(F)F)C2)C)cccc2c3c([nH]c12)CCC3 c1(C(N(CC(=O)N(C(c2ccccc2)C(=O)O)C)CC)=O)ccc(F)cc1Cl C1(CNC(CCC(=O)NCC)=O)CC2(CC2)CN1C(c1coc(Cl)n1)=O c1(OC)nc(=NC2CC(NC(c3c(Cl)ccc4cccnc34)=O)C2)nc(OC)[nH]1 CC1(C)CN(C(C2(C)CC2(C)C)=O)CC(CNC(c2coc(Cl)n2)=O)O1 C(=O)(C1CCCn2cnnc21)NCC1(CNC(=O)Cc2n[nH]cc2Br)CCC1 c1(C(N(C2CCN(C(CCOCCC)=O)C2)C)=O)cc(Cl)nnc1O N1(C(CNC(c2cc(OC)n(C)n2)=O)=O)C2CCCC1CN(C(C1CC1C)=O)C2 c1(-c2n(CC=C)nc(CC3(C)CC3)n2)cnc2c(c1)OCCN2 N1(C(c2cc(Cl)sc2Cl)=O)CCc2c(C(N3CCC(CO)C3)=O)n[nH]c2C1 C1(CNC(C(CC)OCC)=O)CC2CCC1N2C(=O)Cn1cnnc1O c1(C(=O)NCC2CN(C(c3c(CC)cno3)=O)C(C)C2)c(Cl)ccc(F)c1N C(C1CCCC1)=C(C)C(=O)NC(C)CNC(=O)CC1(C)CCCO1 c1(-c2c(F)ccc(OCC)c2)ccc2c(c1NCc1cc(Cl)ccc1Br)OCO2 C1(NC(c2ccc(Br)o2)=O)CC2C1CCN2C(C1CC2(C1)CC(O)C2)=O CN1CCC(N=c2[nH]ccc(=NCCc3cnn(-c4ccccc4)n3)[nH]2)CC1 N1(C(C(Cc2cccc(OC)c2)O)=O)C2CCC1CN(C(C)=O)C2 C(=O)(CN=S(C)(C)=O)NCC1C(NC(C(c2nc(C)sc2)=O)=O)C1 Cc1cc(C(=O)NCC(C2CCC2)NC(C2(C)C=CCC2)=O)nn1C(C)C1CC1 c12cnc3ccccc3c1C(=O)N2.C1(NS(C)(=O)=O)CCN(CCn2cnnn2)C1 C1(C(N2C(CC#C)CCCC2)=O)CC(O)CCN1C(=O)C(CSC)OC C(CC(C)CCNC(=O)CSC(C)(C)C)NC(c1cc(C)sc1)=O C1(CNC(CCC(C)C)=O)CC(C(C)(C)C)CCN1C(=O)CCc1cscn1 n1(CC(C)C)c(-c2ccc(C#N)c(F)c2)csc1=Nc1cc(C#N)ccc1Cl C(=O)(CCCCC(N)=O)N1CC(C)C(CNC(=O)CC2(O)CCCCC2)CC1 CC(=Cn1ccnn1)C(=O)N1CC(C)CN(C(c2ccc(C)cc2F)=O)C(C)C1 CCC(CC)C(F)C(=O)NC1C2CN(C(=O)C(O)CC(C)(C)C)CC12 C1(N(C(c2cnc(SC)s2)=O)C)CN(C(=O)CCSCC2CCCCO2)CC1O CC1=C(CNC(CCCCCO)c2nnnn2-c2ccccc2)S(=O)(=O)CCO1 C(=O)(C(C)(C)C(C)(C)C)NC(C1CCN(C(CNC(CCC)=O)=O)CC1)CO C(=O)(C1=CCCC1C)N(CCCCN(C(=O)CNC(c1cccc(Cl)c1)=O)C)C c1(OCC(=O)NC(C2CC(C)C2)C)cccnc1 N1(C(C(C(=O)OCC)F)=O)CC2(C1)OC1(CNC(=O)C(C)N(C)C)CC2(CO)C1 c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)CO)ccn2ccnc2n1 CC1CCCC1(C)C(=O)N(C1CCN(C(C2CC(C#N)C2)=O)CC1)C C1(C(=O)O)(NC(c2cnc(OC)c(C)c2)=O)CCc2ccccc2C1 CC(CCCc1cccnc1)NC(c1cnnn1C1CCC1)c1nnnn1C N1(C(C(C)CNC(c2ccco2)=O)=O)CCN(C)CC1CCO C1(CNC(c2ccc(N(C)C)nc2)=O)CN(C(=O)CCc2cccs2)CC12CC2 N1(C(c2cnc(CC)s2)=O)CCC(O)C(N(C)C(C2CC2C(F)F)=O)C1 C12(C(=O)NCC(N(C(c3ccc(COC)s3)=O)C)C3CC3)CCC(C)(C1)OC2 C1(C(N(C)CC2CCC(CNC(C(CC)F)=O)CC2)=O)CC2CC2CC1C CC1CC(NC(=O)CCSc2ccccc2F)CN1C(=O)CC1CCC1(C)C C(C(CC(C)C)C(=O)NC1(C)CCCN(C(c2ccnn2C(C)C)=O)C1)OC C(=O)(CCCCCC(C)C)NC1C(NC(c2n(CC)nc(C)c2)=O)COC1 Cc1nc(Cl)[nH]c(=NC2CCCCC2CNC(c2[nH]nnc2C)=O)c1Cl c1(C(=O)NCCOCCN(C(=O)CC2(C#N)CCC2)C)cccc(F)c1OCF N1(Cc2cc(C)cc(Br)c2O)CC2CCC1CN(C(c1nccnc1Br)=O)C2 c1(C(c2nnnn2CC2CCCO2)Nc2ncc(C)s2)ccc(CO)cc1.CO N1(C(C(COCC)NC(C2CCS2(=O)=O)=O)=O)CC2(CC(C)CO2)C1 N1(C(CN(CC(C)(C)C)C)=O)CCC2C(C1)CN2C(=O)C=CC1CCOCC1 c1(CC)ccc(C(N2CCCCC(NC(c3ccc(C)nc3)=O)C2)=O)c(C)c1 N1(C(CCCCOC)=O)CC2=C(C1)CN(C(c1cc(O)nc(OC)n1)=O)C2 C(=O)(C(CC(C)C)NC)N1CC(n2cc(-c3cccc(SC)c3)nn2)C(C)C1 C(C(C)(C)C(=O)NCCCCCOCC1CCCCCC1)OCC C1(NC(C(C)OC)=O)Cc2ccccc2N(C(c2cnn(C(F)F)c2)=O)C1 C1(C(=O)NCc2cnn(CCO)c2)CN(C(C2CCCOC2)=O)CC1(F)F CC(C(=O)NCC(c1ccccc1)N(C(=O)Cc1cccs1)C)S(N)(=O)=O C(=O)(C(C)CS(C)=O)N(CCCNC(c1c(C)nc(CO)o1)=O)C(C)C N1(C(c2c(C)cc[nH]2)=O)CC(NC(c2cccc(C3(C)CC3)c2)=O)CCC(O)C1 C1(CC)(NC(=O)C(c2cnn(C(C)(C)C)c2)C)CCN(C(=O)CO)CC1 C1(N(C)C)(C(=O)NCc2c(O)cc(Br)cc2F)Cc2ccccc2C1 CC1(C)OCCOC1C(=O)NCC1CC(NC(c2cn(C3CC3)cn2)=O)C(O)C1 c1(SC)ccc([N+](=O)[O-])c(C(=O)NC(c2ccccc2)CNC(=O)C2=NOCC2)c1 C(=O)(CCCCC(=O)N1CCC(NC(c2cnc3c(c2)COC3)=O)C1)OCC N1(C(c2cc(C)nn2C)=O)CCC2(CC(C(=O)NC(C)C(=O)NC(C)C)C2)C1 Cc1cc(=O)c(C(=O)NCC2CCCN2C(c2ccc(F)c(F)c2)=O)c[nH]1 c1(CNC(C(=O)Nc2ccc(C)cc2F)C)ccc2c(Br)cccc2c1 CCC(O)C(C)C(=O)NC1CCC(CNC(=O)Cc2cncc(C)c2)CC1 C1(NC(CNC(C)=O)=O)CN(C(C)C(=O)Nc2cccc(C)c2C)CCC1(F)F C(=O)(C(C)(C)CS(N)(=O)=O)N(CCN(C(c1cc(C(=O)OC)sn1)=O)C)C CC(C)C(O)CC(=O)NC1CCN(CCOCC(F)(F)C(F)(F)F)CC1C N1(C(CCCc2c(C)ccs2)=O)CC(CNC(=O)C(=O)NC(C)C)C(F)(F)C1 C1(COC)CN(C(=O)CCc2cccc(F)c2)CCN1C(C1C=CC=CC=C1)=O c1(C(N2CCC(C(N3C(C(C)C)COCC3)=O)C2)=O)n[nH]cc1[N+](=O)[O-] C1(N(C(CC)C(N)=O)C)CCN(C(c2ccc(C)c(C)n2)=O)CC12CC2 CC1CC2CN(C(c3cnc(CCN)nc3)=O)CCCN2C1 c1(C(N2CC(SC)C(n3cc(C4CCOC4)nn3)C2)=O)ccc2c(c1)NC(=O)C2 C#CC1(C(=O)NC(C)(C)CF)CCN(C(c2[nH]cc(C)c2C)=O)CC1 c1(C(=O)NC2(C(=O)NCCC(C(C)C)C)CCN(C)C2)cc2cc[nH]c2cn1 C1(NC(c2c(C)cc(SC)o2)=O)CC(NC(=O)CC2OCCCO2)C12CCC2 c1(C(N(CCNC(COc2ccn(C)n2)=O)C2CC2)=O)ccnc2ncccc12 C1(C(C)NC(c2cc(F)n[nH]2)=O)CCN(C(c2cnc(Cl)s2)=O)CC1 C(=O)(C1=C(C#N)CCC1)N1CCC(C=C)(C(=O)NC2CCC(N(C)C)C2)C1 C1(O)(C(C)NC(CCC(C)OC)=O)CCN(C(C2(CO)CC(F)(F)C2)=O)CC1 c1(C(N2CCC(C)(NC(=O)CSCC(N)=O)CC2)=O)ccc2c(c1)CNC2=O Cc1nc(C(N2CCCC(N(CCO)C(C3(C)CCOCC3)=O)C2)=O)[nH]c1C CC1CN(C(c2csc(S)n2)=O)C(C)CN1C(=O)CNC(c1cccs1)=O N1(C(C)C(=O)NC(c2ccc(N(C)C)cc2)=O)CCC(CC#N)C1 C1(NC(C=CCC)=O)CCCCN(C(c2cc(Br)ccc2SC)=O)C1 Cc1ccc(C(N2CCCC2CNC(c2cc([N+](=O)[O-])c[nH]2)=O)=O)c(C(C)C)n1 C(=O)(C(C(C)(C)C)N1CCNC1=O)N1CCC(C)(NC(c2c(C)nncc2)=O)C1 c1(C(N2C3(c4cn(CC5(C)CC(C)C5)nn4)CC(C2)C3)=O)cc2c(cc1O)OCO2 c1(C(N2C3C(CNC(c4c(OC)cccn4)=O)C(C3)C2)=O)cc(C)cc(C)c1N Cc1cnc(CNC(=O)C(Cn2cccn2)NC(=O)CN2CCCC2)cn1 c1(C(N2C(CCC(N3CCC(OC)C3C)=O)CCCC2)=O)ccc(C#N)c(C)n1 CCC(C)C(O)CC(=O)N1CCCCC1C(=O)Nc1ccc(C)cc1C c1(CC)ccsc1C(=O)NC(CNC(=O)C(CO)OC)CO Cc1c(C(=O)NCCC2(O)CCN(C(=O)C(N3CCOCC3)C)C2)cncc1Cl N1(C(C(CCC)F)=O)CCN(C(=O)C(N2CCCCC2=O)C)C(C(C)C)C1 C(=O)(C(CC(C)C)ONC(c1cn[nH]c1)=O)N1CC(C(=O)NC)C(OC)C1 N1(C(c2nc(C(=O)NCC=C)sc2)=O)CCCC(CCC)(NC(=O)CC(C)F)C1 c1(C(=O)NC(CN(C(C(CC)OC)=O)CC)C)ccc2c(c1)CCCS2 CCCC(CC)NC(c1ncc[nH]1)Cc1ccccc1 c1(COC(c2ccn(CCOC)n2)=O)cc(C)n(C2CC2)c1C c1(Oc2c(C(=O)OC)c(C#N)c(F)cc2)ccc2c(c1F)NC(=O)CO2 c1(-c2cc(CNC(c3cc(CO)cc(Cl)n3)CCOC)no2)ccc(F)c(F)c1 c1(OC)ccccc1C(CNC(c1cccc(CCNC(=O)NC)c1)=O)N(C)C C1(CC(=O)N(CCN(C)C)CC)(NC(=O)CCn2cnnn2)CCCCC1 c1(C(CNC(CC(C)OC)=O)NC(=O)CCN2CCOCC2)ccc(F)cc1F CC1CC(C(=O)NC2CCCC2C(N)=O)N1C(=O)CSc1nc[nH]n1 C1(C(N(CCCC(=O)NC)C)=O)CCC2CCC1N2C(c1ccc(C2CC2)o1)=O c1(SC)cc(C(=O)NCC(C(C)C(C)C)NCc2ccc(CF)cc2)ccc1F C(CC(C(C)(C)C)NC(=O)CC1(O)CCC1)N(C(CC1CCN(C)C1=O)=O)C C(N=c1nnn(C)[nH]1)C1C(NC(C(C(C)C)OCC(C)C)=O)CCCC1 N1(C(c2n(CC)nnc2)=O)CC2CN(C(=O)CCC3CCCN(C)C3)CCC12 c1(Cc2ccccc2)ccccc1C(=O)NC1CC(CNC(C=CC)=O)C1 c1(C(N2C(CNC(C(C3CCOC3)NC(C)=O)=O)CC2)=O)cc2n(n1)CCO2 c1(C(=O)NC2CC(O)(CNC(c3cccc(=O)o3)=O)C2)cc2sc(Cl)cc2s1 c1(C(N(CC(C)C(F)(F)F)C)=O)coc2c1CN(C(=O)C(=O)NCC1CC1)C2 c1(C(NNC(=O)Nc2cc(C(O)C(F)(F)F)ccn2)=O)ccc(Cl)cc1F c1(C(=O)NC2C(CC)N(C(C3CC(=O)NC(=O)C3)=O)CC2)cncc(F)c1C C(=O)(CC(C)(C)CC(F)F)N1CCC(O)(C(C)NC(c2cc(N(C)C)ccn2)=O)C1 c1(C(=O)Nc2ccc(C(=O)NCC)cc2C)cccc2c(C)csc12 c1(-c2ccnc(C)c2C)c(C)ccc2ncccc12 C1(C(N2C(CN(C3CCCCC3)C)CCCC2)=O)CCc2nnnn2CC1 c1(OCC)cc(N2CCC(CO)(NC(=O)C(C)S)CC2)nc(C)n1 C(=O)(C1=C(Cl)CCCC1)N1C(CNC(c2ccc(CC(C)C)s2)=O)CCCCC1 c1(C(C(=O)NCC(=C)C)N(CC(F)Br)C)ccc(OC)c(O)c1 c1(C(N2CCN(C(=O)CCn3ccnn3)C(CF)C2)=O)cncc(Cl)c1Cl N1(C(c2c(C)nncc2)=O)CC2(C1)CN(C(C1CC3(C1)CC(O)C3)=O)CCO2 Cc1cc(F)c(Cl)cc1NC(C1CCC(NCc2cc(I)c[nH]2)C1)=O C(=O)(C(CC(F)F)NC(=O)C(F)CC1CCOC1)N1CCC(SC)CC1 N1(C(COCCSC)=O)CC2(C1)CN(C(c1ccn3ncnc3c1)=O)CC2CO c1(C(=O)NC2C(CNC(C(C)NC(CC)=O)=O)COC2)cc(Cl)ccc1F N(C1CCc2c(O)cccc21)C(=O)NCc1nc(CC2CC2)no1 c1(C(=O)NCC(CCNC(=O)CC(C)(C)C)OC)nccc(Cl)c1F N1(C(CCC)C(=O)Nc2ccccc2OC)CC2CS(=O)(=O)CC2(C#N)C1 CN1CCCC(CNCC2CC(O)(C(F)(F)F)C2)C1c1ccc(C(F)(F)F)cc1 c1(C(=O)Nc2cccc(OCCC(C)F)c2)cccc2ccccc12 C1(N(C(C(C)OCC)=O)CC2CC2)CCN(C(C2(n3cncn3)CC2)=O)CC1 c1(OCC=C)cc(OC)ccc1C(=O)NC(C)CN(C(=O)CC#N)C C1(NC(C)C(=O)N2CC(CC(C)NC(C3CCOCC3)=O)C2)CCOCC1 CCC(C)C(C)N=c1[nH]c(CC(N2CCCN(C)CCC2)=O)cs1 c1(NC(CSCCNC(C(C=C)(F)F)=O)=O)cccc(Cl)c1O C1(CC)C(C(N2CC(=O)CC2C(=O)NCC(F)(F)Cl)=O)CCN1C Cc1cn2c(n1)CCC(N=c1nc3sccc3c(NCC(C)S(N)(=O)=O)[nH]1)C2 C1(C(=O)C(=O)C2CC2)C2CCC1CN(NCc1ccc(OC(F)F)cn1)C2 C1(C(CO)NC(=O)C=CCF)CCCN(C(=O)CCc2ccccc2Cl)C1 N1(C(C(C)S(N)(=O)=O)=O)CCCC(O)(Cn2cc(CCN3CCCC3)nn2)CC1 C1(OC)CCCC(C(=O)NC2(C)CC(NC(c3cc(C)[nH]c3C)=O)C2)C1 CCC(C)C(O)C(C)C(=O)NC1CC2(C1)CN(C(c1n[nH]cc1C)=O)C2 C(CC(=O)NC(c1ccn(C)c1)C)(C(F)F)NC(Cc1cn(CC)nc1)=O C1(C)(C(N2CC(C)(NC(c3c(OC)cc(C)cn3)=O)C2)=O)OC(C)(C)OC1C C1(C(=O)NCC(CNC(C2(NC(C)=O)CCOCC2)=O)OC)CCCCNC1=O Cc1onc(O)c1C(N1CC2C(CNC(C3CCC(CO)CC3)=O)C2C1)=O c1(C(=O)NC2CC2NC(C2CC2F)=O)ccc(C(F)(F)C(F)(F)F)cc1 c1(N(C)CCc2cccc3ccccc23)cc2c(s1)C(C)(C)CCC2 C1(C(N2C(CN(C(c3c(C)con3)=O)C)CC(F)C2)=O)CC2(C1)CC21CCC1 C1(C(=O)NCC(C)(CNC(C2CC(C(C)C)C2)=O)OC)CCC(O)CC1 C1(CCOC)CN(C(c2ccc(Cl)cc2N)=O)CCN1C(=O)C1=CC(C)(CC)C1 c1(CNC(c2ccc(OC)nn2)=O)ccc(CNC(C2CCCN2C)=O)cc1F CC(C)(CC(F)(F)F)C(=O)NC1CN(C(=O)C=CCO)CC(F)(F)C1 c1(N(C)Cc2ccc(C)cc2)ncc(C)cc1S(=O)(=O)NCc1ccc(Cl)cc1C C1(C(=O)NC(CCC=C)(C)C)CC(F)CCN1C(C1CC(C2CC2)=NO1)=O c1(C(N2CCOCC(NC(CC=C=C)=O)C2)=O)ccc2ncc(=O)[nH]c2c1 n1(CC)nc(C)c(C(=O)NC2CC3CC(NC(=O)C(CC(C)C)OC)CC23)c1Cl C(c1cncnc1O)=CC(=O)NC1CC2CC1N(C(C1CCCOCC1)=O)C2 C1(NC(C(CC)C)=O)CCN(C(=O)C=CSc2ccccc2)C1C(C)C c1(OC)cc(C(N2C3CCC(C3)C2CNC(=O)C(C)CO)=O)ccc1O N1(C(C(C)(C)CO)=O)CCCC(O)(CN=c2[nH]nc(CO)s2)C1 C1(C(N2CC(NC(COC(CC)C)=O)C(C)C2)=O)CC2C(C1)C2(F)F CC1CC(C(=O)NCCC(C)(C)NC(c2sc(C#N)cc2Cl)=O)CC(=O)N1 C1(CNC(c2c(C)cccn2)=O)CC2CCC(C1)N2C(C1CCCCN1C)=O C=CCCC(C(=O)OCC)NC(C1CSCN1C(=O)CCCCC)=O CC(C)(CNC(=O)C=CCF)C(=O)N(C1CCCC1)CC(N1CCC1)=O c1(C(N(C(CNC(C2C(C=C)OCC2)=O)C)CC)=O)cc(C)nc2[nH]nc(O)c12 c1(C(N(C2CCN(C(=O)C(O)CCC(C)C)C2)CC)=O)cc2cccnc2cn1 c1(CC)ccc(C)cc1NC(c1cccc(F)c1)c1nnnn1C1CCOCC1 C1(CNC(c2[nH]cc(CC)c2)=O)CCCCC1NC(=O)C(C)(C)c1ccccn1 c1(N(CCOC)C)cc2nc(n1)COCCN2C.C(CF)OC c1(COC(c2cnc(Br)c(O)c2)=O)cccc2nonc12 C1(C2CC2)(C(=O)NCC(CN(C(C(CC)NC(N)=O)=O)C)(C)C)CCOCC1 C1(NC(c2cnn(C(C)C)c2F)=O)CCN(C(=O)C(C)(C)CC#N)CC1F C1(F)(C(=O)NC2C(CC)CCC2)CCN(C(c2cncc(CO)c2)=O)C1 c1(OC)c(C(N2CC(CNC(C3CC34CCCC4)=O)C2)=O)ncnc1C C(=O)(C1=NOC2(CCOC2)C1)N1CC(CCNC(C2(SC)CCC2)=O)OCC1 C1(CCOC)CN(C(C2(n3ccnn3)CC2)=O)CCN1C(c1cccc(F)c1)=O N1(C(C)C)CCOC(C(=O)NCC(C2CCCCN2C(=O)CN(C)C(N)=O)O)C1 C1(C(=O)NCCN2CC3CCC2C3)CCOCCN1C(=O)CCC(F)(F)F N1(Cc2c(OC)c(Cl)ccc2)CCC(N=c2ccn3ncc(C#N)c3[nH]2)C1 C=Cc1ccc(C(N2CCC(CNC(=O)C(O)CCN(C)C)C2(C)C)=O)cc1 C1(CC=C)(NC(C2CC(C)CO2)=O)CCN(C(c2csnn2)=O)CC1 Cc1ccc(NC(c2sccc2CNC(C2(C)CNC(=O)C2)=O)=O)c(C)n1 c1(C(=O)NC(CN(C)C(C2CCCCN2S(C)(=O)=O)=O)(C)C)cc(N)c(F)cn1 C1(C(=O)NC(C2N(C(c3c(CC)n(C)nn3)=O)CCC2)C)CCC=CCCC1 c1(C(=O)NCCC(C(N2C(COC)CCCC2)=O)O)c[nH]c2nccc-2c1 C1(CC)(CNC(C2(NC(=O)CN3CC=CC3)CC2(C)C)=O)CCC(=O)N1 C1(CNC(C)COC(F)F)CCCN1C1CC1(F)F N1(CC)CCCC(C(=O)NCC2(F)CN(N3CC(CC(=O)OC)(OC(C)=O)C3)C2)C1.O.OC.O CCC(C)(CO)C(=O)NCc1ccnc(C(N2CCOCC2CO)=O)c1 C1(CNC(C(C)(C)C2CC2)=O)CN(C(=O)CCC2CCC(=O)NC2)CC(C)(C)O1 c1(C(=O)NC(C2CCCN2C(=O)C(CO)c2ccccc2)(C)C)ncccc1O C1(NC(C2(OC(C)=O)CC2)=O)CN(C(=O)C(C2CCCCC2)C)CC1C c1(OC)c(C(N2CCCCC2CN(C(=O)COC)C2CC2)=O)cccc1[N+](=O)[O-] CN1CCN(C(=O)C#CC2CC2)CC1c1cn(Cc2ncoc2C(F)F)nn1 C1(C(=O)NC(CO)C(F)(F)F)CC12CCN(Cc1cccc(I)c1F)CC2 C(C(F)(F)CCCNC(c1c(C(=O)O)ccn1C)=O)n1cc(CCC(C)C)nn1 C1(O)(C(CN(C(C)=O)C)N(C)C)CCN(CC=CBr)C1 C(=O)(C1Cc2ccc(Cl)cc21)NC1CC(n2cc(-c3cnc(C)o3)nn2)C1 C(CC(O)CO)NC(CCC1(NC(CC2CC(N(C)C)C2)=O)CCC1)=O c1(OC)cc(C(=O)NCC2(F)CN(C(=O)CC3CCCC34CC4)C2)sc1Cl c1(C(=O)NC(C2CCOC2)CNC(c2cnc(SC)[nH]2)=O)cccc(F)c1C Cc1cc(C(=O)NC(C)(C)CNC(=O)C(C)C(C)C)cnc1O C12(CCC(=O)N(C3CCCCC3)CCNC(=O)Cc3ccsn3)CCC(CC1)C2 N1(C(C(c2ccccc2)OC)=O)CCCN(C(=O)Cc2ccc(Cl)cc2)CC1 N1(C(CC2(NC(C)=O)CC2)=O)CC2CN(C(C3(O)CCC3)=O)CC2(C)C1 N1(C(CC(CC)C(C)C)=O)CC(CO)C2(C1)CN(c1ncnc3n[nH]c(C)c13)C2 C1(C(=O)NC(C)CCCNC(=O)C=Cc2ncco2)OCCOC1C C12(C(N(C(C=C)C3CC3)C)=O)C(NC(c3nccnc3C)=O)C3CC1C2C3 Cc1c(C(=O)NCC2(C(F)F)CCN(C(=O)CCn3cnnn3)C2)cccc1O C(=O)(C(F)C(F)(F)F)NC(C1(O)CN(C(=O)CCn2cccc2)C1)C c1(N2C(CCNC(c3ccc(COC)[nH]3)=O)CCCC2)nc(C)nc2[nH]ccc12 N1(C(C2(CC)CCCOC2)=O)C2CCC1CC(c1cn(C3CCCC3)nn1)C2 CC1(CNC(c2cnc3n2CCC3)=O)CN(C(=O)CCC2OCCO2)CCO1 c1(C(N2CC(NC(CN(C)C(N)=O)=O)C(CC(C)(C)C)C2)=O)ccc(O)nc1Cl Cc1[nH]nc2ccc(C(N3CC(O)(CNC(C4(CO)CCC4)=O)C3)=O)c(Cl)c12 c1(SC)cccnc1C(=O)N(C)CC1CCN(C(=O)C2=CCCS2)CC1 C1(O)(CNC(C=CCC)=O)CCCN(C(=O)C(C(C)C)NC(=O)OCC)C1 c1(C(=O)NC2C(NC(C3C(CCC)C3)=O)CCC2)sc2nccn2c1C C#CC1CCCCN1C(C1(CC=C)CCN(C(=O)CCc2cnoc2)C1)=O C1(C(=O)NCCCCNC(C(c2ccccc2F)(C)C)=O)CC1C1CCCC1 N1(C(CCSCC(C)C)=O)CCC(CNC(C2(Cl)CC2)=O)C(O)C1 CC1CCC(CNC(=O)CC2CC(C)(C)C2)CN1C(=O)CCOCCN(C)C CC1(C)CN(C(=O)CC=O)CCC1C(N1CC(CO)C2(CC2)C1)=O.C(C)(C)(C)N Cc1ccc(CC(N2CCC(N(C(=O)C(C)C3(O)CCC3)C)C2)=O)s1 C(=O)(CC(C)(C)C(F)F)NCc1ccc(C(N2CCCC(N(C)C)C2)=O)s1 N1(C(COc2ccc(C)cc2)=O)CCC(C)C(CNC(=O)C(O)CN2CCCC2)C1 CC1CN(C(c2cscn2)=O)CC(C)C1NC(=O)CN1CCN(C)CC1 N1(C(c2c(C)ccnc2C)=O)CC2COCCC2(NC(c2nn[nH]c2Cl)=O)C1 c1(CC)c(C)c(C(=O)C(C#N)OCC2CC3(CN2)OCCO3)n2ccccc12 c1(CC)ccc(C(CNC(=O)COC(C)C(=O)O)C(=O)OC)cc1 C1(NC(CC=CC)=O)CCCC12CCN(C(c1cc(CC)on1)=O)CC2 C1(c2nc(CC)nn2Cc2cccc(Cl)c2)CCc2nncn2CC1 c1(C(C(=O)N(C)CCNC(c2cn(C(F)F)cn2)=O)(C)F)ccccc1F N1(C(C(=O)N)=O)CCC2(O)CCCCC2C1.CS(=O)(=O)C(CN)C1CC1 C1(C(=O)NCCOCCC=C)CCN(C(=O)C#CC(C)(C)O)CC1O c1(C(N2CCC(NC(C(C=CC)O)=O)C(F)C2)=O)cc(N=S(C)(C)=O)ccn1 C1(NC(C2N(CC)CC2)=O)CC2CC(C1)N(C(c1ccn(C)c(=O)c1)=O)C2 c1(C(N2C(CN(C(=O)C(F)(F)C3CCC3)C)CCCC2)=O)ccc(N)c(Cl)c1O C1(N(C(c2c(C(C)C)con2)=O)C)CCC(NC(c2ccn(C)n2)=O)CC1 N(C1CN(C(C2(CCF)CCOCC2)=O)Cc2ccccc21)C(C=NOC)=O c1(C(=O)OCC)cc2n(n1)CCCN(c1nc(C)nc3c1CCC3)C2 C1(CNC(CS(=O)(=O)NC)=O)CC(C)(C)CN1C(=O)C(=O)C(F)(F)F C1(NC(=O)Cc2c(F)cccc2F)CC2CC1N(C(=O)CCc1ccon1)C2 c1(N2CC(C)C(C)(CO)C2)ncc(S(=O)(=O)NCc2ccns2)cc1Cl CCC(CC(=O)NC(C1CCOCC1)C)NC(C1(COC)CCCC1)=O C1(C(=O)NCc2ccc(C)nc2)(CNC(C(C)OCC#C)=O)CCCCC1 C1(COC(c2cncc(C(C)(C)O)c2)=O)COc2ccccc2O1 Cc1cc(Cl)ccc1C(=O)NCCC(C)N(C)C(C1CCN(C)C1C)=O CCCCCC(F)C(=O)NCCCCCCC(=O)NCC1(COC)CCCC1 C1(CCNC(c2c(C)sc(Br)n2)=O)CCN(C(=O)Cn2cnnn2)C(C)C1 n1(CC(=O)NCC2N(C(c3c(OC)c(Cl)sc3)=O)CC(F)C2)cc(C)ccc1=O N1(C(C(C)c2cccs2)=O)CCC(C)(C)C(C(=O)NC2(C)CC(C)(C)C2)C1 C1(C(=O)NC(COC)C(=O)NCCCC(C)(C)C)CCC(F)CC1 CC1(C)CC(NC(=O)C(C)(C)N2CCOCC2)CCN(Cc2cccnc2)C1 C(CC(C)(C)C)(C(=O)N1CCCCC1CCC(=O)NCCCOCC(F)F)OC c1(C(=O)NCC(C)N(C)C(c2ccc(F)s2)=O)cccc(-n2cccn2)n1 C1(C(=O)NCC2(CN(C(C3(CCC)CCC3)=O)C)CC2)CC2(C1)CC(F)C2 CN1CCC(CN(C(=O)CSc2ccnn2C)C)CC1 N1(C(=O)CCN2CCCCC2=O)CCNC2(CCNCC2)C1 N12C(=O)CC(C1c1cccnc1)NCC(O)C2.O=C(O)C.C1(C)CC1 c1(C(=O)NC(C2CCCN(C(C)=O)C2)C)sc2cc(Br)ccc2c1Cl c1(C(=O)OC)ccc(NC(=O)NCC2(C(=O)OC)COC2(C)C)c(Br)n1 C(=O)(C(C)CC(C)C(C)=O)N1CC2C(C(=O)NCc3ncc(CC)s3)C2C1 CCCCC(C(=O)NC1CCC(CNC(c2c(F)cccc2F)=O)C1)N(C)C N1(C(C2CCN(C(C)=O)C(c3nn[nH]n3)C2)=O)CCC2CC1C(=O)O2 N1(C(Cc2c(C)cco2)=O)CCC(O)C(N(C)C(c2cc(C(C)C)nn2C)=O)C1 C#CC(C(C)C)NC(C1(CNC(=O)CCCOCC)CCCC1)=O c1(C(=O)NC2CCC3CC2CN3C(=O)CCC(F)(F)F)cnc(O)c([N+](=O)[O-])c1 CN1CC2(CCN(S(=O)(=O)CC3CCC4(CCNCC4)C3)CC2CO)C1 c1(-c2cc(C(=O)NCC(C3CCOC3)NC(C=C(C)Cl)=O)no2)ccccc1F CC12CN(N3CCN(C(c4cc(C5(O)COC5)on4)=O)CC3)C(CO)(C1)C2 c1(OC)cccc(CNC(=O)C(c2sccc2I)N2CC3CC3C2)c1 C(CC(C)C(=O)NC(CC1CCCC1)C(=O)NCCc1cnnn1C)=CC N1(C(C(CC=C)(C)C)=O)CCC(C2CCN(C(c3[nH]c(C)nc3C)=O)C2)CC1 Cc1nn(CC(=O)N(C)CCNC(=O)Cc2ncsc2Cl)c(=O)o1 C(C(C)(C(=O)NC1CC(O)C1CC(=O)Nc1ccccc1CCO)OC)OC N1(C(C2C(C)C2)=O)CCN(C(=O)OC(C)(C)C)CC1CF CC(C(=O)NCCCOCCN(C)C(C1(C)CC1C)=O)OC(C)(C)C.C(CO)O c1(C(=O)NCC2N(C(C=NOC)=O)CCN(C)C2)cc(OC)c(OC)c(Cl)c1 C(C(CC1CC1)C(=O)N=c1cc2ccccn2[nH]1)NC(Cc1cc(C)on1)=O C1(CC(=O)NC2(C)CC2)CC(NC(c2ccc[nH]2)=O)C1(C)C N1(C(c2c(CC)cccc2)=O)CCC2(CCOC2)C(CNC(C2(C)CCC2)=O)C1 N1(C(c2c(C)scc2)=O)CCOC(CC(N2CCC(CN=[N+]=[N-])C2)=O)C1 C(C(F)(C(=O)N1CC2CC(C1)C2CO)C(C)C)NC(C(CC)(CO)OC)=O CC1(C)CCCN(C(=O)C#CC2CCC2)C1C(=O)N(C(CO)C(=O)OC)C.CCO C(=O)(C(C)(C)C(F)F)NC1CC(OCC(=O)NC(c2ccoc2)C)C1 N1(CC(O)CF)CCN(CCCNCc2ccncn2)CC1 c1(C(=O)NC23CC(CNC(C4CC4Cl)=O)(C2)C3)cccc(Oc2ccccc2)c1 c1(NCC2(CNC(c3cnn(C(CC)C)c3C)=O)CC2)nccc(C#N)n1 C1(CCC2N(C(CCOCC#C)=O)CCC2)CCCCN1C(C1(Cl)CC1(F)F)=O C1(CCNC(Cc2cc(C)sc2)=O)C(C)CCCN1C(=O)CC1CC2(CCC2)C1 C1(C(N(C)CC2(OC)CCCC2)=O)N(C(=O)C2=CCC(C)CC2)CC12CCCC2 C(=O)(CCCC(=O)N1CC2CC1(C(=O)Nc1cc(C)cnc1O)C2)OCC c1(CC)ncc(C(=O)NC2CCCC2NC(=O)CS(N)(=O)=O)c(C)n1 N1(C(C(CC#C)O)=O)CCN(C(=O)CC2CC(O)C2(C)C)C(C#C)C1 N1(CCN(C)CCC(N2C(C)CCC2)=O)CCC2(CCCN(C)C2=O)C1 C1(C(=O)NC(C(=O)NCC)C)CC1C1CN(C(c2cc(C)c(C)cn2)=O)C1 c1(C(N2C(CNC(c3c(COC)cco3)=O)C(C)CC2)=O)cc(N)c(Cl)c(O)n1 c1(C(C)(C)OC)nc(=NCC(C2CC2)NC(c2cnc3cnccc3c2)=O)s[nH]1 C1(CC)(CC)CC(NC(C2C(Cl)(Cl)C23CC3)=O)CN1C(=O)CC1(CSC)CC1 c1(C2(C(N3CCC(C4N(C(C5CC5(F)F)=O)CCC4)C3)=O)CC2)ccccc1Cl c1(CC(=O)NC2CCCC(n3cccn3)C2)nc2cc3c(cc2[nH]1)OCCO3 C1(CNC(C)=O)CN(C(=O)Cc2ccc(Br)cc2C)CC2(CCC2)O1 c1(C(N(C)CC2(CNC(C(C)n3cncn3)=O)CC2)=O)ccc(CO)s1 c1(C(=O)NC2CN(C(C(CC)SC)=O)CC2C)coc2c(C)cccc12 CC1CN(C(C2(C)CC(O)CN2C(C23CSCC2C3)=O)=O)C(C)C(C)(C)O1 c1(C(N(C2CN(C(c3c(CC)nco3)=O)C2)C)=O)cccc(N2CCNC2=O)c1 C(C)(C(=O)C(F)(F)F)OC(C(CCN(C)C)NC(C)=O)=O C(CC(F)F)(C(=O)NC(c1nnc(C)s1)C)N(C(c1nc(C)oc1)=O)C C1(C#N)(CC(=O)NC(CNC(C(C)OCCC=C)=O)CC)CCCCC1 C#CCCCCC(=O)NC1(C)CCN(C(c2cc(OC)ccc2N)=O)CC1 CC(C(=O)NC1(CC(=O)N(C2CCC2C)C)CC1)c1cc[nH]n1 C1(C)(CNC(c2cc(C)cc(O)n2)=O)COCCN(C(=O)C(C)(O)C2CCC2)C1 N1(c2ccc(C#N)cn2)CCC2(NC(c3conc3C(F)(F)F)=O)CCCC12 C1(NC(c2c(C)ncs2)=O)CCC2CN(C(c3cccc(C(F)F)c3)=O)CC2C1 N1(C(c2c(CC)nccn2)=O)CCCC(NC(=O)CC2CC2CC)CC1 N1(C(C(=CC2CCCC2)C)=O)C(CC(=O)NCC(O)CC(F)(F)F)C2CCCC12 C1(CN(C)C(c2csnn2)=O)CCCCN1C(c1ncncc1Cl)=O c1(NC)ccc([N+](=O)[O-])cc1C(=O)NC1CCC(CNC(=O)Cc2cnns2)C1 N1(C(C(F)=CC)=O)CCN(C(c2cc(C(N)=O)ccc2C)=O)C2CCCCC2C1 N1(C(C(COC(C)C)(C)C)=O)CC2CCC2(NC(c2cccc3sccc23)=O)C1 c1(C(N2C(C)CC(NC(CC3CC(OC)C3(C)C)=O)C2)=O)ccc2c(c1)CCN2 N1(C(CC=CCC)=O)Cc2n[nH]cc2C1C(=O)NOCCC1CC1 c1(C(N2CCC(C)(C)C2)C(=O)NCC(=C)C)ccc2cc(F)cc(Br)c2n1 C1(CNC(c2ccccc2F)=O)CN(C(C2(O)CCC2)=O)CC1(F)F C1(CNC(CCCC#C)=O)CN(C(=O)CN2CCC(O)CC2)CC12CCOCC2 C(=O)(N1CCCc2ccnn21)C12C(NC(=O)CC(Cl)Cl)C3CC1C2C3 C1(NC(CCC)=O)C=CCC(C(N2CCOCC2CC(C)C)=O)C1 C=C=C(C)CC(=O)NC(C)C(C(C)C)NC(c1cc(OC)n(C)n1)=O C1(C(=O)NC(C)(C)CN2CCCC2)(NC(CSCC)=O)CC1(C)C C1(C(=O)OC)CCC(CN2CC(F)CC2C(N2CCC(N3CCC3)CC2)=O)CC1 C(CC(C(=O)NC(C)(C)C1(c2ncon2)CC1)NC(=O)CCN(C)C)=CC S(=O)(=O)(c1ccc(Br)cc1NC1(CO)CCOC1)N1CCCC(N(C)C)C1 c1(N2CCC(N(C(C(CCC)OC)=O)CCC)C2)nnc(C)cc1C(=O)OC c1(C(=O)NCC2C=CCC2)cc2c(F)c(Cl)c(Br)cc2[nH]1 N1(C(c2cc(C(C)C)no2)=O)CCC(C(F)F)(CNC(C2C=CCCC2)=O)C1 n1(CC)nccc1C(=O)NCC=CCNC(c1cnccn1)=O C1(C(=O)NC23CN(C(CCSCC)=O)C(COC)(C2)C3)(OC)CCCC(C)(C)C1 CC(C)C(O)CC(=O)N1CCC(C(=O)NOC2CCN(C)CC2)O1 c1(NC(c2c(OC(C)C)nccn2)=O)cccc2ncnn12 c1(NC(Cc2nc(Nc3ncc(C(=O)OC)s3)sc2)=O)c(Cl)c(C(C)C)nn1C Cn1cc(C(=O)NC2CCCN(C(=O)CC3CC4CC4C3)C2)cc1Br N1(C(c2nnn(C)c2N)=O)CCCC(C2(NC(=O)CC3CC4CCC3O4)CC2)C1 C12(CNC(c3c(CCC)occ3)=O)CCCC1CCN2C(c1cccnn1)=O N1(C(CCC=C=C)=O)CC2(CCN(C(c3cnc(Cl)s3)=O)CC2)C1 N1(C(c2c(C#C)c[nH]n2)=O)CCCOC(CCNC(c2cc(C)co2)=O)C1 O=C(CS(=O)(=O)N1CCCCC1)NCCc1ccc(CNC(=O)C(O)C(F)F)cc1 C#CCC(C(=O)NCC1(O)CCN(C(=O)C(C2(O)CCOCC2)(F)F)C1)C1CC1 c1(C(N2CC(C(C(=O)NC3CC(O)C(O)C3)O)C2)=O)cnc(S)nc1 c1(OC)c(C(=O)NCCCC2CCCN2C(C2C3CCC(=O)C23)=O)cnn1C C1(C(=O)NC(C(=O)Nc2c(OC)ccnc2)(C)C)CC2COCC2C1 CC1CC(C(=O)N2CCC=C(CNC(C3CC(CF)C3)=O)C2)=NO1 C1(C(=O)NCC2OCCN(C(C(C)(C)F)=O)C2)CS(=O)(=O)CC(=O)N1 N1(C(C(C)CC(F)(F)F)=O)CCC2(CC1)CCN(C(C1CC3CCC3C1)=O)C2 C(C1=CCN(C(=O)C(O)CCn2cncn2)CC1)NC(=O)CN1CCCC1=O c1(N2CCC(C)(NC(CCCOCC=C)=O)C2)cc(C)nc2c(C)cnn12 c1(SCC(=O)NC2(CCNC(C=CC(=O)N(C)C)=O)CC2)cccc(Cl)c1 c12nnn(n1)CCOC2.C1(N(C)CCN(C)C)CC(F)(F)C1 C(CCC)(C(=O)N1CCC(N(CCO)C(C2CC(F)C(=O)N2)=O)CC1)=CCC CC(C)(CNC(c1cc(O)ncc1F)=O)CC(=O)NC1CNC(=O)C1(C)C C12(NC(c3cncs3)=O)CCOCC1CN(C(c1ccc(=O)n(CCO)c1)=O)C2 N1(C(C(CC2CN(C(COCC=C)=O)C2)F)=O)CCOC(C(=O)OCC)C1 c1(C(C(=O)NCCOCC)N(c2cc(C)cc(C)c2C)C)cc(Cl)c(F)cc1F C1(C(N(C2CCN(C(C3CCCOCC3)=O)C2)CCO)=O)CC2(C1)CC(F)(F)C2 c1(OC)c(C)cc(C(=O)NCC(O)CCNC(=O)C(C)n2cnnn2)cc1Cl C12(NC(c3cc(C)c(C)o3)=O)CC3CCC(C1C2)N3C(C1CCCN1C(C)C)=O CCCCCC(O)C(C)C(=O)OC(C)C.c12ccccc1N2 Nc1ccc(C(=O)NC2(CNC(C3CC3(F)Cl)=O)CCCCCC2)c(F)c1 C1(C(=O)NCCc2ncc(C)o2)CCCCN(C(c2ccoc2C)=O)C1 N1(C(CCC=CC)=O)CCN(C(C2C(C)(C)C2(C)C)=O)CC1CCOC N1(C(C2C(c3ccc(C)o3)C2)=O)CCCC(CNC(=O)Cc2ccoc2C)CC1 O=C1CC(NC(=O)C(c2cccnc2)NC(=O)CN2CCCC2)CO1 N1(C(C=CCC)=O)CC2COCC2(C(=O)NCc2ccc(C)c(O)c2)C1 C1(C(=O)NC23CCCC2C3)(CC)CCN(C(C2CC(C)N(C)C2)=O)C1 CCCCCC(C)(c1nnnn1-c1ccc(OC)cc1)NCCCc1ccsc1 C(=O)(CCCC(=O)N1CC(C(=O)NCCCCCCF)C(C)(C)C1)OCC CC1CN(C(c2cncnc2)=O)CCCN1C(=O)CC1CCCCCC1(F)F C1(Cn2cc(CN(C(C)=O)C)nn2)CCCCN(C(C2CC2(Br)Br)=O)C1 c1(C(C)CC(=O)NC2CC(C)(NC(=O)CCN3CCC(F)C3)C2)ccc(F)cc1 C(=O)(C1=COCCC1)NC1C=CC(CC(=O)NCC2=NOC(C)C2)C1 c1(C(=O)NC2CCN(c3c(Cl)ccc(C)c3)CC2)nncc2ccccc12 Cc1nn(-c2ccnc(F)c2)cc1CNC1CCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NCC2C(NC(C(C)OCCCC)=O)COC2)nccc(Cl)c1Cl C(=O)(CCCC=O)NCC(=O)NCCOCC.C1(C)(CC)CCCC1 N1(C(c2n(C)ncc2Br)=O)CC2CC(CNC(c3ccc(Cl)c(F)c3)=O)C2C1 C1(NC(C(CC)F)=O)COC2(C1)CN(C(c1ccc(OC3CCCC3)nc1)=O)C2 c1(C(=O)NC2CC3CC2CN3C(c2cccc(=O)o2)=O)cc2c[nH]cnc-2n1 CCCC(CC(=O)NC1C(C(=O)OC)CC1)C(=O)N1CCC(CC(=O)NC)C1 Cc1cc(C(=O)NC(C)(CC2CCCN2C(=O)C2=CCOCC2)C2CC2)ccc1Cl C1(CCC)CN(C(c2ccncc2COC)=O)CCN1C(=O)C(CC1CC1)OC C(C)(CSC)(C(=O)NC1(CSC)CCC1)NC(C(C)OCCC=C)=O c1(C(CN(C(=O)CN2CC3CC3C2)CC(F)F)=O)cccc2c1OC(F)(F)O2 N1(C(CS(C(C)C)(=O)=O)=O)CCC2C(CCCN2C(C2CC(=O)C2)=O)C1 c1(CCC(=O)NC(CNC(CCSC)=O)C(C)C)ccc(C(C)C)cc1 CCC(F)(F)CC(=O)NC1CC1NC(c1ncccc1OCCOC)=O N1(C(c2n(CC)c(O)nc2)=O)CC(CN(C(=O)Cn2nnnc2C)C)C2(CC2)C1 N#CC1(C(N2CCCC(CNC(C3(c4cc[nH]n4)CC3)=O)CC2)=O)CC2(CC2)C1 N1(C(CC2(OCC)CCC2)=O)CCN(C(C2CC2(C)CCOC)=O)CC(C)C1 C1(C(=O)NCC2CCN(C(C(C(C)C)NC=O)=O)CC2C)CC2CCCCN2C1 Cc1ccc(C(N2CC3CC2CN3C(c2ccc(O)nc2)=O)=O)c(C)c1 CCCCC(CCCC)C(=O)NC1CC(C)(NC(C2CC(F)C(=O)N2)=O)C1 C(=O)(C1=CC2C=CC(C1)C2)NCC1(CNC(=O)CN2CCCC2CO)CC1 C1(NC(C(C)(C)C2CCCC2)=O)CN(C(=O)C=CC2CC2)C2(CCOC2)C1 c1(C(=O)OC)cc(C(=O)NCC(c2ccncc2)C)c2cnccc2c1 c1(OCC)ccc(C(N2CCCC2C(C)(C)NC(=O)Cc2ccno2)=O)cc1 CC1=C(C(=O)NC(C)(C)C(=O)NCc2ccn(C(C)C)n2)COCC1 C(CC)(CC)(CCNC(=O)CCC1CCCC(C)(C)C1)NC(COCCC=C)=O c1(CC)cc(F)c(C(=O)NCCNC(=O)CCc2cnc3ncccn23)cc1F CCC(C)(CO)C(=O)NCC1CCN(C(c2c(C)nn(CCCC#N)c2Cl)=O)C1 c1(C(N2CC(C(C)(C)C)C2)=O)c[nH]nc1CNC(=O)CCC1CC1(C)C N1(C(C2(OC)CC2)=O)CC2CCC(C1)N2C(=O)C(c1ccc(OC)c(OC)c1)C CC(C)C(O)C(C)C(=O)NC12CC(CNC(c3cnc(O)cc3O)=O)(C1)C2 N1(C(C2(C(CC)=O)CC2)=O)CCC(C)C(CC(=O)NCC2(C#N)CC2)C1 CCC(CC)CC(F)C(=O)N(CC(C)NC(c1cc(F)c(C)cc1O)=O)C Cn1c(C(=O)NC2CC(NC(=O)Cc3ccsc3)CC2O)cnc1O C1(CCC)(NC(c2cc(COC)cs2)=O)CCCNC1 C=Cc1cncc(C(=O)N(CCNC(=O)C(C)CC(F)F)CCOCCO)c1 c1(N2CCN(C(C)C)CC2)nc(=NCCCCCCO)[nH]c2c(F)cc(F)cc12 C1(C)(C(=O)NC(CNC(c2c(CCC)[nH]cc2)=O)C(C)C)CC(C#N)C1 C1(C(N(C(C)C(=O)N2CC(OC(c3ccccc3)=O)C2)C)=O)CCC(=O)N(C)C1 c1(NC(C2CCN(S(Cc3cccc(C)c3)(=O)=O)CC2)=O)c(C)c(C)nn1C c1(OCCC(=O)OC)ccc(-c2ccccc2N2CCC(O)C2)cc1 N1(C(COC(CC)C)=O)CCC(O)C(N(C(=O)C(C)Cn2ccc(C)n2)C)C1 c12ncc(Cl)c(n1)N(C(c1ccncc1)=O)CCN2C.CC(=O)N(C)C CCCCCCCCOCC(=O)NC(C)(C)CN(C)C(c1cscc1C(C)C)=O CN1CCC(n2cc(C(=O)N(CCCC(=O)OC(C)(C)C)CCO)nn2)C1 CCCC(C1CC1)NC(=O)C(C1CCCO1)NC(=O)CNC(=O)CN(C)C Cc1cc(CNC(=O)C(C2CCCO2)NC(=O)CN2C(C)CCC2C)cc(O)n1 c1(C(=O)Nc2cc(I)ccc2F)n[nH]c2c1CN(C(c1ccc(O)nc1)=O)C2 N1(C(C(N)=O)=O)CCC2(CCCCN(C(C3CC4CC4C3)=O)C2)C1 C#CCCCCCC(=O)NC1CC2(C1)CC2NC(C12CC(C)(C1)C2)=O c1(N(CC(=O)NC)C)nc(C)cc(=NCC2CCCC(CCOC)C2)[nH]1 N1(C(C2(C(C)C)CC2)=O)C(C(N2CCCCC2CF)=O)CCC12CC2 C1(N(C(c2c(C)coc2)=O)C)CN(C(=O)CCCc2csc(=N)[nH]2)CC1O N1(C(c2c(COC)noc2)=O)CCC(C2(NC(=O)C(C)CCO)CC2)C1 c1(N(CC=C)C)nc2c(c(=NCC3(C)CC=CC3)[nH]1)CC(C)CC2 C(C)(CO)(CC(C)C)NC(COC1CC(NC(c2cc(C)sc2)=O)C1)=O Cc1sc(C(N2CC(CNC(=O)C(c3ccccc3)O)C(O)C2)=O)cc1Br C(=O)(C(CCCC)ON=C(C)C)ONC(=O)C(C)ONC(=O)C=CC1CCCC1.C#CCSCC Cc1ccc(C(=O)Nc2c[nH]nc2C(=O)NCCN(c2ccccc2Cl)C)cc1 c1(C(=O)NCC(CNC(C2CC3CCCCC23)=O)OC)cc(O)ccc1F c1(C(=O)Nc2cccc(C(=O)NCCC)c2)cc(OC)c(OC)c(OC)c1 C1(F)(C(N(C(CCCC)C)C)=O)CCN(C(C2(C#N)CC(=O)C2)=O)CC1 N1(C(CC2(C)CCCC2)=O)CCC(NC(c2cc(CO)ccn2)=O)C1C1CC1 c1(C(=O)NCC(C)NC(C2(F)CCOC2)=O)cc(O)nc(N(C)C)n1 C1(C(=O)NC(CCCC)CO)CCCCN(C(=O)CC2CCC(C)CO2)C1 C(C(=O)NC(C1(n2cccn2)CC1)C)(C(C)(C)C)n1cc(C(C=C)O)nn1 C(=O)(C(C)CC(=O)N1CCC(C)C(NC(c2oncc2C)=O)C1)OC N1(C(CC)=O)CC2(NC(=O)CC(=O)NCC3CC3)CC1C2 C(=O)(C(C)(C)CC(C)C)NC(C1CCN(C(Cc2cc(C)c(CO)cc2)=O)C1)C C1(NC(CNC(C(CC)CC)=O)=O)CN(C(c2cn[nH]c2)=O)CC2CC12 c1(C(=O)NC2C(C(N3C(C#N)C4CC4C3)=O)CCCC2)n[nH]c2ccccc12 N1(C(CN(C(C)Cc2cccs2)C)=O)CCN(C)C2(CC2)C1 N1(C(C(CC=C)NC(c2cnc(O)c(F)c2)=O)=O)CCC(C2=NOCC2)C1 C1(SC)CCCCN(C(=O)C(C)(C)C(C)NC(C2CCCC(=O)CC2)=O)C1 N1(c2cccc(CNC(N3CCC(OC)(CO)C3)=O)n2)CCS(=O)(=O)CC1 C(CCCC(=O)N1CC(CNC(=O)C=CCN(CC(F)(F)F)C)C(O)C1)OCC c1(C(=O)NC(C)CCCNC(c2ccoc2C(F)(F)F)=O)nc2ncccn2n1 CS(=O)(=O)c1cccc(S(=O)(=O)NNC(=O)CC2NNC2=O)c1.c1(C(F)CCCN)ccc(I)cc1 C1(C(N2CC(OC)C(NC(C3(CC4CC4)CCC3)=O)C2)=O)CCC(=O)N(C2CC2)C1 c1(OCC(=O)NCCCc2cn(CCn3cccn3)nn2)ccccc1Cl Cc1sc2ccccc2c1C(=O)NCCCN(C(=O)CC1(O)CC1)C(C)C c1(C(N2CC(CC(=O)Nc3cccc(F)c3)(OC)C2)=O)ccccc1OC C1(C(=O)NC2C(CNC(c3cc(C)no3)=O)COC2)CNC(=O)CC1(C)C c1(C(N(C2CCC(NC(=O)CC(C)(F)F)C2)C)=O)cc2ccc(Cl)c(F)c2[nH]1 N1(C(C(CC=CC)C)=O)CCC2(CC2)CC1C(=O)NCC1(CC)CC(C)(C)C1 C1(CNC(C2(CC)CCC2)=O)CCCCN1C(c1ccc(O)cc1)=O C1(C(N(C2CCN(Cc3cc(I)c[nH]3)C2)C)=O)CCCN1C C(C(O)(CNC(C1CCC1NC(=O)C(C)(C1(C)CC1)OC)=O)CO)OC Cc1noc(N)c1C(=O)NCCC1CC(NC(c2cccc(OC(C)C)n2)=O)C1 CC1CC(CNC(=O)CCCNC(C2OC3CCC2C3)=O)CC(C)C1 CCC(O)C(C)(C)C(=O)NCC(C)(C)CNC(C1(c2cccc(F)c2C)CC1)=O c1(C(N2C(CN(C(C3CC34CCC4)=O)CC)CCC2)=O)cnc2c(c1)CCC2 c1(C(C)=O)cnn(C)c1F.c1(C(=O)NCC2CC(OCC=O)C2)sccc1OC(F)F CC1(C#CC(=O)NC2CCCC2NC(c2cc3ccsc3s2)=O)CCCO1 C(=O)(C1=NNC(=O)CC1)N(CCCNC(C1CC=CCC1)=O)CCC c1(C(=O)NCCC2(OC)CN(C(=O)C=C(C)C(C)C)C2)ccc2oc(O)nc2n1 C1(C(N(CCC(=O)N(C2CC3CCC2O3)C)C2CC2)=O)C2CCCCC12 C(=O)(C(C)(C)CO)NCCN(C(=O)CCC1(C)CC1(F)F)CC(C)O C1(CC(=O)NC(C2CCN(C(c3cc(C(C)=O)sc3)=O)C2)C)CCC(=O)NC1 N1(C(CNC(C2(n3cc(C4(O)CCCC4)nn3)CC2)=O)=O)CCS(=O)CC1 C(=O)(C(C)(CC)C(N)=O)N(CCN(C(=O)C(F)C(C)(C)O)CC)CC C1(C(N2CC(C(=O)NCCc3n(C)ncc3)C2)=O)CCCN(c2cccs2)C1 CCCC(CC(=O)N1CC2CC1(CO)C2)NC(=O)C(C(=O)OC)SC N1(C(C(C)n2ccnc2)=O)CC2(CCCCN(C(=O)C=CBr)C2)C1 C1(NC(COCCCOC)=O)CCN(C(c2cn(C(F)(F)F)cn2)=O)C(C)C1 C1(C(=O)NCCOCCCN(C)C(c2[nH]cnc2C#N)=O)CCc2nnnn2C1 c1(C(N2C(C)CC(CNC(COCCC)=O)C2)=O)ccc2c(c1)CNC2=O CCCCCCC(C)CC(=O)NC1(C)CCCN(C(c2cccnc2OC)=O)C1 N1(C(CC(C=C)C)=O)CCCC(COC)(NC(=O)C(c2cccc(C)c2)F)C1 c1(OC)cccc(CC(=O)NC(C)C(C)NC(c2c(C(C)C)n[nH]c2C)=O)c1F C1(C(=O)N(C(C)CC(F)(F)F)C)(NC(C(C)N(C)C)=O)CCCCC1 c1(-n2c(C(C)S(C)(=O)=O)nc(CCC(C)C)n2)ccccc1S(N)(=O)=O C(F)(F)(C(F)(F)F)OCC(=O)NC(C1CCCCC1)CNC(=O)CC1CC12CC2 CCC(CCCC(=O)NC1CC2C=CC1C2)NC(=O)CCn1ccc(C)n1 Cn1nccc(C(=O)NC2CC(CCNC(=O)CCCCc3cnc[nH]3)C2)c1=O CCC(C)CCCCC(=O)N1CCCC2CN(C(c3ccc(C(C)=O)s3)=O)CC12 N1(CC(=O)N(C2CCC(NC(=O)CSc3ccccc3)C2)C)CCCNS1(=O)=O c1(SC)ccc(C)c(C(=O)NCCC2CCCN(C(=O)Cc3c[nH]nc3C)C2)c1 CC(CC(=O)NCC(C)N(C)C(C1CSCCS1)=O)NC(c1ccccc1)=O C1(C(N2C(CNC(c3c(CC)con3)=O)CC(O)C2)=O)CCCCC(=O)N1 C1(C(N(C2CN(C(c3nc(NC(C)=O)sc3)=O)C2)CCO)=O)CC(=O)NC1(C)C N1(C(c2cc(C)c(F)cc2)=O)CCN(C(=O)Cc2c[nH]nc2O)C(C)C1C c1(C(=O)NCC(C(C)(C)C)NC(C2C(=C)C2)=O)ccc(OC)c(C)c1OC c1(-c2cccc(C(=O)NCC(=C)CC(F)(F)F)c2)nc2ccccc2o1 C1(NC(c2cc(OC)no2)=O)COCCN(C(=O)CSCc2csc(C)n2)C1 CCC(CC)(C(=O)N1CC=CC1C(=O)NCC(CC(=O)OC)OC)OC CCC(CC)CCNC(=O)CNC(C1CC1C)=O.C(=O)(CCOC)NCC1CCC1 Cc1cc(Cl)c(C(=O)NC(C2CCCCN2C(c2cc(=O)cc(Cl)[nH]2)=O)C)cn1 C1(N(C(=O)COCCF)C)CC(O)CN(C(=O)C(F)(F)c2nccn2C)C1 c1(OC)ccc(O)c(NC(C2CN(C(C3(C)CCCCC3)=O)CCS2)=O)c1 c1(C(=O)NCC2CN(C(C3CC4CCC3O4)=O)CC2O)cc2cccnn2n1 Cc1cc(C(=O)NCCOC2CCN(C(=O)C(C)CC3CCC3)C2)co1 N1(C(c2c(OC)csc2)=O)CC=C(C(=O)N2CCC(C3CCCO3)C2)C1 C1(NC(C(CC)OCC)=O)CCC2(CC1)CCN(C(c1cc3occc3s1)=O)C2 N1(C(C(C2CCN(C(=O)C(F)(F)CO)C2)C)=O)CCC2C(=O)NCC2C1 N1(C(c2c(C)nc(CC)o2)=O)CCN(C(c2cc(C)cnc2N)=O)C(C(C)C)C1 O=C1COCCN1CC(N1CC=CC1C(=O)Nc1cnsc1)=O C1(C(=O)NC(CN(C(c2csc(C)n2)=O)CC)C)COC2COCC2O1 N1(C(C(=O)NC(CC)C)CC2CCCCCC2)Cc2ccccc2OC(C)(C)C1 c1(CC(N2CC3C(N(C(C=C(C)Cl)=O)C)C3C2)=O)ccc([N+](=O)[O-])cc1 C1(F)(C(=O)NC(CNC(CCSCCCC)=O)CC(F)(F)F)CC12CCCCC2 CC1C(C(=O)NCC2(O)CC(CNC(C3(C#N)CCCO3)=O)C2)=NOC1C c1(C(=O)NC2CCC(NC(C(CC#C)C3CC3)=O)CC2)[nH]c2ccccc2c1Cl c1(C(=O)NC(C2N(C(c3c(C)onc3)=O)CCC2)C)c(F)ccc2n[nH]cc12 CC1c2cc(F)c(F)cc2CCN1C(=O)NC(C)Cc1ccccc1F c1(C(=O)NC(C)CCNC(=O)CSc2nncs2)coc2c1C(=O)NCCC2 N1(C(C2(c3cc(C)no3)CC2)=O)CCCC2CN(C(C3CCCO3)=O)CCC12 C1(CCOC)CN(C(=O)Cc2cn[nH]c2)CCN1C(c1cnc(C)n1C)=O C1(NC(C2C(OCC)C2)=O)COCCN(C(C2CC(n3ccnc3)C2)=O)C1 C1(NC(C23N(C(C4COC(=O)N4)=O)CC(C)(C2)C3)=O)CCn2ncnc2C1 C1(CN(C(=O)CCF)C)CN(C(C2CCCCN2CC(F)F)=O)CCO1 N#CC1(C(N2CCOC(CC(=O)Nc3cncc(F)c3)C2)=O)CCCC1 c1(NCCCc2onc(C)n2)ncnc2cc(C(F)(F)F)ccc12 c1(C(N(C2CCN(C(CCCNC(=O)OCC)=O)C2)C)=O)cc(CC)ccc1F C1(O)(CN(C)C(c2ncsc2-c2ccccc2)=O)CCCC(C)(C)C1 N1(C(C23CC(C)(OCC2)C3)=O)C2CCC1CN(C(C1(C)CCCS1(=O)=O)=O)CC2 N1(C(C(CC=CCC)C)=O)CC(NC(c2c(C(F)F)cnn2C)=O)CC(F)C1 C(C)(CCCCNC(C1CC1c1cccc(OC(F)F)c1)=O)NC(C=CCC)=O Cc1c(Cl)sc(Cl)c1C(N1CC(C(=O)NC23CC(C(C)(C)C)(C2)C3)CC(O)C1)=O N1(C(Cc2cc(C)sc2)=O)CCC(CCNC(C2CCC23CCC3)=O)C(F)(F)C1 C(=O)(C1Cc2ccc(F)cc21)N1C(C)C(C)N(C(=O)CCN(C)C(C)=O)CC1 c1(C(=O)NCC2C(NC(c3c(C)csc3)=O)C2)sc2nc(C)nc(C)c2c1C c1(C(=O)NC2CN(C(c3c(C)nccn3)=O)CC(F)C2)coc2ccc(O)cc12 CCC(O)C(C)(C)C(=O)N1C2CC1CN(C(C1CCCN1C=O)=O)C2 C(=O)(C(C)(C)C(C)O)N(CCN(C(CCCn1ncc(C)c1)=O)C(C)C)C C(=O)(C1=CC2CCCC12)NCCNC(CC1C(C)(C)CCCO1)=O N1(C(CN2CCC(OC)C2)=O)CCC2CN(C(c3n[nH]c(C)c3C)=O)CCC2C1 c1(CNC(C(c2ccoc2)NC(C2OC3CCC2C3)=O)=O)cnc2n1CCC2 c1(C(=O)NCCC(C)CCNC(=O)C(C)(F)C(C)(C)F)cccc(S(C)(=O)=O)c1 CC1OC(C)(C)OC1(C)C(=O)N(CCNC(=O)CC1CCCC(=O)N1)C1CC1 c1(C(=O)NC(C2(C(=O)NCCNS(C)(=O)=O)CC2)C)cc([N+](=O)[O-])cs1 C1(C(N2C(CNC(Cc3ccc(COC)cc3)=O)C=CC2)=O)CC2C(C1)C2(C)C c1(C(=O)NC2C(CNC(c3on(C)c(=O)c3)=O)CCC2)cccc2oc(=N)[nH]c12 c1(C2(N)CCC2)cccc(S(=O)(=O)NC2(C3CCCCC3)CC2)c1 N1(C(c2ocnc2COC)=O)CC(O)CC1C(=O)OC C1(C2(O)CCN(C(c3cnncc3O)=O)CC2)(NC(CCCCC=C)=O)CC1 c1(C(N(CCNC(C(C)NC(CC)=O)=O)C)=O)cccc(C#CCO)c1 C1(NCc2nnc(CC)s2)CCOc2cc(Br)ccc2C1 c12ccc(c(F)c1)[nH]2.C(c1cccc(OC(F)F)c1)=CC(=O)NCC N1(C(CCc2n(C)ncc2)=O)CC2CC2(CNC(c2cnc(N(C)C)o2)=O)C1 C1(CC(N2CC(C)OCC2)=O)Cc2ccccc2CN1Cc1cccc(O)c1 N(C1CCc2c(Br)ccc(C)c21)C(c1cc(C)on1)C N1(C(c2nccc(CC)c2)=O)CC2CC1CCN2C(C1CC1(Cl)Cl)=O Cn1cnc2sc(C(=O)NCC(CNC(=O)Cn3cnnn3)C(F)(F)F)cc12 CC1CCN(C(c2cc(Cl)sc2Cl)=O)CC1CNC(=O)CCC(C)(C)O c1(CC)cccc(F)c1C(N1CC(F)(CNC(=O)CCNC(C2CC2C)=O)C1)=O c1(CNc2nccc(-c3cccc(C=C)c3)c2)c(C(F)(F)F)cccc1[N+](=O)[O-] N1(Cc2cncc(C)n2)CC2CCN(C(=O)Cc3cc(Br)ncc3F)C2C1 C1(C(N(CCOC)CCNC(=O)CC=CC(C)(C)C)=O)CC(C)=NO1 N1(C(C(C)(C2CCC2)OC)=O)CCN(C(=O)CC2CCCC(OC)C2)CC1C CCCC(C)(C)CC(=O)NC(CC1CC1)CC(=O)NC1CCC(F)(F)CC1 C1(C(=O)NC2CC(O)(CNC(c3ccc(C)cc3)=O)C2)(CSC)CC(F)(F)C1 Cc1nc2cccc(C(N3CCN(C(C4CCC(C)(C)CC4)=O)C4CC34)=O)n2n1 CC1CC(=O)NCC1C(=O)NCc1c[nH]nc1C(N1CC=CC1(C)CO)=O c1(CC(CC)OC)ccc(C(C)(C)OC(c2cnn(C(F)(F)F)c2)=O)cc1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(C1N(CCC)C(=O)CC1)=O)(CC)CC CC1=C(C(=O)NCC2CC2NC(C2(CC3CC3)CCC2)=O)Cn2ncnc2N1C N12CCN(CC1)C(=O)CCN(C(=O)C=CC1CCCO1)C1(CC1)CC2=O.COC Cc1nn(CC(F)F)cc1C(=O)N(C1CCCN(Cc2ccc(F)cn2)C1)C c1(C(=O)NC2CCN(C(c3c(C)cc(CO)o3)=O)CC2)c(C)c(C)cc(C)c1C C1(F)(CNC(C2(C)ON=C(C)C2)=O)CCCN(C(=O)CC2CC3(CCC3)C2)C1 CCCC(C)(CCC)C(=O)NCC1CCCCC1C(=O)NCc1ncnn1C CCC1=NOC(C(N2CCCC2CNC(c2cncc(O)c2)=O)=O)C1 C1(C(=O)NC2C(NC(c3c(C)sc(Br)n3)=O)C2)CCC(C2CC2)CC1 C(=O)(CCCCCCS(N)(=O)=O)NCCC(C)NC(C1CSCCS1)=O C(CCC(=O)NC(C)CC(C)NC(=O)CSCCOC)=CCC=C C=C(CNC(c1cnn(C(C)(C)C)c1)=O)CCNC(=O)CC1OCCC1C N1(C(CC2C(C)=NNC2=O)=O)CC2CCCC2(NC(c2c(F)cccc2F)=O)C1 N1(C(C(C)C2CCC2)=O)CC2CC1CN2C(c1cn(CC(F)(F)F)nn1)=O c1(C(=O)NC(CNC(c2c(SC)scc2)=O)C(C)C)cc2scnc2[nH]1 c1(C(C)C)noc(C2CC2C(=O)NCCC(F)Cn2cc(C3CCCC3)nn2)n1 C1(N(C(Cc2cc(COC)on2)=O)C)CCN(C(c2cc(C)no2)=O)CC12CC2 c1(C(N(CC(CN(C(=O)CSc2nc[nH]n2)C)O)C)=O)cnc2[nH]nc(O)c2c1 C=CC(CC)C(=O)N1CC(C)(OCC(=O)NC(C)Cc2ccccn2)C1 C=CC(C)(C)CC(=O)NC(C(N1CCCCC(COC)C1)=O)C1CCC1 C1(C(=O)Nc2ccc(NC(c3cscn3)CC)cc2)CCCC2(CNC(=O)C2)C1 c1(C(=O)NC2(CC#C)CCC2)cccnc1CNC(C1CC12CC2)=O C1(CC(N2CCC(O)(CN(C(Cc3cc(C)on3)=O)C)C2)=O)COC(C)(C)CO1 N1(C(=O)C(c2ccccc2I)C23CC(C2)C3)CCN(Cc2ccccc2)C(=O)C1 C1(CNC(CCC#CC)=O)CC2(CCN(C(c3ccc4cc[nH]c4c3)=O)CC2)C1 c1(CN(C(=O)CC2(CO)CC2)C)cccc(CNC(=O)C=CC2CCOC2)c1 CC(=O)CCN=C(NCc1cc(F)ccc1Cl)N(C)Cc1ccc(Cl)s1 N1(C(C(C)(C)n2ccnn2)=O)C2CC=C(C(=O)NCCCn3cccn3)C1CC2 c1(C2N(CCC#N)CCC2)ccc(Br)c(Cl)c1 C1(C(=O)NC(c2nnnn2C)C)(NC(C2CC=CC(O)C2)=O)CCC(C)(C)C1 c1(C(=O)NC2CN(C(CSCCC)=O)C(C)(C)C2)cnn2c1CC(C)CC2 c1(OC)ccc(C(O)CNC(=O)NCC23CC(C(=O)O)(CO2)C3)cc1 N(C(=NCCCN(S(C)(=O)=O)C)NCC)C1CCC(SC)C1.C(C)(C)(C)OC(=O)OC C1(N(C(C(CCCC)N(C)C)=O)CC)CC2CCC(C1)N2C(=O)Cc1ccco1 c1(C(=O)NC(CC(C)NC(C2CC2(Cl)Cl)=O)C)ccc(=O)n(-c2ccccc2)n1 C(C(F)CCNC(=O)NC1(n2cc(CO)nn2)CC1)NC(=O)OC(C)(C)C C(=O)(C1CCCc2c(O)cccc21)NC(C)(C)CCCNC(c1ccc[nH]1)=O N1(C(=O)NCc2n(C)c(Br)cn2)CC2CN(C(=O)OC(C)(C)C)CC2C1 CCCC(C(=O)NCC(O)CCNC(c1sc(Cl)c(Cl)c1C)=O)C(C)C CC1(C)C(NC(C23CCC(CC2)C3(C)C)=O)CC1N=c1[nH]ccnc1F C1(NC(c2c(COC)cccc2)=O)CCN(C(=O)C(Br)=C(C)C)CC1C C1(C)(C(=O)NC(C(=O)Nc2cn(CC=C)nc2)COC)CNC(=O)C1 N1(C(C2CC(=C)C2)=O)CC2CC2(CNC(c2ncoc2-c2ccco2)=O)C1 C1(C(=O)NC2(CF)CCN(C(C(C)NC(CC)=O)=O)C2)CCC(F)(F)C1O c1(C(N2CCC(CC=C)(NC(c3ccnn3C)=O)C2)=O)[nH]c2ccccc2c1Cl Cc1cc(C(N2CC(CCNC(=O)C(C)CS(C)(=O)=O)C2)=O)c2oc(C)nc2c1 N1(C(CC2(SC)CC2)=O)CC2(CCC2)CC1CNC(=O)CN(CC(C)(C)C)C c1(C(=O)NC2CN(C(C3(CC#C)CCCO3)=O)CC2O)c(C)oc(C)c1C N1(C(c2c(CC)csc2)=O)CC2(CC(C(=O)N(C(C)CC(C)C)C)CO2)C1 c1(C(=O)NCC(CN(C(c2ccn(CCCC)n2)=O)C)C)oc(C)cc1C N1(C(C2CCC(OC)CC2)=O)CC2(CO)CC1(C(=O)NCC1(C(N)=O)CC1)C2 c1(C(=O)NCC(O)CCNC(C2(n3nccn3)CC2)=O)ncccc1F c1(C(N(CCNC(CCC=C(C)C)=O)C2CC2)=O)cc(OC(F)F)cc(N(C)C)c1 C1(NC(CC(C)C)=O)CC(NC(c2coc(C(=O)OC)c2)=O)C12CCC2 N1(C(C(C)n2cccc2)=O)CCC2(C=C(C(=O)NCC3C(CO)C3(F)F)C2)C1 c1(OCC)ccc(C(N2CC(F)CC2CN(C)C(C2(C)CC2C)=O)=O)cc1 N1(C(CCCCSC)=O)CCC2(NC(=O)C=Cc3ccc(N(C)C)cc3)CC2C1 C=CCC(C)(CC)C(=O)N(CC(C)N(C(=O)CNC(=O)C(C)CC)CC)CC c1(OCCn2c(C(C3CCOC3)NCC3C(=C)C3)nnn2)ccc(C(F)(F)F)cc1Cl C1(C(=O)NCC(C(C)(F)F)Cl)C2CC3C(C2NC(=O)Cc2ccc(O)cn2)C13 C1(NC(c2cnn3cc[nH]c23)=O)CC2CN(C(c3ccc(O)c(Cl)c3)=O)CC12 C#Cc1cccc(CC(=O)NC(C)CCNC(=O)Cc2ccccc2F)c1 c1(NC)cncc(C(N2CC(C(N3CCC(F)(F)C3)=O)C(C(C)C)C2)=O)c1 c1(NC(C23N(C(=O)CNc4cccnc4)CCC2C3)=O)cncc2ccccc12 n1(CC)ncc(Cl)c1C(N1CC(OC)C(NC(c2cccc(C)c2)=O)C1)=O N1(C(CNC(C(C)(C)C)=O)=O)CCCC(NC(c2ccsc2C#N)=O)C1 Cn1c2ccccc2n(N2CCCC(CNC(=O)C(F)(F)F)C2(C)C)c1=O C1(CC(=O)NC(C)C)C2CCC(C2)N1C(=O)Cc1cccnc1 c1(C(=O)NCC2(NC(C34CC(F)(C3)C4)=O)COC2)ccc(SC(F)(F)F)cc1 c1(C(=O)NCC2N(C(C(C)SC)=O)CC(F)C2)c(O)nnc2c1COCC2 CC(C)CC(C)NC(=O)CNC(C)(C)CNC(=O)CCNC(C1CCCC1)=O N1(c2ncc(C(=O)OC)s2)CCCC(N(C(C2CC23CCOCC3)=O)CC)CC1 Cc1nc(C)c(NC(=O)NC2CN(C3CC(C)OC3=O)C2)s1 c1(CCC(=O)NCC(C)CNC(=O)C#CC2CC2)ccc2ccccc2c1 N1(C(c2c(CC)ccs2)=O)CC2CCC1CN2C(=O)Cc1cccc2nonc12 c1(C(N2CCC(NC(c3coc(Cl)c3)=O)C2)=O)cc2ncccc2cc1Cl C1(NC(C2(CC)CC2)=O)CCCCN(C(=O)C(C)N(CC(F)(F)F)C)CC1 C=CCC(CNC(=O)C=CC(C)(C)C)NC(c1cnn(C(F)F)c1)=O c1(C(=O)NC(CC)CNC(C2CC3CC3C2)=O)cnc2scc(C)n2c1=O Cc1cccc2cc(C(=O)N(CC(C)N(C)C(C3CSCC(=O)N3)=O)C)cnc12 N1(C(c2ccc(CC)s2)=O)CCN(CCNC(=O)C(c2ccc(F)cc2)O)CC1 C1(C(NOCC2CC(=C)C2)=O)CC=CCN1C(=O)C(C1CC1)OC Cc1cc(C)c2[nH]c(C(=O)NC3CC4CC3N(C(c3csnc3C)=O)C4)cc2c1 CC(=O)C(C)CC(C)C(=O)N1C(C)CC2CN(C(=O)C(CO)C(F)(F)F)CC12 C1(NC(C(C)=C2CCC2)=O)CCN(C(=O)C(=O)C(F)(F)F)C12CCC2 C1(NC(CCCOCC=C)=O)CCOCC1NC(C12CCC(CC1)O2)=O N1(C(c2nccc(CC)c2)=O)CC(C)C(NC(c2cocc2C)=O)C(C)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(CNC(=O)Cc2nccn2C)C(C(F)(F)F)C1 N1(C(C(C)OCC(F)(F)F)=O)CCN(C(=O)CC2CC=CCC2)C(C(C)(C)C)C1 C(=O)(N=c1[nH][nH]c2c1CN(C(=O)CCc1cccc(O)c1)C2)c1c(C)nsc1 c1(C(C(=O)N(CC(C)NC(C(CC)=CC)=O)C)C)ccc(C#N)cc1 c1(-c2ccc(C(=O)NC3(C)CN(C(C(C)CSC)=O)C3)s2)c(Cl)cccc1Cl C(CCCC(C)NC(c1conc1C1CCC1)=O)NC(c1cc(CC)no1)=O C1(NC(C2CCC(n3cc(-c4cn(C)nc4)nn3)C2)=O)CC(C)(C)C(=O)O1 c1(C(=O)NC(C(=O)NC(CC=C)CC(F)F)c2ccoc2)ccn2ccnc2c1 c1(C(=O)NC(C)CC(C)NC(c2ccc(C3CC3)s2)=O)cc2nc(=O)ccn2[nH]1 c1(-c2cc(C(N(C3CCC(NC(C4CC(=C)C4)=O)C3)C)=O)sc2)ccc(F)cc1 C12CS(=O)(=O)CC1CC(=O)N2.C1(C)(OC(C)=O)CN(C(C)C)C1=O C1(C(=O)NCCc2cc(C)ncc2)CN(C)CCN1C(=O)CCC1CCOCC1 c1(C(=O)NC(c2c(C)noc2C)C)cc2ccccc2c([N+](=O)[O-])c1N C(=O)(C1=CC2(CCOCC2)C1)N1CCN(CCNC(=O)CC2CS(=O)C2)CC1 c1(CN2C(C(=O)NC(CC#C)C(=O)OC)(C(=O)NC)CCC2)ccc(C)c(O)n1 C#CC1(NC(C2(NC(=O)C(C)CC)CC(F)C2)=O)CCOC1 C(=O)(C(F)(F)C(F)(F)C(F)F)N(CC(CC)NC(c1c(CC)cc(F)cc1)=O)C c1(C(N(CC(C)N(C(C2=NOC(C)C2)=O)C)C)=O)c(Br)ccc(F)c1N C1(NC(C(C)NC(C)=O)=O)CC(F)(F)CC1NC(=O)CC1(C)OCCO1 CCC(O)(CC)CCNC(C=CC1CCCN1C(=O)C(c1cnn(C)c1)=O)=O C1(CNC(CC=CC=C)=O)CC2CN(C(C3(c4ccc(C)s4)CC3)=O)CC12 N(C1CCCc2c1cnn2CC)C(CCCC)(C)C(=O)OC c1(C(=O)NCCC2CN(C(C(CCC)(C)CC)=O)C2)n[nH]c2ccc(OC)cc12 N1(C(C(C)=CC)=O)CC(C2CCN(C(=O)Cc3ccc(O)cc3Cl)CC2)C1 N1(C(CCCSCC=C)=O)CCC2(CC(C3C(=O)O3)C2)C1.C(CCSC)OC CCC(C)(C(=O)N1CCC(C(C)(C)NC(c2coc(COCC)n2)=O)C1)OC C1(CC(=O)NC2(C3CCCN3C(=O)C(O)Cc3cnc[nH]3)CC2)CC=CCC1 C(=O)(CC1CCCc2c(O)cccc21)N1C2C(NC(c3ccccc3)=O)C(C2)C1 c1(C(=O)NC2(CC=C)CN(C(=O)CC3CCCCC(=O)N3)C2)cc(F)ccc1C N1(C(C=CC)=O)CCC(CCNC(C2(C(N)=O)CCC2)=O)C(NC)C1 c1(CN(c2ncccc2OC(F)(F)C(F)(F)F)C(C(CC)C)=O)ccc(NC)cc1 C(=O)(C1OCCc2c(Br)cccc21)NC(CCNC(CCC)=O)C(C)C c1(CCC(=O)NC2CC(N(C(C3C(C(=O)OC)CC3)=O)C)C2)ccc(F)cc1 c1(C2C(C(=O)NC(CN(C(C(F)=CCC)=O)C)C)C2)csc(Br)c1 N1(C(C(C)N2CCC2)=O)CC2CCCC1C2CNC(c1ncccc1Cl)=O C(=O)(C1CCc2c[nH]nc21)N1CCC(NC(C(n2ccc(C)n2)C)=O)C(F)C1 N1(C(CC(C)CF)=O)CCC2(CCOCC2)C(CNC(c2coc(CO)c2)=O)C1 n1(CCCC(=O)N(C2(CCO)CCCCC2)C)cnc(C#N)n1 c1(C(N(C)CCN(C)CCc2ccccc2)=O)ccccc1 C12(CNC(Cc3cc(C)[nH]n3)=O)CCC1CN(C(c1cnn(CC(F)F)n1)=O)C2 N1(CC)CC(C(N2CC(C(O)C(=O)N(C)CC3CCCS3)C2)=O)CC1=O N1(C(=O)C=Cc2ccsc2)CCCC2(C1)CN(C(C1C(F)(F)C13CC3)=O)C2 CN1CCCCC1C(N1CCCC(CNC(=O)CCCN2CCCCC2)C1)=O Cc1[nH]c(=N)sc1C(=O)N(C)CCNC(C1(n2cncn2)CC1)=O N1(C(C(=O)NCC(=C)C)c2nccs2)CCCCC(CC(=O)OC)C1 c1(C(=O)NC2CC(C#N)C2)cccc(CNC(=O)CN2CCNC2=O)n1 N1(Cc2nc(C)sc2)CCC2CN(S(=O)(=O)c3ccccc3C(=O)O)CC2C1 C1(C(N2CCC(CNC(c3c(C)scn3)=O)C2)=O)CCNC(=O)C1 c1(CCC(C)C)ccc(CN(C(=O)C(=O)NC2CCCC2CN)C)cc1 C1(C(=O)NC(c2ccccc2)CC)CCCN1NC(=O)C(C)OCOC CC(C)CCC(=O)C(=O)NC(C)CC(C)NC(C1CCCC(C)CC1)=O N1(C(C=CC(C)(C)SC)=O)CC2CCC2(CCNC(c2nc(C)ccc2F)=O)C1 Cc1cc(C(=O)NCC23CCC2CCN3C(=O)CCC(C)(C)C)nc(O)n1 CC(CCC(=O)NCC1CC(C#N)C1)NC(=O)CCc1nccn1C C12(C(N(CCCCN(C)C(C3COC(=O)O3)=O)C)=O)COCC1C2(F)F n1(CC)cc(Br)cc1C(N1CCCC1C(C)NC(C1CCC(O)C1)=O)=O Cn1c(C(N2CC3CC(NC(c4ccc(F)cn4)=O)C2C3)=O)cc2ccccc12 c1(C(=O)NCC(c2ccc(OC)cc2)NC(=O)CSC2CC2)c[nH]cc(Cl)c1=O C(=O)(C#CC1(C)CCCO1)NCC(CNC(Cc1c(F)ccc(C)c1)=O)CO Cn1nncc1NC(=O)CC1(C)CCN1C(c1ccon1)=O CC1(C)C(NC(c2ccc(Br)o2)=O)CCN1c1ccc(C#N)nc1 N1(C(COCCOCC)=O)CC2CCN(C(=O)C(c3ccc(F)c(C)c3)(C)C)CC12 O(NC(=O)CCCCCNC(C1(C)CCCC1O)=O)CC(=O)N(C)C C(C(=O)N(C1CCN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1)C)(C(C)C)OC N1(C(CCC)=O)CCCN(C(c2ccc(OC(C)CC)cc2)=O)CCC1 C1(CNC(N2C(c3cc(C)cc(C)c3)CCC2)=O)CCCC2(CCC2)C1O N1(C(C(C2CCCC2)NC(CC(C)(C)OC)=O)=O)CCC(O)C(C)C1 N(C1CCCc2ccoc21)Cc1cnc(CC(C)C)s1 Cc1noc2cc(C(=O)NCC(O)CCNC(=O)CS(=O)(=O)N(C)C)ccc12 N1(C(N(C2CC2(F)F)CC)=O)CCCCC1CN c1(C(N)=O)ccccc1S(=O)(=O)N1CC(CC(F)F)C1 O=C1OC2CC(C(=O)NC3CCCN(C(c4ncc5[nH]ncc5n4)=O)C3)CC2O1 N1(CCC)CC(CNCC2CCOCC2OC)CC1=O CC1CC(C(=O)NCC(C(C)(C)C)NC(=O)CC(C)C2CCCO2)CC1 c1(CC(C)C)n[nH]c(=NCC2CCC(NC(=O)C(O)CCN(C)C)C2)s1 c1(C(=O)OCC)coc2cc(C(=O)NC3CCN(C(C4CC4C(F)F)=O)C3)[nH]c12 C(=O)(CC1=CCN(C(c2cc(C#N)cs2)=O)CC1)N1CCC(C)(COC)CC1 C1(CCN(C(COC(c2ccccc2)CCC)=O)C)CCCCO1 c1(-c2cn(C3CCN(C(=O)CC4CCC(C)(C)C4)C3)nn2)cccc(C(C)C)n1 c1(NC(C(CC=C)CNC(C2CC(CC)=NO2)=O)=O)cccc2[nH]ccc12 C1(NC(CCCN(C)Cc2c(C)ncs2)=O)CCCN(C(c2ccoc2)=O)CC1 C1(C(=O)NCCCCC2(NC(C(CSC)O)=O)CC2)CCn2nccc2C1 C#Cc1ccc(C(N2CC(CNC(C3CC(SC)C3)=O)C(C)C2)=O)cc1 c1(C(=O)NC(C(C)NC(c2cc(C)nn2C)=O)CO)c(O)cccc1F C1(C(N2CCC(=CCNC(CCC(C)OCC)=O)CC2)=O)CC2(C1)CC(F)C2 N1(C(C2C(CCC)C2)=O)CCOCC1CCNC(=O)CSc1nnnn1C c1(NC(C(C2CC2)OCC)=O)c(NC(C2CC(OC)CN2C(C)=O)=O)sc(C)c1C N1(C(C2N(CC)CC2)=O)CCN(C(c2cnc(F)c(F)c2)=O)CCC1C C1(n2cc(CC)nn2)CC2CCC1(NC(=O)CSN)C2.c1(OC)ccc(C)cc1 C(=O)(CCCCCCCBr)NCc1nccc(C(N2C(C#N)C3CC3C2)=O)c1 c1(C(N2CCC(NC(c3c(CC(N)=O)occ3)=O)CC2)=O)ccn2cnnc2c1 C1(NC(=O)Cc2nc[nH]n2)CC2(C1)CN(C(=O)C(F)CC1CCCC1)C2 N1(C(c2nc(CCC)sc2)=O)CCC(C)C1CNC(c1cnc(C2CC2)s1)=O Cc1nc(C2CC2)[nH]c1C(=O)NCCC(C)CCNC(c1ncsc1C1CC1)=O Cc1coc(C(=O)NCCC(C)(C)NC(c2coc(Cn3cccn3)c2)=O)c1 c1(C(=O)NC2CC(c3cn(CCOCC)nn3)CC2O)cnc(C)nc1C C(CCNC(C1(N(C)C)CC1)=O)(C(C)C)NC(C(C)=C1CC1)=O c1(OC)cc(Cl)c(C)cc1NC(=O)C(=O)Nc1nc(C(c2ccccc2)O)cs1 N1(C(c2ccc(CC)s2)=O)CC2(CCNC(C3(c4cc[nH]n4)CC3)=O)CCC1C2 CC(C)CCCC(=O)N1CC2C(CC(=O)NC3CCCCC3O)C2C1 c1(C(C)(C)C)nc(=NCC2CCCCN(C(c3ncncc3Cl)=O)C2)s[nH]1 N1(C(C=COCC)=O)CC(C2CCCCN(C(c3c(C)ncn3C)=O)C2)C1 c1(CCC(=O)N(CCN(C(=O)CN2CCNC(=O)C2)C(C)C)C)cccc(O)c1 N1(C(c2cc(C(C)=O)on2)=O)CC=C(CNC(c2cc(C)cc(C)n2)=O)CC1 C1(NC(CCN(C)CC)=O)CC12CCN(C(c1c(OC)ccc(Cl)c1Cl)=O)CC2 Cc1cc(C#N)ccc1C(N1CCC(NC(=O)CSCCN(C)C)C1)=O N1(C(c2cc(Br)co2)C(=O)Nc2ccccc2)CCCC(N2CCCC2)C1 C1(C(N2CC(C)C(NC(c3ccc4oncc4c3)=O)C2)=O)CCC(N=[N+]=[N-])CC1 c1(C(N(CC(C)N(C(Cn2nc(C)c(C)c2C)=O)C)C)=O)cccc([N+](=O)[O-])c1 N1(C(C(Br)=C(C)C)=O)CCCCC1CNC(=O)CC(O)C1(CO)CCC1 N1(C(Cc2c(C)scc2)=O)CCCOC(CCNC(c2ccc(Cl)cc2F)=O)C1 C1(COC)(NC(c2cnn(C3CC3)c2C)=O)CCN(C(=O)COCC(F)F)CC1 N1(C(c2noc3c2CCCC3)C(=O)NCCC)CCc2c(C(C)C)cccc2C1 CCC(C)C(O)C(C)C(=O)N1CCC(c2cccc(F)c2)C1 C1(C(=O)NCC(c2ccc(CC)cc2)=O)CCC(=O)N(C)C1 c1(OC)cnc(C(N2CCCC(O)(CCNC(=O)Cc3ccoc3)C2)=O)c(F)c1 N1(C(C(=O)NCCC)CC(C)SC)CC2CCC(C1)N2c1ccccc1 c1(OC)nc(C)ccc1C(=O)NCc1ccsc1C(=O)NCC(CO)SC c1(OC)c(CN2CC(Oc3cccc(C(F)(F)F)c3)C2)cc(Br)cc1F C(=O)(CC(C)(C)C(F)F)NC1COCCN(C(C2(OC)CCOC2)=O)C1 c1(OCC)ccccc1C(=O)NCC(O)CN(C(=O)CC1CC1(C)C)C C(C(C)(O)CC(=O)N1CC(O)CC1C(=O)N(C)CCC1CCC1)OC N1(C(=O)C=Cc2cccnc2)CCC2(CCN(C(c3cnccn3)=O)CC2)C1 C1(C(=O)NCCCCn2c(C)ncc2)CCS(=O)(=O)C1 Cc1ccc(C)c(NCC(=O)NCC2CN(C(=O)C(c3ccccc3)C3CC3)C2)c1 C1(NC(C(c2c(C)n[nH]c2C)C)=O)CC2CC(C1)CN(C(C1CC1(F)F)=O)C2 C1(C(=O)NCC2CC(C(=O)NC(CC(=O)NC)C3CC3)C2)CCC(O)CN1C CC(CCCC(=O)NC1CCC(O)C1)c1ccccc1 CC(=Cn1ccnn1)C(=O)NCC(CO)NC(=O)CCC1CC1CC1CC1 C1(C)(CNC(C(c2ccoc2)NC(Cc2cn(C)nc2)=O)=O)CCCCC1 CC1CC(CNC(C2(C(F)F)CCC2)=O)CN1C(C1CC12CC(O)C2)=O C(=O)(CCCOCc1ccccc1)NC(C)CN(C)C(C1(C)CC1C(F)(F)F)=O c1(C(=O)NC2C(C(=O)NC(c3ccc(F)cc3)C)C2)cccnc1O C=C(Br)CC(C)(C)C(=O)NC1CCN(C(=O)C(CCC)N(C)C)CC1 C(=O)(CCC(=O)c1ccc(OC)cc1)NC(CNC(C1(CCC=C)CC1)=O)C C1(NC(CCOC2CN(C(CCN(C)C)=O)C2)=O)CC12CCOC2 CC1(C(=O)NCCc2nc(-c3ccccc3F)n[nH]2)CCNCC1 c1(C(N)=O)n[nH]c2c1CN(C(C1CC(=O)N(Cc3ccc(Cl)cc3)C1)=O)C2 C=CCC(F)(F)C(=O)N1CCC(CF)(NC(=O)CNC(c2ccc(F)cc2)=O)C1 C1(NC(C2CC23CCC3)=O)CC(O)CN(C(=O)C(F)(F)c2cncs2)C1 C=Cn1nccc1C(=O)NCCC1(O)CCN(C(=O)CC2(OC)CCOCC2)C1 C1(NC(c2n(CC)ccn2)=O)CC2(C(=O)NC3(C4CC4)CCCC3)COC1C2 C1(C)(NC(C2CN(C(C)=O)C2)=O)CC(C(=O)NCC(C)C2CCC2)C1 C1(C)(C(N2CC(O)(C(C)NC(C3(OC)CCC3)=O)C2)=O)CCCS1(=O)=O C(CCCCC(=O)NCCCCCNC(C1(C)CCC(=O)N1)=O)SC C1(C(=O)NC(c2onc(C)n2)C2CCCCC2)CC2(CCC(CN)OC2)C1 c1(C(C(=O)NCC(CNC(C(c2cccc(Cl)c2)OC)=O)O)=O)cccc(C)c1 C(c1ccc(Cl)s1)=CC(=O)N(CC(C)N(C)C(c1cnnc(O)c1)=O)C C1(C(C)NC(=O)COc2cnn(C)c2)CCCN1C(=O)CCC1CC1(F)F C(=O)(C1CCCc2nc[nH]c21)NC(C)CNC(=O)C(=O)NCC1CC1 c1(C(N(CCCNC(Cc2ccn(CC)n2)=O)C(C)C)=O)cc(Cl)ccc1O n1(CC)ncc(C(=O)NCCC2CCC(NC(=O)CCc3cc(Cl)no3)C2)n1 C1(CNC(C2C(C(C)C)C2)=O)CC2CCC1N(C(c1ccc(Cl)o1)=O)C2 c1(CNC2CCS(=O)(=O)C2)ccc2cccc(Br)c2n1.C1(C)CC1 C(=O)(C(C)(CC)CCC)NCC1C(NC(C2C(=C)C2C(=O)OC)=O)C1 C1(N(C(=O)C(C)NC(=O)Cn2nccc2C(=O)O)C(C)C)CCS(=O)(=O)C1 C12(C(=O)NCC3N(C(CNC(C(C)(C)C)=O)=O)CC(O)C3)CCC(N=[N+]=[N-])C1C2 c1(OC)ccc2c(c1)nc(CSC1C(C)CCN1C(=O)OC(C)(C)C)n2C(F)F N1(C(C(C=C=C)C)=O)CCC2(CC1)CC2CNC(=O)N(C)C CCC(CC1CCCCC1)C(=O)N1CCC1CNC(=O)C(C)(C)NC(C)=O N1(C(C(COC)(C)O)=O)CCOC2(CCN(C(C3CC34CCCC4)=O)CC2)C1 c1(C(=O)NC2C(CNC(C=Cc3cn(C)nc3)=O)CCC2)cncc2ccsc12 c1(OC)ccc(CN2CC(F)CC2C(=O)NCCC(=O)NC(C)(C)C)c(C)c1 C12(CC(=O)NCCOCC(=C)C)CCC1CN(C(=O)CC(C)(C)C)C2 c1(CC)[nH]c(-c2ccccc2)cc1C(=O)N(C1CN(Cc2ccccc2)C1)CC N1(C(Cc2cc(C)sc2C)=O)CCN(C(=O)CCC2CCCN2C)CC1CF C=CCCCC(C(=O)NCc1cc(C)c(C)s1)NC(C1C2CC3C(C2)C13)=O C1(OC)CN(C(=NCCC(F)F)NCCOC)CC1CC1CCOC1 C1(C(N2CC(C(C)OC)C2)=O)CCC(C)(C)N(C(=O)C(N=[N+]=[N-])C(C)C)C1 C(CNC(=O)Cc1ccnn1C)(C(C)C)NC(CCNS(CC)(=O)=O)=O C1(C(N2CCCC(NC(C(=O)NCC(F)F)=O)CC2)=O)Cc2ccccc2CO1 C(=O)(C(CC(N)=O)NC(=O)CC1COCCO1)NCC(C=C)(C)C C(=O)(CC(O)C(C)CC)N1CCC(C(=O)NC(C=C)C(F)(F)F)(CCOC)CC1 Cc1nc(C)c(C(=O)NCC(N2CCN(C(=O)C=C3CCCC3)CC2)C)o1 N1(C(c2c(C)snc2)=O)CCCCC1CC(=O)NCCCC(C)O N1(C(CCC=CC(C)C)=O)CC2COCC2(C(=O)NC(C)CS(C)(=O)=O)C1 C(N=C(NCC1(OC)CCCO1)NC(C)Cc1ccccc1)c1c(CC)n[nH]c1 CC(C)(CN=c1[nH]c(NC2CN3CCC2CC3)nc2c1CCC2)c1ccccc1 c1(C(=O)OC)cc2cc(C)ccc2[nH]1.N12CCC3(CC3C1)CN(C)C1(CC1)C2=O N1(C(c2n[nH]cc2F)=O)CCCN(C(C2CCCS(=O)(=O)C2)=O)CC1 N1(C(C2OCCN(CC)C2)=O)CCC(C)(C(=O)NC2CCC(=O)NC2C)CC1 C1(N(C(CC)C(N2CCCCC(O)C2)=O)CCC(C)=O)C(C)OCC12CCNCC2 c1(C(=O)NC(C2CCCCC2)CNC(=O)C=CC2CCC2)cn2c(n1)SCC2 C1(NC(C2N(CC)CCC2)=O)CC2CCC1C(NC(=O)CCc1ccncn1)C2 c1(C(N(CC(CC)(C)NC(=O)C(=O)NCC)C)=O)ccc(-n2ccnc2)c(C)c1 N1(C(C2CCC(C(=O)OC)C2)=O)CC2CC(NC(=O)Cc3cccs3)CC1C2 C1(NC(C(C=C)O)=O)CC2CN(C(C3CC(=O)N(C(C)C4CC4)C3)=O)CC2C1 c1(N(C)CC2(F)CCCC2)nc(N(C)Cc2cccc(N)c2)nc2c1SCC2 C1(NC(CCCS(N)(=O)=O)=O)CS(=O)(=O)C12CCN(C(C1CCCSS1)=O)CC2 N1(C(C2C(C(C)(F)F)C2)=O)CCC(CO)(CNC(c2cccc(Cl)c2)=O)CC1 C(=O)(C(C(C)C(C)(C)C)N1CCCC(C)(CC)CC1)NCCCCCC N1(C(CCc2onc(CC)n2)=O)CC2(CCC2NC(=O)C(C)CO)C1 C(C1=CCN(C(=O)C(C(C)CC)c2ccccc2)CC1)NC(C1(C#C)CC1)=O Cc1cc(O)c(CN2CCNCC2C(=O)Nc2ccc(CCO)cc2)cc1Cl Cc1ccc(C(N2CCC(NC(c3cc(Br)no3)=O)C(CO)CC2)=O)c(N)c1C N1(Cc2ncc(OC)nc2)CCC(F)(F)C(C(=O)Nc2ncc(SC)s2)C1 N1(C(c2nnc(C)s2)=O)CCCN(C(C2CCCN2C(=O)C(C)(C)C)=O)CC1C C1(N(CC(=O)Nc2nccn2C)C)CN(C(=O)C#CC2(C)CC2)CC1C1CC1 CC1(NC(c2ccc(C#N)o2)=O)CCC(NC(C2CC3(CCOC3)C2)=O)CC1 C1(N(C(=O)Cc2csnn2)C)CCCC(NC(c2ccnc(C(F)(F)F)c2)=O)C1 c1(NC(=O)CC2CN(C(C3CCC(F)(F)C3)=O)CCO2)cnncc1Cl c1(C(N2CCCC(N(C(=O)Cc3cc(C)n(C)n3)CC)C2)=O)cncc(O)c1Cl C1(NC(=O)COCC2CCCCO2)CN(C(=O)C=C2CCCCC2)CC1O N1(C(CC)=O)CCC2CCN(C(=O)Cc3cccc(Br)c3Cl)C2C1 C(C(CO)C(=O)NCCC(CNC(=O)CCC(=O)Nc1sccc1C)OC)OC C1(CNC(C(C)(C)F)=O)CN(C(C2CCSC2)=O)CC1C(F)(F)F C(CCNC(C1CC(=O)N(C(C)(C)C)C1)=O)(C(C)C)NC(c1c(C)con1)=O N1(C(c2cc(C)oc2C)=O)CCC(CNC(C2CC3(C2)CC(O)C3)=O)C(O)C1 C12(CNC(c3ccoc3)=O)CN(C(c3ccc4n[nH]cc4c3)=O)CC1CCO2 N1(C(C)=O)CCN(C(c2cnc(C)s2)=O)CC1.C1(C(NCCOC)=O)(N)CCCC1 CC1CCN2CC1C2.C12(N(c3cc(O)ncn3)C(=O)C(F)(F)F)CCCC1C2(F)F n1(CC)[nH]c(=NC(=O)Nc2cc(C3CCC(=O)N3)ccc2C)c2c(Cl)cccc12 c1(NC(C2CC(=C)C2)=O)cccc(NC(C23CC(C)(CO2)C3)=O)c1 N1(C(c2ccc(Cn3ncc(C)c3)o2)=O)CC(CCNC(=O)CCCF)C(C)C1 c1(CC(N2CCC(C3N(C(C(F)=CC)=O)CCCC3)C2)=O)c(OC)cccc1C c1(OC)cc(C)cnc1C(=O)NC1CCN(C(c2ccc(F)cc2C(F)F)=O)C1 N1(c2n(Cc3cnc(C)o3)nnn2)CCCC(O)(C(F)(F)F)CC1 c12cccc(c1)C2=O.c1(CN(C(CC)=O)CC(C)OC)ccccc1Br C(=O)(CC(C(C)C)NC(C1CN2CCC1CC2)=O)N(CCC(N)=O)CC C1(CN(C(=O)CN2CCCC2=O)C)CCCN(C(=O)CN2CC3CC3C2)C1 c1(OC)oc(C)nc1C(=O)NC(Cc1cnn(C)c1O)C(=O)N(CC(F)Cl)C CCC(C(=O)N1CCC(N(C(=O)C(=O)NC2CC2)CC2CC2)CC1)C(C)O C(=O)(C(O)C(F)(F)F)NC1(CC)CN(C(C2CCN(C)C2C)=O)C1 c1(C(N(C2CCN(C(c3c[nH]c(=O)cn3)=O)C2)CCC)=O)cnc2ccsc2c1 C(=O)(C(C)(C)C(=O)N1CCOCC1C(=O)Nc1cc(Br)ncc1Cl)OCC C(C1CCc2nccn21)NC(C1CN(C(=O)Cc2ccc[nH]2)CC(C)O1)=O C(C)(C(=O)NCC1(O)CCCN(C(=O)C(C)=C2CCCC2)C1)(C(C)C)NC(C)=O Cc1ccc(S(=O)(=O)N2CCN(C(c3ccnc(F)c3)C(=O)NC3CC3)CC2)cc1C C(CC(C)C)(C(=O)NC1CC(NC(=O)Cc2cc(Cl)n(C)n2)C1)NC(=O)OC Cc1ccncc1C(=O)NC1C=CCN(C(C2CC(N(C)C)C2)=O)C1 N1(CCNC(C(CCC)N(C)C)=O)CCCN(C(C2(C(C)C)CCCO2)=O)CC1 CC1=NOC2(C1)CC(C(=O)NCC1CC(NC(=O)Cc3cnoc3)C1)C2 N1(CC(=O)NC(CN(C(CNC(CCC(C)C)=O)=O)C)C)C(=O)NC(C)(C)C1=O c1(Cc2cn(CC(CNC(C3COCC(C)O3)=O)(C)C)nn2)ccc(F)nc1Br CC(C(CO)NC(C1(SS(C)(=O)=O)CC1)=O)NC(=O)Cc1cnn(C(C)(C)C)c1 Cc1ccc(C)c(C(=O)NC2CC2NC(c2nocc2C(C)(C)C)=O)c1O C(C(F)C(F)(F)F)N(C(C(CC)OC)=O)C C1(NC(c2cn(CCN(C)C)nc2)=O)CC12CC(NC(C1CCS(=O)CC1)=O)C2 N1(CC(=O)OC2CCCCCC2c2ccccc2)C(=O)c2ccccc2C1=O C(C(O)C(=O)NCCC1CC(NC(=O)C(C)(C)c2ccc(C(F)(F)F)s2)C1)OC C1(C(=O)NCC(CCOC)NC(C2CC3CC3C2)=O)(OC)CCOCC1 C(=O)(C(F)C(C)(C)O)N1C(CN(C(C(c2ccccc2)SC)=O)C)CCC1 c1(C(=O)NCC2CN(C(c3cc(F)c[nH]3)=O)C3CC23)cc2ccncc2[nH]1 CC1CC=C(C(=O)NCC2CCC(NC(c3ccc(O)c(Cl)n3)=O)C2)CC1 C12(CNC(c3c(C)n(C)cc3)=O)CCCC1CCN2C(=O)CSCc1cccs1 CC(C(F)C(=O)N1CCC(C2CC2)C1CNC(=O)Cc1cn[nH]c1)C(F)(F)F N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCCC(O)(CNC(c2nn(C)cc2C)=O)CC1 C1(C(N2CCC(CC=C)(NC(=O)CC(C)F)C2)=O)CC(C(C)C)=NO1 n1(CC(=O)N(C)CC2(NC(C3CC34CC4(F)F)=O)CC2)ncc(O)nc1=O c1(NC(C2N(c3cc(OC)nc(C)n3)CC(F)C2)=O)ccc2ccsc2c1 C1(C)(CN2C(=O)NC(C)(CC=C)C2=O)Cc2ccccc2C1 n1(CC)cc(-c2n[nH]cc2C(=O)NC2CC2NC(C2CC(N(C)C)C2)=O)cn1 N1(C(c2c(C)cc(C)o2)=O)CCN(C(c2ccccn2)=O)C2COCC12 CC1CCN(CC(=O)NC(C)(C(=O)NCCOCCN(C)C)C2CCC2)CC1 C(=O)(CCCC(C)(C)C)NCC1CN(C(C2=CC(C)(CC)C2)=O)CC1CN(C)C C=CC1CCN(C(C2CC(NC(C3CC4C(C3)C4(F)F)=O)C(O)C2)=O)CC1 C=CCC(CC)C(=O)N1CCOCC1C(=O)NC(C)Cn1cncn1 C(C(=O)NC1(C(=O)NC(C)CCCCO)CC(O)C1)(C(C)C)SC n1(CC(=O)NCC2CN(C(=O)C=CC(F)(F)F)C2)cc(F)ccc1=O c1(NCC2C(C=C)C2)[nH]c(=NCc2cnc(Br)cc2C)nc2c1ncn2C C(=O)(C1=CC2(CCN(C(=O)CC3CC4C=CC3C4)C2)C1)NC(c1cncnc1)C c1(NCC)ccc(C(=O)NCC(C)Sc2cccc(OC(C)C)c2)cc1[N+](=O)[O-] c1(C(N2CC(NC(c3ccccc3)=O)C(C#N)C2)=O)cc(F)ccc1C(F)F CON(C(=O)C(CNC(=O)C=C(C)C)CC1CCCC1)C(C)C C(=O)(C(C(C)(C)C)OCC(F)(F)C(F)F)N1CC(C)CC(COC(C)=O)C1 C1(NC(CCC2(C)CN(C(C3(CC=C)CC=CC3)=O)C2)=O)CCN(C)C(C)C1 c1(C(N2CCN(C(CCOC)=O)CC2)=O)ccc2nc[nH]c2c1F C1(CCNC(C(CC)CC)=O)CCN(C(c2ccn(CC)n2)=O)C(C)C1 Cc1cccc2c(C(=O)N(CC(C)NC(C3CCS(=O)(=O)C3)=O)C)cccc12 C1(C(N2CC(O)(CCNC(CCS(=O)(=O)NC)=O)C2)=O)CN2CCN1CC2C N1(c2snc(COC)n2)CCCCC(NC(c2cc(Cl)cn2C)=O)C1 C12(C(=O)NCc3cn(CC(C)NC(c4cnn(C)c4F)=O)nn3)CCC(CC1)C2 N1(C(c2ccc(SC)o2)=O)CCCC(CCNC(=O)Cc2ccsc2)CC1 C(=O)(C(C)CCN(C)C)NC1(C(=O)NC2(C)CC(=C)C2)CSC1 C12(CC)CCC(C(=O)N(CCNC(C3(NC(N)=O)CC3)=O)CC)(CC1)CO2 C(N=c1[nH]cnc2cc(C)[nH]c12)C1(F)CC(NC(C(C2CCOC2)OC)=O)C1 c1(C(=O)NCC2N(C(C(=O)NCC)=O)CCCC2C)c([N+](=O)[O-])cnn1CC C1(C)(CNC(=O)NC(c2ccc(NC(C)=O)cc2)C)CCC(F)(F)CC1 C1(NC(c2cccn3ccnc23)=O)CN(C(C2C=CCS2)=O)C2CCCC12 C1(C(=O)NCC2C(C)(C)CCO2)CC12CCN(C(=O)CCc1cccnc1)C2 C1(N(C(CC2(OCC)CCC2)=O)CCO)CCN(C(C2(F)CCCC2)=O)C1 C(=O)(CCC(C)(C)F)NC(C1CCCC1)CNC(C(C)OCCCCCC)=O C1(NC(C(CC)NC(N)=O)=O)CCN(C(C2COCCN2C)=O)CC1F N1(C(CNC(=O)OC(C)(C)C)=O)CC2CCC2(NC(C2(C)CCCS2)=O)C1 N1(C(C(F)=CC)=O)CCCOC(CNC(=O)CSc2nncn2C(C)C)C1 C1(O)(C(C)NC(=O)CCc2cnn[nH]2)CN(C(c2cc(-c3ccccn3)ns2)=O)C1 c1(CC(C)C)cccc(C(C)C(=O)NC2CC(NC(c3ccc(C#N)s3)=O)C2)c1 c1(C(=O)NCC=C(C(=O)Nc2cnc(CCC)nc2)C)ccc([N+](=O)[O-])o1 C1(CNC(CSC(C)(C)C)=O)CC12CCN(C(=O)Cn1cnc(C#N)n1)CC2 CC(C)C(=O)C(=O)N1CCCCC1CCNC(=O)C=CCF N#CC1CN(C(C2CN(C(=O)Cn3cc(Cl)cn3)CCC2O)=O)CCO1 C1(C(=O)NCCOC)CN(C(C2(OC(C)=O)CCCCC2)=O)C(C)(C)C1 N1(C(CNC(C(CC)C)=O)=O)CCC2CCCC12C(N1CCC2(CC1)N=N2)=O CC#CCCCC(=O)NCC(n1nnnc1-c1ccccc1)OC c1(CC)nc(C)c(C(=O)NC2CCN(C(=O)COc3ccc(C(C)=O)cc3)C2)s1 N1(C(c2c(CCC)n(CC)nn2)=O)CC=C(CNC(=O)CC(C)CC)CC1 CN1CCCC1CC(=O)NCc1occc1C(=O)NOCCCCF c1(C(=O)OC)sc2ncnc(NCCN(C(=O)CCC3CC3(C)C)C)c2c1C C=C(C)CC(C(=O)N1CCOC(C)C1C(=O)NC(c1c(C)n[nH]c1C)C)OC c1(CNC(C(N2CCCCC2)C)=O)ncccc1C(=O)Nc1cncnc1S CCC(C)C(CN(C)C)NC(=O)CC(CNC(C1(O)CCCCC1)=O)C1CCC1 Cc1cccc2ncnc(N3CCCC(CCNC(=O)C(C)CC(C)C)CC3)c12 c1(C(N(C)CC2OCCN(C(C(=O)NCC)=O)C2)=O)cccc2ncnn12 C(N=c1[nH]cnc(=N)[nH]1)C1CN(C(c2ccc(CSCC)cc2)=O)CC1C N1(C(C(C)OCC)=O)CCN(C(=O)CSc2nncs2)C(C2CCCC2)C1 Cc1ccc(S(=O)(=O)CNC(c2ccc(P(C)(C)=O)cc2O)=O)cc1 C1(C(=O)NCC(CC(C)C)NC(C(C2CCCC2)OC)=O)COC2COCC2O1 c1(CNC(CC2(OC)CCC2)=O)ncc(C(=O)N(C)Cc2nncn2C)cn1 N1(Cc2cn(C3CN(C(C(CC)(C)CO)=O)CC3O)nn2)CCc2ccccc21 C1(CC(=O)NC(C(C(=O)OCC)C)C)CC2(C1)CN(C(=O)C1=CCCCC1)C2 N1(C(C=CSC)=O)CCCC(N(C)C(c2cn(Cc3ccccn3)nn2)=O)CC1 C1(CC=C)(C(=O)NCCC(=O)N(C)C)CCCN1C(=O)CC1(O)CCCOC1 c1(CNC(C2CC(NC(CN(C(=O)OC)C)=O)C2)=O)cc(C)cc(C)n1 c1(CC(=O)N(CC(CNC(C2N(CCC)CCC2)=O)(C)C)CC)nnc(S)n1C Cc1nc(N2CCN(C(=O)CCc3ncccn3)CCC2C)c2c(C)csc2n1 C1(C(N2CC3(CN(C(Cc4cc(OC)no4)=O)C3)C2)=O)CNC(=O)CC12CCC2 C1(CNC(C(CCC)OC)=O)CCCCCN1C(c1ccnc(CO)c1)=O c1(NC(CC2(C)CCC2)=O)ncc([N+](=O)[O-])cc1F Cc1n[nH]c(=NC(CCN(C(=O)CC2CCCOC2)C)C(C)C)o1 C(=O)(CC1=NNC(=O)C1)NC1C(CNC(c2[nH]cc(CC(C)C)c2)=O)C1 N1(C(CCC(CCC)CC)=O)CCC2(CC1)CCN(C(=O)C(C)(C)C(N)=O)CC2 c1(C(=O)NC2CC3CN(C(C(CC)(C)O)=O)C2C3)ccc2c(n1)OCC(=O)N2 C(C#CC1CCCCO1)NC(CC(C1CCC1)NC(=O)OC(C)(C)C)=O CC1CCC(CCC(=O)NC2(CNC(=O)C=Cc3cscn3)CCC2)O1 Cn1ccc2cnc(Nc3cccc(-c4cnn5c4CCCC5)n3)nc12 N1(C(CC)C(=O)NC2CCC(CNC(=O)CCCSC)C2)CCN(C(C)C)CC1 C1(CN(C(Cc2cc(CC)no2)=O)CC)CCCN(C(C2CC2(C)C)=O)C1 C12(NC(c3c(CNC(CC(C)(C)OC)=O)ccs3)=O)CCC(C1)OC2C N1(C(C(CCC)(C)C)=O)CC2CCC(C1)N2C(c1cc(=O)c(O)c[nH]1)=O C(CN=c1[nH]nco1)N(CCC)CCN(c1[nH]c(O)nc1C)C1CCCC1 N1(C(C=CC(=O)OCC)=O)C2CCC1CC(NC(=O)Cc1cccnc1OC)C2 c1(NCC2CC(C)NC(=O)C2)[nH]c(=NCC2CC2(F)F)nc2scnc12 C1(OC)CC(NC(=O)Oc2cc(C(C)C)ccc2C)C12CC(F)(F)C2 CC1OCCCC1C(N1CC(N2CCCC2)C1)=O.C1C(=O)N1 C1(CN(C(C(CC)NC(C)=O)=O)CC)CCCCN1C(c1ccncc1)=O C1(C)(C(N(CCC)CCNC(C2(N(C)C)CCC2)=O)=O)CC(O)CN1C S(=O)(=O)(c1c[nH]ccc1=NCC1(CO)CC(F)(F)C1)N1CC(C)CS(=O)CC1 c1(C(C)=O)ccc(C(=O)N(CCCNC(=O)CN2CCC(C)CC2)CCO)cc1C C12(CNC(c3cc(CC)on3)=O)CCCC1N(C(c1ccco1)=O)CC2 O=C(C1=NOC2(CCCN(CC(N3CCOCC3)=O)C2)C1)Nc1cnc(Br)o1 c1(OC)cc(C(=O)NCCC2COCCN2C(=O)CC2CCCOC2)ccc1F C12(NC(=O)COc3ccon3)CCCC1N(C(=O)Cc1ccc(O)c(F)c1)CC2 CCCCC(O)CC(=O)NC(CNC(c1cnn(CCC)c1C)=O)C(C)C Cc1cc(C(N2CCCC2CCNC(C2CC=CC2)=O)=O)ccc1Br C1(CNC(C2(C)CC2(F)F)=O)(CO)CCN(C(c2ccc(F)cc2O)=O)CC1 N1(NC(CCN(C(C2CCC(CC)O2)=O)CCO)=O)CC=CCCC1 c1(OCC)ccc(CN(c2ccc(Cl)nc2)c2nc(CC(N)=O)cs2)cc1 C1(C(=O)NC23CC(NC(CN(CC(C)(C)C)C)=O)(C2)C3)CCCCNC1=O N1(C(C2N(C(C)C)C(=O)CC2)=O)CCC(CNC(C2CCC(O)CC2)=O)C(C)C1 N1(C(C)=O)CC(CO)C(COC)C1.C1C(O)COC2CC2C(=O)N1 C1(C(=O)NC(c2cn(C)nn2)C)CN(C(C2CCCSC2C)=O)CC1C1CC1 c1(CC)nc(N2CC3C(C(=O)NC4COCCC4O)C3C2)c(F)c(Cl)n1 CCCC(C)(O)CC(=O)N(CCC(=O)NCC(C)CC(C)C)CC C(C(C)(C)C(=O)NCC1CN(C(c2occc2C(C)C)=O)C1)OC(C)C C1(CC2CCN(C(C(=O)NCCC)C3CC(OCOC)C3)C2)CC2C=CC1CC2 N1(CC(=O)N(CCCC#C)C)CCN(C(=O)C=CCN2CCC2)CC1 c1(C(N2CC(C(C)NC(C(C)CCO)=O)C2)=O)cccc2nc(O)oc12 N1(C(=O)CC2CC2)CCC2C(C1)CN2CC1(CO)CCCCC1 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCN(C(c2ccco2)=O)C(CCO)C1 C1(C(N2CCC(O)(CNC(=O)Cc3ccc(Cl)cc3)C2)=O)COC2COCC12 CCS(=O)(=O)CC(=O)N1CC2CC2C1C(=O)N(C)Cc1cc(OC)no1 C1(NC(CC(C(C)C)C)=O)C2CCCC1CC(NC(=O)CCc1cnccn1)C2 C12(C(=O)NC3CCC(NC(c4ccc[n+]([O-])c4)=O)C3)CC(F)(CO1)C2 C1(C2CC2)(CNC(C(C)NS(CCC)(=O)=O)=O)CCN(C(=O)CCC2CCC2)C1 Cc1oc(C)c(C(=O)NCCC(C)CCNC(C2CCOC2(C)C)=O)c1C C(CCCCC(=O)N1CCC(C(N2CCC(CC3CC3)C2)=O)C1)=CC N1(C(CC=C)=O)CC23CCCCC2(C1)CN(C(c1ccc2n[nH]cc2c1)=O)C3 c1(SC)cc(F)ccc1C(N1CCCC1C1CCCN(C(c2cnsc2)=O)C1)=O c1(CC)nn(C)cc1CNC(=O)CCCNC(C1(CN)CCCO1)=O.C(C)=O C(=O)(C1=CCCCO1)NCC(Cn1cc(-c2ncc(F)cn2)nn1)OC N1(C(C)=O)C(=O)CCC1C(=O)OC(C)(C)C.C1C(C)NCCO1 C1(NC(CCOC)=O)CC2CC(NC(=O)COc3cccc(C(C)=O)c3)C2C1 c1(CC)cc(C(=O)N(C(C)CCNC(C2(C#N)CC2)=O)C)nn1CCO Cc1cc(C(N2CCN(CCNC(=O)C(C)CN(C)C)CC2)=O)n2ncnc2n1 N1(c2nnnn2CCOCC2CC2)CCC(CN(C(=O)O)CO)(C2(C)C(C)(C)C2)CC1 N1(C(C2CN(C(c3ccc(C)[nH]3)=O)CC2(C)C)=O)CC(C)CCC12CC2 c1(C(N2C(CC(=O)N(C3C(OC)CC3)C)CC2)=O)nc(C)ccc1F N1(C(C2(NC(c3nc(Cl)cs3)=O)C(C)(C)C2)=O)CCCNC(=O)C1 CC1CC1N=c1[nH]c(=NCC23CCC(CC2)O3)[nH]c2cccnc12 c1(CNC(=O)Nc2onc(C)n2)ccc(N2CCNC(=O)C2)c(F)c1 N1(C(C(CF)NC(C=CCN(C)CC)=O)=O)CC2CC1CN2C(C)=O C(=O)(C(CCCC)C(C)C)NCc1nc(CNC(CC(C=C)CC)=O)sc1 c1(C(N(C(CC(N2CC(C)OC(CO)C2)=O)(C)C)C)=O)ccc(N=[N+]=[N-])cc1 c1(C(=O)NC(C)CCN(C(=O)C(O)CC(N)=O)C)n[nH]c2c1CS(=O)(=O)CC2 C(C(C)(C)CCNC(=O)C(C)C(F)F)NC(c1n(C(CC)C)ncc1)=O C1(NC(Cc2c(CC)nn(C)c2CC)=O)CN2CCC1(F)CC2 c1(OC)ncc(C(=O)NC(CNC(c2ccncc2)=O)CO)cc1C c1(C(N2CC(NC(c3cc(OCC)n[nH]3)=O)C2)=O)cc2ccc(F)cc2[nH]1 C1(NC(c2ccc(CC)s2)=O)CCCC(N(C(=O)COCCCC(C)C)C)C1 N1(C(C(=O)NC(CC)CC)C)CCC(C2CCCN(C(C3(O)CCCC3)=O)C2)C1 N1(C(CC2N(C(C3C(C)=CCS3)=O)CC(F)C2)=O)CCCCN(C)CC1 c1(C(N2CC(C)(C)C(NC(c3cc(Cl)ns3)=O)CC2)=O)coc2ccc(O)cc12 N1(C(c2c(C)ccc(N)c2)=O)CC2CC(NC(C3C(F)(F)C34CC4)=O)CC(C2)C1 c1(SC)cccnc1C(=O)N(CCCN(C(=O)C(C)C(C)O)C)C C1(NC(Cc2ccc(OCC=C)cc2)=O)CCN(C(=O)C(F)=CCCF)C(C)C1 CC1CCCN1C(C(=O)NCC1CCC1)C1CC1c1ccco1 C=C1CC2CC1CN2C(=O)C1=CCN(C(=O)CCNC(=O)COC)C1 N1(CC(=O)NCC2C(C(=O)NC3N(C(=O)OC(C)(C)C)CC3)C2)CC(=O)NC1=O N1(C(c2cc(C)oc2)=O)CCC(C(N2CC3CCC(C2)N3C(C)C)=O)CC1(C)C N1(C(c2c(-c3c(F)ncc(COC)c3)cncc2)=O)CC2CNCC1COC2 c1(CC)cc(OC)ccc1C(=O)NC1CCCCC1NC(=O)CCOCC1CC1 c1(CC(=O)NCC(=C)CCNC(=O)C(COC)NC(C)=O)ccc2n[nH]cc2c1 n1(CC(=O)NCCCN(CCCOC)C)nc(C)ccc1=O.c1(C=O)cc(=O)cc[nH]1 C12(CNC(C(CC=C)CC)=O)CCCC(CN1C(=O)Cn1nccn1)C2 c1(C(=O)NCC(CNC(c2cc(C)n(CC(F)(F)F)n2)=O)F)cn2ccnc2s1 C(N=c1[nH]c(=N)[nH]c2[nH]ccc12)c1cn(CC)nc1C C(=O)(C(C)C(C)S(C)(=O)=O)N1C2CN(C(C(c3ccc(CC)s3)=O)=O)C(CC2)C1 N1(Cc2c(OCC(=C)C)cccc2)CC2OCCN(C(c3cc(Br)cs3)=O)C2C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CC(C)N(C(=O)C(n3cc(C)cn3)C)C2C1 CCCC(CC(=O)NC(c1cccc(O)c1)C)NC(C1CC=C(C)CC1)=O C1(C(=O)NCC2N(C(C3C(C(=O)OC(C)(C)C)C3)=O)CC=C2)Cc2cscc2C1 c1(NC(C(c2coc(C)n2)N(C2CCCCC2)C(CC)=O)=O)ccc(CC)cc1 N1(C(C(C(C)C)C)=O)CCOCC(F)(CNC(c2ccc3nonc3c2)=O)C1 c1(NC(CC)C)ccc(Br)cc1S(=O)(=O)NC1COCC1N Cc1cc(C(=O)NCc2nc(C)c(C(=O)NCC(O)C(C)(C)O)o2)c(C)cn1 C1(NC(N(C)Cc2ccc(C3C(C)C3)o2)=O)COC2(CCC2)C1O CC(=O)CCCC(=O)NCC1(F)CCC(NC(=O)Cc2cc(C)[nH]n2)C1 c12ccccc1[nH]c(=O)[nH]2.C(C(C)C(=O)OC)N(C(CN(CCC)C)=O)CC c1(NC(C2CC2C(=O)Nc2ccc(-n3cccc3)cc2)=O)cccc(Cl)c1Br c12ncnc(Cl)c1CC(C)N2.c1(CC)ccc(CN(C)C(=O)OC(C)(C)C)cc1 Cc1sc(=O)n(CCC(=O)N(C2CCCN(C(=O)C(C#N)CC3CC3)C2)C)c1C N1(C(c2cnc(C)[nH]2)=O)CC2=C(C1)CN(C(C1CC3(CCC3O)C1)=O)C2 Cc1cc(C(=O)NC2CC(CNC(c3c[nH]cc(C)c3=O)=O)C2)ccc1Br c1(C(=O)NCCC(C)NC(c2cc(C)cc(C)c2O)=O)cccc(P(C)(C)=O)n1 C=CC1(CC(=O)NCCN(C(c2nnn(C)n2)=O)CC)CCOCC1 c1(CC(N2C(CNC(c3n[nH]c(C)c3Br)=O)CC2)=O)nc([N+](=O)[O-])n[nH]1 C1(CNC(C=Cc2ncc(C)[nH]2)=O)CN(C(=O)CCCc2cccs2)CCC1C C1(CC#C)(C(=O)NCc2cccc(NC(C3CCCO3)=O)c2)CCCOC1 C(CC(C(=O)NCC1CCOC1)NC(=O)CC1CC=CCC1)N(C)C c1(CCSC)nc(-c2ccc(CSC)cc2)n(C2CCCCC2C)n1 N1(C(c2c(C)nn[nH]2)=O)CCOCCC1C(=O)NCC1(CF)CC1 c1(C(N(C(CNC(C(CCC)N(C)C)=O)C)C)=O)c(C)cc(C)nc1O CN(S(=O)(=O)N1CCOCCC1c1noc(-c2ccsc2)n1)Cc1ccccc1 C(C)(CCC(C)C)NC(CC1(N(C(C(C)OC)=O)C)CC1)=O Cc1nc(S(=O)(=O)N2CC(O)C(O)C(C)C2)ccc1C(=O)O C=CC(C)(C)CCCNC(c1cc(CNC(C2CC2C#N)=O)on1)=O c1(CCC)[nH]ccc1C(=O)N(CCCNC(=O)C(n1cc(C)cn1)C)C1CC1 CC(C)CCCCC(=O)NCCC1CCCCN1C(c1ccc2nc[nH]c2n1)=O C1(C(N2CCCN(CCNC(CC3CC(SC)C3)=O)CC2)=O)CC2(C1)CC(F)(F)C2 CC1CN(C(=O)CCOC2CCCC2)CCC1NC(c1cc[nH]n1)=O c1(C(=O)NC(C2(O)CCCCC2)C(=O)OC)sc2nccc(C)c2c1C C1(C)(CNC(C(C)CN(C(=O)CCN2CCCC2=O)C)=O)CNC(=O)O1 N1(C(c2c(CNC(C3(C(=O)NC)CCC3)=O)cnn2C)=O)CCCN(C)CC1C c1(OC)cc(O)ncc1C(=O)NC1CC12CC(NC(=O)C(C)NC=O)C2 Cc1scc(C(=O)NC2(CNC(=O)CC3CCC(O)C3)CCOCC2)c1C c1(C(=O)NCC(CNC(c2c(C)onc2)=O)C)[nH]c2c(c1C)CCCC2 C1(c2nnnn2CC2CCCC2)(Nc2sc(CC)c(C)c2)CC2CSCC2C1 C1(C)(C(=O)NCC(C(=O)NCCS(=O)(=O)NC)O)CC(F)(F)C1 C1(C(C)NC(c2cocn2)=O)CCN(C(=O)CCC2CCCCCC2)CC1 CON1CCC(C(=O)NCC2(c3ccnc(Cl)c3)CC2)CC1.C12CC(C1)NC2=O Cc1cc2cc(C(=O)NC3(CO)CN(C(C4CC45CCOC5)=O)C3)c(Cl)cc2[nH]1 C=CC(CCC)CC(=O)NCCN(C(=O)C(C)CCC)CC O(NC(=O)CC1CCCN1C(C1CC2CC2C1)=O)CCCN(C)C N1(C(CNC(=O)NC)=O)CCN(C(C2CCCC(C)(C)C2)=O)C(CO)C1 N1(C(Cc2cc(C)no2)=O)CCN(C(=O)COc2ccc(F)cc2Cl)C2CC12 C1(CC(=O)NCC(CNC(c2c(C)csc2Cl)=O)O)CC(C)(C)OC1=O c1(OC)ncc(C(=O)N(C)CC2CCCN2C(c2cc(Br)no2)=O)cn1 N1(C(C2CC(OC)C2)=O)CC2CC(C1)CN(C(C13CCC(CC1)C(C)O3)=O)C2 CCCCC(C(=O)N1CCN(C(C2CCN(CC)CC2)=O)CC1CC)NC(N)=O C1(NC(C=Cc2n(C)cnc2)=O)CCC2CC1CN2C(=O)CCCc1cccs1 c1(CC)ncc(Cl)c(C(=O)NC2CC3CCC2N3C(c2cn3c(n2)SCC3)=O)n1 N1(CCC(=O)NC(C2N(C(CCC#C)=O)CCC2)(C)C)CCCCCC1 C1(NC(C(CO)OC)=O)CCCN(C(c2cc[n+]([O-])cc2)=O)CC1 S(=O)(=O)(c1ccc2sc(Cl)nc2c1)NC1C(C2C(C)C2)C1 N1(C(CCN(C(c2ccc(F)s2)=O)CC2CC2)=O)CCC2CCC(O)C1C2 O=C(N=c1cc(-c2cccc(Cl)c2)o[nH]1)C#CC1(O)CCN(C(=O)OC(C)(C)C)C1 C(=O)(CC(C)(C)CN(C)C)N(C(C(N1CC(C)C(CO)C1)=O)C)C c1(C(=O)NCC(CC)NC(=O)CC2CC(C)=NO2)ccnc(OC)n1 c1(C(=O)NC(CN(C(C(C)OCCOCC)=O)C)CC)cc(O)cc(N)c1C CC(CC(=O)NC(C(=O)NCc1cc(O)cc(F)c1)C1CC1)C(F)(F)F CCCCC(C(=O)NC(c1cccc(C)c1)C)NC(=O)C(O)CC1CC1 c1(CNC(C(C)NC(c2ccc(O)cc2)=O)=O)nnc2n1CCCC2C(F)(F)F c1(C(=O)NC(CNC(CCC(C)C)=O)CC(F)(F)F)c(Cl)cc(C#N)cc1Cl c1(CN(C(C)C)C)cn(Cc2ncoc2CNC(c2ccsc2Cl)=O)nn1 c1(C(=O)NCc2c(CCNC(c3cn(C)nn3)=O)ocn2)coc2c1CCCC2 C=C1CC(C(=O)NC(C)Cc2ccco2)(CN)C1 C1(CNC(=NCC)NCc2nnc(COC)s2)CCC(C#N)CC1 C12(NC(c3cc(Cl)c[nH]3)=O)CCC(CC1n1cc(CN3CCCSCC3)nn1)C2 C(=O)(CC(C)CC(=O)NC(CC1CC1)C(=O)NCCCC1(O)CC1)OC C1(NC(COCCC)=O)CCC(NC(=O)C=CC(c2ccccc2)=O)CC1 C1(CC)CC(O)CCN1C(=O)C(C1(O)CCC1)NC(c1cc(C#N)[nH]c1C)=O c1(C(N2CCC(NC(CCc3cc(OC)no3)=O)C2)=O)ccn2ccnc2c1 C1(C(=O)NCc2c(CCNC(c3cc(C)no3)=O)ocn2)CN(C)CC(C)O1 c1(OC)cc(C(=O)NCC2CC2NC(C2(F)CCOC2)=O)ccc1C(F)(F)F N1(C(C(C)NC(=O)NC)=O)C2CCC1CC(NC(C1(C(C)(F)F)CC1)=O)C2 CN=C(NCCOC(C)=O)N1CCC(Cc2ncccn2)C1 C1(N(C)C(c2ccc(CNC(c3sccc3Cl)=O)o2)=O)CNC(=O)C12CC2 C1(NC(c2cn(C(C)C)nc2)=O)CC2C(NC(c3ncc(C(F)F)s3)=O)C2C1 O=C1CCN(CC(=O)NC2(CCCNC(C3CCCC(F)C3)=O)CC2)C(=O)N1 c1(CN2CCC(C(=O)NCc3cccc(C(F)(F)F)c3)C2)ncc(Cl)nc1Cl C1(CC)CN(C(c2ncc(N)cc2C)=O)CCC1NC(c1cc(C)cs1)=O c1(C(N2CCN(CCN(C(=O)CNC=O)C)CC2)=O)cnn2cccc(Cl)c12 N1(C(=O)NCc2cccc(-n3c(C)ccn3)c2)CC2CCCN2C(=O)C1C N1(S(C(CC)C)(=O)=O)CCC2(CC1)CC2NC(C1COCCO1)=O C(=O)(CC(C)(C)C)NC1CC(NC(c2ccc(CN(CCC)C)o2)=O)C1 N1(C(c2c(C)nccn2)=O)CCCN(C(=O)C(CC(C)C)n2ccnc2)C(C)C1 C#Cc1cc(C(=O)NC2CC(S(C)(=O)=O)C2)ccc1Cl C=C(C)C(CC(=O)NC(CCCNC(C1CCN(C)C1=O)=O)c1nn[nH]n1)OCC N1(C(C2CC(C)OCC2)=O)CCOC2(C1)CN(C(C1(CC3CCC3)CC1)=O)C2 N1(C(C2N(CC)CCC2)=O)CCC(C)(C)C1CC(N1CC(C)(C)C1CN(C)C)=O c1(C(N2CCC(N(C(C(=O)NC)C(C)(C)C)CC)C2C)=O)cc2ncccn2n1 n1(CCNC(C2(CC)COC2)=O)ccc(C(=O)NC(c2noc(C)n2)C2CC2)c1 Cc1cnc(C(=O)NC2(CO)CN(C(c3cnn4cc[nH]c34)=O)C2)c(C)c1 CC1CC(NC(c2cc(CCO)on2)=O)CCN1C(=O)COC(F)(F)C(F)(F)F C1(CC#C)(C(=O)Nc2cccc(Nc3nccc(OC)n3)c2)CCCOC1 n1(CC(=O)NC2C(NC(c3ccc(CC)s3)=O)CC2)nc(C)ccc1=O N1(C(CC(C)c2ccco2)=O)CCCCC(N(C)C(c2cnn[nH]2)=O)C1 CCC(CC(=O)NOCC(N1CCC(OC)CC1)=O)CC(C)C Cc1c(NCC(c2ccsc2)C)ncnc1N1CC2CCC1CNC2 C1(CCC)CN(C(=O)C=Cc2cccnc2)CCN1C(=O)CNc1cccnc1 N1(C(C(c2ccn(C)n2)C)=O)CCN(C(c2c[nH]nc2C)=O)C2(CC2)C1 C1(OC(c2nc(Br)cs2)=O)CCCC(c2ccc(F)cc2)C1 c1(C(=O)NCCCNC(C2(C)CC=CCC2)=O)ccc(OCCF)cc1F c1(C(=O)NCCOCCN(C(C(C)NC(N)=O)=O)C)ccc(F)c(Cl)c1F CC#CCCCC(=O)NC1CCN(C(=O)Cc2c(C)nn(CC)c2C)C1C CCCCCCCCC(=O)NCC1(OC)CCN(C(=O)CC(CN(C)C)CC)C1 CC1CN(C(C2CCC(C(C)(C)O)CC2)=O)CCCN1C(=O)C1=CSCCO1 c1(C(=O)NC2CCC(NC(C(C3CCC3)OCC)=O)C2)c(OC)cccc1C N1(C(c2cc(CC)no2)=O)CCN2CCN(C(=O)C(=O)NC3CC3)CC2C1 c1(OC)cc(C(N2CCC(C(C)NC(=O)COc3ccon3)C2)=O)cc(C)n1 C(CN=c1[nH]nc(C(F)(F)F)o1)C1CCCN(C(c2cn3ccccc3n2)=O)C1 Cc1cccc2cc(C(=O)NC3CN(C(c4cc(O)nn4C)=O)CC34CC4)oc12 C1(CN(C)C)CN(C(=O)Cc2ccc(Cl)s2)CCC1NC(=O)CN1CCOC1=O N1(C(COC(C)(C)C)=O)CC2CC1CCN2C(c1cnc2nccn2c1)=O c1(NCCCCC=C)cc(N2CCN(CCN)CC2)nc(C2CC2)n1.C(N)=O C(=O)(C1=CCCCO1)NC1C(C)CN(C(C23CCC(C2)C3(C)C)=O)C1 C(CC(=O)NC1COCC1NC(=O)CC1CCCCC1)(C1=CCCC1)OCC CCC(C(=O)N1CCC(CNC(=O)CCCc2ccccn2)C1(C)C)C(C)(F)F c1(OC)cccc(C(=O)NC(C)C(C(C)C)NC(c2ccncc2)=O)n1 N1(C(C2C(C(C)C)C2)=O)CC(=O)NCC1C(=O)NCCc1nc[nH]n1 c1(C(N2CC(CC(C)NC(C3CCC(COC)C3)=O)C2)=O)cnccc1C C1(O)(CC(NOC2C(C)C2)=O)CCN(C(C23CC(C)(CCO2)C3)=O)CC1 S(=O)(=O)(CC(=O)NC1CN(C(=O)C(C)(Cl)Cl)CC1O)N(C)C C1(C(=O)NC(C2CC(NC(c3cc(O)n(C)n3)=O)C2)C)CC(F)C(=O)N1 N1(C(C(CC#C)NC(=O)CCc2cnoc2)=O)CCN2CCCC2C1 c1(C(N(C(C(=O)N(CC(=O)NCCC)C)C)CC)=O)cc(CO)[nH]n1 c1(C(=O)NCC2CN(C(C(F)=C(C)C)=O)C(C)C2)cccn2nnnc12 Cc1ccc2sc(CNC(C(=O)N)=O)nc2c1.c1(C)ncc(C)s1 C(=O)(C1=CCCCCC1)N1CCC(C(C)NC(C2CC(C)SCC2)=O)C1 N#Cc1c[nH]c(=NC2CN(C(C3CSC3)=O)CC23CCOCC3)c2sccc12 C1(C(=O)NCC2C(C)CCNC2=O)CN(Cc2ccccc2)Cc2ccnn2C1 C1(CCC(=O)NC)COCCN1C(=O)N(C1(c2cc(C)[nH]n2)CC1)C C1(N(C(=O)C(O)C2CCCC2)C)CCN(C(=O)CSC(F)(F)F)C1 C1(NC(C(C(C)C)(C)C)=O)CN(C(C2C=CC=CC=C2)=O)C2(CCOCC2)C1 C1(NC(C(C)Sc2ccccn2)=O)CCC(CNC(C2(F)CCC2)=O)CC1 CC1(C)CCCC1CCNC(=O)CCCn1cc(COc2ccc(F)cc2)nn1 C12(C(=O)NC(CNC(C3(CC4CC4)CC3)=O)C3CC3)CCC1CC2 c1(C(=O)NC2(CO)CCN(C(C3(F)CCS(=O)(=O)C3)=O)C2)csc2cncn12 c1(C2(CNc3nccc(OC(C)C)c3)CCCC2)ccc(F)cc1C(F)(F)F N1(C(CC2(COC)CC2)=O)CC2(CCC(CNC(C3Cc4nccn4C3)=O)O2)C1 C1(C(=O)NC2C3CN(C(c4n(CCC)nc(C)c4)=O)CC32)CNC(=O)CC1C C12(CC(=O)NCCCN(C(C=CC)=O)CSc3ccccc3)COCC(C1)C2 c1(CC)ccc2c(c1)CCN2C(=O)NC(C)CCOC N1(C(C(CC)N(C(=O)C(c2ccccc2)C)C)=O)CC2CC=CCC2C1 C(C1CCCN1C)=CC(=O)NC1CCC(NC(c2cc(C)on2)=O)C1 c1(C(=O)NCC23CC2CN(C(=O)C(F)C2CCC2)C3)ccc(=O)n(CCO)c1 c1(CC(=O)N(CC(C)(C)NC(Cc2c(C)scc2)=O)C)ccccc1OC(C)C N1(C(c2cccc(OC)c2)=O)CC2CCCC(C1)N2C(=O)C(N1CC2CC2C1)C c1(C2C(C(N3CCC(C(=O)NC4(CC=C)CCCC4)C3)=O)C2)ccc(F)c(Cl)c1 NC(=O)CC(C(=O)NCc1ccccc1)NC(c1n[nH]c(=N)[nH]1)=O CCCCCCC(COC)(c1nnnn1C1COC1)NCC(C)(C)OCCO c1(-c2cncc(C3CC(NCCN4C(O)CCC4)C3)c2)ccc(Cl)nc1 C1(C)(CNC(C(CNC(c2c(CC)noc2)=O)C)=O)CCC(=O)N1C C1(C)(C(=O)NCCCN(CC(c2ccccc2C)O)CC)CCCOC1 C(=O)(C1CCOc2c(F)cccc21)NC(CNC(CCC(=C)Cl)=O)(C)C(C)C Cn1nc(C(C)(C)C)cc1C(N1CC2CC2(CNC(C2CC2C(F)F)=O)C1)=O C12(C(=O)NC3CC(NC(c4cnns4)=O)C3)CCCN1CC(O)C2 CC(O)(C(=O)N(C1CC2CC1CN2)c1ccc(OCC(F)(F)Cl)nc1)C(F)(F)F C1C(C)(C)C#CC(=O)N1.C(C)(CC)(CC)N.N12CCC1C2=O.CC N1(C(CN(C(C)=O)C)=O)CCC(NC(C2C=CCC2)=O)C1(C)C n1(CCOC)nccc1NC(c1nnnn1C1CCC1)C1(C(F)(F)F)CC1 N1(C(C2SCCS2)=O)CC(C(=O)NCC2(C3CC3)CCCO2)C2(CCOCC2)C1 c1(N(C)CCCOC(c2nc(C)oc2)=O)nccc(-c2cnccn2)n1 C1(CNC(c2cn[nH]c2)=O)C(C2CC2)CCN1C(=O)CN1CCC(F)(F)C1 N1(C(Cc2ncc(C)o2)=O)CCC(NC(=O)C=Cc2ccc(Cl)s2)C(F)C1 CC(CC(C)(C)C)C(=O)N1CCN(C(=O)Cc2csc3nccn23)C(CCO)C1 c1(C(N2CC(NC(c3cncc(C(C)=O)c3)=O)C2)=O)c(C)cncc1C c1(CC(C)C(N2CCCC(C(F)(F)F)C2)=O)ccc([N+](=O)[O-])cc1 CCCC(O)C(=O)NCCNC(C1CN(C(=O)Nc2cnn[nH]2)C1)=O Cc1nc2ncnn2cc1C(=O)NCCOCCNC(C1CN2CCN1CC2)=O c1(CC(N2CC(NC(c3ccc(CC)cc3)=O)C(C)C2)=O)ccc(C)cc1F C1(NC(=O)Cc2ccc(CO)cc2)CC(F)CN(C(=O)Cn2nccn2)C1 C1(CC)C(NC(C2CC(=O)N(C)C2)=O)CCCN1C(c1oc(C)nc1C)=O c1(C(=O)NCC2CN(C(c3c(C)nsc3N)=O)CC2C)ccnc2[nH]nnc12 C(CCCCC(=O)N(C1CCCCN(C(=O)C(F)(F)C2CCOCC2)C1)C)=CC N1(C(C(CCCOC)C)=O)CC2(COC(CNC(=O)CCc3cscn3)C2)C1 n1(CCC(=O)NC(C2(O)CCN(C(=O)CCC3CC3)C2)C)ccc2cccnc12 N1(C(Cc2cc(C)no2)=O)CCCC2CN(Cc3csc(Br)n3)CC12 c1(OC)c(Cl)cc([N+](=O)[O-])c(Cl)c1NC(N1CCN(C(c2nccs2)=O)CC1)=O N1(C(CC(C=C)(C)O)=O)CCc2ccccc2C(NC(=O)CCc2cc[nH]n2)C1 c1(C(C(=O)NC)N(C2(C#N)CC2)C)ccc2c(c1Cl)OCO2 Cc1cnc(C(=O)NC2(CNC(=O)C3=CCCCO3)CCCCC2)cc1C#N C1(NC(c2cccc(CC)c2C)=O)CC(C2CCN(C(c3ccco3)=O)C2)C1 Cc1ncc(NC(C2CCCC2NC(c2ocnc2C2CC2)=O)=O)cn1 c1(OC(C)=O)ccc(C(N2CCC3C(C(F)(F)F)C23)=O)c(F)c1 c1(SC)nc(NC(=O)NC(c2ccccc2Br)CF)cc(C#N)n1 c1(OC)ccc(NCc2ccc(-n3cc(C(F)(F)F)cn3)cc2)cc1 c1(C(N2CC(CN(C(C3C(C)OCC3)=O)C)C2)=O)cc(F)cc([N+](=O)[O-])c1 CN1CC=C(C(=O)NCCCNC(c2conc2C(C)(C)C)=O)C1 C1(CNC=O)CCCC(CNC(c2cc(Cl)no2)=O)C1.C(C)(C)(C1CC1)OC C1(C(=O)OC(C)(C)C)CN(Cc2cc(-c3cn(C)nn3)on2)CC1C(F)F C(=O)(C1=C(C)OCCS1)NCC1CCCC(C(=O)NCC2(OCC)CCC2)C1 N1(C(CCCN(C(C)C)C(c2coc(C(N)=O)c2)=O)=O)CCCCC(C)(F)C1 C=CCC(F)(F)C(=O)NC1CCCC1CNC(C1C=CCS1)=O CC1CCC(C(N2CC(CO)C(O)C2)=O)N1C(=O)CC(C)(C)O C1(CNC(c2cncc(OC)n2)=O)CN(C(=O)C(F)C(C)C)CCN1C C(C(COC)C(F)(F)F)Nc1c(C(C(=O)OCC)(F)F)cn(C)n1 Cc1nc(C)c(CNC(C2CC(C)N2C(c2cc[nH]c2)=O)=O)s1 c1(C(=O)NCCCC(C)NC(=O)C=Cc2cnccn2)cccn2ncnc12 N1(C(c2cnc(C)nc2C)=O)CCC2(CC(NC(=O)C(C)n3cccn3)C2)C1 c1(C(N2C(C(=O)NCCC3(OC)CCC3)CC(F)C2)=O)cc(F)cc(Br)c1 C(=O)(C#CC1CCCO1)N1CCCC(O)(CNC(c2c(OC)c(F)ncc2)=O)C1 N1(C(n2ccnc2)=O)CCCC1CCCn1cc(CCO)nn1.C1(C2CC2)CCOC1 c1(NC(C2COCCN2C(C2CCCCO2)=O)=O)ccc(O)cc1 C12(C(N(C3CCN(C(C(C)n4cnnn4)=O)CC3)CCO)=O)CCCC1C2(F)F N1(C(C2N(C(C(=Cc3ccncc3)C)=O)CC=C2)=O)CC2CCC2(C)C1 N1(C(C(N2CC(C)C2)C)=O)CC(NC(c2cnc(-c3ccccn3)s2)=O)C(O)C1 C(=O)(C#CC1(C)CCCO1)N(CC(=O)NCC(C)O)CCC Cc1cc(C(=O)NCC2CCC(C)CN2C(=O)CN2CC(C)C2)nc(C)c1 CC1CN(C(c2cccc(CO)c2)=O)CC1NC(=O)Cc1cn(C)nc1Cl C1(CN(C(c2cnccc2OC)=O)CC)CCCN(C(C2CC2[N+](=O)[O-])=O)C1 CC12COC(C(=O)NCC3CN(C(=O)CSc4n[nH]c(O)n4)CC3O)(C1)C2 N1(C(C(N)=O)=O)CCC2C(NC(=O)CCCNC(c3c(F)cccc3Cl)=O)C2CC1 C1(N(C(CSCC)=O)C)CCCC(N(C(=O)CCC=C(C)C)C)C1 C1(NC(Cc2c(OC(C)C)cccc2)=O)CN(C(C2C=C2C)=O)C2CCCCC12 N1(CC(=O)OC)CCN(C(c2cc(Br)ncc2F)C(=O)NCCC2CC2)CC1C CCC(C)CN=C(NC1CCCCC1)N(C)CC1CCOC1 Cc1ccc2c(c1)N(C(=O)C(=O)NCC(C)CN1CCCC1=O)CCO2 Cc1nc2c(C(=O)N(CCNC(=O)C(C)CC3CCCO3)C3CC3)cccc2o1 CCCC(CNC(C1C2COCC12)=O)NC(=O)C=C1CCSCC1 c1(NC(C2=CCCN(c3ncnc(C)c3F)C2)=O)c(Br)cc(Cl)cc1C#N N#Cc1cc(C(=O)NCC23CC2CN(C(c2ccc(O)nn2)=O)C3)c(F)cc1F C1(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CN(C(=O)C(F)(F)CO)CC1O CCCCC(=O)N1CC(C(=O)NC(C(O)CO)C2CC2)(CC)C1 CC1(C(=O)NC(C2CCCC2)CNC(c2ccnc(S)c2)=O)CC(C2CC2)=NO1 c1(C(=O)NCC(CC)NC(=O)Cn2cc(Cl)cn2)cc2ccc(F)cc2nc1C C=CCCC(C)(C)C(=O)NCC1CC2CCC1N2C(c1ccc(CO)cc1F)=O c1(C(N2C3CC(NC(C(CC=CC)C)=O)CC2CC3)=O)cc2c(nc1N)CCC2 C1(C)(CC)CC(NC(c2n[nH]c3c2CCC3)=O)CN1C(c1ccnc(C)n1)=O C1(C(N2CC(C(CC)CC)C2)=O)CCN(C(=O)Cn2cnnc2O)CC1 Cc1ccc(C(=O)NC2CC(C)(NC(c3ccccn3)=O)C2)cc1Br C(=O)(C(CO)C(C)(C)C)N1CC2(CC(CC(N3CCC(OC)C(C)C3)=O)C2)C1 C1(C(=O)NCCCC)C2CN(C(=O)CCc3ccc(N(C)C)nc3)CC12 C1(CNC(C2(C(C)N)CCC2)=O)CC2(C1)CC2(F)F C1(C(=O)NCCCc2c(C)n[nH]c2)CCC(C(C)C)N1C(C1CC(C2CC2)C1)=O Cc1cc(NC(c2cnn(CCNC(=O)C(C)SC(C)C)c2)=O)c(O)c(C)c1 C1(C(=O)NC(CC(=O)OC)C)CCC(C)(C)N(C(C2CCC3(CC3)C2)=O)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCCCC(NC(C(C)Sc2ccc(C)cc2)=O)C1 CC1=NOC(C(N2CC(C)(NC(c3cc(CC4CCC4)c[nH]3)=O)C2)=O)C1 C#Cc1cccc(C(=O)NCC2(F)CCN(C(=O)C(C)C(F)(F)F)C2)c1 c1(C(N2CC(C)C(NC(=O)C=CBr)C2)=O)ccnc2c(F)cccc12 c1(C(N(CC(=O)NCC(F)Cl)CC2CC2)=O)c[nH]ccc1=O N1(C(C(C2CCOCC2)C)=O)CC2CC2(NC(=O)CCc2ncccn2)C1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(c2ccc(F)c(C3CC3)c2)=O)CC1CO S(=O)(=O)(c1[nH]c(=NCCC2(C)CC2)ccc1Br)NCC(=C)CC C1(NC(c2ncc(OCC)nc2)=O)COC2(C1)CN(Cc1nnnn1C1CC1)C2 c1(NC(c2nc(N3CCCC3)n[nH]2)=O)cc(N2CCNC2=O)ccn1 Cc1cc(=NC(=O)C2CN(C(c3c[nH]c(=N)o3)=O)CC2C2CC2)[nH]n1C1CC1 c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)CC2N=[N+]=[N-])n[nH]c2ccc(Cl)cc12 C1(NC(CC(CC)O)=O)CCCCC12CCN(C(c1sccc1F)=O)C2 C1(C)(c2onc(C)n2)CCN(C(=O)Cc2noc(-c3ccc(C(C)(C)C)cc3)n2)C1 c1(C(=O)NCCNC(=O)C#CC2CC2)c(Br)ccc(C(F)(F)F)c1F c1(C(N(C(C)CN(C(=O)CC2COC(C)(C)C2)C)C)=O)cc(F)ccc1Cl Cc1ccc(Cl)c(S(=O)(=O)Oc2cc(C)cc(C)c2[N+](=O)[O-])c1 c1(NC(C2(F)CCN(C(C3(CC=C)CCC3)=O)CC2)=O)ccc2nccn2c1 CC1CC(C)OC1C(N1CCCCC1C1CCCN(c2nccc(Br)n2)C1)=O c1(CCCCC)ccc(C(=O)NCC(C)(CO)NC(c2cnsc2)=O)cc1 N1(C(c2ncc(OC)nc2)=O)CCC(C(N2CCC(C(F)F)C2)=O)C12CC2 C1(NC(c2cnc3c[nH]nc3c2)=O)CC2CC(C1)N(C(C1CCCC(O)C1)=O)C2 c1(C(N2CCC(C)(C(=O)Nc3cncnc3Br)C2)=O)ccnc(Br)c1Cl c1(C(N2CCN(C(C(CCCC)CC)=O)CC(O)C2)=O)cnn2c1OCC(O)C2 N1(C(COCCCOC)=O)CCN(CC2CSCC(=O)N2)CC1 c1(C(=O)NCCCCCN(C)C(C2C3CS(=O)(=O)CC23)=O)ccc(F)c(O)c1F CC(CC(C)NC(c1ccn(C2CCCC2)n1)=O)NC(=O)C(C)(C)C C12(CNC(C(CC)OCC)=O)CCC(C1)N(C(=O)Cc1ccc(C)s1)C2 CC1CN(C(=O)C(C)(C)C(C)(C)C)CCCN1C(C1CCn2cnnc2C1)=O C(CC(N)=O)(C(=O)N(C)CCN1CCOC1=O)NC(c1cc(CC)[nH]n1)=O c1(C(=O)OC)csc2c1CCN(C(=O)N(C)CCc1ccccn1)C2 C1(C(=O)NC2CN(C(=O)CCn3ccc(C)n3)CC2O)(OC)CCCOC1 Cc1ncc(CCC(N2CC3(CC3)CC2CNC(C2C=CCCC2)=O)=O)c(O)n1 N1(C(CCN(C(C2C(CC)OCC2)=O)CC)=O)CC2(C=C(C(=O)NC)CO2)C1 c1(CC)ncncc1C(=O)NCC1(F)CCC(NC(=O)C(C)(CO)OC)C1 C(=O)(CCCC#N)NCC(CC)NC(=O)Cc1nc(Br)sc1C n1(C(C)C)ccc2cc(C(=O)NC(C)CN(C(=O)CSC(F)F)C)ccc12 C#CCCC(O)C(=O)NC(C)(CNC(c1ccc(C)n1C)=O)CC(C)C N(C)(S(=O)(=O)N1CC(C)(C)OC2(CCCCC2)C1)C(C(=O)NCC=C)CN(C)C c1(C(C(N2CC(c3oc(C(=O)NCC)c(C)n3)C2)=O)=O)cc(Cl)ccc1OCC C1(C(=O)NCC(CC)NC(=O)C(c2cccnc2F)(C)C)CC(=O)N(C2CC2)C1 N1(C(CN2CC(C)(OC)C2)=O)CCC2CCCC12C(=O)NC1CCSC1 N1(C(C2(C(C)C)CC2)=O)CC(NC(c2ccn(-c3cccnc3)n2)=O)C(O)C1 Cn1cc(C(=O)NC2CN(C(c3cnc(C#N)s3)=O)C2)c(-c2cccc(F)c2)n1 c1(C(=O)NC(CC)CN(C(=O)C(C)n2ccnn2)C)nn(C2CC2)cc1C C1(C(N(CCC)CCNC(=O)Cc2c(F)cccc2Cl)=O)CCN2CCCC2C1 N1(C(C(C)=CC)=O)CCC2(COC(CNC(c3cc4cnn(C)c4s3)=O)C2)C1 c1(C(N2CC(n3cc(C4(Cl)CC45CCC5)nn3)C2)=O)cccc2c[nH]nc12 N1(C(C(COCC)C)=O)CCCC(CC)(NC(c2ccc(Cl)cc2)=O)C1 CCC(C)(C(=O)NCC(C(=O)NCc1ccc[n+]([O-])c1)OC)OC c1(C(C(=O)OCC)(C)C)cccc(C2(CNC3CCOC(C(C)C)C3)CC2)c1 CCCC(CCCO)C(=O)NC(C1CN(C(=O)CC(C)(O)c2ccccc2)C1)C Cc1ccc(C(C)COC(=O)C(Cc2cn[nH]c2)N(C(=O)OC(C)(C)C)C)cc1 c1(CC(=O)NCCNC(C2C(C)C2)=O)ccc2sccc2c1 C(CC(CC)C(=O)N(C)CC1CN(C(c2ccc(C(C)C)cc2)=O)CCO1)=CC C=CCC(C)(C(=O)NC1(C)CCN(C(=O)Cc2n[nH]c(=NC)s2)CC1)N(C)C C=CCC(CC(C)C)C(=O)NCC(C)(O)CNC(=O)CC1=CCOCC1 N1(C(C(=O)NCCC2CC2)c2ccco2)CCC(C2CCC2)C1 C(CC(CC)C(=O)NCCC1CCCN(C(c2cc(CC)[nH]n2)=O)C1)=CC Cn1nnc(CNC(=O)CCC2CCCOC2)c1C(=O)NC1CCCC(CO)C1 C#Cc1cccc(C(=O)NC(C2CC(NC(=O)CC3CCCCO3)C2)C)c1 C12(CNC(C3C(C)CC3)=O)CCC(C(=O)O)(CC1)CO2 CC(CCC(=O)N1CC(CC(C)NC(C2CCCC(C)C2)=O)C1)c1ccccc1 N1(C(CCC2CC(OC)C2)=O)CCN(C(c2cn3ccsc3n2)=O)C2COCC12 C1(F)(C(N2CCC(CCNC(C3C(C)CCC3)=O)CC2)=O)CCN(C)CC1 c1(OCC(=O)NCC(C)(CO)NC(C2C(CCOC)C2)=O)cncc(Cl)n1 c1(C(=O)NCC#CCNC(=O)CC2CCC3CC23)c(F)ccc(F)c1F C(C(F)(F)C(=O)OCC(=Cc1ccccc1)C)OC c1(C(c2n(CC(=C)C)nnn2)NCC2CC2[N+](=O)[O-])ncc(OC)cc1F c1(CCCC2C(C)C2)ccc2cc(S(=O)(=O)NC3C=CC(C)(C)CC3)ccc2n1 C1(CNC(CCC=CCC=C)=O)CCN(C(c2cnnc(C)c2C)=O)CC1O Cc1ccc(C(=O)NCC2CCN2C(=O)C=Cc2cc[nH]n2)cc1Br N1(C(CC(C)NC(N)=O)=O)CC2(CCN(C(=O)C(C)(C)F)C2)C1 C1(CNC(c2cncc(C)n2)=O)CC(C)(C)CN1C(=O)C(O)C(C)C c1(C(=O)NC2CCCN(c3ncc(C(F)F)cn3)CC2)ccc(F)c(F)c1F C1(C(=O)NC2C(CNC(CCNS(CC)(=O)=O)=O)C2)CC(S(N)(=O)=O)C1 c1(NC(c2nc(-c3cnc(OCCC)nc3)sc2)=O)c(OC)ncc(Cl)c1C C1(NC(C=CCOC)=O)CC2CN(c3nc(OC)c(F)c(C)n3)CC2C1 N1(C(CC2OCCN(C(CNC(CC)=O)=O)C2)=O)CC2CCCCC2C1C C=CCC(C(=O)NCCC1=CCN(C(c2ccc(Br)c(C)c2)=O)CC1)C(C)C C#CC1CCCN1C(=O)C(=O)Nc1ccccc1NCC C1(NC(C=CCOCCOC)=O)CCC2CN(C(C3CC(=O)NC(=O)N3)=O)CC12 CC1CC(C(=O)NC2CN(C(c3ccc(-c4cnn(C)c4)o3)=O)C2)CC(C)C1 Cc1ccc(CN(CCCN=[N+]=[N-])C=O)cc1C1CC1 C#CCCCCN=C(NCS(C)(=O)=O)NC1CCS(=O)(=O)C1 N1(C(C2CC(=O)N(C3CC3)C2)=O)CCCCC2C1CCCN2C(=O)C1=CCC1 Cc1nc2cc(-c3ccc4oc(NCc5c(F)cccc5Br)nc4c3)ccc2s1 N1(C(C2C(OCC)C2C)=O)CCCC(CCNC(=O)CCC2CCOC2)C1 C(=O)(C(O)CC1CCCCC1)NC(C)CNC(C1(Cc2cnn[nH]2)CCCC1)=O C1(CNC(C2(C(C)C)CCC2)=O)CCCCC1C(=O)NCc1c(C)nsc1 c1(C(=O)NC(CC(=O)NCC(N(OC)C)=O)C)cc(O)ncc1F c1(CCCC(N2C(CNC(C3N(CC)CCC3)=O)C=CC2)=O)cc(C)ccc1C C1(NC(=O)Cc2ccc(O)nc2)CC2CCC(C1)N2C(=O)CN1CCC1 N1(C(C2N(C(c3cc(Cl)no3)=O)CCC(=C)C2)=O)CCc2nocc2C1 C12(NC(CCC=C)=O)CCCCC1N(C(C1CCC(C)CC1)=O)CC2 C12(NC(C(N3CCSCC3)C)=O)CCOC(CNC(=O)C3=NNC(=O)C3)(C1)C2 C1(NC(Cc2nc(CC)sc2)=O)CS(=O)(=O)CC1NC(=O)C=NOC C1(C(=O)NC(C2CCOC2)CO)CN(c2ncc(F)cn2)CCC1O N1(C(C2C(C#N)C2)=O)CC(C(F)(F)F)CC1CNC(c1coc(Br)c1)=O N1(CC)N=C(C(=O)N2CCCC2CNC(C2CC(=O)N(O)C2)=O)CCC1=O C1(C(N(C)CC2CCN(C)C2)=O)CCN(C(=O)CC2OCCO2)C(C)(C)C1 C1(C(N(CC(C)(C)C(=O)NC(C)CCCCO)CC)=O)OCC2CCCC12 CCCCC(O)CC(=O)NC1CCC(C(=O)NCCc2nnc(C)n2C)C1 C1(CCNC(C2CCC2C)=O)(NC(C2CN(S(CC)(=O)=O)C2)=O)CCCC1 c1(C(N2CC(CC(C)NC(CN(CC)CC)=O)C2)=O)cnc(C)nc1C C=CCCCCC(C(=O)NCC)N1CCCCC(Cn2cncn2)C1 C1(OC)CC2(CCN(C(=O)CCC=C(C)C)C2)C1.C12CC1COC2=O CC1(C(N2CCC(O)(CNC(c3nccnc3N)=O)CC2)=O)CCCC(F)(F)C1 c1(C(=O)NC(C2CCN(C(c3cccc(SC)c3)=O)C2)C)cccc(F)c1O c1(CC)cccc(C(N2CCCC2(C)CNC(=O)CCc2cn[nH]c2)=O)c1F C(N=c1nc(C2CC2)[nH]s1)C1CCC(NC(=O)CCOc2cccc(F)c2)C1 C(=O)(C(CC(C)C)NC(C1(C)CCN(C(C2CN(C(N)=O)C2)=O)C1)=O)NC N1(C(c2ncc(C)cc2F)=O)CC(CNC(c2c(C)nsc2N)=O)C2(CCC2)C1 C1(C(=O)O)CC12CCc1cc(Br)ccc12.c1(C[SH](=O)=O)cc(Cl)ccc1Br C1(C(C)NC(=O)CC2OCCC2C)CN(C(c2ccncc2Cl)=O)CCO1 c1(C(=O)NC(CC(C)NC(=O)C(C)(C)n2ccnn2)C)ccc2[nH]ccc2c1 c1(C(N2CCC(N(C(c3cc(Br)c(C)s3)=O)CC)C2)=O)c(C)ccc(C)c1O C1(N(C(=O)CC2OCCO2)C)CCCN(C(C2(C3CCC3)CC2)=O)CC1 CC1(C)CC(=O)N(CC(=O)NC2CC(C)C2(C)C)C1=O.C1(C(=O)N)CC(=C2CC2)C1 C(=O)(C(CC(C)C)C(N)=O)N1CC(OCC)C1.c12ccc(Cl)nc1NC2=O C1(NC(C2(C(C)(F)F)CC2)=O)CCCC1CNC(=O)COC1CCOC1 C1(CC#C)(NC(c2occc2CNC(=O)C(O)CC2CCCC2)=O)CCOCC1 C1(NC(C(C)OCOC)=O)CCCN(C(=O)CCN2CCC2)C1 C1(CC(=O)NCCCO)CN(C(c2cn(C3CC3)nn2)=O)CC12CC2 c1(CC(=O)NCCN(CC(C)O)C(C2CC3CC3C2)=O)cccnc1F c1(C(N)=O)cc(=NCC2CC(C)(C)CCC2NC(=O)Cc2cnsc2)[nH]cn1 CCCCCC(F)C(=O)NCC(CCC)NC(C1(S(N)(=O)=O)CC1)=O O=C(N=c1cccn[nH]1)C1CC12CCN(C(=O)Cc1ccc(Cl)c(F)c1)C2 N1(C(C(CC)CCOC)=O)CC(C)(C)OCC1CNC(=O)CC(C)(C)C1CC1 C=CC(CC)CC(=O)NCC1(C(C)(C)C)CCN(C(=O)CCC2CCC2)C1 c1(NC(CN(C(c2ccc(OC)cc2)=O)CC)=O)ccc2cccnc2c1 Cc1nnc2n1CC(NC(N1CC3CC4CC3C1C4N)=O)CC2 C1(CNC(C2CC(CNC(=O)COCCC3CCCC3)C2)=O)CC2CCCC2C1 C1(NC(CC(C)=C(C)C)=O)CC2(C1)CC(C(=O)NC(C)C(C)n1cccn1)C2 C(=O)(CC(C)(C(F)F)N(C)C)NC1CC(NC(c2c(C)scn2)=O)C1 Cc1nc(CC(=O)NCCCC2(NC(c3ccn(CCO)c3C)=O)CC2)c(C)s1 N1(C(C(C(=O)OCC)(C)C)=O)CC(NC(=O)C=CC2CC2)C2(CCOCC2)C1 c1(N2CC(C)(C)C(NC(=O)C=CCN3CCCC3)CC2)nc2cccc(Br)c2o1 Cn1nc(C2CCC2)cc1C(=O)NCCCCNC(=O)CC1(O)CCC1 C(=O)(CCS(=O)(=O)N(C)C)NCC(CNC(C(C)Oc1ccc(C)cc1)=O)F C1(OC(C)C)CC(C)CC1n1cccn1.N12CC1C(c1cncn1C)CC2 C(CN=c1[nH]c(Cl)c(C#N)s1)(C1CC1)NC(C1C2(CC(C)(C)C2)C1)=O CCC(CC(=O)NCC1COCC(C)O1)N(C(=O)CN1C(=O)CCC1=O)C N1(C(C2(F)CCN(C(Cc3c(C)cccc3)=O)CC2)=O)CC2CCC(C1)N2C C(c1ccccc1NC(C(=O)NC(C#C)(C)C1CCC1)=O)=CCCN c1(C(=O)NC2(C)CCCN(C(Cc3n[nH]c(=NC)s3)=O)C2)ncnc2c1CCC2 CC(C)CCCC(c1cnc(OCC(N2CC(NC(=O)OC(C)(C)C)C2)=O)s1)C c1(C)ccc(OC)cc1.c1(C(c2nnnn2C2CC2)NC(COC)C)ccccn1 C(=O)(N=c1ccn(C)[nH]1)c1cc(CNC(c2cncc(C)c2)=O)ncc1 c1(C(=O)NCCCCCCNC(C2C(C)(C)C2(F)F)=O)ccc(Cl)cc1N c1(C(N2CCC(C(C)NC(CSc3nc(C)[nH]n3)=O)C2)=O)cn(C)[nH]c1=N c1(C(=O)NCC2(C(=O)NC(c3cnccn3)C)CC=CC2)cc2cnccc2[nH]1 C1(C)(NC(C=C2CCN(C)CC2)=O)CCCN(C(C2CCNC(=O)C2)=O)C1 CC1CN(C(=O)C(=O)NCc2ccc(CO)o2)CCN1C(C1CCC1)=O C1(CC(=O)NCC2(NC(C34CCC3CC4)=O)CCC2)CCS(=O)(=O)C1 N1(C(C(C)NC(C2CCCC2)=O)=O)CCC(NC(c2ccc(Cl)[nH]2)=O)C12CC2 N1(C(c2c(C)noc2C)=O)CCC12CN(C(C1(C#N)CCCC1)=O)C2 Cc1ccc(F)c(C(c2nnnn2C(C)C)Nc2cc(N(C)C)nc(Cl)c2)c1Br Cc1cc(=N)[nH]cc1C(=O)NC1CCC(N(C(=O)CC(C)C2CC2)C)CC1 C1(C(=O)NCc2ccoc2)CC2CCCC2N1C(=O)Cn1c(O)nnc1O Cn1ncc(C(=O)NCCC2CC(NC(c3ccc(Br)o3)=O)C2)c1F C(=O)(NNc1ncnc2sccc12)c1cn(C)nc1 c1(C(=O)NCC(CN(C(=O)Cc2cc(Cl)n(C)n2)C)O)cc(Cl)cc(Cl)c1 C(=O)(C1CCc2cccc(Cl)c21)NCC1C(C)C1 Cc1c(C(=O)NCC(C)CNC(=O)CCc2cn(C)nn2)nnn1C(C)C C(=O)(C(C)(C)CC(F)(F)F)NC1CN(C(c2cc(OC)c(C(N)=O)cc2Cl)=O)C1 CC(C(=O)N1CC(F)(F)CC1CNC(C1CC1(C)C)=O)S(C)(=O)=O c1(C(CC(C)C)NCC2C(C(=O)OC)CCC2)cc(OC)cc(OC)c1 C(=O)(C(C)(C)CC(F)F)N(CCC(=O)NC1CC(O)C1OC)CCC C1(C(N2C(CNC(=O)C(C)(C)CN(C)C)CC(OC)C2)=O)CCc2nc[nH]c2C1 C(=O)(CC(F)(F)CC)N1C(C2CCN(C(c3cnc(SCC)s3)=O)C2)CCCC1 C#Cc1cc(C(=O)NCC(CC)NC(=O)C(O)c2ccsc2)cc(Br)c1 c1(C(=O)NC2(C(C)(C)C)CCCCC2)ccc(Cl)c(I)c1 C1(NC(CC2C(C)CN(C(C3(N(C)C)CCOC3)=O)C2)=O)CC(F)(F)C1(C)C c1(C(=O)N=c2ccn(CCC3CC3)[nH]2)cn2cc(Cl)cc(Cl)c2n1 c1(C(N2CC(O)(C(C)NC(=O)C=CC3CC3)C2)=O)c(F)ccc(F)c1Cl c1(C(=O)NCCOC2CCN(C(CC=C(C)C)=O)C2)c(C)nn(C)c1Cl C1(N(C(c2ccsc2)=O)CC)CCN(C(C2CC3CCC2O3)=O)CC1 c1(C(N2CC(CNC(C(C=C)(C)O)=O)C(C)CC2)=O)ccc2c(c1)CN(C)C2 c1(OC)nc(C)c(Br)cc1C(=O)NC1CC(NC(=O)CSC2CC2)C1 N1(C(CCCc2cn(C(C)C(=O)N3CCCC3)nn2)=O)CCn2ncnc2C1 C1(CNC(COCCCOC)=O)CN(C(=O)C(N2CCOC2=O)C)CC1C(F)F C1(C(N2CCC(C(C(=O)N(CCCC(C)(F)F)C)F)C2)=O)CC(O)CN1C S(=O)(=O)(CCCCS(=O)(=O)NC12CCCC1CS(=O)(=O)C2)NCC#CCOC C1(C(=O)Nc2c(C(=O)OC)ccc(C)n2)CCC2(CN(C(=O)CNC(N)=O)C2)O1 c1(OC)ccc(-c2nc(CC(N3CCC(NC(=O)C(F)C4CC4)C3)=O)cs2)cc1 C1(F)(CNC(c2ccc(Cl)s2)=O)CN(C(=O)CCOC2CCCOC2)C1 C(=O)(C1Cc2ccccc21)NC(C1CN(c2nc(C)nc(Cl)c2C)C1)C c1(C(=O)NCC2(C)CN(c3ccnc(OC)n3)C2)cc2[nH]ccc2cc1Cl C1(CN(C(C2(CC)CC2)=O)C)COCCN1C(C1CSCN1CC(C)C)=O c1(OC)ccc(C2CC2)c(C(=O)NCC(C)(CO)NC(c2nocc2Cl)=O)c1 CCCCCCC(=O)NCCN(C(=O)C(c1c(F)cccc1F)C)CC N1(C(C(CC)C(=O)OC)=O)CCC2(CC1)C(NC(=O)C(C)C(C)O)CS2(=O)=O C1(N(C(=O)CC2(O)CC2)C)CCN(C(C2(n3cccn3)CCC2)=O)C1 C1(C(=O)OC)CC=CCC1CC(=O)NC(c1snc(C)c1N)=O n1(CC(C)O)cc(C(N2CCC23CN(C(c2scnc2C)=O)C3)=O)ccc1=O c1(C(=O)NCC(=C)CCNC(C2CCC(=O)O2)=O)cc(C)nc2[nH]nc(O)c12 Cc1c(C(=O)N(C)CC2CCCN2C(C2NC(=O)OC2C)=O)ccn1CC1CC1 C1(N(C(C(C)OCC=C)=O)C)CCCN(C(=O)Cn2cncn2)C1 N1(C(C=CC=CC)=O)CCCCCC1CNC(=O)Cn1cnccc1=O C(=O)(C(O)CC(N)=O)NC1(C(=O)NC(C(C)(C2CC2)OC)C)CSC1 c1(C(N2CC(C(=O)Nc3c(Cl)ncc(Br)c3Cl)SCC2)=O)ccc2cc[nH]c2n1 C=C(C)CC(C)C(=O)NC1CC1CNC(=O)Cn1cnc([N+](=O)[O-])n1 C1(CC)C(C(=O)NCCN2C(=O)CCC2=O)CCN1C(=O)CC1CCCN1C c1(CC)ccccc1C(F)(F)F.c12cnn(C)c1CN(C1CC1)C2C(=O)NC C1(c2c(N(CC(C)(C)C)C)c[nH]n2)CCCN(C(=O)C(=O)N)C1.C(C)(C)(C)OC=O c1(-c2n(C(CC)CC)nc(-c3nc(C)cs3)n2)ccc2nc[nH]c2c1 c1(-c2c(C(=O)NC(C(C)NC(=O)CSCCC#N)C)cno2)cccc(Cl)c1Cl n1(CC(N2CC(CC(=O)NCc3c(C)nns3)C(C)C2)=O)ccc([N+](=O)[O-])n1 c1(C(C)=O)ccsc1C(=O)NC1CC(F)(CNC(c2ccc(Br)s2)=O)C1 c1(C(=O)NCC2(O)CC(NC(C(CCC#C)O)=O)C2)[nH]c2c(C)cccc2c1C c1(CCC(=O)NC(CN(C(c2csc(C3CCCO3)n2)=O)CC)C)cncn1C C1(C(N(CC(C)NC(=O)CS(C)(=O)=O)C)=O)COCCN1CC(F)F c1(N(C)Cc2cccc(C)c2)nc(=NCCn2cnnc2)[nH]c2cc(F)ccc12 C(=O)(CC1=CCOCC1)NCC1CN(C(c2c(C)sc(C)c2C)=O)CC1C C(=O)(C(CC(C)C)NC(C1(OC)CCC1)=O)NCC(COC)C(C)C c1(C(N2CC(NC(C(C3CCC3)OC)=O)(COC)C2)=O)cc2nc(C)[nH]c2cc1F CC1CC(C(=O)N2CC3CC3(CNC(=O)Cc3cncnc3)C2)=NO1 c1(C(NON2CC(C=O)(CO)C2)=O)cc(OC)c(C)c(OC)c1.N(C)(C1CC1)CC C(CCN=c1[nH]ncs1)NC(C1CCN(C(C(COC)OC)=O)CC1)=O c1(OC)ccc(C(=O)NCC(C(C)C(C)C)NC(c2cccn2C)=O)nc1OC N1(C(c2c(C)onc2Br)=O)CCC(C2CCN(C(=O)CC3CC3)CC2)CC1 N1(C(C(C)(C)SC)=O)CCCC2(C1)C(NC(c1ncncc1Cl)=O)CCN2C C12(NC(=O)CC(C)O)CCCC1N(c1c(-c3nc(C)sc3)c[nH]c1)CCC2 CCC(CNC(C1(SC)CC1)=O)NC(=O)COC(C)C N1(C(CSCC#C)=O)CC2(CC(NC(c3ccc(=O)n(C)n3)=O)C2)C1 C1(N(C(c2cnc(COC)s2)=O)C)CCCN(C(C2(CF)CC2)=O)CC1 CC1CCC(CNC(c2cc(Cl)c(Cl)[nH]2)=O)CN1C(c1ccncc1)=O N1(C(c2c(OC)cc(Cl)cc2)=O)CC(NC(=O)C(C)CC(C)C)C(C2CC2)C1 Cc1cc(C(N2CCC(C)N(C(=O)C3=NOCC3)CC2)=O)n2ncnc2n1 CC1CC(CNC(=O)C(C)(O)C2CC2)CCN1C(c1coc(C2CCC2)n1)=O CCCC(O)CC(=O)NC(C)(C)CN1CCN(C(=O)C(C)(C)CC2CCC2)CC1 N1(C(CCCNC(N)=O)=O)CCOCCC1C(=O)NCC1CC12CC2 c1(CC(N2CC(NC(c3c(COCCOC)ocn3)=O)C2)=O)c(F)cccc1F C#CCC(C)(C(=O)N1CCSC(C)(C)C1)NC(=O)C(C)NC(N)=O C1(=CC(=O)NC(CNC(=O)C(c2ccccc2)O)C2CC2)CN2CCC1CC2 CCC(C(=O)NC1(CNC(C2(CF)CC(=O)C2)=O)CC1)n1cncn1 C=CCCC(O)CNC(=O)CCN(C(=O)C=Cc1ccccc1)CCOC C=CC(CCC)CC(=O)N1C(CNC(c2ccc(CN(C)C)cc2)=O)CC2CC12 CC(O)(C(=O)NC1CCCC(C(=O)Nc2nc(Br)cs2)C1)C(F)(F)F c1(CC(C(=O)NCCC2CC2C)NC(c2c(CC)c[nH]n2)=O)ccc(Cl)cc1Cl N1(C(C(C)C2CCCOC2)C(=O)NC2COC2)CCC(O)C(F)(F)C1 c1(C(=O)NCC(CNC(CC(COC)C)=O)OC)cc2sc(Cl)cc2s1 C1(C(N2CCC(F)(F)CC2)=O)CC2(CC2)CN1Cc1ccc(Cl)cc1C(=O)O S(=O)(=O)(c1ccc(N2CCCC(C3CC3)CC2)c2cnccc12)NC(CC)CC C12(NC(c3c(NC)scn3)=O)CCC(CC1)N(C(=O)C(C1CC1)OC)C2 c1(OCC(=O)NCCN(C(=O)CN2CC(=O)NC2=O)C)cc(Cl)cc(Cl)c1 C1(NC(C(C)(CO)OC)=O)CC2CCCC(C1)N2C(c1cc(C)n(C)c(=O)c1)=O c1(C(=O)NC2CN(C(C(C(C)C)O)=O)CC2O)cn2cccc(Br)c2n1 Cc1nccc(C(N2CCC(C)C(CC(=O)NC3CCN(C)CC3)C2)=O)c1N N1(C(C(=O)N(C)Cc2ccc(OC)cc2C)C)CCC2(CCCCO2)CC1 C1(C(=O)NCCC(CC)(C)NC(c2cnsc2)=O)CC2C=CCC(C1)C2 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCc1cc(F)ccc1Br C(C(CC(C)C)C(=O)N1CC(F)(CNC(C2CCCN2c2nccs2)=O)C1)OC N1(C(c2c(OC)oc(C)n2)=O)CCN(C(c2cc(Cl)sc2Cl)=O)CC(C)(F)C1 C1(COC)CN(C(=O)C#CCNC(=O)CC2CC(O)C2(C)C)C1(C)C C=CCCC(CC(C)C)C(=O)NCc1cccc(N(C(=O)C2=C(C)CCC2)CC)c1 Cc1nc(N2CC3(CCCC3NC(C3CC=CCO3)=O)C2)c(F)c(C)n1 Cc1cc(C)n(CCCN(CCN(C)C)Cc2ccc(C)o2)c1 CC1CC(CC(=O)N(C(C)(C)C)C(C2CCCN(CC#N)C2)=O)CCC1C CCCCCCC(C)(C)C(=O)N1CCC(CNC(C2CCN2CC)=O)C1 C(CC(C)(C)C(=O)NCC(C)NC(C1CCCN1c1nc(C)cs1)=O)OC C1(CNC(COC)=O)CC(CNC(=O)CNC(C2CCC2)=O)CO1 C(=O)(C(F)(F)C1(O)CCC1)NCC=CCNC(C1CC1F)=O C1(N(C)C(c2cc(O)nn2C)=O)CN(C(C2(N(C)C)CC2)=O)CC12CC2 c1(OC)c(C(=O)NC(C)CC2CN(C(c3ccc(C)s3)=O)C2)cccc1F N1(C(C2COC(=O)O2)=O)CC2(CCC2)CC1CNC(=O)Cn1ccnn1 C(CN=c1cc(C)nc(CO)[nH]1)(C1CCCC1)NC(C(C(CC)O)C)=O c1(CC)ccccc1C1C(=O)OCC(C)N1C1CCOC1.C(C)(=O)NCC C1(C(=O)NCC2N(C)CCC2)CN(C(=O)CC2C=CCC2)CC12CCC2 N1(C(C(C)SCCCC)=O)CC2CC(C1)N(C(c1ccc(C)n1C)=O)C2 CC1CN(C(c2nn(C)cc2Br)=O)CCN1C(C1CCC(C(N)=O)CC1)=O C(CCCCC(=O)NC(C)CCCC(=O)NC1(CCO)CCCCC1)=CC N1(C(C2C(C)C2C)=O)Cc2ccc(Br)cc2C1 N1(C(CSC(C)C)=O)CCOCC(F)(CNC(c2nnn(C(C)(C)C)n2)=O)C1 N1(C(c2c(Cl)nc(OC)s2)=O)CC(NC(c2cnoc2C2CCC2)=O)CC(O)C1 Cc1ccnc2c(C(=O)N(CC(C)NC(=O)C(F)(F)CN(C)C)C)cnn12 C(=O)(CCC(=O)NCC1CN(C(=O)CCc2cnc(Cl)nc2)CCO1)NC C1(NC(=O)C(C2CCOCC2)F)C2COCC1CN(C(c1ccnnc1)=O)C2 CCC(CC)C(C(=O)NCC1(C)CCCN1C(C12CCCN1CCC2)=O)OC c1(OC)ccc2cnc(Sc3ncnc4ccoc34)nc2c1 C1(C(N2CCC(NC(COC)=O)C2C(C)(C)C)=O)CC(C)(C)OC(C)(C)C1 C1(C(N(CC(C)NC(C2SCCS2)=O)C)=O)CCCOC1C Cn1nc(C2CCCC2)cc1C(N1CCCC1Cc1cn(CC(C)(C)O)nn1)=O C1(C(=O)NCC)CCCN(C(=O)C(c2ccc(Br)cc2)OC)C1C CC1CN(C(C2CCCNS2(=O)=O)=O)CC(C)N(C(=O)CCC2(O)CCC2)C1 c1(SC)nc(Cl)c(CNC2C(F)(F)CCN(C(c3ccc(O)nc3)=O)C2)c(Cl)n1 C1(n2cc(C3(C)CC3)nn2)CCCNC1C1CC1.C(=O)NNC(=O)c1ccccc1F C(=O)(C#CC1CCOC1)C(CCC#C)=O.C12(C(CN)N)CCC(CC1)C2 C(=O)(CC(CC)(C(F)F)NCc1cnc(-c2cnccn2)s1)OCC N1(C(C(CC)=CC)=O)CC(C)N(C(C2CN(C(=O)CC)C2)=O)CC1C.OCC CCC(O)CC(=O)NCC1(C(=O)N(C2CCOCC2C)C)CCC1 N1(C(=O)CCC2CCCC2)CCCC(NCc2ccc(O)nc2)C1 Cc1cc(=NC2CC(c3ccccc3Cl)C2)[nH]c(=NCCCc2ccncc2)[nH]1 C1(CNC(CC(=C)C)=O)CCCN(C(c2ccncc2O)=O)CC1 n1(CC)ncnc1C(=O)NCC(C1CCCC1)NC(C1CCC(=O)N1)=O c1(OC)ccc(NC(=O)C(c2cn(C)nc2C)N(CC(C)COC)C)cc1 c1(CC)nc(C)oc1C(=O)NCCC(O)CNC(=O)CC(c1ccccc1F)C c1(-c2nc(CC)on2)cccc(C(=O)N(CCOCC)CC2CCOCC2)c1 C(C1c2ccsc2CCN1C(=O)C(C)CC(C)C)NC(C(COC)(F)F)=O C1(C(=O)NC(CNC(c2cnc(COC)s2)=O)(C)CO)CC(C(C)C)=NO1 Cc1nc(Cl)[nH]c(=NC2CCC(NC(=O)CCCC(=O)N(C)C)CC2)c1[N+](=O)[O-] c1(C(=O)NCCC(=C)CNC(c2nnc(S)n2C)=O)c(C)ccc(C)c1N C1(NC(CCC(=O)OCC)=O)CCCCCN(C(C2(C(F)(F)F)CCCO2)=O)C1 C#CCCCCCC(=O)N1CCC(C2CCCN2C(=O)CN2CCCCCC2)C1 C1(F)(CNC(C(C)c2ccsc2)=O)CCC(CNC(=O)CNC=O)C1 C1(C2CCCC2)(CNC(C2CCN(C(c3c(C)n(C)cn3)=O)O2)=O)CC1 C12(NC(=O)NCc3coc(-c4cc(Cl)ccc4Cl)n3)CCCC(CO)(C1)C2 c1(C(=O)NC2(C(=O)NCc3cnco3)C(C)C2)nsnc1O CCCCCC(C)(C)C(=O)NC(C1CN(C(=O)C(CC)c2ccccc2)C1)C C(CC(C)C)(C(=O)NCC(C1CC1)N(C)C(C1(c2ccccc2Cl)CC1)=O)OC CC1=C(C(=O)NCCC(O)CNC(=O)CC2CN(C)C2)SCCO1 CC1(C)CCN(C(c2cccc3c2COC3)=O)CC1NC(C1CC=CCC1)=O C1(NC(C(c2c(C)cccc2)C)=O)CC(F)CN(C(c2ccn(C)n2)=O)C1 C1(NC(C(CN(CC)CC)F)=O)CCN(C(=O)CC2CC(C)=NO2)C1(C)C c1(C(N2CC(CC(CNC(C(CC)C)=O)(C)C)C2)=O)cc2cccc(N)c2cn1 c1(NC(Cc2cccc(OCC#N)c2)=O)ccc(N)cc1[N+](=O)[O-] N1(C(c2c(C)cc(F)s2)=O)CC2(CCCCN(C(=O)C(C)Cn3ccnc3)C2)C1 CCCCCCC(C)(CC)C(=O)N1CCCC(N(C(=O)C(=O)N(C)C)CC)C1 N1(C(C2C(=C)CC2)=O)CCCC(N(C)C(c2cccc(CNC(C)=O)c2)=O)CC1 C=CC(C)(CCOC)C(=O)N1CCCC(C(=O)NOC(C)C(=O)OC)C1 N1(C(C2(SCC)CC2)=O)CCCC(COC)(NC(=O)C(C)(C)c2cnco2)C1 C1(C#N)(CCC(N2CC(CNC(=O)OC(C)(C)C)C2)=O)CCC1 CCCCCC(=O)N1CC(COC)CC1CNC(C1CC1CCC)=O C1(C(=O)NC2C(C)N(C(=O)CCOCC3CC3)CCC2)Cc2ccccc2CO1 CC1CN(C(C2CCSCC2)=O)CC(C(=O)NCC2(C)COCCO2)O1 C1(NC(C(CCN(C)C)NC(C2CC(CF)C2)=O)=O)CC12CCCCCC2 C(C)(CCC(=O)NCC1(CNC(c2ccc(N)cn2)=O)CC1)OC C1(c2nnnn2CC2CC2)(NC(C(C(=O)O)C2CCCC2)=O)CCC(F)(F)CC1 C=CCCCCCC(=O)NCC(c1ccccc1)N(C(=O)C=CC1CC1)C c1(C(N2C(CNC(C(C=C)O)=O)CC(OC)C2)=O)cccc(F)c1Cl CC1C2CCCCC2CN1C(=O)CN(C1CCC1)C(C1CCC(O)CN1C)=O C1(CC(N2CCCC(CF)C2)=O)C2CCC(C2)N1C(=O)CNc1ncccn1 N1(C(C2C(C)(C)C2)=O)CC(NC(c2cccc(P(C)(C)=O)n2)=O)CC12CCOC2 Nc1c(O)ccc(Cl)c1C(N1CC2C(CNC(C3CCCN3C=O)=O)C2C1)=O Cc1cc(C(=O)N(C(C)C(=O)NCc2nc(C)sc2C)C)n(C)n1 C1(C(=O)NCCCN(C(=O)C(C2CCS(=O)(=O)CC2)(C)C)C)C(F)(F)C12CCC2 n1(CC(=O)NCCCCN(C(c2cn(CC)nc2)=O)C)cccc(C)c1=O CN=c1ccc(C(N2CCCC(CNC(=O)C=C3CCC(C)C3)CC2)=O)c[nH]1 CC1CN(C(C2CC23CCCC3)=O)CC(C(F)(F)F)O1 N1(C(C2N(C(=O)NC)CCC2)=O)CC(NC(c2cc(Br)co2)=O)CC(F)C1 C1(NC(C2(C(N)=O)CCC2)=O)CC2CC(C1)N(C(c1cccc(N)c1F)=O)C2 CC1CN(C(c2ccc(C(C)(F)F)cc2)=O)CCC1CNC(C1CC(C)C1)=O N1(C(CCCSC(C)(C)C)=O)CC=C(C(=O)N2CC(CO)C(C)(C)C2)C1 n1(C(C)C)nccc1C(N1CCC(CN(C(=O)C(O)CC2CCCC2)C)C1)=O c1(C(N2C(C(=O)NCCCSC)CC(=C)C2)=O)c(Cl)ccc(Br)c1Cl Cc1nc(C2CCN(CC3CNC(C)C3)CC2)nc2c1CCC2 CCC(C)(C)CCCC(=O)NCC1CCCC1NC(c1nc(Cl)oc1C)=O C(C1CCOC1)=CC(=O)NCCN(C(=O)C=CSc1ccccc1)C c1(C(N(CCN(C(=O)C(=O)NCC(F)F)C)C)=O)ccc(P(C)(C)=O)cc1 c1(C(N(CC(C)NC(c2c(C)cc(C)[nH]2)=O)C)=O)ccc2nnc(C)c(C)c2c1 N1(C(=O)CCC2CCCO2)CCC2C(NC(C34CCCN3CCC4)=O)CC12 c1(CC)ccc2[nH]c(C(=O)NCCCC3CCCN3C(=O)C(O)CF)c(C)c2c1 C1(C(=O)NC(CC)CN(C(=O)CC2CCC2)C)CCC(=O)N(c2ccccc2)C1 c1(OC(C)C)cc(NC2(c3nnnn3C)CCOCC2F)ccc1N1CCCC1 C(=O)(C#CC1CCCCO1)NCC1(CCNC(CN2CCN(C)C(=O)C2)=O)CC1 N1(C(C(CCSC)O)=O)CC(C2CN(C(C3COC4(CCC4)C3)=O)C2)C1 C1(C)(NC(c2c(CC)n[nH]c2)=O)CCCCC1C(=O)NC12CC=CC(C1)OC2 C1(C2CN(C(=O)C(F)CC(C)C)C2)(NC(c2c(C)nsc2)=O)CC1 C(=O)(C1=CCOC1)NC(CC=C)CNC(=O)CC1CCC(=O)N1 C1(CNC(Cc2cc(C)[nH]n2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C Cn1cnc(C(=O)NCC2CCC2C(=O)NCc2ccsc2)c1 CC(CC(C)(C)C)C(=O)N1CCN(C(=O)C(C)(F)F)CC1CF C1(C(=O)NC2(C(N(OC)C)=O)CC2)CC(N=[N+]=[N-])CN1C(=O)C=Cc1cc[nH]c1 CC1CCN(C(=O)C(CO)NC(N)=O)C(CNc2cc(Cl)ccc2Cl)C1 c1(C(=O)NCC(CC=C)NC(=O)CCc2cnco2)cc2cccc(F)c2s1 O(NC(=O)C1CC(CC(=O)OC)C1)CC(=O)NC(COCC)CO C1(C(N2CC(C)(C)OCC2)=O)Cc2ccc(O)cc2C(=O)O1 C=C(C)CCC(C)NC(=O)CCC1CCC(NC(=O)C(C)N(CC)CC)C1 C=Cn1nccc1C(=O)NC1(C(=O)NC(CC)C(C)(C)C)CCOCC1 CC1(C(=O)NCC2CN(C(=O)CCNC(=O)CO)CC2C(F)(F)F)CC(C#N)C1 C1(C(=O)NCC2(O)CCN(C(=O)CSCc3ccncc3)C2)CC2CC1C1CC21 N1(C(C2C(OCC)C2)=O)CCC(C2CC2)C1CNC(=O)C(F)C(C)C c1(N2C(=O)CC(NC(=O)NC3CC3c3ccccc3F)C2)cc(F)cc(F)c1 C1(COC)CC(O)CN1C(c1cc(CNC(=O)CC2CCOC2C)nn1C)=O CC(CN1CCCC1)CN=C(NCc1ccccc1Cl)N1CCC(C2CC2)C1 N1(C(CC(=C)C)=O)CCC(CNC(=O)Cc2cncnc2O)C12CCC2 c1(NCC)cc(C)nc(C)c1.C(=O)(CCC(=O)NCC1CC(C)N2CC12)NCC Cc1c[nH]c(C(=O)NC2COCC2NC(=O)C(C)CC2CCC2)c1 CCC(CCC(=O)NC(c1nccs1)C)NC(c1ncncc1Cl)=O c1(C(=O)NCC(C2CC2)NC(C(COC)O)=O)cc(NC2CCCC2)ncc1Cl c1(C(C(=O)NC2CC(NC(c3cn(CC)nn3)=O)C2)(C)F)ccccc1F CC1(CNC(=O)Cn2nnc(C3CC3)n2)COCCN(C(C23CCC(C2)C3)=O)C1 CCCCC(F)(F)C(=O)N1CCC(O)(CNC(=O)CS(=O)(=O)N(C)C)CC1 OC1CCc2cc(Br)c(N3CCC4(CCCOC4)C3)nc21 C12(NC(C(C)n3cccn3)=O)COC(CNC(C3(C#N)CC3)=O)(C1)C2 c1(C(N(C2CCC(NC(C3(F)CC=CC3)=O)C2)C)=O)ccc2ccccc2c1O C(C(CNC(=O)Cn1cc(CN(C)C)nn1)C(F)(F)F)NC(CCC=C)=O c1(C(=O)NCC2C(CNC(C3C(OC)CCCC3)=O)C2)cc(C)ncc1Cl C1(C(C)CNC(=O)C=CCO)CCN(C(=O)C(c2ccc(Cl)cc2)(C)O)CC1 C1(NC(CS(CC)(=O)=O)=O)C(C(=O)Nc2nc(SC)cc(C)n2)CCC12CCC2 C1(C)(CC(=O)N(C2CCC2)C(C)C)CCN(C(=O)Cn2ncnn2)C1 CC1CN(C(=O)CCC2CC2)CC1CNC(c1cocn1)=O C1(C2(O)CCN(C)CC2)(C(=O)NC(C2CCCN(C(=O)C=C3CCCC3)C2)C)CC1 c1(COC)nc(C)c(C(=O)NC(CNC(C2CC(Cl)(Cl)C2)=O)C2CC2)s1 c1(CC(=O)N(C2CCN(C(c3nc(C)c(C)s3)=O)C2)CCC)ccnnc1O O=S(=O)(c1cccnc1NC(C1CCCC1)CO)NCCn1cnnn1 c1(C(N2CCC(c3ccc(C#N)s3)C2)C(=O)NC(C)C)cnn(C)c1F C#CCC(C(=O)N1CCCC(N(C(=O)CC(F)(F)F)C)C1)C1CC1 N1(C(C2CN(CCC)C(=O)C2)=O)CC2(CCN(C(=O)CS(N)(=O)=O)C2)C1 CC(C)C(Cc1ccccc1)C(=O)NC1CCN(c2cccc(F)c2Cl)C1 C(=O)(CCC(C)(C)O)N1CCC(NC(CC(C)c2ccccc2)=O)(CF)C1 C1(C)(CC)CCC(C(=O)NC(C)(C)CNC(c2cc(C3CC3)nn2C)=O)O1 O=C(O)C1c2ccccc2CCN1Cc1cnn2c1OCCC2 CC1CN(C(c2c[nH]cc2Br)=O)CCC1NC(C1(F)CCOC1C)=O Cc1coc(C)c1C(=O)NC1CC(CCNC(=O)CCc2cncn2C)C1 C1(C(=O)NC(CCCNC(CCCC#C)=O)CCC)OCC2COCCC12 C1(CNC(c2cnc(CC)[nH]2)=O)CCC(NC(=O)Cc2cnc(C3CC3)[nH]2)CC1 C1(C(=O)NC(C2CCCC2)CNC(C2(O)COC2)=O)CC1C1CCCC1 CC(C(=O)NCCN(C(=O)Cn1nnnc1-c1ccccc1)C1CC1)C(C)(F)F C1(CNC(C=CSC)=O)CCN(C(=O)C(c2ncc(Cl)n2C)(F)F)CC1C C1(C(N(C(CC)CNC(=O)C=CC2CCC2)C)=O)CCC(=O)N1C C1(C(=O)NC(c2cccnc2)CC)CCCC(NC(c2cc(C#N)cs2)=O)C1 N(C1CCc2cc(CNC(C3(C)CCC(=O)C3)=O)ccc21)C(Cc1c(C)nc[nH]1)=O C(=O)(C1Cc2c(Cl)cccc21)NC(C(C)NC(c1cncc(N(C)C)c1)=O)(C)C c1(CN2C(c3cn(C)nc3C(=O)O)CCC2)ccc(Br)c2c1CCC2 Cc1ccc(C(=O)Nc2ccc(O)cc2C)c(-n2cc(CC3CCCC3)nn2)c1 C1(OC(CCSC)=O)CCCC(C)(C)C1=O c1(C(=O)NCCOCCN(C)C(c2cnccc2Cl)=O)n[nH]c2ccc(Cl)cc12 O=C(NN1CCc2ccccc2C1=O)C1CCCCC1.c1(O)ccccc1C=O n1(CC)cnc2c(N3CC(C)C(C)C3)nc(=NCCCCN3CCCCC3)[nH]c12 N1(C(=O)Cc2nc[nH]n2)CCCC1C1CCCN1C(c1coc2c1CCCC2)=O C(Cc1cc[nH]n1)(C(=O)NCC1CCCSC1)NC(C1CC(N(C)C)C1)=O CCC(CN(C)C)CC(=O)NCCN1CCCN(C(c2nocc2C)=O)CC1 CCC(C)C(CC(=O)NCC1CC2(CCCO2)C1)NC(=O)C=C1CCC1 c1(CNC(=O)C(F)=C2CNC2)ccnc(N2CCC(O)CC2)c1 c1(C(=O)NC2CCC(NC(C=NOC)=O)CC2)ccc(Br)cc1F c1(C(N2CCC(C)(O)C(C(=O)OC(C)(C)C)C2)=O)cc2c(=O)[nH]ccn2n1 C(=O)(C(C)CCC(C)(C)C)NC1(CNC(C=CCCC)=O)CCOCC1 C1(NC(Cc2c(C)cco2)=O)CN(C(=O)CN2CCC(N(C)C)CC2)CCC1C N1(C(C(c2ccccc2)OC)=O)CC(F)CC1CN(C)C(c1cc(C)ncn1)=O C1(OC)CN(C(c2cc(Cl)cn2C)=O)CCC1NC(c1sccc1C1CC1)=O c1(C(=O)NC(C(C)NC(c2c(C#C)cnn2C)=O)C)cc(Cl)c([N+](=O)[O-])[nH]1 C(CN=c1[nH]c(C(C)C)ncc1Br)C1CCC(NC(C2(C#C)CC2)=O)C1 N1(C(C)=O)CCC(Cn2cc(-c3cccc(CN)c3)nn2)C(CO)C1 c1(NCC2(O)CN(C(c3ccns3)=O)C2)ncnc2[nH]c3ccccc3c12 N1(C(Cc2nc(C)sc2)=O)CCCC2CN(C(C3(C)CC(C)C3)=O)CCC12 c1(C(=O)NC(C2CCN(C(=O)CC(C)(C)F)CC2)C)nnn(C)c1N c1(C(N(C2CC(NC(CC(=O)NCC)=O)C2)CC)=O)cc2cccnc2cn1 c1(C(=O)NCCC(O)CNC(C2C3CCCC23)=O)cn2ccc(F)cc2n1 c1(C(=O)NCCC(C)N(C)C(C23CSCC2C3)=O)cnn2ccc(Cl)c(F)c12 CC(C)C(CN(C)C)C(=O)N(CCCCNC(=O)CC1(O)CCOC1)C C1(C(=O)NC2CC(NC(C(C)CC3CC3)=O)C(O)C2)CC2(CCCC2)C1 n1(CCCC)nc(C)c(C(=O)NCC2CCCCC2Nc2cc(O)ncn2)c1Cl CCC(COC)C(=O)NC(C)(C(=O)Nc1cn(C)nc1O)C1CCC1 c1(C(=O)NCC2(O)CN(C(=O)CC3CCCCC3)C2)cccn(C2CC2)c1=O C1(C(N2CC(C(C)NC(C(CC(C)C)NC(N)=O)=O)C2)=O)CC2(COC(=O)N2)C1 N1(C(Cc2c(C)scc2)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC2(CC2)C1 C1(c2nnnn2CCC2(C)CC2)(NC(CC)C)CCCC(C(F)(F)F)C1 C1(NC(C2C(OCC)CC2)=O)CC(NC(c2ccc(C(C)C)s2)=O)C(O)C1 N1(C(C(=O)NCC2CCC(C)(C)N2)=O)CC2CCC(C1)C2N C1(CNC(CCSCCC)=O)CN(C(C2(c3cccc(F)c3)CC2)=O)CC12CC2 c1(SC)cc(=NC(=O)C2CC(C)CCN2C(c2cnn(C)c(=O)c2)=O)[nH]n1C c1(C(=O)NC2CN(C(COC)=O)CC(F)C2)cccc2oc(N(C)C)nc12 CCCC(CNC(C1(C)CC(O)CN1C(=O)Cc1nocc1C)=O)CCC C12(CNC(C=CC)=O)CCC1CCN2C(c1ccc(N2CCCCC2=O)cc1)=O c1(CC)occc1C(N1CCC1COC(C)=O)=O.C12CCCC1Cn1cc2nn1 Cc1cc(NC2(CO)CC2)ncc1S(=O)(=O)NCC1(C)CCCCCC1.C1(C)CC1 N1(C(C(C(C)C)CO)=O)CCOC2(C1)CN(C(=O)CC1CCCCC1C)C2 c1(SC)ccc(O)c(C(=O)NC2CC3CN(C(=O)CCc4cn(C)nn4)CC23)c1 Cc1cc(S(=O)(=O)N2CCCC(C(=O)Nc3ccc(O)nc3)C2)c(F)cc1Cl c1(-c2cccc(CC(=O)NCC3CCS(=O)(=O)C3)n2)c[nH]c2ncccc12 N1(C(c2c(C)nnn2C)=O)CCC(NC(=O)C2=C(Cl)CC2)C(CO)CC1 c1(NC(C2N(C(C(C)(C)OC)=O)C3C(C2)C3)=O)ncc(Cl)cc1F c1(NC(=O)NC2(CC3CC3)NC(=O)NC2=O)cnc2ccnn2c1C(F)F c1(-n2ncc(CNC(C3CC4(CNC4)C3)=O)c2)c(Cl)cccc1Cl N1(C(C2N(C(C)=O)CCC2)=O)C2CCC1CC(N(C)C(C1CCS1(=O)=O)=O)C2 c1(OC(C)C(=O)NCC2COCC2NC(=O)Cc2csc(Cl)c2)ccccn1 CC1C2CCC(C2)C1C(=O)NCCC1(C(=O)N(C)CC2(C)CCCC2)CCCC1 CC(C)(CCC#N)C(=O)N1C2CCC1CN(C(=O)CC1CNC(=O)C1)C2 n1(CCOC)c(N2CCCC(C)C2)nnc1C(C)(C)C#N.C(F)F C1(C(N)=O)CCC(C(=O)NCCOCCNC(=O)Cn2nnc(=O)[nH]2)CC1 CC1(C)C(=O)NCC1NC(=O)CC=CCNC(c1ccsn1)=O Cc1nn[nH]c1C1CN(C(C2COCC2NC(=O)CN2CSCC2=O)=O)C1 C#CCC(C)(C(=O)NC1(C(C)C)CC1)NC(C1OC2CCC1C2)=O CCC(C)(C)C(O)C(=O)NCCC1(OC)CN(C(=O)C(c2cccc(C)c2)C)C1 C1(NC(=O)CN(C)C(=O)NCC)CCC(C=O)CC1.C(C)(C)(N(CC)CC)C1CC1 N1(NCCCC2OCCN(C(=O)OC(C)(C)C)C2)CCC=Cc2ccc(Cl)cc21 N1(C(C2CC3CCC2O3)C(=O)NCc2c(OC)cccc2)CCC2(CC1)CC2 C1(C(C(=O)N(C)CC2(OCC)CCC2)C)CCCN(C(c2n[nH]cc2CC)=O)C1 c1(C(N2CC(F)(CNC(c3cnc(C4CC4)nc3)=O)C2)=O)c[nH]nc1[N+](=O)[O-] CC(C)C(C)(C)C(=O)NCC(C)CNC(c1cnn(C)c1F)=O C1(C(=O)NCCCCNC(Cc2n(C)ccn2)=O)CCN2CCC1C2 C1(C2CN(C(c3ncsc3C(C)C)=O)C2)(NC(c2n(CCC)ccc2)=O)CC1 C1(NC(CC(CCC)(C)O)=O)CCCC2CN(c3nc4ccc(C)nc4s3)CC12 C1(CCNC(Cc2c(C)scc2)=O)CCCN(Cc2nnnn2C)C1 C1(NC(c2cnc(OC)nc2)=O)CC(F)(F)CC1NC(=O)CCC(=O)N(C)C N1(C(c2n(C)ccn2)=O)CCCC(NC(=O)C(O)CCCc2ccccc2)CC1 c1(C(=O)NC2(CNC(C(C)C(C)(F)F)=O)CCC2)cc(=O)n(C)cc1Br c1(CC)cc(O)ccc1NC(C12CCC(CC1NC(=O)CCCCCF)C2)=O CC1SCCN(S(=O)(=O)Cc2ccc(C3CC3)cc2)C1C CCCCC(O)CC(=O)N1CCN(C(c2ccnc3[nH]cnc23)=O)CC1CCO c1(CC)nc(C(=O)NC(CO)C(C)NC(=O)C(C)OCC(F)(F)F)cs1 C1(C)(CN(C(=O)CN2CCC(COc3ccc(C)cc3)CC2)C)CCC(O)CC1 c1(C(=O)NC2(CNC(C3CC=CCC3)=O)CCCC2)ncc(Cl)nc1Cl N1(C(c2cnncc2O)=O)CCN(C(=O)Cc2cc(F)ccc2F)C(CF)C1 C1(C(=O)NC2CC(C#C)C2)(CC=C)CCN(C(=O)C=Cc2cnn(C)c2)C1 c1(CNC(C2C(C(=O)OC)CC2)=O)ccc(CC(C)NC(=O)C=CC2CC2)cc1 c1(CC(N2CCCC2CCC2CCNCC2)=O)ccc(Br)s1 C(=O)(CCCC(C)(C)CC)N1C(CC)(CC)CC(NC(=O)CNC(=O)C2CC2)C1 n1(-n2c(C)ncc2)nc(-c2ccc(Cl)cn2)nc1C(C(C)C)C(F)F c1(OC)cc(OC)cc(C(N2CCOC(CCN(C)C)C2)C(=O)NC2CC2)c1 C1(C(=O)NCC#CCC)CCCN(C(=O)C(C)CC#N)C1 C1(C(N(CC(C)(C)C)CC)=O)CCC2(CC2)N1C(=O)C=Cc1ccncc1 N1(C(c2cn(CC)nn2)=O)CC(CNC(=O)C(C2CC2)OC)OC(C)(C)C1 n1(CC(=O)N(CCC(C)NC(CN(C2CC2)CC)=O)C)cc(Cl)c(O)nc1=O CC1(C)Cc2cccc(CC(N3CC4(NC(C5CC(F)C5)=O)CC3C4)=O)c2O1 N1(C(CCC)=O)CCC(c2cccc(F)c2)C(NC(=O)Cc2ccsn2)C1 Cc1nc(C(C)(F)F)ccc1C(=O)NCC1(C)CCCN1C(C1CCCCO1)=O C=CCCCCCCC(=O)N(CC(=O)N(C)Cc1ncco1)C CCCCC(O)CC(=O)NC(C1(O)CN(C(=O)CSc2ccc(C)cc2C)C1)C Cc1cc(C)c(C(N2CCC(N(C(=O)C=CC(=O)N(C)C)CCO)C2)=O)s1 C12C3CN(CC13)C2=O.C1(CC(=O)N(CC(C)(C)C)CC)CC=CCN1C N1(C(C(CCC)F)=O)CCC(C2(CNC(C3CC(O)C3)=O)CCOCC2)CC1 CCCCC(C)CCC(=O)NCC(C1CCCC1)NC(C1CN(C)CC(C)O1)=O CC1CCCN(C(=O)C(=O)NCC2CC2)C1CN1C(=O)CNC1=O C=C(Cl)CCC(=O)N1CC(CC(N2CC(CC)C(O)C2)=O)C(C)C1 N1(C(C(=O)NC(CCC(=O)OC)C)=O)CCC(S(=O)(=O)N(C)C)C1 C1(NC(C(COC)(C)C)=O)CN(C(c2ccnc(C(F)F)c2)=O)CCC1C c1(-c2cn(C3CC(C(N(C)CC4CC5CCC4C5)=O)C3)nn2)ccc2c(c1)CC2 C1(C(=O)NC(c2nc(=O)o[nH]2)CC)CN(C(=O)C(c2ccc(C)o2)C)CC(C)O1 C1(N(C(=O)CCSc2nccn2C)CC)CCCN(C(c2cnc(O)o2)=O)CC1 C1(CCC(=O)NCC2(CN(C)C)CC2)CCCN1C(C1CC(=O)C1)=O O=C1CC(C(=O)NC2(C(=O)NCc3ccccc3)CC2)c2cccnc2N1 C(C)(C)(CC(=O)NC(=O)NC1CC(=O)N(c2cn[nH]c2)C1)N(C)C N1(c2nccc(N3CCC(CC(N)=O)CC3)n2)CC2(CN(CC(F)F)CCO2)C1 C1(N(c2nccc(N3CCCC(c4nnc(C)o4)C3)n2)C)Cc2ccccc2C1 c1(CCN2CCC(C)(CC)C2)cccc(C)c1C n1(CC(=O)NC(CC=C)CNC(C2(CF)CCOCC2)=O)ccc(C)cc1=O C1(C(N2C(CNC(CSc3cccc(C)c3)=O)CC2)=O)CCCNS1(=O)=O c1(C(=O)NC(C)CNC(=O)C(C)C2CCCO2)cn(C2CC2)nc1C(F)(F)F c1(C(=O)NC2CCC(NC(C(CC)C)=O)CC2)cc(Br)cc(Br)c1 C1(CC(=O)N(C)CC2CCCCN2C(c2cnnn2C)=O)CC2(CCC2)CO1 C12(NC(C(CCCC)NC(C3CSCC(=O)N3)=O)=O)CC3CC(CC1C3)C2 C1(C(N2CCCC(CCCO)C2)=O)C(C2CC2)CCN1C(=O)CCc1cncs1 C(=O)(C(S(C)(=O)=O)C1CC1)NCCN(C(c1conc1C(F)(F)F)=O)CC Cc1c(Cl)ccnc1C(=O)NCC(O)CCNC(C1(C(C)C)CNC(=O)C1)=O CCC(CC(=O)N(C1CN(C(=O)CC2COCC2(C)C)CC1(C)C)C)C(C)(C)C C(C(C(=O)NCCc1nccs1)C(C)(C)C)NC(c1scc(C)c1)=O c1(C(=O)NC2C(CNC(c3c[nH]c(=N)o3)=O)CCC2)cc(Cl)ncc1F c1(CC)noc(CCC(=O)NCC2CCN(C(=O)C=Cc3cscn3)C2)n1 N1(C(CCCCCN(C)C)=O)CCC2CC2(NC(c2coc(C(F)F)n2)=O)CC1 Cc1nc2cncc(C(N3CCCN(C(c4nc(O)sc4C)=O)C(C)C3)=O)c2[nH]1 N1(CC(=O)NC(c2ccccc2)C(=O)NCC2(C(=O)OC)CC2)CCOC1=O C1(NC(c2c(CC)c[nH]n2)=O)CC2CC1CN(C(=O)C(O)C(C(C)C)OC)C2 c1(C(N2C(CNC(C3CCCS3(=O)=O)=O)CC2)=O)ccc(CO)c(F)c1 CC1CCN(C(C2CC(F)(F)CCC2(C)C)=O)CCN1C(=O)CCn1ccnc1 N1(C(C)Sc2c(OCCOC)cccc2)C(=O)NC(CO)C1=O CC1CCCC=C1C(=O)NC1(C(=O)NC2CC(C(F)(F)F)C2)CCSC1 c1(CN(C(c2nccnc2C)C(=O)NCCOC)C)ccc2nsnc2c1 C1(O)(CNC(C(C#C)(C)C)=O)CCCN(C(=O)C(CCSC)NC(C)=O)C1 C1(C(=O)NC(C2CCN(C(=O)CCn3cc(Cl)cn3)CC2)C)CCC2(CC1)CC2 c1(C(N2CC(O)(CN(C(=O)C(C3CCCCCC3)O)C)C2)=O)cc2n(c1)CCC2 Cc1nn(C)c(C)c1C(C)C(=O)NC1CCCC1NC(C1(C)CC1)=O c1(C(N2CCN(CC(C)NC(c3c(OC)cco3)=O)CC2)=O)ncc(Cl)cc1Cl C1(NC(CCN(CCC)C)=O)CN(C(=O)C=C2CCSCC2)CC1(C)C c1(C(N2CCC(CN(C(=O)COC(C)(C)C)C)C2)=O)cnnc2ccccc12 n1(CC)cnc2c(N3CC(=O)NC(=O)C3)nc(=NCc3cc(Br)ccc3Cl)[nH]c12 c1(OC)cccnc1C(N1CCC(CCCNC(c2ccncc2)=O)CC1)=O Cc1cnc2ccc(C(=O)NC3CN(C(=O)C4=CCCC4)C4CC34)cn12 CN1CC(NC(C2(CNC(=O)CC3CCC(O)C3)CC2)=O)CC(C)(C)C1 N1(C(c2nn(CC)c(O)c2)=O)CCCN(C(c2sccc2SC(F)F)=O)CC1C C(=O)(C1=CNC2=NCCC2=C1)N(C1CCN(C(C2(C)CCCS2(=O)=O)=O)C1)C N1(C(C(Cc2ccc(C)cc2)C)=O)CCN(C(=O)COc2ccsc2)C(C)C1 c1(OCc2n(C(C)(C)C)ncc2)ccc(Br)cc1OCF.N12CC(C(F)C1)C2=O CCC(C)C(O)C(=O)NCC1(NC(=O)C(C)CCOC)CCCC1 C1(O)(C(C)NC(CC2(CSC)CC2)=O)CN(C(=O)C(N2CCOC2=O)C)C1 c1(C(N2CCC3CCC(C2)N3C(=O)C=C2CCCC2)=O)csc2c(O)ccnc12 C#CC(C)(C)C(=O)NCC(C)(C)CN(C)C(c1conc1-c1ccccc1)=O C(=O)(CC(C)(C)C(=O)OC)NC(C(C1CCCCC1)NC(C=CC(=O)OCC)=O)C c1(C(=O)NCC2CN(C(c3c(COC)cco3)=O)CC2C)cc2ccncc2s1 N1(CC(=O)NC(CC)CN(C(=O)C=C(C)C(F)F)CC)CCCCC1C N1(C(c2ccc[nH]2)=O)C2COCC1C2.C1CCN1CCO.C=O c1(CC)ncc(C(=O)NCC2CCN(C(c3nc(Br)c[nH]3)=O)C2)o1 Cc1ccc(C2(C(=O)NC3(c4csc(S(C)(=O)=O)c4)CCC3)CC2)cc1C#N C(CCN(C)C)(C(=O)NC(c1nc(C)oc1C)C)NC(CCC)=O C#CC1(NC(C2CSCCN2C(=O)C(=O)N(C)C)=O)CC2CCCC12 N1(C(C(C)OCCN(C)C)=O)CCOC2(C1)CN(C(=O)C=CC1CCCO1)C2 N1(C(c2cc(OCC)ns2)=O)CC(NC(C2CC2[N+](=O)[O-])=O)CC(F)C1 C(CC(C)C)(C(=O)NCC(F)CNC(C1(c2c(F)cccc2Cl)CC1)=O)OC c1(OC)noc(C)c1C(=O)NC1CCCC1CC(=O)NOCc1cccnc1 C1(C(N2CCC(Cn3cc(-c4c(C)noc4)nn3)C2)=O)CCCC(=O)C1 C(C(F)(F)C(=O)N(CCCN(C)C(c1ccn(-c2ccccc2Cl)n1)=O)C)OC c1(C(N(CCC)CCNC(C2(C)CCCCO2)=O)=O)cccc(C)c1C c1(C(c2n(CCCNCC(C)OCC)nnn2)CC)ccc(S(N)(=O)=O)cc1Cl C(=O)(CC(CC(=O)O)C1CCC1)NC1C(c2ccn(C(C)C)n2)C1 Cc1cc(C(N2CCC(C(=O)NCCc3ccccc3O)CC2)=O)sc1C O=C(C1=C2CCN=C2NC=C1)NC1CCC1NC(c1ccc2nc[nH]c2c1)=O c1(C(=O)NCC(C)N(C)C(c2cccc(N3CC=CC3)c2)=O)cn(C)[nH]c1=N c1(C(N(C2CN(C(C3CC3CF)=O)C2)CCC)=O)ccccc1N=S(C)(C)=O C(=O)(C(CC(C)C)ONC(c1ccc(O)c(F)c1)=O)N(C(C)C(C)C)CC N(C1c2ccccc2CC1NC(c1cc(O)nc(O)n1)=O)C(C(C)(CO)CO)=O N1(C(CC2=NNC(=O)C2)=O)CCC2(CO)CN(C(c3ccc(CO)o3)=O)CC2C1 C=CCC(F)(F)C(=O)NCCOCCOCCCNC(C1CCCC1(F)F)=O C(=O)(C(C)(C)C(=O)N(C)C)NCC1(CNC(C2(OC(C)=O)CC2)=O)CC1(F)F CC(C)C(CCNC(=O)CC1CC1(Cl)Cl)N=c1[nH]c2ccc(O)cc2s1 N1(C(C2CC(C#C)(O)C2)=O)C2CCC(C2)C1CNC(=O)CC(C)F N1(C(=O)C)Cc2ccccc2C1.C1(NC(C(F)=CCC)=O)CCNC(C2CC2)C1 c1(OCC(=O)NCC2(C(=O)Nc3nn[nH]c3C(F)(F)F)CC2)cccc(F)n1 C(=O)(C(CNC(=O)C(=O)NCC(F)F)C(C)(C)C)N1CC(CC)SCC1 c1(C(N2C(CNC(c3c(O)cccc3Cl)=O)C=CC2)=O)nnc(O)cc1O c1(C(N2CCCC2Cn2cc(CCN3CCCC3)nn2)=O)cc(Cl)sc1Cl c1(N(c2ccc(C)c(F)c2)C)n[nH]c2ccc(C(F)(F)F)cc12 c1(C(N(C)CC2CCN(c3nccc(C)n3)C2)=O)cc(=O)c2cc(F)ccc2o1 N1(C(C(=O)NCC(CC)(N)CC)=O)CC2CCC1CC2 c1(C(CC)C)ccc(C(C(=O)NCCCSC)N(C)CC2(C)CCCC2)cc1 C1(C(=O)NCCS(=O)(=O)NC)CC12CCN(C(=O)C(C)(C1CC1)OC)C2 C(=O)(C1CCCn2nccc21)N(CCNC(c1c(C)nn(C(C)C)c1)=O)C1CC1 CC(C)C(C)C(C)CC(=O)N1CCC(CO)(CNC(=O)C#CC2(C)CC2)CC1 N1(C(C(CCCC)O)=O)CC2CCN(c3cc(C(F)(F)F)nc(C)n3)C2C1 c1(C(=O)NC2CC(NC(C3(OC)CCCC3)=O)C2)cc(Cl)ccc1C(F)(F)F c1(C(=O)NCC2CCN(C(CC)C)CC2)cnc2ccc(Br)cc2c1 Cc1cccnc1CCCNC(c1ccnn1C1CCCC(C)C1)=O c1(C(N2CC3(CCN3C(c3cccnc3)=O)C2)=O)c(F)cc(Cl)cc1F CC(=O)CCCCC(=O)N1CCCC1C(=O)NCC1CCS(=O)(=O)C1 N1(C(C2C(CNC(c3cccc(C(N)=O)c3)=O)OCC2)=O)CC(CO)CC(C)C1 N1(C(c2c(CC)nn[nH]2)=O)CC(NC(=O)Cc2csc(=N)[nH]2)C(CO)C1 C1(OC)CN(C(=O)CCOCC(C)C)CC1NC(c1ccc(N)cn1)=O c1(CC)ccccc1NC(c1cnn(-c2ccccc2F)c1C)c1nnnn1C N12CCC3(CCC(OC3)NC1=O)CC2.Cc1cc(CC2(C3CC34CC4)CC2)no1 c1(C2C(C(=O)NC3CC(c4ccccn4)C3)C2)cnnc2ccccc12 c1(N(C(C(C)c2cccs2)=O)C(c2cc[nH]n2)=O)ccc(F)cc1O.C1C(=O)O1 C(C1c2ccsc2CCN1C(=O)C(C(C)C)OC)NC(CN(CCC)C)=O N1(C(C)(C)C)CCC2(C1)CC2(F)F.c1(C2CCNC(=O)C3N2CC3)ncccn1 CCC(C(=O)NCCCN(C(=O)C(c1ccc(OC)c(F)c1)C)C)C(F)(F)F N1(C(C2CC(C)OC2)=O)CC2(c3nc(-c4c(F)cccc4F)no3)CC1(CO)C2 S(=O)(=O)(c1cc([N+](=O)[O-])c(Cl)cc1Cl)N(C1CCCNC1)C CC(C)[Si](CC(C)(C)C)(CC(=O)NC1CN(S(=O)(=O)C(F)F)C1)OCC(F)(F)F C=CC1(NC(C2(F)CCN(C(=O)C(C)CCOc3ccccc3)C2)=O)CCOCC1 C#CCCC(O)C(=O)NCC(C)(CC)NC(c1c(C)ncnc1C)=O C1(NC(C2(OCC)CCC2)=O)CCCCCC1C(N1CCOCC1CC)=O c1(C(=O)NC2C(CO)CCN(C(c3ccc(CC)o3)=O)C2)cccc2ncnn12 C1(C)(NC(C(C(C)C)c2ccc(F)cc2)=O)CCCN(C(c2nncn2C)=O)C1 CCCC(C(O)C(=O)N=c1ccn(C2CC2)[nH]1)NC(=O)C(CC1CCCC1)C(C)C N1(C(Cc2cc(OC)ncc2)=O)CCN(C(=O)COC2CCCOC2)CC1C CCC(O)(CC)CC.c1(C(N2C(C(NCC)=O)CCC2)=O)occ2c1CCC2 C1(CCC)CN(C(c2conc2C)=O)CC1C(=O)N(CCC(C)(C)C)C c1(CC(=O)NCc2c(C(=O)NC(CCCCC)C)c[nH]n2)cc(C)ccc1O C1(C(=O)NCC2(c3ccccc3)CNC2)(CCl)CN(c2ncns2)C1 C(c1cc[nH]n1)=CC(N1CCC(N(C(C2CC2F)=O)CC2CC2)C1)=O CCC(CC(=O)NC1(CN(C)C(C2CC(n3cnnc3)C2)=O)CC1)C(C)C CCCC(C(=O)N1CCC(N(C)C(c2ccc3c(c2)OCCN3)=O)C1)S(N)(=O)=O c1(C(N2CC(NC(c3ccoc3)=O)C2)=O)nccc2nc[nH]c12 N1(C(COCC)=O)CCC2(CO)CN(C(c3ccc4cccnc4n3)=O)CC2C1 CCC(C)(F)C(=O)NCCC1COCCN1C(=O)CCCOc1ccc(C)cc1 c1(C(C(N2CC(CNC(C3(CC#C)CC3)=O)C(O)C2)=O)O)cccc([N+](=O)[O-])c1 N1(C(C2CN(C)C2)=O)CCCC2(CCC2NC(=O)CS(C)(=O)=O)C1 c1(N2CC(O)(C(C)NC(=O)CC3(C)CCCCC3)C2)ncnn2cccc12 Cc1ccnc(C(=O)NCC2CCCN(C(=O)C(c3cccnc3)C)C2)c1N C1(C(=O)NCCCN(C(=O)C=C2CCOCC2)C2CC2)CCC2C(CC1)C2(F)F C1(C(=O)NCCC2(O)CCN(C(CC(C)=C(C)C)=O)C2)Cc2nccn2C1 C12CCC(CC1)NC(=O)CS2.C1(CC(=O)NN(CCS)C(C)C)(CC)CCC1 c1(CC(=O)NCC(CNC(c2cc(C)c(O)cc2)=O)F)ccc2c(c1)NC(=O)C2 CC(Cl)(Cl)C(=O)NCC1CC(F)(CNC(c2ccc(C(N)=O)[nH]2)=O)C1 C(=O)(C1CC(=O)Nc2ncccc21)NC(CN(C(CC=CC=C)=O)C)(CO)CO Cc1nn(CC(=O)NC(CCNC(=O)C(C)C(C)C)C(C)C)cc1Cl C1(C(N2CC(CNC(C(CSC)O)=O)C2)=O)CCN(C(C)=O)CC1 N1(C(CCCC)(C)C)CCCCC(C(=O)NCCCN2CCCCC2)C1 C(=O)(CC(O)CC(C)(C)C)N1CCC(CC=C)(NC(c2ncccc2Cl)=O)C1 N1(C(C(C)SCC)=O)CCc2sccc2C1CNC(c1cccc(CO)c1)=O c1(N(C)CCNC2CSC2)ncc(S(=O)(=O)N2CCCC(OC(F)F)C2)cc1Cl N1(C(CCCC(=O)OC)=O)CCN(C(c2ccc(F)cc2)=O)C(C)CC1C Cc1cc(C)c(C(=O)NCC23CC(CN2C(=O)CN2CC4CC4C2)C3)[nH]1 c1(C(CNC(N(C(C)Cc2cnsc2)CC)=O)C)ccccc1 C1(N(C(C2C(=C)C2)=O)C)C2CN(C(=O)CSc3nnc(CC)o3)CC12 c1(-c2n(-c3c(C)ccc(F)c3)nc(C(C)C)n2)c[nH]c2cc(F)c(F)cc2c1=O c1(OC)ccc(O)c(C(=O)NC2CCCCCC2NC(=O)Cc2ncc(Cl)s2)c1 c1(NC(=O)NCC(C)(C)CCC2CC2)ccc(Cl)cc1CC(F)(F)F C1(C(N(CCN(C(CCC(CC)C)=O)C)C(C)C)=O)CS(=O)(=O)CC12CC2 C1(F)(CNC(CC(=C=C)C)=O)CC2CCC(C1)N2C(c1ccc(OC)nc1C)=O c1(Nc2snc(OC)c2Br)cc(O)nc2cccnc12 C(=O)(CCCC(C)(C)C#N)NCC1(CNC(CN(S(C)(=O)=O)C)=O)CC12CCC2 C1(NC(C(C)Oc2ccccn2)=O)CCN(C(c2cnc(Cl)s2)=O)CC1(C)C C(C)(CCP(C)(C)=O)(c1nnnn1CC(F)F)NCc1c(OC)cccc1Br N1(C(C(CC(C)C)NC(C)=O)=O)CC(C2CN(C(=O)Cc3ccns3)C2)C1 CCC(C)(C)C(=O)N1CCOC(C(C)NC(=O)CN2CCCC2)C1 C(C)(CCN=c1[nH]ccc(=NCCCSC)[nH]1)c1cccc(OC)c1 C1(C(C)(C)C)C(=O)NCCCC2CCCN2C1=O.c1(SC)cnn(C(C)(C)C)c1 c1(OC)cc2c(cc1F)CCC2NC(=O)C(C)CS(C)(=O)=O.C12(COC1)OC2 c1(OC)c(C(N2CC(N(C(=O)C(c3ccccc3)F)C)C(O)C2)=O)ccnc1Cl N(C1COc2c(F)cccc21)C(=O)NCC1CC(=O)N(C)C1=O c1(C(=O)NCCC2(O)CN(C(C(CCC#C)O)=O)C2)ccc(N)c2ccncc12 C1(NC(=O)NC(CCSC)(C)C)C(C)(C)C1(F)F C1(C(=O)OC)CC12CCN(C(CCC=C(C)C)C(=O)NC1CCCCC1)CC2 c1(SCC2C(C(=O)OC)CCO2)cccc(NC(N2CCN(C)CC2)=O)c1 c1(N(CCOC)C)ncccc1S(=O)(=O)N1CCC(C(C)(C)C)C1 C(CC(C(=O)N1CCC(F)(C(N)=O)C1)NC(=O)CC1NC(=O)NC1=O)OC c1(C(=O)OC)cnc(O)c(C(N2CCCC2(c2ccccc2)C(N)=O)=O)c1 C1(N(C)Cc2c(C)nco2)CCN(C(=O)C(C)CSC(F)(F)F)CC1C c1(NC(C2(C(F)F)CCNC2=O)=O)cn2c(n1)CCC(C(F)(F)F)C2 N1(C(CC(=O)NCC)=O)CC(O)CCC1C(N1CCC(C(C)O)CC1)=O c1(C(N(CCC(C)NC(C2C(C)C2C)=O)C)=O)n[nH]c2ccccc12 C1(CNC(C(C)O)=O)CCC(CNC(c2ccccc2F)C2CCC2)CC1 C1(CNC(Cn2c(CCC)ncc2)=O)CC(NC(=O)Cc2ccco2)C1(C)C Cc1nc(Cl)sc1C(C(=O)NC1CCOC1)N(C1CC1)Cc1ncc[nH]1 N1(C(c2nc(CC)sc2N)=O)CC2(CNC(=O)CCC(C)OC)CCC1CC2 CC1CCCN(C(C2CCCC23CC3)=O)C1CNC(=O)CCC(C)(F)F c1(CNC(c2cnsn2)=O)ccc(CNC(C2CC3CC2C3)=O)cc1 CC1CN(C(c2ccc(SC(F)F)cc2)=O)CCN1C(=O)CC1COCCN1C c1(C(=O)NC2(CF)CCN(C(=O)C3=CCCC3)C2)ccc([N+](=O)[O-])cc1 C12(NC(C3CCCN(CCC)C3)=O)CCCC1N(C(C1CCOC1)=O)CC2 CC(C(O)C(=O)N(CC(C)(C)NC(c1ccc[nH]1)=O)C)c1ccccc1F C12(NC(CN(C(=O)C(O)C(F)(F)F)C)=O)CCC(CC1)C2(C)C Cn1cnn(CC(=O)NCCC2CN(C(c3cccc(Br)c3)=O)C2)c1=O c1(C2(C)N=N2)ccc(S(=O)(=O)NC2CC(C(=O)O)(CC3CC3)C2)cc1 CS(=O)c1ccccc1CC(=O)NC12CC1CN(C(=O)C(=C1CCCCC1)F)C2 CCCC(C)CC(C(=O)NC(C)(C)C)N1CCNC(=O)C1(C)C C(C(=O)NCCN(C(=O)CNC(=O)OC(C)(C)C)C)OCC CC(C)C(F)(F)CC(=O)NCC(C)(C)CNC(c1cc(C(C)(F)F)on1)=O C1(CCN(C)C(C2(C)CCC2)=O)CCN(C(c2cc(C(F)F)cs2)=O)CC1 N1(C(CC2(C#N)CC2)=O)CCCC2(CC(NC(=O)C3=CCOC3)C2)C1 C(=O)(C1Cc2ccccc21)NC(CNC(c1c(C)nc(C(C)C)nc1O)=O)CO N1(C(c2scc(C)c2)=O)CCC2(CCCC2C(=O)NC(c2ccno2)C)C1 c1(OC)cc(C#N)ccc1C(N1CCC2(NC(c3ccc[nH]3)=O)CCCC12)=O N1(C(C2CCN(C(=O)C3COCC(C)O3)O2)=O)Cc2cccc(C#N)c2C1 Cc1ccc(C(N2CCN(C(c3cn(C)ccc3=O)=O)C(CO)C2)=O)cc1Cl N1(C(=O)C=CC2CCCN2C(=O)COc2ccsc2)CC2(CCOCC2)C1 N1(C(C(CC)(C)O)=O)CCC(C2CCN(C(C3CCC=CCCC3)=O)CC2)C1 c1(C(=O)NC2CCC(C)N(C(C3CC3F)=O)C2)cc(C#N)ccc1O N1(C(C(C)n2cccc2)=O)CCC(C)CC1C(N1CCC(CO)C1)=O c1(C(C)C)nn(C)c(Cl)c1C(=O)NCC(O)CNC(C1CCC(=O)O1)=O N1(C(c2cc(C)sc2)=O)CCN(C)CC1CNC(C1(CC2CC2)CCCO1)=O N1(C(C2N(CC)CCOC2)=O)CCCC2CN(c3ccc(C(C)=O)cn3)CC12 c1(C(=O)OCC2C(C)OCC2)cccc(OCCN2CCOCC2)c1 C1(C(=O)NCC2(C(N(CC)Cc3ncc[nH]3)=O)CC2)CCOC1(C)C C(C)(C(C)C(=O)NCC(N)=O)NC(c1cnc(OC)s1)=O c1(NCC(CNC(c2cnc(CC)[nH]2)=O)C)nc(C(C)CC)ccc1C#N c1(C(=O)NCC(C(C)C)NC(C2CCCC2(C)C)=O)cc2cccnc2[nH]1 C(=O)(C(C)CCC(=O)OC)N(C1CCN(C(=O)C(F)(F)CO)CC1)CCOC N(C1c2ccccc2CC1O)C(C1N(C(c2cccc(OC)c2Cl)=O)CCC1)=O c1(C(N(C)Cc2ccc(C(=O)NCC)cc2)C)nc2ccccn2c1F C#CC1(NC(=O)CCCCCNC(C2CC2Cl)=O)CCCOC1 O=S1(=O)c2ccc(cc2Cl)NCCN1.C1(C2C(SCCO)COC2)COCCO1 C1(NC(c2c(C)snn2)=O)CCN(C(=O)Cc2cnns2)C1c1ccccc1 Cc1ccc(C(=O)NCC(N2CCN(C)C(c3nccn3C)C2)=O)cc1F c1(C(=O)NC2C(NC(C(CO)NC(C)=O)=O)CC2)ccc(Cl)c(S(C)(=O)=O)c1 CCC(C(=O)NC1(C)CCCCC1C(=O)NCc1nnn(C)c1C)C(C)(C)CC c1(OC)ncc(Br)cc1NC(C1CSCCN1C(=O)C(C)OC)=O C1(C(=O)NCCCN(C)C(C23CC(F)(C2)C3)=O)CC2OC(C)(C)OC2C1 N1(C(C(CC)N(C)C)=O)CC(CNC(=O)CC2CC3CC3C2)CC1C c1(CC(=O)NC2CN(C(Cc3ccc(C)nc3)=O)C(C)C2)cccc([N+](=O)[O-])c1 C(=O)(C1=C2CCN=C2NC=C1)NC1C(CNC(CSCC(C)C)=O)CCC1 C(c1csc(Br)c1)=CC(=O)OC(C)C(=O)NC1CCCS(=O)(=O)C1 c1(N2CC(O)(C(C)NC(=O)CC3CCCS(=O)(=O)C3)C2)nccc(S(C)(=O)=O)n1 C12(CC)CN(C(=O)CCCN3C(=O)CCC3=O)C(CNC(=O)C(O)C3CC3)(C1)C2 c1(CC)nc(C)sc1C(N1CC2CC2(NC(c2scnc2C)=O)C1)=O N#CC1CCCC(C(N2CC=CC2C(=O)Nc2cccnc2)=O)C1 CS(=O)(=O)CCC(=O)N1CC(F)(CNC(=O)C=Cc2ccco2)C1 CC(CCC(C)(C)C)NC(=O)C(CC1CC1)NC(=O)CC(C)c1ccco1 Cc1cccc2cc(C(N3CC(NC(C4CC(=O)N(C)C4)=O)C(F)C3)=O)[nH]c12 c1(C(=O)NC(C(C)(C)NC(C)=O)C)cc2nc(C)[nH]c2cc1F c1(C(=O)NCC2CCN2C(C2CC(C3CCC3)C2)=O)ccc2c[nH]nc2c1 C=CCCCC(=O)NCC1CC1CNC(C1CCN(Cc2cccnc2)CC1)=O c1(C(CC(=O)NCCC2N(C(Cc3ccc(C)o3)=O)CCC2)C)ccccc1F Cc1ccc(OC2CCN(CC3(CCO)CCC3)C2)cc1.C1C(=O)O1 C1(NC(c2cncc(-n3ccnn3)c2)=O)C=CCN(C(C2CC2[N+](=O)[O-])=O)C1 C1(C(=O)NCc2c(C)nc[nH]2)CCN(C(c2ncccn2)=O)C1C(C)C CCC(C)CCC(=O)N(C)CC1(O)CCCN(C(c2ccc(N(C)C)nc2)=O)C1 N1(C(C(CSC)(C)C)=O)CCC2C(CCN2C(=O)Cn2cc(C)cn2)C1 Cc1nc(N(C)C)sc1C(=O)NC1CC(C)N(C(c2cnn(C(C)(C)C)c2)=O)C1 n1(CCC(=O)N(C(C)CNC(=O)CC2C(C)(C)C2(C)C)C)cnc2ccccc12 N1(C(C2(C=C)CC2)=O)CCC(C(C)NC(c2cn(C)nc2C(C)(C)C)=O)CC1 c1(C(=O)NC(CCCC)CNC(=O)C=CC2CCCN2C)cc2scc(Cl)c2[nH]1 C1(C)(C(=O)OC)CCC1(C)C(=O)NC1CCN(C(c2cnncc2O)=O)CC1 c1(COC)ccccc1C(=O)N(C)CC1(NC(=O)CC2CC(C)(C)C2)CC1 C12(C(=O)NCC3(F)CCN(C(CC4(C)CCOC4)=O)CC3)CCCCC1OCC2 Cc1cc2[nH]c(C(=O)NCC3CC(CNC(=O)CSc4cccnc4)C3)cc2o1 C1(CC)CCCN(C(C2Cc3nccn3C2)=O)C1C(=O)NC1CCCCC1(C)C c1(C(N(CCNC(C(CN(C)C)N(C)C)=O)CC2CC2)=O)cn(C)c(C(F)F)n1 C1(NC(c2ncn(CC)n2)=O)CC2CCC1CN2C(C1CC=CCC1)=O C(=O)(C(O)CCCc1ccccc1)NC1CC(OC)CN(C(=O)CC(C)C)C1 c1(CC)nn(C)c(CC)c1CNC(C1(CS(C)(=O)=O)CC1)=O C1(CNC(c2c(SC)n(C)nc2)=O)CC(F)(F)CN1C(c1csc(O)n1)=O c1(C(C2CCC2)NC(C2CCC2)=O)cc(O)c(O)c([N+](=O)[O-])c1 c12nc3ccccc3cc1-c1cnc(nc1)CN2.C1(N(C)C)CNCCC1C#N c1(SC)ccc(C(=O)N(C)CC2CN(c3ncc(Br)cn3)CCO2)cc1 C1C(F)C(=O)N2CC1C2.C1(CCC=C)CCCCC1.C(C(=O)NC)OCC#C c1(C(=O)NCC(CNC(=O)C(F)(F)C(F)(F)F)CO)cnc2c(c1)C(=O)NC2=O O=C(CCCCc1ccc(Cl)cc1)NC1CC(NC(c2cc(C3CC3)no2)=O)C1 N1(C(=O)OC(C)(C)C)CCC2(CCC(CC(=O)NCCc3ccon3)O2)CC1 C1(C(=O)NC(c2ccccn2)CC)C=CC(NC(c2ccnnc2)=O)C1 CCC(CCO)NC(=O)C(C1CN(C(c2ncn(CC)n2)=O)C1)OC c1(C(=O)NCC2C(C)CN(C(c3c[nH]cc3Br)=O)CC2)nc2cnccc2s1 CCCC(CC(C)C)C(=O)N1CCCC1CNC(C1CC(OC)CN1S(C)(=O)=O)=O c1(NC(C2(COC)CCC2)=O)cccn(CC(=O)OC)c1=O Cc1ccc(C(F)(F)F)cc1C(=O)NCCNC(C1CCCC1C)=O Cc1cccc(C(=O)NC2CCC(NC(=O)C(CO)NC(N)=O)C2)c1Cl CC(C(=O)N1CCCCC(CNC(=O)CN2CCC2)C1)C(C)S(C)(=O)=O CCC(C(=O)NC(C)CCN(C)C(C1(COC)CC1)=O)SC C1(C(N2CCN(C(c3c(C)cnnc3)=O)C(C)CC2)=O)Cc2cccc(C)c2O1 N1(C(c2c(C)n[nH]c2C)=O)CCN(C(C2CC2c2ccc(Br)cc2)=O)CC1C#N C1(NC(C(C=C)(C)C)=O)CCCN(C(=O)C(C2CCCCCCC2)O)CC1 C(=O)(C1CCCc2nncn21)NC(CCN(C(c1c(SC)nn(C)c1)=O)C)C N1(C(C#CC)=O)CCN(Cc2ccc(-c3ccc(N)cc3)cc2)CC1 CC(C)(CC(=O)N1CCCC(CCN=c2nc[nH]s2)C1)C(=O)Nc1ccccc1 N1(C(C2(OCC)CCCC2)=O)CCC(CCc2cn(C(C)CC)nn2)CC1 C1(C(N2C(C)CSCC2)=O)CCN(Cc2cc(O)nc(O)n2)CC1O c1(C(=O)NC2(C3N(C(C(CCC)F)=O)CCCC3)CC2)ccc(C)c(C#N)c1 N1(C(C(C)C2CCC2)=O)CCOCC1CNC(c1cc(C(C)(F)F)n[nH]1)=O N1(C(C(C)(C)OC)=O)CC2CCC(C1)C2CNC(c1cccn1C(C)C)=O C1(CNC(COCCCC)=O)CCN(C(c2cnco2)=O)C12CCC2 C1(O)(CCCC)CCCN(C(=O)CCCOCCNC(C2(Cl)C(C(C)=O)C2)=O)C1 C1(O)(CNC(c2coc(C(F)F)n2)=O)CCN(C(C2CC(O)C2)=O)CC1 C1(C)(C(=O)NC(CC(=O)NC(C)C)C)CCN(C(c2ccnnc2O)=O)C1 Cc1nc2cc(C(=O)NCCC3CC(NC(c4nsnc4O)=O)C3)ccc2s1 N1(C(c2c(C)nn(CCO)c2)=O)CC2CCCC(C1)N(C(=O)Cc1cn[nH]c1)C2 C(=O)(C(Cn1cncn1)NC(c1ccncc1)=O)NC1C(C)C1C C(C(C)(O)CNC(c1cnnn1C1CC1)=O)NC(CCC1CC(OC)C1)=O c1(C(N(C2CCCCN(C(C3CCC(=C)CC3)=O)C2)C)=O)cc2c(s1)COCC2 c1(C(N(CCC(N2CC(CC)(CO)C2)=O)CC#C)=O)cccc(C)n1 c1(CNC(C(C(C)C)O)=O)nn(C)c2c1CN(C(=O)CCC1CC1(F)F)CC2 C(CCCCC(=O)N1CCC(C(F)C(=O)NCCc2ccsc2)C1)=CC C12(C(=O)OC)CCC(C(N3CCC(O)(C(C)NC(c4ccoc4Cl)=O)C3)=O)(C1)C2 C1(NC(c2c(C)snn2)=O)CCN(C(=O)CCCC2CCCCC2)CC1C(C)C c1(NC(c2n(CCC(=O)NCC=C)nnn2)C2CC2(Br)Br)cccc(CCF)c1 c1(N2CCCC(COC(C)C)C2)nc(=NCC(C)(C)CC(C)O)[nH]c2c1CSC2 N1(C2CN(C(C3CC(=C)C3)=O)C2)CC(NC(c2ccncc2SC2CC2)=O)CC1=O N1(C(CN(C)C2CC2)=O)CC2CC1CCN2C(c1ccc(-n2cccn2)cc1)=O N1(C(CCC(=O)NC)=O)CCCC1C1CCCN1C(=O)COCc1nc[nH]n1 C(=O)(CCC1=CCCCC1)N(C1COC(CNC(C2(C)CCCO2)=O)C1)C c1(C(=O)NCC2C(NC(C(C=C)(C)CC)=O)CCC2)cccc2c1CCN2 C1(NC(c2cncc(C)n2)=O)CCCCN(C(=O)CCC(=O)c2cnn(C)c2)C1 N1(C(Cc2c(OC)cccc2)=O)CC2CCC1CN2c1ncnc(Cl)c1CO C1(NC(C(CNC(C2(COC)C=CCC2)=O)(C)C)=O)CC=C(C(C)C)CC1 c1(CC(=O)NCC(CNC(Cn2c(C)csc2=O)=O)C)cnn2c1CCCC2 c1(NC(C2C(CC)CCCN2C(C2CCCC(=O)N2)=O)=O)cn(C)c(=O)nc1O C1(C(N2CC(C=C)(O)C2)=O)CC2CCC(C1)N2C(=O)CC1CCC(=O)C1 C#CC1(C(=O)NCCC2CCN(C)C2)CCN(C(=O)CCc2nc[nH]n2)CC1 c1(C(NC(N(CC(CC)C)CC)=S)C)ccc(F)cn1 C1(NC(=O)NCC2CCC(C)C2)CC12CC(C)(C)C2 c1(C(N(CC(C)NC(c2c(C)ccc(C)c2)=O)C)=O)cncc(N=[N+]=[N-])c1 C1(C(=O)NC)CCN(C(=O)NC2CC2(C)C(N2CC(OC)C2)=O)C1(C)C C(=O)(CC(C)CC(C)C)N1C(C)(CCC(=O)NCCC=C)CCC1 C1(CC)CN(C(=O)CC2CCC3(CC3)CO2)CCC1NC(c1csc(C)c1)=O C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NCC(CNC(CCSC)=O)O c1(CC)ccc(O)c(C(N2CCC(CNC(=O)Cc3cncn3C)C2(C)C)=O)c1 C1(CNC(c2cn(C(C)C)nc2)=O)CN(C(=O)CO)CCC1(C)C c1(C(=O)NC2CN(C(c3ccc(C(CC)C)cc3)=O)C2)ccc(Cl)c(N)c1 C(=O)(CCCC(C)(C)C)NC1C(CO)CCN(C(c2occ(C)c2C)=O)C1 C(c1cc2ccccc2o1)=CC(N1C2CN(Cc3nccc(OC)c3)C(C2)C1)=O Cc1cccn2cc(C(N3CCC(NC(=O)CCSCC(C)C)C(O)C3)=O)cc12 C1(NC(C2(SC)CN(C(=O)Cc3ccc[nH]3)C2)=O)CCC(N=[N+]=[N-])CC1 CC(CS(C)(=O)=O)C(=O)NCCC(O)CNC(C1(S(N)(=O)=O)CC1)=O C1(NC(C(CC)OC)=O)CN(C(=O)CCc2cn(C)nn2)CC2(CCC2)C1 c1(OC)ccc(C(C)(C)C(=O)Nc2ccc(CN(CCCCCC)C)o2)cc1 CC(C)CC(C(=O)NC(C(=O)N(C1(CO)CC1)C)C(C)C)C(N)=O CCC(CC)C(F)C(=O)NC1CN(C(=O)Cc2ccc(F)c(F)c2)C(C)(C)C1 N1(C(C(C2CC2)NC(c2cc(OC)ncn2)=O)=O)CCCCC(C)(F)C1 CCCCC(=O)C(=O)N1CC2CC(N(C(=O)C(C)C(F)(F)F)C)C1C2 CONS(=O)(=O)c1ccc(C(=O)NC2CC2CNC(C2(CO)CC=CC2)=O)cc1 C(=O)(CCC(=O)NCC1CCCC(NC(=O)C(F)(F)c2nc(C)cs2)C1)NC N1(C(CCC(C)O)=O)CCCC2(CCN(C(c3cnc4occc4c3)=O)C2)C1 C1(C(=O)NC2CN(C(C3CCC(C)O3)=O)C(C)(C)C2)CCc2n[nH]cc2C1 c1(C(N2CCOCC2CNC(c2sc(Br)nc2Br)=O)=O)cc(O)c(Br)c(O)c1 c1(CNC(C(C)(C)OCC)=O)cc[nH]c1C(=O)NC(CN(C)C)CO N1(C(C(CC)SC)=O)CCN(C2CN(C(c3csnc3C)=O)C2)CC1 N1(C(C2(CCC)CCC2)=O)CCC2(CC1)CC2C(=O)NCCc1noc(C)n1 N1(C(C(C(=O)OCC)OC)=O)CC=C(C(=O)NC(C)(CO)C2CCC2)C1 CC1(C)CCCCC1C(N1CCCC1CCCNC(C1(C)CC1(F)F)=O)=O c1(CC(=O)NCC2CN(C(c3cnccc3Cl)=O)CCO2)ccc(I)cc1 c12cc(ccc1N)OC2.C(CNCCSCC#N)NC C1(C(C)C)CN(C(=O)C=Cc2cscn2)CCN1C(=O)Cc1cc(O)nc(O)n1 Cc1nsc(N(CC(=O)NC2CCC2)C(C2CCC(O)CC2)C2CC2)c1C#N N1(C(c2ccc(C(C)C)o2)=O)C2CCC1C(CNC(=O)CCc1n[nH]c(=N)s1)C2 N1(C(N)=O)CCC(C(N2CCC(CCNC(c3cccs3)=O)C2)=O)CC1 C1(NC(c2coc(C3CCCC3)n2)=O)CN(C(=O)Cn2cccn2)C2(CCC2)C1 N1(C(CCN(C(CC2C(C)(C)OCC2)=O)CC2CC2)=O)CC2CSCC2C1 c12csc(n1)CC2.C(CCOCCOC)N1CCOCCNCC1.N(C)C.OC c1(C(=O)OC)cc(CC(=O)NC2CN(C(N)=O)C2)cc(Cl)c1.C12CC(C1)CC(=O)N2 c1(C(N2C(C(=O)Nc3ccc(Br)cc3I)COCC2)=O)cc(Cl)c(Cl)nc1Cl CCC(C)C(O)C(=O)N1CCCCC1C(=O)N(C)Cc1nc(C)cs1 CC1CN(C(C2CN(C(c3cccc(OC(F)F)c3)=O)CCC2O)=O)CCN1C c1(C(=O)NCC2N(C(C(COCC)C)=O)CCC2)ccc(COC)cc1 Cc1nc2ncc(C(=O)NCC3COCC3NC(C3(C)CCCO3)=O)cc2o1 C(=O)(CCC(=O)c1ccccn1)NC(CC)CN(C(=O)C(C)C)C C1(CC)CCCC1C(=O)N(CCN(C(=O)CN1CC2(CC2)C1)C)C(C)C c12cc3ccccc3cc1S(=O)(=O)N2.C(=O)(C(=O)N(CC(C)N)C)OC CCC(C)CCCCC(=O)NC(CNC(=O)CCc1nnc(C)n1C)C(C)(C)C c1(NC(CNC(C2(OC)CCCOC2)=O)C2CCC2)nc(C(C)C)cc(C)n1 c1(OC)cc(C)c(C(N2CCN(C(=O)CC3CC4CC4C3)C(CO)C2)=O)cc1Cl c1(NC)cc(Cl)ccc1C(=O)NCCOC1CCN(C(=O)C#CC(C)(C)C)C1 N1(C(CC(CC)C)=O)CCN(C(c2ccc3nc[nH]c3c2)=O)CC12CCC2 c1(C(=O)NCC2CN(C(CCCOCC=C)=O)CC2O)cn2cccc(F)c2n1 C1(C(=O)NCC(F)CNC(C2(C=C)CCC2)=O)CC(O)CN1C(=O)OC(C)(C)C c1(C(=O)NC2CN(CC(C(C(=O)OC)F)C)CC2(C)C)c[nH]c2nccc-2c1 C#CCC(C)C(=O)N1CCOC(CN(C)C(c2cnn(CCN(C)C)c2)=O)C1 c1(C(N2CCC3CCC(C2)N3C(=O)C(O)C2CCC2)=O)cn2cccc(Cl)c2n1 N1(CC(CN2CCN(CC)CC2)C)CC(=O)N(CC(C)C2CC2)C1=O C1(C(=O)NCCOC2CCN(C(=O)Cc3ccno3)C2)CCC2(CC2)C1 C1(F)(NC(=O)CCCc2nc(-c3ccccc3)no2)CCCCCC1 C#CCCCC(C)C(=O)c1cccc2c(scc1)N1CCCC1CN(CC)C2=O C1(C(=O)NC(COC)(C)CO)CCCN(C(=O)CCc2ccn(C)c2)C1 c1(C(=O)NC(C2CCCCN2C(=O)C2=C(Cl)CC2)C)ccc(C(C)(F)F)cc1 c1(OCC(=O)NCC2C=CC(NC(c3c(CC)onc3)=O)C2)cccc(Br)c1 c1(C(=O)NCC2CC(C)(C)CN(C(C3CC3C#N)=O)C2)c(Cl)ccc2c[nH]nc12 C1(CC(N2CCC(CCOC)C2)=O)CCCCN1C(=O)CCC(=O)C1CC1 C(=O)(C1=CCC(F)(F)CC1)N(C1CCCC(N(C)C(c2cc(=O)n(C)o2)=O)C1)C N1(C(c2cnc(OCC)nc2)=O)CCC(NC(c2cnc(F)cc2C)=O)C(C)C1 C12(CNC(C3C(CCC)CCC3)=O)CC1CN(C(C1COCCN1C(C)=O)=O)C2 C1(NC(C2C(=C)C2)=O)COC2(CCN(C(c3cnc(Cl)cc3OC)=O)CC2)C1 C=CCCCCCC(=O)N1CCC(C(N2CCC3OCCC3C2)=O)(C(C)C)C1 C(=O)(C1CCc2ccc(C)cc21)NCC(C1CCCC1)NC(C1C(OC)C1)=O N1(C(c2cccc(SC)c2)=O)CC2(C1)CN(C(=O)CCc1ccco1)CCO2 C(=O)(CS(=O)(=O)CCO)NCC(CNC(CN(C(C)=O)C)=O)O Cc1cc(C(=O)NCC(C2CC2)NC(C2CCCN2N=O)=O)c(N)cc1F Cc1cc(F)cnc1C(=O)NC(C(=O)NCc1cnc(O)nc1O)C1CCCC1 C(=O)(CCC(C)CCCC)N1CC(C)CC(C(=O)NC(C#C)(C)C2CCCC2)C1 c1(C(N2CC(O)(CN(C(C3C(OCC)C3)=O)C)C2)=O)n[nH]c(C)c1C(F)(F)F c1(C(CNC(=NC)NCc2nc(N(C)CC)on2)(F)F)ccc(Cl)cc1 C1(C(N(CCCNC(=O)COCC(F)F)C)=O)CC12CCC1(CC1)CC2 C1(NC(c2cc(OC)no2)=O)C2CCC(C2)C1C(=O)NC1CCCCCCC1 N1(C(CSCCC)=O)CCCC(O)(CN(C(=O)C(n2cnc(C#N)n2)C)C)C1 c1(C(C)=O)cc(=NCC(O)CNC(=O)Cn2ccc(O)nc2=O)[nH]cn1 C1(CNC(CCSCC)=O)C(C)CCN1C(=O)CC1OCCCO1 c1(C(=O)NC(C)(F)F)ccc(-n2cc(C(C)(C)CC(=O)NC3(O)CC3)nn2)cc1 c1(CN(C(=O)NC(c2cccnc2)COC)CCO)ccc(Br)cc1Cl C1(C(N2C(C)CC(NC(C3(C)CC(=O)C3)=O)C2)=O)C2C3CCC(C3)C12 c1(CC(N2C(c3cn(CC)nc3)C(C)CCC2)=O)cccc2c1OCCC2 c1(C(=O)NCCCCC(=O)N(CCCO)CC#C)ccnc2cc[nH]c12 C1(CNC(C2CC23CC(NC(C2(CO)CCOC2)=O)C3)=O)CCS(=O)(=O)C1 c1(C(N2C(C)CCCC2)c2nnnn2C(C)(C)C)cc(Cl)c(Cl)c(Cl)c1.C1CN1 c1(SCC)ccc(CC(N2CC(CCNC(c3nocc3Cl)=O)C(C)C2)=O)cc1 C12(C(=O)NC(C(C)C)CNC(=O)CCc3nccs3)CCN(C1)S(=O)(=O)C2 C(=O)(C1=NOC2COCC12)NC1CN(C(C=C(CC)CC)=O)CC(C)C1 C(CCCCC(=O)N(C1CCC(CNC(C2CCSC2)=O)CC1)C)SC c12cn(C)nc1OC1CCN(C1)C2=O.C=C1CN(C(=O)NC)C1.OC c1(CC)nc(C(N2CCCCC2CCNC(=O)C(O)CCSC)=O)c(C)o1 c1(C(=O)OC)ccc(OC)c(OC)c1CNC(=O)NCCC1CCOCC1 N1(C(COCCC#C)=O)CCC(C2CCCN2C(C2CCOC2(C)C)=O)CC1 CC1CCCC(CC(=O)N(c2ccccc2F)CCCNCCN2CCCC2)C1 C(=O)(C1=CC2(CN(C(=O)CNC(=O)CCCCC)C2)OC1)N(CCCC#C)CC S(=O)(=O)(c1ccc([N+](=O)[O-])cc1)NCC(C)(C)C(=O)N1CCCC1CCC#N.SC S(=O)(=O)(c1cnc(NCCCNS(C)(=O)=O)c(Cl)c1)NCC(C)(C)C(F)(F)F C1(NC(c2c(C)nc(C3CC3)o2)=O)CCCC12CN(C(=O)CC1CCNC1=O)C2 c1(C(N)=O)ccc(NC(=O)COC(=O)CC23CCC2CCN3)cc1 N1(C(c2cc(C)[nH]c2C)=O)CC2CCC(C1)N2Cc1cc(O)ccc1F C1(CNC(C(C)=C2CC2)=O)CC2(CCC2)CN1C(=O)CC1(C(F)F)CC1 C(C(CC(C)C)C(=O)NC1CN(C(c2ccc(C#N)cc2F)=O)CCC1F)OC C(N=c1nc(Cl)[nH]c(C)c1C#N)C1CCN(C(CC(C(F)(F)F)NC(C)=O)=O)C1 CC(C(=O)NCc1c(C(N2CCCC(O)C2)=O)n[nH]c1)C(F)F C1(CC(=O)NC(C)(C)CCNC(=O)Cc2ccsc2)CC2CCC1C2 N1(C(c2ccc3sncc3c2)=O)CCCC1C1CCCN1C(c1ccsn1)=O C1(N(C(c2cncc(OC)n2)=O)C)CCN(C(c2c(C)noc2N)=O)CC1C C(=O)(C1=CCCCO1)NC1(C)CCN(C(C(Cc2c(C)cccc2)C)=O)C1 c1(OC)ccc2c(c1)CC(C(=O)NC1CCC(N(C(=O)C3=CCCC3)C)CC1)O2 C(CC(C)(C)C)(C(=O)N1CCCC1C1(C(=O)NCC2OCCC2(C)C)CC1)OC C(CC(C)(C)C(=O)N1CCC(CNC(c2ccc(O)cc2C)=O)C(C)C1)OC c1(C(=O)NCCCCNC(C2CC3CCC3C2)=O)ccc2nc(C(F)F)[nH]c2c1 N1(C(Cn2c(C)ccn2)=O)CC(C(=O)N(C)C)CC(C)C1 N1(C(CNC(C=C)=O)=O)CC(C2CCN(C(c3ccc(OC)c(C)c3)=O)CC2)C1 c1(C2(O)CC(C(N3CC(N(C(C4N(CC)CC4)=O)C)C3)=O)C2)ccc(F)cc1 C1(C#CC(=O)NCC2CCC2NC(C2(CC3CC3)CCOCC2)=O)(CC)COC1 C1(NC(COC(C)C)=O)CC(CNC(=O)C(C)C2(O)CCC2)C1 c1(C(N2C3CC(CC(NC(CC(CCC)C)=O)C3)C2)=O)ccc2oc(=N)[nH]c2c1 S(=O)(=O)(c1ccccc1F)NCCC(=O)NC12CC(CNC(C(C)C#N)=O)(C1)C2 C(=O)(C#CC1CC(F)(F)C1)NC1CCN(C(c2c(F)ccc(C)c2)=O)CC1 C1(CNC(CC)=O)CC2(CCN(C(c3ncc(-c4ccccc4)nc3O)=O)C2)C1 N1(C(C(COC)C)=O)CCC(CC(=O)Nc2cccc(F)c2F)C1(C)C C1(C(N2CC(OC)(CNC(c3cc(C(C)C)no3)=O)C2)=O)CCCC12CC2 CCC(CNC(=O)C=CCNC(C12CCC(CC1)C2)=O)C(C)C CN1CCN(c2nc(C3CC3)ns2)CC1CNc1cn[nH]c1 c1(OC)ccc(Br)c(C(=O)Cc2nc(C3CC3)cs2)c1 c1(C(N(C(C)C)Cc2onc(CCC(C)C)n2)=O)nc(Cl)cc(N)c1Cl C12(CNC(c3n(CC#C)ccc3)=O)CCC1CN(C(=O)C(C)(O)CCC)C2 CCCC(C)CCCC(=O)OCC(=O)N(C1CCOCC1)C(C)C N#CC1(CC(N2CC3C(C(N4CC5C(C4)C5(F)F)=O)C3C2)=O)CCCOC1 N(C(=NCc1ccnn1C)N1CCC(N2CCCCC2)C1)CC(CC)C(C)(F)F CC1CN(C(C2CC2c2ccccc2F)=O)CCN1C(C1CCC(=O)N1)=O N1(C(C(CC(C)C)(F)F)=O)CCC2(CCC2CNC(=O)C2=CCCC2)CC1 N1(C(C=CCC)=O)CCC2CN(C(=O)C(C3CCCCC3)CC)C2C1 c1(C(N2C3CCC2CC(N2CCCC2)C3)C(=O)NC)cc2c(s1)CCOC2 N1(C(CCC2CC(NC(c3c(C)cccc3)=O)C2)=O)CC2CN(C)CC2(C)C1 c1(C(=O)NC2(C)CC(NC(c3c(CC)ocn3)=O)C2)ccncc1N N1(C(COCC(=O)OC)=O)CCCCCC1CNC(C1CC(C)(F)C1)=O CCC1=C(C(=O)NCC2COCCN(C(C3CCCC(O)C3)=O)C2)CCCO1 c1(N(C(C2CN(C(C3(Cl)C(C(C)=O)C3)=O)C2)=O)Cc2ccccc2)cnnc(O)c1 N1(C(c2c(C)nsc2)=O)CC(N(C)C(c2cnsn2)=O)C(F)C1 CCC(O)C(C)(C)C(=O)N(C)CC1CN(C(=O)Cn2ccc(C)n2)CCO1 C1(C(=O)NCC(CN(C)C)(C)O)CC(=O)CN1C(c1ccc(CN(C)C)o1)=O N1(C(C2(C)CCN(C)CC2)=O)CC2CCC(CNC(C3(C(C)(F)F)CC3)=O)(C2)C1 N1(C(C(CCSC)NS(CC)(=O)=O)=O)CCCN(CC(=O)OC)CC1C(C)C C#CCC(O)C(=O)N(C1CCN(C(=O)CN(S(C)(=O)=O)C)CC1)CC C1(C(=O)NCC=CCNC(c2c(C)nn[nH]2)=O)CC2(CCCCC2)C1 C1(C(CNC(Cn2cc(CC(OCC)OC)nn2)=O)=O)CS(=O)(=O)CC1O C(=O)(C(CO)NC(C1(NC(=O)CC2(OC)CCC2)CC1(C)C)=O)OC C1(N(C(C2(O)CC(NC(c3c(COC)ccs3)=O)C2)=O)C)CCC(O)CC1 Cc1cccc(CNC(C2OCCC2CNC(C2CCC(N(C)C)C2)=O)=O)c1F C(=O)(C1SCc2cccnc21)N1C(C)CCN(C(=O)COCCN(C)C)CC1 c1(C(=O)NC(CC)(CNC(=O)C#CC2CC2)CC)ccc(CO)cc1F Cc1cc(C(N2CCN(C(=O)CC3(O)CCCOC3)C(C)C2)=O)cn(C)c1=O N1(C(c2c(C)scn2)=O)CC(O)CC1C(=O)NCC(C)O C=CC(CC)CC(=O)N1CCC1CC(=O)NCCCN(CC(C)C)C Cc1nc(C2CC2)sc1C(=O)NCCC(C(C)C)NC(=O)Cn1cnc(C#N)n1 N1(C(C2C(C(C)(C)C)C2)=O)CCC(C(CO)NC(C2CCS2(=O)=O)=O)CC1 c1(C(N2CCC(N(C(C3CC3c3cncn3C)=O)CC)C2)=O)cc(C)ccc1O N1(C(C(C)(C)C)=O)CCN(C2CCN(C(C3CC34CCOC4)=O)CC2)C(=O)C1 c1(CN2CC3CN(C(CS(C)(=O)=O)=O)CC3C2)cncc2ccccc12 c1(CC(=O)NCC(C)N(C)C(c2ccc(C(C)(C)C)o2)=O)ncsc1Cl C1(NC(CC(C)SC)=O)CC=CCC1C(=O)NCCCOC1CCCC1 c1(C(N2CCCC(N(C(C(n3c(C)ncc3)C)=O)C)C2)=O)cccc2c[nH]nc12 c1(C(=O)NCC2C(NC(C3(C)CCNC(=O)C3)=O)CCC2)cc(N)c(F)c(F)c1Cl C1(NC(CC2N(C)CCC2)=O)CCCCCC1C(N1CC(C#N)C1)=O Cc1c(NC(c2ccc(OC(F)(F)F)cc2Cl)=O)cccc1-n1cnnc1 c1(C(=O)NC2CCN(C(C(CC=C)C(C)C)=O)C2C)cccc2c1CC(C)(C)C2 C#Cc1ccc(OC(F)F)c(OCC(=O)NC23CC(NC(C4CC=CC4)=O)(C2)C3)c1 N#CC1(CNC(=O)C(CN(C)C)NC(=O)C(F)C(F)(F)F)CCCCC1 CC1(C)CN(C(=O)Cc2ccc(Cl)s2)CC(CNC(c2cc(O)ncn2)=O)O1 c1(OC)c(C(=O)NC2CC(O)CN(C(C3CCS(=O)(=O)C3)=O)C2)cccc1Cl C(=O)(C(C)CC(=O)NCC1(F)CCN(C(c2cc(F)ccc2C(C)C)=O)C1)OC C1(C(=O)NC(c2cn(CC3C=CCC3=O)nn2)(C)C)COCCC1(F)F N1(C(C=C(C)C(C)C)=O)CC(NC(=O)C=CC(F)F)CC12CCCOC2 C(CC(=O)N1CCC(NC(=O)C(n2cc(Cl)cn2)C)CC1)(C(N)=O)NC(C)=O Cc1nc2ccccc2cc1C(=O)NC1(C)CN(c2nc(C(F)F)nc(=N)[nH]2)C1 CC1CN(C(c2ncoc2-c2ccc(F)c(F)c2)=O)CCN1C(=O)CC1CC1C C1(CC)CC(C(=O)NC2CC(CCC(N3CCOCC3C(F)F)=O)C2)CCO1 CCCCC(F)C(=O)N1CCC(C)CC1C(N1CCOCC(O)C1)=O c1(CCC(=O)NCC(=O)NCC2(C)CCC2)cnc2n1CCNC2 Nc1ccc2c(c1)N(C(=O)CCC1CC1CC1CC1)CCCC2 c1(CC)nnc(C)cc1C(N1CCC2(NC(=O)CCc3ccncn3)CC2C1)=O N1(C(C(CO)N(C)C)=O)CCN(C(C2CCC(C)(C)CO2)=O)CC1CO Cc1cccc(COCC(=O)NC(C)(CNC(=O)CSC2CC2)C2CC2)c1 C(=O)(CC(C)(F)F)NCC1C(NC(CC(=C)Br)=O)C1 Cc1cc(C(=O)NC(CC(=O)N(CC(C)CO)C)C2CC2)ns1 N1(C(C2(COC)CCCO2)=O)CC2(C1)CN(C)C2.C12CCC1C(=O)NC2 c1(CSCC(=O)NC(C2CCN(C(c3ccncc3)=O)CC2)C)ccccc1Cl CC1CN(C(C2(CC3CCC3)CC2)=O)CC1CCNC(=O)CCc1cccs1 C1(CC)COCC1N=c1[nH]c(=NCC2CCN(C)CC2)[nH]c2ncn(C(C)C)c12 N1(C(C(C2CCCN(C(c3cnsc3)=O)C2)C)=O)CCN(C)CC(O)C1 c1(N)ccc(OC(C)CN(C(=O)C(=O)NC2CCC(CC)CC2)C)c(Cl)c1.OC N1(C(C(C)=C2CC2)=O)CCC(C(F)(F)F)CC1CNC(=O)C=Cc1ncc[nH]1 c1(OC)cccc2c1C(C(=O)NCC1(NC(=O)C3=CCCS3)CCOC1)CC2 n1(CC)nncc1S(=O)(=O)N1CC(CO)C(c2cncn2C)C1 C1(NC(C(CC#C)O)=O)CN(C(C2CCc3nc[nH]c3C2)=O)CC12CCCC2 Cc1cc(C(N2CCOCC2CNC(=O)Cn2ncccc2=O)=O)cc(O)c1 C1(NC(C2CCC(C)O2)=O)CN(C(=O)Cc2cnccn2)CC2(CC2)C1 C1(C#N)(C(N(CC(N2CCN(C(c3cc(C)oc3)=O)CC2)=O)C)=O)CCSCC1 c1(C(C)C)cccc(CC(=O)NCC(C)CNC(=O)C(C)n2ccnn2)c1 CC(C)C(C(=O)NCCCN(C(=O)Cc1ccc(-n2ccnc2)cc1)C)N(C)C S(=O)(=O)(CCC(=O)N1CCCC(C)(CNC(C2CCC(=O)C2)=O)C1)N(C)C c1(OCC=C)ccc(CC(=O)N(CC(C)N(C(=O)C=CC2CCC2)C)C)cc1 CCCCC(C(=O)NCCC1=CCN(C(=O)C2=CCC(C)CC2)CC1)C(C)C N1(CC(=O)NCC2CCC(NC(C(C)(C)c3cnsc3)=O)C2)CCCCCC1=O CC1(CNC(=O)C(CC2CCCO2)NC(=O)CN2CCCCC2)CC2(CC2)C1 C1(NC(CCNS(C)(=O)=O)=O)CC2CCC(C1)N2C(c1nocc1Br)=O c1(C(=O)NCC2(CNC(C3C(OC)CCCC3)=O)CC2)cnn2ccsc12 C(=O)(CCS(N)(=O)=O)NC1CCC(CNC(CCSCC)=O)CC1 C1(CNC(CC(C)(O)c2ccccc2)=O)CC2CN(C(C3CC(F)C3)=O)CC12 N1(C(c2cc(CC)nn2C)C(=O)NCC)CCc2ccc(N(C)C)cc2C1 C(=O)(CC(C)(C)c1ccccc1)N(C1CN(C(=O)Cn2cc(Cl)cn2)CC1F)C c1(C(=O)NC2(C)CCN(C(=O)CN3CSCC3=O)C2)cnc2nccnc2c1 c1(C(N2C(C)CC(CNC(C3(C4CCC4)CC3)=O)C2)=O)cc(Cl)cc(Cl)c1N C(=O)(C1=CC(C)(CC(=O)OC)C1)NC(C1CCCCC1)CNC(CCC#C)=O C12(C(=O)NC3CC(C)(NC(C(C)=CC4CC4)=O)C3)CCCC(C)(C1)OC2 N(C(=NCCF)NC1CC1c1ccccc1Br)C(c1ncn(C)n1)C C(=O)(C1=C(C)OCCS1)N1CCCC(NC(c2c(OC)ncnc2C)=O)CC1 Cn1ncc2cc(C(N3CCC(NC(c4ccoc4Cl)=O)C(F)C3)=O)ccc12 N1(C(COCCC=C)=O)CC(CNC(c2ccc(Cl)nc2OCC)=O)CC1(C)C CCCC(O)C(=O)N1CC(CC(=O)NC2CCCN2C=O)(OC)C1 C12(COC)CCN(C1)C2=O.c1(CN(C(CC)C(=O)NC)CC)ccc(OC)nc1 N(C(=NCCCc1ccc(Cl)s1)NC1CCCC1)CC1N(C)CCOC1 Cc1ccc2c(c1)CC(C(N1CCN(c3cc(C(C)C)ncn3)CC(O)C1)=O)S2 c1(C(=O)NC2C(C)CN(C(=O)CC3CC=CC3)CC2)cnc2c(=O)[nH]ccc2c1 Cc1nccc(C(=O)N(CC(C)CNC(C2(CC(F)F)CCC2)=O)C)n1 C(=O)(C(C)(C)C(=O)OC)NCC1CCN(C(C2C(C(C)C)(CC)C2)=O)C1 C1(NC(=O)NCc2nnc(COc3ccc(F)cc3)s2)CC2CNCC12 c1(CC(N2C(C)CC(NC(C3(C(N)=O)CC3)=O)C2)=O)cc2ccccc2oc1=O C1(NC(C2(C(=O)NC)CC2)=O)CCC(O)CN(C(c2c(C(C)C)cnn2C)=O)C1 C1(c2nnnn2C2(C)CC2)(NCC(C(OCC)OCC)O)CC2(CCCC2)C1 c1(CC)ccc(C(=O)NC2(CO)CCCN(C(C3CC4(C3)CC4F)=O)C2)c(O)c1 Cn1cc2c(C(=O)NC3CN(C(c4cncc5ccsc45)=O)C3)cccc2n1 N(C(=NCC(C)C)NCC1(c2ccccc2C)CC1)C1CC(OC)C1 N1(C(CC(C=C)c2ccccc2)=O)CCC(C)CC1CNC(C1(C)COC1)=O C12(CNC(c3c(CC)ncs3)=O)CC(CNC(=O)C(C)OCOC)(CO1)C2 c1(CC(N2CCN(C(C3CC(C)C3)=O)CC2CC(F)F)=O)ccc2nonc2c1 C(=O)(C(C)C(C)S(C)(=O)=O)NC1CN(C(c2cccc(OCC(=O)OC)c2)=O)C1 c1(C(N(S(=O)(=O)C2CCCCC2)C2(CN)COC2)=O)ccc2ccncc2c1 c1(OCC)ccccc1C(=O)NCCC(C)NC(C1(CF)CC1(F)F)=O N1(CCN(C(=O)CC=CCNC(C2CC2C2CCCO2)=O)C)CCCCC1 C12(C(=O)NCC=CCNC(C(C(C)O)N(C)C)=O)CCC(CO)(CC1)CC2 C1(NC(COC(C)C)=O)CC2CCC1C(NC(=O)CS(C)(=O)=O)C2 Cc1ccc(C(C(=O)NCC2CCC=CO2)N(CC(F)(F)F)Cc2ccco2)nc1 C1(C(N(CC(C)NC(C2(COC)CCC2)=O)C)=O)CCCCC1(C)C c1(C(=O)OC(C)=O)cc(NC(C2CC2CN)C2CCC2)ccc1F C=CCC(C(=O)NCC1CN(C(=O)CCCCC2CC2)CC1OCC)C(C)C N1(C(CCOCCCOC)=O)CCC(C2CC2)C1CNC(=O)Cc1nnc(C)o1 CN1CCCC(F)(C(=O)NCCN(C)C(c2ccccc2Cn2cccn2)=O)C1 C1(CNC(=O)C=CC2CCOCC2)CCCN(C(c2cc(O)no2)=O)CC1 N1(C(CCC)=O)CCC2(CC1)CC2NC(C1CC12CCCC2)=O C(=O)(CC(C)(C)C(C)(F)F)NC(CC(C)NC(CN(C(COC)=O)C)=O)C C1(C(=O)NCCCN(C(=O)Cc2cncc(C#N)c2)C(C)C)CC2CCC1CC2 N1(C(c2ccc(C#N)o2)=O)CC2C=CC1C(C(=O)NCc1cccnc1O)C2 CN1CCC(=CC(=O)N(CCNC(C2(C)CC2F)=O)CC2CC2)C1 c1(CC)cc(C)ccc1NC(=O)C(C)N(C(C1CC=C(C)CC1)=O)C1CC1 C1(C(=O)NC(CNC(c2cncc(C)n2)=O)(C)C2CC2)CCn2cc(C)nc2C1 C1(NC(=O)C2=COCC2)CCCCCN(C(c2cc(C(F)F)ccc2F)=O)C1 C1(C2CCN(C(c3nnn(C)c3N)=O)CC2)(NC(c2cnc(C)o2)=O)CC1 c1(Nc2c(C)scc2)nccc(=NC2CC2c2ccccc2C#N)[nH]1 C1(C(N2CC(=C(CNC(c3c(Cl)nsc3Cl)=O)F)C2)=O)Cc2ccncc2C1 C(=O)(CCCC(=O)Nc1cccc(CNC(c2cc(Cl)ncc2C)=O)c1)OCC c1(C(=O)NCC2(C(=O)Nc3n(CCOC)ncc3)CC2)ccc(Cl)c(O)c1 c1(SC(C)C(=O)NC(c2ccccn2)c2ncc[nH]2)ccc(F)cc1 C1(NC(C(CCC#C)O)=O)CCC2(CC1)CN(C(=O)COCC1CCCOC1)C2 c1(OCC(=O)NCC2(F)CCN(C(=O)CC3CCCCO3)C2)ccccc1F C(CC(C(=O)NCC1(CO)CCOC1)NC(c1cc(C)sc1C)=O)=CC c1(C(=O)NC2CCC(CC(=O)N(C)Cc3ncn(C)n3)C2)cccn2ccnc12 C1(C(=O)NC2CCN(C(C3C(=O)NCC3)=O)CC2)CC2CC1CC2O CCC(CC)CC(=O)NCCc1n[nH]cc1C(=O)NC(C1(CO)CC1)C C(=O)(CCCCCC(C)C)N1CC(O)(C(C)NC(C(CC)OCC)=O)C1 Cc1nnc2n1CC(C(N1CC(CNC(=O)CC(C)(C)O)CCC1C)=O)CC2 c1(CN(C(C#C)C)CC(=O)OC)ccc(C(c2ccoc2)=O)cc1 Cn1cc([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)C(O)C(F)F)CCC1CO CN1C(=O)c2ccccc2C1CC(=O)N1CC=CC1CNC(=O)COC(F)F N1(C(C(C)SCC)=O)CC2(C1)SCCC2NC(=O)Cc1cccc(Cl)c1F c1(CC)occ(C(F)(F)F)c1C(=O)NCC(C)(C)NC(c1nn(C)cc1Cl)=O c1(C(=O)NCCN(C(c2ccc(NC)cn2)=O)C2CC2)cc2ccccc2cn1 c1(OC)ncc(-c2ccc(CNC(c3cc(C)cc(C)n3)=O)cn2)cc1C CC(C)C(C)CC(=O)NCC1CN(C(=O)CC2CC(C)OC2C)CCCO1 CC1(CNC(N2CCC(O)(c3c(F)cccc3Cl)CC2)=O)Cc2ccccc21 C1(N(C(=O)CC2(C)CC2)C)CN(C(c2ccnc(O)c2F)=O)CC1(C)C CC(C)(C)C(CCO)NC(=O)COC1CC(NC(C2CC(=C3CCC3)C2)=O)C1 N1(C(CCCOCC=C)=O)CCC(F)(CNC(c2coc(SC)c2)=O)C1 CC1(C)C=C(C(=O)NCCCCC2CCCC2)C1.C12(CCC1)CC(=O)N2 N1(C(CC2N(CC)C(=O)CC2)=O)CC(C)N(C(c2ncn(C(C)C)n2)=O)CC1C C(=O)(C(O)Cc1[nH]cnc1C)N(CC(CC)NC(C(C)=CC)=O)C C(CC(C)(C)C(=O)NOC1CC1)NC(=O)OC(C)(C)C c1(C(=O)NCC2CN(C(C3C(=C)C3)=O)C(C)C2)ccc2c(c1)CC(C)O2 C1(C(C(=O)NC2(C)CC2)N(CC(F)F)CC)CCC2CC1C2(C)C c1(N(C2CCCN(C(C3CCC(F)C3)=O)C2)C)ncnn2c(Br)ccc12 CC(C)CCCCC(=O)NCC1CC(CNC(=O)C=CC2CCOCC2)CO1 c1(CN2CCCC(NS(CCC)(=O)=O)CC2)cccc(S(C)(=O)=O)c1 CC(CC(=O)NCCC1(O)CCN(C(=O)CSCCN(C)C)CC1)C(C)(C)C CCCCC(CC)C(=O)N(CC(C)(C)NC(=O)Cc1cc(C)cs1)C CC1CCC(SCC(N2CCCC2C(=O)N(C(C)(C)C(F)(F)F)C(C)C)=O)CC1 C1(C(=O)NCc2c(C)ccnc2)CCN(C(C23CSCC2C3)=O)CC1C N1(C(c2n(COC)ncc2)=O)CC(NC(c2cccc(C#N)c2)=O)C(C2CC2)C1 c1(OC2CC2)ccc(C(N(CCO)CC)=O)cc1OC.C12CC1CNC2=O c1(OC)ccc(S(=O)(=O)NC(C)C(=O)NCCCCC(C)(F)F)cc1 C(=O)(C1CCc2c[nH]nc21)NC1CN(C(C23CCC(C)(OC2)C3)=O)CC1C1CC1 c1(N2CC(NC(c3csc4ccccc34)=O)C(F)C2)ncnc2[nH]ccc12 C1(CNC(C=NOC)=O)CN(C(c2cc(C3CC3)n(C)n2)=O)CCN1C CN1CCOC(=O)C1CNc1cc(CO)ccc1F c1(C(N(CCNC(=O)Cc2ccccc2O)CC)=O)cc(Cl)c2ccncc2n1 C1(OC)CCC2(C(=O)NC3CC(C)N(C(=O)Cc4nncn4C(C)C)C3)CC12 Cc1cn2cc(C(=O)NCC3CCCN(C(c4ccc(C)s4)=O)C3)ccc2n1 N1(C(c2cc(CC)n(C)n2)=O)CC(C(=O)NCCN2CCC2)CC(C)C1 N1(C(Cc2ccn(C)n2)=O)CCC(COC2CN(C(C3CC3(F)Cl)=O)C2)CC1 N1(C(CC(C(C)C)OCC)=O)CCC2(CC(NC(=O)CC3(O)CCOCC3)C2)C1 C#CC1CN(C(=O)CC(CN(C)C)CC)CCN1C(=O)C=Cc1cnc[nH]1 C12(NC(Cc3nnc(C)o3)=O)CCC(C1)N(C(=O)CSCC(F)(F)F)C2 C1(NC(=O)C=Cc2ccccc2)CC2CN(C(c3cnc(O)s3)=O)CC2C1 c1(C(=O)NCC2(NC(C(C)NC=O)=O)CC2)cc2c(Cl)cncc2s1 c1(C(=O)N(C2C(C(=O)NC3CN(C(C)=O)C3)C2)CCO)[nH]c2ccc(F)cc2c1Cl c1(NCCOC2CN(C(CN(C)C(C3CCCO3)=O)=O)C2)ccnnc1 C1(CNC(CC(c2cccs2)NC(N)=O)=O)CCCCCN1C(c1cncnc1)=O C(C(O)C(F)(F)F)NC(C(=O)N(C)C(c1n(C(C)C)cnc1)c1ccccc1)=O CCCCCCCCCC(C)CC(=O)NC1CCC1NC(c1cc(Cl)c[nH]1)=O CC1=CC(C)CN(C(=O)C(=O)NC2CC(C)(C)CN2Cc2ccccc2)C1 C(=O)(C1=CCCCC1)N1C(C(=O)NC2CC(C)SCC2)CSCC1 CC(C)CCC(=O)NCC(C1CCN(C(C2(C)CCC2)=O)CC1)(C)O c1(C(N2CCCC(CCNC(CP(C)(C)=O)=O)CC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 N1(C(C)=O)CCC(C)(C(N2CCC2CNC(=O)CCn2ccnc2)=O)CC1 CCCCCCC(C)(CC)C(=O)NC(C)C(C)NC(c1cc(C)ccc1F)=O C1(CC=C)CCC(NC(=O)CC2(NC(=O)C(c3ccco3)OC)CCC2)C1 Cc1nnc2cc(NC3CCN(C(=O)C(N4C(=O)CCC4=O)C)CC3C)ncn12 C1(C(C(=O)NCCN(C(=O)COc2cncc(Cl)n2)CCC)F)CCCCCC1 N1(CCCN(CCCC)C)CCC(=O)N(CC(c2cccs2)OCC)C1=O C=C1CCN(C(c2ocnc2CC)=O)C1C(=O)NCCCNC(=O)NC Cc1cccc(C(=O)NC(C)CCN(C(=O)CC2CCCN2C)C)c1[N+](=O)[O-] c1(N(C)C)cccc(C(=O)NC2CCCC2NC(=O)CNC(=O)C(C)(C)C)n1 N1(C(COCC#C)=O)CCCCC1CC(=O)NOCc1ccnc(C)c1 C1(C(=O)Nc2cccc(CC(=O)OC)c2)CCN(C(=O)COCC(C)C)C1(C)C C1(C(=O)NCC(C)C2CCC2)(SC)CN(C(=O)Cc2nc[nH]n2)C1 C1(CC(=O)NC(CN(C)C)CCO)CC2(CC2)CN1C(C1CCOCC1(C)C)=O c1(C(=O)NCC(CC)(C)NC(=O)CCCC(=O)NCC)cc(Cl)c(OC)c(Cl)c1 c1(C(=O)Nc2ncccc2OCC(F)(F)F)ccccc1[N+](=O)[O-] c12ccc3c(c1)CC(=O)N3CC(=O)Oc1cccc-2c1.CCCOC(=O)OCC n1(CCCC(=O)NCCC(C)NC(c2cc(SC)oc2)=O)c(O)nnc1O C1(C(=O)NCC2(NC(c3nccnc3C(=O)O)=O)C(C)C2)CC2(CC2)CN1C C(=O)(C1=NN2CCCN=C2N1)NCC(CN(C)C(c1cnc2nccn2c1)=O)O C1(C(=O)NCCN(C(=O)C(c2ccnn2C)O)C)CCCN(S(N)(=O)=O)C1 C1(F)(C(=O)NC2CC3(CN(C(c4cc(C)c(C)s4)=O)C3)C2)CC12CCCCC2 c1(C(C=CC)O)nc(Cc2cnn(C)c2)nn1-c1ccnc(Br)c1 N1(C(c2onc(C)c2C)=O)CCCN(C(=O)C(C)Cn2ccnc2)CC1C c1(C(=O)NC(C2CN(C(=O)C(C)(C)n3cccn3)C2)C)ccnnc1Cl C1(CNC(c2csc(Cl)c2)=O)(NC(C2CCC3CCC23)=O)CCCCC1 c1(C(C(N2CCCC(CCNC(CC(=C)Br)=O)C2)=O)=O)c(C)nn(C)c1C N12CCOC(C1)CC2.c1(-n2cc(C3C(=C)C3)nn2)ccccc1Cl.C1(C)C(C)C(=O)N1 S(=O)(=O)(C1CC(c2ccccc2)C1)NC(Cc1cc(C)nn1C1CCC1)C C1(CNC(c2ccc(C(C)=O)o2)=O)CC(NC(c2ncoc2C)=O)C1(C)C c1(C(=O)NCCN(C(C2N(C(CCC)=O)CCC2)=O)C2CC2)cnc(O)c(F)c1 C1(CC(=O)NC(C2(O)CCC2)C)CCCN(C(c2cocc2C(N)=O)=O)CC1 n1(C(C=CC(=O)NCC2CCC(NC(=O)OCC)O2)C)cc(C(F)(F)F)cn1 N1(C(C2(CC(C)C)COC2)=O)CC(NC(=O)CN2CCC(C)CC2)C(C)C1 C(=O)(CCC1=CCc2ccccc21)N(C)CC1(CNC(CN(C(C)=O)C)=O)CC1 c1(OC)nc(NC2(CNC(c3c(F)ccc(Br)c3Cl)=O)COC2)ncc1C#N C12(NC(C(CC(C)(C)C)O)=O)CCCC1N(C(C1CC3(C1)CC3F)=O)CCC2 c1(C(=O)NCCCN(C(=O)CCCN(C)C)CC)cccc2oc(C)nc12 C1(CC(N2CC3CC(C2)N(C(c2ccc(CO)o2)=O)C3)=O)CCn2cncc2C1 C1(C)(C(N(CC(CN(C(CSCC#C)=O)C)O)C)=O)CCC(C)CC1 CC(C)C(C(=O)NCC1(NC(=O)C(C)SCC2CC2)CCCCC1)n1cnnc1 Cc1scc(C(N2CCOC(CCCNC(=O)C=C3CCN(C)C3)C2)=O)c1N c1(C(=O)NCC(CNC(c2cc(C)nn2C)=O)(C)O)ccc2cc[nH]c2c1 CCC(C)C(CC(=O)NCC1CCOC1)NC(C1(C)CNC(=O)N1)=O C1(C(=O)NC2CCCCN(C(c3c(C)noc3N)=O)C2)CCCCC1C1CC1 C1(CNC(C2C(C(C)(C)C)C(=O)C2)=O)CC(OC)CN1C(=O)C(F)C1CCCC1 N1(C(CCC2C(C)C2)=O)CCC2(NC(c3coc(C4CCCC4)n3)=O)CC2C1 C=CCCC(C(=O)NC(c1ncn(C)n1)C)NC(c1sc(F)cc1C)=O C(=O)(CCC(=O)NN(C)C)NCCNC(c1c(C)cc(N)cc1)=O CCC(CC(=O)NCC1(O)CCN(C(=O)CCCCN(C)C(C)C)C1)C1CCC1 C1(NC(C(C)O)=O)CCC(C)N(C(c2ccc(Cl)cc2F)=O)C1 C1(NC(C2CSCCS2)=O)C2CN(C(=O)C(F)CC3CCCCC3)CC12 Cn1c(C(=O)NC2CCCC2NC(C2(c3cccs3)CCCC2)=O)nnc1S c1(C(N2CC3(CC(NC(C4CN(C)C4)=O)C3)C2)=O)ccc(Cl)c2ccccc12 c1(C(N2CCC(Cn3cc(C(C4CCCO4)(C)C)nn3)C2)=O)cccc(N)c1Br N1(C(C2(OC)CCCN(C(C(CC(=O)OCC)C)=O)C2)=O)CCC2CC1C(=O)O2 c1(C(=O)NC2(CNC(C3C(C4(C)COC4)C3)=O)CC2)cc(Cl)c(F)cc1O c1(N(C)CC2CCN(C(c3ccc(C)cc3Cl)=O)CC2)ncnc2c1cnn2C c1(NC(N2C(C)CC(C3CCCCC3)C2)=O)ccccc1S(=O)(=O)N1CCCC1 c1(CC(=O)NCCCn2cc(CC=C)nn2)cccnc1C(=O)OC c1(C(=O)NC(CCCC)CNC(C2CC(C)(C)O2)=O)nnc(O)nc1O CCCC(O)CC(=O)N1CCC(CCOC)(NC(c2ccno2)=O)C1 C1(NC(C(C=C)(C)C)=O)CC2(C1)CC(CNC(=O)C(C(C)(C)C)C1CCC1)C2 C1(CNC(C(c2ccco2)NC(CSCC=C)=O)=O)CC2(CCCO2)C1 c1(OC)ccc(C=CC(=O)NCC(C(C)(C)C)NC(=O)C(C)N2CCC2)cc1 C(C(CNC(C1(NC(=O)CCSC)CC(O)C1)=O)C(C)C)OC C(=O)(C(O)CCSC)N1CCC(C(=O)NC(COC)(C)C2CC2)C1 CN1CCN(C(=O)C(C)(C)CC#N)C(CNC(C2CCOC2)=O)C1 C=CC(C)(O)C(=O)N1CCC(C)(NC(=O)Cc2ccnnc2O)C1 CCS(=O)CC(=O)NCCCCC1CN(CC(=O)NC2CC(C)(C)C2)C1 c1(C(N2C(CC(=O)NC(c3c(C)nns3)C)CC2)=O)cc[nH]c2nccc1-2 C1(N(C(c2cc(C(C)=O)[nH]n2)=O)C)CCN(C(c2ccnc(N(C)C)n2)=O)CC1 c1(N2CCC(CNC(c3n(C)ncn3)=O)CC2)ccn2ncc(I)c2n1 C1(CNC(CCCOCCOC)=O)CC(F)CN1C(c1oc(CO)nc1C)=O N1(CCC(=O)NC2CCC3CC3C2)Cc2ccccc2C1=O Cc1ccc(C(=O)NC2CCN(Cc3ncccc3C)C2)c2ccccc12 C(=O)(C(O)C(F)(F)F)N1C(C)(C(=O)NCCCOC)CCC1 N1(C(C=COCC)=O)CCCC(C(=O)Nc2cc(F)ccn2)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)C=Cc2cncs2)c2c(nn1C)CCSC2 N1(C(c2cn(C)c(=O)cc2)=O)CC2(CC(NC(C3(C)COCCO3)=O)CO2)C1 Cc1noc(C)c1C(=O)NC1CN(C(c2cc(-c3ccccc3)cs2)=O)CC1F N1(C(CCC2C(C)(C)C2)=O)CC=C(C(=O)N(CCF)C2CC2)C1 N1(C(C(C(C)C)(C)O)=O)CCCC(C2CCN(C(c3ncnn3C)=O)CC2)C1 C(=O)(N=c1ncn(CCC(=O)N2CCCC2)[nH]1)SC1(C)CC=CCO1 N1(C(C(CCN(C)C)O)=O)CCC2CCCC12C(=O)NCC1CCCOC1(C)C C1(O)(CNC(CC2(C=C)CC2)=O)CCN(C(=O)CC#N)C1 C1(C)(C(=O)NCC(CN(C)C(C2CCSC2)=O)O)CCSCC1 C1(CC(=O)NCC(F)CNC(=O)C(C)N(C)C)(COC)CCOCC1 C(=O)(C1CN(C)C(=O)c2ccccc21)N1CC(C=C)C(NC(=O)CNC(C)=O)C1 N1(C(COC(CC)=O)=O)CCCN(C(=O)Cc2cc(OC)ccc2F)CC1CO N1(C(C(C)O)=O)CC2(C1)CN(C(=O)C=Cc1ccc(Br)s1)CC2CO c1(CC2(CO)CCOC2)ccc(CNCC2CNCCO2)cc1 CCC(CC(=O)N1CCN(C(c2cc(C)nn2CC)=O)CC1C1CC1)C(C)C CC(C)(C)C(C)(C)C(=O)N1CC(NC(=O)Cc2ccc(F)c(Cl)c2)C(O)C1 C1(C(CNC(C2(OC)CCSC2)=O)(C)O)CCN(C(=O)CCC(=O)N(C)C)CC1 N1(C(CCCC#CC)=O)CC(C)(C)OCC1CNC(=O)CCc1ccc(C(=O)O)[nH]1 C1(CCNC(C2N(C)CCC2)=O)CCCCN1C(C1CCCC(C(F)(F)F)C1)=O c1(CC)cc(C(=O)N(CCNC(c2nocc2C)=O)C(C)C)cc(F)c1 C#Cc1cccc(C(N2CC(NC(C3CCCCO3)=O)C(N=[N+]=[N-])C2)=O)c1F c1(NC(C2(C(=O)OC)CC2C(C)C)=O)cccn1C(C)COC1CCCC1 c1(CC)cc(C(N2CCCC(CN(C3CCCC3)C)C2)=O)cc(O)n1 c1(NC(C(CC2CN(C(C3CC(OC)C3)=O)C2)F)=O)cnn2c1CCCC2 C1(NCc2cn(C(CC)CC)nc2C)CCC2CNCC12 Cc1oc(C)c(C(=O)N(C2CCN(C(C3CC(C4CCC4)C3)=O)CC2)C)c1C c1(NC(CC2CCN(C(c3cc(C)oc3C)=O)CC2)=O)ccc(C(C)C)cc1F c1(CCC)ccc(CC(=O)N(C(C)CCNC(c2nnc(S)n2C)=O)C)cc1 C(=O)(C(C)S(C)(=O)=O)N(CC(C)NC(=O)CC1CC(C)OC1C)C Cc1nc(C(=O)NC2CC(c3ccccc3)(NC(C3(C)CCCC3)=O)C2)sc1C C1(CCNC(CC(=C=C)C)=O)CCN(C(c2nn(C)c(N)c2C)=O)C(C)C1 c1(CCC(=O)NCC(CC=C)NC(=O)Cc2cncc(C)c2)cc(F)cc(F)c1 CON(CCC(=O)N(C1CCC1(C)C)C)C(=O)C1Cc2ccccc21 c1(COCC(N2CC(CC(C)NC(=O)C(O)CN(C)C)C2)=O)cccc(Cl)c1 N1(C(C=Cc2cc(C)no2)=O)CCC(CNC(=O)C(C)n2cncn2)C1(C)C N1(CC)CC(C(=O)NC(C(N2CCOCC2CCO)=O)C2CC2)CC1=O Cc1ccccc1CNC(=O)COc1cccc(CCN2CCCC2)c1 CC(C)C(C(C)NC(c1cc(Cl)sc1Cl)=O)NC(c1cc[nH]n1)=O C(CC(=O)NCC(CNC(=O)COCP(C)(C)=O)CO)(C(F)(F)F)OCC C1(C(=O)NCCC)CCN(C(C2CCCN2C(C)C)=O)C1 C1(CC(=O)NC(c2ncnn2C)C)CCCN1C(=O)CCc1cnoc1 CC(C#N)CCC(=O)NC(C)(C)CNC(c1ccc(N2CCCC2)cc1)=O Cc1[nH]nc(C(=O)NC(C2CCCN2C(=O)CC(C)C2CC2)C)c1Br C1(NC(CC(COC)C)=O)CC2CC(NC(=O)CCc3ccccc3C)CC2C1 C=CC(C)(C)CC(=O)N(CC(C)(C)CNC(=O)CC1COC(C)(C)CO1)CC C(=O)(C(C)(C)NC(=O)CC1CCCO1)N(CC=C)CCO c1(OC)cc(NCC2CCCC(NC(=O)C3CC3)C2)nc(C(F)(F)F)n1 CC(C)C(C#N)C(=O)N1CCCC(CO)(CNC(=O)C(C)NC=O)C1 C1(F)(CNC(C(=O)NC(c2nc(C)[nH]n2)C)=O)CCCOC1 CC1CCCCCN1C(c1cc(Br)cs1)C(=O)NCC(F)F N1(C(COCCC(C)C)=O)C(C(N2CC(C)(F)C2)=O)CC1C c1(C(N2CCC(NC(=O)Cn3nccn3)C(F)C2)=O)cc([N+](=O)[O-])ccc1Cl C1(C(NOCCC=C)=O)CCCCCCN1C(c1[nH]ccc1CC)=O c1(C(=O)NC(C(c2ccccc2)NC(C2(COC)CC2)=O)C)sc(CO)nc1C N1(C(c2c(C)c[nH]c2)=O)CCOC(C(=O)NCC(O)CCC2CC2)C1 CCC(CC)(CC)C(=O)N1CCN(C(=O)C(c2ccnn2C)O)CC(C)C1 C1(OC)CCC(C(N2CC(CNC(=O)C(=O)NCC(F)(F)F)C2)=O)C1 N1(C(C2C(=C)CC2)=O)CCC(C(C)NC(C2OCC2(C)C)=O)C1 c1(CNC(C(C2CC(=C)C2)N2CCC2C2CCOCC2)=O)ccc(Br)s1 CC1CCC=C1C(=O)N1CCN(C)C(C(=O)Nc2cnccc2C2CC2)C1 Cc1cnc(C(=O)NCC2CC(NC(C3CC34CCC4)=O)C(O)C2)nc1 c1(C(=O)NCC2C(NC(c3scnc3Cl)=O)CC2)cnc2n1CCOC2 Cc1ncnc(C)c1CC(=O)NCC1CCN(C(=O)CC(=O)Nc2nccs2)C1 N1(C(C2C(C)CCCC2)=O)CCC2(CC1)CC(NC(=O)CN1CCN(C)CC1)C2 c1(CNc2c(C(=O)Nc3c(OC)ccc(F)c3)scc2)c(Cl)cc(O)cc1Cl Cc1cc(C(N2CCC(F)(c3cn(CCN(C)C)nn3)C2)=O)c(C)cn1 c1(NC(CO)Cc2cscn2)cccc(CC(F)(F)F)c1 C(CCCCC(=O)N1CC(F)CC1CNC(c1cnc(C2OCCO2)s1)=O)SC c1(C(N(C2CCCN(C(c3cccc(Cl)n3)=O)C2)C)=O)ccc(O)nc1 C1(C(=O)NC2CN(C(CCC(=O)NC)=O)CC2C)CCc2nnnn2CC1 CC1(NC(c2cnc(-c3ccco3)s2)=O)CCN(C(=O)CNC=O)CC1 CC12CCC(C(N3C4CCC3CN(C(C35CC3CCC5(F)F)=O)C4)=O)(CC1)CO2 c1(N2CCC(C=C)(CO)CC2)nc(=NCCCCS(C)=O)[nH]c2cc(C)ccc12 C=C(C)CC(C(=O)N1CC(C(=O)N(C2CC3CC3C2)C)CC(C)C1)OC c1(NCC2N(C(=O)C=CCN3CCCCC3)CCC2)ncnc2scnc12 N1(C(CC(=C)C)=O)CCN(C)CC1CNC(c1ccc(OC)cc1F)=O c1(C(N2CC(CN(C(c3nc(C)[nH]n3)=O)C)OCC2)=O)ccc(Cl)c(F)c1N S(=O)(=O)(c1ccc(N(C)CC2CC2(F)F)cc1Cl)N1CC(C)C(O)C(C)C1 N1(Cc2cnc(C)s2)C2CCCC1CC(NC(c1cc(Br)cc(Br)c1)=O)C2 c1(CCC(=O)OCC)ncc(C(N2CCCC2C2(C)CC2)=O)s1 C1(CC(N2CCC(CCOC)(NC(C3CCC3C)=O)C2)=O)OCCCC1(C)C c1(C(=O)NCCC2N(C(C3N(C)C(=O)NC3)=O)CCCC2)c(O)ccc(Cl)c1F Cc1cc(CO)ccc1NC(C1CC(C)N1C(c1ccc(N)c(F)n1)=O)=O C(CN=C(NCC1CCCC(C2CC2)O1)N1CCC(O)C1)OC(C)(C)C C1(C(=O)NCCOC2CCN(C(c3cnccn3)=O)C2)CCCCCS1(=O)=O n1(C(C)C)c(O)nc(N2CCCC(NCC34CCCC(CO3)C4)C2)cc1=O C1(NC(CCCCCn2cc(C(C)(C)OC(=N)O)nn2)=O)CN2CCCN1CC2 C(=O)(CCCCC(N)=O)N1CCCC(CNC(C(c2ccccc2F)C)=O)CC1 C(=O)(C(F)CCC(C)C)NCC1(CC(N2CCC(C)(CCC)C2)=O)CC1 c1(C(c2n(C(CC)C)nnn2)NCCC(CO)CO)cc(C(C)C)nn1C c1(C(=O)NC(CN(C(C2C(CC)CCCC2)=O)C)C)cc2cc(OC)cnc2[nH]1 c1(C(=O)NCCN(C(C2(C(=O)OC)CC2)=O)C2CC2)ccnc2c1CCC2 CC1CN(C(=O)Cc2ccc(Cl)cc2)CCCN1C(=O)C1=CC(O)CCC1 C1(C(=O)NCCC(=O)Nc2ccc(F)cc2Br)CC2CCCCN2C1 C1(NC(c2cnc(C(C)=O)s2)=O)CCCC(NC(C2CCCC2)=O)CC1 C1(O)(C(C2CCCCC2)NC(=O)NCC(C2CCOCC2)(C)C)CCCNC1 N1(C(CC=C)=O)CCC(N(C(=O)CCn2cccn2)CCO)CC1 c1(CC)ncc(C(=O)NC2COCCN(c3cnnc(C)n3)C2)c(C(F)F)n1 N1(C(C)C)CCC(C(N2CCCC(NCC3CCC(F)(F)C3)C2)=O)CC1 N1(C(CN(S(CC)(=O)=O)C)=O)C2CCCC1CN(C(c1ncccc1CO)=O)C2 C1(C(c2ccc(Cl)cc2)NC(=O)Nc2cnc3ncnn3c2)Cc2ccccc2O1 c1(CNC(C(=O)OCC(C)(C)COC(N)=O)Cc2ccccn2)ccc(Cl)cc1 N1(C(=O)C2=CCCOC2)CCC2(CC1)CC2(CO)CNC(C1(C(F)F)CC1)=O n1(CC(=O)NC(c2cccnc2N(C)C)C)ncc2nc(Br)ccc12 CCCCCCCC(F)C(=O)N(CCCNC(c1ccc(C(C)C)o1)=O)CC C=C=CCCC(=O)N1CC(CC(=O)NCCC2CC2C)C(C)C1 N1(ONC(=O)Cn2cnnn2)CCCCC1C1CCCCC1.n1(CC=O)ccnn1 C1(CNC(CNC=O)=O)CC(C(F)(F)F)CCN1C(=O)C(F)CC1CCC1 C1(C2CCN(C(C3(N(C)C)CC3)=O)CC2)(NC(C2C(C)=C2)=O)CC1 C1(NC(C2CCC(=O)N2)=O)C2CC(O)C1N(C(C1C3(CCC3)C13CCC3)=O)C2 CCC(C)CC(C)C(=O)N(C)CCOCCNC(=O)C(=Cc1cccs1)C CC(CC(=O)c1ccc(F)cc1)C(=O)NC1CCN(C(C2CCOCC2)=O)CC1 C1(=O)C(C)(C)N1.C1(C)(OCC(=O)N(CCOC)CCO)CCCC1 c1(C(=O)NC(C)CNC(=O)CCCF)ccc(C(F)(F)F)nc1O C1(O)(CNC(CC=CC=C)=O)CCN(C(=O)CC2(O)CCOCC2)C1 C1(C(=O)NC(c2ccc(C)cc2)C)CC(C)CCN1C(=O)CN(C)C C1(C(=O)NC(C2CN(C(=O)CN(C)C(N)=O)CCO2)C)(CO)CCNC1=O C(=O)(CCC(CC)CC)CC#C.C1CC(=O)NCC(=O)NCC(C2CCCC2)O1 c1(NC)cnc(Cl)cc1C(=O)NCC1CN(CCOc2ccccc2Br)C1 C1(C(N(C(C)C)CCNC(C2CC(O)C2)=O)=O)CCCC(=O)N1 CC(C)C1=NOC(C(N2CCCC(NC(c3cccnc3C(F)F)=O)C2)=O)C1 N1(C(C)=O)CCN(C(C2CN(C(C3C4CCC(F)C34)=O)CCO2)=O)CC1 C(=O)(C(C)CCCOC)NCC1(CNC(CC=CC=C)=O)CC1 C1(C(=O)NCC#C)CC(C)CN(C(=O)CSc2ccc(F)c(F)c2)C1 N1(C(c2cc(OC)c(C(F)(F)F)cc2)=O)CCC(C(=O)O)C12CCOCC2 c1(C(=O)NC2CCC(CCNC(c3scc(C(C)=O)c3)=O)C2)nc(=O)n(C)[nH]1 N1(C(=O)NC2(C=C)CCCC2)CCC(C2CCC2)C1 C12(C(=O)NCCC(=O)NCC)CC(CN1C(=O)C(C(=O)OC)OC)C2 C1(N(C(=O)CCCC2CCOCC2)C)CCN(C(=O)CN2CC(=O)NC2=O)CC1 CCCCCC=CC=CC(N1CCC(NC(c2ccsc2Br)=O)C1)=O c1(NC)snc(C)c1C(=O)NC1CC(C)(CNC(=O)CN2CCSCC2)C1 C1(CC(=O)OCC)CCCC2(CCN(C(=O)CC3CC4CC3CO4)C2)O1 n1(CC(=O)NC2C(CNC(CC(C)CN(C)C)=O)CC2)cc(F)ccc1=O CS(=O)c1ccccc1-c1noc(CNC(=O)C(C)(C)CC2CC(F)(F)C2)n1 C1(C(=O)N(c2c(OC)noc2C)CCC#N)CCN(C(C2CC(C#N)C2)=O)C12CC2 C1(CC(C)C)CCCCN1C(C1C=CCN(C(=O)C(F)F)C1)=O CCN=C(NCC(C)OC)NCc1ncccc1Oc1ccccn1 c1(C(=O)OC)ccc2c(NC34CC(C(=O)N=c5[nH]nc(Br)s5)(C3)C4)nccc2c1 C(=O)(C1COc2ccccc21)N(c1nc(C)nc(Cl)c1F)C(C)(C)C CCCCCCCCCCCn1nc(CCC2CCCC2)nc1-c1c[nH]cc1C c1(CCN(C(c2cnn(C)c2F)C(=O)NC2COC2)C)ccc(F)cc1 n1(CC)ncnc1C(=O)NCC1C=CC(NC(=O)C(O)C2CCCC2)C1 c1(N(C2CCN(C(=O)CN(C3CCCCN3C)C)C2)C)ccnc(Cl)n1 c1(C(=O)NCC(CNC(C2(CCC=C)CCCC2)=O)O)ccc(Cl)nc1OCC CC1CN(C(c2ccc(C(F)F)cn2)C(=O)NC2CCOCC2)Cc2c[nH]nc21 CC(C(=O)N1CCC(C(=O)NC(C)(C)C(C)(C)O)C1)C(C)(C)C c1(C(=O)NCC2(CNC(C(CCSC)O)=O)CCCC2)nsc2ccc(C)cc12 C1(C(=O)NCC2CCC(C(=O)NC3(C=C)CCC3)CC2)CCOC(C)(C)C1 CCC(C)C(O)C(C)C(=O)N1CC(F)(C(=O)NCc2nc(N(C)C)n[nH]2)C1 c1(CNC(C23CCC(OC)C2C3)=O)ccc(O)c(F)c1F C(N=c1[nH]c2c(c(=NC3CCC4CC4CC3)[nH]1)CCC2)c1nn(C)c(Br)n1 C(=O)(N1CCC(C(N2CC(n3ccnn3)C2)=O)O1)C1C(OCC)CC1 N1(C(C=CC(=O)OCC)=O)CC2CCCC(NC(=O)Cc3ccn(C)n3)C2C1 N1(C(C(C(C)NC(COCC#C)=O)C)=O)CCC(C)(CO)CC1 CC(C)(C)CC(O)C(=O)NC1CCN(C(c2occ3c2CCC3)=O)C1C(C)(C)C C1(C)(CC)CCN(C(C2(NC(C3CCC(=O)N(C)C3)=O)CC2(C)C)=O)CC1 c1(C(=O)NCC2(NC(C3COCC4(CCC4)O3)=O)CC2)c[nH]c2cccc(F)c12 C1(C(=O)NCc2c(CNC(CC3(CC)CCC3)=O)c[nH]n2)CCCC1C(C)(C)C Cn1c(C(=O)NCC(CO)NC(=O)Cn2cccn2)cc2ccc(O)cc12 C(=O)(CCCCCCC(=O)NCC(O)CNC(C1CC(=O)OC1(C)C)=O)OC N1(CCNS(CC)(=O)=O)C2CCC1CC(NC(c1cc(Cl)c(F)cc1O)=O)C2 C(=O)(C#CC1CCOCC1)N1CCC(C(=O)NCC2CCOC2C2CC2)(CC)C1 c1(C(N(C(C)C)CCNC(C2CCC(C)O2)=O)=O)ccccc1-c1ncc[nH]1 c1(C(C)NC(=O)NCC2CCC2)sc(Br)c2c1OCCO2 C12CCC(CC1)OC(=O)C(c1cccnc1)N2.NC(=O)COC(=O)C1CC1 CC(C)(C)CC(=O)NC1CCOC1C(=O)NCc1cccc(O)n1 N1(C(CC(C)SC)=O)CC(CNC(C2(Oc3ccccc3)CC2)=O)CC1(C)C c1(C(C=CC(=O)NCCNC(C2CC2(F)F)=O)=O)cccc(O)c1 CCC(CC)(CO)C(=O)NCC1CN(C(C2CCOC(=O)CC2)=O)CC1(F)F Cc1c(CNC(=O)CC2CCN2C(=O)C(N2CCCCC2)C)cno1 c1(C(=O)NCC(C)NC(C=C(CC)C)=O)cccc(COC)c1 Cc1ncc(C(N2CC3CC(C2)N(C(=O)C2=CCCSC2)C3)=O)cc1C#N N1(C(=O)CCC2CCC(C(=O)O)N2)CCOC(c2cccc(Cl)c2)C1 C1(NC(C23N(C(C(C(C)C)F)=O)CC(C2)C3)=O)CC(C)N(C)CC1C c1(CC)cc(=NC(=O)C2(CNC(=O)COC3CCOC3)CC=CC2)[nH]n1C c1(C(=O)NC(=O)CC2CCN(CC3C(C(=O)OCC)C3)C2)ccc(C(C)=O)cc1 c1(NC(C2(C)CCN(C(C(CC)C#N)=O)C2)=O)cc(Br)cnc1OC N1(C(c2c(N)nccn2)=O)CC(NC(=O)C(F)(F)C2CCOCC2)CCC(O)C1 C1(CNC(CC(=O)NC)=O)CCN(C(C2(C)CC(OC)CN2C)=O)C1(C)C CN(C)S(=O)(=O)NCC(=O)NCCC1CN(C(C2CCC=CCC2)=O)C1 c1(CC)ccc2ccc(C(N3CCN(C)C(CF)C3)=O)nc2c1 c1(C(N2CCC(N(C(CC(n3c(CCC)ncc3)C)=O)CC)C2)=O)[nH]c(C)cc1C Cc1cc(Cl)ccc1CC(=O)N(C(C)CNC(=O)Cc1cocn1)C c1(-n2cc(C(C)OC)nn2)ccc2c(c1)CCN(C(=O)C(C)(C)CF)C2 c1(SCC)cccnc1C(N1CC(C(C)NC(c2nn(CC)cc2Cl)=O)C1)=O n1(CC)ncnc1CNC(=O)NCC1CC(C)C1 n1(CC(C)C)cccc(C(N2CC3C(CNC(=O)CCCCCF)C3C2)=O)c1=O N1(C(Cc2cc(C(=O)OC)ncc2)=O)CCN(C(C23CCC(C2)C3)=O)C2CCC12 Cc1cccc(C)c1NC(=O)C(=O)Nc1ncc(NCC(N)=O)cc1Cl c1(C(C)=O)ccc(C)c(C(N2CC(C(C)NC(=O)CN3CCOC3=O)C2)=O)c1 Cc1cc(C(=O)NC2CC2NC(=O)Cc2ccsc2C)cnn1 C1(CC(=O)NC2(c3ccccc3)CC2)(OC)CN(C(c2conc2C)=O)C1 C1(NC(c2c(C(C)=O)ccs2)=O)CS(=O)(=O)CC1NC(c1cncn(C)c1=O)=O c1(C(N2C(CNC(=O)CN3CCSCC3)C=CC2)=O)cc(Cl)c(Cl)cc1O c1(OCC(=O)OC)ccc(S(=O)(=O)NCC2CC2Cl)cc1 c1(C(N2C(CNC(c3cc(F)c[nH]3)=O)C=CC2)=O)cccc(Cl)c1O c1(C(=O)NC2C(CNC(C(N3CCN(C)CC3)C)=O)COC2)c[nH]cc(Cl)c1=O N#Cc1cccc(C2CC2C(=O)NC2CC(O)C(O)C2)c1 C12(C(=O)NCC3CCN(CCC)C3)CC(CN1C(=O)Cc1cnn(C)c1)C2 c1(C(C)OC(=O)N(C)C)cn(CC(N2CCCC2C2CCCOC2)=O)nn1 N1(C(CC2N(CC)CCC2)=O)CC2CCC(C1)N2C(=O)CC(C)P(C)(C)=O c1(OCC)ccc(NC(=O)C(C)OC(=O)Cn2c(C)csc2=O)cc1 CCC(C)CCCC(=O)N(C)CC1CCCCN1C(c1ccoc1)=O c1(NC(CC2CCCN(C(C#CC(=O)O)=O)C2)=O)cc2ccccc2cn1 c1(OC)ccc(C(=O)NCCN(C2CCCCC2)C(c2cn(C)nc2Cl)=O)nc1 CC1CCN(CCC(C)NC(=O)NCC(c2ccc(CO)o2)N2CCCC2)CC1 c1(SCC(N2C3(CNC(c4c(C)nco4)=O)CC(C2)C3)=O)cc(F)cc(F)c1 N1(C(C2C(C(C)C)OCC2)=O)CC(C(=O)NC(CO)C(C)(C)C)C(F)(F)C1 c1(C(=O)NCCCN(C(CC(CCC)C)=O)C)ccc(S(N)(=O)=O)cc1N c1(-c2ccn(C)n2)nc(C23CC(C)C2C3)n(CC2CCOC2)n1 S(=O)(=O)(c1cccnc1NCC1(C)COC(C)(C)C1)NCCCC(COC)(C)C N1(C(c2cnc(C3CC3)o2)=O)CCCCCC1CNC(C1(CC(F)(F)F)CC1)=O C1(CC)CCCCCC1.c1(C(C)(C)CCn2cc(CO)nn2)ncoc1C(=O)N CC(CCc1cccc(F)c1)C(=O)NCC(C)(CO)NC(c1nc(=N)cc[nH]1)=O c1(C(=O)NC(CNC(C2(c3ccon3)CCC2)=O)CO)cc2ccccc2o1 C(C(C)CN(C(=O)COCCF)C)N(C(COCCOCCCCOC)=O)C N1(C(C2CCCC(OC)C2)=O)CCCC(F)(CNC(=O)CCCN(C)C)CC1 O=C1CCCC(C(=O)NCc2nc(CNC(=O)CC3CC4(CC4)C3)cs2)N1 Cc1cn2cc(C(=O)NCC3C(C)CCCN3C(=O)CCc3cnc[nH]3)nc2s1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC(O)C1 N1(C(C(C2(C)CC2)NC(c2c(C)oc(Cl)n2)=O)=O)CCC(CO)C(C)C1 c1(CCC)cc(C(=O)NCC2CC(O)CN2C(=O)C(C)C(F)F)c(C)o1 C1(CNC(C2N(CCC)CCC2)=O)CCCCN(C(=O)CCC2(C)CC2)CC1 C(=O)(C#CC1CCOC1)NC(CC(C)NC(c1ncc(C(N)=O)cc1Cl)=O)C C1(C(=O)NC2C(NC(CCCN(C)C)=O)CCC2)CCOC(C)(C)C1 N1(C(c2c(CC)cco2)=O)CCN(C(c2ccc(C)nn2)=O)C(CC(F)(F)F)C1 c1(C(=O)NCCNC(=O)CC2CCCCO2)ccc(NC2CCCCC2)nc1 C1(CN(C(c2cnc(O)[nH]2)=O)CC)CCN(C(C2CC(O)CN2C)=O)CC1 c1(C(=O)NC2CCC(CC(=O)NCCCC(=O)OC)C2)nc(C)c(C)s1 C1(C)(CNC(C2C(C)C2)=O)CN(C(c2ccc(F)cc2Br)=O)CCO1 N1(C(C(c2cn(CC)nc2)(F)F)=O)CC(NC(=O)CN(C)CCO)C2CC12 CS(=O)c1ccccc1COC1CCN(CC(O)COCc2ccco2)CC1 C1(CCNC(c2c(C)ocn2)=O)CN(C(=O)C(F)(F)CC2CC2)CC(C)O1 CN1CCC(O)(CC(N2CC(O)(CNC(=O)CCNC(=O)C(C)(C)C)C2)=O)CC1 CCCCCC(O)CC(=O)N1CCC(CC(N2CC(O)(C3CC3)C2)=O)CC1 c1(C(=O)NCC23C(CN(C(CC(C)SC)=O)C2)CC3)[nH]c2ccccc2c1C CCC(C)(CNC(=O)CCCOCC(C)(C)C)NC(c1ccc(SC)o1)=O Cc1ccccc1C(=O)NC1(C(=O)NCc2cccc(Cl)n2)CCN(C)C1 CC(C)C(C)(C)C(=O)NCc1occc1C(=O)NC1C2CCCCCC12 C1(CNC(C2(C=C)CC2)=O)CN(C)CCN1C(c1c(OC)cccc1O)=O C1(CN(C(CC2(OC)CC2)=O)C)CC(F)CN1C(=O)Cc1cccn1C C(C(O)CCNC(=O)CNC(=O)OC(C)(C)C)NC(C(C)n1cccn1)=O Cc1cc(C(N2CC(NC(=O)Cc3ccc(O)c(O)c3)CC(C)C2)=O)cnc1F C1(CNC(Cc2cc(C)on2)=O)CC2(CCN(C(=O)C=CC(F)F)CC2)CO1 C1(C(N(CCCCN(C(c2nc(C(=O)OC)oc2)=O)C)C)=O)CCC(C)(C)OC1 N1(C(C(C(C)(C)C)O)=O)CCC2OCCN(C(c3cc(CCCO)on3)=O)C2C1 c1(C(C(=O)NCC)N(CC(C)(CC)OC)C)cccc(C)c1[N+](=O)[O-] c1(CC)cccc(CC(=O)NCCOCCNC(c2cnc(OC(F)F)s2)=O)n1 N1(C(C(C2CCOC2)NC(C)=O)=O)CC(C)OC(C)(C)C1C N1(C(C(OC)OC)=O)CCC2CN(C(=O)CCCc3cncs3)CC2CC1 c1(OC(C)C(=O)N(C(CNC(c2ccc(Br)o2)=O)C2CC2)C)ccccc1 c1(CC)ccc(F)cc1C(=O)NCC1CC1NC(c1ocnc1C(F)F)=O C=Cc1cncc(C(=O)NC(CN(C)C(C2CCN2CC)=O)(CO)CO)c1 Cc1oc(C)c(C(=O)NCCCOCCNC(=O)C(F)OC(F)(F)F)c1Br c1(C(N(CCOCCNC(c2c(C)cc(F)s2)=O)C)=O)cn2cccc(Cl)c2n1 C1(CNC(=NC)NC(C)COC)CCCC1(COC(C)(C)C)OC C=CCC(C(=O)N(C(CO)C1CC1)C)NC(C1CC2(CCC2)C1)=O C(N=c1[nH]cc2ncnc-2[nH]1)C1N(C2CCCN(C)C2=O)CCC1 C#Cc1ccc(C(=O)NCC(C)NC(C2CCOCC2(C)C)=O)cc1 N(C(=NCCC1(C)CC1(Cl)Cl)NC1CCCCC1)CC(C)C#N c1(C(=O)NC(C2CCN(C(C(C)c3ccsc3)=O)CC2)C)nccc(N)c1Cl N1(C(C2(OC)CCC2)=O)CCOCC(CNC(C2(c3cc(C)on3)CCC2)=O)C1 C1(C)(C(N(C(C)C(=O)NOC(C)C(=O)OC)CC)=O)CC(F)C1 C1(NC(C(C)OC)=O)CCN(C(c2csc(-c3nc[nH]n3)n2)=O)CC1 C(c1nc2ccccc2o1)=CC(=O)NC1(CC=C)CCN(C(=O)CC(C)O)C1 C(C(C)(C)CC1CC1)NC(C(C1CCCCO1)NC(C1C(C)C1)=O)=O N1(C(C(c2ccccc2F)C)=O)CC2(C1)CN(C(=O)CN1CCCCCC1=O)C2 C1(NC(Cc2cc(C)on2)=O)CC2(NC(c3coc(C)n3)=O)COC1C2 c1(C2(C(N(CCNC(C3C(C)CCS3)=O)CC3CC3)=O)CC2)ccccc1F N1(C(c2c(C)nc(C)s2)=O)CC2C3CCC(C2C1)N(C(=O)C1=CCCC1(C)C)C3 Cn1cc(-c2cc(C(=O)NC3(CCNC(C45CCCC4C5)=O)CCC3)on2)cn1 C1(NC(Cc2c(C)nn(C)c2)=O)CCN(C(C2CC2F)=O)CC1O N1(C(C(C)S)=O)CCC(O)(CNC(c2cc(O)ccc2Cl)=O)CC1 c1(C(C)C)ccccc1CC(=O)N(C(C)CN(C(=O)CC#N)C)C C(C(C)(C)C(C)(C)C)NC(C1C(CNC(CCCCOCC)=O)C1(C)C)=O c1(CC(N2CC(O)(CN(C)C(C3CC3Cl)=O)C2)=O)ccc(Br)cc1 C1(C(C)C)(CO)CCN(C(=O)CC(C)NC(c2cn[nH]c2)=O)C1 CC(CCCC(=O)NCCCCF)NC(=O)CCC1CCOCC1 N1(C(C2CCCC2)=O)CCC2CN(C(=O)Cc3ccccc3F)C2C1 N1(C(=O)Cn2nccn2)CCN(C(=O)CCc2ccc(Cl)cc2)C(CC(F)F)C1 CCCCC(O)CC(=O)N1CC2CC2(CNC(=O)CCC(=O)N(C)C)C1 C(CC(C)C)(C(=O)NCC1CCCCCN1C(c1ccncc1F)=O)NC(C)=O c1(C(N2CC(C)C(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)=O)ccc(C2CC2)c(Cl)c1 C1(C(=O)NC23CN(C(c4n(C)cnc4)=O)C(C2)C3)CCOC2(CCCCC2)C1 c1(OC)ccc(Cl)c(C(=O)N(C2CC(NC(C3(C4CCCO4)CCC3)=O)C2)C)n1 c1(NC(C2(CNC(C3N(C(CCC)=O)CCC3)=O)CC2)=O)c(OC)cccc1C CN1CC(C(=O)N(CC(N2CC(CN=[N+]=[N-])C2)=O)C)CC1=O C=C(Cl)C(C)(C)C(=O)NCC1C=CCN1C(=O)C(C)C1CCCC1 C#CCCN=C(NCCS(=O)(=O)C1CC1)N1CCc2nn(C)c(=O)cc2C1.CC c1(CCCCC(=O)NC(C)=O)ccc(OCc2ccccn2)c(OC)c1 N1(C(C(C)OC)=O)CC2CCC(CNC(=O)C(F)C3CCCC3)C2C1 C(=O)(C1=C(C)OCC1)NCC=CC(N1CCC(NC(C)=O)C1)=O N1(C(c2c(CNC(=O)C(F)C3CCCC3)ocn2)=O)CCC(C2CC2)(CO)C1 Cc1cnc(Cl)[nH]c1=NCCN1CCN(CCNC(=O)C2=CCCS2)CC1 N1(C(CCCC#C)=O)CCN(C(=O)C(N2CCOCC2=O)C)CC1CC(F)F C1(C(N(CCN(C(c2[nH]cc(CC(C)C)c2)=O)C)C)=O)CCCCN1C1COC1 Cc1cc(=NCC2COC(C)C2)c(F)c[nH]1 Nc1c(C(N2CCOC(CCC3(CO)CC3)C2)=O)cnn1CC(F)(F)F c1(CN2CCN(C(C(CNC(C)=O)(C)C)=O)CC2)ncnc2c1CCC2 N1(C(CSC)=O)CCCC(NC(c2cccc(OCC(C)C)c2)=O)C1C N(C(=NCc1ccc(OCCO)cc1)NCCF)CC1CN(S(C)(=O)=O)C1 Cc1cc(CN2CCC(F)(CNC(c3cc(I)ccc3F)=O)CC2)c(F)cc1Br c1(C(N(CCCC(=O)NC(C)Cc2cccnc2)C)=O)ccc(F)nc1 CC(O)C(F)(F)C(=O)N1C(CNC(=O)C(Cl)=CCl)CC2CC12 C1(NC(CCC(C)O)=O)CC2CCC1N2C(=O)CN(C)C(=O)C1CC1 c1(NC(C2CCN(C(C(F)=CCC)=O)C2)C)nc(C)ccc1C(=O)OCC C(=O)(C1=CCOCC1)NC(C(N1CCCC(CC(C)C)C1)=O)C1(C)CC1 c1(C(=O)NC2CC(C)N(C(=O)C(CO)C(C)(C)C)CC2)cc2cc(F)ccc2[nH]1 C1(C(=O)NC(c2nc(CC)on2)C)CC2(CCC2)CN1C(C1CN(C(C)=O)C1)=O C=CCCC(C(=O)OC)NC(C1(C)CCN(C(c2ccc(CC)cn2)=O)CC1)=O N1(C(C=CC(CC)C)=O)CCC(CF)(NC(=O)COC(C)=O)C1 O=S(=O)(c1cnccc1F)N1CCCC(c2ccccn2)C1 c1(OC)ccc(F)cc1C(=O)N(C1CCN(C(=O)C(C)(C)C2CCOC2)C1)CC C12(CNC(c3ccoc3)=O)CCC(CC1)N2C(C1(C(F)(F)F)CC1)=O C1(C(=O)NCC2C(OC)CCC2)CN(C(=O)CSC(F)F)CCC1(C)C C=CCCCC(C(=O)N(C(C)C(F)F)C)NC(=O)CCc1cscn1 CC1OC2(CNC(=O)CC3CC4C=CC3C4)CC1(NC(=O)Cc1cccnc1)C2 CC1=CCN(C(=O)C(c2ccccc2)NC(=O)C(C)N2CCCC2)C1 C1(C(=O)NC2CC(C(=O)NCCCCOC)C2)CCCOC1 Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)C(C)CN(C)C)c(C)s1 C(C)(C(C)(C)OC)NCCOCCOCCN(C(COC)=O)C c1(C(=O)NC2CN(C(C=Cc3cc(OC)ns3)=O)C2)ccc(C#N)c(O)c1 c1(NC(C2N(C(C3C(OCC)CC3)=O)C(C)C2)=O)cnc(CC)nc1 N1(C(CN(C)CC)=O)CCC2CC(NC(c3cnco3)=O)CCC2C1 N1(C(Cc2ccc(C)cc2N)=O)CCN(C(=O)C=C2CCC(C)C2)C2CCCC12 n1(CC(=O)N(CC(CN(C(C(COC)(C)OC)=O)C)O)C)nc(C)n(C)c1=O C1(NC(C(C)OCC(F)(F)F)=O)CN(C(=O)CSCC(F)(F)F)CC(C)(C)C1 c1(C(=O)NCC2CC(NC(c3n(CC#C)ccc3)=O)C2)ccc(Cl)c(C)c1OC C1(NC(C2C(C(=O)OC)C2)=O)CC(F)CN(C(c2cccc(C(C)(F)F)c2)=O)C1 N1(C(C)C)N=C(C(=O)NCC(C)(C)CNC(C2CCCCN2N=O)=O)CCC1=O c1(C(=O)NCC(CN(C(CN(C)CC)=O)C)C)cc(OC)c(C2CC2)nn1 N1(C(C2C(C=C(C)C)C2(C)C)=O)C2CCCC1CN(C(=O)C=C(C)C)C2 c1(C(=O)NC(C)CNC(C2CC(C)C2)=O)cc2n(n1)CC(F)C2 c1(CC)cccc(C(CC)(C(=O)O)NC(=O)CCCC2CCCS2)c1 C(=O)(CC(CCC)CCC)NCC(C1CCOC1)NC(c1n(CC#C)cnn1)=O c1(C(N(CC(CN(C(c2cc(C)sn2)=O)C)O)C)=O)cnc(N)c(N)c1 N1(c2c(C)cccc2)CCN(C(=O)C(O)C2(N)CC2)C(C)C1=O C(CNC(C1CCN(C)C(=O)C1)=O)(C(=O)NOCCCF)OC N1(C(c2csnc2C)C(=O)NCC=C)CC(C)OC(C)(c2ccccc2)C1 C1(C(N(CCCNC(c2cc(CC(C)C)on2)=O)CC)=O)CCC(C)=C(C)C1 C=C=CCCC(=O)NCc1c[nH]nc1C1CCN(C(C2CCCN2CCC)=O)C1 c1(SC)c(NC(C2(NC(=O)CC(C)(C)C3CC3)CC2(C)C)=O)cnn1C c1(C(=O)NCCC2CCN(C(c3ccc(C(C)=O)[nH]3)=O)C2)sc(F)cc1Cl c1(NC2CN(C(C3(CC)CC3)=O)CC2C)cc(C)c([N+](=O)[O-])cc1Br N1(C(c2ccc(CNC(C(CCCC#C)C)=O)cc2)=O)CC23CCC2(COC3)C1 N1(C(C2(CC)COC2)=O)CC2CCN(C(c3cccn4cnnc34)=O)CCC2C1 C1(C(=O)NC(c2cn(C)nn2)C(=O)NCC(=O)OCC#C)CC2CC(=O)C1C2 N1(C(CS(=O)(=O)NC)=O)CC(NC(C2CNC(=O)CC23CCC3)=O)CC(C)(C)C1 C(=O)(C(CCC(N)=O)N=[N+]=[N-])N(CC(C)NC(=O)C#CC1CCCC1)CC c1(CNC(=O)C2=CCCS2)ccc2c(c1)CCN(C(c1ccns1)=O)C2 CCC(CC)C(C(=O)N1CCCC1CNC(=O)CCCCOC)N1CCOCC1 C1(C(=O)NC(C(C)C)CNS(C)(=O)=O)C2CCC1C(F)(F)C2 Cc1cccc2c1OC(C(N1CCCCC1CNC(=O)Cn1ccc(=N)[nH]1)=O)C2 c1(NC(C23N(C(C(CC)C(C)C)=O)CC(C2)C3)=O)cc([N+](=O)[O-])ccc1SC N1(C(C(C(=O)OCC)(C)F)=O)CCC2(CCCC2NC(=O)Cc2nc[nH]n2)CC1 CCC(C#N)C(=O)NC(c1cccnc1)C(=O)NCCc1ncccn1 Cc1cccc2cc(C(N3CC(C)(NC(=O)CN4CCC(C)C4)C3)=O)sc12 Cc1[nH]c(C)c(C(=O)N(CC(O)CN(C)C(C2CCC2CF)=O)C)c1C N1(C(C(C)CO)=O)CCCC(C)(C)C1C(=O)NC1CCN(C)CC1(C)C c1(C(=O)NCC2N(C(Cc3nc(C)[nH]n3)=O)CC(O)C2)cc(C#N)c(F)cc1F Cc1sc(S(N)(=O)=O)cc1C(=O)NC1CCCCN(C(C2(C)CCCCO2)=O)C1 N1(C(=O)C(O)CC2CCCCC2)CC2(CCCC2)c2cc(Br)ccc21 C1(C(N2CCC(=C)C2)=O)CCC(C)CN1C(=O)COCCN(C)C c1(-c2ccc(CN(C(C)=O)C(C)C)s2)ccc(NC(=O)C(O)C(C)CC)cc1F C1(C(N2C(C(=O)NC(CC)C(N)=O)CCC2)=O)CCCC(C#N)C1 C1(NC(C(CCCOC)(C)C)=O)CC2(CCCN(C(c3cccn3C)=O)C2)C1 C1(CC)(NC(c2cc(C)cs2)=O)CCN(C(=O)C(c2cccc(Cl)c2)SC)CC1 N1(C(C(C(C)C)O)=O)Cc2ccccc2CC1CNC(=O)C(C)(O)C(C)(C)C c1(OC)c(C)cc(NCc2ccc(Sc3ccccc3)cn2)cc1I c1(SC)nc(C)c(CC(N2CC(NC(C3CCOC3)=O)C(C)C2)=O)c(O)n1 c1(C(N(CCC(=O)NC(C)Cc2cnc[nH]2)CC=C)=O)cc(C)cs1 c1(OCC#C)cccc(C(=O)NCC(CC(C)C)NC(C2NC(=O)OC2C)=O)c1 C(CC(F)(F)Cn1cc(C2CCCCCC2)nn1)NC(C(CC)n1cncn1)=O c1(C(C)=O)cccc(C(=O)NC2COCCC2NC(C2CC=CCC2)=O)c1 C1(C)(CNC(c2cc(C)nn2C)=O)CCCN(C(c2ccnc(C(N)=O)c2)=O)C1 CN1N=C(C(=O)N2CCCCC(NC(=O)CCCN=[N+]=[N-])C2)CCC1=O C=CCC(CC(C)C)C(=O)N1CC(CNC(=O)CC2CCN(S(C)(=O)=O)CC2)C1 c1(CC(=O)NC2(COC)CN(C(=O)C(C)(C)SC)C2)c(C)[nH]c2ccccc12 c1(C(=O)NCCCOCCCNC(C(c2cn(CC)nc2)=O)=O)cc(O)ncn1 N1(C(C(C)OCCC=C)=O)CC(NC(=O)Cc2cncc(C)c2)C(S(C)(=O)=O)C1 CCCCC(C(=O)N1CCC(Nc2nccnc2F)CC1)C(C)C N1(C(CCC(C)(C)F)=O)CCN2C(=O)C(NC(c3cc([N+](=O)[O-])n[nH]3)=O)CC2C1 N1(C(C(C)=C(C)C)=O)CCN(C(C2CC2c2ccc(Cl)s2)=O)CC1CC(=O)N(C)C N1(C(CCC2(NC(C(C)SC)=O)CCCC2)=O)CC(=O)NCC1C C1(CNC(C(C)NC(N)=O)=O)CC(O)CN1C(=O)CCCC1CCCC1 N1(C(CN(C)C)=O)CCCC(C)(C)C1CNC(C1CC1C1CC1)=O C(C(C)C(F)C(=O)NCc1nncn1CCC)NC(c1c(CCC)nco1)=O N1(Cc2ccc(C(C)C)nc2)CCNCC2(CCC2)C1 C(c1sc(Cl)nc1Cl)=CC(=O)NC(C)CNC(c1c[nH]nc1Br)=O N1(C(C2C(C)SCCC2)=O)CC(C2CC2C(=O)NCC2(F)CC2)C1 c1(C(N(C)CC2CC(F)CN2C(=O)CC2CCCO2)=O)ccn2cncc2c1 Cc1ccc(NC(c2c[nH]nc2CCNC(C2(C)CCCS2)=O)=O)c(O)c1 CC1CN(C(C2CCC(=O)N2C)=O)CC(C)CN1C(C1CSC1)=O C1(C)(NC(C2C(NC(Cc3ccn(C)n3)=O)CC2)=O)CC2(CC2)C1 C1(C(N2CCC(O)(CNC(CSCC(N)=O)=O)CC2)=O)CCN2CCOCC12 C1(NC(CSCC=C)=O)CCN(C(=O)C=Cc2ccncc2C)CC1C(C)C c1(C(=O)NCC(CC)NC(c2cc(O)n(C)n2)=O)ccc2ccccc2c1F Cc1cc(C(N2CC3CC3(CNC(=O)CCSC3CCC3)C2)=O)ncc1C(F)F C1(NC(C2CC3CCC(C2)O3)=O)CCCCCN(C(c2cccn2C2CC2)=O)C1 Cn1cc(C(=O)NCC(O)CNC(c2ccc(CCC#N)cc2)=O)n(C)c1=O CN1CCN(C(C2CC=CC(O)C2)=O)C(C(=O)NC(C(O)CO)C2CC2)C1 c1(NC(N2C(Cn3cc(C4(SC)CC4)nn3)C=CC2)=O)c(F)cccc1[N+](=O)[O-] c1(C(N(C)CCC2CCN(C(=O)C3=CC(C)(C)C3)CC2)=O)ncc(C#N)cc1Cl C1(C(N2CC(CC(=O)NCC3(C)OCCO3)(OC)C2)=O)CC(C)(C)CO1 C#CC1(O)CCN(C(C)C(=O)NCC2CC(NC(=O)C(F)C(C)(C)O)C2)CC1 c1(OS(=O)(=O)CC2CC3CC3C2)cc(Cl)cc(I)c1 c12ccncc1NC2.N1(C(C(N2CCC(SC)C2)=O)=O)CCS(=O)CC1 CCCCC(C)CCC(=O)NC(CCN(C)C)C(=O)NOC(C)C(=O)OC c1(CCC(=O)NCCC2CCCN2C(=O)C=Cc2ccco2)cccnc1 c1(C(=O)NCC2(NC(C(C3(OC)CCCC3)(F)F)=O)CC2)ccnnc1O c1(CC)nc(C)oc1C(N1CCC(CF)(NC(=O)CCOCC(C)C)C1)=O n1(-c2ccnc(C)n2)cc(S(=O)(=O)N2C(C)CCC2C)cn1 c1(C(=O)NC(C2CCCN2C(=O)CC(=O)N(C)C)C)ccc(CCF)cc1 c1(COCC)nc(C)c(C(=O)NC2CC(NC(=O)CCOC)C2)s1 N1(C(C(C)c2ccsn2)=O)CCC(C)(CNC(C2CCCC3(CC3)C2)=O)CC1 CCC(CC(=O)NCC1CC2CC2N1C(c1cnc(-c2cccs2)o1)=O)OC C1(CNC(C(C(C)O)C)=O)CC(C)CCN1C(=O)CSC1CC1 C1(C(=O)NCC2(C)C(C(=O)OC)C2)CC(F)CN1C(=O)CC1CCOC1 C1(C(=O)NC2CCC3CCC23)(CNC(COCCOCC)=O)CC(F)(F)C1 N1(CCCNC(CNCC(=O)NC)=O)CCOCC1 C=CC(C)(CC)C(=O)NCC1(CCCNC(=O)Cc2ccns2)CCCC1 CCCCCC(F)C(=O)N1CC(OC)CC1(C)CNC(=O)CC1(O)CCC1 C1(CNC(C2C(OC)C2)=O)CCC(F)(CNC(=O)CSC2CC2)C1 CS(C)(=O)=Nc1ccc(C(=O)NC2CN(C(=O)CNC=O)C3(CCC3)C2)s1 c1(NC(C)=O)cccc(C(=O)NC2CCCC(NC(=O)Cc3nc(C)no3)C2)c1 C1(N(C)C)Cc2ccccc2N(Cc2ccc(-c3cn[nH]c3)s2)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)N(CC)CC1CCCN1C(=O)C1=C(C)OCCS1 C1(C(=O)NCc2nc(=O)o[nH]2)CC2C=CC1N(C(=O)CCc1nc[nH]n1)C2 c1(C(=O)NCC2C(C)CCCN2C(=O)Cn2ccnn2)nccc2ccsc12 c1(OCC(=O)NCC2CCCN2Cc2ccc(Cl)cc2)cccc(Cl)n1 c1(C(=O)NCC2C3N(C(C(C)OCCC=C)=O)C(CC3)C2)cnc2[nH]nnc2c1 CC(C)CCN=C(NCC1CCOC1(C)C)NC1CC1C(F)F N1(C(CNS(N)(=O)=O)=O)CC(NC(=O)CCN2CCCC2=O)C(O)C1 C(c1cnn(C)c1C)=CC(=O)N(C(C(=O)N)c1ccsc1)CCC#N.CN C1(C(=O)NC(C)CCN2CCCC2)CC12CCN(C(=O)Cc1ccns1)C2 C(=O)(C(C)(C)CCC#N)NCc1c(CCC(=O)NC(CC=CC)CO)cccc1 C1(NC(c2c(Cl)cnc(C)n2)=O)CCN(C(=O)C(=O)N=[N+]=[N-])CC(C)(C)C1 CCCCC(CC(=O)N1CCC2(CSC2)C1)NC(c1cccs1)=O N1(C(CCCCCSC)=O)CCC2(CC1)CC2C(=O)N(C)Cc1cocn1 C(=O)(C(C)CC(C)C(C)=O)NC(CCC(=O)NCCc1cn(CC)nn1)(C)C C12(C(N3CCC(C=C)(O)C3)=O)CC(CCO1)N(C(c1cnn(C)c1OC)=O)C2 C1(CN(C(=O)CN2CCCC2CO)C)COCCN1C(c1sccc1F)=O c1(C(N2CCC(CC)C2C(=O)N(C(C)C(C)SC)C)=O)cccc(C)c1N c1(C(=O)NC2CCC(n3cc(CCC(=O)NC)nn3)CC2)cc(C)cc(C)c1 c1(C(N2CCN(C(C(CC)(C)O)=O)CC(O)C2)=O)cc2c(C)cccn2n1 C1(NC(C=Cc2c(C)ncs2)=O)(CO)CCCN(C(=O)C=CBr)C1 c1(OC)cc(CNC(c2cc(C)cc(Br)c2)C)c(F)cc1F C#CC1(O)CCCC(NC(=O)CCc2nc3ncccn3n2)C1 C1(CNC(C2(OC)CCOC2)=O)CN(C(C2CCCOC2)=O)CC(C)(C)O1 C(=O)(C(C)C(O)C(C)C)N1C(C(=O)Nc2c(O)ncc(C)c2)CCCC1 N1(C(C(C2CN(C(=O)C=Cc3cc[nH]n3)C2)OC)=O)CCC(O)(C(N)=O)C1 N1(C(c2c(C)sc(-c3ccccc3F)n2)=O)CCC(C)(C)C1C(=O)O C1(NC(c2n(CC)ccc2)=O)C2CC(NC(=O)C(n3ccnc3C)C)CC12 C1(O)(CCNC(C2N(CC)CCOC2)=O)CCCN(C(=O)C=Cc2cn[nH]c2)C1 C=CCCCCCC(=O)N1CCN(C(=O)CCCS(N)(=O)=O)CC1CCC N1(C(C2(CCNC(Cn3c(C)cc(C)n3)=O)CCC2)=O)CCC(C2CCCC2)C1 c1(C(=O)NC(c2ccccc2)C(C)NC(C(C)=CC)=O)c[nH]c(C(=O)NC)c1 C1(CNC(CNC(CC)=O)=O)CC(O)(CNC(=O)CN(C)CC)C1 C1(NC(C2(C)CC(C)C2)=O)CCC(F)(CNC(c2nc(C3CC3)cs2)=O)C1 Cc1nc(NCC(C2CC2)NC(C2CC(=O)N(C(C)(C)C)C2)=O)cc2nncn12 C1(CNC(C2(N(C)C)CC2)=O)CCCCN1C(=O)CCc1cccnc1 C1(N(C(CS(=O)(=O)NCC)=O)C)CN(C(c2ccc(C(C)=O)cc2)=O)CCC1C C1(O)(c2cn(CC(N3C(C)(CC)CC(OC)C3)=O)nn2)CCC(C)(C)CC1 C#CCC(CC(=O)NCCC(O)CO)NC(C1CCC(=O)N(C)C1)=O C(CC1=CCN(C(=O)C=Cc2cccc(N(C)C)c2)CC1)NC(CC=CC=C)=O N1(C(C(C)NC(C)=O)=O)CCCN(C(C2CCC3(CC3)C2)=O)C(CO)C1 N1(C(C=CSC)=O)CC(CCNC(c2ccn(C)c(=O)c2)=O)OC(C)C1 Cc1ccc(C(=O)NCC2(NC(=O)Cc3ccoc3C)CCC2)cc1 CN1CCCCC1CC(=O)NCC1CN(C(c2cccnc2C(F)F)=O)CC1O c1(C(=O)NC2CC(CNC(c3cnc(CCCC)s3)=O)C2)oc(CC)nc1C C1(C(=O)NC(C)CCNC(=O)CCc2ccc(Cl)s2)NC(=O)CC1C(F)(F)F c1(C(=O)NCc2nc(CNC(C(C)(C)O)=O)sc2)cn2c(n1)CCCC2 CC#CCC(C(=O)NCc1cnc(C)o1)NC(=O)C(C)CC CC1(C)CCC(CNC(=O)Cn2nccn2)N(C(c2cc(F)c(F)cc2O)=O)C1 c1(N2CCCC(C(C)C)C2)nc(Nc2cccc(OC(C)C)n2)c2ccsc2n1 C12(NC(c3ncc(F)cc3F)=O)CCN(C(=O)Cc3cn[nH]c3)CC1C2 C12(C(=O)NC(CC=C)(C)C)CCCC1CCN2C(=O)CC(O)C1CCCC1 C(=O)(CCCCC(F)(F)F)NC(CNC(C(CC(=C)C)OC)=O)C1CC1 c1(C(=O)NCCONC(C2N(C(C)=O)CC2)=O)n[nH]c(C)c1COC(C)(C)C c1(OC)cccc(CN2CCCC(C(=O)NC3COCC3O)CC2)c1C C(CCCC(=O)NCC1CC(OC)CN1C(C1CC1C)=O)OCCC=C c1(C(=O)NC2C(O)CCN(C(c3nc(C(C)(C)C)on3)=O)C2)cc(Cl)cc(Cl)c1N c1(C(=O)NCC(CC)NC(=O)C(c2cncnc2)C)ncc(F)cc1C C1(C=O)CN(C(=O)Cc2cnns2)CCC1(C)C.c1(OC)ncc(C=CC)cn1 Cc1cc(CCCC(=O)NCCC2CCC(NC(=O)CCOC(C)C)C2)c(C)s1 C1(C)(CC)CC(NC(=O)CSCCN(C)C)CN1C(c1ccc(C2CC2)o1)=O C1(CNC(CS(CC)(=O)=O)=O)CN(C(=O)CCC2COC(C)(C)O2)C2COCC2O1 CCC(C)(CC(=O)N1CCOCC(NC(=O)Cc2ccc(C)s2)C1)C(=O)OC N1(C(c2nc(CCCC)sc2)=O)CC(CNC(=O)C=C(Cl)Cl)C(C)C1 C1(C(=O)NC(CCC)C(F)(F)F)CCC(C)(C)N(C(C2CC3CCC(C2)O3)=O)C1 c1(NCC(C)NC(C2CCC2c2ccccc2)=O)ccccc1[N+](=O)[O-] C(C(C)(O)CCO)NC(C1C(CNC(CN(CC)CC)=O)CCO1)=O c1(C(N2CC(OCCC(=O)NC3CCC(O)C3)C2)=O)cnc(O)c(F)c1 c1(-c2cn(CC#N)nc2)ccc2nc(CC(=O)NCC(O)CO)cn2c1 CC1CCN(C(=O)CC2CC(C)(C)CO2)CC1NC(=O)C=C(C1CC1)C1CC1 C(=O)(CC(C(F)(F)F)N1CCOCC1)NCC(C)NC(c1cn(C)ccc1=O)=O c1(C(=O)NCCCC(C)NC(C(CC=C)(C)C)=O)c(C)c2ccccc2oc1=O c1(CC)cc(C(N2CCC(O)(CCNC(=O)CN3CC=CC3)CC2)=O)cc(F)c1 c1(NC(CC2N(C(C=CCCC)=O)C3CCC2C3)=O)cc(OC)c(F)cc1Br CCCCC(F)C(=O)N(C1CN(C(c2cnc(C)nc2C)=O)CC12CC2)C C12(C(N3CCC(CNC(C4C(C(C)(C)C)C4)=O)CC3)=O)CCC(C1)C(C)(C)O2 Cc1ncc2c(n1)CCC(NC(C1OCCOC1(C)C)C)C2 N1(C(C2(OCC)CCCC2)=O)CC2(C)CC1(C(=O)NC1(C3CCCO3)CC1)C2 c1(NC(=O)NC2C(CC(C)C)CC2)cnn(C(F)(F)F)c1 c1(OC)ccc(CO)cc1C(=O)NCC1CC(O)CN1C(=O)Cc1cc(C)[nH]n1 C1(OC)CC(CN)N(C(C2(c3ncco3)CCCC2)=O)C1 Cc1cc(=O)ccn1CC(=O)NC(C)CC1CN(C(C23CCC(CC2)CO3)=O)C1 N1(C(CONC(CC2(OC(C)=O)CC2)=O)=O)CCC(C2(O)CC2)CC1 C(=O)(C(F)C(C)(F)F)NCCSCC(=O)NC(CC(=O)OC)C1CC1 C1(C(=O)NCC(C)N(C)C(c2cc(C3CC3)[nH]n2)=O)COCCN1C c1(C(=O)NCCC2(O)CN(C(Cc3c(C)scc3)=O)C2)ccc2nn[nH]c2c1 Cc1cccc2c(C(N3CC(C4CN(C(C5CCNC(=O)C5)=O)C4)C3)=O)c[nH]c12 C1(NC(c2ncc(C(F)(F)F)s2)=O)CC2CN(C(c3cc(Cl)sc3Cl)=O)CC12 C1(OC)CCCC(CC(=O)NC(C)(C)CCNC(c2cc(CO)[nH]n2)=O)C1 CN1CCC(C(=O)NC2CCCC2NC(c2ccnc(CC(F)(F)F)n2)=O)C1=O CC(C)(O)C(C(=O)NC1CCCC1CN=[N+]=[N-])NC(=O)C(O)C1CCCC1 c1(CCCC)cc(C(=O)NCCC2CCN(C(C3(C)CC=CCO3)=O)C2)c(C)o1 O=C(Cn1cc(C#N)cn1)NN1CCCC1C(=O)NC1CCCC(O)CC1 c1(C(=O)OC(C)(C)C)ccc(C(=O)CN2CC3C(CN=[N+]=[N-])C3C2)cc1 CCC1=C(C(=O)NCC(COC)NC(c2[nH]ccc(=O)c2C)=O)CCCO1 CCCCCC(O)C(=O)N1CCC(O)(CNC(c2cccc(OCC)c2)=O)C1 c1(C(=O)NCC2N(C(C(CC#C)C3CC3)=O)CC=C2)cccc2ncnc(O)c12 c1(C(=O)NC2CCN(C(C3C(=C)C3)=O)CC2O)ccc(S(=O)(=O)NC)nc1 C1(NC(C(C)Sc2ccncc2)=O)COCCC1NC(c1sccc1C(F)F)=O C1(CNC(C2CC(=C)C2)=O)CC2CN(C(c3n[nH]c(CC)c3Cl)=O)CC12 c1(C(=O)NCC(C)CN(C(=O)CCCC2CCCO2)C)cncn(C)c1=O C(CC(=O)N1CCOCC1C(C)O)(C(F)F)NC(C1CC(CC)C1)=O CC1(C)CN(C(C2(O)CC2)=O)CC(CNC(c2cc(C(C)(F)F)on2)=O)O1 C1(CNC(Cc2c(-c3ccc(C)cc3)nc(C)s2)=O)CCCN(C(=O)CCF)CC1 S(=O)(=O)(c1cccs1)Nc1cccc(-n2c(C)cc(C)n2)c1.C12CON(C1)C2 c1(C(N2CCC2CNC(C23CCC(C2)OC3)=O)=O)cnc(OCC(F)F)cn1.O=CCO C(C(=O)N1CC(C)(C)C1Cn1cc(CCCCO)nn1)(C(C)(C)C)OC(C)(C)C N1(CC)C2CCC1CN(C(=O)CCCCNC(C1CS(=O)(=O)C1)=O)C2 N1(C(C(CNC(C2(OC)CC(C)C2)=O)CC(C)C)=O)CCC2(CCCN2C)C1 CCC(C)CC(C(=O)NCc1cscc1C)NC(=O)CC(=O)OCC CCC(C)(CCC(C)C)C(=O)NCC(C1CC1)NC(=O)CC1CCC(F)(F)CC1 c1(CNC(c2cc3occc3s2)=O)nc2c(s1)CN(C(C1CC(CF)C1)=O)CC2 C(=O)(C(CCCO)c1ccccc1)N1CCCC(CNC(=O)CC2(CO)CC2)C1 c1(C(N(C2CCN(C(c3ccc(CCC)s3)=O)CC2)CC#C)=O)cccc(O)n1 c1(C(N2CC(NC(c3c(CC)non3)=O)C2)=O)sc(CC)nc1NC(=O)OC CC1(C)Cc2nc[nH]c(=NCCNC(=S)Nc3nc4c(s3)CCCC4)c2C1 N1(C(C)=O)CCC(N(C(C2CCCCCC2)=O)Cc2sncc2C)C2(CC2)C1 c1(C(=O)NCC2CN(C(CCCC(=O)OC)=O)C(C)C2)nccc2ncccc12 c1(NC(C(N2CC(CC(=O)OC)OCC2)=O)=O)cnc(C#N)c(OC)n1 c1(OC)ccc(F)c(C(=O)NCC(C2CC2)NC(=O)CC(C)CF)c1F Cc1ccc(CCC(N2CC(NC(C3(C#N)CCCO3)=O)C(C)C2)=O)c(C)c1 Cc1noc(SC)n1.C(C)(C(C)(C)NC(=O)COCC1CCCO1)NC(CC)=O C(=O)(C(CC(N)=O)NC(c1ccc(C)n1C)=O)NCC(CC=C)(C)O C1(C(=O)NCC2CC(NC(=O)CCc3nccs3)C2)CCC2C(C1)C2(F)F C1(NC(c2c(C)[nH]nc2C(F)(F)F)=O)CCCN(C(=O)C2=CCCCC2)CCC1 CC(=O)CCCC(=O)NCC(C)(C)CN(C(=O)Cn1cc(Cl)cn1)C N1(C(=O)CSC2CC2)CCC(NC(C2(O)CCOCC2)=O)CC1C1CC1 Cc1ccc(I)c(C(=O)NC2CCNC2Cc2ccccc2)c1 C(C)(C)(CC=CC(=O)NC1CC(C(=O)OC)C1)NC(CC1C(CC)C1)=O C(CC1=CCN(C(=O)CNC(=O)C2CC2)CC1)NC(c1ccn(C(C)(C)C)c1)=O c1(C(=O)NC(CNC(COCC)=O)(C)C2CC2)oc(Br)nc1C(F)(F)F C1(NC(C=CC(C)=O)=O)CCCC1NC(=O)CCc1cscn1 CCC(C)C(O)C(=O)N(C1CCCN(C(c2cc(C3CC3)on2)=O)C1)CCF C(=O)(C1=NNC(=O)C1)NCCSCC(=O)NCC(CCC)OC N1(C(c2ccc(COC)o2)=O)CCCC(NC(=O)CC23CCC(CC2)OC3)C1C C1(O)(C(N2CC(CC(=O)NCC(CC)(C)COC)C(C)C2)=O)CCCCCC1 c1(C(N2CC(C(=O)NC3CC(=O)OC3)NCC2)=O)c(Br)ccc2c1OCO2 c1(CNCc2cncc(C(F)(F)F)n2)sc2c(c1Br)CNC2 N(C1CC(C)n2ccnc21)C(=O)NCc1cccc(-n2ccc(C)n2)c1C C1(C(N(CC#CC)C)=O)C2CC(O)C(C2)N1C(c1ccc(C)nn1)=O N1(C(C)=O)CCN(C(=O)C(F)(F)C2CCN(C(=O)CCc3cc(C)n(C)n3)C2)CC1 O=C(C1CCc2c(Br)cccc21)NC1CCCN(C(C2(F)CC2)=O)C1 C(=O)(CCN=c1[nH]c(Cl)nc(=N)[nH]1)NC(c1ccccc1Cl)C CC(C)C(CNC(=O)CC1CCCOC1)C(=O)N(C)CC1CC(F)C1 C1(CC(=O)NCCCNC(=O)C2CC2)OCCC1NC(C1CCOC1)=O Cc1cc(CN(C2CCN(C(=O)COC3CCOCC3)CC2)C)cc(F)c1 N1(C(C(C(=O)OC)(C)C)=O)CC2CCCC(N(C(=O)CC(C)C)C)C2C1 N1(C(c2cnc(C)nc2)=O)CC2(CC(CC(=O)Nc3cccc(Cl)c3I)C2)C1 c1(CC)ncc(C(=O)NC2CN(C(=O)C(F)n3cccn3)CCC2CO)c(C)n1 CC(C)(C)CC(O)C(=O)NCC(c1ccc(F)cc1)NC(=O)C(F)C(C)(F)F c1(C(=O)NCC(=C)CCNC(C2CC(=O)N(C)C2)=O)cnc2c(c1)CCCC2 N1(C(CN(CCC)C)=O)CCCCC1CCN(C(=O)C(=O)C=Cc1cccs1)C C=CC(C)(CCOC)C(=O)NCC1CN(C(c2cc(C#N)c[nH]2)=O)C2(CCC2)C1 c1(C(=O)NC2C(CNC(C(CCC)C)=O)COC2)nnc2ccccn12 N1(C(COCC=C)=O)CCOC2(CCC(NC(=O)C(C)C(F)(F)F)CC2)C1 N1(C(=O)C2=CCC2)CC2(C1)CN(C(C1CCCCN1C1CCCC1)=O)C2 CCC(C)(O)C(=O)NCC1(O)CCN(C(c2ccccc2-c2nc(C)no2)=O)C1 c1(CNC(CCOCCCNC(CC=CCC)=O)=O)cccc(F)n1 C(CC)(C(=O)NC(CC(=O)N1CC(O)(C(=O)OC)C1)C1CC1)OCC c1(C(=O)NCCCCCN(C)C(c2ccc(F)cn2)=O)c(S(N)(=O)=O)cnn1C C1(O)(C(=O)NC2CC(CNC(=O)Cc3ccc(Cl)cc3Cl)C2)CN2CCC1CC2 c1(C(=O)NC(CCC2N(C(C(=O)N(C)C)=O)CCCC2)(C)C)ccnc2c1CCC2 c1(NC(=O)NCCC23CNCC2C3)cccc(COc2ccccc2Cl)n1 C(CC(=O)NCCCn1cc(C)cn1)(C(C)(C)C)NC(COC(CC)C)=O CC1(C)C(CC(=O)NC(c2ccccc2OCC(F)F)CC(=O)O)CC1O C(=O)(CCC(C)(C)F)N1CC(NC(c2c(C)ccs2)=O)C(C(F)F)C1 N1(C(C(C)P(C)(C)=O)=O)CC(C)(C)OCC1CNC(C1CC2CCC1CC2)=O c1(-c2cn(CCC(C(=O)NC3C(CSC)CCC3)O)nn2)c(C)cccc1F C1(CNc2cn(CC(=O)O)nc2-c2ccccc2)CCc2ccccc2CC1 N(C(=NCC1CCCOC1)NC1CCCC1)CC1C(=O)CCC1 c1(NCC(c2ccccc2Cl)OC)nccc(=NCC(C)(C)N2CCCC2)[nH]1 N1(C(C(CC=CC)NC(=O)CCc2nc(O)n[nH]2)=O)CCC12CN(C)C2 N#CC1CN(Cc2cc3ccccc3o2)CCN1C(c1cc(=O)cco1)=O c1(CC(=O)NC2C(NC(CNC(COC)=O)=O)CC2)ccc(C)cc1C Cc1cc(C)c(C(=O)NCC2CC3CC3N2C(=O)C(C)Cc2ccco2)c(S)n1 C(=O)(CC(C)C(C)(C)C)NC1CCN(C(c2cc(C)cc(C(F)F)c2)=O)C(C)C1 c1(CC)cncc(C(=O)NC(CCOC)C(=O)N2CCC(CN(C)C)C2)c1 C(=O)(C(C)(C)C(=O)NC(CNC(=O)C(C)(C)CNC(C)=O)CC(F)(F)F)OCC C1(NC(c2cnc(OCC)s2)=O)CCC12CN(C(c1ncc(F)cc1F)=O)C2 N1(C(c2sc(C)c(Br)c2)=O)CCCC(F)(CNC(=O)C(C)C(F)F)C1 N1(CC)CCN(C(=O)NC2CCC(c3ccc(C)cc3)C2)C(C)(C)C1 c1(C(=O)NC2CC(C)(NC(C(C(C=C)C)C)=O)C2)[nH]cc2c1CCS2(=O)=O c1(C(=O)NCCCCCCNC(C2(C)COC(=O)N2)=O)cccc2nccn12 C1(CC)CN(C(c2csc(Cl)n2)=O)CCN1C(C1C2CC(=O)CC12)=O C=CC1(C(=O)NCCC(O)CCC)CCN(C(=O)C=Cc2ccoc2)CC1 Cc1ccc(C)c(C(N2CCC2(C)CC(=O)NCCC2CCCN2C)=O)n1 c1(-n2cc(C3(C)CCN(C(CC(CC)O)=O)C3)nn2)cnc(Cl)c(Cl)c1 c1(C(=O)NC2CCN(C(C3(C=C)CCC3)=O)CC2O)cn2cc(C)sc2n1 C1(C(N(C)CC2N(C(CCCOC)=O)CCC2)=O)CCCCC1C1CC1 c1(C(=O)NCCC2(O)CN(C(c3c(C)nc(O)s3)=O)C2)cc(C)c2n[nH]cc2c1 CC(C)(C)C(CNC(c1ccnnc1O)=O)C(=O)N1CC2CC2(CO)C1 CC(CC(N)=O)C(=O)N1CC(C)(NC(=O)C(C)Cc2ccc(F)cc2)C1 C1(NC(=O)NC(c2nc(C)[nH]n2)CO)COCC1(F)F c1(C(=O)NCCN(C(c2coc(O)n2)=O)CC)ccc2c(c1)CC(C)(C)O2 C1(CNC(c2ccc3ocnc3c2)=O)CC2COCC2N1C(c1ccoc1Br)=O N1(C(C2OCCN(C)C2)=O)CC(N(C)C(c2cn3c(n2)CCC3)=O)C(C)(C)C1 CN=c1ccc(C(=O)NC(CO)C(N2CC(O)CC2C(C)C)=O)c[nH]1 C#CC(C)(C)C(=O)NCCCC(C)NC(=O)C#CCc1ccccc1 N1(C(C(c2cn(CC)nc2)=O)=O)CCCOC(CNC(C2CCCC2(F)F)=O)C1 CCS(=O)(=O)CC(=O)N1CC2CC2(CNC(C2(C(N)=O)CC2)=O)C1 N1(CC(=O)N(CC)CC2C(C)C2(F)F)CCC(C(C)NC)CC1 C(N=c1nnn(C)[nH]1)C1CCCC(CNC(COc2c(C(C)C)cccc2)=O)C1 N1(c2cc(NC(C)C(F)F)nc(COC)n2)Cc2ccncc2C1 C(CCOCCO)(C(=O)NC1(C)CC(C)(C)C1)NC(C(F)=CCC)=O C1(NC(CC2OCC(C)(C)C2)=O)CC2CC1CN(C(=O)C=C1CCC1)C2 N1(C(C(F)=C(C)C)=O)CCCC12CCN(C(C1CC(=C3CC3)C1)=O)CC2 N1(CCC2C(C)(C)CCC2)CCN2c3ccccc3CCC2C1 Cc1cc(C)c(C(=O)N(C(C)CCNC(=O)C(C)OCCN(C)C)C)o1 C=CC(C)CC(=O)N(C(C)C(=O)N(C)Cc1cn(C)nn1)CC C1(CNC(C2C(C)CC(=O)N2)=O)CC(C)(C)CN1C(=O)CCF c1(OCCC#C)ccc(C(=O)NCC(O)CN(C(=O)CC2C=CCCC2)C)cc1 N1(C(CCS(N)(=O)=O)=O)CCC2C(CCCN2C(C2CC3(C2)CC32CC2)=O)C1 N1(OCCCCCCCCN(c2n(C)ccc2)CCO)CC2CC1C2N1CCNCC1 c1(NC(C(=O)NCC2(C)CC(C)(C)OC2)=O)cc2n(c1)CCOC2 Cc1ccn(C)c1C(=O)N(CCC(C)(C)NC(C1CC1(C)C(F)F)=O)C c12cccc(c1F)CNC2C.C1(N2CCOCC2)(C(F)(F)F)CCCCC1 N1(C(C(CC)N(C)C)=O)CC2CCC(CNC(c3cn(C)c(C)n3)=O)(C2)C1 C1(NS(C(C)C)(=O)=O)CN(C(=O)CCN2C(=O)C=CC2=O)CCC1O C1(C(N(CCC(=O)NCc2cc(C(C)C)on2)CC2CC2)=O)CCN(C)C(=O)C1 c1(OC)ccc(NC(C)C)cc1S(=O)(=O)Nc1c(F)cccc1Br N1(C(C(C)NC(CC)=O)=O)CCC(O)(CCNC(c2oc(CO)nc2C)=O)CC1 C1(CNC(CCCCC)=O)CC2(CCN(C(c3cccc(F)c3O)=O)C2)CO1 C(=O)(C(C(C)NC(=O)C1=C(C)OCC1)C(C)C)N1CCOCC(CC)C1 C1(NC(C(N(C)C(c2cnns2)=O)C2CC2)=O)CNC(=O)C12CC2 C(C(O)CCS(C)(=O)=O)NC(CC(=O)OCC)c1ccccc1 N1(C(c2cc(C)ns2)=O)CC=C(CCNC(=O)C(c2ccccc2)N(C)C)CC1 C1(C)(NC(CN(CCOC)C(C2CCOC(C)C2)=O)=O)C(C)(C)C1(C)C N1(C(C2CC2C(=O)Nc2c(CC)nc[nH]2)=O)CC2CC2(C(=O)OC)C1 c1(CC)cn2c(n1)CC(C(=O)NCC1CN(C(=O)C(C)Cn3cccn3)C1)CC2 C(CC(=O)NCCCCCNC(c1nnn2c1CCC2)=O)(C(F)(F)F)OC CC(CC(=O)N1CCOC(CNC(c2ccn(C(C)(C)C)c2)=O)C1)C(F)(F)F CC(CN=C(NCC(=O)NCC(F)(F)F)NCC1CCCCO1)c1cccs1 C(=O)(C(C(C)C)N(C(=O)C(CCc1ccc(F)cc1)N1CCCC(O)C1)C)OC C(=O)(C(COC)NC(=O)CC(C1CC1)C1CC1)NCCOCC(=C)C Cc1ccncc1C(C)NC(c1ccc(CNC(c2cnccc2C)=O)s1)=O N1(C(c2cnc(OC)s2)=O)CC2CCN(C(c3cc(C)c(C)c(F)c3)=O)C2C1 C1(CNC(c2cc(Cl)c[nH]2)=O)CC(F)(CNC(C23CC(CC(F)(F)F)(C2)C3)=O)C1 CCC(C)(C1CC1)NCc1nnnn1C(C)C.C12CC(C1)CCNC(=O)COC2=O C1(C(N2CCC(C(C)NC(c3nccnc3N)=O)CC2)=O)CCCCC(C)(C)C1 C1(F)(CNC(C2(CCCC)CC2)=O)CN(C(c2nnn(C(C)(C)C)n2)=O)C1 N1(C(CC(C)CF)=O)CCN(C(=O)CCc2ccccn2)CC1c1ccccn1 CCC(C)C(O)C(C)C(=O)NC1C2CC3C(C2)C13C(=O)NCC1CC2(CCC2)C1 c1(C(N2CCC3(NC(COCC)=O)C(C2)C3)=O)cncc2c1CCC2 N#CC1(C(N2CCC(CNC(C3CC3F)=O)CC2)=O)CCSCC1 C1(O)(CCNC(c2c(C)oc(Cl)n2)=O)CCCN(C(=O)CCC2CC2(F)F)C1 c1(CC)c[nH]nc1C(=O)NCCCN(CCCNC(=O)C(C)(C)NC(C)C)C C1(CC(=O)NCC(C)CN(C)C(c2nc(=O)n(C)[nH]2)=O)(CC)CCOCC1 N1(C(CC(=O)OC)=O)CCCCC(NC(C2CC(=O)NC2(C)C)=O)C1 N1(C(CC(=C=C)C)=O)CCC12CN(C(c1ccc(COC)cc1)=O)C2 c1(C(NON(C(=O)C(F)=CCCF)C(C)C2CC2)=O)cc(F)ccc1OC N1(C(c2cc(CCCC)oc2C)=O)C2CCC1CC(CNC(=O)CC1(O)CC1)C2 Cc1nccn1C(C)C(=O)N1CC(CC(C)NC(=O)CC2CCOCC2)C1 c1(C(N(C2CN(CC3CCCO3)C2)C)=O)cc(Cl)cnc1O.C12CCN(CC1)C2 c1(C(N(c2cc(Br)ccc2I)C)=O)ccnc2c1CNCC2 c1(OC)ccc(C(N2CC3(NC(=O)CN(C)C)CCC2C3)=O)cc1C C1(CCNC(CN(CCC#C)C)=O)CCN(C(=O)C(CO)N(C)C)C1 N1(C(C(c2ccc(C)s2)C)=O)CC(C2CCCN(C(=O)CN3CC(C)(C)C3)C2)C1 c1(C(C)C)ccccc1NC(=O)C(N1CCCC(c2cn(C)nn2)C1)C C#CCC(CC#C)C(=O)NCC(CNC(C1C(OCC)C1C)=O)CO c1(C(=O)NC2C3(CC(NC(C(COC)N(C)C)=O)C3)C2)cc2cccc(O)c2[nH]1 O=C(C1=CCCSC1)N1CCN(C(c2cnc(C3CC3)nc2)=O)C(CCO)C1 C1(NC(CSCCC)=O)CS(=O)(=O)CC1NC(c1cncnc1C)=O CC(N=c1[nH]c2c(c(=NCC3(Cl)CC34CCC4)[nH]1)CCC2)c1nc(O)n[nH]1 c1(C(=O)NCCC(C)N(C(C(C)NC(COC)=O)=O)C)cnccc1OC C(C(O)C(F)(F)F)NC(=O)CC1(CNC(=O)C(O)c2ccsc2)CC1 C(C(CC(C)C)C(=O)NC1CCC2(CC2)C1)NC(C(n1ncc(C)c1)C)=O c1(N2CCN(C(C3CCCC(NC)C3)=O)CC2)nc(C)ncc1I C1(C(=O)NC2CCC(NC(CC(CCSC)O)=O)CC2)CCc2ncnn2C1 CC1CC(C)(C(=O)NCC(C)(C)CN(C(=O)C=C2CCCC2)C)CCO1 N1(C(CCOCCC)=O)CCC2CN(C(=O)C(O)C(C)C)CC2C1 C(CN=c1nc(OC)cc(C)[nH]1)NC(C(C=C)(C)CC)=O N1(C(CC(=O)NC)=O)CCC(NC(c2csc(O)n2)=O)C12CCCC2 N(C1CCCn2ccnc21)C(C1N(C(c2cc(C)ncc2)=O)CC1)=O CC(C)(O)CC(=O)N1CCN(C2CCC(NC(C3CC3F)=O)C2)CC1 c1(C(N2CCC(NC(C(F)=C(C)C)=O)C2C(C)C)=O)cc(F)c(F)c(Cl)c1F c1(C(=O)NCC(CC)N(C)C(c2cnncc2OC)=O)cc(C)c(=O)n(C)c1 Cc1nc(C(=O)NC(C)CCNC(c2cc(-c3cccs3)[nH]n2)=O)n[nH]1 CC1(C)CN(C(C2CCCC2c2nc[nH]n2)=O)CC1C#N C1(CC(=O)OC)CS(=O)(=O)CC1c1nc(N2CCNCC2)no1 N#Cc1ccc(CC(CO)NC(c2nnnn2CCC2CC2)(C)C2CC2)cc1 N1(C(CC2(C)CC2(Cl)Cl)=O)CCCN(C(=O)CC2CCC2)CCC1 Cc1ccc(OC(C)C(N2CCC(N(C(=O)CSC3CC3)C)C2)=O)c(Br)c1 CCN=c1[nH]c(C)c(C(=O)NC(C)(C)CCCNC(c2cn3c(n2)CCC3)=O)s1 Cc1ncc(F)c(N2CCC(C(C)NC(c3ccccc3-c3nc[nH]n3)=O)C2)n1 O=S(=O)(c1ccc2[nH]c(=NCCC(O)C3CCCC3)ccc2c1)NCC(F)CO CS(C)(=O)=NC(=O)C(=O)NCC12CC(NC(c3cc4ccccc4[nH]3)=O)(C1)C2 c1(NC(=O)OCC(=C)C)cccc(NC(c2ccccc2C)C2CC2)c1 c1(CC)ccccc1CC(=O)NC1(CO)CN(C(=O)CCCN(C)C)C1.C(C)(=O)O C1(C(=O)NCC2(C)CC2)CC(F)(F)CN1C(c1cc(C2CC2)on1)=O.C1(CO)CC1 CC(C)(C)CC(O)C(=O)NC1CCC(NC(C2CC3(CCCC3)C2)=O)C1 c1(N2CC(C)C(CNC(c3cccc(C4CCOC4)c3)=O)C2)ccc(C#N)nn1 c1(C(C)=O)ccc(NC(C2CC3(CC3)CN2C(c2cnc(Cl)s2)=O)=O)c(C#N)c1 c1(C(N2CCC(CF)C2)=O)cccc2cc(-c3ccc(CO)cc3)[nH]c12 N1(C(C(F)=C(C)C)=O)CC(NC(c2oc(Br)nc2C(F)(F)F)=O)C(C)C1 O=C(CS(=O)(=O)CCO)NC1CC1NC(c1ccc(-n2cccn2)cn1)=O C1(NC(=O)CCc2ccco2)CN(C(=O)Cc2ccno2)CC1C1CC1 C1(OC)(CNC(C2(CO)CC(C)(C)C2)=O)CCN(C(=O)C=Cc2ccc[nH]2)CC1 c1(CC)ncc(C(=O)NC2(CCC(=O)NCCC3CCCO3)CCCC2)o1 C1(C(=O)NC(C)CN2CCCC2=O)(NC(=O)C=CC2CCC2)CCCC1C C1(C(N2CC(C(C(=O)NC3CC(C)(OC)C3)OC)C2)=O)CC(O)CCO1 N1(C(CC#N)=O)CCC(C2(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)CC1 N1(C(=O)CC2CCN(C(C3SCCS3)=O)CC2)CC2CCOCC2C1 C(=O)(CC(C(F)(F)F)NC(=O)C1=CCCCO1)NC(C1CC(CF)C1)C C#Cc1cccc(C(=O)N(C2CN(C(=O)C(C)NS(C)(=O)=O)CCC2C)C)c1F N1(C(c2cc(C)nnc2)=O)CC(C(=O)NC(C(N)=O)C2CCCC2)CC(C)(C)C1 CCC(C)(CCNC(c1[nH]cc(C)c1C)=O)NC(c1cnc(C)s1)=O CC(C)CC(F)(F)C(=O)N1CCCC(C(C)NC(=O)CSC(C)C)C1 Cc1cnc(NCC2(C)CCOC2)c(S(=O)(=O)NCc2c[nH]nc2C)c1 Cc1ccnc(C(N2CCC(C)C(CNC(=O)CC(=O)NC3CC3)C2)=O)c1O C(c1ccc(F)cc1)=C(C)C(=O)NCC(C)CNC(c1[nH]nnc1C)=O C1(CNC(C(CC=C)N(C)C)=O)CN(C(c2cnn(C)c2)=O)CCC1C N1(C(c2scc(C(N)=O)c2)=O)CCC(C2CC2)(CNC(C2CCCCO2)=O)C1 C1(NC(c2ccc(C(C)=O)[nH]2)=O)CN(C(=O)CCC(F)(F)F)CC(C)(C)C1 Cn1cnn(CCN2CCN(C(c3cccc(Cl)c3)Cc3ccccc3)CC2)c1=O C1(CC(=O)NC)CN(C(c2cncnc2)=O)CCN1C(c1cnc(C2CC2)[nH]1)=O CN1CC2(CCN(C(C3CCN(C(c4cccc(Br)c4O)=O)CC3O)=O)CC2)C1 Cc1cnccc1C=CC(N1CC(O)(CCNC(=O)C(CC)C(C)O)C1)=O c1(C(=O)NCC(CNC(C(CC2CC2)OC)=O)C)cncc2nc[nH]c12 N1(C(=O)NCC(=C)CC)CCC(NC(=O)CCN(C(=O)C(O)C(C)C)C)CC1 Cc1c(C(N2CCC(C)C2C(=O)NCc2cc[nH]n2)=O)cccc1C#N c1(C(N(CCCCN(C)C(C2(C)CCCO2)=O)C)=O)cc(F)ccc1S(C)(=O)=O C(N=c1[nH]c(N2CCc3c(nnn3C)C2)nc2c1COCC2)C1OCC(C)C1 c1(SC)ccc(NC(=O)C(c2cccnc2)NC(c2nc(=N)cc[nH]2)=O)cn1 C1(C(=O)NC2(C)CN(C(C(COC)N(C)C)=O)C2)CCCN(C)C1 N1(C(c2cccc(C)c2F)=O)CCC2CN(C(c3cc(C)n(C)n3)=O)CCC2C1 C1(N(C(C2CCCN(C(=O)CC3(OC)CCC3)C2)=O)CC)CCOC(C)(C)C1 c1(C(=O)NC2CCN(C(C(C3CC3)OCC)=O)CC2)ccc2[nH]cc(C#N)c2c1 C1(Cl)(C(=O)NC2CC(CNC(c3c[nH]nc3C(F)(F)F)=O)C2)CC12CCOCC2 N1(c2n(CC3CC(CC)C3)nnn2)CCC(c2ccccc2C)CC1 C1(CC)C(C)CCN1C(=O)CC1C2CN(C(c3coc(CC4CC4)n3)=O)CC12 N1(C(Cn2cc(C(C)O)nn2)=O)CCCC(NC(C2COCCO2)=O)C1C CCC(CC)C(C)C(=O)N(C1CCCCC1NC(=O)Cc1c(C)nn(C)c1Cl)C C(CN=c1nc2c(ncn2C(C)C)c(N2CCC(F)CC2)[nH]1)OCC(=C)C c1(C(=O)OCc2ccc(Cl)c(C)c2NS(C)(=O)=O)c(C)sc2ccc(Br)cc12 C1(C(=O)NCC(CNC(C(C)(C)NC(=O)OC)=O)C)CN2CCN1CC2 Cc1cnc(Cl)nc1N1CCOCC(NC(C2C3CCCC23)=O)C1 C12CCN(CC1)C(=O)C(C1CCCCC1)OC2=O.O(C=CC(=O)NCC)CC C(=O)(CS(=O)(=O)C(C)C)N(C1CN(C(c2nc(OC)c(F)cn2)=O)CC1(C)C)C c1(C(N(CC(C)NC(c2cocn2)=O)CC)=O)cc(C(N)=O)cs1 C1(NC(c2ncccc2Oc2ccccc2)=O)CCCCN(C(=O)C=C(Cl)Cl)C1 N1(C(c2c(C)non2)=O)CC2(CCCC2CC(=O)NCC(N)=O)C1 N1(C(C2CCC(C)O2)=O)CCc2ccccc2C1CNC(C1(O)CCSC1)=O C1(CNC(c2ccc(OC)s2)=O)CCN(c2ccnc(COC(C)=O)n2)C12CC2 N1(C(=O)Nc2cc(-c3ccccc3)ccc2[N+](=O)[O-])CC(O)C2(CCOCC2)C1 C(=O)(C(O)CCCNC(C1CC2CC(=O)C1C2)=O)NCCCC(C)(C)C CC1CN(C(=O)OC(C)(C)C)CCN1C(=O)C(c1ccccc1)Nc1cccs1 c1(C(=O)NC2C(C)CN(C(c3cnsc3)=O)CC2C)cc(O)c2ccsc2c1 C(CC(C)(C)C(=O)N1CC(CNC(=O)CCc2nnc(C)n2C)C2(CC2)C1)OC c1(NC2(C)CC(NCc3ccc(F)cc3)C2)ncc2cccc(O)c2n1 N1(C(c2cc(CN(C)C)on2)=O)CCCC(F)(CNC(c2snc(O)c2Cl)=O)C1 c1(C(=O)NCC2C(NC(c3c(C)oc(C)c3C)=O)C2)ccc2c(c1)CNC2=O Cc1cc(O)c(N(C)C)cc1CNCC(O)(CO)CO CC(C)C(C)(C)C(=O)N1CCCC1CNC(C1(c2cccc(F)c2F)CC1)=O N1(C(CC(=O)OC)=O)CCCCC(NC(=O)C(c2csc(C)n2)=O)C1 CC(O)C(F)(F)C(=O)NCC(CNC(C1SCCCS1)=O)C(F)(F)F N1(CCCC)CCOCC1C(=O)N(CC(C)O)CCNC(=O)C(F)(F)C1CC1 C1(CNC(C2(C(=O)NC)CCC2)=O)CC2(C1)CN(C(c1nnn(C)c1C)=O)C2 C1(NC(C=C(C)Cl)=O)CN(C(c2ccnc(C(C)(F)F)c2)=O)CC1C C1(C(C)OC)CN(C(=O)C(C)SC)CCN1C(=O)CC1CCN(C(=O)OC)CC1 CCCC(CCC)C(=O)Nc1ccc(C2CC2)cc1 C(CC(=O)NCCc1ccc(O)cn1)(C(F)(F)F)NC(c1c(C)c[nH]n1)=O c1(C(N2C(C(=O)NC(CCSCC)CO)C(O)CC2)=O)ccc(Br)nc1F Cc1cc(CC(=O)NCC2CN(C(C3CCNC3=O)=O)CCO2)ccc1Br c1(C(N(C2CCCN(C(=O)C(C)(C)N3CCCC3)C2)C)=O)cnccc1Cl C12(NC(=O)CCC3CCOCC3)COC(C1)C(NC(c1ccc([N+](=O)[O-])o1)=O)C2 c1(N(CC=C)C)nc2cccnc2c(=NCCCOCCCC)[nH]1 C(=O)(C(C(C)C)NC(=O)Cn1nnnc1C)N1C(CCCC)CCC1 Cc1ccc(C(C)C(=O)N2CC(N(C)C(C3CCOC3C)=O)C2)cc1 c1(C(=O)NC(CCOC)CNC(=O)CC2CC=CCC2)ccc(C(N)=O)cc1 Cc1cnc(C(N2CC(NC(=O)C(F)CC3CC3)CC2C)=O)c(O)c1 c1(C(N(C2CCN(C(C3(C(C)(C)C)CCC3)=O)C2)C)=O)c(F)ccc2occc12 N1(C(C2COCC2C(F)F)=O)CCN(C(=O)Cc2cscn2)C(CO)C1 N1(C(C2C(C(C)(C)C)C2)=O)CCC(NC(=O)Cn2nnc(C3CC3)n2)C(C)(C)C1 N1(c2nc(SC)c(C)cn2)CC2CCC1C1CN(C(=O)Cc3csnc3C)CC21 C1(C)(CCC(=O)NCCC=CCCC)CN(C(c2ccc(C)o2)=O)C1 N1(C(C(C)C2CC2)=O)CCCN(C(=O)COCc2ccccc2)C(C)C1 C12(N(C)C)CCC(C(N3CC(NC(=O)C(C(C)(C)C)NC(N)=O)C3)=O)(CC1)CC2 c1(CN(C)Cc2cn(C)nn2)cnccc1-c1ccccc1 S(=O)(=O)(c1ccc2c(c1)CC(=O)N2C)Nc1c(C)ccc(=O)n1C C1(NC(c2cc(OC)ncc2)=O)CC2CC(NC(C3(OC)CCOCC3)=O)CC12 C1(C(=O)NC2CCCOC2)(NC(c2ccc[nH]2)=O)CCCC1 c1(OCC(N2CC(CN(C(C3CCC(C)(CC)O3)=O)C)C2)=O)c(C)cccc1C c1(OCC)nc(N(C)CC2CCCCN2C(c2occ3c2CCC3)=O)ncc1C C(=O)(CC(O)C(Cl)(Cl)Cl)NCCCCNC(c1cc(C(=O)OC)c(C)cc1)=O c1(C(=O)NC2C(NC(C(CCC)NC(C)=O)=O)C2)ccc2nc(C)oc2c1 C(=O)(C(C)C(F)(F)F)N1CCC(C(=O)NCCCP(C)(C)=O)(CC)C1 Cn1nnnc1SCC(=O)NCCN(C1CCCCC1)C(=O)Cn1ncnn1 C1(CC(=O)NOCC2CCCO2)CCCN(C(=O)C#CC2CC2)C1 CC1CCCC=C1C(=O)NCCc1ocnc1CNC(C1(n2cccn2)CC1)=O C1(C)(C(N2CC(C(=O)N(C(c3ccno3)C)C3CC3)OCC2)=O)CCN(C)CC1 c1(C(=O)NCC(CC)NC(=O)CN2CCOCC2=O)cc(C2CC2)oc1C1CC1 C1(OC)CCN(C(=O)Cn2cc(OC(C)(C)C)cn2)CC1C.C(C(=O)OC)N C(C(C)N=c1nc2scnc2c(NCC(Br)=C(C)C)[nH]1)OCC N1(Cc2ccc(C(C)C)cc2)CCC(C)(C(=O)NCC2CCC(=O)N2)CC1 N1(C(=O)Nc2c(C)con2)CCN(C(CO)CO)CC1 C1(C)(NC(CC2CCCC(OC)C2)=O)CCN(C(=O)Cc2cncn2C)CC1 C1(CCNC(c2c(OCC)ccs2)=O)CCN(C(=O)C2=CCC2)C(C)C1 C1(CNC(Cc2c(C)cccc2)=O)CCC12CN(C(c1cn(C3CC3)nn1)=O)C2 CC1CCNCCC1N(C(=O)CCSC1CCCN1C(=O)OC(C)(C)C)C1CC1 C1(C)(NC(c2n(C)nc(C(N)=O)c2)=O)CCN(C(=O)CC2CCCCCCC2)CC1 N1(C(c2c(C)ccc(Br)c2)=O)CC2CC1CCC2NC(=O)COC1CCC1 c1(C(=O)NC2CN(C(C(C)Oc3ccccc3Cl)=O)C2)n[nH]c2c1CC(C)CC2 C1(C(=O)N(C2C(=O)NCCC2)C2CCC(O)C2O)CCC(C2CC2)C1.C1(O)CCCCC1 C1(C(N(CCNOCC2COCCOC2)C)=O)(C(=O)OC(C)(C)C)CC2CCCC12 N1(C(c2cnc(CC(C)(C)C)s2)=O)CCN(C(=O)C=C2CCCC2)CC1CO C(=O)(C(C)S(=O)(=O)c1ccc(F)cc1)N1CC(O)(C(C)NC(CC(C)C)=O)C1 N1(C(c2cnn(CC)c2Br)=O)CC2CCC1C(CNC(C1COC1)=O)C2 CCC(O)C(F)(F)C(=O)NCCOC(C)(C)CNC=O.C1(C2CC2)CCCCC1 c1(NC(C2CCN(C(C3(C(C)C)CCC3)=O)CC2O)=O)c(Cl)cc(Br)c(Cl)c1Br CC(C)CCC(C)N(C(=O)Cn1cc(CNC(C2(C)CC(C#N)C2)=O)nn1)C CCC(C(=O)N1CCN(C(c2cn3c(n2)CCC3)=O)CC1CC(=O)NC)C(C)C c1(-n2c(-c3c(OC(=C)C(=O)OC)cccc3C)ncc2)nc(Cl)c2c(n1)COC2 C(=O)(CC(C(F)(F)F)P(C)(C)=O)N1C(C(=O)OC)CC(n2cc(CCO)nn2)C1 C1(NC(C2(CCN(C)C)CC2)=O)CC(C(=O)NOCC(F)(F)F)CC1O C(=O)(CCC(C)C#N)N(CCNC(=O)C(c1ncc(Cl)n1C)(C)C)CC C(=O)(C1OCCc2c(O)cccc21)N(C)CC1CCN(C(=O)CC(C)(C)O)CC1 c1(C(=O)NC2CC3CN(C(CNC(=O)NC)=O)CC32)ccc2cc[nH]c2n1 C1(N(C(=O)C(F)OC(F)(F)F)CCC)CCN(C(=O)CNc2cnn(C)c2)C1 C12(C(=O)NC3C(NC(C4(CC#C)CC4)=O)CCOC3)CCC(N=[N+]=[N-])C1C2 C1(CCCC)(C(=O)NC2(CC(=O)N(C(C)CN(C)C)C)CC2)CCC1 O=S(=O)(c1ccc(CC(F)(F)F)cc1)NCC1CC2CCCCC2N1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(CN(C(CN(CCC)C)=O)CC)C1 N1(C(C2CCC(CNC(C3(OCC)CC3)=O)O2)=O)CC2CCCC2C1 C(=O)(CCC(=O)CC)NC(CCOCC)C(=O)N(C)CCC1CCCN1C c1(CNc2c(C)cc(C(N3CN(C(C)C)CC3C)=O)cn2)ccc2sccc2c1 CC(CCCNC(=O)C(C)CO)NC(c1cnn(C2CC2(F)F)c1)=O c1(OC)ccc(Cl)cc1CC(=O)NC1COCC1NC(C1(C)CC1(C)C)=O N1(C(C=CC)=O)CC2(CCCC(CNC(c3cc(-c4ccccn4)[nH]n3)=O)O2)C1 N1(C(=O)CCc2ccc(C(F)F)cc2)CC2CCC(C1)N2C(=O)CC(F)F c1(CC)nc(C(C)NC(=O)CC2CCCC2NC(C2CCC2(F)F)=O)no1 c1(OCC)ccc(CC(=O)N(CCCCNC(=O)NC2C(C)CC2C)C)cn1 C1(C(N(CC(C)OC)C)=O)CN(C(=O)C(F)OC(F)(F)F)CC(C)(C)C1 O=S(=O)(c1ccc(N2CCC(Cc3ccccc3)C2)nc1)NCCN1CCCC1 CC1(C)CN(C(C2CCC3(CCC3)C2)=O)C(CNC(c2cnc[nH]2)=O)CO1 C1(NC(C(C)OCCOCC)=O)C2CN(C(=O)C(C)(O)c3ccccc3)CC12 n1(CCC(=O)NCC2N(C(c3nc(C)n(C)c3)=O)CCCC2)cc([N+](=O)[O-])cn1 CC(C)CCCC(C)NC(=O)CCSCc1ccc(Cl)s1 N1(C(c2ccc(SC)o2)=O)C2CCCC1CN(C(=O)CC(C)(C)C(F)F)CC2 C1(CNC(C(C)=C2CCCC2)=O)CN(C(c2cc(Cl)ccc2O)=O)C(C)(C)C1 C1(C)(CCC)CCN(C(c2ccnc(CNC(=O)Cn3cccn3)c2)=O)C1 C1(C(N)=O)CCN(C(C2(NC(c3ccnnc3O)=O)CCCCC2)=O)CCO1 c1(C(=O)NCC2OCCN(C(CC=CCC)=O)C2)ccc(I)c(F)c1 c1(C(N(C(C)CNC(=O)C(C)O)C)=O)ncn2cc(Br)sc12 C(=O)(CCCCF)NCCC1ON=C(C)C1 CCC(C)(C)C(O)C(=O)NC(C)CCN(C)C(c1ccc(=O)oc1)=O c1(CC(=O)OCc2nc(Cc3ccccc3)cs2)coc2ccc(Cl)nc12 C(=O)(CC1=CCCCC1)N1CC(C)(C(=O)NCc2c(C)nco2)C(C)C1 C12(NC(c3ccc(CCC)cc3)=O)CCC(CC1)N(C(=O)C(CC)(CC)OC)C2 C1(O)(C(C)NC(C=CC(C)C)=O)CN(C(=O)C(c2ccccc2)NC(N)=O)C1 c1(NC(c2csc(NC(c3ccsc3)=O)n2)=O)cccc(S(=O)(=O)O)c1 Cc1ncc2n1CC(C(=O)NC1CCCN(C(=O)Nc3ncns3)C1)CC2 C(=O)(C(O)C(F)(F)F)NC(CSC)(C)C(=O)N(CC(=O)NC(C)C)C Cc1cnc(NCC(C)C)c(S(=O)(=O)N2CCCC(C(F)(F)F)C2)c1 CC(C)CCCC(=O)N1CC(C2CCCN2C(=O)C(O)CC)C1.C12(N)CCC(C1)OC2 c1(NC(N(C2(C)CN(C(=O)OCC3CCO3)C2)C)=O)cc(F)cc(F)c1 N1(C(C2C(F)(C(=O)OCC)C2)=O)CC2CC2(CNC(C2(CO)CCCO2)=O)C1 C12(NC(=O)Cc3cccc(O)c3)COC(C1)C(NC(C1CCCC13CCC3)=O)C2 N1(CC(C)NC(C2CC2C#N)=O)CCN(C(c2cccc(=O)o2)=O)CC1 C(=O)(C1CCc2c(Cl)cccc21)N1C(CNC(c2cnc(O)o2)=O)CC2CC21 C12(CCCCC1)C(=O)N1CCCC(C1)c1cn(nn1)C2.c1(SN)cnn[nH]1 CCC(F)(C(=O)OC)C(=O)NCC12CCCC1CN(C(c1cc(C)ccn1)=O)C2 c1(OC)ccccc1C1CCCN1c1nc(C(=O)OC)c(C)s1 c1(N(C(=O)COCCC(C)C)CC)cccc(-c2c[nH]c(=N)s2)c1 C1(NC(CCSC)=O)CCN(CCNC(=O)CCc2cccnc2C)CC1 C1(C2CN(C(C(C)CC3CC3)=O)C2)CN(C(C2CC2c2nc[nH]n2)=O)CCO1 C1(NC(=O)CSCC(F)F)CCC(C)(OC)CC1.c12ccc(cc1)n2CC.C1CC1 S(=O)(=O)(c1ccc(C)c(C)c1)NCCOC(C(C1CC1)OC)=O.c1ccccc1 C1(C)(NC(N2CC(C(=O)NC(Cn3ncc(C)c3)C)C(F)C2)=O)CCN(C)CC1 S(=O)(=O)(C1CCCCC1)N1CCC(N(C)C(C2(Br)CC2(F)F)=O)CC1 N1(C(C(CC)OC)=O)CCC(C2CC2NC(=O)Cn2cc3ccccc3n2)CC1 C#CCC(C(=O)OCC)NC(=O)COC1CC(NC(C2CN(C)C(=O)N2)=O)C1 c1(CCC(=O)N(C(c2ccccc2)Cn2cccc2)C)nccn1C C(c1cc(C)ccc1OC)=CC(=O)NC(c1cc(OCC)cc(F)c1)C(=O)O C(=O)(CC(CN(C)C)C(F)(F)F)N1C(C)CN(C(=O)CSCC(F)F)CC1 C(=O)(C(CNC(=O)C(c1cnn(C)c1)O)C(C)C)N(CCC#C)C N1(C(C(C(C)C)SC)=O)CC(CNC(c2coc(SC)n2)=O)C(F)(CO)C1 C(=O)(CC(C(C)C)NC(c1ccncc1)=O)NCC(C#C)(C)C CC1CCC2(CC2)N(C(c2c(CNC(c3ccc(CO)s3)=O)nnn2C)=O)C1 CCC(C(=O)OC)C(=O)N1CC(F)(F)CC1CCNC(=O)Cn1ncc(Cl)c1C C=CC(C)CCNC(C1(C(C)NC(C2CC(F)C2)=O)CC1)=O C(CCC(=O)NCc1nc(C(=O)N(C2CN(C)C2)C)co1)OC(C)C c1(C(N2C(C)CC(NC(c3nn(CC)c(C)c3)=O)C2)=O)ccc([N+](=O)[O-])o1 C1(NC(=O)CC2CCOCC2)CCN(C(C2CC2c2ccccc2)=O)CC(O)C1 c1(C(=O)NC2CC(CCNC(c3[nH]cc(C)c3)=O)C2)sc(CC(F)(F)F)nc1C Cc1cc(N(CCCNC(=O)CCCCCF)C)n2ncnc2n1 C1(N(C(C=CCN(C)CC)=O)C)(C(N2CCC(CF)C2)=O)CCS(=O)(=O)C1 N12CCN(C(C)C1)CC2.c1(C(=O)OC)cccn1SC(F)(F)F c1(C(=O)NC2CN(C(c3c(C)cnnc3)=O)C(C)C2)ccc2c(c1)CCCCN2 c1(CNC(=NCCC)NC(c2ccnn2C)C)ccc(S(=O)(=O)N(C)C)cc1C C1(C(=O)NCCN(C(=O)Cc2cnns2)CCOC)CC=CCC1C C1(NC(CCCCCOC)=O)(CNC(C2CC2OC)=O)CCC(C)(C)CC1 CC(C)CS(=O)(=O)CC(=O)NCCCCNC(=O)C(c1cc2ccccc2o1)C C(CNC(=O)C(C)(F)F)(C(C)(C)C)NC(C(c1ccccc1)C)=O C(=O)(C1=CCCCO1)N1CCC(O)(CCNC(c2c(C)c(C(F)(F)F)n[nH]2)=O)C1 c1(C(=O)NC2CCN(C(c3c(N)cccn3)=O)CC2CO)c[nH]c2cccnc12 C(=O)(N1CC(O)CCO1)C1(CCCN)CCCC1.CC(C)(C)OC(N)=O c1(C(=O)NC2C(CC)N(C(=O)CCCOC(C)C)CC2)ccn2ccnc2c1 C1(NC(=O)COC2CCCOC2)CC2(CCC(NC(c3cncnc3)=O)CC2)C1 N1(C(CCn2c(C)ncc2)=O)CCN(C)CC1C(=O)NOCC1CCCC1 c1(NC(=O)NC(C)CNC(C2(CN(C)C)CC2)=O)cc(F)c(Cl)cc1F c1(C(=O)NC2CCN(C(C=C3CCC(C)CC3)=O)C2)ccnc2ccncc12 Cc1nc(C2CCCN(C(C3CN(C(c4ccccc4)=O)CCO3)=O)C2)[nH]c1C Cc1cncnc1C(=O)NCC1CC1CC(=O)NCC1CC(O)C12CCC2 C=C(C)CC(C(=O)N1CC(C)(C(=O)OCC)C1)NC(=O)C(N1CCOCC1)C C1(NC(C#CC)(C)C)CCN(C(=O)C(CC)OC)CC1 c1(CNC(c2c(NC(=O)CC3CC3C3CC3)c[nH]n2)=O)cc(Cl)ccc1Cl C1(NC(C=C(CC)C)=O)CCC(CNC(c2ncoc2-c2cnn(C)c2)=O)C1 N1(C(C(C)(C)NC(c2ccc(Cl)cc2)=O)=O)C2CCC1CSC2 c1(C(=O)NC2CCN(C(c3c(C)[nH]c(=N)s3)=O)CC2F)ccc2c(c1)CCOC2 c1(C(C(=O)NC(C)C(=O)N(CC(C)(C)O)C2CC2)C)ccnn1C Cn1c(C(N2CCC2CNC(C2CC(CCO)C2)=O)=O)cc2c(O)cccc12 C1(C(=O)C(C2CCCO2)OCCOC)(NC(C=CC(C)(C)SCC)=O)CCCC1 C1(CC)(CC)CCCN1C(C1COC(CNC(=O)CCCn2cccn2)C1)=O C(C)(CSC)(C(=O)NCC(c1cnc[nH]1)C)NC(CCSC)=O N1(C(c2c(OC)ccnc2)=O)CCCCC(NC(c2cn[nH]c2)=O)C1 C1(C)(CN(C2CCSCC2)CC(=O)N(C(C(C)C)c2nn[nH]n2)C)CCCCC1 C1(C(N2CC(C)C(C)C2C)=O)CC12CCN(C(=O)CC1C=CCCC1)CC2 c1(C(N2CCC(NC(c3ccc(C(N)=O)[nH]3)=O)C2)=O)cncc(Br)c1 N1(C(Cc2c(C)nc(S)s2)=O)CC2(CCCC2NC(C2CC2C(C)O)=O)C1 c1(CC(CC)C)nc(-c2cnsc2)n(C2COC(C)(C)C2)n1 C1(C(C(=O)NCCC(=O)OC)N(CCC(C)(C)C)C)C2CCCCCC12 Cc1nn(C(C)C)c(C)c1NC(=O)C(N1CCCC(Cc2cccc(Cl)c2)C1)=O c1(C(=O)NC2C(CNC(CC(C)c3ccncc3)=O)C2)cccc2c1CCN2 N1(C(CSCCC(C)C)=O)CCC(c2n[nH]c(CNC(=O)CC3CC3C)n2)CC1 C(CCCCC(=O)NCC(CO)C(F)(F)F)N(C)C(c1ccco1)=O CC(C)S(=O)(=O)CC(=O)NC(c1ccccc1)CNC(c1cc(Cl)c(Cl)[nH]1)=O C1(C(F)F)(N(c2cccnc2)c2nnnn2-c2ccccc2)CCCCC1 c1(N2CCC(N(C(c3c(CC)scc3)=O)CC)C2)ncnc2cccc(OC)c12 N1(C(Cn2c(C)nnn2)=O)CCC2CC1CN(C(C1CC3CCC(C1)C3O)=O)C2 CCC(O)C(C)(C)C(=O)N1CCC(C(=O)NCC2(CO)CC23CCC3)O1 O(NC(=O)C(CCF)NC(=O)C=Cc1cncs1)CC(=O)N(C)C C1(NC(C(=O)C(Cc2c(NCC)cc(C)nc2)=O)=O)CC(C)CC(C)C1 c1(CC(N2CCC(C)(NC(C3C(OCC)C3)=O)C2)=O)c(F)c(F)cc(F)c1F c1(C(=O)NCC2CN(C(CC)=O)C2)sc2ncc(C(=O)OC)cc2c1C Cc1nc(C#N)cc(=NCC2CCCCN(C(c3cccc(O)n3)=O)C2)[nH]1 C1(OC)(CNC(=O)CC2CCC(C)(C)C2)CCN(C(C2CC3(CCC3)C2)=O)C1 C(=O)(C(C)(CC)CO)NCC(C(C)C)NC(CC=CC)=O CC1(C(N2CCOCC(CNC(C3C=CC=CC=C3)=O)C2)=O)CCNC(=O)C1 C1(NC(c2c(NC(C)=O)ccc(F)c2)=O)CC2CN(c3ncncc3I)CC2C1 C(=O)(CCCCC(=O)N1CCN(C(c2cnc(OC(C)C)cn2)=O)C2CC12)OC C1(C(=O)NCC=CCNC(=O)CC2CCSCC2)CCc2nc[nH]c2C1 [N-]=[N+]=NC1CCC(NC(C2(CO)CN(C(=O)C(=O)N(C)C)C2)=O)CC1 C12(C(=O)NCCCOCCN(C(COCC(C)C)=O)C)CCCC1C2Br c1(-n2cc(CN(C)CC=Cc3ccnn3C)nn2)ccccc1C(=O)O C=C1CCN(C(c2cc(CC)n(C)n2)=O)C(C(=O)Nc2cn(C)c(=O)nc2O)C1 N(C1CCCc2c(F)cc(Cl)cc21)C(CCCNS(N(CC)CC)(=O)=O)=O c1(C(=O)NC(CN(C(c2cc(O)n(CC)n2)=O)CC)C)cccc(F)c1C C1(N(C(C(C)SC)=O)C)CCCN(C(=O)Cc2ccc(OCC(F)(F)F)cc2)C1 N1(C(CSCC#C)=O)CCC(CC(=O)NCC=CCCOC)C1 O(N(C)C(=O)CNC(=O)C(C1CCN(C(=O)CCc2nccn2C)C1)F)CC C1(COC(CC2(C=C)CCOCC2)=O)CCC2(CCCC2)C1 C#CC1(C(=O)NC2CCCCC2CC(=O)NCCc2ccco2)CCCC1 C1(NC(=O)C=Cc2ccoc2)CN(C(C2CC2F)=O)CC(F)(F)C1 N1(C(c2cccc(OC)c2)=O)C2CCC1CC(N(C(=O)C(C)(O)C1CCC1)C)C2 c1(C(=O)NC2CCC(N(C)C(C3CC(N(C)C)C3)=O)CC2)c[nH]cc(F)c1=O C1(CNC(c2cncc(N)n2)=O)CN(C(C2(Cl)CC23CCC3)=O)CCCO1 C12(NC(CCC=CC)=O)CC(CNC(=O)C(Cc3ccccc3)CC)(C1)OC2C c1(C(=O)NCc2nc(C)sc2)cnn2cc(-c3ccc(O)cc3F)ccc12 c1(C(=O)NC2CC3CC(NC(CCC)=O)C2C3)cnc2c(C#N)cnn2c1 C(=O)(C(C)(CCCF)N(C(=O)CSC)C)NC(c1ccncc1)CC C(c1ccccc1F)=CCC(=O)NCC1C(NC(=O)C=C2CCC2)CCCC1 N1(C(c2cc(OC)c(F)c(F)c2)=O)CCCC(N=c2ccnc(C3CCC3)[nH]2)C1 CC1(C(N2CCC(c3ncco3)C2)=O)CCCN(C(C2CNC(=O)N2)=O)C1 C1(CC(=O)OCC)CCC2(CC1)CCN(C(c1cccc(Br)c1)C(N)=O)CC2 C1(CNC(CSC)=O)COCC1n1cc(CNC(=O)CCC2CCC(C)O2)nn1 C1(C(c2c(C#C)cnn2-c2ccc(NC(=O)CS(=O)(=O)C3CC3)s2)=O)CCc2[nH]nc(O)c2C1 C1(NC(CCCNC(N)=O)=O)COCCN(C(C2CCC=CCC2)=O)C1 N1(C(N(C(CC)(C)CO)c2ccccc2)=O)CCOC(C)C1CO C12(C(N3C(CCC)SCC3)=O)CCCCC1(CO)CNC2 C(=O)(C(C)C1=CCCC1)NCCC1CCN(C(c2c(C)c(N)cnc2)=O)CC1 C1(CNC(C2(C)CCN(C(C)=O)C2)=O)CCN(C(=O)Cn2cnnc2)C12CCC2 N1(c2n(CCC3(COC)CC3)nnn2)CCc2c(C)cnc(O)c2C1 C1(OCC)CC(c2nc(C3C(C4CC4)C3(F)F)no2)C12CCC2 N1(C(c2ccn(C(C)C)n2)=O)CC(CNC(c2cn(C)nc2C2CC2)=O)CC1C c1(C(=O)NCCCC(C)NC(C(F)=C(C)C)=O)ccc(=O)n(C2CC2)c1 C(=O)(C(C)(C)C(=O)NC1CCCCC1C(=O)NCCC(O)CO)OC C12(CNC(c3cccc(=O)o3)=O)CCC1CN(C(C1CCC=CCC1)=O)C2 N1(C(C(Cc2cnc[nH]2)NC(c2c(C)nns2)=O)=O)CCC(O)CC(C)(C)C1 C1(NC(=O)Cc2nc(C3CC3)cs2)C2COCC1CN(C(=O)C1=COCCC1)C2 C12(CNC(C3CCC(CNC(c4nc[nH]n4)=O)C3)=O)CCN(CC1)C2 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC2C(C1)NC(=O)CN2C(=O)C(C)COC CCC(CC1CCCCC1)C(=O)N(C)CC1CCCN1C(=O)COC(C)C C1(CNC(Cc2nc(C)sc2)=O)CN(C(=O)Cc2ccc(O)nc2)CCO1 C1(N(C(=O)CCC(=O)N(C)Cc2ccccc2)C)CS(=O)(=O)CC1O C1(C(=O)NCC(CO)NC(c2c(N)ccc(C(C)C)c2)=O)CCCC(F)(F)CC1 CCCC(C)(CC)C(=O)NC1CC2CN(C(=O)C=C(C)c3ccco3)CC12 CCCCC(CC(=O)N1CC=CC1(C)CO)NC(=O)CC(C)(C)C N1(C(c2n[nH]c(C)c2Br)=O)CCCC(CCNC(C23CCC2C3)=O)CC1 N1(C(C=CC)=O)CCC(NC(c2cc(Cl)ccc2Br)=O)C(CO)CC1 c1(C(=O)NCC2C(CNC(C(CC)=CC)=O)C2(F)F)ccc(C)nc1N C1(OC)CC(NC(=O)CSCC(c2ccc(Cl)cc2)C)CN(C(=O)C(C)OC)C1 N1(C(c2c(C)cc(CO)o2)=O)CCOC2(CCN(C(C3(CO)CCCC3)=O)C2)C1 N1(C(CSC(C)C)=O)CCN(C(=O)C(C)(O)c2ccccc2)CC1C C1CN=C2NC(C)=CC(=NC3CC3CO1)N2.c1(OC)cccc(C(C)(C)C)c1 CC(C)CC(C)(O)C(=O)N(C)CC1CCN(C(=O)C=Cc2cn(C)cn2)C1 c1(SC(C(=O)N(CCNC(C2CC(OC)C2)=O)CC)C)ccccc1Cl C=CC(C(=O)NC(C1CCCO1)C(=O)NCc1cc(C(N)=O)co1)OC c1(C(N(CC(CN(C(c2c(C(=O)OC)c[nH]n2)=O)C)O)C)=O)cc(C)cc(C)c1 Cc1nccc(Cl)c1C(=O)NCCN(C(=O)C(F)C1CCOC1)C C#Cc1cncc(C(=O)NC2CCN(C(C3CCN(C)CC3)=O)C23CC3)c1 c1(C(N2CCCC(CNC(CCCC(N)=O)=O)C2)=O)ccc(Cl)c(Cl)c1N Nc1ccc(C(=O)NCC2CCCC2NC(c2ccnnc2Cl)=O)cc1O N1(C(C(=O)N(C(CCCC)C)c2ccccc2)=O)CC(C)OC2(CCCC2)C1 c1(C(=O)NC2CCN(C(c3cnc(C)n3C)=O)C(C)C2)cc(Cl)cc2c1CCC2 Cn1c(C(=O)N(CCNC(C2CC3(CCC3)CO2)=O)CC2CC2)ccc1[N+](=O)[O-] c1(CNC(C(C)C(C)(C)C)c2n(CCCSC)nnn2)cc(C)c(F)c(C)c1 C(=O)(C1=CC2(CCOC2)C1)N1CC(C)C(CNC(C2CC2c2cnn(C)c2)=O)C1 N1(C(C2(COC)CC2)=O)CCC(C)N(C(=O)Cn2[nH]cnc2=N)CC1 C1(NC(c2ccc(OCC)nc2)=O)CC(C)CN(C(C2CC3C=CC2C3)=O)C1 C(=O)(C1COc2ccc(F)cc21)NCC1(O)CN(C(C(CC=C)CC(C)C)=O)C1 N1(C(c2c(SCC)cccn2)=O)CCOC(C)(CNC(=O)C(C)(CO)OC)C1 N#Cc1c(NCCCCNC(c2cscn2)=O)nnc2c1CCCC2 C1(CNC(CCNC(c2ccoc2)=O)=O)CCCN(C(C2CCCO2)=O)C1 N1(C(c2cc(C(N)=O)[nH]c2)=O)CCOCC1CCNC(=O)CC(F)(F)F C1(C(N(CC(C)NC(c2coc(N(C)C)n2)=O)CC)=O)CCC(C(C)C)CC1 N1(C(CCC#CC)=O)CCN(C(=O)C(C)Sc2nncn2C)C(CCO)C1 C=C(C)C(C)(O)C(=O)NCC(C1CC1)NC(c1ccc(F)cc1SC)=O Cc1ccc(N)c(C(N2CCCC2C2CCN(C(=O)C(C)S(N)(=O)=O)C2)=O)c1 c1(OCC)cc(CNC2CC(NC(c3ncc(Cl)cc3C)=O)C2)ccc1OC(F)F C(C(=O)N1CC(C)(NC(c2cccc(C)c2)=O)C1)(C(C)C)NC(C)=O c1(C(=O)NCC#CCNC(c2ncn(CC)c2)=O)ccn2c(C)cnc2c1 CC(CC(N)=O)C(=O)NC(C)CCCNC(c1cccn(C(C)(C)C)c1=O)=O N1(CCOC)CC(C(N2CCC(O)(CNC(=O)C=Cc3cnc[nH]3)C2)=O)CC1=O n1(CCOC)ccc(C(N2CC=CC2CNC(=O)C(C)(C)c2ccn(C)n2)=O)n1 N1(C(CCC(=O)NC)=O)CC2CCC2(NC(=O)CCOC)C1 c1(C(C(=O)NC2CN(CC)CC2CC(C)(C)C)N)cccc(C)c1Br C(CCCC(CO)NC(=O)C=C1CCCCC1)NC(c1c(NC)cnnc1)=O c1(C(=O)NCC(CN(C(c2nc(COC)oc2)=O)C)O)cc(F)cc2c1CCC2 N1(C(c2cccc(C(C)=O)c2)=O)CC2(CC(NC(C3CC3CC(C)C)=O)CO2)C1 c1(C(N2CCC(N(C(=O)C(F)CC3CCC3)C)C2)=O)cnc2ccccc2n1 c1(C(N2CC(F)CC(NC(=O)CC3CCCO3)C2)=O)cnc2c(c1)CCCO2 C1(OCC)CC(N(C)C(c2cccc(Cc3nccs3)c2)=O)C12CCCCC2 N1(C(C2CCC(=C)CC2)=O)CCN2C(=O)C(NC(=O)Cc3ccnn3C)CC2C1 C1(NC(C2(CCOC)CC2)=O)CCOC(C(=O)NC(C2CCCC2)CO)C1 C(=O)(CCCCCN1CCC(O)CC1)N(C)CC1(NC(C=C(C)C(C)C)=O)CC1 Cn1nc(CNC(=O)CC2CNC(=O)O2)cc1C(=O)N(C1CCOC1)CCO c1(CNCCN2CCN(C(C=CC)=O)CC2)c(Cl)cc(C)cc1Cl C1(NC(c2scc(OC)c2)=O)CCC12CCN(C(c1nccn1C)=O)CC2 C(=O)(C1=CC2C=CC(C1)C2)N1C(C(C2=NOCC2)NC2(C)N=C(C)SC2)CC(O)C1 C1(NC(C(C)(Cl)Cl)=O)CCC2CC1CN2C(=O)CCc1ccon1 C1(NC(C23CC(OC)C2C3)=O)CCCN(C(=O)Cn2ccnn2)C1 c1(C(=O)NCCNC(CCNC(COC)=O)=O)cccc(C#Cc2ccccn2)c1 CCCC(C)C(CO)NC(C1C2CC3C(C2NC(=O)C(C)(C)COCC)C13)=O c1(C(=O)NCC(CC)NC(c2cc(=N)[nH]c(=N)[nH]2)=O)cncc(OC)c1C C1(OCC#C)CCCN(C(=O)C(C)CNC(=O)CSC(F)(F)F)C1 Cc1cc(N)ccc1C(=O)NCCCC(N1CCC(O)CC1)=O C(C(C)(CC(C)C)NC(=O)C=C(Cl)Cl)Nc1c(NC(C)=O)nccc1 Cc1csc2c(C(=O)NCC(C)CC(C)O)cccc12 C(=O)(CC(C)C(C)C)NC(CC#C)C(=O)N(C)C(C)C C1(O)(C(C)NC(=O)C(Cl)=CCl)CCN(C(c2cc(N)ccn2)=O)C1 c1(NC(c2n[nH]cc2NC(c2c(O)cccc2O)=O)=O)nc2c(s1)CCCC2=O CC(C)C(O)C(O)C(=O)NCCCN1CC(C)OC(C)C1 C1(C(=O)NCCCC(=O)NC)CC(C(=O)OC)CN1C(=O)C(C)CNC(C)=O c1(C(N2CC3(C2)CN(C(c2cc(Cl)ccc2F)=O)C3)=O)ccc2c(c1)CCC2 N1(C(CCOC(C)=O)=O)CCC2C(CCCN2C(c2ccnc(C)c2)=O)C1 CC(C)C(C(=O)NC1CC1NC(c1cnc(Cl)s1)=O)c1cccnc1 N1(C(CC(C)C(C)(C)NC(=O)CCC(C)(C)C#N)=O)CCC2(CCOC2)CC1 C1(CCOC)(NC(=O)C2CC2)CCN(C(C2CC2C(N)=O)=O)CC1 Cc1ccc(N2CCCC(C(=O)Nc3nccnc3NC(=O)C3CC3)C2)nc1 C(=O)(C(F)(CNC(=O)COC1CCOCC1)C(C)C)N1C(CCOC)CCCC1 c1(N2CCN(C(c3cn(C)nc3)=O)C(CO)C2)ncnc2ccc(I)cc12 c1(CC(=O)NC(C)CNC(C2CCOC(=O)N2)=O)c[nH]c2cnccc12 c1(C(=O)NCCCN(C(C(c2ccccc2F)C)=O)C2CC2)nc(Cl)sc1Cl C(=O)(CC(=O)NC1CC1)N(C)CCn1cc(C2CCOC2)nn1 c1(C(N(CCCN(C(c2cc(OC)n(C)n2)=O)C)C)=O)cc2cccc(C)c2s1 CCCCCC(C)(c1nnnn1C)NCc1cc(C(N)=O)co1 C(CCN=c1[nH]c(C2CC2)nc2c1CCC2)N(C(CCOC(CC(C)C)C)=O)C Cc1ccc(F)cc1C(N(C(c1cccc(F)c1)C(=O)NC1CCNC1=O)CC)=O CCCCC(C)CCC(=O)NC1CCC12CCN(C(=O)C(C)(C)CC(F)F)CC2 CCC(C)C(O)C(C)C(=O)NCC1(NC(c2ncoc2C)=O)CCC1 C1(CC(=O)NCC2N(C(CCC=C)=O)CC(O)C2)CCCC2(CC2)C1 C1(CCN(C)C(C2CCC(=O)NC2)=O)CCCCN1C(c1ncn(C)n1)=O c1(C(=O)NC2CC2)ccc(I)cc1OC(F)F c1(C(N(CC(CC)NC(c2cc(O)c(Br)s2)=O)CC)=O)ccc(F)cc1F Cn1ccc2ccnc(C(=O)NCC3CC(F)(CNC(C4(C)CCCO4)=O)C3)c12 Cc1ncc(CN2CCNCC2C(N2CCCCC2CCO)=O)c(C)n1 C(=O)(CC(C)C1CC1)NCCCN(C(=O)C=CC(=O)NC1CC1)CC c1(CC(=O)NC2CC(CCNC(C=C(C)C)=O)C2)csc(Cc2ccccc2)n1 C1(NC(c2n(CCC)ccc2)=O)CC(NC(c2cc(F)cc(Cl)c2)=O)C12CCC2 N1(C(C(C(C)C)n2cccc2)=O)CCC(NC(=O)CC(C)n2cccn2)C(F)C1 N1(C(CCC)=O)CCCC(C(C)NC(=O)COCc2nccn2C)CC1 C(=O)(C(C)(C)n1ccc(C)n1)N(CC(CNC(CC1(C=C)CC1)=O)O)C N1(C(=O)NC2C(C(N(C)C)=O)CCCCC2)CCC(C)(C2CC2)C1 C#CCCC(C(=O)N1CCOC(CCC)C1)NC(c1cc(CC)no1)=O Cc1cc(C2C(CNc3cc(C4CN(OC(F)F)C4)no3)C2)ccc1Cl c1(C(N(C2(C(=O)NCCS(N)(=O)=O)CC2)C)=O)cc(C#N)c[nH]1 C1(F)(C(N2C(CNC(c3cccc[n+]3[O-])=O)CC2)=O)CS(=O)(=O)CC12COC2 N1(C(C=CC(C)(C)C)=O)CCN(C(=O)C=C2CCCCC2)C2CCCCC12 N1(C(CCOCCOCC)=O)CCC2(NC(c3cnc(Cl)cn3)=O)CCCC12 C(=O)(C(Cc1cccc(Cl)c1)CCCO)NCC1(F)CN(C(CCC(N)=O)=O)C1 CC1CCCCCCN1C(=O)C(C1CCCC1)NC(=O)COCC1CCCC1 C(=O)(CCS(=O)(=O)N(C)C)NCCC1(OC)CN(C(C2CCCC(F)C2)=O)C1 C1(N(C(C(C(C)C)C)=O)C)CCCC2CN(C(C3CCCC3F)=O)CC12 C1(OC)CC(CNC(=O)C(c2cccc(C)c2)=O)N(C(c2cc(C)no2)=O)C1 C(=O)(C(=O)CCC(C)C)N1CCC(CC#C)(C(=O)NC(CC)C(C)(F)F)C1 N1(C(C=COCC)=O)CCC(=CCNC(C2ON=C(C)C2C)=O)CC1 C(=O)(C(C)(C)C(=O)NCCCn1cc(CN2CCS(=N)(=O)CC2)nn1)OCC C1(CC(=O)NCCCC=CCNC(CN(C(C)=O)C)=O)CCOC1(C)C c1(C(C23CC(CO2)C3)NC(=O)NCc2cccc(-n3cnnn3)c2)cncc(O)c1 C1(C)(CNC(C2=CC(C)(CC)C2)=O)CC(F)(F)CN1C(=O)C(c1csc(C)n1)=O Cc1ccc(S(=O)(=O)N2CCC2(C)C(=O)Nc2cc(C(F)(F)F)nn2C)s1 C(=O)(CCCC(=O)NC(C)C)NC(C(C(C)C)NC(=O)Cn1ccc(C(F)F)n1)C CC(C)CC(CC(C)C)C(=O)N(C)CCOCCNC(=O)C(C)(C)C1CCCO1 C1(C(=O)OCCn2cncn2)CSCCO1 C(C)(CN=c1nc2c(cnn2C)c(N2CCCC2)[nH]1)(C1CCOCC1)OC c1(CC)cc(CC(=O)NCCC2(NC(=O)Cc3cn(CC)nn3)CCC2)no1 C(=O)(CCCOCCN(C)C)N(CC(=O)NCCCF)C(C)C N1(C(CC2N(C)C(=O)CC2)=O)CCN(C(=O)Cc2ccccc2Cl)CC1C1CC1 N(C(=NCCC(C)F)NCC1(C)CCC(C(C)(C)C)CC1)C(COC)C Cc1cc(CNc2cc(Cl)ccc2NC(c2ccccc2F)=O)c(C)n1C1CC1 N1(C(CN(C)CC)=O)CCN(C(C2C=CCCC2)=O)CC1CF c1(C(=O)OCC)cc(Br)cc(F)c1NC(=O)CNc1nncn1C C1(CNC(C2CC3(CSC3)C2)=O)CN(C(=O)Cc2ccnc(O)c2)CC12CC2 Cn1ncc2c1CC(NC1CCOCC1OCc1ccccc1)CC2 CC(C)CCC(=O)N1CC(O)(CN(C(=O)C(C2CCN(C)C2)N(C)C)C)C1 c1(CC(=O)NCC2(CN(C3CCCC3C)CC)CC2)cnn2c1CCCC2 N1(C(c2c(C)cc(C(=O)OC)o2)=O)CCCCC(NC(c2ccnc(S)c2)=O)C1 c1(C(=O)NC2CC(OCC(N3C(C)(CCC)CC3)=O)C2)ccc(CC)cn1 N1(C(C(C)OCOC)=O)CC(O)CC1CC(=O)N(C1COC(C)(C)C1)C CCC(CC(F)(F)F)C(=O)NCC1(C)CCN(C(c2cccn2C(C)C)=O)C1 c1(OC)ccc(CN(C(C)CNC(=O)Cn2cc(I)nn2)C2CC2)cc1Br N1(Cc2nc(COC)sc2)CCC2C1CCCN2C(=O)CO N1(C(C2(C(C)(C)O)CC2)=O)CCC(C)(C)C1CC(N1CCC12CCCC2)=O C=CCC(C)(C)CC(=O)N1CCOC(C(=O)NC(C)CC2CCC2)C1 CC(C)(C(=O)NCC1CCC(NC(c2cc(CO)ccn2)=O)C1)C(N)=O S(=O)(=O)(c1ccc(C)cc1)N(C(=O)C(c1cccc(I)c1)C)CCN(C)C.CS C12(CCC(C)(Cn3cccn3)NC(CCCCSC)=O)CCC(CC1)CC2 CC(O)CCCC(=O)NC1CC(CNC(c2n[nH]cc2Cl)=O)C1 c1(C(=O)NC2CC3CC2CN3C(=O)Cn2ccnc2)c[nH]c2ncccc12 c1(OC)ccc(CO)cc1NC1(c2nnnn2CC(F)F)CC(C)(C)C1 N1(C(C2(OC(C)=O)CC2)=O)CCN(C(=O)CC2CCCOC2)CC(C)(C)C1 CC(C(=O)NCC1CN(C(=O)CCC2CCCN2C)C1)C(C)(C)C C#CCC(C)C(=O)N1CCC(C)(CCNC(=O)CN2CC(=O)NC2=O)C1 CC1CCN(CC(=O)NC23CC(CNC(=O)CC4CCCCC4F)(C2)C3)CC1 Cc1nn(CCO)cc1C(=O)NC12CC(CNC(=O)CC3(C)CC3(Cl)Cl)(C1)C2 C1(CNC(COCP(C)(C)=O)=O)CN(C(C2(C)CC=CCC2)=O)CC12CCC2 N1(C(CC)=O)CCC(F)(C(=O)NOCC(c2ccc(C)c(C)c2)=O)CC1 C12(NC(CCCN(C)C)=O)CCCC1N(C(c1cnc(C(F)F)cn1)=O)CCC2 c1(C(=O)NCC2C(C(N(CC)Cc3cccs3)=O)CCO2)cc(F)cnc1O CC1(C)CCC(C(=O)NC(C)(C)CNC(=O)CNC(c2ccoc2)=O)C1 c1(C(=O)NC23CN(C(C(CC)Oc4ccccc4)=O)C(C2)C3)nc(F)ccc1Cl c1(C(=O)NCC2N(C(C(CC)=CC)=O)CCCCC2)cnc2cnn(C)c2c1 C1(C(=O)NC(CCNC(c2cn(CC(CC)O)nn2)=O)C)CCCC(C)(C)CC1 CCS(=O)CC(=O)NCCN(C(=O)CCc1ccc(OC)cc1)CCOC c1(CNC(c2c(Cl)nsc2Br)=O)ncccc1C(F)(F)F c1(OC)ccc2c(c1)OCC(C(=O)NC(C)CNC(=O)Cc1ccccc1Cl)C2 C12(CNC(c3ccc[n+]([O-])c3)=O)CC(NC(C3CCOC3C(F)F)=O)(CCO1)C2 [N-]=[N+]=NC1CCC(C(N2CC(O)(CC(=O)NCCc3cocn3)C2)=O)C1 N1(CC(=O)N(C(=O)Cc2nnc3n2CCOC3)C)CC(C(C)(C)C)c2ccccc21 N1(C(c2csc3nccn23)=O)CCC2(CCN(C(C3C=CCC3)=O)C2)C1 c1(C(N2CCC(CC(=O)NC(CO)C3(O)CC3)CC2)=O)cc(F)ccc1O C(=O)(CN=c1cc[nH]cc1)N1CC(CC(=O)Nc2c(C)c(F)ccc2)OCC1 Cc1cc(=NCCC#CBr)[nH]cc1S(=O)(=O)N1CCCC(C)C1C N1(C(Cc2c(C)nc(CC)nc2C)=O)CCC2(CC1)COC(=O)N2 Cc1oc(S(N)(=O)=O)cc1C(=O)NC(c1cn(C2CNC2)nn1)C1CCCCC1 CC1CCN(C(=O)CC2CC(CF)C2)CC1NC(c1ccnnc1O)=O Cn1c(C(=O)NC2CCN(C(c3cnc(S)n3C3CC3)=O)CC2)nnc1S CC(C)C(C(N)C(=O)Nc1ccc(Br)cc1-n1cccn1)c1ccccc1 N1(C(c2nc(OC)oc2)=O)CCC(C)(C(=O)NCCOCCCCOC(C)C)C1 CC(C)(C)CCC(=O)N1CC2(C)CC1(C(N1CCCC(C)(O)C1)=O)C2 N1(C(C2(N(C)C)CCC2)=O)CCC(N(C(C2C3CNC(=O)C23)=O)CC2CC2)CC1 c1(CC)[nH]nc(Cl)c1C(N1CC(O)(CCNC(=O)CCC2C(=O)ON=C2C)C1)=O c1(C(=O)NCCN(C(=O)CCC2CCCOC2)CCOC)nc(Cl)c(Cl)s1 c1(C(=O)NC(CN(C(CC(CC)SC)=O)CC)C)cccc(N)c1C N1(C(CN(C(COC)=O)C)=O)CCN(C(c2nnc(S)n2C)=O)C2CCCC12 C1(F)(C(=O)CC2(C#N)CC2)CCN(C(c2cc(C(F)(F)F)cc(F)c2)=O)CC1 C(c1ccc(F)c(F)c1)=CC(=O)NC(CNC(C(CC#C)C1CC1)=O)(C)CO c1(CNC(CC2CCC(NC(CC3(OC)CC3)=O)C2)=O)ccc(C)cc1 c1(C(N2CC(CCC)N(C(=O)Cn3cncc3C)CC2)=O)cc(F)c(F)cc1N c1(C(=O)NC(C2CN(C(=O)CN3C(C)CCC3C)C2)C)cc(C2CCCO2)n(C)n1 C1(NC(c2ccc(C)o2)=O)CCCCC1NC(=O)CN(C)Cc1nnc(C)n1C c1(C(=O)N(CC2(O)CN(C(c3cncc(OC)c3)=O)C2)C2CC2)cc(I)ccc1F c1(C(=O)NC(C)CNC(=O)CC(C)C(C)(C)C)c[nH]c2ccc(Br)cc12 N(C)(C1CN(C(c2cc(C)on2)=O)CCc2ccccc21)C(CCCOCC)=O CC(CN(C)C(c1nccs1)=O)C(=O)NC1CCOCC1 c1(OC)cccc(F)c1C(=O)NCC1CN(C(=O)C(O)C(F)F)CC1O c1(-n2c(C(c3nc(C)cs3)C)nc(-c3scc(C)n3)n2)ccc(S(C)(=O)=O)cc1 c1(C(C(=O)NCCN(C(CCC(=C)Cl)=O)CCC)(C)C)ccc(Cl)cc1F Cn1nccc1C=CC(=O)N(C1CCC(NC(=O)CC2CCCCC2F)CC1)C N1(C(C2C(C)C2)=O)CCCCC(C2CN(C(c3occ4c3CCC4)=O)C2)C1 Cc1cnc(CNCCN2CCN(C(c3cc(Cl)cnc3O)=O)CC2)cc1Br c1(C(=O)NCCC2CN(C(C3CCCS3)=O)C2)nn[nH]c1C(F)(F)F C=CC1(C(=O)NCC23CCC(F)(CC2)C3)CCN(C(=O)CN2CC(=O)NC2=O)C1 C#CCC(C)(CC)C(=O)N1CCN(C(c2cc(F)c(F)cc2O)=O)C(C)C1 C1(CC)(NC(=O)C=C(C)C2CCCCC2)CCCN(C(c2ccoc2Cl)=O)C1 c1(C(N(C2CCN(C(=O)C(C)SC(C)C)C2)CC#C)=O)cccn2ccnc12 C1(NC(C2(CSC)CC2)=O)CCC(NC(c2cnc(-c3ccccc3)s2)=O)C1 c1(C(N2CC(NC(C(C(C)O)N(C)C)=O)C(F)C2)=O)ccc2c(c1)C(=O)CCS2 c1(C(N2CCCC(O)(CNC(C(C)C3CC3)=O)C2)=O)csc(S(N)(=O)=O)c1 C(CCC(C(=O)NCc1ccc(F)cn1)NC(c1ncccc1O)=O)OC C1(N(C(C2CCN(C)C2)=O)C)CCC2CN(C(C3CC4(CSC4)C3)=O)CC12 C(=O)(C(O)CCNC(C1(C)COCCO1)=O)NC(C#C)C(C)OC N1(C(C=CC=CC)=O)CCOCC(NC(C2CC3(CC3)CN2C)=O)C1 Cc1cc(-c2nc(C(C)C)nn2C2CCOC2C)c(F)c(Br)c1 c1(C(C)C)ccc(N)c(C(N2CC(NC(=O)C=Cc3ccc(Cl)s3)C(C)C2)=O)c1 c1(CN(C)C(=O)Nc2ccc(O)c(F)c2)noc2c1CCCC2 c1(C(C)=O)c(CCC(N2CC(CNC(=O)CNS(N)(=O)=O)C(O)C2)=O)c[nH]c1C C1(C(C)C)CCOCCN1C(=O)NC1CCCCC1(C)C c1(C(=O)NC(CN(C(=O)CC2CC(OC)C2)CC)C)cc(C)c(C)o1 c1(OC(N(C)OCC(F)(F)F)=O)cc(O)nn1-c1ccccc1F c1(C(C(=O)NC)N(c2cnn(C3CCC(N)CC3)c2)C)cc(Br)c2ncnn2c1 c1(C(=O)NCC(CC=C)NC(c2snnc2C)=O)snc(O)c1Cl CC1ON=C(C(=O)NCCN2CCC(NC(=O)C(F)F)CC2)C1C c1(CC(=O)NC2(C3N(C(C=CC(=O)OCC)=O)CCC3)CC2)ncc(F)cc1F c1(C(=O)NCC2CCC(C(N3CCC(C(=O)NC)C3)=O)C2)cc2cnccc2[nH]1 c1(C(=O)NC(CN(C(C2CC2F)=O)CC)C)cnc(OC(C)C)cn1 C#Cc1ccc(C(=O)NCCC2CCC(NC(C3CC(Cl)(Cl)C3)=O)C2)cc1 N1(C(C(CC)NC(=O)CNS(C)(=O)=O)=O)CC(OC)C2(CC2)C1 C(=O)(C(N)CCC(C)(C)C)NCC(C(=C)C)(C)C C1(C(=O)OC)(NCC2C(COC)C2)CC(C(F)F)C1 CCC(C)C(CC(=O)NC(C1CCCO1)C)NC(=O)CCN(CC)CC C1(CNC(C(C(C)C)OCC)=O)CN(c2ncc(C#N)cc2C)CC2(CCC2)O1 Cc1[nH]nc(C(=O)NC2CCCC2NC(=O)Cc2ccncc2Cl)c1Cl c1(NC(C2c3n(nc(C)c3)N2C)=O)ccc(Cl)cc1F.c1(CC)ccc(C)c(Br)c1 C=CC1(C(=O)NC2CC3C=CC2C3)CCN(C(=O)Cc2ccc(C)s2)CC1 N1(C(c2c(F)ccc(OC)c2Br)C(=O)NC2COC2)CCOc2ccc(F)cc21 CCN(N1CCC(N(c2ccccn2)C(=O)C(C)(C)C)CC1)N1CCCC1 CC1CCN2CC1NC(=O)C2.C(=O)(CC(C)(C)O)N.O(C(F)(F)F)C(C)(C)C c1(OC)ccc(C(N2CC(C3(NC(c4cc(N)nc(Cl)c4)=O)CC3)C2)=O)cc1F c1(C=O)sccc1S(N)(=O)=O.c1(C=O)ccccc1C(=O)NC1CN(N(C)C)C1 CC1CCN(C(=O)CC2OCCC2C)CC1CNC(c1ncc[nH]1)=O C(=O)(C1SCc2cccnc21)N(CCCN(C(=O)CNC(=O)C(F)(F)F)C)C c1(OCC=C)ccccc1C(=O)NCCN(C(=O)C(O)C(C)OC)C(C)C c1(C(=O)NC2(CO)CN(C(=O)C3=CCCCO3)C2)cc2ccsc2c(O)n1 N(C1CN(C(=O)C2=C(Cl)CCOC2)CCc2ccccc21)C(C1C(C#N)C1)=O c1(C(=O)NCC(CC)NC(=O)C(C(C)C)NC(=O)NC(C)C)cncc(Cl)c1 C1(NC(Cc2c(OC)ccc(Cl)c2)=O)CN(C(c2cnn[nH]2)=O)CC1C1CC1 N1(C(c2c(C(C)(C)C)ncs2)=O)CCC(O)(CNC(C2CCC3CC23)=O)C1 C(CC(C(=O)NCCC12CC(CCO1)C2)NC(=O)CC(=O)NC1CC1)OCC c1(C(N2CCN(C(C=C(CC)CC)=O)CC2CF)=O)cc2cccc(F)c2s1 N1(C(C(CC(C)C)ONC(CC(C)C(C)(F)F)=O)=O)CC2CCOC(=O)C2C1 C1(NC(Cc2nc(C)[nH]n2)=O)CN(C(c2ccc(S(C)=O)cc2)=O)CC2(CC2)C1 C(C)(CCC(=O)N1CCC(C(=O)N(C2CCCC2)C(C)C)(CO)C1)SC c1(CNC(CC2CCN(C(CC3C(C)(C)C3)=O)C2)=O)cc(Cl)ccc1O Cc1cc(Cl)c(C(=O)NCC(C)(C)CNC(C2(C3CCCO3)CCC2)=O)cc1F N1(C(C(C)OCCC(C)C)=O)CCCC(C2CCCN(Cc3ncnn3C)C2)C1 C1(CNC(CC(C)(C)SC)=O)CCC2CN(C(=O)CC(C)C3CC3)CC12 C(=O)(C1=CC2CCC=CCCC12)NCCCN(C(c1cnc(OC)nc1C)=O)C N1(C(C2C=CCC2)=O)CC2CCOC2(CNC(=O)C(F)(F)c2ccncc2)C1 C1(CCNC(=O)CC2CCC(=O)N2)CCN(C(c2ccnc(O)c2)=O)CC1(F)F C1(C(=O)NCCN(CC(C)O)C(c2n(CCC)ccc2)=O)CC2CCC2C1 C1(C(=O)NCC2(CN(C)C(c3cccc(OC(F)F)c3)=O)CC2)CCCC12CC2 C(=O)(C1CCCn2cncc21)N1CCC(C(C)(C)C)CC1CNC(=O)C=CCO C(=O)(C(C)Cc1ccccc1)NC(C1CCN(C(C2CCCC2O)=O)C1)C C(=O)(CN=c1cc[nH]cc1)N1C(C)CC1C(=O)Nc1cnc(CN(C)C)nc1 C(CCCC(CO)NC(C1CCCN1C)=O)NC(C(C#C)(C)C)=O c1(CN(CCCNC(C2(C3CCC3)CC2)=O)C(C)C)cc(C#N)ccc1F N(C1CCCOc2ccccc21)C(C=C)C C(C(C)CC(=O)N1CC(NC(=O)C=CC(=O)N(C)C)C(C)C1)OC c1(NC(=O)NCC(CCCOC)C)ccc(OC)c2ccnn12 CCCCCC(O)C(=O)N1CC=C(CCNC(C2CCN(C)C2C)=O)CC1 c1(OC)cc(Cl)ccc1C(CO)OC(F)F.C1(=O)NCCN1 C1(C(=O)NC(C(=O)NC(c2n(CC)ncc2)C)c2ccoc2)C2CN(C)CC12 c1(C(=O)NCC(CC)(CC)NC(C2CCN(C)C2=O)=O)cc(N)c(O)c(F)c1 c1(CCC)nc(CN(CCn2cc(CO)nn2)C(C2(C)C=CCC2)=O)cs1 c1(C(=O)NCCN(C(COC(CC)(C)C)=O)C(C)C)ccccc1NCCOC c1(C(N(C)CC2CCN(C(c3cc(C)on3)=O)C2)=O)ccc(C(F)(F)F)nc1 N1(C(C(C2CC2)OC)=O)CC2(CCCC2)C1C(=O)NC1(C)CCC(=O)NC1=O Cc1c(C(N2CC3(CC(NC(c4nc(C(C)C)cs4)=O)C3)C2)=O)cccc1F Cn1nc2nc1C(c1nnnn1C)NC2c1ccncc1.C1(C)CCC1 CCCC(O)CC(=O)NCC(C1CCCC1)NC(c1c[nH]nc1-c1ccsc1)=O c1(C(=O)OC)ccc(C(=O)NCCOc2ccc(Cl)cc2)c(F)c1 c1(N2CCC(C)C2CNC(c2cc3c([nH]2)CCCC3)=O)ncc2ncn(C)c2n1 c1(C(N2CCN(C(CC3C(CC)C3)=O)C(C)CC2)=O)cc2c(nc1O)CCC2 CC1CCN(C(=O)Cn2ncnn2)CC1CNC(c1csc(Br)n1)=O N1(C(CNC(=O)NC)=O)CCN(C(C2CCC3(CCC3)OC2)=O)CC(CO)C1 C(CC(C)(C)C(=O)N1CCC(CNC(c2ncccc2N)=O)C(C)C1)OC N1(C(Cc2nnc(C)o2)=O)CCC2(CC1)CCN(C(C1CC3CC3CC1C)=O)C2 N1(C(C2(C(N)=O)CCC2)=O)CCCN(CCNC(C2CCC3C2C3(F)F)=O)CC1 c1(NC(C2(OC)CCN(C(=O)CCSC3CCCC3)C2)=O)ccc(CO)c(C)c1 c1(C(N2C(C(N3CCC(CCO)CC3)=O)CC(O)C2)=O)cnc2cc(Cl)ccn12 N1(C(C2(OC)CCCC2)=O)CCCC(C)(CNC(C2CC2c2ccn(C)n2)=O)C1 N1(C(C=C2CCC(C)CC2)=O)CCC2(CCCC2NC(C2SCCS2)=O)CC1 C12(NC(C=C(CCC)CCC)=O)CCCN(C(c3ccc(F)c(N)c3)=O)CC1C2 c1(C(C(=O)NCCNC(C2CN(C(=O)COCC(=O)N(C)C)C2)=O)O)ccccc1 C(C(CC(C)C)NC(=O)CCc1cnccn1)n1cc(C(C2CC2)OC)nn1 C1(C(=O)NC2C(NC(C3C(c4n(C)cnn4)CC3)=O)C2)CC(C2CC2)=NO1 Cc1cnoc1NC(=O)COC(=O)CC1(c2ccon2)COC1 N1(C(c2ccccc2)C(=O)Nc2c(C)cccc2C)C2CCC1CC(F)C2 c1(CCC)ccc(C(N2CC(CNC(C3(Cl)CC3)=O)C2)=O)c(O)n1 CC1(C)CN(C(=O)Cc2ncc(F)cc2F)CC1NC(=O)C#CC1CC1 N1(C(C2CC3CCC(C2)S3)=O)CCN(C(c2nncs2)=O)C2COCC12 N1(C(CC(C)F)=O)CC(CNC(c2ccccc2C2CC3CC3C2)=O)CC1(C)C C1(C(N(C2CCCCC2NC(=O)CCc2cncs2)C)=O)CC1C1CCC1 C#Cc1ccccc1CNC(C1CC(CCNC(C2CCC2)=O)C1)=O n1(CCC)cc(C(=O)NCC2(NC(=O)CC3CC(C(N)=O)C3)CCC2)nn1 c1(C(N2C(CNC(c3ccsc3)=O)CC(OC)C2)=O)coc2c(F)cccc12 N1(C(COCC(=O)NC)=O)CCC(CCN(C)C(=O)OCC(F)F)CC1 c1(C(N2CC3C(NC(CC(CCC)C)=O)(C3)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(COCC=C)=O)CCCCC(CNC(C23CCCC(CO2)C3)=O)C1 CCCCC(C(=O)NC1CN(C(c2cc(OC)cs2)=O)CCC12CCC2)C(C)C N1(C(Cc2c(C)ccc(C)c2)=O)CC2CCC1C(NC(C1CN(C)C1)=O)C2 CC(C1=NOC2COCC12)NC(C1CCCNC(=O)O1)=O C1(CC)CN(C(=O)CCCn2ccnc2)CCC1NC(=O)C(c1cccnc1)O c1(C(=O)NCC(C)(CO)NC(C(CC(=O)OC)C)=O)cc2ccnc(Cl)c2s1 CN1C2CCC1CC(c1nnnn1C(C)(C)C)(NCC1CC1(Br)Br)C2 C=CC1OCCCC1C(=O)NCCN(C)C(C1CCN(CC(F)(F)F)C1)=O C1(NC(c2cc(C)n(C)n2)=O)CN(C(c2cc(C(F)F)no2)=O)CCC1O C1(C(=O)O)(NC(=O)COCCn2cc(COCC3CCCCO3)nn2)CCCC1 Cc1cc(C(F)F)c2nc3n(c2n1)CCC(C(F)(F)F)(C=O)C3.N1CCCC1 N1(C(CC(C)(O)c2ccccc2)=O)CCCCC(NC(C2CC2F)=O)C1 N1(C2CCN(C(CC(C)C)=O)CC2)CCN(C(=O)C=CCCCN=[N+]=[N-])C1=O N1(CC)CC(C(N2CCCC2C2(NC(=O)C3=CCCC3)CC2)=O)CCC1=O N1(C(C2CCC(=C)CC2)=O)CC(C)(C)OCC1CNC(=O)C(C)(C)C#N C(=O)(C(C)(C(C)C)NC(C)=O)N1CCC(CN(C(C=CCN(C)CC)=O)C)CC1 N1(C(c2c(C)n(C(C)C)nc2)=O)CCCN(C(C2CC3CC3C2)=O)CC1C C1(C(N2CC(OC)(CNC(C3C=CCCC3)=O)C2)=O)CC(=O)N(C(C)C)C1 C#CCCCC(C)C(=O)N1CCC(CC(=O)Nc2cncnc2C)CC1 Cc1cn2ccnc(C(N3CCCC3CN(C)C(C3CCC(=O)N3C)=O)=O)c2n1 c1(NC(C2C3(CCN(C(c4cc(C)[nH]n4)=O)C3)C2)=O)ncc(I)cc1[N+](=O)[O-] CC1(C)OC(=O)C(CC(N2CCCC(CCCCNC(=O)C3=CCCS3)C2)=O)O1 CCCC(C)(CO)NC(=O)CCC1CCCN(C(=O)C(C2CC2)C2CC2)C1 c1(C(=O)NCC2(CNC(C)=O)CC2(F)F)nn(C)cc1Cl c1(C(N(C)Cc2cccc(CNC(c3cnc(C)[nH]3)=O)c2)=O)cc(N)c(Cl)cn1 N1(C(C(C2CN(C(=O)Cc3ncccc3F)C2)OC)=O)CCC(F)CC1 C1(NC(c2ccn(CC)n2)=O)CC2CC1CN(C(=O)Cc1nc(C)sc1C)C2 CC1CC(C(=O)N(C(CF)CF)C)CN(C(c2ncc[nH]2)=O)C1 N1(C(CN2CC(C)C2)=O)CCC(C)C(CNC(=O)Cn2cccnc2=O)C1 c1(OC)cc(OC)c(NC(C2(C)CCN2c2nc(C)cc(C(F)(F)F)n2)=O)cn1 c1(OC)ccc(C(=O)N(C2CCCC2)CCNC(C23CC(F)(C2)C3)=O)cc1 C=CCC(CNC(=O)CCCC1CCC1)C(=O)NC1CC(O)C(F)C1 CC1Cc2c(Cl)cccc2C1NC(c1c[nH]nc1C1CNC1)=O c1(C(N(CC(=O)NCc2nc(C(C)C)on2)CC2CCC2)=O)cccc(F)c1F C(=O)(C1=C(Cl)CCCC1)NCC(C(=O)NC1C(OC)CCC1)N(C)C CC1CC(NC(=O)Cc2ccc(Br)cc2O)CN(C(C2C3COCC23)=O)C1 c1(NCCc2cc(C)no2)cc(N(C)Cc2csc(C(C)(C)C)n2)ncn1 CC1CCN(C(=O)OC(C)(C)C)C1CNC(=O)CNC=O.C12CCCN(C1)C2=O c1(CC(=O)NC(C)CNC(=O)C(N2CCP(C)(=O)CC2)C)ccc2nsnc2c1 C1(C(=O)NCCNC(C2CC(C)N(C)C2)=O)CCCC12CCC2 c1(C(=O)NCCC(C)N(C(=O)CCCC2CCCO2)C)ccnnc1O C1(NC(c2c(OCC)ccs2)=O)CCN(C(C2(C)COC(=O)OC2)=O)CC1C C12(NC(c3c(C)snn3)=O)CC1CN(C(C1CCCN(C(C)C)C1)=O)C2 c1(C(=O)NCC=CCNC(=O)OCCOCC)nn(C)c2ncc(S(C)(=O)=O)cc12 CC(O)C(F)(F)C(=O)N1CCOC(C(=O)NCCCS(C)(=O)=O)CC1 c1(OC)ccc(C(=O)NCCC2CSCCN2C(=O)CC(O)C(C)C)nc1Cl c1(C(=O)NC2CCN(C(C(CC)NC(N)=O)=O)C2)c(Cl)ccc(OC)c1N CC(C(=O)NCCC(c1c(OCC(F)(F)F)cccn1)=O)S(=O)(=O)C1CCOCC1 c1(C(N(C2CN(C(CC3C(C)OCC3)=O)CC23CC3)C)=O)ccc2nn[nH]c2c1 C=CCCCC(=O)NCC(CC(=O)Nc1cccc(OC)c1)C1CCC1 N1(C(c2cn(CC)nc2C)=O)CCCN(CCCCNC(=O)C#CC2CC2)CC1 c1(NC(C)=O)ccc(C(N2CCC(O)(CNC(=O)C(C)CF)C2)=O)c(Cl)c1 c1(C(C)=O)cc(NC(=O)C(C)C(C)NCC2(c3ccno3)CC2)ccc1F Cc1cc(C(=O)N(C)CC2(O)CCN(C(=O)CCC(N)=O)C2)cn1C N1(C(C(Cc2ncn(C)c2)O)=O)CCCCC(NC(=O)C=C2CCOCC2)C1 c1(C(=O)NCC(CNC(C(CC)n2ccc(C3CC3)n2)=O)O)nnc(O)nc1O N1(C(C2(OCC)CCCSC2)=O)CCC(N2CCCC2)CC1c1ccccc1 N1(CC(CCCC)CC)C(=O)CCN(Cn2cc(C3CC4(C3)OCCO4)nn2)C1=O O=C(C(O)CCNC(=O)C(O)C1CCCC1)N1CCC2CCC12 N1(C(CC=CCNC(c2nn(C)c(CO)c2)=O)=O)CCC2(CCSC2)C1 C1(CNC(C2C(OC)CC2)=O)CN(C(C23CC(CN2C2CC2)C3)=O)CC(C)(C)O1 c1(N2CCCCC(SC)C2)nc(N2CCN(C)C(C(C)C)C2)c2c(n1)CCOC2 C1(NC(CCC(CC)=O)=O)CCSC12CN(C(c1cc(C)n(C)c1C)=O)C2 c1(C(=O)OC)cc(F)c(C(F)(F)F)cc1S(=O)(=O)N1CCCC1CC1CCC1 C1(NC(CC(C)(C)OC)=O)CCC2CC1CN2C(c1cc(C)n(C)n1)=O C1(C(=O)NCCN(C(C)C)C2CC2)(NC(C2CC23CCOC3)=O)CCCCC1 CC1(C)COC(CCC(=O)NC2COCCC2NC(=O)CC(C2CC2)C2CC2)C1 C1(CN(C(=O)CCNC(=O)CO)C)CCCN1C(=O)CC(C1CC1)C1CC1 N1(C(c2cnn(CCF)c2)=O)CCC2CN(C(C3CC=CCC3)=O)C2C1 C1(C(=O)NC2C(OC)C(O)C2)CC=CCC1NC(=O)CC1OCCCO1 C(C(=O)N(C(C)C(=O)N(C(C)CO)C)C1CC1)(OC)OC CC1C(NC(=O)C(C)N2CCC2)CCCN1C(c1ccnc(F)c1N)=O N1(C(CCNC(C)C)=O)CC2CC1CN2C(c1ncc(-c2ccccc2)s1)=O c1(C(=O)NC2CN(C(C(=O)NCCC(N)=O)=O)C2)ccc(F)c2c1CCC2 CC(CC(=O)NC1CCOC1C(=O)N(CC(F)(F)Cl)C)N(C)C C1(CC(=O)N(c2ccccc2-c2ccccc2)CC=C)CC2COCC12 c1(C(N(C2CCN(C(=O)CCCn3cncn3)C2)CC)=O)sc([N+](=O)[O-])cc1Cl C1(OC)CN(C(C2(F)CC2)=O)CC1NC(c1cnn(CCO)c1N)=O C12CCCN(C1)C(=O)c1cc(oc1C)-c1cccc(c1)N2C=O.CCO.OC c1(C(N2C(C)(C(=O)NC3(CCC)CC3)C=CC2)=O)ccc(C)cc1O CC1CCN(CCCNC(=O)NCCN2CCC(O)CC2)CC1 n1(CC(=O)NCC(CCC)NC(c2n(CC#C)cnn2)=O)nnc2c1CCCC2 C(CS(=O)(=O)C(F)F)NC(=O)NC1CCN(CC(=O)NC(C)(C)C)C1 c1(C(N(CCNC(C=CC)=O)CCSS(=O)(=O)CC)=O)cc(COC)oc1C C(c1ccncc1)=CC(=O)NC1CC1NC(c1cc(C(F)F)ncn1)=O c1(CNC(CCc2cccc(OC)c2)C)ccc(Br)c(C)c1F c1(CN2C(COC)CN(C(=O)Cc3cccn3C)CC2)cc(C)c(OC)c(C)c1 C1(CC#C)(C(N)=O)CCC1.C(=O)(C=CCOCC)NCCOCCOC c1(NC(CC(C)C)CNC(=O)C(c2cnn(C)c2)O)nc2cc(Cl)cc(Cl)c2o1 C1(NC(C2CC(NC(=O)Nc3cncnc3)C2)=O)CCOC12CCOCC2 C(c1ccccn1)=C(C(=O)NCCCCNC(C1(CC)CCC1)=O)C C1(NC(CCC(=O)OC)=O)CCCCC1N=c1ccc(C#N)n[nH]1 Cc1nn(CC(=O)NC2C3CC(NC(c4cc(Cl)ccn4)=O)CC23)c(=O)n1C N1(C(CCN(C(=O)CCc2cncn2C)CC)=O)CCCCCC1C Cc1cc(C(N2CC(O)(C(C)NC(=O)Cc3c(C)cccc3F)C2)=O)cc(Cl)c1 c1(OC)ccc(C(=O)NC2CCOCC2C(=O)NCc2ccc(C(N)=O)s2)nn1 C12(CNC(COc3ccc(CC)cc3)=O)CCC(CC1)N2C(c1ccc(C)o1)=O Cc1cnc(C(=O)NC(CNC(=O)Cc2ccc(Br)cc2C)C2CC2)c(F)c1 C(CC(=O)N(CC(O)CNC(c1nn(CC)cc1Br)=O)C)(C(C)C)OCC C1(C(N(C)CCNC(=O)CSc2ccccn2)=O)CCC2(CC1)CC2 CCC(C)CC(CO)NC(C1(F)CN(C(C2CC(OC3CC3)C2)=O)C1)=O C=CC(C)(O)CC(=O)NC1CCC1NC(=O)Cc1cccc(C2CC2)c1 N1(C(CCSC)=O)C(C(=O)NCc2ccc(F)c(F)c2F)CC2CCCCC12 CCCC(CCc1ccccc1)C(=O)NC(C)(CNC(C12CC(F)(C1)C2)=O)CO N(CP(C)(C)=O)(CC(N1CCC(OC(C)(C)C)C1)=O)C(C1C2(CC2)C12CC2)=O CC1CC(CNC(C2CCC(NC(Cc3cncs3)C(=O)O)CC2)=O)CCS1 N1(C(c2n(CC)nnc2)=O)CCC2(C1)CN(C(C1CCC(F)CC1)=O)CCO2 C1(CCC)CN(C(=O)COCC2CCC2)CCN1C(c1cncc(SC)c1)=O N1(C(C(CS)(C)C)=O)CCC2(CC1)CN(C(=O)C=CC(C)(C)C)CC2CC1CC1.CO CC1(C)C(CNC(=O)CC23CCCC2C3)CCN1C(=O)CCP(C)(C)=O C(CC1=CCN(C(=O)CC2CCCC(=O)N2)CC1)NC(C1(C)CCCCO1)=O CC1(C(=O)NC2COCCC2NC(C2(O)CCC2)=O)COc2ccccc21 c1(C(N)=O)cccc(NCC(N2CC(O)(CCNC(C3OCCCO3)=O)C2)=O)c1 C1(NC(=O)C(c2ccccc2)O)CN(C(C2(c3ccno3)CC2)=O)CC1O C1(CNC(CCc2cc(C)n(C)n2)=O)CN(C(c2ccncc2Cl)=O)CC1(C)C NS(=O)(=O)N1CC(C(N2CCN(C(C3CCC34CCC4)=O)CC2)=O)C1 n1(CC(=O)N(C2CN(C(C3(OC)CCC3)=O)C2)CCO)nc2n(c1=O)CCOC2 C1(C(C)C)CN(C(C2CCS(=O)CC2)=O)CCN1C(c1nccn1C)=O CCCC(CNC(=O)CCN1CCC(C(C)CO)CC1)CC(CC)CC C12(C(=O)NC3C(CNC(=O)CC4CCCOCC4)CCC3)CCC(CC1)OC2 n1(C(C)C)cnnc1CC(=O)NC1CC1CNC(=O)C(C)(Cl)Cl n1(CCC(N2C(CNC(C3CC(OC)C3)=O)CC2)=O)c(C)csc1=O C(CC)(C(=O)NCC(C)(O)CNC(c1cnc(C2CCC2)o1)=O)=CC c1(C(=O)NC(CNC(CC(C=C)CC)=O)C(C)C)cnc2nc(O)nc(O)c2c1 C1(O)(CNC(N(c2ccc(C)cc2Br)C)=O)CCCN(C)C1=O N1(C(c2ccc(Cc3ccccc3)cc2)C)C(=O)NC(C)(c2cc(F)cc(F)c2)C1=O c1(OC)ccccc1C(CNC(=O)C(C)(F)F)NC(=O)CC1C=CCC1 C(=O)(C(CNC(C1(F)CCCCCC1)=O)C(C)(C)C)NC(c1ccc(C)s1)C C1(COC)CN(C(=O)C(N2CCC(CSC)CC2)=O)CCCO1 CC(CC1CCCC1)C(=O)NCC(C)CN(C)C(C1CCCS1)=O C(=O)(C1COc2ccc(Cl)cc21)N1CC(O)(CN(C(c2c(C)ccnn2)=O)C)C1 c1(C(N2C(CCCNC(C3CC3F)=O)CCC2)=O)ccc(C2CCCO2)nn1 C1(NC(C2CC(C)(CC)C2)=O)CCC2CC1CN2C(=O)OC(C)(C)C Cc1nc(C(=O)NC(C)CCCNC(c2cc(C(C)(C)C)c[nH]2)=O)cc(O)n1 c1(NC(CC)CN(C)C)nc(N2CCCC(OC)C2COC)nc2scnc12 C1(C(N2CC(OCCNC(C(C(C)C)n3cccc3)=O)C2)=O)CCC(C)C(C)C1 c1(C(=O)NC(C2CCN(C(=O)C=CC3CCCN3C)CC2)C)cnc2n1CCC2 N1(C(C(Cc2c(C)nn(C)c2C)C)=O)CC(C)CN(C(C23CC(C2)C3)=O)CC1C c1(C(=O)NCCN(CCC)C(c2nnc(C)s2)=O)nccn2cc(C)nc12 CC(CF)C(=O)NCCNC1CC1.C1(C(=O)O)CCCN1S(C)(=O)=O C1(n2cc(CSC)nn2)CCCCC1NC(c1cc(I)ccc1Cl)=O Cc1cc(N)c(C(=O)NCCCCCNC(=O)Cc2ccsc2C)c(Cl)c1 c1(OCC(=O)NCc2cn(CC(C)Nc3cc[nH]n3)nn2)cc(Cl)ccc1Cl C1(NC(Cc2n(C)ncc2Cl)=O)CC(NC(c2nc(Cl)cs2)=O)C12CCOCC2 C1(C(N2CC(C)(OCC(=O)NCCC3(OC)CCC3)C2)=O)CCC(F)(F)C1 N1(C(C2(CC=C)CC2)=O)CCCC(CC(=O)NCCN2CCCC(OC)C2)C1 N1(C(CC2C(C)(C)C(O)C2)=O)CC2CCCN(C(c3ccccc3)=O)C2C1 c1(OC)ccc(C2CC2)c(C(=O)NCCCC2CCN(C(=O)C(C)CO)CC2)c1 N1(C(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)CCn2cnnn2)C2CCC12 C12(CNC(CCNS(C)(=O)=O)=O)CCCCC1N(C(C1C3(CC3)C13CC3)=O)CC2 c1(CC)cc(NCC2CC(C)N(C(=O)OC(C)(C)C)C2)n(C)n1 c1(OCC)cc(C(=O)NCCC2CCCN2C(=O)C(C)CC)ccc1OCC CCCCC(O)CC(=O)N1CCC(C)(CNC(c2cn3ccnc3s2)=O)C1 N1(C(c2c(C)snc2)=O)CCC(NC(=O)CSCc2cccs2)C(C)(C)C1 n1(CCC(C)(C)OC)nc(-c2nc(C(F)(F)F)cs2)nc1C1CC2(CNC2)C1 n1(CC)ccc(C(=O)NCC2CCN2C(C2C=CCC2)=O)cc1=O C(=O)(CCCCC(F)(F)F)N1CC(C)C(NCc2conc2Br)CC1 c1(C(=O)NC2CC(NC(=O)CCc3cnoc3)C2)cccc(Cl)c1Br CCCCCC(O)C(=O)NCCC1CN(C2CCCC2)CCS1(=O)=O Cc1ccc(Cl)cc1C(=O)NC1CC(CCNC(=O)C(c2cccn2C)=O)C1 c12cccc3c1CCN(C3)C2=O.C(C)(C(C(=O)OC)C(=O)OC)COC C1(F)(C(=O)NCC2CC(=C)C2)CCN(C(=O)C(C)SC)C1 C(=O)(CCCC(=O)c1ccc(Cl)c(Cl)c1)NCCNC(C(C)(C)NC(=O)OC)=O CCC(CC(=O)NC1COCC1C(N1CC(OC(=O)N(C)C)C1)=O)OC Cc1ccncc1CNC(C1CC(NC(C2(C)CC3CC3C2)=O)C1)=O c1(C(=O)NC2CC(C)(CNC(=O)C3CC3)C2)ccc(-c2ccncc2)nc1 c1(CN=C(NC(c2ncn(C)n2)COC)NC2CCCC2)ccc(O)c(F)c1 C(=O)(CCCCCN(C)C)NCC1(C)CCC(NC(c2c(C(C)C)cco2)=O)C1 N1(C(C2CC(=C)C2)=O)CC2CC(C)N(C(c3ccoc3CC)=O)C2C1 C=CC(CC)C(=O)N(C)CCOCCN(C(=O)CCCc1cccs1)C c1(CC)cccc(OCC(=O)NCC(C)CNC(=O)CCC2(C#N)CCC2)c1 C1(C(=O)NCCNC(C=C(C)I)=O)Cc2cccnc2C1 CCC(F)(F)C(=O)N1CC2CC2(CNC(=O)Cc2ccc(Cl)cc2)C1 c1(C(=O)NCC(C)NC(C2(CC#C)CCCOC2)=O)ccn2c1CS(=O)(=O)CC2 C(CCC(C(=O)C(=O)C(n1cc(-c2ccc(C(C)=O)c(F)c2)nn1)C)N)OC N1(C(CCC=C)=O)CCN(C(=O)C(C)OCCc2ccccc2)C(CO)C1 CC1CCC=C1C(=O)N1CCC(N(C(=O)Cn2nc(C(=O)OC)cc2O)C)C1.CCO CC1(C(N2CC(O)(C(F)C(N3CC(S(C)=O)C3)=O)C2)=O)COC(=O)C1 N1(C(Cn2c(C)ncc2)=O)CC(CNC(=O)Cn2ccnc2C(C)C)C(C)C1 C1(C(C)(C)C)CCN(C(=O)C(C2CCC2)NC(=O)C=CC2CCC2)C1 C1(NC(CCCCOCC)=O)COCCN(C(C2CC(C(F)F)C2)=O)C1 C(=O)(CS(=O)(=O)CC(=O)N(C1CCCC(NC(=O)CSC(F)F)C1)C)OC N1(C(CSS(C)(=O)=O)=O)CC2(C1)SCCC2NC(C1CC12CCCCCC2)=O C1(OCC(=O)NC23CC(CNC(COC(C)(C)C)=O)(C2)C3)C#CCCCCC1 N1(C(CN(C)CC)=O)CC(F)CC1CNC(c1ccnn1C1CC1(F)F)=O c1(N2CCC(COC(c3cnn(CC(C)C)c3C(F)F)=O)C2)ccc(F)c(Cl)c1 c1(C(=O)NC2C(NC(c3nc(CCC)sc3)=O)C2)cc(C)c2c(c1)CCCN2 C1(C(N(C2(F)C3CCCC23)CC(C)(C)CNC(COC)=O)=O)CCCN(C(C)=O)C1 C1(CNC(CN(C)CCc2cccs2)=O)CCCN1C(=O)COc1ccccc1 N(C1c2ccccc2CC1NC(C1CCS(=O)(=O)C1)=O)C(=O)CCCCO C(CCN=C(NCC1CCCN(C2CCCC2)C1)NCC1(CO)CCC1)OC C1(OCC)CC(N(C)C(=O)NC(C2CCCOC2)CN)C1(C)C c1(C(=O)NC(C2CCN(C(c3cc(O)cs3)=O)C2)C)ccc2c(c1)CCOC2 C1(CC(=O)NCC(CC)O)C(NC(C2CC2C(F)(F)F)=O)CC1O N1(C(c2ccc(C)c(O)n2)=O)CCN(C(C2CC3CCC(C2)C3)=O)CC(C)C1 CC1CN(C(C2CCN(C)C2)=O)CC2(CCN(C(c3cc(CF)on3)=O)C2)O1 CC(C)CCCC(=O)N1CC(NC(=O)Cc2cscc2Br)C(O)C1 C(CCCCC(=O)NC1CC1NC(=O)Cn1ccc(Br)n1)OC C1(CNC(C(C)=C2CC2)=O)CCC(C)CN1C(c1cc(N2CCCC2)ccn1)=O C1(C(N(C)Cc2cc(C)on2)=O)CC2(CCN1C(=O)CC1CCCSC1)CC2 c1(C(=O)NC(COCC)C(=O)NCC(C)N=[N+]=[N-])ccc(C)nc1 C1(NC(c2c(C(C)C)ncnc2)=O)CC2CC1N(C(=O)C(C#N)C(C)C)C2 C1(NC(C(c2ccco2)NC(C2N(C)CCCC2)=O)=O)CC2(CCCC2)C1 c1(C(=O)NC2(CC(n3ccnc3)=O)CCC2)ccc(CNC(=O)CC=C(C)C)[nH]1.CO C(=O)(CS(=O)(=O)CCO)N1CCC(N(C(C(CCC)F)=O)CCO)CC1 C1(C(N2CCC(C)(CNC(c3c(CC)nns3)=O)C2)=O)CC2OC1C1CC21 c1(CC(=O)NCCNC(CC(C)C2CC2)=O)cccnc1OC(F)F N1(C(C2CC(O)(CC#C)C2)=O)CCCC2C1CCCN2C(=O)CC(=C)C CN=c1nc(C(N2CCCOC(CNC(C3CC(CC)=NO3)=O)C2)=O)cc(C)[nH]1 N1(C(CCOCC)=O)CCC(NC(c2cnn(CC(C)C)c2)=O)C(F)(F)CC1 c1(C(=O)NCC23OCCC(NC(c4c(C)ccs4)=O)(C2)C3)ccnc2ncnn12 C=CCCCC(N=c1nc2sccc2c(NCCCS(N)(=O)=O)[nH]1)c1ccccc1 C1(C(=O)NCC2(CNC(C)=O)CC2)CN(C(C)C)CC1C.N12CC(C)(C1)C2=O C1(CS(C)(=N)=O)(COC(C(C)OC2CCCCCC2)=O)CC(F)(F)C1 CC(C)C(C(=O)NCC(O)CNC(=O)CSCCC#N)c1ccc(Cl)cc1 C1(NC(CN2CCC(C)(O)C2)=O)CC(F)CN(C(c2ccc(F)c(N)c2)=O)C1 C1(CNC(C(C)CC2CC2)=O)CCCCN(C(=O)C=Cc2cn(C)cn2)CC1 c1(NCCCC(C)NC(C(C)C2CCOC2)=O)nc(C(F)(F)F)ccc1C#N C1(OC)CC(C(N2CC3CC3(NC(=O)COCP(C)(C)=O)C2)=O)CC1OC CON1CCC(C(=O)NC2C3CCN(C(c4ccc(C(C)C)cn4)=O)C23)CC1 C1(NC(=O)CCNC(C2CCC2)=O)CC2CC1N(C(c1nn[nH]c1Cl)=O)C2 N1(c2ncnc(C)c2Br)CCCC2C1CCN2C(c1ccc(Cl)s1)=O C1(C(=O)NC2CC(OCC)C2)CCC(CNC(c2ccncc2Cl)=O)CC1 C(=O)(CCCCN(C)C)N(CCCNC(CCn1ncc(C)c1)=O)C(C)C Cc1ccc(C(=O)NC(C2(C(=O)NC3(CCF)CC3)CC2)C)cc1 c1(C(=O)NC2CC(N(C(C(C)c3cc[nH]n3)=O)C)C2)ccc2c(n1)OCCO2 c1(C(N2CC(CNC(C(F)=CC)=O)CC2(C)C)=O)ccc2c(c1)NC(=O)CCS2 C1(CNC(C2CC(C#N)C2)=O)(CNC(=O)Cc2cnc[nH]2)CC(F)(F)C1 C1(NC(c2ccc(-c3ccccc3)o2)=O)CN(C(=O)C(F)CC2CC2)CC1O CCCC(C)(O)CC(=O)N1CCC(NC(COC2(C)CC(O)(CO)C2)=O)C1 C#CC1(NC(c2ccc(CNC(c3[nH]cnc3CC)=O)o2)=O)CC2CCCC12 C1(C(=O)NC(CC(=O)OCC)C)C=CCN(C(=O)CC2(O)CCOCC2)C1 C1(C(=O)NC2(CC)CCN(C(c3c(CC)c[nH]n3)=O)CC2)CCC2(CCOC2)O1 c1(C(=O)NC2(CNC(c3c(C)coc3)=O)CC3CCC2C3)cn2ccccc2n1 c1(C(=O)NCCC2(O)CN(C(COCC)=O)C2)ccc(C2CCOCC2)nc1O C1(CNC(COC(C)C)=O)CC2CCC1N(C(C1CC1(F)F)=O)C2 c1(C(N(CC(CC)NC(=O)C(C)Cc2ccncc2)CC)=O)coc(N(C)C)n1 Cc1cc(CNC(=O)CONC(=O)C(O)Cn2cncn2)cnc1C S(=O)(=O)(c1cccc2cnccc12)N1C(C(=O)NCc2cc[nH]n2)CC(O)CC1 c1(-n2ncc(C)c2)cc[nH]c(=NCCCOCCOC2(CO)CCCO2)n1 N1(C(C2CCC(C)(C)C2)=O)CC2CCC2(CC(=O)NC2CCOCC2O)C1 C1(C(=O)NCCC2(NC(C3C(=O)NCC3)=O)CC2)CC2(C1)CC(F)(F)C2 c1(OC)ncc(C(N2CC3CC3(NC(=O)C=C3CCN(C)CC3)C2)=O)cc1F N1(C(C2C(NC(c3c(OC)nsc3)=O)CC2)=O)CCCOC(C2CC2)C1 Cn1cnnc1CCC(=O)NC1CC(NC(=O)CNC(C2CC(C#N)C2)=O)C1 C1(C(=O)NC(C2CC2C(=O)NC2CCC(O)C2)C)(CC)CCCCO1 C1(NC(C2C(NC(C3N(CC)CC3)=O)CC2)=O)C=CCCC1CO C1(NC(C2CC(C)(C)C(=O)CC2)=O)CCN(c2cc(Cl)c(O)nn2)CC12CCC2 CC1(C)CN(C(=O)CN2CCC3CC23)CC1NC(=O)CCC1CCCCO1 N1(C(CCc2ccc(=N)[nH]c2)=O)CCC2C(NC(c3cn(CCO)nn3)=O)CC12 c1(C(CNC(c2cn(C)cn2)=O)NC(C(C)CN(C)C)=O)ccc(F)cc1 CC(C(CO)NC(c1csc(C(N)=O)n1)=O)NC(=O)CC1CC(F)(F)C1 Cc1ccc(F)c(CNC(=O)C=CS(C)(=O)=O)c1.N1(C2CC2)CCC(C(N)=O)CC1 O=S(=O)(c1ccc(N2CCC(CSc3ccncc3)C2)c(Br)c1)N1CC2CC1C2 c1(OC)ccc(C2CC2C(=O)NCCC(C)NC(C2COCCN2CC)=O)cc1 C(C(C)(O)C(C)C)NC(C1(NC(COCCCC)=O)CC(O)C1)=O c1(NC(C2CC23CCN(Cc2cc(F)cc(Br)c2F)C3)=O)ncnc2occc12 c1(C(=O)NCC2C(NC(CC=CC=C)=O)CCC2)cnn(CC2CC2)c1Cl c1(C(=O)NCCCC(C)NC(=O)CC(C)CF)ccnc2c(F)cccc12 c1(C(N2CCC(N(C(C3ON=C(C)C3)=O)CC3CC3)C2)=O)cc(N)c(C)cc1C N1(C(c2cccc(CC)c2)=O)CC2CCC1CN2Cc1nccnc1C Cc1cc(F)c(C(C)NC(=O)C(F)(F)F)c(F)c1.N12CCC(CC1)C(C)C(=O)O2 Cc1nc(CNC(=O)N(C)CC2(CN3CCCC3)CC2)n2ccccc12 Cc1[nH]nc2ccc(C(=O)NCC(C)NC(C3(C)CCCCC3)=O)c(Cl)c12 N1(C(Cn2c(C)nnn2)=O)CC(C)(C)CC1CNC(c1cc(Cl)cc(Cl)c1)=O CC(CC(=O)NCC1(O)CC(CNC(=O)CC2CCC3(CC2)CC3)C1)C(F)F c1(C(=O)NCC2CCCN(C(c3coc(CO)c3)=O)C2)n[nH]c2c1C(=O)CCC2 C=Cn1nncc1C(N1CSCC1C(=O)NC(C1CCCCC1)CO)=O C#Cc1ccc(Cl)c(C(=O)NCCC2CN(C(c3cnc[nH]3)=O)CCO2)c1 Cc1nc(CNC(=O)N(C2CCN(c3ccccc3)C2)C)n(C)c1C C1(CNC(CCCC=C)=O)CCCN(C(C2(C)COC(=O)OC2)=O)CC1 N1(C(CCC(=C)C)=O)CCC(CNc2ncnc(Cl)c2Br)C(C)C1 C(CC(C)(C)C(=O)NC1CC2(C(N3CCCC3CN(C)C)=O)COC1C2)OC C1(N(C(=O)C=Cc2cccs2)CC)CCCN(C(=O)C(C)=C2CCC2)C1 C1(C(=O)NCC2C(OC)CCC2)(NC(=O)CC2CCC2)CCC(C)(C)C1 Cc1nc(CC(=O)NCC2CC(NC(=O)CCC(=O)N3CCOCC3)C2)[nH]c1C N1(C(c2c(OC)scc2)=O)CC(NC(=O)CC2(C)CC2(Cl)Cl)C(F)C1 c1(C(N2C(CNC(COc3ccc(C)cc3)=O)CCC2)=O)cc2ncccn2n1 CC(C)CC(C)(C)C(=O)N1CC=C(C(=O)NCC2COCC(C)O2)C1 N1(C(C(C2CCCC2)NC(C)=O)=O)CCC(C)N(C(c2csc(C)n2)=O)CC1 Cn1c(-c2ccccc2)c(C#N)c(=O)n1C1CCOC1 Cc1cc(NC2CCCC23CN(C(c2nn(C)cc2Cl)=O)C3)ncc1[N+](=O)[O-] C1(C(=O)NCC2C(N(C)C)COC2)CCCCC1NC(C1C2COCC12)=O C1(CCNC(=O)NCC2(CS(C)(=O)=O)CC2)(CCN)CC=CC1 c1(C(=O)OCC)cc(F)cnc1NC(C1CC1NCc1cc(Br)cc(Br)c1)=O CCCCCCCCNC(CCCCCC1CCN(C(=O)CCS(C)=O)CC1)=O C(CCC(N)=O)(C(=O)N1CCC1c1ccccc1F)NC(C)=O c1(C(=O)NCCc2ncc(C)o2)oc(CNC(c2nocc2C)=O)cc1C C1(CC(=O)NCC2CCCC2C(N2CCC3(CC2)CC3)=O)Cc2ccccc2C1 c1(NC(C2SCCN(C(C=COCC)=O)C2)=O)ccc(Cl)c(C(F)(F)F)c1 N1(C(C=CC=CCC)=O)C2CCC1CC(O)(CNC(c1ccc(SC)cc1)=O)C2 N1(CC)C(=O)CN(CCC2CCN2CCNC(c2cccc(C(F)(F)F)c2)=O)C1=O C(=O)(CC(C)(C)C(F)F)N1C(CC)C(C(N2CCN(CCO)CC2)=O)CC1 CC(C)CC(CNC(=O)CSCC#N)NC(c1ccnc(N2CCOCC2)c1)=O c1(N(CC(CCC)C)C)ccnc(NCc2ccc(OCCO)cc2)n1 Cc1nc(C(N2CC(CC(=O)Nc3sncc3C(N)=O)C(C)C2)=O)ccc1Br N1(C(CC2(CNC(c3ccnc([N+](=O)[O-])c3)=O)CC2)=O)CCN2CCCC2C1 C(=O)(CCP(C)(C)=O)NC(C(CO)NC(c1c(SC)nn(C)c1)=O)C CC(C)(C)CCC(=O)N1CC(NC(c2cc[nH]c2)=O)C(CO)C1 N1(C(CCCC(C)C)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC1.C(=O)(C(C)O)OCC C1(C(=O)NCC2C(NC(CCn3c(C)ncc3)=O)C2)CCC(=O)N1C1CC1 CC1CN(C(=O)C(C2CCCO2)NC(C2CS(=O)(=O)C2)=O)C(C)C1C C12(C(=O)NCCCCC)CC(CN(C(C3CCC(CC)O3)=O)C1)C2 N1(C(c2c(C)cno2)=O)CCN(C(=O)C(F)(F)C2(O)CCC2)CC(C)(F)C1 CCCCCC(O)CC(=O)NC1CC(CCn2cc(CC3CCNC3=O)nn2)C1 C1(OCC)CC2(C1)CC2NC(=O)C(CO)NC(c1ccnc(O)c1)=O c1(C(=O)NCC(CCNC(c2ccn(C(C)C)n2)=O)O)c([N+](=O)[O-])c(C)nn1C c1(C(N2CCC(C)C2CNC(=O)C=C(Cl)Cl)=O)cc(Cl)ccc1Cl C12(NC(c3c(C)nc(C)s3)=O)CCC(N=c3[nH]c(Cl)nc4c3CCC4)(CC1)C2 CN1C2CCC1CC(C(=O)NCC1C=CCN1C(c1cc3ncccc3s1)=O)C2 C(=O)(C1COc2cc(C)c(C)cc21)NCCN(C(CCCCN(C(C)=O)C)=O)C c1(C(=O)NC2(C)CC(NC(=O)Cc3ccns3)C2)ccc(C2CCCOC2)cc1 c1(C(=O)NCC2(NC(C(CC)=CC)=O)CCCC2)cc(N)ccc1OCC n1(CC)cnnc1CN(CCCN(C(=O)CC1(C)CC1(F)F)C)C C1(C)(C(=O)NC(CC)CN(C(=O)C(C)NC(c2ccoc2)=O)C)CCCS1(=O)=O Cc1cc(C(N2CC(O)(CN(C(=O)CC3CC(=O)NC3=O)C)C2)=O)cc(O)c1 N1(C(c2cc(C)sc2)=O)CC(C)CN(C(c2ccc3cc[nH]c3n2)=O)C(C)C1 c1(C(=O)NCC(C)CC(=O)NCCN2CCOC(C)C2)ccccc1C#N c1(C(=O)NCC2CC(OC)CN2Cc2c(I)ccnc2F)cccc(C)c1C C1(O)(CCNC(C(N)=O)=O)CCN(C(C2CC23CCC3)=O)C1 C(CCC(=O)NCCCCCNC(=O)Cc1csnn1)OCCOC Cc1ccc(NC(C23CCC(N)(CO2)C3)=O)cc1NC(c1ccccc1)=O c1(C(=O)NC2C(NC(Cn3cc(C(C)O)nn3)=O)COC2)coc2ccccc12 C1(C2(C)CC2)CCC1(c1nnnn1C1CC1)NCc1nnnn1CC1CC1 C1(C(C(=O)NCCCC(=O)OC)N)CCCC(=O)N1 N1(C(CNC(=O)OCC)=O)CCC2(CCC2CNC(c2[nH]c(O)nc2C)=O)CC1 CCCC(C(=O)N(C)CCC1CCCCCC1)c1cccc(Cl)c1 N1(C(c2ccc(NC(C)=O)s2)=O)CCC(CNC(C2(C)CC2(F)F)=O)C12CC2 c1(N2CCC(C(N3CCC(C(C)O)CC3)CC)C2)ncc(C(=O)O)cc1C C1(CNC(CN(C(C)=O)C)=O)CC2(CCN(C(=O)C(O)C(C)C)C2)CO1 C1(O)(CNC(=NCc2n(C(C)(C)C)ncn2)NC2CC2)CC2CCC1CC2 CCC(C)CC(=O)N1CC(CCNC(=O)C(F)(F)CC2CCCO2)C1 N1(C(c2c(OC)ccs2)=O)CC2CC2C1CNC(c1ccc(C2(C)CC2)cc1)=O CN1CCCN(C(C23CCCC2CCN3C(=O)Cn2[nH]cnc2=N)=O)CCC1 c1(C(=O)NC2COCCN(C(C3C(C)(CC)C3)=O)C2)cnn2c(C)cccc12 O=S(=O)(c1cnc(N2CCC(C3CC3)C2)c(Cl)c1)NCC1CC1c1ccccn1 c1(CC)nc(N2CC3C(C(=O)NC45CCCCC4OCC5)C3C2)c(C#N)cc1C c1(C(=O)NC2(c3cn(Cc4c(C)cccc4)nn3)CCC2)ccc([N+](=O)[O-])o1 C1(C(=O)NC(CC=C)CNC(c2c(C)coc2C2CC2)=O)CCOC(C)(C)C1 C1(NC(c2c(C)cc(CCC#N)cc2)=O)CN(C(=O)C(C)N(C)C)CC1C1CC1 N1(CC(N2CC(C(C(=O)N(CC(CC)O)C)O)C2)=O)CC(=O)NC1=O C1(C)(C(=O)NCC(C)N(C(=O)CCc2nc(-c3ccncc3)no2)C)CC1(C)C c1(C(=O)O)cccc(CNc2nc(-c3ccc(Cl)s3)cs2)c1.C12CCN1C2=O c1(N(CCOC)CCNC(c2nnc(C3CC3)s2)=O)ccc(C#N)cc1C Cc1cc(F)sc1C(=O)NCCC1COCCN1C(=O)CCOCCN(C)C c1(CC)c(C(=O)NC2CN(C(=O)C=CC(C)C)CC2(C)C)cnc2cc(O)nn12 c1(NCC(Br)=C(C)C)ncccc1S(=O)(=O)NCC(C)F c1(CN2CCC(c3c(C)cccn3)CC2)cccc2c1OCCC2 Cc1cc(O)c(C(=O)NC(C)CCNC(=O)CCSCC2CCCC2)nn1 N1(C(CN2CC(C)(OC)C2)=O)CCC(CNC(=O)CN2C(C)CCC2C)C(C)C1 c1(C2(C(N3CCCC(n4ccc(C)n4)C3)=O)CCCC2)ccc(F)cc1F C(C(C)C(C)C(=O)N1CC(F)CC1CNC(=O)CCCSC(C)(C)C)OC c1(C(=O)NCCNC(C(C)NC(C2CCC2)=O)=O)ccn(C2CC2)n1 CC(CN(C)C)CN=c1[nH]c(N2CCC3CCCCC3CC2)nc2ccccc12 C1(CNC(C=CSC)=O)CC2(CC2)CN1C(c1sccc1Cl)=O CC1(C)COCC(C(N2CC(NC(=O)C(c3ccc(Cl)cc3)(F)F)C(O)C2)=O)O1 C(=O)(CCC(C)(F)F)N1CCC(C(F)F)(CNC(CCC=CCC=C)=O)C1 C1(C2CCN(C(c3ccc(CCC)cc3)=O)C2)(NC(CCCCC=C)=O)CC1 c1(C(N2CC(CC(=O)NC)N(C(=O)C3=CCSC3)CC2)=O)nccn2ccnc12 C1(C#N)(C(CCC)=O)CCOCC1.C(=O)(C(C)(C)NC(C1COC(C)C1)=O)OC C1(NC(c2ccc(N)c(F)c2)=O)CN(C(=O)CN2CC(=O)NC2=O)CC1C1CC1 c1(C(=O)NC(CN(C(=O)C(=Cc2cn(C)cn2)F)CC)C)cccc(C(C)C)c1 C(=O)(C(C(C)(C)C)NC(=O)CC1(C(=O)NC)CCC1)NC(CCC)CO N1(C(c2c(OC)cncn2)=O)CCOCCC1C(=O)N(C1CCCC1)C c1(-c2ccc(SC)c(F)c2)ccc2cc(C(=O)NCc3ccc(C)cn3)[nH]c2c1 N1(CCC2N(C)CCC2)CCC(=O)N(CCc2ccccc2[N+](=O)[O-])C1=O C1(CNC(C2(COC)CC2(F)F)=O)CN(C(C2CCC2)=O)CCC12CCC2 c1(C(N2CCCCCC2)C(=O)NCCOC)ccccc1OC(F)F N1(C(c2n(CC)nnc2)=O)CCCC(NC(c2ccc(F)c(C)c2)=O)C1C c1(OC)ccccc1CCC(=O)Nc1sc(-c2ccccc2CN(C)C)nc1C c1(C(=O)NC2CC3C(NC(c4c(N)ncc(O)c4)=O)C3C2)noc2ccc(Cl)cc12 c1(-c2nc(CCNC(CNC)C)on2)ccc(C(F)(F)F)cc1 c1(C(CN2CCC2CSC2CCCCC2)OCC)ccc(N2CCCC2)cc1 c1(C(=O)NCCc2cn(CC)nn2)sc(S(N)(=O)=O)c(OC)c1OC C1(C)(NC(c2cc(CC)on2)=O)CCC(NC(C2CC(OC)C2)=O)CC1 c1(C(=O)NCCCOCCN(C(c2c(C)csc2)=O)C)cc(F)cc(C)c1N c1(C(=O)NC2CCN(C(c3cnc4[nH]ncc4c3)=O)C2)coc2c1C(=O)NCC2 C1(NC(c2nc(C(=O)OC)sc2)=O)CN(C(c2sccc2N(C)C)=O)CC1C CC1CN(C(c2cc(CNC(=O)C(C)CC(C)(C)C)[nH]n2)=O)C(C)C(C)(C)O1 C(=O)(C(C)(C)C1CCC1)NCC=CCC(=O)NCC1CN(C(C)=O)C1 C1(C)(NC(C(C)C)=O)CCN(C(c2cc(N3CCC(O)CC3)ccn2)=O)C1 C(=O)(CS(=O)c1cccc(OC)c1)N1CC(NC(c2ccc(SCC)cn2)=O)C1 CCN(OC)C(=O)CNC(C1C=CCCN1C(=O)C(CO)OC)=O c1(C(=O)NC2C(NC(C3(c4c(C)cccc4)CC3)=O)C2)cc2n(n1)CCNC2=O c1(CCOC(C)=O)ccc(NC(N2CCC(N3CCOCC3)C2)=O)cc1 C1(C)(OC)CC(NC(=O)NC(c2ccc(C)c(F)c2)C2CCOC2)C1(C)C C12(OC)CCC(C(=O)N(C)CCNC(c3nnn(C)c3N)=O)(CC1)CC2 CCCC(CC)C(=O)NCC1CCCN(C(c2cnc(O)cc2O)=O)C1 c1(N2C(C)CC(CNC(c3ccc(SC)o3)=O)C2)ccc([N+](=O)[O-])c(O)n1 Cc1ccc2occ(C(=O)NC(CNC(=O)C=C3CCC(C)C3)C(C)C)c2c1 C(c1ccc2c(c1)OCO2)=CC(=O)NC1(CC(=O)NC(C)C(C)NC(N)=O)CCC1 c1(C(=O)NCC2CC(C)N(C(=O)Cc3nccn3C)C2)cccc2nc(S)oc12 Cc1cn2nc(C(=O)NC3CCN(CC4CC(C)C4)CC(C)(C)C3)cc(C)c2n1 N1(C(CC(C)(CO)C2CCC2)=O)CCCCCCC1NCCNC(C(CC)C)=O N1(C(C2=NOC(C)C2)=O)CCC2(C1)CN(C(c1ccc(C(O)CF)cc1)=O)C2 c1(C(=O)NCC2C(CNC(C(F)=CCC)=O)C2)cc(C(N)=O)no1 c1(CC)cc(C(=O)NCCC(C)(C)NC(=O)CC2CC(O)C2(C)C)cc(F)c1 CC1=C(CO)C1CNC(C1CCC1CNC(c1ncc[nH]1)=O)=O c1(C(=O)NC(C)CCc2cccc(C(F)(F)F)c2)n[nH]c2c1CCC(=O)C2 c1(SC)ccc(C(=O)NCC2(NC(=O)CCc3nccn3C)CCC2)c(C)n1 N1(CCCC)CCN(C(C2CN(Cc3ncccc3Br)CCS2)=O)CC1 C(N=c1[nH]cnc2ccsc12)C1N(C(=O)COCCc2ccccc2)CCCC1 C1(CC(=O)NC(CC=C)CC=C)CC(C)(C)CN1C(=O)Cc1ccn(C)n1 c1(N2CCC(CC(C)C)CC2)nc(=NC2CCCC(C)C2)[nH]c2c1COC2 N1(C(c2c(COC)cc[nH]2)=O)CCN(C(=O)CN2CCNC2=O)CC1CCO S(=O)(=O)(c1ccc(N(C(CC(C)C)C(N)=O)C)cc1Cl)N1C(CCC)CCCC1 N1(CC(=O)NC2CN(C(C(C)c3ccco3)=O)C2)CCCCC1C Cc1nc(C(N2CC(CO)(NC(c3nc(O)c(C)s3)=O)C2)=O)n(C)n1 N1(C(c2cc(CNC(CC3OCC(C)(C)C3)=O)no2)=O)CC2C(C1)C2(C)C C(=O)(C(C(=O)NC(C1CN(C(C2CC3(CC3)C2)=O)CCO1)C)OC)OC c1(C(N(CC(C)CNC(=O)C(C)(C)C(C)O)C)=O)ccc([N+](=O)[O-])c(Cl)c1 C#CCC(C)(C(=O)NCCOCCO)NC(=O)C(O)CC1CC1 C(C(C)NC(N(C1(OC(C)(C)C)CC1)C)=O)(C(F)(F)F)OC c1(C(=O)NCC2CN(C(CC(CC)SC)=O)C2)nc2sc(C)cn2c1C c1(C(=O)NCC23CC(NC(CS(N)(=O)=O)=O)(C2)C3)c(Cl)ccc(Cl)c1O C12(C(=O)Nc3nccc(-n4ccc(C)n4)n3)CCN(C1)S(=O)(=O)C2 CC(C)CCCCCC(=O)N1CCC2CCCC12NC(=O)CC1=CCN(C)CC1 C1(C#N)(N(C(C(COCC=C)c2ccccc2)=O)C)CCCOC1 C1(CNCC2(C(N(OC)C)=O)CCCC2)CC(C)(C)CCO1 Cc1cc(N)c(C)nc1C(=O)NC1CCN(C(=O)C(c2ccncc2)C)C1C N1(C(Cc2nnc(C)o2)=O)CCN(C(C2CN(C)CCN(C)C2)=O)C2COCC12 c12ccc(NC)c(c1)O2.C1(C(=O)OC)C(CC(=O)OC)CCN1OC.C1(CF)(C)CC1 c1(NC(CCN(c2ccncc2)C)=O)ccc2c(c1)OC1(CCCCC1)O2 C1(C(N2CCCC(CCNC(=O)CC3(C)CC3)C2)=O)(COC)CCC(=O)N1 Cc1cc(C(=O)NCCC2CN(C(=O)C(O)C3CC3)CCO2)nn1C(C)(C)C C1(CC)CCCN(C(c2cnn(C)c2)=O)C1C(N1CCSCCC1C)=O C(=O)(C(C)(C#N)CC(=O)OC(C)(C)C)NCCN(C(=O)C(F)C1CCC1)C(C)C C1(C(=O)NC(C(C)C)CNC(C2(Cc3ccccc3)CC2)=O)CCS(=O)(=O)N1 c1(C(N2CCC(CC=C)(NC(C3CC(C)(C)C3)=O)C2)=O)c(F)cccc1Cl N1(C(CC(=C=C)C)=O)CCCN(C(=O)C(c2ccc(O)cc2)=O)CC1CO c1(C(=O)NCCN(CC(=O)NCC(F)(F)F)CC)cccc(C)n1 c1(C(=O)NCCC2(O)CN(C(c3n(C)nc(O)c3)=O)C2)nnc(O)cc1O C1(OCC=C)CCN(C(=O)CC(C)NC(c2cscn2)=O)C1 CCC(C)(C)C(C)CC(=O)NC1(C)CN(C(c2ccc(NCC(C)C)nc2)=O)C1 C(=O)(CC(C(F)(F)F)c1ccccc1)N1CC(NC(CSC(C)C)=O)C(C)C1 C1(CN(C(=O)COC)CC)CCCN(C(=O)CCSc2cnsc2)C1 C1(CNC(C(CC)n2nccc2C)=O)CN(C(=O)CCCC(N)=O)CCN1C Cc1ccc(NC(=O)C(C2CCN(C(=O)CC3CCC(C)(C)O3)C2)F)c(CO)c1 N1(C(C(CC)n2nccc2C)=O)CCN(C(=O)CC2OCCCO2)CC1CF Cc1cccc2cc(C(=O)NCCOCCNC(c3ccc([N+](=O)[O-])[nH]3)=O)oc12 CCC(F)(F)CC(=O)NC(C)(C)C.C12CC(C1)CC(=O)OCCC1(CC1)NC2=O N1(C(C(C=C=C)C)=O)C2CCC1CN(C(c1cnc3n1CCCC3)=O)C2 C1(NC(C(COC)C)=O)CN(C(=O)Cn2nccc2C)Cc2ccnn2C1 C1(C(=O)NCC(CC)NC(c2ccn(CCF)n2)=O)CCCC(=O)CC1 Cc1ccc(O)cc1C(=O)NCC1CN(C(=O)CC2CC2)CC1C(F)F c1(C(=O)NC2(CO)CCN(C(C(C)C3CCC3)=O)CC2)ccc2n[nH]cc2c1F Cc1cc2ncn(CC(=O)N(CC(C)NC(=O)C(=O)CCC(C)C)C)c2cc1C C1(CC)CCC(C(=O)NCC2(OC)CN(C(C3CC(O)C3)=O)C2)C1 N1(C(c2c(CC)csc2)=O)CC2CCC2(CC(=O)NCCc2ncon2)C1 C1(CC)CN(C(C2C3CC2N(C(=O)C(C)(C)n2cncn2)C3)=O)CCO1 N1(C(COCCC#C)=O)CCCC(CNC(=O)C2=CCCC2C)CC1 C(=O)(C1CCCc2nncn21)NCCC(C)N(C(c1c(N)cnc(SC)n1)=O)C C1(NC(CC(CC)OC)=O)CC1C1CCN(C(=O)C(C)=C2CCCC2)CC1 C1(C(=O)OCC)CC2(CCC2)CN1C(c1ccc(OCC)c(C(F)(F)F)c1)=O CC(CC(C)(F)F)C(=O)NC1CCN(C(c2cc(N(C)C)ccc2Cl)=O)C1 CCN=c1[nH]c(C)c(C(N2CCC(NC(C3(CCS(N)(=O)=O)CCC3)=O)C2)=O)s1 c1(CCNC(N2CC3C(C(=O)OC)(CNC3)C2)=O)nc2ccc(F)cc2[nH]1 N1(C(=O)Nc2cccc(SCC)c2)Cc2ccc(Br)cc2OC(C)C1 C=Cc1cccc(-c2cnccc2C(=O)N(C2CCS(=O)(=O)C2)C(C)C)c1 N1(C(c2cnc(OC)nc2C)=O)CC(NC(=O)C(C)N(C)C)C2CCCCC12 N1(C(C2CCCC3CCCN23)=O)CCCC(O)(C2(C(=O)O)CCC2)C1 C1(NC(CNC(N)=O)=O)COC2(C1)CN(C(C1CCCS1(=O)=O)=O)C2 Cc1ncc(NC(=O)CC2CCN(C(=O)CC34CCC(CC3)C4)C2(C)C)c(C)n1 S(=O)(=O)(c1ccc(Br)cc1F)CC1(CNC(=O)OC(C)(C)C)CC1(F)F c1(C(=O)NC(CNC(CCC(=O)NC)=O)C(C)C)cc(C)c(F)cc1N C1(N(C(c2c(C(=O)CN3CCCC3=O)cccc2)=O)CCO)CC2C(O)C(O)CC12 C1(C(=O)NCC2N(C(CN(C3CCCC3)C)=O)CC2)CCC12CCOCC2 C(=O)(C(C(C)(C)C)N(C)C)NCC(CC(C)C)NC(CCNC(C(C)OC)=O)=O c1(C(=O)NCc2c(OC)ccnc2)cc(NC(N)=O)ccc1Cl C1(NC(c2cnc(CC)[nH]2)=O)CC12CC(NC(C1CC1C1CC1)=O)C2 C(N=c1[nH]cnc(C)c1Br)C1CCC(NC(C(CC)CCOC)=O)C1 N1(C(c2cc(Cl)ncc2NCc2ncc(Br)cc2F)=O)CCn2nccc2C1 c1(CC)c(C(=O)Nc2csnc2C)ccn1C.C1=CCN(C2CC2)C1=O Cc1nn(CCF)cc1NC(C1(CCNC(C2CCCS2)=O)CCCC1)=O C1(C(=O)NOCc2cn[nH]c2)(CC=C)CCN(C(=O)CSC(C)(C)C)C1 C1(CNC(c2n(C)c(S)nc2)=O)CC(NC(c2cnn(C3CC3)c2)=O)C12CCC2 c1(CN(C(=O)CNC2CCC(C)(O)CC2)C)ccc(Br)cc1Br Cn1c(C(=O)NC2CCCC(NC(=O)CCSCc3nnnn3C)C2)nnc1S C1(C(=O)NCCN(C(C2CN(CCC)C2)=O)CCC)CSC(c2ccccc2)=N1 N1(C(CCN(CCC)C)=O)CCCC(O)(CCNC(c2ccccc2OC)=O)C1 c1(C(N2CC3(N(C(c4c(CC)nn[nH]4)=O)CC3)C2)=O)cc2ccncc2o1 C1(NC(c2c(CC)cncc2)=O)CN(C(c2cccc(SC)n2)=O)C2(CCC2)C1 C(N=c1cc(C#N)nc(C)[nH]1)C1CN(C(C2(C(=O)OCC)CC2)=O)CC12CC2 c1(C(=O)Nc2ccsc2C2CCCCN2)nc(Br)ccc1OC(F)F C#Cc1cc(C(N2CC(O)CC2(C)C(=O)NCC2CC2Cl)=O)ccc1C C(=O)(NNC(=O)N1CCCC(C(C)N(C)C)C1)c1cc(OC)n[nH]1 C1(C(=O)Nc2ccc(OC)c(F)c2)CC2(CCC2)CN1C(=O)C(F)=CC1CC1 C1(c2cn(CC)nc2)CN(C(C2(SC)CCSCC2)C(=O)NC(C)(C)C)CCO1 N1(C(C(C)C2CC2)=O)CC2(CCN(C(=O)C(C)(C)S(C)(=O)=O)CC2)CC1C C1(C(=O)NC(C)CCNC(c2cn(C3CC3)nn2)=O)CN(CP(C)(C)=O)C1 c1(-c2c(C(N(CCNC(c3occc3F)=O)CC)=O)c[nH]c2)ccc(C)cc1 N1(CCC(N)=O)CCN(CC2CC(=O)N(CC(F)(F)F)C2)CC1 C(CC(C(=O)NC1CC=C(C)CC1)NC(=O)Cc1ccoc1C)OCC c1(C(=O)NCC2(CNC(c3c(CC)nco3)=O)CCCC2)cncc(Cl)c1 C(C(CNC(=O)CC1COCCOC1)C(F)(F)F)NC(CC1N(C)CCOC1)=O C1(CC)CCCC(C)N1C(=O)NCC(=O)N(c1ccccc1C)C C#CC1(C(=O)NC(C)CN2CCCC2=O)CN(C(=O)C2=CCCC2)C1 C1(NC(CCN(C(CCC)C)C)=O)CCN(C(=O)CCc2cncc(C)c2)CC1 c1(CNC(C2(CC)CC2)=O)ccc2c(c1)CCN(C(=O)CC1NC(=O)NC1=O)C2 CC(O)C(C)(C)CNC(C1(NC(C2CN(C(N)=O)C2)=O)CCSC1)=O c1(CC)cccc(C(=O)NC(CO)C(C)NC(c2nc(C)oc2C)=O)c1 c1(C(=O)NC(C(C)NC(=O)C=Cc2ccsc2)(C)C)sc(Cl)cc1Cl CC1COc2ccc(C(N3CC4CCCC4(NC(C45CC(F)(C4)C5)=O)C3)=O)cc21 Cc1[nH]c(=NCc2cc(OC(C)C)c(O)c(Br)c2)sc1C(=O)NC1CC(O)C1 CC1CNc2c(C(=O)NC3CC3CNC(=O)C(F)=C3CCC3)cnn2C1 N1(C(C(C)NC(=O)NC)=O)CCC(NC(=O)CCn2ccnc2C)C(C)C1 C1(C)(NC(CC=CCC)=O)CCN(C(C2CCC(OC(C)=O)C2)=O)CC1 N1(C(c2onc(CC)n2)=O)CCOC2(CCN(C(c3cncc(Cl)n3)=O)C2)C1 N1(c2cncc(OC)n2)C(=O)NC(c2ccc(Br)cc2)C1=O CC1=NS(=O)(=O)NC=C1C(=O)NC1CCN(C(C23CC2COC3(C)C)=O)CC1 N1(C(Cn2nc(C)oc2=O)=O)CC(CNC(C2(C)COC(=O)C2)=O)CC1(C)C N1(C(c2c(OC)c(Cl)c(Cl)cc2)=O)C2CCCC1CC(=O)NC2 c1(C(=O)NCCN(C(CSCC=C)=O)C)ncnc(O)c1Br N1(C(C2=NOC(C(C)(C)C)C2)=O)CC2(C1)SCCC2NC(=O)CCS(N)(=O)=O c1(CC#C)conc1CC(=O)N(C1CC(C#N)C1)CC(=O)NC(C#C)C(C)OC c1(N(C)CC2CCCCC2)nc2ccc(S(=O)(=O)N(C)CC3CC3(F)F)cc2s1 Cc1ncc([N+](=O)[O-])cc1C(N1CCC(CNC(=O)C(=O)C(F)(F)F)CC1C)=O c1(C(=O)NCC2C(CNC(C(CC)O)=O)C2)cc(F)cc(F)c1O C(=O)(C(Cc1cc[nH]n1)NC(C1CN(C(N)=O)C1)=O)NCC(C)(O)C1CCCC1 CCS(=O)(=O)CC(=O)NC(CC1CC1)C(=O)NC(C)Cc1nn[nH]n1 c1(C(N2C(CNC(C3CC4C=CC3C4)=O)CC(OC)C2)=O)ccc2c(c1)COC2 CC1(C)CC(C)(NC(=O)CC2CN(C(C3CCC3(F)F)=O)C(C)(C)C2)C(=O)O1 Cc1nsc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCCc2cnn(C)c2)c1N C(C(=O)N(C)CCNC(=O)CCc1c(C)noc1Cl)(C(C)(C)C)NC(C)=O C(C(=O)NNc1ccccc1S(C)(=O)=O)Oc1c(-n2cnnc2)ccc(C)c1 N1(C(C(F)=CC)=O)CC=C(C(=O)NC2(CC3CC3)CCC2)CC1 c1(C(N2CCC(CCNC(=O)CCOC3CCCC3)C2)=O)ccc2[nH]ccc2n1 C1(NC(c2c(C)cnn2C)=O)CC2CC1N(C(=O)C(O)Cc1cn(C)cn1)C2 C1(C(N(C2CN(C(=O)CCCc3ccncc3)C2)C)=O)CC(F)C(=O)N1 N#Cc1c(-c2cn(CCCC(=O)NCc3ncc(F)cn3)nn2)cccc1N C(=O)(C#CC1CCCOC1)N1CCCC(NC(CCc2ccc(C)s2)=O)(CO)C1 C#CC1C2CCC(C2)N1C(COCC)C(=O)Nc1ccccc1 N1(C(C(c2n(C)ncc2)(C)C)=O)CC(NC(=O)Cn2cnnc2O)C(O)C1 C1(c2cn(CC)nc2)CS(=O)(=O)CCN1C(=O)SC1CCC(C(C)C)CC1 C=CC(C)(CC)C(=O)N1CC=CC(NC(=O)C=Cc2cn(C)nn2)C1 N1(C(CC=C)=O)CC(C(=O)N(C(C)C(=O)NC)C)C(F)(F)C1 C1(C(C(=O)N(CC(C(C)C)C)C)C)CCN(C(=O)Cc2ccns2)CC1 C1(CC(=O)NC)CN(C(=O)CC(C)CF)CCN1C(c1cc(N)c(F)cn1)=O C1(C(N(C(CNC(c2nc(CC)sc2)=O)C)C)=O)Cc2cc(Br)ccc2O1 C1(OC)CN(C(=O)CC(C)(C)O)CCC1NS(=O)(=O)Cc1ccc(Cl)nc1 Cc1cc(C(=O)NC2CCC(CNC(=O)CC3(C)OCCO3)C2)sn1 C1(NC(C2N(C(CC)=O)CCCC2)=O)CC2CN(C(=O)C(C(C)C)OC)CC2C1 C1(C2CCN(C(C(C)C)=O)C2)CN(C(c2c[nH]nc2C2CCC2)=O)CCO1 N1(CC)CC(C)N(C(=O)C(CNC(=O)Cc2cnnn2C)CC2CC2)CC1C C(CC(C)(C)C)(C(=O)N1CC(F)(F)CC1(C)CNC(c1cocc1C)=O)OC C(C)(CNC(c1c(C)ncn1C)=O)(C(C)C)NC(CC1(OC)CCCC1)=O C1(CC(=O)N(C)CC2(NC(CCC=C(C)C)=O)CC2)CCCC(C)O1 N1(CC(=O)NC2CCN(C3CCOCC3)C2=O)C(=O)NC(c2ccc(F)cc2)C1=O CCC(C)C(C)(O)CNC(=O)C(O)CCNC(c1cc(C#N)n(C)n1)=O c1(CC(N2C(CNC(C3(C)CCCC3)=O)CCCC2)=O)ccc2c(c1)CCC2 c1(C(N2CC(CNC(c3c(C)cc(N)cc3)=O)C2)=O)cccn2c(O)nnc12 Cn1ncc(C(N2CCOC(CCNC(c3cc(Cl)ccc3F)=O)C2)=O)c1C#N c1(OC)nc2ccc(Cl)cc2c(=NCC(F)(F)Cl)[nH]1.CCS(=O)CCSC CCS(=O)(=O)c1ccc(CC(=O)NC23CCC(CC2)N(C(=O)C(C)(C)F)C3)cc1 N1(C(CCCCC=CC)=O)CCC(C2CC2)C1CNC(=O)CCc1cccs1 N1(C(c2c(C)cc(C)nc2)=O)CC2CCC(NC(C3CC(F)C(=O)N3)=O)(C2)C1 c1(OC)ccc([N+](=O)[O-])c(C(N2CC(NC(c3sccc3Cl)=O)C2)=O)c1 C=CC(C)CC(=O)NCc1cncc(C(=O)NCc2cc(C(C)C)n[nH]2)c1 Cc1ccc(O)c(C(=O)NC2CCN(C(c3c(C)nn(CCO)c3C)=O)C2)n1 c1(C(N2C(CCNC(=O)COCC3CC3)CCC2)=O)nc2ccccc2[nH]1 Cc1ccncc1N1CCC(C2CCCCN2C(=O)CSC(F)F)C1 N1(C(C2(O)CCN(Cc3cc(C(C)C)no3)CC2)=O)Cc2cccc(O)c2C1 CN1C(=O)CCC1C(=O)NCC1CCCC1NC(c1ocnc1C1CC1)=O c1(OC)cncc(C=CC(N2CCC(NC(=O)C(C)C3CC3)C(F)C2)=O)c1 N1(C(CCCCCOC)=O)CCN(C(c2ncc(C#N)cc2Cl)=O)CC12CCC2 C12CN(CCC1(F)F)C(=O)CC1CCCC(C1)N2.C(C)(C)(C)OC(=O)OC CC1(C(=O)NC(C2CCCCC2)CNC(c2nc(=N)cc[nH]2)=O)CCC(=O)N1 c1(C(N(C2CCN(C(=O)CNC(=O)OC(C)(C)C)C2)C)=O)ccncc1 Cc1cc(Cl)cc(C)c1NC(=O)C(=O)NCC1CC(Cn2cccn2)C1 CC(C)CCC(O)C(=O)N1CCC(NC(c2cncc(C(N)=O)c2)=O)CC1C C1(CNC(c2c(C)nc[nH]2)=O)(NC(c2ccc(C(C)(C)C)[nH]2)=O)CC2CCC1C2 C=C(C(=O)N1CC(NC(C2(C(C)C)CCC2)=O)C(F)C1)C(F)(F)F c1(C(=O)O)cccc(CN2CC3CN(C(=O)Cc4cccnc4)C3C2)c1[N+](=O)[O-] S(=O)(=O)(c1cc(C(=O)O)ccc1F)NC(c1ccc(N(C)C)cc1)C1CC1 C12(NC(CC(C)SC)=O)CCC(CNC(=O)CCn3cc(C)cn3)(CC1)OC2 c1(OC)ccc(C(=O)NCCCN(C)C(C23CCCC2C3(F)F)=O)c(N)c1 n1(CC)ncc2c1CCCC2NC(=O)CCc1nc(-c2ccc(F)cc2)no1 N1(C(C2CCCSC2)=O)CCC2CCN(C(=O)Cn3ncc4ncccc34)C2C1 c1(NC(=O)C(n2cc(C(C)OCCOC)nn2)C)ccc(C(C)SC)cc1C CC#CC1CCN(C(=O)CCOCCNC(c2cc(C(F)F)[nH]n2)=O)C1 CCC(C)CCCCC(=O)NC1(CNC(c2ccc(C)s2)=O)CC1 c1(C(=O)NCCC2N(C(CC(CC)(C)C)=O)CCSC2)cc2cc[nH]c2cn1 c1(C(=O)NCC2C(NC(c3cnc(C)[nH]3)=O)CCC2)c(C)cccc1N C1(NC(CC2CC(OCC)C2)=O)CCCN(C(=O)Cc2ccc(Cl)c(F)c2)C1C N1(CCCN2CCN(C(c3c(C#N)ccs3)=O)CC2)CCCC(N=[N+]=[N-])CC1 C1(NC(C(C)NS(C)(=O)=O)=O)CCC2CN(C(=O)C=Cc3ccncn3)CC12 c1(C(C)OCCOCCOCCNCC(=O)C(=O)OC(CC)C)ncccn1 C1(CCC)(NC(=O)C=Cc2cnc[nH]2)CCCN(C(c2cc(CC)nn2C)=O)C1 N1(C(C(CNC(=O)OC(C)(C)C)N(C)C)=O)CC(O)Cc2ccccc21 C1(NC(C(C#N)C2CC2)=O)CS(=O)(=O)C2CN(C(c3cccnc3O)=O)CC12 N1(C(C(CC)(C#N)CC)=O)CCC2(CC1)CN(C(=O)CC=C(Cl)Cl)CCO2 N1(C(CSC(C)C)=O)CCC2(CC1)CCN(C(C1CC13CCC(F)(F)CC3)=O)C2 C1(C(N2CCCC(N(C(=O)Cc3ccn(C)n3)C)CC2)=O)CC2CCCCCC12 c1(OCC(N2CCCC(N(CCF)C(c3cn[nH]c3)=O)C2)=O)cc(F)cc(F)c1 CC1(C)CCC(CNC(=O)CN2CSCC2=O)N(C(C23COCC2C3)=O)C1 c1(SCc2cccc(OC)c2)nc(C)c(C(=O)NC2CC2C(F)(F)F)s1 C(=O)(C(CC(C)(C)C)NC(=O)CC(O)CC(C)C)NCCc1c(C)ocn1 CCCCC(C(=O)N1CCC(C)(C)C1CNC(=O)CCC(=O)OCC)C(C)C c1(C(=O)NC2CCC2NC(C2CCN(C3COC3)C2)=O)cccc[n+]1[O-] C1(NC(c2ccc(Sc3ncccn3)o2)=O)CC2CN(c3ncncc3I)CC12 C(=O)(C1CCCc2scnc21)N1CC(N(C)C(C2(C)CCC(=O)N2)=O)C1 S(=O)(=O)(c1ccccc1)NCCC(F)(F)F.N12CCCN(CC1)CCC2=O c1(C(=O)NCC(CNC(c2n(CC=C)ccc2)=O)O)cc(C2CCCO2)n(C)n1 C(=O)(CC(C)C(C)(C)NC(c1ncncc1N)=O)N1CCC(CCOC)C1 C1(CNC(C(CC=C)C)=O)C(O)C(O)CN1C(c1nc(Cl)sc1C)=O CC(C)C(C)(O)C(=O)N1CCC2C(C(=O)NCCC(C)F)C2C1 N1(C(c2onc(C)n2)=O)Cc2nccn2CC(NC(=O)CC2CCCCC2C)C1 c1(SC)cnn(C)c1C(N1CCC(CO)(NC(=O)C=C(C)Cl)C1)=O N1(C(C(C)CC2CC2)=O)CC(CNC(c2ccncc2F)=O)OC2(CCC2)C1 C(=O)(C(C)(C)CC=C)NC(CNC(C1(CC#C)CCC1)=O)C1CCC1.C(=O)OC c1(N(CCCNC(=O)C(C2CCCCCCC2)O)CC)cc(O)nc(C2CC2)n1 Cn1nccc1C=CC(=O)NCc1ccc(C(=O)NCCNC(=O)CO)cn1 N1(C(CC(OCC)OCC)=O)CC(NC(=O)CCSC)CC(C)(C)C1 c1(OC)ccc(CNC(C2CC2C(=O)Nc2ccc(F)c(C#N)c2)=O)c(F)c1F C1(C(=O)NCC(CCCC)NC(=O)Cc2cc(C)cc(C)c2)CC(S(C)(=O)=O)C1 N1(C(C(C(C)C)OCC)=O)CCCC(CNC(c2nncn2CC)=O)CC1 C1(NC(c2cc(COC)sc2)=O)CC2CC(C1)N(C(C1CSC1)=O)C2 C#Cc1ccc(C(=O)N(C2CN(C(=O)Cn3cccnc3=O)CC2F)C)cc1C c1(NCC2(C)CC2Br)ccc(S(=O)(=O)N2CCCCCC2)cc1Br C1(C2CC2)(C(=O)NC2CCN(C(c3nn(C(CC)CC)c(C)c3)=O)C2)CC=CC1 n1(CC(=O)NCC2(CCNC(c3cc(=O)cc(Cl)[nH]3)=O)CC2)ccc(O)nc1=O C1(N(C(C2(COC)CN(C(C=CCCC)=O)C2)=O)CC)COCC1C1CC1 C1(N=[N+]=[N-])(C(=O)NC2C(C)NC(=O)CC2)CCN(C(=O)Cc2ccccc2F)C1 c1(NC(CC)=O)cncc(C(N2CC(C(C)NC(c3cnc(CC)s3)=O)C2)=O)c1 c1(C(=O)NC(CNC(c2cccc(CNC(C)=O)c2)=O)C)ccc(F)cc1F N1(C(Cn2c(C)csc2=O)=O)CC2CN(C(C3CCC(=O)N(C4CC4)C3)=O)CCC12 c1(OC)cnc(N(C2CCNCC2F)C(c2sc(C)cc2N(C)C)=O)nc1 N1(C(c2cnon2)=O)CCOC(C2CN(C(c3cc(O)ncn3)=O)C2)C1 C1(C(N2CC=C(C)CC2)=O)CN(C(c2ccccn2)=O)CC(C)O1 c1(C(=O)NCC2C(C(=O)NCC(C)SC)CCC2)cn(C)ccc1=O c1(C(N2CCCCC(NC(C3C(C=C)C3)=O)C2)=O)ccc2ccsc2c1 N1(C(CSCC=C)=O)CC(C2CCN(C(=O)CCNC(=O)CC(C)C)C2)C1 Cc1oc2cc(C(=O)NC(CNC(C3CC(C(F)F)C3)=O)CO)[nH]c2c1C c1(C(C(=O)NC2(CNC(C(C(CC)O)C)=O)CCC2)=O)c[nH]c2cc(F)ccc12 N1(C(CCNC(CC(C)C)=O)=O)CC2CC(NC(=O)Cc3cnn(C)c3)C1C2 c1(C(=O)NC2(CO)CCN(C(CCCCC)=O)C2)cc(Cl)cc(Cl)c1F Cc1ccc2oc(N3CC4CCCC(NC(C5CC(C)(F)C5)=O)C4C3)nc2c1 C1(C(C)NC(c2cn(CC)nn2)=O)CN(C(=O)CCCCNC(N)=O)CCO1 CCCCC(C(=O)NCC1(C)CCCN1C(c1ccccc1OC)=O)C(C)C Cc1cc(=NCc2nncn2C2CC2)[nH]c(C)n1 C1(C)(C(C)C)CCN(C(=O)C(C)Oc2ccc(N3CCCC3)cc2)C1 C1(NC(C=CC)=O)COCCC1NC(c1ccc(C)nc1)=O c1(C(=O)NC2CCC(NC(CS(=O)(=O)NC)=O)C2)cc2c(s1)CCCC2 c1(OC)cccc(CC(=O)NC2CN(C(=O)CCc3cncs3)C3CC23)c1 C1(CCC)(NC(c2sccc2C)=O)CCCN(C(=O)C(C)(C)N(C)C)C1 C(CCCC(=O)NC(CO)C1CCC1)NC(C=CC(C)C)=O c1(C(=O)NCCCN(C(C2CCCC2C2CC2)=O)CC)cc(N(C)C)ccc1N c1(CC)[nH][nH]c(=NC(=O)N2CCN(C)CC2CC)c1-c1nn[nH]n1 c1(C(=O)NCC2(Cn3cc(CO)nn3)CC2)c(O)ccc(Br)c1Cl O=C(CCCNC(=O)C(N1CCCC1c1nccs1)=O)Nc1ncc[nH]1 N1(C(c2cc(=NC)[nH]cc2)=O)CCC(NC(=O)C(C)C2CCOC2)C12CCCC2 Cc1[nH]cc(C(=O)NC2CCCCCN(C(C3(F)CCOC3)=O)C2)c(=O)c1Cl Cc1cc(C(=O)NC(CNC(=O)Cc2cc(F)ccc2O)C2CC2)c(F)cc1Cl N1(C(CCOC)=O)CCC(NC(C2CCN(C)C2=O)=O)CC(C)(C)C1 C(=O)(C(F)CCC(C)C)N1CCC(C(=O)NCC(CC)(C)C)(C(C)C)C1 N1(C(C2(CC(C)=O)CC2)=O)CC(C(N2CCC2(C)C(C)C)=O)CCC1(C)C N1(C(CC(=O)NCC#C)=O)CCC(C(=O)NCCC(C)CCC)C1C.C1(C)CC1 N1(C(c2cc(C)no2)=O)CCC=CC1C(=O)NC(C)Cc1ccco1 c1(C(=O)NC2C(C)N(C(c3cc(CCO)on3)=O)CCC2)ccc2ccsc2c1 N1(C(CCCOCC=C)=O)CCN(C(=O)C2=NOC(C)C2)CC(C)(F)C1 c1(CC)ccccc1C(CNC(=O)C(C)n1ccnc1)NC(=O)CNS(N)(=O)=O C1(NC(CCCc2c(C)ccs2)=O)CCN(C(=O)C(C)N(C)C)C(C)C1 C1(NC(C2(C=C)CCOCC2)=O)CCC2CN(C(=O)C3=CCCOC3)CC2C1 c1(CC)nc(C)c(C(=O)NCCOC2CN(C(C3(C4(C)CC4)CC3)=O)C2)o1 C1CCC2(N3C(C)C(=O)NC3=O)CC12.C(=O)(CSC(C)(C)C)OC.C(=O)O.C(C)=O c1(C(=O)NC(C)CNC(C2CC2C2CCCO2)=O)ccccc1N1CCOCC1 C#Cc1cncc(C(N2CCC(O)(C(C)NC(c3csc4nccn34)=O)C2)=O)c1 C1(NC(CCCCC)=O)CCN(C(C2CCN(CC(F)(F)F)C2)=O)CC1O c1(-n2c(C)ncn2)ccc(NC(c2ccc(C3(C)CCO3)cc2)=O)cc1 N1(C(c2csc(O)n2)=O)CC2OCCN(C(c3cccc4cncn34)=O)C2C1 c1(N(C)C)ccc(NC(=O)CCC2(NC(C3(O)CCSCC3)=O)CCC2)cn1 c1(C(N(CCNC(c2ccn(C)c2)=O)C2CC2)=O)cc(O)nn1C c1(C(N2CC(C(=O)NC3CCC(F)(F)C3O)(COC)C2)=O)cccc2nn[nH]c12 c1(OCC(=O)N(C2CC3CN(C(CCC)=O)C2C3)C)ccc(C(F)(F)F)nc1O c1(C(N2CCC(C(C)(C)NC(c3cnn(C)n3)=O)C2)=O)cc(O)cc(=O)o1 C=CC1(NC(=O)C(C)CN(C(=O)C(C)(COC)OC)C)CCCC1 C1(C(=O)NC2CC(C)(NC(c3cc(C(CC)C)no3)=O)C2)CCS(=O)(=O)N1C C1(C(C)(C)C)CN(S(=O)(=O)CCc2ccc(C(=O)OC)o2)CCO1 C1(NC(C2CCC(C)O2)=O)CC2CCCC(C1)N2C(c1cc2cn[nH]c2cn1)=O c1(C(=O)NCC2OCCC(NC(C(CC#C)O)=O)C2)c(N)cc(OC)cc1F c1(C(N2CCC(CC=C)(NC(c3cnnn3CC)=O)C2)=O)cc(=N)[nH]c(Cl)n1 C(C(C)(C)CNC(=O)CN(C(c1cnccn1)=O)CC1CC1)SC C(CCC(=O)O)(C(N)=O)C(N1CC(c2ccc(C)cc2)C(C(=O)O)C1)=O C1(C(=O)NCC2CC(F)(CNC(C3(C(=O)NC)CC3)=O)C2)Cc2cccnc2C1 c1(Cc2n(CC)nc(-c3ccccc3C(F)F)n2)cccc(Cl)c1 C#CCC(C)(C)CNC(=O)C(C)(C)C1CCN(C(c2cc(OC)n[nH]2)=O)C1 C(C(C)C(C)(F)F)NC(c1n(CCC)ccn1)c1nnnn1CCC(=O)OCC C1(C(=O)NC2C3CN(C(C4(C#N)CC=CC4)=O)C2C3)CCCN(S(N)(=O)=O)C1 c1(C(=O)NC2C(NC(c3c(C)ocn3)=O)CCOC2)c(Cl)cccc1[N+](=O)[O-] C=CC1(C(=O)NCC2(CO)CC23CCC3)CCN(C(C2CCC(=O)N2)=O)C1 C1(NC(C=NOC)=O)CCN(C(c2csc(-c3ccco3)n2)=O)CC1O N1(C(C(=O)NCC2(CC(=O)N(C3CN(C(C)C)C3)C)CCC2)C)CCOC1=O C(CC(O)CNC(c1cncn1C(C)C)=O)NC(C(C)OCC#C)=O C1(C(C)(C)NC(C2C(OCC)C2C)=O)CCN(C(C2CN(CC(F)(F)F)C2)=O)C1 C12CCCN(C1)C(=O)c1ncccc1NC2=O.C(C(F)(F)F)C(N)=O C1(C(=O)NC(C2CCN(C(C3CCC4CC34)=O)C2)(C)C)CN(CP(C)(C)=O)C1 N1(C(c2c(C)c(N)ccc2)=O)CCC2(C1)CN(C(=O)CC(F)F)CCO2 N1(C(C(C2CCCC2)OC)=O)CCC2C(NC(=O)CCCC3(OC)CCC3)C2C1 C(=O)(C(C)(C)N=[N+]=[N-])N1C(CC(=O)NCCCCCN(C)CC)CCCC1 c1(CC(=O)NCC2C=CCN2C(c2ccc(O)c(Cl)n2)=O)ccc2c(c1)COC2 c1(C(=O)NCCCNC(c2ccn(CCF)n2)=O)c[nH]c(=NCC(F)(F)F)cn1 c1(C(N(C2CCC(NC(=O)Cn3cnc(=N)[nH]3)CC2)C)=O)ccc2cccnn12 N1(C(C)=O)CCOC(N(C(c2ccc(C)s2)C(=O)NCc2ccc(C)cc2)C)C1 C(=O)(C#CC1CC1)NCCOCCC(=O)NC(C1CCC1)C N1(CCNC(CCN(C(CCC)C)C)=O)CCCC(C)(O)CC1 N1(C(C2(N(C)C)CCC2)=O)CC2C(C(=O)NC3CCC(O)CC3)C2C1 c1(OC)ccc(C(C)CC(=O)NC2CC(NC(c3cnc[nH]3)=O)C2)cc1 C1(C2CCCN(C(c3ccc(Br)s3)=O)C2)(NC(=O)Cc2ccno2)CC1 N1(C(CCC(C)OCC)=O)C2CCC1CN(C(C1CN3CCCC3CO1)=O)C2 C1(C)(CNC(CNC(=O)NC)=O)CCN(C(C2(C(C)C)CNC(=O)C2)=O)C1 c1(CCC(=O)N(C2CN(C(c3cnsc3)=O)C2)C)cnc2c(Br)cccn12 c1(CN(C2(O)CN(C(=O)OC(C)(C)C)C2)CC)cc(F)ccc1CC(=O)OCC N1(CCC)C(=O)NC(c2cccc3c[nH]nc23)C2=C1CC(C)CNC2=O C(=O)(C(CC)(CC)C(C)C)NC(c1cn(CC(=C)CC)nn1)Cn1ccnc1C C1(C(N2CC(CO)CC2)=O)(NC(C(C)OC)=O)CCN(C)C1.CO c12ccc(cc1)NC2C.Cc1ccc(C(C)OCc2cc[nH]n2)o1 C1(NC(C2(C(=O)OC(C)(C)C)CCCC2)=O)CC(F)CN(C(=O)CC2(O)CC2)C1 N1(C(c2c(C(C)=O)c[nH]n2)=O)CCCCC(CNC(=O)CN2CCNC2=O)C1 c1(C(C(=O)N(CC(CC)NC(=O)CN2CC(C)(C)C2)CC)C)ccccc1 c1(OCOC)ccc(Br)c(S(=O)(=O)NC(=O)C(C(F)(F)F)n2cnnc2)c1 O(Nc1nc(-c2ccccc2)nc2scnc12)CC(=O)NCCON C(=O)(C(CO)N(C)C1CC1)N(CC(=O)NC(CC1CC1)C1CC1)CC#C c1(CC(C)C(=O)NC2CCN(C(=O)OC(C)(C)C)C23CC3)ccc(F)c(Cl)c1 N1(C(Cn2nnc(C)n2)=O)CCCC(NC(C2(O)CC2)=O)CCC1 c1(C(=O)NCC(CC)(C)NC(=O)C(c2cn(C)nc2C)C)cc(C)nn1C1CC1 c1(C(N(CC(C)(C)CNC(C2CCCN(C(N)=O)C2)=O)C)=O)cc2c(s1)CCC2 C1(N(C(c2c(OC)csc2)=O)C)CCCCN(C(=O)Cc2cscn2)C1 CC(C)(C(=O)N1CCC(C(C)(O)CNC(=O)CC2CCCO2)CC1)C(F)F c1(C(=O)NC(C(=O)OC)C2CC(N)C2)ccc(C(F)(F)F)c(Cl)c1 CC1(C)CCOC1C(=O)NC(c1cccnc1)C(=O)NCc1cnsc1 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCC(NC(c2cccnc2)=O)C(O)C1 c1(C(N(C2CCN(C(C=C(C)C)=O)C2)CCO)=O)cn2c(n1)COCC2 C1(C(=O)NC(C)C(=O)N2CCCC2)CCCN(C(C2(F)CC2)=O)C1 C12(C(=O)NCC(C)C(=O)NC(C)(C)CCCF)CCC(CC1)CC2 C1(NC(c2cnc(C)[nH]2)=O)CC2CC1CN(C(=O)C1=CCCC1C)C2 C1(OC)CC(C(N2CC3C(CNC(=O)CCC4(C)CC4)C3C2)=O)CC1OC c1(OCC)nc2ccc(C(=O)N(CCNC(=O)CCC(N)=O)C(C)C)cc2[nH]1 CCC(CC)(CC)C(=O)NC(C1CCOC1)CNC(C1CC(=O)NC(=O)N1)=O C#CCC(CC(F)F)C(=O)N1CCC(C(=O)NCC23CCCN2CCC3)C(C)C1 C1(N(C(C(CC)C(F)(F)F)=O)C)CCCC2CN(C(c3c[nH]nc3Cl)=O)CC12 Cn1ncc(C(N2CCCCCC2c2ccco2)=O)c1S(C)(=O)=O N1(C(c2ccn(CC)c(=O)c2)=O)CCN(C(=O)C(N2CCSCC2)C)CCC1C c1(C(C(=O)NC2CN(C(c3c(C)cno3)=O)CC2C(F)F)O)ccc(Cl)c(Cl)c1 C12(CNC(C(C)NC(N)=O)=O)CC1CN(C(=O)CCOC1CCOCC1)C2 Cc1ccc(CC(=O)NC(C)CC2CN(C(c3cc(=O)c(C)c[nH]3)=O)C2)cc1C CCN=c1[nH]c(C(=O)NC2CC3CC(NC(C45CCCC4OCC5)=O)C2C3)cs1 C(=O)(C(C)C(C)C)N(CC(C)C)CC(=O)NCC1(NC(N)=O)CC1 [N-]=[N+]=NCCCCC(=O)N1CCC(C2CC2)C1C(=O)N1CC(O)CCO1 c1(C(N(CC(C)N(C(C=CCOC)=O)C)C)=O)ccccc1-c1nnc(C)o1 C1(C)(C(N(CCC(C(C)(C)C)NC(=O)CC#N)C)=O)CCc2ccccc2C1 N1(C(C)C(=O)NC2CC(F)(CNC(c3csc(Cl)n3)=O)C2)CCC(O)CC1 c1(COC)nc(NCCCN2CCCC2=O)cc(=NC(C)CS(C)=O)[nH]1 C1(CC=C)(NC(=O)CC2CCCCN2C(C2CC(=O)C2)=O)CCN(C(C)=O)CC1 c1(C(N2CCC(NC(C(CC=C)CC)=O)C2C2CC2)=O)cnc2c(c1)COCC2 N#Cc1ccc(COCC(=O)NC2CCN(C(=O)CCC3CC3(F)F)C2)cc1 N1(C(C=NOC)=O)CCC(CC(C)NC(=O)CC2CCC3CC23)CC1 C(=O)(CC(C)CC(C)C)N1CCC(C(C)NC(CC(CCC)O)=O)C1 N12CCCC(F)(C1)CNC(=O)NCC2C.N1(C(C)(C)C)CCCCC1 N1(C(C(N2CCC(C)C2)=O)=O)CCC(OC(=O)Cc2cccs2)CC1 C1(C(=O)NC2(CN(C)C)CC2)(NC(=O)C(c2ccccc2)F)CCN(C)C1 c1(C(=O)NCC(CNC(c2c(C)nn(C)c2)=O)(C)O)cc(F)ccc1N C1(C(=O)NCC2N(C(CN(C)C(N)=O)=O)CCCCC2)CCc2nn[nH]c2C1 CCC(C)CC(C)C(=O)NCC#CCNC(c1ccc2c(n1)NCC2)=O Cc1onc(C(N2CCCC(NC(c3cc(F)cc(F)c3O)=O)C2)=O)c1[N+](=O)[O-] C1(F)(CNC(C(c2cncc(F)c2)C)=O)CCC(CNC(C2(O)CC2)=O)C1 C1(CCNC(C(CC)F)=O)CC(F)(F)CN1C(c1ccn(C)c(=O)c1)=O N1(C(CN(CC)CC)=O)CC(CNC(=O)CCc2nc(C)no2)CC(C)(C)C1 N1(CC(=O)NCCOCC#C)CCCCC1 C12(C(N3CCSCC3C(F)(F)F)=O)CC=CCN1CCC2 S(=O)(=O)(c1cccc(Cl)c1)NCC(N1CCCC(NC(C2(O)CCSC2)=O)C1)=O C1(C(=O)N(C2CC(NC(c3nn[nH]c3-c3ccccc3)=O)C2)C)(OC)CC(C)C1 C(=O)(C1=NNC(=O)C1)NC(CC(=O)NC(CC=C)C1CC1)CC1CC1 c1(OC)cc(C(N2CC(NC(c3csc(C)c3C)=O)C(C#N)C2)=O)cc(O)c1O Cn1ncc(C2CC2)c1C(=O)NCC(C1CCC1)NC(C1CCS(=O)(=O)N1)=O C(C(C)C(C)C(=O)N1CCC(C)(CNC(C2CN(C3CCOC3)C2)=O)CC1)OC C1(C2(C)CC2)COCCN1C(=O)COC1CN(C(C2CCOC2C2CC2)=O)C1 c1(OC)ccccc1S(=O)(=O)N1CCCC1CNC(c1nc(Br)cs1)=O c1(CCNC(C(=O)NC(C#C)CCC)=O)cccc(F)c1F c1(CN(C(=O)CCNCC(F)(F)F)C2CC2)ccn(C2CCOCC2)n1 CCC(C)C(O)C(=O)NCCC1CC(C(N2CCC(N3CCC3)CC2)=O)C1 c1(CCC)cccc(C(=O)NCC(C2CC2)N(C(=O)C(O)C2CCC2)C)c1 c1(CC(=O)NCCC(C)(C)NC(C2CCC3CC23)=O)ccc(Cl)nc1 Cc1ccnc(C)c1C(=O)NC1CC(C(F)F)(NC(C2CCC(C)O2)=O)C1 C1(C(N(CCCNC(C(CCC)(C)C)=O)C)=O)CCN2CCCC2C1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(C2CCCSC2)=O)cn1C C(=O)(C(C)O)NCCCNC(CNCCOCC)=O.C1(CC(=O)NCC)CCOC1 c1(C(N(CCN(C(C2CCCN(C)C2)=O)C)C)=O)ccc(N)cc1O C(c1cccc(F)c1F)=CC(N1CCN(C(CCC(CC)C)=O)CC1C1CC1)=O N1(C(c2cn(CCN(C(CC3(OC)CCC3)=O)C)nn2)=O)CC2CCC2(C)C1 c1(C(=O)N(C2CC2)CC2CCCN2C(=O)Cc2ccco2)cncc(Br)c1 c1(C(=O)NCC(CC=C)NC(=O)CC(C)n2cccn2)cccc(C)c1[N+](=O)[O-] N1(C(c2c(C)ccc(O)c2)=O)CC2OCC(NC(=O)Cc3ccc(Cl)cn3)C2C1 C1(CC)(NC(C2CC(=O)N(CC)C2)=O)CCN(C(=O)CC(C)N(C)C)CC1 C(=O)(C(C)(CC)CC)NCC(CNC(C(CSC)O)=O)(C)O C(C(C)=Cc1ccccc1)(C(=O)NC1CCCC1)N(CCC)Cc1ccccc1 c1(C(=O)NCCOCCNC(C2(SC)CC2)=O)c[nH]c2nc(F)ccc12 C1(C(=O)NCCN(C(C(C2CCOCC2)OC)=O)C(C)C)CCC(C)O1 C=CCC(C(=O)NC1CC2(CCC2)C1)NC(C1OCCC1C)=O CN1CCc2cc(C(=O)NCC3CC4(CCC4)CN3C(C3C=CCC3)=O)ccc21 C1(C(=O)NCC=CC(=O)NC(c2ncc[nH]2)CC)(CC)CCCCO1 c1(CO)cccc2c1CN(CC1CCCCN1CC(F)F)CCC2 c1(OC)cccc(C=CC(=O)NC2CC(OC)CN(C(C3CCC3(C)C)=O)C2)c1 c1(C(N2CCC(C(C)C(=O)NC3(C)CCNC3=O)CC2)=O)ccc(Cl)c(C#N)n1 c1(C(=O)NC2CCCN(C(CCNC(=O)NC)=O)C2C)cnc2n[nH]c(C)c2c1 Cc1cncc(C(N2CCC=CC2C(=O)Nc2cncnc2O)=O)c1 N1(C(Cc2nc(C)[nH]n2)=O)C2CCC1CC(NC(c1ncnn1C)=O)C2 C1(F)(C(N(CC#N)CC)=O)CCCN(C(=O)C(C)CC(C)=O)C1 c1(OC(C)(C)C)ccc(C(N2CCC(CF)(NC(c3cscn3)=O)C2)=O)cc1 C(CCN(C)C(c1ccc(-n2ccnc2)nc1)=O)(C(C)C)NC(C(CC)C)=O CC(C(=O)NC1CC2CCC1CC2NC(=O)CC1CCC(=O)N1)C(F)(F)C(F)F C=C(Cl)C(=O)NC1CC(N(C(C2CCCC2)CC)C(c2nccs2)=O)C1 c1(C(=O)NCC2C(NC(C3(C)CC3)=O)CCCC2)noc2c(F)cccc12 C1(NC(C(C)Oc2ccccc2F)=O)CN(C(C2(CF)CCC2)=O)CC12CC2 c1(OC)ccc(S(=O)Cc2ccc(Br)cc2)cc1 N1(C(C(N2CCCCC2)C)=O)CC=CC(C(=O)NC2CC(=O)N(C)C2)C1 Cn1ncc2nc(O)c(C(=O)NCC(CNC(c3cccc(O)c3)=O)CO)cc12 CCC(C)CCC(=O)N(C1CCN(C(=O)CC2CCCOCC2)CC1)CCO N1(C(C(C)N(C(=O)CCc2cccn2C)CC)=O)CC(C)CCCC1C C(=O)(C1OCCn2ccnc21)NCC(C)(CC(C)C)NC(C=C(C)Cl)=O c1(CNC(C2CC3CC2C3)=O)nnc(O)n1C1CC1 c1(C(C)NC(=O)NCC2CCCC2N2CCCC2)c(F)cccc1F c1(OC)cc(C(N2CCC(CO)(NC(C3(n4ccnn4)CC3)=O)C2)=O)ccn1 c1(C(N2CC(CCOC)N(C(=O)C(C)COC(C)=O)CC2)=O)cccc2sncc12 CC1=C(C(=O)N2CC(c3nc(C)no3)C2)SCCO1.C12CCN(CC1C)C2=O Cc1ccsc1C(c1nnnn1Cc1ccco1)NCc1ccn(C)n1 c1(C(N2C(CNC(CC3C(C)(C)C3)=O)CCCCC2)=O)cc2c(Cl)cncc2s1 c1(NC(C(=O)NC2(C)CN(C(C3CCCC(=O)O3)=O)C2)=O)ccccc1CO c1(C(N2CCC(CNC(c3ccc(SC)o3)=O)C2(C)C)=O)cc(C)c(C)cc1C N1(C(C2(S(C)(=O)=O)CC2)=O)CCCC(NC(=O)CCN2CCP(C)(=O)CC2)CC1 c1(SCCNC)cc(O)c2ccccc2c1.C12CCN(CC1)C2=O N1(C(C2C3(CC(NC(COC)=O)C3)C2)=O)C2CCC1CC(C)C2 c1(C(=O)NCC(CNC(c2ccc(CNC(C)=O)s2)=O)C)ccc2nonc2c1 C1(NC(=O)COCC2CCOC2)CCC2(CCN(C(=O)Cc3ccon3)CC2)C1 C1(N(C(c2cn(CCCSC)nn2)C(=O)Nc2ccccc2)C)CS(=O)(=O)CC1O C1(CNC(c2cc(C)sn2)=O)C2CC2CN1C(c1csc(-c2ccccn2)n1)=O C#CCN(OC)C(=O)CC1(CNC(c2cc(=O)cc[nH]2)=O)CC1 C1(O)(C(=O)NC2C(NC(CN(C3CCC3)C)=O)CC2)CCC(C)(C)C1 CC1(C)CCC(CC(=O)NCC(CNC(=O)CNC(N2CCCC2)=O)CO)OC1 C1(C(N2CCC(CCN(C(=O)C=CCF)C)CC2)=O)(OC)CCC(C)(C)C1 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)N(CC(CC)NC(=O)C(CC)SC)C C#Cc1ccc(CNC(=O)CC2C3CN(C(=O)C(C)NC(N)=O)CC23)cc1 C(=O)(C1CCCc2n[nH]cc21)NC(C1(O)CCN(C(=O)Cn2ncnn2)C1)C N1(C(CC2CC(CC)C2)=O)CC(=O)NCC1C(=O)NC(CC1CCC1)CO N1(C(CCOCCC)=O)CCCC(CCCCNC(C2(O)CCC2)=O)C1 N1(C(C2C(NC(=O)OC(C)(C)C)C2)=O)CC=C(c2ccccn2)C1 C1(C(C)NC(c2nnc(-c3cnccn3)s2)=O)CCN(C(=O)C(C)(O)CO)CC1 C1(C(=O)NCCCNC(c2c(SC)c(F)ccc2)=O)Cc2cc(C)c(C)cc2O1 C(=O)(CC(C)C(=O)NCC1OCCC1C(=O)NC1(C)CCSCC1)OC C(=O)(C1CCCc2scnc21)N(CCN(C(c1n(C)nc(C)c1Cl)=O)C)C(C)C CC(CNC(=O)C=CC(=O)NC1CC1)CNC(=O)CC1(C(F)(F)F)COC1 CN=c1cc(C(=O)NC2CCC(C)N(C(=O)CC(F)(F)Cl)C2)cc[nH]1 CCC(C)C(O)CC(=O)N1CCCC(N2CCN(C(=O)CCCC#N)CC2)C1 Cc1cnn(C)c1S(=O)(=O)N1CCCC1COC(C)(C)C c1(C(=O)NCC(CNC(c2ccc(C)o2)=O)C)cc(F)c(C(F)(F)F)c(F)c1 C1(O)(C(=O)NCC=CCNC(Cc2n(C)cnn2)=O)CCCCCC1 c1(C(=O)NC(c2ccc(OC)c(Br)c2)C(=O)OC)ccc(C)c(I)c1 C1(NC(C2(CCC=C)CC2)=O)CC2CCC1CN(C(=O)C(C)OC)C2 c1(C(N2CC3CC(CN(C(CC(CC)C)=O)C3)C2)=O)ccc2cccc(O)c2c1 CC(C)(CCC(=O)NC1COCC1CNC(=O)CCc1cn[nH]c1)[N+](=O)[O-] C1(NC(c2cn(CC)nc2)=O)C2CCCN(C(=O)C(C)n3cncn3)C2C1(C)C C12(NC(C(N3CCCCC3)C)=O)CC1CN(C(c1cccnc1C(F)F)=O)C2 C1(NC(c2c(SC)scc2)=O)COC2(CCCN(C(=O)Cc3nonc3C)C2)C1 C1(C2(C)CC2)(C(N2C(C)CC2C(N2CC(C)(C(N)=O)C2)=O)=O)CC1 CCC(CC(=O)NCC1(C(=O)NCCN2CC=CCC2)CC2(CC2)C1)CC(C)C Cc1cc(=O)ccn1CC(N1CC(N(C(=O)CCC2CCCCO2)C)C1)=O N1(C(c2cnc(C(C)(C)CF)o2)=O)C2CCC1CN(C(=O)CC1=CCCC1)C2 C1(NC(C(CCCC)O)=O)CC(N=c2nc(O)c3cnn(C)c3[nH]2)C1 C1(C(c2n(CCOC)nnn2)NC2(CF)CCC2)CCCC(F)(F)CC1 c1(C(=O)NCC2CCCN2C(c2cnc[nH]2)=O)cc2ccncc2s1 Cc1cc(C)nc(SCC(=O)NCC2CCN(C(=O)CC3CCOC3=O)CC2)n1 C1(NC(C2CN(C(C)=O)C2)=O)CC(NC(=O)C(C)(F)F)C12CCC2 N1(C(C(CCC)F)=O)CCCC12CCN(C(C13CC(CCC)(C1)C3)=O)C2 C1(COCC(=O)NCCN(C(=O)C(C)c2ccco2)CC)CCCOC1 c1(OCC)cccc(C(=O)NC2CCCC2NC(c2cnc(OC3CC3)s2)=O)c1 c12cccnc1N1CCC(C1)N(C)C2.n1(CCC)ncnc1CNCC(F)(F)F N1(C(CC(COC)C)=O)CCC2CCN(C(c3ccc4nc(C)cn4c3)=O)CC12 C12(NC(CN(CC)CC)=O)CC1CN(C(c1nocc1Cl)=O)C2 C(=O)(C1=CCCS1)NCCCCN(CC(=O)NCCOCc1cnn(C)c1Cl)C c1(CN(CC=C)C)cn(C(C)C(=O)NCC)nn1.C1(=O)C(C)N1Cc1ncsn1 C(=O)(CCCC(=O)N1CC(CNC(=O)CNC(=O)OC(C)(C)C)CC1(C)C)NC c1(C(=O)NC2CCN(C(C3(C)CCCCCC3)=O)C2)cccn2nccc12 c1(C(N(CCNC(c2cc(CCO)on2)=O)CC)=O)cc(Cl)c2n[nH]cc2c1 c1(CNC(CC=C)=O)ccc(CCNC(C2CCCOC2C)=O)cc1 c1(N2CCC(F)(C(=O)NC)C2)nccc(=NCC2CCOC2)[nH]1 C12(C(=O)NC(C)C(c3ccccc3)NC(c3cc(Br)co3)=O)CCCC1OCC2 C(C(C)(C)CNC(C1CC1Cl)=O)N(C(CCN(C)CCO)=O)C N1(C(c2c(C)nc(C)s2)=O)CCC2(CCCN2C(=O)C(C(C)C)C2CCC2)CC1 C(=O)(CC(O)CCS(C)=O)NC1(C)CN(C(c2nc(C)c(C)s2)=O)C1 c1(C(=O)NCC2(O)CN(C(C(CCOC)C)=O)C2)ncc(OC2CC2)cc1F C(C1CN(C(=O)CN(C)C)CC1C(=O)NCCC(O)COC(C)=O)=CC N1(C(CC=C)=O)CCC(NC(C2CCCN2CCC)=O)C1(C)C c1(C(=O)NCCC2N(C(c3csc(C)c3N)=O)CCSC2)ccnc(C)c1C c1(C(N2CC(O)CC(NC(CC=CCC)=O)C2)=O)cc2cc(Cl)ncc2[nH]1 CC(c1ccccc1)=CC(N1CC(O)(C(C)NC(=O)CCc2ccon2)C1)=O S(=O)(=O)(c1ccc(N2CCCC(OCC(F)(F)F)C2)cc1Br)N(CC(C)SC)C N1(C(C(C=C)O)=O)CCN(C(c2ccc(OC)nc2)=O)CC1c1ccc(CC)cc1 c1(NCCCC(N)=O)cc(NC2COCCOC2)ncn1 C1(C(N2CCC(N(C(C34COCC(C3)OC4)=O)CC)CC2)=O)CC2CCCC(C1)C2 CN1C(=O)CCCC1C(=O)NC(C1CCN(C(=O)CC(C)(C)O)CC1)(C)C C(=O)(C1=NNC(=O)C1)NC1CC(OCc2cn(C)nn2)C1(C)C C1(C(=O)NCC(=C)CCNC(=O)CCSCC)CCC2(CCC2)CO1 c1(N(CCOCC)C)ccc(Br)cc1C(=O)OC.C1(=O)C(c2cn[nH]c2)N1 N1(C(c2ncc(C(=O)OCC)nc2)=O)CCCC(O)CC1.C1C(=O)N1CC N1(C(COCC)=O)CCC(NC(=O)CCC(F)F)C(C(C)C)C1 N1(C(CC(CC(C)C)NC(CC(CC)C(F)F)=O)=O)CCc2ccc(F)cc21 C1(C(C23CC(NC(CC(=O)N(C)C)=O)(C2)C3)NC(C2CCCC2)=O)CCC(C)(C)C1 c1(N(C)C)ncccc1C(=O)NCC1COCC1NC(c1nnsc1C(F)F)=O C12(C(N3CCC(F)(CNC(C(C)OCCC#C)=O)CC3)=O)CC=CCN1CCC2 C1(F)(CNC(c2cnn3c2OCC3)=O)CCCN(C(=O)C=CCF)C1 N1(C(CC)=O)CCN(C(=O)C(N2CCOCC2)OC)CC12CC2 N1(C(c2c(C)csc2Cl)=O)CC(CNC(c2cccnc2)=O)CC(C)(C)C1 C(=O)(C(C)C(O)C(C)C)N1CC(C)C(=O)N1.C(C)(C(=O)OC)=C(CC)C c1(NC(=O)NCC2CC(NC(C(=C(C)C3CC3)F)=O)CC2O)c(Cl)cccc1Cl C12(CNC(COC)=O)CCC1CCN2C(c1cc(=O)n(C)o1)=O C1(C(=O)NCCOc2cccnc2)CN(C(c2ccnc(Br)c2)=O)CCC1(F)F C(=O)(C1Cc2c(Cl)cccc21)N1C(C)(C)C(CNC(=O)CSC2CC2)CC1 C1(CNC(C(C)(C)F)=O)CC2(CCN(CNC(=O)C(F)(F)C(F)(F)F)CC2)CO1 Cc1c(C(=O)NC2COCC2NC(C2(C#N)CCCC2)=O)nnn1C c1(NC(C2CCCN(Cc3ccc(Cl)nc3)C2)=O)cccnc1OC(F)F c1(C(=O)NCC2CCCN(C(CC(C)(C)OC)=O)C2)ccnc(C)c1Cl c1(NC(C(N2C(COCC)CCC2)CSC(C)=O)=O)ccc(F)cc1 CCCC(C(=O)NCC1(C)CCN(C(c2n[nH]c(=N)s2)=O)CC1)S(N)(=O)=O c1(C(N2C(CC#N)CC(F)(F)C2)C(=O)NC2CCCCC2)cc(F)c(F)c(F)c1 Cc1ncc(C(N2CCC(CC(=O)NCc3cc(C)c(C)s3)C2(C)C)=O)c(C)n1 c1(C(N(C(Cc2cccc(C)c2)C)C)=O)cncc2cccnc12 C(=O)(C1=CC2C=CC1C2)NC(C(C)NC(c1cnc(C(C)(C)C)[nH]1)=O)C CCCC(C#N)C(=O)N1CC(NC(=O)Cc2cnccc2Cl)C(O)C1 c1(CN(CC(CC)C)CC)nnc2n1CCCC2C(F)F C(=O)(C(CC(F)F)NC(c1cn[nH]c1)=O)NCC1(NC(N)=O)CCC1 c1(CC)ccc(OC)cc1C(N1CCCC1C(C)NC(=O)C(C)CC(C)(C)C)=O C(=O)(C(O)CCc1cnc[nH]1)NCC(C(C)C)NC(=O)C(C)(O)C1CCC1 c1(OC)ccc(NC(C2CC2C(N2CCS(=O)CC2)=O)=O)c(Br)c1 N1(CCC(C)(C)NC2C(OC3C(C(=O)OCC)COC3)CCC2)CCC(C)CC1 C(CCC(=O)N(CC(C)(C)CNC(=O)COc1ccsc1)C)OCCC c1(NCC)cncc(C(N2CCOC(CNCC(=O)NS(=O)(=O)C3CC3)C2)=O)c1 c1(C(N(CCN(C(C2CCCN(C(C)=O)C2)=O)C)C)=O)cc(N)c(C)cc1C N1(C(C=CCN(C(c2c(CC)nn[nH]2)=O)C)=O)CCN2CC(C)CC2C1 C1(NC(C2CCN(CC)C2)=O)CN(C(=O)Cc2cncc(C)c2)CC2(CCC2)C1 C(=O)(C1=C(Cl)CCOC1)NC1(C)CCN(C(CN2C(C)CCC2C)=O)CC1 c1(C(=O)NC2CC(C)N(C(=O)C(c3ccccc3)F)CC2)c(F)ccc(F)c1N N1(CC)CCN(CC(N2CC(CCNC(c3nccn3C)=O)C(C)C2)=O)CC1 CC1(C)CCC(=CC(N2CCCC(n3cccn3)C2)=O)CC1 N1(C(c2nc(CCC)sc2)=O)CCN(C(=O)CNS(N)(=O)=O)CC1CC C1(C(=O)O)(OC)CCN(C(C2CCC(C)(C)CO2)=O)CC1 C1(CNC(C(C)C2CCC2)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC1O c1(CNC2CCN(C(c3ccncc3Cl)=O)C2)c(Cl)cnc(Cl)c1Cl C(=O)(C1CCc2c[nH]nc21)NCC(CNC(c1ccc(=N)[nH]n1)=O)F c1(CC)cnccc1C(N1CCC(C(C)(C)C(=O)N2CCCC2CC(C)C)C1)=O c1(C(=O)NCCC(C)N(C(C(CC)CO)=O)C)ccc(OC)cc1Cl c1(C2OCCN(C(=O)Nc3nnc(C(C)N)s3)C2)cccc(Cl)c1Cl c1(C(N2CCC(NC(C3(C)CC(C)(C)C3)=O)C2)=O)ccc2occc2n1 N1(C(c2cc(C)sc2)=O)CCN(C(C2CC2(Cl)Cl)=O)CC(C)(C)C1 c1(C(=O)NC2CC(CNC(=O)C(O)c3ccco3)C2)ccc(=O)n2c1CCCCC2 N1(C(c2c(OCC)cccn2)=O)CC2(CCCC2NC(=O)C(C)CC)C1 C1(N(C(=O)Cc2cnn(C)c2)C)CCN(CCCc2ccccc2)CC1 c1(CNC(C)=O)ccc2c(c1)CCCC2NC(C1COCC(=O)N1C(C)C)=O c1(C(N2C(C3(O)CCN(C(c4cc[nH]c4)=O)CC3)CCC2)=O)ccc(F)c(Cl)c1 c1(OC)coc(C(=O)NCC2CCCC(NC(c3cccc(F)c3)=O)C2)cc1=O c1(C(N(C2CCN(C(C(C(C)C)(C)C)=O)C2)CCO)=O)cc2cccc(Cl)c2[nH]1 N1(C(C(=O)N(CCNC(C2(F)CN(C(C)=O)C2)=O)CC2CC2)C)C(=O)CCC1=O CCCC(O)CC(=O)NCC(CCNC(c1ccc(C(C)C)s1)=O)C1CCC1 C1(CC(=O)N(C(CN(C(CNC(CC)=O)=O)C)C)C)CCC(C)(C)CO1 c1(NC(C=C(CCC)CCC)=O)ccc(NC(C2CCCC2CC)=O)cc1C c1(CN2CCN(C(c3c(C)cc(F)nc3)=O)C3C2C3)ccc(C#N)cc1[N+](=O)[O-] c1(N(C)C)ccc(C(N2CC(F)(CNC(C3CC3C(F)F)=O)C2)=O)c(F)c1 CC(CC(C)(F)F)C(=O)N1CCC(CCNC(c2c(N)cc(Cl)cc2Cl)=O)C1 N1(OC)CC2CN(C(C34C5C6C7C5C3C7C46)=O)CC(C1)O2.c12cccc(c1)S2 C1(OCC)CCOCC1NC(=O)CC1CC(C)N(C(=O)CCc2nncn2C)C1 C1(CCNC(c2scc(C)c2)=O)CCCN(C(=O)CCC2CCCN2C)CC1 c1(CCC(=O)NC2CCN(CCC3CCOC3)C2)ccc(O)nn1 c1(C2(Cn3c(N(C)C(C4C=CCN4C4CC4)=O)nnn3)CC2)ccc(Cl)c(Cl)c1 CCCC(CNC(C1CCOC(C)(C)C1)=O)C(=O)NCC(C)C(=O)OCC N1(C(C(C)OC2CCOC2)=O)CCN(C(c2cc(CO)on2)=O)CC1CC(F)F C(=O)(C1=CCCOCC1)NCC1(C(N)=O)CN(C(C2CCC(C)CC2)=O)C1 N1(C(C(C)SC)=O)CCC(CC(N2CC(C(N)=O)C2)=O)C1 C1(C(N(C(CNC(CC2CN(C(C)=O)C2)=O)C2CC2)C)=O)CC(C)(C)CN1C C(=O)(C(CC1COCCO1)C(F)(F)F)NCC1CN(C(CNC(C)=O)=O)C1 c1(C(N2CCN(C(CC(COC)(C)O)=O)C3C2CC3)=O)ccc2c(c1)CCCO2 C1(c2n(C(CC)C)nnn2)(NC(C)CCOc2ccc(F)cc2)CCCSCC1 CC(C)(C)CCC(=O)NC1CC1NC(C1(F)CN(C(=O)OC(C)(C)C)C1)=O N1(C(C(F)=CCC)=O)CCC(N(C(c2cc(C(F)(F)F)c[nH]2)=O)C2CC2)C(C)C1 Fc1cc(SCC2CC(CCl)C2)c(F)c(F)n1 N1(C(C(CC=C)C)=O)CCC2(C1)CN(C(C1OCCOC1c1ccccc1)=O)C2 c1(C(=O)NCC2CC(NC(CCCc3onc(C)n3)=O)C2)[nH]c(C)c(C)c1C C1(C(=O)NC2CCC(NC(C(C)CN3CCOCC3)=O)CC2)CCC(=O)N(C)C1 Cc1ncccc1-c1cn(CC2C(CNC(C3CCCC3CF)=O)C2(F)F)nn1 N1(C(CCc2ccc(N(C)C)cc2)=O)CCOC(C)(CNC(C2CC2CF)=O)C1 c1(C(N2CC3(CCN(C(CC4CCN(C)C4)=O)C3)C2)=O)cccc(S(C)(=O)=O)c1 N1(C(c2c(C)nn[nH]2)=O)CCCC(C(C)NC(=O)CCc2ccon2)C1 c1(OC(C)C(N2CCC(OC(F)(F)F)C2)=O)ccccc1-c1ccccc1 c1(CC(=O)NCC(CNC(Cc2ncc(C)s2)=O)F)cc(F)cc([N+](=O)[O-])c1 C(=O)(CC(C)(C)O)NC1(c2cn(-c3c(OC)nsc3)nn2)CCC1 c12ccccc1NC(=O)C1(CC1)O2.C1(N(C)C)CC(N(C(=O)C(=O)N(C)C)C)C1 c1(OCCC)cccnc1C(=O)NC(CN(C)C(c1cnc(OCC)s1)=O)CC C(=O)(C1CCCc2c[nH]nc21)N(CCCCCCNC(C(CCC(C)C)O)=O)C c1(NCC2C(C)CN(C(=O)CCn3cnnn3)CC2)ccc([N+](=O)[O-])cc1C(F)F N1(C(C(C=CC)O)=O)CCN(C(c2cc(O)cnc2N)=O)C(C)C1 C(=O)(C1=Cc2ccccc2OC=C1)NCC(CN(C(Cc1c(C)ccs1)=O)C)O c1(C(=O)NCCCN(C(=O)C(F)C2CC2)CC)ccc(S(C)(=O)=O)cc1 N1(C(C=CCOC)=O)CCCC(C2CCN(C(=O)C(O)CSC)CC2)C1 C1(NC(C(C(CC)C)=O)=O)CC2CC1CN(C(c1ccc[nH]1)=O)C2 C1(NC(CC(CC)C)=O)CCS(=O)(=O)C12CN(C(C1(c3ccncc3)CC1)=O)C2 CN1C(=O)CSC1=CC(=O)NCC(CO)NC(C1CCCCC12CCC2)=O C(CCCC(C)C)NC(C(c1cn(C)nn1)NC(c1cc(OC)no1)=O)=O c1(CC(=O)OCC)ccc(C(=O)COC(=O)C(C)COC)cc1 C(C(CC(C)C)NC(=O)CSCC1CCCO1)NC(C(SC)SC)=O c1(SCC(=O)NC(CC)CN(C(=O)CC(C)SC)C)ccc([N+](=O)[O-])cc1 c1(SCC(N2CCC(C)(CNC(C3CCC(=O)N3)=O)C2)=O)ncnc2[nH]cnc12 N1(C(c2nnnn2C2CC2)C)CC2CCCN(C(C3CCC(=O)N(C)C3)=O)C2C1 CCCCCC(=O)NCC(N1CCC(N(C)C(C2CC3(C2)CC3F)=O)CC1)=O c1(C(=O)NC2C3CCN(C(CC(C)C(C)(C)C)=O)C32)nc2ccccn2c1F C(=O)(N=c1cc[nH]c2cccnc12)c1cc(OC)c(C(=O)OC(C)(C)C)cc1 c1(N2C(CNC(c3ccc(F)cc3F)=O)CC3(CC3)C2)ccc([N+](=O)[O-])cc1 N(C(=NCCOCC(F)(F)F)NC1CCCCC1)C1CCC(=O)NC1 Cc1cc(C(=O)NCC2OCCC2C(=O)NC2CC3C=CC2CC3)ncc1N C1(NC(c2cc(CO)on2)=O)C2CCC1CN(C(=O)C1=CC3CCC1C3)C2 c1(NC(C2CCCN(C(C3(C)CCCO3)=O)C2)=O)ccc(O)c(F)c1 C1(NC(CNC(=O)NC)=O)CC(F)(CNC(C2CCN(CC(C)C)C2)=O)C1 N1(C(C2(OCC)CCCC2)=O)CCCC(C2CCN(C(=O)CC3CC=CC3)C2)C1 C1(CC(=O)NCCCC(=O)NC2CN(C(=O)C3CC3)C2)CC2(CCOCC2)CO1 N1(C(c2nccc(C)c2)=O)CCC(C(=O)Nc2cc(C(C)O)ccc2I)C(O)C1 N1(C(CCCC(=C)C)=O)CCCC(C2CN(C(c3cc(CO)c(C)o3)=O)C2)C1 N1(c2nc(SC)c(F)cn2)CCCC2C1CCN2Cc1cc(Br)c[nH]1 C1(F)(CNC(CC2C(C)(C)C2)=O)CC(NC(C2CC2(Cl)Cl)=O)C1 C(=O)(CCCC(c1nnnn1C)NC1CCCCC1c1cccc(C)c1)OCC C=C1CCN(C(=O)CCCCN(C)C)C(C(=O)Nc2ccc(N(C)C)cc2C)C1 C1(NC(C(CCOC)NC(=O)CN2CCC(F)CC2)=O)C=CC(C)(C)CC1 c1(CNC(CNC(C=C)=O)=O)ccc(Cn2cc(C3(O)CCOC3)nn2)cc1 C1(C(=O)NC2(c3cccs3)C(C)C2)CCCN(C(=O)CCN2CCCC2)C1 C1(C)(C(=O)NCCCCCN(C(CC(CCC)(C)O)=O)C)CC(C(F)(F)F)=NO1 C(CNC(C1CNC(=O)C1)=O)(CC(F)(F)F)NC(CS(=O)(=O)NC(C)(C)C)=O C1(CC(=O)NC23CC(F)(C2)C3)C2CN(C(=O)COC3CCCCC3)CC12 c1(CC(N2CCC(N(CCC)C(c3ccc(F)o3)=O)C2)=O)ccc(F)cn1 C1(NC(C2C(C)CC(=O)NC2)=O)CC2CC(C1)N(C(C1(C3CCCO3)CC1)=O)C2 N1(C(C(CC2CCOCC2)NC(COCCSC)=O)=O)CCC(C2=NOCC2)C1 S(=O)(=O)(c1ccc(C(=O)NC2C(O)C3CCCC23)cc1)NC(c1cccs1)C N1(C(C2(CC)COC2)=O)CCN(C(=O)CC2CC(C)(C)CO2)CC(O)C1 CC(C)CCC(O)C(=O)N1C2CCC1C(C(=O)NCC1CC(C)(C)CCO1)C2 CN1CCC(N(C)Cc2ccnc(-c3cccc(NCCO)c3)c2)CC1 c1(OC)ccc(Br)c(F)c1C(=O)NC1CC1C(=O)NCC#N CC(CN(C)C)CCC(=O)NCC=CCNC(=O)CCCOCc1ccccc1 Cc1cc(OCC(=O)NC2CC(C)(NC(=O)Cc3cncnc3O)C2)cc(C)c1 C1(CCNC(CCNC(=O)NC)=O)(NC(c2cc(C(C)(F)F)on2)=O)CC(=O)C1 c1(N(C)C)c(F)ccc(C(=O)NC2C3CCC2CN(C(C2(N)CC2)=O)C3)c1F CCCCCCC(C)(CCC)C(=O)N1CCC(N(C(=O)CCOC)CC)C1 CCCC(O)CC(=O)N1CCN(C(=O)C(C)=C2CCCC2)CC1c1nccn1C C12(C(N3CCC(C(C)(C)NC(c4cc(O)ncn4)=O)C3)=O)CC3CC1C2C3O c1(CN=C(NC(COC)C)NC2CC2(C)C2(C)CC2)ccc(C#N)c(F)c1 C1(NC(C2CCC(C)C2)=O)CC2CCCC(C1)N2C(C1CC(CC(C)(C)C)C1)=O C1(C(=O)NCc2n(C)ccn2)CCC(C)(C)N(C(c2ncccc2N)=O)C1 C1(N=[N+]=[N-])(C(=O)NCCCc2nc(C)[nH]n2)CCN(C(=O)C#CC2CC2)C1 N1(C(C(C)C2(O)CCC2)=O)CC(C(=O)Nc2cc(OC(F)F)ccn2)CC(F)C1 C[S+](C)CCC(O)C(=O)N1CCC(C)(CNC(=O)C(C)(C)NC(=O)C(F)(F)F)C1 c1(NCC(CSC)OC)[nH]c(=NCCS(N)(=O)=O)nc2c1ncn2C(C)C CCC(C)CC(=O)N1CCCCC1C(=O)Nc1[nH]cc(O)c1-c1ccccc1 N1(C(C=CCCC(C)C)=O)CCC2(CC1)CN(C(C1CC1CF)=O)C1COCC21 Cc1cc(C(=O)NC2(C)CC(NC(C3CN(C(C)C)C3)=O)C2)c2ncccc2c1 c1(C(=O)OC)c[nH]c(C)cc1=NCC(CNC(=O)CCc1cnn[nH]1)C(F)(F)F C(=O)(CC1OCCc2ccccc21)NC(CNC(C1(CC)CCOCC1)=O)CO N1(C(C)=O)CCC2CN(C(=O)CCCCCc3cccc(O)c3)CC2CC1 C1(NC(c2cc(Br)n[nH]2)=O)CC1C1CCN(C(=O)COc2ccon2)CC1 C(=O)(C(O)CC(F)(F)F)NC(CN(C(c1cncnc1C1CC1)=O)CC)C c1(C(N2CC3(CN(C(CC(C)C4CC4)=O)C3)C2)=O)ccnc2[nH]ncc12 C=CCC(C(=O)NCCC1(CNC(=O)C(C)C=C)CC1)c1ccccc1 C(=O)(C(C)(O)Cc1cn[nH]c1)NCC(CC)NC1(Cc2ccc(F)cc2)CCOCC1 Cc1cccc(C(CNC(=O)C(c2ccnn2C)C)NC(c2csc(C)c2)=O)c1 N1(CC(=O)N(C2CCN(C(=O)C=CCO)C2)CC)CCC(NS(C)(=O)=O)CC1 C1(OCC#C)CCN(C(=O)C(C)N(C(c2cc(OC)n[nH]2)=O)C2CC2)C1 N(C(=NCC1CCC(C(N)=O)CC1)NCC(F)C(F)(F)F)C(C)(C)C N1(C(C(c2cnsc2)NC(C2(CO)CC2)=O)=O)CCC(CCCCO)CC1 C1(NC(C(F)OC)=O)COCCN(C(=O)C2=COCCO2)C1 N1(C(c2c(C)cc(CO)o2)=O)CCN(C(=O)CN(C)C2CC2)C2CS(=O)(=O)CC12 C(CCC(C)C(=O)NC1C2CC1N(C(c1ccc(Br)c(O)c1)=O)C2)OC C(=O)(CCCC(=O)N1CC(C)(NC(C2CCC(NC(N)=O)CC2)=O)C1)OC C=C(C)c1ccccc1NC(=O)CCC1(C)CN(C(=O)CCN(C)CC)C1 C(CC(F)F)(C(=O)N(C)CC1(C)CCC1)NC(c1c(C)nn[nH]1)=O c1(C(=O)NCCN(C)C(C2COC(=O)O2)=O)cc(=O)c2ccccc2o1 c1(CCC)nnc(-c2cccc(OC)c2)n1C(c1cccc(Cl)c1)C1CCCO1 C1(C(=O)NCCCN(C(=O)CCc2ccc(OC)cc2)CC)C2CC2C2CC12 C1(NC(CC(=O)NCC)=O)(CNC(=O)Cn2cc(C(F)F)cn2)CCOCC1 C(c1ccc(C)nc1)=CC(N1CCC(N(C(C2CCCCN2CC)=O)CC)C1)=O C1(NC(c2c(C)cc[nH]2)=O)CCN(C(c2conc2-c2ccccc2)=O)CC1C N1(C(C(C)n2cccc2)=O)CC2(C1)CN(C(=O)CNC(C1CCC1)=O)CC2CO N1(C(CCCc2ccc(CC)cc2)=O)CCN(C(=O)CCS(C)=O)C(C)C1 N1(C(c2cc(F)cnc2Cl)=O)CC2CC(C1)N(C(=O)C(O)Cc1ccccc1)C2 CN1CCOCC1C(=O)NC1CCOCC1NC(C1CNC(=O)O1)=O C1(CNC(c2nnc(O)nc2O)=O)CC(F)(F)CN1C(=O)C(C1CCOCC1)F C1(NC(CS(CC)=O)=O)CCCC12CCN(C(C1CC(F)(F)C1)=O)CC2 c1(C(N(CC(C)N(C(=O)CC2CC2(Cl)Cl)C)C)=O)cc(Cl)ccn1 C1(CNC(c2cccnc2CO)=O)CN(C(C2CC3(CC(=O)N3)C2)=O)CCCO1 c1(C(=O)NCC2CN(C(c3c(C)ncnc3C)=O)CC2C)coc(S(C)(=O)=O)c1 C(C(C)(C)CC(=O)NCC(C)(C)N(C)C)NC(c1c(COC)cco1)=O c1(CC(=O)NC(C(CO)NC(c2nc(CC)oc2)=O)C)cc(Cl)n(C)n1 CC(C)C(CNC(C1(NC(c2ccc(F)c(F)c2)=O)CC1C)=O)C(C)C c1(C(C)C)cccc(OCC(=O)NC(CNC(C2CC3CC3C2)=O)CO)c1 C1(CC)CC(C(=O)N(CCCNC(=O)C=C2CCCCC2)CC2CCCC2)CCO1 c1(C(=O)NCCN(C(=O)C(C)C(F)(F)F)CCCCCC)coc2c1C(=O)NCCC2 C(CC(=O)N1CC2CC(CO)C2C1)(C(F)F)NC(C(c1n(C)cnc1)O)=O C#CCC(CC(F)F)C(=O)N1CCC2(CC(C(=O)NCCCOC)C2)C1 S(=O)(=O)(c1ncccc1Br)NC1CC(OC(C)(C)C)C12CCC2 N1(C(C(C)C(=O)NOCCCN(C)C)=O)CC=CC1CN(C)C C(=O)(CC(O)CC(C)C)NC1CC(C)(CC)N(C(=O)CCCC(C)C)C1 FC1COCCC1N=c1[nH]c(N2CCC(F)(F)C2)nc2c1CSC2 C1(CC)CN(C(=O)CNc2nc(C#N)c(Cl)s2)CCC1NS(=O)(=O)CC C1(NC(C(C)OCCC#C)=O)(CO)CN(C(c2ccc(CC)o2)=O)C1 C1(NC(C(C)CN(C)C)=O)CCC2(CC1)CN(c1ncc(Br)cc1C#N)C2 c1(C(N2CC(F)(C(N)=O)C2)=O)ccc(CNC(c2cc(CO)ccn2)=O)cn1 c1(CC(C)CN2CCOC(c3nnnn3CCCF)C2)ccc(O)cc1 c1(C(CO)NC(CN(CCOC)C(C2CCC2C)=O)=O)c(C)cccc1Br C1(CC(N2CC(CC)N(C(c3csc(C)c3C)=O)CC2)=O)NC(=O)CN(C)C1=O c1(C(N2CCN(C(C3(CC)CCC3)=O)CC2)=O)ccc2c(n1)CCC2 C1(C)(COC)CC(NC(=O)C(=O)N(C)C)CN1C(c1cc(OC)nnc1O)=O N1(C(C(=O)OCCC(C)(C)O)=O)CCCCC1c1ccc(Cl)cc1 C1(C)(COC)CN(C(=O)C(c2ccc(OC)c(F)c2)C)CCO1 c1(NC(c2ccc(CC)cc2)c2nnnn2C2COC2)cnc2n1CCOC2 c1(-c2cn(CCC)nc2)ccc(C(=O)NC(C)C)c2[nH]ccc12 S(=O)(=O)(c1cccc(C(=O)NC2CCN(CC(F)F)C2)c1)NC(C(C)C)C(=O)O Cc1nc(N(C2CC3CCC(C2)N3)Cc2ccc(OCF)c(F)c2)cc(O)n1 N1(C(c2c(N(C)C)nccc2)=O)CC2=C(C1)CN(C(C13CCC(CC1)C3)=O)C2 Cc1cccc(CC(=O)NCC2C=CCN2C(=O)COCCCC(C)C)c1Cl C1(CC(N2CCC(c3ccc(F)c(F)c3)C2)=O)CC2(C1)CN(C(=O)CC(F)F)C2 N1(C(CN(C)C)=O)CCCN(CCC(=O)CCN)CC1.C(c1cnc[nH]1)=CC(=O)N C1(NC(C2CC(=O)CN2C(=O)CNC=O)=O)CNC(=O)C12CC2 C1(NC(CSCC#C)=O)CN(C(C2CC(n3ccnc3)C2)=O)C2CCCCC12 CC1(C(=O)NCCNC(C23CC(C2)C(C(F)(F)F)O3)=O)CCC(F)(F)C1 CC1=CC(C)CN(C(C2CCN(C(=O)C(C)(C)N3CCCC3)C2)=O)C1 C1(CNC(C(CN(C)C)N(C)C)=O)COCCN(C(=O)Cc2cc[nH]n2)C1 Cn1nc2c(c1C(=O)Nc1ncco1)CN(Cc1ccc(F)c(F)c1Cl)CC2 N1(C(COCCC=C)=O)CC2(CC(CC(=O)Nc3ccc(Cl)c(C)c3)C2)C1 C1(O)(CCNC(CC2(OC)CCC2)=O)CCCN(C(=O)CC(C)n2ccnc2)C1 CCCCC(=O)C(=O)NCCCCC(=O)NCc1cc(F)ccc1F C(=O)(CC(C)(C)C1CC1)NC(CN(C(=O)CC(=O)NCC1CC1)CC)C C(=O)(CC(C)C(C)(C)C)N1CC2C(C(N(C3CCCC3)CC#C)=O)(C2)C1 c1(C(=O)NCC2(NC(C3C(C=C)CC3)=O)CC2)cc(Cl)c(O)c(Cl)c1 C(CCCC(=O)N(C(C)CCNC(=O)C(C)C#N)C)NC(C)=O c1(SC)cccc(C(=O)NCC2CC(NC(=O)C=C3CCCC3)CC2O)c1Cl Cc1c(Cl)ccc(C(=O)NCC2C(C)CCCN2C(c2nncs2)=O)c1N c1(OC)ccc(C(=O)NCC2CC2NC(c2ccnc(F)c2OC)=O)c(OC)n1 Cc1cc(=NC2CCC(OC(F)F)CC2)[nH]c(CN2C3CCC2CC(O)C3)n1 c1(C(=O)NC(C)CCNC(c2ccc(O)c(O)c2)=O)ncn2ccccc12 Clc1nc2ccc(CNC(c3nnnn3C3CCOC3)c3cscn3)cc2o1 N1(CC(=O)NC(CCN)C(=O)NCc2nc(=N)[nH][nH]2)CC2COCC2(CO)C1 c1(C(=O)NC2CC(CNC(C(C)SC(C)C)=O)CC2O)ccnc2[nH]c(C)nc12 c1(OC(C)C(=O)NCC2CCCN2C(c2cocn2)=O)ccc(CC2CC2)cc1 C(c1ccccc1)=CC(=O)NC1(C)CC(NC(c2ccc(C(C)=O)[nH]2)=O)C1 N1(C(C)C(=O)N(C)C)CCC(C)(CNC(c2csc(-c3ncccn3)n2)=O)CC1 C=CCC(CNC(c1ccncc1F)=O)C(=O)NC1(CSC)CCC1 C(=O)(C(C)(C)CCCC(=O)N1CC(O)(CNC(C2CCS(=O)(=O)CC2)=O)C1)OC C#Cc1cccc(C(=O)NC2(CCC)CCCN(C(C3CCOCC3)=O)C2)c1 c1(OCCNC(C(=O)N(CC(c2ccccc2)(C)C)C)=O)ccc(C#N)cc1 N1(C(C2(C)CCCN(C(C(N3CC(C)C3)C)=O)C2)=O)CCOC2C(O)CC12 C(=O)(CS(=O)(=O)CC1CCCO1)NC(CCNC(C(C)Oc1ccccn1)=O)(C)C c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2C(C)(C)C)ccc(C(C)=O)c(F)c1 CC(C)(C)CCCCCC(=O)N1CC(NC(=O)Cn2cnnc2)CC(F)C1 CCC#CCCNC(=O)CCC1CCCN1C(=O)CC=C(C)C CC(C)CC(C)(C)CNC(=O)CCC1CCC(NC(c2cc(CO)[nH]n2)=O)C1 CC(CC(=O)NC1(c2cc[nH]n2)CC1)C(C)(C)NC(C1CS(=O)(=O)C1)=O c1(N2C3CC(COC)CC2CCC3)nc(Cl)c2c(ccn2C(=O)OC(C)(C)C)n1 C1(CNC(=O)COC2CCOC2)CCCCN(C(c2cn3c(n2)CCC3)=O)C1 c1(C(=O)NC(CC(C)NC(C(C)SCCCC)=O)C)cnn(CCO)c1N C1(C(=O)NC(C)CNC(C2CCC(C#N)CC2)=O)CCCC2(C1)CC2(F)F CC(C(=O)NC1(C(=O)NC2COC(C3CC3)C2)CCOCC1)C(F)(F)F CCCC(CNC(=O)C1=C(Cl)CCOC1)C(=O)NOCC1(C)CC1 c1(C(=O)NC(CNC(CCc2c(C(=O)OC)nco2)=O)C)ncnc2cc[nH]c12 c1(C(=O)O)cncc(C2CCN(C(c3cc(C(F)(F)F)ncn3)=O)C2)c1 N1(C(CC2(C)CC2)=O)CCN(C(=O)CCNc2cnccn2)C2COCC12 c1(OC)ccc(-c2c(C)noc2C)cc1CN1CCN(c2cc(Br)ccn2)CC1 N#Cc1ccc(C(N2CCC2C(=O)Nc2cccc(Cl)c2F)=O)c(F)c1 C1(C(N2CCC(C)(NC(c3cn(C)c(=O)n3C)=O)C2)=O)CCCC2CCCCC12 Cc1c(NC(c2ncc[nH]c2=O)(C)C)ncnc1N1CCOC(C)(C(F)(F)F)C1 C(C)(C)(CCCCNC(C1CCN(C)CC1)=O)NC(C(N1CCN(C)CC1)C)=O c1(C(=O)NCCC2(NC(c3c(COC)cc[nH]3)=O)CCC2)ccc2nncn2c1 CCCCC(O)C(=O)N(CCCN(C)C)CCNC(=O)C(C)(C)CSC CCCCC(CNC(=O)C=C(C)c1ccsc1)NC(c1ccc(COC)cn1)=O C1(NC(CN(C(CNC(C2N(C(CCC)=O)CCC2)=O)C)C)=O)CCCC(C)C1C C1(C)(C(N2CCCC(N(C(C3CCCO3)=O)CC)C2)=O)CCCCC1(F)F C(C(C)(C)C(=O)N1CCC1(C)CC(=O)NCCCCNC(N)=O)OC Cc1c(C(=O)NC2CN(C(c3cnsn3)=O)CC2F)nn2ccccc12 c1(C(N2CCN(C(c3cnsc3)=O)C3C2CC3)=O)ccc2c(c1)OCCNC2=O c1(OC)cccc(S(=O)(=O)N2CCC(C(=O)Nc3ccc([N+](=O)[O-])cc3I)C2)c1 Cc1cnc2c(C(=O)NC3CN(C(c4sc(F)cc4Cl)=O)CC34CC4)cnn2c1 CC(C)C(CO)C(=O)N1CC(F)CC1CNC(=O)CC1OCCC1C N1(C(C2CC(=O)NCC2)=O)CC2CCC1C2NC(C1CCN(CC2CC2)CC1)=O CCCCCC(=O)NCC1C2CC1N(C(c1c[nH]nc1C)=O)C2 O=C(C1=C(F)CN(C(c2ccc(Cl)cc2)=O)CC1)NCCC1(O)CCC1 c1(N(C)CCF)nc2cccc(F)c2c(=NC2CN(c3ccccc3)C2)[nH]1 c1(C(N(CCN(C(C2CC3(CC3)CO2)=O)CC)CC)=O)cncc2cnccc12 C1(C(=O)NC2CCC(NC(Cc3cn(C)nn3)=O)C2)(CNC(N)=O)CCCCC1 N1(C(C=CC=CC)=O)CC(C)CN(C(=O)Cn2nc(Cl)ccc2=O)CC1C C1(C(N2CCC(CC)(Nc3ncnc(=N)[nH]3)CC2)=O)CCOC2(CCCC2)C1 C1(C(=O)NCC2(CC)CCOC2)CCCCC1NC(=O)C(O)CSC c1(NC(c2c(OC)cccn2)C)ccc(S(=O)(=O)N2CCCCC2C)cc1Cl C(=O)(CC(C)C(C)(C)C)N1CCC(C(C(=O)NCc2cc(C)sc2C)(C)C)C1 c1(OC)ccc(C(c2nnnn2C2CC2)NCC2CC(=O)N(C)C2=O)c(F)c1 N1(C(C2CCCC(CC(F)(F)F)C2)C(=O)NCCC#N)CCC(O)CC1C1CC1 C(C)(C)(CC(=O)N(C)Cc1cn(CC2(O)CCC2)nn1)OC N(C1CCc2cc(CNC(=O)Cn3nc(O)ccc3=O)ccc21)C(=O)C1CC1 c1(C(N2C(CC(=O)OC)CCC2)=O)cc(C(=O)O)n2ncccc12 c1(NC(C2N(S(C3(CC=C)CC3)(=O)=O)CCCC2)=O)ccc2nnsc2c1 c1(C(=O)NCC2CCC(NC(C#CC(C)(C)C)=O)C2)ccnc2[nH]ncc12 C1(NC(c2c(CC=C)cccc2)=O)CN(C(=O)CCC(=O)N(C)C)CC2(CC2)C1 C1(C(=O)NC2(C)CC=CC2)CCC(C)(C)N(C(=O)CC2CCCC(=O)C2)C1 c1(C(N2CC(C)(NC(C=CC(=O)OCCCC)=O)C2)=O)n[nH]c(C)c1[N+](=O)[O-] c1(C(N2CC3(CC(O)CO3)C2)=O)cc(O)nc2c1CN(C1CC1)CC2 C(c1ccc(F)cc1)=CC(=O)NCCN(C(=O)C=CC(=O)N(C)C)C(C)C c1(CC(=O)NC(c2ccccc2)CNC(c2c(C)noc2)=O)ccc(F)c(F)c1 n1(CC(C)OC(C)C)cc(C2(NC(CNC(CSCC)=O)=O)CC2)nn1.CC c1(OC)c(F)cc(C(=O)NC2CC3CC2CN3C(c2ccc(O)cn2)=O)cc1Cl C(=O)(C(F)C(F)(F)C(F)(F)F)N(CC(CNC(c1c(C)ccc(C)n1)=O)C)C C1(CO)CN(N2CCCC3=C(Nc4c(F)ccc(F)c4O3)C2)C1 C1(CCN(CC)Cc2cnoc2C)CCCN1C(=O)C(C)N1CCCC1 c1(OC)cccc(C(N2CC3CC(C2)N3C(C2(OC)CCC2)=O)=O)c1NC(C)=O N#CC1(C(=O)NCCNC(c2ccc(OC3CCCCC3)nc2)=O)CCCO1 C=CC(C)(C)CC(=O)NC(C1CCOC1)CNC(c1ccc(C(F)F)cn1)=O C1(Nc2cccc(OC)c2C)COC2(CCN(C(=O)OC(C)(C)C)C2)C1 c1(C(=O)NCC(C)NC(C(C(=C)C)(C)O)=O)c([N+](=O)[O-])ccc(C)c1C C1(=C(C)NC(C)C2CC2)CCN(c2cc(-c3ccccc3)ncn2)CC1 C1(NC(c2cncc(F)c2Cl)=O)CCN(C(=O)Cn2ccc(O)nc2=O)CC1O C#CCCCC(C)C(=O)N1CC2(CNC(=O)C(F)C3CCC3)CC1CCO2 c1(C2C(NC(N3CCC(NC(c4ccco4)=O)CC3)=O)CC2)ccc(F)c(Cl)c1 C1(CNC(c2cc(CCC)ncc2)=O)C2CCC1CN(C(=O)Cc1cccs1)C2 C1(CN(C(C=NOC)=O)C)CCCN(C(c2sc(N3CCCCC3)nc2Cl)=O)C1 C1(CNC(C2CCC(C(C)C)CC2)=O)CN(C(=O)C=Cc2ccsc2)CC12CC2 Cc1ccc(CN=C(NCC2CCC23CCC3)NC2CCS(=O)(=O)C2)c(C)c1 c1(CC(=O)NC2CCCC(NC(C3C(C)C3)=O)C2)coc2c(F)c(F)ccc12 CC1(C(=O)NC2CCN(C(c3sncc3Br)=O)C2)CC=CCO1 CCC(O)C(F)(F)C(=O)NCC1CC1NC(=O)C(=O)N=S(C)(C)=O Cc1nc(C)c(CCC(=O)NCCC2CCCN2C(=O)C(C)(C)CF)c(O)n1 CC1C(NC(=O)CN2CSCC2=O)CCCN1C(=O)C1=NOC(C(C)(C)C)C1 CCC(CNC(=O)C=CC(C)(C)SC)(CC)C(=O)N1CCOC(CCF)C1 N1(C(C(=O)Nc2cc(C#C)c(C)cc2)=O)CC(C2CCC2)CCC1C Cc1ccc(C(=O)NC2CC(CCNC(=O)C(C)c3cccs3)C2)c(C)c1 C1(N(C(CCc2cncc(OC)c2)=O)C)CCCN(C(C2CC2CF)=O)CC1 c1(C(=O)NCC2(NC(=O)CC3COC(=O)C3)CCCC2)cc2nc(=O)ccn2[nH]1 c1(OC)cc(C(N2CCC(O)(CNC(C34CC3CCC4(F)F)=O)C2)=O)cc(F)c1 c1(OCC)cccc(C(=O)NC2CCCC(NC(=O)Cc3ccoc3)CC2)c1N CC#CCCCC(C)(c1nnnn1CC1CCOCC1)NCCC1C=CCC1 C1(CNC(C(CCN(C)C)NC(=O)CSc2nc[nH]n2)=O)NC(=O)OC1(C)C C1(C(=O)NC2(C)CCC2)CN(C(=O)NC2CC2)Cc2nccn2C1 C1(NC(C2(c3cccc(C)c3)CC2)=O)CN(C(=O)CCC(C)(F)F)CCC1O N1(C(C2N(C(C)=O)CC(F)(F)C2)=O)CC2CCC(C1CO)N2C(C1C=CCC1)=O C1(NC(CCCNCC(F)(F)F)=O)CCN2CC1NC(=O)C2=O.CN(C)CCO c1(C(N2CCC(C(C(F)(F)F)NC(CC=C)=O)CC2)=O)noc2c1COCC2 N1(C(C2CCN(C(c3c(C)cco3)=O)C2(C)C)=O)CCC2(CC1)CC2C#N CN1C(=O)CCC1(C)CNC(=O)CC(C)(C)N(C(=O)C=C1CCCCC1)C N1(C(CN(C2CCC2)C)=O)CCC2(CC(NC(=O)C(N3CCCC(C)C3)=O)C2)C1 n1(CC)nnc2cc(C(=O)NC3CCCC(NC(c4cnn(C)c4)=O)C3)ccc12 c1(C(=O)NC2CN(C(CCc3ccc(C)nc3)=O)CC2C)cccc(C)c1F C(=O)(C(F)C(F)(F)F)NCCC1(NC(C2C=CCC2)=O)CC1 c1(CN2C(OCC)CCCC2)cc(C)cc(C#N)c1 CC(CC(=O)NCC=C1CCN(C(=O)CC(C)(C)C(F)F)CC1)C(F)(F)F c1(COC)ncc(C(=O)NCC2(O)CC(NC(C3(C#N)CC3(C)C)=O)C2)c(O)n1 C1(C(=O)NC(C(=O)NCC2(F)CCC2)C2CCC2)COCCO1 Cc1cc(C(=O)N(CC(=O)NC2CCC(F)(F)C2)C(C)C)c(C)n1C c1(C(=O)NC(CC)CNC(c2cnc(COC)s2)=O)c(C)ccnc1O Cc1cnc(C(=O)NC2CCCC2CNC(=O)Cc2ncoc2C)cn1 C1(NC(c2ncc(CC)nc2)=O)(CO)CCCN(C(=O)C(C)(O)CC)C1 c1(C(=O)NCC(CNC(c2cccc(O)c2F)=O)OC)cc(F)cc2ccoc12 C(c1nc2ccccc2o1)=CC(=O)NCC=CCNC(=O)CC1CCCC1O c1(C(=O)NC(C(=O)NCC(CC)CC)C(C)C)ccc(C)c(C#N)c1 N1(C(C2(CC=C)CC2)=O)CC(CNC(=O)CN2C(C)CCC2C)C(C)C1 c1(CC(=O)N(CC(CNC(CCC)=O)O)C)ccccc1OC C1(F)(C(N(CC#C)CC2CC2)=O)CCCN(C(C2CN(CC)CCO2)=O)C1 C=CCC(C)(C)CC(=O)NC1COC2(CNC(c3ccc(O)cc3)=O)CC1C2 Cc1cc(C)c(C(=O)OC(C)C(=O)Nc2ccc(Br)cc2)s1 c1(NC(C2C3CN(c4cc(SC)nc(C)n4)CC32)=O)nc(Cl)c(Br)cc1I CC1CCC(C)(C(=O)NCC23CC(NC(=O)C(C)C(C)n4cccn4)(C2)C3)CC1 C1(C(=O)NC(c2cccnc2)CC)CN(C(c2sc(Br)nc2C)=O)CCC1O CC1CCc2onc(C(N3CC(NC(c4cccc(S(C)=O)c4)=O)C3)=O)c2C1 c1(CC)cc(C(N2CCC(COC)(NC(c3cc(O)ncn3)=O)C2)=O)ccc1C C1(N(C(CC(C)SC)=O)C)CCCCN(C(=O)CC(=O)OCCC(C)C)C1 c1(C(=O)NC2C(NC(C3CN(C(N(C)C)=O)C3)=O)CC2)ccc(F)o1 CC(CCC(=O)NCCNCC(=O)NCC(c1ccco1)O)S(C)(=O)=O c1(CC)nccn1CC(=O)NC(C(=O)N(C)CC1CCCCO1)C1(O)CCC1 N1(C(COC)=O)CCCC(C(=O)OC)C(F)C1.c12cc(ccc1Br)CCC(=O)O2 Cc1cc(C(=O)NCC2(F)CC(CNC(=O)CC3CC(O)C3(C)C)C2)c(C)[nH]1 C1(CC(=O)NC(C2CCCN2C(=O)CSCC(N)=O)C)C(C)(C)C1(C)C N1(C(CN(C(=O)CC2CCCOC2)C(C)C)=O)CCC(C(F)F)C1 c1(C(=O)NCC(CC=C)NC(c2cccc(OC)n2)=O)cccc(C)c1 C1(CC)C(NC(c2nnn(C)c2N)=O)CCCN1C(=O)CC1CC1(Cl)Cl Cc1cc(C(N2CC(O)CC2C(N2CC(CC3CC3)C2)=O)=O)c(C)cn1 Cc1c(C(=O)NCC2CC(C(=O)NC3(CC4CCC4)CC3)=NO2)cccc1O Cc1cc(Cc2nc(C(C)N(C)C)nn2-c2ccn(C)n2)[nH]c1C#N c1(C(N2CCOC(COC)C2)C(=O)NC)cc(OC)cc(Br)c1.c1(C)ccc(F)cc1 c1(C2(C)COC2)ccc(C(=O)NC2CN(C(c3cccs3)=O)C2)cc1 N1(C(CNS(CC)(=O)=O)=O)CCC(c2ccccc2)C(NC(c2ccsn2)=O)C1 c1(C(N2CC(C3(NC(C4CCN(C(C)=O)C4)=O)CC3)C2)=O)cc2occ(C)c2[nH]1 C(F)(C(=O)N(CC(O)CN(C(=O)C(C)n1ccnc1)C)C)=C(C)C c1(C(N(CCCCNC(C2(CF)CC2)=O)C)=O)ccc2c(c1)SCCN2 c1(C(N(CCCNC(C2=CC(C)CC2)=O)C)=O)cnn2cccc(Cl)c12 C1(C(C)(C)C)C(=O)N1.C(CC(=O)NCC1(CF)CCC1)NC(=O)OC N(C1CN(C(=O)COCCF)CCc2ccccc21)C(c1c(Cl)nc(OC)s1)=O Cc1nnc2n1CCN(C(=O)C(N1CCNC(CO)C1)=O)C2C CN1CCCC(C(N2CCC(C(F)F)(CNC(=O)CC3CCC(=O)NC3)C2)=O)C1 C1(C(=O)NC2(CN(C(=O)CCc3nccs3)C)CC2)CCCC(O)C1 C1(C(N(CCN(C(C2CC(OC)C2)=O)C)C(C)C)=O)CC(C)(C)CCO1 c1(C(N2CCC(NC(C3C(C=C)OCC3)=O)C(O)C2)=O)ccc2c(c1)CCOC2 N1(C(=O)CC2(O)CCC2)CCC2C(CCN2Cc2n[nH]c3ccc(Br)cc23)C1 N1(C(C)C)CCN(C=O)CC1.c1(CCNc2cc(C)no2)cccnc1Br c1(C(N2CC(C(C)NC(COC)=O)OCC2)=O)c[nH]c2cccc(C)c12 Cc1cc(Cl)c(Cl)cc1C(N1CCCC(NC(=O)CSc2nncn2C)C1)=O N1(C(C(CC)N2CCCC2=O)=O)CCC(O)(CO)CC1 c1(C(=O)NCCC2CN(C(C3(C)COC(=O)C3)=O)C2)cc2cccnc2cc1F C(=O)(C(C)CC(C)(C)C)NC(CN(C(COCCCCOCC#C)=O)C)C N1(C(C2CC(SC)C2)=O)CCCCC2(CCN(C(c3ccnc(C)c3)=O)C2)C1 c1(C(=O)OCC)cc(NC(=O)NC2CCCC(C(N)=O)C2)cc(F)c1 C=CC1CN(C(=O)C(C)(CNC(=O)CCC(CC)OC)CC)CCO1 C(=O)(CC(C)C(F)(F)F)N1CC(OC)C(NC(=O)CN2CCC(CO)CC2)C1 c1(C(N(CC(=O)N(CCC(=O)OC)CC#C)C)=O)cc(F)ccc1F C12(C(N(C(C)CCNC(=O)CN(C)S(N)(=O)=O)C)=O)CCC(O)(CC1)CC2 c1(COC)ccoc1C(=O)NC1CCC1NC(c1csc(CCC(F)(F)F)n1)=O C1(C(N(CC=C)CCO)=O)CCC(C)CN1C(=O)C=Cc1ccccc1 C(C)(CO)(C(=O)NC1CC(CN(C)C)C1)NC(C1C(C)=CCS1)=O N(C(=NCCC(C)=O)NCCc1ccccc1NC(C)=O)C1CC(=C)C1 c1(CC)cc(F)c(C(=O)NCC2COCC2NC(c2[nH]cnc2C)=O)c(F)c1 c1(C(CNC(CCCC)=O)N(C(=O)CCc2scnc2C)CC)ccc(C)cc1 C1(CC=C)(NC(=O)C(O)C(F)(F)F)CCN(C(=O)CO)CC1 c1(NC(C(=O)OC)Cc2ccccc2)ncnc(N2CCCC2)c1N C1(CC)CN(C(=O)C(C)(C)SC)CCN1C(=O)C(C)C=Cc1ccccc1 C1(CNC(C2N(C(=O)NC)CCC2)=O)C(C)CCCN1C(c1ocnc1C)=O c1(C(=O)NC2CCN(C(=O)C3=NOCC3)C2)n[nH]c2cc(Br)ccc12 c1(C(=O)NCC(CC)NC(c2cnnc(Cl)c2)=O)cc([N+](=O)[O-])cn1C C(=O)(C1CC(=O)Nc2ncccc21)N1CCC(C(C)NC(c2ccco2)=O)CC1 CCC(C)(C)C(O)C(=O)NC1CCN(C(c2cc(C(F)F)ccc2F)=O)C1 c1(C(=O)OC)ccn(CC(F)(CN)C(C)C)c(=O)c1 CC1CC(C)CCN(C(C2(NC(c3sccc3C#N)=O)CC2(C)C)=O)C1 N1(C(C2(N(c3ccccc3)C)CC2)=O)CCC(NC(C2(C)CCCS2)=O)C1CO C(=O)(C1=CN=C2N=CNN2C1)NC1C=CCN(C(c2n(CCC)ccc2)=O)C1 c1(C(N(C)CC2(NC(C3CCCCC(=O)N3)=O)CC2)=O)ccc2ccc(O)nc2n1 c1(N(C(C(=O)NCC2(COC)CC2)c2ccco2)C)cccc2ccoc12 N1(C(C2CC(=C)C2)=O)CC(OC)CC1(C)CNC(=O)C(=Cc1cn(C)cn1)F C1(NC(Cc2cc(C)sc2)=O)CN(C(=O)CCC(C)(C)N(C)C)CC2(CC2)C1 CCC(CC(=O)NCCC1(NC(=O)C(C)(C)c2cscn2)CCCC1)SC c1(C(N2CCC(OCCNC(C(C)SC)=O)CC2)=O)cccc(=O)n1C C1(NC(C(CCC)N(C)C)=O)CS(=O)(=O)C12CCN(C(C1(CF)CC1)=O)CC2 C=CC1CCCCN1C(C1CCCC(C)C1)=O c1(CC)cc(NC(C2CCCCN2C(c2ccc(C3CC3C)o2)=O)=O)ccc1Cl N1(C(c2c(CC)ccs2)=O)CCC(C)(C)C1C(=O)NC1CN(C)CC1(F)F C1(C2CC2)(NC(C2(CS(N)(=O)=O)COC2)=O)CCN(C(c2ncccc2Cl)=O)C1 c1(C(C)=O)cc(N2CC3CC(NC(=O)CC(C)C4CC4)CC2C3)ccc1[N+](=O)[O-] C1(c2onc(CC(=O)NC3CCN(C)CC3)n2)CCOCC1(C)C c1(C(=O)NCC(CNC(C(CC)CO)=O)O)cnc(C)nc1COC Cc1csc(C(F)(F)C(=O)NC2CC(C)(NC(=O)C(n3ccc(C)n3)C)C2)n1 Cc1cc(C(=O)NC(C2CCCN2C(c2cc(=O)cc[nH]2)=O)C)oc1C C1(C(C)(C)NC(=O)C(C2CC2)C2CC2)CCN(C(C2(CO)CCCO2)=O)CC1 C1(NC(=O)CCCc2ccsc2)CN(C(c2cc(Cl)c[nH]2)=O)C2CC12 C1(C(N2CC(C(C(=O)N(C(C)C)CCN(C)C)O)C2)=O)CCCCCN1C C1(C(=O)NCCC(C)(CC)NC(c2c(CC)nco2)=O)OCCCC1(C)C C1(CNC(CC)=O)CC2(CCN(C(=O)Nc3c[nH]cc3C(C)(C)C)CC2)CO1 C1(C(=O)NC(CC)CN(C(=O)CCc2nccn2C)C)(CC)CCOCC1 C(=O)(C1=CCCC1C)N(CCC(=O)N(C)Cc1ncc(C)o1)C1CC1 CC(C(=O)NCC(O)CCNC(=O)Cc1cc(F)cc(Cl)c1)C(C)(F)F N1(C(C(C)OCCCC)=O)CCC(NC(=O)C(O)COC)C12CCCC2 C1(C(=O)O)C2C=CC2CN1C(c1ccc(Br)cc1Br)=O CCCC(C(F)(F)F)NC(C1(F)CCN(C(C2SCC=C2C)=O)CC1)=O C1(C2CN(C(=O)C=C3CCCC3)C2)(N(C(CC(C)(C)C)=O)C2CC2C(F)F)CC1 Cc1[nH]nc(CO)c1C(N1CCC1C(N1CC2CC2C1)=O)=O c1(C(=O)NCC(CC)(CC)NC(c2c[nH]c(C(N)=O)c2)=O)ccc(OC)c(C)c1 N1(C(c2cn(CC(=O)OC)nn2)=O)CCC(NC(C2CCCC2)=O)C(C)C1 c1(C(C)(C)C)nnc(N2CCCC2C(=O)NCC2C(C(F)(F)F)C2[N+](=O)[O-])o1 C(=O)(CCCCC(C)C)N(C(CC)C(=O)NCCCC1CCOC1=O)C N1(C(C2(C(C)C)COC2)=O)CC2(C1)CN(C(=O)COc1ccc(F)cn1)C2 c1(CC)nn(C)c(CC(=O)NC2(CCNC(c3ccsc3Cl)=O)CC2)c1Cl c1(C(N(CCC)CCNC(c2cnn(CC)c2)=O)=O)cc(COC)cn1C c1(C(=O)NCCCCNC(c2cc(OC)cc(F)c2)=O)cc(O)cc(N)c1Cl CC(CN(C)C)CCC(=O)N1CC(C)(C)CC1CNC(C1CC12CCSCC2)=O C(C(C)C)(C(O)C(=O)N1CC2(C1)CN(C(=O)CCNC(C1CCC1)=O)C2)OC C1(C(N2CCC(C=C)CC2)=O)CC12CCN(C(=O)C(COC)N(C)C)CC2 S(=O)(=O)(c1ccc(N(C)CC2C(C)(C)C2(C)C)cc1Br)N(C1C(C)CCCC1)C c1(OC)cccc(C(N2CCC(NC(c3c(C)ncn3C)=O)CC2C)=O)c1C N1(C(C(C)(C)NC(C)=O)=O)CC(O)CC1C(N1CCN(Cc2ccoc2)CC1)=O C1(CCC(=O)NCC2(OC)CN(C)C2)CCN(C(=O)C(C)n2ccnn2)CC1 CCC(C)(CN=C(NC(c1ccc(C(C)C)cc1)C)NC1CCCCC1)OC c1(C(N2CC(C(C)NC(Cc3c(C)nn(C)c3)=O)C2)=O)ccc(O)c(F)c1F Cc1ccc(Cl)c(C(=O)NCC(C2CC2)NC(c2ccc(OC(C)C)cc2)=O)c1 C=CC(C)(C)CC(=O)N1CCC(O)(CCNC(=O)C(CCC)OC)C1 Cc1ncc2n1CCN(C(C1(CCNC(c3cnc4n3CCC4)=O)CC1)=O)C2 Cc1nn(C)cc1C=CC(N1CC(N(C)C(C2CCCC(C(F)(F)F)C2)=O)C1)=O C1(CN(C(CCCN(C(C)=O)C)=O)C2CC2)CN(C(=O)C2CC2)CC1C CC1(C)OC2(C(=O)NC3CCN(C(c4c[nH]c5ncccc45)=O)C3)CCC1CC2 CCC(CC(=O)NCC(C(=O)NCCc1ccnn1C)OC)C1CCC1 c1(C(=O)NC2CCC(C(N(C(C)CN(C)C)C)=O)C2)cncc(Cl)c1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2CCN(C(=O)C(C)(C)SC)CC2C1 C(C)(C)(CCC(=O)NC1(CCCCNC(=O)CCN2CCCC2=O)CC1)OC C1(NC(C2C(C)(C)C2C#N)=O)CCCC12CN(C(c1cnc3[nH]ccc3n1)=O)C2 c1(C(=O)NC(CC)(C)CNC(C2(C(=O)NC)CCC2)=O)cnn2ccncc12 C=CC1(CC)COCCN1C(=O)C(n1cnc(C#N)n1)CC c1(NCC=C(C)C)cc(C)c(S(=O)(=O)NCC2CCC(C)(C)O2)cn1 Nc1c(C(=O)NCC2CC3CCC2N(C(c2cnoc2)=O)C3)ccc(F)c1F Cc1cc(N)c(C(=O)NCC(C)NC(C2CCCN2C)=O)nc1C N1(C(N2CCC(C)OCC2)=O)CC2(CCCCC2)CC1C O=C(CC1NC(=O)NC1=O)NNC(=O)c1cccnn1 c1(C(=O)NCC(CO)NC(Cc2c(C)ccs2)=O)ccc2c(c1)COCCN2 Cc1cnncc1C(N1CCCC(C(=O)Nc2ccc(C(N)=O)nc2)C1)=O CN1CC(C)(NC(C2(C)CN(C(=O)CN3CCNC3=O)C2)=O)CCC1=O c1(CC)ccc(CNc2ccn(C3CCC3)n2)c(C)c1 CC1CC(NC(=O)C=CCO)CN1C(c1cnc(S)n1C)=O C1(C(=O)NCCN(C(CCCOC(C)C)=O)CC(C)O)CC2CCCCC12 c1(C(=O)NCCSCCO)cccc(-n2cc(-c3cncnc3)nn2)c1 C(CN=C(NCC(C)(O)C(F)(F)F)NCc1cccc(C(C)C)n1)OC c1(CNC(C2(CCC=C)CC2)=O)cc(C(=O)NCC(C)C(C)C)ccn1 c1(C(N2CCCC(NC(C)=O)C2)C(=O)NCCSC)cc(OC)c(OC)cc1C N1(C(C(C)n2cccc2)=O)CCCC(C2CC2NC(=O)Cc2cnn(C)c2)C1 c1(C(=O)NC2CC(C)N(C(c3ncc(Br)cn3)=O)C2)cc(F)cnc1O c1(OC)cc(CC(=O)NC2CC(C(C)NC(=O)CC3CC(C)=NO3)C2)on1 C1(CNC(CC2(C=C)CC2)=O)CC(NC(=O)CCCc2ccccn2)C1(C)C CCC(O)CC(=O)NCCCC(=O)NCCc1cccnc1F C1(NC(C2CCS(=O)(=O)N2)=O)CC2C1CCN2C(c1cnc2sccn12)=O c1(C(=O)NC23CC(C(=O)NC(C=C)(C)CC)(C2)C3)cnc(O)c(F)c1 CCS(=O)(=O)c1ccc(F)c(C(=O)NC23CC2CN(C(=O)C2=CCCC2)C3)c1 N1(C(CCCN(C(C2C(C)CCCC2)=O)C)=O)CCC2CCCC2CC1 C1(CNC(C(C)CCO)=O)CC(F)(F)CN1C(c1ncc(Cl)n1C)=O CCC(C)(O)C(=O)N(CCc1cn(-c2ccnc(C(=O)O)c2)nn1)C1CC1 C12(Cc3ccc(C(=O)OCc4cnn(C(F)F)c4)o3)CC3CC(CC(C3)C1)C2 C1(C(C)C)CC(CC(=O)N(C2CCN(C(=O)CC=C(Cl)Cl)CC2)CCO)CCO1 C(N=c1[nH]c2cccc(F)c2s1)C1N(C(C2CC=CCC2)=O)CCCC1 c1(C(=O)NC2CN(C(c3c(CC)nc[nH]3)=O)C(C)CC2)nc2ncccn2n1 c1(C(=O)OC)c(C(=O)NC(CNC(C2CN(C(C)C)C2)=O)CO)n[nH]c1C C1(C(=O)NCCN(CCC)CC)CN(C(C2(C#N)CCCO2)=O)CC1F c1(C(=O)NC2(C)CCN(C(C(C(C)C)NC(N)=O)=O)C2)ccc(F)cc1N c1(C(=O)NC(C)CCCNC(c2ccc(CN=[N+]=[N-])o2)=O)n[nH]c2c1CCOC2 c1(C(=O)NC(c2cc(C)c(C)s2)CC)cccnc1Nc1cccnc1 c1(C(=O)NCC(CNC(=O)COCc2ccncc2)F)ccc(F)c(O)c1F C1(N(C(Cc2ccc(C)o2)=O)C)CN(C(C2CC(F)(F)C2(C)C)=O)CC12CC2 C1(CC)(CO)CCOCC1.C12(NC(C3N(CC)CC3)=O)CC(C1)NC(=O)C2 Cc1ccccc1-n1ccc(C(=O)NC(CNC(c2cnn(C)n2)=O)C(C)C)n1 C#CCCC(O)C(=O)NCC1(C(N)=O)CN(C(=O)C(C)(C=C)CC)C1 c1(OC)cnc(F)c(C(=O)NC(C)CC2CN(C(C3(OC)CCCOC3)=O)C2)c1 C1(NC(C2(C)CC2(F)F)=O)CN(C(c2nonc2N)=O)CC1c1ccccc1 Cn1nc(C(=O)NC2(C)CCC(NC(=O)CCC(C)(C)F)C2)cc1C#N c1(C(=O)NCC2N(C(C3NC(=O)OCC3)=O)CC2)ccc(=O)n(CCF)n1 Cc1ccc(N)c(C(=O)NCc2ccc(C(C)NC(C3CC3(F)F)=O)cc2)c1F n1(CCC)nnnc1C(c1cncs1)NCCSC(F)F c1(SC(C)C(=O)NCC(CNC(C2(C)CC=CC2)=O)CO)ccc(F)cc1F c1(C(=O)NC(CCCCNC(CCC(C)OCC)=O)C)n[nH]c2c1CCCCC2 c1(C(=O)NC(C2CN(C(=O)CC3CCOC3=O)C2)C)cc(F)c[nH]1 c1(C(=O)NC(c2cn(-c3nonc3C(=O)O)nn2)C)ccnc2c1cnn2C c1(CC(=O)NC2C3CN(C(c4cnco4)=O)CC23)cn2cc(F)ccc2n1 c1(NC(C2(C)CN(C(CCn3ccc(C)n3)=O)C2)=O)cc(F)cc(Br)c1 C1(OC)CCC2(CCN(C(=O)CN(C3CCCO3)C(C3CCCC3)=O)C2)C1 n1(CC)nccc1C=CC(=O)NCCC1(O)CCN(C(C2CC2C(F)(F)F)=O)C1 C1(CN(CC(=O)NCC)CC)CCN(C(C2CC(n3ccnc3)C2)=O)C1 C(C(F)(C(=O)NCC(C)(O)C1CC1)C(C)C)NC(C1(OC)CCCCC1)=O c1(C(=O)NCC2(F)CCN(C(CC(C)C(F)F)=O)C2)ccc2c(c1)CCO2 C(CCCc1ccccc1)(C(=O)OC)c1nnc(-c2cccc(OC)n2)o1 N1(C(C(C(C)O)(F)F)=O)CCC2(CCC2)C(NC(=O)Cn2cnnn2)C1 N1(C(=O)NCC2NC(=O)CN(CC)C2)CCC(S(=O)(=O)NC)CC1 N1(C(c2c(CC)ocn2)=O)CCC(CNC(c2[nH]c(=N)ccc2C)=O)C(C)C1 c1(C(=O)NC(CNC(C)=O)C2CC2)cnc2n(c1=O)CCS2 N1(C(=O)OCC(C(=O)OC(C)(C)C)Cc2cncs2)CCC(C2CC2)CC1 Cc1cccc(C(C)C)c1C(N1CCOC(CNC(C2(P(C)(C)=O)CC2)=O)C1)=O C12(C(C)NC(C3CCNN3C(C3CCCS3)=O)=O)CCC(CC1)C2 C=C(C)C(CC(=O)NCCCOCCNC(c1ccon1)=O)OCC N1(C(CCC(C)OC)=O)CCCCC(NC(=O)C=Cc2cnn(C)c2)C1 c1(C(=O)NC2CC(NC(Cc3ccc(C)c(O)c3)=O)C2)cc2sc(Cl)cc2s1 C1(C(=O)NOCC2CCOC2)CCCCN(C(C2CN3CCC2C3)=O)C1 C1(CNC(C(CC(C)C)C)=O)CC2COCC2N1C(=O)CSCCC(F)(F)F C(=O)(C(F)CC(C)(C)NC(C1CC2C=CC1C2)=O)N(C1CCN(C)CC1)C N1(C(C(C)N(C)C)=O)CCCC2(CCC(NC(C3CCCCCCC3)=O)C2)C1 N1(C(CCC)=O)CCN(CCNC(C2CCC(=O)N2C)=O)C2(CCC2)C1 C1(CNC(CCCSC)=O)(NC(=O)CCOCCOCCCO)CCCCC1C c1(CC)cccc(C(=O)N(C)CC2CCCN2C(=O)CC2CCOC2)c1 c1(C(=O)NCC2N(C(C=CC)=O)CCOC2)cc2cncn2c(O)n1 CCC1=NOC(C(=O)N(CCCNC(c2coc(-c3ccccc3)n2)=O)C)C1 c1(C(=O)NCCC(CCNCc2scc(C(=O)OC)c2)C)n[nH]c2c1COCC2 c1(C(N2CC3C(NC(C4C(C(N)=O)C4)=O)(C3)C2)=O)cc2ccc(Cl)cc2c(O)n1 CN1CCCCC(NC(=O)CC2CC(NC(C3(C#N)CCCO3)=O)C2)C1=O Cc1cc(C(=O)NCCCCCN(C)C(C2CC23CCOC3)=O)cc(C)c1C C1(OC)CC(NCC(C)OC)C12CCNCC2 c1(-c2cccc(-n3c(C)cc(C)n3)c2)ccc(S(=O)(=O)CCO)cc1 C1(C(=O)OCCSc2ccc(Cl)cc2)CC(F)(F)C12CCC2.CN1C(=O)O1 C1(C(=O)NCC(C)(C)NC(=O)CC2CCC(=O)NC2=O)CCCCC(F)(F)C1 C1(C(=O)NC(CN(C(c2cc(C)c(F)cn2)=O)C)C)CC=C(C(C)C)CC1 N1(c2nc(C#C)c(C)cn2)CCC(CC(N)=O)C(C2CC2)C1 Cc1sc(C)c(C(=O)N(C)CCNC(C2CCC3CC3CC2)=O)c1Br CC(O)C(C)C(=O)N(CCCCNC(C1(c2ccccc2)CC(F)C1)=O)C Cc1ccc2cccc(NC(=O)C(F)(F)C3=CCOCC3)c2n1 C1(NC(C(C(C)C)c2cc(C)no2)=O)COC2(CCN(C(=O)C=CCF)CC2)C1 N1(C(C2C3(CC(NC(CN(C(COC)=O)C)=O)C3)C2)=O)CCCCCCC1 n1(CCOCC=C)c(N(C2CC2)Cc2ccc(CC(C)C)cc2)nnc1C1CC1 N1(C(COCCOC)=O)CCC(CNC(c2nc(C)nn2C)=O)CC1 c1(CCC(=O)NCCC(C)N(C(C(CSC)O)=O)C)c(F)cccc1F c1(NC(C(=O)OC)=O)cc(Cl)c(C)c(C(C)NC2CC=CCC2)c1 N1(C(C=C(CC)C)=O)CCN(C(c2cn(CC)nn2)=O)CC1CCOC C1(NC(C(CC)N(C)C(c2ccc(C#N)[nH]2)=O)=O)CCCC(O)C1 c1(C(=O)NCC=CCNC(c2c(C)nns2)=O)ccc(O)cc1F Cc1ncc(CCC(=O)NCC(O)CCNC(c2nocc2Cl)=O)o1 N1(C(CCC2(NC(C(C)c3cc[nH]n3)=O)CCC2)=O)CC2CCCC1C2 N1(C(CSCC)=O)CC(CNC(c2ccc(Cl)cc2C(F)F)=O)CC1(C)C C1(C(N2C(C)(C)C(NC(=O)CC3CC4CC4C3)CC2)=O)CCCC(F)(F)CC1 C1(NC(C23CC(CN(C(C4CCCSC4)=O)C2)C3)=O)CC2COCC(C1)C2 CC1C(=O)N2CC(CO2)n2cc1nn2.N1(CC2CCCCC2)CCCCC1 C1(COC)(NC(c2ccc(-c3cscn3)cc2)=O)CCN(C(=O)CS(C)(=O)=O)C1 C(=O)(C(CNC(C1C(C)C1C)=O)N(C)C)NCCC N1(C(C(c2nccc(C)c2)(F)F)=O)CC2(CC2)CC1CNC(=O)C1=CCCC1C C(=O)(CC(O)CC(C)(C)C)NCC1(CNC(C(CC=C)CC)=O)CCC1 N1(C(c2scc(OC)c2)=O)CC(NC(=O)CCC2CCCCO2)C2CCCC12 c1(CNC(COCC=C)=O)cncc(C(N2CCCC2CC(C)C)=O)c1 S(=O)(=O)(CCN=c1cccc(S(=O)(=O)N2CC(C)OCCC2C)[nH]1)NC O=C(CCN(C(=O)CCn1ccnn1)CCCO)NCC(O)CC1CCC1 Cc1ccc(S(=O)(=O)NC(c2cnc3n2CCOC3)=O)cc1C(F)(F)F C1(C(=O)NC(CC(C)C)CNC(=O)C(C)(C)C2CC2)CCCCC12CC2 c1(C(=O)NCC(O)CC(=O)NCc2ccncn2)cnc(O)c(F)c1 C1(NC(=O)NC(CCOC)COC)COc2ccccc2NC1=O C1(C(=O)OC)C2CN(C(=NCCCCCF)NCC(c3ccccc3)O)CC12 C1(NC(C(COC)C)=O)CN(C(=O)CNC(C)=O)CC2(CCC2)C1 c1(C(=O)NC(CC)CN(C(=O)C2=C(C)CCC2)CC)cccc(P(C)(C)=O)c1 c1(C(N(C(C(=O)NCCC(C)SC)C)C2CC2)=O)cc(C2CC2)no1 C1(CNC(=NCc2ncc(F)cc2F)NC2CC2)CCC2C(CC1)C2(F)F N1(C(c2cc(N)ncc2)=O)CCN(C(c2conc2C2CCCO2)=O)CC12CC2 C1(N(C(CC(CC)C2CC2)=O)C)CCCN(C(=O)CCOCC2CC2)CC1 N1(C(C23CCC(C(F)F)(CC2)C3)=O)CCC(CNC(C2CC2CC)=O)C12CC2 CC(C)C(=O)NCCC(C)N(C(=O)CCC1CCCC1)C C#CCCCCCCC(=O)NC1CC12CC(NC(c1cccc(O)n1)=O)C2 C(CC1=CCN(C(=O)COCC(=O)OC(C)(C)C)CC1)NC(c1c(F)ncc(C)c1)=O Cc1nnc(C(=O)NC2(CNC(C3(c4ccccc4)CCC3)=O)CCCC2)s1 C1(S(N)(=O)=O)(C(=O)NSCC(=O)NC(C)(C)CC)CC1.C#CCCCOC.NO N1(C(c2nnc(C)s2)=O)CCN(C(c2cc(C(F)(F)F)ncn2)=O)C(C)C1 c1(SC)ncc(N)c(C(=O)NCCN(C(=O)C(CO)NC(=O)C(F)(F)F)C)n1 C12(CNC(C3CCCCS3)=O)CC1CN(C(=O)Cc1ccc(C(F)(F)F)cc1)C2 N1(C(C2C(C)CCO2)=O)CC2(CC(S(C)(=O)=O)C2)C1 c1(OC)cc(Br)cc(C)c1C(=O)Nc1ncc(-c2cc(C)nc(C)c2)cc1O CCCCCCCC(=O)NCC(C(C)C)NC(=O)Cn1cnc([N+](=O)[O-])n1 N1(C(C2CCC(C(=O)OC)C2)=O)CC(CNC(C2(F)CCC2)=O)OC2(CCC2)C1 C1(NC(c2cncc(C(C)C)c2)=O)CCC12CCCN(C(=O)CNC=O)C2 c1(CC)cc(NC(=O)C(CC2CCC2)NC(c2cnc(C3CC3)o2)=O)ccc1F C1(CNC(C2CCCN(CC)C2)=O)CCN(C(=O)C#CC2CC2)CC1(F)F C(=O)(CS(C)(=O)=O)N1CC(CCNC(=O)C(O)CC2CCOCC2)(OC)C1 N1(C(C2(Cl)C(C)(C)C2)=O)CC(C2CN(C(c3cc(NC(N)=O)ccc3Cl)=O)C2)C1 c1(C(N2CCN(C(C(C)Oc3ccccc3)=O)CC2C)=O)cnn2c1N(C)CC2 Cc1cccn2cc(C(N3CCN(C(C4CCC(=O)C4)=O)CC(CO)C3)=O)cc12 C#Cc1ccc(C(N2CC(C(C)NC(c3cnn(C(F)F)c3)=O)C2)=O)o1 c1(OC)cc(F)cc(C(=O)NCC2(OC)CN(C(=O)C(O)c3ccsc3)C2)c1N CCC(C(=O)NC1CCC(NC(C2CC(C(F)F)(OC)C2)=O)CC1)C(C)(F)F c1(C(N2CCC(CCNC(c3ccco3)=O)C2)=O)cc(O)nc(Br)c1 N1(CC)CC(C(=O)NCC(COC)NC(c2cn(C)cn2)=O)CC1=O CC(CS(C)=O)C(=O)N(CCCNC(=O)CCCCN1CCOCC1)C(C)C Cc1cc(F)cnc1C(N1CC=CC(C(N2CCOCC2CC(C)C)=O)C1)=O CC(C)C(C#N)C(=O)NC1(CNC(c2ccn(C(C)C)n2)=O)CCCCC1 C1(C(N2CC(C(N3CC(n4c(C)ncc4)C3)=O)OCC2)=O)Cc2nccn2C1 C1(C(C)NC(c2cocn2)=O)CCCN1C(c1c[nH]c(-c2ccccc2)c1)=O CC1CN(C(=O)CC2CCN(C(=O)CCC3(C)N=N3)C2)CCC1CO N1(C(C(C)(C2(C)CC2)OC)=O)CCCC(C(=O)N(C)CC2C(C)(C)C2(C)C)CC1 C1(C(=O)NC2CCCC23CC3)(CC)CCCN1C(=O)CCn1ccnn1 C(Cc1ccoc1)(C(=O)NCC(F)C1CCC1)NC(C1C=CCC1)=O Cc1cnc(C(=O)NC2CCC(NC(C3CC4(C3)CC4F)=O)CC2)cc1Br C1(NC(CCN(C(C(C(CC)C)N(C)C)=O)C(C)C)=O)CCC(=O)NC1(C)C c1(C(N(CCC(C)NC(c2ncc(C)nc2)=O)C)=O)cc2ccc(C)cn2n1 C1(C(n2cc(C3(N(C)C)CCC3)nn2)C)CCN(C(c2ccc(F)cc2)=O)CC1 C1(C(=O)NC(C(=O)NC)C2CC2)C2CCC(C2)C1NC(=O)CS(=O)(=O)N(C)C C1(CC(=O)NCCCCNC(c2ncn(CC)c2)=O)CC(OC)C1(C)C C1(NC(CSC(c2ccccc2)C(=O)OC)=O)CCN(C(=O)OC(C)(C)C)CC1 CC(=O)CCCCCc1cccc(OC2CC3(C(C(=O)OC(C)(C)C)C3)C2)c1 c1(C(=O)NCC2N(C(c3c(C)sc(Cl)n3)=O)CC2)cnc2ncnc(O)c2c1 c1(NCC(C(C)C)(C)NC(C23CCOC(C)(C2)C3)=O)ncnc2cc(Br)sc12 C(=O)(C1=C(F)CN(C(=O)Cn2[nH]cnc2=N)CC1)N(C(C)CC(N)=O)C CCC(C)CC(CO)NC(c1cn(CCNC(c2ccoc2C)=O)cn1)=O C1(CC(=O)NCC(CC)N(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C)CCCC1O C(=O)(C1=CCCOCC1)NCC(CC(C)C)NC(=O)Cc1ccc2occc2c1 Cn1cnc2nc(Cl)nc(N3CCC(Oc4ccccn4)C3)c12 N1(C(c2scc(C(C)C)n2)=O)CC2(CCCCN2C(=O)CCCCCl)C1 C1(CC(=O)NC2(C(C)(F)F)CCC2)CCN(C(C23CC2CNC3=O)=O)CC1 C12(NC(CCCC)=O)CCCCCC1N(C(c1cnn(C(F)F)c1)=O)CC2 C(=O)(C(N)CC(=O)O)NCCCSCCC(N)=O C(CC(C)(C)CC(=O)N(CCC(C)NC(c1ccc(C)c(C(C)=O)c1)=O)C)OC C(C(CC(C)C)C(=O)N1CC2CCCC2(CNC(=O)C=Cc2cc[nH]n2)C1)OC c1(C(=O)NC2(CCNC(CN(C(C)=O)C)=O)CCCC2)cc(C)cc(F)c1N N1(C(c2c(CC)noc2C)=O)CCC2C(C1)CN2C(=O)C(C(C)(C)C)N(C)C c1(C(=O)NC2(CNC(c3c(N)nccc3)=O)CC2)cc2cccnn2n1 N1(C(C(N2CCNC2=O)C)=O)CCCC(C2CN(C(C3(C)CC(C#N)C3)=O)C2)C1 N1(C(c2c(-c3nc(C)sc3)c[nH]c2)=O)CCCN(C(C2CCCO2)=O)C(CO)C1 C(=O)(CC(C)(C)F)NC1(OCC)CCN(C(=O)C(F)C(=O)OCC(C)(C)C)C1 O=C(CCC(CF)CF)NCC1CCCN1C(=O)CCc1ccc(CO)cc1 c1(CC)ncccc1C(=O)NCC1(C)CCCN1C(=O)CCC1CCCOC1 C1(C(N2CCCC(C)C2CN=c2nc[nH]s2)=O)CCCC2CCCN12 CC1=CCC(C(=O)NCc2ocnc2C(=O)NCCN2CCCOC2=O)CC1 CC1CC(N)CCN1Cc1ccc(=O)n(C)c1 C1(NC(CN2CCC(C)(O)C2)=O)CC2CCC1N(C(=O)C1=CCCOC1)C2 c1(NC(C2CCN(C(c3c(C)ccs3)=O)CC2)C)ncnc2sc([N+](=O)[O-])cc12 C1(CNC(C(C(C)C)O)=O)CC(C)(C)CN1C(=O)Cc1coc(C(F)F)n1 c1(C(=O)NCC(C)N(C(c2cscc2C)=O)CC)cncc2nc[nH]c12 N1(C(CC(C(=C)C)OCC)=O)CCC2(CCC2)C(CNC(C2CCCO2)=O)C1 c1(C(=O)NCc2ccc(C(=O)NCC(=O)NC3CCC3)s2)cnn2c1CCC2 CCCCC(C)C(=O)NC1CCC(CCNC(=O)CSc2ccccc2)C1 Cc1cc(OCC(=O)N(C2CN(C(=O)C(C)OCC3CC3)C2)C)c(C)c(C)c1 C(C)(CNC(c1cnc(S)[nH]1)=O)(C(C)C)NC(CC1CC(=C)C1)=O Cc1nc(C(=O)NCCN(C(=O)C2=CC(O)CCC2)C(C)C)c2ccccn12 CCC(C(=O)N(CC(O)CNC(=O)CCC1CCCCCC1)C)C(F)(F)F c1(C(=O)NCC(CC)NC(=O)C(CSC)c2ccccc2)cn(C)c(=O)nc1O CC(c1ccco1)=CC(=O)NCCNC(c1cnn(CCO)c1C)=O C1(C(N2CCCC(Cn3cc(CC(O)CO)nn3)C2)=O)CCC(O)C1O N1(C(c2[nH]cc(C)c(=O)c2C)=O)CCC2CN(C(=O)OCc3ccccc3)C2C1 C(C(=O)NCC1CN(C(=O)COCC2CC2)CC1O)(c1ccccc1)=C(C)C C12(CNC(=O)CN3CCNC(=O)C3)CC(CN1C(=O)COc1ccccc1)C2 N1(C(CCC#C)=O)CCN(C(=O)Cc2ccn(C)n2)CC1C1CCC1OC C12(C(=O)OC(C)(C)C)CN(N(CC(C)C)CC)CC1(C)C2.C(CSC)OC=O C1(C)(NC(c2c(CNC(C(C(C)(C)O)F)=O)n[nH]c2)=O)CCC(=O)NC1=O C(=O)(C1=CCCC1)N(CC(=O)NCCC=C=C)CCOC N1(C(CC(CCC)NC(C2(C(C)(C)O)CC2)=O)=O)CC2(CCC2)OCC1C c1(CC(=O)NCC(CNC(C(CO)N(C)C)=O)CO)ccc(Cl)cc1F C#CCC(C)(C)C(=O)N1CC(O)(C(C)NC(=O)CCn2ccc(=N)[nH]2)C1 C1(NC(c2ccc(C3CC3)o2)=O)CC2(C1)CC(NC(C1CCC(F)C1)=O)C2 C1(NC(C(CC)CC)=O)CC12CCC(NC(c1cnc(C(C)OCC)s1)=O)CC2 CC(CC(C)(F)F)C(=O)NCCCCN(C(=O)CN(C)Cc1ccccc1)C c1(SCC(=O)NC2CC(NC(C3C(C)(C(F)F)C3)=O)C2)ccncc1 C1(C)(CCC(=O)NC(C2CCOCC2)C)CCCN1C(=O)CN1CCCCC1=O C=CCC(CC=C)C(=O)NC1(CC=CC(N2CCN(C)C(C)C2C)=O)CCC1 c1(C(N2C(C3(NC(c4n(CC)ncn4)=O)CC3)CCC2)=O)ccnnc1C N1(C(C=CC)=O)CC2CCN(C(c3cscc3C(F)F)=O)CC12 N1(C(C(CC)(F)F)=O)CC2CC(C1)CN(C(=O)CC13CCC(C)(C1)OC3)C2 C=CCCCCCCCC(=O)NCC1CC1NC(c1cc2sc(Cl)cc2[nH]1)=O N1(C(CCC2(NC(c3cc(C)nc(O)n3)=O)CCCC2)=O)CCC(F)(F)C(F)C1 c1(CC)cnn2ccc(C(=O)NC3CCOCC3NC(C3CC(C)(F)C3)=O)nc12 C(=O)(C1CCCc2nccn21)NC(CCC)CNC(c1cncc(C(C)=O)c1)=O C1(C(C(N2CC(O)(C(=O)OC)C2)=O)(C)C)CCCN(C(c2cc(C)co2)=O)C1 c1(SCC(=O)N(C(C)CCNC(=O)CNC(N)=O)C)ccc(Br)cc1 C(=O)(C1=NOC(CNC(c2cc[nH]c2C)=O)C1)NC(CC)(C)COC C1(C(=O)NCCC2CCC(NC(CCc3n(C)cnc3)=O)C2)CCC2CC2CC1 C1(OC)(CNC(C2CCC2C)=O)CCN(C(c2cccnc2N(C)C)=O)CC1 CC1CN(C(C2CCC2)=O)CC2(CCN(C(c3nnc(Cl)cc3N)=O)C2)O1 N1(C(CCOCC#C)=O)CC(C)N(C(=O)CC(C)(C)C)CC1C C1(CNC(C2(C)CCCC2)=O)CCCCN(C(c2cnc(C(F)F)nc2)=O)C1 n1(CC)nc(C(=O)NC(CNC(=O)CC2(CSC)CC2)CO)c(C)n1 c1(NCc2ncc(C)o2)ccc(S(=O)(=O)NC2CC2C(C)C)cc1C#N C1(C2N(C(C(C)N(C)C)=O)CCC2)CCN(C(c2ncn(C)n2)=O)CC1 c1(C(=O)NCCCCCN(C(CCCCC=C)=O)C)cnc2[nH]nnc2c1 N1(C(C(Cc2cn[nH]c2)NC(C(C=C=C)C)=O)=O)CCOCC(C)C1 c1(CS(=O)(=O)NC(C2C(C#N)CCNC2)=O)nc2ncc(Br)cn2n1 C1(C(=O)NC2(CC=C)CCC2)CCCCC1(C)NC(c1cccn1CCC)=O C(N=c1[nH]c(NC2CC3CC3C2)nc2c1CCCCC2)c1n(CC)ncn1 C1(C(N2C(CC=C)(C(=O)NC3CC(O)C3)CCC2)=O)CCCC(=O)N1C c1(CC)cc(C(=O)NC2(C3CCCCN3C(=O)CC(C)SC)CC2)cc(O)n1 CCC(C)(CC(=O)N1CCN(CC(C)NC(=O)C=C(C)C)CC1)C(=O)OC N1(C(CNC(CCC)=O)=O)CCN(C(C2Cc3nccn3C2)=O)C2CCCC12 CC(C)(C)C(C(=O)NCC1CCN(C(=O)CC2COC(=O)N2)C1)NC(N)=O C1(N(C(C(C)OCCCC)=O)C)CCC2CN(C(=O)C=C(C)c3ccco3)CC12 CC#CCCCC(=O)N1CC(OC2CCN(C(=O)C3=NOC(C)C3)CC2)C1 C(=O)(C(CO)C(C)C)NC(CNC(c1cc(C)c(C)s1)=O)(C)C Cc1ccc2c(c1)SC(C(N1CCCC(O)(CNC(C3(CO)CCC3)=O)C1)=O)C2 C1(Cl)(C(N2CC(C=C)(CC(N3CCC(O)CC3)=O)C2)=O)C2CCC(=O)C12 c1(C(=O)NCC2CCN(Cc3c(SC)cccc3)C2)cccn2cc(C)nc12 C1(NC(COCC=C)=O)CCCCCC1NC(c1c(C)nsc1NC)=O CC1(C(=O)NCCCCNC(c2csc(C#N)c2)=O)Oc2ccccc2NC1=O C(=O)(CC(C)(C)CC=C)NC1C(CNC(C(C=C=C)C)=O)COC1 C1(C(=O)NCC2(O)CN(C(c3cc(C)nc(C)c3)=O)C2)CCc2ccccc2O1 N1(C(C2C(C)C2)=O)CC2COCCC2(NC(=O)CS(C)(=O)=O)C1 c1(C(=O)NC2CCCC(NC(c3ncc(C)cc3F)=O)C2)[nH]nc2ncccc12 C1(NC(c2ccc(CCC)[nH]2)=O)CCN(C(=O)C(C)CF)CC1 N1(C(CNC(C)=O)=O)CC(N(C(=O)Cc2cccc(C(N)=O)c2)C)C(F)C1 CC(Cl)(Cl)C(=O)NCCC(O)CNC(=O)Cn1ncnn1 C(N=c1[nH]c(=NC(C)C2CC2)[nH]c2c1CCC2)c1c(C)nc2ccccc2n1 C1(NC(c2ccsn2)=O)CCC2CN(C(C3Cc4cccnc4C3)=O)CC2C1 c1(N2CCC3(C)C(C)(C2)C3(F)F)nccc(=NCCCCC#N)[nH]1 CCCCCCCCc1cn(CCCCC2CCCN2Cc2csnn2)nn1 c1(OC)ccc(C(=O)OCC2CCN2C(=O)Cc2nnc(C)s2)c(N)c1 c1(-n2c(-c3cn(CC=C)nc3)nc(C3CCOC3)n2)ccc2ncsc2c1 CC(C)CCC(C(=O)N1CC2(C=CCO2)C1)NC(=O)CSC(C)(C)C S(=O)(=O)(c1cc(Cl)cc2cccnc12)NCC(c1ccco1)O C=CC(C)C(C)C(=O)N1CCC(CN(C)C(c2ccc(C#N)o2)=O)CC1 C1(NS(C)(=O)=O)CCCC1CNC(=O)Nc1csc(C(N)=O)c1 Cc1cc(N)cnc1C(N1CC(NC(c2ccnc(C3CC3)n2)=O)C2(CC2)C1)=O C(=O)(C1=NOC(C)C1)NCC(C)N(C(CC(=C=C)C)=O)C C1(C(C)NC(C2(C)COC2)=O)CN(C(C2CC2(c2ccccc2)F)=O)CCO1 CC(C)S(=O)(=O)CC(=O)NC1CCCC1NC(c1snnc1C1CC1)=O c1(CC)cnc(C)c(NC(=O)C(c2cccs2)NC(C2CNC(=O)N2)=O)c1 S(=O)(=O)(c1ccc(Cl)nc1C)N1CC(F)CC(C(=O)NC(C(=O)OC(C)C)C)C1 C1(NC(CCc2scc(C)n2)=O)CCC2(CCN(C(=O)C(O)CN(C)C)C2)C1 c1(C(N2CC(CCNC(=O)CCCN(C)C(C)=O)(OC)C2)=O)ccc(C)cc1 CCCCCCCc1ccc(CC(=O)NCC(C)(C)NC(=O)C(C)C(C)O)cc1 C1(C)(C(=O)NCCCCNC(CC2C(C)(C)C2)=O)CC=CCC1 c1(C(=O)NC2(CC3CC3)CC2)ccc(C(F)C(N2CC(COC)(CO)C2)=O)cc1 C(=O)(C(F)(F)CC(C)C)NCC1(O)CN(C(CCCCNC(=O)OCC=C)=O)C1 c1(OC)ncnc(C(N2CC(NC(c3cn(C(C)C)nn3)=O)C(C)(C)C2)=O)c1F N1(C(CC2CCCCC(=O)N2)=O)CCN(C(=O)C=C(Cl)Cl)C2CCCC12 c1(C(C)C)cccc(C(=O)NC2CC(N(C)C(c3c[nH]c(=N)s3)=O)C2)c1F C1(C)(C(N2C3CN(C(C4=NOC(C)C4)=O)CC2CC3)=O)COc2ccccc2O1 N1(C(C)=O)CC2CC1CN2C(=O)CCOCCNC(=O)Nc1nnc(O)nc1O N1(C(C(C)OCC)=O)CCCCC1CCC(=O)NCc1nncn1C c1(SCC(=O)NCC2CCCN(C(CCS(C)=O)=O)CC2)nc2ccccc2s1 C=CCCC(C)(C)C(=O)NCC1CCC1C(N1CC(C)(C)C1C(=O)OC)=O C1(C(N2CCC(N(C)C(c3ncc(F)cn3)=O)C2)=O)CN2CCCN1CC2 C1(NC(C2(NC(CCCC#C)=O)CC2(C)C)=O)CC(C)N(C)CC1C c1(C(N(C2CCCN(C(c3ncccc3O)=O)C2)C)=O)ccc(C(C)(F)F)cc1 N1(C(=O)NCc2ccc(COC)cc2)Cc2cccn2C(C)C1 c1(CNC(C(c2ccccc2)C)=O)cn(C2CN(C(C3(CO)CC3)=O)C2)nn1 CC1CCCN(C(=O)Cc2csc(Cl)n2)C1CNC(c1cnccn1)=O c1(NCC2CCC(CC)O2)[nH]c(=NCc2ccc(N)cc2C)nc2scnc12 C1(CNC(CC=CC=C)=O)CC2(CC(NC(=O)C(O)C(C)C)C2)C1 c1(NC(C2C(NC(c3ccc(OC(C)(C)C)cc3)=O)C2)=O)ncc(I)nc1Cl c1(C(=O)NCC(CNC(=O)CCn2ccc(C)n2)OC)ccc(Cl)[nH]1 C1(N(CC(=O)NCC(CN(C(C2C(CCC)C2)=O)C)O)C)CCCCC1 O=C1CCc2cc(S(=O)(=O)N3CCCC(C4CCCO4)C3)cc(F)c2N1 C1(N(C(Cc2c(C)n(C)cn2)=O)C)CCN(C(c2cnc(O)n2C)=O)CC1C Cc1cnc2c(C(N3CCCC34CN(C(=O)C(O)C(C)(C)C)C4)=O)cnn2c1 CCS(=O)CC(=O)N(C)CCC1CCN(C(C2CC(F)C(=O)N2)=O)CC1 c1(-c2ccc(CC)c(F)c2)ccn2cc(C(=O)NCc3cnn(CC)c3)nc2c1 c1(C(=O)NCCC(C(C)C)NC(c2cn(CC)nn2)=O)cccc2c1C(=O)NC2 C(=O)(CCCCNC(=O)C(C)SC(C)C)N(CCOCCO)CC c12ncccc1S(=O)(=O)NCCCN2.c1(C(N(CCC)C)=O)ccc(Cl)cc1 N1(C(CC)C)C(=O)NC(c2cc(Br)cc(OC)c2O)C2=C1CC(C(=O)O)NC2=O N1(C(C(COC)OC)=O)C(CNC(=O)C(=Cc2cn[nH]c2)C)CC2COCC12 c1(OCC(=O)NCC2C3CCC(C3)N2C(=O)CC2CCC2)ccc(F)cc1F C(CCNC(=O)Cc1cncs1)(C(=O)NC(c1nn[nH]n1)C1CC1)OC C1(CCC)CCC(C(=O)NCC2CCN(C(=O)CCc3nccs3)C2)CC1 N1(C(c2c(C)nn[nH]2)=O)C(C(N2CCN(CCN(C)C)CC2)=O)CC2CC12 C(=O)(CCCN=[N+]=[N-])N1CC(C)C(CC(N2CCC3(CSC3)C2)=O)C1 C1(O)(CCNC(CN(C(C)=O)C)=O)CCCN(C(=O)CCc2cnn(C)c2)C1 c1(C(=O)NCCN(C(C2CN3CCC2(C)C3)=O)CC)occ2c1CCC2 C(=O)(CC(C)(C)NC(C1CCCC1(C)NC(C12CC(C(=O)OC)(C1)C2)=O)=O)OC CC1(C)CCN(C(c2cnsn2)=O)C1C(N1CC(n2cccn2)C1)=O c1(NC(CC2(OC)CN(C(c3c(C4CC4)noc3C)=O)C2)=O)c(C)cnnc1O Cc1csc(=O)n1-c1ccc(NC(=O)C(=O)NC2CCCOC2C(C)(C)C)cc1 C1(CC(=O)N(CCN(C(c2cc(C)ncc2)=O)C)C)CCn2cncc2C1 N1(CCN(C(CC2CC(=C)C2)=O)C)CCN(C(=O)C(F)CCC)CC1 CCC(CNC(c1cn(C2CC2)cn1)=O)(CC)NC(c1nnn(C)n1)=O C(CCC(C)C(=O)N1CCN(C(c2ccc(C(C)=O)cc2)=O)CC1CCO)OC c1(C(=O)C=O)ccc(C#N)cc1.c1(NC(C(c2ccn(C)n2)N)=O)ccc(F)cc1CO CN1CCC(NC(c2cnn(C)c2-n2cnnc2)=O)c2ccccc21 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(NC(c2cc(Cl)ccc2C)=O)C(O)C1 N1(C(C(CC(C)C)ONC(c2cc(C)c(O)nc2)=O)=O)CCc2ccccc2C1 CCC(Cc1ccccc1)CC(=O)N(CCCN(C)C(c1cccnc1F)=O)C N1(C(C(C(C)C)OCC)=O)CCOC(C(=O)NCc2cccc(F)c2)CC1 C1(NC(CC=CC=C)=O)CC2CCC(C1)N2C(=O)C(C(C)C)NS(C)(=O)=O CC1CCc2c(C(=O)NCC(O)CNC(C34CC(C3)C4)=O)c[nH]c2C1 C1(C(C)C)N(C(=O)CC2CCC2)CC12CCN(C(C1C3CCC(F)(F)C13)=O)CC2 c1(CC(N2CC(CC(C)NC(c3cncs3)=O)C2)=O)ccc(O)cn1 N1(C(c2cccnc2Cl)=O)CCc2cccc(-c3cccc(C4CCC4)c3)c2C1 c1(C(N2CCCC(N(CCC)C(C3CC3CC)=O)C2)=O)c(C)nn(C)c1C c1(C(=O)NC2CC(CCNC(c3nc(C)sc3C)=O)C2)nc(C)n(C)c1C c1(CC)cccc(C(N2CCC(NC(c3ccc(C)c(O)c3)=O)CC2C)=O)c1F C1(OC)CCC2(C(=O)NC(C3CCOC3)CNC(c3cc(C4CC4)no3)=O)CC12 C1(CNC(CCN(CCC)C)=O)CN(C)CCN1C(c1cccc(F)n1)=O N1(C(C=C(CCC)C)=O)CCC(c2cn(-c3ccccn3)nn2)(N(C)C)C1 C#CC1(C(=O)NCC2(CO)CCCO2)CCN(C(=O)CCCOCCOC)C1 C(=O)(C1(C)CCCc2ccccc21)NCC1N(C(CC=CCC)=O)CCCC1 n1(CC(=O)Nc2cn(C3(C(=O)O)CC(OCC)C3)nn2)cnccc1=O c1(COC)cc(C(=O)NC2CCC(CCNC(=O)CCC3CCCCC3)C2)no1 O=C(C(F)(F)CO)NCC1CCCN(C(=O)CCOC2CCOCC2)C1 C(CC(=O)N(C)CCN(C(=O)C(C)n1cccn1)C)SC CCC(CCOC)C(=O)N(C1CCCN(C(=O)C(CC(C)C)NC(N)=O)C1)C C1(CCC#C)CCN(C(C2(CNC(=O)C(O)CCSC)CCC2)=O)CC1 C1(NC(CSCC(N2CC(C)(F)NCC2)=O)=O)CCCC2CCCCC12 C(C(C)(CC(=O)OC)C(F)(F)F)NCc1ccc(NC23CC(CC)(C2)C3)cn1 c1(C(=O)NCC2C(CNC(c3c(C)occ3)=O)C2)cc(=O)n(C)cc1Br c1(N(C(c2cc(C)n(C)n2)C(=O)NCCCCCC)C)nc2c(s1)CCCCC2 N1(C(=O)Cn2cnnn2)CCN(C(=O)CN2CC3CC3C2)C2CC12 c1(NCC2CN(C(CNC(CC(C)(C)C)=O)=O)C2)ncc(S(C)(=O)=O)cc1Cl Cc1n[nH]cc1C(=O)N(CCCNC(c1ccc(COc2cnn(C)c2)o1)=O)C c1(OC)nc(C(N2CC(CNC(=O)Cc3ccns3)CC2C)=O)cc(O)n1 c1(NC2(C)CC(NC(C(CC)OC)=O)C2)ncc(S(C)(=O)=O)cc1Cl C(C(C)(CC)CO)NC(C(CSCC)NC(c1cnsc1)=O)=O N1(C(CC2N(C(C34CCC(OC)C3C4)=O)CC2)=O)CC2CC3CC2C1C3 C1(C(N(C)Cc2nnc(CC)o2)=O)CCC(O)CN1C(=O)CC1(O)CCOCC1 CC1=NOC(C(=O)N(C2CCCC2)CCCN(CC(=O)N(C2CCSC2)CC)C)C1 C1(CNC(C(CCC)C#N)=O)CN(C(=O)C(F)=C(C)C)C2(CCC2)C1 c1(CC)ccc(CCC(N2C(CNC(C3(C)CCC(=O)N3)=O)CC3CC23)=O)cc1 C1(NC(CSC)=O)CN(C(=O)COc2cnn(C)c2)C(C)(CO)C1 c1(C(N(CC(CNC(c2cc(C)oc2C)=O)C)C)=O)cc(F)c(N)cc1F N1(C(C(CCC)(C)C)=O)CCCC(C2CN(C(=O)C(O)CCC(F)(F)F)C2)C1 C1(C(N2C(C3CCN(C(=O)C=CI)C3)CCC2)=O)CCN(CCO)C(=O)C1 N1(C(C(CCSC)OC)=O)CCC2(CCN(C(c3cc(CC(C)C)on3)=O)C2)C1 C1(NC(C(Br)=C(C)C)=O)CCCCC12CCCN(C(C1CCC1(C)C)=O)C2 C12(CNC(c3c(OC(C)C)cccc3)=O)CCC(CC1)N(C(C1(Cl)CC1)=O)C2 c1(SC)nc(=NC2CC(C)N(C(C3CN4CCC3CC4)=O)C2)s[nH]1 C1(CC(C)(C)C)CN(C(=O)CC(C)(F)F)CCN1C(=O)C(F)CC1CCOC1 c1(CC(=O)NC2(C)CN(C(C3CN(S(CC)(=O)=O)C3)=O)C2)c(C)noc1Cl CCCCCC(C)CC(=O)NC1CN(C(=O)Cc2nc(=N)[nH][nH]2)CCC1CC1CC1 CCCCCC(=O)NC1CC(F)(CNC(=O)CC2CC(C(F)F)C2)C1 C1(NC(c2cn[nH]c2)=O)CCC2CN(C(c3cccn4nncc34)=O)CC2C1 C1(C(N2CC(C)(C)C(NC(C3CC(F)(CO)C3)=O)C2)=O)CCc2ncncc2C1 c1(-c2n(C3C(C)CCCC3C)nc(CC(F)(F)F)n2)ccc(F)c2cccnc12 C12(C(N3CCC(CCNC(C(C)CC4CCCC4)=O)CC3)=O)CCC(CC1)CO2 C(CC(=O)NC1(CN(C)C)CC1)(CC(C)C)NC(CCC=C)=O n1(CC2CN(C(C(C)C3CCCO3)=O)C2)cc(CN(S(C)(=O)=O)C)nn1 C1(C(=O)OCC)(CN2CCCC(c3nc(C)c(C)s3)C2)CCOCC1 c1(C(=O)NCCCCNC(C2(CC(C)C)CCC2)=O)cn(C)nc1C(C)C N1(C(C(C(C)C)SCC)=O)CCCC12CCN(C(c1nccc(C)c1O)=O)C2 CON(CCC(=O)NCC(=O)NC1CCOCC1)C(=O)C(C)Cn1cccn1 c1(CCN(C)C)ccc(-c2nc(-c3cccnc3)nn2-c2ccc(F)cc2)cc1 C=CCCC(C(=O)OC)NC(C1CC(C)(C)CN1C(=O)C(CC)N(C)C)=O CC1CCN(C(C2CSCN2C(N)=O)=O)CCN1C(=O)Nc1ccncc1F Cc1c(F)ccc(N)c1NC(=O)OC(C)(C)C.C12CN(C)CCN1C(=O)C=CCS2 CCCC(C(=O)NCCN(C(C1CCC1(F)F)=O)CC)c1ccccc1 CC(C(=O)NC1CCCC(CC(=O)NCCc2ccncc2)C1)S(N)(=O)=O C(=O)(C1=CCC(NC(c2cc(F)ccc2F)=O)C1)N(C)CC1CCC(F)(F)C1 c1(SC)cc(C)ccc1C(=O)NC(CNC(C1(C)CC=CCO1)=O)C(C)C N1(C(C(=O)NCCOCC)C(CC)CC)CCN(C)c2ccc(F)cc21 C(=O)(CCCCCC#N)N1CC(NC(CCc2cccc(OC)c2F)=O)C(C)C1 c1(CC)nc(=N)[nH]c(=NC(CNC(=O)Cc2cccnc2C)C2CC2)[nH]1 C(C)(C)(C(=O)NC(C)C(=O)NCC(O)Cn1cccn1)OC(C)C Cn1cc2c(n1)CCCC2C(=O)NCCOCCCNC(=O)CCC1CCCO1 N1(c2ncc(C)cn2)CCC(C(C)NC(=O)C=Cc2cnccn2)CC1 N1(C(C=CC(=O)N(C)C)=O)CCN(C(C2CCCCO2)=O)CC1c1cn[nH]c1 CON(CCC(=O)NC1CCNC(=O)CC1)C(=O)c1c[nH]cc1C C1(CC(=O)N(C(C)C)CCN(C)C)CCCCN1C(C1CNC(=O)O1)=O N1(C(C2(C#C)CCN(C(=O)CP(C)(C)=O)C2)=O)CCC(F)(F)CC1C C1(CNC(c2c(C)con2)=O)CCN(C(c2cccc(C#N)n2)=O)C12CC2 c1(C(N(CC(CC)NC(c2cc(C)sn2)=O)C)=O)ccc(=O)n2c1COCC2 N1(C(CNC(CN(C)C)=O)=O)CCC2(CCCC2NC(C2(C3CC3)CC2)=O)C1 N1(c2cc(NCCCc3cnc[nH]3)nc(C)n2)CCC(C2CC2(F)F)CC1 c1(C(=O)NCC2CCCNCC2)cccc(SC(F)(F)F)c1Cl C1(C(N(C2(c3cccc(F)c3)CC2)C)=O)CC2C=CCC(C1)C2 C=CC(CC)CC(=O)N1CCOC(CNC(=O)COc2ccc(OC)c(C)c2)C1 C12(NC(CC3CC(OC)C3)=O)CCC(CN(C(=O)C(C)=C3CC3)C1)C2 C1(CCC)CN(C(C2CN(C3CCOC3)C2)=O)CCN1C(=O)Cn1nnc(C)n1 c1(C(=O)NC2CCC(NC(C3(C)CCOC3)=O)C2)cccc(N)c1Br CC1CN(C(=O)C=Cc2cc[nH]n2)CCCN1C(C1CC2CCC2C1)=O C1(NC(C2CCn3ccnc3C2)=O)CCN(C(c2ccccc2)=O)C12CCCC2 Cc1nc(F)ccc1CN1CCC2(CC2C(=O)NC2CCC(=O)NC2=O)C1 N1(CC(=O)N(C)CC2CCN(C(C3(C4CC4)CC3)=O)C2)CC2CCC1C2 CCC1C(=O)NC(C)(CC)CNC(=O)CC(SC)CCC1CCC(=O)N C1(C(=O)NCCN(C(=O)CC(C)P(C)(C)=O)C(C)C)CCc2n[nH]cc2C1 c1(CC(=O)N(C2CCC(NC(=O)Cc3cnn(C)c3)C2)C)cc[nH]c(=N)c1 C=CC(CC)CC(=O)NCC1(CNC(c2scnc2C)=O)CCC1 C1(NC(Cn2cc(C(=O)OC)nn2)=O)COCCN(C(=O)C=CCn2cncn2)C1 N1(C(C(Cn2cncn2)NC(CCSCC)=O)=O)CCSCCC1C Cc1cc(C(N2CCCCC2CN(C)Cc2noc(C)n2)=O)c(C)c(C)c1 CC1CN2CCN1C(C(N1C3CCC(C3)C1CNC(=O)CC1CCCO1)=O)C2 C1(NC(CC(C=C)CC)=O)CN(C(=O)CSCCOC)C2(CCCCC2)C1 CCCCC(CCC)N=c1[nH]c(=NCCC(=O)NC)[nH]c2c1CC(C)CC2 C1(C(=O)NCc2cc(C)no2)CCN(C(C2CCC2(F)F)=O)C(C)C1 c1(COC)cc(CNC(CCCO)c2ccccc2)on1 c1(N(CCOC)CCNC(=O)C=CCCC(C)C)nc(OC)cc(OC)n1 N1(C(CNC(CNC(c2ccc(C(C)C)o2)=O)=O)=O)CCCC1(C)C1CC1 c1(OC)ccc(C(N2CC(NC(=O)Cn3ncnn3)C(C)(C)C2)=O)c(N)c1F N1(C(c2nccc(N)c2)=O)CCCC(NC(c2c[nH]cc2C(F)(F)F)=O)C(F)C1 C1(CCC)(NC(c2coc3c2COC3)=O)CCN(C(=O)Cc2nc(C)cs2)CC1 C(C1CCc2ccccc21)NC(c1n(CCC)nnn1)c1cc(CC)on1 C1(N(C(=O)CC(=O)OC(C)(C)C)C)C2CN(C(=O)C(F)CC3CC3)CC12 C(C(O)CN(C(=O)CSCc1ccco1)C)N(C(C=C(COC)C)=O)C N1(C(c2n(CC)ccc2)=O)CC2(CCCC2NC(c2cn[nH]c2)=O)C1 C(=O)(C(=O)NOC)NCC(CCNC(=O)CCCn1cccc1)OC C(=O)(C1=COCCC1)NCC1C(CC)CCN1C(=O)CC(F)(F)c1ccccc1 c1(NC)cncc(C(N2CC(CCNC(c3cc(SC)oc3C)=O)C(C)C2)=O)c1 CC(C)CCC(O)C(=O)NCC1(CNC(=O)C(C2(O)CCCC2)F)CCCCC1 CCCC(CC(C)C)C(=O)NCc1cccc(CNC(C2CNC(=O)N2)=O)c1 C1(NC(CC(C)OC)=O)COC2CN(C(c3ccc(SC)cc3Cl)=O)CC12 CC1(C)CC(=O)NCC1C(=O)NC1C2CC1CN(C(=O)CNc1ncccn1)C2 C1(O)(CNC(c2ccccn2)=O)CCCN(C(c2cccc(C(F)(F)F)c2)=O)C1 c1(CNC(c2c(Cl)n[nH]c2CC)c2n(CC(=C)C)nnn2)ccc(Cl)nc1C c1(NC)cc(C(N2CC(C)C2C(=O)NCCCOCCOC)=O)ccc1NC C1(CNC(C(CC=C)C)=O)CC2CCC(C1)N2C(C12CC(C)(C1)OC2C)=O C1(NC(C2(C)CC(NC(C3CC(OC)C3)=O)C2)=O)CC2CC1OC(=O)N2 c1(NC(C(=O)NCCc2cc(OC)c(C)c(OC)c2)=O)cc2ccc(Cl)nc2s1 C=CC(C)(O)C(=O)NCCC(C(C)C)NC(c1ccn(C(C)(C)C)n1)=O C(CC(=O)NC1CCCN(C(c2cnc3c[nH]nc3c2)=O)C1C)(C(F)(F)F)OC C(=O)(CCC1CC1)NCCN(CC(C)O)C(C1CCN1C1CCCC1)=O N1(C(c2nccc(C)n2)=O)CCC2(CC1)CC2CNC(C1CCC(C(N)=O)C1)=O C1(CCN(C(=O)CC(C)(C)O)C)CCCCN1C(=O)CC1CCCOCC1 C1(C(=O)NCC2CCCC(C)O2)CN(C(c2cc[nH]c(=N)n2)=O)CC1(F)F C1(N(C)C(C2CCS2(=O)=O)=O)CCC(CNC(=O)C(O)CC2CC2)CC1 c1(OC)ccc(CC(=O)NC2CCN(C(c3cc(SC)on3)=O)C2(C)C)cc1F C1(CNC(c2nc(C)nn2C)=O)CC2OCCC2N1C(c1ccc(C)c(F)c1)=O C1(C(N2CC(C(=O)NC)C2)=O)C(O)CCN1C(=O)Cc1csnc1C Cc1nnc(O)c(C(=O)NCC(C)(CO)NC(=O)CC2CC2(C)C)c1C c1(C(=O)NC2CN(C(c3ncn(C(C)C)n3)=O)CC2C)cccc(F)c1C#N CN1CC2CCCC(C1)N2C(=O)CCN(C(=O)C1Cc2ccccc21)C1CC1 Cc1nc2ncnn2c(N2C3CCC2CN(C(c2cn(C4CC4)cn2)=O)C3)c1C c1(C(=O)NCC(CC=C)NC(c2cc(CC)[nH]n2)=O)cccc2nc(CC)[nH]c12 Cc1ccc(C(C)C)cc1C(=O)NC(C)CCN(C(=O)C(=O)C(C)C)C c1(C(=O)NCC2C(NC(C3C(CC)OCC3)=O)CCC2)ccc(C)c(C(C)=O)c1 N1(C(C(ONC(C2=CCCC2C)=O)CC(C)C)=O)CCC(C)OC(C)C1 C#Cc1cc(Br)cc(Cl)c1NC(C1CC(c2ccccc2Cl)C1)=O C=CCC(CNC(=O)Cc1coc(C)n1)NC(=O)Cc1cc(OC)no1 N1(C(c2nc(CC)oc2C)=O)CC(NC(=O)Cc2c(C)cccc2C)CC(O)C1 Cn1cnc(CC(=O)NC(Cc2ccco2)C(=O)NCC2CCC(C(N)=O)O2)c1 CCCC(C(O)C(=O)NC(C)CN(C)C(C)C)NC(c1nccn1CC)=O c1(NC(=O)CC2CCN(C(c3cc(Br)ccn3)=O)C2)nccn2c(Br)cnc12 CC1CN(C(c2cn(CCO)nn2)=O)CCC1NC(C12CCOC(C)(C1)C2)=O Cc1cccc2nc(C(=O)NC3COCCC3NC(=O)CC34CCCC3C4)cn12 c1(CC(=O)NC2CCC(N(C)C(C3CCCC3)=O)C2)ccc2c(c1)CCCS2 S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NCC(C(C)C)F CCC(C)CC(C(=O)N1CCC2CCCC12)NC(=O)COC(C)=O CC1(C)C(C(=O)NCC2(C)CC2(F)F)CCN1C(c1ccc(=N)[nH]n1)=O Cc1csc(CCNC(c2sccc2CNC(c2cnco2)=O)=O)n1 N1(C(C(C)(F)F)=O)CCN(C(C2CCC(F)(F)CC2)=O)C(c2ccccc2Cl)C1 c1(CC)ccc(C2CCCN2Cc2ccc(C3C(C(=O)OC)C3)cc2)cc1 CS(=O)c1cccc(C(=O)NCC2CCCCN2C(=O)C2=CCCC2)c1 c1(C(=O)NCCN(C(C(CC=C)F)=O)CC(C)O)cccc2c1nc(O)n2C CCCC(C)CCCC(C)N(C)Cc1nccn1CCc1ccccc1 C1(CC=C)(NC(=O)CNc2nccs2)CCCN(C(C2CCN(C)C2)=O)C1 c1(N2C(CCC(=O)NC(COCCOC)C(=O)O)CCC2)ncc(F)cn1 Cc1oc(C(C)(C)C)cc1C(=O)NC1CCC(NC(=O)C(C)(C)n2ccnn2)C1 C(N=c1cc(C)nc(Cl)[nH]1)C1CCC(NC(c2c(CC)nc[nH]2)=O)C1 N1(C(C2C(C=C(C)C)C2(C)C)=O)CC2(CC2)CC1CNC(=O)C(C)O CCC(CC)(CC)C(=O)N1CC2CCC(CNC(=O)CCC3(C)CC3(F)F)C2C1 CCC(C)CC(=O)N1CCN(C(CNC(c2cc(C)c(C)s2)=O)C(F)F)CC1 c1(C(=O)NC2CCC(CNC(C(CCSC)N(C)C)=O)C2)ccn2ccnc2c1 N1(C(c2ncccn2)=O)CCCCC2(CCN(C(=O)C(O)C3CCCC3)C2)C1 Cc1ccc(Br)cc1CC(=O)NC1CC2C(NC(=O)CC3CCCO3)C2C1 Cc1c[nH]c(CNC(C2CCC2C(F)F)=O)c(C)c1=O C1(C)CCC(=O)N1.N1(CCOC)CCC(NC(C23CCC(CC2)C3)=O)CC1 CC1CC(CCC(=O)NCC2CCC2C(N2CCC2)=O)C1.C12(CC1)CS2 C(=O)(CCC(C)(C)C#N)N1CCCC(C(C)NC(c2c(O)cccc2F)=O)C1 c1(CC(=O)NC(C(C)NC(=O)C=CC(=O)N(C)C)CO)cc(F)ccc1Br N1(C(CC=C=C)=O)CC(NC(c2ccc(O)cc2)=O)C2(CCOCC2)C1 C1(C(=O)Nc2c(N3CC(C)(C)OCC3)cccc2)CCC2CCCCC2C1 Cc1ccc(CCC(=O)NC2(CCCNC(C3C4(CC4)C34CC4)=O)CC2)cc1 C1(C(=O)NC(COCC)C)(NC(c2nc(O)sc2C)=O)CCN(C)C1 Cc1ncc(Cl)c(C(=O)NC2(C)CCN(CCOCCC(C)C)C2)n1 C1(NC(c2cc(COC)cn2C)=O)CCN(C(=O)CC2COCC2O)C(C)C1 C(=O)(CS(=O)CCC(F)(F)F)NCCN(C(C(C(C)(C)C)(C)O)=O)C1CC1 C1(C(N2CCCC(NC(c3cccs3)=O)C2)C(=O)NC)CC2C=CC1C2 C(=O)(C(F)C(F)(F)F)N(CCCNC(c1cc(CCCCC)[nH]n1)=O)C(C)C C(=O)(CC(C)C(C)(C)C)NCC(C1CC1)NC(C(C)(C)SC)=O O=S(=O)(c1ccc(F)cc1F)N1CC2CCC(C1)N2Cc1ccc(Cl)c(Br)c1 N1(C(C(CCCC)C)=O)CCC(C)(C)C(NC(=O)CC2CCCCCC2)C1 N1(C(c2ccn(C(C)C)c(=O)c2)=O)CC2CN(C(c3csc(Cl)c3)=O)CC2(C)C1 C(=O)(C(C(C)C)OCC(C)C)NCCCCCNC(C1(CCOC)CCCC1)=O C1(NC(C(C2CCCCC2)OC)=O)CCN(C(c2csc([N+](=O)[O-])c2)=O)CC1F N1(C(C(C)n2cncn2)=O)CC2(CNC(C3(C(C)(F)F)CC3)=O)CC1CO2 C(=O)(CCC(C)(C)C)OCCNC(C1CN(c2cccc(OC)c2)C(=O)C1)=O C(=O)(C1CC(N)c2ccccc21)N(C1CC(C)(NC(=O)OC(C)(C)C)C1)C CCC(CO)(C(=O)NC(CO)C(C)NC(c1cc(=O)cc[nH]1)=O)OC c1(C(=O)NC2C(NC(C(C3CCOCC3)OCC)=O)CC2)cc(N)cc(F)c1 c1(NC(C2C(NC(c3cc(CC)[nH]n3)=O)CCCC2)=O)ccccc1N(C)C c1(C(=O)NCCC2CC(NC(c3c(CC)c[nH]c3)=O)C2)cncc(O)c1 C(=O)(C(C)CC(=O)N1CCOCC1CN(C(=O)C=Cc1ccccc1)C)OC C#CC1C(C(=O)N(c2ccc(NS(C)(=O)=O)cc2)CCC)C1(C)C C1(CCCC)CN(C(=O)CCC(C)(C)C)CCN1C(=O)C(CCSC)NC(N)=O CC(C)(CCNC(c1ccc(C2CCCCC2)o1)=O)NC(c1cnc(Cl)s1)=O C1(C(=O)NC(C2CCN(C(C3(C)CCC3)=O)CC2)C)CC2(CCCC2)CO1 c1(CNC(CC(c2ccc(OCC)cc2)NC)=O)nnc2n1CCNC2 CCC(C)C(O)C(=O)NCC1(O)CC(NC(=O)CC23CCCC2C3)C1 CCCCCCCCC(=O)N1CCC(N(C(=O)C=CCN2CCCC2)C)C(C)C1 Cc1nn(C(C)C)c(NC2CC(C)N(C(=O)Cn3nnnc3C)C2)c1[N+](=O)[O-] c1(C(=O)NCC2CCN(C(c3ccc(CC)[nH]3)=O)C2)cc(C)n(C(C)C)n1 n1(CC)nc2c(c1C(=O)NC(C)C(C)NC(=O)CCC1CCCC1)CCCC2 Cc1cc(=O)ccn1CC(N1CCC(NC(c2snnc2C(C)C)=O)CC1C)=O CC1(C)CN(C(=O)Cn2ccc([N+](=O)[O-])n2)CC1NC(c1nsnc1O)=O C1(C)(NC(Cn2cc(CN(C(C3C(C)NC(=O)N3)=O)O)nn2)=O)CCC(C)CC1 c1(CC)cc(NC2CCCN(C(=O)CC3CCC4(CCC4)O3)C2)nc(C)n1 c1(C(=O)NCC2COCCN(C(c3c(C)occ3)=O)C2)cc2ccccc2[nH]1 N1(C(C(C)CCN(C)C)=O)CCC(NC(c2nccnc2Cl)=O)C(C)(C)C1 C1(C(=O)NCCC(C(C)C)NC(c2ccc(C#N)cc2)=O)CCc2nncn2C1 N1(C(C(N2CC(C)C2)C)=O)CCCCC1CNC(c1cccnc1C(F)F)=O CC(CC(F)(F)F)C(=O)NC1CC2CC(NC(C3CC(=O)CC(=O)C3)=O)C1C2 Cc1ccc(C(=O)NCC2CN(C(=O)CCCc3ccccc3C)C3CC23)cn1 c1(CN(C(Cn2cc(CCCC=C)nn2)=O)C)cccc(C)c1 C1(C(=O)NC2C(NC(c3ccc(CCC)s3)=O)CC2)Cc2ccccc2C1 C1(CNC(Cc2nnc(C)o2)=O)CC2CCC(C1)N2C(=O)Cc1ccnc(F)c1 c1(C(=O)NC(CN(C(C(=O)NCC#C)C)C)C)cc(-c2ccc(C)s2)[nH]n1 C(=O)(C(O)CC(C)(C)C)N1CCC(OC2CN(C(C(C(=C)C)(C)O)=O)C2)CC1 C1(COCC)CN(C(=O)Nc2cc(C)nn2-c2ccc(C)cc2)CCO1 CCCCC(CC(=O)N1CCCC1(C)C1CC1)NC(c1nocc1C)=O C=CC1CC(NC(C2(CC=C)CCN(C(=O)CCC(C)CC)C2)=O)CCO1 C1(C(NOCCCSC)=O)CN(C(=O)CC=CCCCCC)CC1C c1(C(=O)NC2(C(N)=O)C(C)CCC2)ccc2c(c1)CCC2(C)C c1(Cc2c(C)oc(S)c2)cc(Cl)c(Cl)c(Cl)c1O.CO C(C(F)(F)Cn1cc(-c2cscn2)nn1)NC(CCSCC)=O Cc1nn(CCC(=O)N(C(C)CN(C(=O)C(c2ccccc2)C)C)C)c(C)c1C c1(N(C2CCN(C(C(CCC)OC)=O)CC2)C)ncnc2c1cnn2C c1(CCC(=O)NCC(CNC(c2c(C)ncs2)=O)F)c(C)nc2ncnn2c1C N1(C(C(c2ccn(C)n2)C)=O)CCCC1CC(=O)NC1CCN(CCCO)C1 C1(CC)CSC(C(N2CC(C(c3cn(CCC(=O)NC)nn3)C3CC3)C2)=O)C1 C1(C)(NC(c2n(CC)nnn2)c2cnn(CC(F)(F)F)n2)CCC(C)=C(C)C1.OC C(=O)(C(C)CC(F)F)Nc1ccc(CNC(C=CC(=O)OCC)=O)o1 C1(CC)C(C(=O)NCCC(O)C(C)C)CCCN1C(=O)COC(C)C c1(CC(=O)N(C(c2nn[nH]n2)C)Cc2cccc(F)c2)c(Cl)cc(Cl)cc1Cl N1(C(Cn2ccc(C)n2)=O)CC2CCC(C1)C2CNC(c1cc[nH]c1C)=O C1(NC(=O)CN2CCCCC2)CCCC(C(=O)NCC2(CCO)CCCC2)CC1 CC1(C(=O)NC2CCC3CC2CO3)CCN(C(c2cc3n(n2)CCO3)=O)CC1 CN1CC(=O)N(CC(=O)N(C)CC2CC(F)CN2C(=O)C(CO)N(C)C)C1=O CC1CN(C(C2(C#N)CCCOC2)=O)CCN1C(n1cc(C(F)F)ccc1=O)=O C1(c2onc(-c3ccc(OC)cc3)n2)CC(C)(C)CN1CC1CC1c1ccncc1 c1(OC)nc(Cl)nc2c1CN(C1(C(F)(F)F)CC3(CCC3)C1)CC2 C(CCCCCCn1cc(-c2cccc(OC(F)(F)F)c2)nn1)NC(C(C)O)=O C1(NC(C#CC)=O)C2CN(C(=O)Cc3coc(-c4ccc(Cl)cc4)n3)CC12 CC(C)(C)CCC(=O)NCCC(C)(C)CNC(c1cnn(-c2ccccc2)n1)=O C(=O)(C1=CCC(F)(F)CC1)N(CCNC(c1c(N2CC(C)(C)C2)cccc1)=O)CC c1(C(=O)NCCCCN(C)C(C2(CCO)CC2)=O)ccncn1 c1(C(N(CC(=O)NC(c2ccnn2C)COC)C)=O)ccn(CCF)n1 C1(NC(C=CC(C)(C)C)=O)CCC2(CCN(C(C3(C4CC4)CC3)=O)CC2)C1 N1(C(=O)NCc2c(C)nn(CC(=O)OC)c2C)CCc2c(Br)ccnc2C1 C1(CC(=O)NCC2CN(C(C3CN(C4CCOC4)C3)=O)C2)(COC)CCOCC1 C1(OC)CC2(C(=O)N(C)CCOCCN(C(=O)CNC=O)C)CC12 Cc1ccc2[nH]c(-c3ccc(CNC(c4nc(Cl)c(Br)cc4I)=O)nc3)cc2c1 C(=O)(CC(C(F)(F)F)NC(=O)CCn1cccc1)NCCC(CC)CO Cn1ccc2sc(C(=O)NC3CCOCC3NC(=O)CN(C3CCCC3)C)cc12 C(=O)(CCC(CC)OC)NCCn1ccc(C(=O)NC(CCCC)CO)c1 N1(Cc2c(OCCOC)cccn2)Cc2ccc(O)cc2CC1C(=O)OC.C(=O)O c1(NCC(C2CCOC2)OCC)cccc(N2CCOC2=O)c1 c1(OC)cc(C=CC(=O)N(C2CCCN(C(C3(CF)CC3)=O)C2)C)sn1 N(C(=NCCCF)NCC1CCOC(C(C)C)C1)CC(C)(C)OCC(F)(F)F c1(C(=O)OC)cccc(NC(=O)COC(=O)CC2CNC(=O)C2)c1F C1(C)(CNC(C(C)(F)F)=O)CN(C2CCN(C(C34CCCCC3C4)=O)CC2)C1=O N1(C(C(C)CBr)=O)CCCC2(CCCN2C(=O)CNC(=O)C2CC2)CC1 C1(C(=O)NCCCCN(C)C(C2C(F)(F)C23CC3)=O)CN2CCCN1CC2 c1(C(=O)NC2CN(C(CSCC(C)=O)=O)C(C)C2)ccc2scnc2c1 C(=O)(C(C)C(F)(F)C(F)F)NCc1c(C(=O)NC(=O)OC(C)(C)C)con1 Cc1cc(=O)oc(C)c1C(=O)NC1CN(C(=O)CN2CCOC2=O)CCC1CO Cc1cccn2ncc(C(=O)NC3CN(C(=O)CC(C)C)CC3C#N)c12 C(=O)(CC(C)C(C)(C)C)NCC(C)CNC(c1cccc(N2CCCC2=O)c1)=O Cn1ccnc1CCC(=O)NC1(CCNC(C2(C(N)=O)CC2)=O)CCC1 c1(C(=O)NC(CC(C)NC(C(CC)(C#N)CC)=O)C)cnn2ccc(Br)cc12 CC(C)CC(C(=O)N1CC2CC1C2CNC(=O)C(F)C(C)(F)F)C(C)C Cc1nc(C(=O)NC(C2CCCC2)CNC(=O)C=CC(F)(F)F)co1 N1(CC(C2CCC2)OC)CCC(C2(NC(=O)Cc3ccon3)CCC2)CC1 N1(C(C2(CC)COC2)=O)CCCC2(C1)CN(C(C1(CC)CC(C)(C)C1)=O)C2 c1(C(N2CC(NC(c3ncn(CC)c3)=O)(CF)C2)=O)ccc2cnoc2c1 CC1CCN(CCC(=O)N(CCCCNC(=O)C(C)Cn2ccnc2)C)CC1 C1(n2cc(COCC(=O)NCc3cc[nH]c3)nn2)CON(C(=O)C2CCCC2)C1 CC1(C)c2[nH]nc(O)c2CN1C(C1CCC(c2ccccc2)O1)=O c1(SCC(=O)N(CCN(C(=O)C(F)CCCC)CC)CC)nnc2ccccn12 c1(O)c(C)nc(C)nc1O.c1(CC(=O)OCC)nnc(OCS(=O)CC)s1 N1(C(c2ccn(C)n2)=O)CCC(NC(=O)Cc2cc(F)cc(F)c2)C12CC2 C1(CNC(CCOCCCOC)=O)CCCN(C(c2cccc(C)c2O)=O)CC1 N1(C(C2CC(C#N)C2)=O)CCC2(CC1)CC2CNC(=O)CC1CCCCC1O c1(C(N2C(C(C)C)C(=O)N(C)CC2)=O)cnc2c(c1)nnn2O N1(C(C2CCC(F)(F)C2O)=O)CCC2CCC(C1)N2C(C1CCOCC1)=O C(=O)(C1=C(Cl)CCCC1)NC1CN(C(c2[nH]cc(OC)c(=O)c2)=O)C2C1C2 Cc1cnccc1C(C)C(=O)N(C)CCNC(C1CCNC(=O)C1)=O c1(CN2CC(NC(c3cc(OC)ncc3)=O)C(F)C2)cc(Cl)ccc1Cl c1(C(=O)NC(C2CCN(C(c3c(C)nc(O)[nH]3)=O)C2)C)cc(N)nc(Br)c1 C12(N(C(c3cn(C)cn3)C(=O)NC(CC)C)C)CCC1CC2.c1ccccc1 N1(C(C)=O)CSCC1C(N1CCC(N(C(=O)Cc2ccc[nH]2)CC)C1)=O.C1(C)CC1 C1(C(=O)NC2CCN(C(CC(C(C)C)(F)F)=O)C2)CCOCC12CCCCC2 N1(C(C(C)OCC)=O)C2CCC(C2)C1CC(=O)NCc1cc(F)cc(F)c1 C1(C(N2CC(CCCCNC(CN3C(C)CC3)=O)C2)=O)CCCSC1 c1(C(=O)NCC2CC(F)(CNC(c3cccnn3)=O)C2)cccc(C2COC2)c1 CC(C)C(CCNC(c1cn(C)nc1Cl)=O)NC(=O)C(C)(C)O C12(C(=O)NC3C(CC)CN(C(Cc4ccc(CC)cc4)=O)C3)CCCC1CCC2 N1(C(C)=O)CCOCC1CC(=O)NCCc1nccc(O)n1 c1(C(=O)NCC2C(C)CCN(C(CCC=C(C)C)=O)C2)ccc2nc[nH]c2c1F C=Cc1ccc(C(=O)NCC2CCN(C(=O)Cn3nccc3C(=O)O)CC2)cc1 c1(C(N2CCC(NC(CC(COC)C)=O)C(F)C2)=O)cc(C)c2c(c1)CCCN2 c1(CNC(c2ccccc2)C(=O)N(C)Cc2cccs2)ccc(Br)nc1 N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(C2(C)CC(C3CC3)=NO2)=O)CC(O)C1 CCC(CC(F)(F)F)C(=O)NCC1CC(NC(=O)Cn2cc(C(=O)NC)nn2)C1 C1(C(N(CCCCC=C)C)=O)CCC(C)N1C(c1ccnc(CO)c1)=O N1(C(CCCOC)=O)CCN(C(c2c(C3CC3)cnn2C)=O)CC1c1cn[nH]c1 c1(CC)nn(C)c(Cl)c1C(=O)NC1CCCN(C(=O)C(O)CC(F)F)C1 C1(C(=O)NC2CC(C)CO2)CCCCC1n1cc(CC2(CC)CCC2)nn1 C(=O)(C1CCc2ccc(C)cc21)N1CC2(CCC(CNC(C(COC)C)=O)O2)C1 N1(C(CCCC(C)NC(C(C(=O)OCC)(C)F)=O)=O)CCC(C2(O)CC2)CC1 C(C(C(C)(C)C)NC(C1CN(C(C)=O)C1)=O)NC(Cn1cc(C(=O)OC)nn1)=O C1(C(N(C2CCN(C(c3cc(=O)cc[nH]3)=O)C2)CCC)=O)CC(=O)C12CCC2 c1(CC(=O)NC2CN(C(CCSc3n(C)nnn3)=O)C2)c(F)cncc1Cl N1(C(C(CCC)=CCC)=O)CCOCCC1CNC(=O)Cc1cccc(O)c1 n1(CCOCC=C)c(N(C2CCCC2CF)C)nnc1CCCS(C)(=O)=O C1(NC(=O)NCc2ccc(OCCCC)nc2)CCCC(CC)C1 N1(C(CN(CCC)C)=O)CC2CCC2(CNC(c2cccc(C(C)(F)F)c2)=O)C1 c1(CNC(C(CCC=C)C)c2nnnn2CC(=C)C)sc2ccccc2c1Br CCCN=C(NCC1CC1C(C)(F)F)NC1CCCN(c2cc(C)nn2C)C1 CN1CC(N(C)C(c2occc2CNC(=O)CCCN=[N+]=[N-])=O)CCC1=O c1(C(=O)NC2C(C)CN(C(=O)CCc3ccn(C)n3)C2)nc(Cl)ccc1Cl C(C(CC(F)(F)F)NC(C1CC1C(=O)OCC)=O)NC(Cc1ncc(CC)[nH]1)=O c1(CN2CCCN(C(=O)Cc3ccnc(Cl)c3)CC2)ccc2c(c1)CCO2 C(=O)(C(C)CNC(=O)CC1OCCO1)NCC1CN(C(C)=O)C1 C1(NC(C(CC)NC(C)=O)=O)COC2C(NC(=O)CCc3ccoc3)COC12 Cc1ccc(C#N)cc1C(=O)NCC1CN(C(=O)C=Cc2cocn2)C1 c1(OC)ncc(C(N2CCCC2C(=O)Nc2ccc(I)c(C)c2)=O)cc1Br N1(C(C2C(CC(C)(C)C)C2)=O)CC(NC(C2CS(=O)(=O)C2)=O)CC2(CC2)C1 C(=O)(C(F)C(C)(C)O)N1CC(C(N)=O)(CNC(C(C2CCOCC2)OC)=O)C1 CCCCCCCC(=O)N(C)CCNC(=O)C(C)(C)Cc1cc2ccccc2o1 C1(NC(C2(OCC)CCCCC2)=O)CC2(CCN(C(C3CC3C#N)=O)CC2)C1 C1(C#N)(C(=O)NC2C(NC(CCC3(C)CC3)=O)CCC2)CCCO1 CC(C)(C(=O)NC1CCN(C(=O)C2CC2)C1)c1ccc(-c2cn[nH]c2)s1 c1(C(=O)NCCC2(OC)CN(C(=O)Cc3ncc(C)s3)C2)nc(C)c(C)[nH]c1=O N1(C(CC2CCCC(C)O2)=O)CC2CC(C)N(C(=O)CC(F)(F)C(F)(F)F)C2C1 CCCCN=C(NCCNC(c1ccoc1C)=O)N(C)Cc1c(F)cccc1F C1(C(N2CCCC(NC(=O)CN3CCCC3)(CO)C2)=O)C2C3CC4C1C1C2CC3C41 c1(C(=O)NCC=C2CCN(C(CCC3CC(C)C3)=O)CC2)cc2cccnc2[nH]1 n1(CC=C)cc(C(=O)N(C(CC)C(=O)NCCn2cnnn2)C)nn1 N1(C(CCCCOC)=O)CC(C)(C)OCC1CNC(c1cc[nH]c1C1CCC1)=O N1(C(Cc2cccc(C(C)C)c2)=O)CCC(C)CC1CNC(=O)C(C)S(C)(=O)=O c1(CC(C(=O)NCCCC#C)F)ccc(NC(=O)OC(C)(C)C)cc1 c1(CNC(CC2ON=C(C)C2)=O)nc(C(=O)NCC2CCOC2=O)c(C)o1 C1(C(=O)NC(C)(CNC(=O)COc2ccsn2)C2CC2)CC2CCCCN2C1 C1(C(=O)NCCCOCCN(C(=O)CCc2ccoc2)C)CCC(F)C1 CC(C)CC(CNC(=O)C(C)Cn1ccnc1)C(=O)N1CC(O)CC1C(C)C CC1C(=O)NCCCN1N(C)Cc1ccc(Oc2ccccc2)cc1 C1(NC(COCCCOCC)=O)CN(C(=O)C(C2CCOCC2)F)CCC1(C)C C1(C(N2CCN(CC)C(=O)C2)=O)C2CCCC2CCN1C(=O)C(F)(F)F C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCCC(CN(C(CSCCC)=O)C)C1 N1(C(c2cnc(S)nc2)=O)CCC2CN(C(c3scc4c3OCCO4)=O)CC2C1 c1(C(=O)NCCCC(C)(C)NC(C=C(CC)CC)=O)cc2c(C)cc(C)cc2[nH]1 c1(C(=O)NCC(CNC(c2ncc(OC)nc2)=O)C)cccc2c1C1CCC2O1 N1(C(CC(C)(C)C)=O)CCC(C2CC(NC(=O)CC3CC(n4cnnc4)C3)C2)C1 N1(C(CC)=O)CCN(C(=O)C(C)(C)C2CCCN2C(=O)CC(CC)C2CC2)CC1 C1(NC(=O)COCCF)CC(CNC(=O)C(=O)NC2CC2)C12CCC2 c1(C(CCCC)OCCC)nc(-c2ccco2)nn1CCC c1(C(N2CCC(C(N(CCC=C)CC)=O)CC2)=O)cccc(C#N)c1C C1(N(C)C(c2ccc(O)nc2)=O)CCCN(C(=O)C(C)(C)c2cccnc2)C1 C1(C(=O)NC2CCCC(NC(CC3C(C)OCC3)=O)C2)C2CC3CC(C2)CC1C3 N1(C(C2ON=C(CC)C2)=O)CCCC(C)(C(=O)NCc2cnc[nH]2)C1 C1(C(=O)OCC)CC2(CC(NC(C34CCC(CC3)C4)=O)CCS2(=O)=O)C1 C1(C(=O)NCCC(C)C(F)F)CCOCCN1C(=O)CCC1CCOCC1 c1(NCC(=O)NC2CC3CCC2(CNC(C2CC2F)=O)C3)cccc(Cl)c1Cl C(=O)(CC(CSC)NC(C12CCN(CC1)C2)=O)NCCCN(CC)CC c1(C(=O)NCC2CCCN(C(C3(OC)CC3)=O)C2)ccc(=O)n2c1CCC2 N1(C(Cn2ncc(CC)c2)=O)CCN(C(C2C=CC=CC=C2)=O)CC12CC2 C1(NC(c2c(C#C)c[nH]n2)=O)CC2CCC1(NC(C1CC(=C3CCC3)C1)=O)C2 c1(CCNC(c2nnnn2-c2ccc(C)cc2C)CCC)cnn2c1CCCC2 C12=CC=C(C=C1)C2c1cn(CCOC)nn1.C=C1CCCC1C(=O)OC(C)(C)C C1(C(=O)NCC(C)N(C)C2CC2)CC2CCC(C1)N2C(c1ccc(F)cc1O)=O C1(CC=C)(C(N2CCCC2CN(C(=O)C(CC)OCC)CC)=O)CC=CC1 Cn1nnc2cc(C(N3CC4(C3)SCCC4NC(C3CC=CCC3)=O)=O)cnc12 c1(C(N2CCC(CCN(C(C(CC)C(C)O)=O)C)CC2)=O)ccc2ccoc2c1 C1(C(=O)O)C[Si]2(CCCC2)CN1C(c1nc2n(c1Cl)CCCC2)=O c1(C(=O)NCC2CN(C(CC(C)OC)=O)C(C)(C)C2)nc2ncccn2n1 C1(C2CCN(C(C3(F)CCCC3)=O)CC2)(NC(c2ccc(NC)cc2Cl)=O)CC1 C1(C(N2CCC(O)(CNC(=O)CC(C)F)CC2)=O)(COC)CCCNS1(=O)=O c1(C(=O)NCC2C(NC(=O)CCc3csnn3)CC2)ccc(C(F)(F)F)o1 c1(NC(C(C)C2CCOC2)=O)cccc(NC(=O)C(=O)NCc2ccccc2)c1 C1(NC(c2c(Cl)cn(C)n2)=O)CC(O)CN(C(=O)CCSCC(N)=O)C1 N1(CCOCC)CCN(CCCCCNC(C2(C)CCCN2C(C)=O)=O)CC1 c1(C(N2CCC(N(C(CN(CC)CC)=O)C)C2)=O)cc(N2CCOCC2)ncn1 N1(C(C2(CC#C)CC2)=O)CCCC(C2CN(C(C3CCC=CCCC3)=O)C2)C1 c1(NC(c2c(-c3c(C)cncc3)ncs2)=O)ccc(C(F)(F)F)c(O)c1 c1(C(CO)NC(C2C(NC(C3CC(=O)NC3)=O)CCC2)=O)ccccc1Br C(=O)(N=c1[nH]c(Cl)ncc1O)c1cc(-c2c(SC)c(F)cc(F)c2)[nH]n1 c1(C(c2nnnn2CCC2CC2)NCC2C(C)C2C)cc(-c2ccco2)on1 CC(CS(C)(=O)=O)C(=O)N(C)CCOCCNC(c1cnn(C)c1F)=O N1(C(c2c(C)nccn2)=O)CC2OCCN(C(=O)CC3OCCOC3(C)C)C2C1 CC1CCN(C(c2cnc3ccccn23)=O)CCN1C(c1cc(Cl)ccc1O)=O C(CCC(=O)NC(C1(Cc2nnc(O)s2)CC1)C)SCC.C1(=O)CN1C1CC1 CC1CN(C(=O)C=CC2CCCC2)CC1(C)CNC(=O)C(O)CC1CC1 C1(CNC(C2CCC(C)(C)O2)=O)CN(C(=O)C#CC2CC2)CCCO1 C(=O)(C#CC(C)(C)C)NC(C(C)C)C(C)NC(c1csc(-c2cnccn2)n1)=O CC1(C)CN(C(=O)CSc2ccccn2)C1C1CCN(C(=O)C2=CCCO2)CC1 c1(NC(C(C=C)O)=O)cccc(CNC(=O)COCc2ncnn2C)c1 N1(CCC)CCCC(C(=O)NCC2CN(C(C34CCC(CC3)C4)=O)CC2O)C1 CCC(CCC(=O)NCc1ccc(F)c(O)c1)NC(=O)C(C#N)CC Cc1cn2c(n1)CCC(C(=O)NC1CC1CNC(C1(CC(C)C)CC1)=O)C2 C1(C(=O)NCC2(CCOC)CC2)CN(C(c2ccon2)=O)CCC1(C)C CC1C(O)CC2CCC1N2C(=O)C(=O)NC1(Cl)CCOCC1 N1(C(CCCCCC(C)C)=O)CCC2CCCN(C(=O)CCOCCN(C)C)C2C1 N1(C(c2cc(C)c(O)nn2)=O)CCCC(C2CC2NC(=O)C#CC(C)(C)C)C1 n1(C(CN(CCCO)C)C)cc(SCCNC(=O)COC(c2ccco2)C)nn1 N1(C(C(C)=C2CC2)=O)CCN(C(=O)CCN(c2ccccc2)C(=O)CO)CC12CC2 c1(OCC)cc2c(=NC(CN(C)C)CCO)[nH]cnc2cc1F c1(CC)nnc2n1CCCC2C(=O)NCCOC1CCN(C(c2cc[nH]n2)=O)C1 c1(NC2(CS(C)(=O)=O)CCC2)nccc(=NCCC(CC2CC2)C2CC2)[nH]1 C=CCCCCC(=O)NCC(C1CC1)NC(C1(C(=O)N(C)C)CC1)=O C(=O)(CCS(=O)(=O)N(C)C)NCCC(C)NC(=O)CC1CCCCC1(F)F N1(C(C=CC=CCC)=O)CC2CC(C)N(C(c3ccnc(F)c3OC)=O)C2C1 CCN=c1[nH]cc(C(=O)NC2CCC(NC(=O)COCC3CCOC3)CC2)s1 C(=O)(C1CCCn2c(C)nnc21)N1C(CNC(c2ccc(C)c(O)c2)=O)CCC1 c1(C(N2CCC(F)(CNC(C(C)S)=O)CC2)=O)ccc(Br)c(Cl)c1F C=CC(C)N=c1[nH]c(N2CCC(C3CCS(=O)(=O)CC3)CC2)nc2c1COC2 CCC1=NOC(CNC(=O)CC2(NC(=O)Cn3cccn3)CC2)C1 c1(C(=O)OC)cn2cccc(NC(c3cc4cc(Br)sc4[nH]3)=O)c2n1 C1(C(C)NC(=O)CSc2nncs2)CCCN(C(C2CCC(=O)C2)=O)C1 C(c1cc(F)c(F)c(F)c1)=CC(=O)NC1COCCN(c2ncc(Br)cn2)C1 C(CC(C(=O)N1CC(CCNC(=O)Cc2nn(C)cc2Cl)C1)NC(C)=O)SC C(CS(=O)(=O)c1ccc(Br)cc1)NC1(c2ccc(Br)cc2)CCN(C)C1 CCCC(O)C(=O)NC1CC(C)(C(=O)NCCC2CCN(C)CC2)C1 C1(S(C)(=O)=O)(C(=O)NCC(CC)NC(C(C=CC)O)=O)CC1 c1(CCNC(c2cnc(C)s2)=O)ccc(F)cc1Cl N1(C(c2cc(OCC)n[nH]2)=O)CCCC2(CCN(C(C3CC(F)C3)=O)C2)C1 C#CC1(NC(=O)COC2CN(C(c3cncc(C#N)c3)=O)C2)CCC(C)CC1 c1(OC)ccc(N2CCC(C(=O)NC3(c4ccccc4)CC3)C2)c(C#N)c1 N1(C(C(C)N(C)C)=O)CC2(CNC(c3cnc(Br)s3)=O)CCC1CC2 N1(C(C2CC(OC)C2)=O)CCCC1(C)CNC(c1c[nH]c(=O)cn1)=O c1(SCC)cc(C)c(-c2nc(C3CCCCC3)nn2-c2cccc(C(N)=O)c2)o1 c1(N2CCC(NC(C3CCCO3)=O)C(F)C2)nc2ncc(Cl)cc2s1 C1(C(=O)OC)C(OC)CCCN1C(=O)NCCS(C)(=O)=O.C(C)(C)(C)O C(=O)(C(C)(C)C(=O)N1CCOCC1CNCc1cncc(Cl)c1Cl)OC c1(OC)c(O)cc(C(N2CC3(CCN3C(c3cnccn3)=O)C2)=O)cc1O C1(CSC)CN(C(c2sccc2Cl)C(=O)NC2COC2)CCO1 N1(C(c2ccc(C(C)=O)o2)=O)CC2CCC1C1CN(C(=O)C(C)=CC3CC3)CC21 CC1(C)CCCCC(C(=O)NCCC2CSCCN2C(=O)Cc2csc(Cl)c2)C1 n1(CC#C)cccc1C(=O)NCC(=O)N(C1CN(C)C1)C Cc1cc(Cl)ccc1N(C(=O)COC(C)(C)CNC(=O)CC1CC=CC1)C1CC1 C1(C(C)C)CC(C(=O)NCC#CCNC(=O)CCc2cncs2)C1 C1(C(N(CC(CC)NC(c2c(C(F)(F)F)cnn2C)=O)CC)=O)CN(C)C(=O)N1 C12(CCOC(C34CC(C(=O)O)(C3)C4)=O)CCC(CC1)CC2 C(=O)(CC(C)(C)C(=O)NC1CN(C(=O)C=Cc2cc[nH]n2)CC1OC)OC C(=O)(C(C)CCC(C)(C)C)N1CCN(C(CC2(C(C)=O)CCC2)=O)CC1C(C)C c1(OC)cccc(Cl)c1C(=O)NC1CCCN(C(C2CCC(=O)N2C)=O)CC1 c1(C(=O)NC2CN(C(=O)COc3cccnc3Cl)CC2O)cccc2[nH]ncc12 N1(C(C2(SC)CCC2)=O)CCC(C2CCN(C(C3CS(=O)(=O)C3)=O)C2)CC1 n1(CCC=C=C)cc(CC2CCCN2C(c2nccn2C(C)C)=O)nn1 CC1CCN(C(C2(n3cccc3)CCCC2)=O)CCC1(F)F C(CCCCCC(=O)NC(c1cncs1)C)NC(C1C(C)C(=O)OC1)=O N1(C(CCc2cnc(C)o2)=O)CCC(C2CCN(C(=O)C(F)(F)CO)C2)C1 S(=O)(=O)(c1ccc(C(=O)O)cc1)N1C(CC(=O)Nc2c(C)nc[nH]2)CCC1 C=CCC(F)(F)C(=O)N1CC(CNC(=O)C(c2ccc(Cl)c(F)c2)O)C2(CC2)C1 C1(CCC(=O)N(CC(C)O)CC)CCN(C(=O)Cc2csnn2)C1 N1(C(C2(C)CCOCC2)=O)CC2(CCC(C(=O)NCC3(CC4CC4)CC3)O2)C1 N1(C(C(C(=O)OCC)(C)F)=O)CCC(C)N(C(c2cc(CC)cc(Cl)c2)=O)CC1 c1(CNC(C2(CNC(C(c3ccn(C)c3)C)=O)CC2)=O)ccc(C#N)cn1 O=C1CN(C(=O)NC2C3Cc4c(Br)cccc4C23)c2cc(Br)cnc2N1 C1(NC(CCc2ccc(C(N)=O)cc2)=O)CCN(C(C2(O)CCCC2)=O)CC1O Cc1cc(=NCCc2ccc(N(C)C)cc2)[nH]c(=NCc2ccc(N)cc2F)[nH]1 S(=O)(=O)(c1ccc(Cl)cn1)N(C(CCO)C(C)(C)F)C c1(CNC(CCCn2cc(CC)nn2)=O)ccc(OCCN2CCOCC2)nc1 CC(CCCNC(=O)C(C)(NC(=O)SCCC1CC1)NC(N)=O)OC(C)(C)C C(CC(O)C(=O)NC(Cc1cn[nH]c1)C(=O)NCC1(O)CCSC1)N(C)C CC(C)CCC(O)C(=O)N1CCC(C(=O)NC(C)Cc2cccnc2)O1 N1(C(C(C)Oc2ccccn2)=O)CC2CC1CN2C(c1cc(I)cnc1Cl)=O c1(OC)ccc(C)cc1Cc1cc(C(=O)OCC)no1.C12(C)CC(C1)CNC(=O)N2 c1(C(C(N2CC(CC=C)(NC(C3CCSC3)=O)C2)=O)=O)ccc(C(C)C)cc1 N1(C(Cc2nc(C)sc2)=O)CCC2C(NC(c3ccnc4c3CCC4)=O)C2CC1 CC1(C)CC1(O)C(N1CCC(CNC(c2csc(N3CCCCC3)n2)=O)C1)=O N1(C(CCC2CCC(=O)N2)=O)CC2CCC1CC2NC(c1cccc(O)n1)=O N1(C(c2c(C)oc(CNC(=O)CCNS(C)(=O)=O)c2)=O)CC(F)(F)CC1CO C(=O)(C(C)C(C)C(C)(C)C)N(CCCNC(Cc1ccc(C(C)C)cc1)=O)C c1(C(=O)NC2(C)CCCN(C(C(C)C(F)(F)F)=O)C2)cc2c(F)cccc2s1 c1(NC(C2CN(C(=O)CCc3ccco3)CCC2(F)F)=O)ccc2c(c1)CCC2 CC(CCCCNC(c1cnc(-c2ccco2)s1)=O)NC(C1CC(C)(C)CO1)=O C1(C(N2CC(C(N3CC(CC#C)OCC3)=O)(CC)C2)=O)CCCC2(CC2)C1 c1(OC)cccc(C(N2CC3CC2C3CNc2csc(NC(=O)C(C)O)c2)=O)c1 N1(C(CC2ON=C(CC)C2)=O)CCCC(C(=O)NCC2(CCO)CC2)(CC)C1 N1(C(c2ccc(O)c(F)c2)=O)CCC2(CC1)CN(C(C13CCCC1C3)=O)C2 C1(CC=C)(C(=O)NCC(n2cnnn2)C)CCCN1C(=O)CC c1(C(=O)Nc2cc(Cl)cc(Br)c2C)ccc2c(NC(C(CC)C)=O)n[nH]c2c1 CN1CCC(N=c2[nH]c(=N)[nH]c(=NCc3cc(O)n[nH]3)[nH]2)c2ccccc21 N1(C(C(CC)(C)CC)=O)CCC2CCN(C(C3CC(n4cnnc4)C3)=O)C2C1 Cc1cc(O)c(Cl)cc1C(N1CCCC1CN(C(=O)CN1CC2CCC1C2)C)=O Cc1cc(NC(=O)C(c2cccnc2)NC(=O)Cc2cscn2)cnc1O N1(C(c2c(C)ccs2)=O)CCC2(CC1)CC2NC(c1c(C)cncc1C)=O C=CC(C)(CC)C(=O)N1CC(O)(C(F)C(=O)NCCC2(CO)CCC2)C1 C(C(C)(C)CCCO)OC1CN(C(CCCNC(c2c(CC)n(C)nn2)=O)=O)C1 C1(CNC(C2(CC)CC2(F)F)=O)CCN(C(=O)CC2CCOC2(C)C)CC1 N1(C(C2(NC(C)C)CC2)=O)CCC(NC(=O)CCc2ccc(Cl)cc2F)C(C)C1 Cc1cc(C(=O)NC2CCCC2CNC(=O)CSC2CC2)c(C)cn1 CC1CC(N(C)C(C2(CNC(c3ccc(C#N)s3)=O)CCCC2)=O)CC(C)C1 CC1(C)CC(NC(c2ccnc(OCCO)c2)=O)CN1C(c1[nH]cnc1C#N)=O Cn1nnc2c(N3CCOC(CNC(C45CCCC4C5(F)F)=O)C3)ncnc12 N1(C(C2(CC#C)CCOC2)=O)CCC(C)(NC(=O)C(F)C2CCCC2)CC1 N1(C(CC2CC(=C)C2)=O)CCCCC1C1(NC(=O)C=CC2CCCO2)CC1 C1(C(=O)NC2CC(CC(=O)OC)C2)(CNC(=O)NCC(F)(F)F)CC(C)(C)C1 c1(C(=O)NCC2(NC(c3ccccn3)=O)CCC2)ccnnc1Cl c1(C(=O)NCCC(C)NC(=O)C(C2CC2)C2CC2)cc(F)c(Br)cc1N C1(C(=O)NC2(CC#C)CC(F)(F)C2)CCN(C(=O)CC(C)n2cccn2)CCO1 c1(C(=O)NC2CCC(C)(NC(C3CC4(C3)CC4F)=O)CC2)occ2c1CCCC2 N1(C(CCc2onc(CC)n2)=O)CCCC(C)(C)C1CNC(=O)CC1CC1(Cl)Cl n1(C(CC)C)nnnc1C(c1cnccn1)NCCCOC(C)(C)C c1(-c2n(CCC(C)(C)OC)nc(C3CCOC3)n2)cc2c(s1)CCSC2 N1(C(C(CCOC)OC)=O)CCCC(NC(c2cnsc2)=O)CC1 C1(NC(c2c(C)coc2)=O)CN(C(=O)Cc2cn(C)cn2)CC1N=[N+]=[N-] c1(C(C)=O)ccc(C(=O)NCC(C)CNC(c2cc(C)oc2C(F)(F)F)=O)nn1 C#CC1CCCCN1C(c1ccnc(CNC(C2(SC)CC2)=O)c1)=O C1(C)(CNC(C(N2CCCCC2CO)CC)=O)CCN(C(=O)CNC2CC2)CC1 C1(c2cn(CC(=O)N(C3CCS(=O)(=O)C3)C)nn2)(OC)CCCCCC1 c1(C(N2CC(CC)C(C(=O)O)C2CC)=O)csc(=NC2CC2)[nH]1 O=C1CC2(C1)CC(C(=O)NCCC1CC(C(=O)N(c3cnsc3)C3CC3)C1)C2 C(CC1=CCN(C(c2nncn2C)=O)CC1)NC(C=Cc1cnc(OC)nc1)=O n1(CC(C)O)cc(C(N2CCC(NC(c3cc(N)cc(F)c3)=O)C2)=O)ccc1=O C12(NC(CNC(N)=O)=O)CCCCCC1N(C(C1CC=CCO1)=O)CC2 C1(NC(C2CC(SC)C2)=O)CCN(C(c2coc(C3CCCCC3)n2)=O)CC1C C1(F)(CNC(=O)CCC2CC2(F)F)CCN(C(C2(c3ccno3)CC2)=O)C1 c1(C(=O)NCCCN(C(c2cc(C)[nH]n2)=O)CC)cn(C)nc1C(F)(F)F C(=O)(C#CC1(C)COC1)N1CCC(N2CCN(C(CC=CC)=O)CC2)C1 c1(OC)cccc(C(=O)NC2CC(F)(CNC(=O)COCC3CCOC3)C2)c1F N1(C(Cc2c(C)non2)=O)CCOCC1CC(=O)NCC1(C)CCOC1 C1(C(=O)N(C2CC2NC(C23CSCC2C3(F)F)=O)CCO)CCC(F)(F)CC1 C(CCC)(C(=O)NCC12CC1CN(C(=O)CCc1n[nH]c(=N)s1)C2)=CCC N1(C(CC(n2c(CC)ncc2)C)=O)CCC(CNC(c2cc(C)sn2)=O)CC1C CCS(=O)(=O)CC(=O)N1CC(NC(c2c(C)cnn2C(C)C)=O)CC(C)C1 C(=O)(C(CSCC)NC(=O)CSc1nc[nH]n1)NC(C(=O)N(C)CC)C C1(NC(C2(OC)CC2)=O)CN(c2cc(Cl)nc(SC)n2)CC2(CCC2)C1 Cc1cc(C(C)C)ccc1OC(C)C(=O)NCCCNC(=O)C(F)(F)C(F)F N1(C(C(C=C=C)C)=O)CCC2(CCC(CNC(c3cscc3Cl)=O)CC2)CC1 c1(CNC(=O)C(=O)N2CC(Cc3ccnn(C)c3=O)C2)nn(C)c2c1CCCC2 c1(N2C3CC(=C)CC2CC3)nc2cc(CC)ccc2n1CC1CNCC(C)O1 C(=O)(CC1OCc2ccccc21)NCCCN(C(C1CC(=C)C1)=O)CCO c1(C(N2C3C(C(=O)NC(CC)CO)C(C3)C2)=O)ccc(OC)cc1O C1CCCCC(N=c2[nH]c(N3CCC4(CC3)COC4)nc3c2CCCCCC3)C1 C1(CNC(CCCC)=O)COCC2(CCN(C(=O)CN3CCCC3)C2)O1 c1(C(C)NCCc2ncccc2F)cc(Cl)cc(Cl)c1.n12nnnc1C2(C)C C(CCCCC(=O)NCC1CCN1C(=O)C(C)CF)NC(=O)OCC c1(C(=O)NCCCCCN(C(C(N2CCC(O)CC2)C)=O)C)cc2sccc2[nH]1 c1(C(N2CC(OCCNC(=O)CC3CC=CC3)C2)=O)ccc(C2CC2)nc1O c1(C(=O)NCC2N(C(C(CC)SC)=O)CC3(CCC3)C2)ccc2oc(C)nc2c1 C(=O)(CC(C)C(C)(C)NC(=O)C(C)NC(C)=O)N1CCC(CC=C)C1 c1(CNC(CC2ON=C(C)C2)=O)nnc2n1CCN(C(C1C(C)C1(F)F)=O)C2 C1(CNC(C(C)C2CCCC2)=O)CCC(NC(C2(C(N)=O)CCC2)=O)C1 C1(C(=O)NCCCN(C(c2csc(Cl)n2)=O)CC)(CCN(C)CCO)CCCC1 N1(C(CCC(=O)N(C(C)C)C)=O)CCN(C(c2cccc(O)c2)=O)C2CCC12 C(=O)(C(C)CC(N)=O)NCC(C)=CC(=O)NC1C(=O)OCC1CO C(C)(C)(CC(=O)NCC1(C)CCN(C(=O)CCC2CC(F)(F)C2)C1)OC C1(NC(CCCC2C(C)C2)=O)C2CC3C(C2)C13C(=O)N(CCO)Cc1cn(C)nn1 C=CC1(C(=O)N(C)Cc2csnc2C)CCN(C(=O)CC(C)C(F)F)CC1 C(CC(=O)N1CCCC1(C)CNC(c1cnsc1)=O)(C(C)C)OCC c1(C(=O)NCC(=C)CCNC(C2SCCCS2)=O)ccc(-n2cc(C)cn2)cc1 N1(C(c2ccc(CC)s2)=O)CCC2CN(C(c3ccccn3)=O)CC2CC1 N1(C(c2cccc(CCC)c2)=O)CC(F)(F)CC1(C)CNC(=O)C=CCF N1(C(C2C(CC)CCC2)=O)CC(NC(C2CCC(C)O2)=O)C(C)(C)C1 N1(C(C(CCC)(C)C)=O)CC(C)OC2(CCN(C(c3n[nH]c(CC)c3Cl)=O)C2)C1 n1(CC(=O)N(C(C)CNC(C2CC2(F)F)=O)C)cnc2c1CCCC2 c1(OC)nc(C(N2CCN(C(c3cc(OC)ccc3F)=O)C3CC23)=O)cc(O)n1 c1(CCC(=O)NC2CCC(CC(N3CC(O)C(F)C3)=O)CC2)cccc(Br)c1 C(CCC(C)(C)C(=O)N(C)CC1CC1C)NC(C=CCCC)=O C(=O)(C(C)(C)C(=O)N(C)C)NC(CC)CC(=O)N1CC(C(N)=O)C(C)C1 c1(C(N2CC(NC(CC=CC(C)(C)C)=O)C2)=O)ccc([N+](=O)[O-])c2cccnc12 N#Cc1cc(C(=O)NC2CC2CNC(=O)CSC2CC2)c(F)cc1F C(CCCCCN(C)C(C1CC1CCC)=O)NC(C1(CC#C)CCOC1)=O N12CCC(CC1)C2=O.C(CNC(=O)Cc1ccoc1)(CNC(C)=O)OC c1(CC)cc(C(=O)NC(c2ccccc2)CNC(C2(C#N)CCOC2)=O)nn1C c12ccc(Cl)c(c1)N(CC1N(C(CCC=C)=O)CC1)C2=O.c1(NC)ccc[nH]1 N1(C(C=CC(C)NC(=O)C(c2cccnc2)O)=O)CCC(C2CC2)CC1 C1(CCC(=O)N(C)CC2CCCN2C(=O)CC2OCCCO2)CCCC(=O)N1 N1(C(C=CCC)=O)CCN(C(=O)CCC(C)(C)C)CC1C(C)C C1(CN(C)C)(CNC2(C)CN(CC(=O)NC)C2)CCCC1 N1(C(CCC)=O)CC(N(C(=O)CCCCNC(c2ccccc2)=O)C)C(F)C1 C1(C(N(CCCC)C(C)CC)=O)OCCC1NC(C1(C)CC1)=O C1(CNC(c2cnc3[nH]cnc3c2)=O)CCC2(CN(C(c3cn[nH]c3)=O)C2)O1 C(=O)(CCCCCF)NCC(C(=O)NCC(N(OCC)C)=O)C n1(CC(N2C3(CNC(C(C)N(C)C)=O)CC(C2)C3)=O)c(=O)cnc2ccccc12 C(=O)(C(C)(C)C(C)(F)F)N(CC(C)C(=O)NC(C)C(=O)NO)C N1(C(c2ncn(C(C)C)n2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1C(F)F C1(F)(C(N2CC3C(NC(C(c4c(C)cccc4)(F)F)=O)(C3)C2)=O)CCS(=O)(=O)C1 c1(C(=O)NCCCCNC(c2[nH]cc(C)c2)=O)c(C)ccc2n[nH]cc12 C1(C(N2CC=C(C)C2)=O)N(C(c2ccc(O)cc2)=O)CCC1(C)C C12(C(=O)NC3C(CC=C)CCC3)CCC(CN(C(=O)CN(C)C(C)C)C1)C2 N1(C(C2(NC(N)=O)CC2)=O)CCC(C2CC2)(CNC(=O)C2=CCSC2)C1 Cc1cnc(N)c(C(=O)NC2CCOCC2NC(c2coc(C)c2)=O)c1 C1(O)(C(=O)NC(CCNC(c2c(C(C)C)noc2)=O)C)CCC(C)(C)CC1 C12(NC(C(F)=CCC)=O)CC(CNC(=O)CC(O)C3CCCC3)(C1)OC2(C)C C1(NC(CC2CCC(COCC)O2)=O)CCC(CC)CC1.C123CC(C1)(C2)NC3=O C1(CC(=O)NC(C(=O)OCC)C2CC2)C(NC(=O)CCc2ccccc2)CC1O c1(-c2nc(NC(CNC(c3c(C)scn3)C)=O)on2)cccc(F)c1 C1(CC(C)C)CCC(NC(=O)CCCN(C)C(c2c[nH]nc2C2CC2)=O)C1 c1(C(N2C(CCNC(=O)C(c3ccccc3Cl)O)CCC2)=O)ncncc1F c1(OC)nc(C(=O)N(CC(C)NC(c2ccc(C(C)(C)C)cc2)=O)C)ncc1F N1(C(CC(C)C)=O)CC(CNC(C2CN(c3ccccc3F)C2)=O)OC2(CCC2)C1 c1(OC(CC)C)cc(N2CC(NC(=O)CSC3CC3)C(C)(C)C2)nc(C)n1 CN1CC(C(N2CCC2(C)CC(=O)NCc2ccc(CO)o2)=O)CCC1=O C1(C(NOCC(C)(C)O)=O)CN(C(=O)CCCC#N)CC1(F)F Cc1ccc(C(=O)NCCc2n[nH]cc2C(=O)NC2CC2(C)C(F)F)nc1O N1(C(C2N(C(CCC(C)N(C)C)=O)CCC2O)=O)CCn2ccnc2C1 C1(CC(=O)NC(CC=C)CNC(c2ccnc(Cl)c2O)=O)CC2(CCCC2)CO1 N1(CC2CN(C(CCC)=O)C2)CCN(C(C2(COC)CCCCO2)=O)CC1 C1(CCCCC)CCCN(C(c2ccc(NCC(N)CO)cc2)=O)C1 c1(C(=O)NC2C(C)N(C(=O)C(CCO)N(C)C)CC2)[nH]nc2ncccc12 C(CC(=O)NCCN(CCCC1CC1)CC)(OCC)NC(C1OCCC1C(C)C)=O c1(NCC)cncc(C(=O)NC23CC2CN(C(c2ccncc2Cl)=O)C3)c1 c1(CN2CCCC(C(N3CCC(F)(F)C3)=O)C2)cc(Br)c(F)cc1F N=c1[nH]c(=NCCc2cc(Cl)ccc2Br)[nH]c(=NC2CCN(CC(F)F)C2)[nH]1 c1(C(=O)NCC(C)(CO)NC(c2c(CC)nc(C)[nH]2)=O)cccc2c1ncn2C Cc1nnc(O)c(C(N2CCCC(CNC(=O)C=CC3CCC3)C2)=O)c1C c1(NC(C(c2cncnc2)=O)=O)cnc(Cl)cc1C(N1CCSCC1)=O c1(C(N2CC3CCC(C2)C3O)C(=O)NCCOCC)ccc(C#N)c(F)c1 c1(NC(c2c(F)ccc(Cl)c2Cl)=O)cc2c(cc1Cl)OCCO2 C(CC(C(C)(C)C)NC(=O)CCc1c(Cl)cccc1Cl)NC N1(C(C(CCCC)O)=O)CCC2CCCC12C(=O)NCc1cnn(CCO)c1 C(C(C(=O)N1CC(C)(C)CC1CNC(=O)CC1(CO)CC1)C(F)(F)F)OC c1(C(N2C(C3(O)CN(C(C(C=C)O)=O)C3)CCC2)=O)cccc(C2(C#N)CC2)c1 C=CCCCCCC(=O)N1CCN(C(c2coc(Cl)n2)=O)C(c2ccncc2)C1 Cc1cnn(CCCNC(=O)C(O)C2CN(C(=O)C(O)CN(C)C)C2)c1 C1(CCC(=O)N(CCCCNC(=O)Cc2cnc[nH]2)C)CCCC(O)C1 C(=O)(CCCCC(N)=O)N(C1CC(NC(c2cn3c(n2)CCC3)=O)C1)C N1(C(c2c(CCC)nns2)=O)CCCC(NC(C23CC(CO2)C3)=O)C1C C1(C(C)C)CN(C(=O)CSc2nncn2C(C)(C)C)CCCN1C(=O)C(C)O c1(C(=O)NC2CC3(CN(C(C(CC(N)=O)O)=O)C3)C2)cccc2c1CNC2=O C1(NC(CCS(C)=O)=O)CC2CN(C(=O)CC3CC(O)C34CCC4)CC12 C(=O)(C(C)C(C)NC(C1(n2cc(SC3(C)CCC(=O)N3)nn2)CC1)=O)OCC c1(C(N(C2CCCCC2)CCNC(C(COC)(F)F)=O)=O)nccc(Cl)c1Cl Cc1cnc(CN2CCCC(O)(CNC(C3C4COCC34)=O)C2)cc1Br C(=O)(C(C(=O)NC(C)CN(C)C(C1CCC(C)O1)=O)OC)OCC C1(CC)C(C(=O)NCCOC2CC2)CCN1C(=O)C(COC)N(C)C c1(C(=O)NCC(CNC(C(CC=C)OC)=O)F)ccnc(F)c1OC Cc1csc(CC(N2CCCC2CN(C)C(c2cnn(CCO)c2)=O)=O)n1 C#CCCCCC(c1nnnn1CCC)NCC1CCC(C(F)(F)F)O1 c1(C(=O)NC2C=CCC(C(N(CC(=O)N(C)C)C)=O)C2)cnc2ccccn12 c1(C(=O)NCC(CC=C)NC(=O)C(C)CN(C)C)cnncc1C(F)(F)F S(=O)(=O)(c1c[nH]c2ccccc12)NC(N1CCC(CC(F)F)CC1)=O Cc1ncc(C(=O)NCC23CC(CN2C(=O)CSCC(N)=O)C3)c(C(C)C)n1 C1(NC(CCSC)=O)CC(C)N(C(=O)CC2C=CCC2)C1 Cc1cc(C(N2CCCC(NC(C3(F)CCOC3)=O)CC2)=O)c(O)c(C)c1 C(CCCC(=O)N1CCC(C(F)C(=O)NOCC(C)(C)C)C1)OC.C1CC1 c1(C(=O)NCCC(C)NC(c2cc(C)c(C)o2)=O)ncc(C(N)=O)cc1Cl C1(C(=O)NCC(n2cccn2)C)CCCCC1CNC(C1CN(C)C1)=O c1(CC(=O)NCCOC2CCN(C(CNC(CC)=O)=O)C2)ccc(Cl)c(C)c1 C#CCC(C)(C(=O)NCC1CC1(F)F)NC(=O)CCOC1COC1 C1(C(=O)NCC(C(C)C)NC(CC2(C(=O)OC)CCC2)=O)CC2C(C1)C2(C)C C(=O)(CCC(F)(F)C(F)F)N1CC(NC(=O)Cn2ncc3ncccc23)C(O)C1 Cc1cc(C)c(C(=O)NC23CC(CNC(=O)CC(O)c4ccccc4)(C2)C3)o1 C(C(C)(C)CC(=O)N1CC(CF)(NC(=O)CC(C)F)C1)OC N(C(=NCCCF)NC(C(C)C)c1cccs1)C(C1CCCCC1)C C12(CNC(c3[nH]cc(C#N)c3)=O)CC(CO1)N(C(C1CCCC3(CC3)C1)=O)C2 C1(C(=O)NCC2(CNC(C3C4CCCC34)=O)CC2)COc2ccccc2O1 C1(NC(c2cnc(-c3ccco3)s2)=O)CCN(C(C2CSC2)=O)CC12CCC2 c1(OCCC(=O)NCC2N(C(C(C)=C3CC3)=O)CCCC2)cc(Cl)ccc1Cl c1(OC)ccc(C(=O)NCC(C2CC2)NC(=O)CC2CC3(CC3)CO2)c(C)n1 CCCCC(=O)C(=O)NC1CCC(CNC(=O)CCc2ccccc2C(N)=O)C1 Cn1ncc2c1CCC(C(=O)NCC1CCN(C(C3CC=CC3)=O)CC1(F)F)C2 Cc1nc(N2CCC(C)C(NC(=O)C(=O)NCC3CC3)C2C)c(F)c(C)n1 c1(NC(C2CN(C(c3c(Cl)cc(Cl)cc3Cl)=O)CCN2)=O)nccn2c(Br)cnc12 C1(NC(CSCCCC)=O)CCCCN(C(=O)C=Cc2cccnc2C)C1 C1(NC(c2c(SC)n(C)nc2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)CC1F C1(C#N)(C(N(CCN(C(=O)CCCC2CCC2)C(C)C)C)=O)CC2C=CC1C2 N1(CC#C)CCN(NC(=O)C(CCOC)c2ccccc2)CC1 C1(CNC(C(=O)NCC)=O)(NC(=O)Cc2ncccc2C)CC2CCC1CC2 C#CCC(C(=O)NCC(C)(O)CNC(c1cccc(C(N)=O)n1)=O)C1CC1 C=CCCCC(C(=O)N(C)Cc1nnnn1C)NC(=O)CCCOC(C)C CCC(C)C(O)CC(=O)NCCC1CCCN(C(=O)CSc2cccc[n+]2[O-])C1 c1(C(=O)NC2CCN(C(C3C(CC)C3)=O)CC2)coc2c1C(=O)CCC2 C1(C#CC(=O)N2CCCC(N(c3cc(O)nc(O)n3)C)C2)(CC)COC1 C1(N2C(C3CCNC3)CCC2)CCN(CCOCC)CC1.c1cccc(Cl)c1 CN1CCC(C(=O)NC2(C3CCCN3C(c3csc(C(C)(C)C)n3)=O)CC2)CC1 c1(C(=O)NC(COCC)C(N2CCC(C#N)C2)=O)cc(C)nn1C C(C)(CC(C)(C)CO)NC(C1(CCC=C)CN(C(=O)C(C(=O)OCC)OC)C1)=O N1(C(c2c(NC)nccc2)=O)CC2CCC(CNC(=O)CCCOC(C)C)C2C1 C(=O)(CS(=O)(=O)C1CC1)NCC1C(CNC(CN2CCN(C)C(=O)C2)=O)C1 n1(C(C)C)ccc(S(=O)(=O)N2CCC(c3ccccc3Cl)C2)n1 c1(OC)cccc(CNC2(CC(=O)NCCC3CCCC(C)C3)CCC2)n1 N1(C(CC(=C)C)=O)CCC2(CCOC2)C(CNC(C2CCSC2)=O)C1 C1(NC(c2c(OC)scc2)=O)CCCC(NC(c2csnn2)=O)C1 C1(C(C)NC(=O)NCC2(c3ccccc3OC)CCCC2)(OC)CCSCC1 C1(NC(C(C)N(C)C)=O)CC2CC1N(C(=O)CCN1CCC(O)CC1)C2 CCC(CC)C(C(=O)N1CC(N(C)C(C2CCC(C)=C(C)C2)=O)C1)OC C1(NC(c2cnc(CC)nc2)=O)CC2CN(NC(c3nc(CC)cs3)=O)CC2C1 C1(C(N(C(CC(C)C)C)C)=O)CN(C(=O)C(C)c2cccs2)CCO1 c1(C(=O)NCC2CCN(C(C3COC(=O)O3)=O)C2)cnc2ccoc2c1 c1(N(C)Cc2coc(CN(C)C)n2)nc(N2CCC(C)(CO)C2)nc2c1CCC2 c1(C(=O)NCC2CCN(C(c3cn(C)nc3)=O)CC2)cnc2ccccn12 C(=O)(C(C#N)C(C)(C)C)N1CCOCC(CNC(Cc2c(SC)cccc2)=O)C1 N1(C(C(CCC)OC)=O)CC(CNC(c2ccc(NC)cc2Cl)=O)C(C)(C)C1 c1(C(=O)NCC(CN(C(C(C2CCOC2)OC)=O)C)C)cc2c(F)cccc2s1 C1(C(=O)NCc2ccc(C(=O)NC(C(=O)N(C)CC)C)cn2)CC(=O)NC(C)C1 N1(S(C)(=O)=O)CCC(CC(=O)OC(C(F)(F)F)C2CC2(C)C)CC1 C(=O)(C(C)CC(C)(C)C)N1CCN(C(C(C)NC=O)=O)CC1C1CCC1 C1(CC(=O)NC2(C(N3CC(O)C(O)C3)=O)C(C)C2)CC2(CCC2)C1 C1(C(NOC)=O)CC(NC(c2ccsc2C)=O)CO1 N1(C(C(C)OCC)=O)CCCC(C(C)(C)C(=O)NCCC(=O)NCC(C)C)C1 C1(CNC(=O)COCCCF)(CNC(C2CCCCO2)=O)CC12CCC2 N1(C(C2CC(C#N)C2)=O)CCC2(CCCCC2NC(=O)CC(C)(C)C2CC2)C1 c1(C(=O)NC2C(CNC(CC(=O)OC)=O)CC2)ccc(SC)c([N+](=O)[O-])c1 CCC(C(=O)NCC1CC(NC(C2CN(C(N)=O)C2)=O)CCO1)C(F)(F)F N1(C(c2cccc(COC)c2)=O)C2CC1CN(C(c1cnc3sccn13)=O)C2 C(Br)(C(=O)N1CC(CC(C)NC(=O)CCn2cccn2)C1)=C(C)C c1(C(=O)NCC(C2CCC2)NC(C2C(C=C)CC2)=O)ccnc(C2CCC2)c1 C#Cc1cccc(COC(=O)C(C)(C)NC(c2ccccn2)=O)c1 c1(C(=O)NCC2CC(OC)CN2C(=O)CCC2CCC(=O)N2)ccc(N)c(Cl)n1 N1(C(c2ccc(C(N)=O)s2)=O)CC2CN(C(=O)C(c3ccc(Cl)cc3)O)CC2C1 c1(N2CCCC(C)(CNC(C=Cc3c(C)cncc3)=O)C2)nn2cc(C)nc2s1 Cc1nnc(NCCN(C(=O)C=C2CCC(C(C)(C)C)CC2)C)c(C#N)c1C N1(C(C(CC)C#N)=O)CCC2(CC1)COC(CNC(=O)CCc1cc(C)on1)C2 N1(C(C(C)C2CC2)=O)CCCC(CCn2cc(CCn3cc(N)cn3)nn2)CC1 C1(N(C(=O)Cc2nc(Cl)cs2)CC2CC2)CCCN(C(=O)COCC(F)(F)F)C1 CCCCC(O)C(=O)NCC1CC1NC(=O)Cc1ccnc(C(F)(F)F)c1 C#CCC(CC(F)F)NC(C1(C(C)C)CCN(C(c2cc(CO)ccn2)=O)C1)=O CN1CCOC(COC(c2ncc(C3CCOC3)s2)=O)C1 CC(C(=O)OC(=O)Cc1cc2c[nH]nc2cc1Br)C(C)C(C)(C)C.C1C(=O)N1 C1(C(=O)NC2CCN(C(CCc3ccn(C)c3)=O)C2)CC(C)(C)OC1(C)C c1(NCC2N(C(c3cc4cc(F)ccc4s3)=O)CC2)ccc(Br)cc1[N+](=O)[O-] c1(CN(C2CCCN(C(CN3CCC(C)(C)C3)=O)C2)C)ccc2[nH]nc(O)c2c1 C(=O)(C(C)(O)CC(F)F)NCCN(C(=O)CN(C)C)CCOC.C1(=O)CN1 N1(CCC(N2C(CCNC(C3(C)CCCC3)=O)CCC2)=O)CCCCCC1 C1(C(=O)NC2(C3CCCN3C(=O)C(F)n3cccn3)CC2)CC12CCCC2 C1(CC(=O)NC(C=C)CO)CN(C(=O)CC2CC3C=CC2C3)CC12CC2 C1(C(=O)NC(CC)(C)CC)CN(C(c2cc(C3CC3)no2)=O)CCO1 CCCC(C(O)C(=O)N(CC(c1nn[nH]n1)C)C)NC(=O)C(CC(C)C)OC C1(C(=O)NCC#CC(=O)OC)CCCN(C(C2C=CCC2)=O)C1 N1(C(=O)CSc2ccncc2)CC(C2CN(C(C3CC4(CCC4)C3)=O)C2)C1 O=C1CCC(N2CCC(CC(N3CCC(CS(N)(=O)=O)CC3)=O)C2)CN1 C1(C)(COC)CC(NC(C2(OC)CCOCC2)=O)CN1C(=O)C=CC(=O)N(C)C C1(C(=O)NCC(C)CNC(c2cc(F)cc(Cl)c2O)=O)CCC2(CCC2)CC1 C1(C(N(C)Cc2cc(C(C)(C)C)no2)=O)CC2(CCC(=O)CC2)C1 CC1CN(C(C2CCC(=O)N(C3CC3)C2)=O)CCC1NC(C1CCS(=O)(=O)N1)=O C(=O)(C(C(C)C)Sc1nccn1C)NCCC(C)N(C(CN(CCC)C)=O)C CC1CN(Cc2ccc3c(n2)CCC3)c2cccnc2O1 C1(C(=O)NC2(C)CC(O)C2)CC(F)CCN1C(=O)CCc1cncnc1 C(=O)(C1=C2CCN=C2NC=C1)NCC1CN(C(c2c(C)c(C(C)C)ccc2)=O)C1 CCCCCC(O)C(=O)NCCCCCC1CCN(C(=O)C=C(C)Cl)CC1 c1(C(N2CCC(CNC(c3ccc(CC)s3)=O)C2)=O)cc(Cl)n(C)n1 c1(SC)nc(=NC23CCCC2CN(C(c2cn4cc(Cl)cnc4n2)=O)C3)s[nH]1 c1(NC(C2C(C)C2)=O)sc2c(c1C(=O)NC1CC(O)C1)CCCC2 C#CCCCCCC(=O)N(CC(C)(C)CNC(=O)CC1CCCNC1=O)CC c1(C(=O)OC)cccc(C(N2CCC(CCCO)C2)C(=O)NCC2CCC2)c1 C1(CNC(C(C)OCCOC)=O)CCCCN1C(=O)CC1CCC1(C)C N12CCC(CC1)c1nc(cs1)C(=O)N(C)CC2=O.C=CC(=O)OCC C1(NC(c2c(C(C)C)onc2)=O)CCCC(NC(c2occc2F)=O)C1 c1(C(N2CCN(C(CC(=C=C)C)=O)C3C2C3)=O)cc2c(cc1F)OCC(=O)N2 CCC(CC)CC(F)C(=O)NC(CC(N1CCC(C)C(F)(F)C1)=O)C(C)C C(C(C)C(=O)NCC(C)CNC(=O)CNC(C1CCCC1)=O)SC C(=O)(CCC(CC)NC(=O)CCc1cncs1)N(CC(=O)NCC)CC C1(NC(C(C(=O)O)n2cc(C3C(C)(C)C3(C)C)nn2)=O)Cc2ccc(Br)cc2C1 C1(C(=O)NCc2cn(C3C4CC5C(C4)C35)nn2)CCC2(CCOC2)O1 c1(CC(=O)NC2CC(CC(N3CC(CC(C#C)C)C3)=O)C2)nonc1C C#CC1(C(=O)N(C)CC2CC23CC3)CN(C(=O)CC)C1 Cc1nn(C)c(CNc2cc(OC(C)C(=O)O)cc(F)c2)c1I C1(c2nnccc2)CCN(N2CCC3(C2)CC3(F)F)CC1 N1(C(c2cc[nH]c2C2CC2)=O)CC2CCN(C(c3n[nH]c4c3COCC4)=O)C2C1 N1(C(c2c(C)cc[nH]2)=O)CCC(CN(C(C2CC2CC(C)C)=O)C2CC2)CC1 c1(C(=O)OC)conc1CC1CN(C(=O)NCC(C)C)C1 c1(C(=O)NCC(N(C(C=CC2N(C)CCC2)=O)C)C2CC2)cc2sc(Cl)cc2[nH]1 C(=O)(CC(O)CC(C)(C)C)NCC(CN(C(=O)C(CCOC)OC(C)=O)C(C)CCN)(C)C C1(CCNC(CSc2nc(C)[nH]n2)=O)CSCCN1C(=O)CN(C)C(N)=O C(=O)(CCCCC(=O)N(C(C)(C)CC(=O)N1CC=CC(OC)C1)C)OC c1(C(=O)NCC(C)(CO)NC(C(c2cnn(C)c2)C)=O)cc2c(s1)CCC2 C(CN=c1[nH]nc(C(F)F)s1)NC(NC1CCCC(C)C1)=S C1(NC(C2(CC)CC(C)C2)=O)CCOC(CC(=O)OC)C1 n1(CC)cnc2c(NCCC3CC(C)(C)C3)[nH]c(=NCCC(C)S(C)=O)nc12 C1(NC(Cc2cccc(OC)c2F)=O)COC2(C1)CN(C(c1cccnn1)=O)C2 Cn1c(O)nc2ccc(NC(N3CC(F)(F)C4(CCCC4)C3)=O)cc12 C1(CC(=O)NC(C2(O)CN(C(CCC(=C)C)=O)C2)C)CCC(F)(F)CC1 c1(C(N(CCCCCC)CCNC(C2CCC2C)=O)=O)cnc(C)cn1 C1(NC(C=CC=CCC)=O)CCN(C(c2cn(C3CCOCC3)nn2)=O)C1 C(=O)(C(CN=c1ccc(S(C)(=O)=O)c[nH]1)OCCN(C)C)NC(C)=O N1(C(C(C(C)C)O)=O)CCN(C(c2cccc(CCO)c2)=O)C(C#N)C1 C(=O)(C(CC(C)C)NC(c1cn(C(C)C)cn1)=O)N(C(C1CCC1)C)CC CC(CC1=CCCCC1)NC(C1(NC(=O)CCN2CCCCC2)CC(F)C1)=O C1(NC(COCCOC)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CC1F CC(C(C)(C)C)=CC(N1CC(=C(F)CNC(=O)C(F)(F)C2(O)CCC2)C1)=O c1(CN=C(NCC)NCC2(CO)COCC3CCCN23)cnc2c(F)cccc2c1 N1(C(=O)Cc2cc(F)cc(Br)c2)CCN(C(c2cc(O)ccc2F)=O)C(C2CC2)C1 CC1CC(=O)NCC1C(=O)NCC(C)(C)C(=O)NCC1C2CCCOC12 c1(C(N2C(=O)NC(C(C)C)C2=O)C)cc2ccccc2o1 C#Cc1ncc(F)cc1NC(N1CCC(CCC)(CO)C1)=O CC1CC(NC(C2(CNC(=O)Cc3ccon3)CC2)=O)CC(C)(C)C1 C=CC(C)(CC)C(=O)N(CCCCN(C)C(c1c(OC)cccc1F)=O)C Cc1ccc(C=CC(=O)NCCCCC(=O)NCC2(O)CC2)o1 c1(C(N2CC(OCCNC(=O)CC3CCCOCC3)C2)=O)cccc2occc12 c1(OC)ccnc(C(=O)NCC(C)(C)NC(c2n[nH]c(C)c2O)=O)c1F C1(NC(CCCNC(C(C)(C)C)=O)=O)CC2CC(NC(=O)CN3CC=CC3)C2C1 c1(C(C2N(C(C)=O)CCC2)NC(=O)Nc2nn[nH]c2C(C)C)cccc(Cl)c1 N1(C(C2CCOC2)=O)CCCC2CN(C(C3(C4CCCO4)CCC3)=O)CCC12 C1(C(N(CCOCC)CC)=O)CC12CCN(C(=O)C(C)CC(F)F)CC2 CC1(C)c2[nH][nH]c(=NC(=O)c3cn[nH]c3)c2CN1Cc1ccnc(F)c1Cl c1(C(N2C(C(=O)NCC3CC3C3CCC3)CSC2)=O)cccc(F)c1 N1(C(C2N(C(c3c(CC)cco3)=O)CCC2CC)=O)CC(O)C(O)C1CO C1(C)(NC(c2cccc(C)n2)=O)CCCN(C(=O)COc2cccc(Cl)c2)C1 C1(NC(C2(C#C)CCCC2)=O)CN(C(=O)CC(=C)Br)C(CC)(CC)C1 C12(N(C(=O)CSc3nncs3)C)CCCC1N(C(=O)CCCc1csc(=N)[nH]1)CC2 CCCCC(CCCC)C(=O)N1CC2(COC(CNC(=O)C(C)CC(F)F)C2)C1 N1(C(N2C3CCC2CC(NCc2c(C)ncs2)C3)=O)CCCC2CN(C)CCC12 c1(C(=O)NC2C3CC(O)C2N(C(C2CC(O)C2)=O)C3)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NCC2C(NC(C3C(C=C)OCCC3)=O)C2)[nH]c2ccccc2c1C C1(NC(=O)CN(C(C2CCC(=O)N2)=O)C2CC2)CCc2nncn2C1 N1(CCN(C(=O)C(=O)N(C)C)CCCC)CCCC1CSC C1(NC(c2n(CC#C)ccc2)=O)CCN(C(c2cc(C(C)C)nn2C)=O)C(C)C1 C1(C(N)=O)(C(=O)NCCC2(NC(C3CC3Cl)=O)CC2)CC1 c1(C(=O)NCC23N(C(c4ccc(C)c(C)n4)=O)CC(C2)C3)c(C)nc2sccn12 N1(C(C(CCC#C)O)=O)C2CCC1CC(CNC(C1(CC3CC3)CC1)=O)C2 c1(OC)cccc(C)c1C(=O)NC1CC1CNC(=O)C(C(C)(C)C)OC C1(C(N2CC(CNC(c3ccc(C(F)F)s3)=O)C2)=O)CCCC1C1CC1 c1(C(=O)NCc2c(Cn3cc(CSC)nn3)nco2)cc2cnn(C)c2s1 c1(C(=O)NCC2(CNC(C3C(C)CC(=O)N3)=O)CCCC2)cnn2c1N(C)CC2 CCCS(=O)(=O)CC(=O)N(CCCNC(c1cccc2cncn12)=O)CCO CC(C)CC(C(=O)N1CC2CCN(C(=O)CCc3ccncc3)C2C1)C(C)C N1(C(CNC(C)=O)=O)CC2(CCC(NC(c3nn(C)c4c3CCC4)=O)C2)C1 N1(C(Cc2c(C)n[nH]c2)=O)CC(F)CC1CC(=O)NCC1CCOC1C N1(C(CCN(C)CCO)=O)C(CC(N2CC(C3CC3)C2C2CC2)=O)C2CCCC12 C1(C(C)(C)NC(C2CCCC2O)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1 C1(C(=O)NC2(CCCNC(c3cn(C(C)C)nn3)=O)CC2)CC(C)CC(=O)N1 N1(C(c2cc(C)no2)=O)CC2(CC(NC(=O)CCc3cnn[nH]3)CO2)C1 CCC(C)CCCC(=O)NCC(O)CCNC(c1cscc1C#N)=O c1(C(N2C(CNC(C(CC=CCC)C)=O)CCC2)=O)cnc(C)[nH]c1=N N1(CCOc2ccc(OC)cc2)CCCC2(CCCCC2O)C1 CCCCCCC(=O)N1CCCC1(C)C(=O)NCCCC(C)(C)CO N1(C(C(C(C)(C)C)C(Cn2cc(C(CC)(C)O)nn2)=O)=O)CC2C(C1)CS(=O)(=O)C2 C1(C(N(CC(C)N(C)C(c2cc(C(C)(C)C)no2)=O)C)=O)CN2CCCN1CC2 N1(C(C(C)=C2CC2)=O)CC(C)CN(C(c2cnc3n2CCCC3)=O)C(C)C1 c1(CCCC(=O)NC(c2ccc(C)cc2)COC)ccc(Cl)cc1 Cc1ccc(CNc2ccc3c(c2)CN(C2CCC2)C3)c([N+](=O)[O-])c1 Cc1cc(Cl)ncc1NC(C1CCCC1NCc1cccc(C#N)c1)=O C1(N=[N+]=[N-])(C(=O)NCCCCCCC#C)CCN(C(C2CC(=O)NC2(C)C)=O)C1 C(C(N=[N+]=[N-])C(=O)NCC1(OC)CN(C(=O)C(C)C(=O)OC)C1)OCC N1(C(C(n2cc(-c3cc(OC)ns3)nn2)C)=O)CCCC(CN)C1 N1(C(C=CC)=O)CCC2(CC1)COC(CNC(=O)CC(O)Cc1ccccc1)C2 C1(C(=O)NC2(CC)CCC2)CCCN1C(=O)CCN(C)CCO C1(CCN(C(c2c(OC)c[nH]n2)=O)C)CCCCN1C(=O)C(O)Cn1cncn1 c1(N(C(CC2CCN(C(=O)OC(C)(C)C)C2)=O)CCC#N)cnc(N)c(Br)c1 N1(C(c2c(CC)nn[nH]2)=O)CCCCCC1CC(=O)NC(C)CC(C)(C)OC CC1(C)CCc2c1n[nH]c2C(=O)N(C1CCCCC1)C(=O)CC1CCOC1.C(C#N)N N1(C(c2cc(C)c(C(F)F)nc2)=O)CCN(C(=O)C2=CCOC2)C2CCCCC12 C#Cc1cccc(CC(N2CC(OC)CC2(C)CNC(=O)CCC)=O)c1 N1(C(CCC2C(C)C2)=O)CC(C)CN(C(c2ccccc2SCCO)=O)CC1C c1(C(C)C(=O)NCC2CCC2C(=O)NCCCC2CCC2)ccn(C)n1 C(c1cscn1)=CC(=O)NC1CC(CNC(C2OCCCO2)=O)C1 C1(NC(C(n2cc(-c3ncccc3N)nn2)C)=O)CC(N(C)C)C1(C)C O=C(CCCCC(F)F)N1CCC2CN(C(=O)C(F)C(F)(F)F)C2C1 N1(C(CSCCOC)=O)CC(NC(=O)CCc2nc(C)c(C)[nH]2)C(C2CC2)C1 c1(N(CCCO)C(c2ncc(C)s2)C2CC2)cnc2ncccc2c1 c1(C(=O)NC(CCNC(CC(C=C)CC)=O)C)nc(S(C)(=O)=O)n2ccccc12 Cn1ncc(C(=O)NCCCNC(C2(C)CC(C#N)C2)=O)c1C(C)(F)F c1(C(=O)NC2CN(C(CNC(=O)NC)=O)CC2C)cc(Cl)c(F)cc1C C1(C(=O)NC2C(NC(c3c(C)ncn3O)=O)COCC2)CCc2ccnn2C1 c1(CC(N2CCCC(N(C(C)=O)CCO)CC2)=O)ccc(S(=O)(=O)N(C)C)cc1 C(C(C(=O)NC(C1CCCC1)CO)NC(=O)CC1CCCC1O)OC N1(C(C(C)OCC=C)=O)CC2CC(NC(=O)CCCCC(C)C)CC(C2)C1 c1(C(N(CC(C)NC(c2c(C)cc(C)nc2O)=O)C)=O)ccc2c(C)noc2c1 C1(C(N2CCC(C)(F)C2)=O)CCCN1NC(=O)CC1CC(F)(F)C1 Cc1onc(CC(=O)N(C2CCCC(NC(=O)Cc3cnnn3C)C2)C)c1C#N c1(C(N(C2C3CN(C(C4CCOC4)=O)CC23)C)=O)cccc2c1OCCN2 c1(CNC(COC2(C)CN(C(c3cc(C)sc3)=O)C2)=O)cncc(O)c1 NS(=O)(=O)N1CCCC(C(N2CC3CCC(C2)N3C(C2(CO)CCCO2)=O)=O)C1 c1(C(N2C(C(N3CCC(N4CCCCC4)C3)=O)CCC2)=O)c(I)ccnc1F C(C)(C(C)(C)C)=CC(=O)NC(CN(C(c1ccnn1C)=O)CC)C c1(C2C(C(N(CC(CCC)O)C)=O)C2)cc(F)ccc1F c1(OCC)ccc(C(=O)NC2CCCN(C)C2)cc1[N+](=O)[O-] c1(C(C)NC(C2CC2C(C)NC(C2CC(C)(C)C2)=O)=O)nnc(O)o1 C1(CN(C(=O)CSc2ccccc2)C)CC(O)(CNC(=O)CC2CC(F)C2)C1 c1(C(N(C(CNC(C2(C(=O)NC)CC2)=O)C)C)=O)cc(C(F)F)ccn1 Cc1sccc1C(=O)NCC(n1cc(CN2CCSCC2)nn1)C c1(NC(C2CCC(C(=O)O)N2)=O)c(Cl)c(Cl)cc(Cl)c1Cl C(=O)(C(C)(C)C(=O)NCCCC(C)NC(=O)CCN1CCSC(C)(C)C1)OC c1(C(N2C(CNC(CCc3c(C)n(C)nc3)=O)CC2)=O)[nH]nc([N+](=O)[O-])c1Cl C(CNC(=O)CC1(c2ccccc2)CC1)(CC(C)C)NC(CC=CC=C)=O c1(C(=O)NCC2C(NC(c3c(CCC)occ3)=O)COC2)c(C)ccnc1N c1(C(=O)NCC2(OC)CN(C(=O)C(N3CCC(C)C3)=O)C2)cn(C)c(=O)c(C)n1 c1(C(N(C)CC2CCCCN2C(C2CCC2(C)C)=O)=O)ccc2[nH]c(=N)sc2c1 c1(CC(=O)NC(C)(C)COCCCNC(c2ccoc2)=O)cccc(F)c1Cl c1(CCC(=O)NC2(CF)CCN(C(C(C(C)C)O)=O)C2)ccc2c(c1)OCCO2 c1(C(N2CCC(C(C)(C)NC(C3CC(C)C3)=O)C2)=O)cccc2scnc12 C1(O)(C(C)NC(C(CC)N(C)C)=O)CCN(C(C2(CSC)CCC2)=O)C1 C1(C(N2CCC(CC(N)=O)CC23CC3)=O)CCCC2(CCOCC2)O1 C(N=c1[nH]cnc(Cl)c1C(C)C)C1CCCC(NC(c2cc(CC)n(C)n2)=O)C1 c1(CNC(c2n(CC(=C)C)nnn2)c2coc(C)n2)cc(O)nc2ccccc12 C(=O)(CC(C)C(=O)NCC1CC2(C1)CN(C(=O)C(C1CCCCC1)C)C2)OC N1(C(C2(CNC(C(C=CC)O)=O)CC3(CC3)C2)=O)CC2CCC2(OC)C1 c1(C(=O)NCC2CC(C)N(C(c3ccoc3)=O)C2)ccc2cnoc2c1 C1(CC(=O)NC2CC(N(C(CCSCCCC)=O)C)C2)COCC(C)(C)O1 C#Cc1ccc(CC(N2CCN(C(C3CCC(=O)O3)=O)C(C3CC3)C2)=O)cc1 C1(C(N2CC3(CC(CNC(COC(CC)(C)C)=O)C3)C2)=O)OC(C)(C)OC1(C)C N1(CC(N2CCC(NC(c3cnc(CC)s3)=O)C2)=O)CCC(C)(C)C1 c1(C(N2CCN(C(C3(C)C(CC)CCC3)=O)CC2)=O)cnc2cc[nH]c2c1 c1(OC)ccnc(NCC2CCCN2C(C2CC(F)(CO)C2)=O)n1 S(=O)(=O)(CCC(=O)NC1CS(=O)(=O)CC1NC(=O)C1=CCCC1)NC C(=O)(CCCCC(N)=O)NC(CC(=O)NCC(CC)(C)C(N)=O)C1CC1 C1(C(=O)NC(c2cnnn2C)C)CCc2nnc(Br)n2C1 N1(c2c(NC3CCCC(F)C3)cccc2)CCc2ccc(Cl)cc21 c1(CCNC(CC(C)(C)OC(C2C(CCC)C2)=O)=O)ccc(CC)cc1 CC(=O)CCCC(=O)NCC(C)N(C(=O)C(Cc1ccccc1)n1cnnn1)C C1(CCNC(C(C)O)=O)CCCN1CC.C1(NC(=O)C)CCCC1 CC1(C(=O)NCC(O)CNC(c2ccn3ccsc23)=O)CCC(F)(F)C1 CC1(C)CC(CC(N2CC=CCC2)=O)N(C(=O)C#CC2CC2)C1 c1(N(CC(N2CC(C)(NC(=O)C(F)(F)CC3CCCO3)C2)=O)C)ccc(Cl)cc1 N1(C(c2ccc3c[nH]nc3c2)=O)CCC2CCCN(c3cc(F)ncn3)C2C1 C(=O)(C(C)(O)CC(C)C)NCCC(C)(C)NC(c1c(CCC)[nH]cc1)=O C(=O)(C1CCCn2c(CC)nnc21)NCCC(=C)CNC(=O)CCCCN(C)C CC(C)CC(C(=O)NCC(O)CNC(c1c(F)cccc1Br)=O)C(C)C N1(C(c2nc(C)c(CC3CCCC3)s2)=O)CC(N=[N+]=[N-])C(S(C)(=O)=O)C1 c1(OC)ccc(C(=O)N(C(C)CN(C(=O)CCCc2cc(C)no2)C)C)cc1 c1(C(=O)NCC2(CNC(C3(CF)CC3(F)F)=O)CC2)cc2n(c1)CCOC2 C1(CC(=O)NC2(CCC(=O)NCC3CC(F)(F)C3)CCCC2)COCCO1 c1(OC)ccc(S(=O)(=O)CCC(=O)N2CC3C(NC(=O)C(C)C(C)O)C3C2)cc1 CC(=O)NNC(=O)C(C)SCC1CNC(=O)CO1 C(C)(CNC(=O)CC(C)Sc1ccc(F)cc1)(CC(C)C)Nc1ncc(C)cn1 C(=O)(C(F)(CNC(=O)CC1CCOC1(C)C)C(C)C)N(C1(O)CCC1)CC C1(NC(C(COCC)C)=O)(CF)CCN(C(c2ccoc2Cl)=O)C1 c1(C(=O)NC(CC(C)NC(C2CSCCS2)=O)C)ccnc(-n2cccn2)c1 C(CN=c1[nH]ccc(=NC2CC3(C=CCO3)C2)[nH]1)c1c(C)cc(Br)cc1 c1(C(=O)Nc2n(CCN(C3CCCCC3)C)ncc2)cc(C#N)no1 C1(C(N2C(CC)CC2)=O)CCN(C(=O)COCCCF)CC1O C12(CNC(c3c(CCC)occ3)=O)CC(CN1C(C1CC3CC3C1)=O)C2 N#Cc1cncnc1C(=O)NCCOCCNC(c1cccc(=O)o1)=O C(=O)(N(CCC(=O)OC)OC)C1N(C(c2ccoc2CC)=O)CCC(=C)C1 c1(C(N(C)CC2CN(C(c3cncc(C)c3)=O)C2)=O)cc2c(=O)[nH]ccn2n1 N1(C(C(C(C)C)N(C)C)=O)CCCN(CCCCNC(c2ccsc2)=O)CC1 O=C(C1CCc2c[nH]nc21)NCC1CCCCN(C(=O)C2CCc3c[nH]nc32)C1 CC1CCc2ncc(C(=O)NCC3C4CN(C(=O)CCc5cn[nH]c5)CC34)n2C1 C1(NC(C2C(C)CC(C)O2)=O)CCN(C(c2ccc(O)c(F)c2F)=O)CC1(C)C c1(CN(C(=O)Cc2c[nH]nc2O)C)ccccc1CNC(c1ccoc1)=O Cc1cc(C(=O)NC2(CNC(c3csc4nnsc34)=O)CCOCC2)nc(C)n1 c1(C(=O)NCC(C)(C2CCC2)NC(CCOC)=O)ccc(C)c(OC)c1 CC1COC(C(=O)NCC#CCNC(c2cnn(Cc3ccccc3)c2)=O)C1 C(=O)(N(CCC(=O)N1CC(O)CC1C1CC1)OC)C1(CC)CCOCC1 c1(OC)cccc(O)c1CNCC1CCCN(C(=O)C=CC(C)C)C1 C1(NC(CCN(C)CC)=O)CC2CN(C(C3(C4CC4)CC3)=O)CCN2C1=O c1(CC(=O)N(CCN(C(C2CC2F)=O)CC)CC)ccsc1Br C1(CC)CN(C(=O)Cc2ccon2)CCC1NC(=O)CC1CCC2(CC1)CC2 N1(C(Cc2c(C)nc[nH]2)=O)CC2(NC(=O)Cc3ccccc3Cl)CC1C2 Cc1cc(CC(C(=O)OCC(F)C2CCC2)NC(=O)OC(C)(C)C)nn1C C1(NC(c2cc(C)on2)=O)CS(=O)(=O)CC1NC(=O)COC1(C)CCC1 C(=O)(C(O)CC(N)=O)NC(C)CC1CN(C(=O)Cn2ccc(C3CC3)n2)C1 C(=O)(CC(C)(C)N(C)C)NC1(CC=C)CN(C(c2ccc(SC)o2)=O)C1 c1(OC(C)C)ccc(Cl)cc1NC(=O)CNC1CC1(c1cccc(Br)c1)F N1(C(C(C(C)C)NC(CCCC#C)=O)=O)CCC(NC(C)=O)C(C(N)=O)C1 C1(CC(=O)N(CCNC(=O)CCC2CCCN(C)C2)CC)OCCCC1(C)C C1(N(C(=O)CC(C)(C)F)C)CC2CCC(C1)N2C(C1(N(C)C)CCCC1)=O N1(C(CC=CCC)=O)CCC2CCN(C(c3cc(C)nc(O)c3)=O)CC12 c1(OC)ccccc1C1(C(N2CCOC(CCCO)C2)=O)CCC1 C(c1cn(C)nn1)=CC(=O)NCCCN(C(C1N(CC)CC1)=O)CC1CCCC1 C1(C(NOCC=C)=O)CC12CCN(C(=O)C(C)(C)CC(F)F)CC2 CCCC(F)(F)C(=O)NC1CC(C)CN(C(c2ccncc2NC)=O)C1 C(=O)(N=c1cc(C(C)NC(C(COCCOC)C(C)(C)C)=O)n(C)[nH]1)c1cn(C)nn1 C1(C(=O)NC(CC=C)CNC(=O)CSc2nnnn2C2CC2)CCN(CC)CC1 N1(CC(=O)NC2CC(C)(C)N(C(=O)CC3(O)CC3)C2)C(=O)C2C3C=CC(C3)C2C1=O c1(NC(C2CC(C)CN2Cc2ccc(F)cc2)=O)ccc(Cl)nc1C#N CC1(CC(=O)NC2CC(CO)N(C(c3ccc(C(N)=O)o3)=O)C2)CCS(=O)(=O)N1 c1(-c2cc(C(=O)NC(C(C)NC(=O)Cc3ccco3)C)no2)ccccc1O Cn1nncc1C(=O)NCCOC1CCN(C(=O)CCNC(N)=O)C1 c1(OC)c(C(=O)NC2CC(NC3CC(=O)NC3=O)C2)c(C)nn1C N1(C(C2CCC(=C)CC2)=O)CC2(COC(CNC(=O)C(CC3CCC3)OC)C2)C1 C=CCCC(C)(O)c1nc(-c2ccccc2)nn1C12CC(C1)C2 N1(C(c2cn(CC(C)NC(=O)CC)nn2)C)CCC(O)(CO)C1 N1(C(c2ccc(C#N)o2)=O)Cc2ccc(CNC(=O)C(F)=C3CCC3)cc2C1 c1(CC)nc(C)c(C(N2CCCC(CNC(=O)C(C)SC(F)(F)F)C2)=O)s1 N1(C(c2ncn(C)c2)=O)CCC2(CCC2)C(CNC(C2(C)CCOC2)=O)C1 C(=O)(C1=NOC2COCC12)NCC1N(C(Cc2c(F)ccc(OC)c2)=O)CC1 C(CCCC(C)(C)C(=O)NNC(=O)CSc1cccc(F)c1)NC(C(C=C)O)=O c1(NC(C(C)(C)CNCCCOCCN)=O)ccc(F)cc1F C12(CNC(c3oc4ccc(C)nc4c3)=O)CN(C(=O)CCF)CC1CS(=O)(=O)C2 N1(C(c2nnc(C)o2)=O)CC(CC2(n3cc(C4CC4)nn3)CCOCC2)OC(C)C1 N1(C(CC=CCC)=O)CC(O)CC1CNC(C1(OC)CCOC1)=O n1(CCCNC(=O)Nc2ccc(N(C(C)=O)CC)cc2)cc(C#N)c(O)nc1=O N1(C(C2(OC)CCOC2)=O)C(C(=O)NCC(C)C(=O)OC)C2CC(O)C1C2 C1(CNC(c2ccc(C(C)=O)o2)=O)CC(C)N(C(=O)COC2CCOC2)C1 C1(CNC(CC2N(C(C3C(C(C)(C)C)C3)=O)CC(F)C2)=O)CC2(CCOC2)C1 C#Cc1cccc(CNC(=O)CCN(C(=O)CCn2ccnc2)C)c1 Cc1cccc(C(N2CC(CCNC(C3CCCN3C(C)C)=O)C(C)C2)=O)c1C C1(CC=C)(NC(C2CCOCC2)=O)CC2CCC(C1)N2C(C1(C)CCCO1)=O Cc1cnc(N2CCCC(CC(=O)NCC3CCN(C)C3=O)C2)nc1C C(=O)(CC1=CCCCC1)NCCC1CC(NC(C(c2c(OC)cccc2)O)=O)C1 N1(C(C)=O)CCCC1(C)C(N1CC2CC2(NC(=O)C(C)(C)c2cccnc2)C1)=O CCC(CC)CC(=O)NC(C1CCN(C(C2(CC)CCCC2)=O)CC1)C Cc1cc(C(=O)NC(C2CN(C(C3(c4ccno4)CC3)=O)CCO2)C)nc(O)c1 Cn1c(C(=O)N(C2(C(=O)NCCC3NC(=O)NC3=O)CCC2)C2CC2)nnc1S N1(C(C2CCC(CNC(c3c(C(C)C)n[nH]c3)=O)C2)=O)CCC2(CCN(C)C2)C1 c1(C(N(CCCNC(c2ccc(SC)s2)=O)CC)=O)ccc(F)c(F)c1N N1(C(CCOCCOCC)=O)CCC(C(C)NC(c2ccc(NC)cc2)=O)CC1 C1(C2CCOCC2)(C(=O)NC2CN(C(CS(C)(=O)=O)=O)CC3C2C3)CC1(F)F N1(C(Cn2c(C)ncc2)=O)CCC(F)(F)C(NCc2cc(I)ccc2Br)C1 c1(OC)cccnc1N1CCC(N(C)C(=O)NC(c2ccccc2F)C)C1 C(CCC(=O)NCc1ccc(C(=O)NC(C)C(C)SC)o1)=CCC=C Cc1nc(N(C)CC2CN(C(=O)C(C)OC3COC3)CCO2)ccc1[N+](=O)[O-] c1(OC)cnc(C(N2CC(CO)(NC(C3(C)CCNC3=O)=O)C2)=O)c(OC)n1 N1(C(C(C)SCCCC)=O)CCN(C(=O)C(c2ccc(F)c(F)c2)C)C(C)C1 C(C(F)(F)CCC(=O)OC)n1cc(C(=O)NCC(c2ccccn2)N(C)C)nn1 c1(C(=O)NCC23CC(CO2)N(C(C2(CO)CCCO2)=O)C3)cccc2nncn12 Cc1oc2ncnc(O)c2c1C(=O)NCC1CC(NC(c2cccnc2S)=O)C1 N1(C(CN(C(C)C)C)=O)CCCC2(C1)CN(C(C1CCCSC1)=O)CCO2 Cn1ccc2nc(N(c3ncnc4[nH]ccc34)CC3CC4(C3)CC(N)C4)nc(Cl)c12 N1(C(C2(OCC)CC2)=O)CCCC(N(C(=O)C2=C(C)OC2)C)CC1 CC1CN(C(c2cc3ccccc3o2)=O)CCCN1Cc1ccncc1O C1(CNC(c2occ(C)c2)=O)CN(C(=O)C(F)(F)c2ncccn2)CC1(C)C C1(C(N2C(C3(O)CN(C(=O)C=Cc4ccsc4)C3)CCC2)=O)CCCC(O)C1 C1(C(C)O)CCN1C(=O)CC1(NC(c2cnsn2)=O)CC1 c1(C(N2CCC(NC(COCCC=C)=O)C(F)C2)=O)oc2c(Cl)cccc2c1C C(=O)(C1=C(C)OCCS1)NCC(CC(=O)NCC(C(=O)OC)OC)C C1(O)(CCNC(C2OCC(C)(C)C2)=O)CCN(c2ccnc(C(C)(C)C)n2)CC1 C=CCC(F)(F)C(=O)N1CC(CNC(=O)CCC2CC2(F)F)C(C)C1 C(C1CSc2ccccc21)NC(c1cc(C(C)(C)C)c(O)cc1)=O C12(NC(=O)CNC(=NC)NCC#C)COCC(C1)C2 c1(OC)ncc(C(=O)NC2(C)CCN(C(=O)C(C)c3cncs3)C2)cn1 N1(C(C2(C)C(C)CN(C(C(COC)N(C)C)=O)C2)=O)CCC2(CCC2)C(O)C1 CC1(C)OCC(CCC(=O)NCC2CC(F)(c3ccccc3)C2)O1 C(=O)(C(F)CCCCCC)NCC1N(C(c2ccc(C#C)c(C)c2)=O)CC(F)C1 c1(C(=O)NCCCOCCNC(C2(OC)CCC2)=O)cc(-c2ccco2)nn1C CCC(C)C(O)C(=O)NC1(C(N2CC(C)CCC2CC)=O)CC(O)C1 C#Cc1ccc(C(N2CCCC2CCC(=O)NCc2conc2C(F)(F)F)=O)o1 c1(C(=O)NCC2CCC(NC(c3c(N)cc(Cl)cc3)=O)C2)cnc2[nH]cnc2c1 c1(N(C2CN(C(C3CC=CCC3)=O)C2)C)ncc2ccc(Br)cc2n1 C1(C(C)NC(c2cc(C)oc2)=O)CN(C(C2(c3ccno3)CC2)=O)CCO1 c1(C2(C(N3CCC(CN=[N+]=[N-])C3)=O)CCC2)ccc(Cl)cc1 c1(CN=C(NC(COC)C2CC2)NC(c2ccncc2Cl)C)ccc(F)cc1O N1(C(C(CNC(C)=O)CN=c2cc[nH]c(C#N)n2)=O)CCc2c(cnc(C)c2C#N)C1 c1(CC(N2CC3C(NC(=O)C4=CCC4)(CC3)C2)=O)cc2cc(Cl)ccc2[nH]1 S(=O)(=O)(c1c(C)nc2sc(C)cn12)N1C(c2ccc(C)cc2)CCCC1 N1(C(c2c(CNC(C(C)NC(=O)NC)=O)noc2)=O)CCC12CCSCC2 N1(C(C2(F)CCN(C(c3cn(CC=C)nc3)=O)C2)=O)CC(C)OC(C)(C)C1 C1(C(=O)OCC)CCOC1NC(C1CN(C(=O)C(c2cncn2C)C2CC2)C1)=O C(C(CC(C)C)C(=O)N1CCCC1C1CCCC1)NC(CCCC)=O C#CCCCC(C)C(=O)N1CC=CC(NC(C2(O)CC(C)(C)C2)=O)C1 N1(C(c2cc(C)oc2)=O)CC2CC(C1)N(C(=O)CNc1ncccn1)C2 C(CC(C(=O)NCCCN(C)C(C)=O)NC(c1n[nH]c(C)c1C)=O)SC C1(NC(=O)C=CC=C(Cl)Cl)CC2CC(NC(c3cncc(F)c3Cl)=O)C2C1 N1(C(C2(C=C)CCOCC2)=O)CC(C)N(C(=O)OC(C)(C)C)C(C)C1 C1(CNC(C2(C(C)C)CC2)=O)CC(C(=O)NC(C)Cc2cccs2)=NO1 C1(CN(C(=O)C(C)(C)CSC)CC)CCN(C(=O)C(c2ccn(C)n2)C)CC1 c1(C(N2CC(CO)OCC2C)C(=O)NC)cc(OC)cc(OC)c1C C1(C(=O)NC(C(=O)Nc2cn(CCOC)nc2)CCSC)CC(=O)NC1(C)C C1(N(C(C=CC(=O)N(C)C)=O)CCO)CCN(C(=O)C=CC(=O)N(C)C)C1 C1(C)(CC(=O)N(C)CC2CCCCN2C(C2(CF)CC2)=O)CCS(=O)(=O)N1 c1(OCC)ccc(C(=O)NC(CN(C(c2ncncc2F)=O)CC)CC)cc1 c1(C(=O)NCC(=O)N(CCN(C(=O)OC)C)C)c(OC)cncc1Br c1(NCC(c2ccc(OCCC(C)C)cc2)C)nc2ccc(O)cc2s1 C(=O)(C(C)CC(C)C(C)=O)NC1CC(CCC(=O)NC(CC#CC)CO)C1 C(CN(C)N1CCNc2c(C(N)=O)cccc2C1)c1ccc(OC)cc1 N1(C(C)=O)CCCC(CC(=O)NC(C)CCC=C(C)C)C1 c1(CC(C)C)nnc(-c2ccncc2Cl)n1CCC#N N1(C(C(C)CC(F)F)=O)CCOCC(C)(CNC(c2cccc([N+](=O)[O-])c2)=O)C1 C(=O)(C(C)(CSC)NC(=O)C(C)CCOC)NCC(CC)n1cccn1 C1(CNC(c2c(C)occ2)=O)CN(C(C2CCC3CC3CC2)=O)CC12CCC2 C1(CC(N2C(CN(C(c3ccc(O)nc3)=O)CC)CCC2)=O)OCCC1(C)C C1(CNC(C2(CCCC)CC2)=O)CCC(C)N(C(c2nn[nH]c2CC)=O)C1 C1(CNC(C=COCC)=O)C(C2CC2)CCN1C(c1sccc1OCC)=O C1(NCC(=O)N(CCCNC(c2cccc(N(C)C)n2)=O)C(C)=O)CCS(=O)(=O)C1 CC1CN(C(=O)C(c2ccccc2Cl)O)CC1NC(c1cnc(=NC)[nH]c1)=O C(=O)(C(C)(C)C(C)(F)F)NC1CC2CC(NC(C3CCC(C)CC3)=O)C1C2 C=CCC(C)(C)CC(=O)NC1COC2(CNC(C3CCOC3(C)C)=O)CC1C2 c1(C(=O)NC2COCC2NC(C2(F)CCC2)=O)ccc2c(c1)NCCC(=O)N2 C(=O)(C(c1ccccc1)=Cc1ccccc1)NC1C(NC(COCC#C)=O)CC1 c1(C(C)C)nc(NCCCF)cc(N(C(C)CCN2CCOCC2)C)n1 Cc1ccc(CCCNC(c2n[nH]c3c2CCC3)=O)c(O)c1 C1(C(=O)NC(C(=O)NC(C=C)COC)C2(C)CC2)CCCCCC1 c1(NC)snc(C)c1C(=O)NCC1CC(CNC(C2CC3CCC3C2)=O)CO1 c1(NC(=O)Nc2ccn(C3CCN(c4nccs4)CC3)n2)ccc2c(c1)OCO2 C12(C(=O)NCC3(C(N)=O)CN(C(C(C(=O)OC)(C)C)=O)C3)CCC(C)(CC1)OC2 C(N=c1cc(Cl)c(O)n[nH]1)C1CC(NC(C2(F)CCCCCC2)=O)C1 C12(C(=O)NC(CC(N)=O)C3CC3)CC(CN(C(c3n[nH]c(O)n3)=O)C1)C2 Cc1cc(NC(c2sc(CS(C)(=O)=O)nc2C)=O)cc(C)c1S(N)(=O)=O C1(=O)C(CC(C)C)ONC(=O)C2CCC(C2)N1.C(=O)(CCC(C)N(C)C)OC C1(C(C)C)CN(C(c2coc(CNC(=O)Cc3ccns3)n2)=O)C1C(C)C C(=O)(C(CCC(N)=O)N=[N+]=[N-])NCC1C(C)(C)C1C(F)F N1(C(c2c(C)nc[nH]2)=O)CCN(C(c2ccc(Cl)s2)=O)C(CC#N)C1 N1(C(CCC(=C)Br)=O)CC2CCC(C1)C(NC(=O)C(C(C)(C)C)OC)C2 C1(NC(c2nc(CCCC)sc2)=O)CCC2(CCCN2)C1 C1(NC(=O)Cc2cncs2)CC2CCC1CC2NC(C1CCc2nc[nH]c2C1)=O c1(C(=O)NC2C(NC(c3cn(CCC(C)C)nn3)=O)C2)cnc(N(C)C)nc1 c1(OCC)ccc2nc(O)n(CC3CCCC(N(C)C)C3)c(=O)c2c1 C1(C(=O)NCCn2ncc(CC)c2)C=CCN(C(c2cn(C)nn2)=O)C1 c1(C(N(C(C)CNC(=O)C(C2CCCCC2)F)C)=O)cc(-c2cc[nH]n2)ccn1 N1(C(C2(CC=C)CC2)=O)CCCN(C(c2ccc(F)c(C(C)=O)c2)=O)C(C)C1 N1(C(C(C(C)(C)C)SC)=O)CC(NC(C2(C3CC3)CC(=O)C2)=O)C(C2CC2)C1 C1(C(N2C(CCCNC(C=CCCC)=O)CCC2)=O)CCCCCS1(=O)=O c1(CNC2(CC(=O)Nc3cccc(OC)c3)CCC2)ccc(Br)nc1Br c1(C2CCC(=O)N2)ccc(CCC(N2CCCC2CO)=O)cc1 C12(CNC(Cn3c(C)c(Cl)cn3)=O)CCC1CCN2C(=O)CN(C)CCO c1(CC(=O)N(CC(O)CN(S(C)(=O)=O)C)C)nnn(C(C)(C)C)n1.C1(C)CC1 c1(CNC(=O)Cc2cncs2)ncccc1CNC(c1ccnnc1)=O Cc1cc(NC2CCCCCCC2CO)ncc1S(=O)(=O)NCCN(C)C1CC1 C(C)(C#CC(=O)N=c1cc(C)n(C2CC2)[nH]1)OC.c12ccoc1C(=O)NC2 c1(C(=O)NCC(CNC(C(C=C)(F)F)=O)(C)C)sc2cccc(C)c2c1Cl S(=O)(=O)(c1ccc(Br)c(C#N)c1)N(c1ncc(F)cc1F)C Cc1ccc(C(=O)NCc2csc(CNC(C3COC(=O)O3)=O)n2)c([N+](=O)[O-])c1 CC(C)S(=O)(=O)CCCNC(=O)CN(C1CCN(C(=O)C(C)n2ccnc2)CC1)C C1(NC(COCC(C)(C)C)=O)CC1C1CCN(C(C2CC2(F)F)=O)CC1 C1(NC(C(C2CCCN(C(=O)C=Cc3ccnn3C)C2)C)=O)CC(F)(F)C1(C)C c1(C(=O)NC2C3(CCN(C(C=CC)=O)CC3)C2)cc(S(=O)(=O)NCCOC)c[nH]1 c1(C(C(=O)NCCCF)N(CCCN(C)C)C)ccc(SC(F)F)s1 C#CC1(O)CC(C(=O)NCC2(O)CN(C(C3C(C(F)(F)F)C3[N+](=O)[O-])=O)C2)C1 C1(C#N)(C(=O)NC2(C)CCN(C(C34COCC3C4)=O)C2)CCS(=O)(=O)CC1 c1(C(N2C(CNC(C(C)=C(CC)C)=O)CCC2)=O)ccc2[nH]ccc2c1 C1(C(N2CCCC(N(C)C(C3CC(O)C3)=O)CC2)=O)CCCC2(CCC2)O1 CCC(C)CCCC(=O)NCC1CC1CC(=O)NCC(C)C(C)CC C1(NC(Cc2[nH]n(CC(C)C)c(=O)c2)=O)CCCN(C(=O)CN2CCCC2)CC1 c1(C(=O)NCCN(c2ccc(NC(C=CC)=O)cc2)CC)ccc(F)nc1F c1(CC)cccc(C)c1NC(=O)CNC(=O)CC1C=CCCC1 C1(C(=O)NCC(C)(C2CC2)NC(c2ncc(Cl)cc2Cl)=O)CC(=O)CC12CCC2 C1(C(=O)NCc2cccc(CN(C)Cc3ccc(Cl)cc3)c2)CC(=O)OC1(C)C N1(C(C(C)OCCCC)=O)CCCC(CN(C)C(c2nocc2C)=O)C1 CC(CCC(=O)N(C1CCC1)CCO)NC(=O)C(C)(C)O CCCC(C)(C)CC(=O)N1CCCCC(C(=O)NC2CCCC2(C)C)C1 C1(C(=O)NC(C(N)=O)C(N)=O)CC12CCN(C(c1cnn3c1OCCC3)=O)CC2 n1(CC)ncc(C)c1C(=O)N(CCCCN(C(=O)CC1OCCO1)C)C N1(C(c2ccc(-c3cccc(Cl)c3)o2)=O)CC2CN(Cc3ccc(F)cn3)C2C1 C1(NC(CCOCCN(C(C2(CC(C)C)CC2)=O)C2CC2)=O)C=CC(C)(C)CC1 c1(C(=O)OCC)cc(CCOC(c2cc(-c3csc(C)n3)cn2C)=O)oc1C N1(C(C(n2ncc(C)c2)C)=O)CCOC2CN(C(=O)CC(C(C)C)C(C)C)CC12 c1(N2CC(C(C)C)OCC2)nc(=NCCc2ccoc2)[nH]c2c1CCCCC2 c1(C(=O)NC2CCC(C)(CNC(CCN(CCC)C)=O)C2)nc(C)c(C)nc1C c1(CC)ccc(CCNCCC2CC2)nc1 Cc1ncc2n1CCC(c1nc(C3CCCO3)nn1CCS(N)(=O)=O)C2 C12(C(=O)NC(CNC(c3ccc(C(=O)OC)nc3)=O)C)CCCC(C1)C(=O)N2 S(=O)(=O)(c1sc2ccccc2c1C(=O)OC)NC(CSC)Cc1ccc(F)cc1F N1(C(C2(C)CC=CCC2)=O)CCCC2(CCN(C(C3CCNC3=O)=O)C2)C1 C1(CNC(c2cncc(C)c2)=O)CN(C(=O)Cc2ccsn2)CCC12CCC2 Cc1oc(CO)cc1C(=O)NC(C1CCCC1)CNC(c1ccc(N)cc1)=O N1(C(C(C)SC)=O)CCC(C2CC2NC(c2ccc(F)c3c2OCC3)=O)CC1 C1(C2CCCN(C(c3nnsc3C)=O)C2)(NC(C2C(CCC)C2)=O)CC1 C1(C(N2CCC(OCCNC(c3c(Cl)cn(C)n3)=O)C2)=O)CCn2ncnc2C1 Cn1nc(C(=O)Nc2ccsc2C#N)c2ccc(-c3c(F)cccc3F)cc12 N1(C(c2cc(C)[nH]c2C)=O)CCCC(C)(C)C1C(N1CC2(CNC(=O)C2)C1)=O C1(C(=O)NCC(O)Cc2ccccc2)CSCCN1C(c1cncc(O)c1)=O C1(C(N2CC(C)C(NC(=O)C(C)(C)n3cccn3)C2)=O)CCCCC12CC2 c1(NC(C2CN(C(=O)C=Cc3cccs3)CCO2)=O)cnc2ccccc2c1Cl c1(OC)cccc(-n2nnnc2C(CSC2CCCC2)Nc2cc(C)sc2C)c1 N1(C(C2CCCN(C(CC=C)=O)CC2)=O)CC2CCCC(O)C2C1 Cn1cc(C=CC(=O)NC2(CNC(C3CCNC(=O)C3)=O)CCOC2)nn1 C1(O)(Cn2cc(C(C)O)nn2)CCN(C(=O)CCc2ccnn2C)C1 O=C(CCC1C(=O)Nc2ccccc21)NC1CCCN(C(=O)CO)CCCC1 CC1(NC(=O)Cc2cccc(C(F)F)c2)CCN(C(=O)Cc2csc(=N)[nH]2)C1 C(CC(=O)NC(c1ccco1)CO)OCCN(C)C(c1ccco1)=O C(=O)(C1CCCc2nc[nH]c21)N1CC(CC(C)NC(c2ncn(C(C)C)c2)=O)C1 C1(NC(c2cc(C)on2)=O)CCC(NC(C2(C)CC3(CC3)C2)=O)CC1 c1(C(N2CCC(O)(CN(C(CSCC=C)=O)C)C2)=O)ccn2nnnc2c1 C(=O)(CCCC(C)(C)C#N)NC(C(N1CCC(O)(C(C)C)C1)=O)Cc1ccoc1 N1(C(CCOCCC)=O)CC2CC(C1)N(C(C1CC13CCSCC3)=O)C2 CC#CCCC(=O)NCC(O)CN(C)C(c1cnn(CCOC)c1)=O Cn1nc(C(C)(C)C)cc1C(N1CCOC(CNC(=O)CC(C)(C)O)C1)=O C1(NC(c2c(CC)nc[nH]2)=O)(COC)CCN(C(c2nn(C)cc2SC)=O)CC1 C1(OC)CC(CNC(=O)CCC2(C)CCC(=O)N2)N(C(c2cc(Cl)cn2C)=O)C1 c1(C(=O)NC(CCOC)CNC(C2(F)CCCC2)=O)ccc2c(c1)CC(C)O2 CC1OC2(C(=O)N(C)CCN(C(=O)CCOc3cccnc3)C)CC1C2 O=C(C(Cn1cccn1)NC(C1CC12CCC2)=O)NCCCc1nncs1 c1(C(=O)NCC(C2CC2)NC(C(CC)O)=O)ccc(Cl)cc1C(F)F Cc1cc(C(=O)NCC(C)(CO)NC(c2cc(C3(C)CC3)n[nH]2)=O)cc(F)c1 C1(OC)CC(CNC(=O)CC23CCC(CC2)C3)N(C(=O)C=CCN2CCC2)C1 N1(C(CCCC(C)=O)=O)CC2OCCN(C(=O)C3Cc4ccccc43)C2C1 c1(C(N2CC(N(C(C(C)n3ccnn3)=O)C)C2)=O)ccc(Cl)c2ccccc12 C(=O)(CCCCC(C)(C)C)NC(CNC(C(CSC)C)=O)CC(F)(F)F c1(C(N2CC(NC(c3cnn[nH]3)=O)CC(OC)C2)=O)cc2cccc(O)c2[nH]1 Cc1nnc2c(C(N3CCC(NC(c4ccc(F)cc4)=O)CC3C)=O)cccn12 CCC(C(=O)NC(C)CNC(=O)CCC1CCOC1)SC C1(CC)CN(C(c2cc(Br)ccn2)=O)CC1NC(=O)CC1COCCO1 C(C(C(=O)N(CC)Cc1ccccc1)C(C)C)NC(COCCCC#C)=O CC1CCN(C(C2C3CNC(=O)C23)=O)CC1NC(c1cc(C(C)(C)C)on1)=O Nc1ncc(Br)nc1C(=O)NC1CN(C(C2C=CC(=O)N=N2)=O)C1 C1(C(=O)NC(C)C(C)(C)C)CCC2(CC2)N1C(c1cccc(C#N)c1)=O CCCC(CC(=O)NCCC1(C)CCCC1)NC(c1cc(C(C)=O)[nH]n1)=O C(C(F)(C(=O)NCCC1(C)CC1)C(C)C)NC(CC1CCC(C)CO1)=O C1(CNC(CNC(C)=O)=O)CC2(CCOCC2)CN1C(=O)C(C)OCOC Cn1c(C(N2CCC(C)(NC(C3CC3[N+](=O)[O-])=O)C2)=O)cc(Cl)c1Cl C1(C(=O)N(CCCCN(C)C(C2CCCS2)=O)C)(OC)CCCC(C)(C)CC1 C1(C(=O)NC(C#C)CCC)CC(=O)N2CCCCC12 C(=O)(CCC(=O)N(C)CCOCCC(=O)NCC1(O)CCCC1C)NCCC C(C(CC(C)C)C(=O)NC(C)(CNC(c1csc(F)c1)=O)CC(C)C)OC C(CC(O)CCC)NC(C1(CCC=C)CN(C(=O)CCOCCC)C1)=O c1(N(C)C)ccc(-c2ccnc(C(=O)NCc3cccc(O)c3)c2)cc1Cl C=CCC(C(=O)NC1(C)CN(C(C2(CC)CCOC2)=O)C1)NC(C)=O C#Cc1cccc(C(N2CCC3(CC2)CC3NC(=O)C(C)CC2CC2)=O)c1Cl C(C)(CCCCNC(C1(N(C)C)CCOC1)=O)NC(c1ccc(C(C)C)s1)=O N1(C(C=Cc2ccc(SC)s2)=O)CCN(C(c2coc3c2COC3)=O)C(C)C1C n1(CCCOCC)c(N2CCOC(C(C)C)C2)nnc1C(c1ccncc1)C C1(NC(c2c(CC)cco2)=O)CN(C(c2cnn(C)c2C)=O)CC1OC C1(F)(CNC(C(C2CC2)OC(C)(C)C)=O)CCN(C(=O)CSc2cscn2)C1 C(CC(C)C(=O)N1CCCC1C=CC(=O)NCC(=O)N(C)C1CC1)=CCC c1(C(N2CC(O)(CNC(C(C)N(C(C)=O)C)=O)C2)=O)ccc(Cl)c(N)c1 N1(C(C(C(C=C)C)C)=O)CCC2(CCC(CN(C(=O)C(C)CCC)C)C2)C1 c1(SC)ccc(O)c(C(=O)NCC2CCN2C(C2(CC3CCC3)CC2)=O)c1 c1(CC)nc(C)[nH]c1C(N1CCCC1C(C)(C)CNC(c1ccoc1Br)=O)=O C1(OC)CC(CNC(c2cc(C)n(C(CC)CC)n2)=O)N(C(=O)CNC(N)=O)C1 Cc1cc(C(=O)NCC2CC(C)N(C(=O)CCS(C)=O)C2)ncc1C#N CCC(C)CCCC(=O)N1CCC2C(C1)CN2C(c1cc(Cl)cc(Cl)c1OC)=O c1(-c2c(OC)ccc(F)c2)cc(C(N2CCCOCC2)=O)cc2c[nH]nc12 CC1(C)CCCCNC(=O)CN(C)CCN(S(C)(=O)=O)C(CC)C1=O N1(C(C2C(C)C2C)=O)CCCC(C2CC2NC(C2CCOCC2)=O)C1 C12(CNC(CC(C=C)C)=O)CCCC1CN(C(c1[nH]ccc1C1CC1)=O)C2 C(CC(F)F)(C(=O)N(CC(C)C#N)C)NC(c1c(C(C)C)c[nH]c1)=O c1(OC)cc(C(=O)NCC2CC2NC(c2cnoc2C)=O)cc2c(C)c(C)[nH]c12 N1(C(Cc2c(C)cnn2C)=O)CCC(NC(C2CNC(=O)N2)=O)C(C(N)=O)C1 c1(C(N(C(CNC(C(CC#C)C2CC2)=O)C)C)=O)cnc(O)c2ccccc12 CC1CN2CCN1CC2C(=O)NC1CN(C(C2(F)CCC(F)(F)CC2)=O)CC1C c1(C(=O)NC2CC(NC(c3nn(CC)c(C4CC4)c3)=O)C2)ccc2n[nH]cc2c1 c1(NC(N2C(C)(CC(C)C)CCC2)=O)ccccc1N=[N+]=[N-] c1(CC2(C(=O)NC(c3cc(C)oc3C)=O)CC2)c(C#N)oc2ccccc12 CC(C(=O)NCCCCNC(c1ncccc1O)=O)S(N)(=O)=O C12(C(N3C(C4(NC(C=CCC)=O)CC4)CCCC3)=O)CCCC1OCC2 C12(NC(c3c(CC)nc(C)o3)=O)CCCN(C(C3(CC)CCCO3)=O)CC1C2 C12CCCN(C1)C(=O)N(C(=O)NN(CCCC(C)C)C)CC2.C(C)(C)(C)O.CCS CC1CCCCC1(CNC(=O)C(C(C)(C)C)C1CCCC1)NC(=O)C(C)CO N1(C(Cc2cc(OC)no2)=O)CCC(O)(C(C)NC(=O)C#CC(=O)N(C)C)C1 C1(C)(C(=O)NC2CC(C)OC2)CCCN(C(=O)CCNC(=O)OC(C)(C)C)C1 N1(c2n(CC=C=C)nnn2)CCN(C(C)CC)CC1 Cn1ccc(C(=O)NC(CC2CC2)C(=O)NCc2ccc(Cl)o2)c1 C=CC(CC)CC(=O)N1CC2CC(CNC(=O)Cc3nc(C)c(C)s3)C2C1 N1(C(C2(CCC=C)CC2)=O)CCC(NC(C2CCN2CC)=O)C12CC2 c1(C(=O)NCCCCC2(NC(C(OC)OC)=O)CC2)cc(O)ccc1Br c1(C(=O)NC2CC(N(C)C(c3cn(C(C)(C)C)nn3)=O)C2)cnn2ccncc12 N1(C(Cc2c(C)noc2)=O)CCCOC(CNC(c2nc(O)c(C)s2)=O)C1 c1(CCC)ccc(CC2(CNC(=O)OC(C)(C)C)CC(C(=O)O)C2)o1 c1(C(N(C)CC2CCN(C(C=C(C)Cl)=O)C2)=O)n[nH]c2c1CC(C)(C)CC2 c1(C(=O)NC(CNC(C2CC(OC)C2)=O)C(C)C)cc(OC)c2c(cnn2C)c1 c1(NC(CCC2N(C(c3nn(C)c(Cl)c3)=O)CCC2)=O)ccnc(O)c1[N+](=O)[O-] c1(C(=O)NCC2C(NC(Cn3c(C)cnc3)=O)CCC2)cccc2cc[nH]c12 c1(OC)cc(Cl)ccc1C(N1CCC2(NC(c3cc(Cl)c(C)cn3)=O)CC2C1)=O N1(C(CC(=C=C)C)=O)CC(C)C(C)(CNC(c2c(Cl)nn(C)c2C)=O)C1 N#CC1(C(=O)NCC2C3CN(C(=O)Cc4cnccc4Cl)CC23)CC2C=CC1C2 C1(C)(CCC(=O)NCCSC(C)C)CN(C(=O)CN2CCCC2)C1 c1(CC(C)NC(C2(CCNC(c3csnc3Cl)=O)CCC2)=O)ccncc1 C1(NC(C(C)NCCCC(=O)OC)=O)CC(C2CC2)C1 c1(OC)ccc(CC(=O)NCCNC(C2COCCO2)=O)c(Cl)c1 CCC(CC(=O)N1CC(O)(CNC(=O)CC(F)(F)C(F)(F)F)C1)C(C)(C)C c1(CNC(c2c(CNC(C(C3CC3)SC)=O)c[nH]n2)=O)ccccc1F CC(CC(=O)NCC1CC1)C(=O)c1ccc(Cl)cc1.C1(=O)CCCCCCN1 c1(OC)cc(C2(C(N3CCN4CC3C4=O)=O)CC2)ccc1Cl.C1(OC)CC=CC1 C(=O)(C(F)C(C)(C)O)NC1CC(N(C(C(F)=CC)=O)C)C1 CC(C(=O)NC1CC1CC1CCN(C(c2cnc(Br)s2)=O)CC1)C(C)(C)C Cc1ccc(CCC(=O)NC(c2cn(CCc3ccccn3)nn2)C)cc1Cl C1(C(=O)NCC2CCCN2C(C2CCC2(F)F)=O)CCCCC12CC2 CC1(C)Cc2[nH]nc(C(=O)NCc3cncc(C(=O)O)c3)c2C1 CCCC(O)Cn1cc(CN(C(=O)C(F)(F)c2cccnc2)C(C)(C)C)nn1 CN1CCCCC(C(=O)Nc2csc(C3CCS(=O)(=O)C3)n2)C1=O c1(C(=O)NCC=C2CCN(C(C3(C)CCCCC3)=O)CC2)cc2n(c1)CCSC2 C1(CC=C)(NC(C2CC(=C)C2)=O)CCN(C(=O)CCNC(=O)C=CCl)C1 C(CNC(=O)C(CSc1cn(CCC(=O)O)nn1)OC)(C(C)C)OC C(=O)(C#CC1CCCOC1)NC1CCN(C(c2cc(OC)c(N)cc2)=O)CC1F c1(CN2CC(C(N(CCCNC(C3(CC)CCC3)=O)CC)=O)C2)ccc(Cl)cc1 Cc1cccc(N2CCC(C(=O)NCCN(C(=O)C(O)C3CC3)C)C2=O)c1 CCC(C)(CC)C(=O)NCCC1CCCCN1c1ccnc(CCOC)n1 S(=O)(=O)(c1ccc(Cl)c(F)c1Cl)NC1CN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC2(C)CN(C(C3C4CN(C)CC43)=O)C2)cc(=O)n(C)cn1 Nc1cc(Cl)cc(Cl)c1C(=O)NC1CC(NC(c2noc3c2CCCC3)=O)C1 c1(NC(C2C(C(=O)NC(c3ccccc3F)C)C2)=O)ncccc1Br c1(NC(=O)C=C2CCN(C(c3ccc(F)cc3O)=O)CC2)cc(Br)ncc1F c1(CC(N2C(CNC(c3n(CC)cnn3)=O)CC2)=O)ccc2c(c1)OCO2 C(=O)(C1=CC2CCC(C1)C2)NC(CCC)CNC(c1n[nH]c2c1COC2)=O C1(CNC(CSC(C)C)=O)C(C)CCN1C(=O)C(C)CN1CCCCC1 N1(C(CC(C)n2ccnc2)=O)CCOC(C(C)(C)C)C1 Cc1onc(C2CC2)c1C(=O)NCCNC(C1(C)CC=CC1)=O C(C)(C)(CCC(=O)N1CCOCCC1C(=O)NC(C)CC1CCC1)OC c1(C(=O)NC(C2CCCCN2C(=O)CC(F)(F)Cl)C)cnc2ncccn12 Cn1cccc1CNC(=O)C(CO)NC(=O)CCc1cscn1 c1(NC(C2N(S(CCCC)(=O)=O)CCOC2)=O)c(OC)ncnc1Cl Cn1cc(CCC(c2nnnn2-c2ccccc2)NC(CO)CCF)cn1 c1(C(=O)NCc2cccc(CN=c3ncc(Br)c[nH]3)c2)ccn2ccnc2n1 C1(C(CC)(C)C)CCc2nc(NC(=O)N(CCO)Cc3ccc(Cl)cc3)sc2C1 c1(CC(=O)N(CC(C)NC(c2cc[n+]([O-])cc2)=O)CC)ccc(C)c(F)c1F Cc1onc(CO)c1C(=O)NCCNC(C1CC1F)=O c1(C(N(C)CC2(NC(=O)CC3CCCC(=O)N3)CC2)=O)cc2cccc(F)c2s1 CCC(C)(C)C(C)CC(=O)NCC1(O)CN(C(=O)C(n2nccc2C)C)C1 c1(C(=O)NC2CCCC2CNC(C2C3CC4C(C3=O)C24)=O)ccc2ccoc2c1 Cc1cc(Cl)cc(C)c1C(=O)NC1CCCCC1NC(C1(CF)CCC1)=O N1(C(CC(C)(C)SC)=O)CC(NC(c2coc(C(F)F)n2)=O)C2(CC2)C1 C1(CNC(=O)Nc2cc(F)c(CC)c(F)c2)CCC2C(CC1)C2(F)F c1(CC)cccnc1C(=O)NCC1(F)CCN(C(=O)Cc2ccccc2NC)C1 C1(CC(N2C(C)C(NC(=O)CC34COCC(C3)C4)CC2)=O)CCCC(C)(C)C1 c1(C(N2CCC(N(C(=O)Cc3ccnc(Br)c3)C)C2)=O)c(Br)cc(Br)c(O)c1Br C(=O)(CC(C)(C)C(F)F)NCCC(C)NC(C1(OC)CCOC1)=O C1(NC(C(C)(C)OCC)=O)CN(C(C2CCCN(CC(F)(F)F)C2)=O)CCC1F c1(CCC2CCCC(C(=O)NC(=O)C(c3ccccc3I)O)C2)ccc(Cl)cc1Br C(N=c1[nH]c(N2CC(C)OC(C)C2)nc2cccnc12)c1cnc(CC)s1 N1(C(C(C)Cc2ccccc2F)=O)CC2=C(C1)CN(C(=O)C=C1CCOCC1)C2 C(=O)(C(F)(F)CC(C)C)NC(C1CCN(C(C(C2CCCCC2)OC)=O)C1)C n1(CC)c(C)nn(CC(=O)NC2CCC(NC(c3ccc(C)s3)=O)CC2)c1=O C1(NC(C2(OC)CCOC2)=O)CN(C(c2cnncc2C(F)(F)F)=O)CC1C c1(OC)cc(C(=O)NCC2CC(NC(=O)CC3CCCS(=O)(=O)C3)C2)cc(F)c1 c1(C(N2CCC(N(C(CCCC(CC)C)=O)C)C2)=O)cccc(S(C)(=O)=O)c1F C1(C(=O)NCc2n(CCC)cnc2)CCN(C(=O)C(C)CC(F)(F)F)O1 CC1CCN(C(c2ccccc2)=O)CCN1C(C1(c2ccco2)CC1)=O c1(C(=O)NCC2(C)CCC(NC(C=C(CC)CC)=O)C2)cc2ccccc2[nH]1 N1(C(C2CC2(F)F)=O)CCCC(NC(C2(F)CCCC2)=O)CC1 C1(c2cnn(C)c2)C(=O)N2CCC(O2)C(=O)N1.N1(CC)CCc2cccc(F)c21 N1(C(C(C)(C)OC)=O)CC(C)(C)C1C1CCN(C(=O)CCCc2ncco2)CC1 N1(C(C)C(=O)NCC(O)CN(C(=O)C(C)(C)c2ccccn2)C)CC2CCC1C2 c1(C(=O)NC23CC(CNC(CCC(=O)OC)=O)(C2)C3)ccc(Br)cc1SC n1(CC)cnc2c(N3CCCC(CCO)C3)nc(=NCc3ccsc3)[nH]c12 c1(NC(c2cccc(N)n2)=O)c(Cl)cc(F)cc1Cl c1(SC)ccc(C(=O)N(C)CC2(O)CCN(C(C3CC(C(F)F)C3)=O)C2)cc1 c1(O)cccc(C(=O)N(C2(C(N)=O)CC2)C)c1.CCS Cc1cc(Cl)ccc1NC(c1cc(CCNC(=O)C(C2CCCCC2)O)on1)=O N1(C(c2c(CC)nco2)=O)CC=CC(NC(c2cncn2C2CC2)=O)C1 S(=O)(=O)(c1cccc(=NCCCCCO)[nH]1)NC(COCC)C(C)C C1(CN(C(C(CSC)C)=O)C)CCN(C(C2CC2F)=O)CC1 Cc1cc2occ(C(=O)Nc3cc(OC4CCCC4)ncn3)c2cc1C CCC(C)(CC)C(=O)NCCC1(CNC(=O)C(C2CCCC2)OC)CC1 CC(C)CCCC(C)NC(=O)CCN(CCO)C(c1nc(Cl)cs1)=O CCCS(=O)(=O)c1ccc(C(=O)N(CC(C)NC(=O)CCCC(C)(C)C)C)cc1 C1(NC(c2cc(CC)on2)=O)CCC(NC(=O)CC2CCCN2C)CC1 C1(ONC(N2CCOCC2)=O)CCN(N2CC(OC(F)F)C2)CC1.CO C1(NC(c2c(C(C)C)ccs2)=O)CC(C)CN(C(=O)Cc2csc(Cl)n2)C1 Cc1ncnc(C)c1CC(=O)NCCN(C)C(C1(N2C(=O)CCC2=O)CC1)=O N1(C(c2c(C)nc(C3CC3)s2)=O)CC(O)(C2(CNC(=O)C(F)=CC3CC3)CC2)C1 C1(CNC(COCC)=O)C2CN(C(=O)CN(C)C(c3cccs3)=O)CC12 C1(C(=O)NCC2(C(=O)OCC)CCC2)CC(=O)N(C)C1c1ccc(Cl)c(F)c1 c1(C(=O)NC(CCNC(c2c(SC)cc(F)cc2)=O)C)ccn2ncccc12 CN(C(=NCC1CCOC1)NC1CCS(=O)(=O)C1)Cc1ccc(F)cc1Br c1(OC)ccnc(F)c1C(=O)NC(C)CNC(c1n[nH]c(C)c1F)=O Cc1cc(NC(=O)CC2CC(NC(c3ccc(C(N)=O)o3)=O)C2(C)C)cnc1O C12(C(N)C(N3CCC(c4cccc(OC(F)F)c4)C3)=O)CC3CC(CC(C3)C1)C2 C1(CNC(C(=O)NCCS(CC)=O)=O)NCCC12CCC2 Cc1nc(C)c(C(=O)NC2COC3(C2)CN(C(c2cnc(C)[nH]2)=O)C3)c(C)n1 C1(NC(Cn2c(C)c(Cl)cn2)=O)CCCCN(C(=O)CC23CCC(C)(C2)OC3)C1 CCCC(C#N)C(=O)NCCc1ccc(CNC(=O)C(O)C(C)C)cc1 C1(C2CCCCC2)(C(N2CCC(CNC(=O)C(F)=CCCF)C2)=O)CCCCC1 C(CC(C)(C)C)(C(=O)NC1(CO)CCN(C(=O)CCc2ncc[nH]2)C1)NC(C)=O C1(C(=O)Nc2cccc(-c3noc(C4CC4)n3)c2)CC2(CCC2=O)C1 c1(CC)nc(C(N2CC(SCCNC(=O)Cc3ncc(C)s3)CC2C)=O)c(N)s1 CCC(C)(C(=O)N1CC2CN(C(=O)Cc3csc(C(C)(C)C)n3)CC2C1)C(N)=O C1(C(=O)OC)CC(n2cc(CN)nn2)CN1C(C1(C(F)F)CCCO1)=O C1(N(C(=O)CC(C2CC2)C2CC2)C)CCCN(C(C2CC2C(F)F)=O)CC1 N1(C(c2c(CNC(C(C)O)=O)cco2)=O)CC(O)CC1CO c1(CN(C)CC2CN(C(C3CC(F)(F)C3)=O)C2)cc(Cl)cc(Br)c1 c1(C(=O)NC2(CC)CN(C(=O)COCCc3cccc(F)c3)C2)nn(C)cc1Cl n1(CC(=O)NC2CN(C3CN(C(CC(=O)NC)C)C3)C(=O)C2)cnc([N+](=O)[O-])n1 n1(CCC)ccc2cc(Nc3cnn(CCC(=O)OCCCO)c3)ccc12 C(=O)(C#CC1CCCC1)N1CCC(NC(C(COC)(C)OC)=O)C(C)C1 Cc1c(OOC2C=CCCC2)cccc1NC(=O)Nc1cn(C)nn1 N1(C(CC2C3CN(C(C4C(C)(C)OC(=O)C4)=O)CC32)=O)CC(C2CC2(F)F)C1 c1(CC)c(C(N2CC(CC(C)NC(C3(C)CC4CC4C3)=O)C2)=O)csc1C N1(C(c2c(CC)cco2)=O)CCN(C(c2cocn2)=O)C(c2cccc(F)c2)C1 N(C(=NCC(=O)NC1C(SCC)CCCC1)NCCc1ncc(C)s1)C(C)C Cc1oc(C(C)C)nc1-c1nc(Cc2cccs2)nn1-c1ccc(Cl)cc1 C(=O)(C(CCS(C)=O)CNC(=O)OC(CCc1ncc(C)[nH]1)=O)OC(C)(C)C C1(F)(CNC(C2CCCC2CNC(=O)CCC2CCCCC2)=O)CCOCC1 C1(NC(C2(COC)CCC2)=O)CN(C(=O)CSCC(F)(F)F)CC1S(C)(=O)=O C1(CC)CCCC1C(=O)NCC=CCNC(=O)CC1CC(F)(F)C1 N1(C(C(C(C)C)OC)=O)CCC(N(C(=O)CCOC(C)=O)C)C(C)C1 C(C(C)(C)CNC(=O)Cc1ccco1)N(C)C(c1nc(Br)c[nH]1)=O c1(N2CC(Cn3ncc(C)c3)OCC2)ccc([N+](=O)[O-])c(N)c1C#N N1(C(Cc2cc(OC)c(O)cc2F)=O)C2CCCC1CN(C(C1(F)CCC1)=O)C2 c1(CCCN2CC(N(C)S(N)(=O)=O)C2)ccc(Br)cc1 c1(CCC)cccc(C(N2CC(NC(=O)CCNC(=O)COC)CC2C)=O)c1 c1(C(N2CCC(F)(C(=O)Nc3n(CC)nc(C)c3)C2)=O)cc(O)ccc1Cl C(=O)(C1=CCCC1)NCCC(Cc1ccccc1)NC(C(C)OC)=O c1(OCC(=O)OCC2C(CC(C)(C)C)C2)ncc(Cl)cc1Cl c1(NC(=O)NC2C(C=C)CNC2)c(C)cc(C)cc1C C1(CCC(=O)NCC(C)(C)NC(C2CN(C3CCOC3)C2)=O)CCCCO1 CCCC(CC)C(=O)N(CCCCCCNC(c1ccccc1OC)=O)C C1(C(N2CC(CC(C)NC(C3C=CCC3)=O)C2)=O)CC2(C1)CC1(CCC1)C2 c1(C(N2CC(C)N(C(C3CN4CCN3C(C)C4)=O)CC2)=O)n[nH]c2ccccc12 CN1CC(O)CC1C(=O)NCCC(O)CNC(c1ccc(C2CCCC2)cc1)=O N1(C(CC(COC)C)=O)C2CCC1C(F)C(NC(=O)C1=CCOCC1)C2 c1(C(=O)OC(C(=O)NCC(c2cccc(O)n2)(C)C)=O)csc(S(N)(=O)=O)c1 CCCCCC(C)CC(=O)NCC1CN(C(=O)Cc2sc(S)nc2C)CC1C c1(C(N2C(CO)CC(NC(c3nccc(C)c3)=O)C2)=O)nccc(C#N)c1F c1(CC(=O)NC(C(CO)NC(c2ncn(CC)n2)=O)C)cccc(OC(F)F)n1 C1(C(=O)NCC2(NC(c3csnn3)=O)CCOC2)CC(O)C(F)C1 C(=O)(CC(C1CC1)NC(c1cn[nH]c1)=O)NCC(c1ccco1)SC Cc1cc(C(=O)NC(C)C(CO)NC(C2CN(c3nnnn3C)C2)=O)ncn1 CCCCCC(=O)NCC1(NC(=O)CC2CCCN2CC)CC(OCC)C1 Nc1cc(Cl)c(Cl)cc1C(=O)OCC(N1CCN(c2ccncc2F)CC1)=O c1(C(N2CC(C)C(NCc3cncc(Br)c3)C2)=O)ccc(Cl)cc1F C(=O)(CCCN=[N+]=[N-])NCC1(C(=O)NCc2c(C)n(C)nn2)CCCO1 C(=O)(CCCC(C)(C)C#N)NCC(CNC(C(C)C(C)c1ccc(F)cc1)=O)C C1(F)(C(=O)NC2(CC=C)CCOC2)CCCN(C(C2CCCC3(CC3)C2)=O)C1 CN1CCC(C(N2CCC(CCNC(=O)C(N)=O)C2)=O)(C(F)F)CC1 N1(C(C(C)(Cl)Cl)=O)CC2COCC(C1)C2NC(C1COC2COCC12)=O C(=O)(C(C)(O)C(F)(F)F)N1C(CNC(CNc2cccc(C#C)c2)=O)CC2CC21 C1(CNC(C2N(CC)CCOC2)=O)CN(C(C2CCCCS2)=O)CCN1C C(=O)(CC1OCc2ccccc21)NCCCNC(c1cnc(C)nc1C(C)C)=O CCCC(CCC)CC(=O)NC(CNC(=O)CCNC(C1CCC1)=O)CO C12(C)CCN(C1)C(=O)C(N(C)C)CNC(=O)C2.C1(CCOCC)(OC)CC1 N1(C(=O)NCCn2c(C)ncc2)CC(CC(=O)O)CC12CCC2 c1(NC)c(C(=O)N(C2CCCN(C(=O)C=C(C)C)C2)C)cccc1F C(C1CCOc2ccccc21)NC(=NCCCF)NCCCN1CCCCC1 c1(C(=O)OCC)ccoc1C(=O)N(CC(C)N(C)C(c1ccnn1CC)=O)C N1(C(CCC(C)OC)=O)CCC(CNC(=O)CCc2ccccc2)C12CC2 C1(NC(CC2CCC(C)C2)=O)CCN(C(C2(C)CCC2)=O)CC1(C)C c1(C(=O)NC(CC(C)NC(CC2(C=C)CCC2)=O)C)ccc2nc[nH]c2n1 N1(C(c2cc(F)c(F)c(Cl)c2)=O)CCCC1C1CCCN1C(c1cc(Cl)no1)=O n1(CC(=O)NCCCCN(C)C(c2ccnn2C(F)F)=O)cnc(C#N)n1 c1(C(=O)NC2CC(NC(C(CC)OC)=O)C2)cc(C)c2ccccc2n1 C1(CC=CC)CCCN(C(=O)C(C)(C)CN(C(=O)CCCOC)C)C1 C(C(C)C(=O)N1CC(C)(c2cn(Cc3cnns3)nn2)C1)OCC c1(C(N2Cc3c[nH]nc3C2)C(=O)NCC=C)noc2cc(Br)ccc12 N1(C(c2n(CC)ccc2)=O)CCC(C)N(C(=O)CCn2c(C)ccc2C)CC1 C(=O)(C1=C(Cl)CCCC1)NCC1CC(C)CN(C(c2csnc2Cl)=O)C1 C1(C2CCN(C(c3nn(C)c(Cl)c3Cl)=O)CC2)(NC(c2c(C)ncnc2)=O)CC1 c1(C(C)(C)OC)nc(C)c(C(=O)NCC(C2CC2)NC(C2CC(C)(C)CO2)=O)s1 C(C(=O)Nc1nc(C2CC(F)(F)C2)cs1)(C(C)C)OC(C)=O C1(CCCCC(N2CCC(NC(C(N)=O)=O)C23CC3)=O)SCC2NC(=O)NC12 N1(C(c2cncc(COC)c2)=O)CC2CCC2(CCNC(=O)C(C)(C)CO)C1 N1(C(CC=C=C)=O)CCN(C(C)CNC(=O)CCCCC2CC2)CC1 c1(C(=O)NCC(CN(C(C2(CC=C)COC2)=O)C)C)cnc(C2CC2)nc1C C1(C(C)C)CN(C(=O)Cn2cc(-c3ccc(CC#N)s3)nn2)CCC1CO N1(C(CCCOC)=O)CCc2cccc(C(=O)NC(C)=O)c2C1.C1(=O)CCN1C C1(NC(COCCC)=O)C=CCC(C(N2CCCC(C)C2)=O)C1 CC(C)(C)C(=O)C(=O)N1C(CC(N2CCC(C(C)(C)O)CC2)=O)C2CCCC12 C(=O)(CC(C)P(C)(C)=O)N(CCc1cn(-c2cc(OC)cc(Br)c2)nn1)C C1(Nc2c(C(=O)OCC)cccn2)CN(C(=O)CC2C=CCCC2)C(C)(C)C1 N1(C(Cc2nc(NC(C3CC4CCC3C4)=O)sc2)=O)CCC2(CC2)C1 C1(NC(C2CC(CCC)C2)=O)CC(=O)N(C2CN(C(=O)CCC3CC3(C)C)C2)C1 C#Cc1ccc(C(N2CCC(NC(=O)C3=CCCC3)C2(C)C)=O)cc1C C1(NC(C(C)N2CCCC2)=O)CC2CCC1(NC(=O)Cn1cncn1)C2 c1(C(=O)NC(CCC)CNC(=O)C(O)CN(C)C)ccc2nonc2c1 Cc1cc(C#N)ccc1C(=O)NOCC(=O)N(C1CCCN(C)C1)C1CC1 N1(C(COc2ccc(C)cc2F)=O)CCC(C)N(C(c2cc(C#N)no2)=O)CC1 c1(C(=O)NCCCN(C)C(c2nccc(C#N)c2F)=O)cnc2cccnc2c1 C1(NC(Cc2c(C)noc2Cl)=O)COC2(C1)CN(C(C1CC3CCC(C1)O3)=O)C2 C(C)(CCCC(=O)OC)NC(=O)Nc1ccc(N(C)CC)cc1 c1(C(=O)NCCC(C)N(C(c2ccc(C(=O)NC)nc2)=O)C)cc(C)ccc1F C(C(N=c1cc(C)nc(C2CC2)[nH]1)N(c1cccc(C(N)=O)c1)CCOC)OC C1(C(=O)NCC2C(C(N(C3CC=CC3)C)=O)CC2)CCC(=O)C1 c1(OC)cccc(OC)c1NC(c1cccc(NC(c2c(C)n[nH]c2C)=O)c1)=O c1(C(N(CC(C)NC(=O)C(C)OCCN(C)C)C)=O)ccnc2[nH]cnc12 CCCC(CC(=O)Nc1cc(C)ccc1C)NC(=O)C=Cc1ccc(C)o1 N1(CC(C(C)C)O)CCC2CCC(C1)N2C(c1c(F)cccc1Cl)=O C1(N(C(C)=O)Cc2ccccc2)(NC(c2nc[nH]n2)C)CCOCC1 N1(C(c2c(C)csn2)=O)CCC(NC(c2c(C)cncc2C)=O)C(C)C1 N1(C(c2cnn(CC)c2Cl)=O)CCOC2(CCN(C(C3CC(F)CN3C)=O)C2)C1 CC1C(Cc2ccccc2)CCCN1CCCc1ccc(-c2nn[nH]n2)cc1 C1(CCNC(c2cn[nH]c2)=O)(OC)CN(C(c2cnn(C)n2)=O)C1 C1(CNC(C2OCC(C)(C)C2)=O)N(C(=O)C2=CCCCC2)CCC1(C)C c1(CN2CCC(C(C(F)F)NC(=O)C(F)F)C2)cc(C(F)(F)F)cc(F)c1 c1(C(=O)NCC(C)CNC(=O)C(C)CCO)csc2c1CCCC2 C(=O)(N=c1[nH][nH]c2ncc(Br)cc12)C1N(C(CC(CC)O)=O)CCC1 CC1(C(=O)NCC(CNC(=O)CC2CC3(CC3)C2)CO)CCC2(CC1)CC2 c1(C(=O)NCCCC(C)NC(c2c(C(C)C)con2)=O)cc(C#N)ccc1O C1(CC(N2CC(CCn3cc(CC(C)(C)CO)nn3)C2)=O)CC(O)C12CCC2 C(CCC(C)C(=O)N1CCC(N(CCO)C(c2csc(C#N)c2)=O)C1)OC C(N=c1ncc(O)c[nH]1)C1(NC(C2C(c3cccc(OC)c3)C2)=O)COC1 c1(C(N2C3CN(C(c4c(OC)ccs4)=O)C(C3)C2)=O)c[nH]c2ccccc2c1=N C1(C(=O)N(C2CCN(C(c3n(C=C)nnc3)=O)C2)CC)Cc2ccccc2C1(C)C CC1(C)NC(=O)CCC1NC(C1CCCCC1(C)NC(C1CC(=O)CCO1)=O)=O c1(CC(C)NC(C)C(=O)NC(C)(C)C)ccc(OC(F)(F)F)cc1F c1(C(=O)NC2CN(C(C(CC=C)(F)F)=O)CC(O)C2)c(C)nn2cc[nH]c(=O)c12 S(=O)(=O)(c1ccc2c(c1)C(=O)NCCC2)Nc1c(C2(C)CCO2)cc(Cl)cc1 N1(C(c2c(C)nns2)=O)C(C(=O)NCc2csc(N(C)C)n2)CC2CCCCC12 C1(CC#C)(C(=O)NCC2CCCC2NC(=O)COc2ccccn2)CCCCO1 C=CCCCCC(=O)NC1CCCC1CC(=O)N(C1CC(O)C1)C CCCCCC(C)CC(=O)NCC(F)CNC(=O)C1=CCCC1(C)C Cc1cc(C(=O)NC2(CO)CCN(C(C3CCC(F)CC3)=O)C2)cc(NC)n1 C(N=c1[nH]c(=NCCCCN2CCCC2)[nH]c2c1CCCC2)C1NC(=O)C(F)(F)C1 N1(C(C(CC)c2ccccc2)=O)CC(C2CCN(C(c3cncc(C)c3)=O)C2)C1 c1(C(C)C)nccc(C(=O)NCC(C)(C)CN(C(=O)C(C2CCCO2)OC)C)n1 C1(CNC(C(F)=CCC)=O)CCCC1C(=O)NCC(C)(C1CC1)OC C1(CNC(CCCC#C)=O)CC(F)CN(C(=O)CCc2ccc(C)nc2)C1 C1(NC(c2cccs2)=O)CCCCN(C(=O)CC(O)c2ccccc2)CC1 C1(NC(C(C=C=C)C)=O)CCN(C(C23CCCN2CCC3)=O)CC1OC C1(NC(C(C)(C)SC)=O)CCCN(C(=O)CSc2cc(F)ccc2F)CC1 C12(CC)COC(C(=O)NC3CN(C(C4CC(O)(C#N)C4)=O)CC3OC)(C1)C2 c1(C(=O)NC(CNC(C(CCC)O)=O)C(C)C)ccc(C(F)(F)F)c(C)n1 Cc1nc(N2CCN(C(=O)C(C3CCCO3)C3CC3)CC2C)cc2nncn12 C1(CC(=O)NC(CCN(C(c2n(C)nc(C)c2Cl)=O)C)C)CC2(CCCC2)CO1 N1(C(c2[nH]nnc2C)C(=O)NCCCSCC)CCCC1C1CCCO1 N1(C(C(C=CC)O)=O)CCC(C)(CNC(C2CCCC(C)(C)C2)=O)CC1 c1(C(COC)NC2CCN(C(=O)C(c3ccccc3)C)CC2)ccc(Cl)nc1 C(=O)(C(C)(C)CC(=O)OC)NCC1C2(CC(NC(C3(C)C(CC)CCC3)=O)C2)C1 C(CN=c1[nH]c2ccccc2o1)OCCN(C(C1CC(C)OCC1)=O)C N1(C(CCC)=O)CC2CCCC(C1)N2C(c1nc2c(C(F)(F)F)cccc2s1)=O N1(C(Cc2cc(OC)no2)=O)CC(C)CCC1CNC(=O)Cc1ccon1 C(=O)(C1=CN=C2N=CNN2C1)NC(C)CCCCNC(C1CCSC(C)C1)=O N1(C(C2C(=C)CC2)=O)CCC(F)C(NC(c2cc(C(F)F)ccn2)=O)C1 C(=O)(C(C(C)(C)C)n1ccnn1)NCC(CNC(C1CC(OC)C1)=O)C c1(N(C(C)CNC(c2cccc(F)n2)=O)C)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] N1(C(C2(OC)CCC2)=O)CC2CCC1C1CN(C(=O)CNC(C3CCC3)=O)CC21 C1(C(=O)NCC(C(C)(C)C)NC(C2CNC(=O)N2)=O)CC2CS(=O)(=O)CC2C1 c1(C(=O)NC2CN(Cc3ccc(O)cc3Br)CC2F)cc(Cl)nc(Cl)c1 N1(C(C2N(C(C)C)C(=O)CC2)=O)CC2=C(C1)CN(C(=O)CN1CCCC1C)C2 C1(C)(CNC(CN(C(C)=O)C)=O)CCN(C(C2CC3CC2C3)=O)CC1 c1(C(=O)NCC(=O)N(C2CC=CC2)C)c[nH]c(C#N)c1 C(=O)(C(C)(F)C(=O)N1CC2(C1)CN(C(=O)CC1CN(C)C1)C2)OCC Cc1cn2cccc(C(=O)NCC(C)N(C)C(c3cccc(C)c3C)=O)c2n1 N12CCN1CC21CCCC1.C1CCOCC1F.O=CNCC1CC1 CCCC(O)CC(=O)NCC(Cc1ccccc1)NC(=O)Cc1cc(C)no1 c1(C(=O)NC2CCN(C(C(C)(CO)OC)=O)C2)ccc([N+](=O)[O-])c(C#N)c1 C1(COC)(NC(=O)Cc2ccc(C)nc2)CCN(C(C2CCN2S(C)(=O)=O)=O)C1 CC(CC(N)=O)C(=O)NCCCC1N(C(=O)CC(C)C2CCCO2)CC1 CC(C)CC(O)C(=O)NC1CCC(F)(C(=O)O)C1 S(=O)(=O)(c1ccc(S(=O)(=O)N2CCNC(C)C2C)cc1)NC c1(C(N2CCC(NC(Cc3c(C)cccc3F)=O)C2)=O)ccc2c(c1)CC(=O)N2 N1(C(C#CC(=O)N(C)C)=O)CCC2(CC(NC(=O)C=Cc3cncn3C)CO2)C1 N1(C(C#CC)=O)CCC2C(CCN2C(c2ccncc2Cl)=O)C1 c1(CC)cccc(CNCC2N(C(C3(CC)CCCCC3)=O)CCC2CC)c1O C=Cn1cc(CN(C=O)Cc2cccc(NCCOc3ccccc3)c2)cn1 c1(C(=O)OCC)cnc(NC2CCCN(C(=O)Cc3cc(C)on3)C2)nc1OC c1(N2C3(CNC(c4cc(C)cc(C)c4)=O)CC(C2)C3)ccc(Br)c(C)c1[N+](=O)[O-] c1(C(N(CCOCCNC(C=CC=CCC)=O)C)=O)cc(C)c(F)c(C)c1 c1(C(=O)OC)cc(C)ccc1NC(N1CCC(C2CC3CCC2C3)C1)=O c1(C(=O)NCCC(C(=O)N(C(C)C)CC2CC2)O)ccc2occc2c1 S(=O)(=O)(c1cccc(-c2ccc3ncsc3c2)c1)N1CCS(=O)(=O)NC1 C1(NC(c2n(CC)cc(Cl)c2)=O)CCCC2CN(C(=O)C(C)(O)C(C)C)CC12 Cc1cc(C(=O)NC2(C(N)=O)CCCN(C(=O)OC(C)(C)C)C2)nc(C)c1 c1(C(=O)NCC(C)NC(c2cccc(OCC(F)F)n2)=O)ccc(O)nc1 C1(C(C)=O)CC(CC(=O)NCCN(C)C(c2cccc(Cl)c2)=O)C1(C)C CS(=O)(=O)c1cccc(C(CO)NC(=O)CC(=O)NC2(CC3CC3)CC2)c1 C(N=c1[nH]c(=N)[nH]c(=NC2CCC3(CCCC3)C2)[nH]1)C1(C(=O)OC)CC12CCC2 N1(C(CC(CCC)O)=O)CC(NC(c2ccc3occc3c2)=O)C2(CCC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)NCC(N(C(=O)C(F)C(C)(C)O)C)C1CC1 c1(C(=O)NC2C=CCN(C(c3c(CC)[nH]nc3Cl)=O)C2)cnc2c(n1)CCCC2 C(=O)(CS(=O)(=O)NC1CCC1)N(C1CCCCN1C(=O)OC(C)(C)C)C C1(CCC(=O)NCCN(C(C)C)C(C2CC(=O)N(C)C2)=O)CC(C)(C)CO1 CCCCC(O)CCC(=O)N1CCCC(CNC(=O)CN(CC(=O)NC)C)C1C N1(C(CC)=O)CC(F)(F)CC1(C)CNC(C1CCN(CC(C)C)C1)=O CC(C)C(O)C(C)C(=O)N1CCN(C2CCCN(C(=O)CSC(F)F)C2)CC1 C1(C(N2CC(CCNC(=O)Cn3cc(CO)nn3)C2)=O)(CCOC)CC1(F)F.CC c1(C(c2c(C)n(C)nc2)NC(C2CC(C3CCC3)C2)=O)cc2cc(Br)cnc2o1 c1(-c2n(-c3cccc(CC(NOCC=C)=O)c3Cl)ccc2)cc(F)ccc1OC Cc1ncc(NC(C2CCCN2CCC(C)C)=O)cc1C#N N1(C(CSC)=O)CCCC(C2CCN(Cc3ccnn3-c3cccc(F)c3)C2)C1 c1(OC)cc(C)cc(C=CC(=O)NCCOCCCNC(=O)C(O)CC(C)C)c1 C1(NC(C(C(C)C)C#N)=O)CN(C(c2ncc3ccccn23)=O)CC1C1CC1 c1(CC)cc(Br)c2nc(OC(=O)Cc3cc(SC)c4c(c3)CCO4)sc2c1 c1(C(=O)NC(CC=C)CNC(c2c(C(F)F)n[nH]c2C)=O)cc(N)c(F)cc1F C1(C)(C(N2CC(CC)OCC2)=O)CCN(C(=O)CCc2ccc(C)cc2C)CC1 N1(C(CCOC(C)=O)=O)CCC(NC(c2ncoc2C)=O)CC1C1CC1 N1(C(C2C(CCC)C2)=O)CC2C(CNC(c3cc(C)sc3C)=O)C2C1 C1(C(=O)OC)(NC(=O)CC2(N(C)C)CCCC2)CC(CO)C1.C1(C)CC1 c1(CC)nc(C)c(C(=O)NC2CCOCC2C(=O)N(CC(C)O)C(C)C)o1 C1(CC)CCN(C(=O)C=Cc2cccc(C)c2)C(C(=O)NCCCSC)C1 C1(NC(=O)NCC(C2(OC)CCC2)N(C)C)COC2(CCOC2)C1 C1(NC(Cc2ccc(C)c(Cl)c2)=O)CCC(O)CN(C(=O)CCCCCC#N)C1 C1(CC(=O)N(CC(C)NC(=O)CCn2cnnn2)C)CCCCC1 C(CCCCC(=O)NCC1CC1C(N1CCC(c2ncc[nH]2)C1)=O)OCC C(C(=O)NCC(C)NC(=O)CCn1cc(C)cn1)(C(C)(C)C)SC CC(C)C(C#N)C(=O)N1C2CCC1(CNC(c1n[nH]cc1C(F)(F)F)=O)CC2 Cc1csc2ncnc(Nc3cccnc3C(N3CCOCC3C(C)C)=O)c12 C1(NC(C(C2CCOC2)OCC)=O)CCN(C(c2cccn2C)=O)CC12CCC2 CC1=C(c2ccco2)CN(C(=O)CC2(CN(C)C)CCCCC2)CC1 c1(C(N2CCC(C)C(NC(C3CCC(F)C3)=O)C2)=O)cc[nH]c2nccc1-2 N1(C(C2OCC(C)(C)C2)=O)CCC2(CC1)CC2NC(=O)C(C)(C)N1CCCCC1 c1(NC(c2cnn(C)c2)CC)cc(F)c(N)c(F)c1 c1(C(=O)NC(CC(C)NC(=O)CCc2cnccn2)C)ccc(C2(C)CC2)cc1 C=CC1(NC(=O)C(CO)NC(=O)Cc2cnns2)CCC1 O=C(CCCC(F)F)NCC(CNC(c1cn(CC2CCOC2)nn1)=O)CO C1(N(C(CC)CC)C(c2cc(OCC)ns2)=O)CCCS(=O)(=O)C1 C1(NC(CC=CC(C)(C)C)=O)CN(C(=O)CC2CCCC3(CC3)C2)CC12CC2 c1(CC(=O)NCC(CC)NC(C(CCC)OC)=O)cccc2c1OCO2 c1(C(c2ccccc2)CC(C)NC(CC)(C)C)ccc(Br)s1 N1(c2n(CC=C)c(C(C)(C)COC(C)C3CC3)nn2)CCc2c(OC)cccc2C1 C1(NC(c2cnc(C(C)(C)C)nc2)=O)CC2CC(C1)N(C(=O)C=CC(N)=O)C2 C(=O)(C(C)CCCOC)NCC1(C(N(CCC(F)(F)F)CC)=O)CC1 c1(C(=O)NC(C(C)C)CNC(c2cnc(C3CCC3)s2)=O)ccc2cnnn2c1 C1(CC(=O)NCc2ccc(CC)s2)CC(C)(C)CN1C(c1nc(C)sc1C)=O C(=O)(C(C)(C)C(F)(F)F)NC(CCCC)CNC(C1CCC(O)CN1C)=O N1(C(C(C)(C)CO)=O)CCC(O)C(NC(=O)CCc2ccc(F)cc2)C1 C12(NC(C(C)O)=O)CC(CNC(c3c(Cl)cccc3Cl)=O)(C1)OC2C C1(C(N(C2CC(CCNC(C3C4CC(=O)CC34)=O)C2)C)=O)(CF)CC(F)(F)C1 c1(NC(C(CCCNC(C2CCCCC2O)=O)O)=O)ccc2c(c1)CCC2 c1(C(=O)NCC2(CN(C(COC)=O)C)CC2)ccc(C)c2c1CCC2 c1(C(=O)NC(C)C=CC(=O)NCCCC2CCCCC2)cccc2occc12 C(=O)(C(O)CCC(F)(F)F)N1CCC(CC=C)(NC(C2CCC(O)C2)=O)C1 C1(NC(=O)NC(C)COCc2ccccc2)COC2(CCOCC2)C1 C=CCCCCCCC(=O)N(CCCC(=O)N(CCC=C)CC)C c1(C(=O)NCC(C)(CO)NC(C(CC)CC)=O)cnc2onc(C3CC3)c2c1 c1(C(=O)NC(C(N2CC(O)(CC(=O)N(C)C)C2)=O)C2CCCO2)ccc(O)cn1 c1(NC(C2CCC(CNC(Cn3c(C)ncc3)=O)C2)=O)cc(Cl)cnc1Br C(=O)(CC(C)(C)CCOC)NC(C(=O)NC(C(CCC)O)CO)(C)CO C1(NC(C(C)C(C)(F)F)=O)COC2(CCN(C(c3ccc(F)cc3)=O)CC2)C1 c1(C(=O)NC(CNC(C(CC)C2CCOCC2)=O)CO)ccccc1COC Cc1cnc(C#N)c(NC(c2ccc(NC(=O)CN3CCN(C)CC3)nc2)=O)c1 c1(NC(CC)CN2CCCC2)nccc(=NCCC(C)c2ccccc2)[nH]1 C12(C(N3CCC(CNC(c4c(C)noc4C)=O)C(C)C3)=O)CCCN(CCC1)C2 c1(C(N2CC(CC(C(=O)OC)F)C2)=O)cc2c(F)cc(Cl)cc2[nH]1 c1(C2(C)CC2)ccc(F)c(C(N2CC(NC(C34CCCC3C4)=O)CC(C)C2)=O)c1 C(=O)(C(C)C(O)C(C)C)NCC1N(C(C(c2cccc(C)c2)C2CC2)=O)CC1 Cc1cccn2cc(C(=O)NC3CC(NC(=O)CN=S(C)(C)=O)CC3O)cc12 N1(C(C2C(CC)C2)=O)CCC(CNC(=O)Cn2nc(C(F)F)cc2C)C(C)C1 CC1C(NC(=O)C2=CCCC2)CC2CCC1N2C(=O)CNc1cccc(Cl)c1 Cc1nc(C(C)(F)F)ccc1C(N1CCCN(C(=O)C(C)OCC2CC2)CC1)=O Cc1cc(C(N2CC(C)(C)CC2CNC(C2CCNC(=O)C2)=O)=O)c(O)cc1F N1(C(=O)OC(C)(C)C)CCCC1CCn1cc(CNCC2CCC(=O)N2)nn1 N1(C(CC(CCC)C)=O)CCC(NC(=O)C(CC(C)(C)C)OC)CC(O)C1 C12(NC(c3c(C)occ3)=O)CCC(C1)N(C(=O)C(C)NC(=O)C(C)(C)C)C2 C1(CCC)CN(C(=O)Cn2cnccc2=O)CC1NC(c1sccc1F)=O c1(OC)cc(C)c(-c2c(C)cc(C)o2)cc1S(=O)(=O)N1CCCC(N(C)C)C1 C1(CNC(C2CCN(C)C2)=O)CN(C(=O)NC2(CC(=O)O)CC2)C2COCC2O1.CO c1(OC)nccc(C(N2CC(NC(C3(CF)CCC3)=O)CC2C)=O)c1F C(CC(F)F)(C(=O)NCC12CC(CCO1)C2)NC(c1c(CC)cncc1)=O C12(C(N3C(CNC(CCOC(C)=O)=O)CCC3)=O)CC3CC(C1)CC(CO)(C3)C2 CCC(COC)C(=O)N1CC(CC(=O)NC2C=CC(C(=O)NC)C2)C(C)C1 CC(C)CC(C(=O)NCC(O)Cn1ccnc1)ONC(=O)CCn1cccc1 c1(C(N2CC(Cc3cc[nH]n3)C2)=O)csc(-c2ccsc2)n1 c1(CCC)nc(C)c(C(=O)NCC2CCCN(C(=O)CC(C)n3ccnc3)C2)o1 C1(C(=O)NC(CCN(C)C)C(=O)N2CC3CC2CS3)CC12CCOCC2 Cc1nnccc1C(=O)NCCN(C(C1CC2CCC1O2)=O)CC1CC1 N1(C(c2cc(OCC)ncc2)=O)CCCC2(NC(C3CCC(C)(C)O3)=O)CC2C1 C1(NC(C(=O)NCCOC(C)=O)=O)CCC(CN)C1 C12(C(=O)NCC3(C)N(C(C4C(C)=C4)=O)CCC3)CCCCC(=O)N1CCC2 C(=O)(C#CC1CCCCC1)NCC(CCNC(c1c[nH]nc1C1CC1)=O)OC N1(C(c2ccc(NS(C)(=O)=O)cc2)=O)CCC(CO)(NC(=O)C=C2CCC2)CC1 C(=O)(C1CNC(=O)c2ccnn21)N1CC(CSCc2nc(NC(C)=O)sc2)C1 N1(C(CCC=C)=O)CC(CNC(=O)CC2COC(C)(C)CO2)C(C)(C)C1 CC1(C)C(CC(N2CC(O)CC2CNC(c2cnco2)=O)=O)C1(C)C CC1CN(CCN2CCC(N(C)Cc3nccn3C)CC2)CCO1 c1(C2(C)COC2)nocc1C(=O)NCC1(NC(C2CC(=O)N2)=O)CCOC1 C(=O)(C(C)N=[N+]=[N-])N(C(C)C(=O)NCCCCC1CC1)CCC c1(C(N2C3(C(=O)NC4C(CC)CCCC4)CC(C2)C3)=O)nccc2[nH]ccc12 C(=O)(CCCCCN(C)C(C1(CO)CCOC1)=O)NCC(C#C)CC1CC1 C(C(=O)NCCC1(NC(=O)C=C2CCCC2)CCCC1)(C(C)C)SCC c1(CN2CCC(C(C(=O)NCC)NC(=O)OC(C)(C)C)CC2)ccc(F)cc1F C=CCN=C(NCCN1CCCC1=O)N1CCC(Cc2cnn(C)c2)C1 c1(N(CCSC)C)[nH]c(=NCc2cc(Cl)nc(=N)[nH]2)nc2scnc12 C1(O)(CC(=O)NCC(CC)(C)NC(=O)CCCc2cc(C)no2)CCCCCC1 C1(C(N2CC(CC(C)NC(C=COCC)=O)C2)=O)C(C)(C)CCCC1(C)C N1(C(=O)OC)CCCC(NC(=O)C(n2cc(C(N(C)C(C)C)C)nn2)C)C1 CC(C)CC(C(=O)NCCC(C)(C)NC(C1CC1c1ccn(C)n1)=O)C(N)=O C1(CSC)CCCCN1C(=O)C(C(C)C)Oc1ccccc1.C(=O)C(C#N)Cl CCC(C)C(CC(=O)NC)NC(c1cccn2nnnc12)=O C1(C(=O)NC2(C)CN(C(c3sc4ncn(C)c4c3)=O)C2)CCCCC12CC2(F)F C1(C(N2C(C)CC(NC(=O)C(=O)N(C)C)C2)=O)CC2CC(C1)CC(F)(F)C2 C1(C(=O)NC2CCCC2C(=O)Nc2cncc(Cl)n2)CCc2nc[nH]c2C1 C(=O)(C(CC)CCCC)N1CC2(CN(C(CC3(C=C)CCC3)=O)C2)C1 c1(C(N(C(CC)C(=O)NC)C)=O)ccc(CNC(=O)C(C)OCC2CC2)cc1 n1(CC)ccnc1C(C)NC(=O)C(=O)Nc1nc(C2CCCCC2)ns1 c1(N(N2CCCCC(CN=[N+]=[N-])C2)C)cc(N2CCCC2)cc(C(F)(F)F)c1.CC c1(C(=O)NCCCC(=O)N(CCCCCC)C)ncccc1N c1(CN(C(=O)CC2(NC(C3CCCC3)=O)CC2)CC)cnn[nH]1 Cn1nnc2cc(C(=O)NCC(C3CCC3)NC(c3cocn3)=O)cnc12 C(C1C(C)C1(Cl)Cl)=CC(=O)NCC(CCOC)NC(=O)Cc1ccc(F)cc1 O=S(=O)(c1cnccc1NC(CO)CCC1CC1)N1CCCc2sccc2C1 C1(C(N2CC(=C)C2)=O)CC(NC(C2CS(=O)C2)=O)C1(C)C c1(C(N2CCC(C(=O)Nc3c(C)ncc(C)c3)C2)=O)ccc(F)c(F)c1F C1(C(C)O)CCC(C(=O)NCCCCCCn2cc(C3CCCC3O)nn2)CC1 CCC(CNC(=O)C(C)Nc1ccccn1)(CC)NC(=O)Cn1nc(C)cc1C c1(C(=O)OC)cnc(N(C2CCCN(C(=O)C=CCOC)CC2)C)c([N+](=O)[O-])c1 CCC(CCCC(=O)N1CCC(F)(CF)C1)NC(c1nc(C)oc1C)=O c1(C(=O)NCC2(F)CC(NC(C3C(=C)CC3)=O)C2)c(C)nn(CCC)c1Cl C(=O)(C1CCCc2c1ncn2C)OC(c1nnc(C)o1)C N1(C(C(COC)C)=O)CC(C)(C(=O)Nc2cc(C(N)=O)ncc2OC)C(F)(F)C1 C(=O)(CCCCNC(c1coc(COC)n1)=O)NCC(CC)(C)Cl c1(OCC(=O)NCCCCC(CO)NC(C(CC)(F)F)=O)c(C)cc(Cl)cc1C c1(C(N(CC(O)CN(C)C(C2CCCC2CF)=O)C)=O)cc(C(N)=O)cc(F)c1 Cc1nc(N2CCC(C)(C)C(CNC(c3ccc(O)nc3)=O)C2)c2cc[nH]c2n1 c1(C(N(CCN(C(CC(C)OC)=O)C(C)C)C)=O)c[nH]c2cc(C)ccc12 N1(C(CCC)=O)CC(C)CCC1CNC(=O)CCc1ccc(OC)c(C)c1 c1(C(=O)NC(c2ccccc2)C(=O)NCC2CC(C)C2)ccc(=O)n(C)c1 C(C(C(=O)NC(C(C)C)C(C)(C)O)C(C)(C)C)NC(c1cc(C)on1)=O N1(C(C2N(C)CCC2)=O)CCC(F)C(NC(=O)CC(F)F)C1 c1(NC(C)=O)ccc(C(=O)NCC(O)CNC(C2CCCCN2C(N)=O)=O)cc1 C1(NC(Cc2c(C)n(C)cn2)=O)CC2CC(NC(=O)Cc3ccccc3O)C1C2 CC(C)(C#N)CCCC(=O)NCCCC1CCCCN1C(C1CCNC1=O)=O c1(N2CCC(C(=O)Nc3ccc(F)nc3F)C2)nc(C2CC2)nc2ccccc12 c1(C(C(=O)NCC)N(C(c2ccc3c(c2)OCO3)=O)CC)cnc2c(c1)CCC2 C=C1CC2(C1)CC(C(=O)N(CCNC(=O)CS(C)(=O)=O)C1CC1)C2 C1(CNC(C(C(C)C)O)=O)Cc2ccccc2CN1C(C1(C(F)F)CCC1)=O C1(NC(C(CO)N(C)C)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1CO C1(NC(C(CCC)OC)=O)CC2CCC(C1)N2C(C1CCCCC1OC)=O N1(C(c2c(OC)nccc2)=O)CC(c2cccc(OC)c2)C2(CC2)C1 C1(C(=O)NC2C(NC(c3nc(CCC)oc3)=O)CCC2)CCCC(C)(C)C1 C1(CC)CCCCCCN1C(C1CCN(C(c2csnc2Cl)=O)C(C)C1)=O N1(C(=O)CSC(F)F)CC2(CNC(c3c(CC)noc3C)=O)CCC1CC2 N1(C(c2ncc(C)c(Cl)c2)=O)CC(NC(C2CNC(=O)C2)=O)Cc2ccccc21 C1(CC)CCC(C(=O)NCCCN(C(c2cc(Br)n[nH]2)=O)CC)O1 Cc1cc(F)c(C(N2CCNCC2C)=O)cc1-c1cccc(SC(C)(C)C)c1 c1(CC)ccc(C)cc1NC(C1(C(C)C)CCN(C(=O)CCC2CC2C)C1)=O C1(C(N2CCC3CN(C(c4ccnn4C)=O)C3C2)=O)(OC)CCC(F)(F)CC1 C1(NC(C(C)CO)=O)CN(C(c2cc(C3CC3)cs2)=O)C2(CCC2)C1 c1(C(=O)NCC2N(C(C3C(CC)C3)=O)CCC2)cnccc1Cl CC1C(O)CCCN1C(=O)CCCC1(NC(c2cn(C)nn2)=O)CCC1 c1(C(=O)NCC2CC(NC(C3CC(O)C(F)C3)=O)C2)cc([N+](=O)[O-])cnc1O N1(C(CC2CCC(C)CC2)=O)C2CCCC1CC(NC(=O)CCCN1CCC1)C2 c1(C(=O)NCCN(C(C(C)OCCC=C)=O)C)cnc2nccnc2c1 C1(C(=O)NCn2cc(CC3COC3)nn2)CCCCC1n1cc(CCCO)nn1 C(CCCCC(=O)N1CCCN(CCO)CC1)N(C(C(CCC)NC(N)=O)=O)C CN=c1cc(C(N2C3CCC(C3)C2C(=O)NC2COC(C)(C)C2)=O)cc[nH]1 CC1(C)CCCC(C(N2CC3(CCCCN3C(=O)CCNC(N)=O)C2)=O)CC1 N1(C(CN(C)Cc2nccn2C)=O)CC(NC(C2CCCS2)=O)C(C)(C)C1 C=CC(O)C(=O)N(C)CCNC(c1cnc(N(C)C)o1)=O c1(CN2C(C(=O)NCc3cn(C)nc3)CC3CC32)cc(F)c(Br)c(F)c1 c1(C(N(C2CCCN(C(c3nc(C)sc3)=O)C2)C)=O)cc2n(n1)CC(C)NC2=O CCCC(CCC)CC(=O)NC1C(C)CN(C(c2ccsc2)=O)CC1C c1(C(N2CC(C)(NC(c3cc(CCO)on3)=O)C2)=O)[nH][nH]c(=N)c1Br N1(C(C2(C)CCC2)=O)CCCC(O)(CNC(c2cncc(C#N)c2)=O)C1 CC1OC2(C(=O)NCC3(CCNC(C4(C)CC4(F)Cl)=O)CC3)CC1C2 CC(C)CC(CNC(=O)C=Cc1ccsc1)C(=O)NCC1(C)CC(C)=NO1 C=CC1COCCN1C(=O)COC1CC(NC(=O)C(SC)SC)C1 n1(CC(=O)NC2C(C)CCN(C(c3ncn(C)n3)=O)C2)nc2ccccn2c1=O Cn1ncc(C(=O)NCC2CN(C(=O)CC3CC3)C3(CCC3)C2)c1S(N)(=O)=O N1(CC(=O)NCCCC2C(C=C)C2)CCCC(NC(=O)C2CC2)C1=O C1(NC(C2C(OCC)C2)=O)CC2(C1)CN(C(=O)CCc1csnn1)C2 C(C)(CNC(=O)COC1CN(C(=O)COC2CCC2)C1)(C1(C)CC1)OC c1(C(N2CC=C(C(N3CC(C#C)OCC3)=O)C2)=O)ccc([N+](=O)[O-])nc1 N1(C(C=CC)=O)CCCC(C)(CNC(c2cc(-c3ccns3)on2)=O)C1 C1(C#N)(C(=O)NCC2N(C(c3n(CC)ccn3)=O)CCCC2)CC2C=CC1C2 c1(C(=O)NCC2(CCNC(C(CC)O)=O)CC2)cc2c(s1)CCC(C(C)C)C2 Cc1ccc(CN2CCCC(C(N3CCC(OC(F)(F)F)CC3)=O)C2)c(F)c1 C1(NC(c2ncc(CC)nc2)=O)CN(C(c2ccc(N)c(Cl)c2)=O)CC2(CC2)C1 N1(C(Cc2cc(OC)no2)=O)CCCN(C(=O)CC(C)c2cnn(C)c2)CCC1 c1(N(CCCNC(c2ccc(CN3CCOCC3)o2)=O)CC)ncnc(=N)[nH]1 CC1CN(C(=O)CCCCC2CC2)CCC1CNC(c1cc(C(C)(C)C)n[nH]1)=O CCCCC(C(=O)NCCC[Si](C)(C)C)NC(c1ccccc1CC#N)=O Cc1cccc(C)c1CN1CCCC1C(=O)Nc1ncccc1-c1ccccc1 CCCCC(C)C(=O)N(CCCNC(=O)CCC(C)(C)C)C1CC1 c1(-c2cc(NC(C)=O)c(F)nc2)nc2c(s1)CCN(C(C1(O)CCOCC1)=O)C2 C1(CC(N2CCC(F)(CNC(C(CCC)=CCC)=O)C2)=O)NC(=O)CNC1=O N1(C(c2ccc(C)s2)=O)CC(NC(=O)C(=O)NCCN(C)C)CC12CCC2 c1(NC(C(=O)NCC2(C)CCCS2)=O)cc(F)ccc1Cl c1(C(=O)NC(CNC(C2(COC)CC2(F)F)=O)C(C)C)ncc(C)cc1C CCC(C)(C)C(O)C(=O)N1CCCCC1C1CCCN(C(c2csnc2C)=O)C1 Cc1ccc(NC(=O)CSC(F)F)cc1S(=O)(=O)Nc1ccc(Br)cc1 c1(CC(N2CCC(C)(NC(C=C(CC)CC)=O)CC2)=O)nc2cccc(F)c2[nH]1 c1(C(=O)NCC2(F)CN(C(c3cncc(C#C)c3)=O)C2)cnc2n1C(C)CCC2 C1(F)(CNC(CN2CC(C)C2)=O)CC(NC(C2(Br)CC2)=O)C1 c1(OC)ccc2c(c1)C(NC(=O)C(C)Cc1ccc(F)c(Cl)c1)CC2 C1(NC(=O)Cc2noc(C(F)(F)F)n2)CC2CCC1(CNC(c1cccs1)=O)C2 Cc1[nH]c(C(N2CCN(C(=O)CC3CCOC3)CCC2C)=O)c(C)c1S(N)(=O)=O N1(c2ccnc(NC(C)Cc3ccco3)n2)CCCC2(CCOCC2)C1 C1(CC(=O)NC(CCC2CCC2)C(=O)N2CCOC(C3CC3)C2)CCCC12CC2 c1(C(N2CC(NC(C(COC)O)=O)C(C)C2)=O)sc2ccc(F)cc2c1C N#Cc1ccc(C(=O)NC2CCC(NC(C3Cc4cscc4C3)=O)C2)c(F)c1 CC1CCN(C(=O)CCCc2ccsc2)CC1NC(=O)Cc1ccon1 C(=O)(C(C)(C)C(C)O)NCC1C(NC(c2ccc(CSC)cc2)=O)C1.C1(C)CC1 C1(NC(c2nn(CC)nc2C)=O)CC2CC(NC(=O)Cn3cc(C#N)cn3)C1C2 C1(C)(C(=O)NC2C(C(=O)NC(c3nc(=O)o[nH]3)C)OCC2)CCCN1C c1(NC(C2C(CNC(=O)C=Cc3ccccc3)CCC2)=O)cc2nncn2cn1 N1(C(C(C)SCC)=O)CCOCC(CNC(c2ccc(=O)n(O)c2)=O)C1 c1(OC)ccc(C(=O)NCC(O)CNC(c2cccc(O)c2Cl)=O)c(Cl)n1 C(C(=O)Nc1cnn(C)c1)(C(C)C)n1ccc(C)c1.C12(CCC1)CNC(=O)CO2 N1(C(c2c[nH]cc(C)c2=O)=O)CC2=C(C1)CN(C(c1nccn1C)=O)C2 S(=O)(=O)(c1cnc(N2CCCC(O)CC2)c(Cl)c1)NCc1c(C)cncc1 C(=O)(CC(C)NCc1cnn(C)n1)NCCCN(CC)CC C1(NC(c2cnc(CC)o2)=O)C2CC3C(C2)C13C(=O)NC(c1cc(C)on1)C CCC(C(=O)N1CCC2(CCN(C(c3csc(CO)n3)=O)C2)C1)C(C)(C)CC N1(C(C=COCC)=O)CC(CNC(=O)C(C(C)C)Nc2nccs2)C(C(F)F)C1 C1(CNC(C(C2CCC2)NC(C)=O)=O)CN(C)CCN1C(=O)CCC1(C)CC1 c1(COC)cncc(C(=O)NCC2CC(NC(c3cn(C)nc3Cl)=O)C2)c1 C1(CNC(c2cc(C)on2)=O)CN(C(=O)CSC(F)F)CC12CCC2 N1(C(C2C(OCC)C2)=O)CC(NC(c2ccc(O)c(CO)c2)=O)CC(O)C1 C1(C(=O)NCc2cc(C(=O)NC(C)Cn3cc(C)cn3)no2)(CC)CCCO1 N1(C(CCNC(C2(C)CCSCC2)=O)=O)CCc2ccccc2C1 CCC(CC(=O)N1CCC1C(=O)NCc1cc(C)nc(C)c1)CC(C)C C=CCC(CC=C)C(=O)NC(C(=O)NCc1nncn1C)c1ccco1 c1(C(=O)OC)ccn(CC(=O)OCCC2CC2(Cl)Cl)n1 CON1CCC(CC(=O)NCC(C)(O)CNC(=O)CCn2ccnn2)CC1 c1(C(N(CCC)CCNC(c2cc(Cl)ns2)=O)=O)cc2c(C)cc(F)cc2[nH]1 C(c1ccccc1F)=CCC(=O)NCC(CCCC)NC(c1ncncc1Cl)=O C(=O)(C(C)(C)CN1CCCCC1)NC1(C2N(C(CNC(C)(C)C)=O)CCC2)CC1 N1(C(c2c(C)ncc([N+](=O)[O-])c2)=O)CCC(C2CCCN(CCF)CC2)CC1 C(C(CC(=O)N1OC2C=CC1CC2)C1CCC1)NC(c1cc(O)ncn1)=O C(C(O)CCNC(C1CCCC1C)=O)NC(C(OCC)OCC)=O Cc1nc(-n2nc(CCCO)nc2-c2cscc2Cl)n(C)n1 C(=O)(C(C)CCNC(C1CCC(C)N1C(=O)CCn1cnc(=N)[nH]1)=O)OC C1(N(C(C=CCCC(C)C)=O)C)CCCCN(C(=O)CN2CSCC2=O)C1 CC1CCCN(C(C2(CNC(c3cnn(CCOC)n3)=O)CCCCC2)=O)C1 N1(c2c(OC)cnc(Cl)n2)CCCC2(NC(c3cnc(C)[nH]3)=O)CC2C1 Cc1ccc(CCNC(=O)CNC(c2nc[nH]n2)=O)nc1 Cc1cc(NC(=O)NC2CC(C)(OCc3ccccc3)C2(C)C)c(Cl)cc1Cl S(=O)(=O)(c1cnn2ccc(=NCC(c3cccs3)N(C)C)[nH]c12)N(C)CC C(C)(C)(C(=O)NCC(C)CNC(=O)CN1CC2CC2C1)OC(C)C C(=O)(CCCN(C(=O)C(C)(C)c1ccn(C)n1)C)NCC(CC1CC1)OC N1(C(C(C)N(CC)CC)=O)CC(C)(C)OCC1CNC(=O)CSC(F)F C1(CC(=O)N(C)CC2(CNC(=O)CCc3ccsc3Cl)CC2)CC2CC2C1 O=C1CC(C(=O)NC(Cc2cc[nH]n2)C(=O)NCC2CC23CCC3)CC(=O)N1 N(C(=NCCC(=O)N(C)C)NC(c1cnccc1C(C)C)C)C(C)C c1(C(c2nnnn2CCCSC)NCC(=O)OCC=C)sc(Br)cc1C C1(NC(c2cnc(C(C)(C)C)s2)=O)COC2(CCN(C(=O)CC3CCOCC3)C2)C1 C(CC(C(=O)Nc1cnc(SC)nc1)NC(=O)C(F)F)OCC c1(C(N2C(C)(CNC(c3ccc(Br)o3)=O)CCC2)=O)nc2ccccn2c1F C(=O)(CCC(CC)OC)N(CCCC(=O)N(C(C(CC)(C)C)C)C)C c1(C(=O)NCCCOCCNC(C2C(C)OCCC2)=O)cccc2[nH]cc(Cl)c12 Cc1cc(C(=O)NCC23CC2CN(C(c2ccoc2Cl)=O)C3)cc(C)c1F C1(CNC(C(C)=C2CCC2)=O)(NC(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)CCCC1 N1(CC(=O)N(C)CCNC(c2cn(C3CCCC3O)nn2)=O)OC(C)(C)CC1=O C1(C(=O)NC(C2(O)CCN(C(c3cc(C)sn3)=O)C2)C)CN(C)CCN(C)C1 c1(C(N(C)CC2CCN(C(=O)COCC3CCC3)C2)=O)cc2ccoc2cc1F C(=O)(C1=C(Cl)CCOC1)NC1CCN(C(C(C)CC(F)F)=O)C1(C)C c1ccc2c(c1)CCCC2CNCc1nnnn1-c1ccc2c(c1)OCCO2 C(=O)(C1=CCSC1)NCCC(=C)CNC(c1csc(C(N)=O)n1)=O c1(C(=O)NC2CCC(NC(c3c(CC)ccs3)=O)C2)cccc2c1COCC2 c1(C(=O)NC(CC=C)CNC(=O)C(F)=CCC)ccc2ccc(Br)cc2c1 c1(C(C(=O)NCC(C)C)N(C2CCSC(C)C2)C)nc2c(s1)CCCC2 C1(C(=O)OC)CCCCN(C(=O)C(c2cccnc2)NCCC(F)(F)F)C1 c1(NC2(CNC(=O)C(c3cccc(Cl)c3)O)CCOC2)c(Cl)cncc1[N+](=O)[O-] C1(CNC(c2ccc(OCC)cc2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1C c1(C(N(C2CC(NC(c3ccc4c(n3)CCC4)=O)C2)C)=O)ccc2occc2c1 N1(C(C2C(C)=C2)=O)CCCC(C2CN(C(c3ccc(S(C)=O)cc3)=O)C2)C1 C1(CNC(CC(C(C)C)C)=O)CN(C(=O)Cc2ccns2)CCC1(F)F N1(C(c2ccc(SCCC)cc2)=O)CC(NC(=O)COCCN(C)C)CC(O)C1 c1(C(=O)Nc2ccco2)nccc(C2CC2)n1.O=C1C=CSCCC2CCCN12 C(=O)(C(C)(C)C(=O)N(C)CC1CCCC(NC(c2ncn(C(C)C)n2)=O)C1)NC CCC(CC(=O)N1CCC(N(C)C(C2CCNC2)=O)C1)OC Cc1nnc2n1CCCC2C(=O)NCC(C)N(C(=O)Cc1ccsc1)C1CC1 S(=O)(=O)(c1cc(Br)c(F)cc1F)NC12CCC(NC(CCOCCOC)=O)(CC1)C2 C(=O)(N=c1ccc(N)c(C#N)[nH]1)NC(CCC)CCc1ccccc1 N1(C(C(CCC)N(C)C)=O)CCOCC(NC(=O)CCc2ccn(C)c2)C1 C1(C(=O)OC)C2C=CC(CC2)C1C(=O)NC1CCN(Cc2cccnc2)CC1 CC(C)(C)C(O)CCC(=O)NC1CC(CNC(C23CCC(C)(C2)OC3)=O)C1 c1(C(=O)NC2CC2NC(c2ccc(Cl)s2)=O)cnc2n1CCCC2 C1(CC(=O)NC2CCN(C(=O)C=CC(F)(F)F)CC2)CCCC(=O)N1 N1(C(COC2(C)CN(C(C3CCCCC3F)=O)C2)=O)CCC(C)(C)CC1 N1(C(CCC(=O)NC)=O)CC2(CC(OC)CO2)C1.N12CC3(CC(C3)CC1=O)C2 c1(NCC2C(NC(=O)OC(C)(C)C)CC2)ccc(C2CC2)o1 N1(C(CN2CC(OCC)C2)=O)CC2CC(C(=O)NCCC3(CO)CCC3)C(C2)C1 CC(C)(C)C(CNC(=O)CN1CC(=O)NC1=O)C(=O)N1CC(C)(C)C12CCC2 c1(C(N2C(C(=O)NOCC(C)O)(COC)C=CC2)=O)coc2ccccc12 CCC(C)CCCCC(=O)NC1CC2CN(C(c3cc(Cl)ccc3N)=O)CC12 C(=O)(C1c2ccoc2CCN1C(c1ncc(Cl)s1)C(=O)NCCCC1CC1)OCC C(=O)(C(C(C)(C)C)C1CCC1)N(C1CCCCN(C(C2(C)CCCC2)=O)C1)C Cc1ccc(C(N2CCC23CCOC3)=O)c(N)n1 C1(CN(CCn2cc(C(C)C3CC3)nn2)C(C(F)(F)CC(Cl)Cl)=O)Cc2nccn2C1 C1(CC)CN(C(=O)CN(C2CCC2)C)CCC1NC(c1cc(OC)no1)=O C(=O)(CCS(N)(=O)=O)N1CCCC(N(C(Cc2c(C)n(C)cn2)=O)CCO)C1 c1(OCC)ccc(S(=O)(=O)N(C)C)cc1NC(=O)NC1CCC(C2CC2)C1 CC1OC2CCC1(C(=O)N(C)CCNC(=O)CCNS(=O)(=O)C(F)(F)F)C2 C(=O)(C(O)CCNC(=O)C=C(C)c1ccco1)NC(C#C)(C)C1CCCC1 C(=O)(C(F)C(C)CNC(C12CC(F)(C1)C2)=O)N(c1cccc(OC)c1)C CCCCC(CNC(=O)CCOc1cccnc1)NC(=O)CCOCC(F)F C(C(F)(F)CC(O)CO)N(C(c1ccc(-c2ccc(C)cc2)o1)C(=O)NCC(C)C)C c1(C(N(CC(C)N(C(c2c(OC)cc(C)cc2)=O)C)C)=O)cc2c(ncn2C)[nH]1 N1(C(C(CCC2CCC2)NC(c2c(C)csn2)=O)=O)CC2(C=CCO2)C1 c1(CN2C(C(=O)NCC(C)(C)CC3CC3)COCC2)cc2ccccc2nc1O C(=O)(CCC(=O)NC1CC2(C1)CC2NC(=O)Cn1nnnc1C)NCC c1(C(N2C3C(NC(CC)=O)CC(C3)C2)=O)cn2ccnc2cn1 C1(C(=O)NC(C)CNC(C2CC(n3ccnn3)C2)=O)CCOCC1(C)C c1(C(=O)NC2CCN(C(CC(CC)O)=O)CC2F)cc(Br)cc2c1cnn2C n1(CC(=O)NC2CCCC(NC(c3cc(OC)ncc3)=O)C2)nc(O)ccc1=O CC(c1cnn(C)c1)=CC(N1CCCC(NC(=O)CC2CCSCC2)C1)=O N1(C(CCN(C)CC)=O)CCOC(C(N2CC(COC)C2)=O)CC1 c1(CC(CN(C)Cc2cc(C3CC3)n[nH]2)=O)ccc(C(F)(F)F)cc1 O=C(C#CC1CCCCC1)NCCSCC(=O)NCC(=O)NC1CC1 c1(C(=O)NC23CC(NC(c4c[nH]c(=N)o4)=O)(C2)C3)ccnc2c1CCO2 C1(C(=O)NCC2CC2C(N)=O)CCCC(CCNC(c2nc(NC)sc2)=O)C1 C(=O)(CCP(C)(C)=O)NCCCCNC(C12CC(C(=O)OC)(C1)C2)=O c1(C(=O)OCC)[nH]cc(C)c1C(=O)NCC(O)CNC(=O)CSCC(N)=O CC(C)C(CN(C)C)C(=O)NCC1(CNC(=O)C2=CCSC2)CCOCC1 N(C(=NCCSC)NC1CC1(C)C(F)F)CC.C12CC1C2 C(=O)(N1CCC(C(N2CC=CC2CF)=O)O1)C1(C)CC(C)C1 c1(C(=O)NC2CCCN(C(C3(N(C)C)CCC3)=O)CC2)cccc2c1OCO2 C1(C(N)=O)CCC(C(=O)NCC2(CNC(=O)CCCC3CCOCC3)CC2)CC1 c1(C(=O)NCCC(C)N(C)C(c2cccnn2)=O)c(O)cnc2ccccc12 C(=O)(CCC1=CCCCC1)NC(C(C)C)CC(=O)NCCc1ccccn1 c1(-c2ccc(NC(c3ccc(OC)nc3C)=O)s2)cnn2c1CNCC2 C1(CC)CCc2nncn2C1.C1(CC(F)F)C(=O)NCCSCCC(=O)N1.CSC C(=O)(CCCC(=O)C1CC1)NCCC(=C)CNC(=O)C(N1CCOCC1)C1CC1 N1(C(=O)NCc2cc(C)nc(Cl)c2)CCN(C)Cn2nccc21 S(=O)(=O)(c1cnn2ccc(N3CCN(CCO)CC3)nc12)N(CC(C)(C)CO)C c1(C(=O)NCCNC(C(n2ccc(C)n2)C)=O)cnn2c1SCC2 c1(CC)onc(C)c1C(=O)NC(CCNC(C1C(SC)CCCC1)=O)C(N)=O C(=O)(CCCCCn1cc(NC(c2ccc(OC)cc2)C)nn1)NCCCCC C(=O)(CCCC(=O)NC1CC2(C1)CC(NC(C1CCOC(C3CC3)C1)=O)C2)OC c1(C(=O)NCCC2CCCN(C(c3ccccc3O)=O)C2)c[nH]nc1[N+](=O)[O-] N1(C(CCN2C(C(c3c[nH]cc(F)c3=O)=O)CCCC2)=O)CCCC(F)(F)CC1 n1(CC(=O)NC2C3CN(C(CCCN(C)C)=O)C2C3)ccc2ccccc2c1=O C(CCC(C)(C)C(=O)Nc1cncc(F)c1)NC(C(N1CCOC1=O)C)=O c1(SCC)ccc(C(=O)NC2CC(C)N(C(c3cnc(OC)cn3)=O)C2)cc1 N1(C(C(C(CC)C)=O)=O)Cc2ccc(C(C)NC(=O)CCC(N)=O)cc2C1 N1(C(c2c(OCCCC)cccc2)=O)CC23COCC2(C1)C3 CCCCC(CC)CC(=O)NCC1CN(C(c2cccc(OC)n2)=O)CCC1C CC(C)CCCCC(=O)NC1CCC(CNC(=O)Cc2cnns2)C1 C(=O)(C(O)CCCNC(=O)C(C)S(N)(=O)=O)NC(CC=C)(C)CC=C c1(C(N2CC(OC)C(NC(=O)C=C(C)I)C2)=O)cc(F)ccc1OC Cc1cnc(C)c(NC(C2C3CC3CN2C(=O)C(C)NC(c2cccs2)=O)=O)c1 C(=O)(C(C)(C)C1CCN(C(C2CCN(C)C2)=O)C1)NC N1(S(=O)(=O)c2nccs2)CCCC2C1CCN2Cc1ccc(-c2ccncc2)o1 N1(C(c2c(C)nns2)=O)CCC2(COC(=O)N2)C1.C12CC(C1)OCC(=O)N2 c1(-c2cn(CCNC(C3C(C)(C(=O)O)C3)=O)nn2)ccccc1SC1CCCC1 c1(C(=O)NC2(CC=C)CN(C(c3cc(C)on3)=O)C2)ccc(OC(F)F)cn1 c1(C(=O)NC(CNC(CCC=C=C)=O)(CC)CC)cnc2n1C(C)CCC2 c1(CC)cc(C(N2CCOCC2CNC(=O)C(C)n2cccn2)=O)c(C)o1 C1(CNC(c2c(NC)cncc2)=O)CN(C(=O)CCC(C)(C)N(C)C)CC1(C)C N1(C(c2n(C=C)ncc2)=O)CC(NC(c2cc(Cl)n[nH]c2=N)=O)CC(F)(F)C1 N1(CC(=O)NCCN(CCC)C(c2ncc(C)s2)=O)CCCC1=O [N-]=[N+]=Nc1ccc(C(N2CC3C(CNC(C4CCSC4)=O)C3C2)=O)cc1 c1(NC(C)=O)ccc(F)c(C(=O)N(CC(O)CN(C)Cc2cccc(Cl)c2)C)c1 N1(C(COCC=C)=O)CCCC(NC(C2C(C)C2(F)F)=O)CC1 c1(NC(c2n(CCOCC)nnn2)c2cnc(CC)[nH]2)ccc(SC)cc1 c1(OC)ccc(C(N2CCC3(NC(=O)CCCC(C)=O)CC3C2)=O)cc1OC Cc1nn(CCO)cc1C(=O)NCCOCCCN(C)C(C1CC=CC1)=O C(=O)(CC1OCc2ncccc21)OC(CCOCC)C(=O)OC C1(NC(Cn2c(CCC)nnc2S)=O)C=CCN(C(C2CCCOC2)=O)C1 c1(NCCCC(N)=O)[nH]c(=NCCc2nc3ccccc3o2)nc2sccc12 CC(C)(C(=O)N1CC2CCC1C(NC(=O)C=Cc1cccc(Cl)c1)C2)C(F)(F)F O=C(C1=CC2(CN(C(c3nc(Cl)cs3)=O)C2)OC1)NCC(O)(C1CC1)C1CC1 C1(CNC(c2cnn(C)n2)=O)CCCCC1NC(C1CCC(C(C)(C)C)O1)=O C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N1CCC(NC(C2N(CC)CCOC2)=O)CC1 n1(CC(=O)NC2CCN(C(C(C)(C)c3cncnc3)=O)C2)cnc(C#N)n1 C1(CC(N2CC(c3cn(C4CCCN(C)C4)nn3)(C(=O)OC)C2)=O)CC2(CC2)CO1 C1(CC(=O)NCCCC2N(C(C(N)=O)=O)CCC2)Oc2ccccc2NC1=O c1(C(N2CC(C(N3CCC4(C(C(=O)NC)C4)C3)=O)OCC2)=O)ccc(F)cc1C CC1(C)CCN(c2ncc(F)cn2)CC1CNC(=O)CSc1cccc(F)c1 CCC(C)(C)CCCC(=O)NCCC(O)CNC(=O)CC1CC=CCC1 c1(C(=O)NC2CCC(NC(CN(C3CCC3)C)=O)C2)ccc2c(c1N)CCCC2 Cc1cc(C(=O)NC2CCC2NC(=O)CCc2ccon2)c2n[nH]cc2c1 C(=O)(C(S(C)(=O)=O)C1CC1)NC1C(NC(C(C2CC(F)(F)C2)OC)=O)CCOC1 C1(C)(C(N2CC(C)C(NC(=O)CCS(C)(=O)=O)C2)=O)CC(O)CN1C C1(NC(C(CCN(C)C)NC(=O)C(F)CC2CCOC2)=O)CC2(C1)CC(C#N)C2 c1(OC)ccccc1CN1CCC(NC(=O)NCCc2ccc(Cl)cc2)CC1 C(=O)(C(C(C)(C)C)NC(c1ccc(CC)nc1)=O)N1C(CCC#C)CCC1 CCC1=C(C(=O)NC2CCC2NC(c2cn(C3CC3)c(C)cc2=O)=O)CCCO1 C(=O)(C1=NN(c2cccc(F)c2)C(=O)CC1)NC(c1ccc(OC)c(Cl)c1)(C)C c1(C(N(C2CCN(C(c3ncsc3C)=O)C2)CCC)=O)ccc2ncsc2c1 CC1CN(C(C2(Br)CC2)=O)CCN1C(C1CN(CC(F)(F)F)C1)=O CCCC(C(=O)N1CC2CCC1CN2c1ccc(C#N)cn1)C(C)C c1(C(=O)NCC(C)NC(C(N2CCCCC2=O)C)=O)cc(-n2cnnc2)ccn1 N1(C(c2cnc(C)nc2C2CC2)=O)CCCC2C1CCN2C(=O)CC1CC12CC2 C1(C(C(=O)NCC(C)(C)CC(=O)O)O)CCc2ccccc2C1 S(=O)(=O)(c1ccc(C(N2CCCC2)=O)cc1)NC(C(C(C)(C)N)O)=O C1(C2(O)CN(C(C3CN(C(N)=O)C3)=O)C2)(CNC(C2OCCC(C)C2)=O)CC1 c1(OC)cc(C)cc(-c2cscc2C(=O)NC(c2ccccc2)C2CC2)c1F c1(OC)ccnc(C(=O)NC(C2(CO)CN(Cc3ccc(C#N)o3)C2)=O)c1OC CN1C(=O)COc2ccc(NC(=O)C(=O)NC3CCC3=O)cc21 C1(CN(C(NC(C2CCCO2)C)=NCc2ccsc2)C)Cc2ccccc2C1 CCC(C)C(C(=O)NCC(C)(C)NC(C1C(F)(F)C12CC2)=O)NC(=O)OC C1(CC(=O)NC(C(=O)NC(CCC)c2ccco2)C2(C)CC2)CCN(C)CC1 C1(NC(CCNC(=O)OC)=O)CCCC(CC(=O)NCC2(C)CC(F)(F)C2)C1 C1(C(=O)NC2CCN(CC(=O)N(c3ccn(C)n3)C)C2)CCCCC1CC c1(C(N2C(C)CCC(NC(=O)COCCOCCO)C2)=O)ccn2cnnc2c1 N(C(=NCC1CCCN(CC(=O)NC2CC2)C1)N(C)CC)Cc1c(C)csc1 c1(SCC(C)(CO)OCC)ccnc(F)c1CO C1(NC(C23CC(OC)C2C3)=O)CCCN(C(c2cnc(Cl)c(N)c2)=O)CC1 N1(C(COCc2onc(CC)n2)=O)CC(NC(c2cncc(C)n2)=O)C(O)C1 C(CC(=O)NCc1sc(C)cc1C)(C(F)(F)F)NC(C(CC)n1cncn1)=O C=CC(C)CC(=O)N1CCC1C(=O)N(CC(=C)C)CCO.C1(C2CC2)CCCCO1 C=CCC(CC)C(=O)NC(C1CC1C(=O)NCC(C)N(CC)CC)C N1(C(C(C)OCCOC)=O)CCC2CC1CN2C(c1cc2ncccc2[nH]1)=O N=c1[nH]c(N2CC3CC(NC(=O)CCCNC(N)=O)C3C2)ncc1[N+](=O)[O-] c1(C(=O)NCC(=C)CCNC(c2nccn2C)=O)onc2ccccc12 C(=O)(C(CC1(C(F)(F)F)CC1)NC(=O)C(C)N)NC C(=O)(C(C(C(C)C)NC(=O)OC(C)(C)C)N(c1ccc(C)cc1F)C)NCC C1(CC)(CC)CCN(C(=NCCC2=CCOCC2)NCc2cccs2)C1 Cc1nc(CNC(=O)N(CC(C2CCOC2)O)C)nc2c1CCCC2 c1(C(=O)NC2CCN(C(CCc3nc(C)sc3)=O)C2)cc(S(N)(=O)=O)sc1C C(=O)(CCCC(C)(C)C#N)N(CCC(=O)NC1CCCC(O)CC1)C CC1CCS(=O)CCN1C(=O)C=C1CCCCC1 C=CCCC(CC(C)C)C(=O)N1CCC(OCCNC(=O)C(CC)(CC)CC)C1 C(=O)(C(C)CC(=O)c1ccccc1F)N1CCCC(c2c(OCC)cccc2)C1 c1(C(=O)NC(C(C)NC(c2ccc(CC)cc2)=O)(C)C)cc(C)cc2c1OCC2 C#CCCCCCCC(=O)N1CCCC1C=CC(=O)N(CC(C)O)C CC1CN(C(=O)Cc2cncc(O)c2)CC1CC(N1CCOCC1C(C)(C)C)=O c1(C(=O)NCCOC2CN(C(C(C3CCOC3)OC)=O)C2)ccc(Cl)o1 c1(OC)cc(N)c(F)cc1C(=O)N(C)CCNC(C1C(=O)NN=C1C1CC1)=O N1(C(c2c(N)cnc(Cl)c2)=O)CCCC2(NC(=O)Cn3ncnn3)CCCC12 N1(C(C(C=C)(C)C)=O)CCC(N(C(=O)CCC(C)(CC)CC)C)C(C)C1 C1(CNC(C(C)(C)N2CCC2)=O)CC(F)CN1C(=O)COc1cccnc1 c1(C(=O)NCC2(OC)CCN(C(C3CN(C)C3)=O)C2)ccc(C)c2ccccc12 C(=O)(CS(=O)(=O)C1CC1)N1CCCC2(C1)C(=O)NC2.C1(=CC(=O)OC)CCCC1 CCC(CC(=O)N(CC(=O)NOCc1ccccc1)C(C)C)C1CCC1 CC1CC(C(=O)NCC2(C)CSC2)CN(C(c2nnc(S)n2C)=O)C1 c1(OCC(=O)N(CCNC(C2CC(Cl)(Cl)C2)=O)CC)ccccc1Br S(=O)(=O)(c1cc(C)cnc1NCC1(CO)CC2CCC1CC2)N(CCCSC)C C1(C(N2CC(O)(CCNC(C=C(CC)C)=O)C2)=O)CC2C=CC1C2 C(=O)(C1=CCN(C(=O)OC(C)(C)C)C1)NCC1N(C(C=CCOC)=O)CC1 c1(C(=O)NC(CN2CCN(C(C)C)CC2)(C)C)cnc2ccccn2c1=O CC(C)(CO)C(=O)NC1CC(NC(C2CCNC2c2ccccc2)=O)C1 n1(C(C)CNC(=O)C(=O)NC2CCNCC2)nccc1-c1ccccc1 c1(OCC)cc(C(=O)NC(C)(C)C(C)NC(C2CC23CC3)=O)on1 c1(CC(N2CC(CNC(C3C(COC)CC3)=O)C2)=O)c[nH]c2cnccc12 CCCC(CCc1ccccc1)C(=O)NC1C(O)CC1O C(CCC(C)(C)NC(=O)CCc1scnc1C)NC(CSCC#C)=O C1(NC(c2c(CC)scc2)=O)CN(C(=O)C(c2ccc(F)c(F)c2)O)CC12CC2 c1(C(=O)NC(CC)CN(C(=O)C(O)CF)CC)ccc2c[nH]nc2n1 CC12COCC1CN(C(=O)C(=O)Nc1cncc(F)c1)C2 N1(C(C(CC)Cc2cn(CCC(C)=O)nn2)=O)CCC(C(F)(F)F)(N(C)C)CC1 C1(C(=O)NC2CN(C(c3c(COC)cco3)=O)C(C)C2)CN(CP(C)(C)=O)C1 C1(C(N(c2cccc(O)c2)CC)=O)CCN(C(=O)COCC2CCCC2)C1C c1(Cn2cc(C(CCC(C)C)NC(=O)OC(C)(C)C)nn2)cc(I)ccc1Cl N1(C(C(C)OCC(C)C)=O)CC2CC1CN(C(=O)Cc1noc3ccccc13)C2 C1(N=[N+]=[N-])(C(=O)NCC(C2CC2)NC(C2N(CCC)CCCC2)=O)CCOCC1 c1(OC)ccc2cc(C(=O)OCc3nc(C(C)(C)C)co3)sc2c1 COC1CCOc2c(OC(=O)CCN3CCC(F)(F)C3)cccc21 N1(C(C2CC(OC)(OC)C2)=O)CCCN(C(=O)CCC2CCCOC2)CC1 C1(C)(CC)CCC(C(N2CC3(NC(=O)C(=O)NC)CC2C3)=O)O1 C(=O)(CCC(C)CN(C)C)NC(c1nocc1C(N1CCC(OC)C(F)C1)=O)C N1(C(c2ccc(F)cn2)=O)CCC2(CC1)CN(C(C1CC1c1ccccc1)=O)C2 C1(CNC(C2(OCC)CCOC2)=O)CCC12CN(C(=O)CN(C)CCO)C2 Cc1nsc(N)c1C(N1CC=CC(NC(=O)C=C2CCN(C)CC2)C1)=O C1(C2CCN(C)CC2)(NCCCc2cccc(C)c2)CC1 n1(CC)ccc(C(=O)NCC2(NC(c3cc(C(F)F)no3)=O)CCOC2)n1 C1(CC(=O)N(C(c2ccccc2)C(=O)NC(COCC)CO)CC)CCN(C)C1=O CC1CCn2ncc(C(N3CCN(C(c4cncc(N)c4)=O)C(CO)C3)=O)c2C1 C1(NC(C(C)CC2CC2)=O)CC2(C1)CC(NC(=O)C(c1cccnc1F)(C)C)C2 N1(C(C(C)SCCCC)=O)CCC(CCN(C)C(C2(O)CCOC2)=O)CC1 N1(C(C(C2CCCC2)NC(C(C)NC=O)=O)=O)CCCN(C)C(=O)C1 C1(C(=O)NC(CNC(C)=O)(C)C)CCCCCC1NC(=O)C1=CCSC1 n1(CC)cc(C(=O)NC(CN(C)C)C(=O)NCCNS(C)(=O)=O)nn1 N#Cc1cc(S(=O)(=O)NCC2CCCCC2)ccc1NCc1c[nH]c(=N)s1 N1(C(CCC(C)O)=O)CC2(CCOCC2)CC1CNC(=O)C(C(C)C)NC=O N1(C(N(C)C)=O)CCCC(NC(C2CCCCN2c2ncc(I)cn2)=O)C1 CC1CN(C(=O)NC(C(CSc2ccccc2)(F)F)C2CC2)C(C)CCO1 C1(NC(c2scc(C)c2)=O)CC(F)(F)CC1NC(c1cncc(O)c1)=O CCCC(C(O)C(=O)N1CC(N(C)C)C(C)C1)NC(=O)Cc1ccc(C)o1 C1(NC(C2CC(NC(C(NOC)=O)=O)C2(C)C)=O)CCCCC1N=[N+]=[N-] N1(Cc2cc(C(=O)OC)nn2C)CC2(CC=CC(=O)C2)C1 c1(NC(=O)OC)ccc(C(=O)NC2CC(CNC(=O)Cc3csc(C)n3)C2)cc1 [N-]=[N+]=NCCCCCC(=O)NCC1CCCC1C(=O)NCC1(O)CC=CC1 CC1=NOC(C)(C(=O)N(CCCNC(C2CC(C)N(C)C2)=O)C)C1 N1(C(C(CCOC)NC(c2ccc(OC)cc2)=O)=O)CC(F)CC(F)C1 C1(NC(CNC(CC(C)C)=O)=O)CN(C(=O)C(c2cc(Cl)ccn2)(F)F)CC1O C1(C(=O)NC(CNC(c2cc[nH]c2C2CC2)=O)C2CC2)(OC)CCC12CCC2 C1(CCOC)CN(C(C2(Cl)CC2(F)F)=O)CCN1C(=O)CCc1ccsc1 N1(C(Cc2c(C)cco2)=O)CCCN(C(=O)CCC2CC2(F)F)C(C)C1 N1(C(c2nc(C(C)=O)sc2)=O)CCC2(CCC2NC(C2CC(=C3CC3)C2)=O)CC1 C(=O)(CCCC(=O)N1CCOC(C(=O)NCCNC(N)=O)CC1)NCCC c1(CC)cnc(O)c(C(=O)NC(C)CCN(C(=O)CC2CCC(C)(C)C2)C)c1 c1(C(=O)NC2CN(C(c3n(CC)nnc3)=O)CC(O)C2)ccc2c(c1)CC(=O)N2 N1(C(c2c(C)ccs2)=O)CCCCC1CC(=O)NCCOc1ccccc1 N1(C(CC2C(C)OCC2)=O)CC(O)(C2(CNC(=O)CCC(F)(F)F)CC2)C1 C1(NC(CCCN=[N+]=[N-])=O)CC2CN(C(c3ccc(=N)[nH]n3)=O)CC2C1 c1(NC(C23CC(C(NC4=NCCS4)=O)(C2)C3)=O)ccc(-c2ccccc2)nc1 C1(NC(C=NOC)=O)CC(C)CN(C(c2csc(Br)n2)=O)C1 CC1(C)CN(C(C2(C)CC3CC3C2)=O)CCC1NC(=O)CN1CC=CC1 C1(C(=O)NC(CCC)C(N)=O)CCC2(CC2)N1C(c1ccnn1CC)=O c1(C(=O)NC2(C(=O)NC(COC)C3(C)CC3)CC(F)C2)c(C)nn(C)c1N c1(CC)cnccc1CNC(=O)CC1(NC(c2conc2C(=O)OC)=O)CC1 n1(CCC(=O)N(CCN(C)C)CC2CC2)cnc2c(N)ncnc12 N1(C(c2cc(C)n(C)n2)=O)CCCC(CCNC(C2CCS(=O)(=O)N2C)=O)CC1 C#CCCC(O)C(=O)N(C1CCN(C(=O)C(C)(F)F)C1)CC C=CCCCCCC(=O)NC12CCC(CNC(C3CCCN3C(=O)CC)=O)(C1)OC2 C12(C(=O)OCC)CC3CC(CC(NC(=O)C(c4ccc(C)c(Br)c4)C)(C3)C1)C2 C1(C(=O)NCC(C)NC(c2ccc(CF)cc2)=O)CSc2ccccc2O1 Cc1c(C(=O)NCC2(NC(C3CCN(C)C3)=O)CC3CCC2C3)cncc1N c1(C(=O)NCC2CCCN(Cc3c(C)nc(Cl)cc3)CC2)cc(C#N)ccc1O c1(SC)nc(CO)cc(C2(NC3CCCC(F)C3)CCOCC2)n1 C1(NC(CC2N(C)CCCC2)=O)CN(C(c2c(O)cccc2Cl)=O)CCC1(C)C C12(CC(N3C(CN(C(CC(C)SC)=O)C)COCC3)=O)CCC(CC1)OC2 O=C1CCCC(CC(=O)NCCCCNC(c2csc(Cl)n2)=O)N1 Cc1ccc(COC(C)C(=O)NCCOCCN(C(=O)C(F)CN(C)C)C)cc1 CCC(C(C)Cc1ccccc1)Nc1cccc(-c2nc(O)n[nH]2)c1 C1(C(=O)NCCC(C)NC(=O)CSCCC(F)(F)F)OCCOC12CCC2 O=C(C1=CS(=O)CCC1)NCC1CC(F)CN1C(C1CCCN1c1nccs1)=O N1(C(C(CC)O)=O)CCc2c(C(=O)NCc3cnc(C(F)(F)F)nc3)n[nH]c2C1 C=CC(CCC)CC(=O)NCC1CCCN(C(C23CCC(C2)OC3C)=O)C1 c1(NC(C2N(C(c3c(C)cc(C)o3)=O)C(C3CC3)CC2)=O)ccc2nc[nH]c2c1 C1(C2CCN(C(=O)Cc3cn4ccsc4n3)C2)(NC(c2cc(C)c(Cl)s2)=O)CC1 c1(C(=O)NC2CN(C(c3cc(C)c(C)s3)=O)C2)coc2c(C)cccc12 N1(C(C(c2cc(F)c(F)cc2Br)CC)=O)CCCC(C2CN(c3nncs3)C2)C1 C1(C(=O)OC)N(C(C2C3CC3CN2C(=O)CN(CC(C)(C)C)C)=O)CC1(C)C C(=O)(CN=c1ccc(Cl)n[nH]1)NC1CC(NC(=O)CC2CN3CCC2CC3)C1 CN1CCC(NC(=O)CC2CCN(C(c3ccccc3CC#N)=O)CC2)C1=O N(C1CC2(CCOC2)Oc2ccccc21)C(C(N1CC(F)(CC)C1)=O)=O C1(NC(CN(C(c2cccc(C)c2)=O)CC)=O)CCOCC1(C)C N1(C(C=C(C)C(C)(C)C)=O)CCC(NC(c2ncccc2C)=O)C12CCC2 C1(CNC(c2c(OC)cccn2)=O)CC2CN(C(=O)C(O)CC3CC3)CC12 C1(CC(N2CC(O)(C(C)NC(=O)CNC(c3ccoc3)=O)C2)=O)CCCC(O)C1 N1(C(C)=O)CCC2OCCN(C(c3ncn4cc(-c5ccnn5C)sc34)=O)C2C1 C=CC1(C(=O)NCC(C)CNC(C2SCCS2)=O)CCCC1 Cc1nccnc1C(=O)NC1CC(C)N(C(C2CCC(N(C)C)CC2)=O)C1 N1(C(CCCOC)=O)CCSCC1CCNCCNC1C(c2ccccc2)C1C C1(C(N2C3CC(CNC(Cc4cc(C)sc4)=O)C2CC3)=O)CCC2CCCCN12 c1(CNC(=O)NC2COCCN(C(COC(C)(C)C)=O)C2)nc2ccccc2o1 CC1CC(C#N)CN(N2CCN(c3ccc(C#N)c(F)c3)CC2)C1 c1(SCC(=O)NCC(CNC(C(C)Cc2ccco2)=O)F)nc2ccccc2o1 c1(C(=O)NCCCC(C)NC(c2c(C)coc2C)=O)coc2c(Cl)cccc12 C(CC(C)C(=O)NCc1ccc(C(=O)NC2CC(C)(O)C2)cc1)=CC N1(C(CN(c2cn[nH]c2)Cc2c(C)cccc2)=O)CCCC(O)C1C(=O)O CC1C(O)CCCN1C(c1ncccc1NC(=O)CCC(=O)N1CCCC1)=O C(=O)(C(C)(C)C)NCCCC1CCCN1C(=O)CSc1ccoc1.CC1C(=O)N1 CCCCC(C)(F)C(=O)NC1CCC(NC(c2cccc3scnc23)=O)C1 C1(C(N(C)Cc2n(CC)cnn2)=O)CCC2CCCCN2C1 C(=O)(C(C(=O)N(CC(C)NC(c1cc(F)ccc1CC)=O)C)C(C)C)OCC c1(C(=O)NCCC2(O)CCN(C(=O)C(F)n3ccnc3)C2)ccc2ncccn12 Brc1cc2c(N3CC4(CN(Cc5cnc6n5CCOC6)C4)C3)ncnn2c1 c1(C(=O)Nc2c(NCC)ccc(Cl)c2)ncc2ccccc2c1O C(=O)(C1CCCc2nncn21)NC1(C)CN(C(C2COC3COCC23)=O)C1 C1(C2(O)CCOCC2)(C(N2CC(CNC(C(C)=C3CCC3)=O)N(C)CC2)=O)CC1 C#CCCCCC(=O)N(CCNC(C1CC(=O)NC(=O)C1)=O)CC1CC1 c1(C(N2C(CC)CN(C(C3(CC(C)C)CC3)=O)CC2)=O)ccc2c(c1)CC(C)O2 c1(NC(C2N(Cc3n(C)ccn3)CCSC2)=O)ccc2c(c1)n(C)c(=O)n2C C1(CNC(CC)=O)C(C)CCN1C(C1CC(C)(O)C1)=O CC12CC(NC(C3CCOC3)=O)(C1)C1(CN(C(=O)CC3CN4CCN3CC4)C1)O2 C1(OC)CN(C(=O)CCc2cocn2)C(C)(CNC(C2SCCS2)=O)C1 C(=O)(CS(=O)(=O)CCSC)N1CC(CC(C(=O)NC(CCCC)CO)F)C1 Cc1cc(C(=O)NC(CO)C(C)NC(c2sccc2F)=O)nn1C(C)C1CC1 C1(C(=O)NC2(COC)CCN(C(=O)Cc3sc(C)cc3C)C2)CC12CCSCC2 N1(C(c2nnc(CCCC)s2)=O)CCC(C2=NOC(C(=O)OC)C2)CC1 c1(Cc2ccc(Br)cc2)nc2ccc(NCC3CCC4(CCNC4)O3)cc2[nH]1 CC(C)CC(=O)NCC(N1CCCC1CN(C(C1OCCC1C)=O)C1CC1)=O CC(C)C(C(=O)NC1(CN(C)C(C2CC(n3ccnc3)C2)=O)CC1)N(C)C C1(C(=O)OC)CCN(C(=O)C2CC2c2cncn2C)O1 C(=O)(CC(C)(C)C(=O)N1CC2CC2(CNC(=O)CCN2CCOCC2)C1)OC c1(C(=O)NC2CC(N(C(C=CCN(C)CC)=O)C)C2)ccc(CO)c(F)c1 C(CCN(C)CC1(C(F)F)CC1)(C(=O)NC(c1ccccc1)C)N(CC)CC N1(C(Cc2nc(C)cc(C)n2)=O)CCC2(CCN2)CC1 C(C(=O)NCC1CCCCN1C(=O)COCCOCCO)(C(C)C)OC C(c1cc(C)c(C)cc1C)=CC(N1CCN(C(CCNC(C)=O)=O)CC(O)C1)=O C1(C(N2C(C)C(NC(=O)CN(C)C)CC2)=O)CCCCC1(C)C c1(C(=O)NCc2cccc(OC(CC)C#N)c2)ncc(C)nc1N1CCOCC1 Cc1cc(=NC(=O)C(=O)N2C3CCC32)[nH]o1.c1(C(=O)NC(C)CC)ccc(F)c(N)c1 c1(OC)cnnc(C(=O)NCC2(NC(=O)C(c3ccccc3)C)CCOCC2)c1 c1(C(=O)NC(C)C(C)(C)NC(=O)CCS(C)=O)ncncc1Br c1(OC)ccc(C(F)(F)F)cc1C(N1CCC(F)C(NC(=O)CCC(C)C)C1)=O C1(N(C)C(C2CC3CC3C2)=O)CCCN(C(c2ccc(CNS(C)(=O)=O)o2)=O)C1 c1(CCC(=O)NC2CC(NC(C(COC)C)=O)CC2O)c(Cl)cncc1Cl C(CCCCC(=O)NC1CCCN(C(=O)COCC(=O)OC(C)(C)C)C1)SC C1(C(N(CCNC(COCC(=O)NC)=O)C(C)C)=O)CSCC(=O)N1 CC1CCCn2ncc(C(=O)NC3CC(O)(CCC(C)(C)C)C3)c21 C1(NC(c2oc(CC)c(C)c2)=O)CCN(C(=O)CC2CCCC(C)(C)O2)C1(C)C N1(C(CSCC=C)=O)CCCC(C2CCCN2C(=O)C=CC(c2ccsc2)=O)C1 CC1CNCCC1NCC1(CCN(C)C)CNC1 c1(C(=O)NCC2COCCN(CCC3CCS(=O)(=O)C3)C2)occ2c1CCC2 C1(CN(C(C=Cc2c(C)cncc2)=O)C)CN(C(c2coc(Cl)n2)=O)CC12CC2 c1(NCC2(NC(C3C(C(C)C)C3)=O)CCCC2)cc(O)nc(O)n1 c1(OC)nc(Cl)cnc1NC(c1cc(F)ncc1-c1cncc(N(C)C)n1)=O N1(C(C(C)=C2CCCC2)=O)CCCC(C(N2CC(N3CCCCC3)C2)=O)CC1 c1(CC)nccnc1CNC(=O)CC1CCCCN1C(C1C=CC1C(=O)OC)=O C1(NC(n2c(C)csc2=O)=O)CC(NCC(N)=O)C12CCC2 CCCCC(C(=O)Nc1cc(Cl)ccc1O)NC(=O)C(CN(C)C)CC C(=O)(CC(O)c1ccccc1)NC(=O)CC1CN(C(CC(C)N(C(N)=O)C)=O)C1 N(C(=NCCCOCC1CCCC1)N1CCC(CCNC(C)(C)C)C1)C(C=C)C N1(C(CCn2c(C)nc(C)n2)=O)CC2CN(C(=O)CC3CC4CC4C3)CCC12 C1(CC(N2CCCC2(C)C2CCC2)=O)C2CCCC2N1C=O.C1(CC)CCC1 c1(C(=O)NCC2CCN2C(=O)C2Cc3c(Cl)cccc32)cc2c(F)ccc(F)c2s1 c1(CCc2nc(OC)nn2C2Cc3cc(Cl)ccc3O2)cc2cc(C)ccc2[nH]1 C1(CC#C)(C(N2CCC(F)(CNC(=O)CN(C)CCO)C2)=O)CC=CCC1 c1(C(N2CC(C)C(NC(=O)CC3CC3(Cl)Cl)C2)=O)ccc(N)c(F)c1F Cc1[nH]nc(C(=O)NCCC2CCCN(C(c3ncccn3)=O)C2)c1[N+](=O)[O-] c1(C(N2CC(F)CC(C(N3CC4CC4C3)=O)C2)=O)cccc([N+](=O)[O-])c1I C=CCC(CC)C(=O)Nc1cccc(NC(=O)Cc2cnc(C)o2)c1 CCCC(CNC(C1COCC(C)O1)=O)C(=O)N1CCC(C#N)C1 C12(C(N3CCC(C)(CNC(C(COC)O)=O)C3)=O)CCOC1CCOC2 c1(OC(C(=O)NC(CC)CNC(c2cscc2OC)=O)C)ccc(F)c(F)c1 Cc1sc(C(N2CC(NC(c3ccn(C4CCOCC4)n3)=O)C(C)C2)=O)nc1O C(=O)(CC(O)CNC(c1cccn1C(C)C)=O)NC(C=C)(C)C N1(C(CNC(=O)NC)=O)CC2CC1CCN2C(=O)C(C)Oc1cccc([N+](=O)[O-])c1 CCC(C)C(C)CNC(=O)CC1CC(NC(c2cncc(C)c2)=O)C1 c1(C(=O)NCC2C(NC(C(CC)OCC)=O)CCC2)cn2cccc(F)c2n1 c1(C(N2CCCC(NC(c3ccc(CC)c(N)c3)=O)C2)=O)cc(S(C)(=O)=O)cs1 C1(C)(C(=O)NC(c2ccccc2CC)CNC(CCC#CC)=O)CC(O)CN1C c1(C(N(CCNC(CCCCC=C)=O)C)=O)cc([N+](=O)[O-])ccc1NC(=O)OC C12(CN=c3cc(C)nc[nH]3)CCCCC1CN(C(=O)C(=O)N(C)C)C2 C=CCC(CC)C(=O)N1CCC(C)(NC(=O)CCSc2ccccn2)C1 N1(C(C2C(OC)C2)=O)CC(NC(C23CCC(C)(CC2)CO3)=O)CC12CCCOC2 N1(c2c(C)cncn2)CC2CN(Cc3cccc(C(C)(C)C)c3O)C2C1 C(C)(CCC(=O)NCC1CN(C(C2CC(F)C(=O)N2)=O)CCO1)OC c1(OC)nc(C)ccc1C(=O)N(C1CC2CC1N(C(c1ccc(C)cc1)=O)C2)C CC1=C(C(=O)NC2(C)CCC(NC(=O)CN3C(=O)CCC3=O)CC2)CCCC1 c1(C(=O)NC(CNC(=O)C#CC2CCOC2)C2CCC2)ccc2nc(O)oc2c1 Cc1cc(CC(C)NC(c2[nH]ccc2CNC(=O)Cn2nccn2)=O)n[nH]1 C1(NC(c2n(CC)ncc2)=O)CCCCC1NC(C1CCCN1S(C)(=O)=O)=O C1(NC(COC)C(=O)NC2CN(C(=O)C3CC3)C2)CC(=O)N(C2CCCCC2)C1 N1(C(CCC2C(C)(C)C2)=O)CCC(C)(C)C1C(=O)Nc1cnccc1CO C12(C(=O)NC(CC)CNC(C3CC34CCC4)=O)CCC(OC)(CC1)C2 Cc1ccc(CN2C(C(=O)Nc3cccnc3CO)CC3CC23)cc1Br c1(C(=O)NCC2C(NC(C3CCN(CC(C)C)C3)=O)C2)cc(O)cc(=O)o1 C1(C(N(CCCCNC(c2cc(C)nn2C)=O)C)=O)CC(C)CCC1C(C)C c1(C(=O)NC(CCCC)C(=O)NC2CC2C(F)(F)F)ccc2c(c1)OCO2 C(=O)(C(C)C(F)(F)F)NCCC1(NC(C(c2ccc(C)cc2)C2CC2)=O)CCC1 CCCC(C)(C)C(=O)NCC1CCN(C(c2c(C)nn(C)c2Br)=O)CC1 c1(C(=O)NC(COC(C)C)C(=O)O)cnc2ccnn2c1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCC2(CC(CNC(C=CSC)=O)C2)CC1 C(C(C)(C)CC(=O)NCC1(CC2CC2)CC1)NC(C(C)CN(C)C)=O c1(C(=O)NC(C)C(CO)NC(=O)CCc2cccs2)cc2n(n1)CCC2 C1(C(=O)NC(C2(O)CN(C(C=C(C)Cl)=O)C2)C)CCCN(c2nccs2)C1 C(C1=NOC2(CCC2)C1)NC(C1(COC)CN(C(c2cc(Cl)ccc2O)=O)C1)=O c1(C(N2CCC(C)(NC(C3CC34CCCCC4)=O)C2)=O)ccc2ncnn2n1 C1(C(=O)NC2CC(n3ccnc3)C2)C2CCC1(c1ccc(C(F)(F)F)cc1)C2 C1(CCC(N2CCC3(C(CNS(C)(=O)=O)C3)CC2)=O)CCc2cnn(C)c2C1 N1(C(C2C(CC)OCC2)=O)CC2CCC1C1CN(C(=O)C(C)(C)CF)CC21 c1(OC)ccc(OC)c(CC(=O)NCC(C)CN(C)C(c2cc(C)no2)=O)c1 Cc1c(Br)ccc(C(=O)NCC(c2ccc(Cl)s2)O)c1F C(=O)(C(C)CC(N)=O)NC(C)C(=O)NCC1(O)CN(C)C1 N1(C(C2N(C(C3(CC)CCCC3)=O)CCCC2)=O)CCCCC(CO)C1 c1(C(N2CCCC(F)(C(=O)OC)C2)=O)ccc2c(c1)C(C1CCOCC1)C(=O)N2 c1(C(N(CC(CC)NC(c2ncncc2F)=O)CC)=O)cccc2cncn12 CC1CC=C(C(=O)NC2CCN(C(C3COC(=O)C3)=O)C23CCC3)CC1 c1(C(=O)NC2CN(C(CCc3n(C)ccn3)=O)CC2O)cn2cccc(Cl)c2n1 n1(CC)cc(Cl)c(-c2nc(CC(C)OC)nn2-c2ccccc2)n1 N1(C(c2c(CC)nccn2)=O)CC(C)(C)CC1C(=O)NCC1COCCN1C CC(O)C(C(=O)N1CC(O)(CCNC(=O)CCC2(C)CC2(F)F)C1)NC(N)=O c1(C(C)C)ccc(C(CO)NC(=O)CCc2cccn2C)cc1 c1(CC(=O)NC2(CO)CCCN(C(C3CC34CC4)=O)C2)c[nH]c2ccccc12 CC1(C)CCCCC1CNC(=O)C(C1CN(C(c2cc(C(N)=O)[nH]n2)=O)C1)N.CCCC C(=O)(C(C)(C)C(C)(C)O)N1C(CC(=O)N(C2COCC2O)C)CCCC1 N1(C(C(C2CC2)OC)=O)CCOCC(NC(=O)CCc2ccccc2C)C1 CN=S(C)(=O)c1ccc(C(N2CCC3CN(C(c4cccnn4)=O)C3C2)=O)cc1 CC(C)CC(C(=O)NC1CC(C(=O)N(CCCN=[N+]=[N-])C)CC1O)C(C)C N1(C(c2c(C)cc(C)s2)=O)CC2CCC1C(NC(c1ccc(F)cc1)=O)C2 C1(C(N2CC(OCCNC(c3c(C)snn3)=O)C2)=O)CC(O)CN1C c1(N(CCCCCC)C)ccc(S(=O)(=O)N(C)C(c2ccccn2)C)c(Cl)c1 N1(C(c2cc(CC)on2)=O)CCCC(CC(=O)NC(C)CCn2cncn2)C1 C(=O)(C(O)CC(F)(F)F)N(C1CCN(C(=O)C(F)CC2CC2)CC1)CCOC c1(OC)ccccc1CN(CCCNC(=O)C(N)=O)C.c1(C)sc(COC)nc1C C1(NC(c2c(C)nc(Br)o2)=O)CC(C)CN(C(c2cnccc2Cl)=O)C1 C1(NC(C2CCN(C(c3sc(Br)cc3Br)=O)C2)=O)CCCCC1C(F)(F)F c1(C(=O)NCC2CC(NC(c3cnc4ccoc4c3)=O)C2)cccc2ccoc12 Cc1cn(C)cc1C(=O)NC1CC(NC(C2CCCC3CC23)=O)C1 C1(NC(c2cccc(C)c2Br)=O)CC12CCN(C(c1cnc(O)nc1O)=O)CC2 CCC(C)C(C(=O)N(C)C)NC(=O)C(c1ncccc1C)(F)F N1(CC(N2C(CC(=O)NC(C(=O)OCC)C3CCC3)CC2)=O)CCCCC1C C1(C(N(CCC#C)CC)=O)C2CC(O)C(C2)N1C(=O)C(c1ccc(C)o1)C Cc1nc2cc(C(=O)NCCCCCCNC(=O)COc3ccsn3)[nH]c2s1 NC1CCC(F)(F)CC1C(=O)NCCCNC(=O)Nc1ccccc1 Cc1nn(C)c(Cl)c1-c1cn(C2CN(C(C3CC4CC3CC4=O)=O)C2)nn1 c1(NC(CCc2n(C)ccc2)=O)ccc2oc(=O)n(C3CC3)c2c1 Cc1cc(C)c(C(=O)NCCC2CN(C(C3C4CCCCC34)=O)CCO2)c(O)c1 Cc1cc(NCCCCC2CN(C(=O)C3=CC4CCCC34)C2)n2ncnc2n1 c1(C(N(C2CCN(C(c3cc(C)c(C)o3)=O)C2)CCO)=O)ncc2ccccn12 c1(-n2cc(CCCCC)nn2)cccc(CCNC(C2(C)CCCN2C)=O)c1 c1(C(N(C2CCCN(C(C(CC)F)=O)CC2)CC)=O)cccc2[nH]ccc12 C(=O)(CC(C)SC)NCC(C1CCCCC1)NC(C(F)=CCC)=O C(CNC(c1cnc(C2CC2)[nH]1)=O)(CC(F)(F)F)NC(Cc1cccc(C)c1)=O C1(CNC(c2ccccc2)OC(Cc2nc(COC)sc2)=O)CC(=O)N(C)C1 Cc1ccc2c(c1)CC(C(=O)N(CC13CCC(CC1)C3)Cc1nn[nH]n1)S2 c1(C(=O)NCCCNC(c2cc(C(C)=O)sc2)=O)cc(O)nc2c1CCCC2 c1(C(=O)Nc2c(C)nc(Cl)cc2)cccc(S(=O)(=O)NCC2CCCCCN2)c1 C1(NC(COC(C)C)=O)CC2CC1N(C(=O)CC1CCCC(=O)C1)C2 c1(NC(C(=O)N(CCC#C)CC)=O)ccc(Oc2ccc(F)cc2)nc1 Cc1ocnc1CC(=O)NCCOC(C)(C)CNC(C1CC(=O)C1C(C)(C)C)=O CC1(CC#N)CCN(C(=O)C(=O)NCC2CC2)C1 C12(CNC(C=CCOC)=O)CCCC1CCN2C(=O)C(=Cc1ccncc1)C C1(CNC(CC(n2c(CC)ncc2)C)=O)CCCCN1C(C1CCCN1C=O)=O C12CCCCN1C(=O)C(CC)OCC2.C=CCCC(=O)Nc1ccccc1 c1(C(=O)NC2CCC(N(C)C(c3cnccn3)=O)C2)cnc(O)c2c1NCCC2 C=Cc1ccc(C(N2CCCC(NC(=O)C(CC)=CC)C2C)=O)cc1 c1(C(N2CCCCC(NC(C(C)S(C)(=O)=O)=O)C2)=O)ccc([N+](=O)[O-])cc1O N1(C(c2sccc2Cl)=O)CC2CC(C1)CN(C(c1c[nH]c3ccc(Cl)cc13)=O)C2 CC1C2C(CCN2C(C2CCOCC2(C)C)=O)CN1C(c1ccnc(CO)c1)=O Cn1cnc2c1CCC(C(=O)NC(CNC(=O)CSCCC#N)C(C)(C)C)C2 C1(NC(CCCCC)=O)CC2CCC(C1)N2C(=O)CN(C)CCOCC(F)(F)F c1(SCCC(=O)NC2C(N(C)C3CC3)CCCC2)ncnc2[nH]cnc12 c1(C(CC)NC(=O)CCCc2cccc(F)c2)ccc(F)c(Br)c1 Cc1ncc(CC(=O)NCC2CCC(C(=O)NCC(C)C#N)C2)s1 S(=O)(=O)(C1CN(C(=O)CC(C)(O)C2CC2)C1)N1CCN(C(CN(C)C)=O)CC1 Cc1ccc(O)c(C(N2CCC(NC(c3cn(C(C)C)nn3)=O)C(C)C2)=O)c1 CCC(O)C(=O)NC1CC(NC(=O)OC(C)(C)C)C1.C12CC(C1)CNC2=O C1(CNC(C(C)(C)CF)=O)CN(C(c2cc3ncccc3s2)=O)C2CCN1C2 N1(C(c2n(C)cnc2)=O)CCC2CN(C(c3ccc(C(F)(F)F)s3)=O)CCC2C1 c1(OC)ccc(O)c(NC(=O)CONC(=O)CC(O)c2cncc(Br)c2)c1 C12(NC(c3c(C)nsc3)=O)CCOCC1CN(C(=O)CCc1ccc(Cl)nc1)C2 c1(C(C)C)nn(C)c(Cl)c1C(=O)NCCCN(C)C(C1CC(N(C)C)C1)=O C1(NC(c2cnc(C)nc2)=O)C(CNC(=O)Cc2ccc(C)s2)CCC12CCC2 C1(C(N(C)CC2(NC(=O)CN3CC4CCC3C4)CC2)=O)COc2ccccc2O1 Cn1cccc1C(=O)C(=O)NCC1CC1NC(C1(CC2CC2)CCC1)=O Cc1ncncc1C(=O)NC(C(=O)N1CCC(C(F)F)CC1)C(C)C Cc1cc(SCC(=O)N(C)CCNC(C2(C(O)CO)CC2)=O)cc(C)c1 CCCCC(CCCC)NCC1CCC(C)CC1NC(=O)OC(C)(C)C C(=O)(C(=O)C(C)(C)C)N1CC(C)(CCC(=O)NCCCc2n(C)ncc2)C1 c1(OC)cc(C(N2CCCC(CN(C(=O)C3=CCCCC3)C)C2)=O)c(F)c(Cl)c1 C1(C(=O)NCC(C)N(CC)CC)CC(F)(F)CN1C(C1CC(=O)CC(=O)C1)=O c1(NC(C2(C)CCN(C(c3c(C)cnnc3)=O)C2)=O)c(O)cccc1O Cc1[nH]nc(CO)c1C(=O)NCC(C)C(=O)NCC(O)CC1CCC1 N#CC12CCC(C(N3CC(OCC(F)F)C3)=O)(CC1)CC2.c12coc(c1)NC2=O c1(NC(C2CC2C(=O)Nc2cnccc2CO)=O)nccn2ccnc12 N1(CC(C)(C)NC(CCc2ncc(C(C)C)o2)=O)CCN(c2cnc(F)cn2)CC1 C1(C(=O)NCC(C)(CO)NC(C=CC(=O)OCC)=O)CC2(CCC2)CCO1 C(c1ccc(Cl)cc1)=CC(=O)N(C)CC1N(C(c2nc(CC)oc2)=O)CCC1 N1(C(C(CCC)(C)CCC)=O)CCCC2(CCCN2C(=O)C(O)P(C)(C)=O)C1 C1(NC(c2c(OC)nn(C)c2)=O)CCCN(C(=O)CCc2cnc(N)cn2)CC1 C(c1cccc(F)c1F)=CC(=O)NC1(C2CN(C(Cc3ncc(C)s3)=O)C2)CC1 C(CC(=O)NOCCCF)C1(C)CN(C(CC2(OC)CC2)=O)C1 Cc1occc1C(=O)NC1CCC1CNC(=O)C(c1cccnc1)O c1(C(=O)NCC2(F)CN(C(C(C3CC3)SC)=O)C2)n[nH]c(C(C)C)c1[N+](=O)[O-] C1(CC(=O)NCC2CN(C(c3c(C)ocn3)=O)C(C)C2)CC(C)(C)OC(C)(C)C1 c1(C(=O)NC(CNC(CCOCCC)=O)(C)C2CCC2)cncc2ncn(C)c12 N1(C(C2CCCC2)C)CC(CO)C(C)(C)C1 N1(C(C2C(C(=O)OCC)C2)=O)CCC(N(C(=O)COC(F)F)C)CC1 C1(CC)(CC)CC(O)CN1C(c1oc(NC(c2c[nH]nc2C2CC2)=O)cc1C)=O C(=O)(C(CC)C(=O)NC(C)CCNC(=O)CCc1ccc(C)nc1)OCC C(=O)(C(F)CC(C)(C)NC(=O)C(C)NC(C)=O)N1CCC(N(C)C)(CC)C1 C(=O)(C1CCCc2scnc21)NCCN1CCN(C(Cc2ccn(C)n2)=O)CC1 C1(CC(=O)N(CC(C)NC(=O)CCC2CC2(F)F)CC)CNC(=O)O1 c1(CC(=O)NC2C(NC(c3c(OC)n[nH]c3)=O)CC2)cc(O)nc(O)n1 C(=O)(C#CC1CCCC1)NC(CC=CC)C(=O)NC1CCOCC1(C)C O=C(C1CCc2scnc21)N1CCCCC1Cn1cc(CC(O)C2CC2)nn1 C=CCCC(O)CN(C(=O)C(C)(CO)NC(=O)Cc1cccc(F)c1)C C1(F)(CNC(c2nnn(CC)c2C)=O)CCN(C(c2ncc(N)cc2Cl)=O)CC1 C1(C(=O)NC(C(=O)NC(c2onc(C)n2)CO)C2CCCC2)C2CCC(C2)C1C Cc1cc2ccc(C(=O)NC3CN(C(=O)CCc4nnc(C(F)F)o4)C3)cn2c1 C1(C)(NC(C(C2CCCCC2)NC(C(C(C)C)O)=O)=O)CC2(CCC2)C1 C1(C(=O)NC(c2ccccc2)CNC(C2CCSC2)=O)CCCCC1(F)F c1(C(=O)NC(CC)CNC(c2cccs2)=O)cc(Br)cc([N+](=O)[O-])c1 C1(NC(C2C(C)(Br)C2)=O)COC2(C1)CN(C(c1cccc(N)c1)=O)C2 N1(CCC)CCCCC1C(=O)N(C)CCNC(c1ccc(C(C)F)cc1)=O C1(CNC(C2(OC)CCC2)=O)CN(C(C2(C(F)F)CC2)=O)CCC1C O=C(C1=NN2CCCN=C2N1)NCC(O)CNC(c1nnn2c1CCCC2)=O N1(C(C(=O)NC(C)(C)C)CC2(C#N)CC2)CC2CCCN2c2ccccc21 C1(CS(=O)(=O)N(CC(=O)OCC)Cc2ncc(Cl)s2)(CF)CC(F)(F)C1 C1(NC(C2OCCC(NC(C3(CC)CCCC3O)=O)C2)=O)C2CCC(F)(F)C12 CC1(C)CCCC(C(=O)NC(C(=O)NCC=CCl)C2CCCC2)C1 C#CCN(OC)C(=O)C1CCCN(C(c2cc(C)c(C)cn2)=O)CC1 C1(N(C(C)=O)CC)CCCN(C(=O)C(C)(C)C)C1.c1(C(C=O)(F)F)ncccc1F C1(NC(COCCOCC)=O)CC(C(=O)NOCC(C)(C)C)=CC1O N1(C(c2nc(C(C)C)oc2)=O)CC(CC(=O)Nc2ccccc2C2CC2)CC1C c1(-c2c(C(N3CC(C(=O)OC)C(O)C3)=O)n[nH]c2)ccc(N)c([N+](=O)[O-])c1 C1(COC)CN(C(c2cnc(C)[nH]2)=O)CCN1C(=O)CCC1CCCOC1 C(c1cccc(F)c1)=CCC(=O)NC1C(OC)CN(C(C(C=C)(C)O)=O)C1 c1(CC(=O)N(C2CCCC(NC(C3(CO)CC3)=O)C2)C)cccc(OC(F)F)c1 C1(CNC(=O)CCc2cncnc2)CC2(CC(NC(C3CCCCO3)=O)C2)C1 CCC(CC)C(F)C(=O)NCCc1ocnc1CNC(C1CCCCCCC1)=O N1(C(c2c(C)ocn2)=O)CCOCC(CNC(c2nccn2C)=O)C1 C(C(C(C)C)NC(c1cc(CC(C)C)[nH]n1)=O)NC(C1(OC)CCC1)=O N1(C(C2CC(N3CC(O)C3)C2)=O)CCCC1CCNC(C1CSCCS1)=O c1(C(=O)NC2N(C(=O)C3CC3)CCC2)c(Sc2ccccc2)nnn1C.C12CN(C1)C2 S(=O)(=O)(c1ccc(NC(c2cc(C(=O)OC)cs2)=O)cc1)NCCCC(=O)OC CCCC(C)(CC)C(=O)NC1CCC1NC(c1coc(C2CCCCC2)n1)=O CC1CN(C(C2(NC(=O)C=CCN3CCC3)CCC2)=O)C(C)C(C)(C)O1 C1(NC(CNC(C(CC)C)=O)=O)C2CN(C(=O)C=C3CCCCC3)CC12 N1(C(=O)Cn2cc(Br)cn2)CC2CCC(C1)N2C(=O)Cc1cnn(C(F)F)c1 c1(C(=O)NCC(C)N(C(c2nc(COC)[nH]n2)=O)C)cc(=O)c(OC)cn1C c1(NC(C2(CNCc3cc(Br)ccc3F)CC2)=O)cnccc1[N+](=O)[O-] C(CC(C)C)(CS(C)(=O)=O)NC(C(N1CC2(CN(C(=O)OC(C)(C)C)C2)C1)=O)=O c1(NC2CN(C(=O)Cc3ccnn3C3CCCC3)C2)ccc([N+](=O)[O-])cc1Cl CC(C)C(CNC(c1cnn[nH]1)=O)NC(=O)CSCc1ccccc1 C1(CC(N2CC(CCCCNC(C(C)NC(C)=O)=O)C2)=O)CC=CCN1C c1(C(N(CCC(C)NC(=O)CC(C)C(F)(F)F)C)=O)coc2cc(F)ccc12 c1(NC(c2c(CNC(C(C)NC=O)=O)occ2)=O)ccc(CN(C)C)cc1 N1(C(=O)OC(C)(C)C)CCC(C)(C(=O)C(F)(F)F)C1.N1(C=O)CCN(C(=O)N)CC1 N1(C(C(CC)N(CC)CC)=O)CC2CN(C(c3cc(C)c(Br)c(C)c3)=O)CC2C1 C(=O)(C(C)(O)CC(F)(F)F)N(CCCC)CC(=O)NCCOC(C)O c1(C(=O)NC2CCN(C(CCC(=O)OC)=O)C2(C)C)snc2ccccc12 C(CCCCC(=O)N(C1CCCC1)CCOC)N(C)CC C1(C(=O)NC(C)CCc2ccc(F)cc2F)CCN(C(=O)CN)CC1(C)C C(=O)(C(C)(C)CS(C)(=O)=O)N(C1CCN(C(C2CCC(O)CC2)=O)CC1)C N1(Cc2c(OC)ccc(Br)n2)CC2CCC(C1)C2NC(c1cc2cnccc2[nH]1)=O N1(C(CC2CC(=O)NCC2)=O)CCC2CN(C(=O)CCC3CCCO3)C2C1 c1(C(=O)NC(CC(C)NC(COCC#C)=O)C)cn(C(F)F)c(C)n1 n1(C(CC)C)nccc1C(=O)NCCC(C)(C)NC(C1CC(CC)(CC)C1)=O CCC(CNC(C1(C)CCCO1)=O)(CC)NC(=O)CCSCC(C)C c1(C(N2CC(O)CC(NC(C3(OC(C)C)CCC3)=O)C2)=O)cc2cnn(C)c2s1 Cn1ccc2cc(-c3ccc(C(N4CCOCC4C(N)=O)=O)nc3)cnc12 C1(C(=O)OCC)CCC(C(=O)NCC(C2CC2)NC(=O)CC2C=CCC2)CC1 C(N=C(NCC(C)(C)c1cccs1)NC1CCS(=O)(=O)C1)C1(N(CC)CC)CC1 c1(C(N2CC(NC(=O)Cc3cncs3)CC(C)C2)=O)cc2ccc(F)cc2o1 c1(NC(=O)OC)cc(I)c(NC(=O)C(c2ccc(O)cc2)C)cc1Cl C1(CNC(C2C(C(=O)OC)C2)=O)CN(c2ncc(C(F)F)cn2)CCC1(F)F c1(NC(=O)NC(C)CCCOc2cccnc2)ccc2c(c1)ncn2C c1(CCN(C(C(N(C(=O)CC2=NNC(=O)C2)C)N)=O)CC)ccc2ccc(O)nc2c1 CC(C)(C(=O)NC1CCN(C(=O)CC(Cc2ccccc2)C2CC2)CC1)C(F)F C1(OC)CC(C(=O)NCCC2CC(NC(C3(C#N)CCC3)=O)C2)CC1OC c1(NC(CNC(C(CC)CN(C)C)=O)=O)cnc(Cl)nc1C C12(NC(C=C(CCN(C)C)Cl)=O)CCC(CC1NC(=O)C(=O)c1ccco1)C2 C1(NC(C2(C=C)CC2)=O)CC(CNC(C2CCCN2CCC(C)C)=O)C(O)C1 c1(CN2CCCC(CN(CCN)C(c3ccccn3)=O)C2)ccc(Cl)cc1 c1(-c2ncn(C)n2)ccccc1C(N1CCC(CCNC(c2cocn2)=O)C1)=O Cc1c(C(=O)N(C)CC2CCCN2C(=O)C(C)C2CCC2)nn2ccccc12 N1(C(C2(CC)CC2)=O)CC2CCN(C(c3cccc(C)c3NC(C)=O)=O)CC2C1 C1(CNC(c2ccc(COC)o2)=O)CN(C(=O)C2=CC(C)C2)CCCO1 O=C(N=c1nc[nH]n2cccc12)N1CCn2cncc2C1 Cc1nn(C)cc1CC(=O)NCC1C2CN(C(c3cc(C)n(C4CC4)n3)=O)CC12 N1(C(C2(CC#C)CCOC2)=O)CCC(CCOC(C(=O)C=CBr)=O)(OCC)C1 C=CC(C(=O)NCC1CCN1C(c1ccc(F)s1)=O)NC(=O)OC(C)(C)C c1(C(=O)NC2C(CO)CCN(C(c3c(C)nn(C)c3)=O)C2)cccc2cncn12 CC1(C)CCN(C(c2ccn(C(F)F)n2)=O)CC1NC(=O)CCOC1COC1 c1(C(N2CC(C=C)C(NC(C3COCCO3)=O)C2)=O)cc2sccc2n1C N1(C(c2ccncc2)CC)CCCC(C)(CNC(=O)C(N2CCC(O)CC2)C)C1 c1(C(N2C(CNC(C3C(OCC)C3C)=O)CCC2)=O)nn(CC(F)(F)F)cc1Cl CCCCC(C(=O)NCC(CCC)OCC)NC(c1n[nH]c2c1CCC2)=O C(C)(CCC(=O)N1CC(O)CO1)NC(c1cnc(C)c(C#N)c1)=O c1(C(C(=O)NC(CC)C)N(CC(C)C)C)ncn(C)n1 N1(C(C2(Cl)C(C(C)=O)C2)=O)C2CCC(C2)C1CC(=O)NCCOCC(F)(F)F c1(C(N2CCC3CN(C(CCCOC)=O)CC3C2)=O)coc2c(F)cc(F)cc12 C1(C)(C(=O)NC2CCN(C(CSCC=C)=O)C2CC)CCC(F)(F)C1 c1(OC)ccc(O)cc1C(=O)NCC1C2CCC(C2)N1C(=O)C(C)=C(C)C C(CCF)(C(=O)NCC1C(C)(C)C1(F)F)NC(C=CCCC(C)C)=O c1(NC(C(C)=O)=O)n[nH]c2c1CN(C(c1cc3ccoc3cn1)=O)C2 N1(C(c2nc(CCCC)sc2)=O)CC2(C1)CN(C(=O)C(c1cnn(C)c1)C)C2 c1(C(N2C(CN(C(C3CCCN3S(C)(=O)=O)=O)CC)CCC2)=O)c(C)noc1C c1(C(N2CC3C(C(C)NC(c4nc(Cl)c(Cl)s4)=O)C3C2)=O)cnc(O)nc1O N1(C(C=CC(C)(C)C)=O)CC2CCN(C(=O)COC3(C)CCC3)C(C2)C1 C1(OC)CN(C(=O)CC(C)N(C)C)CC1NC(=O)C(c1ccc(Cl)cc1)C C1(C(=O)NC(CCC)C2CCCC2)CC2(CCN(C(c3cnccc3C)=O)C2)C1 Cn1nc(Br)c2c(CNCCN3CCCC(F)(F)CC3)ncnc12 CC(C)C(O)CC(=O)NCCC(C)NC(C1(C)CCN(C)C1=O)=O N1(C(C(=O)Nc2cc(C(=O)OC)sc2Cl)=O)CC2CCC1(CC(=O)OC)CC2 C(C1=C(C(=O)OC)C(c2nnc(Br)s2)NC(=S)N1CCCF)OC c1(NC(C)=O)ncccc1C(N1CCC1CNC(c1nn(C)cc1C)=O)=O c1(C(N2CCC(NC(CN(C)CC)=O)CC2C2CC2)=O)ccc2c(C)noc2n1 N1(C(C(c2ccc(C)o2)C)=O)CCCN(C(C2(P(C)(C)=O)CC2)=O)CC1 N1(C(=O)NCc2c(C)sc(C)c2Br)CCC12CCN(C)C2 N1(C(CC2C(C)(C)CCO2)=O)CCC(C(=O)NC(CO)C2(C)CC2)C12CCC2 C1(C(=O)NC2(CO)CC(CO)C2)CCCN(C(C2(C(F)(F)F)CC2)=O)CC1 CCC(C(=O)N1CCC(N(C(=O)C=NOC)CC)C1)Sc1nc(=N)[nH][nH]1 C1(NC(c2cc(-c3ccc(C)s3)[nH]n2)=O)CCN(c2nncs2)CC1O C1(OC)CC(NC(=O)C(C)Oc2cccc(Br)c2)CN(C(=O)CC(C)F)C1 S(=O)(=O)(c1cc2c(cc1C)OCO2)NC(c1ccc(CC)cc1C)C N1(CC(=O)NCCN(C2CC2)Cc2ccn(CC)n2)C(=O)C(C)C(C)C1=O C#CCC(C)(C(=O)N(C1CCCCCC1O)C)NC(C1CCC(C)(C)OC1)=O c1(C(=O)NC2C(NC(Cc3cnn(C)n3)=O)CCCC2)c(F)cccc1[N+](=O)[O-] c1(C(=O)NCC(C2CCC2)NC(C2C(C(=O)OC)C2)=O)ccc2nnc(S)n2c1 C(CC(C)C(=O)N(C1CCN(C(c2cncc(N)n2)=O)CC1)C)=CCC O=C1CC(N=c2ccnc(N(c3ccc(Br)cc3F)CCO)[nH]2)CN1C(F)(F)F N(C1CCc2cccc(F)c21)C(N=c1c(C(C)C)c[nH][nH]1)=O C1(NC(C(CC)SC)=O)CC2CC1CN(C(C1(C)CCC(OC)CC1)=O)C2 CC1CCC(C2OCCO2)N(C(c2ccc(Oc3cccc(F)c3)cn2)=O)C1 c1(C(N2C3C(C(N4CCC5(CCC5)C4)=O)C(C3)C2)=O)ccc(F)c(Br)c1F C1(C(N(C)CC2CCN(C)CC2)=O)CCN(C(=O)CCC2CC2)C1(C)C c1(N(C)C)cc(C(=O)NC2CC(CNC(c3nocc3C3CC3)=O)C2(C)C)ccn1 C1(C(C)C)CN(C(=O)C2=CCOCC2)CCN1C(=O)CCCCCNC(N)=O CCCCCCC(C)CC(=O)NC1(CNC(C2CCCCCC2(F)F)=O)CC1 c1(CNCC2(C)N(C(CSC(C)=O)=O)CCC2)cccc2c1CCCC2 C1(NC(=O)C(O)C2CC2)CC2CCC1N(C(c1ncccn1)=O)C2 N1(C(C(CCC)F)=O)CCCCC2(CCN(C(=O)CCNC(=O)COC)C2)C1 N1(C(CC=CCC)=O)CCCC(COC)(NC(=O)Cc2ccnc(C(N)=O)c2)C1 N1(C(c2scc(C)c2)=O)CC(C(=O)Nc2cscc2C)CC(C)(C)C1 C1(C(=O)NC(c2ccsc2)C)CCN1C1CCCC1 Cc1ccc(C(=O)N(C2CCCN(C(=O)C(C)Cc3cnc[nH]3)C2)C)c(N)c1Cl N#CC1CC2(CC(NC(c3cccc(-c4nc(O)n[nH]4)c3)=O)C2)C1 Cn1cc(NC(c2ccnc(C(F)F)c2)=O)cc1C(=O)NC(C1CCCC1)CO c1(NCCc2cc(O)cc(F)c2)cc(=NCC2CC2Cl)[nH]cn1 C(=O)(CCCCCCn1cc(-c2conc2C2CC2)nn1)NC(CCC)C N1(C(C2(CC)CCCC2)=O)CC2CS(=O)(=O)CC2(NC(=O)Cc2cnsc2)C1 c1(C(N(CC(CN(C(C(OC)OC)=O)C)O)C)=O)cc(F)c(F)cc1C(F)(F)F c1(C(CC)C)ccccc1C(=O)NC(C)CNC(=O)CSC1CC1 C1(NC(=O)NC(C2CCC(OC)CC2)COC)CC2CCCCC2C1 C(C)(C)(C(C)CC(=O)NCc1nnc(O)o1)NC(C(C)CC(N)=O)=O Cc1ccc2cc(C(=O)NC3CCN(C(C4CC(O)C4)=O)CC3F)cn2c1 CCC(CC(=O)NC1CCC(C(=O)NCCC(=O)NC(C)(C)C)CC1)C(C)C C1(C(=O)Nc2cccs2)CCCCCN1C(c1ccncc1C(F)(F)F)=O C1(NC(c2c(C)nccn2)=O)CCN(C(c2cc(F)ccc2F)=O)CC1O C(=O)(CC(C)C(=O)N1CC(NC(c2ccccc2SC)=O)C(C)C1)OC c1(OC)cc(C)ccc1CC(N1CCCOC(CNC(=O)CN2CCCC2)C1)=O Cc1cnc(CNC(C2COCCN2C(=O)OC(C)(C)C)C)n1C Cc1nc(C)c(C(=O)NC2CC3(C2)CC3NC(=O)C=CI)o1 C1(C(N2CCC(CCN(CC(F)(F)F)CCCOC)CC2)=O)CCS(=O)(=O)C1 c1(C(N2C(C(C)NC(CCCCCC)=O)CCC2)=O)cc(Cl)c(F)cc1O N1(C(C2(C#C)CCC2)=O)CC(NC(C2COCCN2CC(F)(F)F)=O)C(O)C1 c1(C(=O)NC2CC(O)(CNC(C3CC4(CC(=C)C4)C3)=O)C2)cccc2sccc12 Cc1cnc(C(=O)N(C2CCCC2)CCNC(c2csc(Cl)n2)=O)cc1C c1(CCC(=O)NC2CC(F)(CNC(C3CC3F)=O)C2)ccc(Cl)cc1Cl c1(OC)cccc2nc(CNCC3(C)CCN(C(=O)OC(C)(C)C)C3)sc12 N1(C(c2cn(CC)nn2)=O)CC2C3CCC(C2C1)N(C(C1(CCF)CC1)=O)C3 c1(C(=O)NCCOCCCNC(=O)CCC2CCOC2)ccc(OCF)cc1F c1(OC)ccc(OC)c(CN2CCOC(C)C2)c1.c12cccc(c1)NC2=O Cc1nc2c([nH]1)CC(C(N1CC(OCCNC(=O)Cc3cccnc3)C1)=O)CC2 c1(C(=O)NC(C)CCNC(=O)CCc2ccc(O)cc2)n[nH]cc1[N+](=O)[O-] Nc1ccc(C(=O)NC2(CNC(c3cccnn3)=O)CCCCC2)c(F)c1F c1(C(=O)Nc2cc(C(=O)OCC)oc2C)cc(F)ncc1OC c1(OC)cccc2c1CCC(NC(C13CCC(C1)C(C)O3)=O)C2 c1(C(=O)NCC2=CCN(C(C(CC)(C)OC)=O)CC2)c(C)ccc2n[nH]cc12 C#CCCCCCC(=O)NCC1(C)CCC(NC(=O)C=CC(C)C)CC1 c1(C(=O)NCC(c2ccc(Cl)c(Cl)c2)C)ccc(F)cc1C1CC1 Cc1cc(F)ccc1C=CC(=O)NC(C1CCCCN1C(=O)C(F)=CCCF)C N1(C(COC(C)(C)C)=O)CCC2(CC(NC(=O)Cc3cccc(Cl)c3Cl)CO2)C1 CCC(CC)(CCOC)C(=O)NC(c1ccccc1)C(=O)OCC(C)C N1(C(C(C)NC(=O)NC)=O)CCCN(C(c2cc(C#N)on2)=O)CC1 CC1(C)CCC(C(=O)Nc2ccc(O)c(CO)c2)CN1C(=O)CC1CC2CC2C1 Cc1nc2cc(C(=O)NCCC(O)(CC)CC)cc(Br)c2o1 c1(CNC(=NCC)NCCOCC(F)F)cnc(C)cc1C CCCCC(C(=O)N1CCC(C(N2CC3C(C)C3C2)=O)C1(C)C)C(C)C C(C(C)(CO)CC=C)NC(C1C(NC(CC2CC(=C)C2)=O)COCC1)=O Cc1ccn(C(C)CC(=O)NC2CCC2CNC(c2ccc(C(F)F)s2)=O)n1 Cc1n[nH]c2cnc(C(=O)NC3CC3NC(=O)C(C(C)C)n3ccnc3)cc12 c1(C(=O)NCC2N(C(C(C)(C)NC(C=COC)=O)=O)CCC2)cnc2n1CCC2 c1(C(C(=O)OC)N(C)Cc2nc(CC)sc2)ccc(F)c(F)c1 C1C(C)(NC(C(=O)NCCC(=C)C)=O)C(=O)N1.C(C)(C)(C)O.C(C)(C)(C)O c1(C(N2CC=CC(NC(c3nccc(C)n3)=O)C2)=O)cnc2scnc2c1 C1(C(N(C)CC2(F)CC(C(C)(C)C)C2)=O)CC(C)(C)CO1 CCC(CC)C(C(=O)N1CCC(O)C1C(N1CCOCC1CO)=O)OC c1(C(=O)NCCN(C(=O)CCc2csc(C)n2)CC)ncc(C)cc1OC c1(C(=O)NC2C(NC(CCSCC(C)C)=O)C2)cnn2ccncc12 C1(CC)COC(C)(C)CN1C(=O)CC(CC(C)C)NC(=O)CCn1cccn1 CC(C)(F)CCC(=O)NC1CCC(NC(c2ccc(CCC(N)=O)cc2)=O)CC1 CCCCCCC(C)(CC)C(=O)N1CCC(NC(c2cccc(C(C)C)c2)=O)C1 N1(C(c2cccn3ccnc23)=O)CCN(C(=O)CC2CC2)C2CCCCC2C1 N1(C(C(CC)NC(N)=O)=O)CC(CC(N2CCCCC2)=O)C(O)C1 C1(C(=O)NC2CC(C(C)NC(COCC(C)C)=O)C2)CC12CCC2 c1(C(=O)NCC2CC(NC(c3ccc(C(C)=O)s3)=O)C2)ccc(Cl)nc1 C1(N(C(=O)CC2CCN(C(=O)CC3CCC(C)(C)CC3)C2)C)CCC2(CCC2)C1 N1(C(C(F)OC)=O)CC(NC(=O)CSC(C)C)C(C)(C)C1 N1(C(C(C)NC(=O)C(C)(C)C)=O)CCC2C1CCCN2C(=O)C(F)=C1CCCC1 C1(CNC(c2c(C)nsc2)=O)CN(C(c2cnc(Cl)c(C3CC3)c2)=O)CCN1C n1(C(C)C)ncc(C(=O)NC2CCC(NC(=O)CCN(C)CCO)CC2)c1F C1(NC(C(c2ccc(OC)cc2)(C)C)=O)CCC2CN(C(=O)CO)CCC2C1 C1(NC(C=CC(=O)OCC)=O)CCCCC1C(N1C2CCC1CC2)=O N(C1COCc2c(Br)cncc21)C(C1CN(c2n(C)ncc2)C(=O)C1)=O Cc1oc(CNC(=O)CCn2cnnn2)nc1C(=O)N(C1CCC1)C c1(C(N2CC(NC(C3(OC)CCCOC3)=O)C(O)C2)=O)nc2nc(C)ccn2n1 CN1CCC(NC(=O)C(c2ccc(Cl)cc2)(C)C)C1(C)C C1(NC(Cc2ccn(C)c2)=O)CN(C(C2CCC(=O)CC2(C)C)=O)C2CCCC12 N(C(=NCC(C)C)N(C)CC1CC1)CC1CCN(c2c(OC)cc(F)cc2)C1 C(=O)(C(O)CCC(C)C)NCC1N(C(Cc2cc(C)no2)=O)CC=C1 C1(O)(CNC(C2CCC(=O)N2)=O)CCCN(C(=O)CCc2cnoc2)CC1 C1(C(=O)NCC2C3CN(C(C4(O)CCC(CC)C4)=O)CC32)CN2CCN1C(C)C2 C1(NC(c2ncsc2Br)=O)(CNC(C2(O)CC2)=O)CCOC1 CC(O)C(C)(C)C(=O)NCC(O)CNC(c1cc(F)n(C)n1)=O c1(C(=O)OCC(CCC)(F)F)coc2c1N(C)C(=O)CCC2 Cc1cc(CCC(=O)NC2CC(NC(=O)C(CO)N(C)C)C23CCC3)cc(C)n1 C1(C(N(CCC(N2CCC2(C)CC)=O)CC#C)=O)CCC(C)=C(C)C1 C1(NC(c2cc(C)on2)=O)CN(C(=O)C(O)CNC(=O)OC(C)(C)C)CC1N=[N+]=[N-] c1(C(=O)NC23C(CN(C(C(n4cc(Cl)cn4)C)=O)C2)C3)ccc2ocnc2c1 c1(OC)c(C(=O)NC2CN(C(=O)C(c3ccccc3)O)CC2(C)C)cccc1Cl N1(C(CC2N(CC)CCC2)=O)CCOC(C(C)NC(=O)CNC(=O)OC)C1 N1(C(CCCCCC#C)=O)CC(NC(c2ccnn2C=C)=O)CC12CCCOC2 C1(C(=O)NCCC2CCN(C(CC3(C)CCC3)=O)C2)CN(CP(C)(C)=O)C1 Cc1ccnnc1C(=O)NC1CCCC(CN(C(=O)Cn2cccc2)C)C1 c1(OCC(=O)NC(CCCCNC(CSC)=O)CO)cccc(S(C)(=O)=O)c1 C1(CNC(C(CCC)N(C)C)=O)CN(C(c2cc(C(C)(C)C)no2)=O)CCN1C C1(C(=O)Nc2ccc(Cl)cc2)(C(N2CCOCC2)=O)CC2C=CC1C2 c1(C(N2CCC(N(C(C#CC3(CC)CC3)=O)C)C2)=O)cc2c(OC)cccc2s1 c1(C(N2CCC(NC(C3(Cl)CC3)=O)C(c3ccccc3)C2)=O)c(F)cccc1F C1(CCCCN(C(CC(C)C)=O)C2CC2)CCCN(C(=O)Cc2ccc(Cl)cn2)C1 c1(CC)nc2cc(Oc3cncc(-c4ccccc4)c3)ccc2o1 c1(CC)ccc(N2CC(C(=O)Nc3ccnc(OC)c3)CC2=O)cc1 C1(C(N(CC(C2CCC2)NC(C2CCNC(=O)C2)=O)C)=O)CCC(C)(C)CC1 C1(CCCCNC(C2C(C(C)C)CCC2)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1 c1(C(=O)NCC(C)N(C(c2ccc(F)cc2F)=O)CC)cccn2cnnc12 C1(CNC(C=Cc2scc(C)n2)=O)CC(C)(C)CN1C(C1CCOC(=O)N1)=O c1(C(=O)NCC(CC)NC(C(CC)c2ccccc2)=O)n[nH]c2c1CCOC2 c1(-c2ccc(COCC)cc2)ccc(Cl)c(OC)c1N N1(C(c2c(OC)ncc(F)c2)=O)CC2(CCN(C(C3NC(=O)OC3C)=O)C2)C1 CN=c1[nH]c(=NCc2cc(C(C)OC)nn2C)[nH]c(=NC(CCO)C2CC2C)[nH]1 N1(Cc2cc(C)ncc2)CCC(C(=O)Nc2ccc(I)c(Cl)c2)C(O)C1 c1(OCC(=O)NCCCN(C)CC2(C=C)CCC2)cccc(F)c1F c1(SC)cc(C(N2CC(N(C(=O)CN3CCCCC3)C)C(O)C2)=O)ccn1 c1(C(C)C2CC2)nc(-c2ccn(C)n2)nn1C1CCOC1 Cc1ccc(C2CC2C(=O)NCc2ccc(N3C=CC=C(F)C3)cc2)cc1 c1(C(=O)NCC2CCCCC2NC(C2COCCO2)=O)cc2n(n1)CCCC2O C(=O)(CC(C)CC(C)(C)C)N1CC(N(C(Cc2cc(C)on2)=O)C)C(C)(C)C1 C(=O)(CC(O)CNC(=O)C(F)(F)C1CC1)N1C(CC(C)(C)C)CC1 C1(NC)CCC(C(=O)NCCC(O)CNC(=O)C=C(C)C(F)F)CC1 c1(-c2scc(CC(=O)NC(C)CCCNC(=O)CCF)n2)ccc(Cl)cc1 C(c1cnc2ccccc2n1)=CC(N1C(CN(C(=O)COC2CC2)C)CC(F)C1)=O c1(C(N(CCC)CCc2ccccc2)C2CC2)ccc(C(C)(C)C)cc1Br c1(C(=O)NCC(CO)NC(CCC(C)C#N)=O)cc2ccccc2cc1O N1(CC)C(=O)NC(c2cnn(C3CC3(F)F)c2)C(C(=O)NC)=C1CCl N1(C(CCOC)=O)CCOC(C(C)NC(=O)COc2cccnc2Cl)C1 C(C)(C)(CCCC(=O)NCC1CC1COC)NC(C1(CC)CCCO1)=O C1(C(N(CC(C)NC(=O)C(=O)N(C2CC2)C2CC2)CC)=O)(CC)CC=CC1 C1(C(NNC(c2ccc(N(CC)CC)cc2)=O)=O)CN2CCCN1CC2 n1(CC)ccc(C(=O)NCC2CCCC2NC(c2cc(C)n(CC)n2)=O)cc1=O c1(C(C(=O)NC2CCCN(C(c3csc(O)n3)=O)C2)N(C)C)c(F)cccc1Cl C1(NC)(Cc2cn(CC(=O)Nc3ccccc3)nn2)CCOCC1 c1(NC2CC(NC(N(C)CC)=O)C2(C)C)c(C)ccn(C)c1=O C(=O)(C1=CCCOCC1)N1CCCC(N(C(=O)CCS(=O)(=O)N(C)C)CC)C1 Cc1nonc1CC(C(=O)O)NC(=O)CSc1ccn(-c2ccccc2)n1 C1(NC(C2(COC)CCC2)c2nn[nH]n2)CCC(P(C)(C)=O)C1 c1(Cc2cn(C(=O)NC(c3cn(C)nn3)C3CC3)nn2)nc[nH]c2nccc1-2 C(CNC(=O)CCCN1CCOCC1)(CC(F)(F)F)NC(=O)C=CC1CCCC1 n1(-c2ccc(OC)cc2)cc(S(=O)(=O)N2CC(C(=O)OC)CC2CN)cn1 CC(CS(C)=O)N=c1[nH]c2c(c(=NCCc3cc(O)n(C)n3)[nH]1)COCC2 N1(C(Cc2ccc(SC)o2)=O)CCC(C)C(CNC(=O)C(O)C(C)C)C1 c1(CNC(CC)=O)nc2c(s1)CCN(C(C1CCCN(C)C1)=O)C2 c1(C(=O)NCC2CCC(NC(C3C(C)=C3)=O)C2)n[nH]c2cc(C)ccc12 CC1CC(NC(c2c(Cl)n[nH]c2C2CC2)=O)CN(C(=O)CC2CCOCC2)C1 c1(OCC(N2CC(O)(CNC(c3n(C)nnc3)=O)C2)=O)ccc(C(N)=O)cc1 C1(NC(CN(C(=O)CCCc2ncco2)CC(F)F)=O)CCC(=O)NC1=O Cc1ccc(C(N2CCC(CC(=O)Nc3ncc(Cl)nc3Br)C2)=O)cc1Br N1(C(CCc2scc(C)n2)=O)CC(NC(c2nn(C)cc2C)=O)C2CC12 N1(C(C2CCC(=O)O2)=O)CCC2(NC(c3ccc(Br)nc3O)=O)CCCC12 C1(O)(CNC(C(CCC)O)=O)CCN(C(c2cnnn2C)=O)CC1 c1(C(C(=O)NCC2(F)CC(NC(=O)Cn3ccnn3)C2)CO)ccc(Cl)cc1 C(=O)(C(CCC(C)C)NC(C)=O)NCC1(F)CC(NC(CCSCCCC)=O)C1 N1(C(c2c(C)nc(-c3cccc(Cl)c3)[nH]2)=O)CCN(C(C2CCSC2)=O)C(C)C1 c1(CNC(C(CCC)O)=O)c(C)nn2c1CN(C(C1CC(C)(C)CN1C)=O)CC2 N1(C(C2CCCC(C)C2)C(=O)NCC(C)C)CCC(C)c2ccccc21 CS(=O)(=O)C1CCC(NC(C2CC(=O)N(c3cccc(Cl)c3)C2)=O)C1 Cc1cncc(CNC(C2CC(NC(C3CC(F)(CF)C3)=O)CCO2)=O)c1 N1(C(c2cc(C)sc2)=O)CC2(C1)SCCC2NC(=O)COC1CCCCC1C C1(F)(CNC(c2cc(O)cs2)=O)CCCN(C(C2CCOC2C(F)(F)F)=O)C1 c1(OC)ncc(Cl)cc1C(N1CCN(C(=O)C(F)CC2CC2)C(C)C1)=O O=C(CC1NC(=O)c2ccccc21)NCCN(C(c1csc(Cl)n1)=O)C1CC1 C1(C(N2CCN(C(=O)CC3=CCCC3)C(C(F)(F)F)C2)=O)CC12CCCCC2 n1(CC(=O)N(C(CNC(C2(C)CC(=C)C2)=O)C)C)ncc(O)nc1=O c1(C(=O)NCC2CN(C(C3C(F)(C(=O)OC)C3)=O)C2)cc2n(n1)CCCO2 c1(CNC(COCCNC(CC2CC(=C)C2)=O)=O)cc(C)nc(C)n1 c1(C(CC2CC2)NCc2cccc(C(C)C)n2)ccc(F)c(Cl)c1 N1(C(C2(F)CCCC2)=O)CCN(C(C2CC2C(F)(F)F)=O)C(c2ccccn2)C1 N1(C(=O)Nc2cc(Cl)nc(Cl)c2)CCCC(CO)(Nc2nccc(CC#N)n2)C1 c1(CNC(C(CNC(C2COC(=O)N2)=O)OC)=O)cc(C)cc(F)c1 Cc1cnn(C)c1C(=O)NCC(C)CC(=O)N1CC(c2nncs2)C1 C1(C(=O)NC(CC)CN(C(C2(CCOC(C)C)CCCC2)=O)C)C(C)(C)C1(C)C N1(C(C=Cc2cc(C)no2)=O)CCC2CN(C(=O)C(O)CC(C)C)CC2C1 N1(C(CC=C)=O)CCc2ccccc2C1CNC(c1ncccc1C)=O c1(C(=O)NC(COC(C(C)SC)=O)=O)cc(-c2cccnc2)nn1C CN=S(C)(=O)c1cccc(C(N2CCCCC2CNC(c2nccn2C)=O)=O)c1 C1(NC(C=CC=CCC)=O)CCN(C(=O)C(C)(C)c2sccc2Cl)CCC1CO c1(C(N2C(CN(C)C(c3ncoc3Br)=O)CCCC2)=O)ccc(F)cc1F C1(CC(=O)NCCOCC(F)F)CCCCC1NC(=O)CC1CCOCC1 C(=O)(CC(O)CC(C)(C)C)NCC12N(C(C(C)NC(CC)=O)=O)C(CC1)CC2 C1(NC(C=CC(C)(C)SC)=O)CC2(C1)CC2C(=O)NC1C(C#N)C1(C)C c1(N2C3(CN(Cc4nccc(C)c4)C3)CC2)nc(C)nc2ccsc12 C(=O)(C(C(C)(C)C)NC(C)=O)N(C)CC1N(C(CNC(C)=O)=O)CC(F)C1 N1(C(c2c(C)nco2)=O)CCN(C(=O)C(CN(C)C)C(C)C)C(CC(F)F)C1 C1(C)(C(N2CC(=C(CNC(c3cc(SC)oc3)=O)F)C2)=O)CCC(F)(F)CC1 CC(CNC(C1CCC1(F)F)=O)(Cn1cccn1)NC(=O)CSC(F)F C(C(=O)NC(C1(OC)CCC1)C)(C(C)C)NC(COCC(=O)OC)=O N1(C(C2C(=C)C2CO)=O)CC2(NC(=O)CN3C(=O)CCCC3=O)CCCC2(F)C1 N1(C(CC=CCC)=O)CCOCC1CCNC(=O)C(C1(O)CCCC1)OC CN1C(=O)CSC1=CC(=O)NCC1CCN(C(=O)CCC2CCCC(=O)N2)C1 C1(CC=C)(NC(=O)C(C)C(C)O)CCCN(C(c2c(Cl)cnn2C)=O)C1 c1(OC)cc(C(=O)NCC2CCC(C)CN2C(=O)CN=S(C)(C)=O)cc(Cl)c1 C(CC(C(=O)N1CCC(C(N2CC(OC)CC(C)C2)=O)O1)OC)OC N1(c2nccc(OC)n2)CC2CC1CN2C(c1cc(Br)cnc1OC)=O c1(C(N2CC(OC)CC(NC(C(CC=C)CC)=O)C2)=O)ccc2oc(C)nc2c1 N1(CC(=O)N(CCC(C)NC(=O)CC(=O)Nc2ccncc2)CC)CCN(C)CC1 CCC(CC(=O)N1CCOCC1CNC(=O)C(F)OC(F)(F)F)CC(C)C C1(CN(C(=O)CCCN(C)C(C2CCCO2)=O)C)CCCOC1 N1(C(Cn2c(C)cc(C)n2)=O)CCCC(NC(c2cnc(C(F)F)nc2)=O)C1C C1(C)(C(=O)NCc2cccc(N(C)C)n2)CCNC(=O)C1 c1(C(N2CCN(C(c3c(C)cco3)=O)CC2CF)=O)cc(F)cc2ccncc12 c1(C(N2C(C)C(NC(=O)Cc3csnn3)CC2)=O)cc2cccnc2s1 C1(CNC(c2c(C)oc(Cl)n2)=O)CN(C(=O)COC2(C)CCC2)C2CCCCC12 c1(C(N2C(C(=O)NC(COC)(C)C)CC3CC32)=O)cc(C)cc([N+](=O)[O-])c1 C12(CNC(c3ccc(Br)cc3)=O)CC1CN(C(C1C(F)(F)C13CC3)=O)C2 C1(N(C(=O)CSc2cccs2)C)CCN(C(C2(C3CCCO3)CC2)=O)C1 C#CC1(C(=O)NCCCCCCOC)CCN(C(c2cnc(N)cn2)=O)C1 C(=O)(C(CNC(c1cnnc(O)c1)=O)C(C)(C)C)NCc1ncn(C)c1 Cc1cc(C)c(C(=O)NCCCCC(C)NC(C2CCCC(=O)CC2)=O)cn1 C=CCC(C)(C)C(=O)NC(CNC(c1ncsc1C)=O)C(C)C(C)C C1(CNC(c2ccc[nH]2)=O)CCN(C(=O)CC2CCSCC2)CC1(F)F c1(C(=O)NC2CC(N(C(C3(CC)CCNC3=O)=O)C)C2)ccc2c(C)noc2c1 C(C)(C(CC(=O)NCC1CNC(=O)C1)NC(=O)C(F)(F)C1CC1)OC CC(C)(CC(=O)N1CCOCC(NC(=O)CC2CC(=O)NC2=O)C1)C(F)F CCC1=C(C(=O)N2CC(CNC(c3[nH]c(C)cc3C)=O)CC2C)SCCO1 c1(CC(N2C(C(C)(C)NC(C(CC)F)=O)CCC2)=O)ccc2nonc2c1 c1(C(N(C(CCNC(C(C=C)(C)C)=O)C)C)=O)cc2cc(F)cc(F)c2nc1C CCC1=C(C(=O)N2CCCC(CN(C(=O)C(O)C(C)C)C)C2)SCCO1 O=S(=O)(Cc1cc(Br)ccc1Cl)C12CC(C1)C2 C(=O)(C(F)(F)C(C)O)NCC1C(NC(c2c(COC)cco2)=O)C1 c1(NCC(C)NC(=O)NC(COC(C)(C)C)CF)ccccc1 c1(C(=O)NCC(CC)N(C(C(C)NC(CC)=O)=O)CC)cc(CC)on1 c1(CC(N2CCCCC(NC(C3CC(OC)C3)=O)C2)=O)cnc2n1CCCC2C CC1(C)OCCC1NC(c1ccc(CNC(C2(C#N)CCCO2)=O)s1)=O n1(CC(=C)C)nnnc1C1(NCCCCN2CCCC2=O)CCCC1C(C)(C)C c1(C(=O)NC2CC(C)N(C(C3CCC(=O)C3)=O)C2)cc(C2CC2)nc(Cl)c1 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CCN(C(=O)C=CC3CCCO3)CC(C2)C1 O(NC(=O)C(C)CNC(C1(F)CC=CCC1)=O)CCOCCOC c1(OC)ccc(C(=O)NC2CCN(C(c3cc(C)n(C(F)F)n3)=O)CC2)nc1 C(=O)(C(C)(F)CC1CCCC1)NC1C(CNC(CCCn2c(C)ncc2)=O)C1 C(=O)(C(F)C(C)(F)F)N1CC(C)(C(N(C(C#C)(C)C)C2CC2)=O)C1 N1(C2CN(C(c3nnn(C)n3)=O)C2)CCN(C(C2CCN(C3CC3)C2=O)=O)CC1 c1(-c2ccc(F)c(C)c2F)cnc2c(cnn2C2CCCCO2)c1 C=CCC(C)(C)CC(=O)NC(CC1CC1)C(N1CC2(CCC(=O)O2)C1)=O C1(=O)C2=CCCN(C2)C(=O)CCN1C(C)(C)C.C1(C(C2CSC2)C)CCCC1 c1(C(N(CCN(C(=O)CC2CCC(=O)N2C)CC)CC)=O)cc(C)c(C)c(C)c1 C(=O)(C#CC1(C)CCCO1)N1CCCC(NC(C2(C)CC=CC2)=O)CC1 C1(Nc2scnc2C(=O)NC2C=CC(CC(=O)NC)C2)CCCCC1CO c1(OCC)cccc(NC(c2nc(C(=O)Nc3ccc(C)cc3)cs2)=O)c1Cl C(=O)(CC(CC)CCCC)N1C(C(=O)NCc2nccc(CC)c2)C2CC2C1 N1(C(c2occ(C)c2C)=O)CC(C2CCCN(C(=O)C(C)(C)C3CC3)C2)C1 N1(C(CN2C(C)CCC2)=O)CCCC(CCCCNC(C23CC(C)(CO2)C3)=O)C1 c1(OCC)cc(Cl)ccc1C(=O)CNC(C1CC1c1ccco1)=O c1(CC(=O)NCC=CCNC(C2CN(C)C(=O)N2)=O)cn2c(n1)CCCC2 CCCC(CNC(C1(NC(=O)CC(C)(C)OC)CC(F)(F)C1)=O)CCO C(N=c1cc(C)nc(N2CCC(C3CCCO3)CC2)[nH]1)C1C(COC)C1 C(=O)(C1=NOC2COCC12)NC1(CC)CN(C(C2CC(C)(O)C2)=O)C1 C(=O)(C(C)C(C)C)NCC(=O)NCC(=O)NC(CCC)C1CCC1 c1(NCc2n(C(C)C)ncn2)[nH]c(=NC2CCCC2N(C)C)nc2ncn(C)c12 n1(CC)c(C)c(C(N2CC(OC)CC(O)C2)=O)c2cc(OC)ccc12 c1(C(=O)NCC2(O)CC(NC(CCC=C(C)C)=O)C2)ccc(Br)c(C)n1 C1(CC(=O)N(C2CCN(C(c3ccc(C)nc3)=O)CC2)CC)CCC(C)CO1 c1(OC)ccc(F)cc1NC(C1CC1NC(c1nc(C)no1)=O)=O N1(C(CC(=O)NC)=O)C2CCC1CC(NC(=O)COCC1CCCOC1)C2 N1(C(CCN(C(C)=O)C)=O)CCC(OCCNC(C2CC=C(C)CC2)=O)CC1 C(CN=c1[nH]c(C)cc(=NC2CC(C)C2)[nH]1)c1n[nH]c2ccc(NC(C)=O)cc21 C1(NC(CC=C)=O)CCN(C(c2ccccc2OCCN2CCCC2)=O)CC1C C(=O)(CC1=CCN(C(c2cc(C(C)C)no2)=O)CC1)N1CCC(OC(C)=O)C1 Cc1nn(C)cc1CN1CC(NC(=O)C#CC2CC2)C(F)C1 O=C(CCC(=O)NC(=O)CC1CC2(COC2)C1)NCC(C1CCCC1)C1CC1 Cc1[nH]c2ccccc2c1CC(=O)NCC1CCN1C(C1CC(=O)N(O)C1)=O C(C(C)(CC(C)C)NC(c1cc(C(C)C)oc1C)=O)NC(C(CC)C#N)=O C1(O)(CNC(CC(C)OC)=O)CC2CCC(C1)N2C(=O)C(=O)N=S(C)(C)=O C1(N(C(=O)CC2CC(F)(F)C2)C)CN(C(=O)C=CCN2CCCCC2)CC1(C)C c1(CNC(C2(c3ccc(OCC)cc3)CC2)=O)oc2c(C)cccc2c1C c1(NCCC(CC)(C)C)[nH]c(=NCCC2CC=CC2)nc2c1cnn2C(C)C N1(C(c2scc(C(C)=O)c2)=O)CC(C)OC2(CCN(CC3CCCC3)CC2)C1 C(=O)(C1CCc2nccn21)N1CCC(CC(=O)NCC(C)C)C1 N1(C(C=C2CCC(C)C2)=O)CC2(COC(CNC(c3ccccc3)=O)C2)C1 C1(C(N2CC(C(C(=O)Nc3cnn(C)c(=O)c3)OC)C2)=O)CC(=O)N(OC)C1 c1(OC)ccccc1C(C)C(N1CC(CNC(c2c(C)coc2C)=O)C(C)C1)=O O=C(Nn1nnc2c1CCCC2)C1CC=CCN1.n1(CC(=O)N)cccn1 N1(C(CC(C)N(C)C)=O)CCCC(NC(=O)CS(=O)(=O)NC(C)(C)C)CC1 CCCC(C)(O)CC(=O)NC1(C)CC(NC(C2CC(=O)N(CC)C2)=O)C1 CC1(C)CNCCN1CC(=O)NC1CCN(c2ccccc2)S1(=O)=O c1(CC)c(NC(=O)C(CC(C)C)NC(=O)CC2=CCCC2)cccc1F c1(C(N2CC3C(NC(C(C)O)=O)(CC3)C2)=O)cc2cc(C#N)ccc2[nH]1 c1(CC(=O)NCC(C)NC(C(C)NS(CCCC)(=O)=O)=O)nc2ccccc2s1 C(=O)(C(C)(C)CCC#N)NCC(C)CNC(C1CCCC2C1C2(F)F)=O N1(C(CN(C)CC)=O)C2CCC1CC(CNC(c1ccsn1)=O)C2 Cc1cc(C(C)NC(N2CC(=CCC(=O)O)C2)=O)cc(F)c1 N1(C(CCCN(C(C)C)C)=O)CCC(O)(CNC(C2CCCCN2N=O)=O)CC1 c1(NC(C(c2ccccc2)N(C)C)=O)coc(C=CC(=O)OC(C)(C)C)c1 N12CCOCC1C2=O.c1(OCC)ncc(C(=O)Nc2cnn(CC3CC3)c2)s1 C1(CC)CCCC(NC(c2sccc2CNC(c2cccn2C2CC2)=O)=O)C1 C1(C(=O)NC(CCNC(C2(COC)CCC2)=O)C)CSc2ccccc2O1 C(=O)(CCC(C)NC(N)=O)NC(C)CCCNC(C1CCCN1C(=O)C(C)C)=O CC1C(O)CCCN1C(=O)CCCNC(C1CCNC(=O)C1)=O C(C#CC(=O)N1CCCc2nccn21)NC(C(C)(C)C#N)=O c1(N(CCC2CN(C)C2)C)nc(=NC2CCOC2)[nH]c2c1SCC2 C(=O)(C1=CCN(c2ccccc2)CC1)N1CCN(C(=O)Cc2ccc(=N)[nH]c2)CC1 C1(C(=O)NCC(C(N2CC(CC)(CO)C2)=O)N(C)C)CCOC1(C)C C1(NC(C(CCSC)NC(C)=O)=O)CN(C(c2cnoc2C2CC2)=O)CCC1F N1(CC(=O)NCCOCC(=O)NC(C(C)n2cccn2)C)CCOCC1 C1(CNC(c2ccc(Cl)s2)=O)(CNC(=O)C(C2CCCCC2)O)CC12CCC2 c1(C(c2nnnn2C2CCOC2)NCC2C(C(=O)OC)CC2)cc(C)ccc1Cl C(=O)(C(CCN(C)C)NC(=O)CC1COCCO1)NCC(C1CCC1)OC CCCCCCCCCC(=O)NC1CN(C(c2cn[nH]c2)=O)CC2CC12 Cc1cc(F)ccc1CC(N1CCCCC(CNC(c2cncnc2)=O)C1)=O c1(C(=O)NC(CCOC)CNC(C2CC23CC3)=O)ccc(C)c([N+](=O)[O-])c1 C(CC(C)(C)C(=O)N1CCC(NC(=O)C(O)CC2CCOCC2)C1)SC C1(C(=O)NC(C)CCNC(c2ccncc2O)=O)CC2CCCCCC12 C1(C(=O)NCc2ccc(C(=O)NC3(CC#C)CCC3)nc2)CC2CC(=O)C1O2 C(=O)(C(CC)CC(F)F)N(C1CCN(C(c2c(CC)cc[nH]2)=O)C1)C c1(C(=O)NC(CNC(c2c(Cl)c(C)n(C)n2)=O)C(C)(C)C)cn2c(n1)CCCC2 C1(C(=O)NCC2(COC)CN(C(=O)C=CC3CC3)C2)CC2CC(O)CC(C1)C2 N(C1CCc2cc(CNC(c3cnco3)=O)ccc21)C(CC(CC)OC)=O N1(C(c2ccnc(CC(C)C)n2)=O)CCN(C)C(CNC(c2cscc2Cl)=O)C1 N1(CC(=O)N(CCNC(CNC(CCC)=O)=O)C(C)C)CCC(F)CC1 C=C(C)C(C)(O)C(=O)NCC1(NC(c2sc(COC)nc2C)=O)CCOC1 c1(OC)ccccc1CCN(CC(O)CN1CCN(C)CC1)C c1(CSC)ccc(CNC(c2c(CC(=O)COCC3CC3)nnn2C)=O)cc1 C1(C(=O)NCCC(C(C)C)NC(=O)CCC2CCN(C)C2)CC2(CC2)CN1C C#CC1CN(C(=O)C=C(C)C(C)(C)C)CCN1C(=O)CCCOC(C)C c1(C(=O)O)cc(-c2cn(CC3CCCN3C(C3SCCCS3)=O)nn2)ccc1F Cc1ccc2c(c1)CCC(C(=O)NCCN(C)C(C1CCC(C)O1)=O)O2 N1(C(c2c(OC)csc2)=O)C2CCC1CC(NC(c1n[nH]c3c1CSCC3)=O)C2 c1(C(=O)NC2C3N(C(c4cn(CCC)nc4)=O)C(CC3)C2)ccc2c(c1)CCC2 c1(-n2c(C(c3cc(C)no3)NCCC(F)F)nnn2)ccc(Cl)cc1F c1(C(=O)NCC2(O)CN(C(c3n(CC)ncc3)=O)C2)ncccc1Cl CCCCC(C(=O)NCC(C)OCCO)NC(=O)C(c1cccn1C)=O N1(C(CCC=C)=O)CCCC(N(CCO)C(c2ccc(OC(F)F)cn2)=O)C1 N1(C(C(C)(C)O)=O)CC2OCCN(C(=O)CCC3(C)CCC(=O)N3)C2C1 c1(C(N(CCCNC(CCCSC)=O)C)=O)cccc(C(F)F)c1F N1(C(C2N(C(=O)OC)CSC2)=O)CC=CC(NC(=O)CCC(=O)N(C)C)C1 C(=O)(C(C)(C)CC(F)F)NC1CCN(C(CC(COC)(C)C)=O)C(C)C1 C1(CCC)CN(C(C2CCC3(CC3)C2)=O)CCN1C(c1cscc1SC)=O CC1C(NC(c2cccc(=O)o2)=O)CCCN1C(c1cc(C(F)(F)F)ccn1)=O Cc1ccc(O)c(CC(=O)NCC2CCC(NC(=O)C(C)(C)CC3CC3)C2)c1 C1(NC(c2cn(C3(C(=O)O)CC3)nn2)=O)CCN(C2COC2)CC1O N(C(=NCCc1cnn(C)c1C)NCc1cc(C)ccc1Br)CC(=C)C N1(C(CCCCC)=O)CCC(NC(c2ccc(OC)cn2)=O)C(CO)CC1 C(=O)(C1COc2ccccc21)NCC1(O)CCCN(C(COCCCCC)=O)C1 C1(Cn2ccc(C(=O)OC(C)(C)C)n2)CCCNC1=O.C1(N2CC2=O)CCCO1 c1(C(C)Cn2cc(CC(C(=O)O)NC(c3cc(C4CC4)no3)=O)nn2)nncn1C N1(C(C(COC)N(C)C)=O)CCN(C(c2cc(O)n(C)n2)=O)C(CC(C)(C)C)C1 C1(C(=O)NC(C)C)CC(NC(=O)C=Cc2cnn(C)c2)C1(C)C C=CCCCC(C(=O)NC(C)(C)CC=C)NC(c1nccnc1N)=O C12(NC(=O)CC3CCC(O)C3)CCCC1N(C(C1CC3(CC3)C1)=O)CCC2 c1(OCC(=O)NC2CCN(C(C(CC)C#N)=O)C2)ccc(F)cc1O C(=O)(C(O)CC(F)F)N1CC(NC(CC2CC(=O)NC2=O)=O)(CO)C1 N1(C(c2ccc(SC)s2)=O)CCC(NC(C2CCN(C)C2=O)=O)C(CO)C1 Cc1cc2cc(C(N3CC4OCC(NC(C5CC5F)=O)C4C3)=O)[nH]c2cc1Cl c1(NC(CN(CCC2=CCCCC2)C(CC)C)=O)cnn2cccnc12 c1(C(=O)NC2(CNC(Cc3c(OC)nccc3)=O)CC2)cc(F)c(SC)cc1F C(=O)(C1=CCCCC1C)NC1(CC=C)CCN(C(=O)CCCC(F)(F)F)C1 N1(C(C=CC(C)(C)SC)=O)CC2CC2(CNC(c2cn(C)nc2C(F)F)=O)C1 c1(C(=O)NCC2C(NC(CC=C)=O)CC2)ccccc1S(=O)C(F)(F)F C(=O)(C(C(F)(F)F)C(F)(F)F)N(CCNC(C(CC)NC(N)=O)=O)C(C)C CN1CC=C(CC(=O)NCC2(NC(c3cccc4c3C(=O)NC4)=O)CCC2)CC1 C1(NC(c2nc(C)c(C)s2)=O)CN(C(C2(C(N)=O)CC2)=O)CCC1C C(=O)(CCC(CF)CF)NC1CCOCC1.C12CN(C1)C(=O)C=CC=C2C C1(NC(C(F)=C(C)C)=O)CC2CCC(C1)N2C(c1ncc(C(F)(F)F)cc1N)=O C1(CC(=O)NC2CC(NC(C34CCCC3C4)=O)C2)CCS(=O)(=O)CC1 CC(O)CCCC(=O)NCC1CN(C(=O)CSCc2cccs2)CCO1 c1(NC(CN2C3CC(NCC(CC)(C)C)(C3)C2)=O)ccc(C#N)cc1 C1(NC(C2(C=C)CCC2)=O)CCCN(C(C2CCC(C(F)(F)F)O2)=O)C1 C=C(C)CC(=O)NC(C)(CNC(=O)C(C)COCC)Cn1cccn1 N1(CC(=O)NC2C(NC(C(C)SC)=O)C2)CC(=O)Nc2ccccc21 CN1CCCC(C(=O)NCC(C(=O)N2CCC(c3ccon3)C2)N(C)C)C1 C1(C(=O)NC(CCCC)C)C=CCN(C(C2CCOCC2)=O)C1 C=CCC(CC(C)C)C(=O)N1CC2CC1CN(C(=O)C(C)(C)COCC(F)F)C2 C(=O)(C1=NN(C)C(=O)CC1)N1CC(C(c2cn(CC3C4(C(C(=O)O)C4)C3)nn2)C)C1 C1(C)(CNC(Cc2ccc(C)cc2)=O)CN(C(=O)C=C2CCC2)CC1C Cc1cc(C(=O)NCC2CCN(C(c3c(C)[nH]c(C)c3C)=O)C2)ccc1Cl c1(COCC)nnc2n1CN(C)C1CCN2CC1.c1(C(=O)OC)ccsc1 C(=O)(C1CCc2c(Cl)cccc21)N1CCC(C(CNC(C2(SC)CC2)=O)F)CC1 CC1(C)CN(C(=O)C=CC(F)(F)F)CC1C(N1CCC(C)(O)C1)=O Cc1c(C(=O)NCC2CC2NC(=O)CN2CCCC2=O)cnn1C1CC1 C(=O)(C1Cc2ccccc21)NC(C1(O)CN(C(c2c(N)ncc(C)c2)=O)C1)C c1(CNC(c2n(C(CC)C)nnn2)c2ccsn2)ccc2c(c1)CCCC2 c1(CC)cccc(NC(=O)NC(C)CC2CCN(C)CC2)c1C c1(OC)cccc(CN(C)CC2CC(O)CN2C(=O)C(C)OC)c1SC c1(OCC(=O)NCC2(Oc3c(C)nc(Cl)cc3)CCC2)cccc(S(C)(=O)=O)c1 CN1CCCC12CN(C(C1CC=CCN1C(=O)COC1CCC1)=O)C2 c1(NC(=O)C(N2CCC(CNC(c3csc(O)n3)=O)C2)=O)ccccc1 C1(CC)(NC(C2CCC(O)CC2)=O)CCN(C(=O)C(n2cc(C)cn2)C)CC1 C1(CC)CCN(C(C2CC23CCN(C(=O)CC(O)CN(C)C)C3)=O)C1(C)C c1(CC)nc(C(N2CCC(CF)(NC(=O)CCC3CCOC3)C2)=O)c(C)o1 CCC(C)C(CNC(=O)CCOCCCNC(=O)C=C1CCC1)CO CC1(C)C2CCC1(C(=O)NCCC(O)C(=O)NCCc1ccccc1O)C2 CON(CCO)C(=O)C1CCCCN(C(=O)CC2CNC(=O)O2)C1 C1(COC)(CNC(=O)CC2CCCN(C)C2)CCCN1C(=O)CCc1csnn1 C1(CNC(CN(C2CCCC2)C)=O)COCCN1C(=O)C(C1CCOCC1)=O N1(C(c2cc(CCC)n(C)n2)=O)CCCC2C1CCN2C(c1cncc(C)c1)=O CCCC(C)(CC)C(=O)N1CC(CCNC(c2ccc3cnnn3c2)=O)C1 N1(C(C(c2ccnn2C)C)=O)CCCCCCC1C(=O)NC1(CO)CCOCC1 C1(CNC(CSCCC)=O)CC(C)(C)CN1C(C12CC(OC)C1C2)=O S(=O)(=O)(c1cc(-c2ccc(C#N)c(F)c2)c(C)cc1C)NCCCOCC Cc1nc(N2CCC(c3cccc(F)n3)C2)c2cnn(CCO)c2n1 C1(C)(C(=O)NCc2scc(CNC(COCC(=O)NC)=O)n2)CC(C#N)C1 C1(NC(C(CSC)O)=O)C2CN(C(C3CCOC3c3ccc(Cl)cc3)=O)CC12 c1(C(=O)NCC2CC(NC(C(CC)C(C)(F)F)=O)C2)cccc2c1OC(F)(F)O2 Cc1cc(CCC(N2CCC(Cc3ccccn3)C2)=O)on1 C1(CCOC)CC(Oc2ccccc2)CCN1 C1(NC(N2C(NCc3n(CC)ncc3)CCC2)=O)CCC2(CC1)NC(=O)NC2=O C#CCC(O)C(=O)NCCCCNC(=O)Cc1cnc(C(F)(F)F)s1 c1(NC(CCNC(C(C)OCC#C)=O)(C)C)ncnc2[nH]cc(CC)c12 N1(C(c2n(C(C)C)ccn2)=O)CC(CNC(c2nc(=O)n(C)[nH]2)=O)C(C)(C)C1 N1(C(C2C(NC(c3c(C)cccc3)=O)CCC2)=O)CC2CC=CCC2C1 CC1(C(=O)NCCCCC2CN(C(=O)C=Cc3ccc(Cl)s3)C2)CCNC1=O N1(C(=O)Cn2nccc2N)CCCC(C(C)NCC2(C#C)CC2)C1 CCCC(CCCNC(=O)CCCC1CC1)NC(=O)CC(=O)NCC N1(C(=O)Nc2nc(C(C)C)nc(O)c2)CC2CC(C1)C1CCCC(=O)N1C2 CCCC(C(O)C(=O)N(CC(O)C1CC1)C)NC(=O)CC1=CCOCC1 C1(NC(c2c(OCC=C)cccc2)=O)CN(C(=O)CCCC(C)C)CC1C=C c1(CN(C)C(C2(CNC(=O)CCC3CCOC3)CC2)=O)cccc(C(F)(F)F)c1 C1(CC(=O)NC(COCC)C(C)C)CC(O)CN1C(c1cscc1CC)=O N1(C(CC(=O)Nc2nccs2)=O)CCC2(CCC(NC(c3cc[nH]n3)=O)C2)C1 N1(C(C)C(=O)NCC(c2ccccc2F)NC(C2(O)CC2(C)C)=O)CCCCC1=O c1(N2C3CC(CNC(C(C(CC)C)O)=O)(OC3)C2)ccc([N+](=O)[O-])c(C)c1 N(C(=NCC1(N(C)C)CC1)NC1CCCc2nc(C)sc21)C(COC)C C(=O)(CC(F)(F)CC)N(C(CC(=O)NCC1CN(CC)C(=O)O1)CC)C N1(C(C2CCC(C(=O)OC)O2)=O)CCCC(NC(c2cnc(C)cn2)=O)CC1 N1(C(C(c2c(Cl)cccc2Cl)C)=O)CCN(C(c2c[nH]nc2F)=O)C2(CC2)C1 C(=O)(C1=CCCCCC1)N1CCC(C(=O)NCC(O)CC2CCCC2)OCC1 c1(-c2ccnc(CN3CC(C)(C)OCC3)n2)ccc2ccccc2n1 c1(C(=O)NCCC2CC(OC)CN2C(=O)C=CC2CC2)cccc2oc(O)nc12 C1(C)(C(N(CC(C)(C)CNC(C2CC2C(C)(C)C)=O)C)=O)CC(C)(C)C1 c1(C(=O)NCC(CO)NC(=O)CSCc2ncc[nH]2)sc(F)cc1Cl c1(OC)ccc(CCCNC(=O)C(=O)NCCC2CCC(N)C2)cc1 N1(C(C2(F)C(C)C2)=O)CC2C3CCC(C2C1)N(C(c1cnn2c1CCC2)=O)C3 C(=O)(CCCCNC(=O)CCC1NC(=O)NC1=O)OC(C)CSC C1(NC(C2COCCN2)=O)CCCC2(C1)CC(O)C2 C1(NC(CN(C(=O)C(C2CCC2)OC)CC)=O)CC(C)(C)O1 c1(C(N2C(CNC(c3cnc(OC)nc3)=O)COCC2)=O)c(Cl)ccc(F)c1N c1(CC)cc(C(N2CC(O)(C(C)NC(=O)C3=CCSC3)C2)=O)ccc1Cl CCCC(O)CC(=O)NCCN(CCOC)C(C1(C(F)(F)F)CCN(C)C1)=O c1(C(N(C)CC2CC2(C)C)=O)c(Br)ccc2ccccc12 c1(C(=O)NC(CC)CNC(C2CC(O)C2)=O)c(S(N)(=O)=O)ncn1C C1(O)(C(N2CCC(NC(c3cc(OC)ncc3)=O)(CF)C2)=O)CCCCCC1 c1(C(N2CC=CC(NC(C(CC#C)O)=O)C2)=O)nc(Cl)ccc1OCC N1(C(CCC(C)c2ccccc2)=O)CCC2(CCC2)C(NC(=O)CCC(C)(C)F)C1 Cc1[nH]nc(C(=O)Nc2ccc(CCS(C)=O)cc2)c1F c1(CN2CC(CC(=O)OCC)N(Cc3ccccc3)CC2)cc(I)c(C)c(I)c1 C1(NC(c2c(C)nn(CC(F)F)c2)=O)CCC(C)(CNC(c2csnn2)=O)CC1 C1(NC(c2c[nH]cc(Cl)c2=O)=O)CN(C(C2CCCC2F)=O)CCC1CO C1(CNC(CCC2(C)N=N2)=O)CCCN(C(=O)CC(C)n2ccnc2)C1 C12(COC)CC(CNC(=O)C(CCO)N(C)C)(CN1C(=O)CCC(=O)N(C)C)C2 N1(CC(=O)NCC2CC(NC(C(=O)NCCNC(C)=O)=O)C2)CC(C)OC(C)C1 c1(OC)c(C(=O)NCC(C)(C)NC(=O)CSCc2cccs2)cccc1Cl c1(C(C(=O)NCC(CNC(C(C=C)O)=O)CO)(F)F)ncccc1Br Cc1c(C(N2CC=CC(NC(=O)C=C3CCC(C)C3)C2)=O)cnn1C(C)C c1(C(N2CCC(C(C)NC(c3ccc(C#N)o3)=O)C2)=O)onc2c1CCCC2 c1(C(N2CC(O)(C(C)NC(=O)CC3(N4CCCC4)CC3)C2)=O)cnn2ccccc12 CN1CC2(CC2)CC1C(N1CCC(F)CC1C(N1CCC1(C)CCO)=O)=O C1(O)(CN(C(=O)CSc2nc[nH]n2)C)CCN(C(=O)C(C)(C)C2CCCCO2)C1 c1(-c2cn(CC(=O)Nc3cccc(C4CC4)c3)nn2)cnc2ccccn12 C(=O)(CCS(=O)(=O)C(F)(F)F)NC(C1CN(C(=O)CC2CCC(=O)C2)C1)C O=C(C1CCc2ccccc21)NC1C2CC1N(C(c1cscc1Br)=O)C2 C(=O)(C(C(C)C)N(C)C)NC1CC(CCNC(c2ccn(CC(C)C)n2)=O)C1 c1(NC(C2CCNC2)=O)ccc(F)c(Nc2cc(-n3cncn3)ncn2)c1 C1(c2c(OC)nn(C)c2)CCN(N2CCc3[nH]c4cc(Br)ccc4c3C2)C1 C(=O)(C(C)(C)CC(F)F)NC1CN(C(C(C)OCCC=C)=O)CC(O)C1 C12(C(=O)NCC(CN(C(C(C)(C)OC)=O)C)O)CC3CC(CC(C3)O1)C2 c1(C(=O)NC2C(N(C(C(C=C=C)C)=O)C)CCCC2)cc(C)cc([N+](=O)[O-])c1N c1(C2(Cc3c(C(N(CC(=O)NCC)C)=O)c[nH]n3)CC2)ccc(OC)cc1OC CC(C)(C)C(C(=O)NC1(CNC(C2(CO)CC2)=O)CCCCC1)C(O)C(F)(F)F C1(CC)CCC(CNC(C2(NC(C3CC4(CC4)C3)=O)CC(O)C2)=O)O1 CC1COc2c(C(=O)NC3CC3CNC(c3snnc3C3CC3)=O)cnn2C1 C(=O)(C(C)S(N)(=O)=O)N1C(COC)(CNC(=O)CC2CN3CCC2CC3)CCC1 N1(C(c2ncn(CC)c2)=O)CCC(C)CC1C(=O)NCC1(CC)CCOC1 n1(CC(C)NC2CC2(c2ccccc2)C)c(=O)ccc2ccccc12 c1(OC)ccc(C(N2CCSC(C(F)(F)F)C2)C(=O)NC2CCOC2)c(Cl)c1 c1(N(CCS(=O)(=O)NC)C)nc2cc[nH]c2c(=NC(C)c2ccc(Cl)c(C)c2Cl)[nH]1 c1(CC(N2CC3CCC2CN3C(C2CCOCC2)=O)=O)cc(F)ccc1[N+](=O)[O-] C=CCCC(F)(F)C(=O)NC1CC(F)(CNC(=O)Cc2cc(F)ccc2Cl)C1 CCC(C)(C)CC(=O)N1CC(C)(C)CC1C(=O)NC(C)C(C)C(=O)OC C1(C(=O)NCCC2(CNC(=O)CC3OCCO3)CC2)COc2ccc(Cl)cc2C1 C(c1c(C)nn(CC(C)C)c1Cl)=CC(=O)NCCNC(C(C)OCC)=O Cc1cc(Cl)c(C(N2CCCC2Cn2cc(C3(O)CC3)nn2)=O)cn1 c1(C(N2CC(CNC(C=C(C)Cl)=O)C(C)C2)=O)nc(C)ncc1Cl C1(CC(=O)NC(c2ccco2)CNC(CSC)=O)COC(=O)N1 c1(C(C(=O)N(C2(CN)CC(F)(F)C2)CC)(C)C)ccc(F)c(C)c1 C1(C(N(CC(=O)NCC(C)C)C(=O)N)=O)C2CCC(C2)C1C.C1CC12CCC2 c1(C(N2CC(OCCNC(C34C(C)(C)OCC3C4)=O)C2)=O)nc2ccccn2n1 C1(C(=O)OC)CCC(CC(=O)NC(C)C(C)(C)NC(C2(C)CS(=O)(=O)C2)=O)CC1 C1(C(N2CC(CCC=C)(C(=O)NCCCc3n[nH]c(C)n3)C2)=O)CCCCC1C c1(C(=O)NCCC2CCCN(c3cnc(F)cn3)C2)cc2c(nc1O)CCC2 C1(CNC(C(=O)Nc2cccc(-c3cn(C)nc3)c2)=O)CCC2(CC1)CC2 C(=O)(CCCCC(F)(F)F)NC1C(C(C)NC(=O)CCCCC)CCC1 CC1CN(C(=O)OC(C)(C)C)CC1N=c1[nH]nc(-c2ccccc2)s1 C12(C(N3CC(NC(C4OCC(C)C4)=O)C(C)C3)=O)CCCC(C)(C1)OC2 c1(NC(=O)NC(C#C)(C)C2CCCC2)cc(-n2cccn2)ccc1Br N1(C(C(CC(C)C)=O)=O)C2COCC1CC(NC(c1coc3c1COC3)=O)C2 C=CC(C)(C)CCCNC(=O)C(C)(C1CC1)N(C(=O)CCCCSC)C C(C(COC)CC(=O)NCC(CNC(=O)C(C)NC(C)=O)C(F)(F)F)OC C(C(C(=O)NCCCCCN(C(=O)CCCc1nncn1C)C)OC)OC C1(C)(C(=O)NC2CN(C(C(C)Sc3ncccn3)=O)C2)CCC(=O)CC1 N1(C(C(CN(CC)CC)F)=O)CCC(C)(NC(c2ccnc(OC)n2)=O)C1 C1(c2nnnn2CC2CC2)(NC2(C=C)COC2)CC2C(Br)C(O)CC12 Cc1cc(Br)cc(C(N2CCN(C(=O)CCNC(=O)CC3CC3)CC2)=O)c1N Cc1cn2cc(C(=O)N(C(C)CNC(c3cc(N)cc(F)c3)=O)C)nc2s1 CCC(C)C(=O)C(=O)NCCn1ccc(C(=O)NCc2cnn(C)c2C)c1 N1(C(C(C)SC(F)(F)F)=O)CCn2nc(CNC(c3cccc(O)n3)=O)cc2C1 c1(C(N2C(C)CC(CNC(c3c(C)cccn3)=O)C2)=O)ccc(F)c(O)c1 c1(C(=O)NC2C(OC)CN(C(C3CCSC3)=O)C2)cnn2cnnc2c1 c1(CC)[nH]nc(C(N2CCC2C(=O)Nc2ncccc2C)=O)c1F N1(C(=O)NC(c2ccc(C#N)cc2)CC(=O)NCCCCl)CCN2CC(O)CC2C1 c1(C(C(=O)NC(C)C)C)cc(NC(C2(C(F)(F)F)CC2)C)ncn1 c1(C(N2CCC(O)(C(C)NC(CC(C)C)=O)C2)=O)cc(N)nc(Br)c1 C(CCC(=O)N1CCCC1CNC(C1CC1(C)C(F)(F)F)=O)OCCC C1(C(N(CCNC(C(C)c2ccco2)=O)C)=O)CCCCS1 CC(C)C(CN(C)C)C(=O)N1CCC(CO)(CNC(=O)CC2CCSC2)CC1 c1(NC(c2ccc(C(=O)Nc3n(C)ncc3Br)[nH]2)=O)ccc2ccccc2n1 O(C1CCCc2ccc(Br)cc21)C(c1nncc(OC)c1)=O CC1CC(C(N2CCC(O)(C(N)=O)CC2)=O)CN(C(c2cnn(C)c2)=O)C1 C1(CNC(c2cnccc2Cl)=O)CN(C(c2nc(C3CC3)cs2)=O)CC12CC2 C1(NC(=O)CC23CCCC2C3)CCC(NC(c2cncc(F)c2)=O)CC1 Cc1ccc(S(=O)(=O)N2CC(C(F)(F)F)C(F)(c3ccccc3)C2)c(C)c1 c1(C2(CC(=O)NC3CC3NC(=O)C(F)C3CCC3)COC2)ccccc1 c1(NC(CCC=C)c2nnnn2C(C)(C)C)cnc2c(O)cccc2c1 CC(C)C(C(=O)Nc1[nH]nnc1C1CCNC1)NCCNC(=O)OC(C)(C)C CC1(C)CCCN(C(=O)CC2CCCC3CC23)C1C(=O)NOCC1CCOCC1 C1(NC(c2cc(OC)no2)=O)CCN(C(=O)C(C)O)CCC1CO C1(C(=O)NCc2cccnc2O)CN(C(=O)CCN2CCCCC2)C2(CCC2)C1 C1(CCC(=O)NCC2C(NC(C(C)O)=O)CCC2)CCCCN1C C#CCC(CC#C)C(=O)N1CCN(C(c2cccc(O)n2)=O)C(CS(C)(=O)=O)C1 C(=O)(CCCn1nnnc1C1C=CC(CNCC(C)(C)NS(N)(=O)=O)C1)OC CN1CCOC(C(=O)N(C)CC2COCCN2C(C2CCCC23CC3)=O)C1 N1(C(c2cn(C)nc2O)=O)CCCN(CCCCNC(C2CCCC2O)=O)CC1 C(=O)(C(C)(C)C(=O)NCC(C)(O)CNC(c1cncc(N(C)C)n1)=O)N(C)C Cc1ccc(C(N2CCCC(CCNC(C3CCC(=O)N3)=O)C2)=O)c(C2CC2)c1 N1(C(CC(=O)NCC)=O)CCCC(C)(C)C1CNC(c1ccc(N)cc1OC)=O C1(CCNC(C(C=C)O)=O)CSCCN1C(c1cc[nH]c(=N)c1)=O c1(CC(=O)NCCC2N(C(CCC(=O)OC)=O)CCCC2)ccc(F)cc1F c1(CC)cc(F)ccc1C(N1CC(CCNC(=O)CC(F)F)OC(C)C1)=O c1(N(CC(C)NC(C2(c3cc(C)on3)CCC2)=O)C)ncnc2scnc12 C12(NC(C(C)=C(C)C)=O)CCCC1CN(C(=O)Cc1csc(-c3ccoc3)n1)C2 C1(C)(NC(c2cnc(COC)s2)=O)CCN(C(c2cccc[n+]2[O-])=O)C1 C1(NC(COCC)=O)CCC2CN(C(c3ccnn3CC)=O)CCC2C1 C1(N(C(=O)Cn2cccc2)C)CN(C(C2CC(=O)N(C(C)(C)C)C2)=O)CC1(C)C N1(C(c2cnccn2)=O)CC2CCC2(CNC(C2(Cl)CC23CCOCC3)=O)C1 c1(C(N2CC(NC(C(CC)O)=O)C(C3CC3)C2)=O)cc2nc(Cl)ccc2o1 c1(C(NOCC=C)=O)cc(CNC(=O)Cc2[nH]cnc2C)[nH]n1 c1(C(N2CCCC(NC(CCC)=O)C2C)=O)ccc(C(F)(F)F)c(Cl)c1Cl N1(C(C(C)(F)F)=O)CCC2(CCC(CNC(c3ccnnc3S)=O)OC2)CC1 Cc1cc(C(=O)NCCCCN(C)C(C2(C)CCCNC2=O)=O)cc2c1CCC2 C1(NC(c2scc(C(N)=O)c2)=O)CC(NC(C2CCC(=O)NC2)=O)C(O)C1 CC(c1ccccc1Cl)=CC(N1CCC(CF)(NC(=O)C(O)C(F)(F)F)C1)=O C1(NC(=O)CN2CCC2)CCN(C(=O)CCOC2COC2)C12CCC2 N1(C(C(CC)C2CCOCC2)=O)CCN(C(C2CC(O)CN2C)=O)C(C(F)F)C1 c1(NC(C2CN(c3ccc(F)cc3)C(=O)C2)=O)nccc(Cl)c1I c1(NC(c2ccccc2-n2cccn2)=O)cc(Cl)ccc1CO c1(C(N2CCN(C(=O)CCc3cscn3)C(CCO)C2)=O)csc2nnsc12 N1(C(CC(C)(C)F)=O)CCCC2(C1)CN(C(c1nccnc1C(N)=O)=O)C2 n1(CCCN(CCCC)C)c(N2CCC(c3nncn3C)C2)nnc1C(C)OC N1(C(CC2CCC(OC)CC2)=O)CC2(CCN(C(=O)COC(F)F)C2)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CC(OC)CN(C(C2(C#C)CCC2)=O)C1 c1(C(=O)NC(C2CCN(C(=O)CCC3CC3(Cl)Cl)CC2)C)ccnc(CO)c1 C(=O)(C(C(C)(C)O)NC(=O)CCCc1ncco1)N1CC(S(C)=O)C1 c1(OC)cc(C(=O)NC2CN(C(c3ccon3)=O)CC2C)c(Br)c(F)c1 c1(C(=O)NC2(C(=O)NC(C#CC)(C)C)CC2(C)C)c(C)noc1C C(=O)(C#CC1CCOCC1)N(C)CCN(c1ncc2c(n1)COC2)C O(N=C1CCCCCC1)CC(N1C(C)CC(CNC(c2ccsc2C#N)=O)C1)=O C(=O)(CCCC(F)(F)F)NC1CC(NC(c2ccc(C(CC)(C)C)cc2)=O)C1 C(=O)(C(CC)C(C)(C)CC)NCC1(COC(C)=O)CCN(C(C(CCC)OC)=O)C1 C1(C(N(CC(C)CNC(C2(C)CC=CCC2)=O)C)=O)CCC2(CC1)CC2(F)F N1(C(C)C(=O)NCCNC(C2(C)CC2(C)C)=O)C(=O)CCC1=O c1(C(N2C(CC(=O)NC3(CSC)CC3)CC(C)(C)C2)=O)cc(C#N)ccc1N Cc1ncc(Br)cc1C(=O)NCC1(O)CCN(C(C2CN(C)CCO2)=O)C1 c1(OC)cc(SC)cc2c1OCCO2.N12CCOCC1(C)NC(=O)C2 c1(C(C(F)(F)F)C(=O)NCC(C)CN2CCOC2=O)cc(Cl)cc(Cl)c1 Cc1c(C(N2CCN(C(C3CCC(C)O3)=O)CC(O)C2)=O)cnc2ncnn12 C(=O)(CC1=CCN(C(=O)C(C)CC2CCC2)CC1)Nc1cn(CC)c(=O)cc1 Cc1cc(C(=O)NC2CCCN(C(c3csc(=N)[nH]3)=O)C2C)cc(C)c1F C1(CC)CN(C(c2cnc(F)c(Cl)c2)=O)CCC1N=c1cc(C)nc(OC)[nH]1 c1(C(=O)NC2C(C(N3CCN(C)C(CO)C3)=O)CC2)cc([N+](=O)[O-])nn1C C(=O)(CCC1CCc2ccccc21)N1CC(NC(=O)CCC2CCC2)C2(C1)CC2 N1(C(c2cncnc2)=O)CC(C2CCN(C(c3ncncc3Br)=O)CC2)C1 Cc1ccc2ncn(CC(=O)NC3CCCC3NC(c3ccnc(S)c3)=O)c2c1 c1(C(=O)NC2CC(NC(CCCNC(C)=O)=O)C2)cc2sc(Br)cc2[nH]1 c1(C(=O)NCC2CC(NC(c3ccc(CC)cc3)=O)C2)cc2cc(C)ccc2s1 C1(c2n(CC(F)F)nnn2)(Nc2ccc(-c3ncc[nH]3)nc2)CCCC2CC12 C(=O)(CCC(C)S(C)(=O)=O)N(C1CCCN(C(C=C(C)C)=O)CC1)C CC(C(=O)NCC1CCN(C(C2CC3(C2)CC2(CC2)C3)=O)C(C)C1)C1=CCCC1 Cc1cnc(Br)cc1NC(C1CC(F)CN1C(=O)CCc1cc(Cl)ccc1Br)=O c1(C(N(C)CC2N(C(C=CCCC)=O)CC(F)C2)=O)cc2c(s1)CCSC2 N(C(=NCCC(O)c1ccccc1)NCC1CNC(=O)O1)CC(C)C C1(C)(NC(C2(NC(CC(C)OC)=O)CC(F)C2)=O)CCCC1(C)C C(c1nccs1)=CC(=O)N(C(C)C(=O)NCC1(O)CCSC1)CC Cc1cc(C(=O)NC(C)(CO)C(=O)NC(C)CC(N)=O)ccn1 C(=O)(C1CCCCc2ccccc21)N1CCC(NC(COC)=O)(CO)CC1 CC(C)C(CCNC(=O)CC(C)C1CC1)NC(=O)CSCc1cccs1 c1(COC)cccc(C(=O)NC2(CNC(=O)CC(C)n3cccn3)CC2)n1 c1(CN(C)C(c2cnc3cc(F)ccn23)=O)cn2cc(Cl)ccc2n1 c1(C(c2nnnn2CCCSC)NC(C=C)C2CCC2)csc(CCC)n1 Cc1ccc(C(=O)NC(C)(C)C(=O)N(C2CC2)CC2CCOC2)o1 CN1CCN(C(C2CCOC2C(F)(F)F)=O)CC1CNC(C1C2CC3C(C2)C13)=O CCCCCC(O)C(C)C(=O)NCC1CC(NC(C2(C3CC3)CC2)=O)C1 CCCCN=C(NCCCOC1CCCCC1)NC1CCCSC1 N1(C(Cc2c(C)scc2)=O)CCN(C)CC1C(=O)N(C)Cc1ccns1 C(CCC(C)NC(=O)COCC1CCC1)NC(CSCCC(C)C)=O CCCC(CCC)C(=O)N1CCN(C(c2cnsc2)=O)CC(C)C1 c1(SC)ccc(C=CC(=O)NCCCC(C)NC(=O)CN(C)CCO)cc1 C=CCC(CC=C)CS(=O)(=O)N1CCC2CCCC12CO C1(CC(=O)NC(C2(CNC(C=CC(C)(C)SC)=O)CC2)C)CCCCO1 C1(C)(CCC)CCCN(C(=O)C(CCC2CC2)N(C(C2(SC)CCC2)=O)C2CC2)C1 N1(C(c2cc(C)[nH]c2C)=O)CCCC(NC(c2coc(O)n2)=O)C1C N1(C(C2C(C=C)CC2)=O)CCC2(CCCN2C(=O)Cc2cccc(F)c2O)C1 N1(C(C=CC=CC)=O)CC2CC(N(C(=O)C(C)P(C)(C)=O)CC)C1C2 C12(C(=O)NCC3CCC(C(=O)NCCC(C)(C)O)CC3)CCC(CC1)CO2 c1(C(C(=O)OC(C2CCCCO2)C)(F)F)ncccc1Br N1(C(C2(C=O)CCC2)=O)CC2C(CN)C2C1.c1(C(N)=O)cc(C(=O)N(C)C)co1 Cc1cc(N)c(C(=O)NC2CCC3CC23CO)cc1C C1(CNC(c2on(C)c(=O)c2)=O)CC2CCC1N(C(=O)COC1CCCOC1)C2 N1(C(C#C)=O)CCC2(CC2C(=O)NC2(C(F)(F)F)CC2)C1 C(=O)(C(O)CCC(C)C)N(CCCNC(C1C(C)(C(=O)OCC)C1)=O)CC CC1=CCC(C(=O)NC(C)C(=O)N(C)Cc2cc(C)nn2C)CC1 c1(C(=O)NC2CN(C(C3CC34CC(O)C4)=O)CCC2O)cccc2c1CCC2 c1(-c2cnc(SC)c(C)c2)ccc2c(C(=O)NCc3ccc(Br)cc3)noc2c1 N1(c2ncnc(OC)c2OC)CCn2ncc(CNC(=O)C=C(C)C)c2C1 C1(C(=O)OC)CN(C(=O)C(CC(N)=O)Sc2ccccc2)C2(CCC2)C1 C(C(C(F)(F)F)N1CCN(C(c2cn[nH]c2)=O)CC1)NC(C=CCOC)=O c1(CCOCCOC)cccc(CC)c1C.C1(=O)C(=O)NC12CC2.C(C(=O)NC)OC CCC(CCCC(=O)NC(C)Cc1ncn(C)n1)NC(C1(O)CCCC1)=O N1(C(=O)NCCc2ccc(C)cc2Cl)CCC(C2CCCC2)C1 N1(C(c2cc(C)sn2)=O)CC2(CCNC(C3CC34CC4)=O)CCC1C2 CCCCCCCCCCCn1nc(CSC)nc1-c1nn[nH]c1Cl C1(C(N2C(C(C)(C)OC)CCC2)=O)CN(C(=O)C2=CCCC2C)CCN1C CCCCCCCCCC(=O)N1CCCC(CNC(=O)C(F)CC(C)C)C1 O=C1CCCC(CC(=O)NCC2(C(=O)NCCC(F)=C(F)F)CCCCC2)C1 C=C1CC2(C1)CC(C(N1CCN(C(=O)CCN3CCOCC3)C(CCC)C1)=O)C2 N1(C(C=CCOC)=O)CC(NC(c2snc(O)c2Cl)=O)CC(O)C1 CC(c1ccco1)=CC(=O)N(CCCNC(c1ccnc(C2CC2)n1)=O)CCO C1(O)(CNC(CCOCC)=O)CCCN(C(=O)CNC(c2cccc(C)c2)=O)C1 c1(C(=O)Nc2nc(C(N3CC4CCCC4C3)=O)cs2)ccc(O)c(Br)c1 CC1(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CC(C(=O)O)C2(C)C)=O)CC1 C1(C(=O)NCCC(COC)(C)C)CCCN1NC(=O)C(F)(F)CO c1(C(=O)NC2CCN(C(c3scc(C)c3)=O)C2C2CC2)sc2ccccc2c1C C1(NC(C(C)OC)=O)CCCC1NC(=O)CCCc1ccccn1 C(=O)(C1=CCCOC1)N1CC(CCC)C(C(N2CCC(c3cc[nH]n3)C2)=O)C1 N1(C(C(C(=O)OCC)OC)=O)CCC(C(=O)NCC(CC)CCO)C12CCC2 c1(C2CN(C(CSCC=C)=O)C2)cc(CC)no1.C123CC(C1C2)NC3=O CCCC(C)(C)CC(=O)NC12CCN(C(c3cnc(C4OCCO4)s3)=O)CC1C2 c1(C(=O)NCC2C(CNC(C3(C)CC=CCO3)=O)C2)ccc(CO)c(Cl)c1 C12(NC(C(C)C(F)(F)F)=O)CCCCC1CN(C(c1cnc3n1CCCC3)=O)C2 C1(C2CCC2)(C(N2CC(O)CC(NC(c3c(C)nncc3)=O)C2)=O)CC1(F)F CC#CCCC(=O)NCC=C1CCN(C(c2cccc(C(C)(C)C)n2)=O)CC1 CC(C)CC(Cc1ccn(C)n1)C(=O)OCC(=O)N(C1CC1)Cc1cscc1Br c1(CC)ccc(C(=O)NCC(O)CC(=O)NCCN2CC=C(C)CC2)cc1 C1(C(N2CCC(CNC(CCc3nnc(C(C)C)o3)=O)C2)=O)CC2(C1)CC(O)C2 C1(C)(COC)CC(NC(C2(S(N)(=O)=O)CC2)=O)CN1C(=O)COC1(C)CCCC1 C(=O)(C1CCCn2nccc21)OCc1nccc(C)n1 CC1(C)C(NC(C2CCCCN2N=O)=O)CCN1C(c1csnc1Cl)=O N1(C(c2ccc(OC)cc2)C(=O)NC)CC2C(C(=O)NCCC#N)(C1)CS2(=O)=O N1(C(COCCCC(C)C)=O)CCN(C(C2CCCCN2N)=O)CCC1C c1(C(=O)NC(C2CN(C(C(C)=CC)=O)C2)C)ccc(NC(C)=O)cc1Cl N#CC1(C(=O)NCC2CCCN2C(c2ccc(C3CCOC3)s2)=O)CCCCC1 N1(CC)CCOC(C(=O)N(C(C)CN(C(=O)CCC(=O)c2ccccn2)C)C)C1 C(C(C)(O)CC(=O)N1CCN(C(c2cnc(F)c(C)c2)=O)CC1C)OC CC(C)(CO)C(CO)NC(=O)C(Cn1cncn1)NC(c1csc(Cl)c1)=O C(=O)(C(C)C(C)n1cccn1)NCC1C(NC(CSCCCC)=O)COC1 C1(CC(c2nnnn2CCCOC)NC(C=C)(C)C)CC2CCC1C2 C1(NC(c2ccno2)=O)CCOC12CCN(c1nnc(C(F)F)o1)CC2 c12cccnc1CNC2=O.N1(CC(=O)NCCOC(=N)O)CCSCC1 CCC(CCCC(=O)N1CC2COCC2(CO)C1)NC(=O)CSC(F)(F)F c1(C(N(C)CC2N(C(CNC(=O)OC)=O)CC(F)C2)=O)cc(N)cc(F)c1 c1(C(=O)NCC2C3CN(C(CCCC(N)=O)=O)CC32)ccc2c(c1)COB2O Cc1cc(C(=O)NCCNC(c2nc(OCc3ccccc3)c(C)s2)=O)n(C)n1 N1(C(c2cncc(SC)c2)=O)CCC(C2(NC(C3CC(F)(CO)C3)=O)CC2)C1 C(N=c1cc[nH]cc1S(=O)(=O)NC1C2C3CCC(C3)C12)c1c(C)occ1 C(C(CC(=O)NCC1CCC(C)C1)NC(=O)CC1CCCC(=O)C1)OC Cn1ncc(C#N)c1C(N1CC2CC(NC(c3ccc(F)c(F)c3)=O)C1C2)=O N1(C(C(=O)NC(CC)(C)C)c2cnsc2)CCC(C2CCCOC2)CC1 n1(CC)nnc2cc(C(N3CCC(C)CC3CNC(C3CC3C#N)=O)=O)ccc12 N#Cc1cc(NNC(=O)c2cc(Br)ccc2S(N)(=O)=O)ccc1F C(C)(CNC(c1onc(C)c1C(F)(F)F)=O)(C(C)C)NC(C=CC=CC)=O Cc1cc(C)c(C(=O)NCC2(C(C)NC(C3(C(F)(F)F)CCOCC3)=O)CC2)o1 C1(C(N(C(C(C)C)CO)C)=O)CCCCN(C(=O)C(O)CCN(C)C)C1 C1(NC(CC(COC)(C)O)=O)COC2(C1)CN(c1ccnc(C3CCCC3)n1)C2 N1(C(C(C(C)C(F)(F)F)F)=O)CCCC2(CCN(C(c3cccn3C)=O)CC2)C1 C=C(C)CC(C)C(=O)N1CC(NC(c2cc(NC(C)=O)ccc2N)=O)C2(CC2)C1 c1(C(C(=O)NCCOCCCN(C)C(c2cn(C)nc2O)=O)F)ccc(F)cc1 CC1CCCc2cc(C(N3CC(NC(c4cn(C)nn4)=O)C(F)C3)=O)nn21 c1(OC)ccc(-c2ncc(C(=O)OCc3nnc(C)o3)cc2C(C)C)c(OC)c1 Cc1cc(Cl)c(C(N2CCC(C(C)(C)CNC(c3ncoc3C)=O)CC2)=O)cn1 N1(C(CC2CCN(C)CC2)=O)CCC2C(CCCN2C(C2CC2C(F)(F)F)=O)C1 c1(NC(C2CC(NC(C3CCCC(O)C3)=O)C2)=O)cc2ccccc2nc1Br C1(CC)C(C(=O)NCCN(C(=O)C(c2ccc(Cl)cc2)N(C)C)C)CCN1C c1(C(=O)NC2CN(C(C(C(C)C)C#N)=O)C(C)(C)C2)cncc2sccc12 c1(-n2cc(C(=O)NCC(CN(C)C(c3ns[nH]c3=O)=O)O)nn2)ccccc1Cl c1(C(=O)NCC(C2CCC2)NC(Cc2n(C)ccn2)=O)cc(S(N)(=O)=O)n(C)c1 c1(C(N2C(C)CC(NC(CCN(CC)CC)=O)C2)=O)cnc2[nH]ccc2n1 C(=O)(CCC1=CCCCC1)N1CCCCC(N(C(=O)C(F)C2CCCC2)C)C1 C(CNC(c1c[nH]c(=N)o1)=O)(C(=O)NCC(C)CC1CC1)OC C1(CC(=O)NCC(CC)(C)CO)N(C(c2sccc2Cl)=O)CCC1(C)C c1(C(=O)NCCCN(C)C(c2cnn3c2NCCC3)=O)cnc2[nH]nnc2c1 C1(CCNC(c2c(CC)c(C)sc2)=O)C(C)CCCN1C(=O)C(N)=O c1(OC)ccc2[nH]c(C(=O)NCCN(C(=O)CCC(C)(C)F)C(C)C)cc2n1 c1(C(=O)NC(CNC(CC2ON=C(CC)C2)=O)C)nccn2ccnc12 C1(NC(c2c(OC)cc(C)s2)=O)CCC(O)CN(C(C2CC23CC(C)(C)C3)=O)C1 c1(C(=O)NC2C(C)N(C(=O)C(CO)NC(N)=O)CC2)nccc(F)c1Cl N1(C(C(CC)C(=O)OC)=O)CCC2CC(C1)CN(C(c1cc(C)sc1C)=O)C2 Cc1cc(C(=O)NC2CCC(NC(=O)C=Cc3cccs3)CC2)nc(O)c1 C1(CC(N2CC(NC(CN(C)C)=O)C(O)C2)=O)Cc2cc(C(F)(F)F)ccc2O1 N1(C(c2ccc(Cl)s2)=O)CCC2(CCCCN(C(C3(C(F)(F)F)CCO3)=O)C2)C1 CCCCCC(C(=O)NCC1CN(C)CCN1C(c1cscc1OC)=O)C(C)C N1(C(c2cnc(C(C)C)s2)=O)CC2CC1CCC2NC(=O)COc1cnn(C)c1 c1(NC(C(=O)N(C2CN(C(C(C)SC)=O)C2)C)=O)ccccc1C.C1CC1 c1(CC(=O)N(C(CNC(C2CC(C)(C)C2)=O)C2CC2)C)cncn1C1CC1 c1(CC(=O)NCC2N(C(CCOC)=O)CC(C)C2)ccc([N+](=O)[O-])c(N)c1 N1(C(CCOCC#C)=O)CCN(CC2CCCN(C(c3cnn(C)n3)=O)C2)CC1 C1(NC(c2c(CC)noc2)=O)CC(F)CN(C(=O)CC2(O)CCCN(C)C2)C1 c1(CN(c2ccccc2C)CC(C(=O)OC)C)nc(C)cc(C)c1C#N C(=O)(C1=C(F)CN(C(=O)CCOCC2CCC2)CC1)N(C1C(C)C1)C CC1CC(C2CN(N(C)Cc3ccncn3)CC2)C(C)O1 N1(C(c2c(C)ccnc2)=O)CC(NC(c2ccc(O)c(Cl)n2)=O)CC(C)C1 c1(NC(C2C(CNC(C3C(C)=CCS3)=O)CCCC2)=O)cnc(F)cc1C N1(C(C(=O)Nc2cccs2)c2cncs2)CCN(C(C2C3COCC23)=O)CC1 C(N=c1[nH]c(Cl)ncc1F)C1C(NC(c2c(C)nccn2)=O)CCCC1 c1(C(N2CCC(NC(C3(C=C)CCC3)=O)C(O)C2)=O)ccc(S(=O)(=O)N(C)C)o1 Cc1cccc2cc(C(=O)NCCC3CCCN(C(c4cscn4)=O)C3)nn12 CC(C)(C(=O)N1CCC(NC(c2csc(C3CC3)c2)=O)C1)C1CCCCO1 C1(NC(c2ccc(CNC(=O)CC3CCC3(F)F)s2)=O)(CO)CC(F)(F)C1 c1(C(=O)NCC2CC(NC(C3CC34CC4)=O)C2)nc(N2CCOCC2)ncc1Cl C1(C)CCC2(CC2)CO1.c1(CC)cc(C)c(C(=O)NC23CC(NC(=O)C4CC4)(C2)C3)o1 N1(C(CC2(OC)CCCCC2)=O)CC2CCN(C(C3CC3C#N)=O)C2C1 N1(CCNC(C2C(=C)C2)=O)CCN(C(c2cc(C)nnc2CC)=O)CC12CCC2 C1(F)(CNC(C2CCC2)=O)CCCN(C(C2CC2(F)F)=O)C1 C1(N(C(C(=O)N(C)C)=O)CCNC(=O)C(C)(C)C)CCC2CCCC1O2 N1(C(C2CN(C(N)=O)C2)=O)CCC2CC12NC(C1CCCC1)=O c1(CC)nnc2n1CCCC2C(=O)N1CC(NC(=O)CCN2CCC2)C(C2CC2)C1 c1(C(N2CCC(C(C)NCc3cnn[nH]3)CC2)=O)cnc(C(F)F)nc1 C1(CC=C)(NC(=O)C(C)Oc2cccc(C)c2)CCN(C(c2cc(O)cs2)=O)C1 Cn1ccnc1CCC(=O)NCC=CCNC(C1(C)CC1(C)C)=O C(CC(F)F)(C(=O)N1CC(CO)CC1CO)N(C(C(CC)SC)=O)C C(CC(=O)N1CCC(C(N(CC(=O)OC)C)=O)O1)SCC N1(C(CSCCC)=O)CC2C(CC(=O)N(CCOC)CCOC)C2C1 C1(C(C)C)OCCC1C(=O)NCCCCNC(c1cc(C2CC2)no1)=O C1(C(=O)NCC2CCCO2)CC(=O)N(C2CN(CCc3nccs3)C2)C1 c1(C(N(CC(CN(C(C(C)CO)=O)C)O)C)=O)ccc(F)cc1[N+](=O)[O-] CCCC(CC)CC(=O)N1CCCC1(CNC(c1cc(O)nc(O)n1)=O)COC c1(N2CC3C(N(C)CC4Cc5ccccc5C4)C3C2)c(C#N)cccc1[N+](=O)[O-] C(=O)(C(F)C(C)(C)O)NCc1ccc(C(N(CC(C)(O)C)C2CC2)=O)o1 C(=O)(C1=NOC(C)(C)C1)N1CCC(C#C)(C(=O)N(CCC(C)C)CCO)C1 CC(C)C(C(=O)NCCCN(C1CCCCC1)C(=O)C(C)NC=O)C(C)C C1(C(=O)NC2(C(=O)NC3C(C)COCC3)CCCCC2)CCCC(C#N)C1 C1(C(N(C)CC2CCCN(C(c3ccc(COC)o3)=O)C2)=O)CC12CCCCC2 N1(CCC)CCCC1C(=O)NC(CNC(=O)CC1(SC2CC2)CC1)C1CC1 CON(CCC(=O)NCC1(C)CCC(C)O1)C(=O)CN1CCOCC1=O c1(CC)nc(C)c(C(N2CCOCC2CC(=O)NCC2CC(CC)C2)=O)o1 c1(OC)nc(=NCCCN(C(=O)C2=NN(C)C(=O)CC2)CCO)nc(OC)[nH]1 c1(C(=O)NC2C(CC)N(C(c3nc(C)sc3C)=O)CC2)nccn2nccc12 C1(C(N2CCN(c3cc(C(C)C)ncn3)CC2C(C)C)=O)Cc2ccccc2O1 C(=O)(CC1CCCc2ccccc21)NCC1CN(C(c2c(C)nn(C)c2F)=O)C1 CC1=C(C(=O)NCCC2CN(C(c3cc(C)c(N)cn3)=O)CC2C)CCC1 C1(C(N2CC(C(C)(C)C)C2)=O)CCN(C(C2(C)CCC(=O)NC2)=O)CC1O C(=O)(C(C(C)C)C(C)C)NC1CN(C(c2cnc(OC)c(C)n2)=O)C(CO)C1 Cc1cc(NC(C2CC(O)CN2C(c2cccc(F)c2C)=O)=O)ccc1Br C1(C(N2CC(C(N)=O)(CNC(C(C)OCCC=C)=O)C2)=O)COCCOC1 C12(NC(c3ccc(C)nc3O)=O)CCCC1N(C(c1c(C)[nH]c(C)c1C)=O)CC2 C1(C(N2C(C(C)C)CCCC2)=O)CN(C(c2ccc(C(F)F)o2)=O)CC(C)(C)C1 N1(C(CC(=O)N(C)C)=O)CC(O)CCC1C(=O)NCCC1(C)CCOC1 C1(NC(CN(CCOC)C)=O)CC(C(=O)NCCCSC)C12CCC2 c1(C(=O)NC23CC(CNC(C(CSC)O)=O)(C2)OC3C)cccn2cc(C)nc12 c1(C(N2CCC(O)(C(CNC(CCCOC)=O)C)C2)=O)c(C)ccc(F)c1N c1(C(=O)NCC2(CF)CC2)ccc2c(c1)CCC2.CC1(C)C2CC1CCN2 C(C(C)(CC(C)C)NC(=O)CC1CC=CCC1)NC(CC1(OC)CC1)=O c1(CC(N2CC(C)C(NC(=O)C(F)(F)C3CC3)CC2)=O)cccc2ccsc12 C1(NC(Cn2nc(C)oc2=O)=O)CCN(C(=O)COc2ccccc2)C12CCC2 c1(NC(C2(NC(C(CCOC)OC)=O)CCCC2)=O)ccc(Cl)cc1C S(=O)(=O)(c1ccc(C(=O)OCc2ccc3c(c2)OCO3)cc1)N1CCC(C)(C)C1 c1(NC(C(C(=O)OCC)(F)F)=O)nc2cc(S(N)(=O)=O)ccc2o1 O=C1CC(NC(C2CC3CC2CC3NC(C2CN3CCC2CC3)=O)=O)CC(=O)N1 c1(OCCC(=O)NC2CN(C(C3CC4CCC3C4)=O)C2)cccc(-n2nccn2)c1 C1(C(=O)NCC2(OC)CN(C(c3csc(S)n3)=O)C2)CC2C=CC1CC2 Cc1cccc2[nH]cc(C(=O)NCCNC(=O)CCCCc3cccc(O)c3)c12 C1(CC)CC2CCC(C1)N2C(C1(C)CN(C(=O)C(F)OC(F)(F)F)C(C)(C)C1)=O N1(C(C=CC(CC)C)=O)CC2(CCC(CNC(c3noc4c3COCC4)=O)O2)C1 c1(C(N2C3COCC2C3)=O)c(NCc2ccc(Br)nc2Cl)nn2ccccc12 CC1(C)CCOC1CC(N1CCC(NC(c2cccnn2)=O)C1)=O c1(C(N2C(CNC(C(C)(C)N3CCCC3)=O)CC3CC32)=O)ccc(Cl)c(O)c1 c1(CC)[nH]nc(C(=O)N(C)CCN(C(c2ccnc(C)n2)=O)C(C)C)c1[N+](=O)[O-] C(C)(CO)(C(=O)N1CCC(CC(=O)NC(c2ccnn2C)C)CC1)OC C#Cc1cccc(C(=O)NCC2CCN2C(=O)COC(C)=O)c1C C1(C(=O)NCC(CO)NC(C(C)CC2CCC2)=O)CC(C2CC2)C1 C(=O)(N1CCC(C(N2CC(CO)C3(CC3)C2)=O)O1)c1cc(C)[nH]n1 c1(CC(N2CCC(O)(CNC(C(CC)SC)=O)CC2)=O)c[nH]c2ccc(F)cc12 C1(C(=O)NC2(C(=O)NC)CCC2)CN(C(=O)C#CC2CCOC2)CC1C1CC1 N1(C(c2cc(CC)ncc2)=O)CCC(C(=O)N(OC)C(C)CC)C(C)(C)C1 C1(CNC(c2cc(CC)c(C)cc2)=O)CC12CCN(C(=O)C(C)(F)F)CC2 c1(C(=O)NC2(C)CCCCC2C(N2CCCC2)=O)nnn2c1CCCC2 N1(C(C2(NC(CC(CC=C)(C)C)=O)CCSC2)=O)CCc2nnnn2CC1 c1(N(C(c2ccc(-n3c(C)ncc3)cc2)C)C)cc2n(n1)CCCN(C)C2=O C(=O)(C(COC(C)=O)C(F)(F)F)NC1(CO)CN(C(C2C(C(=O)OC)CC2)=O)C1 Cc1cc(=NCC2CN(Cc3ccn(C)n3)C2)[nH]c(N2CC(C)CC(C)C2)n1 CN1CCC(C(N2CC(O)CC2CC(=O)NC2(C)C(C)(C)C2(C)C)=O)CC1=O N1(C(N(C2CCCOC2)C)=O)CCCC(n2ccnn2)CC1 C1(C(C)NCCCOC(CC(C)C)C)CC(=O)N(c2ccccc2)C1 Cc1[nH]c(-c2ccccc2)cc1C(=O)NC(C)CN(C(=O)C=CC1CCC1)C C=Cc1cncc(C(=O)NC(C)CCCC(=O)NC(C)(C)C)c1 Cc1cc(Cl)ccc1C(=O)NC1CCC(CNC(c2cc(O)ccc2F)=O)C1 CC1CC(=O)NC1C(=O)Nc1cnn(CC(F)(F)F)c1C1CC1 c1(C(=O)NC(c2onc(-c3ccc(OC)cc3)n2)C(C)C)cc(C)ccc1SC c1(OCCOC)ccc(-c2nc(C(C#N)C(C)(C)C)n(C3CCOC3)n2)cc1 C=C1CCCN(C(=O)C(CCNC(=O)CCSCC)OC)C1 c1(NC(c2cccc(-c3n(C)ncn3)c2)=O)ncc(F)cc1C#N C1(CNC(c2nnnn2CCOCC)CCC)CC(C)(C)CC(C)(C)C1 C12(C(N3CC(NC(c4ccn(C)c4)=O)C4(C3)CC4)=O)C3C4C1C1C2C3C41C N1(C(C2C(OCC)C2C)=O)CC(CO)C2(C1)CN(C(c1cnc3n1CCC3)=O)C2 c1(COC)ccoc1C(N1CCC(n2cc(C(=O)NC3(SC)CCC3)nn2)C1)=O NC1CCCC2(CC(C(N3CCN(Cc4ccc(F)cc4)CC3)=O)C2)C1 c1(CNC(c2n(CC=C)nnn2)c2cccn2CC(C)C)ccc(OC)nc1 C=CCCC(C)(C)C(=O)NCC12CC1CN(C(=O)Cc1cc(C)[nH]n1)C2 C1(CCC(=O)NC2(CCOC)CC2)CCCN(C(=O)CCn2ccnn2)C1 C1(n2cc(-c3cc(OC)ns3)nn2)CCC(C)(C)N(C(C2(C(C)(F)F)CC2)=O)C1 Cc1cc(=NCCCCCF)[nH]c(NC2COC3(CCC3)C2)n1 N1(CC)CCCC1C(N1CC(COC)(NC(c2ccno2)=O)C1)=O C(=O)(CCCCCC#N)N1C(C(=O)NC)(CC)C=CC1.C1CS(=O)(=O)N1.NC c1(C(=O)NC(CCCNC(C=CCCC)=O)C)cc(C(N)=O)ccc1OC CC1CN(C(=O)CCC(C)(F)F)CC2(CCN(Cc3ccc(Br)o3)CC2)O1 CC#CC1CCN(C(C23CC(CO)(CN2C(=O)CC2OCCCO2)C3)=O)C1 CCCCC(CC)(c1nnnn1CCCOCC1CC1)NC(CC)C(C)(F)F C1(NC(c2ccccc2F)=O)CN(C(C2CC3(CCOC3)C2)=O)CC12CC2 c1(OC)cccc(C(=O)NC(CNC(C2(C3CCCO3)CCCC2)=O)C2CC2)c1 N1(C(Cn2cccc(N)c2=O)=O)CCC2CCN(C(c3cscc3Cl)=O)C2C1 C1(N(S(=O)(=O)C2CCN(C(=O)OC(C)(C)C)C2)C(C)C)CCCCN(C)C1=O C12(C(=O)NCc3scc(C(C)=O)c3)CC1CN(C(=O)C(C(C)C)N(C)C)C2 C12(C(=O)NC(C#C)(C)C)CC(CO)(CN1C(c1cc(OC)n[nH]1)=O)C2 Nc1nccnc1C(=O)NCC1(C(=O)NCCCc2ccccn2)CC1 CC1C(=O)N(CC(=O)NCC2CCC(C)CN2C(=O)CCCCCF)C(=O)C1C c1(N2CCOCC(NC(C3N(C)C(=O)NC3)=O)C2)nc2c(cc1C#N)CCCC2 c1(C(C)C)ccc(C(N2CC(NC(=O)Cc3cscn3)C3CC3C2)=O)c(O)n1 N1(C(C(CC)C(C)C)=O)C2CCC1CC(N(C(=O)C1=CCCS1)C)C2 C(=O)(C(F)CCC(C)(C)C)NCC(C)N(C(c1cc(SC)oc1)=O)C N1(C(CC2(OC)CCCC2)=O)CCN(C(C2CN(C)C2)=O)C(CO)C1 CC1(C)C(CC(=O)NCC2(NC(c3cncc(C(F)F)c3)=O)CCCC2)CC1O c1(C(=O)NCC(C)N(C(CC(=O)NCC#C)=O)CC)nc(C)n(C)n1 c1(C(=O)NCC(CNC(c2cn3c(n2)CCC3)=O)F)ccc(F)cc1F C#CCC(C)(CC)C(=O)N1CCC(CN(C)C(c2cc(C)cs2)=O)C1 CCCC(C)CC(=O)NCC(C)(C)CNC(C1(CSC)CCOCC1)=O C(CCC1CC1)(C(=O)NCCc1cnoc1)NC(COCC(=O)NC)=O c1(C(N(C2CCCN(C(CC(C(C)C)O)=O)C2)CCO)=O)nnn2c1CSCC2 C(C(C)(CNC(=O)CN1CCN(C(C2(SC)CCOCC2)=O)CC1)CO)OC c1(NC(CCC2N(C(c3nn(CC)c(C)c3)=O)CCC2)=O)cc(C)cc(C)c1O N1(C(C2(N(C)C)CC2)=O)CC2C(CNC(=O)CC3C=CS(=O)(=O)C3)C2C1 C1(O)(CNC(CCC(CO)NC(Cc2cc(C)sc2)=O)=O)CCN(CC(C)C)C1 c1(SC)cccc(CC(N2CCCC2C2(NC(=O)CC(CCO)CF)CC2)=O)c1 N1(c2nnc(CCSC)s2)CCCC(C(=O)NCCCCn2ccnc2)CC1 Clc1ccc(Sc2csc(=NCc3cnoc3)[nH]2)c2ccccc12 C1(COC)(CNC(=O)C(C(C)C)SC)CCN(C(C2(C)CC3CC3C2)=O)CC1 c1(C(=O)NC)ncccc1NC(=O)CCC1CCCN1C(=O)C(O)CCSC c1(NC(C(CC)NC2CC(OCC)C2n2cccn2)=O)cnc(C#N)c(Cl)c1 C1(NC(c2ccc(C)c(F)c2)c2n(CCCSC)nnn2)CC12CCCCCC2 CCC(C)(CC)C(=O)N1CC2CC2(NC(c2cnn(C)c2OC)=O)C1 c1(OC)c(C(=O)NC2CCCC2CNC(=O)C=Cc2cocn2)cc(Cl)cc1Cl c1(OC)nc(C(N)C(=O)N(C)C)cs1.C12CC(C1)C(=O)N2 N1(C(c2cc(OC)n[nH]2)=O)CCC(CNC(=O)C(C)CN2CCCCC2)CC1 c1(C(=O)NC(CC=C)CNC(=O)CCC2CCC(=O)NC2)cc(C)nc(C)n1 CCCCCCC(C)C(=O)NC(Cn1ccnn1)C(=O)NC(c1c[nH]ccc1=O)C N1(C(C(=O)NCC2CCC(OC)(OC)C2)=O)CCc2cnc(C)nc2C1 c1(C(C(=O)NC(C)C(F)F)NC(CC=C)=O)cnn(C)c1O c1(OC)cc(CC2CCN(c3ccccc3OC(F)(F)F)C2=O)ccc1C CCCC(C(=O)N(C1CCN(C(c2c(Br)cnn2C)=O)CC1)CC)OCC N1(C(c2cn(CC)nn2)=O)C(C(=O)N(C)CC2CCC2)C2CC(O)C1C2 c1(C(N2CC=C(CCNC(C=NOC)=O)CC2)=O)ccnc2[nH]c(O)nc12 c1(CC)ccccc1C(=O)NCCOCCN(C)C(C1(C(C)C)CC1)=O C(=O)(C(CCC(N)=O)N(C)C)NC1CCCCN(C(c2ccc(C)cn2)=O)C1 C1(CNC(C(N2CC(C)OC(c3ccsc3)C2)=O)=O)CC1C1CCCCC1 N1(C(C2(C#C)CN(C(c3cc(CC)ccn3)=O)C2)=O)CCCC(O)C1C c1(N2CC(C(C)NC(c3scc(C)c3)=O)OCC2)ncc2ccsc2n1 C=CCCC(C)(C)C(=O)NC1CCCN(C(c2cccc3c[nH]nc23)=O)CC1 CC1CCOC(C(=O)Nc2cccc(NC(=O)Cc3nc[nH]n3)c2)C1 c1(CC)nn[nH]c1C(=O)N(CCC(=O)NCC1CSC1)CCCO c1(C(=O)NCCCOC(=N)O)ccc2c(n1)CN(C(=O)CCOC1CC1)CC2 C(C(=O)NOCCc1ccccc1)(C(C)(C)C)NC(CC1C(C)(C)CCCC1)=O c1(C(N2CCC(Oc3ccccc3C)C2)C(=O)NCC=C)ccc(C2CC2)cc1 C1(C(N2CC(O)(C(C)NC(C3C=CCC3)=O)C2)=O)CC(C2CCOCC2)=NO1 C1(NC(C(C)CC2CC2)=O)CC=C(C(=O)N2CCCCCCC2)C1 C1(CC(=O)NCC(C=C)O)CCN(C(=O)CC2OCCC2(C)C)C1(C)C CCC(C#N)(CC)C(=O)N(C1CCCC1)CC(C(=O)CCN1CCNC(=O)C1)=O.N Cc1cc(C(=O)NC2CC(CNC(=O)CN3CCC(F)CC3)C2)nc(C)c1 c1(NC(c2ccn(CC(C)C)n2)=O)cccc(CNC(c2ccc(O)cc2)=O)c1 c1(C(N2CCC(CN(C(CC3(C=C)CC3)=O)C)C2)=O)c(C)oc(C)c1Br C1(CC(=O)OCC)CCCN1C(=O)CC1CCN(C(=O)Cc2cncnc2)C1 N=c1ccc(C=CC(=O)NCC2CN(C(=O)Cc3c(Cl)cnn3C)CCO2)c[nH]1 C1(C(=O)NC(CC)(CC)CC)CN(C(=O)CC2CCC3CC23)C(C)(C)C1 c1(C(NNC(c2ccc(OCC)c(OCC)c2)=O)=O)cccc2c1NC(=O)CC2 C1(OC)CN(C(=O)Cc2cc[nH]c2)CCC1NC(=O)C1=CCN(C)C1 C1(N(C(=O)COCC(C)(C)C)CCC)CCN(C(=O)Cc2ccn(C)n2)C1 CC1=C(C(=O)N(C2CCC(NC(=O)CC3(C)CCC3)C2)C)Cc2ccccc2O1 C1(COC)(NC(=O)C(C)Sc2ccncc2)CCC(F)(F)CC1 C1(C(N2C(C)(CNC(C3(SC)CC3)=O)CCC2)=O)CS(=O)(=O)CC12CCC2 C1(C(=O)NCC(C)OCC#C)CCN(C(C2COCCN2C)=O)CC1C N1(C(C(C)NC=O)=O)CCCC2C1CCCN2C(=O)C(=O)N=S(C)(C)=O N1(C(c2cc(CNC(c3c(C)c(F)cnc3)=O)no2)=O)CCOC2CCCCC12 CCC(CN(C(=O)CN(C)C(C)C)C)OC.C12(CCC1)CC(=O)N2 C1(C(C(=O)N(C)Cn2cc(C)nn2)OC(COCC)=O)CCC(F)(F)CC1 C#Cc1ccccc1CC(N1CCCC(O)(CCNC(=O)C(CC)OCC)C1)=O CCCC(CCCNC(C1CC2C=CC1CC2)=O)NC(c1nnn(C)c1C)=O CN1CCN(C)CC(C(=O)NC(CNC(C2CC23CC3)=O)CO)C1 CC1OC2CCC1(C(=O)NCCC1CCN(C(c3cncc(Cl)c3)=O)C1)C2 N1(C(C(CC=C)C)=O)CCN(C(C2CC(F)(CO)C2)=O)C(c2cn[nH]c2)C1 c1(C(=O)NC(COCC)C(=O)NCCS(=O)(=O)NC)coc2ccccc12 CCC(C(=O)NC1(c2ccccc2)CN(C(=O)CCCCCO)C1)C(C)C CC1(C)CN(C(C2CCC(C(N)=O)O2)=O)CC1NC(=O)CC12COC(CF)(C1)C2 c1(C(=O)NCCCCN(C(CC(C)NC(N)=O)=O)C)cc2ccsc2c(O)n1 N1(C(C(C)OC(C)=O)=O)CCCC(C)(C)C1C(=O)N(C)Cc1ccon1 C1(CCNCC(C)Oc2ccc(Cl)c(Cl)c2)CC2(CCC(F)(F)CC2)C1 N1(C(C(CNC(C)=O)C)=O)CCC2(CC1)CCN2C(c1ncccc1Br)=O CC1(C)CCC(CNC(c2cncs2)=O)N(C(=O)Cn2cc(F)ccc2=O)C1 N1(C(CCCC2C(C)C2)=O)CCOCC1CCN(C)C Cc1nc(C)c(C(=O)NC(C(N2CC(C)(CF)C2)=O)c2ccoc2)s1 c1(N2CCC(N(CCC)C(c3cccc(F)c3F)=O)C2)cc(C)nc(C2CC2)n1 C12COC3(CCC3)CN1C2.n1(CC)cc(Br)cc1C(=O)OC(C)(C)C C1(C(=O)NC(CC)CNC(c2sccc2Cl)=O)CCCC(=O)O1 N1(Cc2ccc(N(C)C)nc2)CCC(F)(F)C(NC(c2csc(Cl)n2)=O)C1 C1(NC(C(CCC#C)O)=O)CCN(C(=O)CN(C)C(=O)C2CC2)CCC1(F)F C=CC(C)(CCOC)C(=O)NC1CC2CCC1CN2C(=O)C(O)CCC c1(OC)cc(C(=O)NCC2CCC2NC(=O)C(C)(C)C#N)ccc1OCC(N)=O N1(C(C2(c3cccs3)C(C)C2)=O)CCN(C(=O)CC2(N3CCCC3)CCC2)CC1 CCCC(C(=O)NCC1(C)CCN(C(c2cnc(C)[nH]2)=O)C1)c1cccc(Cl)c1 C(=O)(C1=NOC2COCC12)NC1C(NC(c2c(C)nccn2)=O)CCC1 C1(NC(c2cnc(OC)c(Cl)c2)=O)CCCC12CN(C(c1ncc(F)cn1)=O)C2 c1(C(=O)OCC)ccc(C(=O)NCCCC(C)NC(C2CCOCC2)=O)cc1 N#Cc1ccc(C2(NCCCN3CC4CC3(c3ccccn3)C4)CCC2)cc1 C1(C(=O)NCC2C(C)OCC2)CC12CCN(C(c1cccn1C)=O)C2 N1(C(CN2CCCC(CC)C2)=O)CCC(C(C(C)C)NC(C2CCC2)=O)CC1 C1(CNC(CCC(=C)C)=O)N(C(=O)CSc2nc[nH]n2)CCC1(C)C C(C(F)(F)C(=O)NCC(CNC(c1cnc(O)n1C)=O)OC)OC C(=O)(C(C(=O)OCC)C(C)C)N1CC(O)(C(C)NC(C(CCC)O)=O)C1 Cc1cc2sc(C(N3CCCC3CCNC(c3cncs3)=O)=O)cc2s1 c1(NCCn2cncn2)nccc(=NCCCC2CCC3CC23)[nH]1 c1(C(C(=O)NC)N(C)CC2CCCC2(C)C)ccc(Br)nc1 c1(C(=O)OC)cccn(CC(=O)NC2(CNC(C3CN(C)C(=O)N3)=O)CC2)c1=O N1(C(C2N(C(CNC(=O)C3CC3)=O)CC(O)C2)=O)CC2CC=CCC2C1 CC(C)(O)C(F)C(=O)N1CCC(CNC(=O)CCC2OCCO2)C1 c1(NC(=O)NC2CCN(CCS(C)=O)CC2)cc(N)ccc1O c1(C(N2CCC(CNC(CCC(=C)Cl)=O)C2)=O)ccn2cc(C)nc2c1 N1(C(C(C)(c2ccccc2)NC(=O)CSC)=O)CCN(C(COC)C(F)(F)F)CC1 C(=O)(C(C)(C)CC(F)(F)F)NCC1CN(C(c2c(C)ccnn2)=O)C(C)C1 C(c1cnc(O)nc1O)=CC(N1CCC(N(C(=O)C(O)C(F)(F)F)C)C1)=O C(=O)(C(C)(F)C(=O)N1CCCCC(CNC(C2CSCN2C(C)=O)=O)C1)OCC C(CC(C)(C)C)(C(=O)NCC1(CCNC(C2CC3(CC3)C2)=O)CC1)OC Cc1ccc(OCCCN)cc1.N12CCC(C1)N(C)C(=O)C2.c1cc(C)sn1 C(=O)(C(C(C)C)c1ccc(F)cc1)N1CCC(N(C(C(C2CC2)OC)=O)CC)C1 C(=O)(CS(=O)CCC(F)(F)F)NCCCN(C(CCC=C)=O)C1CCCC1 C1(CNC(C2(COCC)CC2)=O)(CO)CCN(C(C2CC2F)=O)CC1 C12(NC(C(C)Cc3ccccn3)=O)CCOCC1CN(C(C1(O)CCCC1)=O)C2 C1(OC)CCN(C(=NCCC(C)(C)F)NCc2ccco2)CC1C Cc1cc(Br)cc2cc(CNC(=O)NC3CC34CC(F)(F)C4)oc12 C1(O)(C(CNC(C2(OC)CCC2)=O)C)CCN(C(=O)Cc2nc(C)cs2)C1 c1(C(=O)NCC(C)(CC(C)C)NC(Cc2c(C)ccs2)=O)c(C)ccc(C)c1N C(CCNC(=O)C(=Cc1ccco1)C)(C(C)C)N(C(Cn1ncc(CC)c1)=O)CC N1(C(Cc2cc(C)no2)=O)CCC2(CCN(C(c3cc(C(F)(F)F)n[nH]3)=O)C2)C1 C(=O)(C(CNC(=O)NC(C)(C)CN(C)C)c1ccccc1)OC C(C(=O)N1CCC(CN(C(c2ccc(=N)[nH]c2)(C)C)C)CC1)(C(C)C)SCC C1(C)(C(=O)NC(C(C)NC(=O)CCc2ncoc2C2CCCC2)C)CCCCC1 c1(C(=O)NCCN(C(=O)CSC)CCC)cc(Br)n2ccccc12 c1(CNC(c2ccc(-c3ccc(-c4cnco4)cc3)cc2)=O)ccc(F)nc1F c1(OC)nc(C)ccc1CN1CCCC(NC(=O)CCC(=O)SC)CC1 c1(CC(=O)NC(CNC(C(CC)n2cncn2)=O)COC)ccc(C)cn1 Cc1c(C(N2CC3(CC(NC(C4CC4Cl)=O)C3)C2)=O)oc2cc(Cl)ccc12 C1(NC(C(CC=C)C)=O)CC2CCC(C1)N2C(c1cscc1-c1ccccc1)=O c1(OCC)ccc(OCC(=O)N(C(C)CNC(=O)C(F)n2ccnc2)C)cc1 c1(C2C(N(CC(C)C)CCN)CCC2)cccc(Cl)c1 O=C(CCCCC(F)F)NC1CC2CCC1CN2C(c1ccc(CCO)cc1)=O c1(CC(=O)NCC2CN(C(CCC=C=C)=O)CC2O)cc(C)c(Cl)c(C)c1 c1(OC)ccc(Cl)c(Cc2noc(-c3ccsc3OC)n2)c1 N1(C(Cc2cnc(C)s2)=O)CCC(C2CC(NC(c3nc(Cl)cs3)=O)C2)C1 N1(C(CCN2CCN(CC)CC2)=O)CCCC1C1CCCN1C(C1CC=CC1)=O c1(CCC(=O)NCC2CN(C(Cc3cnc(C)o3)=O)C(C)C2)cccc(C#N)c1 N1(C(c2nc[nH]c2C(F)(F)F)=O)CCC2CCC(C1)N2C(C1(CO)CC1(F)F)=O c1(SC)cccc(C(=O)NC2CCC2NC(=O)CCCN(C)C(C)=O)c1 C(CN=c1[nH]c2c(c(=NC(C)c3c(Cl)cccc3Cl)[nH]1)COC2)C1(C)CC1CO C1(NC(C(COC)NC(C)=O)=O)CCC(NC(c2nnsc2C)=O)CC1 Cc1cc(CN2CCCCC2CNC(=O)CCc2nccs2)ccc1F CC(CC(=O)NC1CCN(C(c2ccc3c(c2)CCC3)=O)C1(C)C)C(F)(F)F C(CC(F)(F)C(=O)NCC1CCC2(CCC2)O1)n1cc(CCNC(C)=O)nn1 c1(C(=O)NC2CCN(C(c3ccco3)=O)CC2)cc2ccc(Cl)nc2s1 c1(C(c2nnnn2C2CCCC2)NC(c2nc[nH]n2)C)nn(C)c2c1CCCC2 c1(C(=O)NC2CCC(N(C(C3C(C)OCCC3)=O)C)CC2)cc2scc(Cl)c2[nH]1 C(=O)(C(C)C(C)(C)C)NCCC(C)(C)NC(C(c1cccnc1)C)=O n1(CC(=O)NC(C)C(C)NC(=O)Cc2cncn2C)nc(C(F)F)cc1C1CC1 c1(C(=O)NC2CCC(N(C(C=C(C)C(C)C)=O)C)C2)cc(N)c2ccccc2n1 N1(C(COCCC#C)=O)CCN(C(=O)CSc2ccccc2)C2CC12 C1(O)(C(=O)NC(C)CCCNC(=O)CCC2CC2(F)F)CCCCC1 Cc1cc(Br)ccc1S(=O)(=O)N(C1CC2CNC1C2)C(=O)C1CC1 c1(C(N(C2CCN(C(CC=CC=C)=O)C2)C)=O)ccn(CC(F)(F)F)c(=O)c1 c1(-c2cn(C)nc2)ccc(C(=O)OC2CC3CCC2C3)cc1 c1(C(C)Nc2ncnc(NCc3c(C)nco3)c2C)ccc2c(c1)CCCO2 O=C(C1=CC2CCCC12)NC1CCCCC1NC(c1ccc(Cl)s1)=O C1(N(C(=O)CC2SC(=N)NC2=O)C)CCCN(C(C2OCCO2)=O)CC1 N1(C(CC(CCC)C)=O)CC(C2CN(C(c3ccccc3SC(F)F)=O)C2)C1 c1(CCC(=O)NCC(CC)NC(c2ccn(C)c(=O)c2)=O)c(O)nc(=N)[nH]c1C c1(CNC(=O)NC2CCN(C(c3ccsc3)=O)CC2)ccnc(Cl)c1 CCC(CNC(C1CC(NC(=O)COCCSC)C1)=O)CCO C1(NC(CCOC(C)C)=O)COC2CN(C(c3nc4ccccc4[nH]3)=O)CC12 N1(C(CCSCC(=O)OC)=O)CCC(NC(c2[nH]nnc2C)=O)C12CC2 c1(C(N2C(C(=O)NC(CC)C(C)O)CC(C)C2)=O)c(C)cc(OC)cc1C c1(C(=O)NC(C2N(C(CC(=C)C)=O)CCC2)(C)C)cc(Br)ccc1OC c1(C(N2CC(C)C(NC(C3CC(=C(F)F)C3)=O)C2)=O)cccc2nc[nH]c12 N1(c2[nH]c(=NCCC(=O)NCC)nc(COC)n2)CCS(=O)(=O)C2(CCCCC2)C1 c1(COC)ccccc1NC(=O)CC1CCN1C(=O)Cc1ccnn1C c1(OC)cc(C#N)cc(Cl)c1OC(=O)C(O)CC(=O)O N1(C(C2N(C(C)C)CCC2)=O)CCCC(C(=O)NCc2nc[nH]n2)CC1 C1(CC)CCCN(C(=O)CC2CCCCO2)C1CNC(=O)CCc1cn[nH]c1 Cc1cccn(CC(=O)NC(C2(CNC(C3CCOC3(C)C)=O)CC2)C)c1=O CC(C)C(O)CC(=O)N1CC2(CCN2C(=O)CCC(C)(F)F)C1 c1(C(N2CCC(C)(NC(c3n(CC)ncc3Cl)=O)C2)=O)cc(S(N)(=O)=O)oc1C c1(NC(CN2CCCC(NCc3n(C)ccn3)C2)=O)c(F)ccc(N)c1F c1(NCCC2CCCN(C(CC(COC)(C)O)=O)C2)nc[nH]c2ncnc1-2 C1(CNC(C(c2n(C)ncc2)(C)C)=O)CC(C)(C)CN1C(=O)CC1COC(=O)C1 N1(C(=O)CC2CCCCC2I)CC(CO)Cn2nccc21 c1(CC(=O)NCC2C(C)(C)CN(C(C3CC34CC4)=O)C2)cccc2ccoc12 C1(C)(CC)CC(NC(=O)CNC=O)CN1C(=O)CC1CNC(=O)O1 C(=O)(C1=CCCCO1)N1CC(CCNC(c2cc3[nH]ccc3s2)=O)C1 CCC(C(=O)N1CC(NC(=O)CN(c2cc(C)no2)C)C1)N(C)CC.OCC C1(NC(c2cnn(C)c2Br)=O)CC2(C1)CC(N)C2 CC(C)CCCC(C)C(=O)N1CCC(O)CC1C(=O)N(C1CCN(C(C)C)C1)C c1(N(C(C(=O)NC(Cc2cc(C)[nH]n2)(C)C)=O)CC(F)F)cnc(Cl)c(N)c1 c1(CC)nc(N(C)Cc2ccc(N3CC(SC)C3)s2)cc(C#N)n1 C#CCCCCCCC(=O)N1CCC(F)CC1C(=O)NC(c1cccs1)C C(CCCC(CO)NC(C1(OC(C)C)CCC1)=O)NC(c1onc(CC)c1C)=O N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(NC(c2cnn(C)n2)=O)C(C)(C)C1 c1(C(N2C(CCNC(C3(CC)CC3)=O)CSCC2)=O)cc(C)nc(N(C)C)n1 c1(N2CC(NC(COc3ccc(C)cc3)=O)C(C)CC2)ncc(C#N)cc1Cl Cc1c(NCC2CN(CC(C)C)CCO2)ncnc1N1CCOC(CCO)C1 C(=O)(C(F)C(C)(C)O)NCC(CCOC)NC(=O)C(C)(C)C(C)C CC1(C)CN(C(c2cc(F)c(Br)cc2F)C(=O)NC2CCCCC2)CC(CO)O1 CN=S(C)(=O)c1cccc(C(=O)NC2CCCN(C(C3CSC3)=O)CC2)c1 C1(C)(CC(N2CCC(C(C)NC(C(CCOC)C)=O)CC2)=O)CCCCCC1 c1(C(=O)NC(CCNC(CCN(CCC)C)=O)C(C)C)cc2ccnc(Cl)c2[nH]1 C12(C(N3C4C(N(C(C(C)OCCN(C)C)=O)C)CC(C4)C3)=O)CC(=O)N1C2(C)C C1(NC(=O)OC(C)(C)C)CC(NCCn2ccnn2)C12CCC2 n1(CC)ccc(C(N2CCCC2CCC(=O)NC2CC3CC3C2)=O)c1C N1(C(C(C)CC2CC2)=O)CC(F)CC1C(=O)NCCS(C)(=N)=O c1(OC)c(Br)ccc(C(c2nnnn2C2(C)CC2)NCC2(CC(C)C)CC2)c1F N(C1CCc2c(F)ccc(F)c21)C(=O)NCc1c(C(C)(F)F)cccc1 N1(C(c2c(C)csc2)=O)CC2(C1)OC1(C)CC2(NC(=O)C(C(C)C)NC=O)C1 C1(OC)CN(C(=O)CC(C)(C)C)C(C)(CNC(=O)Cc2c[nH]nc2C)C1 C1(C(=O)NCC(CNC(C2C(C)(C(=O)OCC)C2)=O)O)CNC(=O)N1 N1(C(C(C2CCCCC2)N)=O)CCC(C2CCCCC2)C1 C1(NC(=O)C=C2CCOCC2)CCSC12CN(C(c1cccc(C(F)F)c1)=O)C2 N1(C(c2c(Br)ccc(C)c2)=O)CC(S(=O)(=O)CC(F)(F)F)C1 N1(C(=O)Cn2ncccc2=O)CC2CC(C1)N2C(=O)CC1=CCCC1 C1(C(N)=O)C2CCN(C(=O)CNC(c3cc(C(=O)NC4CC4C)ccn3)=O)CC12 c1(OC)ccc2c(c1)OCC(C(N1CCCC(c3cn(CC(N)=O)nn3)C1)=O)C2 c1(C(=O)NC(CCNC(CSC)=O)(C)C)ccnc(N2CCCC(C)C2)c1 C=CC1(C(=O)NC2CC(C(C)(C)C)C2)CCN(C(C2C(C#N)C2(C)C)=O)CC1 C1(NC(C2C(CC)CCN2C(=O)Cc2ccc(F)nc2)=O)CN(C)CC12CC2 c1(NC(C2CC3(CC3)CN2C(=O)CN2CCCC2)=O)cc(Cl)cc2[nH]ccc12 CC1CCN(C(c2cccc3occc23)=O)CCN1C(c1ccc(F)s1)=O N1(C(CNC(=O)OC)=O)CCC(CC(C)NC(C2(CO)COC2)=O)CC1 N1(C(CCCCCCCC)=O)CCC2OCCN(C(C3CCCCN3C)=O)C2C1 C1(C(N2CC(O)(CNC(c3n(C)nnc3)=O)C2)=O)CCc2n[nH]cc2C1 Cc1cc(-n2ccnc2)ccc1C(=O)N(C1CN(C(c2cnns2)=O)CC1O)C C1(NC(C2CCN(C(=O)C3CC(c4ccccc4)C3)O2)=O)CCc2n[nH]cc2C1 Cc1ccc(C)c(CCCC(=O)NCCC(O)CNC(C2(C)CC2(F)F)=O)c1 c1(C2(C(=O)NC3CCC(NC(C4C(OC)C4)=O)CC3)CC2)cc(F)cc(F)c1 C(=O)(CCC(C)(C)NC(c1ncncc1Cl)=O)NCCC(C)C N#Cc1ccc(NC(C2CN(C(c3cccc(Cl)c3)=O)CCC2O)=O)c(O)c1 C1(CNC(C(C(COC)C)C)=O)CN(C(=O)CCCCC#N)CCC12CCC2 n1(CC(=O)NC(CC=C)CNC(=O)C=Cc2cn[nH]c2)cnc2c1CCCC2 N1(Cc2c(C)nc(CC)o2)CCC2C(CCCN2C(=O)CCc2cnn[nH]2)C1 C1(NC(CCCOCC)=O)COCCC1C(=O)NC1C=CCCC1 C(N=c1cc(Cl)c(O)n[nH]1)C1(CCNC(C23C(C)OC(CO)(C2)C3)=O)CC1 N1(CCSC)C(=O)CN(CCC(C)(c2nnnn2C)SC)C1=O C=CC1(NC(=O)CCN(C(=O)C(=O)NC(C)C)C(C)C)CCOCC1 c1(C(C)CC(=O)NCC(C)N(C)C(C2CCSCC2)=O)ccccc1F c1(C(N2C(CN(C(=O)CCc3cc(Cl)no3)C)CCC2)=O)coc2c1COC2 c1(NC(CCN2CCN(C(C)C)CC2)=O)nccn2nnnc12 C1(NC(CC(COC)C)=O)(CNC(=O)C(C)OC)CC2CCC1CC2 CC1(C)CN(C(C23CCC(CC2)CC3)=O)CC1CNC(c1n[nH]cc1Cl)=O CC(=O)n1cc(CSc2ccc(CC(=O)O)c(O)c2)c2ncccc12 CCC(C)CC(C(=O)NC1CC2(CCOC2)C1)NC(=O)CCCC(C)C N1(C(CC(C)O)=O)CCN(C(c2cc(Br)ccn2)=O)C(c2cnn(C)c2)C1 Clc1ccnc(N2CCCC(OC3CC3)C2)c1I c1(C(=O)NC2CN(C(CCc3nnc(C)n3C)=O)C(C)C2)cccc2nc[nH]c12 c1(C(=O)NCc2c(CNC(C=CSC)=O)cncc2)ccc(C(C)=O)c(F)c1 N1(CCCC(=O)NCC23CC2CN(C(=O)Cc2cncnc2)C3)C(=O)CNC1=O N1(C(C2C(C)C2C)=O)CC2CCC1CN2C(c1ccc(Cl)o1)=O C1(CC(=O)NC2CCN(C(c3ccc(F)o3)=O)CC2F)CCCC2(CCC2)O1 c1(C(N2CC(NC(=O)C(F)(F)CC3CC3)C(O)C2)=O)cc(F)ccc1Br c1(C(=O)NC(C2CC3(CCC3)C2)C)ccc2c(n1)CN(C(C1CC(F)(F)C1)=O)CC2 C1(O)(C(C)NC(COCCCCOCC#C)=O)CN(C(=O)C(F)CC2CCC2)C1 C#CC1CCCN1C(C1COCC1NC(c1ccc(Cl)cn1)=O)=O c1(C(=O)NC(C2(O)CN(C(COCC#C)=O)C2)C)cc(F)cc(Br)c1 c1(OC(C)C(=O)NC2CC(OCC(F)(F)F)C2)cc(C(F)(F)F)ccn1 c1(C(=O)NC2(C)CCCN(C(CCC(C)OC)=O)C2)cc(C#N)c(C)cn1 CCC(C)C(C)C(=O)N(C1(C(N2CC3C(C2)C3(C)C)=O)CC1)C C1(CC)CNC(=O)CN1C(=O)CCC1CCCCN1C(c1n[nH]cc1C)=O c1(NC(C2CCCCCC2)COC)cnc(N2CCOCC2)nc1 Cc1c(C(=O)NCC2CCN(CC3CCOCC3)C2)oc2ccc(F)cc12 N1(C(C(C)OCCC=C)=O)CC(NC(C2(C)CCSCC2)=O)Cc2ccccc21 N1(C(CNC(C)=O)=O)C2CCC1CC(CC(C)NC(=O)C(C)(C)C(C)O)C2 c1(C(=O)NCC2C(NC(c3cc(Br)co3)=O)CC2)cccc2[nH]ncc12 N1(C(C=C(CCC)C)=O)CCCC1CNC(=O)CSSC C1(NC(C(C(C)C)SCC)=O)CN(C(=O)CCOC)C(CC)(CC)C1 c1(C(=O)NC2C(C(N(C(C)C(=O)NC)CC)=O)CCOC2)cccc(C)c1O c1(C(=O)NC(C)CC(C)NC(C2CCS2(=O)=O)=O)ccc(-n2cccn2)c(F)c1 N1(C(C2(C(=O)O)CCOC2)=O)CCC(C2(O)CCOCC2)CC1 c1(NC(C(=O)NCCOc2ccccn2)=O)cccc(OC2CCOC2)c1 N1(C(C(CCC)N(C)C)=O)CC(NC(C2CCC3(CCC3)CC2)=O)C2CCCC12 c1(-c2nnc(CCC(=O)N(C)Cc3ccnc(Br)c3)o2)ccc([N+](=O)[O-])cc1 C(=O)(C(C#N)C(C)(C)C)NC(C)CCNC(=O)CCS(C)(=O)=O C1(CNC(CC(C)F)=O)(CO)CCN(C(=O)CCC2CCCN2C)CC1 N1(C(=O)Cn2ccc(C(F)F)n2)CCN(C(C2CCCC(F)C2)=O)C(CCO)C1 c1(C(=O)NCC2N(C(C(C=C)OC)=O)CCC2)ncc(C#N)cc1C Cn1ncc(C(N2CCCCC2CCNC(c2ccc(Cl)nc2)=O)=O)c1C1CC1 N1(C(c2ccc(OC)cc2OC)=O)CCC2CN(C(C3CC3CF)=O)C2C1 CC1(C)CN(C(=O)CN2C(=O)CCC2=O)CCN(C(=O)C#CC2CCCCO2)C1 Cc1nc(C)c(C(=O)NC2CCCN(C(=O)CSC3CCOC3=O)C2)[nH]1 CC(C)C(F)(CNC(c1cc(F)cc(F)c1)=O)C(=O)NCc1ccc(F)c(F)c1 c1(NC(C(=C)CN)=O)cccc(CC(=O)NCC(C)C)c1 CC(C)(C)CCCCC(=O)NC1CCC(NC(=O)CC2CC(=O)C2)CC1 c1(N(C)CC2CCC2)ccnc(N2CCOC(CC(N)=O)C2)n1 Cc1nc2c(s1)CC(C(N1CC(CNC(=O)C(CC#N)c3ccccc3)C1)=O)CC2 C(c1cn(C)c(=O)n(C)c1=O)=CC(=O)NCC(CC=C)NC(c1csnn1)=O c1(C(N(C2CCCN(C(=O)CCCCN3CCCC3)C2)C)=O)ccc(CO)nc1 c1(C(=O)NCC(CC)NC(C2CCCN2C(C)C)=O)cccc2occc12 CC(C)C(C(=O)NCC1CCN1C(C1(O)CCOC1)=O)NC(c1ccccc1)=O c1(NC(C2C(C(=O)NCC)C2)=O)ccc(OC)nc1Br C=CCC(C(=O)NCC=CC(=O)NC(C)CO)NC(C)=O c1(CNC(C2(NC(c3c(CC)c[nH]c3)=O)CCCCC2)=O)ncc(F)cc1F CCC(CC)(C(=O)N1CCC(C)(C)C(NC(C2(OC)CCCOC2)=O)C1)C(C)C Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC1CCC(C)(NC(C2CCCC2)=O)CC1 C(=O)(CC1NC(=O)c2ccccc21)NC1CN(C(COCC)=O)CC1C C=CC(C)(C)C(=O)NC1CC1CNC(c1cc(Br)c[nH]1)=O N1(C(CCCCC(=O)NC)=O)CCC(NC(=O)C=Cc2cnc[nH]2)C2(CCC2)C1 C(CC(C)(C)C(=O)N1CCC1C1CCC1)NC(C(SC)SC)=O Cn1cnn(CCC(=O)NCC2COCCN2C(=O)C2=NOCC2)c1=O Cc1cccc2c1CN(C(=O)C(c1ccoc1)NC(=O)CC#N)C2 c1(CC)ccc(C(=O)NC23COC(C2)C(NC(=O)C(C(C)C)SC)C3)cc1Cl c1(-n2cc(CN(C)C(c3cc(Cl)sc3Cl)=O)nn2)ncc(Cl)cn1 C1(N(C)C(C2CCC3CC3CC2)=O)CCCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 CCC(CC(=O)N(CC(CC(C)C)C(C(=O)N=c1ccn(CC)[nH]1)=O)C)C(C)(C)C c1(C(N(CCC(=O)NCC(=O)OCC=C)CC=C)=O)sccc1C#N C1(OC)CC(NC(c2cccc(F)c2)=O)CN(C(=O)CN2CCCC2)C1 Cc1noc(C)c1CC(=O)NC1CCC1NC(=O)CC(C)(F)F C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(c2cc(Br)n[nH]2)=O)CC2(CCC2)C1 c1(SCC)ccccc1NC(=O)CCNC(C1CN(Cc2cccnc2Cl)C1)=O C1(NC(COCC)=O)CC12CCN(C(=O)CCC1CC(C)(C)CO1)CC2 c1(C(N2CC(C)(NC(c3cccc(OC)c3F)=O)C2)=O)cc(S(N)(=O)=O)co1 C(C(C)CC(=O)N(CC(C)(F)F)C)NC(C(C)OCC)=O C1(CNC(Cc2c(C)ccs2)=O)CC2CC2N1C(=O)CCCC1CCCCC1 C1(C(N2CCC(N(C)CC)C2)=O)CN(C(=O)CC2CCCC(C)O2)CC(C)O1 c1(C(=O)NC2CC(CNC(C(C)S(N)(=O)=O)=O)OCC2)cc2ccccc2s1 C1(CNC(Cc2cc(CC)no2)=O)(NC(=O)C(=O)NCCC(N)=O)CCCCC1 c1(C(=O)NCC2CC(NC(C(CC)N(C)C)=O)CC2O)cn2c(C)cccc2n1 CCCC(C)C(=O)NC1CC(NC(c2c[nH]c(=O)cn2)=O)CC1O Cc1cc(C)c(C(=O)NC(c2ccnn2C)C(N2CCOCC2CO)=O)s1 c1(OC)ccc2c(c1)CCC2C(=O)NCC(C)N(C(=O)CC1=NN(C)C(=O)C1)C c1(CC(=O)NC2CC(NC(c3c(C)cc(F)s3)=O)C2)c(C)nn(CC(C)C)c1C CC(C)C(CC(=O)N1CCCC(C)(CNC(c2cnc(O)s2)=O)C1)c1ccon1 c1(C(N2CC(NC(C(CCC)N(C)C)=O)C(C)(C)C2)=O)ccc(Cl)c(N)c1Cl C1(CNC(C(F)=CCC)=O)C(C2CC2)CCN1C(=O)Cc1c(C)noc1CC CCC(c1cccc(Cl)c1)=CC(=O)NC1CN(C(c2occc2F)=O)CCC1C n1(CC(=O)OC)cnc(C)c1C(=O)NC1CCOCC1NC(=O)C(C)CSC N1(C(c2c(CC)n(C)nc2)=O)C(C)CN(C(=O)C(=O)N=S(C)(C)=O)CC1C c1(C(=O)NC(CC)CO)cn2c(n1)CN(Cc1ccnc(C(=O)OC)c1)CC2 C1(C(=O)NCCC(C)NC(c2cc(C3CC3)ncn2)=O)(COC)CCC(=O)N1 C(C(C)(C)CNC(=O)CCc1cnc(C)s1)N(C(C1(OC)CCSC1)=O)CC CC(C)CC(CNC=O)CC(=O)N1CCC1CNC(c1cscc1S(C)(=O)=O)=O C1(CC=C)(C(=O)OC)CCCN(C(c2cnn(-c3cc(C)ccc3F)c2N)=O)C1 C(CN=c1nc(C#N)[nH]cc1C)C1CCC(NC(CN(CC)CC)=O)C1 C1(n2cc(C(C)N(C)C(c3cc(C(F)F)no3)=O)nn2)CCCCCC1 N1(C(CN(C(C(C)=CCC)=O)C2CCC2)=O)CC2(CCN(C)CC2)C1 N1(C(=O)C=Cc2cccnc2)CCC2(COCCN2C(c2ccc(O)cn2)=O)C1 N1(C(C(CO)NC(N)=O)=O)CCC(=CCNC(C2CC23CCOC3)=O)CC1 CC1(C)CC(NC(=O)Cc2ccoc2)CN1C(c1cc(COC(C)(C)C)[nH]n1)=O Cc1cc(S(=O)(=O)NC(C2CCCC2N(C)C)=O)c(C(=O)N(C)C)cc1Br Cc1csc(Cl)c1C(=O)NCC1(CO)CCN(C(C2(CC(C)C)CC2)=O)C1 C1(C(=O)NC(C(=O)NC)CC2CCC2)CC2CCC1N2C(=O)CCCCCSC N1(C(CCOC)=O)CCC=CC1C(=O)NCCCOCC(C)C N1(C(COCCCC)=O)CC2COCC2(C(=O)NC(C)CCC(F)(F)F)C1 Cn1ncc2c1CC(C(=O)NCCC1COCCN1C(=O)OC(C)(C)C)CC2 C(CC(=O)NCc1ccc(OC(F)F)cc1F)(C(C)C)C1C(C)CNCC1 Cc1nc2n(n1)CCC(C(=O)OCc1cnccc1C(F)(F)F)C2 CC(C)(C#CC(=O)N1CC2CSCC2C1)CNC(C1(C)CC=CCC1)=O Cc1ccc2c(c1)C(NC(=O)C(=O)NCCOC1CCN(C)CC1)CC2 CC1NC(=O)CCC1NC(C1CC(O)(CN(C(C2CCO2)=O)CC2CC2)C1)=O c1(CC(=O)NCCCN(C(CCCCC)=O)CC)c[nH]c2cccc(C)c12 c1(NCc2cn(C3CCN(C(c4[nH]cc(C)c4)=O)C3)nn2)ccccc1Br C1(CN2C(=O)NC(CCCCC)C2=O)(NC)Cc2ccccc2C1 C1(NC(CCOCC(C)C)=O)CN(C(c2ccnn2C2CCOCC2)=O)CC1C c1(C(C)(C)C)ncnc2cc(I)sc12.N12CCN(CC1C#N)c1ccnc2n1 C#Cc1ccc(C(=O)N(CCNC(=O)C(c2ccc(C)s2)C)C(C)C)c(F)c1 N1(C(C(C=C)(F)F)=O)CCN(C(c2cccn2CC)=O)C(CS(C)(=O)=O)C1 NS(=O)(=O)c1ccc(CNc2ccc(I)c(F)c2F)nc1 Cc1cc(OCC(N2CC(c3nccc(C)n3)C2)=O)cc(F)c1 C(c1cccc(O)c1)=CC(=O)N(C1CCN(C(c2cn(C)nc2C2CC2)=O)C1)C Cn1c(C(N2CCCCC(NC(c3ccn(C(F)F)n3)=O)C2)=O)ccc1[N+](=O)[O-] C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1CN(C(C2(CCCC)CC2)=O)CC1F CCC(C(=O)N1CC(C(C)(C)O)(CNC(=O)C(F)n2ccnc2)C1)NC(C)=O c1(C(=O)NCC23C(CN(C(C4CN(C(C)=O)C4)=O)C2)C3)cc2c(Cl)nccc2o1 Cc1cc(C#N)nc(N)c1NC(N1CC2(CO)CCC1(CO)CC2)=O C(=O)(N1CCCc2nncn21)C1CCN(C(Cc2cnc(C)s2)=O)CC1(C)C C(C)(C(C)C(=O)NCCC(C)(C)CO)NC(C(N1CC(C)C1)C)=O c1(C(CN)O)ccc(C)cn1.N1(C(C(Cn2cncn2)N(C)OCC)=O)CCCC1C c1(C(N2C(CC(=O)NC3(C)C(C)(C)C3(C)C)CCCC2)=O)coc2ccccc12 Cc1ccc(C(N2CCCC2Cn2cc(CNC(C3CC3(F)F)=O)nn2)=O)nn1 Cc1cc2sc(C(=O)NC(C3CCCN3C(C3CC34CCCC4)=O)(C)C)cc2s1 c1(-n2c(C(C)(C)C)nc(CC(=O)NC)n2)ccc2c(c1)CCO2 c1(CNCC(CC(=O)OCC)(C)C)cccc2c(C)coc12 N1(C(C(C=C=C)C)=O)CC2(CCC2)CC1C(=O)NCC(=O)N(C)C1CC1 c1(N2C(C3CCN(C(c4cc(C)ns4)=O)C3)CCC2)nc(C2CC2)nc2[nH]ccc12 C=CC1(C(N2CCC(N(C(C3CC4(C3)CC(O)C4)=O)CC)C2)=O)CCCCC1 N1(C(C(C)c2cccs2)=O)CC2C(NC(c3c[nH]c(C(F)(F)F)n3)=O)C2C1 C12CCCC(C1)NCC(=O)N2C.C1(C(CC#C)=O)CC2(CSC2)C1.C1CCCO1 Cn1cc(S(N)(=O)=O)c(C(=O)NC2CN(C(=O)COC3(C)CCCC3)C2)n1 c1(CC(=O)N(CC(CNC(C2(OC)CCOC2)=O)O)C)cnn2c1CCCC2 Cc1nn2ccccc2c1C(N1CC(CNC(c2ccc(O)cc2O)=O)C1)=O c1(OC)ccc2c(C)c(C(=O)NC3(C)CCC(F)(F)C3=O)oc2c1 c1(C(C(=O)NC2C(C)CN(C(c3cnn(C4CC4)c3)=O)C2)=O)ccc(F)c(F)c1 C1(C(c2n(C(CC)C)nnn2)NCc2oc(C3CC3)nc2C)CCS(=O)(=O)CC1 C1(NC(c2cnc(OC)nc2)=O)CC(O)CN(C(c2ccsc2Br)=O)C1 C(=O)(C1Cc2ccc(F)cc21)NCC1CC(NC(=O)Cc2c[nH]nc2O)C1 C1(CC(N2CCC(CN=c3[nH]ncs3)(CC(F)F)CC2)=O)CC2(CCC2)CO1 C1(C(N(CCCNC(C(C)SC)=O)CC2CCCC2)=O)CCN(S(C)(=O)=O)C1 c1(CC(=O)NC2CC(NC(C(CCC)OCC)=O)C2)cc(C)cc(C)c1 C(CCN=c1[nH]c(=NCCC(=O)N2CCCCC2)[nH]c2cc[nH]c12)OCC(C)C c1(C(=O)NC(CC=C)CNC(=O)C(C(CC)CC)OC)c[nH]c2cccc(Cl)c12 Cc1ccc(CC(=O)NCCC2CCN(Cc3ccccc3OC(F)F)C2)cc1 CCC(C)(C)C(O)C(=O)N1CCOC(C(=O)NCC(Cl)C(C)(F)F)CC1 C1(NC(C(C=C)(C)O)=O)CN(C(C2CN(C(=O)N(C)C)C2)=O)C2(CCC2)C1 N1(C(COCC(C)(C)C)=O)CC(NC(C2CC3(CCCO3)C2)=O)C(C)(C)C1 C(=O)(C(C)(F)c1ccon1)N(CC(C)NC(C1CSCCS1)=O)C C#CCCN=C(NCCCNCC1(O)CCN(C(N)=O)C1)N(C)CC C(=O)(CC1=NNC(=O)C1)NCC(C)NC(c1ccc(CNS(CC)(=O)=O)cc1)=O N1(C(CC2C(C)OCC2)=O)CCCCCC1C(=O)NOCc1nc[nH]n1 N1(C(CCSCCC)=O)CCCCC(C(=O)NCCC(O)COC)C1 c1(C(=O)NCC2CN(C(CC(C(C)C)O)=O)CC2(C)C)cc2ccccc2[nH]1 c1(C(N2CC(O)(CNC(c3c(C)coc3)=O)C2)=O)ccc2ncsc2c1 CC1(C)CC(CNC(=O)Cc2nc(C3CC3)nn2C)CN(C(=O)CSC2CC2)C1 C1(C(N(C2CN(C(=O)C3=C(Cl)CCC3)CC23CC3)C)=O)Cc2ccccc2S1 Cc1ccc(O)cc1C(N1CCC(C)C(NC(c2ccc(C3CC3)nc2)=O)C1)=O N1(C(CCN(C)CC)=O)C2CCC1C(NC(=O)CSc1nc(C)cc(C)n1)C2 c1(C(=O)NCC2C(C)(C)C(NC(=O)CCCC3CC3)C2)c(N)cccc1[N+](=O)[O-] c1(OC)ncc(C(=O)NC2(CO)CCN(C(=O)C(C)C(F)F)C2)cc1Cl N1(C(C)=O)CCC(NC(=O)CCN(CCO)C(c2cnoc2C(F)(F)F)=O)C1 Cc1nn(C)c(C(=O)NC(c2ccccc2)CNC(c2cc(Cl)cn2C)=O)c1Cl Clc1ccc(OCCNC2CCC(Nc3cc(-c4ccccc4)ncn3)C2)cc1 c1(C(=O)NC2CC(NC(Cc3cc(C)on3)=O)C2)nc2ccc(Br)cn2n1 C(C(C(=O)N(C1CCCCCC1)C)C(C)(C)C)NC(COCC(C)C)=O C1(C(=O)NC2(C)CN(C(c3c(C)noc3C3CC3)=O)C2)C2CC3C(C2=O)C13 C1(C(N2CC3C(CNC(c4c(C(=O)OC)coc4)=O)C3C2)=O)CC(=O)OC1(C)C N1(C(C2(CC#C)CC2(F)F)=O)CCC(N(C)C(c2cc(C(C)CC)no2)=O)CC1 C1(C(C(N2CC(=CCC)C2)=O)C)CCCN(C(C2(C)CCOC2)=O)C1 C1(C(=O)NC2C(NC(C(C)(C)SC)=O)CCOC2)CCCCNC1=O CCC(CC)(C(=O)N1CCC2(CC(C(N3CCSCC3C)=O)C2)C1)C(C)C Cc1ccc(C(F)(F)F)cc1C(=O)NCC1CN(C(=O)Cc2cnsc2)CCO1 C(C)(C)(CCCN=c1[nH]cc(Cl)c(C)c1C#N)NC(COCCCOC)=O C(=O)(C(C(C)C)NC(C1CCCOCC1)=O)N1CC(C)(CC=C)C1 c1(C(=O)NCC2(CO)CCN(C(CC3C(C)CCO3)=O)C2)nnc(O)nc1O c1(C(=O)NC(CNc2nccc(OCC)n2)(C)C2CC2)cccc2scnc12 C=CC(C)(CCOC)C(=O)N1CCN(C(c2cccc(CN(C)C)c2)=O)CC1C Cc1cc(N)c(C(=O)NC(CCNC(c2ocnc2C)=O)C(C)(C)C)nc1C C(=O)(CCC(C(=O)NCc1nc(-c2ccccc2)oc1C)N(C)C)OC N1(C(C(CC)(C)O)=O)CCC2C1CCCN2C(c1cc(Cl)ccc1F)=O C(C(CN=c1[nH]c(N2CCC(CC(C)C)C2)nc2cccnc12)C(F)(F)F)OC C1(CC(=O)NCC(C(C)C)(C)F)N(C(C2CCCCCN2C)=O)CCC1(C)C C12(NC(C=CC(=O)N(C)C)=O)CCN(C(=O)Cc3cccc(C4CC4)c3)CC1C2 c1(-n2cc(CCC(=O)Nc3ncc(CC)s3)nn2)ccc(F)cc1F c1(OCC)ncccc1C(=O)N(CCCCCNC(c1nnn(CC)c1C)=O)C C(=O)(C(C)(C)CN1CCOCC1)N(CC(C)N(C(=O)CNC(N)=O)C)C C1(NC(=O)COc2ccc(Cl)cc2)CCCC12CN(C(C1(F)CCC1)=O)C2 S(=O)(=O)(c1ccc(Br)cc1F)NCC1CCCN(C(C2CCC(CO)CC2)=O)C1 C1(C(=O)NC2C(CNC(CC(C)(O)C3CC3)=O)CCCC2)CCCCCCC1 C1(C(=O)NC(c2ccc(I)cc2)C)CC2(CCN1)CCOCC2 C1(NC(CSc2c(OC)cccc2)=O)CCC(C)N(C(=O)C2=CCCOC2)C1 C(=O)(C1=C(C)CCOC1)NCCC1CC(C(N2CCC(OC)C2(C)C)=O)C1 C(=O)(C(C)CC(C)CC)N(CCCCc1c(OCC)nccc1)C(C)C N1(C(CC2(OC)CN(C(C34CCC(CC3=O)C4)=O)C2)=O)CCCCN(C)CC1 c1(C(=O)NC2CN(C(c3c(C)nsc3)=O)C2)c(C(F)F)nc2n1CCCC2 C(C(C(=O)NCC(=O)N(C)C)C(C)(C)C)NC(CCC(C(C)C)N(C)C)=O N1(C(CCC(=O)NCC)=O)CCN(C(c2cc(F)c(CO)c(F)c2)=O)CCC1C c1(CNCC(=O)NC(c2ccc(O)cc2)C(F)(F)F)ccc([N+](=O)[O-])cc1F S(=O)(=O)(c1ccc(Br)c(Cl)c1Cl)NC(c1ccccc1Cl)COC CCCS(=O)(=O)CC(=O)NCC1CC1NC(=O)CCCCC=CC C(c1cccc(F)c1)=CC(=O)NCCC(C)NC(=O)C(=Cc1cnc[nH]1)F c1(C(N2C(C(=O)NC(C3CCCC3)C#C)CC(C)(C)C2)=O)ccc2c[nH]nc2c1 CC1CN(C(=O)COC2CCCOC2)CCCN1C(c1cncc(Br)c1)=O c1(C(N2CC(CNC(CCCOC)=O)N3CCC2C3)=O)n[nH]c2nccc(Cl)c12 c1(C(=O)NC(CC=C)CNC(=O)CNS(=O)(=O)C2CC2)cnc2snc(C)c2c1 C1(C(=O)NCCC(=O)NC(C)C)(NC(C23CC(F)(C2)C3)=O)CCC(C)(C)C1 C1(C)(COCC)CCCN(C(C23CC(n4cc(C(=O)OCC)nn4)C2C3)=O)C1 c1(C(=O)NCC(C)(O)CNC(=O)COCc2ccncc2)ccc2cccnn12 C(N=c1[nH]c(=NCCNC(C)=O)[nH]c2ccsc12)C1C(CCC)C1 C(=O)(C1CCc2nccn21)N1CCCC(CC(=O)NCC2CC(C(F)(F)F)C2)C1 c1(C(=O)OC)ccc(N(C(C)CCNC(=O)Cn2cnccc2=O)C)nc1 C1(C)(C(=O)NCC(N(C(CN(S(C)(=O)=O)C)=O)C)C2CC2)CCCN1C C(C)(CCN=c1[nH]c2ccc(Br)cc2o1)NC(C1(C)C(CC)CCC1)=O Cn1[nH]c(=NC(=O)NCCc2ccncc2)cc1C1CCCC1 Cc1ccc(OC(C)C(=O)NCCC2CC(NC(=O)CCOC=O)C2)c(C)c1 N1(CCCCCNC(C2(CC=C)CCCC2)=O)CCN(C(=O)C(O)C(F)F)CC1 S(=O)(=O)(c1ccc(Br)s1)N1C(CC(=O)Nc2c(OC)cccc2Cl)CCC1 Cc1cc(N2CCC(N(C)C)CC2)ncc1S(=O)(=O)NCC1CCCC1CCO C(=O)(C1CCc2c[nH]nc21)N1CCN(C(c2c(C)ncc(C)c2)=O)C(C)CC1 C(=O)(CCN=c1[nH]c2ccccc2s1)N1CCC(CNC(C(C)(C)F)=O)C1(C)C c1(SCC)ccc(NC(C2CC(Cn3cc(C4(F)CCOCC4)nn3)C2)=O)cn1 C=CC1(C(N2CCCC2CC(N)=O)=O)CCN(C(C2C=CC=CC=C2)=O)C1 N1(C(C2(OC)CC2)=O)CCC2CCN(C(=O)C=Cc3cc(Cl)cc(Cl)c3)CC2C1 CCCC(C)CCCC(=O)N(C1CCCN(C(c2cccc(N)c2O)=O)CC1)C c1(C(N2CCCN(C(C(CC)(C)O)=O)CC2C(C)C)=O)nn(C)c2c1CSCC2 O=C(C1=CC2CCCCCC12)NCC1CCN(c2ccnc(Cl)n2)C1 c1(C(N(C2CN(C(CN3CC(C)(OC)C3)=O)C2)C)=O)ccc2nn[nH]c2n1 Cn1cnnc1C(CO)NC(c1ncoc1CNC(c1cncs1)=O)=O CCC(O)C(C)C(=O)NC1CC(OCC(=O)NC23CC(F)(C2)C3)C1 N1(C(c2cc(C(C)=O)sc2)=O)CCN(C2CCN(C(=O)CC(C)C)CC2)CC1 CC(C)C(CC(=O)N1CCCC(C)(N(C)C)C1)NC(=O)C(C)N1CCCC1 C1(C(=O)NC(CN(C(CCN(CC)CC)=O)C)C)COC(C)(C)C1 c1(C(N2CCC(C)(C(N(CC(C)OC)C)=O)C2)=O)cc2c(=O)[nH]c(C)cn2n1 Cc1cn2c(n1)C(C)CC(C(=O)NC1CN(C(c3ccn(C(C)C)n3)=O)C1)C2 N1(C(COCCC)=O)CCC2(CNC(=O)C3CC3)CCCCC12.OCC c1(C(N2C(CC)C=CCC2)C(=O)NCCCSC)ccc(C2CC2)c(F)c1 C12(C(=O)NC3C(NC(=O)C4=NOCC4)CC3)CCCCC(=O)N1CCC2 c1(C(=O)NC2(C)CC(NC(Cc3cc(C)sc3)=O)C2)ccc(CC(C)(C)C)cc1 C1(CNC(Cc2cnc(C)[nH]2)=O)CC(F)CN1C(=O)C(C)Oc1cccnc1 N1(C(c2cc(C)c(C)o2)=O)CCC(C)N(C(=O)Cc2nc(=N)[nH][nH]2)CC1 C(=O)(C1CCOc2c(F)cccc21)NCC(C(C)C)NC(=O)C(F)(F)CN(C)C C(CC(CC)C(=O)NC1CN(C(=O)COc2cccnc2)CCC1O)=CC CC(C)(CC(F)C(=O)NC1CC(CO)C2CC12)NC(C1C=CCCC1)=O C(=O)(C(C)(C)CC(F)(F)F)N(CC(C)NC(C1CCC(C)C1)=O)C c1(C(N(CCNC(C(CC)CC(F)F)=O)C(C)C)=O)cnc2ccncc2c1 c1(CC(=O)NCC(CNC(=O)C(F)=C2CCCC2)F)cccc(N2CCCC2)c1 c1(C(=O)NC2CCN(C(C34OC(C)C(C3)C4)=O)C2)ccc2nc(C(F)F)[nH]c2c1 c1(C(=O)NCC2(O)CN(Cc3c(C)nccn3)C2)cc(O)nc2ccccc12 c1(C(N2CCC(CCNC(CCC(C)(C)C)=O)C2)=O)ccccc1-c1cn[nH]c1 c1(OC)c(C(=O)NC2CC3C2CCN3C(C2COC2)=O)cc(Br)cc1F c12cnc3cc(ccn13)[nH]c2=O.C(=O)(C(CC)C(C)C)N1C(CO)CC(OC)C1 N1(C(C(C)SCCCCCC)=O)CCN(C(=O)C(C)(C(C)C)OC)CC1C(C)C C12(C(=O)NC3CCN(C(CC4N(C(C)C)CC4)=O)C3)CC3CC(CC(C3)C1)C2 CCC(C)(O)C(=O)NCC(O)CNC(=O)C(c1ccc(SC)s1)=O Cc1ccc(C(=O)NCC2CCCCN(C(c3cnnn3C)=O)C2)cc1O C(c1c(O)ccc(Cl)c1O)=CC(=O)N(CC(C)NC(c1ccnn1C)=O)C c1(C(=O)NCC(C2CCC2)NC(Cc2c(C)ocn2)=O)nn(C)cc1Cl C(c1ccccc1)=CC(=O)NC(C)(CNC(C1CC1c1ccoc1)=O)CO C1(C(=O)NC(CC)CSC)CC(=O)N(CCc2ccccc2-c2nc(C)no2)C1 O(C=CC(O)(CNC(=O)NC(Cc1ccccc1)C(C)=O)C(F)(F)F)CC N1(C(C)=O)CCCC(O)(C(=O)NC2CC(NC(c3c[nH]nc3C3CC3)=O)C2)C1.N(C)C O=C(N=c1cc[nH][nH]1)C1(C(=O)O)CC1.N12CCC(CC1)C(=O)N1CCC2C1 c1(N(C)C)ccc(CNC(=O)C(=O)NCCN2CCNC(=O)C2)cc1 c1(NC(CN2CC(CNC(C(CC)C)=O)C2)=O)ccc(Nc2ccccc2)cc1 c1(C(=O)NCCC2CC(NC(=O)Cc3cnsc3)C2)ccnc2ncccc12 C1(C)(C(=O)NC(CN(C(=O)CCc2cn[nH]c2)C)Cc2ccccc2)CC(F)(F)C1 CC1CC(COC(C2(Nc3ccccc3)CCCCC2)=O)CCO1 C12(C(=O)NCCCNC(C)=O)CC1CN(C(C1CCC(CO)CC1)=O)C2 C(=O)(C(CC)(CC)c1ccccc1)NCCCC1N(C(C=CCC)=O)CCCC1 C(C1CCN(C(c2ccco2)=O)CC1)=CC(N1C(C)(C(=O)OC)CCC1)=O c1(C(=O)NC2CCN(Cc3ccc(NC(C)=O)cc3)C2)cccc2ccnn12 C(=O)(CCS(=O)(=O)CC(C)C)N1CCN(C(CCCCCOC)=O)C(CO)C1 c1(C(=O)NCCCCN(C)C)cccc(-n2cc(COC(=N)O)nn2)c1 C1(CC(=O)NCCCC(C)NC(C2(C(N)=O)CCC2)=O)CCC12CCC2 N1(C(C(c2c(OC)cccc2)O)=O)CC2(C1)CN(C(c1cc(Cl)nc(=N)[nH]1)=O)C2 c1(C(=O)NCCc2nnco2)ncncc1Cl Cc1c(O)c(=O)ccn1CC(N1CC(NC(C2CC2(C)C)=O)C2(CC2)C1)=O N1(C(=O)Nc2c(CC)c(Br)ccc2)CCN(C)c2ncccc2C1 C1(C(N2CC(C)(NC(=O)CN3CCCC3CO)C2)=O)CC2C=CCC(C1)C2 N1(C(Cc2cnc(C)[nH]2)=O)CC2(C1)CN(C(c1coc(CC(C)(C)C)n1)=O)CCO2 c1(CC(N2CC(CC(C)NC(=O)COCCN(C)C)C2)=O)ccn(C)n1 CC1(C)CN(C(c2ncnc(O)c2Cl)=O)CCC1NC(C1CC(C2CC2)=NO1)=O C1(NC(CC2CNCC(C)O2)=O)CCN2CCCCC12 c1(C(=O)NCC2(C(=O)NCC3N(CC)CCC3)CCCC2)occ2c1CCC2 CC(C)(C)C(CN)N1CCCC1.S(C(F)(F)F)CC=O c1(C(N2CC(SC)C(NC(c3cnn(CCO)c3)=O)C2)=O)nc(C)c(C)nc1O C(=O)(C1CCCc2nn[nH]c21)N1CCN(C(C=Cc2c(C)nccc2)=O)CC1 c1(CC)ccc(OC)cc1C(=O)N(C1CCN(C(=O)C2=CCCCO2)C1)CCO S1(=O)(=O)c2cc(ccc2C)CN1.c1(OC)ccc(C(C)=O)cc1.C12CC1(C)S2 c1(C(N2CCC(NC(C(c3ccncc3)C)=O)C2C)=O)nc(Cl)ccc1Cl CCCCC(C(=O)N1CCCCC(CNC(=O)COC2CCCC2)C1)N(C)C.C=O Cc1c(F)ccc(C(N2CCC(C)C2CNC(c2cnccn2)=O)=O)c1N C(CC(C(N)=O)NC(C1(CNC(=O)C(C)SC)CCCCC1)=O)OC C1(NC(c2cnc(C)[nH]c2=N)=O)CN(C(=O)C(=C2CCCCC2)F)CC(C)(C)C1 C1(N2CCCC2)(CC)CCN(CC2CCN(c3cc(Cl)ccc3C)C2)CC1 C=CC1(CC(=O)N(CCCNC(c2cc(C(C)(C)C)n[nH]2)=O)C2CC2)CCC1 C(=O)(CCCCCS(N)(=O)=O)NC1C(CN(C)C)CCCC1 c1(C(=O)NC2C(C)CN(C(=O)C(n3cnc(C#N)n3)C)C2)ccc2c(c1)CCO2 c1(OCC)ncc(C(=O)NCCCCCN(C(=O)C(C)c2ccon2)C)s1 N1(C(c2nc(CCC)oc2)=O)CCC2CCN(C(C3(C)CC(=O)N(C)C3)=O)CC12 C(CC(C)(C)C(=O)N1CCC2C(NC(=O)CCCc3cc(C)sc3C)C12)SC c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)CCO)C2)ccc(Cl)c(F)c1F N1(C(C(c2cccc(F)c2)C)=O)CCOC(CNC(C2CC2(F)F)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CCCC(CCNC(Cc2nc(C(C)C)sc2)=O)C1 C(=O)(CCC(C)(C)C#N)NC(CNC(c1n(C(C)C)ccc1)=O)C1CCC1 CN1CCN(C(=O)CC2CCC(O)C2)C(CNC(=O)Cc2cnc(Cl)cn2)C1 c1(COC)nc(C(N2CC(C(C)(C)O)(CNC(c3cscc3F)=O)C2)=O)co1 C12(NC(C(CO)N(C)C)=O)CCCC1N(C(=O)Cc1ccc3c(c1)OCO3)CC2 C(CCCCC(=O)N1CCCC(CO)(NC(=O)C=CC2CCCO2)C1)SC c1(C(=O)Nc2ccc(NS(N)(=O)=O)cc2)cc2c(cc1F)NCCC2 C(C(O)CC(=O)N1CCC(CN(C(=O)CC2CCC(O)C2)C2CC2)C1)N(C)C N1(C(C(CCC(C)C)NC(C2CC3(CC3)CO2)=O)=O)CCC2(CCCCO2)C1 CC1CN(C(C2CCCC23CCC3)=O)CC1(C)C(N1C2CCC1CC2)=O C(C1CN(C(C2(CC(N)=O)CCC2)=O)CC1C(N1CC(OC(C)C)C1)=O)=CC C1(NC(c2nccc(OC)c2)=O)CCN(C(c2ccc(Cl)cc2C)=O)CC1CO CCCC(CNC(C1(C)CC(F)(F)C1)=O)C(=O)N1CC(N=[N+]=[N-])C1 C(c1cccc(F)c1Cl)=CC(N1C(C)(C)C(CNC(=O)C=CC(F)(F)F)CC1)=O C1(NC(c2nncc(OC)c2)=O)CCN(C(c2snc(C)c2N)=O)CC1CO c1(C(C)NC(c2n(CCSC)nnn2)C2(CSC)CCC2)cccc(F)c1F C1(CN(C(=O)Cc2ccc(C)s2)CC)CCCCN1C(c1[nH]ccc1C)=O C1(C(C)C)CC(O)CN1C(=O)C(CNC(C1CN(C(C)C)C1)=O)CC1CC1 C1(NC(C2(C)CC2(F)F)=O)CN(C(C23CC(C(F)(F)F)(C2)C3)=O)CC1C#N C1(NC(CS(CC)(=O)=O)=O)CC2CCC1CN2C(=O)C(C)(F)C(F)(F)F C1(C(N2CCN(C(CCn3ccc(C)n3)=O)C(C)C2)=O)CCc2nc(O)[nH]c2C1 N1(C(C(c2cn(CC)nc2)=O)=O)CC(CNC(=O)C2CC2)N2CCC1C2 N1(C(CNC(c2ccc(C)s2)=O)=O)CCN(C(C2CC3C=CC2O3)=O)CC1CO C1(NC(c2ccc(OC)c(Cl)n2)=O)CN(C(=O)C(C(C)C)SC)CC2CCCC12 C1(NC(C2C(C=C)C2)=O)CCCN(C(c2cccc(-c3nnc(C)o3)c2)=O)C1 c1(C(C(=O)NC2CC2)N(C)CC2C=CCC2)ccnn1C N(C1CCCn2ncnc21)C(C=C)C Cc1ncn2ccc(C(N3CCC(NC(=O)CCCCC#N)CC3)=O)cc12 N1(C(=O)C2CC2)CCCC(C(N2CCC(n3cncn3)C2)=O)C1 N1(C(=O)NC2C(c3n(C)ncc3)C2)CCCc2c(F)cccc21 c1(NCCCC(CC)O)cc(Br)ccc1S(=O)(=O)NCC1CCSC1 C1C(C)CCCN1C(C)=O.C=CC(C(=O)NC)c1ccccc1 C1(N(C(=O)CSC2CC2)C)CCCCN(C(C2(O)CC2(C)C)=O)C1 C1(CNC(C(C2CCC2)OC)=O)CC(O)CN1C(c1cn(CC(F)(F)F)cn1)=O C1(C(N(C(C)CC(F)(F)F)C)=O)CN(C(=O)CN(C)C)CCC1(C)C C1(CC(=O)N(CC(=O)NCC=Cc2cn(C)nn2)CC)CC2(CCC2)CO1 c1(NC(C2CC(C)CN2C(C2CCCCN2C)=O)=O)cc(O)c(F)cc1F c1(CNC(CC2CC(NC(CNC(CC)=O)=O)C2)=O)nnn(C)n1 N1(C(COCC)=O)CCC(CCNC(C2CC(C)(C(=O)OC(C)(C)C)C2)=O)C1 C1(C(N(C(CC)CO)C)=O)(CO)CCN(C(=O)C(=O)N(C)C)C1 N1(C(=O)Cc2cnc(O)nc2O)CCC2(C1)CN(C(C1COC1)=O)CCO2 N1(C(CN2CCC(OC)C2)=O)CC(C)(C)C1C(=O)NC1COCC1C(N)=O C1(O)(Cn2cc(CCc3c(C)nc[nH]3)nn2)CCN(CC2CCOC2)C1 C(c1ccc(C)nc1)=CC(=O)N(C)CC1(O)CCN(C(C(C(C)C)OC)=O)C1 CCC(CC(=O)N1CCC(NC(c2nc(O)sc2C)=O)C(CC)C1)C(C)(C)C c1(C(=O)NC2CCCC2CNC(c2cc(CO)cs2)=O)cnc(O)c([N+](=O)[O-])c1 c1(C(=O)NCCCC(C)NC(=O)CN2CCOCC2)cc2ccccc2[nH]1 c1(C(=O)NCC(CNC(CNC(CC(C)C)=O)=O)C)cccc(N(C)C)c1 C1(C(N2CC(N(CC=C)C)C2)=O)CCCC(NC(C2OCCC2(C)C)=O)CC1 c1(C(=O)NCC(CNC(CCCN(C(C)C)C)=O)C)ccc(-n2cncn2)cc1 Cn1ccc(-c2n[nH]cc2C(=O)NC(CNC(C2CCSC2)=O)CO)n1 C(=O)(C(C)(C)CCC(=O)OC)NC1CC(NC(C(F)=CCC)=O)C1 Cc1nccn1CCC(=O)NCC1(C(=O)NCCCO)CCC1 C1(CNC(C2CCC(C)(C)CC2)=O)CC(C)(C)CCC1NC(=O)CC(F)F N1(C(CCC(=O)OCC)=O)CC2CC(NC(c3cc(OC)ccc3F)=O)CC1C2 c1(C(C)NC(C2CC3CC3C2)=O)nocc1C(=O)N(C)Cc1ncc[nH]1 c1(NCC2(CNC(CN=S(C)(C)=O)=O)CC23CCC3)ccc([N+](=O)[O-])cc1 CCN=c1ccc(C(=O)NC2CCOCC2NC(=O)CC2(N(C)C)CCC2)c[nH]1 C1(C(N2CCC3C(NC(c4cnc(SC)n4C)=O)C32)=O)CCC(=O)N(C)C1 N1(C(c2cnc(C)[nH]2)=O)CC2CCC2(CCNC(=O)CSc2nc[nH]n2)C1 CCCC(CC1CCCC1)C(=O)NC1CC(CNC(C2CC3(C2)CC3(F)F)=O)C1 N1(C(Cc2nc(C)[nH]c2)=O)CC(CNC(c2nc[nH]c2C(C)(C)C)=O)CC1C C(=O)(C(CNC(=O)C(CC=C)OCC)CC(C)C)N(CCC#C)CC O=C(CC1C(=O)Nc2ccccc21)NCCC1(O)CN(C(=O)CCOC(F)F)C1 C(=O)(CCCCCC#N)N1CCCCC(C(=O)NC(CC#C)CC)C1 O=C1CCCC(C(N2CCCCC2C(=O)NCCc2cccnc2O)=O)CC1 c1(C(c2n(CCC)nnn2)NC(C)C(=O)NCCOC)cc(Cl)sc1C C(=O)(C(C#N)C(C)(C)C)NC1(CO)CCCN(C(c2cc(OC)c(O)nc2)=O)C1 c1(C(N2CCC(c3scc(C)n3)CC2)C(=O)NCCC2CC2)sc(C)c(C)c1C N1(C(C2(C)CC(OC)(OC)C2)=O)CC(NC(c2cccn(C)c2=O)=O)CC(O)C1 N1(C(C(CCC)OCC)=O)CCN(C(c2cc(=O)c(OC)co2)=O)C(CF)C1 c1(C(N(CC(N2CCC(CCC)C2)=O)CC)=O)ccn2cncc2c1 c1(NCC)ccc(C(=O)NCCN(C(=O)C(O)C2CC2)C2CC2)cc1 N1(C(C(=O)NC(C)C)=O)CC2CCN(C(C3CCCC(C)(C)C3)=O)CC2C1 C1(OCC(N2C(CNC(c3cc(C(CC)CC)no3)=O)CC2)=O)CCC(C)CC1 C=C1CCCN(C(=O)CC2(CNC(=O)C(C3CCCCC3)O)CC2)C1 c1(C(N2CCN(C(C3CC(C)OC3=O)=O)CC2)=O)cncc2c1CCC2 N1(C(C2N(C(=O)OC)CCC2)=O)CCC(O)(CCNC(C2CNC(=O)N2)=O)CC1 c1(C(=O)NC(C(C)NC(c2cnccc2Cl)=O)(C)C)cccc2c1COCCN2 c1(CN2CCC(CNC(c3cn(C(C)(C)C)nn3)=O)C2)cc(Br)cc(F)c1O CCC(C)CCCC(=O)NCC=CCC(=O)NC(C)(CO)C1CCCC1 C1(Cc2cccc(F)c2)CCCN1N1CCC(Oc2ccccc2Br)CC1 CCCC(C(=O)NC1CCCC1C(=O)NCC)NC(=O)C(CCC)OC C1(C(C)C)C(NC(c2coc(O)n2)=O)CCN1C(=O)COc1ccc(O)cc1 CC(C)CCC(O)C(=O)NCc1cn(CC(=O)N(CC(C)C(C)(C)C)C)nn1 N1(C(C2(CNC(C(C)O)=O)CCCO2)=O)CCOC(C)(C)C1C C12(NCc3c(C)cccc3C)CCC(C(N3CCC3CO)=O)(CC1)CC2 c1(C(=O)NC(CNC(=O)CNC(=O)Cc2cn[nH]c2)CO)ccc(Cl)cn1 n1(CC)nc(C(C)C)cc1C(=O)NCC1CCN1C(C1CCCCO1)=O C(CS(=O)(=O)CC(=O)NC1CC(CNC(=O)C(C)C(C)C)C1)OC N(C1CCCc2cc(F)cc(Cl)c21)C(c1ncc(Br)cn1)C c1(CC(=O)NC2(C)CCN(C(C3CCN(C(C)=O)C3)=O)C2)ccc2ocnc2c1 CC(C)CCC(O)C(=O)N1C(C)CC2CCCC12.c1(C(=O)NC)cc2n(n1)CCO2 Cc1csc(=NCC(=O)NC(CNC(c2ccn(CC(F)F)n2)=O)CC(C)C)[nH]1 n1(CC)c(C)nn(CC(=O)NC2CCC2NC(=O)C(F)(F)CN(C)C)c1=O C1(NC(C(CCCOC)C)=O)CCN(c2cc(O)ncn2)C12CCC2 n1(CC#C)cccc1C(=O)NCCN(C(=O)C(C)Cc1ccccn1)CC(C)O c1(NC)scnc1C(=O)NCC(C)(O)CNC(=O)CNS(N)(=O)=O C#CC1(O)CC(C(=O)N(CCCCN(C)C(C2(C(C)(C)C)CCCCC2)=O)C)C1 C1(OC(C)C)CCCN(C(=O)CCCCN(C(=O)C(N2CCOCC2)C)C)C1 CC1(C(=O)OCCC23CCC(C2)C3(C)C)CC2CCC(C1)S2 c1(C(C(=O)NC2(CCNC(CNC(C)=O)=O)CC2)O)ccc(F)cc1 C(N=c1[nH]c(=NCCS(=O)(=O)CCOC)[nH]c2ccncc12)c1n(CC)nnn1 O=C(CCCCCc1ccccc1)NCCC1CCN(C(c2cscn2)=O)C1 C1(N(C(=O)C(F)=C2CCCC2)CC)CCCN(C(c2csc(C3CC3)n2)=O)CC1 CC12CCC(CC1)SCCOCC(=O)NC2.c1(CC2(C(=O)OC)CC2)cccs1 c1(C(=O)NC2CCN(C(c3ncn(C)n3)=O)C2)csc2ccc(C(F)(F)F)cc12 S(=O)(=O)(CCC1CNCC2=C1C=CC=NN2)N(CCCOCC)C C(=O)(CC(C(F)F)C(C)(C)C)NC1C(C)N(C(=O)C(C)CSC(F)(F)F)CC1 C(C(C)CN=c1cc(C2CC2)nc[nH]1)C1C(C)CCCN1C(=O)C(O)C1CCC1 c1(NC(N2CCC(CN(C(=O)C(Cl)=CCl)C)C2)=O)ccc(CO)c(Cl)c1 C(CC(F)F)(C(=O)NCC1(O)CCC(C)C1)NC(c1c(C)csn1)=O C12(NC(CN(C)CCn3cncn3)=O)CCC(CC1)N(C(=O)COC(=O)CO)C2 N(C1CN(C(=O)C(C2CC2)OC)CCc2ccccc21)C(C(CCCC)O)=O C1(NC(c2ccc(CCF)cc2)=O)CCN(C(=O)CCc2csnn2)C12CC2 C1(C(=O)N(CC(C)NC(c2sc(-c3ncc[nH]3)nc2C)=O)C)(OC)CS(=O)(=O)C1 c1(C(N(C)CCN(C(=O)C(C)(C)Oc2ccc(F)cc2)C)=O)[nH]cc2c1CCC2 c1(C(C(=O)N(CCn2cc(CCSCC)nn2)CC)F)cccc(C)c1 Cc1ccc(C)c(NC(=O)C(CNC(C2CN(C(C)C)C2)=O)CC2CC2)c1 C1(N(C(=O)CCN2CCCC2)CC)CCN(C(=O)C(C)(C)N2CCCCC2)C1 c1(-c2c(C(=O)NCC3CCC(CCC)CC3)n[nH]c2)ccc(S(C)(=O)=O)cc1 Cc1cccc(CCNC(C2CC(C)N2C(=O)CC2CCCC2O)=O)c1 N1(C(=O)CCc2cccc(Cl)c2)CCN(C(c2cc(O)ncn2)=O)C2CCC12 N1(C(=O)NC2(N(C)C)CCN(C)CC2)CCCN(CCF)CC1(C)C CC1=CCN(C(=O)C(C2CCCC2)NC(c2c[nH]c(=N)o2)=O)C1 C=CCC(C(=O)NCC1(CNC(=O)C(C)(C)c2cccnc2)CCC1)C(C)(C)C c1(OC)ccc(O)cc1C(=O)NCC1CCN(Cc2cncc(C)n2)C1 c1(C(N2CCCN(C(C3CCN(C)S3(=O)=O)=O)CC2)=O)ncc2n1CCCC2 c1(C(N2C(CCN(C(CCCCC)=O)C)CCCC2)=O)c[nH]c2cccnc12 c1(NCC(=O)NC(C)(C)CNC(C2CC3CCC2C3)=O)ccc([N+](=O)[O-])[nH]1 C1(CNC2(c3nnnn3C)CC(C)(CC)C2)(CC)CCCCCC1 C1(NC(=O)Cn2cnnn2)CCC(NC(c2cnc(C3CCC3)o2)=O)CC1 N1(C(=O)CC2(c3ccccc3)CCCO2)CCCCC1Cc1ccccc1Br C12(NC(C=COCC)=O)CCCC1N(C(c1n[nH]c3c1CC(C)CC3)=O)CCC2 c1(C(=O)NC(c2ccc(OC)cn2)C)c(OC(F)(F)F)ccc(Br)c1F C(=O)(C1CCCc2ccnn21)N(CCN(C(C1OCCN(C)C1)=O)C)C N(C(=S)N1CCCC1c1c(C)ccc(C)c1F)CCC N1(C(C=CC(CC)C)=O)C2CCC1CC(NC(c1cccc(Cl)c1C)=O)C2 C(C)(C)(C(=O)NCc1ccc(C(=O)NC(c2ncc(C)s2)C)s1)OC(C)=O C(C)(CCCC(=O)N1CC(N2CC(O)C2)C1)NC(C(C)N(C(C)=O)C)=O c1(C(=O)NC2(C)CC(NC(=O)CC3C=CS(=O)(=O)C3)C2)cccnc1SC(F)F Cc1cc(C(N2CC(CNC(=O)C(C)C(O)C(C)C)C(O)C2)=O)c(O)cc1F c1(CNC(C2C(NC(=O)OC(C)(C)C)C3CCC2C3)=O)ccc2[nH]ccc2c1 N1(C(C(C=C)(F)F)=O)CCC(C)(C)C(C(=O)NCCN2CCOCC2C)C1 c1(OC)ccc(F)c(CN2CC(CO)CC2C)c1Cl C1(NC(C(C)SC(F)(F)F)=O)CC2CCC1N(C(=O)Cc1ccn(C)n1)C2 n1(CCC(=O)NC(CCNC(C2(C)C(C)C2)=O)(C)C)ncc2ccccc12 N1(C(C2N(S(C)(=O)=O)CC2)=O)CCCCC2(C1)CN(C(=O)C=C(Cl)Cl)C2 c1(C(=O)NCC(C(C)C)Nc2cccc(C(=O)OC)n2)cnc(OC)c(Cl)c1 c1(OC)cnc(C(N2CCOC(C(C)NC(=O)CC(C)O)C2)=O)c(F)c1 CCCCC(CN=c1nc(OC)cc(OC)[nH]1)NC(c1cnc2c(c1)CCOC2)=O N1(OCC(=O)Oc2ncc(-c3c(C)cccc3)o2)C(=O)c2ccccc2C1=O C1(CCNC(C2CC23CCCC3)=O)CC(F)(F)CN1C(=O)C1=CSCCO1 N1(C(C)C)N=C(C(=O)NC2C=CCN(C(c3cc(O)n(C)n3)=O)C2)CCC1=O C(=O)(CCCCC(C)(C)OC)NC(c1c(OC)cccc1)C(C)SC C1(C(=O)OC(CCOCCCC)C)CC(=O)N(C2CCC(OC)CC2)C1 N1(c2sc(C(=O)OC)c(C)n2)CC2CCN(C(=O)OC(C)(C)C)C2C1 C12(C(=O)NCC3(O)CC(NC(c4ccccc4)=O)C3)CC3CC(CC1C3)C2 CCC(C)C(O)C(=O)NCCOCCN(C(=O)CN1CCCC(CC)C1)C N1(C(C2(C#C)CCC2)=O)CCOC(C)(CNC(C2C3CC4C(C3=O)C24)=O)C1 c1(C(=O)NC2(CNC(C(C)OC)=O)CCOC2)ccc(C(C)CC)nc1O CC1(C(=O)NC2CCS(=O)(=O)CC2)CC12CCN(C(CCC(=O)O)C(=O)O)CC2 C1(C(=O)NC2CCN(C(=O)CCOC3CCC3)CC2O)CCn2c(O)nnc2C1 N1(C(c2c(C)ncn2O)=O)CC2CCC2(CNC(c2c(F)cncc2Br)=O)C1 CCCCCCCC(=O)NCC1(NC(c2ccn(C)c(=O)c2)=O)CCCCC1 CC(CC(=O)NCCc1nc(C2CCCCC2)n[nH]1)c1cnn(C)c1 c1(OC)ccccc1CCC(=O)NC1CC(CO)N(C(C2COC(CF)C2)=O)C1 CC1(C(=O)NCC2CC3CN(C(C4CC(O)C4)=O)CC23)C2Cc3ccccc3C12 c1(C(C(=O)NCC(=C)CCNC(=O)C=CC(=O)N(C)C)C)c(Cl)cccc1Cl Cc1[nH]c(C)c(C(=O)NCC2CCC(NC(=O)C(C)(C)C(F)F)C2)c1C c1(C(C)=O)cc(C(=O)NCC2(F)CC(NC(=O)COc3ccccc3)C2)oc1C c1(NC(C(C2N(C(C(CC)OCC)=O)CCC2)(C)C)=O)ccc(F)c(CO)c1 C1(CC(=O)N(C(CNC(=O)C#CC2CC2)C2CC2)C)CCC2(CCOCC2)CO1 c1(N(C)Cc2nc(=N)[nH][nH]2)nc(N2CCC(n3cncn3)C2)c2ncn(C)c2n1 CC1CN(C(=O)CNc2ccccc2Cl)CC1NC(=O)CC1CC(=O)NC1=O N1(C(c2ccncc2Cl)=O)CCC2(CC1)CCN(C(c1cnnc(Cl)c1)=O)C2 C(=O)(C(CCCC#N)N1CCN(C)C2CC12)Nc1c(C)cccc1 C1(C(=O)NCCNC(c2ccc(CN3CCCCC3)o2)=O)CCS(=O)CC1 N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(=O)CC(=O)NC)C1(C)C N1(C(c2cc(C)n(C(C)C)n2)=O)CCCC2(C1)CN(C(=O)CCC1CCOC1)C2 C1(NC(CCc2cn(C)nn2)=O)CN(C(C2CC23CC3)=O)CCC12CCC2 c1(CC(N2C(C(=O)Nc3ncccc3OC(F)F)CC2)=O)cccc([N+](=O)[O-])c1 S(=O)(=O)(C1CC2(CC(F)C2)C1)N(C(c1ccc(NS(C)(=O)=O)cc1)C)CCO c1(C(N2C(C(=O)NCCOCCOC)CC2C)=O)cc(C)ncn1 CC(O)CCCCCC(=O)N1CCN(C(=O)CC=C(Cl)Cl)C2(CC2)C1 c1(NC2CCCC(NC(C(CC(C)C)C)=O)C2)cccc(F)c1[N+](=O)[O-] c1(CNC(=O)Nc2n(CC)ncc2)cnc(NC)nc1 N1(C(c2cnc(C(C)C)n2C)=O)CCN(C(=O)C=CCN(C)C)C(CF)C1 C1(C)(C(N(C)CC2CCCCC2O)=O)CN(C(=O)CCC(CF)CF)C(C)(C)C1 c1(C(N(C2CCN(C(CCCCC#C)=O)C2)CC)=O)cccc2ncsc12 c1(OC)c(C(N2CCC(C3CCCN3C(=O)CC(C)(C)C#N)C2)=O)ncnc1C C12(C(N(CCOC)CCNC(=O)COCc3ccncc3)=O)CCCCC1C2 Cc1nn(CCO)c(C)c1C(=O)NCC1CCCC1NC(C1(C)CC=CCC1)=O N1(C(C2C(OC(C)=O)C2)=O)CC2C(CNC(C3CCCN3C)=O)C2C1 Cc1nncc(CNC(=O)N(C)CC2CNC(=O)N2)c1C c1(OC)ccc2c(C(=O)NCCCCCCN(C)C(c3cnn[nH]3)=O)c[nH]c2c1 N1(C(C2N(C(C(C)N=[N+]=[N-])=O)CC(C)CC2)=O)CCCC(C)(C#N)C1 c1(OC)ccc(F)c(C(=O)NC2(C)CCCN(C(c3cc(C(C)=O)cs3)=O)C2)c1 c1(C(=O)NC(C2N(C(C=NOC)=O)CCCC2)C)cc([N+](=O)[O-])ccc1SC C(=O)(CCCCCF)N1C(CCNC(c2ccccc2F)=O)CCC1 C1(O)(C(CNC(c2cc(SC)oc2)=O)C)CCN(C(c2cnn(C(F)F)c2)=O)C1 CCCCCCC(CC)C(=O)NCCCC1CCCN1C(C1CC2(CSC2)C1)=O C(C(CC)(CC)C(=O)NCc1cccnc1)NC(C1N(CC)CCC1)=O C12(CNC(c3c(N)ccc(CC)c3)=O)CN(C(=O)C(CC)C(C)C)CC1CCO2 c1(C(N(C(C)C)C2CC2)=O)cc(CNC(C2CCCC2F)=O)nn1C CC1(C)CC(CC(=O)Nc2cccc(C3CC3)c2)N(C(=O)CC2CCCCC2)C1 c1(OC)cccc(F)c1CN1CCSCC1C(=O)NCCCSC c1(C(N2C(CNC(C3CCCS(=O)(=O)N3)=O)COCC2)=O)cn2ccccc2n1 c1(CNCc2ccc(-c3cc(OC)cc(COC)c3)nc2)ccc(C)c(C#N)c1 C(=O)(CN=c1[nH]c(=NCCCNC2CC2)c2ccccc2[nH]1)N(CC)CC C1(NC(COc2cc(C)on2)=O)Cc2ccccc2C1NC(C1CC(CF)C1)=O C(=O)(C1CCOc2ccccc21)N1CC(NC(c2c(C)oc(Cl)n2)=O)C(C)CC1 c1(OC(C(=O)NC2CCC(NC(c3c(CC)onc3)=O)C2)C)ccc(C)cc1C c1(NC(=O)NC23CC2C3)ccc(O)nn1.C1(CN)CC(O)C(O)C1.C(F)F C(=O)(CCS(=O)(=O)N1CCCCC1)NC1C(NC(CSC)=O)CCCC1 CON1CCC(NC(=O)NCC(=O)OC(C)(C)C)CC1.C12CC1N2 c1(C(=O)NCc2ncn(C)n2)ccc(CNC(C2CC3(CCC3)C2)=O)cc1 Cc1nc(NC(C2CCN(C(C3CCCN(C)C3)=O)C2)C)c2cc[nH]c2n1 C1(C2CCC2)(C(N2CCC(C)(NC(C=CC(C)(C)SC)=O)C2)=O)CC1(F)F CC1CN(C(=O)CC2N(C(=O)CC3CCOCC3)CCC2(C)C)CCCO1 C(=O)(CCCn1cccc1)N(CC(c1ccccc1)O)C(c1ccccc1)C CC(C)C1=NOC(C(=O)NCCC(C)N(C)C(c2cc(O)cc(=O)o2)=O)C1 CC1CCCC(CCNC(=O)CC2CCCC2NC(C2CCC2)=O)C1 Cc1cc(C(=O)NCC(C)CNC(C2(N(C)C)CC(O)C2)=O)cc(O)n1 c1(NC(c2ccc(OC(F)F)cc2)=O)cn2ccc(-c3cccnc3F)cc2n1 C(=O)(CN=c1[nH]c2ccccc2s1)N1C2CN(C(C3(C)CCOC3)=O)C(CC2)C1 N1(C(c2cc(C)c(C)s2)=O)CC2(CC(C(=O)NCCOC3CCC3)CO2)C1 N1(C(c2cccc3c2CCO3)C(=O)NCCCC)CCCCC12CCOC2 C1(NC(C(C=CCCC)O)=O)CC(C)N(C(=O)C(CC)n2ccnc2)C1 c1(OCCC(=O)NCCC2CN(C(=O)COCC(=O)NC)C2)ccccc1F c1(C(=O)OC)sc(NC2CCC(NC(C3CCC(C)CC3)=O)CC2)nc1Cl C1(NC2(C(=O)NCCC(=O)N(CC(=O)OC)C)CCC2)CC2(C1)CC(C#N)C2 N1(C(C(=O)NCSCCSC)CC2CCC(C(C)C)CC2)CC2CCC(C1)N2C C(CCCCCCO)NC(=O)CCCNC(C1CC12CCCCC2)=O c1(CC)nccnc1C(=O)NC(C1CCCCC1)C(=O)NCC(O)CO c1(C(N2CCC(C(=O)NCc3ccncc3F)C(O)C2)=O)cc2cccnc2s1 c1(CN2CC(NC(=O)Cc3ccc(Br)nc3)C(O)C2)cccc(O)c1O Cc1cccc(Cl)c1C(=O)NC1CCN(C(=O)C(c2cccc(Cl)c2)O)CC1F N1(C(c2cnc(CCC(F)(F)F)s2)=O)CCN2CC3(CC3)CC2C1 CCC(CC(=O)N1CC(C(C)NC(C2CC(O)CN2C(N)=O)=O)C1)OC Cc1cc(=O)oc(C)c1C(=O)NC1CN(C(=O)COCC2CCCC2)CCC1F c1(CC(N2CC(N(C(C3C(CCC)CCC3)=O)C)C2)=O)c(C)nc(CC)nc1C c1(C(=O)NCCC2CCCN(C(c3cn(C)nc3)=O)C2)cc(N)c(Cl)c(O)c1 C(N=c1nc2c(c[nH]1)COC2)C1(NC(C2CCC3C(C)(C)C2C3)=O)CCOCC1 c1(CCC(=O)NC(CNC(CC=C)=O)CO)cc(Br)ccc1C N#CC1(CC(N2C3CCC(C3)C2CNC(=O)CCC2CC2)=O)CCOCC1 c1(C(=O)NC2C(NC(C(C=C)O)=O)CC2)c(F)c(C)cc(N)c1F c1(NC(C2N(Cc3c(OC)ccc(Br)c3)CC3(CC3)C2)=O)c(O)cccc1C#N c1(OC)ccc(C(=O)NCC23CC2CN(C(=O)C(N2CCCCCC2)C)C3)cn1 C1(NC(c2nc(CC)sc2)=O)CN(C(C2CCOC(C)(C)C2)=O)CC1(C)C c1(C(=O)NCC(C(C)(C)C)NC(c2cc(O)cc(Cl)c2)=O)ccc2nccn2c1 C12(C(N3C(C(C)(C)NC(CCC=CC(C)C)=O)CCC3)=O)CCC(N=[N+]=[N-])C1C2 N1(C(CC(C)(C)OC)=O)C2CCC1CC(CNC(C1CC3C=CC1C31CC1)=O)C2 C(=O)(C#CC1(C(F)(F)F)CC1)NC1CCCN(C(c2cc(C)sc2C)=O)C1 C1(NC(=O)CNC2CC(=O)N(C3CN(Sc4cocn4)C3)C2)CCCCCC1 C1(CC(=O)NCC(C)(C)NC(C(C)Cc2cccnc2)=O)CC=CCN1C c1(C(=O)NCCCCCCNC(c2ccc(OC)s2)=O)[nH]cc2c1CCS2(=O)=O Nc1ccc(C(=O)NC2CCCC23CCN(C(=O)C(N)=O)CC3)c(S(N)(=O)=O)c1 CCC(C(=O)N(C(CNC(=O)CC1CCOC1)CC)C1CC1)N(C)C N1(C(c2c(OC)csc2)=O)CC(NC(=O)C(c2cccc(F)c2)(C)C)C2CC12 c1(OCC(=O)NCC(C)CNC(c2nc(=O)n(C)[nH]2)=O)ccc(F)cc1O c1(C(N(C2CCN(C(=O)C(C)c3cc[nH]n3)C2)CCC)=O)ccnn(C)c1=O c1(CC(N2CCC(NC(c3c(CC)nn(C)c3)=O)C2)=O)cc(Br)ccc1F c1(C(N2CCCC(F)C2)=O)cc2c(C(F)(F)F)cccc2s1 N1(S(c2cccc(C(=O)NC)c2)(=O)=O)CC(C)Oc2cc(F)ccc21 C(=O)(C1Cc2c(Cl)cccc21)N1CCCC(N(C(C2(COCC)CC2)=O)C)C1 Cc1nc(Cl)cc(Cl)c1C(N1CCCC1(C)C(=O)Nc1c(Br)ccc(F)c1F)=O N1(C(C2CC(=C)CN2C(=O)Oc2ccccc2)=O)CCc2cc(F)ccc2C1 Cc1cc(C(=O)NC2CC3CC2N(C(c2nc(C)oc2C)=O)C3)cc([N+](=O)[O-])c1 N1(C(CNC(CCOCC=C)=O)=O)CCCN(C(=O)COCCSC2CC2)CC1 c1(C(=O)NC(C2(O)CCN(C(=O)C3=CCS(=O)(=O)C3)C2)C)ccc(S(N)(=O)=O)o1 C(C(=O)NC1CCOC1)(C1=CCSC1)NC(=O)CN1CCCCC1 c1(NCCC=C)ncnc(N(C)CC2CCOC2c2c(OC)cncc2Cl)c1C c1(C(=O)OC(CC2N(CC)CCS(=O)(=O)C2)=O)ccc2c(c1)nnn2CC CC(O)C(C)(C)C(=O)NCC1CC(F)(CNC(=O)C2=CCCCC2)C1 Cc1csc(C(N2CCCCC2c2ccco2)C(=O)NCCC2CC2)c1C N1(C(c2c(C)nns2)=O)CC2CC(NC(c3nc4ccccn4n3)=O)CC2C1 C12(NC(CCn3ncn(C)c3=O)=O)CC3CCC(C1C2)N3C(=O)CC1(O)CC1 CC(C)CC(C(=O)NCCC(C)CCO)ONC(=O)CC1CC(C2CC2)C1 N1(C(c2ccc(CC)s2)=O)CCC2(CC1)CC2C(N1CC(CO)C(CO)C1)=O c1(C(=O)NC2CCC(C)(NC(c3cccc(O)n3)=O)CC2)cc2nc[nH]c2cn1 Cc1nc(C)c(C(=O)NC2CCCC(CNC(=O)CSc3cccc(F)c3)C2)[nH]1 C1(C(N2C(C3(NC(C=CC=CCC)=O)CC3)CCC2)=O)C2CCCCCC12 c1(CC(=O)NC2(CCO)CN(C(C(CN(C)C)(C)C)=O)C2)c(N)nc(C)nc1O N1(C(CC(C)SC)=O)CC2(CCCC(CNC(=O)CCN3CCCCC3)O2)C1 C1(CNC(c2nccnc2Cl)=O)(OC)CCN(C(=O)CSCC(F)(F)F)CC1 c1(C(=O)NC2CCC(NC(C3CC(C#N)(OC)C3)=O)CC2)cccc2c1CCC2 C=CCC(C)C(=O)N(CC(=O)NCC(C)(CO)OC)CCOC C12(C(=O)OC3CC(OC(=O)C4CC4)C3)CC3CC(CC1C3)C2 C1(C(=O)NCC2N(C(CC(C)O)=O)CC2)CCCCC1c1nc[nH]n1 c1(C(=O)OC)ccc(CN2CCCC2CC(=O)NCc2cncs2)nc1 Cc1cc(C(N2CCC(C)C2CNC(c2ccc(CO)nc2)=O)=O)sc1C CC(C)CCC(=O)N1CC(O)(CNC(=O)C(O)Cc2cnn(C)c2)C1 N1(C(CSCC#C)=O)CCN(C(=O)C=CCF)CC1c1ccc(OCC)cc1 C#CCCCC(C)C(=O)NC(C)(C)C(C)CC(=O)N1CCCC(CN(C)C)C1 c1(CC)nc(-c2ccc(-c3nccn3CCO)s2)c2n1CCCC2 C1(CN(C)C(C2(C)CC2C(F)(F)F)=O)CCCCN1C(c1cc[nH]n1)=O N1(C(c2nc(C(C)=O)sc2)=O)CCC(NC(=O)C(C)CC2CCC2)C(C)(C)C1 CC1(C)CN(C(C2(C)CC2Br)=O)CC(CNC(c2ccn(C(F)F)n2)=O)O1 c1(C(=O)NC2CN(C(C(C)OCOC)=O)CC2C2CC2)ccc(Cl)cc1[N+](=O)[O-] N1(C(C=CC2N(C)CCC2)=O)CCC2(CC2)CC1C(=O)NC1CC12CCC2 N1(C(C(CO)OC)=O)CC2(CCN(C(c3cscc3Cl)=O)CC2)C1 CCCC(C)CC(=O)NCCCCCC(=O)NC(C(=O)OC)C(C)OC N1(C(C(CC=C)C)=O)CCOCC2(COCCN2C(=O)C(O)CCCC)C1 CCCCC(F)C(=O)NCC1(C)CN(C(=O)CCn2ccccc2=O)CCO1 Cc1nc(NCC2CCCCC2O)cc(N2CCCC2c2ccccc2Br)n1 C(CC1=CCN(C(C2(C3CC3)CC2)=O)CC1)NC(CC1CCN(C)CC1)=O CC(C)C(CC(=O)N1CCCC(NC(C2CSc3ccccc3O2)=O)C1)C(C)C CCCC(CC)C(=O)N1C2CCC1C(C(N1CC3CC3C3CC13)=O)C2 N(C1CCCc2ccoc21)C(C(CC(F)F)N(C(=O)CSC(F)F)C)=O C1(CNC(c2n(CC)cnn2)=O)CCCC2(CN(C(=O)CC3CC(F)(F)C3)C2)O1 C=C(C)C(C)(C)C(=O)NCC1CCCN(C(=O)CC2COC(C)(C)CO2)CC1 C1(CNC(c2cc(C)[nH]c2)=O)CCC(C)CN1C(c1ncoc1C)=O C1(CNC(CCC=CC)=O)CN(C(=O)Cc2cc(C)[nH]n2)CC1(C)C N1(CC(=O)NC2CCCN(C(C3C4CC5C(C4)C35)=O)CC2F)CCc2ccccc21 c1(N2CCC(C)(CN(C)C)C2)nc2c(c(=NCCC(O)C3CC3)[nH]1)CCC2 C=C1CCN(C(c2nccnc2C)=O)C(C(=O)NCCC(O)C2CCCC2)C1 CCCCC(CNC(C1(C)CCCC1C)=O)NC(=O)C1=NOCC1 c1(C(=O)NCCC(C)(C)CNC(c2ccncc2Cl)=O)ncnc(O)c1F Cc1cc(C#N)ccc1NC(c1ccc(C2CCCCC2N)cc1)=O c1(NC(C(=O)NC2CC(SC)C2)=O)c(Br)cc(Cl)c(Br)c1Cl CC(C)C(O)C(F)(F)C(=O)NCC1CN(C(=O)C(C)NC(=O)C2CC2)CC12CC2 CC1C(C(=O)Nn2ccnn2)CCCN1C(=O)COCCN(C)C C1(C(=O)NCC(C(=O)NC)O)CCCN(C(=O)C(C2CCCCC2)C)C1 CC(C)CCCCCC(=O)NCC1CCCCC1NC(c1cccnc1)=O C1(C(=O)NCC(CC(C)C)NC(CSCC=C)=O)CCCC2(CCCCC2)C1 CC1(C)c2ccccc2CN1CC(=O)NC(c1ccccc1)=O C1(N(C(CC2N(C(c3cncc(CC)c3)=O)CCOC2)=O)C2CC2)CC2CCC1CC2 C1(NC(=O)CC2OCCCO2)CCN(C(c2cnnc(O)c2)=O)CC1 c1(C(=O)NCC(C(=O)NC(c2c[nH]ccc2=O)C)(C)N(C)C)ccc2c(c1)CC2 c1(C(=O)NCC(C)NC(=O)CSCCN(C)C)cccc2nnn(C)c12 C(=O)(C(C)(C)C(C)(C)C)NC1C(C)N(C(c2ccc(CS(C)(=O)=O)o2)=O)CCC1 C1(C(=O)OC(C)(C)C)CC(C(N2CCC(c3ccccc3)CC2C)=O)CCC1O n1(CN(C2CCC(Nc3nnccc3C#N)CC2)C(C)=O)ccc(=O)c(O)c1C CN1CC(C(=O)NCC2CCN2C(=O)Cc2ccc(-n3cccc3)cc2)NC1=O CC1CC(C(N2CC(CN(C)C(C3CC(F)C3)=O)C2)=O)CCS1 C(CC(C(=O)NCCC1CCCC2CC12)NC(=O)Cc1cnc(C)s1)OCC N1(C(COC)=O)CC2CCC(CNC(c3cccn3C)=O)(C2)C1 C1(C(=O)NC(c2ccc(Cl)cc2)C)CCCN(CCS(=O)(=O)NC2CCOC2)C1 CC(CCC(C)(C)C)C(=O)N1CCC(C(N2CC=CC2CN(C)C)=O)C(O)C1 C1(C(N2CC(C)CC(NC(c3c(C)occ3)=O)C2)=O)CC2(C1)CC1(CC1)C2 N(C1CCCc2occc21)C(C(C)(CO)NC(c1ccc(C)nn1)=O)=O C1(C(C)NC(=O)C(C)NC(N)=O)CCCN1C(c1cnccn1)=O.CC(F)(F)F C1(OC)CCCCC1NC(C1(F)CN(C(=O)Cn2nnc(SC(C)CCCl)n2)C1)=O C1(CNC(CCCC=C)=O)CCC(C)(C)CN1CCC1CC1OC c1(C(=O)NC2CN(C(C(CC)(F)F)=O)CC(C)C2)cncc2ccc(F)cc12 C1(CC(N2CC(C(C)(C)O)(CNC(C(C)n3ccnc3)=O)C2)=O)CCS(=O)(=O)C1 C1(C)(CNC(C=C(C)CNC(c2ccnn2C)=O)=O)CC2CCC1C2 CCCCCC(O)CC(=O)NCCC1CCN(C(C2CC3(C2)CC2(CC2)C3)=O)C1 Cc1ccc(C(=O)N(CCCN(C)C(C2CCCC3(CCC3)O2)=O)C)cc1C#N c1(C(N2CCCC(CC=C)(NC(C3CC3CCC)=O)C2)=O)nc2ccccc2[nH]1 C1(C(F)(F)F)(OC)CC(C(=O)NC2CCC(NC(=O)CC3(O)CCC3)C2)C1 C1(CC(=O)NC(c2c[nH]ccc2=O)C)CCCN(C(C2(O)CCCC2)=O)C1 N1(C(COCCC)=O)CCN(C(=O)CCC2CCCN(C)C2)C(CC(C)(C)C)C1 C1(NC(=O)CN2CCCCC2=O)CC(C2CCN(C(=O)C3=CCC3)C2)C1 c1(-c2cn(-c3cccc(C4CC5(C4)CC(F)C5)c3)nn2)ccccc1P(C)(C)=O.CC C1(N=[N+]=[N-])(C(=O)NCc2ccc(C)nc2)CCN(C(c2cc(C)n(C)c2C)=O)C1 C1(CCCCCNC(C(CC2CC2)OC)=O)CCN(C(=O)CC2(O)CCC2)CC1 c1(N2CCCCC(CNC(c3c(C)ccs3)=O)C2)ncnc2c1nnn2C(C)C N1(C(C(C)n2cncn2)=O)CCC(OCCNC(=O)Cc2ccccc2)CC1 c1(C(N2CC(NC(=O)Cc3ccc(Cl)s3)C(F)CC2)=O)cnc2c(c1)CCCO2 c1(C(=O)NC2(CCNC(=O)Cn3cc(Cl)cn3)CCC2)ccc(O)c([N+](=O)[O-])c1 Cc1cc(F)sc1C(=O)N(C1CCCN(C(=O)C(F)(F)C2CCCC2)C1)C C(=O)(C1c2ccccc2C2CC1C2)N1C(C(=O)NCC(CCOC)OC)CCC1 Cc1cc(C(C)(C)C)ccc1C(N1CC2CC2(NC(=O)C2=COCCO2)C1)=O C1(CCNC(c2ccsn2)=O)CCCN(C(c2coc(CO)c2)=O)C1 C1(C(N2CCCC(C)C2CNC(=O)CC2=CCCC2)=O)CCc2nncn2CC1 n1(NCC)cnc2nc(=NCc3nnc(C(C)C)s3)[nH]c(NS(=O)(=O)C3CC3)c12 C#CCC(CC(F)F)C(=O)N1CC(C(C(=O)NC(c2cccc(C)n2)C)OC)C1 C1(NC(c2c(C)cc(O)cc2)=O)C(CNC(c2sccc2C)=O)CCC12CCC2 C1(C(=O)NC(C2CC(NC(C3CN(C)C(=O)N3)=O)C2)C)CCCC2CC12 c1(CC)ccoc1C(=O)NC1CCC1NC(c1cc(COC)on1)=O Cc1cc(CNc2ccc(OC(F)(F)F)cc2Cl)cc(O)n1.Cc1ncsc1C=O c1(OC)c(C(=O)NC2CC(NC(C3CN(C(C)=O)C3)=O)C2)ccc2c1CCC2 C=CC(C)(C)C(=O)NC(CO)C(C)NC(C1(c2cc[nH]n2)CC1)=O N1(C(CCSC)=O)CCCOC(CNC(=O)Cc2ccc(NC(C)=O)cc2)C1 N1(C(c2csc(-c3ccc(Cl)cc3)n2)=O)CC2COCC(C1)C(=O)N2 n1(CC)cc(CC(N2CCC(NC(c3cnnn3C3CC3)=O)C2)=O)nn1 c1(C(N2C(CNC(c3c(C)nc(CCC)o3)=O)C(C)CC2)=O)ccc(F)nc1F N1(C(C(COC)NC(C)=O)=O)CCCC2(CCN(C(c3ccnn3CC)=O)C2)C1 c1(C(N2CCC(NC(C3C(C)CCC3)=O)CC2C)=O)cc(O)c(O)c(O)c1 C1(C(=O)Nc2cc(OC(C)C)ncn2)CCCN(C(C2CCCC23CC3)=O)CC1 CC1CCn2c(C(N3CC(O)(C(C)NC(c4occc4Cl)=O)C3)=O)cnc2C1 N1(C(c2cccc(OC)n2)=O)CCC(C(=O)N=c2ccn(C(F)F)[nH]2)C12CCC2 CS(=O)(=O)C1(C(=O)NC2CC3(CCN(C(=O)COCC4CCC4)C3)C2)CCCC1 Cc1c(C(N2CCC3(C2)CN(C(=O)CN(C)C)C3)=O)[nH]c2cc(F)ccc12 N1(C(C2(CNC(CC3(N(C)C)COC3)=O)CC2)=O)CCC2CCC12 Cn1ccc2cccc(CN3CCC(C#N)(NC(c4cc(I)ccc4F)=O)C3)c12 c1(C(N(C(C)CCNC(=O)CCc2nc(O)n[nH]2)C)=O)ccccc1O C1(C(F)(F)F)(CNC(c2cc(C)sn2)=O)CC2CCC1CC2.C12CCN1C2=O C1(C(=O)NCCN(C(C(=O)NC2CC2)C2CCCC2)CCCO)CCCOCC1 Cc1cc2cc(C(N3CCN(C(C4CCC=CCC4)=O)CC3C)=O)oc2cc1C O=C(C1=CC2(CN(C(=O)CCCC3CC3)C2)OC1)NCCc1ccnc(O)c1 c1(C(=O)OC)ccnc(N(C(Cc2ccc(O)cc2)C(N)=O)C)c1I Cc1ccc(C=C2CCN(C(=O)Nc3ncc(F)nc3C)C2)cc1 C(CCCCCN(C)C)NC(C1(C)CN(C(C(c2scc(C)n2)C)=O)C1)=O C(=O)(CC(C)(C)n1cc(-c2cc[nH]n2)nn1)NCC(C)OC C1(C)(NC(C=CC(C)(C)SC)=O)CCN(C(=O)NC(C)C)C1.C12CCCN1C(=O)N2 C1(CC)CNC(=O)CN1C(=O)C(C)(C1CC1)N(C(=O)C(C)n1ccnc1)C N1(CC)CCC2CN(C(c3ccsc3C)=O)CCC12.C1(C(=O)N)(CO)COC1 C1(CC=C)(C(=O)N(C(C)C(C)SC)C)CN(C(C23CSCC2C3)=O)C1 c1(C(=O)NCCC(=C)CNC(C2(O)CC2)=O)cncc(C(C)(C)C)c1 C=CCC(F)(F)C(=O)NCCC1CCCN(C(=O)C(C)C(C)(F)F)C1 CC1(C)CCC2(CC1)CC2NC(N1CCOC(C(F)(F)F)(C(=O)O)C1)=O CCC1=C(C(=O)N(C)CC2CCCCN2C(c2ccn(C)c2C)=O)SCCO1 CC(CC(=O)NC1CCN(C(c2cc(C(F)F)cs2)=O)CC1F)P(C)(C)=O C(=O)(CC(C)(c1cccs1)N(C)C)NCC1N(C(CCC2C(C)C2)=O)CC1 C1(C(CNC(C)=O)NC(=O)CC2COC3CC2C3)CCc2ccccc2C1 C=CC1(C(=O)NC(C)CC(C)NC(C2CCC(CC)CC2)=O)CCOCC1 c1(CNC(C2(C(C)C)N(C(CC(=O)OC)=O)CCC2)=O)cn(C)nc1C(N)=O C=CCC(C)(C)C(=O)N1CCC(CNC(c2ccc(C(C)(C)C)[nH]2)=O)(OC)CC1 Cc1cc(C(=O)NCCCCCN(C(=O)CC(C)c2ccccc2)C)ccc1O C(C(=O)Nn1nnc(C)c1C)N(CCOC)C(C1CC(=O)N(OC)C1)=O C(=O)(CC(C)C(C)C(C)C)OCCOc1c(C(=O)OCC)cc(Br)cc1 C1(NC(C(C)CN(C)C)=O)CC=C(C(=O)NCCc2cccc(O)n2)C1 c1(C(=O)NCC2N(C(c3ncc(N)nc3)=O)CCC2)cc2c(F)cccc2[nH]1 N1(C(C(C)SCC)=O)CC2C3CCC(C2C1)N(C(=O)C(=Cc1cccnc1)C)C3 N1(C(C2N(CC)CC2)=O)CC(C)(C)CC1CNC(=O)Cc1c(C)cccc1F N1(C(c2cccc(F)c2)=O)CCC(F)(C(=O)NC(c2ccccc2)CO)CC1 CC(C)(C(=O)NCC(=C1CN(C(c2coc(O)n2)=O)C1)F)C1(C)CC1(F)F c1(OC)ncc(C)c(C(=O)NC2CC(F)(CNC(=O)CC(C)N(C)C)C2)c1Cl c1(CN(CC)CC)c[nH]c2cc(F)ccc12.c12cc(c(O)c(OC)c1)OC2=O C1(C)(C(N(C(C2CCCO2)C)C)=O)CN(C(C23CSCC2C3)=O)C1 C1(CN)CCN(CC)CC1.CCCCCCN(C(=O)CC(=O)OC)CC(=O)NCC c1(C(N2C(C(C)NC(c3cnoc3-c3ccoc3)=O)CCC2)=O)c(Cl)cnn1C N1(C(CNC(C)=O)=O)Cc2ccccc2CC1CC(=O)Nc1ccc(C)c(O)c1 C1(C)(CNC(CC2C(OC)COCC2)=O)CCN(C(=O)C(F)C(C)C)CC1 N1(C(C2CC(NC(COC)=O)C23CCC3)=O)CCCC(C)(C)CC1 C1(COC)(NC(C23CC(C2)C(C)O3)=O)CCCN(C(c2cc(C)ccc2Cl)=O)C1 CN(C)S(=O)(=O)N1CCC(C(=O)NC2CCC2NC(c2csnn2)=O)CC1 Nc1cc2c(cc1C(=O)NCC1CN(C(=O)CNC=O)CC13CCC3)CCC2 N1(C(C(CC)C#N)=O)CCCC(O)(CCNC(c2cnc(-c3ccsc3)s2)=O)C1 CC(C)C(F)(CNC(C1(CC2CC2)CC1)=O)C(=O)NCC1(CO)CC1 C1(NC(c2cn(C(C)C)nn2)=O)C2CCN(C(C3CC=CCC3)=O)C12 c1(OCC)ncc(CN2CCC(c3n[nH]cc3C(=O)O)C2)cn1 C(C)(c1ccc(OC)cc1)=CC(N1C(C)CC(NC(CCCC)=O)C1)=O N1(C(=O)C(C2CCCCC2)O)CC2CCCC2(CNC(C23CCC(CC2)C3)=O)C1 c1(OC)[nH]c(=N)nc2sc(C(=O)NC(C)C(C)NC(=O)C=Cc3ccco3)cc12 c1(CN2CC(NC(C3CCC4(CC3)OCCO4)=O)C2)ccc2ncccc2c1 N1(C(C(CC=C)CNC(=O)C(O)CC(C)C)=O)CCCC(C)(C#N)C1 c1(C(=O)NC(CC)CNC(C2(CF)COC2)=O)cscc1S(C)(=O)=O CC(C)CC(CN=c1[nH]nc(-c2ccsc2)s1)c1cccc(F)c1 c1(CN(c2nc(OC)c(F)cn2)C23CC(N)(C2)C3)cc(C)c(F)c(F)c1 c1(NC(CN2CCN(Cc3cc(C)[nH]c3C)CC2=O)=O)ncnc2scc(C)c12 N1(C(C(C)CO)=O)CCC(C(F)(F)F)C(NC(C2(C#N)CCCOC2)=O)C1 c1(C(=O)NCC2C(CNC(C(CC(C)C)O)=O)C2)cc2c(C(F)F)nn(C)c2s1 c1(C(N2CCCC(N(C)C(c3cnsc3)=O)CC2)=O)cc(F)c(F)cc1O C(=O)(C1CCCn2nccc21)NC(CCCC)CNC(=O)CCc1cc(Cl)cs1 c1(C(=O)NCCN(C(C23OCC(COC)(C2)C3)=O)C(C)C)cccc(N)c1O c1(C(c2n(CCCC)nnn2)NC(CCOC)c2ccco2)cncc(Br)c1C N1(C(CC2N(C)CCCC2)=O)CC2CCC1CN2C(=O)CS(N)(=O)=O CON(CCC(=O)N(C(C)CO)CCO)C(=O)CC1CCSC1 N1(C(=O)OC)CC2CC2(C(N2CC(CNC(=O)C(c3ccccc3)O)C2)=O)C1 C(=O)(C1=CCc2ccccc21)NCC=CCNC(C1(OC)CCC(C)C1)=O C(=O)(C(N=[N+]=[N-])C(C)C)N1CC(F)CC(N(CC(CC)(C)O)c2ccccc2)C1 CC(CC(=O)NC1CC2C1CCN2C(c1nncs1)=O)C(F)F c1(CC)cnoc1C(=O)NCC(C)C(=O)NC(c1ccnn1C)C C(=O)(CC(C)C(C)C)N1CC(C(=O)NCC(C#C)OC)(C(=O)OC)C1 N1(C(CN(C(C)=O)C)=O)CCC2(COC(CNC(c3ncc(Cl)cc3F)=O)C2)C1 N1(C(C(C2(C)CC2)NC(CCOCCC)=O)=O)CC(C2CC2(F)F)C1 C1(CNC(c2c(COC)ccs2)=O)(NC(c2cc(F)n(C)n2)=O)CCCCC1C c1(C(=O)NC(C2(O)CN(C(COCCC(C)C)=O)C2)C)ccc(=O)n(C(C)C)c1 C(=O)(CC(C)CNC(C1C=CCCC1)=O)NC(c1nc[nH]n1)C CCCC(CC)C(=O)NCC1(CC(N)=O)CCN(C(=O)CC2CC(SC)C2)CC1 C(=O)(C(F)C1=CCCCC1)NC1CC(NC(C(C)N(C)C)=O)C12CCC2 c1(C(=O)NC(C2N(C(CS(CCC)(=O)=O)=O)CCC2)C)ccc2oc(=O)oc2c1 c1(C(N(CCCCCNC(C(CC)CC)=O)C)=O)ccc(F)c(S(C)(=O)=O)c1 C1(C(=O)NC(c2ccc(Br)cc2)CC)CC(O)CN1C(c1cc(Br)cs1)=O Cc1ccc(NCc2nncn2C)cc1.C1CCCC(=O)N2CCCC(C2)CO1 c1(OC)c(NCc2nnnn2-c2ccc(F)cc2F)cccc1Cl CCC(C)CCC(=O)NC1CN(C(=O)Cc2cnn(C(C)C)c2)CC1C Nc1nccnc1C(=O)NCC(CC1CC1)C(=O)NC1CCN(C(N)=O)C1 c1(-c2nc(COC)nn2C2CCCC(C)C2)cc(C)ccc1Cl C12(Cc3cn(C(COCC)C(=O)NCc4nc(Cl)cs4)nn3)CCC(CC1)CC2 N1(C(CC=CC)=O)CCOCC1CNC(c1n[nH]cc1OC)=O C1(O)(CCNC(C2CCC(=O)C2)=O)CCCN(C(C2(c3cc[nH]n3)CC2)=O)C1 Cc1nc(CC(=O)NCC23CC2CN(C(=O)CCc2cncs2)C3)c(C)s1 N1(C(CCC)=O)CCCCCC1CNC(C1CCC(CCC)CC1)=O c1(C(N(CC(C)C(=O)O)C)=O)ccc(-c2cncc(F)n2)cn1 c1(C(N2CC(CC=C)(NC(=O)C3=CCC(C)CC3)C2)=O)cnc2n1C(C)CCC2 C(=O)(C(F)CCC(C)C)N1CC(CC(=O)NCC)OCC1 C1(NC(CC=CCC)=O)C(C)CN(C(c2cccc3cnsc23)=O)CC1C C(C(C)(C(=O)N1CC2C(NC(=O)Cn3cnnc3C)C2C1)OC)OC c1(C(=O)NC23CC(NC(C(C(=O)OC)C)=O)(C2)C3)cccc2c1COCC2 C(CCc1ccccc1)(C(=O)O)SC.n12cc(cn1)CCNCC2 c1(C(=O)NCC(CC)NC(=O)Cc2ccoc2)cc(C(N)=O)cn1C N#Cc1cc(F)c(NCC2CCCN2C(=O)CCc2cnc[nH]2)c([N+](=O)[O-])c1 c1(C(N(C)CCN(C)C(C2CC=CCC2)=O)=O)cc(F)ccc1F CCCC(O)CC(=O)N1CC(NC(C23CC(CC(F)F)(C2)C3)=O)CCC1C CC(C)C(C(=O)N1CCC(C(=O)NCC2CNC(=O)C2)O1)NC(N)=O C1(C(=O)OC2CCOCC2)CCN(c2ccccc2Br)C1=O N1(C(c2noc(CC)c2C)=O)CCC(CNC(C2CCN2CC)=O)C(C)C1 C1(NC(CC(C)(C)OC)=O)CCC(O)CN(C(=O)CC2COCCO2)C1 CC(C)C(C#N)C(=O)NCC1(NC(c2ccc(OCC(N)=O)cc2)=O)CCCC1 c1(C(=O)OC)ccc(CC(=O)NCC2CCC2NC(C2CC3CC2C3)=O)cc1 N1(C(C2CCC(C#C)CC2)=O)CC2CCC1CN2C(=O)CC1CCCO1 c1(CCCNC(=O)NC(C2CCOC2)CC2CC2)csnc1Cl N#Cc1c[nH]c2cc(C(N3CCc4ccccc4C3)=O)ccc12.C1(=O)CCO1 N1(C(CCCCCN(C(C(C)c2ccco2)=O)C)=O)CCOCC(C)(C)C1 N1(C(Cc2cc(C)nn2C)=O)CCC2CN(C(=O)C(C)CC3CC3)CCC12 Cc1ccc(F)cc1C(C)NC(c1cc(-c2ccccn2)on1)=O c1(C(=O)NC2CN(C(C(CC)O)=O)CC2(C)C)c[nH]c2cc(F)c(F)cc12 c1(C2C(NC(C(N3CCC(C(C(=O)OCC)F)C3)=O)=O)C2)ccc(F)c(Cl)c1 C1(CC)CC(NC(=O)NC2CC(=O)N(c3ccc(OC)cc3)C2)CCO1 C1(C)(C(=O)NCCN(C(=O)CCCc2ccsc2)C(C)C)CC1(F)Cl N1(C(CCc2cccc(C#C)c2)=O)CC(NC(c2csc(Cl)n2)=O)C2CCCC12 N1(C(COCCOC)=O)CCN(C)CC1CNC(C1CCCCCN1C)=O c1(C(N(CCN(C)Cc2cn(CC)nc2)C)=O)cn(C(C)(C)C)nc1C c1(OC)ccc(C)c(C(N2CCC(C)N(C(=O)C(O)CSC)CC2)=O)c1N C1(NC(c2cn(C)[nH]c2=N)=O)C2CCCN(C(c3csnn3)=O)C2C1(C)C c1(C(N2CCN(C(c3c(O)ccc(Cl)c3F)=O)CC2)=O)cnc2ccccc2c1 c1(CC)ccc(-n2ccc(-c3cccc(C4(C#N)CC4)c3)n2)cc1 Cc1ccccc1C=CC(N1CC(CNC(c2cnn[nH]2)=O)C2CC12)=O N1(C(C(c2cccc(Cl)c2)C)=O)CC2C(NC(=O)CC3(CN(C)C)CCC3)C2C1 Cc1c(C(N2CCOCC2CCNC(=O)C=CC2CC2)=O)cc(C2CC2)n1C C12(CC(N3C(C4(NC(=O)Cc5cc[nH]n5)CC4)CCC3)=O)COCC(C1)C2 C1(C)(CC(=O)NCCSCC(C)C)CCN(C(c2ncnn2C)=O)C1 C1(NC(c2c(OC)cncc2)=O)CN(C(c2cccc(=O)o2)=O)CCC1(C)C CCCCN=C(NCC(=O)NCC1CC1)NCC1(C)CCC(=O)N1 C#Cc1ccc(C(=O)NCCN(C)C2CC2)cc1C.c12ccnc(c1)NC2=O c1(N2CCC(C(C)NC(=O)CCN3CCCC3=O)C2)nc2ccc(Br)cc2o1 Cc1c(C(=O)NC(CNC(c2cc([N+](=O)[O-])n[nH]2)=O)CO)sc2ccc(F)cc12 Cc1cc(C(=O)NC(C)C(CO)NC(=O)CC2CC2)c(C)n1-c1ncccn1 C1(NC(COCC(C)C)=O)CN(C(c2ncsc2Br)=O)CC1C N1(C(C(C2CC2)OCC)=O)CCC1CC(=O)NCCNC(=O)CO Cc1cn2cc(-c3ccccc3C(N3CCCC(C)C3)=O)cc2c(C)n1 C1(NC(c2c(C)csn2)=O)CC2CC1CN(C(=O)CN(CC(C)(C)C)C)C2 C1(CC(N2C(CNC(c3cc4ccoc4cn3)=O)CC2)=O)CCn2cncc2C1 c1(C(=O)NCC2CN(C(CCCSC)=O)CC2C)noc2cc(Br)ccc12 O(C1CCCc2ccccc21)CC(=O)NCC1C(C(=O)NC2(CC)CCCC2)C1 c1(N(CC)CC)nnc(C)n1CSc1ccccc1C CON1CCC(C(=O)NCC2CC(C)N(C(=O)C(N3CCOC3=O)C)C2)CC1 N1(C(C2ON=C(C)C2)=O)CCC2(CC1)CC(NC(C1CN(C(C)C)C1)=O)C2 O=C(CCC[N+](=O)[O-])NCC1CCCC1NC(c1cc(Cl)ccc1F)=O C1(OC)CCCC(CC(=O)NC(C2CN(C(=O)C(O)C(C)C)C2)C)C1 c1(NC(c2cccc(C3(CC)CCC3)c2)=O)ccc(OC)c(C#N)c1 C(=O)(C(C)CCCC(C)=O)NC1C(C(=O)NC(CCC=C)C)CCCC1 C1(CC(=O)NCC(CNC(C2CC(CC)(CC)C2)=O)O)NC(=O)CNC1=O Cc1cc(C(=O)NC2CN(C(C34CC5CC3C4C5O)=O)CC2C)cc(=O)n1C C1(NC(C(C)=CC)=O)CN(C(=O)C(C)Sc2ccc(C)cc2)CC2CC12 c1(CC)ccc(N)c(C(=O)NCC2(F)CCC(NC(=O)C(C)n3cccn3)C2)c1 N1(C(C(=O)N2CCCC2)=O)CC2(C1)CN(C(C1CC(=C3CCC3)C1)=O)C2 CC(C)CCC(C(=O)N1CCC(C)(C(N)=O)C1)NC(=O)C(=O)CC(C)C N1(CC(=O)NC2CN(C(C(C3CCC(=O)N3)C)=O)CC2C)C(=O)C(C)C(C)C1=O C(=O)(C1=CCCCCC1)NC(C(=O)N1CC(CCC)OCC1)CCCOC N1(C(C(COCC)n2cc(CC(C)O)nn2)=O)CCC(c2ccsc2)CC1 C1(C(N(CCNC(Cc2cc(C)ns2)=O)C(C)C)=O)C(F)(F)C12CCC2 C1(COC)(CNC(=O)CC(C)SC)CN(C(=O)CCCN(C)C(C)=O)C1 c1(CC(=O)NCC(=C2CN(C(CC(C)C3CCCO3)=O)C2)F)ccc(F)cc1F N1(C(c2nc(CC)sc2)=O)CCC(O)(C(C)CNC(c2cnc(Cl)[nH]2)=O)C1 c1(NC(C(N2CCS(=O)CC(C)C2)c2nc(C)[nH]n2)=O)ccc2c(c1)OCO2 N1(C(c2nn(CC)c(C(F)(F)F)c2)=O)CC2(CCCN(C(=O)C(F)CC)C2)C1 c1(CCNC(c2coc(CNC(C3CCC4CC34)=O)c2)=O)cccc(F)c1 C(CCC(O)CO)NC(C1C=CCN(C(C2COCCO2)=O)C1)=O C(CCC(C(=O)N1CC2CC1CN2C(C)C)NC(=O)CCc1cnn[nH]1)OC N1(C(C2CC(C(=O)OC)C2)=O)CCCCC1CN(C)C(C1COCCO1)=O c1(CNC(C2C(CC)C2)=O)ccc2c(c1)CCN(C(c1c(C)cncc1F)=O)C2 CN1CC(C(=O)N2CCC2CNC(=O)Cc2ccn(C)n2)c2ccccc2C1=O C1(CC)CN(C(C)=O)CCC1NC(c1conc1CSc1ccccc1)=O N1(C(C2CCC(CC)CC2)=O)CC2=C(C1)CN(C(=O)COc1cccc(N)c1)C2 C=CCCC(F)(F)C(=O)N1CC2CCC2(CCNC(c2ccc(Cl)cc2)=O)C1 C12(CNC(C(CNC(C)=O)(C)C)=O)CC(CO1)N(c1nccnc1F)C2 C(=O)(CC(CNC(=O)CC1CCC(=O)C1)C1CCC1)N(C(C)C(=O)OC)CC Cc1oc(C(=O)NC2CCCC23CCN(C(c2cscn2)=O)C3)cc1S(N)(=O)=O C1(NC(Cc2c(CC)noc2CC)=O)CC(C)N(C(c2cc(C)[nH]n2)=O)C1 N1(c2ccc(NC(c3ccco3)=O)nn2)CCCC(O)(C2CC2)C1 C1(NC(C2(CC)CC(C)(C)C2)=O)CC2(C1)CN(C(=O)C(C(C)C)NC(N)=O)C2 C1(CC(N2C(C)(C(=O)OCC)CC2)=O)CCCCN1C(C1CCC2CC12)=O c1(CCC)cc(=NCCCCC(C)NC(=O)C2=Cc3ccccc3OC2)[nH]c(Cl)n1 N1(C(CCCOC(C)=O)=O)CC(F)CC1CNC(C1CC(C)(F)C1)=O CC1(C)CC(C(=O)NCC2CC3(C2)CC(O)C3)CN(C(=O)C(C)(C)N(C)C)C1 Cn1ncc(C(=O)NC(CC(N)=O)C(=O)NCCCC2C=NNC2=O)c1C#N c1(CC)cc[nH]c1C(=O)NC(C(=O)NCC(O)CCOC)c1cccs1 C1(C(=O)NCc2nnc(C)o2)CCN(C(c2cnc(Cl)n2C)=O)CC1O C1(C(N2CCC(CNC(C(C)(C)C(F)F)=O)C2)=O)CC(c2ccncc2)=NO1 C1(C(N2CCC(C(N3C(C#C)CCC3)=O)(C(C)C)C2)=O)CCC2(CC1)CC2 CCC(CC)CCC(=O)NCC(C1CC1)NC(c1ccc(F)c(F)c1N)=O C1(CN(C(CC2(OC)CCC2)=O)C)CCCN1C(c1cc(CC2CC2)on1)=O C1(N(C(c2cc(Cl)on2)=O)CC)CCCN(C(=O)C(c2ccncc2C)C)CC1 c1(OC)cccc2c1CN(C(=O)CC1CC(Cc3cccc(Br)c3)C1)C2 C1(CNC(CN(C(C)C)C)=O)CC(C)N(C(=O)Cc2ccccc2O)C1 c1(C(=O)NC23CC(C(N4CC(N5CCC(O)CC5)C4)=O)(C2)C3)ccc(Br)cc1F C1(C(=O)NCC2(C)CCCN2C(=O)CCCC2CCC2)CC2CCCCN2C1 C(=O)(C1=C2CCCN=C2NN1)NC1C(NC(C(C(CC)CC)OC)=O)COC1 Cc1cc(C(N2CCOCC2)=O)ccc1NCc1ncc(C(C)(C)C)o1 C1(C(=O)NCC(CC)O)(CC)CCN(C(=O)C=Cc2cc[nH]n2)C1 O=C1CC(C(=O)NC2CC(c3ccccc3)(CNC(=O)COC(F)(F)F)C2)CN1 C(CNC(=O)C=CC(=O)NC1CC1)(CC(=O)N1CCSCC1C1CC1)OC C1(O)(CC#C)CC(C(=O)NC(C)CCCNC(=O)C(CC)SC)C1 Cc1cccc2c1CC(C(=O)N(C(C)CNC(C1CCSC1)=O)C)N2 n1(C(CC(=O)NC(CN(C(c2ccc(CC)o2)=O)C)(C)C)C)nc(C)cc1C c1(C(=O)NCC2(O)CCCN(C(C(C=CC)O)=O)C2)cc2c(F)cc(F)cc2[nH]1 N1(C(C(F)=CC)=O)CC2CCCC2(NC(c2cc(=O)n(-c3ccccc3)[nH]2)=O)C1 N1(C(=O)CCC2(O)CCC2)CCCCC(C(=O)NC2(c3cccnc3Cl)CC2)C1 c1(C(N2C(CNC(c3csc(Br)n3)=O)CCCC2)=O)nc2ccccc2[nH]1 C1(C(=O)NCC(CCOC)NC(=O)C2=CCCC2(C)C)CCCN2CCCCC12 c1(CC(N2CC(CC=C)(NC(=O)C(O)C3CCCC3)C2)=O)c[nH]c2ccccc12 C1(CC)CN(C(=O)CCC#N)CCN1C(C1CC=CC1)=O CN=c1cc(C(=O)NC2(CN(C)C(C3(C4CCCO4)CCC3)=O)CC2)cc[nH]1 N1(C(c2cn(CC)nn2)=O)CC(C2CC2)(C(=O)N(C2CCOC(C)C2)C)C1 c1(C(N2C(C)CCC(NC(=O)CCc3ccncn3)C2)=O)cc2ccccc2[nH]1 CN1CCCCC(CNC(c2nocc2CNC(=O)CC2(C)CCOCC2)=O)C1 N1(C(CCC(C)SC)=O)CCCCC(NC(=O)CC2CCOC2)C1 C1(C(N=c2cnn(C)[nH]2)=O)COCCC12CN(C(=O)NC(c1ccccc1)=O)C2 c1(C(C(N2CCC(NC(c3c(C)cns3)=O)C2)=O)O)ccc(OC(C)C)cc1 S(=O)(=O)(c1cccs1)NCCC(=O)NC(CNC(C=C(C)C(C)(C)C)=O)C C1(NC(=O)CCc2nncs2)CC(F)CN(C(c2sccc2SC(F)F)=O)C1 N1(C(CCCOC)=O)CCCC(F)(CNC(=O)C(c2ccc(F)c(F)c2)C)C1 c1(C(=O)NC2C(NC(C3C(OC)(OC)C3)=O)CCCC2)cnn2cccc(Cl)c12 c1(C(=O)NCC2(CNC(C(C3CC3)SC)=O)CCC2)cnn(CC(C)C)c1 CN1C(=O)CCC(C(N2CC(NC(c3ccc(Cl)s3)=O)C2)=O)C1c1ccccc1 Cc1c(Cl)c(C(=O)NC2CCCC2Cc2ccccc2)cn1C(C)C N1(C(CCSC)=O)CCC2(CC1)OCCC2NC(=O)Cc1ncnc2sccc12 c1(C(=O)NCC2CN(C(CCC#CC)=O)C(C)(C)C2)cccc2nccn12 C1(F)(C(=O)OCC)CCCN(C)C1.C(C1C(=O)N1)OCC N1(C(C(C)(C(C)C)OC)=O)CC2(CCC(NC(=O)Cc3cnccc3C)CC2)C1 c1(C(N(C2CCN(C(c3nnn4c3CSCC4)=O)C2)C)=O)cc2ncccn2n1 C1(NC(C2(CC)CCOC2)=O)(CNC(c2ncn(C)n2)=O)CCCCC1 c1(NCC(C(=O)NC)(C)C)nc2ccccc2nc1NCc1ccc(Br)c(C)c1 C1(CC(=O)NCC2CN(C(c3cn(CC)nc3)=O)CC2C)OCCCC1(C)C C(=O)(C(F)CCC(C)C)NCCN(C(c1c(C)nc(CC)o1)=O)C CCC(C)C(O)C(C)C(=O)NCc1cc[nH]c1C(N1CC(C)(C(F)(F)F)C1)=O N(C1CN(C(=O)C2=COCCO2)Cc2ccccc21)C(c1ccnn1CCF)=O c1(C(=O)NCC(CNC(C2(C)N(C(C)=O)CCC2)=O)C)cnn2c1CCCC2 CC1CC(CN(C(=O)CCCCNC(C2CC(O)C2)=O)C)CC(C)O1 C12(C(N3CCC4(CN(C(C(CC)CO)=O)C4)C3)=O)CCCCC(=O)N1CCC2 C(=O)(CC(C(F)F)c1ccccc1)N(C1(CC(=O)NCc2c(C)n[nH]c2C)CC1)C Cc1c(C(N2CCN(C(=O)C(C(C)O)N(C)C)CCC2C)=O)ccc2c1CCC2 CC1CN(C(=O)CC(O)C2CCCC2)CCC1NC(C1(S(C)(=O)=O)CC1)=O CC1(C)OCC(CN=C(NCc2ccc(CN3CCOCC3)s2)NC2CC2)C1O N1(C(c2c(C)[nH]nc2C(C)C)=O)CC2(CCN2C(c2cc(F)n(C)n2)=O)C1 N1(C(CCc2c(C)nccc2)=O)CCCCC(CNC(C2(S(N)(=O)=O)CC2)=O)C1 C1(NC(C(C2CC2)OC)=O)CN(C(C2CCC3CC3C2)=O)CC1C c1(C(=O)NC2C(NC(c3cnc(COC)s3)=O)CC2)c(C)ncc2ccccc12 C1(C(=O)NC(CSCC)C(=O)NC2CC(C)OC2=O)C2CCC(F)(F)C12 C(=O)(C#CC(C)(C)COC(c1ccc(C)cc1F)=O)N(C(c1ccccn1)=O)C1CC1 c1(NC)ccc(C)cc1C(=O)NCCc1cn(C2CCC2)nn1 Cc1c(NC(=O)NCCC(C)c2cn[nH]c2)ccn1CCO N1(C(CN(C)C2CC2)=O)CCOCC(NC(=O)CNC(C2CCC2)=O)C1 c1(C(N2C(C(N(C)Cc3ccc(Br)o3)=O)CC2)=O)cccc(Cl)c1O N1(C(N(CC)CC)=O)CC2(C1)CN(C(=O)NCCN(C)C)C2 c1(C(=O)NCC(C)N(C(C(C2CCCC2)OCC)=O)C)cc(Cl)sc1NC(C)=O Cc1cc2c(C(N3CCN(C(=O)C(CO)C(C)(C)C)C(C)C3)=O)cccc2[nH]1 N1(C(c2cn(CC)nn2)=O)CCCC(F)(CNC(=O)C=C2CCN(C)C2)C1 C(C(O)CCC(F)(F)F)NC(C1C(CC(C)(C)C)CN(C(=O)OC(C)(C)C)C1)=O c1(SCC)cncc(C(=O)NC(C)C(C(C)C)NC(=O)C(C)(C)c2cccs2)n1 N1(CCC(=O)NC2C(c3ccc(OC)cc3)C2)C(=O)c2ccc(Br)cc2C1=O c1(C(C)C(=O)NCCCCNC(C2CC2C(C)(F)F)=O)cccc(Br)n1 C(=O)(C(C(C)NC(C12CSCC1C2)=O)C(C)C)NCc1c(C)ocn1 c1(C(=O)NCC(C)N(C(CC(CC=C)(C)C)=O)C)cc2cccc(C)c2s1 N1(C(CCNC(CC(C)C)=O)=O)CCCCC(C(=O)NCC(Cl)=CCl)C1 N1(C(C(c2ccccc2)N(C)CC)=O)CC(O)(CNC(C2CCC(C)O2)=O)C1 c1(NC(C2(c3ccc(Cl)cc3)CC(C)C2)=O)cccc(C(C)(F)F)n1 c1(C(N2CCC(NC(C34COCC3C4)=O)C(O)C2)=O)cccc2sccc12 N1(C(C(CC)(C)C)=O)CC2CC1CN2C(=O)CNS(=O)(=O)N(C)C CCCCC(C)C(=O)N(CC(C)NC(=O)CC1CC2CCC1CC2)CC C1(C(N(C)Cc2cc(C(C)C)no2)=O)C2CCC(C2)N1C(C1CC(N)C(O)C1)=O c1(C(=O)NCC2C3N(C(CC4(OC)CC4)=O)C(CC3)C2)cccc2oncc12 N1(C(C2C(CC)C2)=O)CCCCC12CC(NC(c1ccnn1C1CC1(F)F)=O)C2 c1(CCC)nc(C(=O)NCc2ccc(C(=O)NC(CC)C(N)=O)s2)co1 CC1CCN(C(C(=O)NCC(F)CNC(c2nc(=O)n(C)[nH]2)=O)C(C)C)CC1 N1(C(C2(COC)CCOC2)=O)CCC(CC(C)NC(=O)CC=C(Cl)Cl)CC1 c1(-n2c(C)ncc2)ccc(C(=O)NCCNC(c2cnc(Cl)[nH]2)=O)cn1 N1(C(C2CC(C)(CC)C2)=O)CC2CC2(CNC(c2cc(C)c(C)[nH]2)=O)C1 Cc1nc(F)ccc1CNC(C1COCCN1C(=O)C(C)C#N)=O Cc1cc(NC(C2CN(C(=O)C(O)CN(C)C)CC23CC3)=O)c(C)cc1F c1(C(N2C3CC(CNC(C4CC=CC4)=O)C2CC3)=O)ccn2cccc2c1 N1(C(C2CC(C)(C)OCC2)=O)CCC2C(C1)CN2C(=O)Cc1cccc(F)c1O N1(C(C2C(C(=O)OC)C2)=O)CC(=O)NCC1C(N1CC(C(C)OC)C1)=O C(=O)(C(C)(C)C1=CCN(C(C2CCC(C3CC3)C2)=O)C1)NC N1(C(CC(CCC)C)=O)CC(CNC(=O)Cc2ccnn2C)OC2(CCC2)C1 Cn1cc([N+](=O)[O-])c(S(=O)(=O)N(CCCO)C2CCC2)n1 c1(C(N2C(C(=O)NC(C(C)F)C)CCCCC2)=O)ccc2[nH]nc(Cl)c2c1 N1(C(C(C(C)O)N(C)C)=O)CC2=C(C1)CN(C(c1ccc(N)cc1Cl)=O)C2 Cc1cnc2n1CCC(C(=O)NCCC1=CCCCC1)C2 Cc1cc(Cl)cc(C(N2CCOC(CN(C)C(C3(C)CCOCC3)=O)C2)=O)c1N CC1(C)NC(=O)C2N(C(=O)COCC3CCCOC3)CC12 C1(C2(O)CCN(C(=O)C3=CCCCC3)CC2)(N(C(=O)CCCCCF)C2CCC2)CC1 N1(C(C)=O)CCC2CC(NC(=O)COCC(F)F)CCC2C1 C1(NC(CC2(OC)CC2)=O)(CNC(=O)CC2CC(C)(C)CO2)CCCCCC1 C(=O)(C1=CC2(CCN(C(=O)C=C3CCC3)C2)C1)N1CC(C)(C)C(CO)C1 C1(CC(=O)NC(c2ccccc2)CO)COCC1NC(=O)C(O)C1CCC1 N1(C(c2[nH]ccc2-c2cccs2)=O)CC2CC1CN2C(C12CCCC(C1)OC2)=O N1(C(c2c(C)cc(Cl)c(F)c2)=O)CCC2C1CCCN2C(c1conc1C)=O C1(CC(=O)Nc2ccn(CCC)n2)CC(C)(C)CN1C(C1CCOC1)=O Cc1nn(C)c2ncc(C(=O)NCC(C)(C3CC3)NC(=O)CC3(C)CCC3)cc12 N1(CCOCCCOCC(=O)NCCN(C(C2C(CC)C2)=O)C)CCCC1 N1(C(C2(C#C)CCC2)=O)CC2CCN(C(=O)C(C)CC(F)(F)F)C(C2)C1 C1(c2cn(C(C)CNC(c3cc(CN(C)C)on3)=O)nn2)CCC(=O)CC1 N1(C(C2C(Cl)(C(=O)OCC)C2)=O)CC2CC(NC(=O)Cc3csc(CC)n3)C2C1 CCCCC(O)CCC(=O)NC(C1CCN(C(=O)CCn2nc(C)cc2C)C1)C C1(C)NC(=O)NC1=O.c12ccn(c1)c(=O)n2C.C(=O)(CCCOC(C)=O)NCCN C1(Cc2ccc(OC)c(OC)c2)CN(C(=O)Cc2nn[nH]n2)CC(C)O1 N1(C(C(c2ccccc2)C)=O)C(NC(=O)Nc2nnc(O)s2)CC1C NC(Cc1ccccc1)CCC(=O)N1CCCC(OCC2CCCO2)C1 C1(C(N(CCC(=O)NC2CN(CCC)C(=O)C2)C)=O)CCC2(CCC2)C1 CCCC(CCC)CC(=O)NCC(C)(C)CNC(=O)C1=CCCC1C N1(C(=O)CC2COCC2O)CCN(C(c2cc(C(F)F)cs2)=O)C(CO)C1 C1(NC(c2c(C)scn2)=O)CN(C(c2cc(Cl)ccc2F)=O)CC1N=[N+]=[N-] c1(C(=O)NC2C3N(C(c4cnn(C)c4N)=O)C(CC3)C2)cc2c(=O)[nH]ccn2n1 N1(C(=O)C(F)=C2CCC2)CCCCC1C1CCCN1Cc1ccoc1Br c1(C(N2C3(CNC(CC4C(C)=NOC4=O)=O)CC(C2)C3)=O)ccc(F)c(C)c1N C1(NC(c2cc(C(N)=O)[nH]c2)=O)CCCCC1CNC(=O)C(=O)Nc1ncc[nH]1 Cc1ccc(NC(=O)C(O)CNC(=O)CCC(C)CN(C)C)c(Cl)c1 CC(CC(N)=O)C(=O)NCC12CC(CO1)N(C(=O)CCN1CCC(C)CC1)C2 C1(CNC(=O)Cn2nnc(C(F)(F)F)n2)CCCN(C(=O)C2=CCC2)C1 N1(C(CCn2cc(C(C)N(C)C)nn2)=O)CCC(C(N2CCSCC2)=O)CC1 C1(NC(C(C)n2cnnn2)=O)CN(C(c2cc(C#N)ccc2O)=O)CC2(CC2)C1 C1(CC=C)(C(=O)NCC2CCCN2C(N)=O)CCN(C(=O)C(C2CC2)OC)C1 c1(C(N2CC(C)C(CNC(c3ccc(Cl)cn3)=O)CC2)=O)cccc2ccoc12 c1(C(=O)NCC(C)(C2CCC2)NC(CSCCOC)=O)coc2c1C(=O)CCC2 Cc1c(N2CCCC(C#N)C2)ncnc1N1CCC(CN(C)C)C1 c1(NC(CC2C(C)CCCC2)=O)cnc2ccc(C(F)(F)F)cn12 Nc1cccc(C(F)F)c1C(N1CC=CC(NC(C2CCCC3(CC3)C2)=O)C1)=O C1(C2CCCO2)(C(=O)NCCCNC(c2ccc3sccc3c2)=O)CCCO1 C1(C(N2CCC(CCNC(C(CC#C)(C)C)=O)C2)=O)CCOC2(CCCCC2)C1 c1(CNc2c(C(=O)NCCC3CCCCCC3)n[nH]c2)cccc(Br)c1[N+](=O)[O-] c1(CNC(c2n(CCOCC)nnn2)c2cc(CC)cs2)cnc(F)c(C)c1 N1(C(CN(C(C)=O)C)=O)CCC(C)(C)C1CNC(=O)Cc1c(Br)cnn1C N1(C(c2c(Br)ccc(C)n2)=O)CCC2(C1)CN(c1ccn3nccc3n1)C2 C#CCC(CC#C)C(=O)NC1CCOCC1NC(c1cccc(CC)c1O)=O N1(C(C)C(=O)O)CCC(O)C(CNC(c2c(Br)c(C)nn2-c2ccccc2)=O)C1 C1(C(C)NC(C2(CO)CCOC2)=O)CCN(C(C2CCC(=O)O2)=O)CC1 c1(C(=O)NC2(CN(C(C(C)SC(F)(F)F)=O)C)CC2)csc([N+](=O)[O-])c1 c1(C(=O)NC2COCC2NC(C2CC23CCOCC3)=O)cc2ccccc2s1 N1(C(C2CC(C(C)C)C2)=O)CCCC1C(c1ccccc1)=O c1(C(=O)COC(C2CC23CCOC3)=O)ncc(F)cc1F c1(C(N2CC(CNC(C3(C)N(C)CC(OC)C3)=O)C2)=O)ncc2cc(Cl)ccn12 C(=O)(C(C)(O)C(C)(O)C(=O)O)Nc1cn(C)c(=O)cc1 n1(CC(C)Nc2cccc(Cl)c2C#N)ccc2cc(Cl)ccc12 C1(C(C)CC2CC2)C(=O)Nc2cccc(c2)N1C1CC1.C(CCOCC)NCC C[S+](C)CCC(O)C(=O)N1CCN(C(=O)CC(C)(C)C)CCC1C C(C(C)(CC)CC)NC(C(C1(O)CN(C(C(CC)N(CC)CC)=O)C1)(C)C)=O CCC(C)CC(C(=O)N1CCC(C(=O)N(C)C)C1)NC(=O)Cc1cccnc1 C1(C(N2CC(N(C)C(c3csc(-c4ccoc4)n3)=O)C2)=O)CCCCC1(F)F Cc1nc(-c2cc[nH]n2)sc1CC(=O)NCCC1(C)CC1(F)F C1(C)(CNC(CN(C)C2CC2)=O)CN(C(=O)CCN2CCC(C(N)=O)CC2)CCO1 N1(C(C2(CC)CCC2)=O)CC2CCN(C(c3cc(C(F)F)ccn3)=O)C2C1 N1(C(C(C=C)C)=O)CCOC(C(=O)Nc2c(CC)noc2C)CC1 C#CC1CN(C(c2csc(O)n2)=O)CCN1C(C1CCN1C1CCCC1)=O C(N=c1[nH]cnc(I)c1Cl)c1cnc(CN(C)C)n1C N1(C(C2N(N=O)CCCC2)=O)CCCC2(NC(=O)CN3CCOCC3)CCCC12 C1(C(N2C(CCNC(CC3(C)CCCC3)=O)COCC2)=O)Cc2ccccc2O1 Cn1c(CCC(=O)NC(C)(C)CC(=O)NCCn2ccnc2)nnc1S CCS(=O)(=O)c1cccc(CC(=O)NC(CNC(C2CCO2)=O)C(C)(C)C)c1 C1(CNC(c2cn(-c3ccccc3)nn2)CO)CCCC12CC2 C1(NC(CC(C=C)C)=O)CN(C(c2cccc(=O)n2C)=O)C2(CCC2)C1 C1(C(=O)NCCCn2cc(-c3cncc(OC(C)C)c3)nn2)CC2CC1CC2O N1(C(C(c2ccccc2)SC)=O)CCC(CO)(NC(c2nocc2Cl)=O)C1 c1(OC)ccc(C(=O)NC(C)CNC(C2(O)CC2(C)C)=O)c2cnccc12 C1(C(=O)NCCCC(C)=O)C2CC2CN1C(=O)CN1CCCC1=O c1(C(F)(F)F)ccc(-c2nc(-c3cccnc3OCC3CC3)no2)cc1 CC1CCN(C(=O)CC(O)CN(C)C)CC1CNC(C1(C)COC(=O)OC1)=O C1(NC(C2OCC(C)C2)=O)C2CC1N(C(c1ccc(CS(C)(=O)=O)o1)=O)C2 N1(C(C(=O)NC2C(C)(CO)CC2)=O)CCC(c2ccccc2)C(O)C1 C1(=CC(=O)NC(C)C(F)(F)F)CCN(C(C2C=CC(=O)N=N2)=O)CC1 CC1CN(c2cc(C(C)(C)C)nc(Cl)n2)CCC1NC(=O)C=CCO Cc1cc(C(N2CCCC(NC(C3(CC#N)COC3)=O)C2)=O)cc(N)c1 CC(O)CC(=O)NCC1(C(=O)Nc2cc(-c3n[nH]c(=N)s3)no2)CC1 C1(CNC(c2ccccn2)=O)CCN(C(=O)CSCC(F)(F)F)C12CCC2 c1(C(N2CC(NC(c3n(CCOC)ncc3)=O)C2)=O)cnc2cc(OC)ccn12 C1(F)(C(=O)OC(C)(C)C)CCN(C(c2cccnc2Nc2cc(C(N)=O)[nH]n2)=O)C1 N1(C(C2(C)CCC(=O)N2)=O)CCCC2(CC(NC(c3ccoc3I)=O)C2)C1 N1(C(C(C)(C)C#N)=O)CCC(NC(c2cc(CO)[nH]n2)=O)C(F)C1 c1(CC)ccc([N+](=O)[O-])cc1C(C)NC(CCOC(C)=O)C(=O)O c1(C(=O)NCC2(OC)CN(C(c3csc(C)n3)=O)C2)cc2c(F)cccc2s1 c1(NC(=O)CC2CN(C(c3ccc(Br)cc3)=O)C2)cc(F)cc(F)c1Cl c1(NC(C#C)CCCC=C(C)C)ccc(C2CCCN2N=O)cc1 C1(NC(C2(OC)CC2)=O)CCCCN(C(=O)CC2(O)CCCN(C)C2)C1 C1(C2CCN(C(c3cncc([N+](=O)[O-])c3)=O)C2)(NC(c2coc(Cl)c2)=O)CC1 c1(C(N2C(C(C)NC(=O)C(C3CCOCC3)O)CCC2)=O)cnc(O)n(C)c1=O N1(C(C2C(C=C)CC2)=O)CC(F)(F)CC1CCNC(C1CC(O)C1)=O C(=O)(CCS(C)(=O)=O)NC(CN(C(C1CCCS1)=O)CC)C N1(C(C2C3CC(NC(c4c(CC)cc[nH]4)=O)C(C3)C2)=O)CCCC(N=[N+]=[N-])C1 N1(CCNC(=NCc2cnc(CCC)o2)NC(C)CC)c2ccccc2CC1C C(CC(C)(C)C(=O)NC1(C)CSC1)NC(C(CC1CCC1)OC)=O C1(N(C(C(C)(C2CCC2)OC)=O)C)COCC1(C)C.c12cc(on1)C(=O)NC2 CCC(C)CC(=O)NCCCN(C(C1CC2CC1C2)=O)Cc1ccccc1 c1(C(=O)NCC(C)(CC(C)C)NC(C2C(=C)CC2)=O)cnc2cc(C)ccn12 C1(NC(c2cc(C3(C)COC3)no2)=O)CCC(NC(=O)Cn2cncn2)CC1 C1(NC(CCN(C(CC)CC)C)=O)C2COCC1CN(C(=O)CCCC1CC1)C2 N1(C(c2nc(CC)oc2)=O)CC(CNC(=O)Cc2ccccc2Cl)C(C)(C)C1 N1(C(C=C(CC)C)=O)CCC(n2cccn2)C(NC(=O)CCSC)C1 C1(C(N(CC=C)CCC)=O)CC2CC2N1C(=O)Cc1cc(C)cs1 C1(C(C)=O)COCC1C(=O)N(CC(C)C(=O)N1CCC(n2ccnc2)C1)C N1(C(CS(C(C)C)(=O)=O)=O)CCC2(CCCC(CNC(c3ccns3)=O)O2)CC1 c1(OC)cc(Cl)ccc1C(=O)NCC#CCNC(C1CCCN1N=O)=O C1(CNC(c2ccc(C(N)=O)[nH]2)=O)CC2(CCN(C(=O)C=CBr)C2)CO1 c1(C(c2nccc(C(=O)OC)n2)C)c(Cl)ccc(C)c1N.C12CCCCC1N2 Cc1cc(Cl)ncc1CC(N1CC(N(C(=O)CCCn2c(O)nnc2O)C)C1)=O C12(CNC(C(CC)OCC)=O)CN(C(c3cnnn3C)=O)CC1CCO2 CC1C(NC(=O)C=Cc2cccc(F)c2)CC2CCC1N2C(=O)C1=CCCO1 C=CCC(C)(O)C(=O)NC1CCC(C)(CNC(=O)CCc2cccnc2)C1 N1(C(COCC#C)=O)CCN(C(=O)C(c2ccc(F)c(Cl)c2)C)CC1CO c1(C(C(=O)NCC(C)C)N(C(COC)C2(C)CC2)C)nscc1Br C1(N(C(C=C=C(C)C)=O)C)CN(C(=O)CCc2ccc(=N)[nH]c2)CCC1O CC1CC(NC(c2coc(C3CCC3)n2)=O)CN1C(c1ncn(C)n1)=O c1(OC)cncc(C(=O)NCC(n2cc(CC(OC)OC)nn2)C)n1 C(CC(C(C)(C)C)NC(c1nccnc1N)=O)N(C(C(CC)F)=O)C c1(OC)ncnc(C)c1NC(=O)CC1(C)CCN(C(=O)Cc2ncoc2C)C1 C1(NC(c2nc(C(C)C)sc2)=O)CCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1O n1(CCC)cncc1CNC(c1ccc(Cl)s1)c1nnnn1CC1CCCO1 N1(C(C2C(CCC)C2)=O)CCN(C(c2ccc(C#N)cc2F)=O)CC(CO)C1 C12(CNC(Cc3ccc(CCCC)cc3)=O)CCC(CC1)N(C(=O)C(C)(C)O)C2 Cc1c(C(=O)OCC(=O)CC(C)c2ccccc2)noc1C1CC1 N1(C(CC2N(C)CCCC2)=O)CCCC(F)(CNC(c2cc(CO)on2)=O)C1 N1(C(C(CCC)C)=O)CCN(C(c2nc(C)no2)=O)C(c2cn[nH]c2)C1 N1(C(CNC(=O)OC)=O)Cc2ccc(C(C)NC(c3sc(C)cc3C)=O)cc2C1 C1(CC(=O)NCCCC(C)NC(=O)CC2CCCNC(=O)C2)CCC2(CCC2)O1 N1(C(c2cccc(CF)c2)=O)CCCC1C1CCCN1C(c1ncncc1Cl)=O Cn1nc(C(=O)NCC(C2CCCCC2)NC(C2CC2(F)F)=O)cc1C1CC1 CC1=NNC(=O)C1CC(=O)NCCNC(=O)CC1CC=CCN1C CCC(CC)(CC)C(=O)N1CCOC(C(N2CCCCC(O)CC2)=O)CC1 C1(NC(Cc2nc(C)[nH]n2)=O)C2CC3CN(C(c4cc(O)cc(Cl)c4)=O)C1C3C2 N1(Cc2c(NC(C(CC)(C)O)=O)cccc2)CCCN(c2ccccc2)CC1C CCCCC(C(=O)NCc1cccc(Cl)c1)N1C(C)CCC1(C)C c1(NC2CCCN(C(c3occ(C)c3C)=O)CC2)cc(C#N)ccc1[N+](=O)[O-] C(c1ccc(C)cc1C)=CC(N1CC(CCNC(c2ncccn2)=O)(OC)C1)=O C1(OC)CCC2(C(=O)NCCC3(C)CCN(C(C4CC45CCC5)=O)C3)CC12 C(=O)(C(C)(C)CC1CCOCC1)NCC=CCNC(CCOC(CC(C)C)C)=O Cn1[nH]c(C(N2CC(NC(=O)CC3CC=CC3)C(CC(C)(C)C)C2)=O)nc1=O C1(O)(C(N(C(C)CNC(=O)CCC2CCOC2)C)=O)CCCC(C)(C)CC1 c1(CNC(c2c(C)cc[nH]2)=O)ncccc1CNC(c1ccc(F)cn1)=O Cc1nn(C)c2sc(C(=O)N(C3CCCC3)CCNC(=O)CC(C)CF)cc12 C1(C(=O)Nc2cc(C(F)(F)F)ccc2Br)CCC2(CN(S(=O)(=O)C(F)(F)F)C2)O1 C(=O)(C(C)(C)S(C)(=O)=O)N1CCC(CN(C(c2ccc(OC)s2)=O)C)C1 N1(C(C=C(C)C2CC2)=O)CCC(CNC(c2cc(C(N)=O)[nH]n2)=O)C1 Cc1cc(C)c(C(N2CCCC(C(C)NC(c3csc(C)c3C)=O)C2)=O)c(=O)o1 C1(CCC)CN(C(=O)Cc2cc(C)no2)CCN1C(=O)C(C(C)CC)N(C)C c1(C(=O)NC(c2cn(Cc3ccccc3Cl)nn2)COC)cc(=O)n(C)cn1 N1(C(c2c(C)cc(F)cn2)=O)CC2CCN(C(c3cc(N)nc(Cl)c3)=O)CC2C1 c1(OCCCC)ccc(C(N2CCN(C(c3ccsn3)=O)C(C)C2)=O)cc1OC C12(C(=O)NCC=C)CC(n3cc(CC(C)(C)CCN(C)C)nn3)C1C2 c1(SC)cc(C(=O)NCCCCCN(C)C(C23CC(C)C2C3)=O)oc1C C(CC(C)CCNC(C1CCCS1(=O)=O)=O)NC(CONC(=O)OC(C)(C)C)=O c1(CC(=O)NCC(CO)NC(C(C)OC)=O)nnc(S)n1C N(C(=S)N1CCCCC1)C1C(C(=O)O)OCCC1 C1(NC(C(C=C)c2ccccc2)=O)(CNC(C2CCC2C(N)=O)=O)CCOCC1 N1(c2cc(C)ncn2)CCC2(CCCC2C(=O)NCCOc2cccnc2)C1 C1(C(=O)NC2OCCN(C)C2)N(C(C2CCC3(CC3)C2)=O)CCCC1(C)C CC1(NC(=O)Cc2csc(-c3cccnc3)n2)CCCN(C(=O)C(O)C2CC2)C1 c1(NCC2(CNC(=O)OC(C)(C)C)CC2)cc(C2CC2)on1 c1(C(=O)NCC2(C(C)(C)C)CCN(C(CCC(C)OC)=O)C2)ccc(C)c(N)c1 C1(C(N(C2CCN(C(=O)Cc3cccnc3)C2)CC#C)=O)CCCC(=O)N1C c1(OC)cncc(C(N2CCC(CN(C)C(c3ccc(N)c(N)n3)=O)C2)=O)c1C c1(C(N(CCCNC(Cc2c(CC)con2)=O)C(C)C)=O)csc(C)c1N S(=O)(=O)(c1cc[nH]n1)NC(c1cc(C(C)=O)[nH]n1)=O C1(NC(CCOCCNC(c2c(CCC)nco2)=O)=O)CC(C)(OC)C1(C)C C12(CNC(CC(CN(C)C)O)=O)CC(CO1)N(C(=O)COCCCN(C)C)C2 c1(N(CCC)CC)ccc(C(=O)NC2CC2CNC(=O)CCc2ncnn2C)cn1 C(=O)(CC(C)CC(=O)N1CC(C(O)C(N2CC3(CCC(=O)N3)C2)=O)C1)OC c1(C(CNC(c2c(CC)ccs2)=O)NC(c2c[nH]cc2CC)=O)ccccc1F c1(C(N2CCOCC2CC(c2ccccc2)O)=O)ccc2c(c1)CCO2 CCC(C(=O)NC1(CCNC(=O)CCc2cnc(C)o2)CCCC1)C(C)(C)CC c1(NC(C(C)NC(=O)C(C)OCc2ccccc2)=O)ccc(Cl)cc1C(F)(F)F N1(C(=O)NCC(C(CC)C)CO)CCc2ccncc2C1C CC(CC(C)(C)C)C(=O)NCC1(NC(=O)CC2COCCO2)CCC(F)(F)CC1 C1(C(C)(C)NC(N)=O)CCN(C(=O)CSC2CCOC2=O)CC1.c12cn(nn1)C2 N1(C(c2c(C)c[nH]c2)=O)CCCCC(CNC(c2c(C)n[nH]c2C)=O)C1 N1(C(C(C(C)C)O)=O)CCCN(C(C23C4CC(CC24)C3(F)F)=O)C(C)C1 C1(NC(C(C)NC(N)=O)=O)CN(C(c2nc3ccccc3[nH]2)=O)CC1C1CC1 C12(CC(=O)NCCC(C)NC(=O)CCS(C)=O)CC3CC(C1)CC(F)(C3)C2 CC1CN(C(c2ccc([N+](=O)[O-])s2)=O)CCC1NC(C1(N(C)C)CCCCC1)=O C(=O)(CCCC(CC)CC)NC1C(NC(CC(CC=C)(C)C)=O)CCC1 C1(NC(=O)CCC2CCC2)CN(C(=O)CSCc2ccncc2)CCC12CCC2 C1(CC(=O)N(CCNC(C(c2ccccc2)OC(C)=O)=O)C)CCOC1(C)C Cc1cc(C)c(S(=O)(=O)N2CCc3[nH]nc(C(N4CNC(=O)C4)=O)c3C2)c(C)c1 c1(OC)cc(C)cnc1C(N1CC2(CC2)CC1CNC(=O)CCCCCF)=O c1(CN(CC(O)CO)Cc2ccc(-c3n(C)c(O)nn3)cc2)ccc(F)c(Br)c1 c1(C(N2C(CNC(CCOCC)=O)CC(F)(F)C2)=O)ccc(C#N)c(Cl)c1 N1(C(C(C)SCC)=O)CCC(NC(=O)Cn2nc(C(F)F)cc2C2CC2)C(F)C1 C(=O)(CC1=CCN(C(c2cnco2)=O)CC1)N1CCC(OC)CC1 c1(CC)c(C(=O)NCCC(O)CNC(c2nn(CC)cc2Cl)=O)cccc1F CCCCCCC(F)C(=O)N1CCC(CCNC(c2ccc(COC)s2)=O)CC1 Cc1ccc(C#N)cc1C(=O)Nc1cccc(Br)c1F c1(C(N)=O)cc(C(=O)NCC(F)CNC(c2cnc(N)cn2)=O)ccc1O Cc1cnc(-n2cc(C3CCN(C(C4(n5nccn5)CC4)=O)C3)nn2)s1 C1(C(=O)OCC)C=CCN(C2CCCSC2)C1 N1(C(c2n[nH]c(C)c2Cl)C(=O)NC(CC)C)CCOCC1(C)C N1(C(c2cc(C)n(C)c2)=O)CC2CCCC(N(C(=O)CN(C)C3CC3)C)C2C1 N1(C(C(c2ccccc2I)(C)N)=O)CC2(CCC2)C2COCC12 S(=O)(=O)(c1ccc(I)cc1Br)NC1C(OC)Cc2ccccc21 CC1ON=C(C(=O)NCCOCCCNC(c2cccc(=O)n2C)=O)C1C N1(C(c2c(C(CC)(C)C)cccc2)=O)CCN(C(c2cc(=O)n(C)o2)=O)C(C)C1 c1(OC)nc(C(N2CC(NC(=O)CN3CCCCC3=O)CC(O)C2)=O)ncc1F CC1CN(C(=O)Cn2nnc(=O)[nH]2)CC1NC(=O)Cc1cc(Cl)sc1Cl C1(C)(C(=O)NCC2C(C)CN(C(c3cc(Br)nn3C)=O)C2)CCC2CC2C1 C(=O)(C(C(C)C)NS(N)(=O)=O)NC(CN(C(c1c(OCC)scc1)=O)CC)C n1(CC)nc(C(=O)N(C2CCC(NC(=O)C(=O)NCC(F)(F)F)C2)C)cc1C N1(C(C(C)NC(CC)=O)=O)CCC2(CC1)CC(C)N(C(c1cc(F)n[nH]1)=O)C2 N1(C(c2nc(CC)sc2N)=O)CC2CCCC(C1)N2C(C1CCCC(C)(C)C1)=O c1(OC)ccc(C(F)F)cc1C(=O)N(C1CN(C(c2ccon2)=O)CC1F)C C1(O)(CN(C(=O)Cn2ccc(O)nc2=O)C)CCCN(C(C2CC=CCO2)=O)C1 c1(N(C(CCSC)C(=O)NC(C)(C)C)CC2CC2)ccc(Cl)c(C)c1 N1(C(C(=O)NC(C)C)=O)CCCC2(NC(=O)C(C)S(C)(=O)=O)CCCC12 O=C(C1CCCn2c(Br)cnc21)NC1C2CCC3C(C2)CC13 c1(C(=O)NCCN2CCN(C(c3nccc(C)c3)=O)CC2)cccc2occc12 C(=O)(C(C#N)C(C)(C)C)NC(C(=O)NCC1CCN(C(C)=O)C1)(C)CO c1(C(N(C(C(=O)N(C(CC)C)C)C2CC2)C)=O)csc(C)c1C c1(C(N2C(C)CC(NC(=O)C(C)(C)c3cnco3)C2)=O)ccc(C(N)=O)c(Cl)c1 C1(N(C(CCOCC)=O)C)CC2CCC(C1)N2C(c1sccc1S(C)(=O)=O)=O N1(C(c2n(CC=C)ccc2)=O)CCCC(C)(NC(C2(CC)CCCC2O)=O)C1 C1(CNC(C(C(C)O)NC(=O)OC)=O)COCCN(C(C2C(C)(C)C2(F)F)=O)C1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Br)NCCOCC(=O)NCC1CCC1 C(=O)(C(CO)C(C)(C)C)NC(C)C(C)NC(c1cccc(NC(C)C)c1)=O C1C(=O)N2CCC(O2)C(=O)O1.N1(C(CC)=O)CCCCC1COC CCCC(CNC(=O)CCOC(C)C)C(=O)Nc1cnc(Cl)nc1 C12(C(=O)NC(CC#C)CC#C)CCCC1CCN2C(C1CC(O)CN1C)=O c1(C(=O)NCC2(NC(CC3C(C)CCC3)=O)CCOCC2)ncnc2sccc12 N(C1CCOc2ccc([N+](=O)[O-])cc21)C(N1Cc2c([nH]c(=N)s2)CC1)=O c1(CC)nc(C(=O)NCC2C3CN(C(C4(SC)CCC4)=O)CC23)c(C)o1 C1(C)(C(=O)NC(CC)C(=O)Nc2cnc(OC)c(C)c2)NC(=O)NC1=O C(=O)(CC(C)C(C)(C)NC(C1CC12CCC2)=O)OC Cn1cc(Cl)c(CC(N2CC3CC3(NC(C3CC3(F)F)=O)C2)=O)n1 c1(NC(=O)OC(C)(C)C)ccc(CC(=O)N)cc1.C(C(F)(F)CC1CC1)NC(N)=O N1(C(CC(CC)C)=O)CCC(NC(C2CN(C)C2)=O)CC(C)(C)C1 N1(C(CCSCC(C)C)=O)CCC(NC(C2CCS2(=O)=O)=O)C(F)C1 N1(C(C(c2cncnc2)C)=O)CCC(CNC(c2ncoc2-c2ccccn2)=O)C1 C1(S(C)(=O)=O)(C(=O)Nc2c(C)[nH]nc2C(=O)O)CCC1 Cc1ccccc1-n1c(SCCCO)nnc1-c1nccn1C1CCC(N)C1 c1(-c2cn(CCNC(CCc3cncc(OC)c3)=O)nn2)ccc(C#N)c(F)c1 O=C(C1Cc2ccccc21)NC1CN(C(=O)CC(Cl)Cl)CC1O C(=O)(CCCC(F)(F)F)NC1CC(C(N2CCC(C(C)C)CC2)=O)C12CCC2 C1(CNC(C2CC(CC)C2)=O)CN(C)CCN1C(c1cc(Cl)n[nH]1)=O c1(C(N2CC(NC(C(CC)(C)OC)=O)C(CO)CC2)=O)cn2cccnc2n1 Cc1cc(CC(=O)NCC2(NC(C3COCC3(C)C)=O)CCCC2)ccc1O S(=O)(=O)(c1ccc(F)c(C(=O)O)c1)N1CC2C(CN(C(CC=CCC)=O)CC)(C2)C1 N1(C(C(C2CCCOC2)OCC)=O)CCC(NC(=O)CCc2cnoc2)CC1 C1(C#N)(C(=O)NCCCCC(C)NC(=O)C(C)(C)c2ccno2)CC2(CCC2)C1 N1(C(C(c2ccn(C)n2)C)=O)CC2CCN(C(C3CC4CC(=O)C3C4)=O)CC12 C1(CC#C)(C(N2CCC(C)(COC)C2)=O)CCN(C(=O)C=Cc2ccc(C)o2)C1 Cc1nc(NC(=O)CC2CCN(C(=O)Cc3cccnc3C)C2)sc1Cl c1(C(N2CC3CCN(C(=O)CCN4CCC4)CC32)=O)cc2ccc(Cl)cc2[nH]1 Cc1cc(O)n2ncc(CC(=O)NC3CCCN(C(C4(SC)CC4)=O)CC3)c2n1 N1(C(=O)OC(C)(C)C)CCCC(C(=O)NC(C)C(C)(C)c2ccccc2)C1CO CC1(NC(=NCC2CCCCC2)NC2CC(C)(F)C2)CCCOC1 c1(CC(=O)N(C)CC2(O)CCN(C(C(C)=C(CC)C)=O)C2)cc(F)ccc1F N(C)(C1CS(=O)(=O)c2ccccc21)C(c1cncc(OC)c1)C(=O)NCC(F)F C(=O)(C(C)(C)CCC#N)N(C1CCN(C(Cc2c(CC)noc2CC)=O)C1)CC C(=O)(CC(C(F)(F)F)c1ccon1)NC(CNC(CCC(C)(C)C)=O)C1CC1 c1(C(=O)NC2CC(C)N(C(=O)CCSc3nnnn3C)C2)ccc(N)c(Cl)c1 Nc1cc(F)ccc1C(=O)NCC(O)CNC(=O)CS(=O)(=O)NCC1CCCO1 N1(C(C2(C)CC=CCO2)=O)CCC(COC)C(NCC(c2c(C)coc2C)=O)C1 c1(CNC(C)(CCC(C)(C)O)c2n(CCC)nnn2)ccc2ccc(O)nc2n1 N1(C(c2c(C)ccnn2)=O)CCC(C)CC1CNC(=O)COCc1ccccn1 CCC1=C(C(=O)NCCOC(C)(C)CNC(=O)C2=CCCC2C)CCCO1 C1(NC(c2ccc(SCC)nc2)=O)CCN(C(=O)Cc2cnns2)CC1O c1(C(N(CCCCNC(C2CC2c2ccccc2)=O)C)=O)cc(Br)cs1 c1(CSCC(=O)NCCCOCCNC(C2CCCS2)=O)cccs1 N1(C(C2=NNC(=O)C2)=O)Cc2cnn(-c3ccccc3)c2C1.C12CC(C1)C2=O N12CCCC(O)(CC1)C2.C1(CCC(C)C)CCC(C(N(C)CC(C)C)=O)CC1 N1(C(CC(C(=O)OC)C)=O)CCC2(C1)CN(C(=O)CCC1CC1)C2 CCCCC(O)CCC(=O)N(CCN(C)C(c1ccc(NC)cn1)=O)C(C)C c1(C(N(CCC(C)C)C2CC2)=O)cc(CNC(=O)Cc2cn(C)nn2)ccn1 c1(C(=O)NC(C)(CO)C(=O)O)ccc2ccncc2c1 c1(C(=O)NC2CC(F)(CNC(Cc3cc(C(C)C)no3)=O)C2)c(Cl)nn(C)c1Cl C1(CC(=O)NCCN(C(C)C)C(c2cc(Br)cs2)=O)CCC(C)(O)CC1 Cc1cccc(C(=O)N(CC(C)N(C)C(C2CCC(C)(C)OC2)=O)C)c1C#N c1(C(=O)NC(C(C)NC(=O)Cc2nnn(C(C)(C)C)n2)(C)C)ncc[nH]c1=O C(CC(C)(C)CNC(=O)C(N1CCCC(Cn2ccnn2)C1)=O)OC N1(C(CC2CC(SC)C2)=O)CCCC(C(=O)NCC23CC(CCO2)C3)CC1 O=C(C1=CC2(CCOCC2)C1)NC1CCC(NC(=O)C(c2ccccc2)O)CC1 c1(N2CC(CNC(c3cccc(C(=O)NC)n3)=O)C2)nc2ccc(OC)nc2s1 C12CCCCCN1C2=O.N1(C(C)=O)CCOC(C=C)C1.C1CCCN1C=O Cc1cc(S(=O)(=O)N2CC(F)CC2CO)ccc1-c1cnsc1 C(C(C(=O)NC1(CO)CCCC1)C(C)(C)C)NC(CC(C)n1cccc1)=O c1(OC)ccc(C(CF)NC(C2(CF)CCN(C(=O)OC(C)(C)C)C2)=O)cc1 N1(c2cc(C)nc3c2nccc3)CCOC2(CCC(C(=O)OC(C)(C)C)CC2)C1 N1(C(C)=O)CCC(C)(C(=O)N(C)CC2CCN(C(c3sc(C)cc3OC)=O)C2)C1 C(N=c1[nH]c(=NC2CCC2C(F)(F)F)[nH]c2c1SCC2)C1CCCC(C)(C)C1 C1(OC)(CNC(c2ccccc2Br)C(C)C)CCC(C)CC1 N1(C(C2N(C)CCC2)=O)CCOC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 c1(C(=O)NC(C2CCCCN2C(c2cc(CO)on2)=O)C)cc(C(F)F)ccn1 c1(N2CCN(C(c3c(Cl)ncc(C)c3)=O)C3(C2)CC3)ncnc2cc(F)ccc12 N1(C(CN(C(C)C)C)=O)CCC(C(C)C(=O)NCC(C)(C)OCCOC)CC1 c1(C(=O)NCCCOCCNC(C23CC(O)C2C3)=O)cc2cccnc2[nH]1 N1(C(C(C=CC)O)=O)C2CCC1C(F)C(NC(c1cc(C)cc(C)c1)=O)C2 CN1CCC(C)(C(=O)N(C)CC2CCCN2C(C2CCCC(F)C2)=O)C1=O N1(C(c2c(OC)scc2)=O)CC2CCN(C(c3cc(C)ccc3C)=O)CC12 c1(CNC(=O)Nc2scc(C(=O)OCC)c2OCC)c(Br)nnn1C Cc1nccc(Cl)c1C(N1CCN(CCN(C(=O)CCCCCF)C)CC1)=O CC1CC(CC(=O)NC23CCN(CC2)C3)CN1C(=O)CCc1cnoc1 Cc1nc(O)c(C(=O)NC2CC2CNC(=O)Cc2ccco2)cc1Br c1(OC)ccc(C(CNC(=O)CNC(=O)C(C)(C)C)NC(C2CC2C#N)=O)cc1 CCCS(=O)(=O)CC(=O)NC(C)CC(C)NC(c1ccc(C2CC2(F)F)cc1)=O c1(C(=O)NCC2(F)CC(CNC(c3ccc(CO)o3)=O)C2)ccccc1Cl CC(=O)C(C)CC(C)C(=O)NCc1occc1C(=O)NC1CC2CC1CC21CC1 C1(C(N2C(COC)CN(C(=O)CC3(C#N)CC3)CC2)=O)Cc2ccccc2S1 Cc1cc[nH]c(=N)c1C(=O)NCC(C)(C)CN(C(=O)CC1(CS(C)(=O)=O)CC1)C C1(NC(N2CCC(Oc3cc(C)ncc3)C2)=O)CCC(=O)N(C)C1=O C(=O)(C1=CC(C)(CC)C1)N1C(CNC(C(CC)c2ccccc2)=O)CC(F)(F)C1 C(CN=c1[nH]c(Cl)c(C#N)s1)N(C(CCCCCCSC)=O)C C1(COC(C(C)(Cl)Cl)=O)NC(=O)OC1(C)C Cc1cc(C(=O)NC2CC3CN(c4cc(C5CC5)ncn4)CC23)cc2nn[nH]c12 CC1OC2CCC1(NC(=O)C(c1ccnn1C)NC(C1CCCC(CF)C1)=O)C2 C1(C(N2CCC(C(C)OC)CC2)=O)CC(C)(C)CCN1C(C1C(C)C1C)=O c1(CC(=O)NC2CCN(C(C3(C)CC3)=O)CC2)ccc2sccc2c1 c1(CC)nn(C)c(C(=O)NC2CCN(C(=O)Cc3cccc(C)c3C)C2)c1Br c1(OC)ccc(C(c2nnnn2C2COC2)NCCSC(F)(F)F)c(C)n1 Cn1cc(C#N)cc1C(N1CCN(C(=O)C(O)CC(F)F)CC1CCO)=O N1(C(C(CC=CC)CC)=O)CCC2C(C1)CN2C(c1nn(C)cc1Cl)=O N1(C(CCCC(CC)NC(c2nc(C)c(C)s2)=O)=O)CCC2(CCOC2=O)C1 C1(C(C(N2CC(C(C)NC(C3C(C)(CC)C3)=O)C2)=O)F)CCC(=O)CC1 N12CC3CCCC3C1C2=O.C1(C(=O)NCCN(CCC)CCC)CCCC(C)CC1 c1(CCC)cnnc(C(=O)NCC(C)NC(c2c[nH]cc2C2CC2)=O)c1 [N-]=[N+]=NC1(C(=O)NCC23CCC(CC2)OC3)CCN(C(=O)CCCF)C1 N1(C(C(C)=C(CC)C)=O)CC2(C1)CN(C(=O)C(C(C)C)Sc1ccccc1)C2 c1(NC(C2CCN(C(C3(OCC)CCCC3)=O)C2)C)ncc(C(C)=O)cn1 c1(NC(C2N(Cc3cc(C)nc(C)c3)CC(O)C2)=O)cccc2cc(Cl)cnc12 N1(C(c2cccc(OCC#C)c2)=O)CCCCC12CN(C(C1(F)CCC1)=O)C2 C(=O)(CC1=CCOCC1)NCCC(C)NC(c1ccc(NCCF)cn1)=O CC1CN(C(C2COCCN2C(c2cccc(O)c2)=O)=O)C(C)C1C c1(C(N2CCCCC(N(C(CC=C=C)=O)C)C2)=O)cnc2n1C(C)CCC2 CCCCCC(O)C(=O)NNCCCC(N1CCC(N(C(C)=O)CC)(CC)C1)=O.C=O Cc1nc(Cl)[nH]c(=NC2CCCN(C(C3CCC4C(C3)C4(F)F)=O)C2)c1[N+](=O)[O-] C#CCCCCCC(=O)NC(C)CNC(c1c(O)cc(Cl)cc1F)=O N1(C(CC2CC(NC)C2)=O)CCCC(C)C1CC(=O)NCC#CCCO N1(C(C)C(=O)O)CC(NC2CCOC(C)(C)C2)C(C)(C)C1 C1(N(C(CN(C)CC)=O)Cc2ccccn2)CCCN(C(=O)CCN(C)C)C1 c1(C(N(C(CNC(C2CC(CC)(CC)C2)=O)C)C)=O)ccc2c(=O)ccoc2c1 C1(N(C(C(C)N(C(CCC(C)SC)=O)C)=O)C)CCCC(C)C1C C1(CNC(c2c(CC)cns2)=O)CN(C(c2cc[nH]c2C2CC2)=O)CC1(F)F c1(C(=O)NC2CN(C(c3n(CC)nnc3C)=O)CC2COC)cccc(Cl)c1F C1(NC(c2c(CC)nc(C)o2)=O)CCC2CC1CN2C(c1ccncc1Cl)=O CC1=C(C(=O)N2CC(CNC(c3cn[nH]c3)=O)C(F)(F)C2)Cc2ccccc2O1 C1(Nc2nnc(C)c(C)n2)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC1(C)C c1(NCc2ccc(N)cn2)ccc(S(=O)(=O)N2CC(N3CCCC3)C2)c(Br)c1 c1(C(=O)NCc2ccc(CN=c3nnn(C)[nH]3)cc2)cn2ccncc2n1 C1(CNC(=O)CC2CCOC2)CC2CCC1N(C(=O)Cc1sc(O)nc1O)C2 c1(C(N2CCCCC(NC(=O)CC3C=CCC3)C2)=O)c(F)c(F)c(F)c(F)c1F N1(C(C(CC)O)=O)CC(OC)CC1CNC(c1cn(CC2CCCO2)nc1C)=O C1(O)(C(N2CCC(C(C)NC(CCc3ncc(C)[nH]3)=O)C2)=O)CCOCC1 CP(C)(=O)c1ccc(C(=O)NC2CN(C(C3CC34CCOCC4)=O)C2)nc1 Cn1nnc2cncc(C(=O)NCCOCCCNC(C3(F)CCCC3)=O)c12 c1(CC)oc(C)cc1C(N1CC(O)(CNC(=O)CC2CSCCO2)C1)=O N1(C(C2(C)CCOC2)=O)CCC2(CCC2)C(NC(=O)Cc2ccsc2)C1 C(=O)(C#CC1CCCOC1)NC1(CC=C)CCCN(C(C2(CN(C)C)CC2)=O)C1 C(=O)(CC(F)(F)C(=O)O)N1CC(CNC(c2cn3cccnc3n2)=O)OCC1 CC1(NC(c2cnc(N)c(CO)c2)=O)CCN(C(=O)C=CC2CCCO2)CC1 C#CCCCCCCCC(=O)N1CCC2(CCC2)C(NC(=O)C(O)C(C)CC)C1 C1(NC(c2cc(C)nn2CCO)=O)CC2CCC1CN(C(=O)CCC(F)(F)F)C2 C=CCCC(CC(C)C)C(=O)N1CCCOC(CNC(c2ccc(C#N)o2)=O)C1 N1(C(C(CSC)OC)=O)CCCC(O)(CCNC(c2ncnc(O)c2F)=O)C1 c1(C(=O)NCCN(CCOC)C(c2ccc(C#N)s2)=O)cnc2c(c1)CNC2=O c1(C(=O)NC(c2cnn(C)c2)COC)ccc(CCN)cc1 c1(C(=O)NC(CN(C(c2cc(C)ncc2C)=O)C)C)cc2c(C)ccc(C)c2[nH]1 c1(C(=O)NC2C(NC(C(C)NC(=O)OC)=O)CCC2)c(C)ccc2n[nH]cc12 C1(NC(C(OC)OC)=O)CCCC12CCN(C(C1CC1C1CCCC1)=O)CC2 N1(C(C(c2cccnc2)NC(C2C(C)(C)C2)=O)=O)CC2C3CCC(C3)C12 C1(C(C(=O)NC(c2ccccc2)C)=O)CCN(C(c2cc(O)n(C)n2)=O)CC1 C1(CC(=O)NCCC2CN(C(CCCN(C(C)=O)C)=O)C2)CCCC(F)(F)C1 c1(NC2CC(C)(CSC)N(CC(=O)Nc3ccccc3)C2)ncc(C(N)=O)cc1C C1(NC(c2c(C)onc2-c2ccccc2F)=O)CCCCN(C(=O)C2CC2)C1 n1(CCC(=O)NCC2(COC)CN(C(=O)CCC(C)(C)F)C2)c(C)c(C)sc1=O c1(C(=O)OC)cc(NC(=O)NCc2c[nH]c3nccc-3c2)c(Cl)c(Cl)c1 N1(C(c2c(C)cnc(F)c2)=O)CCC2CN(CCN(S(C)(=O)=O)C)CC12 CC1CCCCN1CC(=O)NCCC(C)NC(c1ccc(O)cn1)=O C(=O)(CCCS(=O)(=O)N1CCCC1)NC1C(C)N(C(=O)C(C)N2CCCC2)CC1 c1(OC)cc(C#N)ccc1CN1CCC(F)(F)C(NC(C2(C#N)CC2)=O)C1 N1(C(C2(CCC=C)CC2)=O)CC(CNC(=O)COc2cccc(F)c2)C2(CC2)C1 c1(C(=O)NCC2(CNC(CC3CC(C)C3)=O)CC2)ccc(=O)n(C)c1 C1(CNC(CCCC#C)=O)CCCCN(C(c2nc(C)sc2Br)=O)C1 N1(C(COCC#C)=O)CCC2C(C1)NC(=O)CN2C(c1cccc(CC)c1N)=O N#Cc1ccc(CC(=O)NC2CCC(NC(=O)C(=O)NCC(F)F)C2)c(F)c1 C1(C(=O)NCC2CCN2C(c2ccncc2F)=O)CCCC2(CCOCC2)O1 C12(C(N(CCC#C)CC)=O)CCCC1CCN2C(=O)CC1(OCC)CCOCC1 CC(c1cnn(C)c1)=CC(N1CCC(C(C)(C)NC(C2CSC2)=O)CC1)=O S(=O)(=O)(c1cccnc1NCc1cc(C(F)(F)F)ccn1)NC(C(C)O)(C)C N1(C(C2(CC=C)CCC2)=O)CCN(C(=O)CC(C)(O)C2CC2)C(C)C1 c1(NC(c2ncccc2F)C)ccc(S(=O)(=O)N2CCOCC2)cc1C(N)=O c1(CC(=O)NC2CC(F)CN(C(C3CC4(C3)CC43CC3)=O)C2)ccc(F)cc1Cl CC1CN(C(c2nn[nH]c2Cl)=O)CC1NC(=O)C(C1CC1)N(C)C C1(OC)CN(C(=O)Cc2ccns2)CC1NC(C1(O)COC1)=O CC1(CNC(C2(C)C=CCC2)=O)CCN(C(c2cc(Br)no2)=O)C1 N1(C(CC(CN(C)C)(C)C)=O)Cc2n[nH]cc2C1C(=O)NC1CC(C(N)=O)C1 Cc1nc2c(s1)CN(Cc1cocn1)C2C.C(C)(C)(C)C(=O)O.C1CC1 N1(C(C2C(CNC(=O)C=Cc3nccs3)CCC2)=O)CC=CC12CCOCC2 C1(C(=O)NC(CCC)CCO)CCCC(NC(C2(c3cc[nH]n3)CC2)=O)CC1 C(CN=[N+]=[N-])(C(=O)NC(C)CN1CCCC1=O)NC(CCC(=O)NCC)=O N1(C(c2snc(C)c2N)=O)CCN(C(=O)C=NN2CCCCC2)C2CCCC12 c1(C(=O)NC(CC)CNC(c2cc(OC)n(C)n2)=O)c(C)ccc(Cl)c1O c1(C2C(CC)CCO2)nc(CC2CC2)nn1-c1ccc(-c2ccccc2)cc1 c1(C(=O)NC2(CC=C)CN(C(c3cnnn3C3CC3)=O)C2)ncsc1S(N)(=O)=O N1(C2(C)CC2)CC(NC(=O)C(CC2CCC2)NC(=O)CCNC(N)=O)CC1=O c1(CCC(=O)NCCNC(CC2CCC(C)O2)=O)cncc(F)c1 C(CC(C(C)C)NC(=O)C=CCN1CCOCC1)NC(C(C)=C1CCCC1)=O c1(C(=O)NCC2C(NC(C3(COC)CC3(F)F)=O)COC2)cccc(N)c1F c1(C(N2CCCC(NC(CSC)=O)C(F)C2)=O)n[nH]c2c1C(=O)NCC2 c1(OC)ccc(NC(=O)COC(c2conc2C2CCCO2)=O)cc1 C12(CNC(CC3CCCN(C)C3)=O)CN(C(C3CC(N(C)C)C3)=O)CC1CCO2 CC(C)(C)CCCCC(=O)N1CCCC2(CCN2C(=O)OCCOC(C)(C)C)C1 C1(NC(C(=O)NCc2cccc(CN(C)C)c2)=O)CCOC12CCS(=O)(=O)CC2 c1(Cc2onc(CN)n2)ccc(C(=O)Nc2ncccc2C(F)(F)F)cc1 c1(OCCC(=O)NC2CN(C(C(F)=C(C)C)=O)C(C)C2)cccc(Cl)c1Cl N#CC1CN(C(=O)CCOC2CN(C(=O)CCC3CCOCC3)C2)C1 C12(C(=O)OC)CC1CCN2C(c1sccc1CNC(C1CC(F)(F)C1)=O)=O CN=c1[nH]c(C(=O)NCC2CCCC(NC(=O)CSCC(C)C)C2)cs1 C1(C)(NC(C=C(CCC)C)=O)CC(NC(=O)C(c2ccccc2)OCC)C1 C(=O)(C1CCCc2ccccc21)N1C(CC(=O)NC(C(C)O)CO)COCC1 C1(C(N2CC(CN(C(=O)CS(N)(=O)=O)C)OCC2)=O)CCc2cc(F)ccc2O1 C1(C(C)NC(C=COCC)=O)CCN(C(=O)CN2CCOCC2=O)CC1 N1(C(C(=O)Nc2ccccc2)=O)CC(C2CCCN(C(c3cscc3F)=O)C2)C1 N1(C(C(COC)NC(C)=O)=O)CCOC(CNC(=O)CC(C)(C)SC)C1 CCC(CC(=O)NCC1(NC(=O)CCc2ncc(F)cn2)CCC1)C1CCCC1 C1(NC(CC=C)=O)C=CCCC1C(=O)NCC(O)C(C)C N1(C(CC=C(C)C)=O)CCC(C(C)CNC(=O)CSc2n[nH]c(=N)s2)CC1 N1(C(C(CCOC)C)=O)C(C(=O)NC2CN(C3COC3)C2)CC2CCCC12 N1(C(C=CC(CC)=CC)=O)CC(NC(=O)C(C)Oc2cccnc2)CC1(C)C C(CC(C)(C)C(=O)N1CC(NC(c2ccc(F)c(CN(C)C)c2)=O)C(C)C1)SC c1(N2CC(C)C(CNC(C3(C)CCC3)=O)CC2)nc(O)c2ccccc2n1 C1(CN(C(=O)CCCc2ccsc2)C)CCCN(C(=O)Cc2ccon2)C1 C(=O)(CCCS(N)(=O)=O)NC(C)(C)C1CC1.CN1CCOC(C(N2CCCC2C)=O)C1 c1(CC(C(=O)N(C2CC2)Cc2ncc(C)nc2)N)ccc(Cl)cc1C(F)(F)F N1(C(c2nn(CC)nc2C)=O)CCCC(F)(C(=O)NCC(N2CCCCC2)C)C1 Cc1c(C(=O)NC2CC2c2ccnn2C)nnn1CC(N)=O c1(-c2n(-c3ccc(OC)cc3)nc(-c3ccn(C)n3)n2)cccc(Br)c1C C1(C(=O)NCC2(NC(COC)=O)CC2)COCCC1NC(c1cc[nH]n1)=O C(=O)(CC(C)C(C)(C)NC(=O)C1CC1)NC(C)CCF C1(OC)COc2c(C(=O)NCCCNC(=O)C(C)OCC(F)(F)F)cnn2C1 CC1=C(C(=O)NC(C)CN(C)C(c2cc(-c3cccnc3)on2)=O)CCCC1 C1(C)(CNC(C2(CC=C)COC2)=O)CCCN1C(=O)CC=CCC N(C(=NCCCC(F)(F)C(F)(F)F)NCC(C)(C)C)CC1(C)CCN(C)C1 C(CC(=O)N1CC(O)(C(C)NC(c2[nH]ccc2C2CC2)=O)C1)(C(N)=O)NC(C)=O c1(C(=O)NC2C(C)CCN(C(C3(C#N)CC=CC3)=O)C2)cc2cccc(Cl)c2o1 c1(SCC)nccnc1C(=O)NC1CC(NC(C2CC(N3CCOCC3)C2)=O)C1 C(CS(=O)(=O)CC(=O)N1CC(CC(=O)NCc2ncc(C)cn2)CC1C)OC c1(CC)nnc(C)cc1C(=O)NCC1CCC(NC(C2COCC(C)(C)O2)=O)C1 CCC(C)C(C(=O)NC1CC(F)(CNC(=O)Cn2cc(C3CC3)nn2)C1)OC c1(C(N)=O)ccc(O)cc1C(=O)NCCCCNC(C1(C2CCC2)CCC1)=O N1(C(CCOC(C)=O)=O)CCC(C(N2CCC(C(C)C)C2)=O)C(C)(C)C1 c1(CNC(C23C(CN(C(c4ccc(C)cc4)=O)C2)C3)=O)ccc2nc(Cl)sc2c1 C1(N)CC2CCC2C1.c1(C(=O)O)cc(OCc2ccccc2)cnn1 C(CCC(C)C(=O)N1CC2CC1(C(=O)NC(C1CCC1)C)C2)OC Cn1nnc2c1C(C(=O)N1CC3C(CNC(=O)CC4CC(F)C4)C3C1)CCC2 CC1CC(CNC(C2CCCCC2(C)C)=O)CCN1C(CCN(C)C(=O)CCO)=O c1(C(=O)NCC2(OC)CN(C(=O)CCOC3COC3)C2)cc(C)c(C(N)=O)cn1 N1(C(C(=O)NCc2nc(N(C)C)sc2)=O)CCC2C(C1)C2(F)F C(C(CC(C)C)C(=O)N1CCS(=O)C(C)C1)NC(C1C(COC)CC1)=O C1(C(=O)NCC=CCNC(C=CCCC=C(C)C)=O)CCCN(CC(F)(F)F)C1 N1(C(CCc2c(C)n[nH]c2C)=O)CCC(NC(C2CCC3CC23)=O)C(O)C1 C(=O)(C(C)(C)C(=O)NCC(c1ccccc1)CNC(=O)C(C)(C)CO)OC N1(CC(C)(C)Nc2ccc(F)cc2)C(=O)CCN(CC2(n3nccn3)CC2)C1=O CCC(CCOC)C(=O)N1CC(O)CC1CNC(C1(CC2CC2)CC1)=O C1(CN(C)C(C2CC(=C3CC3)C2)=O)CCCN(C(C2CC2C2CC2)=O)C1 N1(C(c2ncn(CC)n2)=O)CCCC(N(C)C(c2ncc(Cl)cc2O)=O)CC1 CCCCCC(C)(CC)C(=O)N1CC(C(C)NC(=O)CC(C)C(=O)OCC)C1 N1(C(c2scc(C#N)n2)C(=O)Nc2ccc(F)cc2)CCn2nccc2C1 c1(CC)cc(C(=O)NCC(C)C(=O)NC(C)CN2CCCC2=O)ncn1 C1(NC(NNC(c2cccc(C)c2F)=O)=O)CCCC2(CCOC2)O1 C1(NC(C2(CN(C)C)CCCCC2)=O)CCN(C(=O)CCC2CCCC2)CC1O C(=O)(CC1=NNC(=O)C1)NCC1CC(C)(CNC(=O)CN2CCN(C)C(=O)C2)C1 c1(C(=O)NCCOCCCNC(C2(OC)CCCC2)=O)c(OC)cc(C)nc1O.CC C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(C)CN(C(=O)C(N)=O)C(C)C1 CC#CCC(CO)NC(=O)C(C)(C)C1CCCN1C(C1CC1Cl)=O CC1CCCC1C(=O)N(C(C)CCN(C)C(c1cn(C2CC2)cn1)=O)C1CC1 N1(Cc2c(NC(C)=O)nc(Cl)cc2)C2CCC1CC(NC(c1ccccn1)=O)C2 N1(CC(=O)Nc2ccc(C3CN(C(C)=O)C3)cc2)C(=O)C2C=CCCN2S1(=O)=O N1(C(C)CNC(N2CCOC(CN3CCC3)C2)=O)CCc2ccccc21 n1(C(C)C)ncc(C(=O)N(CC(C)CNC(=O)CC(C)F)C)c1N C(=O)(C1=CCS(=O)(=O)C1)NC(C)CCCNC(c1cncc(O)c1)=O c1(NCCOC)ncnc(N2CCOC(C3CC(F)(F)C3)C2)c1C C12(NC(CCCC(N)=O)=O)CCOCC1CN(C(c1onc3ccccc13)=O)C2 c1(C(=O)NC2CC(N(C(=O)CCC3CC3(C)C)C)C2)ccc(Cl)c(N)c1 N1(C(=O)C2=NOC3(CCC3)C2)CCN2C(=O)C(NC(C3SCCS3)=O)CC2C1 N1(C(c2cccc(C)c2)=O)CCCC(NC(C2CCCC2(C)C)=O)CC1 c1(N2C(C)CCN(C(CS(CC)=O)=O)CC2)ncnc2c(Br)nn(C)c12 c1(C(=O)NC(C2CCOC2)CNC(c2c(C)cco2)=O)cnc2[nH]cc(C)c2c1 CCC(C(=O)NC(CC1CCC1)C(=O)NCC(F)CO)NC(N)=O c1(OC)cc2nn[nH]c2cc1C(N1CC2CCC1CN2c1nc(C)nc(=N)[nH]1)=O CN1CC(CC(=O)N2C3COCC2CC(NC(=O)CC(Cl)Cl)C3)c2ccccc21 C(=O)(C1Cc2ccccc21)NC1(CCNC(C=Cc2oc(Cl)c(C)c2C)=O)CC1 N1(C(C(C)=C2CCCC2)=O)CCC(NC(c2cc(C)cnn2)=O)CC1C C1(C(N2CC(CC)(NC(c3ccon3)=O)C2)=O)(CC)CC1(F)F c1(C(c2ccccc2Cl)OC)nc(-c2ccc(Cl)s2)nn1C1CSC1 CC1(CC(=O)NC(CO)C(=O)Nc2ccn(C3CC3)n2)CCOC1 c1(N(C(C)=O)C(N2CCC(Oc3ccc(C)cn3)CC2)=O)c(F)ccnc1Cl c1(C(=O)NCC(CNC(C(COC)(C)O)=O)C)nn(C)c2c1CS(=O)(=O)CC2 C12CCN(CC1)C(=O)CNC(=O)N2.C1(COC)CC1NC(C)=O N1(C(CC2(CC(=O)OC)CC2)=O)CCC(NC(C2CC=C(C)CC2)=O)C(C)(C)C1 N1(CC(=O)N(CCCN(C(=O)CC2CSCCO2)C)C)CCCCCC1 Cn1c([N+](=O)[O-])cnc1C(=O)NCCOCCCNC(=O)CC1C=CCCC1 N1(C(C2C3C(NC(Cc4c(C)scc4)=O)C4C(C3)C42)=O)CCCC(C)(O)CC1 c1(C(=O)NCCC(C(=O)N(CC(C)(C)CN(C)C)C)OC)cc(C)c(C)cn1 C12(CNC(=O)CC3CCC(F)(F)C3)COCCN1CCN(C(c1ccon1)=O)C2 C1(C(=O)NC(C)CNC(c2ccoc2Br)=O)CCCCCS1(=O)=O c1(C(N(CCN(C(=O)C(F)C(C)(C)O)CC)CC)=O)cc(Cl)c2c(c1)OCCO2 c1(OC)cnc(C(=O)NCC2CC3CC2CN3C(c2cnn(C)n2)=O)c(OC)n1 C1(NC(C)(C)C2CC2)CN(C(c2c(C)ncn2C)=O)CCC1C1CCCO1.C(F)(F)F Cc1c(C(N2CCC(NC(=O)CN(C)C(C)C)C2C)=O)cnn1CCO C(=O)(C1=C(Cl)CCC1)NC1(CO)CN(C(c2ccc(N(C(C)C)C)cc2)=O)C1 C(=O)(C1CCSc2ccccc21)N1CCCC(N(C)C(C2CC3CC2C3)=O)C1 O=C(CCCCOC1CCCC1)NCC1(NC(C23C=CC(CC2)C3)=O)CC1 Cc1ccc(C)c(CN2CCOCC2CC(=O)NCC2CCCCO2)c1 Cc1cc(F)c(C(N2CCC(C(C)NC(c3nccn3C)=O)CC2)=O)c(Cl)c1 C1(CNC(CCC=CC)=O)CCC12CCN(C(=O)C(CN(C)C)CC)CC2 C1(CC)COCCC1NC(=O)C(F)(F)Oc1ccc(C(N)=O)cc1 C1(NC(C2N(C(C)=O)CSC2)=O)CN(C(c2nccnc2C)=O)CC1C c1(CC)c(OC)cccc1C(N1C2CCC1C(CNC(=O)C(C)(C)C)C2)=O C1(C)(C(=O)NCC(CN(C(COCCCCC)=O)C)O)CC2CCC1O2 C(=O)(C(CC(C)C)C(N)=O)NC(C(=O)NC(c1nnc(C)o1)C)(C)CO C1(NC(c2ccc(CC)o2)=O)CCCCC1NC(=O)C=C1CCC(C)CC1 C1(NC(C(CC)OC)=O)CN(C(c2cc(CN(CC)CC)cs2)=O)CCC1(C)C C1(C(N2CC(NC(c3n(CC#C)cnn3)=O)C(C)(C)C2)=O)CCCCC12CCC2 c1(C(=O)NC2(CN(C(C3(N(CC)CC)CCOC3)=O)C)CC2)cc(C#N)[nH]c1C C12(C(N(C(C)C(F)F)C)=O)CCN(C(=O)CNC(=O)C(C)(C)C)CCC1C2 C1(C(C)C)CN(C(=O)Cc2ccncc2)CCN1C(c1cc2c(s1)CSC2)=O c1(SCCC(=O)NC2C(OC)CN(C(C3CC(C#N)C3)=O)C2)cc(F)ccc1F N1(C(CCCC(C)=O)=O)CCC2(CCCC2NC(c2cc(Br)n(C)n2)=O)C1 C(C1=CCN(C(C2(C)CC2Br)=O)CC1)NC(c1n(C(C)C)ncc1)=O N1(C(CCCn2c(C)csc2=O)=O)C2CCC1CN(C(=O)Cc1ccnn1C)C2 N1(C(c2ccc(C(C)C)o2)=O)CCC(CNC(c2ccncn2)=O)C(F)(F)C1 c1(C(=O)NCC(CC)N(C)C(c2cc(OC)n[nH]2)=O)nc2cccnc2s1 c1(-c2n(C)cnn2)ccc(S(=O)(=O)NC(C2CCC3C2C3(F)F)=O)cc1 C(N=c1[nH]nc(C(C)(C)C)o1)C1CN(C(c2cnc(CC(C)C)s2)=O)C1 C1(C(N(CCC(C)NC(c2csc(C)c2C)=O)C)=O)CN2CCCN1CC2 Cc1cccc(NC(C2CC(C)N(C(c3ccc(N4CCCC4)nc3)=O)C2)=O)n1 C(=O)(CC(C)C(=O)N1CCC(OCC(=O)N(CCCc2ccco2)C)C1)OC O(NC(=O)C(C1(O)CCCCC1)NC(=O)CC1NC(=O)NC1=O)C(C)C S(=O)(=O)(c1ccc(NC2CCC(O)CC2)cc1Br)NCCC(C)N(CCOC)C C(=O)(CCOCCNC(=O)Cc1nc[nH]n1)NC1(N(C(C)=O)C)CC1 CCCC(C)(C)CC(=O)N(C1CN(C(=O)C=Cc2cncc(C(F)(F)F)c2)C1)C CCCCCC1C(=O)OCCN1CC(C)CC.C(C)(C)(C)OCC C1(NC(COCCCC)=O)CCC(C)N(C(c2ccnc(N3CCC3)c2)=O)C1 C(=O)(C(CNC(c1ccoc1Cl)=O)(CC)CC)NC(C#C)C N1(C(C2(C)CCN(C(CC(COC)(C)C)=O)C2)=O)CCC(C2CCCC2)C1 c1(C(=O)NCC2COCCN(C(C(CC)SC)=O)C2)cc2c(cc1Cl)NCC2 C1(CNC(C2CCN(C(CC)=O)C2)=O)CCCCN1C(=O)Cc1nc(=N)[nH][nH]1 O=C(CCCCC(F)(F)F)NC1CCCN(C(C2CC(F)(F)C2(F)F)=O)C1 C(=O)(C(C)(C)c1cnsc1)NCC1C(NC(CN(C2CCSC2)C)=O)C1 CCC(CC)(CC)C(=O)N1CC(NC(=O)C(F)C(F)(F)F)C(C)C1 CCC(CCC(=O)N(C1CN(C(=O)Cc2ccc(O)nc2)C1)C)OC C(=O)(C1=C(C)OCC1)NC(CNC(C(CC)N1CCCC1=O)=O)CC(C)C c1(C(=O)NC2C=CCC(C(=O)NCC=C=C)C2)nc(C)ccc1C C(=O)(CCC(C)CC)N1C(CN(C(c2c(CC)noc2)=O)CC)CCC1 Cc1cc(=NC2CCN(C3CC3)CC2C)[nH]cc1C#N c1(C(CC(=O)NC)C)cccc2ccccc12.C(=O)(CCCCCF)O N1(C(CCn2c(C)cc(C)n2)=O)CCCC(C)C1CNC(c1ccc(CO)o1)=O C(=O)(C(F)(F)CC(C)C)NCC1CC(NC(c2c(OC)c(Cl)ncc2)=O)C(O)C1 C1(CN(C(CC2(OCC)CCC2)=O)C)CN(C(c2cncc(OC)c2)=O)CCO1 CC(CCCNC(=O)CCC1CCCO1)NC(=O)CCc1ccccc1 C1(NC(c2cc(C(F)(F)F)ns2)=O)C2CCC1N(C(c1ncncc1Cl)=O)C2 CC(CC(F)F)C(=O)NCc1ncccc1C(N1CC(CN(C)C)C1)=O C1(N(CC(C)C(=O)OC)CC)CC2CC1CN2C(=O)CN1CCCCCC1 C1(C(=O)NCCCN(C(=O)C(O)C2CC2)CCC)CCCC1C1CC1 C12(NC(CCN(C(C)=O)C)=O)CC3CC(C1)CC(NC(=O)CC1OCCO1)(C3)C2 CCC(C)C(CC(=O)NC1(CO)CCSC1)NC(c1cncs1)=O C1(C(N2CCC(O)(C(C)NC(=O)CSCC(N)=O)C2)=O)CC2(C1)CC21CCC1 C(CCCOC)(C(=O)N1CC=CCC1)NC(CC1CC(CC)C1)=O C#Cc1ccccc1CC(=O)NCCCC(C)NC(=O)C(CCSC)NC=O CC(CCN=c1[nH]c2c(c(=NCCCCN3CCCC3)[nH]1)CC(C)CC2)N(C)C C1(NC(COCCC)=O)CN(C(=O)C(C(C)C)NS(C)(=O)=O)CC(C)(C)C1 C1CC2(C1)CCOC2CNC1(c2nnnn2C2CC2)COC2(CCC2)C1 c1(OC)ccc2c(C(N3CCC(C)(CNC(=O)CNS(N)(=O)=O)C3)=O)c[nH]c2c1 C1(C)(NC(COCC(C)C)=O)CC(NC(=O)C=Cc2ncc[nH]2)C1 CC1(C)Cc2ccc(C(=O)N=c3ccn(CCN4CCOCC4)[nH]3)cc2O1 c1(C(=O)NC(C)C(C)NC(c2cnc(C3CCCCC3)s2)=O)cc(C(F)F)n[nH]1 C(=O)(C(C)(CCC)CCC)NC(CN(C(CC(C=C)(C)C)=O)C)C c1(C(N2C(C)C(NC(=O)CC3CC4(CC4)C3)CC2)=O)ccn2cnnc2c1 c1(OC)ccc(C)cc1CC(=O)NCCCC(C)NC(C1COC(=O)O1)=O O=C(CC1CCc2ccccc21)N1CC(O)C(O)C1 c1(CC(=O)NCC(C2CCC2)NC(CC(=C)Br)=O)ccc(C)c(Cl)c1 C1(C(=O)NC2CCC(NC(c3c(C)nc[nH]3)=O)C2)CCc2cc(F)ccc2O1 Cc1ccc2c(N3CCCC3(C)C(=O)NCCC3CCCCN3C)ncnc2c1 CC(C)(C)CC(=O)NCCCNC(C1C2CCC(=O)C12)=O C1(CNC(CCSCCC)=O)CN(C(=O)C(C)c2cc[nH]n2)CC2(CCC2)O1 c1(C(=O)O)c(NC(N2CCC2CO)=O)sc2c1CCOC2 C1(CC(=O)NC23CC(CNC(C(CCC)=CCC)=O)(C2)C3)CC2(CCC2)CO1 c1(CNC(c2n(CCC)nnn2)c2ccnn2C(C)CC)cccnc1Br C1(CC(=O)NC2C3(CC(NC(c4c(CC#N)ccs4)=O)C3)C2)CC(=O)NC(=O)C1 c1(OC)ccc(C(=O)NCC2CCCCCC2C)cc1OCC(=O)O C1(C(=O)NC2(CCNC(c3ncccn3)=O)CCC2)CC(F)(F)CS1 N1(C(C2(C)C(C)OC(C)(C)O2)=O)CCOC2(C1)CN(C(=O)CCC(C)(F)F)C2 N1(C(=O)CC2CSC2)CCC2CCC(C1)N2C(=O)CC1CC1 Cc1cc(NC(=O)CCc2nc(C)c(C)[nH]2)ccc1NC(C1(O)CC1)=O C(=O)(C(O)CC(F)(F)F)N1CCC(CCNC(c2cc(N)cc(O)c2)=O)C1 CCCCC(C)CCC(=O)N(C1CN(C(C2COCCC2(F)F)=O)C1)C CC1C(NC(c2ccc(N)cn2)=O)CCN1C(c1ccnc(-n2cncn2)c1)=O N(C(=NCC1CCCCO1)NCc1cnccc1Cl)CC1(CF)CC(F)(F)C1 C1(C)(C(=O)NCCC(C(C)C)OC)CCCN(C(c2cc(C)cc(F)c2)=O)C1 C1(CC(N)=O)(NC(CCOCCC)=O)CCN(C(=O)CN(S(C)(=O)=O)C)C1 N1(CC(=O)N(C)CC2CCCC2)CCN(CCc2cnccn2)CC1 N1(C(C(C(=O)OCC)OC)=O)CCOCCC1C(N1CCC(C(=O)OC)CC1)=O C(CC(O)CC(=O)NCC=C1CCN(C(C2CC2(C)C(C)C)=O)CC1)SC c1(C(N2CC(C(C(=O)NCC3(C(N)=O)CCC3)O)C2)=O)cccc([N+](=O)[O-])c1 C(=O)(C1Cc2ccccc21)N1CCC(F)(CNC(c2c(C)noc2C)=O)C1 Cc1cccc(C(=O)N(C)CCN(C)C(C2CCC3CC3CC2)=O)c1Cl CC1CCCC(CCNC(C2CCC(NC(=O)C3=COCC3)C2)=O)C1 C1(CC#C)(C(N2CC=CC(NC(c3ccc(F)s3)=O)C2)=O)CC=CCC1 C1(C(C)=O)CC12CCN(Cc1cc(C)n(-c3cccc(F)c3)n1)CC2 C=C1CC(C(=O)NC2CCCC2OCC)(CNC(=O)COC2(C)CCC2)C1 c1(CCC(=O)NC(c2cn(CC3(CO)CC3)nn2)C)ncc(C(C)(C)C)o1 N1(C(C(CCC)C(C)C)=O)CCOC2(CCC(NC(=O)C(C#N)C(C)C)CC2)C1 C1(O)(C(=O)NC2CC(NCc3cccc(OCC)c3)C2)CCOCC1CC N1(C(C(C)c2cc[nH]n2)=O)CCC(CCC(N2CCCC(CC3CC3)C2)=O)CC1 CCC(CCC(=O)NC1COCC1NC(C1(F)CCCCC1)=O)OC c1(CCN2CCC(CNC(C3CCC(COC)C3)=O)CC2)cc(Cl)ccc1F c1(COC)csc(C(=O)NCC(C2CCCC2)NC(=O)CCCNC(N)=O)c1 c1(CC(=O)NC2(C)CN(C(Cc3nccc(C(=O)OC)c3)=O)C2)ccc(Cl)c(C)c1 C1(CC(=O)NCCN(C(C2CC(C)OC2=O)=O)CC)(N(C)C)CCCCC1 c1(C(=O)NC(C2(C(=O)NCC(F)(F)Cl)CC2)C)cocc1C(N)=O Cc1nn(C2CCC2)cc1C(=O)NCC(C)CNC(=O)C(C)(O)c1ccccc1 c1(COC(C2(O)CCN(C(=O)OC(C)(C)C)C2)=O)cccc2c1CCC(=O)N2 C12(NC(C(C)Sc3ncccn3)=O)CCCC1N(C(=O)CCC(C)(C)O)CC2 C1(NC(CCOC(C)C)=O)CN(C(c2cccc(N)c2O)=O)C2(CCC2)C1 c1(CC)ncc(C(=O)NC2CC2CNC(=O)C(C)CC2CCCCC2)cn1 O=C(C(Cc1cccc(Cl)c1)=NO)NC1CCC1NC(c1coc(Cl)n1)=O c1(CC)ccc(OCCC(=O)NCC=CCNC(C2CNC(=O)N2)=O)cc1 CC1(C(=O)NCCC2(NC(=O)OC(C)(C)C)CCC2)CC=CCC1 C1(c2nnnn2C)(NS(CC(=O)OCC)(=O)=O)CCC(C)(CC)CC1 C(=O)(CC(C)CC(C)(C)C)NCC(CC=C)NC(C1CC(n2cnnc2)C1)=O C(CCC(=O)N(C(C)C(=O)NC(CO)C1(C)CC1)CCC)=CC n1(CC)ncc(C(=O)NC2CCN(C(=O)C(C(C)C)n3cnnc3)CC2)c1Cl C1(CNC(c2cncnc2)=O)CC2(CO1)CN(C(C13CC1COC31CCC1)=O)C2 N1(C(C(CC(=O)OC)(C)C)=O)CCC2(CC1)CC(NC(=O)CC1(C)CC1)CCO2 c1(C(=O)NCC(CN(C(C(n2c(C)ncc2)C)=O)C)C)ccc(OC(C)C)cc1 C(=O)(C(CC(C)C)N(C)C(C1CC(=O)NC1(C)C)=O)NCC1(OC)CCC1 c1(C(N2CC3(C(NC(C=CSC)=O)CCS3)C2)=O)ccc2ccccc2c1 C1(C(N2CCC(N(C(c3c(C)nc[nH]3)=O)CCO)C2)=O)CC2(C1)CC21CC1 Cc1c(Br)ccc(NCCCS(C)(=O)=O)c1[N+](=O)[O-] C1(NC(C(C)NC2(C3CC3)CC2)=O)CC(C)CC(C)(C)C1 N1(C(CCSCCCC)=O)CC(CNC(c2nccc(Cl)c2F)=O)CCC1C CC1(NC(c2cccnc2CO)=O)CCN(C(C2CCCS(=O)C2)=O)CC1 Cc1cnc2c(C(=O)NC3CN(C(=O)C(C)C(C)(C)C)CC3O)cccc2n1 Cc1nc(C)c(CC(=O)NC2CCC(NC(c3ncncc3Cl)=O)C2)s1 C(C(C)C(=O)NC1(C(=O)NCc2ccc(Cl)o2)CSC1)SC C1(C(=O)Nc2c(CC)csc2)CN(C(C2CC(C)(C)CO2)=O)CC(C)O1 C(=O)(C1CCc2snnc21)N1C2CN(C(CCC(CC)C)=O)CC1CC2 N1(C(C(CCOC)(C)C)=O)CCC(C2CCN(C(=O)CN3CC4CC4C3)C2)CC1 c1(C(=O)NC2CCN(C(c3ccco3)=O)CC2F)cc2ccc(Cl)cc2o1 C1(F)(CNC(CC(CC)C2CCC2)=O)CCCN(C(C2(C)CCCN2C)=O)CC1 c1(C(N2CC(c3ccccc3)(C(=O)OC)C2)=O)cn(CCOCCO)nc1C C(=O)(CC(C)(C)CC(F)F)NCC1N(C(c2c(C)nsc2)=O)CC=C1 CC(C(=O)N(CC(O)CF)C)N(C(=O)Cc1cnoc1)C1CC1 N1(C(CC2N(C)CCCC2)=O)CCOCC(CNC(c2cnoc2C2CC2)=O)C1 C1(CC(=O)NC(CC2CN(C(COC)=O)C2)C)COCCN1Cc1ccncc1 C1(C(C)NC(c2coc(C3CC3)n2)=O)CN(C(C2COC(=O)OC2)=O)CCO1 N1(C(c2cc(CC)ncn2)=O)CCC(C2CC2)(NC(C2CC2C(F)(F)F)=O)C1 CCC(C)(C(=O)NCCC(C)NC(c1ccc(-c2ccncc2)o1)=O)OC c1(CCCNCc2c(CCCCCC)ccs2)ccc(Br)cc1OC C1(NC(c2ncn(C)c2)=O)CCOCC1NC(=O)CCc1ccon1 Cn1cc(C=CC(=O)NC(C)(C)CCNC(C2CCC(F)C2)=O)cn1 C(=O)(C1CCCc2c[nH]nc21)N1CCN(C(=O)CC2COCCO2)CC(C)(C)C1 CC(CN=c1ccnc(NCc2c[nH]nc2C(C)(C)C)[nH]1)C(F)F N1(C(c2n(C)cc(Cl)c2)=O)C2CCC(C2)C1C(=O)NCC1(O)CCCCC1 C(=O)(C1CCc2c[nH]nc21)NC1C(NC(c2nc(OC)c(F)cn2)=O)COC1 C(C)(CCC(=O)N1CCOC(CCNC(=O)C=Cc2ncc[nH]2)C1)OCC C(C)(CCC(=O)NCCN(C(C1CCCSC1C)=O)C(C)C)SC C1(OCC)(CNc2cc(C(C)(F)F)ccn2)CCC(COC)CC1 c1(SCC(=O)NCc2cnc(SC)s2)ccc(S(=O)(=O)C(F)(F)F)cc1 N1(C(c2c(SC)cccc2)=O)CCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C(C)C1 C1(COC)(OCCOC)CCCN1C(C1(C)CCCCC1)=O.C1(=O)NCCOC1 c1(N2CCC(CNC(CCc3c(C)n(C)nc3)=O)C2)ccc(S(C)(=O)=O)cn1 c1(C(=O)NC2C(O)CCN(C(c3n(CC)ccc3)=O)C2)nc2cccnc2s1 C12(C(=O)NC3CC(F)(CNC(c4c(C)csc4)=O)C3)CC(C)(C1)OC21CCC1 Cc1nc(C2CC2)sc1CC(=O)NC1CC(CNC(=O)CSCCN(C)C)C1 CCCC(CCCO)C(=O)N1CCC(CNC(=O)CCC(C)OC)(OC)CC1 C1(CNC(=O)NCC2(CC(C)(C)C)CCC2)CC2CCCC1CC2 C(Cc1ccccc1)(C(=O)NCC(CO)NC(c1cnco1)=O)NC(CCC)=O C1(N(C(=O)CCc2nccn2C)CC)COCCN(C(C2C(F)(F)C23CC3)=O)C1 c1(C(N(CCC(=O)Nc2cn(CC=C)nc2)C2CC2)=O)nnc(O)nc1O C(=O)(CCCN=[N+]=[N-])NC(CC(C)NC(c1c(C)oc(C(C)C)c1)=O)C c1(C(N(CCC)CCNC(c2cnc(C)nc2)=O)=O)c(Cl)nn(C)c1C N1(C(Cc2c(C)ncs2)=O)CCC=C(CNC(C2CCCC(C)CC2)=O)C1 N1(C(C(CC)O)=O)CCNC(C(=O)NC(c2ccccc2)CC)C1 c1(C(N2CC(N(C(Cc3n(CCC)cnn3)=O)CC)C2)=O)nc(OC)ccc1Cl C(=O)(CS(=O)(=O)CC(F)(F)F)N(CCC(C(C)C)NC(=O)C(C)N(C)C)C C1(C(N2CCC(NC(C3C(C)C3)=O)C(CO)CC2)=O)CC12CCC(C)(C)CC2 c1(OC)ccc(C(O)C(=O)NCC23CC(NC(c4cccnc4N)=O)(C2)C3)cc1 c1(C(N(CC(CN(C(c2c(C)coc2)=O)C)O)C)=O)cc2ccccc2[nH]c1=N N1(C(c2c(OC)cncc2)=O)CC2CCC2(NC(=O)C(C)CC(N)=O)C1 c1(C(=O)NCC2(CO)CCN(C(C(CC#C)O)=O)CC2)cc2cccnn2n1 O=C(CCC1CCOC1)NN=c1[nH]nc(-c2ccccc2)s1 Cc1cncc(-c2cn(CCCC(=O)NC(c3nc(=O)o[nH]3)C)nn2)c1 c1(NCCC2CN(C)C2)ncc(S(=O)(=O)NC2COc3cc(Br)ccc32)cc1Cl CCCC#CC(C)(C)NC(=O)C(C)(CSC)NC(=O)CCc1csnn1 C1(C(=O)NCC(CCCC)NC(c2ccnnc2O)=O)Cc2nnc(C)n2C1 C1(NC(C2ON=C(C)C2)=O)CCOCC1NC(=O)C=Cc1sccc1C C1(NC(C(C)NC(C)=O)=O)CCCC(NC(=O)Cn2nnc(C)n2)C1 N1(CC23CC(C)(OC2)C3)C(=O)CCN(Cc2nc(C(F)(F)F)n[nH]2)C1=O C1(CC(=O)NCCN(C(=O)CSc2nncs2)C(C)C)CCOC1C(=O)OC c1(CC)ccc(NC(C2CCC2CNC(c2cc(CO)[nH]n2)=O)=O)c(C)c1 N1(C(CC(C(=O)OC)(C)C)=O)CCC2CN(C(=O)Cc3cncn3C)CC2C1 N1(C(C(c2ccncc2)C)=O)CCCC1CNC(c1cnn(C2CCC2)c1)=O c1(-n2c(C(N3CCC(CNC(C4(CC)CCC4)=O)C3)=O)cnc2)cccc(F)c1 N1(Cc2cnnc(C)c2C)CCC(=O)N(CCC=CC(C)C)C1=O c1(C(N2C(CNC(CCCC=C)=O)C=CC2)=O)coc2c(Cl)cccc12 O=C(CCCn1cncn1)NCC(C1CC1)NC(C1CSC1)=O C(=O)(CC1=NN(C)C(=O)C1)N(C1CCCCN(C(c2c(C)nc(C)o2)=O)C1)C C1(CC)C(=O)NCCCN1C(C1C(C)CCN1C(=O)COC(C)=O)=O C1(NC(CC(CC)CC)=O)CCCC12CCN(C(c1ccnn1CC1CC1)=O)C2 c1(C(=O)NCC2C(NC(C(n3ccc(C4CC4)n3)C)=O)C2)ccnc(C(F)(F)F)c1 c1(CCN(C(C(CCC)OCC)=O)C)ccc(Cl)cc1Cl c1(C(=O)NC2(C(=O)NCC(C)OCCO)CSC2)cncc(F)c1 Cc1cc(C(=O)NC2(C(=O)NCC3=NOC(C)C3)CC(O)C2)sc1C N1(C(C2=C(C)CC2)=O)CC2CCC(NC(=O)CC3CCCNC(=O)C3)(C2)C1 c1(C(=O)NC(C2CN(C(c3ccon3)=O)C2)C)cc(C2CCOCC2)[nH]n1 CC1=C(C=O)CCCC1.c1(-c2cn(CC3CC(OCC)C3)nn2)cccc(C)c1F C(=O)(C1=CCC(F)(F)CC1)NCC(C1CCCC1)NC(C(C1CCC1)OCC)=O C1(CCNC(c2c(C)cccc2)=O)CN(C(=O)COCC(F)F)CCCO1 S(=O)(=O)(c1ccccc1F)N1CCN(Cc2c(C)non2)CC1 N1(C(c2c(C)cncc2C)=O)CCC(NC(=O)C=C2CCC2)CC(C)(C)C1 c1(NC(c2nc(-c3cnc(C)nc3)sc2C)=O)cn2cc(F)ccc2n1 c1(NC(C(=O)NCC2CN(C(C(C)c3cccs3)=O)C2)=O)ccccc1C(F)F c1(C(N2CC3C(CNC(C4CC(F)C4)=O)C3C2)=O)cnc2ccccn12 C1(C(=O)NC2CC(C)(NC(=O)CC3CCC3)C2)COCC2(CCC2)O1 N1(C(CC2(OC)CCCC2)=O)CCCCC12CN(C(C1(C)CCCNC1=O)=O)C2 C(=O)(CC(C)CC(C)(C)C)NCCCCCNC(C(CCC)F)=O C1(OCC=C)CCN(C(=O)NC(c2cccc(Cl)c2)C)CC1C N1(C(C2N(C(C(CO)OC)=O)CC(O)C2)=O)CC2C=CCC(C2)C1 c1(C(=O)NC2CN(C(C)=O)C(C)CC2)cc2cccc(C)c2nn1.c1(=O)[nH]oo1 C1(C(C(=O)N(C)Cc2cn(-c3cccc(CO)c3)nn2)F)CCS(=O)(=O)CC1 n1(CC(=O)N(C(CN(C(CC=CCC)=O)C)C)C)cc(Br)c(O)nc1=O c1(C(=O)NC2CN(C(C(C)(Cl)Cl)=O)CC(O)C2)ccc2c(c1)C=CCC2 O=S(=O)(c1sccc1C1COC1)NC1CCN(CC2CCCC2)C1 C1(F)(CNC(C=CC(=O)NC)=O)CCN(C(=O)C(c2nc(F)ccc2Cl)C)CC1 N1(C(CCCC(Cl)Cl)=O)CCOC(c2cn(CC3(COC)CC3)nn2)C1 C1(NC(C2(CCC)CC2)=O)CCCCN(C(=O)C(CC)OC)C1 N1(C(CCCOC(C)C)=O)CCCCC1CCNC(c1nc(Cl)sc1Cl)=O C1(C(N2CC(CNC(c3cc(C)nc(C)c3)=O)C2)=O)CC2(CCCC2)CO1 C1(C(=O)NCC2CC(F)CN2C(C2(C3CCC3)CC2)=O)CCc2[nH]nc(O)c2C1 c1(C(=O)NC(C)CC2CN(C(c3coc(O)n3)=O)C2)cnc(N(C)C)cn1 c1(N(CCN(C(C(C2CCOCC2)OC)=O)C)C)ccc2c(c1)CC2 c1(CC)cc([N+](=O)[O-])ccc1C(=O)Nc1cccc(NC(=O)C2=CSCS2)c1 CC(C)C(C)(O)C(=O)N1CC2CCC2(CNC(=O)Cn2ncc(Br)n2)C1 N1(CC)CC(CNC(=O)COC2CC(CNC(c3nc(=N)cc[nH]3)=O)C2)CC1=O c1(C(N2CCCC(CN(C)C(C3CCC(F)(F)CO3)=O)C2)=O)cc(N)ccc1Cl C(=O)(C1CCc2c(Cl)cccc21)N1CCC(COC)(NC(=O)CSC2CC2)C1 Cc1nc2ccc(C(=O)NC(CC(N)=O)c3cn(CC4CCOC4)nn3)cc2s1 C(=O)(C(C)(O)CC(F)F)N1CC(CN(C(CCCc2ccc(C)s2)=O)C)OCC1 C1(CNC(c2c(CC)ncnc2)=O)CN(C(c2cc(CCO)on2)=O)CCC1C Cn1nc(C(=O)NCC2CCCC2NC(c2cncn2C2CC2)=O)ccc1=O c1(C(N2C(CNC(c3c(SCC=C)cccc3)=O)C=CC2)=O)ccc(O)c(Cl)n1 C1(COC)(NC(c2ccccc2O)=O)CCCN(C(=O)CCc2ccc(C)s2)C1 c1(C(=O)NCCOc2cccnc2)cc(Cl)c(Cl)c(Cl)c1.c1(N)ccccc1O c1(CNCC2CCCN(C(c3c(C#N)ccnc3)=O)C2)ccc(F)c(F)c1Cl c1(OC)nccc(CNC(=O)C(C2CCCO2)NC(C2CC=CCC2)=O)n1 c1(C(=O)NC2CCN(C(c3scnc3C3CC3)=O)C2)c(F)cncc1Br Cc1ccc(F)c(CNS(=O)(=O)CCBr)c1.C12CC(F)CN1C2=O c1(N(CCCNC(COCCNC(CCOCC)=O)=O)C)cc(OC)ccc1Br c1(CC(N2CCCC(NC(C3CC(C#N)(O)C3)=O)C2)=O)cccc2cnccc12 C1(NC(Cc2c(CC)con2)=O)CCCN(C(=O)CCNC(=O)CC(C)C)CC1 c1(C(=O)NC2CC(C)N(C(c3nccnc3Cl)=O)C2)cccc2c1NC(=O)CC2 C(=O)(C1CCCc2cncn21)N(CC(CC)NC(=O)Cc1ccnc(Br)c1)CC c1(CN2CCN(CCN3C(C)(C(=O)OC)CCCC3)CC2)ccc(C#N)c(C)c1 N1(Cc2c(F)cc(-c3sccc3Cl)cc2)CCC2(CCC(O)C2)CC1 C(C)(CC(=O)NC1CCN(C(c2ccoc2)=O)C1(C)C)(C(F)(F)F)N(C)C N1(C(C2(CC=C)CCC2)=O)CCC(O)(CNC(c2cnn(CCCC)c2C)=O)C1 c1(CSC(CC(C)C)C)nnc(-c2cc[nH]n2)n1-c1ccccc1 c1(C(=O)NCC(CCNC(Cn2c(=O)ccc(C)c2)=O)O)cccn2ccnc12 c1(C(=O)NCCC2CN(C(c3csnc3Cl)=O)CCO2)cc2c(Cl)cccn2n1 N1(C(c2c(C)snc2)=O)CC(C)(C)CC1C(N1CCC(F)(CO)C1)=O c1(CCC2OCCN(C(C(=O)NCCCC3CC3)=O)C2)cccc(F)c1 CC1CN(C(=O)CCn2ccnn2)CCC1NC(=O)C(C)(C)COCC(F)F Cc1cc(C(=O)NC(CC2CCC2)C(=O)NCC2C=CCCC2)c(C)o1 C1(C)(CNC(C2CCCN(C(c3c(C)n(C)nn3)=O)C2)=O)CC2CCC1C2 C(CC(O)C(=O)NCCNC(C1CCCCN1C(C1CCCCCC1)=O)=O)SC c1(SCC(=O)NCC(C)NC(=O)C(C)n2cccn2)cnc2ccccc2c1 c1(N(CCNC(=O)CSc2cnn(C)c2)CC)cc(C(F)F)nc2ncnn12 C(=O)(C(C)C(C)C(C)(C)C)NCc1c(C)c(C#N)ccc1 c1(CC(=O)NC2CC(C)(CNC(c3c(CC)c[nH]n3)=O)C2)ccc2nc[nH]c2c1 c1(NC)ccc(F)cc1C(=O)NCC12CCC(CC1)N2C(C1(SC)CCC1)=O c1(NC(CCSC)C)ncc(S(=O)(=O)NCC2COCCN2C)cc1Cl N1(C(c2ccc(N)c(Cl)n2)=O)CCC2CN(C(c3cc(C(F)F)cs3)=O)CC12 c1(C(N2CCCC(CCNC(CNS(C)(=O)=O)=O)C2)=O)cc(Cl)c(F)cc1F CCCCC(C)CCC(=O)NCC1CC(CC(N2CCC(C)(CCO)C2)=O)C1 CCCC(CCCNC(c1snnc1C(C)C)=O)NC(C1CCCC1(F)F)=O N1(C(CCc2cnc(C)o2)=O)CC(NC(=O)CC(C)(C)O)C(C)C1 Cc1ccc(C(O)C(=O)NCC(CNC(=O)CN2CCSCC2)CO)cc1 N(S(=O)(=O)N(C)CCC1CC1)CC1(OC)CCC1 C(C(C(=O)N1CC2(CNC(=O)O2)C1)C(C)(C)C)OCCOC C1(NC(C(N2CCCCC2C(N2CCCC2)=O)=O)=O)CCC2CCCC2C1 CC(C)C(C#N)C(=O)N1CC(NC(=O)CC(c2cccc(F)c2)O)C1 c1(C(C)C)conc1C(=O)NC1CN(C(c2ncoc2-c2cccs2)=O)C1 C1(C(=O)N(CCCNC(C2(CCC)CC2)=O)C(C)C)CN(C2CCC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC2CCC(NC(=O)Cn3ccnn3)CC2C1 O=C1CNC(C(=O)NCCC2(CO)CCOCC2)CN1 c1(NC(CC2C(CC)C2(F)F)=O)ccc(NC(c2c(C)nsc2Cl)=O)c(C)c1 Cc1cnsc1C(=O)NC1CCC(CNC(=O)CSc2n[nH]c(=N)s2)C1 C(=O)(C(O)CN1CCCC1)NCCC1(C(=O)NC(COC)C2CC2)CC1 c1(C(N(CC(C)NC(=O)CC2CCCCC(=O)N2)C)=O)cnn2cccc(Cl)c12 [N-]=[N+]=NC1CCC2(C(=O)NCC3CCC(CNC(=O)C(O)C(F)(F)F)CC3)CC12 c1(C(c2nnnn2C2CC2)NC(C)CCC(F)(F)F)ccc2c(c1)NC(=O)CO2 c1(C(=O)NC(CCOC)CNC(C2CC3CCC3C2)=O)n[nH]c2c1COCC2 O(P(C)(=O)CNC(C1CCC(C2CC2)N1C(=O)C(C)C(C)C)=O)CC c1ccc(Cl)c(OC)c1.CCC(CC)C(c1nnnn1C1COC1)N N1(C(C2CCC(=C)CC2)=O)CCC2CN(C(C3CC(C(C)(C)C)=NO3)=O)CC12 c1(CN2CC(CCNC(c3c(C)coc3)=O)S(=O)(=O)CC2)c[nH]c2ccc(Br)cc12 c1(C(N2CCC(OC)(CNC(c3cnc(C)[nH]3)=O)C2)=O)cscc1S(C)(=O)=O c1(CC(N2CCC(Cn3cc(CN4CCCC4CO)nn3)C2)=O)ccncc1Cl Cc1cn2c(n1)CC(C(N1CC3(CC3)CC1CNC(c1coc(Cl)n1)=O)=O)CC2 c1(OC)cc(C=O)c([N+](=O)[O-])cc1OCc1nc(C2CCCCO2)no1 C1(NC(CCCCNC(N)=O)=O)CCC2CN(C(=O)C=C(C3CC3)C3CC3)CC12 c1(CNC(=O)CNC2(C)CN(C(=O)C(F)(F)CC3CC3)C2)ccc(F)cc1 c1(CCC)cc(C(=O)NCCCCN(C)C(C2CC3C=CC2C3)=O)n(C)n1 C(=O)(C(C(C)(C)C)N(c1cc(-c2ccc(Cl)cc2)[nH]n1)C)OC.C12CN(C1)C2=O C1(C(=O)NCCc2csnn2)CCCN(C(=O)CC2CC(F)C2)C1 c1(C(=O)NCC2(C)N(c3nc(C)cc(CC)n3)CCC2)nccc2[nH]ccc12 C1(C(=O)NC(C2CCN(C(=O)CCCN(C)C)C2)C)CCSCC1 c1(C(=O)NC2CCCN(C(c3c(CC)nn(C)c3)=O)C2)cnc2c(c1)CCCC2 C(=O)(C(C)N1CCCC1)N(CC(=O)N(C(C)C1CC1)C1CC1)C C(=O)(C(C)C(O)C(C)C)NC(C=CC(=O)N(C(CCC)CCC)CC)(C)C c1(CC)ccc(C)cc1C(=O)NCC1(C)CCN(C(=O)CCNS(=O)(=O)CC)C1 c1(SC)nc(Cl)c(NC(=O)CC2CCCN2Cc2cc(Br)c(C)c(Br)c2)c(Cl)n1 CCCCCCCCC(C(=O)Nc1cccc(Cl)c1C)N1CC(C)CC(C)C1 N1(C(C(c2ccc(F)cc2)C)=O)CC(NC(c2ccnn2C)=O)CC2(CC2)C1 n1(CC)cc(C(=O)N(CCCN(C)C(C2(COC)CC2)=O)C)nn1 C1(NC)CCCN(C(C2(C)CC3CC3C2)=O)C1 C1(NC(C)=O)CCN(C(=O)CCC2CCN(C(=O)CCC3CCCO3)C2)CC1 c1(C(C)(C)C)ccc(Br)cc1Cl.C1CCN(C(C(C(=O)NC)=O)=O)C1 N1(C(C2C(C)C2C)=O)CC2CC2C1C(=O)NCCCN1CCCC1=O N1(CC(=O)Nc2cccc(C)c2)CC2(CCCC2)C1C(=O)O Cc1ccc2c(c1)CN(C(C1Cc3nncn3C1)=O)CCN2C(C1CCCO1)=O N1(C(CC(=O)NC2CC2)=O)CCC(C(N2CCC(C3(C)N=N3)C2)=O)(CF)C1 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(Cc2ccc(C)o2)=O)CC1CCO c1(CC)cc(C(=O)N(CCNC(=O)COC2CCC(C)CC2)CC)n(C)n1 C1(C(N2CC(CC)N(C(=O)CCc3nc(C)no3)CC2)=O)CCC2CCCCN12 C1(COC)(NC(c2ccc[nH]2)=O)CCN(C(c2cnc(O)n2C)=O)CC1 C1(C(N2CC(c3n(C)cnc3)C(C(=O)O)C2)=O)Cc2nccn2C1 C(CC(=O)NCC1CCCCCN1C(c1cc(Cl)ncc1O)=O)(C(C)C)OCC N1(C(c2ccc(C(=O)OCC)o2)C(=O)NCCC2CC2)CC(C)SC(C)C1 c1(CC)c(C(=O)NCc2ccsc2C(=O)NC2(C)CCOC2)nnn1C C1(NC(c2coc(C(C3CC3)=O)c2)=O)COC2(CCCN(CC3CC(=C)C3)C2)C1 N1(C(c2c(C)c[nH]c2)=O)CCC2(CC1)CC2(CO)CNC(=O)CC1NC(=O)NC1=O N1(C(Cc2c(C(C)C)con2)=O)CC(N(C)C)C(F)C1.C1(=O)CC(O)CN1 Cc1cccc2cc(C(=O)NC3CCCC3c3cccc(Br)c3)nn12 C(CCC(C(=O)NCC1CCCO1)N1CCC(c2nncn2C)CC1)OCC N1(C(C2CC(C#C)(O)C2)=O)CCC(C)C(CC(=O)N(CC(N2CCCC2)=O)C)C1 C1(NC(CCc2cc(C)on2)=O)CCC(F)(CNC(=O)C(=O)NCC(F)(F)F)C1 c1(OC)cc(C(=O)NCCOC2CCN(C(=O)CCC(F)(F)F)C2)ccc1F C(CC(N)=O)(C(=O)NC1CCC(C)CC1)N(CC)CC.C12C=CC(C1)C(=O)N2 C(CCCCC(=O)NCCc1cncs1)N(C(C1CC=C(C)CC1)=O)C N1(Cc2cc(OCC)ncc2F)CCC2(CCC(CC#N)C2)CC1 C1(CCN(C)C(c2cccnc2S)=O)CCCCN1C(=O)C1=CCOC1 Fc1cc(NC(c2ccccc2)c2nnnn2CC2CC2)cc(F)c1Br c1(C(N2C(C)CN(CCOc3ncc[nH]3)CC2)=O)ccccc1[N+](=O)[O-] Cc1cnn(C)c1CC(=O)NC(C)CC(C)NC(=O)Cc1cc[nH]c1 CCCCC(CCCC)SC.C(=O)(C(CC(C)(C)C)OC)NC12CN(C1)C2=O Cc1c(C(N2CC(n3cc(C(C)(O)CC(C)C)nn3)C2)=O)ccc(CO)c1F C(=O)(C1=CC2(CCOC2)C1)Nc1cccc(NC(C(C)Cc2cnco2)=O)c1 N1(C(C(CNC(C2(CC(C)=O)CC2)=O)N(C)C)=O)CCCC(O)C1 Cc1c(C(N2CCCC2CNC(c2cccc(CO)c2)=O)=O)cnn1C C(=O)(CCCCC#N)NC1CCN(CCCNC(C(C2CCCN(C)C2)(C)C)=O)C1 CCN=C(NCC1C(C)C1(F)F)NCC(c1ccccc1)OC C1(CNC(C(c2n(C)cnc2)O)=O)CCN(C(C2CC3CCC3C2)=O)C1(C)C CC(C)CC(C)CNC(=O)C(O)CCNC(c1cn(CCO)nn1)=O C1(CC(=O)N(CCCCNC(=O)CCC2CCCO2)C(C)C)CCCC12CC2 c1(OCC)ncc(NC(=O)C(C2CCCN(C(=O)CC3(N(C)C)CC3)C2)C)cn1 C1(C(C)C)CCCC1C(=O)NC1CCC(NC(=O)COC2CCC2)C1 C1(CNC(C(COC)(C)O)=O)N(C(c2sc(C)cc2Cl)=O)CCC1(C)C C1(C(=O)NC2(CNC(c3n(CC#C)ccc3)=O)CC2)CC(c2ccncc2)=NO1 c1(C(N2CCC(CO)C(O)C2)C(=O)NCCC#N)ccc2ccc(Br)cc2n1 C1(C)(C(N2C(CCC)CN(C(=O)C(C)C(C)(C)C)CC2)=O)CCC2(CC1)CC2 CCC(C)CCC(=O)NCc1csc(CNC(=O)C(C)CC(=O)OC)n1 C(=O)(C(C(C)(C)C)C1CCCC1)NC1C(NC(C2(OC)CCCCC2)=O)C1 CC(C)S(=O)(=O)C(C)C(=O)N1CCOCC1CNC(c1cnc(S)[nH]1)=O C(=O)(C1c2ccccc2CN1CC1CC1)N(CC=C)Cc1cc(Br)ccc1OC c1(OC)nccc(C(=O)NC2CCCCC2CNC(c2cc(=O)n(C)o2)=O)c1F N1(C(Cc2n(C)ncc2C2CC2)=O)CCC2(NC(c3cnn(C)c3)=O)CC2C1 c1(C(=O)NCC(C)CN(C(=O)Cc2cncs2)C)ccnc(S)c1 C1(C(=O)NC(C2CCCN2C(c2cc(O)cs2)=O)C)C=CCCC1 CCC(COC)C(=O)N1CCC(OCC(=O)NCC2(O)CC=CC2)C1 N1(C(C2N(C)CCC2)=O)CC(F)(F)CC1(C)CNC(=O)C(C)(C)C(N)=O n1(C(C)C)ncc(C(N2CC(N(C(=O)CCC3CC3)C)C(F)C2)=O)c1N C1(CNC(N2C(C(C(=O)OC)(C)C)CCC2)=O)CC2C(C1)C2(C)C O=C(CCCC#Cc1ccccc1)NCCNC(C1CC12CCOC(C)C2)=O C12(C(=O)NCCN(C(C(CN(C)C)(C)C)=O)C)CC1COC21CCC1 C(=O)(C(C)(C)n1ccnn1)NCCN(C(=O)Cc1cnc(C(F)(F)F)s1)CC c1(OC)ccc(C)nc1C(N1CCN(CC(C)(C)NC(C2CCCS2)=O)CC1)=O CC1=C(C(=O)NC2COCC2CNC(c2oc(CO)nc2C)=O)C(C)(C)CCC1 N1(C(c2c(NCC)cccn2)=O)CC(C)N(C(=O)C(C)=C2CC2)CC1C Cc1cc(C(=O)NCC2CN(C(=O)CC#N)CC2(F)F)c2nccn2c1 C#Cc1cccc(CC(=O)N(C(CC(C)C)C(=O)N(C2CC=CC2)C)C)c1 c1(CC)cc(C(=O)N(C2CCN(C(=O)C(C)OCC3CC3)C2)CC)cn(C)c1=O N1(C(c2ccc(C)c(Cl)c2Cl)=O)CCC2CN(C(C3(C)CCNC3=O)=O)CC2C1 Cc1cc(C(=O)NCCCC(C)NC(=O)Cc2cnns2)cc(C)c1C#N N1(C(C=CC2(C)C(CC=C)C2)=O)CC(NC(=O)C(CC)CCC)C2(CCCC2)C1 CC1CCC(C(C2(NC(CCC3CCC3)=O)CCC2)N2CCC2C2CCCC2)O1 N1(C(C(CC#C)(C)CC)=O)C(C)CC2CN(C(C3CC4(CCO4)C3)=O)CC12 c1(CNC(=O)CC2(NC(C3C(c4ccccc4)C3(F)F)=O)CCC2)ncccn1 c1(OC)cc(C)c(C(=O)NC2CCOCC2NC(=O)CN2CCC(C)CC2)cn1 N1(C(C2(C)CC2(F)F)=O)CC2(CCC2NC(c2nnc(C(C)(C)C)s2)=O)C1 C1(NC(C2N(C(C)(C)C)CC2)=O)CCC(CC(=O)NC2(C(O)CO)CC2)CC1 c1(CCN(C(C(C)C2CC2)=O)C(C(=O)O)C2CC2)ccccc1 N=c1[nH]c(=NCC2(CO)CCCCC2)[nH]c(=NCCC(O)C2CCC2)[nH]1 CCC(C)CCC(=O)N1CC=CC1(C(=O)NCCC(O)C(C)C)COC Cc1nc(C)c(-c2ccc(CN3CCCC3(C)c3cccs3)o2)s1 C1(C(=O)NC(CC=C)CO)CC(C)(C)CN1C(c1ccc(F)s1)=O C1(C)(CCNC(C2CCC(C)(CC)O2)=O)CCN(C(c2nc(=N)cc[nH]2)=O)CC1 CC1COC2(C1)CN(C(=O)C1=CCN(C(C3COCC3C(N)=O)=O)C1)C2 N12CCN(C(c3ccccc3)C1)C2=O.CC1(c2noc(C3CC3)n2)CCSCC1 C1(COC)(CNC(c2cc(C)ns2)=O)CCCN1C(c1nc(O)sc1C)=O O=C1CN(C(C2(C(=O)O)CCOCC2)=O)CCN1Cc1ccccc1Cl c1(C(C(=O)NC(C(=O)OC)C)N(C(C)CS(C)(=O)=O)C)sc(Br)nc1Cl C1(CC(=O)NC(C)CNC(=O)C(C)(C)Oc2ccccc2)COCC2(CCC2)O1 Cc1nc(=N)[nH]cc1C(=O)NC1CC1NC(=O)Cc1c(O)ncnc1O c1(C(=O)NC(C(C)C)CCNC(C2(S(N)(=O)=O)CC2)=O)ccc(N)c(Cl)c1 c1(C(=O)NC(CNC(C(CCC)OC)=O)CO)c(C)[nH]c(C(=O)OC)c1C C(=O)(CCCC(C)(C)CC)NC(CC)CNC(=O)Cn1nnc(C)n1 CC(CO)(C(=O)NC1COC(C2CC2)C1)NC(=O)Cn1cnnn1 c1(C(N2CCC(NC(CSCC=C)=O)CC2C)=O)ccc(Cl)c2ccccc12 C(=O)(CC(F)(F)F)NCCC1N(C(C(=O)Oc2ccccc2)=O)CCC1.C1CN(C)N1 N1(C(c2cnc(C)s2)=O)CC(NC(=O)Cc2coc3ccccc23)C(C2CC2)C1 CC1CC2CN(C(=O)CCF)CC2N1C(=O)C(N1CCc2ccccc2C1)C CCC(CC)(C(=O)NCC1CCN(C(c2nnn(C)c2N)=O)C1(C)C)OC CCCCCC(O)CC(=O)N1CCOCC1CN(C(=O)CC(C)(F)F)C C1(C(=O)NC23CC(C(=O)NCC(CC)CO)(C2)C3)CCC=CCC1 C(N=c1cc(NCc2cn(C)nc2Br)nc[nH]1)c1cc(C(C)C)no1 N1(CC)CCC2=C(C1=O)C(c1ccc(Br)cc1Br)NC(=O)N2CC(C)C c1(OC)ccc(NC(C2CCCCC2NC(C2(C(F)(F)F)CCC2)=O)=O)nc1C C1(F)(C(=O)NCCCCCNC(C(CC)=CCCC)=O)CCCCC1 Cc1cc(C(=O)NC(C2CCN(C(c3occc3C)=O)C2)C)cs1 c1(C(=O)NC2CCC(CNC(C3CC(N(C)C)C3)=O)C2)cncc(F)c1Cl CCC(C)(O)C(=O)NCC1(OC)CCN(C(=O)C(=Cc2ccccc2)OC)C1 C1(NC(c2c(C)[nH]cc2)=O)CCOCC1NC(C1CC1CC(C)C)=O C1(O)(CCNC(CC(C=C)C)=O)CCCN(C(C23CCC(C2)OC3C)=O)C1 c1(C(N2C(C(N(CCC(F)(F)F)C)=O)C=CC2)=O)cc2cccn2cn1 N1(C(c2c(C)cno2)=O)CC(CNC(=O)CCCc2ccncc2)C(C)C1 N1(C(C(N2CC(O)(c3cc[nH]n3)C2)=O)C2CCCC2)CCC(F)(F)CC1 c1(COC)cc(CN2CCC(O)CC2C(=O)NCC2CNC(=O)CO2)cc(Br)c1 C(=O)(C1CCc2cc(F)ccc21)NCCOCCN1CCN(C(C)=O)CC1 C1(C)(C(=O)NCC(C2CC2)NC(C2N(CC(C)C)CCC2)=O)CCOCC1 c1(CCC)ccc(C(=O)NCCCCNC(=O)C(O)c2cnc[nH]2)cc1[N+](=O)[O-] C1(C)(C(c2n(CCC)nnn2)(C)NC(C)CC2CC2)CCCCO1 C1(C)CCCC1(F)F.c1(C(=O)NC(C2CCCC2)CNC(CNC)=O)cnoc1 C1(CNC(c2cccc(C(F)(F)F)n2)=O)COCCN1C(=O)CSC(F)(F)F CC1=NOC(CCNC(c2cc(CNC(=O)CCc3cncnc3)on2)=O)C1.C1(C)CC1 c1(C(N2CCN(CC=C)CC2)=O)coc2c1CN(C(=O)CC1CC(O)C1(C)C)C2 c1(C(=O)NCC(CN(C(CC)=O)C)C)nc(OC)ccc1C Cn1nc(C(=O)NC2(C)CC(NC(C3CCC34CCC4)=O)C2)c2cc(F)ccc12 C#CCC(C(=O)NCCN(C(c1cnc(C(F)(F)F)nc1)=O)C(C)C)C1CC1 C1(CC(=O)NCCN(C(c2csc(-n3ccnc3)n2)=O)CC2CC2)CC2(CC2)C1 C1(C(=O)NC(CC=C)C(=O)N2CC(CC)C(O)C2)CCC(C)(O)CC1 C1(Cn2cc(C3(CN)CCOCC3)nn2)CCC(F)(F)CC1 CC1C(NC(=O)C(c2cccc(Br)c2F)C)CCS1(=O)=O C1(C(=O)NC(CCCC)CNC(C2CNC(=O)N2)=O)C2Cc3cc(Cl)ccc3C12 N1(C(CCSC)=O)CCC(C(F)CNC(c2snc(Cl)c2Cl)=O)CC1 Cc1ccc(C(C)(C)C(=O)NC2CN(C(=O)C(=O)NC3C4CCCCC34)C2)cc1 C(N=c1ccn2nccc2[nH]1)C1N(C(c2ccc([N+](=O)[O-])s2)=O)CCC1 C1(NC(COC(CC)C)=O)CC2CCC1(C(=O)NCC1C(C)(C)C1(C)C)C2 C(N=c1nc(N2CCC3(CC2)CC3C#N)c2c([nH]1)CCCC2)C1N(CC)CCC1 C(=O)(C(CNC(c1cc(C)cc(F)c1)=O)CC(C)C)NCc1cc(C(C)C)on1 C1(NC(CC2CC(=C)C2)=O)CCCN(C(c2ccc(C(=O)CC)cc2)=O)C1 C1(C(N(C)Cc2c(C)cncc2)=O)CN(C(c2cn(C)cn2)=O)C(C)(C)C1 c1(C(N(CC(CNC(c2nc(OC)c(C)s2)=O)O)C)=O)nc(C)[nH]c2nccc1-2 C1(CN(C(C2CC2(C(C)C)CC)=O)CC)CN(C)CCN1C(=O)C=CC(=O)OC n1(CC=C)nnnc1C(C)(CCc1ccccc1)NCC1(OC)CCSC1 c1(OC)cc(C(O)CNc2cc(-c3cccnc3)[nH]n2)c(F)cc1O C1(NC(=O)C=Cc2cccnc2)CCN(C(C2CC3(C2)CC(O)C3)=O)C12CCC2 N1(C(=O)OC(C)(C)C)CCN(Cc2snc(Cl)c2Cl)CC1Cc1ccccc1 C1(C(N2CCC(CC=C)(NC(=O)CC(C)N(C)C)C2)=O)CC2(CC2)CN1C C(=O)(C(=O)NCCC(=O)N(C)Cc1nc[nH]n1)NC(C)C CC1CCN(C(=O)CN(C2CCSC2)C)CC1N(C(=O)CC1(N(C)C)CCC1)C C(=O)(CC(O)CCC(C)CC)NC1(CC)CN(C(c2c(CC)occ2)=O)C1 Nc1cc(C(=O)NCCC2(O)CN(C(=O)COC3CC3(F)F)C2)cnc1Cl C1(C(N(C(C)(C)CC(=O)N2CCCC2CC(N)=O)C)=O)CCC(=O)N(C)C1 N1(C(COCCCC)=O)CCCC(CC(=O)NC2(CC)CCOC2)CC1 Cc1ccc(C)c2[nH]c(C(=O)OCCCC(Cl)Cl)cc12 N1(C(C(CN(C)C)NC(=O)CCc2nc(=N)[nH][nH]2)=O)CC2C(C1)C2(F)F N1(C(C=C(CC)C)=O)CCC(NC(=O)CSCCN(C)C)C1 C1(CNC(C=C(COC)C)=O)CC2CCC1N2C(c1csc(C(C)(C)C)n1)=O c1(NC2(CNC(CC=CC=C)=O)CCCC2)nc(C)nc2c1cnn2C C(=O)(C1=CCC(F)(F)CC1)NC(C)CN(C(=O)CCSCCN(C)C)C C1(NC(c2cc(Cl)cnc2O)=O)C2CC(O)C1N(C(c1csc(C3CC3)n1)=O)C2 N1(C(C2C(C)(C)C2)=O)CCCC2CN(C(c3cccn4cncc34)=O)CC12 C1(C(=O)NC(c2cccnc2)CC)OCCC1NC(=O)CC1CC2(CC2)C1 C(N=c1[nH]nc(Cc2ccccc2)s1)C1(NC(C#CC)=O)CCOC1 C1(C(=O)NCCCN2CCC(NC(Cn3c(C)ccn3)=O)C2)CCCCS1(=O)=O C(c1ccc(Br)s1)=CC(=O)NC(C)CN(C(=O)CC1OCCCO1)C C1(NC(C2N(CCC(C)C)CCC2)=O)CN(C(=O)C2=CCCCC2)CCC1(F)F C12(C(N3CCCC(C)(NC(C(C)O)=O)C3)=O)CCC(C(F)(F)F)(CC1)CC2 C1(NC(c2ccn(C)c2C2CC2)c2n(CCC3(C)CC3)nnn2)CC12CC(O)C2 N1(C(c2ccn(CCCC)n2)=O)CC2CC1CCN2C(=O)CCN(C)CC c1(C(=O)NC(C2CCCCC2)CNC(CC(=O)OC)=O)cn2cccnc2n1 N1(C(=O)OC(C)(C)C)CC2COCC(C1)C2NC(=O)CCc1ncc[nH]1 N(C(=NCc1sc(C)nc1C)NCC(=O)NCc1ccccc1)CC c1(C(=O)NCCCCN(C(C(=O)NCCOC)=O)C)cc(S(C)(=O)=O)cnc1O CC(C)CC(F)C(=O)Nc1nnc(N2CC(CC3(O)CCCC3(C)C)C(C)(C)C2)s1 C1(C2CNC2)CN(C(c2ccn(C3CC3(F)F)n2)=O)CCO1.CCC=O.C(F)(F)F c1(CCC(=O)NC2C(NC(CC3(CSC)CC3)=O)COC2)c(C)nc(S)nc1C CC(CN(C(=O)C(Cc1cc[nH]n1)NC(C1CC12CC2)=O)C)C(C)(C)C c1(C(=O)OC)ncc(C(=O)NCC2COCC2NC(C2(F)CC2)=O)s1 c1(OC(C)C(=O)NC2CC(Cn3cc(CC(C)O)nn3)C2)ccccc1Cl C(CC(C)C(=O)N1CCC(N(C(=O)CCC=C(C)C)CCC)C1)=CC N1(C(C2CN(C(C)(C)C)C(=O)C2)=O)CCC(CNC(=O)CCF)C12CCC2 C(=O)(C1=CCOCC1)N1CCC(NC(c2n[nH]cc2C2CCC2)=O)C1 n1(CCC(=O)NCC(CO)NC(C(CCSC)N(C)C)=O)ccc(O)nc1=O c1(NC(=O)OC)cccc2c1CCCC2NCC(C)COCCO Cc1cc(F)cc(C(=O)NCC(CNC(=O)CC2=CCOCC2)OC)c1N N1(C(c2scc(C(C)=O)c2)=O)CCC(C)(C)C(CNC(=O)C(C)CN(C)C)C1 c1(C(C(=O)NCCCNC(=O)C(O)c2ccco2)O)ccc(F)c(Cl)c1 C=CCC(C)(CC)C(=O)NC1CC2(C1)CC2C(N1CCCCCCC1)=O C(=O)(CC(O)C(C)C)NC(CC)CNC(C1CC2CC1C2)=O N1(C(CCOCCOCC)=O)CCOCC1CNC(c1cc(C)nn1C(F)F)=O C1(C(=O)Nc2ccc(OC(C(=O)OC)C)cc2)Cc2nccnc2C1 Cc1ccc(CC(C)C(=O)N(CCC(C)NC(c2ccon2)=O)C)cc1 C(CC(C(=O)N(C)Cc1ccc(C)cc1)NC(C1CC1(C)C)=O)SC N1(c2cc(NC(CC(=O)NC)C)nc(C)n2)CCC2OC(=O)NC2C1 C(CCCCC(=O)NC(CNC(=O)CC(O)Cc1ccccc1)C(C)C)OC C1(CNC(c2c(C(=O)OC)cccc2)=O)CCN(C(=O)C(C)(C)CSC)CC1O N1(C(COC)=O)CCN(C(=O)CCNC(=O)C=CCl)CC1C.C1C(=O)N1 Cc1ccc(NC(=O)Nc2ccccn2)c(SC2COC2)c1 N1(C(CC2CCN(C(c3c(C)cc(O)nc3)=O)C2)=O)CCC2(C1)CC2(F)F CCCCS(=O)(=O)NC(C)C(N1CCC(NC(=O)COC(C)=O)C1C(C)(C)C)=O CCCC(C)CC(=O)NC1CC1NC(=O)C(C)(C)CO C1(N(c2ccccc2)C(C)=O)COCCN(C(C)C(=O)NC2CCCC2C)C1 n1(CC(=O)NCC2C(NC(c3c(N(C)C)nccc3)=O)C2)ncc(C#N)c1N c1(CN(C)C(C2(CNC(c3ccccn3)=O)CCC2)=O)ccccc1O Cc1ccc(C)c(OCCOC(c2c(CO)n[nH]c2C)=O)c1 CCC(C)(CC)C(=O)C(=O)COC1CC(F)(F)C1.C1(C(CN)NC(=O)CO)CCOC1 C(N=c1cc(C(F)(F)F)nc[nH]1)C1(NCCCN2C(C)CCCC2)CCC1 c12ccc(cc1)C(=O)NCCn1cc-2nn1.C(C(=O)N(C)C)SCCN(C)C C1(CNC(CCS(=O)(=O)NC)=O)CC2COCC2N1C(=O)CC12CC(C1)C2 N1(C(C)=O)CC2(C1)CN(c1ccc(C#N)nc1)C2.c12nc(cs1)C(=O)N2 Cc1cscc1C(=O)NCC(C1CC1)N(C(=O)Cc1ccc(Br)s1)C c1(C(N2C(CO)CC(NC(C3CC3(F)F)=O)C2)=O)c[nH]c2ccc(O)cc12 CCC(C)CCC(O)CC(=O)N1CCN(C(C2(CCF)CC2)=O)CC1C c1(C(=O)NC2C(C)CCN(C(CCOCCOC)=O)C2)n[nH]c2c1CCCCC2 c1(CC)nc(C(=O)NC(C)C(C)NC(c2cc(O)ncn2)=O)c2ccccn12 C1(NC(C(CC)n2nccc2C)=O)COCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCOCC1CCNC(C12CCC(C1)OC2)=O c1(OCCCC(=O)NC2(CC(=O)OC)CCC2)cc(C)ccc1C c1(C(=O)NCC(CCOC)NC(=O)CN(C)S(N)(=O)=O)ccc2nccn2c1 C12(NC(c3cc(CCO)on3)=O)CCCC1CN(C(=O)Cc1ccno1)C2 Cc1cc(C(=O)NC(C)C(=O)NCC2(N(C)C)CCOC2)c(N)s1 C1(CNC(N(C2CC(F)C2)CCC)=O)CCCCC1OC c1(C(=O)NC(CNC(C(C)SC)=O)CC(C)C)ccn2cccc2c1 CC1CCN(C(=O)CC(C)(C)C2CC2)CC1CNC(=O)CNC(=O)C(C)(C)C C1(C2CCCCN2C(=O)CC2OCCO2)(CNC(CCSC)=O)CCOCC1 CC(C)CC(C(=O)NCCCCNC(C1CCCN1C=O)=O)N1CCCCC1=O c1(OC)c[nH]c(C(N2CCC(N(C(=O)C=Cc3ccc(C)cn3)C)C2)=O)cc1=O C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(=O)C(F)OC(F)(F)F)CCC1(F)F c1(N2CCC(NC(N(C3CCC(C)CC3)CCC)=O)CC2)nccc(C#N)n1 C1(C(=O)NC(CNC(c2ccnn2C2CCC2)=O)C2CC2)Cc2ccccc2N1 N1(C(Cn2ccc(C(=O)OC)n2)=O)CCC(F)C(NC(c2cc(Cl)c[nH]2)=O)C1 C1(C(=O)NC2C3(C)CN(C(CCC)=O)C2C3)CC(C)(C)OC1(C)C N1(C(C2(CCC)CCC2)=O)CCC(O)C(NC(=O)Cc2sc(C)nc2C)C1 C1(CN(C(Cc2c(C)occ2)=O)C)CCCC(NC(C2(F)CCC2)=O)C1 C1(C(=O)NC2CC(NC(c3cc(SC)oc3)=O)C(O)C2)CCC(=O)N(C)C1 C1(=O)NN2CCCC2OCn2ncc1c2.N1(C(N2CCCC2)=O)CCCC(F)CC1 n1(C(CC(=O)N(C(CC)CN(C)C(=O)OC)CC)C)nc(C)cc1C c1(CNC(c2cccc(C)c2)CNC(=O)CC(C)C(C)C)ncn2ccccc12 C1(C(=O)NC(CCC)C2CCCC2)(CNC(=O)COC2CCC2)CC(C)(C)C1 c1(CC)cc(C(=O)NC2(C)CC(NC(C3(C)CCOCC3)=O)C2)ccc1O CCC(C)CCCCC(=O)NCc1ccc(C(=O)NC(c2cnsc2)C)cc1 C1(O)(CCNC(C(C)c2cccs2)=O)CCN(C(=O)Cc2nncn2C)CC1 c1(OS(C)(=O)=O)ccccc1Oc1ccc(Br)cc1 c1(C(=O)Nc2nc(C)c(C(N3CC(F)(F)C3)=O)s2)cc2n(n1)CCCC2 C1(CC=C)(C(=O)NC(CNC(=O)C(=O)NC2CC2)CCC)CC=CCC1 c1(CC)ccc(C(=O)NCC2CCN(C(=O)Cc3csc(CC)n3)C2)s1 C1(NC(CCC(C)N(C)C)=O)CC2CC(NC(C3(c4ccno4)CCC3)=O)C2C1 c1(C(=O)NC(C)CCNC(C2(C)CCCC2(F)F)=O)n[nH]c2ccccc12 c1(C(N(CC(C)NC(=O)CC(O)C2CC2)C)=O)cc(C(N)=O)co1 C(=O)(C1CCN(C)c2ccccc21)NC1(CNC(C(C)OCC)=O)CCCC1 N1(C(=O)C=CSc2nc[nH]n2)CCC2(C1)CN(C(C1(F)CCCOC1)=O)CCO2 N(C(=NCCc1cccs1)NCC1CCN1C)C(c1ncc(C(C)(C)C)o1)C CCC(CN(C)C)CC(=O)N1CCC(CNC(C2CCCCN2C(C)C)=O)C1 c1(C(=O)NC(c2ccccc2)C(=O)NC2CC(C)(F)C2)ccnc2cc[nH]c12 c1(CCC(=O)NC(C)CCN(C(=O)C(C)NC(N)=O)C)ccc(N(C)C)nc1 c1(C(=O)NCCN(CCC)C(c2cccc(CC)c2)=O)ccc2nccn2c1 Cc1c(C(F)(F)F)nc(N2CC3C(CNC(C4CCOC4)=O)C3C2)nc1Cl c1(CC)ccc(C(N2CCCC2CN(C(=O)C(C)C(F)(F)F)C)=O)c(C)n1 C1(CCNC(C(CSC)O)=O)CCN(C(=O)C(C(C)C)N2CCCCC2)CC1 C1(NC(c2cccc3ccccc23)=O)C2CC(O)C1N(C(c1occc1F)=O)C2 C1(NC(C2(CC)CCC2)=O)CC2(C1)CC(NCc1c(O)n[nH]c1C)C2 C1(CC=C)CCCC1NC(C1CC1CNC(=O)CC1CCSC1)=O C(=O)(C(O)(C(C)C)C(F)(F)F)N1CC(CCNC(C(C=C)(C)C)=O)OCC1 C(CCCC(C)NC(=O)C(COC(C)C)NC(C)=O)NC(CCOCC#C)=O C=CC(CC)CC(=O)N1C2CCC1C(CNC(C1(NC(C)C)CC1)=O)C2 N1(CC)CCOCC1C(=O)NC1(CCCC(=O)N2CC(C)(CF)C2)CCC1 C1(CC)CCC(C(=O)NC2(CCOC)CCN(C(C3(CO)CC=CC3)=O)C2)CC1 c1(C(=O)NCC2(C(=O)NCC(O)CN(C)C)CC(C)(C)C2)cncc(C#N)c1 N1(C(C2C(C)CCS2)=O)CCC2(CCC(NC(=O)CCC3(C)CC3)C2)C1 c1(C(N(C2CN(Cc3ccc(Cl)o3)CC23CC3)C)=O)cc(Cl)ccc1Br C1(C(C(N2CC3C(CNC(C4(C=C)CCC4)=O)C3C2)=O)OC)CCCCC1(C)C CC1(C)C(C(N2CC=C(CCNC(=O)Cn3ccnn3)CC2)=O)CCS1(=O)=O C1(OC)CC2CC(NC(=O)C(C)N(C(=O)CCc3cnn(C)c3)C)CC12 CCCC(C)(C)C(=O)NCC(C)NC(=O)C(C)(O)CCC C=CCCCCC(=O)N1CCOCC1C(=O)NC1CCC(O)C1 CC1(C)C(NC(c2ccc(Cl)cc2)=O)C2CCCN(C(=O)C(F)n3cccn3)C12 CN1CCN(C(C2CCN(C(=O)c3cc([N+](=O)[O-])n[nH]3)O2)=O)CC(O)C1 C1(NC(=O)CCc2cncc(F)c2)COC2(CCN(C(=O)C=CCF)CC2)C1 C1(CC(=O)NCCN(C(C(C)CN2CCOCC2)=O)C)COCCOC1 N1(C(C(C)NC(COC)=O)=O)CCCC(CCNC(c2cncn2C)=O)C1 c1(C(=O)NCC(C)N(C(=O)C2=CC(O)CCC2)C)c[nH]c2cc(F)c(F)cc12 C1(NC(CC=Cc2ccc(C)cc2)=O)CCC(O)CN(C(=O)C(F)(F)C(F)F)C1 Cc1ccc(CC(=O)NCC#CCNC(c2cc(C)n(C(C)C)c2C)=O)c(Br)c1 C1(C(=O)NCC2C(C)CN(C(=O)CC3CCCCCC3)C2)CCCCC1(F)F c1(C(=O)NC2COCCC2NC(C2CC3(CC3)CO2)=O)ccc(N2CCCC2)nc1 c1(N(CCNC(C)=O)C)nc(N2CCCC(C)(F)C2)nc2ccccc12 C(=O)(C1=CC2C=CC1C2)NCCOCCNC(C(C)S(N)(=O)=O)=O CC1CC(NC(=O)CCC=CBr)CCN1C(=O)CC1CC2(CC2)CO1 N1(C(CN2CCN(C)CC2=O)=O)CC2CN(C(=O)Cc3nncn3C)CC2(C)C1 CC(=O)C(C)CC(C)C(=O)NCC(CNC(=O)C#CC1CCCCC1)S(C)(=O)=O c1(C(=O)NCCCC(C)NC(C(N2C(=O)CCC2=O)CC)=O)cnc(C)c(C)c1 n1(CC(=O)NCC(CCNC(CC=C=C)=O)O)ccc(=O)n(C)c1=O C(=O)(C1=CCCOCC1)NC1C2(CCN(C(c3c[nH]c(=N)s3)=O)C2)C1 C1(C)(NC(C(COC)NC(=O)CCc2ccoc2)=O)CCC(C)C1 C(N=c1[nH]c(=NCCCn2ccnc2)[nH]c2c1CSC2)c1cc(C)c(Br)cn1 c1(CC(N2C(C(=O)NCCSCC)CCCC2)=O)c[nH]c2cccc(C)c12 C1(NC(c2c(Cl)cn(C)n2)=O)CC2CN(C(=O)CO)CC12 c1(C(N2CC(COCCCNC(C)=O)C(N(C)C)C2)=O)ccc(C)cc1C C1(C(CNC(C(F)=CC)=O)(C)C)CCN(C(=O)CCC2CCC(=O)N2)CC1 c1(C(=O)OC)ccc2c(c1)C(C(=O)N1CCC3(CC(CCO)C3)C1)CO2 C1(NC(C(CCC)=CCC)=O)CC2CCC(C1F)N2C(c1ccc(O)cc1F)=O N1(C(c2c(CC)occ2)=O)CCC2(CC1)CN(C(=O)COC(C)C)C2 C(CC1CCc2ccccc21)N1CCC(NC(c2n(C)nc(O)c2)=O)C(F)C1 C(c1cccc(F)c1Cl)=CC(=O)NCCN(CCC)C(c1[nH]c(=N)ccc1C)=O Cc1c(NC2CCC(CN)C2)cnn1-c1ccccc1 N1(C(CCc2ccc(C)c(Cl)c2)=O)CC(C)(C)OCC1CNC(=O)C(C)N(C)C C1(N(C(=O)Cc2cncn2C)C)CC2CCC(C1)N2C(c1cnc(Cl)c(N)c1)=O Cc1nc(S(C)(=O)=O)sc1CN1CCC(CCc2cccc(O)c2)C1 N1(C(CSCC=C)=O)CCN(C(=O)CC(C)C(F)F)CC1c1ccc(OC)cc1 CC(F)(F)CCC(=O)N1CCCC(NC(C2CC2(C)C)=O)C1 N1(C(C2C(NC(C3(CCOC)CCC3)=O)CCCC2)=O)CC(C)CC(C)C1 C=CCC(CNC(=O)CCc1cc(C)on1)C(=O)N(CC)CC1CCCO1 C1(C2=CCN(C(=O)C(=O)Nc3ncc(CCO)s3)CC2)(C(=O)OC)CCOCC1 Cc1ccc(F)c(C(F)(F)C(=O)NC(C)CC(C)NC(=O)CCC(=O)N(C)C)c1 C(=O)(CCCCCC(=O)OC)N1CC2C(COCC)(CCC2)C1 Cc1cn2c(n1)CC(C(=O)N(C(CNC(=O)COCC(=O)NC)C1CC1)C)CC2 C1(C)(C(=O)NC(CNC(CNC(=O)OCC)=O)C2CCC2)C=CCCC1 CC(F)(C(=O)NCC(O)CCNC(=O)CCCn1ccnc1)c1ccon1 c1(NC(C2CC(NC(c3ccc(C)s3)=O)C2)=O)cccc(S(F)(F)(F)(F)F)c1 CC1CC(C(=O)NC2CN(C)CC2(F)F)CN(C(c2cc3occc3[nH]2)=O)C1 c1(C(N2CCC(O)(CCNC(CSCC)=O)C2)=O)ccc(Cl)cc1CC CC(C)S(=O)(=O)c1ccccc1C(=O)NCC(F)CNC(=O)Cc1cnoc1 Cc1cnc(C(N2CCCC(F)(CNC(=O)C(C)OCCC(C)C)C2)=O)c(C)c1 c1(C(=O)NCC2CCC(CC)C2)ccc(C(C)(C)CO)cc1 Cc1cccc(C(F)(F)C(=O)NC2CC2CNC(C2COC(=O)N2)=O)c1 c1(OC)cc(C)nc(N2C3(CNC3)C2=O)n1.c1(SC)cnc(Cl)s1 C1(C)(C(=O)NCC(CC)(C)O)CCN(C(=O)Cc2cc(C)no2)C1 C(=O)(CC(C)CC(C)(C)C)N1CCN(C(CC(C=C)C)=O)C(C)CC1 C(=O)(C(CCCC#N)N1CCC(O)CC1)NC1(COC)CC1.c1(C)cccs1 C(=O)(C(C)(F)C(=O)Nc1ccn(C2CCC2)n1)OC.C12CCC(C)N(C1)C2=O c1(OC)ccnc(C(N2CC(N(C(=O)CC3CC3(Cl)Cl)C)C2)=O)c1 N1(C(=O)CCc2ccc(Br)nc2)CCC2C1CCCN2C(=O)Cc1cncnc1 CC1CC(C(=O)NCC2CN(C(c3ccnc(CO)c3)=O)C2)C(C)O1 C1(C(N(CC(=O)NC(C#C)C(C)OC)C2CC2)=O)C2CN(C)CC12 C1(NCc2ccc(C(=O)OC)o2)CC12CCN(C(C1CC1(F)Cl)=O)CC2 N1(C(c2cc(NC(C)=O)n(C)n2)=O)CC2(CC(CC(N3CCCC(OC)C3)=O)C2)C1 C(=O)(CCCCCCCC1CC1)NCC1CCCC(NC(CS(N)(=O)=O)=O)C1 C1(C(N(CC(CC)CC)C)=O)C(C)CCN1C(=O)CNC(=O)CN(C)C N1(C(Cn2cccc(C)c2=O)=O)CC(C)CN(C(=O)C2=CCCC2)C(C)C1 C1(C(=O)NCC2(F)CCCN(C(c3n(C)nnc3)=O)C2)CC12CCC(C)(C)CC2 C12(C(N(CCNC(=O)CCCC(N)=O)CC)=O)CCCC(CCC1)C2O N1(C(C(c2cn(C)nc2)=O)=O)CCC2(NC(c3ccc(Cl)s3)=O)CC2C1 N1(C(C)C(=O)NC(C)(C)CNC(c2ccn(C3CCCC3)n2)=O)CCCC(O)C1 C1(NC(C2C(C)CC(C)O2)=O)CCN(C(c2cocn2)=O)CCC1CO C1(C(N(CC(C)C)CC(=O)NC2CN(C)NC2=O)=O)CC(C2CC2)C1 c1(C(=O)NCCN(C(CC2CC(OC)C2)=O)C)cn(CCO)nc1-c1cccs1 C12(NC(Cc3n(C)ncc3)=O)CCCC1N(C(c1cn[nH]c1)=O)CCC2 c1(OCC)cc(C(=O)NC2CC(NC(c3cncc(N(C)C)c3)=O)C2)ccn1 C(N=c1nc(NC2CCCOC2C(C)(C)C)c2c([nH]1)CCOC2)c1c(C)noc1 c1(NCC(C)(C)C)ccccc1C(N(C(CCSC)C(=O)N(C)C)C1CC1)C N1(C(C2CN(C(C3CC(C)(CC)C3)=O)CC2(F)F)=O)CCCC(C2CC2)CC1 C(C(O)CC(=O)NCCN(C(c1ccc(F)o1)=O)CC1CC1)N(C)C Cc1cc(C)nc(SCC(=O)N(C)CCN(C)C(c2cc[nH]c2C)=O)n1 C=CCCC(O)CN(C)C(C1(CO)CCN(C(=O)CCn2ccc(C)n2)C1)=O C1(F)(CNC(C2(CC#C)CCC2)=O)CCN(C(c2ccnn2C2CC2(F)F)=O)C1 C1(CNC(=O)CN2CCSCC2)CCCN1C(=O)CCSc1ccccn1 CCCCC(O)CCC(=O)N1CCC(NC(C2COCCN2CC)=O)C1 CC(C)CCCCC(=O)NCC(C1CCC1)NC(c1c(Cl)cnn1C1CC1)=O CCCC(CNCC(N=[N+]=[N-])c1ccccc1)OCCC1CC1 CCC(C)(C(=O)NC1CC2(C1)CC2NC(=O)Cn1cnccc1=O)C(N)=O CC(C)(CF)C(=O)NC(CNC(c1cnn(-c2ccc(Br)cc2)c1)=O)C1CC1 C(=O)(C1=C(C#N)CCC1)N1CCC(CN(C(=O)CC2(N(C)C)CC2)CC)CC1 C1(NC(C=CCSC)=O)CCOCC1NC(c1ccc(SC(C)C)cc1)=O C#CCCC(O)C(=O)NCCCN(C1CCCC1)C(c1cc(COC)no1)=O C1(OC)(CNC(=O)CC2COCCOC2)CCN(C(=O)CNC(=O)CN(C)C)C1 c1(C(=O)NCC(CN(C(C(C)NC(COC)=O)=O)C)O)nccnc1C CCCC(C(=O)N1CCOCC1C)NC(=O)Cn1ccnn1 N1(C(c2cn(C(C)C)nc2)=O)CC2CC(C(=O)NC(C3CCOC3)C)(C2)C1 C1(C)(CNC(Cc2nnc(C)s2)C(=O)O)COC(C)(C)O1 c1(NC(=O)NC(C)C(C)n2cncn2)ccc(I)cn1 N1(C(c2ccc(C)[nH]2)=O)CCCCC1C1CCN(C(c2ncc(C)cn2)=O)C1 O=C1CCc2ccc(C(=O)NCC3CCN(C(c4ccc(Br)cn4)=O)C3)nc2N1 c1(CC)nnsc1C(=O)N(CCOCc1cccnc1)Cc1ccccc1 C1(C(C)C)C(=O)N1.C(CCC(=O)N1CCC1CNC(c1ccc(SC)o1)=O)OC C1(C(=O)NCC(C)CN(C)C(c2noc3ccccc23)=O)CC2C=CCC(C1)C2 c1(C(=O)NC2(CNC(CCCOCC=C)=O)CCOC2)cccc([N+](=O)[O-])c1N C1(C(=O)OCC)CCC(C(c2nnnn2C2CC2)Nc2ccsc2)C1 C(=O)(C(C)C(O)CC(C)C)N(CCN(C(c1cc(C)cc(O)c1)=O)C)C N1(C(CN2C(C)CC2)=O)CCOC2CN(C(c3cc(CCO)on3)=O)CC12 Cc1cc(C)n(CCC(=O)NCC(C2CCOC2)NC(c2nocc2Cl)=O)n1 c1(CNC(c2n(C(C)C)cnc2)=O)cnn(C)c1C(N1CC(COC(N)=O)C1)=O C1(CCNC(C(C)SCC)=O)CCCCN1C(=O)CCC1C(=O)ON=C1C C(CC1CCc2ccccc21)NC(=NCCCCC=C)NCC1(C#C)CC1 c1(OC)cncc(C(=O)NC(CO)C(=O)NCC(O)C(C)(C)O)c1 CCCCC(CC)OCCNCCOC(C)(C)C.C1CN(C)C(=O)O1 O=C1CCC2CN1CC(CN(CC(F)(F)F)Cc1cccn1C1CCCC1)O2 c1(C(=O)NCC2N(C(COCC=C)=O)CCCC2C)nnc2n1CC(=C)S2 C1(C(N2CCC(N(C)C(C3(CC4CCC4)CC3)=O)CC2)=O)CC2CCC1CC2 Cc1nn(C)nc1C(=O)NCCC1CN(C(c2conc2C2CCC2)=O)CCO1 c1(C(=O)NC)ccc(O)c(CNC23CC(NC(=O)CSCC(F)(F)F)(C2)C3)c1 C(=O)(C1=Cc2ccccc2OC1)NCC(CNC(Cc1c(O)ccc(C)c1)=O)F N1(C(C(CCOC)C)=O)CCOCC(NC(C2(COC)CC=CC2)=O)C1 c1(C(=O)NC2CN(C(CC3CC(=C)C3)=O)C3(C2)CCC3)cc2ccc(O)nc2s1 c1(C(=O)NC(C(=O)OCC)CS(C)(=O)=O)ccc(F)c2ccncc12 c1(C(N2CCC(OC)(CO)C2)C(=O)NC2COC2)cn2ccc(C)cc2n1 c1(C(=O)NC2CN(Cc3c(C)scn3)CC2C#N)ccc2cccnc2c1 c1(CNC(C(c2cnn(C)c2)C)=O)nc(C(=O)NCCCc2ccncc2)co1 C(=O)(C(C)P(C)(C)=O)NCCCN(C(c1nc(OC)oc1)=O)C(C)C C(=O)(C1=CCC(C)CC1)NC(C1CCN(C(C2CC=C(C)CC2)=O)CC1)CO N1(C(CC2CC(OC)C2)=O)CC(NC(C2(C)CC3CC3C2)=O)C(SC)C1 N1(C(=O)Nc2cnc(F)cn2)CCC(C2CCNC2)C1 C(=O)(C(CC)ONC(=O)C1(NC(=O)C2CC2)CC1)N(CC(=O)N(C)CC)C C1(C(=O)NC2(C)CCCN(C(C(C)C)=O)C2)CCn2nnnc2C1 c1(C(=O)NC(CCCC)CNC(=O)CSCC(=O)NC)ccc(CC)cc1Cl CCC(CC(=O)N(C(C)CO)C1CC1)NC(C1COCC1(C)C)=O CCC(C(=O)OC)C(=O)N(C(C(=O)NC1CC(F)C1)C1CC1)C c1(C(CO)NC(C2C3CCC2(c2ccnn2C2CCCC2)C3)=O)ccccc1F c1(-c2n(CC)nc(CCc3cnn(C)c3)n2)cc(SC)ccc1C c1(OC)ccc(OC)c(C(N2CCC(CCNC(=O)CCC3CC3(Cl)Cl)C2)=O)c1 c1(C(CC)CNC(C2(CNC(=O)OC(C)(C)C)CC2)=O)ccnn1C CCCCC(CC)CC(=O)N1CCOCC1CNC(c1cc2n(c1)CCOC2)=O c1(CSCCC)ccc(C(N2CC(NC(=O)CCCC3CC3)C2)=O)o1 CN1C(=O)C(F)CC1C(=O)NC1C2CN(C(C3CC4C=CC3C4)=O)CC12 C1(F)(C(=O)NC2CC(N(C(C3CCC(CC)CC3)=O)C)C2)CCN(C)CC1 c1(C(N2CCOCC(CNC(C3C(C)CCCC3)=O)C2)=O)nccc2[nH]ccc12 C1(CC(=O)N(C2CN(C(c3cc(C#N)on3)=O)CC2O)C)CCOC(C)(C)C1 C1(CCCCNC(C2C3CCCCC23)=O)CCCN(C(=O)Cc2cnc[nH]2)C1 C1(C(N(C23CC(C2)C3)CC)=O)CN(C(=O)CC2C=CCC2)CC1C(C)C c1(NC)cncc(C(=O)NCC2(CCO)CCCC2)n1 c1(CC)ccc(Br)cc1C(=O)NC1CC(NC(=O)C(c2cnn(C)c2)=O)C1 C1(=O)C(C)N(C)C(=O)C2(CC2)CCCN1CC(=O)NC.C(C)(C)(C)OC(=O)C1CC1 C(=O)(CCCC(=O)N1CC2CC(CNC(C3COCCO3)=O)C2C1)N(CC)CC C1(C#CC(=O)N2CC(C)(NC(=O)CCc3nccs3)C2)(CC)CC1 C1(CC(N)=O)(NC(C(C2CCCO2)OC)=O)CCN(C(=O)Cc2cncs2)CC1 C1(NC(C(C)(C)F)=O)CN(C(=O)CCc2cc(F)ccc2Br)CCC1CO CC(C)CC(CNC(C1CCCSC1C)=O)C(=O)N(CC(O)CO)CCO c1(C(=O)NC(C(C)C)C(C)NC(=O)CN2C(=O)CNC2=O)nccc(N)c1Cl c1(OC)ccc(S(C)(=O)=O)cc1C(=O)NC1CCN(C(=O)CC(O)C(C)C)C1 c1(C(N2CCC(N(C(c3scc(C)c3)=O)C)C(C)C2)=O)c[nH]c2cccc(C)c12 c1(C(N(CCCNC(=O)CCOC2CCC2)C2CC2)=O)c[nH]cc(Cl)c1=O N1(CCC)C(=O)CCC1C(=O)NCCN(C(=O)C(c1cccc(C)c1)O)C1CC1 N1(C(COCCOCC)=O)CCC(CNC(=O)Cc2cnoc2C)(CC)CC1.O Cc1cncc(CC(=O)NCC=CCCCCNC(=O)C=CCO)c1 C1(C(C)C)CNCCN1S(=O)(=O)C(F)(F)F.c1(C)ncccc1Br C12(NC(=O)CC3C=CCC3)CCC(CC1n1cc(C3(O)CC3)nn1)C2 c1(C(N2CCCC(F)(CO)C2)=O)nnc2ccc(-c3ccc(F)cn3)cn12 N1(C(C=CCNC(CC2CC(SC)C2)=O)=O)CCC(C=C)CC1 C(=O)(CC(C)N=c1nc(NCC(c2ccccn2)C)c2c([nH]1)c(C)nn2C)NC C(CC(=O)NCC1(F)CCOC1)(C(C)(C)C)NC(C=CC(N1CCCC1)C)=O C1(NC(C2C(OCC)C2C)=O)CN(C(=O)CCCSC)CC1(C)C c1(NC(CC(=O)NCC)=O)cccc(CNCC(C2CC(C)(C)C2)O)c1 C(C(C(=O)NCC1CCN(C(=O)CCCNC2CC2)C1)c1ccccc1)OC c1(C(N(CCC2CCN(C(C=C(C)Cl)=O)CC2)C)=O)noc2c1CC(C)(C)CC2 c1(OCCC)ccc(C(=O)NCCC2(CNC(c3conc3C)=O)CC2)cc1 Cc1cc(C(=O)N(c2nc(C)c(-c3nn[nH]n3)s2)CC(C)C)nnc1C c1(CC)cc(C(=O)N(C(C)CNC(C2CCC(NC(C)=O)CC2)=O)C)cc(Cl)c1 C1(NC(CCCCC)=O)CCN(C(=O)CC2CCN(C(C)C)CC2)CC(O)C1 CC1(NC(=O)CCC2CCCCC2)CCN(C(=O)CNC(C2CCC2)=O)CC1 Cc1cnncc1C(=O)NC12CC(C(=O)Nc3cccnc3N(C)C)(C1)C2 c1(CCNC(c2ccc(NC(=O)OCC)cn2)=O)c(C)nn2c(C)cc(Cl)nc12 N1(C(C2CC(CC)C2)=O)CC(O)CC1(C)C(=O)NCCCC(F)F C(=O)(C(CC=C)CC(C)C)N1CC=CC(C(=O)NCC(CCC=C)O)C1 Cn1c(O)nc2c(C(=O)NC3C4CN(C(C5(O)CCOCC5)=O)CC34)cccc12 CC(O)C(F)(F)C(=O)NCCN(C(c1cc(CO)cn1C)=O)Cc1ccccc1 Cc1ccc(OCC(=O)NC2(O)CCN(C(=O)C3=NOC(C)C3)C2)c(Br)c1 C1(CN(C(=O)C(F)C2CC2)C)CCN(C(=O)CCc2cncs2)C1 C1(CNC(C=C(C)Cl)=O)(CO)CC12CCN(C(C1CC(CCO)C1)=O)CC2 c1(CC(=O)NCC2C(CNC(CCCSC(C)(C)C)=O)C2)ccc(S(N)(=O)=O)s1 c1(NCCN(C(CC2C(CC)C2)=O)CC)ncc(C(N)=O)cc1Cl C#CCC(C(=O)NC(C)(C(=O)NC(CC1CC1)CO)C1CCC1)C1CC1 C12(CNC(c3ccc(CCC)cc3)=O)CCCN(C(c3ccncc3C)=O)C1C2 c1(NC2(CNC(c3cnn(CCF)c3)=O)CCOCC2)c(F)cccc1[N+](=O)[O-] C1(CC(=O)NC(C)CC2CCOC2)CN(C(C2CC2C(C)(C)C)=O)C(C)(C)C1 C1(C(=O)NCC2(NC(=O)CC3(n4ccnc4)CC3)CCC2)C2CC2C2CC12 C1(NC(COCC=C)=O)CC(C2CCN(C(=O)C(C)(C)CF)C2)C1 C1(C2CCN(C(c3cc(C(=O)OC)oc3C)=O)C2)(NC(C(CC#C)C)=O)CC1 Cc1ncncc1C(=O)NCC1CN(C(=O)C(c2ccc(Br)s2)C)CCO1 NC(=O)CCCCC(=O)NCC1CCCN1C(C1CC(c2ccc(O)cc2)C1)=O C(=O)(C1SCc2cccnc21)NCC(CC)NC(c1cccc2ncnn12)=O C1(CNC(CSC)=O)CC2(C1)CN(C(c1ccc(OC(C)=O)cc1)=O)C2 Cc1cc(C(=O)NC2CCC(CNC(=O)CSc3ccc(Cl)cc3)C2)nc(O)n1 c1(C(=O)NCC(C(C)C)NC(=O)C(=O)C(C)(C)C)cc2c(o1)CCCNC2=O c1(C(=O)NC2(C)CCN(C(C(C=C)O)=O)CC2)cn(C)c2ccc(Cl)cc12 CC1CCCN(C(=O)Cn2cnnc2O)C1CCNC(c1cc(Br)no1)=O c1(N2CC(C)(C)C(NC(=O)COCC3CC3)CC2)ncc2c(n1)CCOC2 N1(c2cc(OC)c([N+](=O)[O-])cc2)CC(C)CN(C(=O)CCC(C)(C)C)CC1C N1(C(C2(COC)C=CCC2)=O)CCOC2(C1)CN(C(C1C=C(C)CS1)=O)C2 C1(CN(C)C(c2noc(C3(C(F)(F)F)CC3)n2)=O)CCN(c2nnc(C#N)s2)CC1 C1(CC)CC(C(N2CC(NC(c3cnn4ccsc34)=O)CC(C)C2)=O)CC(=O)N1 N1(C(C(CSC)OC)=O)CCC2CN(C(c3cnc(O)cc3C)=O)CC2CC1 c1(CC)nc(C(=O)N(C(C)CNC(=O)CCCC2CCCCC2)C)c(C)o1 Cc1[nH]nc(Cl)c1C(=O)NC(C)CCN(C(=O)CCCC1CCCC1)C c1(OC)ccc2c(C)c(C(=O)NCC3CC(NC(=O)C(C)=C4CCC4)C3)[nH]c2c1 CC1CN(C(=O)C2=CCCC2C)CCC1C(N1CCOCC1)=O c1(NC(C(c2cccc(OCC)c2)C)=O)cc(C)c(C(=O)O)c(C)c1 N1(C(c2nc(CC)on2)C)CC2(CC(NC(=O)COC(C)=O)CO2)C1.O Cc1ncc(Cl)c(C(N2CCN(C(c3ccsc3C(F)F)=O)C3CC23)=O)n1 CCCCCCC(C)C(=O)NC1CCC(NC(c2ccc(C(C)(C)C)cn2)=O)C1 c1(C(C)OCC)cn(CCCN(C(=O)C(CC)N(C2CCOCC2)C)C)nn1 N1(C(c2cnc(CC)s2)=O)CCC(F)(C(=O)N(C)Cc2sccc2C)CC1 N1(C(C(C2CCC(C)(C)CC2)C)=O)CC2CC(C1)N(C(=O)C(=O)N=S(C)(C)=O)C2 CC1CCOCCN1C(C1CC(O)CCN1C(c1cccc[n+]1[O-])=O)=O c1(C(=O)OC)ccc(CC(=O)NCC2(NC(C3CCS3(=O)=O)=O)CCOC2)c(Cl)c1 C1(NC(c2onc(C)c2C)=O)COC2(CCN(C(=O)CCN3CCCC3=O)C2)C1 CC1CN(C(C)C(=O)N2CC(CC(C)NC(=O)COCC(F)(F)F)C2)C1 CC(C)C(O)C(C)C(=O)N1CC2CC(C(=O)NC34CC(F)(C3)C4)(C2)C1 c1(C(N(C2CCN(C(=O)COCc3cc(C)no3)C2)CCC)=O)cnnn1CC c1(C(=O)NCCN(C(=O)C(F)CC2CCC2)CCC)c[nH]c2cc(F)c(F)cc12 C1(NC(CNS(N)(=O)=O)=O)CCN(C(c2ccccc2O)=O)C12CCC2 C1(NC(CNS(NC)(=O)=O)=O)COCCC1NC(C1CC(OC)C(OC)C1)=O C1(CC(=O)NCCCCN(C)C)CC2(C1)CN(C(=O)CCc1ccoc1)C2 C(CC1CCCC1)(C(=O)N(C)C(C1CCCC1)C)OC N1(C(C(CCC2CC2)OC)=O)CC(C2CN(C(=O)Cc3ccoc3C)C2)C1 c1(NCCC2N(C(c3cn(CCC)nc3)=O)CCCC2)ncc2ccnc-2[nH]1 c1(C(C2N(C(=O)Nc3cn(CC)nc3C)CCC2)(C)C)ccc(C#N)cc1 c1(C(C(=O)NC(C)C(=O)OC)N(C(C#C)C)C)ccccn1 N1(C(CCN(C)CC)=O)CCN(C(=O)Cc2ccc(S(C)=O)cc2)C2(CCC2)C1 CCN=c1[nH]cc(C(=O)NC2CCC3(CCC3)C2)s1 N1(C(c2cc(C)n(C)c2)=O)CCCC2C1CCN2C(=O)Cn1cnc(C#N)n1 n1(CC)nc(C)c2cc(C(=O)N(c3cc(Cl)ccc3C)CC(F)F)sc12 C12(CN)CN(C(=O)CSCCC3CCCN(S(C)(=O)=O)CC3)CC1CCCO2 CCC(CC(=O)N1CCN(C)C(C(=O)NC(CC(C)C)C(N)=O)C1)C(F)F Cc1c(C(N2CCC3C(CCN3)C2)=O)cc([N+](=O)[O-])cc1Br O=C1CC(NC(C2(NC(C3CCCC3CF)=O)CC2)=O)CC(=O)N1 C1(CC)C(C(=O)NCC(C)(CO)NC(c2ncccc2C)=O)CCN1C c1(C(N(CCCNC(=O)C(C)n2ccnn2)CC)=O)cc(C#N)ccc1Cl C1(C(=O)NCCN(C2CCCC2)C(c2cc(C)ns2)=O)Cc2ccc(F)cc2C1 Cc1nncc(C(N2CCOCC2C(N2CC(CC(C)(C)C)C2)=O)=O)c1C c1(CC(N2C3CCN(C(CC(C)C(F)F)=O)CC3C2)=O)ccc2c(n1)OCCO2 c1(CN(C(=O)C=CC2CCC2)C)cccc(CNC(C2CCC(=O)N2)=O)c1 c1(CC)nc(Cl)c(CC)c(=NCCC(C)NC(C2(O)CC3CCC2C3)=O)[nH]1 C1(O)(CCNC(c2nncc(C)c2)=O)CCN(C(C2CC(=O)N(C)C2)=O)CC1 C1(NC(COCC(=O)OCC)=O)C2CCC(C2)C1C(=O)NCCCCN(C)C c1(N2CCC(N(C(C3CCCCC3(C)C)=O)CC)C2)nc(O)c2c[nH]nc2n1 c1(C(=O)NC(c2ccccn2)C)ccc(Cl)nc1NCc1ccc(I)o1 Cc1cc(C(=O)NC(C)C(C)NC(c2cc3c[nH]nc3s2)=O)c(C)n1C N1(C(C=CCC(C)(C)NC(c2c(C)occ2)=O)=O)CC(C2CC2)C1C1CC1 CON=CC(=O)NCCC1CCN(C(c2c[nH]nc2-c2ccc(Cl)s2)=O)C1 C#Cc1cccc(CC(=O)NC2C3CC2CN(C(=O)C=CC(C)C)C3)c1 n1(-c2cn(CC)nc2)nc(-c2ccccc2CO)nc1C1CNC(=O)N1C N1(C(CC2(OC)CCC2)=O)CC(NC(=O)C(=O)Cc2ccc(F)cc2)CCC1C N#CC1(C(=O)NCC2(CNC(=O)C(O)C3CCC3)CC2(F)F)CC=CC1 C(=O)(CCCCC(=O)OCCCN(CCC#C)C)OC Cc1ccc(-n2cc(COC3CCN(C(C4CCC(N(C)C)C4)=O)C3)nn2)cc1 CC1(C)CN(C(=O)C=CBr)CC(C)(C)C1NC(=O)CC1CCC1(C)C C1(NC(CCOCCOC)=O)CC(C)(CNC(=O)CC2(OC)CC2)C1 C1(C(N2CCN(C(C)CNC(C3CC4(CCC4)C3)=O)CC2)=O)(CC)CCNC1=O C1(NC(C(N)=O)=O)CC(NC(=O)Cn2nc(Br)c(Br)n2)C12CCC2 C1(C(=O)NCC=CCNC(C2CCCC(N(C)C)C2)=O)CC12CCCCC2 Cc1cccc(C(=O)NC(CO)C(C)NC(=O)CC2SC(=N)NC2=O)c1O C(=O)(CC(C)(O)COC)NCC(C1CCC1)NC(C1(COCC)CC1)=O C1(CNC(c2cc(OC)no2)=O)CCCC2(CN(C(=O)C(C)C3CC3)C2)O1 C1(C(N(CC(C(=O)OC)C)C)=O)(NC(=O)C=Cc2cocn2)CCC(C)(C)C1 CN1CC(NC(C2COCCN2C(c2cccs2)=O)=O)C(C)(C)C1 C1(C(N2CC(CNC(C#CC(C)C)=O)C2)=O)Cc2nccn2C1 Cc1ccc(I)c(C(=O)NC23CC(NC(=O)Nc4ccc(I)cc4)(C2)C3)c1 C1(C(=O)NC2C(C)N(C(c3ccn4ccccc34)=O)CC2)OC(C)(C)OC1(C)C C(=O)(C1CCCn2ccnc21)N1CC2CC(NC(C3CCOC3)=O)C2C1 CCCC(O)C(=O)N(C)CC=CC(=O)NCC(c1ccccc1)C C(=O)(C(F)(F)CCn1cc(C(C)(C)O)nn1)N(C)CCC(CCO)C1CC1 c1(C(=O)NCc2ccc(-c3c(O)cccc3O)cn2)ccc2c[nH]nc2c1 Cc1ccc(CNC(=O)N(CC(=O)NCC2(C)CCC2)C)o1 C=CCC(C)C(=O)N1CC(CNC(=O)C(c2c(C)noc2C)CC)(COC)C1 C1(C(N(CCCCC)CCO)=O)CC2(CCC2)CN1C(=O)CC1CCCSC1 C1(NC(CC2C(C)(C)OCC2)=O)C2CCC(C2)C1C(=O)NCC(O)C1CC1 CC1(CNC(c2ccsc2)=O)COCCN(C(C2CC3CCCC(C2)C3)=O)C1 c1(CNC(c2nc(OCC)sn2)=O)cccc(CNC(C2(F)CCCOC2)=O)c1 c1(C(=O)NCC2CC(NC(C3C(C=C)C3)=O)C2)ccc(CO)nc1 N1(C(=O)NCc2ccc(O)cc2I)CCC2(CCc3ccccc32)C1 c1(OC2CN(C(=O)Nc3c(CC)[nH]nc3)C2)ccc(F)c(Cl)c1.OCC CC(C)C(CC(=O)NCCN(C(=O)CCc1cncs1)C(C)C)c1ccon1 N1(C(C(C(CC)C)N(C(=O)C=C(C)C(C)(C)C)C)=O)CC2(COC(C)(C)C2)C1 c1(C(=O)NCC2CN(c3nc(C(F)F)ns3)CCO2)ccc(O)c(C2CC2)c1 N1(C(Cn2c(C)csc2=O)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C(C)C1C C(CCCC(=O)NCCC1(NC(=O)CCC(=O)c2ccc(N)cc2)CCC1)SC N1(C(C(C(C)C)SC)=O)CCN(C)C(CNC(c2ccc(F)c(F)c2)=O)C1 C1(c2n(CCCOC)nnn2)(NCC2CCC(CO)O2)CCN(C2CC2)CC1 C1(CN(C(=O)CCCn2cccn2)C)CCN(C(=O)C(C)(O)c2ccccn2)C1 C(=O)(CCC(=O)NCCCCCN(C(=O)CSc1ccccc1C)C)NCC C1(NC(c2cc(CC)on2)=O)CN(C(C2CC2[N+](=O)[O-])=O)CCC1O N1(C(C(=O)NC(C2CCNCC2)C)=O)Cc2cc([N+](=O)[O-])ccc2N2CCCC2C1 CC(C)(C(=O)N1CC2CCC1C(NC(=O)CCCCN1CCCC1)C2)C(F)(F)F N1(CCCC)CCCCC1C(=O)NCC(C)(C)CNC(c1ocnc1C1CC1)=O CC1(C(=O)NCC=CCN(CCO)C(C23C(=O)C4CC2C3C4)=O)CC2CCC1C2 C1(c2nnnn2C2CCOCC2)(NCCCCCC)CCC(=C2CCC2)CC1 N1(C(c2c(CC)occ2)=O)CCC2(CC(NC(=O)COC(C)C)CO2)C1 CC(C)(C)C#CC(=O)N1CC2CC1C2C(N1CCC2(CC1)CC2)=O N1(C(Cc2ccc(OC)cn2)=O)CCCCCC1COC(c1cnncc1O)=O CC(C)(C)S(=O)(=O)CC(=O)NCC(C1CCOC1)NC(=O)CCC(F)(F)F c1(C(=O)NCC2C(CNC(C(c3c(C)cncc3)C)=O)C2)cc2c(ncn2C)s1 c1(C(N2CCC(C(N3CCC(CC)C3)=O)CC2)=O)cccc(Br)c1Cl c1(CC(=O)NCCC2CN(C(Cc3cc(C)no3)=O)C2)ccnc(Cl)c1F N1(C(c2ccnn2C)C(=O)NC(C(=O)OC)C)CC(O)CC(O)C1 Cc1ccc2c(c1)SC(C(=O)NC1CN(C(C3(Cl)CC3)=O)CCC1C)C2 N1(C(Cc2nc(=N)[nH][nH]2)=O)C2CCCC1CC(NC(C1CCCCS1(=O)=O)=O)C2 CC1(C(=O)NCc2cc(Cl)cc(Br)c2)CCN(C(=O)Cn2nccn2)CC1 C(F)(F)(C(F)(F)F)OC(C)(C)C(=O)NCC1(F)CCC(NC(S(C)(=O)=O)=O)C1 C(=O)(C(C#N)C(=O)c1ccc(N2CC(C)OC(C)C2)cc1)NCCCOC c1(C(N2CCC(OCC3CC3)C2)C(=O)NC2CCC2)cnn2ccccc12 N1(C(Cc2cn(CC)nn2)=O)CC2(C)CCC1C2.c1(C2C(C=O)C2)ccccc1 C1(CC(=O)NCc2ccncc2)OCC2CCN(C(C3CC=CCC3)=O)CC12 C(=O)(C1CCCc2nncn21)N1CC(NC(=O)CCOCC2CC2)CC2(C1)CC2 N1(C(CC2N(C(C(C)SC)=O)CCC2(C)C)=O)CCC2(CC(F)C2)C1 Cc1ccc(C(C)C)cc1C(N1CC(NC(=O)CC2COCCO2)C(C)(C)C1)=O CN1CC(C(=O)NC2CCCCN(C(=O)CCn3cc(Cl)cn3)C2)OCCC1=O C1(C(N2CCCN(CC=C)CC2)=O)C2CC(O)C(C2)N1C(C1CC1(C)C(F)F)=O c1(C(N2C(CN(C(C(C(C)C)O)=O)C)CCC2)=O)c(F)ccc(C#N)c1F O=C(C1=C(F)CNCC1)NC1(c2cc(Br)ccc2Cl)CCC1 C(=O)(Nn1cnnc1)C1(C)CCCN1C(c1ccccc1CC#N)=O C=CC1CN(C(=O)C(C)(O)C2CCOCC2)CC1NC(C1COCCOC1)=O Cc1cnccc1C(=O)NCC1(C)CCN(C(=O)CSc2nccn2C)C1 c1(C(=O)NC2CN(C(C34CCC(OC)C3C4)=O)CC2O)sc(Cl)c(Cl)c1C C1(CNC(COc2ccn(C)n2)=O)CCCCC1C(N1CCCC(C(N)=O)C1)=O C#CCC(C)(C(=O)NC1(C2CCCCO2)CC1)NC(c1cn(C)c(C)n1)=O CC1=C(C(=O)N2CCC(N(C(=O)C(O)C(C)C)C)C2)S(=O)(=O)CCO1 C1(NC(CC2CCC(C)(C)O2)=O)CN(C(=O)Cc2cc[nH]c2)CCC1F C1(C)(OCCN(CC(=O)NCC)C(=O)CC2CCC3CC23)CCOCC1 C(=O)(C1=CCCCCC1)NC(C(CO)NC(CCOc1c(CC)cccc1)=O)C c1(OCC(=O)NC2CC(OC)C(O)C2)cc(Br)cc(F)c1F Cn1cc(C(=O)NC2CCN(C3CCN(C(=O)C=CC=C(Cl)Cl)C3)CC2)ncc1=O C(=O)(N=c1[nH]n(C)c2cc(Br)cnc12)NC1(CC)CCOCC1 c1(OC)cnc(C(=O)NCC=CCNC(C2CCN(C)C2)=O)cn1 O=C(O)CCC(Cc1ccccc1)NS(=O)(=O)CCC1CCCO1 CCC(CC(=O)N(C)Cc1ccccc1CNC(=O)CCOCC(F)F)C(F)F Cc1n[nH]c(C)c1C(=O)NCC1C(C)CCN1C(=O)C(=O)Cc1ccc(Cl)cc1 CCC(N=c1[nH]c2c(c(=NC(C)c3ncc[nH]3)[nH]1)COC2)c1c(C)noc1C C(=O)(C1=CC2(CCOC2)C1)NC1C2CN(C(CC(C=C)(C)C)=O)C1C2 c1(CC(=O)N(C(C(=O)NC2CC=CCC2)C2CC2)C)ccn(C)n1 c1(C(=O)NC(CC)CNC(=O)C=CBr)ccc(S(=O)(=O)N2CCOCC2)cc1 C1(C(N(CCC2CN(C)C2)C)=O)C(C2CC2)CCN1C(c1cc(Cl)cs1)=O c1(CCN(C)C(=O)NC(c2cccs2)CC2CC2)nn[nH]n1 N1(CC)CCCC(ONC(=O)CN(C)C)C1.c1(C2NOCC(=O)N2)ccccc1 c1(N(CC(C2CC2)OC)C)nc(=NCCC2(CCO)CC2)[nH]c2c(F)cccc12 c1(CC)cc(C(N2CCC(CN(C)C(C3(C#N)CCOC3)=O)C2)=O)cn(C)c1=O c1(C(=O)NCCC2(O)CN(C(CSC)=O)C2)ccc([N+](=O)[O-])c(SC)c1 C=C=CCCC(=O)NCC1CCN1C(c1cc(SC)c(C)o1)=O CC1CCN(C(=O)C=CC(=O)OC(C)(C)C)CC1CNC(c1ncn(C)n1)=O N1(C(Cn2cnc(=N)[nH]2)=O)CC2C=CC1C(C(=O)NCCC1CCC(=O)N1)C2 c1(C(N2CCC(CCNC(=O)CCOCC(F)F)C2)=O)ccc(F)c(O)c1F C1(NC(c2cnsn2)=O)CC2CC(C1)N(C(=O)CN1CCOCC1)C2 C1(NC(c2scc(C)c2C)=O)CS(=O)(=O)C2CN(C(=O)CN(C)C(=O)C3CC3)CC12 C(=O)(CCCCCC#N)N(C(CCNC(c1c(C)ccc(C)c1)=O)C)C CCC(C(=O)NC1CC(CCC(=O)N(CC(C)C(C)C)C)C1)C(C)(C)CC c1(CC)cccnc1C(=O)N(CCCNC(=O)C=C1CCC(C)CC1)C C1(C(=O)NCCc2ccccn2)CCN(N2CCCCCCC2)CC1 Cn1nnc(C(N2CCCCC2Cc2nn[nH]n2)=O)c1-c1ccccc1 C1(CNC(C(CC)F)=O)CCN(C(c2ccc[nH]2)=O)CCC1(F)F C(CS(=O)(=O)CCNC1CCOCC1NC(=O)CN1CC(OC)CC1CO)OC c1(OC)ccc(C(O)C(N2CC(NC(C3(F)CC=CC3)=O)C3CC23)=O)cc1 c1(CN2C(CNC(N(CCCSCC)C)=O)CCC2)ccccc1 C1(C(=O)OCCSC(C)(C)C)CCCCN1C(C1CCCC1c1ccccc1)=O c1(C(N2CCC(N(C(=O)C(C)CF)CCC)C2)=O)c(C)cc(Cl)cc1C N1(C(c2c(C)nc(C)o2)=O)CC(NC(=O)CC2NC(=O)CNC2=O)CCC1C N1(C(C2C(C(=O)OCC)C2)=O)CCC(C)(NC(=O)COCCc2cccs2)C1 C(=O)(N=c1nc(-c2ccccc2)[nH]n1Cc1ccsc1)N1C(CC)C(=O)NCCC1 C#CCCC(C(=O)OC)NC(=O)CC(O)CNC(=O)C(=O)NCC C(C)(C)(CC(F)C(=O)NC1CCCCN(C)C1=O)NC(CC(=O)NCC)=O c1(C(N2CCN(C(C(COC)(F)F)=O)CC2)=O)c(C)cnc2ccccc12 N12CC3(CCN(CC3)CC1=O)C2.Cc1cc(Cc2c(C)cccc2Cl)cc(O)c1 c1(CNc2c(C(=O)OCC)n3c(n2)CCC3)nc(C)c2ccccc2n1 C1(CC)CN(C(C2CC3CCC(C2)O3)=O)CCN1C(=O)C=CC(C)C C1(CNC(C=CS(C)=O)=O)CN(C(C2CC(=C3CCC3)C2)=O)CC2(CCC2)O1 c1(CC)cc(=NCC2CCN(C(C3CC4CC4CC3C)=O)C2)[nH]c(COC)n1 C(=O)(CCCC(c1nnnn1-c1cccc(OC)c1)NCC1(CO)CC1)OC c1(OCC(=O)NCC23CCCCC2C3)ccc(Br)cn1 c1(CC(N2C(C)CN(C(=O)CCC(C)CN(C)C)CC2)=O)cnn2c1CCCC2 c1(C(N2CCC(CCC(=O)NC(c3cnn[nH]3)C)C2)=O)ccn(C)c(=O)c1 c1(C(c2n(CCC)nnn2)NCCCOC2CCOC2)ccn2ncc(Br)c2c1 C=CCN=C(NCCS(=O)(=O)CC)NCC(c1cccnc1C)(C)C Cn1ncc2ccc(C(=O)NCC3CC4CCC3N4C(c3cnns3)=O)cc12 C1(NC(c2ccc(Cl)o2)=O)CCCC(NC(c2ocnc2C(F)(F)F)=O)C1 Cc1c(CC(N2CC(CCNC(=O)C=CC(F)(F)F)C(C)C2)=O)ncn1C C1(C(=O)NC2(CC=C)CCCC2)CCCCCCN1C(=O)C(=O)C(C)(C)C C=CCCC(F)(F)C(=O)NCC1CCC(NC(=O)CCN2CCCCC2)CC1 Cc1nn2c(c1C(=O)NCC(C)CCN)CCCC2C C12(CC(=O)NCC3(SC)CCC3)CCC1CN(C(c1ncccn1)=O)C2 C=C(Cl)CC(C(=O)NCCOCC(C)(C)O)NC(=O)CC(C)CC Cc1ccc(C(=O)N(CC(C)CNC(C2CCN(C)C2)=O)C)c(N)c1Br C1(C(=O)NCC(C)NC(=O)C=C2CCC2)NC(=O)CC1C N1(C(c2nccc(CC)c2)=O)CC2CCN(C(=O)C(F)=CC3CC3)CC12 c1(C(=O)NC2CC(NC(C(CC)OC)=O)C2)c(-c2cccc(OC)c2)noc1C C=CC1(CO)CCN(C(C2C=CCN2C(C2CCC2C(=O)OC)=O)=O)CC1 CN1CCC2C(CCN2C(c2c(C(=O)N(C)C)nnn2C)=O)C1.C12(CC1)C(=O)NC2 c1(C(=O)NC2C(C(=O)NCC(=O)NC3CC3)CCC2)ccc(Cl)nc1Cl c1(C(=O)Nc2c(C(=O)OCC)scc2)nc(OC)c2nc[nH]c2n1 C1(C(c2ccccc2)NC(C)(C)C(N)=O)CC2(CCNCC2)S1(=O)=O C(=O)(C(C)N=c1cncc[nH]1)N1Cc2c(C(=O)NCC(=O)N(C)C)n[nH]c2CC1 c1(C(=O)OCC)cc2cc(S(=O)(=O)NCc3cnn(C)c3OC)ccc2s1 N1(C(c2ccc(C(C)C)o2)=O)CC=C(CC(=O)NC2CCN(CC3CC3)C2)CC1 C1(C(C)C)CC(c2nnnn2C2CCC2)(NCc2nncs2)CCO1 c1(NC(C(c2ccc(F)cc2)(C)O)=O)cccc(-c2cnco2)c1 c1(C(=O)NC2C(C)N(C(C3CCC3)=O)CCC2)nnc2ccccn12 N1(C(c2cnc(Br)n2C)C(=O)NCC(=C)C)Cc2ccc(Cl)cc2C1C N1(C(C2CCCC23CC3)=O)CCN(C(=O)Cc2nc[nH]n2)C(c2ccccn2)C1 c1(C(=O)NCC(c2ccccc2)CNC(CC=CC)=O)c(F)cccc1F CCC(CC(=O)NCC1CC(O)(CNC(c2cnc(O)c(Cl)c2)=O)C1)C(C)(C)C N1(C(CCCCCSC)=O)CC2CN(C(=O)C(O)C(C)C)CC2(C)C1 CC(CN(C)C)CCC(=O)NC1CCN(C(c2cnsc2)=O)C1 Cc1cnc2n1C(C(=O)NCCN(C(=O)CN1CCC(C)C1)CC1CC1)CCC2 C(C)(C(=O)NCC(C1(O)CN(C(=O)Cc2nn(C)cc2Cl)C1)(C)C)(C(C)C)OC N1(C(CCN(C)CC)=O)CCOCC1CNC(c1ccc(C(=O)OC)s1)=O C1(NC(c2c(CC)nns2)=O)CC(F)CN(C(=O)CCC(C)OC)C1 Cc1ccc2cc(C(N3CCC(NC(=O)CC4(C)CCC4)C3)=O)[nH]c2c1 C1(NC(c2cc(F)c[nH]2)=O)CCN(C(C2(c3ncco3)CCC2)=O)CC1F c1(CCC(=O)NC(CNC(c2ccc(C#N)o2)=O)CO)c(Cl)cccc1Cl c1(C(=O)NC(c2ccc(SC)cc2)C(=O)OC)cnc(S(C)(=O)=O)s1 N1(CCC(N2CC(OCC(=O)NC3CCCOC3)(CO)C2)=O)CCC(O)CC1 C(CS(=O)(=O)CC(=O)NCC(C1CC1)NC(c1ncccc1C(F)F)=O)OC c1(C(c2n(C(CC)C)nnn2)NC2(CCOC)CCC2)cccc(C(C)(C)C)c1 C(=O)(C#CC(=O)N(C)C)N(CCNC(C1CCC(C)S1)=O)C(C)C N1(C(C2CCCOCC2)C(=O)NCCCOC)CCCSCC1C c1(SC)ncc(Sc2cccc(NC3CCC(C)CC3)c2)n1C C(C(C)(C(C)C)NC(=O)CCc1cnc(O)[nH]1)NC(C1C(c2ccc(C)s2)C1)=O C(=O)(C1CCc2c[nH]nc21)N(C(CN(C(c1c(C)nn(CC)c1C)=O)C)C)C c1(C(=O)NCC(C)(CC)NC(C(CC)=CC)=O)c(C(F)(F)F)nc(C)n1O C1(CC=C)(NC(C2CC2c2ccnn2C)=O)CCN(C(=O)CC2CCC3CC23)C1 C1(C(C(=O)NCCC2(NC(C(=O)NCC)=O)CCC2)OC)CCCOC1 N1(C(Cc2ccc(C)nc2)=O)CCCC2(NC(C3(F)CCCCC3)=O)CCCC12 C(=O)(C1=CC2(CN(C(C3(OC)CC(C)C3)=O)C2)OC1)NCCSCC#C N1(C(C=C(C)CCc2ccccc2)=O)CC2CC1C2NC(c1ccsc1)=O CCC(C)(C)C(C(=O)NCC(CC)(CC)NC(c1cnoc1C)=O)OC N1(C(=O)C=CC2CCOC2)CCC2CN(C(c3ccccc3O)=O)C2C1 C(C)(N=c1[nH]c(N2CCC3(CCC3)C2)nc2cc[nH]c12)c1c(C)nc(C)[nH]1 c1(OCCCOC)ccc(C(=O)NC(C)C(C)NC(C2(C)CCOCC2)=O)cc1 CCC(C)CCCC(=O)N1CC(NC(C2CC(OC(F)(F)F)C2)=O)C(C)C1 c1(OC)cccc(C(C)C(=O)NCC2CC(O)CN2C(c2ccnn2C)=O)c1 N1(C(c2c(C(C)C)ocn2)=O)C2CCCC1CN(C(C1CC3(CCC3)CO1)=O)C2 C1(CNC(c2ccc(OC(C)C)cc2)=O)CCN(C(c2nc(Cl)cs2)=O)CC1C C(CC(=O)N1CC(O)CC1CNC(c1csc2nccn12)=O)(C(F)(F)F)OC C1(C(N2CCC(C)N(C(c3n[nH]c(=N)s3)=O)CC2)=O)CC12CCC(F)(F)CC2 c1(N2CCN(C3C4CN(S(CC#N)(=O)=O)C(C4)C3)CC2)nc2cccc(F)c2[nH]1 c1(OC)cc(N)c(C(=O)NCC(CO)NC(C2CCCCC2(C)C)=O)c(F)c1 N1(C(c2ncn(C(C)C)n2)=O)CCOCC(CNCCN2CCCC2=O)C1 N1(C(C2N(C(C)=O)CSC2)=O)CCC2C1CCN2C(C1CCCSC1)=O c1(C(N(CC(C)NC(CCCC(=C)C)=O)C)=O)ccc(F)c(C)c1C#N CC1CC(C)OC1C(=O)NC1CC(NC(C2CCC(=O)N2)=O)C1 C1(CNC(CNC(=O)NC)=O)CN(C(c2cc(C3CC3)on2)=O)CC(C)(C)C1 C1(C(=O)NCC=CCNC(c2c(C(F)(F)F)ncn2O)=O)CCC2CC1CO2 c1(C(=O)NCCN(C)C(C2(F)CC=CCC2)=O)ccc2c(c1)CCCO2 Cc1cnc(C=CC(=O)NC2COCC2NC(=O)C(C2(O)CCCC2)F)[nH]1 C1(CNC(C(C(C)C)NC=O)=O)CCCCN(C(=O)C=C2CC2)CC1 CN1CCN(C(=O)CC2(C)CCOC2)CC1CNC(C1CN(C(N)=O)C1)=O c1(C(=O)NCC(CO)C2CC2)coc2c1CN(C(=O)C(O)CC(F)(F)F)C2 n1(C(C)C2CC2)ncc2cc(C(=O)NC3CNCC3C(=O)O)cnc12 C1(CC)CN(C(=O)CC2CCN(C(=O)CCC3CCCN(C)C3)C2)CCO1 Cc1nc(C(=O)NC2CCC(NC(C34COCC3C4(F)F)=O)CC2)ccc1C#N Cc1ccc(CCC(C)NCc2csc(-c3sccc3C)n2)cc1 C1(C(=O)NC2CCN(CC)C2)(COC)CCN(Cc2cccc(C(=O)OC)c2)C1 O(N(C)C(=O)C(C1CCCO1)C1CCC1)CCCOC.C(=O)CC(C)(C)O S(=O)(=O)(c1ccc(I)cc1F)NC(C(C)(F)c1ccccc1)=O CC(Cn1ccnc1)N=c1[nH]c(N2CCOCC3(CC3)C2)nc2c1COCC2 C1(C(N2CCC(C(N3CCCC(C4(C)N=N4)C3)=O)C2)=O)(CC)CNC(=O)C1 c1(C(N2CCCC3CCN(C)CC23)C(=O)NCCOC)nc2ccccc2nc1C N1(C(c2oc(C)c(CO)c2)=O)CCCC(C)(C)C1C(=O)NC1CC2C=CC1C2 C(c1cn(C2CN(C(C3CC(C)(C)CO3)=O)C2)nn1)=CC Cc1cn2c(n1)CCC(C(=O)N(C1CCCN(C(c3cnc(C#N)s3)=O)C1)C)C2 C1(NC(CCc2ccc(OC)cc2)=O)CC2CC1N(C(c1cc(CO)[nH]n1)=O)C2 n1(CC(CC)CC)nc(-c2cncs2)nc1C1CC1(C)C c1(C(N2C(C)CC(NC(=O)C=Cc3cccn3C)CC2)=O)ccn2ccnc2c1 N1(CC(=O)NCCN(CC(C)O)C(=O)CC2(C(F)F)CC2)CCOCC1=O C(=O)(CCCC(C)(C)C)N1C(C)(C(NOCCC(C)O)=O)CCC1 C(C)(C)(CCCNC(=O)CC1C=CC(NC(=O)C=CCN2CCC2)C1)OC N1(C(=O)NCc2n(CCC)ncn2)CCN(Cc2ccccc2)C(=O)C1C c1(NC(=O)NCC2C(CCC)C2)cc(Br)cc2[nH]ccc12 C#Cc1ccc(C(=O)NC2COCCN(C(c3[nH]ncc3C#N)=O)C2)cc1 CC(CO)CCN=c1[nH]c(=NC(C)Cn2cnnc2)[nH]c2c1CCCCCC2 c1(C(=O)NC(CNC(c2cc(SC)oc2)=O)C2CC2)ccc(Cl)c(N)c1 N1(C(C2(SC)CN(C(=O)CC3CC4CCC3O4)C2)=O)CCC=C(F)C1 c1(C(=O)NC(CNC(C2N(CC)CCC2)=O)(C)C2CCC2)ccccc1CC#N N1(C(C(CC)OC)=O)CCCCC(CCC(=O)Nc2cccc(Cl)c2C)C1 c1(NC(N(C2CCCN(C(CCC(=C)Cl)=O)C2)CCF)=O)ccc2nc[nH]c2c1 N1(C(c2c(CC)nc(C)nc2)=O)CCC2CN(C(c3cn(C)nc3SC)=O)CC12 C1(C(N(C2(CCCNC(C3CC3(C)C)=O)CC2)C)=O)CC12CCC(=O)CC2 N1(C(C=CC(CC)C)=O)CCOCCC1C(=O)NCc1cccc(OC)n1 C1(C2(C(N(C)CC3CC=CC3)=O)CC2)CCCCN1C(=O)C(F)CC1CCOC1 C1(NC(C2C(C)C2)=O)CCC(N=c2[nH]cc(C#N)s2)CC1 N1(C(C(=O)NCCCCNC(C(C)Cc2cnn(C)c2)=O)C)C(=O)CCC1=O N1(C(C(C(CC)C)O)=O)CCCC2(NC(=O)Cc3ccc4c(c3)CCO4)CC2C1 C#Cc1ccc(C(N2CCC(O)(C(=O)OC)CC2)C(=O)NCCC2CC2)c(F)c1 C1(C(=O)NCC2N(C(C3(C)CCCCC3)=O)CC2)CCCC12OCCO2 n1(CC(=O)N(CCCN(c2nncs2)C)C)cnc2ccccc12 C(CCC)(CCCNC(=O)CN1CCCNC1=O)NC(COCCCCCC)=O C1(NC(CS(=O)(=O)NCC)=O)CN(C(c2cc3c(s2)CCC3)=O)CC2(CCC2)C1 N1(NC)CCC(C(=O)N(CCCNC=O)C)CC1.c1(C(=O)N)cccnc1.C1CS1 n1(CC(=O)N(C(CC(=O)OC)C(=O)O)C2CC2)cnc2ccccc12 C1(CNC(CCCC)=O)CN(C(C2(C)CC(C#N)C2)=O)CC1(F)F N1(CC(N2CCC(O)(C3CC3)CC2)=O)CCC2(CC1)Cc1ccccc1C2=O C#CCCC(O)CCNC(c1cnc(CNC(=O)C(C)n2ccnc2)nc1)=O C1(OC)CC(CC(=O)NCCN(C(=O)C=CC2CCCC2)C(C)C)C1(C)C N1(C(C2CC(=O)N(c3cccc(Cl)c3Cl)C2)=O)CCC(c2nn[nH]n2)C(F)(F)C1 N1(Cc2cc(C)on2)CCN(C(C2CN(C)C(=O)O2)=O)C(C(F)(F)F)C1 N1(C(C=Cc2nc(C)sc2)=O)CCCC(NC(=O)CC2CCCCCO2)C1C C1(CCC)CN(C(c2ccc(C)c(C)c2)=O)CCN1C(N1CC(C)(C)C1)=O c1(NC(=O)CCc2cccnc2)ccc(C(N2CCC2)=O)cn1 C(=O)(C1OCCn2ccnc21)N1CCCC(CC=C)(NC(=O)Cn2nccn2)C1 CCCN=C(NCC1(OCC)CCCSC1)N1CCC(F)(c2ccc(F)cc2)C1 CCC(CCC(=O)NCC(C)S(C)(=O)=O)NC(c1cn(CC)cn1)=O C1(CNC(CC2(C)CC2)=O)CCCN1C(c1cnc(C2CCCCC2)s1)=O CC1CN(C(C2CCC(N(C)C)C2)=O)CCC1C(=O)NC(c1ncc[nH]1)CO c1(C(N(C2CCN(C(=O)C=CCn3cncn3)C2)CCC)=O)ncc[nH]c1=O c1(C(=O)NC(C(C)(C)NC(c2c(CC)cco2)=O)C)cccc2c1CCC2 c1(C(N(CCC(N2CCC(OCCO)C2)=O)CC=C)=O)cc(CO)[nH]n1 c1(CNC(COCCCC#C)=O)c[nH]nc1C1CC1.C1(=O)CC=CCN1 C1(CNC(c2cc(C)c(C)o2)=O)CCCN(C(c2cc(F)cnc2Cl)=O)CC1 Cc1ncc(C(N2CCC(C(F)C(=O)NCC3C4CCCC34)C2)=O)o1 N1(C(c2nc(C#C)sc2)=O)CCOCC(CNC(c2cc3ccsc3s2)=O)C1 Cc1ncnc(C(=O)NCc2nn[nH]n2)c1C Cc1ccc(C(C)NC(=O)CC2CC=CCC2)c(F)c1 C1(C(N(CC(O)CF)C)=O)CC2(CCC2)CN1C(c1cc([N+](=O)[O-])n[nH]1)=O c1(CC)nc(C(=O)NC(C2CCN(C(=O)CCCSc3ccccc3)C2)C)cs1 C(C(CN=c1nc(C(C)(C)C)[nH]s1)C(F)(F)F)CNC(CC1(CSC)CC1)=O N1(S(CC(C)C)(=O)=O)CCN(C(=O)C(C)(C)N(C)C)CC1CO C(C)(C)(CCC(=O)NC1CC2CCC(C1)O2)NC(C(CCC)=CCC)=O c1(C(N2CCC(F)(CNC(=O)COC3CCOCC3)C2)=O)c(F)cccc1Cl CCCCCC(O)C(=O)NCCC(C)N(C)C(c1cccn1CCC)=O C1(C(=O)NC2CCCC2C(=O)NC2CC2c2ccc(Br)cc2)CCc2nc[nH]c2C1 C1(C2CCN(C(C3CC(C4CC4)=NO3)=O)CC2)(NC(CC(C)(C)C2CC2)=O)CC1 c1(C(=O)NC(C)CCC(=O)NCCCc2ccncc2)ccc(N)c(F)n1 C(C(C)(C)C(=O)NCC1CN(C(=O)CCc2nc(C3CC3)no2)C1)OC CC1(C)CN(C(=O)C2=CCC2)CC1NC(c1ccc(CCC#N)cc1)=O N1(C(CCN(C(C2CN(C)C(=O)CC2)=O)CCO)=O)CCC2(CC=CCO2)C1 C(=O)(C1=C(C)CCOC1)NCC(C(=O)NC(CCCC)CC)CC1CC1 N1(C(=O)CC(O)CF)CCC2(CC1)CCN(C(C1CCCO1)=O)CC2 c1(C(=O)NCC2(CNC(C3(CC#C)CCCCC3)=O)CC2)cc([N+](=O)[O-])c[nH]1 C1(CNC(C2(NC(C)=O)CCOC2)=O)COCCN(C(=O)COC(F)F)C1 C=CCCCCCCC(=O)N1CCC(CCC(N2CCCC(C)(CC)CC2)=O)C1 C1(NC(CSC)=O)CCOC12CCN(C(C1CC(OC)(OC)C1)=O)CC2 c1(C(=O)NC(C)COc2ccc(F)cc2)nccc(-n2cccn2)n1 N1(C(C2(OCC)CC2)=O)CC(NC(C2CCc3nncn3C2)=O)C(C2CC2)C1 N1(C(c2c(OC)csc2)=O)CCCC(CNC(=O)CSCc2cscn2)CC1 C1(NC(C2N(C(CC)=O)CCCC2)=O)CCC2CCN(C(=O)COCCO)C1C2 C1(NC(CC2C(C)CC2)=O)CC2(CCN(C(=O)C(C)(C)N(C)C)C2)C1 C1(O)(C(=O)OCC)CCCN(C(=O)CN2CCC2C(=O)OC(C)(C)C)C1 C(C1CCCc2nccn21)NC(N(CCOC)Cc1ccsc1)=O Cc1nonc1CC(=O)NC(C)(C)C=CC(=O)N(C1CC2(CC2)C1)C c1(C(=O)OC)ccc(C(c2nnnn2CC2CCCO2)NCCCCO)s1 C1(NC(c2c(C(C)C)sc(Cl)n2)=O)CC2CC(NC(=O)CCOC(C)C)CC2C1 Cc1nc(N2CCCC(NC(=O)CCc3ccn(C)n3)CC2)c2ccsc2n1 N1(C(Cc2c(C)non2)=O)CCOCC(CNC(=O)C(C)CC(C)C)C1 C1(NC(C2C(C)(C)C2(C)C)=O)CN(C(=O)C2=NNC(=O)CC2)C2(CCCOC2)C1 CC(C)CC(C)C(=O)N1CCC(C(CO)NC(=O)CC2C=CCCC2)CC1 c1(C(=O)NC2CN(C(C3(F)CC3)=O)CCC2F)cc2cccnc2o1 c1(CN(C2CN3CCC2CC3)CCOCC)cn2cc(Br)ccc2n1 Cc1nc(CC(=O)NCCCOCCOCCNC(C2(C)COC2)=O)[nH]c1C N1(C(CS(=O)(=O)NC)=O)CCN(C(=O)C(C2CCCCC2)O)C2CCCCC2C1 C12(CNC(C=C(C)C(F)F)=O)CC1CN(C(c1ocnc1C1CCC1)=O)C2 CC#CCC(CO)NC(=O)CCN(C(C1CCCCCC1)=O)CC CCC(CC)(CCNC(C1CCCC(O)C1)=O)NC(c1cc(C(F)F)no1)=O C(=O)(CCCCC(C)(C)C)N1C(CC(=O)NCCCS(C)=O)CC2(CC2)C1 N1(C(C(C)(C)OC)=O)CCCC2(CCN2C(=O)C(n2nc(C)cc2C)C)C1 CCC(CC)C(C)C(=O)NCC(F)CNC(c1ncoc1-c1cnn(C)c1)=O C1(C(=O)NC(CNC(c2ncc(C)cc2O)=O)CC(C)C)CCC2CCCCN12 C(CC(=O)NC1CC2CCC1N2C(=O)Cc1c(C)nn(C)c1C)(C(C)C)OCC c1(NCC2(C)CCC(C(=O)OCC)CC2)ccc(OC)cc1N=[N+]=[N-] C1(NC(=O)CCc2ccsc2)CCC(O)CN(C(=O)CN2CCCS2(=O)=O)C1 C1(C)(C(=O)NC2C(N(C(C(C=CC)O)=O)C)CCCC2)CCS(=O)(=O)CC1 C1(CC(N2CC3C(CNC(c4cnc(C)n4C)=O)C3C2)=O)CCCCC12CC2 CC(C)(C#CC(=O)N1CC(N2CCCC2)C1)CNC(c1cnc2ccccn12)=O C=CCCCCCC(=O)N1CC(OC)CC1CNC(=O)C(C)C(O)CC N1(C(N2CC(F)(NC(=O)OC(C)(C)C)C2)=O)CC(NC(=O)C2=CCC2)C2CC12 C1(CSCCNC(=O)NC(CCCC)C)CCCN1S(=O)(=O)N(C)C C(c1c(Cl)cccc1Cl)=CC(=O)NC1CN(C(C2CC(C#N)C2)=O)CC1O C(=O)(C1=COCCC1)NCC1(CNC(C2(CC)CCCC2O)=O)CCC1 N1(C(C(C2CCC2)OC)=O)CCOC(C(=O)NCCC2CC(C)=NO2)C1 C=CC1(C(N2CC(OC(=O)NC)C2)=O)CCN(C(c2ccnn2CCC)=O)C1 C1(NC(C2CC(C)SCC2)=O)CCN(C(c2cc(O)nn2C)=O)CC1F N1(C(Cc2c(Br)cn(C)n2)=O)CCCCC(NC(C2(C)CC=CCC2)=O)C1 C#CC1(F)CCN(C(C2C3CC3CN2C(=O)C(C)OC)=O)CC1 C(=O)(N=c1[nH][nH]cc1C(C)C)C1N(Cc2ccc(C)cc2)CC(OCC(=O)O)C1 C=CCCC(F)(F)C(=O)N1CCC(O)(CCNC(=O)C(C(C)OC)N(C)C)CC1 C(=O)(C1=NOC2COCC12)NCC1(CNC(CC(CCC)C)=O)CCCC1 CC(C)CC(F)C(=O)N(C1CCCCC1N(C(=O)CCSc1ccccn1)C)C N1(C(CC(C)C2CC2)=O)CC2(CO)CC1(C(=O)NCC1CC13CCCCC3)C2 c1(C(N2CCC(O)(C(CNC(C=C(CC)CC)=O)C)C2)=O)cc(C)cc(C)c1N C1(CNC(CCOCC)=O)CCCC(NC(C2CCCC(C)O2)=O)C1 c1(OC)cnc(F)c(C(N2CC(CCNC(C3C4CC4C4CC34)=O)(OC)C2)=O)c1 c1(CC)ccc([N+](=O)[O-])cc1C(N1CCOC(CNC(c2c[nH]cc2Br)=O)C1)=O N1(C(CCN(C)C(C2CCOC(=O)CC2)=O)=O)CCCC(O)(CO)C1 C1(C(C)(C)C(=O)Nc2cccc(CCO)c2)CCCCCN1C(=O)CS(C)(=O)=O CC(CS(C)(=O)=O)C(=O)NCCC1CCCN1C(c1cc(F)c(F)cc1O)=O c1(C(=O)NCC(C)NC(c2ccns2)=O)csc(-c2ccoc2)n1 Cn1nc(CC(N2CC=CC2CNC(c2cscc2Cl)=O)=O)c2ccccc12 N1(C(C2N(C(c3c(C)n(C)cc3)=O)CC=C2)=O)CCCC2(CCOC2)C1 c1(C(=O)NC2(CNC(c3cc(N)cc(F)c3)=O)CCC2)c[nH]c2nccc(Cl)c12 C(=O)(C1CCCc2nc[nH]c21)N(CC(C)O)CCNC(CCCC(CC)CC)=O C(=O)(CCCC(C)(F)F)NC(CC(C)NC(c1n(CCC)ccc1)=O)C N1(C(Cc2cn(C)nc2C(F)(F)F)=O)CC2CC(C1)N(C(=O)CC(C)(C)O)C2 c1(C(C)=O)ccc(O)c(C(=O)NC(CNC(=O)C=Cc2ccc(C)cn2)CO)c1 N1(C(C23N(C(C(C(C)C)OC)=O)CCC2C3)=O)CCC2(CCC2)CC1 C1(C(=O)NC(CC)(CO)CO)CCCN(C(c2ccccc2Br)=O)CC1 S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(C(=O)OCC#C)CC1 N1(C(CC(=C=C)C)=O)CC2(CCCN(C(=O)C(C)CSc3ccccc3)C2)C1 C1(CNC(CN(C)C)=O)CC2CCC1N2C(c1ncc(C(F)(F)F)s1)=O C1(C(=O)Nc2c[nH]nc2C2CCOC2)NCCC1C1CCC1 Cc1ccc(C(=O)NC2CCN(C(C3CC(=C4CC4)C3)=O)CC2C(C)C)cc1F CN1CCC(CCNC(C23CC2CCN3C(c2ccsc2Cl)=O)=O)C1=O CC1CCN(C(C2C3CCCC3CN2C(=O)CCc2ccncc2)=O)CC1(F)F C1(C(=O)N)CCCC(=O)C1.C(CCNC(=O)CN(CCOC)CC)OCC C(C)(CCC(=O)NCC(C(C)(C)C)NC(C)=O)NC(=O)CN(CC(=O)N(C)C)C c1(C(=O)OC)ccc(C(=O)NC2(CNC(=O)CSC(F)(F)F)CCCCC2)n1C n1(CC=C)cc(C(=O)NCCN(C(=O)C(=O)Nc2ncc[nH]2)C2CC2)nn1 C1(NC(C(COC)CC)=O)CN(C(=O)C=NOC)CCC1(C)C c1(C(=O)NCC2OCCC(NC(CCC(=C)Br)=O)C2)ccc(F)c(C)c1 C12(NC(c3ccc(OC)cn3)=O)COC(C1)C(NC(=O)C=Cc1ccc(C)o1)C2 N1(C(C(CSC)C)=O)CC(CNC(=O)Cc2cc[nH]n2)CC(C)C1 c1(CNC(C=CC(CC)C)=O)cc(C(N2CC(OCCO)C2)=O)ccn1 c1(CC)ccc(C)c(C(N2CCN(C(C3CCCOC3)=O)C(CC(F)F)C2)=O)c1 C(=O)(C(C)(C)C(F)c1ccccc1)NC1C(OC)CN(C(=O)CC2(O)CCC2)C1 C1(C(N(CCNC(=O)C(C)Sc2ccccn2)CC)=O)CC=C(C)CC1 N1(C(C2C(C)OC(C)C(C)C2)=O)C2CCC1CC(CNC(=O)Cc1ccon1)C2 C=C1CCN(C(=O)CC2CCCOCC2)C(C(=O)NCCN=[N+]=[N-])C1 c1(C(N2CCCCC2c2ccc(Cl)nc2)C(=O)NC2CC2)cc(Cl)c(Br)cc1F N1(C(c2cn(CC=C)nn2)=O)CCC(NC(=O)C(C)(C)CC#C)C(C)C1 c1(NC(CC2C(CNC(c3ccc(OC)cc3)=O)C2)=O)cnc(OC)cc1C C(=O)(C(CC)C(C)C)NCCC(CNC(c1cncc(C(=O)OCC)c1)=O)O N1(C(c2c(C)nc(Br)o2)=O)CC(CNC(=O)CNC(N)=O)N2CCC1C2 C1(C(N(CC2CCN(C(C(CC)F)=O)CC2)CC(=O)NC)=O)CNC(=O)CC1(C)C c1(C(C(=O)NCCCC2CC2)N(C(c2cccc(O)c2)C)C)nccc(Cl)c1Cl N1(C(C=NOC)=O)CC(C2CCN(C(c3cnsn3)=O)CC2)C1 C1(Nc2ccc(NC(c3ccc(F)cc3)=O)c(Cl)c2)CCCCC12CCNCC2 N1(C(C(c2ccc(CCC)cc2)C)=O)CCCC(CCNC(=O)COCC)CC1 C1(C(=O)NCC(C2CCN(C(C3CCN(C)C3)=O)CC2)C)CCCCC1O CC1CCCCN1C(=O)CC(C)NC(c1cncc(CO)c1)=O Cc1cccn2c(C(=O)NCC(C)NC(c3ccc4[nH]c(=N)oc4c3)=O)cnc12 C1(NC(C(C2CC=CCC2)NC(c2ncc[nH]2)=O)=O)CC2CCC(C1)C2O Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)CCn2ccnc2)c(C)o1 C1(C(N(CCN(C(CCc2c(C)ncs2)=O)C)C)=O)CCC(=O)CC1C C(=O)(C(F)CC(C)(C)NC(=O)OC(C)(C)C)N1CC(CC)C(C)C1C N1(C(CC2CC(OCC)C2)=O)CCC(NC(c2coc(Cl)c2)=O)C1(C)C N1(CC2(COC)N(C(CC(CC)C)=O)CC=C2)Cc2cnn(C)c2C1 c1(OC)cccc(C(C(=O)N(C(CNC(=O)C=CC2CC2)C2CC2)C)OC)c1 C1(C(C)NC(c2c(CC)c[nH]n2)=O)CCN(C(c2ccc(C)s2)=O)CC1 c1(C(=O)NC2(CNC(C3CC(F)C3)=O)CCCC2)c(OC(F)(F)F)cccc1F C(CCNC(=O)CC1CCN1C(c1cccc(CC#N)c1)=O)(C(C)C)OC N1(C(C2N(C(c3ccc(CC)nc3)=O)C3CCC2C3)=O)CCC(F)(CF)CC1 Cc1c(C(N2CC(n3cc(-c4ccncc4)nn3)C(C)C2)=O)cnn1CC(F)F C1(C(=O)NC(c2ccncc2)C(C)C)CCC(NC(=O)C(C)CNC(N)=O)CC1 CC(C)C(C)C(=O)N1CCC(C)(CNC(c2cnnc(Cl)c2)=O)C1 C1(CC=C)(C(=O)NCC2CN(C(=O)C(C)OCC3CCCCO3)C2)CC=CC1 N12CCN(C(=O)CCCCSC)C(C1)Cc1ccc(cc1)C2=O.CC(=O)OCC c1(C(=O)NCC(C)CNC(C2CC3CCC2CC3)=O)cc2ccsc2s1 N1(C(CCC(=C)Cl)=O)CC2CC1CN(C(c1cccc(-c3ccccc3)c1)=O)C2 C1(CNC(c2csnn2)=O)CCC2CN(c3nc(Cl)nc4c3SCC4)CCC2C1 C1(COC)(NC(c2ccc(C)nc2O)=O)CCN(C(c2cnc(C)[nH]2)=O)CC1 CCCCCCCCCC(C)CCNC1CCC(C)C(C)C1 N1(CC(=O)NC(C2CCN(C(=O)CCCCN(C)C)C2)C)C(=O)CC(C)(C)C1=O S(=O)(=O)(c1cccs1)N1CC2(C(C(=O)Nc3cc(C)nn3C(C)C)C2)C1 C#CCC(C)(CC)C(=O)NC(CNC(=O)CS(=O)(=O)CCO)CO C1(C(N2C(C(C)C)C(NC(=O)CCc3cscn3)CC2)=O)OCCOC12CCC2 C1(C(N(CC(=O)NCCc2cnnn2C)CCOC)=O)CCC(C)(CC)O1 c1(CC(C(=O)NC2CC(N(C(=O)CN3CCCC3=O)C)C2)O)ccccc1Cl c1(C(=O)NC2CC3CC(NC(=O)CC4CCCOC4)C2C3)ccc(O)nc1Cl c1(C(=O)NCC2C(NC(CCCC(=O)OC)=O)C2)cc2n(n1)C(C)CCC2 c1(CN(CC(=O)NCC2C(CNC(C3(CC)CC3)=O)C2)CC)ccc(Cl)cc1F c1(CC(=O)NC2CC(CCNC(c3c(CC)ccs3)=O)C2)c[nH]c2cnccc12 C12CC3(C1)CC(C3)NC(=O)CN2.CC1(C)CN(CC(F)(F)F)C1.C12(C(=O)N)CCC1C2 C1(NC(=O)CCc2cc[nH]n2)CC(O)(CNC(c2csc(Br)c2)=O)C1 N1(CC(=O)NCC2CC2Nc2ncc([N+](=O)[O-])cn2)Cc2ccccc2C1=O CC1(C(=O)NCCOC2CCN(C(c3csc(O)n3)=O)C2)COC(=O)C1 CC1C(NC(=O)CN2CCCC(CO)C2)CC2CCC1N2C(C12CC(F)(C1)C2)=O n1(CC)ncc(S(=O)(=O)NC(C2CCN(CC(F)(F)F)CC2)C)c1C C1(C(=O)NC2C=CC(C(N3CC(NC(C)=O)C3)=O)C2)COCCC1C c1(C2C(C(N3CC(O)C(O)C3)=O)C2)ccc(Br)cc1F C1(C(C(=O)Nc2ccccc2C)N(CCCCCC)C)C2(CCC2)C12CCC2 C(N=c1[nH]c2c(c(=NC(C)C3CCC3)[nH]1)COCC2)c1cccc(NC(C)=O)c1 Cc1cncc(CNC(C2(CNC(=O)C(C)c3ccco3)CC3(CC3)C2)=O)c1 CCCC(O)C(=O)NC1CCN(C(=O)Cc2cnn(C)c2)C1C(C)C c1(C(=O)NCCC2N(C(C(C)NC(=O)NC)=O)CCC2)nccn2nc(C)cc12 N1(C(C2C(C(=O)OCC)CCO2)=O)CCC(C)C1CSc1ccccc1 C(CC(CNC(=O)CCc1cnco1)NC(=O)CSC(C)C)OC CN(C)S(=O)(=O)NCC(N1CC(O)CC1CNC(c1nn(C)cc1Cl)=O)=O C1(CC(=O)NCC(C)(C)OCC(=O)NC(CC)COC)CCC(C)(C)C1 Cc1csc(=O)n1CCC(=O)NCC1CC1CNC(=O)Cc1cccc(O)c1 N1(C(c2csc(C3CC3)n2)C(=O)NCc2nnn(C)n2)CCC2(CCCOC2)CC1 CC(N=c1[nH]c2c(c(=NCc3cc(Br)ccc3N)[nH]1)CSC2)C1CSC1 C(=O)(N=c1[nH][nH]cc1C(N)=O)C1CCCN(Cc2cccc(OC)c2O)CC1 n1(CCC)ccc(C(=O)NCC2(OC)CN(C(=O)C(C)Cc3ccnn3C)C2)n1 N1(CCC(=O)NC(C2CCCN2C(=O)C=CCO)C)CCNC(=O)C1 c1(C(CO)SC(C)=O)ccc(-c2ccc(CCCN(C)C)cc2)cc1 N1(C(c2cc(C)c(C)s2)=O)CCC(C2CC2)C1C(=O)NC1(CO)CCC1 C(C(C)C(=O)N(CCC(=O)NC1CC=C(C)CC1)OC)OCCOC CC(CC1CCCC1)C(=O)N1CC(=C(F)CNC(=O)CC2(C)CCCO2)C1 CC(=NO)c1cc(C(=O)N(C2C3CN(C(=O)Cn4cccn4)CC23)C)cnc1O n1(CC(N2CCCN(C(=O)CNc3ncccn3)CC2)=O)cc(F)ccc1=O C(=O)(CCC(=O)C(C)(C)C)N1CCCC(C(C(N2C(CC)CN(C)CC2)=O)C)C1 N1(C(CC2(OC)CCCC2)=O)CCC2C(C1)CN2C(c1sc(F)cc1C)=O c1(CC(N2CC(N(C(CC3(OC)CCC3)=O)C)C(F)C2)=O)ccc(F)cc1Cl c1(C(=O)NC(CSc2cccs2)CO)cnc(N2CCCCC2)s1 C(=O)(CCC(F)(F)Cn1cc(-c2ccc(F)cn2)nn1)N1C(COC)COCC1 C1(NC(C(CNC(c2ncn(C)c(=O)c2)=O)(C)C)=O)CCn2nnnc2C1 c1(OC)cc(Cc2nc(-c3ccccc3)n(-c3ccnc(Cl)c3)n2)ccc1C C1(N(C(c2cc(C(=O)OC)oc2C)=O)C)CCCN(C(=O)CC(C)F)CC1 C1(C(=O)NCCN(C(Cn2c(CCC)nnc2S)=O)C)CCn2c(O)nnc2C1 C1(C(=O)NCCOCC#C)CN(C(=O)C(C)(C)C2CCCO2)CCC1(C)C C(=O)(C(C(C)(C)C)c1cc[nH]n1)NC(C)C(C)(C)NC(c1cnn(C)n1)=O N1(C(CS(C)(=O)=O)=O)CCCC(C2CC2NC(=O)Cc2cccc(C3CC3)c2)C1 N1(CC(=O)NCCNC(C(C)(C)NC(=O)OC(C)(C)C)=O)CCCOC1=O c1(OCC(=O)NC2C(NC(c3c(CC)cco3)=O)CCC2)cc(C)c(F)cc1F C1(NC(C(CSC)OC)=O)CCCC2CN(C(c3ccc4c(c3)OCO4)=O)CC12 C1(CCNC(C(CC=C)(F)F)=O)CCN(C(=O)CCSCC(N)=O)CC1(F)F N1(C(CN(C(=O)OC)C)=O)CCC(C(=O)NCC2CCCO2)(CO)C1 C(=O)(C1CCCc2c[nH]nc21)NC1(C)CN(C(c2ncc(C)nc2)=O)C1 CC(C)CCC(=O)N(C1CCN(C(C2CC3CCC3C2)=O)C1)CCO C#Cc1ccc(F)c(C(=O)NC(C2CCCCN2C(c2cc(Br)n[nH]2)=O)C)c1 CCCCCC(O)CC(=O)NC(C1CCCN1C(c1ccc(C)c(C#N)c1)=O)C C(C)(C)(CCC(=O)NC1(C(=O)NCc2cnccn2)CC1)OC CC1CCN(C(C2CSCCS2)=O)CC1CNC(C1CSCC(=O)N1)=O c1(C(=O)NC2(C)CC(NC(C(CCC)CCC)=O)C2)nccc2c(C)cccc12 Cc1cc(=NC(=O)CC2CC3(C2)CN(C(=O)CCNC(=O)CO)C3)[nH]n1C(C)C Cc1csc(CC(N2CCCC2C(C)(C)C(=O)NCc2cnc(C)s2)=O)c1 C1(C(=O)NC2CCCSCC2)CCC2(CC2)N1C(C1CC(F)(CF)C1)=O N1(C(CCC(C)=O)=O)CCC2(CCC2)C(NC(=O)CCCc2cc(C)sc2C)C1 CC(C)(CCCNC(=O)CCn1cccc1)NC(=O)CC1CCC1 C1(CC=C)CCN(C(C2(CNC(C3C4CCCC34)=O)CC2)=O)C1 c1(C(C)NC(CCC(=O)N(C)C)=O)ccc2c(c1)CCN2C(C1(C(=O)O)CC1)=O CC(=O)C(C)CC(C)C(=O)N1C2CCC(C2)C1C(=O)N(CC(C)O)CCO N(C1CN(C(C2CC2F)=O)Cc2ccccc21)C(c1c(C)nn(CCC)c1C)=O C1(C(=O)NC2CSC2)CN(C(C2CN3CCC2CC3)=O)C2(CCC2)C1 N1(C(c2c(CC)onc2C)=O)CCC(C(=O)NC2CCCNC2=O)C(C)(C)C1 c1(OC)ccc(Br)cc1CNc1cn(C)c(C(N2CCC(C(F)(F)F)C2)=O)n1 C(=O)(C(F)CCC(C)(C)C)NCCN(C(CC(C)CN(C)C)=O)CC1CC1 C(c1cccc(C#N)c1)=CC(=O)NCCN(C)C(C1(C2CCC2)CC1(F)F)=O C(CN=c1[nH]c(N2C3CCC2CC(F)(F)C3)nc2c1CSC2)(C1CC1)OC C1(C(=O)NCCC(C)CCNC(C2(C#N)CCC2)=O)C2Cc3cc(Cl)ccc3C12 C1(C(N2C(C(=O)N(C)Cc3sccc3C)(CC)CCC2)=O)CCCC(=O)N1C N1(C(C2C(C(C)O)C2)=O)CCN(C(c2nnc(O)nc2O)=O)CC1C C1(O)(C(C)CNC(=O)C=CCN(C)C)CCNC1 N1(C(C=CC=CC)=O)CC2CC2(NC(=O)Nc2cccc(I)c2)C1 N1(C(c2coc3cc(F)ccc23)C(N2CCCCC2)=O)CCC2(CCSCC2)CC1 C1(C(N2CC3(C(NC(c4cnc(C)nc4)=O)CC3)C2)=O)CCc2nncn2CC1 CCC(Cc1ccccc1)CC(=O)OC.c12ncnc(OC)c1o[nH]2 N1(C(COCCOC)=O)CCC(CNC(=O)CC2CC(C)=NO2)C1 C(=O)(C1CCCn2nccc21)NCCCC(C)NC(c1ccc(C)c(CO)c1)=O C1(NC(c2cnn(CC)n2)=O)CN(C(c2conc2-c2ccccc2)=O)CC1F C(=O)(C1Cc2ccccc21)N(C1CCCN(C(c2nc(CC)sc2)=O)CC1)C c1(CC)ccc(C(C)C(=O)NCCCCC(C)NC(=O)C(C)CSC)cc1 C1(NC(=O)Cn2ccnn2)CC(O)CN(C(c2cnc(OCC3CC3)c(Cl)c2)=O)C1 c1(N2CCC(C(C)O)C2)nc(N2CCCC(C#N)C2)c2nnn(C)c2n1 Cc1c(C(=O)NCC(C(C)C)NC(C2(O)CCC(C)CC2)=O)cccc1C1CC1 N1(CC(=O)NCCOCCNC(=O)CCOc2cccnc2)CCCCC1=O c1(C(N2C(C)(C(=O)Nc3c(C)cc(F)nc3)CCC2)=O)cc2cnccc2[nH]1 c1(CNC(=O)C(N2CCCC3(CCCO3)C2)=O)cccc2c1CCS2(=O)=O c1(CNC(=O)Cc2ccc(-c3cc(CO)ccc3F)nc2)ccc(F)cc1Cl C1(F)(C(N2CC(O)(C(C)NC(Cn3c(C)ccn3)=O)C2)=O)CCOCC1 C(=O)(CC(C)(C)C1CCCO1)NCC#CC(=O)NCC(=O)N(c1ccccc1)C c1(C(=O)NCC2C(CNC(c3c(C)nsc3)=O)C2)cnn2c(C)ccnc12 c1(NCCc2c(C)[nH]nc2O)nccc(=NC(C)c2ccc3c(c2)CCO3)[nH]1 CC1C(NC(=O)C(N2CCCCC2=O)C)CCCN1C(=O)CC12CCC(CC1)C2 C1(C(N(CC(CC)NC(c2c(OCC=C)cccn2)=O)C)=O)CCCC(C)CC1 C(=O)(CC(CC)C(C)(C)C)NC1CC2(C(C(=O)NC(CC#C)CCOC)C2)C1 C(=O)(CN=c1cc[nH]cc1)N1CCCCC(N(C)C(c2cscc2C(F)F)=O)C1 C1(C(N2CCC(n3ccnn3)C2)=O)C2CC2CN1C(c1coc(C(N)=O)c1)=O C(C(C(=O)N1CCC(N2CCC2)C1)C(C)C)NC(C(CC)C#N)=O C1(C(N2CCSCC2CO)=O)(NC(c2scc(C)c2)=O)CCOCC1 C1(NC(COCCC#C)=O)(CNC(C2OCC3CCCC23)=O)CCCCCC1 c1(N(C)C)cc(F)ccc1CN1CCCC1CCC(=O)NCc1ccncc1 CC(C)C(F)(CNC(=O)CN(C)C1CC1)C(=O)NCc1csc(O)n1 C(=O)(C#CC(C)(C)O)NC(c1n(C)ncc1)C(N1CCOC(C)(C(C)C)C1)=O Cc1nnccc1C(N1CC=CC(NC(=O)CCc2ccsc2)C1)=O C1(CNC(C(CCC)CC)=O)CC2(CO1)CN(C(=O)Cc1ccsn1)C2 C1(C(N(CCNC(C2CC(C(F)(F)F)CO2)=O)CC)=O)CC(=O)NC(=O)C1 C1(C(C)NC(c2c(C(F)(F)F)n[nH]c2C)=O)CN(C(=O)CCSCC(N)=O)CCO1 N1(C(C(C(C)O)(F)F)=O)CCC(C2CC2)(NC(c2snc(Cl)c2Cl)=O)C1 C(=O)(CCCC(=O)NC1CN(C(=O)CSC)CCC1c1ccccc1)NC C(=O)(CN=c1cc[nH]cc1)N(C1CCN(C(c2cc(COC)on2)=O)C1)CCC C1(C(N2C(C(C)(C)NC(=O)COC3CC(F)(F)C3)CCC2)=O)CCCC(=O)C1 N1(C(C(CC)O)=O)CC(CN(C(=O)C2=C(C)CC2)Cc2ccccc2)C2(CC2)C1 CC1(NC(=O)CCCc2ccccn2)CC(NC(c2cc(Cl)n[nH]2)=O)C1 c1(C(=O)NC(COC)CNC(=O)C(C)n2cncn2)cc(C)c(C)o1 CC1OC2(C(=O)N(C)CC3(O)CN(C(=O)CC(C)n4cccn4)C3)CCC1CC2 c1(CCC(=O)OCc2ccc(-c3ccccc3)o2)ccnn1CC1CCC1 C(=O)(C(C)(C)C(=O)N(C)C)NCC1N(C(c2cnc(C)s2)=O)CC1 c1(CC(=O)NC2(C(=O)NCC)CC2)ccccc1.C(=O)CNC(=O)C1CC1 c1(CC)[nH]c(=N)sc1C(N1CCC(N(C(C2CC(F)(F)C2)=O)CC)C1)=O C(=O)(C(C(C)(C)C)NC(C)=O)NC(CCC)CNC(C1(F)CCCCC1)=O N1(C(C=CCC)=O)CC2(C1)C(NC(=O)C(F)=C(C)C1CC1)CCS2(=O)=O N1(Cc2cncc(C)c2)CCCC2(CCN(C(=O)C(C)Cc3ccccc3)C2)C1 c1(OC)cccc(I)c1C(N1CC2(CC(C(=O)Nc3ncc(F)cc3Br)C2)C1)=O c1(CC(C)NC(=O)C(N)Cc2cccc(F)c2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] c1(NC(COC(C=Cc2ccc(C3C(C)C3)o2)=O)=O)ccc(Br)nc1Br c1(C(N(CC(C)NC(c2cccc(NC(C)=O)c2)=O)C)=O)cnc2ccccn12 C1(C(N2C(CCNC(=O)Cn3cccn3)CSCC2)=O)CC2CCC(C1)O2 C1(OC(C(=O)NCC(C2CC2)NC(c2n(CC)nnc2)=O)C)CCCCCC1 Cc1ccc(CNc2ccc(F)c3cnccc23)c2ccccc12 CC1CCC(CNC(c2cc(N)c(Cl)cn2)=O)N(C(c2cc(C(F)F)no2)=O)C1 c1(C(=O)NCCCN(C(C(CC)c2ccccc2)=O)C)ccc(F)c2c1CCC2 N1(C(CCC=CC)=O)CCC(NC(c2noc(C3CC3)c2C)=O)CC1C1CC1 C1(C(=O)NC(c2ccccc2)C)CCc2nnc(-c3ccccc3)n2C1 Cc1cc2c[nH]nc2cc1C(=O)NC1CC1NC(C1CC1C1CCC1)=O C1(NC(CC2CCCC(OC)C2)=O)CC2CCC(C1)N2C(=O)C(C)CS(C)(=O)=O C1(CNC(C2CCN(Cc3ccccc3)C(=O)C2)=O)C2CCCCCCC12 CCN=c1[nH]cc(C(N2CCN(C(C3(C)CCN(C)C3=O)=O)C(C)C2)=O)s1 C(C1=CCC2CC1C2(C)C)(c1nnnn1CCCF)NCc1cncc(C)c1 c1(C(=O)OC)cn2c(n1)CC(C)CC2.c12ccsc1C(=O)COC(=O)C(=O)N2 c1(NC(C)=O)cc(C(=O)NC(CN2CCCC2)CC(C)C)ccc1Cl c1(C(N(CC)CC2CCN(C(=O)CS(N)(=O)=O)CC2)=O)n[nH]c2cccnc12 C1(NCC(C)(C)c2nccs2)(CC(=O)OC(C)(C)C)CCCCC1 c1(C(=O)NC(C2CCCCN2C(c2scnc2Cl)=O)C)nccnc1C(F)(F)F CN(CCCC(=O)NC(C)(C)CNC(C1CN(C2COC2)C1)=O)N=O N1(C(CNS(NC)(=O)=O)=O)CC2CCCC(N(C)C(C3CSC3)=O)C2C1 Cc1csc(C(C)C(=O)NC2(CNC(C3CCC(=O)O3)=O)CC2)n1 C(=O)(CCCCCCCS(C)(=O)=O)NC1C(CC)N(C(C2CC3CC3C2)=O)CC1 C1(C(=O)NCCCC(=O)OC)CC2(CCCC2)CO1 C1(C(N2C(C)(CC)CC2)=O)CCN(C(C2(OC)CCC2)=O)C(C)(C)C1 N1(C(C(=O)NC(c2ccc(C(F)(F)F)cc2)CCC=C)=O)CCCC(C)(C)CC1 CC1(C)CC(C(N2CC3C(NC(=O)CCn4ccnc4)C3C2)=O)C(C)(C)O1 C1(NC(CC2CCC(=O)N2)=O)CC2CC1CN(C(c1cc(F)c(Cl)cc1F)=O)C2 N1(C(C2C(C(=O)OC)C2(C)C)=O)CCCC(O)(CNC(=O)CC2CC=CC2)CC1 c1(C(=O)NC2C(CNC(c3n[nH]cc3F)=O)C2)cc2ccc(Br)c(F)c2[nH]1 N1(C(C(F)OC)=O)CCN(C(C2CCCCC2)=O)C(CS(C)(=O)=O)C1 c1(-c2c(COC)cccc2)cccc2nc(C(N3CCC(CO)C(F)C3)=O)cn12 c1(C(N2C(COC)C=CC2)=O)ccc(F)c(F)c1N.C12(CCCCCC1)C(=O)N2 N1(Cc2c(C)cc(Br)cc2)CCC2CN(C(=O)CCN(C)C)CC2C1 C1(NC(C2C(C)(C)C2)=O)CN(C(C2(C)CCCCNC2=O)=O)CC12CCOCC2 C(=O)(CC(O)CCCC)N(C(CC(=O)NC(CC#C)C)C)C N1(Cc2cn(CCCCCCO)nn2)CC2(CC2)CC1C(=O)Nc1c(C)nc[nH]1 CCCCC(CNC(C1CCCO1)=O)NC(c1cc(-c2cccnc2)n(C)n1)=O C1(C(=O)NC(CCSC)C(=O)NCc2cnccc2Cl)CC(=O)NC1(C)C c1(COCC)nc(N(CCCNC(c2sncc2C)=O)C)cc(C)n1 C(=O)(C1CCc2nccn21)NC1C2(CCN(C(CC=CC)=O)C2)C1 CC1(C(=O)NCc2ccc(C(=O)Nc3cncc(Cl)c3)s2)CCCC1O c1(C(=O)NCCCOCCC(=O)NC(c2nnnn2C)C)coc(C2CC2)n1 c1(CCNC(C2CCOC2C(=O)NCC23CCCC2C3)=O)cccc(F)c1 C1(CNC(=O)CC2CCC2)CN2CCCCC2CN1C(c1ccccn1)=O C1(C(N2CCC(N(C(=O)CCN(CC(F)(F)F)C)C)C2)=O)(OCC)CCCC1 C1(CC(C)CN2CCOC2=O)NC(=O)CCN(Cc2ccccc2)C1=O C(CC(C)C)(C(=O)N=c1cc(C)n(CCO)[nH]1)N(C(C)=O)C CCC(CCCC(=O)N(CCCO)CCO)NC(C1CCC2CC1CO2)=O c1(C(N(C2CCCCN(C(c3n[nH]cc3F)=O)C2)C)=O)cccn2ccnc12 C12(C(=O)NCc3cc(C)c(F)cc3)CC(CN=[N+]=[N-])(C1)OC21CCNCC1 c1(C(N2CC(C)(NC(c3cc(Cl)nnc3Cl)=O)C2)=O)ccc(F)cc1[N+](=O)[O-] C=CC1(CC(=O)NC(C)CC(C)NC(C2(O)CCSC2)=O)CCCCC1 C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NCC2(NC(C)C)CC2)C2CCC1C2 C(CCC(=O)N1CCCC1CNC(=O)CC1(C)CC1)OC(C)C c1(OC(C)C)cnc(NC(=O)C(N2CCCC2Cc2nn[nH]n2)=O)cn1 C1(NC(CCSc2n(C)ccn2)=O)CN(C(=O)C(O)C(F)F)CC12CC2 N1(C(Cc2cnc(C)[nH]2)=O)CC2(CC(NC(=O)CC3CC3(C)C)CO2)C1 N1(C(c2ccc(OC)nc2)=O)CCN(C(c2ccc(C)c(F)c2)=O)C(C2CC2)C1 CC1=C(C(=O)NC(C)(CNC(=O)C(C)C2CC2)C2CC2)SCCO1 C1(C(C)NC(=O)C(c2ccccc2)F)CCCN(C(C23CSCC2C3)=O)C1 C1(C(N2CC3C(C2)CNO3)=O)CCc2nnnn2CC1.C(=O)(COC(C)C)CC N1(C(C(C)OCC#C)=O)CCCN(C(c2cnc(OC)cn2)=O)CC1C c1(C(=O)NC2(CC)CN(C(C3N(CCC)C(=O)CC3)=O)C2)cccn(C)c1=O C1(C(=O)NC2CC(CNC(c3cc(O)cc(O)n3)=O)C2)CCC2(CCOCC2)O1 c1(C(N2C(CCC(=O)NCc3ccc(Cl)cc3)CCCC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nn(C)c2c1C(NC(NC1CCc3ccccc31)=O)CCC2 N1(C(=O)Nc2cccc(CC)c2F)c2ccc(F)cc2CCC1C c1(C(N2CCCC(CC(=O)NCC3CCCCO3)C2)=O)cc2ncccc2o1 C(=O)(C(C)C(O)C(C)C)NC1CN(C(CCc2cncc(C)c2)=O)CC1O Cc1nc(N(C)CC2CCCN2C(c2coc(O)n2)=O)nc2ccccc12 CCCC(C)CNC(=O)C=CC(C)NC(c1c[nH]c(=N)o1)=O c1(NCC(C)=CC(=O)N(C2CC(C#N)C2)C(=O)CN(C)C)snnc1C C1(NC(C(C)CO)=O)CCC2CN(C(=O)C=Cc3cnn(C)c3)CCC2C1 c1(C(C)=O)c[nH]c2cnccc12.C1(=O)C(C)C(C)NC(=O)c2n[nH]cc2N1.C1CC1 CC(C)(C)CC(F)C(=O)NC(CO)C(N1CCCCC1CCO)=O CN1CCn2ncc(CNC(N3CCC(NC(N)=O)CC3)=O)c21 c1(C(N(C2CCC(NC(CCC(=O)NC)=O)C2)C)=O)cc(F)cnc1O Cc1cc(C(N2CCCC(CCNC(c3ncnn3C)=O)C2)=O)c(C)cc1Br c1(C(=O)NCCOCCNC(c2n(C)nc(O)c2)=O)ccc(C#N)c(O)c1 C1(NC(c2ccc(C(F)(F)CF)cc2)=O)C2CC(CN(C(=O)CO)C2)C1CO C1(O)(C(C)NC(CCC=C(C)C)=O)CCN(C(c2cnc(-c3ccco3)s2)=O)C1 c1(C(C)NC(C2(OC)CN(C(=O)Cc3ccc(C)o3)C2)=O)nccc(O)n1 C1(C(=O)NCCC(=O)NC2CC2)CCCN(C(=O)CC2CC3(CC3)CO2)CC1 C(C(CO)CC(C)C)NC(CN(C(C1(CC)CCOC1)=O)C)=O Cc1nc(C)c(C(N2CCN(C(C3CCN(C(=O)C(C)C)CC3)=O)CC2)=O)o1 N1(S(CCCC#C)(=O)=O)CCCC2(CCN(c3ccccc3)C2)C1 c1(C(N2CCC(N(C(=O)CSC(F)(F)F)C)C3(C2)CC3)=O)c(F)ccc2c1OCC2 N1(c2c(C)cccc2)C(=S)NC(C2CC2Br)C2=C1CC1(CCOCC1)NC2=O c12cnc(cn1)c(=O)n2C.C(=O)(NOCC(N)=O)C1(COC)CC1 c1(C(N2C(CCNC(C(C(C)C)C)=O)CC(F)(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl CCCCC(CCC)NC(=O)CCC(C)NC(=O)CCc1nncn1C c1(C(=O)NCCC2CCCN(C(C(CCC)OC)=O)C2)cc2c(C)cccc2[nH]1 N1(c2snc(C(=O)OC)n2)CCC(C)(NC(C2CC(F)(CO)C2)=O)C1 N1(C(c2c(C)c(N)ccc2)=O)CC2CC(NC(=O)C(F)CC3CCC3)CC2C1 Cc1ccc2sc(NC(=O)C(N3CCCC(C(N4CCC4)=O)CC3)=O)nc2c1C C1(NC(c2cc(C)ns2)=O)CCCC(C(N2CC3(C=CCO3)C2)=O)CC1 N1(Cc2c(C)n(C)nc2)CCC(F)(F)C(C(=O)Nc2cnc(Cl)c(C(N)=O)c2)C1 c1(C(=O)NC2(C)CCN(C(C(CCO)N(C)C)=O)C2)cc2ccc(F)cc2o1 N1(C(CCC(C)SC)=O)CC2CC(CNC(=O)C(C)(F)F)CC1C2 CS(=O)(=O)CCC(=O)CNC(CSc1ccccc1)CC(=O)O C1(O)(CN(C)C(C2CC2F)=O)CCN(C(c2cncn2-c2ccccc2)=O)C1 C(C(C)C(C)C(=O)NC1CC1CNC(c1cscc1C)=O)OC N1(Cc2ccc(C)[nH]2)CCC2(CCCC2C(=O)Nc2cc(O)c(Cl)cc2F)C1 c1(C(=O)NC(CC(C)NC(c2ccn(C(F)(F)F)n2)=O)C)ccc(F)c(Cl)c1 c1(OC)ccc(CC(=O)NCC(C(=O)O)C2CCOC2)c(Br)c1 C(C)(CCC(=O)N(C)CC1COCCN1C(c1occc1Cl)=O)OCC N1(C(CC(C)(C)NC(C(C)N(CC)CC)=O)=O)CC2(CCC(=O)NC2)C1 C1(CC(=O)NC2C(CNC(C(c3cn(C(C)(C)C)nc3)=O)=O)CC2)CCCCC1O N1(C(C(COC)C)=O)CC(NC(c2cc(=O)cc(Cl)[nH]2)=O)CC(F)(F)C1 N1(C(c2cnc(CC)[nH]2)=O)CC(NC(C2CN(C)CCO2)=O)C(C)C1 C1(C(=O)N(CCCCCO)CCO)C2CC(O)C(C2)N1C(=O)COCC1CCOC1 c1(C(=O)NCCCCNC(c2cnc3[nH]ncc3c2)=O)cc2cc(Cl)cnc2[nH]1 c1(OC)ncccc1C1CCN(CCn2cc(C3CCCCO3)nn2)C1 c1(CNC(CC2C(C)C2)=O)nnn(C)c1C(=O)N(CCn1cncn1)C1CC1 CCC(CC)(CC)NC(=O)CCC1CCN(C(=O)CCC(C)SC)C1 c1(C(N2CCC(C)(C(=O)OC)C2)C(=O)NC)cc(CC)cc(F)c1.C=CC C(=O)(N=c1[nH][nH]c2c1CCCC2)C1N(C(c2cc(OCC)c(Br)cc2)=O)CCC1 C1(O)(C(C(=O)NC(CC#CC)C)(F)F)CCN(C(=O)OC(C)(C)C)CC1 CN=c1cc(C(N2CCCC2C(=O)OC)=O)cc[nH]1.C12(C(=O)O)CC1C2 C#CC1(C(=O)NCC2CN(C(=O)C(C)=CC)CC2C(F)(F)F)CCCCC1 Cc1c(Cl)ccc(C(N2CCC(C(C)NC(C3CNC(=O)N3)=O)CC2)=O)c1Cl c1(C(N(C2CCN(C(=O)CC3CSCCS3)C2)C)=O)ccnc2c1ncn2C Cc1cc(C(C)NC(=O)NC2(C(c3ccccc3)O)CCCCC2)ccc1Cl CCC(CC)CCC(=O)NC1(C(=O)NC(=O)C2CC2)CC1.n12cc(nn1)CCC2 c1(OC)ccc(C(=O)NC2CCOC(C)(CN)C2)c(F)n1 CCC(CC(=O)NCC(C)NC(=O)OC(c1ccccc1)=O)NN1CCCCC1 C(=O)(C1=CCCC1C)NC(C(=O)Nc1c(C)ccnc1)(C)C1CCC1 c1(NCC(C)OC)ncnc(NC2CC(=O)N(C)C2)c1C c1(C(N2CCOC3CC23)=O)ccc(OCC2CC2)cc1 Cc1cc(F)sc1C(=O)NCC(O)CN(C(=O)CCc1ccncc1Br)C N1(Cc2c(C)cccc2)CCC2C1CCCN2C(c1cnn(C)c1C(F)(F)F)=O N1(C(C=CCSc2ccc(OC)cc2)=O)CCC2CCN(C(=O)C3=CCC3)CC12 C1(CC2CCC(CC)O2)CN(C(c2noc(C3CCCC3)n2)=O)CCO1 CCC(CNC(=O)CCCCCNC(c1c(C)noc1C)=O)CC(C)C n1(CC#N)cc(C2NC(=O)Nc3c(C(N)=O)cc(-c4cccnc4)cc32)cn1 c1(NC(CCC)CCCO)ccc(S(=O)(=O)NC(CC(C)C)CC(C)C)cc1Cl O=C1CCC(=O)NC2CCCCC2N1.c1(NC2CC2)nccc(SC2CCCC2)n1 C(C)(CC(=O)NCC1(C)CCN(C(=O)C(C)(C)CO)CC1)(C(F)(F)F)N(C)C C12(C(=O)NCCC(C(C)C)C)CC(CO1)N(C(=O)CC13CCCC1C3)C2 c1(CNCC2(NC(=O)Cc3ccccc3)COC2)ccc(O)cc1Cl c1(C(=O)OC)ccc(O)c(C(N)=O)c1.c12ccc(cc1)C1(CC1)C(=O)NC(C)C2 N1(C(CCc2cc(OC)no2)=O)CCC(NC(=O)Cc2cc(Cl)n(C)n2)C(O)C1 c1(C(=O)NC(C2(CNC(C3CC(O)C3)=O)CC2)C)cccn1C1CCCC1 N1(C(Cc2cn(CC)nc2)=O)CCN(C(c2[nH]ccc2C2CC2)=O)CC12CCC2 C1(CC=C)(NC(C2CCC(CC)C2)=O)CCN(C(=O)C(O)CC)C1 N1(C(CCc2c(C)nn(C)c2)=O)CCOCC(CNC(=O)C(C)CN(C)C)C1 C1(NC(C(C)(C)OC(C)=O)=O)CCCC(NC(c2csc(Cl)n2)=O)C1 CC(C)CC(C)C(=O)N1CCC(F)(CNC(=O)C(C)(C)C2CCCCO2)CC1 C12(C(N(CCNC(c3noc(CC)c3C)=O)C3CC3)=O)CCOC1CS(=O)(=O)C2 Cc1cc(C(=O)NC2CC(n3cc(Cc4nc(C(=O)O)co4)nn3)C2)co1 C(=O)(C1CSc2ccccc21)NC(CNC(c1c(C)c(O)ccc1)=O)C1CC1 C(=O)(CCCCC(C)(C)C)N1CC(OC)N(C(=O)CCOC)CC1 c1(C(C)NC(=O)NCC2(CO)CCCC2)cn(C)c2cc(F)ccc12 c1(C(CC)(C)C)ccc(C(=O)NCC23CC(NC(C4CC5CC4C5)=O)(C2)C3)cc1 c1(NC2(CCNC(C3N(S(C)(=O)=O)CC3)=O)CCCC2)cc(O)nc(O)n1 c1(OC)c(C(N2CC=CC2CNC(c2nc(Br)sc2C)=O)=O)c(C)nn1C c1(OC)ccc2cc(-c3c[nH]c(=NCCc4ccccc4OC)s3)ccc2c1 C1(N(C)C(C2CNC(=O)C2)=O)CCCCN(C(C2(F)CC=CC2)=O)C1 N1(C(CN2CCC(C)C2)=O)CCN(C(=O)CCC2CCCN2C)CC12CC2 Cc1cc(C(=O)NCC2CCCN(C(c3nc(O)sc3C)=O)C2)ncc1C(N)=O C(=O)(CCCCCS(N)(=O)=O)NCCCCC(CO)NC(C(C(C)C)NC(C)=O)=O c1(CC(=O)N(C2CCN(C(C(CC)N3CCOC3=O)=O)C2)C)cccc(C)c1F N1(C(C2N(C)CCC2)=O)CCC2(CC2NC(=O)CC2CCCCO2)C1 C1(NC(=O)C(=O)NC2CC(c3ccc(F)cc3)C2)COC2(CCCCC2)C1 C12(CNC(c3nc(Br)c[nH]3)=O)CC(CN1C(=O)C=C(C1CC1)C1CC1)C2 CC1CCN(C(c2cn(C)nc2-c2cccs2)=O)CC1NC(=O)C(C)CO c1(NC(c2nc(CNC(=O)C(F)(F)CO)n[nH]2)=O)ccc(C2CCOC2)cc1 CCC(O)C(F)(F)C(=O)NCC=CCC(N1CC(O)(C(N)=O)C1)=O c1(C(=O)NCC2=CCN(C(C3C(C(=O)OC)C3)=O)CC2)cccn2nnnc12 C1(C(=O)NCC2N(C(C(C)(C)C3(C)CC3(F)F)=O)CC2)(N(C)C)CCOCC1 C1(C(N2CC(NC(CC(C=C)(C)C)=O)C2)=O)CCc2nc(C)cn2C1 c1(C(=O)NCC2C(NC(Cc3scc(C)c3)=O)CC2)n[nH]c(C)c1Cl c1(-c2n(CC)nc(CCOC(C)C)n2)cc2cc(F)c(F)cc2[nH]1 C(=O)(CC(C)C(F)F)NCC(Cc1ccccc1)NC(C1C(CC)C1)=O C1(CNC(Cn2c(C)nnn2)=O)COCCN(C(=O)CC2CCC(=O)O2)C1 c1(C(=O)NC(C(=O)NCC(C)(C)C2CCC2)Cn2cncn2)cc2n(n1)CCC2 N1(C(C(C)c2ccco2)=O)CC(C(N2CCOC(C)(C)C2)=O)CC1(C)C CN1C(=O)OCC12CCN(C(=O)Cc1nn(C)cc1Br)C2 c1(C(N(C)CC2N(C(c3nn(CC)nc3C)=O)CCCC2)=O)cc(Cl)ncc1N C(=O)(N=c1[nH]ccc2cc(Cl)ccc12)C1CN(C(Cc2ccc(C#N)cc2)=O)C1 C1(O)(CNC(c2ccnc(Cl)c2F)=O)CCN(c2ncncc2I)CC1 N1(C(c2c(C)cco2)=O)CCCC(C(N2CCCC(CS(N)(=O)=O)C2)=O)CC1 C1(NC(c2n(C)c(O)nc2)=O)CC2CC(C1)N(C(c1cc3c(s1)CCOC3)=O)C2 c1(NC(C2N(CCCC(=O)OCC)CC(C)(C)CC2)=O)ccc2nc(C)oc2c1 Cc1ccncc1NC(C1(n2cc(CSC3(CO)CCC3)nn2)CCOCC1)=O C(CCSC)(C(=O)NCC(C(F)(F)F)N1CCN(C(=O)Cn2cccn2)CC1)OC N1(C(c2cc(OC)ncc2)=O)CC2CN(C(c3cc(O)no3)=O)C2C1 C(=O)(CCCCSC(C)(C)C)N(CCN(C(C(c1cccnc1)OCC)=O)C)C N1(C(CN(C(C)C)C)=O)CCC(O)(CNC(=O)CN2C(=O)CSC2=S)CC1 C(=O)(CCCCCCCS(C)(=O)=O)NCC1C(C)(C)CCN(C(CCC=C)=O)C1 c1(C(N(CC=CC(=O)NCc2ccn(CCC)n2)C)=O)cc(=O)cc[nH]1 N1(C(CN(C(=O)C(C)COC)CCC)=O)CC(N=[N+]=[N-])C1 C1(NC(=O)C(c2ccc(Br)cc2)O)CN(C(c2cc(F)ccc2Cl)=O)CC1(F)F C1(C#N)(C(=O)NCc2cccc(C(=O)NCCS(CC)=O)n2)CCCCC1 O(NC(=O)C(C)C(C)NC(c1c(C)ncnc1C)=O)CCCC c1(C(N2CC(OC)C(NC(c3snnc3C(C)C)=O)C2)=O)cc(C)nc(C)c1O C1(F)(C(=O)NC2(C)CC(NC(c3c(OC)cccc3)=O)C2)CCC(C)CC1 c1(CC(C)NC(CC(C)C)=O)ccc(C2CC2)cc1.c12cc(on1)CNC2=O c1(C(c2nnnn2CC(F)F)NCCc2ncn(CC)n2)ccncc1F C(CC)(C(=O)NC(C)CN(C(c1csc(-c2ncccn2)n1)=O)CC)OCC CCCC(C(=O)NCC(CNC(=O)C=Cc1ccc(F)cc1)OC)S(N)(=O)=O N1(C(c2cnc(CC)nc2O)=O)CCC2(CCC2)C(NC(=O)CCS(C)(=O)=O)C1 c1(C(=O)NCC(CO)NC(C(=Cc2ccncc2)C)=O)cc(Cl)c(C)cn1 Cn1nc(CC(=O)NCC2(C)CN(CC3CC3)C2)cc1C1CCCO1 C1(OCC=C)CCN(C(=NCC2CCC23CCOCC3)NC2CCCC2)C1 CCC(C(=O)N(CCCO)CCO)NC(=O)COc1ccccc1 CCCCC(CNC(C1(CN(C)C)CC1)=O)NC(=O)COC1(C)CCC1 C1(C(=O)NCC(C(C)(C)C)NC(C2C(CC)OCC2)=O)CS(=O)(=O)CC(=O)N1 c1(CC)cc(C(=O)NC(CNC(C2CCSCC2)=O)(CC)CC)nn1C c1(C(=O)NC(CC)CN(C(=O)Cn2cccn2)C)cc(F)c(OC)c(Cl)c1 C1(NC(C2CCC(C)(CC)O2)=O)CC2CCC1CN(C(c1ncc[nH]c1=O)=O)C2 C1(OC)CCCC1C(=O)NCCC1CC(NC(=O)CSCCC(F)(F)F)C1 N1(C(c2cccc(OC)n2)=O)CC(NC(=O)CC2CC(OC)C2)CCC1C n1(CC(=O)NC(CC)CNC(c2snc(Cl)c2Cl)=O)nc(C)c(Cl)c1C C=CC(C)(O)C(=O)N1CCC(Oc2cccc(Cl)c2)C1.C12CCN(CC1)C(=O)C2 C(=O)(C#CC1CCOC1)N1CCN(C(c2c(C)oc(C#N)c2)=O)CC1CC(F)F C1(CCC(=O)N(CCCSC2(C(=O)OCC)CC2)CCC)CCC(=O)N1 CC1CCCC=C1C(=O)N1CCCC(CCC(N2CCC(F)(F)C(O)C2)=O)C1 Cc1nc(N2CCC(C)C2CNC(=O)CC2(O)CCOC2)ccc1[N+](=O)[O-] C12(NC(=O)NCCNc3c(C)c[nH]n3)CC3CC(C(=O)N1)C2C3 Cc1cn2c(CC(N3CCN(CCNC(=O)C(C)C4CC4)CC3)=O)csc2n1 CCN=c1[nH]cc(C(N2CCN(C(=O)CC3CCCSC3)CC2C)=O)s1 C1(NC(c2c(N(C(C)C)C)cccc2)=O)CCN(C(c2csc(Cl)c2)=O)CC1F c1(CC)ccc(C(=O)NCCN(C(=O)CN2CCCC2CO)C)nc1 CC(C)C(O)CC(=O)NCC1(F)CCN(C(=O)CC2CC(C(C)(C)C)C2)CC1 C1(CCNC(C2(CC=C)CC=CC2)=O)CSCCN1C(c1csc(C#N)c1)=O N1(C(c2ccc(Br)c(F)c2)C(=O)NCCOCC)CC(C)Oc2ccccc21 C(=O)(C(C)(CC)CCC(C)C)NC1CCN(C(c2n(CCCC)ncc2)=O)CC1 N1(C(c2c(CC)non2)=O)CCC2CCN(C(=O)C=C3CCN(C)C3)C2C1 C12(NC(C(C)SCCCC)=O)CCC(CN(C(=O)C(=CC3CCCCC3)F)C1)C2 C1(NC(C(CCC)C#N)=O)CC(O)(C2CCN(C(C3CC34CC4)=O)CC2)C1 c1(C(N(C)CC2CC(F)CN2C(=O)C(F)CC2CCC2)=O)ccc2cncn2c1 c1(C(C)(C)C)nc(C(=O)NCCN(C(=O)CCCn2ccnc2)C2CC2)cs1 C(CCC(C)C)(C(=O)NC1(CF)CCN(C(C2(C)CCC2)=O)C1)NC(C)=O N1(C(C2(CNC(CC(C)C(F)F)=O)CC=CC2)=O)c2ccccc2CC1C c1(SC)cnn(C)c1C(=O)NC1CC(C)N(C(c2cccc(=O)o2)=O)C1 c1(C(=O)NC2C3CCN(C(CC4C(CC)C4)=O)C3C2)cnn2cccnc12 C1(NC(C2CCCN(CC)C2)=O)CC2CC(NC(=O)CCC3CCCC3)C2C1 CCC(C)C(=O)C(=O)N1CC2(CCNC(=O)C(C)SC)CCC1C2 C1(c2ccc(Br)cc2)(NC(C(CC)CC)c2nnnn2C2CC2)COCCOC1 C(C1C(C)C1(Cl)Cl)=CC(=O)OC(CC#C)C C(=O)(C(C)C(F)(F)F)N1CC(CNC(c2c(C)nsc2C)=O)OCC1 C1(CCC(=O)NC2(CC(C)C)CC2)CCCN(C(=O)C(N2CCNC2=O)C)C1 CC(C)(F)C(C)(F)C(=O)N1CCCC1CNC(=O)C=CBr Cc1nocc1C(=O)NCC(C)C(=O)NCc1nc[nH]n1 n1(CC)ncc(C(=O)NC2(CCNC(=O)CCCN3CCCC3)CCCC2)c1C c1(C(=O)NCC#CCNC(C2CCCC(OC)C2)=O)ccc([N+](=O)[O-])cc1Cl c1(C(NC(=S)NCc2ccc(Br)c(C)c2O)C)ccc2c(c1)CNCC2 C1(NC(c2cc(C)nnc2)=O)CC2CC(NC(c3cc(C)c(C)o3)=O)CC2C1 CC1(C)CN(C(=O)CCCN2CCCC2)CCC1NC(=O)C=CC1CC1 C=CC1(CC(=O)N(C2CC3CC3C2)CC)CN(C(=O)CN2CCNC(=O)C2)C1 N1(C(c2cncc(NC(C)C)c2)=O)CCN(C(C2(NC(C)C)CC2)=O)CC12CC2 c1(C(C)NC(COC(C)C)=O)nocc1C(N1CCC(CCO)C1)=O C1(NC(C2CCN(C)C2)=O)CC2CN(C(c3cc4ncccn4n3)=O)CC2C1 N1(C(c2cccc(OC)c2O)=O)CCCN(C(c2ncc(Br)cc2C)=O)CC1C C(=O)(CCCCC(C)CC)N(C1CCN(C(C2(F)CCCC2)=O)CC1)CC#C C=C1CCN(C(=O)CCCCCC)C(C(=O)N(C)Cc2ncccn2)C1 C1(C(C)NCC2CCN(C(=O)Cn3cccn3)CC2)CCC(F)(F)CC1 C(CC(COC)C(=O)N1CC(O)CC1(C)C(=O)N(C)CC1(O)CCCC1)OC CC1CN(C(c2ccc(C(N)=O)nc2)=O)C(C)CN1C(C1CCC(=O)O1)=O Cc1cc(C)c(CN(C)C(c2nnsc2C(F)F)=O)cn1 O=C(C1=CC2(CN(C(=O)CC3CSC3)C2)OC1)Nc1ncc2c(n1)CCC2 N1(C(C(c2cnccn2)C)=O)CCOC(CNC(C2CN(C)CCO2)=O)C1 C1(NC(C(c2c(Cl)cccc2Cl)C)=O)CCN(Cc2c(Br)cccc2Br)CC1O c1(OCC)ccccc1C(=O)NC(C1CCN(C(c2ccc(Cl)nn2)=O)C1)C CC1(C(=O)NC2CCOC2CNC(=O)CSC(F)F)CC2CCC1C2 N1(C(C(C)c2cccs2)=O)CC2CN(C(=O)C=CI)CC2C1 CCCCCCCC(=O)N(C1CC2CC1N(C(c1ccc3nccn3c1)=O)C2)C C1(NC(c2c(C(C)C)nco2)=O)CC2C(NC(=O)C(c3ccccc3)C)C2C1 C(=O)(CC(C(F)(F)F)NC(c1snc(C)c1N)=O)NC(CC=C)CO c1(C(=O)NC(CNC(CC(CC)OC)=O)(C)CC)ccc(S(N)(=O)=O)nc1 c1(C(=O)NC2(CNC(Cn3c(C)cc(C)n3)=O)CCC2)ccc2c(c1)ncn2C C1(CNC(C=CSC)=O)CCN(C(C2CC(C(N)=O)C2)=O)C1(C)C Cc1c(NC(=O)C(=O)N(CC(O)Cc2cccc(Cl)c2)C)cccc1F C(CC(F)(F)F)N(C(N1CCC(N2CC(F)C2)C1)=O)CCO Cc1ccc(C(=O)NC2(CO)CN(C(C3CCCCC3F)=O)C2)c(F)c1 C1(C(=O)NCC2CCN2C(c2c[nH]nc2-c2ccoc2)=O)CCS(=O)(=O)C1 C(=O)(C(CNC(=O)CC1CCSC1)CC1CCCC1)N(CCCCC=C)C N1(C(=O)CCF)CCCOC(CNC(c2cc(N3CCCC3)ncn2)=O)C1 C1(NC(c2c(C(C)C)cccc2)=O)CCN(C(c2cnc(O)c(Cl)c2)=O)CC1F Cc1cc(C(=O)O)cc(C)c1NC(=O)C(C)C1CCOC1 c1(CC)ccnc(C(=O)NC(C(=O)NC(C2CCCC2)C)C2CCC2)c1 C1(CNC(C=NOC)=O)CC(F)(F)CN1C(C1CCC(C(N)=O)O1)=O S(=O)(=O)(c1ccc(NC(CO)CCC(C)C)cc1Cl)NCCN(C1CC1)CC C1(NC(CSCC=C)=O)CCN(C(c2cnc(C(C)(F)F)s2)=O)C(C2CC2)C1 C1(N(C(=O)C(C)(O)C2CCC2)C)CCC(NC(=O)Cc2cncnc2)CC1 Cc1ccc(SCCCNC(c2cn(CC3CCCO3)nn2)C(C)C)cc1 c1(C(=O)NCC2CCN(C(C(C(COC)C)C)=O)CC2)c(SC)nc(O)nc1C C1(CC)OCCC1N=c1nc2scnc2c(NCC(C)C(F)(F)F)[nH]1 C(=O)(C(CCF)NC(C1CC(NC(c2ncc(F)cn2)=O)C1(C)C)=O)OC C1(C(=O)NC23CC(C)(C2)C3)CC2(CCN(C(c3cc(S(C)(=O)=O)co3)=O)C2)CO1 N1(C(C2CC2F)=O)CC(C2CCCN(C(c3cnc4ccncc4c3)=O)C2)C1 N1(C(c2ccc(C(C)F)cc2)=O)CCCOC(CNC(=O)CP(C)(C)=O)C1 c1(C(=O)NCC(=O)NCC(CCC)OC)cnn2cccc2c1.COC CCC(CC(=O)N(CC(O)CNC(c1cnn(CCO)c1)=O)C)OC N1(C(c2cc(CC)on2)=O)CC=CC(NC(=O)CN(CC(=O)NC(C)C)C)C1 O(N=C1CCCCCC1)CC(=O)NC1CN(C(c2c(C)nncc2)=O)C(C)C1 c1(C(=O)NCC(C)NC(C(c2ccccc2)OC)=O)cnc2c[nH]nc2c1 c1(C(N2C(C(N(C)Cc3cc(C)no3)=O)CC2C)=O)cccc2c1CCC2 C1(C)(C(N2CC(C)C(NC(=O)C3=COCCO3)C2)=O)CCCCC1(F)F C1(CNC(C(=O)NC(C)C)=O)CC2CCC1N2C(=O)CNc1ccccn1 C1(C2CCN(C(N3CCCS3(=O)=O)=O)CC2)(NC(C2Cc3nncn3C2)=O)CC1 N1(C(c2cccc(OCC(F)(F)F)c2)C(=O)NC)CC2CC(C1)N(C)C2 O=C(CS(=O)(=O)CCCc1ccccc1)NC1CCNC12CC2 Cc1cnc(C(=O)NC(C(N2CCC(CO)C(C)C2)=O)C2(C)CC2)c(F)c1 c1(NC(CC)CNC(=O)CC(c2cccc(F)c2)C)nc(C)nc(=N)[nH]1 CC1CC2(CCC2)CN1C(C1CCC(CNC(=O)Cc2ccccc2O)O1)=O N1(C(C2(CC)CCCC2)=O)CC2CCN(C(c3cncc(Br)c3)=O)C2C1 C1(C2CC2)(CNC(CCCCNC(C)=O)=O)CCN(C(=O)Cn2cc(C)cn2)C1 C1(C(=O)N(C(C)CC(C)C)C)(COC)C=CCN1C(C1SCCS1)=O c1(C(N(CCCNC(C2CCC2C(N)=O)=O)CC)=O)cc(C(F)(F)F)ncc1N N1(C(c2cc(CC(C)C)on2)=O)CCOCC(F)(CNC(c2cn(C)nn2)=O)C1 C1(NC(=O)CCC2CC2)CCN(C(=O)C(c2cccc(F)c2Cl)(F)F)C12CC2 c1(C(=O)NC(CC(=O)OC)(C)C)ccc(S(=O)(=O)NCC2CC2)cc1 CC#CCCC(=O)NC1CN(C(=O)C(c2cnccc2C)(C)C)CC1C N1(C(CC)CC)CC(C(=O)N(C)CCNC(=O)C(C)Cc2ccnn2C)CC1=O c1(C(=O)NC2CCN(C(C3CCC(=O)C3)=O)C23CC3)cc2ccccn2c1 N1(C(=O)C(O)CN2CCOCC2)CC(S(=O)(=O)N2CCN(CC3CCC3)CC2)C1 N1(C(N2C(C(N3CCCCC3)C)CCC2)=O)CC2CCCC1CCC2 c1(C(=O)NCC2COCCN(C(=O)C(CCO)N(C)C)C2)n[nH]c2c1CCOC2 C(=O)(CCCCCSC)N1CC(C#C)(C(=O)NOCC2CC2)C1 C1(CNC(=O)Cc2ccsn2)CCCCC1NC(c1ccc(N(F)F)cn1)=O C1CCCC(=O)NC(C)C(=O)N1.Cc1noc(-c2ccccc2)n1 C(=O)(C1=COCCO1)N1CC=CC(NC(c2[nH]cc(CC(C)C)c2)=O)C1 CC1(C)CC=C(C(=O)N2CCC(N(CCO)C(c3csc(S(C)(=O)=O)c3)=O)C2)CC1 C(=O)(CS(=O)CCC(F)(F)F)NC(C(C)C)Cc1c(F)ccc(Cl)c1F C(CC(C)C(=O)N(CC(O)CNC(=O)CS(=O)(=O)NC)C)=CCC C1(C(=O)NCCN(CCC)CCN2CC=CC2)CCN(S(=O)(=O)NC)CC1.C N1(C(Cc2ccc(C)o2)=O)CCC2CN(C(C3CCS(=O)(=O)C3)=O)CCC12 CC(C)C(C#N)C(=O)NCCc1ocnc1CNC(=O)CSc1ccc(F)cc1 c1(C(N2C(CNC(C(c3ccccc3)OCC)=O)CC2)=O)cc(F)n(C)n1 CC(CC(=O)NCC(O)CNC(C1CCCN1C(c1ccccn1)=O)=O)N(C)C C1(CNC(c2c(CC)onc2)=O)C2CN(C(C3CCC(N(C)C)C3)=O)CC12 C(C(=O)NOCC(=O)OC)N(CCC)C(C1CC1(C)C1CCC1)=O n1(C(C)C)ncc(C(=O)NCC2(CNC(=O)C(N3CCNC3=O)C)CC2)c1N c1(C(C(=O)NC(CC(C)NC(C(C)NC(=O)NC)=O)C)C)cccc(C(=O)OC)c1 N1(C(COCCCC(C)C)=O)CCC(NC(C2CC(F)(F)CS2)=O)CC1C1CC1 c1(C(N(CC(C)NC(c2cnn(C)c2C#N)=O)C)=O)cnc2c[nH]nc2c1 N1(C(CCCC#N)=O)CC(=O)NCC1C(N1CCN(C2CCC2)CC1)=O N1(C(=O)OC(C)(C)C)CC2CN(C(=O)Cc3cnn(C4CC4)c3)CC2(C(=O)O)C1 c1(CC)cc(C)c(C(N2CC(CC(F)C(=O)N3CC(C)(CF)C3)C2)=O)o1 CCC(CC(F)F)C(=O)NCCC(C)(C)NC(=O)C(C)O c1(C(=O)NC(CC(C)NC(Cc2cn(CC)nc2)=O)C)c(C)nsc1C C1(CNC(CC(C)O)=O)CN(Cc2c(F)cccc2F)CCC1(F)F C1(CNC(C2C(C#C)C2)=O)(NC(c2c[nH]ccc2=O)=O)CCCCC1 c1(-c2c(C(N3CC(CNC(C=NOC)=O)OCC3)=O)cno2)ccc(O)c(F)c1 N1(C(c2c(CC)onc2C)=O)CCCC2(NC(c3cn(C4CC4)cn3)=O)CC2C1 Cc1ccc(C=CC(N2CCC(CCC(=O)NCc3cnc(C)o3)C2)=O)o1 C=C(CNC(c1nc[nH]c1C(C)(C)C)=O)CCNC(C1(C)CCCO1)=O c1(NC(c2c(OC)c(F)ccc2)C)ncccc1S(=O)(=O)NCC(C)S(C)(=O)=O O=C1Cc2c(C(=O)NC3CC(NC(C4CCC=CO4)=O)C3)cccc2N1 C1(C(=O)NC(CN(C(C(C=C)C)=O)C)Cc2ccccc2)Cc2nnc(C)n2C1 c1(C(N2CCCC(NC(=O)C=Cc3cncs3)C2)=O)cccn2nccc12 c1(CC)sc(C(N2CCC(C(C)NC(=O)CC(=O)N(C)C)C2)=O)cc1C c1(CC(CN(C)C(C2(c3cccs3)CC2)=O)NC(=O)C=CC2CC2)ccccc1 Cc1ccc(CN2CCCC(N(C)C(c3ccccc3Cl)=O)CC2)c([N+](=O)[O-])c1 C1(C(C)NC2(c3nnnn3C)CC3CC3C2)CCC2(CCOCC2)C1 N(C(=NCc1cc(C)on1)N1CCC(OC)C(C)C1)CC(c1ccccc1)OCC c1(C(N2C(CCNC(C3ON=C(CC)C3)=O)CSCC2)=O)cc2c(s1)CCCC2 C1(C(=O)Nc2cccc(NC(C(C(C)C)F)=O)c2)COc2cc(Cl)ccc2C1 C(=O)(C(O)C1=CCCCC1)NC1C2(CN(C(Cn3nc(C)oc3=O)=O)C2)SCC1 CCCCC(CNC(c1cc(Br)c(Cl)s1)c1nnnn1CC1CCCO1)CC N1(C(C2C(C)C2(F)F)=O)CCCN(C(=O)Cn2ncc3c2CCCC3)CC1C C(=O)(C(CC(=O)N1CCCN(C(=O)CSCCO)CC1C)C(C)=O)OC c1(CNC(C2CC(C)OC2)=O)cc(C(=O)O)ccc1F CC1CN(C(=O)CCCCn2ccnn2)CCC1NC(=O)CC1CCCCC1 c1(C(CC)C)cc(C(=O)N(CCNC(c2cscn2)=O)CCOC)oc1C C1(NC(c2c(CC)cco2)=O)CC2COCC(C1)N2C(c1nnsc1N)=O CC(C)CC(C(=O)NC1CCCCC1NC(=O)CN1CCCOC1=O)C(N)=O c1(C(=O)NC2CN(C(CCCC=C)=O)CC2C=C)cc2c(=O)[nH]ccn2n1 Cn1ncc(C(N2CCC(NC(=O)Cc3ccccc3C(F)(F)F)C2)=O)c1C#N c1(C(=O)NCCC2(OC)CN(C(C(CO)OC)=O)C2)cnnc(C)c1 c1(-c2n(C3CCOC3)ccn2)cnccc1SC1C(Cl)(Cl)C1 CC(=O)CCCC(=O)NC(C)(C)CNC(c1ccnc(Cl)c1N)=O CC(=O)CC(C)(C)C(=O)NC1COCCC1C(=O)NC(C)CN(C)C(C)C N1(C(c2nc(C)sc2)=O)Cc2ccccc2CC1CNC(=O)Cc1ccns1 C1(C(N2CC(C)(NC(=O)C=Cc3cncnc3O)C2)=O)CC2CCCCC2O1 c1(C(N(C2CCCN(C(=O)C(O)Cc3cnc[nH]3)C2)CC)=O)cn2c(n1)SCC2 c1(OC)ccc(C(=O)NCC(c2cc(C(F)(F)F)cc(C(C)C)c2)(C)C)nc1Cl c1(CC)[nH]nc(C(=O)NC(C)C=CC(=O)NC(c2ccccc2)CC)c1C C1(NC(c2n(C)ncc2C2CCC2)=O)CC2CN(c3ncc(F)cn3)CC2C1 c1(OC)ccc(SC)cc1C(N1C(C=O)CCC1C)=O.C(C#N)N(C)C1CC1 c1(OCCC)ccc(C(=O)N(C)CC2(O)CCN(C(=O)CC3CC3)C2)cn1 CC(C)(CNC(C1COCOC1)=O)C(=O)NCC12CC(CCO1)C2 C12(NC(c3c(Cl)cn(C)n3)=O)CCCCC1CN(C(=O)C(C1CCCCC1)O)C2 N1(C(C2ON=C(C)C2C)=O)CCC(CCNC(C2(N(C)C)CC2)=O)C(F)(F)CC1 Cc1cc(F)c(C(=O)NC2CC23CC(NC(c2c(C)nn(C)c2F)=O)C3)cc1F C1(COC(=O)OC(C)(C)C)(NC(N(C(c2nc[nH]n2)(C)C)C)=O)CCC1 CCCCC(CC)CC(=O)NCC(C)NC(=O)C(C)(C)Oc1cc(F)cc(F)c1 C1(CC(N2CCCC(CC(=O)OC)C2)=O)CCC2(CCC2)CO1 CCC(C(=O)NCC(C)(C)NC(c1ccc(Cn2cncn2)cc1)=O)C(C)C N1(CC(N2CCC(N(C(C3CCS3(=O)=O)=O)CC)C2)=O)CC(=O)NC1=O C(=O)(C1CCCn2nccc21)NC1C(NC(CCCN(C)C)=O)CCC1 CC1(C)C(NC(C2CC2C2CC2)=O)C1C(N1CC2(CC2)C1)=O c1ccccc1O.c1(CC(=O)NCC2(F)CC(NC(=O)CS)C2)ccccc1O C1(C(=O)NC2C(CCOCC)C2)N(C(C2CC2C(N)=O)=O)CCC1(C)C C(c1ccncn1)=CC(=O)NCC1OCC(CNC(Cn2c(C)nnn2)=O)C1 N1(C(Cn2c(C)csc2=O)=O)CCC(NC(c2cc(Cl)cs2)=O)C(O)C1 c1(N(CCC)CC)nc(-c2ccccc2)nc(=NCC2CC(C(F)(F)F)CO2)[nH]1 CC1(F)CCN(C(=O)CCn2cc(C3(N4CCCC4)CC3)nn2)C1 C1(CC#C)CN(Cc2cc(C)n(C)n2)C12CCC2 CC1(C)CCCCC1C(N1CCC(CF)(NC(=O)Cc2sc(O)nc2O)C1)=O C1(O)(C(C)NC(=O)COC2CCCCCC2)CCN(C(=O)C(F)(F)C(C)O)CC1 c1(NC(CCC(=C)Cl)=O)c2c(nn1C(C)C)CSC2 Cc1c(Br)noc1C(=O)NC1CCCCC1NC(c1coc(N(C)C)n1)=O Cc1sc(C(=O)NCC2(C(F)F)CCN(C(C3(C)CC=CCC3)=O)C2)c(C)c1C CCC(C)(CC)C1c2n(nnn2)CC(=O)C(=O)C(C)(C)C(C)N1.OC c1(C(=O)NCC(C)CNC(c2cccc[n+]2[O-])=O)c(Cl)nn(C)c1Cl N1(C(c2c(C)cc(F)s2)=O)CCCCC1C1CCCN1CC(N1CCCC1)=O CC1(C)CN(C(c2cocn2)=O)CCC1C(=O)NCC1(C2CC2)CCC1 N1(C(C(C)OCc2ccc(F)cc2)=O)CC(NC(c2ccoc2)=O)C2(CCC2)C1 c1(CC(=O)NCC(C(C)C)N(C)C)ccc(Cl)cc1Br CCCC(C)(O)CC(=O)N1CCN(C(=O)CN2CC(=O)NC2=O)C(COC)C1 Cc1c(C(=O)NC(C)CNC(=O)CCc2ccoc2)[nH]c2c(Cl)cccc12 Cn1nc(C(=O)NC2CCCC2NC(=O)CC2(C)CC2(F)F)cc1Cl N1(CC)CCCC(C(=O)NC(C)CCNC(=O)C(F)=C(C)C2CC2)C1 C1(C(N2CCC(C)(O)C2)=O)CC12CCN(S(=O)(=O)c1nccs1)CC2 N1(C(C2CC(OC(C)(C)C)C2)=O)CCC(CNC(=O)CCC(=O)N(C)C)C1(C)C C1(CC)C(NC(=O)C(C2CCCC2)OC)CCCN1C(c1c[nH]ccc1=O)=O N1(C(CCCOCCOC)=O)CC2(C1)OC1(C)CC2(NC(c2occc2C)=O)C1 N1(C(c2cn(C)nc2)C(=O)NC2(C)CC2)CCC(C)(CO)CC1.n12cc(cn1)C2 C(=O)(C(Cn1cncn1)NC(=O)CC1CNC(=O)O1)N(C)CC1C(C)C1 N1(C(c2cc(C)on2)C(=O)Nc2cccs2)CCN(CC(=O)NCC(F)F)CC1 c1(C(=O)OC)cncn1CNC(C1C(CNC(=O)CC(C)F)C1(C)C)=O c1(OC)ccc(F)c(C(=O)N(C2CC(NC(=O)CCC(C)O)C2)C)n1 C1(n2cc(-c3c(C)cccn3)nn2)COC2(C1)CN(C(c1ns[nH]c1=O)=O)C2 c1(N2CC(C)SCC2)nc(N2CCCC(CCC(F)(F)F)C2)c2c(n1)CSC2 C1(C(=O)NCc2cc(OC)no2)CCC(C)(C)N(C(=O)C(C2CCCCC2)=O)C1 Cc1cc(Cl)cc(C)c1C(=O)NCC(C1CCOC1=O)NC(=O)CC1=NN(C)C1 CCCCC(O)CC(=O)NC(C1CCCN1C(c1cc(C)c(Cl)s1)=O)C c1(C(=O)NC23CC(NC(c4[nH]cc(CC)c4)=O)(C2)C3)c(C(=O)O)n[nH]c1C Cc1ccc(C)c(C(=O)NC2CCC(NC(=O)C3=CCCSC3)CC2)c1 C=CCN=c1[nH]cc(C(N2CC(NC(c3c(OC)ncnc3OC)=O)C2)=O)s1 N1(C(c2[nH]c(=N)sc2)=O)CCC(NC(C2CCCNS2(=O)=O)=O)C12CCCC2 N1(C(COc2ccc(OCC)cc2)=O)CCOCC(NC(=O)CSC2CC2)C1 c1(NC(C2CC(F)CN(C(C3(O)CCCC3)=O)C2)=O)c(Cl)cc(Br)cc1[N+](=O)[O-] c1(C(=O)NCCNC(C2(CC)CCCC2)=O)n[nH]c(C)c1Cl c1(OC)ncnc(C(=O)NCCCN(C(c2cc(CO)cn2C)=O)C(C)C)c1F N1(C(C(CC)C)=O)CC(C)(C)C(NC(=O)CC2CCCN(C)C2)C(C)(C)C1 CC1CCN(C(C2CN(C(C3CC4(CCCO4)C3)=O)CCO2)=O)CC1(C)C n1(CC)cnc2nc(=NCc3cc(Cl)sc3Cl)[nH]c(NCCn3cnnn3)c12 C1(C)(C(N2CC(NC(c3cc(C)n(C4CC4)n3)=O)C(C)C2)=O)CCN(C)C1=O c1(C2(CN(C(c3nn[nH]n3)CN3CCN(C)CC3)C)CCC2)cc(F)ccc1F C1(CNC(c2c(C(C)C)ccs2)=O)CCN(C(c2ccoc2Cl)=O)CCC1(F)F N1(C(C=CCC)=O)CCC(N(C(=O)CCS(=O)(=O)NC)C)C(C)C1 c1(NC)ccc(S(=O)(=O)NC)cc1NC(c1cc(-c2ccco2)[nH]n1)=O S(=O)(=O)(c1ccc(NCC2COC3(CCCCCC3)O2)cc1Br)N1C(C)CCC1 c1(OC)cc(C(N2CC(O)CC2C(=O)Nc2ccc(C(F)F)nc2)=O)cc(F)c1 C1(NC(c2cn(C3CC3)cn2)=O)CCCN(C(c2ncccc2O)=O)C1 c1(C(=O)NCCC(C)CCNC(=O)C=CCO)ccc(Br)cc1Cl C1(CNC(CN2CCC(NC(C3CCC(CC)CC3)=O)C2)=O)CCC(C)(C)CO1 S(=O)(=O)(c1cn(C)cc1C)Nc1cc(OC)c(C(F)(F)F)cc1 S(=O)(=O)(c1ccccc1NC(=O)CCCCC(N)=O)NC(C)(C)C C1(C2CC2)(CNC(CCc2c(C)cccn2)=O)CCN(C(=O)CC2CC2C)C1 c1(CNC(C(SC)SC)=O)cc(C(=O)NCC2CC2(Cl)Cl)n[nH]1 C(C(=O)NCC1(C)CCCN1C(c1cncc(F)c1)=O)(C(C)(C)C)OC C1(NC(CN(C(C2CC3(CC(=O)C3)C2)=O)CC)=O)CCOC12CCOC2 S(=O)(=O)(c1ccc(F)cc1F)N1CCC(CNCc2ccc(OCC)cc2)C1 N1(C(COC(CC)(C)C)=O)CC2CCC1C(C(=O)NCC1CCCCN1C)C2 C(=O)(NNC(=O)c1cn(C(C)(C)C)nn1)NCCc1cn(C)nc1 c1(C(N2CC(C(N)=O)(CNC(c3cc(F)cs3)=O)C2)=O)cccc2oc(=N)[nH]c12 N1(C(=O)NC(c2c(CC)ccc(F)c2)c2nccn2C)CCCC2(C1)CC2(F)F Cc1nn(CCC(=O)NCc2coc3ccc(Cl)cc23)c(C)c1[N+](=O)[O-] C(C(F)(C(=O)NCCC1C=CCC1)C(C)C)NC(C1(C#C)CC(=O)C1)=O c1(N(C)C)ccc(NC(C2C=CC(NC(C3CCS3(=O)=O)=O)C2)=O)cc1 C#CCCCC(=O)NC1CC(NC(=O)C(C(C)O)NC(=O)OC(C)(C)C)C1 Cc1ccsc1C(C(=O)NCCCC1CC1)N(C)CCF C#CC(CC(C)(C)C)NC(C1CCN(C(=O)C2(SC)CC(=O)C2)O1)=O c1(C(=O)NCC(C)NC(=O)C2=CCOC2)ccccc1S(=O)(=O)N1CCOCC1 Cc1ccc(Cl)cc1C(N1CCC2(CC2C(=O)NCCc2ccsc2)C1)=O c1(C(N2CCN(C(C(C)OC)=O)C(C)C2)=O)c(F)ccc(OC)c1F C(=O)(C1=CCCC1C)N1CCC(NC(C=CC=CC)=O)(CO)C1 S(=O)(=O)(c1c[nH]c(C(=O)NCC2CN(C(=O)C(=O)NC3CC3)CC23CC3)c1)NC c1(CN2CC(CNC(c3ccnnc3O)=O)C2)c[nH]c2cc(Cl)ccc12 CCCCC(C)C(C(=O)NC)N1CCC(O)CC1c1ccccc1OC C(=O)(CC1=CCOCC1)N1C(CC(=O)NC(CCCC)(C)C)CCC1 N1(C(C=Cc2c(C)nsc2)=O)CCCCC(NC(=O)C(O)Cn2cncn2)C1 C1(NC(C2CCC(=C)CC2)=O)CC2CC(C1)N(C(c1cc(C#N)c[nH]1)=O)C2 c1(C(=O)NC2CN(C(CCc3ccc(C)o3)=O)CC2(C)C)ccc2ncnn2c1 C1(CC=C)(NC(C2CCN(CC)C2)=O)CCN(C(c2cc(Br)n[nH]2)=O)C1 C1(C)(CNC(CSCCOC)=O)CCCN(C(c2cccc(=O)o2)=O)C1 c1(CCC)onc(C)c1C(N1CC(C(N)=O)(CNC(=O)CC(C)NC(N)=O)C1)=O c1(CNCCc2c(-c3ccc(C)cc3)n[nH]c2)cncc(Br)c1Cl N1(C(C(CCC)N(C)C)=O)CCN(C(C2OCCCO2)=O)C2COCC12 c1(CC(N2CCCN(C(C(CC)n3cccn3)=O)CC2)=O)ccc(F)cc1Cl C(=O)(CC(=O)NC(c1ccc(CNC(C23CCCC2C3)=O)s1)C)NCC#C N1(C(CN(C(CC2(CC)CCC2)=O)CC(C)C)=O)CCC(C2CCC2)C1 N1(C(CCC(N)=O)=O)CCC(F)(F)C(NCc2c(O)cc(O)cc2O)C1 c1(C(=O)NCC(CC=C)NC(=O)C(N2CCSCC2)C)cncc(OC)n1 CCC(C)(C)C(=O)N1CC(NC(C2CC(=O)N(CC(F)(F)F)C2)=O)C(C)C1 O=C(C1CCOc2ccc(Cl)cc21)OCC12COC(CCO1)C2 CC1CN(C(=O)CCc2cnc[nH]2)CC2(CCN(CCOC3CCC3)C2)O1 Cc1cc(C(N2CC(NC(C3(C(C)C)CC3)=O)C3CC23)=O)sc1C c1(C(=O)NCCNC(C(C)Oc2ccc(C)cc2)=O)cc(C#N)[nH]c1C CC1(C)CNC(=O)C1NC(=O)Nc1cccc(OCCC(F)(F)F)n1 CCCC(CO)NC(=O)CCn1cc(C2CC(OC)C2)nn1 C1(C(=O)NCC(C)NC(c2nn(CC)nc2C)=O)CC2CC1C1CC21 C(CCCO)(c1ccccc1)NC(=O)NC(COC)CF C1(NC(C2(C)CC(=C)C2)=O)CCC(CNC(C2CC2C(=O)OC)=O)CC1 S(=O)(=O)(c1cccc(Cl)c1Cl)N1C(CC(=O)Nc2ccc(Br)c(F)c2)CCC1 C1(C(N(CCCCC)CCO)=O)CCC(C)(C)N(C(=O)CC2C(=O)NN=C2C)C1 c1(C(N2CCC(N(C(C(CC)F)=O)CC)C2)=O)cc2ccc(O)nc2s1 C(C)(C(C)C=O)NC(C(COC)N(C)C)=O.C(C(F)(F)F)=CC(=O)N N1(C(c2ccc(N)c(F)n2)=O)CC2CC1CCC2NC(C1CCCC1O)=O CC1CCN(C(c2ccc(Cl)o2)=O)CC1NC(C1CC(CF)C1)=O Cc1ccc(NC(=S)NC2CCCC2C(=O)N(c2ccccc2)C)cc1 C1(OC)(CNC(=O)C2=CC(C)C2)CCN(C(=O)CC(C)c2cccnc2)C1 C1(C(=O)OC)(NCC(=O)C(C(C)C)c2ccccc2)CCCOCC1 c1(OCCC)cccc(C(=O)N(C)CC2CN(C(c3ocnc3C3CC3)=O)C2)c1 c1(C(=O)NC2CCCCN(C(C3(C(CC)=O)CC3)=O)C2)ccc2c(c1)C(C)C(C)O2 N1(C(C(CC)N(C)C)=O)C2CCCC1CC(NC(=O)CCC(C)O)C2 C1(C(=O)NCC(CN(C(CCC#C)=O)C)(C)C)CCOC(c2ccccc2)C1 C1(CN(C(C(C)Cn2cccn2)=O)C)COCCN1C(=O)CS(=O)(=O)N(C)C C1(COCCC(=O)NCC(C)N(C(=O)CCc2ccccc2)C)CCCC2CC12 S(=O)(=O)(c1cc(Cl)ccc1Cl)N1CCC(C)(C(=O)Nc2cncc(C#N)n2)C1 c1(C(N(CCN(C(c2cc(OC)nn2C)=O)C)C)=O)cc2c(ccn2C)s1 N1(C(C2C(C3CN(C(C4(C)CCNC4=O)=O)C3)C2)=O)CC(O)C2(CCCC2)C1 CCCCC(F)C(=O)N1CCCCC(CCC(=O)NC2(C)CC3(CC3)C2)C1 CC(C)(CC(F)F)C(=O)N(C(C1CC2COCCN2C1)=O)CC1(O)CC2CCC1C2 c1(C(=O)NC2(CC=C)CCN(C(c3cc(=O)cc[nH]3)=O)C2)cc(C)ccc1F CC(C)(C(=O)N1CC(=C(F)CNC(=O)CN2CCNC2=O)C1)c1cncnc1 C1(CNC(C2CC23CCOCC3)=O)CCN(C(C2(CCF)CC2)=O)CCC1(F)F C1(CNC(C2CCCS2)=O)CN(C(=O)CCC2CCCCO2)CCO1 C1(C)(C(=O)NC(CCN(C(CCc2cnc(C)o2)=O)C)C)CCCCCCC1 N1(C(CCCCOC)=O)CCN(C(=O)C(c2cc(F)cc(F)c2)C)CC(O)C1 c1(C(N2CC(NC(C(CO)N(C)C)=O)C(O)C2)=O)cnc2c(Cl)cccn12 N1(C(CCc2ccnc(C)n2)=O)CC2=C(C1)CN(C(=O)C=Cc1ccn(C)c1)C2 C12(C(=O)Nc3c(C)nc(Cl)nc3)CCC(NC(C3CCCC(C)C3)=O)(CC1)CC2 N(C(=NCCC(C)=O)NCC1(Cl)CCCC1)C1CCC(SC)C1 C1(CN(C(=O)C(F)=CCCF)C)CCN(C(=O)CC2CNC(=O)C2)CC1 N1(C(C(CCCC#C)C)=O)CCC2(CCN(C(=O)CCOC3CCC3)C2)C1 N1(C(C)C)CCCCC1C(N1CCC(C)(NC(c2cnsc2)=O)C1)=O CN1C(=O)CCCC1C(N1CCC(O)C1C(=O)NC1CC(Cl)(Cl)C1)=O CCCCCCCCNC(=O)C(=O)NC1CN(C(=O)N=CC(C)(C)SC)CC1C N1(C(C2N(CC)CCC2)=O)CCC2(NC(C3CC4(CCC4)C3)=O)CCCC12 N1(C(C(C)OC2CCOC2)=O)CC(C2CN(C(c3ccnn3C(C)(C)C)=O)C2)C1 c1(C(=O)NCCC2(O)CN(C(c3cc[nH]c3)=O)C2)ccc(-c2cscn2)cc1 CCCCC(O)C(=O)N(C1CN(C(C2CC2c2ccccc2N(C)C)=O)C1)C C1(NC(C(C=C)(C)C)=O)CC2(CCC(CNC(C3(COC)C=CCC3)=O)CC2)C1 N1(C(CSC(C)C)=O)CCN(C(=O)CCc2cccc(F)c2)C(CC(F)(F)F)C1 CCC(CC(=O)N1CCC(C)(NC(=O)CS(N)(=O)=O)C1)CC(F)(F)F C(=O)(N=c1nc[nH]s1)C1N(C(C(Cc2ccccc2)NC(C)=O)=O)CC1.C(C)(=O)O c1(C(=O)NC23CCCC2CN(C(c2coc(O)n2)=O)C3)oc2ccccc2c1Cl C1(CNC(CCC#C)=O)CCCCN(C(c2c[nH]c(Br)c2)=O)C1 CCC(C)C(O)C(C)C(=O)NC1CN(C(C2(C)CCC(=O)C2)=O)CC1O C1(NC(C=C(CC)C)=O)CC(C2CCN(C(=O)CCN3CCCC3=O)C2)C1 C1(OC)CC(CCNC(=O)CCNC(=O)CO)N(C(=O)C(F)CC2CCCC2)C1 C(CCCN=c1[nH]c2c(c(=NC(C)CN3CCCCCC3)[nH]1)CCC2)=CC c1(OCC(=O)NC2CCCC(NC(C3C(CC)C3)=O)C2)nn(C)cc1[N+](=O)[O-] C1(CCCCNC(c2ncn(C)c2)=O)CCN(C(C2(C)CCC(=O)N2)=O)CC1 N1(C(C(C)=O)=O)CCC(O)(C(C)NC(=O)C(F)(F)C=Cc2ccccc2)C1 CC1(NC(=O)CCOC2COC2)CCCCC1C(=O)NCC1(F)CCOC1 c1(C(N(CC(C)CNC(=O)CC2CCCO2)C)=O)cc2cccn2c(O)n1 N1(C(C=CC(C)C)=O)CC(F)(F)CC1CCNC(c1n[nH]cc1C(C)(C)C)=O C1(CC)C(C(=O)NCCc2cscn2)CCCN1C(=O)Cc1ccc(F)nc1 C#CCCC(O)C(=O)N1CC2(C1)CN(C(C1CCN(C)C1C)=O)C2 N1(C(c2c(C)snc2)=O)CC(CO)C2(C1)CN(C(c1ccc(N)c(F)n1)=O)C2 C1(C(N(C)Cc2ncnn2C)=O)CCC2CCC1N2C(C1C2CCCC12)=O C1(C(C(C)C)NC(Cn2ncc(CC)c2)=O)CCN(C(C2CSCCS2)=O)CC1 C1(NC(c2c(C)nccn2)=O)CC2(NC(=O)Cc3cnsc3)COC1C2 N1(C(C2N(C(C(C)OC(C)=O)=O)CC=CC2)=O)C2CCC1CC1(CC1)C2 CCC(CC(F)F)C(=O)N1CC2(CCN(C(=O)C(C)Cc3c(C)n[nH]c3C)C2)C1 N(C1CCCc2ccoc21)C(C(C(C)NC(=O)CCC1(C)N=N1)(C)C)=O N1(C(C2(COC)C=CCC2)=O)CC2CCCC(C1)N2C(c1ccsc1Cl)=O C(=O)(C1CCCc2nn[nH]c21)NCC(CCOC)NC(=O)Cc1ccc(F)cc1 N1(C(C(CCO)N(C)C)=O)CC(CNC(c2coc(C(N)=O)c2)=O)CC12CCC2 C12(CC(=O)N(CC(=O)NCc3ccncc3)CC)CCC(CC1)CC2 c1(C(=O)NC2CC(C)(NC(CN3CCC(C)(C)C3)=O)C2)ccc(F)cc1Cl c1(CC(=O)NC2C(NC(CC(C=C)C)=O)CCC2)cccc(S(=O)(=O)CC)c1 N1(C(C(C)CC2CC2)=O)CCC2(CC1)CC(NC(c1cc(Br)cn1C)=O)C2 N1(C(C(CC#C)NC(C2CNC(=O)O2)=O)=O)CCN2C(=O)OCC2C1 c1(NC(C2N(C(C3CN(C)C3)=O)CC(O)C2)=O)cc(C(F)(F)F)c(Br)c(Cl)c1 c1(C(=O)NC2C(NC(c3c(C)n(C)nc3)=O)CC2)c(C#N)cnn1C CC(C)CCCN=c1[nH]c(N(C)CC2(OC(C)C)CCOC2)nc2c1COCC2 C1(CNC(CS(=O)(=O)NC)=O)CCCN(C(=O)CCc2c(C)noc2Cl)CC1 C1(C2N(C(C3C4(CC(OCC)C4)C3)=O)CCC2)CCCCN1C(=O)CCCSC c1(C(=O)NCC2N(C(C3CN(COC)C(=O)C3)=O)CC2)cnc(C2CC2)nc1C c1(OC)ccc2[nH]cc(CN3CCOCC3C(=O)Nc3oncc3C#N)c2c1 C1(F)(CNCCc2nccc(C)n2)CCC2(CC1)CC2 C1(CNC(C2(C)CCCC2O)=O)CC2(CC(NC(c3n[nH]c4c3COC4)=O)C2)C1 C12(CCN(CC(C(C)C)N3CCCCC3)C3CC3)CC(c3ccccc3)(C1)C2F C1(C(N2C(CNC(C(=O)NCCC(N)=O)=O)CC(F)C2)=O)CN2CCC1CC2 Cc1ccc(C(=O)NC2(C)CC(NC(C3CCCN3C3CCOCC3)=O)C2)s1 C1(NC(C(CSCCN(CC)CC)O)=O)CNCC(C)C1 C(=O)(CCCCCCCC1CC1)N1C(CNC(CNC(N)=O)=O)CC1 c1(C(N2CC(CC(C)NC(C3CC3c3cnc[nH]3)=O)C2)=O)cnc2[nH]ncc2c1 CC(CNC(=O)C=CC1CCCN1C)C(F)C(=O)NCC1CCC=CO1 C1(C(=O)NCc2nc(C)c(C)[nH]2)CC2(CCC2)CN1C(=O)CC1CCC=CCC1 N1(C(C2(C=C)CC2)=O)CCN(C(C2CCCN2C=O)=O)C2(CCC2)C1 CC(CN1CCOCC1)N=c1cccc(S(=O)(=O)N2CCOCC(N(C)C)C2)[nH]1 CP(C)(=O)C(CC(=O)N1CC2(CC(NC(c3ccnnc3O)=O)C2)C1)C(F)(F)F C12(CNC(CCC)=O)CC(CN1C(C1(COC)CC1(F)F)=O)C2 c1(C(=O)NC2CCN(C(CCCCCC#C)=O)C(C)C2)n[nH]c2c1CN(C)CC2 C1(NC(c2c(C#C)c[nH]n2)=O)CCCN(C(c2coc(Br)n2)=O)C1C N1(Cc2cccc(SC)c2)CC2(CCC(C(=O)Nc3ccc(Br)c(Br)c3)O2)C1 N1(C(C(CCOCC(=O)NCCO)NCCCN=[N+]=[N-])=O)C2CCC1COC2 CC1(C)CCC(C(N2CCC(c3cc[nH]n3)C2)=O)(NC(C2COCC2CO)=O)C1 N1(C(c2cccc(CNC(c3nn(CC)nc3C)=O)n2)=O)CCC(N=[N+]=[N-])C1 c1(CC(=O)NC(CC(C)NC(c2c(C)occ2)=O)C)ccccc1Cl C(C(C(=O)NOCC(=O)Nc1ccc(=N)[nH]c1)C(C)C)NC(C)=O C1(c2c(C)n(C)nc2)C(NC(N2CCOCC2CNC(N)=O)=O)CCC(=O)N1C n1(CC)nc(C(N2CCCC2(C(=O)N(C)Cc2cnn(C)c2)CC)=O)cc1C c1(NC(C)=O)cc(C(=O)NC2CC2C(N2CCCC2CO)=O)ccc1C(=O)O C1(OC)CN(C)C(C)(C(N2CCC(C)(CNC(=O)Cc3ccc(C)s3)C2)=O)C1 n1(C(C)C)ncc(C(=O)NC2(C(=O)NCc3cnn(CCN(C)C)c3)CC2C)n1 c1(CC2NC(=O)N(Cc3c(C)ncs3)C2=O)cnn2c1C(=O)N(C)CC2 C1(C(C(=O)NCC)N(CC)Cc2cccc(Br)c2)C2CCCCCC12 C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCN(C(c2cccc(=O)o2)=O)C1 C1(C(=O)NCCOCCCNC(C(C)O)=O)COC2(CCC2)C1 c1(C(=O)NC(C(=O)NCC(CC)CC)(C)CO)ccn2ccccc12 Cc1nnccc1C(=O)NCCCC1CCCN1CC(C)COC1CCCOC1 c1(C(=O)NC2C(CNC(CC(C)c3cnn(C)c3)=O)CC2)ncccc1Cl CC1=CCC(C(=O)NC(c2ccnn2C)C(=O)NC2CCC(F)CC2)CC1 C(=O)(C#CC1CCCCC1)N1CCC(C(N(CC(F)(F)F)CC)=O)CC1 c1(C(C(=O)N(CCC=C)CCO)NC(COCC#C)=O)cnn(C)c1 N1(C(COCC#C)=O)CCC(OC)CC1.C(=O)(C1CCO1)NCCCOC c1(C(N2C(CNC(CN(CCCCCC)C)=O)CC2)=O)cccc(N)c1 CC(C)(C)C#CC(=O)N1CCC(OCCCNC(c2cnc(F)c(F)c2)=O)CC1 c1(C(C(=O)NCCN(C(c2c(C)cn(C)c2)=O)C2CC2)C)ccc([N+](=O)[O-])cc1 c1(NC(C2CCN(C(c3cnc(C)[nH]3)=O)C2)=O)ccc(C)c(C)c1C N1(C(C(CCC)O)=O)C2CCC1CC(CNC(=O)C(C)(C1CC1)NC(C)=O)C2 c1(C(N(C2CCN(Cc3c(CC)noc3)CC2)C)=O)occ2c1CCC2 N1(C(C=C(CC)CC)=O)CCC(CNC(c2cnn3c2CCC3)=O)C(F)(F)CC1 C1(NC(c2ccc3c(c2)COC3)=O)CC2CN(C(=O)C3CC3)CC2C1 C(=O)(C(C)S(N)(=O)=O)NCC1C(NC(c2c(C)cn(C(C)C)c2)=O)CC1 C1(CCNC(C(N(C(=O)CCC2CCCO2)C)C2CC2)=O)CCCCC1 C(=O)(C1=C(C)OCC1)N1CC(O)(CNC(CSCC)=O)C1.c12ccccc1S2 N1(CC(C)C)CCCC(C(=O)NCC2CN(C(=O)C(C)CSC(F)(F)F)C2)C1 c1(-c2cccc(CN3CC4C(CO)(C4)C3)c2)cc(O)c(F)cc1F.c1(S)ccccc1 N1(C(CC=C(C)C)=O)CCCC2(CCC(NC(c3cscc3F)=O)C2)C1 c1(C(N2C3C(N(C)C(C4CSCCS4)=O)CC(C3)C2)=O)cccc2c1CCCC2 c1(-c2scc(C3C(=O)N3C3(C)CC3)n2)cccc(Br)c1.C1(CCC#N)CCCC1 S(=O)(=O)(CCC(=O)N1CC(CNC(=O)C=Cc2cncn2C)CC1(C)C)NC C(=O)(CC(C)(C)C#N)NC1C(C(N2C(C(=O)NC)CC(F)C2)=O)COC1 c1(C(=O)NCCN=c2[nH]ccc(I)c2F)ccc2c(c1)C(O)CCC2 c1(C(=O)NC(N)=O)ccc(NC2CNC(=O)C2)c(F)c1.C123CC(C1)(C2)NC(=O)N3 C1(NC(C(CC)NC(N)=O)=O)CN(C(=O)Cn2cnc([N+](=O)[O-])c2)CC2(CC2)C1 Cc1nccc(C(=O)NCc2ccccc2CN(C)C(C2CC23CC(O)C3)=O)n1 C1(NC(C2(CC#C)CCCCO2)=O)CC2CCC1N2C(c1cc(F)cnc1O)=O c1(C(N2CC(OC)C(NC(=O)Cc3cnns3)C2)=O)cnc(N)c(CO)c1 CCC(CC(=O)N1CCCC1(C(=O)NCCc1nncn1C)CC)C1CC1 c1(OC)ccnc(C(=O)NC(CNC(=O)CC(C)OC)C2CCC2)c1C c1(C(=O)NC)cn(C)cc1C(N1CC2(CC2C(=O)OC)C1)=O c1(OC)cc(C(=O)NCC2=CCN(C(c3cc(Cl)on3)=O)CC2)ccc1[N+](=O)[O-] C(=O)(CC(C(F)(F)F)NC(=O)CN(C1CCC1)C)N(C)CC1(SC)CCC1 N1(C(C2(CC=C)CC=CC2)=O)CC(CNC(=O)CCC2CCCCC2)C(C)C1 N1(C(c2c(CC)ccc(F)c2)=O)CC2(CCC(NC(C34CC(OC)C3C4)=O)CC2)C1 C12(CC(=O)NCC3CC(OCC)C3)CNC(=O)C(C1)C2 N1(C(CC(C)C(F)(F)F)=O)CCc2sc(CNC(c3ccncc3)=O)nc2C1 c1(N2CCC(C)C2)ccccc1CNC(=O)N(C1CC1C(F)(F)F)C N1(C(CCCCCNC(C(C)(C)CC#N)=O)=O)CCOCC2(CCC2)C1 N1(C(CC=CCNC(c2c(CC)noc2)=O)=O)CC(CO)OCC1C c1(CC(=O)OC)cc(C(=O)NC2C(CNC(=O)OC(C)(C)C)CCC2)n[nH]1.C1CC1 c1(C(=O)NC(C2CCCN2C(c2ncccc2Cl)=O)C(N)=O)cc[nH]c2nccc1-2 C1(N(C(CN(C(=O)OC)C)=O)C)CCCN(C(C2CC=CCC2C)=O)CC1 c1(NCCCOc2cccc(C)c2)ccc(S(=O)(=O)NC2CC(C)(C)C2)c(Cl)c1 CCCC(C)(C)CC(=O)NC1CCC(N(C(=O)C=CSCc2ccco2)C)CC1 Cc1nc(C)n(CCCCC(=O)NC(C)C(C)(O)c2ccccc2)n1 N(C1CCOc2c(Br)cccc21)C(C1CCCC(O)(c2nccn2C)C1)C C1(C)(c2cn(CC(=O)NCC)nn2)CCCN1C(C1COC(C)(C)C1)=O c1(C(N2C(C(C)NC(C(n3ncc(C)c3)C)=O)CCC2)=O)ccc(C#N)cc1 C12(CNC(C3(CCC=C)CC3)=O)CC1CN(C(C1COCCN1CC)=O)C2 C12(CNC(C(C(CC)C)O)=O)CCC(CC1)N(C(c1cn3ccnc3s1)=O)C2 O=C(C1OCCc2ccccc21)N1CCC(C2CCCN2CCC2CCC2)CC1 C(CCC(C)C)N(C(C1(NC(COCCC#C)=O)CC1)=O)C1CC1 c1(OC)nc(N2CC=C(CCNC(C3(C(C)C)CC3)=O)CC2)nc(C)c1F C(C(CNC(c1coc(C2CCCC2)n1)=O)CO)NC(c1cncnc1)=O N1(C(C2N(C(C3CC(CC)(CC)C3)=O)CC(C)CC2)=O)CCC2(CCCO2)C1 C(=O)(C1CCc2cccnc21)N1CCC(NC(CC2(C)OCCO2)=O)(CO)CC1 C1(CN(CCN(C(C2CCN(C(C)=O)C2)=O)C)C)CCCCN1CC(F)F CC1(C)CCC1(COC1CC1)OC(c1nc(-c2ccc(Br)cc2)sn1)=O C12(NC(c3cc(C)nn3C)=O)CCCC1N(C(c1cnn[nH]1)=O)CCC2 c1(C(=O)NC(C(=O)NC(CCOC)C)C2(C)CC2)ccc(C#N)c(C)n1 C(CO)(CCCNC(c1csc(C2CC2)n1)=O)NC(c1cn(C(C)C)nn1)=O C1(C(=O)OC)N(C(=O)CCN2CCCCC2=O)CC12CCOCC2 C1(CC)CN(C(C2(C)CCCC2C)=O)CCC1NC(C1(C#N)CC2CC2C1)=O Cc1cc(C(=O)N(C2CN(C(=O)C(C)c3cncs3)C2)C)cc(C)n1 N1(CCNC(c2n(CC)nnc2)=O)CCCN(C(=O)Cc2ccc(O)nc2)CC1 C1(CNC(C2=C(C)CCC2)=O)CC2(CO1)CN(C(C1COCCN1C)=O)C2 c1(CNC(C(COCC)NC(C2CCOCC2)=O)=O)cnc(OC)nc1 c1(C(N2CCC(C)C(CC(=O)NOCC3(C)CCC3)C2)=O)cc2ccncc2[nH]1 C(=O)(C(F)(F)C(C)(C)O)NC(CC)CN(C)C(C1CC(C(C)C)=NO1)=O C1(C(C)C)N(C(C2CCCN(C)C2)=O)CC12CCN(C(=O)CC1(C)CC1)CC2 C1(NC(CCCCNC(c2nc(N(C)C)oc2)=O)=O)CC(CO)C12CCC2 C1(CNC(CC2(C)CC2)=O)CC2CCC1N(C(C1COCCO1)=O)C2 CC1(C)CN(C(C23CC2CCN3C(c2cc3ncccc3[nH]2)=O)=O)CCC1O CC(C)C(CC(=O)NC(C1CCN(C(c2cnnn2C2CC2)=O)C1)C)C(C)C Cc1cc(C(=O)NC2CCCN(C(C3CCCC(C)(C)C3)=O)CC2)ncc1F CC1CC1(F)C(=O)N(CCNC(=O)Cn1cnnc1)C1CC1 c1(C(=O)NCC2CCC(CNC(C(COC)C)=O)CC2)cc(C)cc(OC)c1O C1(C(=O)N)CC2CC2CC1C.c1(CC)ccc(C(N2CCC(CCO)(C)C2)=O)nc1 c1(C(=O)NC(C2N(C(c3cc(OC)ns3)=O)CCC2)C)cccc2nc(O)[nH]c12 C1(NC(C(CC)=CC)=O)CN(C(c2cc(Br)sc2C)=O)CC1OC c1(CN2C(C(=O)Nc3nnc(C4CC4)o3)CC(O)C2)c(O)ccc(F)c1F C(=O)(CCCCCF)NC1C(CNC(C23CC(C)(C2)C3)=O)CCCC1 Cc1cc(C(=O)NC23CCC(C(=O)NC4CCCCC4)(CC2)C3)cc(O)c1 c1(C(N2C(C)(CNC(CC(CC)OC)=O)CCC2)=O)cnc2[nH]ncc2c1 C(C)(C)(CCCO)NC(C(C1CN(C(C2CCC2(F)F)=O)C1)OC)=O C1(CNC(=O)Cc2cncnc2O)CCCC2CN(C(=O)C=C3CCCC3)CC12 C12(C(=O)NC(C(C)SC)C)COCC1CN(C(c1cccc(F)c1O)=O)C2 CC1(CNC(c2cc(Cl)c(Br)s2)=O)CCCN1C(c1cc(C#N)c[nH]1)=O C1(CNC(C2CCC(C)(C)C2)=O)CC2CCC1N(C(=O)CS(C)(=O)=O)C2 C#CCC(CC(F)F)C(=O)NC(c1nocc1C(=O)NC1CCC2(CC2)C1)C Cc1cccc(C=CC(=O)NCCN(C(c2cn3ccnc3s2)=O)CC2CC2)c1 N1(C(c2cnc(CC)[nH]2)=O)CC2CCC(C1)C(NC(c1cnc(CC)o1)=O)C2 CC1(C)C(NC(c2nnc(O)o2)=O)CC1CNC(c1coc(OC(F)F)n1)=O c1(N(CCC)C)ccnc(C(=O)NC2CN(C(C3C=CCC3)=O)CC2C)c1 CCCC(C)(C)C(=O)N1CC2(CCN2C(C2(C)CCN(C)C2=O)=O)C1 N1(C(c2n(CC)ncn2)=O)CC(CNC(c2ccsc2OC)=O)CC1C Cc1cccc(Br)c1NC(C1CC(NCc2ccc(N3CCCCC3)cc2)C1)=O C1(NC(c2cc(COC)no2)=O)CCCC(NC(C2(n3cccn3)CC2)=O)CC1 CCCC(C)(O)CC(=O)NC1CCCCN(C(C2C3CCC2(C)C3(C)C)=O)C1 Cc1ccc2c(c1C)OCCC2NC(C1COC1)C c1(N2CC3C(CNC(=O)COC4CCCC4)C3C2)nc2cc(F)ccc2o1 CCC(CNC(c1cccnc1N1CCCCC1)=O)(CC)NC(=O)C(O)COC C1(C)(NC(c2c(C)nco2)=O)CCN(C(=O)CC2CCCCC2C)C1 N1(c2n(CCC=C)c(-c3cocn3)nn2)CCC2(CC1)OCC1CC21 N1(C(C(C(CC)C)O)=O)CCc2ccccc2C1CNC(c1ccon1)=O c1(C(C)C)cccc(C(=O)NC(C2CCN(C(c3ccoc3Cl)=O)CC2)C)c1 CCC(Cc1cn(CCF)nn1)C(=O)OC.C12CCN(CC1)CC1CC1CC(=O)N2 C=CCC(C)(C)CC(=O)NC1CCCCN(C(c2cc(C(C)(C)C)n(C)n2)=O)C1 Cc1nn(CC(=O)NC(CCF)C(=O)N2CCC(CCO)C2)c(=O)o1 C1(NC(CNC(=O)Cc2cscn2)=O)CCCN(C(=O)C(c2cccnc2)O)C1 N1(C(Cc2c(C)n[nH]c2)=O)CCC2CCN(C(c3occ4c3CCCC4)=O)CC12 C(=O)(CCCCCCc1ccccc1)N(CCC(C)NC(c1cnco1)=O)C Cc1ccc(F)c(OCC(=O)NCC2(O)CCN(C(c3ccc(C#N)s3)=O)C2)c1 c1(CC(=O)NCCCN(CCC)C(C2CC3COCC3C2)=O)cc(C)cc(F)c1 CCC(C)C(CC(=O)N1CC2CC(F)CC2C1)NC(=O)C(C)(C)n1ccnn1 Cc1ccsc1CC(=O)NCC(C)(C)CC1CN(C(=O)CCC2CCCOC2)C1 C(=O)(C(CC(C)C)C(C)C)NCC1C(NC(Cn2c(=O)ccc(C)c2)=O)CCC1 C(=O)(C1CCCc2c[nH]nc21)NCc1nc(CNC(C2OCC(C)(C)C2)=O)sc1 c1(NC(N(CC(N)=O)C)=O)cccc(S(=O)(=O)NC2CC3CCC2O3)c1 CC(C)CC(C)C(=O)NC(C)(CO)C(=O)N(C)CCc1ccccn1 CC1(C)C#CC(=O)NC1.C1(C(=O)NC2CCCN(CCO)C2)CC(=O)CCO1 C1(CNC(CCC(C)SC)=O)CN(C(c2nc(C3CC3)c(C)s2)=O)CC12CCC2 C(=O)(C(O)CCC(C)C)NC1C(NC(c2c(C)csc2)=O)CCCCC1 C1(NC(C2C(CC)C2)=O)CCN(C(c2cc(C(F)(F)F)n(C)n2)=O)CC(C)(C)C1 CCC(C)(C#N)C(=O)NCC1CCN(C(=O)CCN(CC(F)(F)F)C)CC1 N1(C(C=CC(CC)C)=O)CCC(C(N2CC(N=[N+]=[N-])C2)=O)(CC)C1 C1(CC)(NC(c2cc(Cl)ccn2)=O)CCCN(C(C2(SC)CC2)=O)C1 C(CCC)(C(=O)NC(C1(CNC(=O)C=CCN(C)C)CC1)C)=CCC C1(OC)CN(C(c2c[nH]c(C#N)c2)=O)CC1NC(C1(C)C=CCC1)=O C=C=C(C)CC(=O)NC1CC(CNC(c2ccn(-c3cccs3)n2)=O)C1 c1(NCC2N(C(C3(C)C(C)CCC3)=O)CCCC2)cc(=O)n(C)cn1 N1(C(C(COCC)(C)C)=O)CCC2CC2(C(=O)NCc2ncnn2CC)CC1 N1(C(CC=C)=O)CC(C2CN(C(C3COC(=O)O3)=O)C2)C1 S(=O)(=O)(c1cn(NC)nc1C)N1CC2N(C(C)=O)C(CC2)C1.c1ccc(F)cc1 N1(C(C(COC)CC(C)C)=O)C2CCCC1CN(C(c1cn[nH]c1)=O)CC2 C(c1ccc([N+](=O)[O-])cc1)=C(C)C(=O)NC(C(C)C)c1nc[nH]n1 c1(C(=O)NCC2CN(C(c3c(C)coc3)=O)C(C)C2)cnc(O)c2cncn12 c1(C(=O)NCC(C)(C2CC2)NC(CC(C)SC)=O)cnn(CC2CCCC2)c1C S(=O)(=O)(c1ccc(NC2C3CC4CC(C3)CC2C4)c(C#N)c1)NCCC(C)SC S(=O)(=O)(c1ccc(C)c(C)c1)NCC(=O)NCC(C(C)C)NC(C1CCCC1)=O C(=O)(C(C)(C)C(C)(C)C)NCC1CCC(C(=O)NCCOC(C)=O)C1 CCC(C)(C)C(C)CC(=O)N1CC(NC(=O)CSc2cnn(C)c2)C2(CCC2)C1 C12(C(N(C3CCN(C(=O)C4=C(Cl)CC4)CC3)CC#C)=O)COCC1C2(F)F c1(C(=O)NCC(CNC(=O)CCn2cccn2)O)ccnc2ccncc12 Cc1ccc(CNC(N2CCC(C(c3ccncc3)O)C2)=O)cc1C C1(C)(CNC(CSC)=O)CCCN(C(c2ccc(C(F)(F)F)cc2N)=O)C1 N1(C(CC(=O)N(CCNC(C(c2cccs2)OC)=O)C)C)CCCCC1=O C1(CNC(C2(C)CCC(C)C2)=O)C2CCCC1N(C(c1csc(=N)[nH]1)=O)C2 C1(NC(CCOC)=O)CCC2CCN(C(c3cc(OC)ccc3C3CC3)=O)C12 c1(C(=O)NC(C2CCCC2)CNC(c2c(C)cn(C)n2)=O)cc(F)c(F)cc1F C1(OC)CC(NC(=O)Cn2cc(CO)nn2)CN(C(=O)CC2CCCCN2C)C1 C1(C(=O)NC2(CCCC(=O)NC(COC)C3CC3)CCC2)CC1C1CCCC1 CCCC(O)C(=O)NCCN(C)C(c1nnsc1C)=O C1(CN(C(C2(C#C)CC2)=O)C2CC2)CCN(C(C2CCOC2C)=O)CC1 N1(CC(N2CC(N(C(CC(C)F)=O)C)C(O)C2)=O)CCC(=O)NC1=O CN=c1ccc([N+](=O)[O-])c[nH]1.CCCCCC(=O)N1CCCC(C2CCCCO2)C1 CC1CCN(C(c2cc(C3CC3)on2)=O)CC1CNC(=O)CC(O)C1CCCC1 C(CCCCCNC(C12CC1CN(C(=O)CNC(N)=O)C2)=O)N(C)C CCCCC(=O)N1CCCC1C(C)(C)CNC(=O)CSc1nncs1 C1(C(N2CC(C(C)NC(=O)CNC(c3ccoc3)=O)C2)=O)CCCOCC1 C1(C#N)(C(=O)NC(C2CCCCC2)CNC(CN(c2cnccn2)C)=O)CCCO1 c1(CC(=O)NCC2CCCC2NC(c2nncs2)=O)cnn2ccccc12 C1(CNC(C(C(C)C)CO)=O)CCN(C(=O)Cc2cc[nH]n2)CCC1(F)F c1(-c2n(-c3ccc(OC)c(OC)c3)nc(C3CCC3)n2)cc(Br)c(F)cc1Cl S(=O)(=O)(c1ccc(NCc2cncc(F)c2)c(Cl)c1)N1CCCCC(SC)C1 n1(CC(=O)NCC(c2cccc(C)c2)NC(C2C=CCC2)=O)nc(C)c(Cl)c1C N1(C(CCC)=O)CCCCC1C(N1CC(NC(=O)Cn2nnnc2C(C)C)C1)=O Cn1c(=O)oc2c(C(=O)N(C3CCN(C(=O)COCP(C)(C)=O)C3)CC)cccc12 CN1CCC(C)(C(=O)NCCOC2CCN(C(c3ccc(N)cc3Cl)=O)C2)CC1 CCCCC(CNC(=O)CC(c1ccccc1F)C)NC(c1cc(CC)on1)=O c1(C(C(=O)NC(CC(C)NC(C2C(=C)CC2)=O)C)OC)ccc(C)cc1 N1(C(c2cc(OC)no2)=O)CCCC(NC(c2cc(C)nc(C)n2)=O)C1C C12(NC(c3c(CC)nc[nH]3)=O)CCC(CC1)N(C(=O)C(C)N(C)C)C2 c1(N(CC(CN(C)C(C2CSCCS2)=O)O)C)nc(Cl)ncc1C(N)=O N1(C(CN(CC(C)C)C(C2CC(F)(F)CS2)=O)=O)CCCOC(C2CC2)C1 c1(SC)cc(C)c(C(=O)NC2(CNC(=O)Cc3ccc(O)cn3)CCCC2)o1 c1(SC)ccc(-c2nc(C(O)C(F)(F)F)n(CC(C)CO)n2)nc1 c1(NCCC(C)(C)NC(C2C(CC)OCC2)=O)nc(C)nc2sc3c(c12)CCC3 CP(C)(=O)c1cccc(C(=O)NCC=CCNC(C2CCN3CCCC3C2)=O)c1 Cc1nc(CC(C)C)c(C(=O)NC(C2CN(C(=O)CC3CCCO3)C2)C)s1 C=C(Cl)C(C)(C)C(=O)N(CCCCCCNC(=O)C(C)(C(C)C)NC(C)=O)C Cc1cc(Cl)cc(C(=O)NCCN(C(C2(C)CC2C(F)(F)F)=O)C(C)C)c1O C1(CC(N2C(C(C)NC(C=C(C)Cl)=O)CCC2)=O)CCCC(C)(C)O1 CC(C)CC(C(=O)NCC1CCN(C(=O)C(c2cccs2)C)C1)NC(N)=O N1(C(=O)OC(C)(C)C)CC2CN(C3CCCCCC3)CC(C1)C2(F)F c1(NC(N2CCN(C(c3ccc(CCC)s3)=O)CC2)=O)c(C)ccnc1Cl N1(C(C(CC)C(F)(F)F)=O)CC2CCN(C(C3CC4(CCCC4)C3)=O)CC2C1 CC(=NO)C1CC(C(=O)NCC2CCCN2C(c2c[nH]cc(Cl)c2=O)=O)C1(C)C C(=O)(C(=O)C(C)(C)C)NC1CC(N(C(=O)CC=Cc2ccccc2)C)C1 C=CC(CCC)CC(=O)NCCCC(CCC)NC(c1c[nH]nc1C)=O C1(NC(C2(NC(c3n(C)c(S)nn3)=O)CCSC2)=O)CC2CCCC2C1 c1(C(c2n(CC(C)C)c(N3CCC(C(N)=O)CC3)nn2)C)nnc2n1CCCC2 c1(C(C)NC(N(C2CCN(C)CC2)CC(C)OC)=O)ccccc1CN(C)C c1(C(C(=O)NCC(C)N(C(C2CC2C#N)=O)CC)(C)C)ccc([N+](=O)[O-])cc1 c1(C(N2CC(CN(C(C(COC)C)=O)C)OCC2)=O)ccc(N)c2ncccc12 C(=O)(CCCCCCS(N)(=O)=O)NC1CCN(C(Cc2cc(C)sc2)=O)CC1F CC(C)C(CCN(C)C(C1CC1C(F)F)=O)NC(C1CC(C#N)C1)=O N1(C(c2c(SCC)ncs2)=O)CC2CC(C)N(C(=O)C(CC)CC)C2C1 c1(CNC(C(C(CC)C)O)=O)cnn2c1CN(C(=O)CCCN(C)C)CC2 CC1(C)CN(C(c2c(O)cc(O)cc2O)=O)CCC1NC(C1(C)COC1)=O c1(OC)ccc([N+](=O)[O-])c(N2CCCC(NC(N)=O)C2)c1F c1(C(C)OC(c2c(C)nc(C3CCCC3)s2)=O)ccc(Br)c(F)c1 N1(C(Cc2c(C)noc2C)=O)CCC(O)C(NC(=O)COc2cc(Cl)ccn2)C1 Cc1cc(-c2nc(COC(C)(C)C)n(C(C)COCc3cccs3)n2)c(C)o1 C1(C(N(C2CCN(C(=O)CN3CC=CC3)CC2)CCC)=O)CCC(C)(C)CC1 CC(CNC(=O)CC1CC2(CC2)CO1)CC(=O)NOC(c1ccccc1)C C1(CC)CCN(C(c2cc(C(C)=O)c[nH]2)=O)C1C(=O)N(CCN=[N+]=[N-])CC C1(N(C)C(=O)C2CC2)COCCN(C(=O)C=CC(=O)NC(=O)CN(C)C)C1 N(C(=NCCOC)N1CCC2(CC1)C(F)(F)C2(F)F)CC1(CC#C)CCOC1 C(=O)(CC1OCc2ncccc21)NC1(C)CC(NC(C2CCCO2)=O)C1 C1(CNC(C2(OC)CCSC2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C12CC2 c1(CC(C)NC(C(=O)N(CC(C)O)CCN(C)C)=O)ccc(O)c(F)c1 C1(C(=O)NC2CC(c3cn(CCOCC)nn3)C2)COCCN1CC(F)F C1(C)(CC(=O)NCCN(CCCCCC)C(=O)C(CO)NC(N)=O)CCCCC1 N1(C(CCSC)=O)CC=C(CCNC(=O)CSCc2nnc3ccccn23)CC1 c1(CNC(C(CC(C)C)NC(C)=O)=O)cccc([N+](=O)[O-])c1C C12CN(CC13CCC3)C2.c1(SC(C)(C)C)cc(C)c(C#N)[nH]1.C1(=O)CSCCN1 CCCC(C(=O)NCc1cccnc1)N1CC(O)(C(=O)OC(C)(C)C)C1 C1(C#N)(CC)CCN(C(=O)C(F)C(C)CNC(C2CC(N=[N+]=[N-])C2)=O)CC1 Cc1cc(CCC(N2CCCC2CCC(=O)NCc2cn(C)nn2)=O)n[nH]1 C1(NC(c2ccc(N)cn2)=O)CC2CC1CN(C(C1CCCCNC1=O)=O)C2 C=CC(C)(CC)C(=O)NCC12CC1CN(C(=O)CC(C)(C)C#N)C2 c1(CC)nccc(=NC(=O)C2CC(F)CN(Cc3ccc(C(F)(F)F)cc3)C2)[nH]1 N#CC1(C(N2CCOC(CNC(=O)COCCO)C2)=O)CC2C=CC1C2 c1(C(N(CC(CNC(CCC2C(C)=NNC2=O)=O)C)C)=O)cc(O)ccc1C N1(C(c2cncc(C=C)c2)=O)CCN(C(c2onc(C)c2C)=O)CC(C)C1 N1(OC)CCC(N(C)Cc2c(-c3c(OC)nccc3)cnn2C)C(C)C1 c1(C(=O)NCCOCCC(=O)NCC(COCC)C)cc(C#N)cn1C C1(C)(NC(C(OC)OC)=O)CCCN(C(C2(C(=O)NC3CC3)CC2)=O)C1 c1(CC)noc(CC)c1CC(=O)NCCCCN(C(=O)C(c1ccc(Cl)s1)C)C C(=O)(CC1=CCN(C(c2cc(F)ccc2O)=O)CC1)N(CC(N)=O)CC(N)=O CC(C)C(CCC(=O)NC1COCC1CO)NC(c1cc(O)nn1C)=O C=CCC(C)(C)C(=O)N1CC2(CC(NC(C3CCNC3=O)=O)C2)C1 C(C(CC(F)(F)F)NC(c1cc(C)nn1C1CC1)=O)NC(C1N(CC)CCC1)=O N1(C(C2(C#N)CCC2)=O)CCC2(COC(CNC(C3CCC(=O)N3)=O)C2)C1 C12(C(=O)NCC3(NC(C(C)n4ccnn4)=O)CCCC3)CCC(N=[N+]=[N-])C1C2 c1(C(N2CCN(C3CCCC3)C(c3ccccc3)C2)C(=O)NC)cccc(Cl)c1C C1(O)CCCCN(C)C1=O.c1(C(N(CC)CC2CN3CCC2C3)=O)sc(O)nc1C C(=O)(CCCCCCC(=O)N1CC(NC(c2cn(C)nc2Br)=O)C1)OC N1(C(C2N(C(C)=O)CCC2)=O)CC2(CCCN(C(=O)COCCOCCO)C2)C1 c1(C(=O)NCC2C(NC(=O)CCF)CCC2)cnn2cccc2c1 c1(C(=O)NCCCCC(C)NC(=O)CC(F)(F)Cl)c[nH]c2ccccc2c1=O c1(CC(=O)NCC2CCCN(C(c3cc(C)nnc3)=O)C2)nc2cnccc2[nH]1 c1(CC)nc(N2CCC(CF)(NC(=O)CC(C)C(C)C)C2)[nH]c(=N)n1 C12(C(N3C(C(=O)NC)CC3)=O)CCN(C(=O)C(C)N(C)C)CCC1C2 C(=O)(C(CC(C)C)C(N)=O)N(CCN(C(c1c(OC)cccc1O)=O)C)C c1(CC)oc2ccccc2c1C(N1CC(NC(=O)CC2CCCCO2)C(C)C1)=O c1(C(=O)NC(C(CO)NC(COCCC)=O)C)ccc2nc(Cl)nn2c1 c1(OC)ncnc(C(=O)NC2CCC(C)N(C(C3CCC4(CCC4)C3)=O)C2)c1F C1(NC(C(COC)OC)=O)CCCC2CN(C(C3C=C(C)CS3)=O)CC12 C1(CCNC(C2CC(C#C)(O)C2)=O)CCCN(C(=O)C(CC)=CC)CC1 c1(C(=O)NC2CC3C(NC(=O)CCc4cccs4)C3C2)cc2cccnn2c1 N1(C(CSCCC#N)=O)C2CCCC1CN(C(=O)CC1CCCCC1F)C2 c1(CC(=O)N(C2CCC2)CC#C)cccc(OC(F)F)c1 N1(C(c2ccc(C)cc2F)=O)CCC2C(CCN2Cc2c(F)ccc(Br)c2F)C1 C1(N(C(C2CCCN2C(N)=O)=O)CC)CCN(C(=O)CP(C)(C)=O)CC1 CC(N=c1ccn(C2CCCCO2)[nH]1)c1nc(C(F)(F)F)cs1 N1(C(c2coc(Cn3cccn3)c2)=O)CC2=C(C1)CN(C(c1cccnc1)=O)C2 c1(C(N2CC(O)CC(NC(C(n3cc(Cl)cn3)C)=O)C2)=O)c2c(nn1C)CCC2 C1(CCNC(c2c(OC)c[nH]n2)=O)CN(C(=O)COC2CCCC2)CC(C)O1 C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(COC(=O)Cc2cn(CC(=O)O)nn2)C1 C1(CC)C(NC(=O)C(C)Oc2ccccc2F)CCN1C(c1cc(Cl)n(C)n1)=O C1(CNC(C(C)(C)OC)=O)CN(C(c2cc(C)cc(C)c2C)=O)C2(CCC2)C1 N1(C(C2CN(C(N(C)C)=O)C2)=O)CCN(C(C2CCC=CCC2)=O)CC(O)C1 c1(C(N2CCC(CC(N3CCOCC3CO)=O)C2)=O)cccc(O)c1 c1(C(=O)OCC)ccc(CO)c(CNC(=O)OC(C)(C)C)n1.C1(=O)C(C)(CF)O1 c1(C(N2CCC(C(N3CCC(CCOC)C3)=O)(C(C)C)C2)=O)cc(C)nnc1O C1(CN(C(c2nncs2)=O)CC)CCN(C(=O)CCN2CCCC2)C1 C1(C(=O)NC(C2(CNC(C3(c4ccno4)CC3)=O)CC2)C)CCCN(C)C1 CC1CCC=C1C(=O)NCC(C1CCC1)NC(c1ccc(Cn2ccnc2)o1)=O c1(OCC#C)ccc(CN(CCCO)C(c2cccc(-n3cnnn3)c2)=O)cc1 N1(C(C=C(CCC)CCC)=O)CCC2(NC(c3cc(O)cc(Cl)c3)=O)CC2C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)(C)C(O)CC)ccn2cnnc2c1 C1(CNC(C(CCSC)O)=O)N(C(c2cncc(O)c2Cl)=O)CCCC1(C)C Cc1[nH]nc(C(=O)NCC2CC3(CC(NC(C4(C)CCC4)=O)C3)C2)c1[N+](=O)[O-] N1(CCC)CCCC(C(=O)NC(C)CC(C)NC(=O)Cc2cc(C3CC3)on2)C1 C(=O)(C1CCCc2nnn(C)c21)NC1CCCN(C(c2c(C)csc2)=O)C1C C1(CS(=O)(=O)NC2CCC3C2C3(F)F)CCC2(CCCOC2)O1 C(N=c1cc(C(=O)NOCC(F)F)nc[nH]1)c1cn(CC(C)C)nn1 c1(C(=O)NCC2CC(OC)CN2C(=O)C=Cc2ccccc2)c(C)cnnc1O C1(C(N(CCOC)C(C)C2CC2)=O)CCN(C(c2cccc(CO)c2)=O)CC1C CC(C)C(C(=O)NC(C1(CNC(=O)CC2CCCC23CC3)CCCC1)C)N(C)C N#Cc1ccc(C(=O)N(C2CCCN(C(C3CNC(=O)N3)=O)C2)CCO)s1 c1(NC(c2ncc(Cl)cc2Cl)=O)cccc2[nH]c(C(=O)NC(COCC)C)cc12 c1(NC(c2cc(-c3ccc(-n4cccn4)cc3)cs2)=O)ncc(C(F)(F)F)cn1 C1(NC(c2ccc(SC)s2)=O)CC2CC(C1)CN(C(c1cc[nH]c(=N)c1)=O)C2 c1(C(=O)NCC2N(C(c3c(F)ncc(OC)c3)=O)CC2)cc(F)c(F)c(O)c1F N(C(=NCc1ccccc1C(F)(F)F)NCC1CC2C(=O)OC12)C(C)C c1(C(=O)NCC2(C)N(C(CC=CC=C)=O)CCC2)ccc2cc(Br)ccc2n1 c1(C(=O)NC2C3CC(O)C2N(C(C2CCC(F)CC2)=O)C3)cccc2nn[nH]c12 n1(CC(=O)N(C)CC2N(C(C(C=C)C)=O)CCC2)nc(C)oc1=O C1(C(N2C(CCC)CCC2)=O)CSCCN1C(=O)CCC1CC(C)C1 C(=O)(CCCCC(F)F)NCC1C(CNC(c2nccc(OC)c2)=O)C1 C1(CNC(CCSCC)=O)CC(C(F)(F)F)CN1C(C1CC12CC2)=O CN=c1[nH]cc(C(N2CCCC2C(C)(C)C(=O)NCCC(O)C(=O)OC)=O)s1 c1(C(N2CCC3CN(CC)C3C2)C(=O)NCC=C)cc(F)cc(F)c1Br c1(C(=O)NC2CC3CN(C(CC)=O)C(C2)C3)cc2c(Br)cccc2cn1 c12ncc(C)c(n1)N(C(c1nccnc1C)=O)C2.C1(SC)CNC1 c1(OC)c(C)cccc1C.N1(C(c2cc(C(F)F)on2)C(=O)NC)CCN(C=O)CC1 C(C(F)(F)C(=O)NCC1(C(C)NC(C2CCCSC2)=O)CC1)OC CC1CC(C#N)(C(=O)NCC2(CNC(=O)CCCn3cncn3)CC23CCC3)C1 c1(C(C#C)OC(C(Cc2ccccc2)C(=O)OC)=O)ccc(F)cc1 N1(C(C(C(=C)C)(C)C)=O)CC(CNC(=O)CCOC2CCOCC2)C2(CCC2)C1 C1(N(C(=O)C(C)n2cncn2)CC)CCCN(C(=O)C(F)(F)CC)C1 N1(C(C(CC)(C)CC)=O)CCC(C(=O)Nc2ccc(SC)cc2)=C(F)C1 N1(C(C2C(OCC)C2)=O)CCCC2(C1)CN(C(C1CCc3n[nH]c(C)c3C1)=O)C2 n1(CC)nnc(C(N2CCOC(C(=O)NCCC3CCCCC3)C2)=O)c1C C(C(=O)NCCNC(c1cccnc1NC)=O)(C(C)C)OCC C#CCC(C(=O)NCC1(SC)CC1)NC(C1CC(C2CC2)C1)=O N1(C(c2c(C)nc(F)cc2)=O)CCN(C(=O)Cc2cncnc2)CC(C)(F)C1 C(=O)(C(C)(F)C(=O)NCCNC(C1(n2cccn2)CCC1)=O)OC N1(C(C2(CC)CN(C(c3ccccc3Cl)=O)C2)=O)C2CCC1CC(=O)NC2 c1(C(N2CCC(CCNC(C3=CC(C)(C)C3)=O)C2)=O)cc(O)ccc1[N+](=O)[O-] c1(NC(C2CC(OC)CN2C(C2CCCSC2C)=O)=O)ccc(C)c(F)c1 c1(OC)ccc2nc(C(F)(F)F)[nH]c(=NCC3(O)CCSCC3)c2c1.N(C)C(C)C C1(CCNC(CCOC)=O)CN(C(=O)C(c2ccccc2F)F)CCCO1 C12(CNC(CCCSC)=O)CC(NC(=O)CCn3cnccc3=O)(CO1)C2 CN=c1[nH]c(C(=O)NC2CCCCC2NC(C2CC2C)=O)cs1 C(CN=c1[nH]c(=NCC2SCCS2)[nH]c2c1CSC2)C1(COC)CC1 C1(C(=O)NCCn2cc(CSC3CCCCC3)nn2)(OC)CCCOC1 c1(CC(N2CCN(CC3CCCN(C(COC)=O)C3)CC2)=O)c(F)cccc1Cl C(=O)(C(C(C)(C)O)NC(N)=O)NCC(C)NC(=O)C(C)C(F)F c1(CNC(C2(CCCC)CCC2)=O)nc(CNC(=O)C(O)c2ccsc2)cs1 c1(C2(NC(c3cccc(C(=O)NCCO)c3F)=O)CC2)ccc2ccccc2c1 N1(C(C=CC)=O)CCC(C(N2CCCC(NC(=O)C3CC3)C2)=O)C1(C)C C1(CNC(C(C)SC)=O)(OCCNC(c2ccn(C(C)C)c2C)=O)CCOCC1 c1(CNC(c2c(C)nc[nH]2)c2nnnn2C)ccnc(Cl)c1Cl c1(N2CCCC(=C)C2)ccc(S(=O)(=O)NCc2c(F)ccc(C)c2Cl)c(Cl)c1 Cc1cc(C(N2CC(O)(CNC(C3COCC(C)(C)O3)=O)C2)=O)cc(C)c1C c1(C(N2CCC(C(N3CC(CCC)C(O)C3)=O)CC2)=O)cc(C)ccc1Cl C(CN=c1cc(C)c(S(=O)(=O)NC)c[nH]1)C1CCN(CC)C1 c1(C(=O)NC(CC(C)NC(=O)C(F)(F)c2cncs2)C)cccc(N)n1 c1(SC)cc(F)ccc1C(=O)NC(C)CCCNC(C1(C)CCCS1)=O N1(C(c2c(OC)c(C)ncn2)=O)CCN(C(=O)C(C)(C)CSC)CCC1C Cc1cccc2[nH]c(=NCC(C(C)(C)C)NC(=O)C(c3ccccc3)O)oc12 C1(N)(C(=O)NC(C(=O)OC)(C)C2CCCC2)CC12CCC2 CC1(C)C=C(C(=O)NCCCN(C(C23CC(CCO2)C3)=O)C2CC2)C1 c1(CC)[nH]ccc1C(=O)N(CCC(C)NC(=O)CSc1nncn1C(C)(C)C)C C123CC4CC1C2C4NC3=O.c1(Cc2onc(COC)n2)cc(F)ccc1OC C1(N(C(C(N2CCC(C)CC2)=O)=O)C)CCCN(C(=O)CCP(C)(C)=O)CC1 c1(SCC(=O)NCC2CCN2C(=O)CC(O)C2CCCC2)c(Cl)cccc1Cl CN=C(NCC1CCN(S(C)(=O)=O)C1)N(C)CCc1ccccc1Cl N1(C(c2c(OC)nsc2)=O)CCN(C(=O)CC2CCN(C)CC2)C(C2CCC2)C1 N1(C(C(CCC)C)=O)CCN(C(C2CC(N(C)C)C2)=O)CC1CCO N1(C(c2c(CNC(C=C(C)C)=O)cnn2C)=O)CC(O)CCC1C CCC(C)(C)C(C)CC(=O)NCC1CC2CC2N1C(c1nccc2ccsc12)=O C(CN=c1cccc(S(=O)(=O)NC2CC(CO)C2)[nH]1)c1nnc(C)n1C N1(N2C(C)C2=O)CCC(=C(F)F)CC1.N1(CC(c2cnn(C)c2)=O)CCCCC1 C1(CNC(CC(C)(C)SC)=O)CC(F)(F)CN1C(=O)C=Cc1nc(C)cs1 N1(C(C(C2CCOCC2)C)=O)C2CCC1CC(NC(=O)CCOC1CC1)C2 c1(C(=O)NCCc2nn(C)c(Cl)c2)ccc(C(F)F)cc1-c1cccn1C c1(CC(=O)N(C(CNC(C(CC)n2ccnc2)=O)C)CC)cccc(C(=O)NC)c1 C1(NC(COC)CNC(=O)OC(C)(C)C)COCCN1CC CC1OC(C)CC1CC(=O)N(CCN(C)C(C1(N(C)C)CCCC1)=O)C(C)CCC c1(CC(=O)NC(CNC(C2C(C(=O)NCC#C)C2)=O)(C)C)nc2ccccc2[nH]1 N1(C(C(C)OCCC=C)=O)CCOCC(CNC(c2cc(C(C)C)on2)=O)C1 c1(N2CCCC(CSC)C2)cc(S(=O)(=O)N2CCSC2C(C)C)ccc1C#N c1(CCC(=O)N(CC(=O)O)CC2CCC2)ccncn1 CC1(C)COCCC1CC(=O)NCCC(O)CNC(=O)CC1(CO)CC1 CC1CCC(CNC(c2cccc(N)c2)=O)CN1C(c1ocnc1C1CC1)=O C1(C(N2CC(C)(NC(C3CCCCC3C(F)(F)F)=O)C2)=O)CC(C2CC2)=NO1 C1(Nc2ncnc(C)c2F)CCC2CN(C(=O)C=Cc3cn[nH]c3)CC12 C1(CC=C)(NC(C2CC(n3cnnc3)C2)=O)CCN(C(C2CCS2(=O)=O)=O)C1 N1(C(c2ccn(C3CC3)n2)C(=O)NC(CC)C)CCC(C)C2CCCCC12 c1(SC)sccc1C(=O)NCCOC(C)(C)CNC(C1OCC1(C)C)=O CCC(C(=O)OC)C(=O)N1CC(C)(C(=O)N(C)Cc2ccncc2C)C1 c1(NC)ccc(F)cc1NC(C1CSC(C)C1)=O C(C(O)C(=O)N(CCCNC(c1cc(-c2ccccc2)[nH]n1)=O)C)N(C)C C=CC1(C(=O)NCC2(C)CNC(=O)O2)CCN(C(=O)Cc2ccc[nH]2)C1 N1(C(C(CC)O)=O)CC2(CCN(C(c3c(C)nn(CC)c3C)=O)C2)C1 N1(C(C(C)=C(C)C)=O)CC(NC(c2cnc(C(C)(C)CF)o2)=O)C2(CC2)C1 c1(C(=O)NC2(CNC(=O)CC3CCCCCC3)CC2)cc(Cl)c(Cl)c(Cl)c1O C1(NC(CNC(CC(C)C)=O)=O)CC12CC(NC(=O)C(c1ccc(Cl)cc1)C)C2 c1(C(N2CCC(C)(CNC(C3(OC)CC3)=O)C2)=O)ccc(S(N)(=O)=O)o1 N(C1CN(C(=O)CN2CCCCCC2)CCc2ccccc21)C(C)=O C1(NC(CCNC(=O)NC)=O)CCC2(CC1)CCN(C(=O)Cc1ccc(C)s1)C2 c1(SCC(=O)NC2(C)CCCN(C(c3cnc(Cl)s3)=O)C2)ncnc2[nH]cnc12 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(c2cc(O)cs2)=O)CC(C)C1 N1(C(CCC=C)=O)C2CCC(C2)C1CNC(c1csnc1Br)=O C1(C(N2CCC(C)(NC(c3c(C)nn[nH]3)=O)C2)=O)CCCCC12CCC2 c1(CN2CC(NCc3cc(C)c(O)c(C)c3)C(C)C2)cc([N+](=O)[O-])cc(Br)c1O c1(C(=O)NCC2C(NC(c3c(C)snc3)=O)CCC2)ncc(F)cn1 c1(OC)cccc(C=CC(N2CCC(C)(CNC(C3CC=CCO3)=O)CC2)=O)c1 c1(CCC(=O)NC2CC(N3CSCCSC3)C2)ccc(SC(F)(F)F)cc1 N1(CC(N2CC(NC(C(C3CC3)OCC)=O)C(C)C2)=O)CCN(CC)C(=O)C1=O C(=O)(C(C)(C)C(C)NC(=O)CCCC1CCCC1)N(CCCC=C)CC N1(C(C2C(=O)NCCC2)=O)CCCC(S(=O)(=O)N2CCCCC2)C1 N1(C(C(F)=CCC)=O)CCC(C)C1C(=O)NCCNC(C)=O C12(CNC(=O)C3=NOCC3)CCC(CC1)N(C(c1cc3cccnc3s1)=O)C2 CC(=O)CCC(=O)NC(C)C=CC(=O)NCCCCCOC(C)C c1(C(=O)NC(CC)C)cn(C)nc1Nc1ccc(C(C)CC)cc1 C(CNC(C1(SC)CCC1)=O)(CCNC(C1C=CCC1)=O)OC C(c1ccncn1)=CC(=O)NC(C1CCN(C(c2c(CC)c[nH]n2)=O)C1)C N1(Cc2c(Br)cc(OCC)c(O)c2)CCC(C)(O)C(O)C1 C1(NC(COCC#C)=O)CCN(C(=O)CNC(=O)C(CC)CC)CC1F c1(C(=O)OCCn2c(C)nc(C)n2)nc(C)n2c1CCN(C)C2.C(C)(C)(C)S C(c1ccc([N+](=O)[O-])s1)=CC(N1CCCCC(CNC(C2N=C(C)SC2)=O)C1)=O N1(C(C2CCC(C)(CC)O2)=O)CCN(C(=O)Cc2ccc(Cl)nc2)CC(O)C1 C12(NC(C3(C)CCCN(C(C4CNC(=O)C4)=O)C3)=O)CCC(C#N)(CC1)CC2 Cc1noc(C)c1CCC(=O)NCC1CN(C(=O)C=CC(C)C)CCO1 C1(CNC(C2(N(C(CCCCC)=O)C)CC2)=O)CCCN(C)CC1 C1(CNC(C(C)(C)C2CC2)=O)CC2(CCN(C(C3(C#N)CC3(C)C)=O)C2)CO1 N1(C(c2cc(C)nc(C)c2)=O)CC2CC(C1)N(C(=O)Cn1cnnc1O)C2 C1(F)(CNC(=O)CSCC2CCCO2)CN(C(C2(C3CC3)CC2)=O)C1 C1(CC)CN(C(C2CCN(C)C2)=O)CC1C(=O)NC1CCC(O)CC1 Cc1ccc(-c2cc(C(N3CC=CC3CNC(=O)C3=CCSC3)=O)n[nH]2)cc1 c1(CNC(=NCC)NCCCCC(C)C)cc(Br)c(OC)cc1F CC1CCn2c(C(N3CC(c4ccccc4)C(C)(C)C3)=O)cnc2C1 n1(CC)ncc(C(=O)NC2CCC(NC(=O)C=Cc3ccc[nH]3)CC2)c1C CCCC(C)(C)C(=O)NCC(CC(=O)NC(C)CCN(CC)CC)C1CCC1 CC1CCN(C(=O)CCCn2cncn2)C(C(=O)NCC2CC(O)C23CCC3)C1 C1(CNC(C(C)SCC)=O)CCCCN1C(C1(C)CCCS1)=O Brc1ccc(-c2ccc(CNC(c3nnnn3C3CCC3)c3cnoc3)o2)cc1 C1(C(N(CCCC)C(C)CC)=O)CCCCC1NC(c1ncccc1O)=O C#Cc1ccc(C(N2CCN(c3ccc(C(C)C)cc3)CC2)C(=O)NC2CC2)cc1 C1(CC)CCC(C)N(C(c2nc(CNC(c3cnc(C)c(C)c3)=O)oc2C)=O)C1 CC1CN(C(C2CC2C(F)(F)F)=O)CCC1CNC(c1c[nH]ccc1=N)=O c1(C(N(CCCCNC(C2=C(C)OCCS2)=O)C)=O)ccc2cccc(O)c2c1 C(=O)(C(CCC)C1CCCO1)N1CC(CC2(C(C)N)CCCO2)C1 c1(C(=O)NCC2N(c3nnc(CC(C)C)s3)CCC2)cccc2[nH]ncc12 C(=O)(C1CCCc2nn[nH]c21)NCCCN(C(=O)CCOC1CC1)CCO c1(OC)cc(C(N2CC3CN(C(c4conc4C)=O)CC3C2)=O)c(OC)cc1Cl C(=O)(CC(C)C(C)(C)C)N1CC2(C(NC(c3n(CC#C)ccc3)=O)CC2)C1 c1(C(=O)NC2CCCC(CN(C(C3(SC)CC3)=O)C)C2)ccc2c(c1)NCCC2 C12(CNC(c3c(C)snn3)=O)CC(NC(C3CCCS3)=O)(CCO1)C2 CS(=O)(=O)c1cc(NC(c2cc(C#N)c(N)cc2O)=O)cc(C(F)(F)F)c1 C1(NC(CNS(N)(=O)=O)=O)COC2(C1)CN(CCCO)C2 c1(CN2CC(C(=O)NCc3ccc(SC)cc3)OCC2)ccc(F)nc1N(C)C c1(NC(C)=O)cc(F)ccc1C(=O)Nc1cccc(NC(=O)C(F)(F)CO)c1 N1(C(c2ccc(SC)cc2)=O)CC2CC(n3cc(CC(N)C(=O)O)nn3)CC2C1 C#CC1CCC(C(N2CCCCC(CNC(C3CC(C)(C)C3)=O)C2)=O)CC1 N(C1CCCn2ccnc21)c1c(C)c(N(C)Cc2nc(C3CC3)n[nH]2)ncn1 c1(C(=O)NC2C(NC(C3(C)C(C)CCC3)=O)COCC2)coc2ccccc12 C(CC)(C(=O)NC(C1CC=CCC1)C(=O)NCCC(=C)C)=CCCC CC(CC(F)(F)F)C(=O)NCC1CCCCC1NC(c1cnn(C)c1Cl)=O C(c1cscn1)=C1CN(C(C2(COC(C)(C)C)C(C(=O)OCC)C2)=O)C1 Cc1c(C(=O)NC2(CNC(C3CCN3S(C)(=O)=O)=O)CCC2)nn(C)c1Br C1(CNC(C=CCOC)=O)CN(C)CCN1C(C1CCC(C)(O)CC1)=O c1(NC(=O)CC2CCCN2C(c2ncc(Br)cc2F)=O)ccc(Br)c([N+](=O)[O-])c1 C#Cc1ccc(CC(N2CC=CC(NC(=O)COc3ccc(Cl)cn3)C2)=O)cc1 c1(OC)ccc(C(N2CCCCC2CNC(=O)C=CCO)=O)cc1F N1(C(C2CC=C(C)CC2)=O)CCC2CCN(C(c3cc4ncccc4[nH]3)=O)CC12 N1(C(C(C)N2CCC2)=O)CC2CC1CCC2NC(C1C2CCC1(C)C2(C)C)=O c1(N(C)C)ncc(CN2CCC2C(=O)Nc2nc(C(C)(C)C)cs2)cn1 c1(CC(=O)NC(c2ccccc2F)CNC(CC)=O)ncn(C)c1C CCC(C)C(O)C(C)C(=O)NC(C)CNC(=O)CC(C)c1cnn(C)c1 C#CCC(CC(=O)NC(C1CCCC1)CO)NC(=O)COCCC C1(NC(C2(CC=C)CC2)=O)CN(C(C2CCCC2n2cccc2)=O)CC2CC12 CC(C)CCC(=O)NCC(=O)NC(C(C)NC(c1cccnc1Br)=O)C(C)C N1(C(C2C(CC)CC2)=O)CC2CCN(C(c3ccc(=O)n(CCF)n3)=O)CC2C1 C1(NC(C2N(C(C)C)CCC2)=O)CN(C(c2nc(C(N)=O)cs2)=O)CC1F CN=c1[nH]cc(C(=O)NCC2CCC2NC(C2C3COCC23)=O)s1 O=C1C2COC3(CCC3)CN2C(=O)N1Cc1ccc2ccccc2n1 C1(NC(C2CCCC3(CC3)C2)=O)CCN(C(C)(C)C)CC1O.c12nc(cs1)CNC2 N1(C(c2csc(C)c2C)=O)CCC(C2CCCC23OCCO3)C1 C1(CC)CN(C)C(=O)CN1C(=O)C(F)C(C)CNC(C1CCN(C)C1)=O N1(C(C(=O)NCCC)C2CCCO2)CCN(C)CC1.N12CCCC1COC(=O)C2 N1(c2nc(N3CCCC(C)(F)C3)c3c(n2)[nH]cc3)CCOC2(CCSC2)CC1 c1(NCc2c(C)nn(C)c2Cl)cc(F)c(F)c(F)c1F.N12CC3CC(C1)N3C2=O c1(NCc2nc(NC(c3cc(OC)n(C)n3)=O)sc2)cc(C)c(Br)cn1 N1(C(c2cc(C(C)C)on2)=O)CCC2(CC(NC(=O)C(F)=C3CCCC3)CO2)C1 C(=O)(CCCCNC(=O)CC1(CC)CCC1)NCC=C=C S(=O)(=O)(c1ccc(Cl)s1)N(C(CCCl)C(=O)O)C(=O)CCCc1ccccc1 C1(NC(C2=C(C)CCCC2)=O)CCCCC12CCCN(c1cc(O)ncn1)C2 c1(C(=O)NCCNC(c2cnc(=NC)[nH]c2)=O)cc(C)cc(OC)c1C c1(C(N(C2CCN(C(=O)CC3C=CCCC3)CC2)C)=O)csc(=NC2CC2)[nH]1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCOCC(C)(CNC(=O)C2=CCCSC2)C1 C1(C(N2CC(N(C)C)C(O)C2)=O)CC2CCC(C1)N2C(=O)CCn1ccnc1 Cc1c(NC(=O)CNC(=O)C2=CC(C)C2)cnn1C1CC1 CC1=C(C(=O)NCc2ccc(CNC(C3CCCC3CN(C)C)=O)cc2)CCC1 c1(N(CCC)C)cc(Br)ccc1S(=O)(=O)NCC(C)C1(CO)CC1 N1(C(c2cccc(C3CC3(F)F)c2)=O)CCCN(C(=O)CC2CCCSC2)CC1 C1(NC(C2(CNC(Cc3cn(C)nc3C(F)(F)F)=O)CC2)=O)CC1C1(C)COC1 C(=O)(C(C)(C)C(C)C)NC(C(C)C)CNC(=O)C(C)Oc1ccc(Cl)cc1 c1(C(=O)NC2CCCCC2CNC(C23CCCC2C3)=O)cc(O)nc(O)n1 C1(CCC)CCCN1C(C1C(NC(=O)COCCCN(C)C)C1)=O Cc1cc[nH]c1C(=O)NC(c1cccnc1)C(=O)NCCC1(CO)CC1 C(=O)(C(C)(O)CC(C)C)NC1CC(NC(Cc2c(C)nn(C)c2C)=O)C(O)C1 N1(C(=O)Cc2ccc(F)c(Br)c2)CC2(CCC(NCc3ccc(Cl)c(O)c3)C2)C1 c1(CC(N2C(Cn3cc(C(C)(C)O)nn3)C(C)(C)C2)=O)ncn2c1CCCC2 C(C(C)C)(C(C)(C)O)NC(CC1(OC)CN(C(C2(C(C)=O)CC2)=O)C1)=O C1(C(=O)NC(CNC(C(C(C)C)NC(C)=O)=O)(C)CO)CN2CCCN1CC2 N1(C(C2C(C)(C)NC(=O)C2)=O)CC2(COC(CNC(C3(O)CCSCC3)=O)C2)C1 c1(C(=O)NC2(C)CC(NC(c3ncccn3)=O)C2)cc2cc(Br)ccc2cn1 c1(C(N2CC(NC(CCc3c(C)n(C)nc3)=O)C2)=O)ccc2c(c1)C(=O)CCO2 N1(C(Cc2ccc(C)cc2)=O)CCC(C2CN(C(C3CN(C)CCO3)=O)C2)CC1 Cn1cnc(C=CC(=O)NCc2nc(CNC(=O)CC3CC4CCC3C4)cs2)c1 C#CC1CCCC(NC(=O)CC2CCCCN(C(C3(COC)COC3)=O)C2)C1 C1(CC(N2CC(C)(CO)C2)=O)C2CCCC2N1C(=O)Cc1ncccc1F C1(C(=O)NCc2c(C(=O)NC(C)C(N)=O)cccn2)CC2CCC(C1)C2 CC1CCCC1CC(N1CC(O)(CCNC(C2CC2(C)C(F)F)=O)C1)=O Cc1coc(C)c1C=CC(=O)NCC1(F)CCCN(C(C2CCC(=O)C2)=O)C1 N1(C(c2ccc(C)cn2)=O)CC2CCCC2C1C(N1CC2C(C1)C2(C)C)=O C(=O)(C1CCOc2c(F)cccc21)N(CCCNC(c1cc(F)n(C)n1)=O)CC c1(OC)ccc(C(=O)N(C2CN(C(=O)C(F)CC3CCC3)CC2F)C)cn1 c1(C(=O)NC2CC(CO)N(C(C3CSCCS3)=O)C2)cnc2[nH]nc(O)c2c1 c1(C(=O)NCCCC(C)NC(=O)CCc2cccn2C)noc2ncccc12 c1(CC(=O)OC)ccc(OC)c(NS(=O)(=O)CC(C2CCOC2)OC(C)=O)c1 C(=O)(C(C)CC(F)(F)F)NC12CC(NC(c3cc(OC)no3)=O)(C1)C2 C1(C(=O)NCCn2nnc(C)n2)CN(C(C2CN(C)C(=O)N2)=O)CC1N(C)C C1(NC(=O)CN2CC3CC3C2)CC(N=c2[nH]nc(-c3ccccc3)s2)C1 N1(C(C(=O)NC(C)C)C)Cc2cc(Br)ccc2CC1C C1(NC(CCNC(C)=O)=O)CN(C(C2CCCC23CC3)=O)C2CCCCC12 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CCOC)NC(=O)CCc1nncn1C c1(C(N2C(C(=O)NCC(=O)NCC(F)(F)F)CC(OC)C2)=O)ccc(F)c(Cl)c1F c1(OC)c(C(=O)NC2CC(NC(c3cncnc3C)=O)C2)cccc1Br N1(C(CCS(=O)(=O)NC)=O)CC(NC(c2nnc(S)n2C)=O)C2(CCOCC2)C1 c1(OC)ccc(S(=O)(=O)N2CC(Cc3cccc(C)c3F)C2)cn1 c1(C(=O)NCC(C2CCC2)NC(C(C=CC)O)=O)ccc(C2CCC2)nc1 Cc1cccc(C(N2CCC(NC(=O)CCc3cnc[nH]3)CC2C2CC2)=O)c1N CCC(C)CCCCC(=O)NC(C)CCC(=O)N(CC(F)Cl)C c1(OC)ccc(Cl)c(C(=O)NCC2CC2NC(c2cnn(C)c2C(C)C)=O)n1 C1(NCC2CCOCC2)CC2(C1)CC(O)C2.C1(c2n(CCO)nnn2)(N)CC2(CC2)C1 c1(N2CCCC(NC(C(CCC)Nc3nccs3)=O)CC2)ncc2ccn(C)c2n1 C1(C(N(CC#C)C)=O)C(O)CCN1C(=O)C(O)CN(C)C c1(C(=O)NCCN(C(C2CC2C(N)=O)=O)CC)cc2c(nc1O)CCSC2 C(CC(C)C(=O)N(CCCNC(=O)Cn1nc(C(F)F)cc1C(F)F)C)=CC C1(NC(Cc2ccc(OC)nc2)=O)CC(O)CN(C(c2sc(C)c(C)c2C)=O)C1 Cc1cccc(C(=O)NCC2N(C(=O)C3=C(Cl)CCC3)CCC2(C)C)c1F N1(C(C)C)C(=O)COCC1C(=O)NCCOCCNC(=O)C(c1ccc(Cl)s1)C C1(COC)CCN(C(=O)C=CC(C)NC(=O)CN2CSCC2=O)C1(C)C N1(N(C)C)CCC(CC2(C)CCCN(CCCN3CCCC3)C2)C(C)(C)C1 CC1(C)CC(NC(=O)Cc2csc(=N)[nH]2)CN(C(=O)Cn2nc(O)ccc2=O)C1 N1(C(c2c(-c3c(OCOC)ccc(C)c3)csc2)=O)Cc2ccc(Br)cc2C1 N1(C(c2ncc(CC)[nH]2)=O)CCN(C(C2CC2c2ccc(Br)cc2)=O)CC12CC2 N1(C(C2C(C3C(C)C3)C2)=O)CCC(C2CCCN(C(=O)C=Cc3cccs3)C2)C1 Cc1ccc(CCC(N2CCN(C(c3cc(Cl)cnn3)=O)C3CC23)=O)c(C)c1 C1(OC)(CNC(=O)CC(F)(F)F)CCN(C(=O)CCc2nc(C(C)OC)no2)C1 C1(C(N(CCCC(=O)NCC(C)CC2CC2)C)=O)CCS(=O)CC1 c1(NC(=O)NC(CC)C(=O)NC(c2cccnc2)C(C)C)ccccc1C N1(C(CCOC(CC(C)C)C)=O)CC(CNC(c2scnc2Cl)=O)C(O)C1 c12ccc3cnc(cc3c1)NC2=O.CC1(C(=O)O)CCSC1 c1(C(N(C(CNC(COCCC)=O)C2CC2)C)=O)n[nH]c2cc(C)ccc12 c1(C(=O)NCC2(CNC(COCC=C)=O)CC2(F)F)ccc2c(=O)ccoc2c1 c1(-c2cc(OC)nnc2OC)ccc2cc(C(=O)Nc3nc(Br)cs3)[nH]c2c1 C(C)(C)(CCC(=O)NC1CCC2CC1CO2)NC(CCN(C)CCO)=O c1(C(N(C2CC3(C2)CC(O)C3)C)=O)ccc(-c2ccncc2)nc1O N1(C(c2snc(C)c2N)=O)CCCC2(CCC2NC(C2CCCN2N=O)=O)C1 C(c1ccc(F)c(Cl)c1)=CC(=O)NC1C(NC(c2c(C)ccc(Cl)c2)=O)CC1 CCCCCC(CCCCC)CC(=O)NCCNc1cnn(C(C)(C)C)c1N N1(C(CS(C)(=O)=O)=O)CCC(CO)C(NC(=O)C(O)Cc2ccccc2Cl)C1 C1(C)(CNC(CCCNC(C)=O)=O)CCN(C(C2OCCC2(C)C)=O)C1 Cc1cc([N+](=O)[O-])c(C)cc1C(N1CCC(CC(=O)Nc2ccc(F)c(Br)c2)C1)=O C#CCC(C)(CNC(=O)C(C)(C)C1CCN(C(C2CCCC(=O)C2)=O)C1)CO C=CCC(C)(C)C(=O)NCC1(F)CCC(NC(C2(C(C)C)CC2)=O)C1 C1(NC(c2c(C)[nH]cc2)=O)CC2(C1)CC(C(N1CCC13CCCC3)=O)C2 CC(C)(CNC(C1CCC2(CCC2)O1)=O)CC(=O)NCC1CCCOC1 c1(C(COC(=O)CCc2nc[nH]n2)NC(=O)OC(C)(C)C)ccccc1 c1(OC)ccc(CNC(=O)CN2CCN(C(=O)Cn3ccccc3=O)CC2)c(C)c1 N1(C(Cc2nc(C)oc2)=O)CCC2CC12C(=O)NCc1cn(C)cn1 c1(C(N2CCN(C(CN3C(=O)CSC3)=O)C3C2C3)=O)cc2n(c(=O)c1)CCS2 c1(C(N2CC(O)(C(C(=O)NC(CC(C)C)(C)C)F)C2)=O)coc2ccccc12 C(=O)(C(C)(C)C(C)(F)F)NC1C(O)CCN(C(CC(=C=C)C)=O)C1 c1(OC)cccc(=NC(=O)CCC2CCCN2C(=O)CC2COCCO2)[nH]1 c1(C(N2CCC(CC(=O)NCCc3c(C)cccc3)C2)=O)ccc(Cl)c(O)c1 CCC(C)C(=O)C(=O)N1CCCC(CC(=O)NCC(O)C(CC)CC)CC1 c1(CC)cnc(C(N2CC(NC(=O)C=C3CCC3)C3CC23)=O)cn1 C1(NC(CCOCC#C)=O)CN(C(=O)CCCC2CCCO2)C(C)(C)C1 C1(C(=O)NCCC(C)SC)(CC)CCCN1C(C1COCOC1)=O N1(C(CSCC#C)=O)CCC2(CCC(NC(=O)C3=CCCC3)C2)CC1 C1(C(=O)NC2CCC(CNC(=O)CSC3CC3)C2)CCCCCCC1 c1(C(N2C3CCN(C(C=CC=CCC)=O)CC3C2)=O)ccc2c(n1)CCC(C)C2 N1(C(=O)NC)CCC2(CC(C(=O)NCC(N3CCCC3C(=O)NC)=O)C2)C1 C#Cc1ccc(Cl)c(C(=O)N(CCCNC(c2csnc2OC)=O)C2CC2)c1 C12(CNC(c3c[nH]c(C)c(Cl)c3=O)=O)CCC(CC1)N(C(C1CC1C(N)=O)=O)C2 N1(C(CCC=C=C)=O)CC(NC(=O)CC2=CCCC2)CCC1C CC(=O)CCCC(=O)N1CCC(C(=O)NCC(C)CC2CCC2)C1 N1(C(C(C)(C)CC(F)F)=O)CC2(CCCCN(C(=O)CCc3ncc[nH]3)C2)C1 C1(NC(c2cnc(CC)[nH]2)=O)CC(O)CN(C(=O)CCc2cncc(C)c2)C1 COn1cnc(C)c1C(=O)NCCC1(O)CCN(C(=O)C(c2csc(C)n2)=O)C1 C1(C(=O)NC(C2(O)CCN(C(C=C(C)C(C)C)=O)C2)C)CC2(C1)NC(=O)NC2=O c1(C(=O)NCCOCCCN(C(C(CCC)C#N)=O)C)nc2n(c1Cl)CCCC2 N1(C(C2(C3CC3)CN(C(CC(C)C(F)F)=O)C2)=O)CCOCC(C)(O)C1 C1(CCC)CN(C(C2CCC(C#N)CC2)=O)CCN1C(C1CC(=C2CC2)C1)=O c1(OC)cc(OC(F)(F)F)c(F)cc1NC(CC(=O)NC(C)(C)C)C(F)(F)F CC1CC(NC(=O)Cn2ccnn2)CCN1C(c1csc(-c2ccncc2)n1)=O c1(OC)cccc(C(C(=O)N(CCN(C(=O)C2=CSCS2)C)C(C)C)C(C)C)c1 CCC(CC)(CC)C(=O)N1CC2CC(NC(C3CCCCN3C(N)=O)=O)CC1C2 C1(CNC(Cc2c(C)nc(C3CC3)s2)=O)CCN(C(c2csc(O)n2)=O)C12CC2 C1(NC(c2c(C(C)C)n[nH]c2)=O)CC(NC(=O)CCC2CCCC(=O)N2)CC1O C1(COC)CN(C(=O)Nc2cnc(Cl)c(C)c2)CCN1C(=O)CCC(C)C c1(SCC(=O)NC2CCN(C(C(C)(C3CC3)OC)=O)C2)nc2ccccc2s1 c1(CNC(c2cccc(-n3c(C)cc(C)n3)c2)=O)ccc(Cl)cc1C(=O)N(C)C c1(OC)cc(C(=O)N(C)CCOCCNC(=O)C(C)C2CCCO2)ccc1OC c1(NC(C2(C)CCN(C(N)=O)CC2)=O)c[nH]c2cccc(F)c12 c1(C(N2CC(O)CC2C)C(=O)NCC)cccc2c1COC2=O Fc1ccc(C2(NCC3CCNCC3)CCOC2)c(F)c1 S(=O)(=O)(c1ccc2c(c1)CCO2)NC1C(OC)CN(C(c2cnco2)=O)C1 C(=O)(CCCCNC(C1CCOC1CNC(=O)CCCC1CC1C)=O)NC C(=O)(C(O)CC(C)(C)C)NC1CC2C(NC(c3c(C)cco3)=O)C2C1 c1(C(C)C)nc(=NCC(C2CC2)NC(=O)CC2(c3ccccc3)CC2)s[nH]1 N1(C(C(CC)N2CCCC2=O)=O)CC2CCCC(C1)N2C(c1cc(C)no1)=O N1(C(CN2C(C)CCCC2)=O)CC(=O)NCC1C(=O)N(C)CC1(O)CN(C)C1 C=C(C)CCC(=O)NC1C=CCN(C(c2cc(C(F)F)ncn2)=O)C1 C1(C(=O)NCC(CNC(C2CN(C(=O)NC)C2)=O)O)CN(C)CCN(C)C1 CC(C)(CC#N)C(=O)N1CCN(C(c2ccc[n+]([O-])c2)=O)C(CCN(C)C)C1 N1(C2CN(Cc3cn(CC(=C)CC)nn3)C2)CCN(C(=O)CC2(C)CC2)CC1 N1(C(=O)C=CCO)CCOC2(CCN(C(c3cc(Br)cc4nn[nH]c34)=O)C2)C1 c1(-c2c(C(=O)N(C)C)ccc(C)c2)coc2c1CN(C(=O)CCc1ccccn1)C2 Cc1ccc(Br)cc1C(C(=O)NCc1ccc(Br)cc1)N1CCC1C(=O)N(C)C c1(OCC)ccc(CC(=O)NC2CC2CNC(c2cncn2C)=O)cc1OC c1(C(N2CCC3(CN(C(c4c(CC)nc[nH]4)=O)C3)C2)=O)cn2c(C)cccc2n1 C1(C(=O)NC2(C)CC(NC(C3(CN(C)C)CCCCC3)=O)C2)CC(=O)NC1(C)C n1(CCC(=O)NCC(C23CC4CC(CC(C4)C2)C3)=O)ccc2cc(Cl)ccc12 N1(C(C=Cc2cnc(OC)nc2)=O)CCNc2ncc(C)cc21 C=CCCC(C(=O)N1CC2(CCC2)C1)NC(C1OCC2CCC1C2)=O c1(CC(=O)NCC2(CCNC(C3(C)CCNC3=O)=O)CC2)cn2ccccc2n1 c1(NC)cc(C(=O)NCCCN(C)C(C2CCC(OC)C2)=O)cc(Cl)n1 CC(C(=O)NCC1CC(C)N(C(c2csc3c2CCCC3)=O)C1)C(C)S(C)(=O)=O Cc1cccc(CCC(=O)NC(C)CCCCNC(=O)CC2CC(C)(C)CO2)c1 c1(C(=O)NCC2N(C(c3[nH]c(=NCC=C)sc3)=O)CC2)cc2c(cn1)CCCC2 C(=O)(CCC(C(C)C)NC(=O)C(F)OC(F)(F)F)NC(CC#C)C(=O)OC c1(C(N(CCCNC(C(C)NC(COC)=O)=O)CCO)=O)ccc(Br)o1 C#Cc1cccc(C(=O)NC2CCCN(C(C3CCC(=C)CC3)=O)C2)c1Cl C1(F)(CNC(C(=O)NC(C)C)=O)CCN(C(=O)CCc2cccc(F)c2Cl)CC1 c1(CN2CC(CC(=O)NCc3cnc(C)s3)OCC2)ccc(O)c(Br)c1 Cc1nnc(O)c(C(N2CC(CNC(c3ccn(CC#N)n3)=O)C2)=O)c1C c1(C(N(CCC(C(C)C)NC(C2CCN(C)C2C)=O)C)=O)ccn2c1CSCC2 C1(NC(=O)NC2(c3ccccc3)C(CC)C2)CC2(C1)CC2F C(C(=O)SC)N(C(=O)C=CC(C)=O)CCN(C)C1CC1.C(C)(C)(C)O CN1CC(CC(N2CCCCC2C2CCN(C(C3CCC(=O)N3)=O)C2)=O)C(O)C1 C1(NC(C2C(C)OCCC2)=O)CN(C(C2CC3(CCC3)CO2)=O)C2CCCC12 N1(C(CCCC)=O)CCCC2(NC(c3cn(CCO)c(=O)nc3O)=O)CCCC12 CC(CC(N)=O)C(=O)NC(C)(CNC(=O)C(C)Cc1cnco1)C1CCC1 C1(OC)CN(C)C(=O)C12CC2.C12CC(C)N(C1)C(=O)C1(CC)CN(C1)C(=O)C2 c1(C(=O)NCC(CNC(C2C(=C)C2)=O)O)ccc(-c2ccccc2C)cn1 n1(CC(=O)NC(C2(C(=O)NC(C(=O)NC)C)CC2)C)cc(Cl)cn1 c1(N(C(N(c2ccc(CC(=O)NC)cc2)C)=O)C)ccc(N(C)C)cc1Cl C1(NC(CCOC)=O)CN(Cc2cc(-c3cccc(F)c3)no2)CCC1C S(=O)(=O)(c1cnco1)N(CC)CC(C)C.c1(OCC(CC)OC)ccccc1OCC C(CCC(C)C)(C(=O)N1CC(N(C)C)C(O)C1)NC(COCC(=C)C)=O CC1=C(C(=O)NC2CCC(CNC(=O)C=CCO)CC2)S(=O)(=O)CCO1 N1(C(=O)OC(C)(C)C)CCC2(CC(NC(=O)Nc3cc(Br)ncc3Cl)C2)C1 CCCN(OC)C(=O)C1(CNC(=O)C(C2(O)CCCC2)F)CC2(CC2)C1 N1(C(CC(C)c2ccco2)=O)CC2(CCCC(CNC(=O)CO)O2)C1 c1(OCCOC(C)C)cccc(N=c2cc(NC(C)C(C)C)nc(OC)[nH]2)c1 Cc1nc2n(n1)CCCC2NC(=O)NC(C)(C)C.c12oc(nc1C)N(C)C2 c1(C(NOCCCOC)=O)ccnc(CNC(c2cc[nH]n2)=O)c1 N1(C(c2nc(C(C)C)no2)C(=O)NCCCC)CCN(C(C2CCCO2)=O)CC1 C1(N(C(CC(C)N(C)C)=O)C)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 c1(OC)cc(-c2ccc(F)cc2CN2CCC(O)(C(N)=O)CC2)ccc1C N1(CC(=O)NCC2(NC(C3CC(CC)OCC3)=O)CC2)OC(C)(C)CC1=O c1(OC)ccc2c(c1)S(=O)(=O)N(C(C)C(c1c[nH]cc(C(F)(F)F)c1=O)=O)C2=O C(CN=C(NCC(C)(C)OC)NC1CCCC1C)NS(CC)(=O)=O C1(C(N(C(C)CCO)C)=O)CCOC1C(=O)NCC1(n2cccn2)CC1 C#CC1CCC(CNC(C2(OC)CCN(C(C3CCC(C)(CC)O3)=O)C2)=O)CC1 c1(C(N2C(CNC(C(CCC)O)=O)CCCC2)=O)ccc(Cl)c(C(F)F)c1 N1(c2snc(CCOC)n2)CCN(C(=O)C(C(C)C)OCCOC)CC(O)C1 N1(C(c2c(C)ccnc2O)=O)CC=C(CCNC(c2cccnc2C)=O)CC1 C1(N(C(=O)CN(CC(N)=O)C)CCC)CCN(C(=O)CCCSCC)C1 c1(-c2cn(CCCC(=O)N(C3CCCC3(F)F)CCO)nn2)ccc2ocnc2c1 C(c1ccccc1)=C(CC)C(=O)NC1(C)CN(C(=O)Cc2nncn2C(C)C)C1 CCCCC(CNC(=O)CCOC(C)=O)NC(C12CC(C#N)(C1)C2)=O C1(CC(=O)N(C)CC2(OCC)CCC2)C2CCC(C2)N1C(=O)C(O)SC C1(C(=O)NC(CCC2CCC2)C(=O)N2CCCCCC2)CC2CCC(C1)S2 C1(NC(C2C(C)CC2)=O)CC2(C1)CC(C(N1C3CSCC1C3)=O)C2 C(=O)(C(F)CC(C)(C)NC(=O)CN(C)CCOC)NC(c1ccccn1)CC N1(C(c2ccc(CC)s2)=O)CC2(C(N3CC(O)CC3(C)C)=O)CCC1CC2 C1(N(C(C)C(=O)N(CC(C)CNC(C23CC(C)C2C3)=O)C)C)CCCCCC1 N1(C(c2ccc(C(C)C)cc2)=O)CC2CCC(NC(=O)C3=CCCCC3C)(C2)C1 C(CCC(C)(C)C(=O)Nc1cnc(F)c(C)c1)NC(CSCCC)=O Cc1sc(C(N2CCCC(N3C(=O)CCC3=O)C2)=O)c(Br)c1C.c12cn-1nn2 N1(C(C2N(CCC)CCC2)=O)CC(NC(c2cccnc2CC)=O)CC(C)(C)C1 C(CCC(=O)NC1CN(C(=O)C(O)CC2CCCC2)C1)=CC c1(C(=O)NC2(CO)CCN(C(C3CC(C)OC(C)C3)=O)C2)cc2ncccc2[nH]1 Cn1cc2ccc(NC(C3CC3NC(c3cc4cccn4cn3)=O)=O)cc2n1 c1(CC)[nH]nc(Cl)c1C(=O)NCC1CCC(NC(=O)CC2CN(C)C2)C1 c1(CC(C)NCC(=O)Nc2cc(Br)ccc2N)ccccc1[N+](=O)[O-] Cc1sc(C(=O)NC(C2CN(C(c3nc(Cl)cs3)=O)CCO2)C)nc1O C1(C(N2CCC(O)(CNC(CSCC)=O)C2)=O)Cc2ccccc2C1 N1(C(c2c(C)c(I)nn2C)C(=O)NCCCOC)CC2CCCC2C12CC2 C1(NC(CC(C)N(C(c2c(C)oc(CO)c2)=O)C)=O)CN2CCC1(C)CC2 n1(CC(=O)NC2(CO)CCN(C(CCOC)=O)C2)nc2ccccn2c1=O N1(C(CCc2ccn(C)n2)=O)CC2CC1CC2CNC(C1CS(=O)(=O)C1)=O C(=O)(C(C#N)C(C)(C)C)NC12CN(C(c3ccc(COC)cc3)=O)C(C1)C2 C1(C(=O)NC2C3(CCN(C)CC3)C2)CCCN1NC(=O)C1=CC(C)(C)C1 CC1(CNC(=O)CN2CCCNC2=O)CCC(NC(C2CC(n3cnnc3)C2)=O)C1 C1(C(=O)NCC23COC(CO)(C2)C3)CCC2CCCCC2C1 c1(OCC(=O)NCCCCCN(C)C(C2CC2C#N)=O)cccc2cccnc12 C#Cc1cccc(C(N2CCN(C(=O)C(Cl)=CCl)CC2C2CCC2)=O)c1 c1(CN2CC(NC(C(=O)OCC)=O)C(F)C2)cc(I)ccc1OC CC1OC(C)(C)OC1(C)C(=O)N(CCCNC(c1cn(C)nc1C1CC1)=O)CCO C(=O)(C(C)(O)CC(F)F)NCC1CC(C)(C)O1 N1(C(c2cnc(C(C)C)s2)=O)CCC2CCC(NC(=O)CN3CCCC3=O)C1C2 N1(C(C(c2ccccc2)N(C(C)C)C)=O)CC(O)CC1CO.N12CCC(C1)C2=O N1(C(c2ccc(C(=O)NCC=C)o2)C(=O)NCC=C)CCCC(O)(C(F)(F)F)C1 C(=O)(C(CC(C)C)NC(C)=O)NCCC1CC(NC(CC2(OC)CC2)=O)C1 c1(C(=O)NC2CN(C(c3scc(C)c3C)=O)C(C)C2)cc[nH]c(=N)c1[N+](=O)[O-] C1(C(N2C(CCC#C)CCC2)=O)CC1C1CN(C(c2cc(O)ccc2OC)=O)C1 Cc1ccc(OCC(=O)NC(C2CCN(C(C3CC4(C3)CC4F)=O)C2)C)cc1C C1(NC(C(C)(O)C2CCC2)=O)COC2C(NC(c3cccc(=O)o3)=O)COC12 C(=O)(C(C)(C)C(C)NC(c1cc(=O)cc[nH]1)=O)NCC1(OC)CCC1 n1(CC(=O)NC(C)C(C)NC(=O)CCC(C)(C)C#N)ccc2ccccc2c1=O C1(C(=O)OC)CC2(C1)C(C(=O)OC)C21CCC1.c12cc(O)c(cc1C)NC(=O)N2 N1(C(C(Cc2cn[nH]c2)NC(C(OC)OC)=O)=O)CCCC2COCC12 c1(C(=O)NC(CCNC(Cn2ccc(C)cc2=O)=O)C)cc2cc(F)ccc2[nH]1 C1(c2nc(C(C)OC)nn2C2CCC2)CC12CCOc1ccccc12 c1(OC)cc2cnc1oc2=O.N1(C)CCC(CN(C(=O)CSCC(N)=O)C)C1 C1(C(NOCCC(=O)OC)=O)C=CCN1C(C12CSCC1C2)=O c1(C(N(C(c2cccnc2)CC)C)=O)nccc2c(C)cccc12 N1(C(C2CN(C(=O)NC)C2)=O)CCC2(CC2NC(c2cc(Cl)c(Cl)s2)=O)C1 C(=O)(CCCC(C)(C)C)N(C)CC1CCN(C(c2nncn2C)=O)CC1 N1(C(C(C)=C(C)C)=O)CCOC2(CCC(NC(=O)CC(C)(C)O)CC2)C1 c1(C(=O)NCCCCC(C)NC(c2ccc(OC)cc2)=O)cccc(N)c1F N1(C(CCC(=C)C)=O)CC2(CCCC(CNC(=O)CCC3CCN(C)CC3)O2)C1 CC1(C)CCN(C(c2sccc2Br)=O)CC1NC(C12CCC1C2)=O C1(C(CC)(C)C)CCCC1(c1nnnn1-c1ccccc1OC)NC1CCCC1 c1(CNCCc2cc(C)cc(C)c2)ccc2oc(O)nc2c1 C(C)(CCN=c1[nH]c(=NC(C)C(c2ccccc2)SC)c2[nH]ccc2[nH]1)OC C1(NC(CCC=CC)=O)CCCC12CCN(C(c1ccc(N)c(SC)c1)=O)C2 C1(CNC(C2C(C)C2)=O)CCN(C(C2(c3ccc(F)cc3)CC2)=O)CC1(F)F C1(N(C(C(C)=CC2CC2)=O)CCO)CCCN(C(=O)C(c2cccc(C)c2)O)C1 Cc1cccc(-c2nccnc2OCC(=O)NCC2CN(C)CCO2)c1 c1(OC(C)C(=O)N(C2CN(C(c3ccc(CO)nc3)=O)C2)C)cc(Cl)cc(Cl)c1 N1(C(c2ccc(C(F)F)s2)C(=O)NCCOC)CCN(CC(F)F)CC1 C1(CCC)(NC(=O)CCCSC(C)(C)C)CCCN(C(C2CC(C)(C)CO2)=O)C1 N1(C(C(C)OC2COC2)=O)CCC2(CCC2)C(NC(=O)CCC2CCC(=O)N2)C1 N1(C(C(C2CCOC2)NC(=O)COC2CC2)=O)CCC(O)C(O)C1 Cc1ccc2c(C(N3CCN(C(=O)CSC4CC4)C(C4CC4)C3)=O)c[nH]c2c1 CCCC(C(=O)NNC(=O)CCc1ccccc1N)OC C1(CNC(CCN(C(CCC)C)C)=O)COCC1NC(c1nnsc1C)=O N1(C(CC=CC=C)=O)CCCC1(CNC(=O)CC1CCOC1(C)C)COC CC(CC(=O)NC1CN(C(C2C3CC4C(C3)C24)=O)C(C)(C)C1)C(C)(C)C.CCO c1(C(=O)NC(C2(O)CCN(C(C3C(C(C)O)C3)=O)C2)C)cnc2c(cnn2C)c1 CC1CN(C(=O)CCF)C(C)CN1C(=O)CN(C)S(N)(=O)=O c1(CNC(C(n2cc(CCC3CCCC3)nn2)C)=O)sc(Cl)nc1Br N1(C(C2C(CCC)CN(C(C3CCCO3)=O)C2)=O)CC2(CCCCCC2)C1 C1(C)(CNC(C=C(C)C(F)F)=O)CN(C(C2CC23CC(F)(F)C3)=O)CCO1 C1(C(=O)NCCC2CCC(C)C2)CCN(C(=O)OC(C)(C)C)CCO1 C(=O)(CCCC(F)F)N1CC(C(C)NC(=O)CSc2cnn(C)c2)OCC1 C1(C(=O)NCCNC(C(CCC)(C)O)=O)CCN(S(=O)(=O)NC)CC1 c1(CC(=O)NCC2C(C)(C)CN(C(=O)CC3CC3)C2)ncn2c1COCC2 CCC(C)(C)C(O)C(=O)N(C)CCC1CCCCN1C(c1ccc(C(C)=O)[nH]1)=O N(C1CCc2ccccc21)C(C(CCCNC(CCCCOC)=O)O)=O C1(CNC(C(F)=C(C)C)=O)CN(C(c2ccc(F)cc2C)=O)CCC1(C)C n1(CC)cnc2nc(=NCc3ccc(C#N)cc3F)[nH]c(NCC(N)=O)c12 c1(C(N(C(C)C(N2CCSCC2C(N)=O)=O)CC)=O)cccc(C)c1 c1(C(=O)NC(c2ccccc2)CO)ccc2[nH]c(-c3ccco3)nc2c1 c1(OC)c(C(=O)NCCC2(O)CCCN(C(c3cc(C)cs3)=O)C2)ccnc1Cl C=CCC(CCCCC)C(=O)NCCN(C(=O)C#CC1CCCC1)C CC1C=C(C(=O)NCC2CCCN2C(=O)CCCn2ccccc2=O)CC1 c1(CC)cc(C(=O)NCCCCc2cn(Cc3cocn3)nn2)cc(O)n1 C1(C(=O)NCCC(=O)NC(CC)C)CCN(C(c2c(C)coc2C(C)C)=O)CC1 C1(C)(NCC(c2csc(C3CCCCC3)c2)C)CCCN(C(=O)OC(C)(C)C)C1 C1(N(C(=O)CCc2cnn(C)c2)CC)CCCN(C(=O)Cc2cc(C)cs2)CC1 N1(Cc2nc(C)sc2)CCN(C(c2cccnn2)=O)CC1 CC1CC2(CCO1)CC2C(N1CC(O)(C2CCN2C(c2nc(Cl)ccc2N)=O)C1)=O c1(OCC(=O)NC2CC(NC(C3(COC)CCC3)=O)C2)cccc(Cl)c1 N1(C(C(C)(C)OCCC)=O)CCC(CNC(C2(C)CC2)=O)C(CC)C1 C#CCC(O)C(=O)N1CCC(C(C)(C)NC(=O)C(C)(C)Oc2ccccc2)C1 CCC(CNC(C1(C)CCCCCC1)=O)N=c1ccc(C(F)(F)F)n[nH]1 C1(CCNC(C2CC(OC)C2)=O)CC(F)(F)CN1C(c1csc(C#N)c1)=O c1(OC)cc(C=CC(=O)NC(CC2CC2)CC(=O)N2CCCC2C#N)ccc1O C1(CC(N2CC(NC(CCCNC(N)=O)=O)C2)=O)CCC2(CC1)CCC2O c1(C(N(C2CCOCC2)C(C)C)=O)ccc2c(c1)CC(=O)NC2 c1(C(=O)NCC23C(CN(C(C4(C)CC(C)C4)=O)C2)C3)cc2c(ccn2C)s1 C(=O)(C(C)(C)C(C)(C)C)N1C(CNC(C2CC(OC)C(OC)C2)=O)CC2CC21 C1(C(N(CC(CC)NC(c2ccccc2O)=O)CC)=O)C(F)(F)C12CCC2 c1(C(N2CC3CN(c4ncnc(C)c4Br)CC32)=O)cc2cc(F)ccc2s1 c1(OCC)c(F)c(C(N2CC3C(CNC(=O)COC(C)=O)C3C2)=O)cc(F)c1F C1(CC(=O)NCc2occ(C(=O)NC(C3CCCO3)CC)n2)C=NN(C)C1=O C(=O)(C#CC1CCCCC1)N1CCC(C(C)NC(CC(COC)(C)O)=O)CC1 CCCCN=C(NCC(C)(C)CC(C)O)N1CCC2(CCCOC2)C1 CN1C(=O)CCC1C(=O)NC(C)(C)CN1CCN(C(C2(F)CCCOC2)=O)CC1 C1(NC(=O)OCC2(NC(=O)OC(C)(C)C)CC2)CCP(C)(=O)CC1 c1(C(N2C(C(C)NC(C(C)OCC)=O)CCC2)=O)cc(C)[nH]c1C CCN(N1CCn2cc(-c3cnn(CC)c3)nc2C1)C(N)=O C1(C(=O)NCCC(=C)C)CN(C(=O)CC(C)(C)CN(C)C)CC12CCC2 CC1CCCc2nc(S(=O)(=O)N3CCC(CN(C)S(=O)(=O)N(C)C)CC3)cn21 c1(C(N(C2CCCN(C(CS(CC)(=O)=O)=O)C2)C)=O)coc2cc(F)cc(F)c12 CCC(C)C(O)CC(=O)NCCNC(=O)CCc1ccc(OC2CCCC2)cc1 c1(CCNC(C2C(C=C)C2)=O)ccc(CNC(=O)CSC(F)F)cc1 c1(C(=O)NC(CC=C)CNC(C2(n3cnnn3)CC2)=O)ccc(C)c(Br)c1 c1(SCC(N(C)C(C2CC(C(N)=O)C2)=O)C2CC2)ccc([N+](=O)[O-])cc1F c1(CN(c2ccccc2)CC(=O)NC(C)(C)CC(N)=O)ccc2c(c1)OCO2 C#CC(C(C)C)NC(=O)Cn1cc(CNC(c2cc(C(N)=O)c[nH]2)=O)nn1 C12(CNC(CN(C)Cc3ccc(C)cc3)=O)CN(C(=O)C(C)(F)F)CC1CCO2 c1(C(N2CC(O)(CCNC(C(CSC)OC)=O)C2)=O)cc(C(F)(F)F)cnn1 C1(NC(c2c(C)onc2Br)=O)CN(C(=O)CC(C)CF)C2(CCC2)C1 c1(C(N2CC(C(=O)CNC(C(F)OC)=O)C2)=O)nc[nH]c1C(C)(C)C C1(NC(c2ccoc2Cl)=O)CCN(Cc2cccc(F)c2Cl)CC1O Cc1cccc(C)c1OCC(=O)N(C(C)CNC(C1CCC(=O)CC1C)=O)C N1(C(C(C)CO)=O)C(CC(=O)Nc2ccc(N(C)C)cc2)C2CCCC12 C=CCC(CNC(=O)C(F)OC(F)(F)F)C(=O)N(C)CCOC1CCCC1 Cc1c(NCCc2ccc(F)c(Br)c2)nc[nH]c1=NCC1CC(CC)=NO1 c1(CC)c(C(=O)NC(C2CCOC2)CNC(=O)CNC(=O)COC)nnn1CC c1(C(C)C)ccc(CC(=O)NC(C)CNC(C2CCCN(S(C)(=O)=O)C2)=O)cc1 C1(OCC)(CNC(=O)C(C)O)CN(C(c2ocnc2C2CC2)=O)C1 c1(N(CCCNC(C(CC)C(C)O)=O)C2CC2)nc2cc(Cl)cc(Cl)c2o1 Cc1cc2c(C(=O)NCCCCCNC(C3CCCC(F)C3)=O)nccn2n1 C1(C(=O)NC2(C)CC2C)CCN(C(c2cn(CCCC)nn2)=O)CC1 O=C(C1=CCC2(COC2)OC1)N1CCOC2CCN(C(C3(CO)CC3)=O)CC12 C(C(CCC)C(=O)NCC1(SC)CC=CC1)NC(C1C(=C)C1C(=O)OC)=O N1(C(c2c(C)nccn2)=O)CCCC2(CCN(Cc3c(O)cccc3F)C2)C1 CN1CCN(C(C2CC(=O)CN2C(c2ccc(=O)n(C)c2)=O)=O)C(CO)C1 C(=O)(C1=CCSC1)NCC1(CNC(C2CCC(C(=O)OC(C)(C)C)C2)=O)CCC1 C(CCC(O)CO)NC(CCN(CC=C)C(C1CCC2(CC2)C1)=O)=O CCCC(C(=O)NCCC1CCN(C(C2CSCCS2)=O)CC1)OCC CCC(C)CCCCC(=O)NCC(C(=O)NCC1(C)CC(O)C1)C(C)C c1(OC)ncnc(OC)c1NC(C1(C#N)CCN(C(=O)CCc2ccco2)C1)=O c1(C(N2C(CNC(C=Cc3n(CC)ncc3)=O)CC2)=O)ccc2nc(S)[nH]c2c1 CC1C(NC(c2cc(Cl)ccn2)=O)CCCN1C(c1ncc(Cl)nc1Cl)=O c1(C(=O)NCC2(F)CCC(NC(CC=CC=C)=O)C2)cc(C(F)(F)F)c(Cl)cn1 C1(C(=O)NC(C2CN(C(C3CCC(CO)CC3)=O)CCO2)C)CCCCCC1 C1(NC(C=C(C)C(C)C)=O)CCCCN(C(C2COC(C)C2)=O)C1 C1(C(=O)NCC2(F)CN(C(CSCC(=O)OC)=O)C2)CCc2nnnn2CC1 CC(C)CC(C(=O)N(C)C(c1cnn(C)c1)C)ONC(=O)C1(F)CCC1 c1(CC(C(=O)OCC)NC(c2ncoc2CC)=O)ccc([N+](=O)[O-])cc1 N1(C(C(CCSC)O)=O)C2CCCC1CN(C(c1cc(Cl)cc3nc[nH]c13)=O)C2 N1(C(C2C3(CCN(Cc4c(OC)cccc4Br)C3)C2)=O)C2CCC1CN(C)C2 c1(CC(C)NC(=O)C=CC(c2cc(Br)sc2Br)=O)nn(C)c2ccccc12 CC1=C(C(=O)N2CCC(C)C(NC(c3cnc(C)cn3)=O)C2)CCCO1 C1(C(N2CCC(C)(NC(CC(C)(C)N(C)C)=O)C2)=O)CCOC(C)(C)C1 C1C(C)(O)CC(=O)N1.c1(C(C(N2CC(O)(CSC)C2)=O)(C)C)cnccc1C N1(C(C(C)NS(CC)(=O)=O)=O)C2CCC1C(CNC(=O)CC(C)O)C2 C1(C(N2C(CC(=O)NC)CC2)=O)CN(C(c2ccc(C)c(F)c2)=O)CC(C)(C)C1 CC1CCCn2ncc(C(=O)NC3CC(CNC(C4CCCC4C(F)F)=O)C3)c21 CCCC(CCCO)C(=O)NCC1(C)CCN(C(C23CCCN(CCC2)C3)=O)C1 CCCCC(CC)CC(=O)N1CC(O)(C2(CNC(=O)C(F)=CCC)CC2)C1 c1(C(=O)NC(C2(O)CN(C(C=CCC)=O)C2)C)cc(S(=O)(=O)CC)cnc1O N1(C(=O)NCCCOC)CCC(C)(NC(C2CC(OC)C2)=O)C1 C=C=C(C)CC(=O)NCc1cccc(CCCCC)c1.C12CCN1NC2=O c1(OC)ccc(F)c(CNCCC(N)CCC(C)C)c1Cl C1(NC(CCC(=C)C)=O)CC(F)CN(C(C2(CCC)CCNC2=O)=O)C1 CC1CN(C(c2cc(C(F)F)cc(F)c2)=O)CCC1N(C(=O)CCC(F)(F)F)C n1(CC)nc(C2CC2)cc1NC(=O)NCC1(O)CC(N(C)C)C1 C1(C(=O)NCC(C)N(C)C(c2ccc(C3(C)CC3)cc2)=O)CCCN1N=O C(CC(C)(C)C(=O)NCC(C)(CC(C)C)NC(=O)CC1CCCN1C(C)C)OC C=CCC(CC)C(=O)NC(C)(CNC(=O)Cc1ccn(CC)n1)C1CC1 N1(C(CCOCCC)=O)CCN(C(=O)C(CC)n2cccn2)C(CC(=O)OC)C1 CCC(CCC(=O)N1CCCCCC1C(=O)N(CCCN1CCCC1)C)OC N(C1CCCc2c(I)n[nH]c21)CCc1c(I)cccc1 C12(C(=O)NCC3(C)CCN(C(C4(C)CC4)=O)CC3)CCCCC1C2(F)F c1(CNC(C2(OC)CCOC2)=O)ncc(C(=O)NCC2CCC2(F)F)cn1 c1(OC)ccc(I)c(NC(=O)Nc2ccc(CCO)c(F)c2)c1 N1(C(C2N(C(CC(CCC)(C)O)=O)CC=CC2)=O)CC2C3CCC(C3)C2C1 c1(OC)ccccc1C(CNC(=O)Cc1cnoc1)NC(c1nc(OC)c(C)s1)=O Cc1ccc2[nH]c(C(N3CCN(C(c4cnco4)=O)CC3CF)=O)cc2c1C C(=O)(C(CNC(=O)C(C(C)C)OCC)C(C)(C)C)NC(CCCC)CO C1(NC(C(CC)O)=O)CCS(=O)(=O)C12CN(C(c1cnn3c1OCCCC3)=O)C2 C1(C(=O)NC2(CC=C)CN(C(c3ccc(C4COC4)cc3)=O)C2)CCC(C)CC1 c1(N2CC3C(CC(=O)N(C4CCC4)C)C3C2)cc(Cl)nc(CS(C)(=O)=O)n1 N1(C(c2cc(C)c(C)o2)=O)CCC2(COC(CNC(C3CC3C)=O)C2)C1 Cc1ccc(C=CC(=O)NC2CC2NC(=O)C=Cc2ccc(O)cc2)c(C)c1 c12cc(Cl)ccc1c(=O)[nH]n2C(C)C.C1(NCC)CCC(C(=O)OC)CC1 C12(C(=O)NCC3C(NC(C=C(C)C)=O)CCCC3)CCC(CC1)OC2 C#CC1CN(C(=O)COC(F)(F)F)CCN1C(=O)C(F)=CCC CC1(C)CC(CCNC(=O)CC(C2CC2)NC(c2cc(Cl)cs2)=O)CO1 c1(CC=CC(=O)NCC(C2CC2)NC(C2CC(OCC)C2)=O)cccc(Br)c1 c1(OC)ccc2c(c1)CC(C)CC2Nc1nccc(N(C)Cc2cn[nH]c2)n1 N1(C(Cn2nc(C)oc2=O)=O)CCN(C(=O)C=CCn2cncn2)C(C(F)F)C1 C1(C(=O)NCCCC)CCN(C(=O)CCc2ncc(C)[nH]2)C(C)C1 c1(CCC(=O)N(CCCNC(Cn2ccc(C)c2)=O)CCO)ncccc1C CCCCC(C)C(=O)NC1CCC1CNC(=O)C(c1cnn(CC(=O)OC)c1)=O CCC(C)C(CNC(C1(C)CCCN1C(=O)C(CC1CC1)OC)=O)CO C1(NC(CC2(C=C)CC2)=O)CN(C(=O)C(F)C2CCC2)CCC1C C(C)(C)(CCC(=O)N1CC(C(=O)NCCNC(C2(CO)CCCCC2)=O)C1)OC C1(CCCNC(CCOCC#C)=O)CCCCN1C(c1nccn1C)=O CC1N(C(=O)CC2CCCC2NC(=O)CN2CCCC2=O)CCC1(C)C CCC(CC(=O)NCCN(C)C(c1cc(O)c2ccsc2c1)=O)C(C)(C)C N1(C(CSc2n(C)cnc2)=O)CCCC(C2(NC(=O)CC3CCCCO3)CC2)C1 N12CC3CCC(C3)(C1)C2=O.CC1CCN(C(=O)CN(C(=O)CC2CCCC2)C)C1 N12CCCC1C(=O)NC(C)CNC(=O)C2.c1(CO)cscc1C(F)F c1(CCC(=O)NCC(CNC(CCSC)=O)F)cnc2n1CCOC2 c1(C(=O)NC(c2ccc(CC)o2)COC)ccc2c(c1)C(=O)CCC2 n1(CCC(N2CC(O)(CNC(CC=C)=O)C2)=O)ccc2c(C)cc(Cl)cc12 Cc1nc(=N)[nH]cc1C(=O)NCC12CC(NC(=O)CC3CCN(C)C3=O)(C1)C2 C1(CCC(=O)NCC(O)(C2CC2)C2CC2)CCCCN1C(=O)COCC1CC1 CC1(C)CN(C(=O)CC2CCCCCCC2)CC1CNC(c1coc(CO)c1)=O C1(C(N(C)CC2CCCCO2)=O)CCCN(C(C2CCOC2(C)C)=O)CC1 Cc1nc(CNC(C2(CNC(=O)CCOCC(C)C)CC=CC2)=O)oc1C c1(CC)cc(C(=O)NCC2OCCC2C(=O)NOCC(=O)N(C)C)n[nH]1 Cc1cncc2cc(C(=O)NC(CNC(c3cnc(C(C)C)[nH]3)=O)C(C)C)sc12 c1(C(N2CC(C)C(NC(=O)C(=O)N(C)C)C2)=O)c(OC(F)(F)F)ccc(F)c1N CN1CCC(CNC(=O)C(C)(C)C2CCOC2)C1 C1(CCOC)CN(C(C2CCN(C)CC2)=O)CCN1C(=O)CSCCC(F)(F)F C=CC(CC)CC(=O)NCC(O)C(=O)N(C1(C)CC1)C.N1(CC)CC=CC1 CC(C(=O)NCC1(NC(c2n[nH]c3ccc(O)cc23)=O)CC1)C(C)S(C)(=O)=O N1(C(C=CC)=O)CCCC(C(C)NC(=O)C(COc2ccccc2)OC)C1 c1(C(=O)NC2CCC(C(=O)NC(C3CCOC3)C)C2)cc(Br)ccc1Br c1(OC)ccc(CNC(C2(CNC(c3cc(O)n(C)n3)=O)CC23CCC3)=O)nc1 C1(NC(c2ccc(OC)nc2OC)=O)CC2(CCCN(CC(F)(F)C(F)F)C2)C1 CC1=C(C(=O)NCC2(NC(c3cc(C4CC4)ccn3)=O)CC2)CCS1(=O)=O C1(NC(CN(C)CC)=O)C(C)CN(C(=O)C(F)(F)C(F)F)CC1C c1(C2(C(=O)NCC#CCNC(C3C(C)OCC3)=O)CC2)ccc(Br)cc1 Cc1oc(C(=O)NCCC2CCCN(C(=O)CC3CCCCC3O)C2)cc1CO Cc1cnn(C)c1C(=O)NCC(=O)NCCN1CC(OCCNC(N)=O)C1 C1(NC(C(C2CC2)OC)=O)CCN(c2nnc(C(F)F)o2)CC1(C)C N1(C(COCCOC)=O)CC(n2cc(C(O)CC(C)C)nn2)C(C)C1 C1(C(N(C(CN(C(C2C(C(C)=O)C2(C)C)=O)C)C)C)=O)CCCCC1(C)C c1(C(=O)NC2CN(C(C(CC)N(C)C)=O)CC3C2C3)ccc(P(C)(C)=O)s1 C1(C(N(CC(=O)NCCN2CCNC2=O)CCOC)=O)CCN(C)C1=O c1(CNC(c2cc(C)[nH]c2)=O)cn2c(Nc3ccsc3C(=O)OC)cccc2n1 n1(CCC)nc(C)c(C(=O)NCCC(O)CNC(c2sc(C)nc2C)=O)c1C c1(OC)ccc(C)cc1C(=O)NCC1(O)CC(CNC(=O)C(C)C#N)C1 c1(C(=O)NC2CC(NC(C3(C#N)CCCC3)=O)CC2O)c(F)ccc2n[nH]cc12 c1(C(=O)NCCNC(C(CC(C)C)NC(C)=O)=O)ccc(C#N)c(O)c1 N1(C(C(CC#C)C)=O)CCC(NC(=O)COc2cc(C)ccc2F)C(C)(C)C1 N1(C(CC2CCC(C(C)=O)CC2)=O)CC(NC(=O)C=Cc2ccoc2)C(C#N)C1 N1(CCCNC(c2n(CC)c(Br)nc2)=O)C(=O)C2CCCCC2C1=O c1(C(=O)NC(C)CNC(c2cccc(C(F)F)c2)=O)cc2ncccc2[nH]1 C1(NC(C=NOC)=O)CC2CN(C(=O)C(C3CCCCC3)C)CC2C1 CC(c1cccs1)=CC(=O)NCC(N1CCN(C(=O)CC2CCC(O)C2)CC1)=O C#CCCN=C(NCCc1cc(OC)ccc1Br)NCC(C)OC(F)F c1(C(=O)NC2CCCCC2NC(c2coc(O)n2)=O)cnc2c(c1)NCC2 c1(C(=O)NC(C(C)NC(Cc2c(C)nsc2)=O)CO)c(C)nn(CCO)c1C C(C1CCCO1)=CC(N1C(CNC(C2CC23CC3)=O)CC1)=O c1(CCC(=O)NCC)ccc(N(C2CCN(C(=O)C(CC)OC)CC2)C)nc1 CC1COCCC1NC(=O)C(c1ccco1)NC(=O)Cc1c[nH]ccc1=O N1(C(c2c(N)ncc(Br)c2)=O)C2CCC1CC(CNC(=O)CCC1CC1)C2 C(=O)(CCCC(C)NC(c1cc(C(C)=O)[nH]n1)=O)N(CC)CC N1(CC(=O)NCCSCC(=O)NCC(C2CCCO2)C)C(=O)CNC1=O c1(N(C)C(C2CC=CCO2)=O)ccc(CC(=O)NC2CCN2S(C)(=O)=O)cc1F c1(CCNC(CC2N(C(C(COC)O)=O)CC2)=O)ccccc1C C1(C(=O)NC2(C(N3CC(C)C(NC(=O)OC(C)(C)C)C3)=O)CC2)CCS(=O)(=O)CC1 C(C)(C(=O)N1CCC1CNC(c1ccc(-c2ccco2)s1)=O)(C(C)C)NC(C)=O C12(NC(C(c3ccc(Cl)cc3)CC)=O)CC1CN(C(=O)Cc1nc(=O)o[nH]1)C2 CC1CCN(C(C2CC3(CC3)C2)=O)C1CNC(=O)CCF C1(C(N(CC(C)O)CCNC(=O)CSCc2cccs2)=O)CN2CCN1C(C)C2 C(=O)(C1=CCN(C)C1)NCc1occ(C(N(CC(C)CO)C)=O)n1 N1(C(COCC)=O)CCC(C)(C)C(NC(=O)CC(C)(C)c2cccs2)C1 c1(C(N(CCN(CC)CC)C)=O)ccc(S(C)=O)cc1.C1(=O)C(F)C(=O)N1 C(=O)(C(C)(F)C(=O)NC1CN(C(c2ccc(N(C)C)cc2F)=O)C(C)(C)C1)OC O=C(C1CCCc2nccn21)NCCc1cn(-c2cc[nH]c(=N)c2)nn1 n1(CC(=O)NC(CNC(CC(C)C(F)F)=O)CO)nnc2ccccc12 N1(C(C2(C)C(C)CN(C(=O)C(C)NC=O)C2)=O)CCNC(=O)CC1C CC1C2CN(C(=O)C(O)CNC(C3(C4CC4)CCCO3)=O)CC12 c1(C(=O)NCCOCCC)conc1CNC(c1ocnc1C)=O C(=O)(C1Cc2ccc(Cl)cc21)NC(CNC(c1nc(Cl)cs1)=O)C1CC1 c1(CC(C)C(=O)NC2CCC2NC(c2nnn(C)n2)=O)ccc(F)cc1 N(C1CCc2ccc(Br)cc21)N1C(=O)NC(C)(C2CC2c2cccc(Br)c2)C1=O N1(C(C(F)OC)=O)CCC(C)(CNC(C2(CO)CC(F)(F)C2)=O)C1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(NC(C(C)=C2CCC2)=O)C1 CC1(C)CC(C(=O)N2CCCC(C(=O)NCCN3CCC4CC34)CC2)=NO1 c1(CC(=O)NCC(CNC(C2C(CC)OCC2)=O)O)cccc(C(F)F)c1 C(=O)(C1=CC2C=CC(C1)C2)NCc1occ(C(N2CCC(C)(C#N)C2)=O)n1 C(=O)(C(CC(C)CC)NC(c1cc(C)sn1)=O)N1CCC(CCC#C)CC1 CC1CC(CNC(c2cc3scnc3[nH]2)=O)CN(C(c2cc(F)ccc2Cl)=O)C1 Cc1cnoc1C(=O)NCC1C=CC(NC(C2(C)CCCO2)=O)C1 C1(C(=O)NCC2CCN(C(=O)CC3CCCCC3O)CC2)COC2CCCCC12 C1(CCC(=O)NC(CC)CO)CCCN1C(c1cscc1Cl)=O.C12CCCN1C2 c1(C(N2CCC(NC(C(OC)OC)=O)C2C(C)C)=O)ccc(=O)n(C)n1 c1(C(=O)NC(CC(C)NC(c2c(SC)cccc2)=O)C)noc(C)c1[N+](=O)[O-] c1(C(N2CCC(C(F)F)(CNC(CCCC#C)=O)C2)=O)cc2cc(Cl)sc2[nH]1 CC1CC(=O)NCC1C(=O)NCCOCCCN(C)C(c1ncc(N)cc1Cl)=O N=c1[nH]c(=NCc2ccsc2)[nH]c(=NC2CC3C(C2)C3(F)F)[nH]1 CC1(C)CCC(CC(=O)NC2CCN(C(c3cnc(C4CC4)nc3)=O)C2)O1 N1(C(C(C)OC(C)=O)=O)CCC(C(O)CNC(C2CC3(CC3)C2)=O)CC1 C1(C(=O)NCC2CCC(NC(CSC(C)C)=O)C2)COC(C)(C)CO1 c1(C(N(C(C)CCNC(=O)Cn2nccn2)C)=O)csc(Cl)c1Cl Cc1cc(N)cnc1C(=O)NCC1CC1CNC(=O)Cc1nn(C)cc1Cl C1(CN(C(c2ccc(F)cc2Cl)=O)C2CC2)CCN(c2ncns2)CCC1(F)F C(=O)(CCCCSC)NC1(CC=C)CN(C(=O)CC2(n3cncn3)CC2)C1 CC(CC(=O)N1CCC(CNC(c2ccc(-c3ccsc3)cc2)=O)C1)C(C)(C)C C1(CC(=O)N(CCN(C(C(C)SC(F)(F)F)=O)C)C)CCCC2(CCC2)O1 O=C(CC1OCCc2ccccc21)NCCNC(C1(C2=CCCCCC2)CC1)=O c1(CC(=O)NC2(CNC(C(CC=C)C)=O)CC2)ccc([N+](=O)[O-])c(N)c1 C1(C(=O)NCC2N(C(C34CCC(OC)(CC3)C4)=O)CCC2)CCc2nc[nH]c2C1 CC1CCc2n[nH]cc2C1C(=O)NCC1(C)CCCC(F)(F)C1 Cc1c(-c2cncn2-c2nn[nH]n2)cccc1N.N1CCC(C)C1c1ccc(F)cc1 c1(CC(=O)N(CCCNC(=O)CC2CC(F)C2)C)cn2ccccc2n1 C1(CCNC(C2(C)CC2)=O)CCCN(C(C2CCC(C)CC2)=O)CC1 C(=O)(CCCCC(C)C)NC(CCC(=O)NC1(COCC)CC1)CC N1(C(C(C)CO)=O)CCCN(C(c2ccc(SC(F)(F)F)cc2)=O)CCC1 C1(C(=O)NC(COC2CC2)CO)CC2(CCN1C(=O)CCc1ccccc1)CC2 c1(C(N(C)CCNC(=O)CN(C(C2CCC2)=O)CC2CC2)=O)ncccc1F c1(OC)nc(C)ccc1C(=O)NCCC1CCC(NC(=O)C(F)(F)CF)C1 C1(CNC(C2(C(C)C)COC2)=O)C2CN(C(c3scnc3C(F)(F)F)=O)CC12 C(c1ccc(Cl)s1)=CC(=O)NC1(CCCNC(C(C2CCOCC2)OC)=O)CC1 C=C1Cn2c(C(=O)NCCC(C)NC(C3OCCOC3C(F)(F)F)=O)nnc2S1 N(C)(S(N)(=O)=O)CC(=O)NC1CC(N(C(=O)CCC2CCCCC2)C)C1 N1(C(C(C)(C2(C)CC2)OC)=O)CC(CC(=O)NCCCN2CC=CC2)C2(CC2)C1 C1(NC(C(C(C)NC(C2(C(=O)N(C)C)CC2)=O)C)=O)CC(C)N(C)CC1C N1(C(C2N(C)CCCC2)=O)CCCC(C)(C)C1CNC(c1ccoc1C1CC1)=O c1(C(C)C)ccnc(NC2CCCC2NCc2ccccc2CO)n1 C(=O)(CCS(N)(=O)=O)NC(CN(C(c1cc(OC)cc(Cl)c1)=O)CC)C C=CC(C)(CC)C(=O)N1CCC(CCCNC(=O)COC2CCCCC2C)CC1 N1(C(c2ccc(F)cc2)=O)CCC2CC12C(=O)NCCN1CCCC1=O CCCCC(O)C(C)C(=O)NCC1CC(C(=O)Nc2ccc(C)c(C#N)c2)=NO1 C1(C(=O)NCC(CC(C)C)NC(C(CCC)F)=O)CCCC(=O)N1C C1(C(N2CC(NC(C3OCCC3CSc3ccccc3)=O)C2)=O)(CC)CC1(F)F C1(NC(c2cc(C(C)=O)cn2C)=O)CC(F)CN(C(=O)CC(C)(C)C)C1 C1(NC(C2CCn3ncnc3C2)=O)CN(c2nc(Cl)ncc2F)CC2(CCC2)C1 C1(N(C(c2cc(C)c(O)nc2)=O)C)CCN(C(=O)CCn2cnnn2)CC12CC2 C1(C(C)(C)C)(CNC(C(CC)NC(C)=O)=O)CCN(C(=O)CCCC2CC2)C1 c1(N(C)CC2CCCN(C(=O)CCC3CCOC3)C2)ccc(Cl)cc1[N+](=O)[O-] N1(C(Cc2ccc(C(C)=O)s2)=O)CCCC(C2CC2NC(c2cnc(SC)[nH]2)=O)C1 C1C(C)C(=O)N1.C(C(F)(F)F)(C1CC1)NC(C1CN(C(C)=O)C1)=O CC(C)C#CC(=O)N1CC=CC1CNC(=O)C(c1ccccc1)C CC1CCc2[nH]c(=NC(Cc3ccccc3)CCO)c(C#N)cc2C1 c1(OC)cc(C(N2CC3(C2)CN(C(=O)C(C)(C)C(F)F)C3)=O)cc(C)c1 c1(C(=O)NCC(CNC(=O)CCN2CCOCC2)OC)nccc(N)c1Cl CCC(CC)CCCC(=O)NCC(CO)NC(=O)C(C)Sc1nncn1C c1(C(C)=O)cnn2ccc(=NC3C4C5CCC(C5)C34)[nH]c12 N1(CC(=O)N(C)CC2N(C(c3n(CCC)ncc3)=O)CCC2)CSCCSC1 Cc1ccn2cc(C(=O)NCC3CC4CCC3N4C(C3CCCN3C)=O)nc2c1 C=CC1(C(=O)NCCC(C)(O)C2CC2)CCN(C(=O)CC2CC3CC3C2)CC1 C1(C(N2CC(CNC(c3c(CC)occ3)=O)C2)=O)CCN(CCO)C(=O)C1 C1(NC(C2C(C)C2)=O)CCN(C)C12CCCN(C(c1ccoc1)=O)C2 CN1CC(C)(C(=O)NC2CC(NC(=O)CSc3ccncc3)C2)CC1=O c1(C(N(C2CCN(C(=O)CC=C(C)C)C2)CCC)=O)ccc2c(c1)CCN2C c1(CC)nccnc1C(=O)NCCN(C1CC1)CC1CC(=O)N(CC(F)(F)F)C1 Cc1cc(C(N2CCCC2CN(C(=O)C(Cl)(Cl)Cl)C)=O)nc2nccn12 N1(C(C2NC(=O)OCC2)=O)CC2CCCN(C(c3cc(Cl)c(Cl)s3)=O)C2C1 c1(CSC)nc(-c2nn(C)cc2Cl)n(C2COC(C)(C)C2)n1 c1(C(=O)OCC)c(C)[nH]c(C(=O)N(CC(C)CNC(=O)C2=CCC2)C)c1C(C)C C1(CNC(C(C)(C)C2CCCN2C(c2cccnc2)=O)=O)CCCC12CCC2 C#Cc1ccnc(C(=O)NCC23CC(C2)C(NC(=O)CC(=O)NC2CC2)CO3)c1 N1(C(c2c(N)cncc2)=O)C2CCC1C(CNC(=O)CN1CC3CCC1C3)C2 C1(CNC(CC(C)F)=O)CC(NC(=O)Cn2cccn2)CC1O C1(CNC(=O)CCC2CCC2)CC(O)CN1C(=O)CCn1cnnn1 N1(C(C2C(C)N(C(c3cocn3)=O)CC2)=O)CCC2CCN(C)CC12 Cc1nc(NC(C2(CNC(=O)C(C)(O)CC)CC2)=O)sc1I C1(OC)CC2CCC(C1)N2C(c1cc(CNC(=O)CCCC2CC2)no1)=O C12(C(=O)NC(Cc3cc[nH]n3)C(=O)NC3CCCC(F)C3)C(=O)C3CC1C2C3 C(C1CCOCC1)=CC(=O)NCCNC(C1C(Cl)(Cl)C12CC2)=O C1(OC)CCOCC1NC(=O)CCN(C)C(c1ccn(C)c1)=O N1(C(C(C(C)C)SC)=O)CC(NC(=O)C(c2csc(=N)[nH]2)=O)C2(CCOCC2)C1 C=C(C)CC(C(=O)N1CCC(N(C(c2nncn2CC)=O)CC)CC1)OC Cc1cccc2c(C(=O)NCC3CC3NC(=O)C=Cc3ccsc3)coc12 C=C1CN2C(=O)CCC2(C(=O)NCC(C)NC(=O)C(CC(C)C)N(C)C)C1 N1(C(c2cc(OC)ncc2)=O)CCC(CO)(CNC(C2C3CC(=O)CC23)=O)CC1 c1(C(=O)NCC(CC)NC(C2CN3CCN2C(C)C3)=O)csc(S(C)(=O)=O)c1 C(CCNC(=O)C(Br)=C(C)C)(C(C)(C)C)NC(C=C(CC)C)=O C1(C(N2CC(C(C)(C)O)(CNC(C3(C4(C)OCCO4)CC3)=O)C2)=O)CCCOC1C C1(OCC(=O)N(C)CCc2ccccc2)CCN(C(=O)COCCC2CCC2)C1 C1(NC(C2C(CCOC)C2)=O)CCN(C(=O)Cc2ccc(F)cn2)CC12CCC2 CCCC(C(=O)NCC(C)CN(C)C(c1cc(OC)no1)=O)N(C)C C(=O)(CC(C)(O)C(F)(F)F)NC12CC(CNC(C3C(C(=O)OCC)C3)=O)(OC1)C2 C12(CCNC(C(C=CC)O)=O)CCC(CC1)N(C(C1CCCCC1C1CC1)=O)C2 c1(C(=O)NC(CN(C(C2C(C)(C(=O)OCC)C2)=O)C)(C)C)sc(C(C)C)nc1C Cc1ccc(CCCCC(N2CC(NC(C3CSCCS3)=O)C(F)C2)=O)cc1 C1(OC)CC(CO)N(C(C2(Cc3ccccc3Cl)CN(C(=O)CN)C2)=O)C1 c1(C(=O)NC(CC)CNC(c2ccc(C(C)F)cc2)=O)noc2cc(F)ccc12 N1(C(CCCN2CCCC2)=O)CCCC(c2cccc(Cl)n2)C1 CCC(C(=O)N1CC(CCO)C1)NC(C1CC1C(C)(C)C)=O Cn1cnc2[nH]c(=NCc3cscn3)nc(N3CCOC(C#N)C3)c12 CN1CCN(C)CC(C(=O)NC2CCCCC2NC(c2cnc(=N)[nH]c2)=O)C1 CCC(CO)CN=C(NCc1snnc1C)NCC1CCOC1 c1(C(=O)NC)c[nH]c2ncc(-c3ccc(SCCF)cc3F)cc12 N1(C(C2CCN(CC(C)C)C2)=O)CCN(C(c2ccc(N)c(N)n2)=O)C(CF)C1 CC(C)C(CCNC(C1(C(C)NC(=O)Cc2csc(=N)[nH]2)CC1)=O)N(C)C c1(CNC(=O)NC(CCC)C(F)(F)F)cccc2c1OC(F)(F)O2 N1(C(CCOCCOC)=O)CCC2CCC(NC(=O)Cc3ncc(Cl)s3)C1C2 c1(CCC(=O)N(CC(C)NC(=O)C(C)(C)N2CCCC2)C)cncnc1 C(c1ccc(NC(N2CC(C=C)C2)=O)cc1)=CCO C1(NC(CNC(C(C)(C)C)=O)=O)CCCCN(C(=O)COC2CCOC2)C1 c1(C(=O)OC)ccc(O)c(C(=O)NCC2C3CCC(C3)N2C(=O)CC(C)OC)c1 N1(C(C2CN(CCOC)C(=O)C2)=O)CCC(C)C(NC(=O)C(C)n2cncn2)C1 c1(OC)oc(C)nc1C(=O)NCC1CCCC1NC(C1CC=CCO1)=O C#CCCCCC(=O)NC(Cc1ccccc1Br)C(=O)NC1CCN(C(N)=O)C1 C12(C(N(CCCN(C(=O)COCc3cccc(Cl)c3)C)C)=O)CCC(CC1)C2 C1(N(C(C(N)CC2CC=CCC2)=O)CCc2ccccn2)CCCC(F)C1 C1(C(=O)NCCN(C(CCN(C(C)=O)C)=O)Cc2ccccc2)COC(C)C1 N(C1CCCc2c(F)cc(F)cc21)CCCN1CC(C2OCC2(F)F)C1.CNC c1(C(N2CCC(N(C(C(CC=C)C)=O)CCC)C2)=O)c(C)cc(C#N)cc1C N1(C(C(CC#C)SC)=O)CC(C)(C)CCC1CNC(=O)CCOCCOC CC(C)(O)C(F)C(=O)N1CCCC(NC(c2ccsc2Br)=O)C1 c1(C(N(CCNC(C2C(C=C)OCCC2)=O)CC)=O)cc(Br)cc(C)c1F CC1(NC(=O)Cc2ccsc2Br)CCN(C(=O)Cc2cncnc2)CC1 C1(CCNC(c2cnnn2C2CCOCC2)=O)COCCN1C(C1CC1(F)F)=O c1(C(=O)NC2C(NC(c3c(C(C)C)con3)=O)CCCC2)nsc2ccccc12 N1(C(C2(COC)CCCC2)=O)CCC(F)(C2(CNC(=O)CN3CC=CC3)CC2)C1 C1(C(=O)OC)C2COC(C(=O)NCC(C)(O)CNC(=O)CN3CCOCC3)CC12 C1(C(=O)NC(c2nnc(C)o2)C)C2CN(C(c3c(C)noc3C)C3CC3)CC12 C1(C(N2C3CC(CC(NC(C#CC(C)C)=O)C3)C2)=O)CCc2nnn(C)c2C1 c1(C(=O)NC(C(=O)NC2CC2F)C2CCCC2)c[nH]c2nccc-2c1 N1(C(C2CCC(CNC(C(C)(F)c3ccon3)=O)CC2)=O)CC2(CCNC2=O)C1 CCC(C)(O)CCNC(C1CCOCC1NC(c1cccnc1C)=O)=O S(=O)(=O)(c1cc(C(=O)NCC(C2CC2)NC(=O)CC(F)(F)F)c(C)o1)NC C(=O)(C1=CCOCC1)O.c1(CCN(C(=O)CNS(C)(=O)=O)CC)csc(C)n1 N1(C(c2nc(CC)sc2)=O)CCC2(N(CC)CC)CCCC12.C(C1CCC1)=CC=O c1(CC(=O)NC2CC(NC(CCCCC#N)=O)C2)c(F)c(F)c(F)c(F)c1F Cc1nn(C(C)(C)C)cc1C(=O)NC1CCCC1CNC(c1ccncc1N)=O C1(C)(C(N2CC3C(CNC(CN(S(C)(=O)=O)C)=O)C3C2)=O)CC(=O)N(C)C1 c1(C(N2CC(C)(C(=O)OC)C2)=O)cc(F)ccc1CC(N1CCC1CO)=O CCCC(O)CC(=O)NCC1(NC(c2cc(OC)cnc2F)=O)CCCC1 C(=O)(C(O)CC(F)(F)F)NCC12OCC(C(=O)Nc3c(F)cccc3F)(C1)C2 c1(NC)ccc(C(=O)NC(C)CNC2CC2F)cc1[N+](=O)[O-] c1(C(=O)NCCCCNC(C(CC)N(C)C)=O)cnn(-c2ccccc2F)c1C N1(C(CC(C)C(F)F)=O)CCC2(CCOCC2)C(CNC(c2coc(O)n2)=O)C1 c1(C(N2CCC(CC=C)(NC(c3cc(C4CC4)sn3)=O)C2)=O)ncc(N)cc1Cl n1(CC(=O)NCC2C3CN(C(=O)CCCn4cncn4)CC23)ncccc1=O c1(C(N(CCCOCCN(C(=O)C(O)C2CC2)C)C)=O)ncc(C#N)cc1Cl Cc1csc(C(=O)NC(C2CCCN2C(=O)CCc2ncc[nH]2)C)c1Cl CC(C)CC(F)C(=O)N1CC(CNC(c2nc(=O)n(C)[nH]2)=O)C1 c1(C(N2CCCC(NC(CCC)=O)(CC)C2)=O)nc2ncc(C)cn2n1 c1(-c2ccc(NC(c3cc(Cl)nc(Cl)c3)=O)nc2)cnn2ccccc12 c1(C(F)(F)F)cc(N2CCN(c3nc4cccnc4s3)CC2)n2ncnc2n1 C12(CNC(c3c(CC)occ3)=O)CC1CN(C(c1nccnc1C(F)(F)F)=O)C2 S(=O)(=O)(c1ccc(C)cc1)NC(C(N1CC(COC)C(C(F)(F)F)C1)=O)C C(C1Cc2ccccc21)NC(c1c(CNC(c2c(C)ccc(C)n2)=O)ccs1)=O Cn1cc2c(n1)CC(C(N1CCC(C)(NC(=O)CN3CC(=O)NC3=O)C1)=O)CC2 C1(C(N2CCCSCC2C)C(=O)NCCCOC)CCS(=O)(=O)CC1 c1(C(N(C2C(NC(CCOCCOC)=O)CCCC2)C)=O)csc2ccccc12 N1(C(C(C)SCC)=O)CCC(C)N(C(c2cccc(OC(F)(F)F)c2)=O)CC1 CC1(C)CN(C(=O)Cc2ccc(F)cc2)CCN1C(C1Cc2ccncc2C1)=O c1(C(=O)NCC(CNC(C(CC)(C)C#N)=O)O)cc2c(F)c(F)c(F)cc2[nH]1 C#CC1CCC(CNC(=O)CCN(C)C(C2CCCC(C)(C)C2)=O)CC1 N1(C(CC(CC)C2CC2)=O)CCCN(C(=O)C=Cc2cn[nH]c2)CC1C(C)C C(=O)(C1=COCCC1)NC1(C)CC(NC(=O)CC2CCC(=O)O2)C1 C12(CNC(c3c(OCCC)cccn3)=O)CCC1CCN2C(=O)CCCSC N1(C(CC(=O)NCCC)=O)CC(c2cccc(C(F)(F)F)c2)OCC1(C)C Cc1cc(Br)cc2c(COC(C3CN(S(=O)(=O)C4CC4)C3)=O)ccnc12 c1(C(N(CCCNC(c2[nH]c(C)nc2C)=O)CC)C)nc2ccccc2s1 N1(C(C(C)=CC)=O)CC2CCN(C(c3sc(Br)cc3F)=O)C2C1 c1(C(=O)NC2CC(N(C(=O)CN3CCCC3=O)C)C2)c[nH]c(=O)c2ccnn12 CC(CN=C(NCC1CCC1)NC1CCCC1)Oc1ccccc1Br CC1CCN(C(=O)Nc2nccnc2N)CC1N1CCOCC1 C(CC(=O)N(C(C)C)CC1CC1)SCCCC.N1(C)CCOCC1 C(=O)(C1CCCc2scnc21)N1CCC(NC(=O)CC2CCOCC2)C12CCC2 CCCC(C(=O)NC(C)(C)CC(N)=O)NC(=O)CCc1nccs1 C1(CNC(C(C)OCCOC)=O)CN(C(c2cnc(Cl)cc2Cl)=O)CCC1(C)C c1(N2CC(C(=O)NC(c3ccc(C(F)(F)F)nc3)C(C)C)C2)ncc(Br)cn1 C1(COC)(NC(=O)CSC)CCN(C(c2ccc(OC)cc2)=O)CC1 C1(Cn2cc(CC(C)O)nn2)C(C2CC2)CCN1C(C1(CO)CCCCO1)=O.CO N1(C(C(n2cc(-c3c(Cl)ccc(OC)c3)nn2)C)=O)CCC(O)C(C)(C)C1 C(CC)(CCCC(=O)N1CC(O)CC(C)(C)C1)NC(CC(CC)C1CCC1)=O N1(C(=O)OC(C)(C)C)CC(NCC(c2cnc[nH]2)O)OCC12CCC2 Cc1cncc(C(=O)N(C(C)CNC(C2CCCCC2)=O)C)c1Cl N1(C(CNC(c2ccccc2)C)=O)CC2(N)CC1C2 N1(C(=O)CSc2ccccn2)CC(F)(F)CC1CC(N1CC(C2CC2)C1)=O c1(-n2cc(C(C)NC(=O)C(c3ccn(C)c3)C)nn2)cc(F)cc(F)c1 N1(C(COCC#C)=O)CC(NC(=O)Cc2ccc(Cl)cc2)CC(C)C1 C1(C(=O)NCC(CO)NC(C2CSC2)=O)Cc2ccccc2S1(=O)=O C(=O)(C1=NOC2COCC12)NCCC(C(=O)NC1C(C)(C)CCC1)O Cc1cc(C)c(C(N2CCC(OCCNC(c3cc(Cl)ccc3F)=O)C2)=O)cn1 c1(C(N(CCC)CCNC(=O)C(F)C(C)(C)O)=O)c[nH]c2cc(F)ccc12 Cc1cc(CC(=O)NCC2CCN2C(c2cn(C3CC3)cn2)=O)on1 c1(NC(c2ccc(-c3c(C(=O)NC)cccc3)nc2C)=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(CC=C)=O)CC2(CCN(C(=O)CN(CCO)CCO)CC2)c2ccccc21 C(=O)(C(C)(C)c1cccs1)NC1CC(CNC(CC2(CN(C)C)CCC2)=O)C1 CC(C)C(F)C(=O)NC1CN(CC2CC2NC(c2ccccc2N(C)C)=O)C1 N1(C(c2cccc(Cl)c2Cl)=O)CCCN(C(C23CC(F)(C2)C3)=O)CC1CO N1(C(C2CC(CC)NC(=O)C2)=O)CC2CCC(C1)N2C(C1NC(=O)OC1C)=O c1(CC(N2C(CNC(c3cnc(CO)cn3)=O)CCC2)=O)ccc2c(c1)CCC2 N1(C(C)=O)CCCC1CC(=O)N(C)CCN(C(=O)CCn1ccnc1C(C)C)C c1(CC)c(C(=O)NCC2(NC(C3CC3C#N)=O)CCC2)sc2ccccc12 C#CCCCCCC(=O)NC1(C2CC(NC(=O)CCNC(=O)C(C)(C)C)C2)CC1 c1(C(=O)NC2C(NC(=O)CCc3cccs3)C2)ccc(-c2ccccn2)nc1O C1(C(=O)NC2CN(C(c3c(C)cn(C)c3)=O)C2)CC2CCCCN2C1 C(C(CC1CC1)C(=O)NCCc1ccns1)NC(c1cc(C)sn1)=O C(N(C)N1CCC2(CC1)OCCCC2CO)c1ccc(OC)c(Br)c1 C(CCCNC(C1(CNC(=O)C(C)OC(C)=O)CC1)=O)OC Cc1ccncc1C(C)(C)C(N1CC(C)(NC(C2COCCO2)=O)C1)=O C1(NC(c2sccc2F)=O)CCC2CCN(C(=O)Cc3ccccc3[N+](=O)[O-])C12 C1(CNC(C(Br)=C(C)C)=O)CCC2(CN(C(C3OCC3(C)C)=O)C2)O1 O=C1CCCC(C(=O)NCC2(O)CCN(C(c3cnc(-c4cccs4)o3)=O)C2)O1 C(=O)(C1CS(=O)(=O)c2ccccc21)N(CCNC(C(CSC)O)=O)CC1CC1 CC1CCn2ncc(C(=O)NCC(C3CC3)NC(C3(C4CC4)CCC3)=O)c2C1 N1(C(c2scc(C)c2Cl)=O)CCC(C)(CNC(=O)CN2CC3CCC2C3)CC1 C1(C(N(C)CCN(C)C2CC2)=O)(NC(=O)CC2CC2(C)C)CCCCC1 c1(C(=O)NC2(CC)CN(C(C3C(OCC)C3)=O)C2)cc(F)cc([N+](=O)[O-])c1 C1(NC(=O)CSC2(CC(=O)Nc3cccs3)CCC2)CC2CC2C1 C1(=O)C(Cc2ccsc2)N1.C(=O)(CN(CC(C)O)C)NCCNC(=O)OC C12(C(=O)NCCCN(C(=O)C(C)CC3CCCCC3)C(C)C)CCCC(C1)OC2 c1(C(c2ccccc2)Cc2onc(C(n3c(C)ncc3)C)n2)cncc(Br)c1 C1(NC(C(N2C(c3cc(C)c(F)cc3)CCC2)=O)=O)CCCCCC1(F)F c1(C(=O)NC2CCCC(NC(CC3(C)CCCO3)=O)C2)cn2cnnc2cn1 CC1CCCC(C(=O)NCC(F)(F)Cn2cc(-c3cnccc3C(=O)O)nn2)C1 c1(C(=O)NC(CCOC)CNC(C2(C)CCOC2)=O)cn(C)ccc1=O c1(CN2CCCC(NC(c3ccc(Cl)cn3)=O)CC2)c(F)cc(O)cc1F C1(C(=O)NC2C=CC(CNC(CCc3c(C)ncs3)=O)C2)CC2(CCC2O)C1 C1(C)(CCNC(C=C(C)C(F)F)=O)CCN(C(=O)CC(C)C2CCCCC2)C1 C12(C(=O)NCC3(F)CCN(C(CCC#N)=O)C3)CC=CCN1CCC2 c1(N(C(=O)C=Cc2cocn2)CC2CCCC2)cc(O)ccc1Cl C1(CNC(c2cc(Cl)cc(Cl)c2)=O)C2CCC(C2)N1C(c1n[nH]cc1Cl)=O c1(NC(c2c(-c3nnc(COC)o3)cccc2)=O)cncc(S(C)(=N)=O)n1 N1(C(CCC(=O)NCCC)=O)CCOC(C)C1C(=O)Nc1ccc(F)nc1 c1(C(N(C(C(CCC)C(C)C)=O)CC(=O)OC)=O)cc2c(C)cccc2[nH]1 N1(C(c2ccn3c(O)nnc3c2)=O)CCC2(CC1)CCN(c1cnc(F)cn1)C2 c1(C2(CNC(c3n(CC(=C)C)nnn3)CCOC(C)C)CC2)ccccc1C c1(CN2CCC(C)(NC(C(C(C)O)C)=O)CC2)cc(Br)c(F)cc1[N+](=O)[O-] C1(CC)CCN(C(=O)C=C2CCOCC2)C1CNC(=O)C(C)Cn1cccc1C N1(C(c2cc(=O)c(OC)co2)C(=O)NCC)CCC2(CCCCC2)C1C c1(CC)ccc(F)cc1C(=O)N(CCN(C)C(c1cc(C(C)C)on1)=O)C(C)C c1(C(=O)NC2C(NC(Cc3cc(C)sc3)=O)C2)ccc(OCC(F)(F)F)cc1 c1(C(=O)NCC2N(C(C(C)O)=O)CCC(C)C2)coc2cc(O)ccc12 C1(C(N2CCCC(C(C)C(=O)NCC3(O)CCC3)C2)=O)(OC)CCOCC1 N1(C(CC(C=C)C)=O)CCC2CN(C(c3scnc3COC)=O)CCC12 C1(C(=O)NC(c2n(C)cnn2)CO)CCCN1NC(=O)C12CC(F)(C1)C2 C1(C(c2n(CCC)nnn2)NCc2cc(Br)cs2)OCCOC1(C)C N1(C(C(C)O)=O)CCC2(CCC(C(N3CCOCC3)=O)O2)CC1 N1(C(c2cc(C(=O)OCC)no2)=O)CCC2CCN(C(c3csc(Cl)n3)=O)C2C1 CCC(CC)CCCN(C)C(C1CC(C)N1C(=O)CN(C1CCC1)C)=O C1(O)(CCNC(c2c(COC)ccs2)=O)CCN(C(c2csnc2C)=O)CC1 C#Cc1cnn(C)c1C(=O)NC1CCOCC1NC(=O)C(C)Oc1ccccc1 N1(C(C2ON=C(C)C2)=O)C2CCC1CN(C(=O)C(c1cccn1C)=O)C2 c1(OC)cnc(C(N2CCCC2(C)CNC(=O)Cc2sccc2C)=O)cn1 C1(OC)CC2(CCC(C(=O)NCC3C4CN(C(=O)CC5(O)CCC5)CC34)CC2)C1 C1(CNC(C(C2CCOCC2)C)=O)CCCCC1NC(=O)CCc1n[nH]c(=N)s1 C1(C(=O)NCC2(NC(c3c(F)ccc(OC)c3)=O)CC2)CCC2C(C1)C2(F)F C1(CNC(C)CN)COC2COCC12.c1(CC(=O)C=O)cccc(OC(F)F)c1 c1(C(N2CCCC(CN(C(c3c(CC)cco3)=O)C)C2)=O)cc(C)c(F)cc1O C(=O)(C(CC(=C)C)OC)NC(CNC(C(C=C=C)C)=O)CCOC C#CCCCCCCNC(C1CC=CC(NC(=O)CCOCC)C1)=O Cc1cnc(NC(C2CCCN(Cc3cnc(Cl)cc3Cl)C2)=O)c(C)c1 c1(CC(=O)NC2C(NC(CC(=O)NC3CC3)=O)CC2)ccnc(F)c1F C12(CCC1)C(=O)OC2.C(=O)(C(C)O)NC C(=O)(CC(CC)CCCC)NC(CC(=O)NCC(CCCC)O)COC c1(C(=O)NC2C(NC(C3(N(C)C)CCCC3)=O)CCC2)cccc2nc(C)[nH]c12 CCC(C)C(C(=O)NCc1ccc(C(=O)N(C)CCc2ccccn2)s1)N(C)C C1(N(CCCC(=O)NCC(CC(F)(F)F)NC(C)=O)C)CCCC(C)(C)C1 C1(C(=O)NCC(C(C)C)(C)NC(=O)C(=C2CCCCC2)F)CN2CCN1C(C)C2 C1(CC2CC2)CCCCN(C(=O)CC2(Cc3ccccc3)CC2)C1.O=C1CCN1C c1(NCC(=O)NCC(CNC(C(C=C)(C)C)=O)OC)ccc([N+](=O)[O-])c(SC)c1 CC1CCCC=C1C(=O)NC(c1cnn(C)c1)C(=O)N1CC(N2CCC2)C1 c1(-c2cn(CCCN(C(C3(C(N)=O)CC3)=O)C3CC3)nn2)ncc(Cl)cc1F C#CC1CC2(CC(C(=O)NC3CCN(C(=O)CCOCCN(C)C)C3(C)C)C2)C1 C1(NC(C(CC#C)O)=O)CN(C(=O)Cn2cc(C)cn2)CC12CCC2 N1(C(CCC(C)(C)C)=O)CCN(C(=O)CCc2nc3cccnc3[nH]2)CC(O)C1 C(=O)(C1CCCc2nc[nH]c21)NCC(C)N(C(=O)CC1CCCO1)C c1(N(CC(C)NC(COCC)=O)C(=O)C=CCOC)ccccc1 C1(COC)CCN2C1C2=O.C1(C(=O)NCC(F)F)CN(C(N)=O)C1 C1(OC)CCCCC1C(N1CC(=C(F)CNC(c2ncsc2C2CC2)=O)C1)=O O=C(N=c1ccnc(N2CCCC2)[nH]1)C1CC1C(=O)Nc1cc(Br)c(O)cc1Br C(=O)(C(CC(C)(C)C)NC(=O)CC1CCN(C)C1=O)NCCC=C=C N(C1CCC(Nc2ncncc2Cl)c2ccccc21)C(C(F)=CCC)=O c1(COC(C)C)cccc(SC2(c3nnnn3C)CC(C(C)C)C2)c1 CC1(NC(=O)CC2CCCOCC2)CCN(C(c2ccoc2)=O)C1 C=CCCCC(C(=O)NCC(C)C(F)(F)F)NC(=O)C=CC Cc1cc2sc(C(=O)NCCCCCCNC(c3cnc(O)c(F)c3)=O)cc2s1 N1(C(C2C(C(=O)OCC)C2)=O)CCC2CCN(C(C3CC(=O)N(OC)C3)=O)CC12 C(=O)(CCCC(=O)NCC1(C)CCN(C(=O)Cc2ccc(C)c(Cl)c2)C1)NCC N1(C(C2(CC#C)CCCCC2)=O)CC2CCCN(C(=O)CCc3nncs3)C2C1 C1(C(=O)O)CCC(C(=O)O)N(C(c2ccccc2NCC2CC2)=O)C1 c1(CC(C(=O)NCC2CC(NC(c3cnc(C)[nH]3)=O)C2)C)cccc(Cl)c1 C1(NC(CCOCCC)=O)CCC(NC(C2(CC3CC3)CC2)=O)CC1 CC(=O)C(C)CC(C)C(=O)NC(c1cccnc1)C(=O)NCC(O)C(C)O c1(OC)noc(C)c1C(=O)NC1CC(CCNC(C2CNC(=O)O2)=O)C1 O=[N+]([O-])c1cccc(N2CCCC(NCCCN3CCOC3=O)CC2)c1 C1(C(=O)OC)CN(C(C)=O)CC1C(F)F.C1(C2CC2)CCCCN1C(=O)C=CCF C1(NC(CCNS(CC)(=O)=O)=O)CCCN(C(=O)CCc2cnccn2)CC1 c1(-c2nc(C)on2)ccc(NC2CCCN(S(=O)(=O)Cc3ccccc3)C2)cc1 C(CNC(=O)Cc1nccn1C)(CC(=O)N(C)OCCC1CC1)OC C(CCCCC(=O)NC1CCCCC1CO)N(C(C1CCC(CC)O1)=O)C c12cccc(n1)S2.C1(CNC(C=CC)=O)C(C)CCN1C(=O)CC1CC(C)(C)C1 C1(C)(SC)CN(C(C2COCC2NC(=O)CNc2ccncc2)=O)C1 C1(NC(C2(CC=C)CC2)=O)CCN(C(=O)C(c2ccc(C)o2)C)C1C1CC1 CCCCC(CC(=O)N(C)C(c1ncccn1)C)NC(=O)C(C)CC N1(C(CN2C(C)CC2)=O)CCC2(CC1)OCCC2NC(=O)Cn1cccn1 C1(C(=O)NC2CC(CNC(C(C(COC)C)C)=O)C2)CCC2CC(C)CN2C1 CC(C1=Cc2ccccc2OC1)NCCc1c[nH]c2cc(F)c(F)cc12 N1(C(CC(CC)O)=O)CC2(C1)CN(C(c1cncc(O)c1)=O)C2 C1(C(F)(F)F)(C(N2CCN(Cc3c(OC)cccc3)CC2)=O)CC2CCC1C2 C(=O)(C(CC)CC(C)C)NCCC(C)(C)NC(c1c(CC)ocn1)=O C1(C(N2CCCC(NC(=O)CS(=O)(=O)NC3CC3)C2)=O)CCC2(CCC2)C1 N1(S(=O)(=O)CCn2nccn2)CC2(CCC2)C1C1CCCO1 CCC(CC(=O)NCC1(C#N)CCC1)NC(C1CC(N(C)C)C1)=O C1(C)(C(c2n(C(CC)(C)C)nnn2)NCC2(CC3CC3)CC2)CC2(C1)OCCO2 N1(C(C2C(C(C)NC(C(CC)N(C)C)=O)C2)=O)CC(F)(F)C1C1CC1 C1(C(=O)OC)CC2CCC(C1)N2C(C1C2CCC(F)(F)C12)C(=O)NCCSC Cc1ccc(C)c(C(=O)NCC(C)(O)CNC(C2CCCC2C(F)(F)F)=O)c1N Cn1nnc2c1CC(C(=O)NCC1(N(C(c3ncc(Cl)s3)=O)C3CC3)CC1)CC2 c1(C(N(C2CN(C(=O)Cn3nccn3)CC2F)C)=O)ccc(Cl)c2ncccc12 C#Cc1ccnc(C(=O)NC(C2CCN(C(=O)Cc3ccc(C)cc3Cl)C2)C)c1 N1(C(C2(CC#C)CC2)=O)CCC(N(C(=O)CCSC(C)C(C)CC)CC)CC1 C1(CCC)CCCN1C(=O)C=CCC(C)(C)NC(=O)C(O)C1CCC1 C(CCCC(C)NC(=O)C(C)N(C)C)OC(CCCC)=O.C1(=O)CC(C)CN1 C1(NC(C(n2cc(Cl)cn2)C)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C(C)C1 C12(CCNC(c3c(CC)cno3)=O)CCC(CC1)N(C(C1(C)CCNC1=O)=O)C2 Cc1c(-c2cc(C(=O)NCC(O)CNc3ccncn3)no2)cnn1C CCC(C)C(O)C(=O)N1CC(O)(C(C)NC(=O)Cc2c[nH]ccc2=O)C1 C1(C(=O)NCCC2COCC2O)CCOCCN1C(=O)CCN1CCOCC1=O C(=O)(C1Cc2ccc(Cl)cc21)N1CCCC(NC(c2c(C)nc(O)[nH]2)=O)CC1 N1(C(C2C(CC(C)C)C2)=O)CCC2(CC2NC(=O)CC2CC(F)(F)C2)C1 CCC(C(=O)NCC1(CNC(=O)COC(C)C)CC12CCC2)C(C)(C)CC c1(C(=O)NCC2(F)CC(NC(C(COC)(C)C)=O)C2)ccc(C)cc1Cl C1(CCC=C)(C(=O)NCC(C)(C)C)CN(C(C2CCC3CC23)=O)C1 C(=O)(C1=NOC2COCC12)NC(CC(C(N1CCC2C(O)C(C)(C)C12)=O)NC)=O c1(NC(=O)Cn2cc(CNc3ccc(C(=O)O)cc3)nn2)cccc([N+](=O)[O-])c1 N1(C(c2c(CNC(c3ccc4c(c3)CCC4)=O)cco2)=O)CCCc2ccccc21 c1(CN(C(=O)CCCN(CCN(C)C)CC)CC=C)cc(Cl)ccc1C(=O)OC C=CC1(C2(C(N3CC4CC3CN4C(=O)CCCSCCC#N)=O)CCC2)CCC1 C(=O)(C(C)(C)C(C)NC(C1CC2(CC2)CO1)=O)NCc1ccc(CC)s1 c1(C(=O)NCC(N(C(CC=C)=O)C)C2CC2)ccc(S(=O)(=O)NCC)cc1 CCCC(O)CC(=O)NC1CCCCCC1NC(c1cccc(C2CC2)n1)=O c1(C(N2CCN(C(C3CCCS3)=O)CC2CF)=O)ccc2c(n1)CCC2 c1(N2CCC(c3sc(C(=O)OC)c(C)n3)CC2)ccccc1S(=O)CC(O)CC C1(NC(C2CCC(=O)NC2)=O)CCC2CC1CN2C(=O)Cc1cc(F)ccc1F C(=O)(CC(C)CC)N1CCC(OCCNC(C=CCCC)=O)C1 C12CCC13CCN(CC3)CCN2C.N1(C(CNC(C)(C)C)C)CCCC1 c1(N(CCCF)C)nc(=NCC(=O)NCc2ccccn2)[nH]c2ccc(Cl)cc12 C12(NC(C(C(C)(C)C)NC(c3cc(C)oc3)=O)=O)CCC(CC1)C2(C)C c1(C(N2CCN(CCN(C(CCCC)=O)C)CC2)=O)[nH]c2c(c1C)C(=O)CCC2 c1(OCC)cccc(CCC(=O)N(C(C)CCNC(=O)C2=COCC2)C)c1 N1(CCCCNC(c2cnc(C)o2)=O)CCCN(C(C2(C)CC(C)(C)C2)=O)CC1 C1(NC(C2CC=C(C)CC2)=O)CN(C(c2ccc([N+](=O)[O-])cn2)=O)CCC1(C)C N1(C(C(CC#C)O)=O)CCN(C(c2cccn2CC)=O)C(c2cccc(F)c2)C1 C1(CC(=O)NCC(=O)NCCC(N)=O)CCC2CC12 c1(C(=O)NC(C)C(=O)NC2CCC2NC(c2ccc(C(F)F)o2)=O)sccc1Cl C1(CC(=O)NCC2(C(=O)NC(C3CCCC3)C)CC2)CC2(CC2)C1 c1(N(c2nc(N(C(=O)C#CC(=O)N(C3CCOC3)C)C)cs2)C)ccccc1F CN1CC(NC(=O)COC2CN(C(=O)CN3CCC(=O)CC3)C2)CC1CO O=C(CC1C(=O)Nc2ccccc21)NCC(F)CNC(c1ccsc1)=O c1(CNCC2CCN(C(C(C)C)=O)C2)cccc2cccc(O)c12 N1(C(c2ccc3nccnc3n2)=O)CCC2(CCCN(C(=O)C3CC3)C2)C1 N1(Cc2cccc(C(=O)OCC)c2)CC2(CCN(C(C3CCCN3C=O)=O)C2)C1 C(=O)(CS(=O)(=O)CCO)N(CCC(C)NC(C1(CC)CCCC1O)=O)C c1(-c2c(C)cc(OC(C)C)cc2)c[nH]c2cc(NCC3COCCO3)ccc12 N1(C(CC(C)c2ccncc2)=O)CCC(NC(=O)CC2OCCC2(C)C)C(O)C1 c1(C(N(CC(C)NC(C2CC(CC)OCC2)=O)C)=O)cn(C)c(C)cc1=O N1(C(c2nncn2C)C(=O)NCCCOC)CC2CC(C)C2C1 CCCCC(O)C(C)C(=O)N1CC(CNC(c2ccc(CC)nc2C)=O)C1 N1(C(CSCCCC)=O)CC2CCCC2C1C(N1CCOC(C(C)(C)C)C1)=O C1(CCC)CCC(C(=O)NCC2(F)CCN(C(=O)Cn3cc(C)cn3)C2)CC1 Cc1[nH]c(C#N)cc1C(=O)NC(CO)C(=O)NCC1CCN(C(C)C)CC1 N1(C(c2ccc(C)cc2)=O)Cc2[nH]nc(-c3ccc(-c4nn[nH]n4)cc3F)c2C1 N1(C(c2cc(CC)ncc2)=O)CCN(C(c2ccsn2)=O)C(C2CC2)C1 N1(C(CCC=CCC=C)=O)CCN(C(c2nnc(C)s2)=O)C(C)CC1C CCCCC(O)C(C)C(=O)N1CC(C(N2CCCC2CC)=O)(CO)C1 c1(CC(N2CCN(C(CC=CCC)=O)C(COC)C2)=O)cccc(S(C)(=O)=O)c1 C1(C(C)C)N(C(=O)CCOC2CNC2)CC12CCS(=O)(=O)CC2 C1(C(N2CCC(N(CCC)C(C3CC(OC)(OC)C3)=O)C2)=O)NC(=O)NC1=O N1(C(c2c(C)cc[nH]c2=N)=O)CCN(C(=O)CSC2CCOC2=O)C2(CCC2)C1 Cn1nc(C(N2CCC(CNC(=O)CC(C)(C)O)C2)=O)c(Cl)c1Cl C(C(C)(O)CC(=O)NCC1CC2(CC(NC(=O)C(C)SC(C)C)C2)C1)OC c1(C(=O)NC2CCC(CNC(COCCSC)=O)C2)cccc(SC)c1 c1(CN2C(CC(=O)Nc3c(C)cc(Cl)nc3)COCC2)cc(F)c(C)c(Br)c1 n1(CCNC(C2N(C(=O)OC(C)(C)C)CCC2)=O)cc(C(N)=O)c2ccccc12 C1(CCO)(C(C2CCCO2)=O)CN(C(C23CC(C)C2C3)=O)C1.CCC(C)(C)OCC=O N1(C(c2sccc2I)C(=O)NCCCSC)CCC(O)CC(C)(C)C1 CCCCCC(C(=O)N1CCCC1CCCNC(C1CCC(F)(F)C1)=O)C(C)C C(=O)(C(CC(C)C)NCCCC(C)N(C(C=CC)=O)C)NC1CCOCC1 CC1CC(CNC(=O)C2=CCOCC2)CCN1C(=O)CSc1nncn1C c1(OC)ccc(F)cc1-c1csc(NC(=O)Cn2cc(CCC(=O)O)nn2)n1 C(CC1=CCOCC1)NC(COCC)(C(C)C)c1nnnn1C1COC1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC2CC(NC(C=CCCC)=O)C2C1 C1(O)(CNC(c2cncc(N(C)C)c2)=O)CCCN(C(C2CCCNC2=O)=O)C1 c1(C(N2CCC(NC(c3cn(CC)nn3)=O)C2)=O)cccc[n+]1[O-] N1(C(CC(C(=C)C)C)=O)CCC2(CCC2NC(c2ncc(F)cn2)=O)CC1 C(=O)(N=c1cc(CC)n(C)[nH]1)C1CCN(C(c2cnc(CC)o2)=O)C1C(C)C c1(C(N2C(C)C(NC(c3ccc(F)cc3)=O)CCC2)=O)cccc(S(N)(=O)=O)c1 N1(C(C=C(C)C(C)C)=O)CCOC2(CCN(C(=O)C=Cc3cc[nH]c3)CC2)C1 c1(C(C)=O)ccc(CC(=O)NC2CCOCC2(C)C)c(Cl)c1 N1(C(N(C)C)=O)CCN(CCCNC(=O)Nc2cc(C(N)=O)cn2C)CC1 c1(NC(CC(CC)C(C)C)=O)ccc(Cl)c2cc(Br)ccc12 c1(NC2CCC(NS(=O)(=O)CC3CC3)C2)ncc2[nH]cc(I)c2n1 C=Cc1cc(C(=O)NCC2CCCCCN2C(=O)Cc2ccc(C)s2)cc(F)c1 n1(CC)ccc(C(=O)NC(C2CN(C(C3CCC(=O)N3C3CC3)=O)C2)C)cc1=O c1(C(=O)NCC2N(C(C(CC)NC(C)=O)=O)CCCC2)n[nH]c2ccc(C)cc12 N(C1CCC(NC(c2ccsc2Cl)=O)c2ccccc21)C(c1c(C)cncn1)=O S(=O)(=O)(CCCOc1ccc(C(F)(F)F)cc1)NC(C)C(C)(C)c1ccccc1 CCC(C)C(O)C(C)C(=O)N1CCCCC1CNC(=O)C(C)(C#N)CC c1(-n2cc(CCC(=O)NC3(C(=O)O)CC(C(=O)OC)C3)nn2)cccc(Br)c1 C1(NC(CNC(=O)NC)=O)CCN(C(=O)CC2CCCC23CC3)C1(C)C N1(C(C(OC)OC)=O)CCCC1(C)CNC(=O)CCCn1cc(C)cn1 Cn1nnc(C(N2CC(NC(=O)CC3CC4(CCC4)C3)C(F)C2)=O)c1C(F)(F)F c1(C(=O)NCC2C(NC(C(C)n3cncn3)=O)COC2)ccc2c(c1)OCC2 Cn1nccc1CC(C(=O)N1CCC(CN2CCCC2)C1)NC(c1cn[nH]c1)=O c1(C(=O)NCC2N(C(C(C=C)(C)CCOC)=O)CC2)cc(S(N)(=O)=O)c(C)s1 c1(COC)ccc(C(=O)NC2CCCC2NC(=O)CCN(S(C)(=O)=O)C)s1 c1(C(N(C2CCN(C(=O)CCCC)CC2)CCCC)=O)ccc(F)c(OC)c1 N1(C(COc2ccc(OC)cc2)=O)CCCC(NC(=O)CCCCSC)C(F)C1 c1(C(N(C(C)(C)C)CC(=O)OC(C)(C)C)=O)ccn(C2CCNCC2)n1 C1(CC)CN(C(=O)CNC(=O)Cn2cc(C)cn2)CCN1C(=O)Cc1ccno1 C=CC(C(F)(F)F)NC(=O)CC1(CNC(=O)CC2CSC2)CC1 Cn1ccc(CCNC(C2(CCNC(=O)CCc3ccccn3)CC2)=O)n1 CC(C)(C)C1=NOC(C)(C(=O)NC(c2ccccc2)CNC(=O)CC2CCC2)C1 c1(NC(CC2CCCN(C(C(C)(C)Br)=O)C2)=O)nc2cc(Cl)ccc2s1 C1(NC(CCC(CC)C)=O)COC2CN(C(=O)CCc3ccnc(C)n3)CC12 C1(C(N(CCC(N)=O)C)=O)COCCN(CC(O)Cc2ccccc2)C1 CCCCCC(O)CC(=O)N(C)CCNC(c1cccc(C(F)F)n1)=O c1(C(=O)NCCC2(C(N(C)CCC3CCCO3)=O)CC2)cccc(C#N)c1 C(CCC(C)(C)C(=O)NCC(O)CC(=O)N(CC(F)F)CCO)OC C1(NC(c2cn(C)nn2)=O)CN(C(C2CCC2(C)C)=O)CCC12CCC2 c1(OCCOC)ccccc1C(=O)NC(CO)C(C)NC(c1[nH]cnc1C)=O C1(C(=O)NCCCOCCC(=O)Nc2ccnc(C)n2)CC(=O)NC(=O)N1 c1(OC)ccc(C(N2CC(NC(=O)COCCCC(C)C)C3(CC3)C2)=O)c(C)n1 c1(C(N2CCN(CCNC(CS(CC)(=O)=O)=O)CC2)=O)cnn2cccc(C)c12 c1(OC)cc(C(=O)N(CCNC(=O)C(C)NC(C)=O)C(C)C)cc2cnn(C)c12 C1(NC(c2ccccc2S)=O)COC2(CCN(C(=O)CN3CCOCC3)CC2)C1 C1(OC)CC2(C1)CC(C(N1CCC1CNC(C1(F)CCOC1)=O)=O)C2 CN1CCCC1(C)C(=O)NCCCc1cn(C(C)(C)C)nn1 N1(C(C(COC(C)C)NC(=O)CN2CCC(=O)CC2)=O)CCC12CC(C)(CO)C2 C1(CNC(=O)C=Cc2ccccc2)CC2(CCN(C(c3csc(Cl)n3)=O)C2)CO1 c1(C(N2CCC(N(C(C34CC(C)(C3)C4)=O)CC)C2)=O)ccc2c(c1)C(=O)CCC2 C1(C(c2nnnn2CCCC2CC2)NCC(F)F)(CF)CC(F)(F)C1 Nc1ncc(NC(C2CCN(C(=O)CC3CC3)C2)=O)cc1CC1CC1.CO C1(CC(=O)NC2CCC(SC)C2)CC2(C1)CN(C(C1C3CCC(C3)C1C)=O)C2 C12CCCCN1CC(=O)N2.N1(C(=O)OC)CCNC(=O)C1 c1(NC(C2N(C(Cc3c(C(=O)OC)cccc3)=O)CC2)=O)cccc(Br)c1C C=CCC(CNC(C1(C2CCCN2C(=O)C(C)C)CCC1)=O)CC(C)C C#Cc1cccc(C(N2CCCCCC2CNC(=O)CCC(C)(C)C)=O)c1Cl C1(CCCCNC(Cc2c(C)n[nH]c2)=O)CCCN(C(c2csc(=N)[nH]2)=O)C1 N1(C(CC2C(=O)NC(=N)S2)=O)CCCN(C(=O)CCCn2cccc2)CC1 C1(CC)CN(C)CCCN1C(C1(C2CC2)CN(C(=O)C(C(C)C)SC)C1)=O c1(NC(C2C(C)N(C(=O)CC3CCOC3=O)CC2)=O)ccc2c(c1)CCC2 c1(C(=O)NCCCNC(C23CC(C(C)C)(OC2)C3)=O)ccc(Cl)c(O)c1 C(=O)(CC1=CCCCC1)NC(C)CN(C(=O)C(c1cccnc1)O)C c1(C(=O)NC(C2N(C(c3c(C)noc3)=O)CCC2)C)cc(P(C)(C)=O)ccn1 C1(NC(=O)NCc2nc(C)sc2)CC(C)(C)C12CC2 N1(C(CN(C(=O)C(C)(C)C2(O)CCOC2)C(C)C)=O)CCc2sccc2C1.CCCl C1(CNC(=O)NC2CCCN(Cc3ccccc3)C2)CC2CCCCC2C1 C1(C=O)(CC)CCCN(N2CCCC(OCC)C2)C1.c1(C=O)cccs1 CC1(NCCNC(=O)CCC2CC=CCC2)CC(C(F)(F)F)C1 c1(N2CCC(N(OC)C)CC2)nc(=NCCC(F)(F)C(C)C)[nH]c2cc[nH]c12 N1(C(C(CNC(=O)OC)(C)C)=O)CCC(C)C(NC(=O)C=CCOC(C)(C)C)C1 CC1(C)CCCN(C(c2cccs2)=O)C1C(N1CCC2(CC(F)C2)C1)=O C1(CNC(C2C(CN(C)C)C2)=O)(CO)CCN(C(c2ccnc(O)c2)=O)C1 CC(CC(N)=O)C(=O)NCC1CC(NC(=O)CSc2cccc(Br)c2)C1 c1(SC(C)C(=O)O)ccccc1C(=O)NCc1cc(-c2cccc(F)c2)on1 O=C(C(C(C1CC1)C1CC1)N(C1CC1)CC1CCC1)NC1CC1 O=C1CC(C(N2CCCC2CC2CCCCCC2)=O)CN1C1CC1.n1(N)ccnn1 CC1C(NC(=O)CC2(N3CCCC3)CC2)CCCN1C(=O)Cc1ccnc(F)c1 C(=O)(C1CCc2cccc(Cl)c21)NC1CC(NCc2ccc(OC)c(I)c2)C1 C(=O)(N=c1cc[nH]c(C(=O)OC)c1)c1c(N)nn(C)c1.CC1CCC(C(=O)CCO)O1 N1(C(CCC(=C)Br)=O)CC(C2CN(C(=O)CC(C)(C)F)C2)C1 C1(CC)C(NC(c2cscc2Cl)=O)CCN1C(C1CCCC1OC)=O C(=O)(C(C)CC(=O)N(C1CCN(C(C2CCC(=O)N2CC)=O)CC1)CC)OCC CCCS(=O)(=O)c1ccc(C(=O)NC2CN(C(c3cn(C4CC4)nn3)=O)C2)cc1 c1(CCNC(=O)Nc2nc(C(C)=O)c(C)s2)nc2ccccn2n1 n1(CC(N2CC(NC(C3CC4C=CC3C4)=O)C(O)C2)=O)ccc(O)nc1=O c1(CC)nnc2cc(NCC(C3CC3)NC(=O)CC3CCCCO3)ncn12 C1(N2C(CCN)N(CCOCC)C2=O)CC2CC(C1)CC(F)(F)C2 N1(C(c2[nH]c(=NC)sc2)=O)CCN(C(=O)CCCCCF)C(C)C1C C1(O)(C(C)NC(c2cnco2)=O)CCN(C(c2c(Br)noc2C2CC2)=O)C1 Cc1cc2sc(C(N3CCN(C(C4CC45CCCCCC5)=O)CC3)=O)cc2s1 CC1(NC(c2ccc(C(F)(F)F)s2)=O)CC(NC(=O)CC2CCC(O)C2)C1 C=CCC(CC)C(=O)NCCCCCCNC(C1CC1c1c(C)cccc1C)=O C1(C(N(C2CCC(NC(C(CC)(C)O)=O)CC2)C)=O)CCc2nncn2CC1 c1(C(=O)NC2C(NC(=O)CC3CCCO3)CC(F)(F)C2)[nH]cc2c1CCS2(=O)=O c1(C(=O)NCC2CCN2C(C23CCC(CC2)CC3)=O)ccnc2ccnn12 C(=O)(C(C)(C)CCS(C)(=O)=O)N1CCCN(C(CCCC(=C)C)=O)C(C)C1 C1(O)(CNC(C2CCO2)=O)CCN(C(=O)C(c2cc(Br)co2)=O)C1 c1(CC)oc(C(=O)NC(CCN(C)C(c2ccc(O)nn2)=O)C(C)C)cc1C C1(N(c2nc(C)c(C)s2)CCO)COC2(CCNCC2)C1 C(=O)(CCCC(C)(C)C(=O)OC)N1CCC(CCNC(C(CC)C(F)(F)F)=O)C1 N1(C(c2cnc(C(=O)OCC)s2)=O)CC2(C)CC1(C(=O)NCCCCN(C)C)C2 c1(NCc2n(C)ncc2Br)ccc(S(=O)(=O)N2CCC(C(N)=O)CC2)c(Cl)c1 Cc1cc(C(N2CC(O)(C(C)NC(=O)C(O)CCc3ccccc3)C2)=O)c(C)s1 c1(C(=O)NC2(CNC(C3C(CC)OCC3)=O)CCCC2)cc(N(C)C)nc(Cl)c1 C1(NC(c2c(CC)nc[nH]2)=O)CCC(C)N(Cc2ccccc2CC(C)C)C1 N1(C(C(CC)F)=O)CC(CO)C2(C1)CN(C(c1ccc(C(F)(F)F)[nH]1)=O)C2 c1(C(=O)NC2(C)CN(C(C3C(CCOC)C3)=O)C2)cccc(C2CC2)c1 C(=O)(CCCCC(C)(C)C)N1CCC(C)C1CNC(C1COC(C)C1)=O CCC(CNC(=O)CN1CCCNC1=O)(CC)C(=O)NC(c1nnc(C)s1)C C1(CNC(c2[nH]ccc(=N)n2)=O)CC(NC(c2ccsc2)=O)C12CCC2 c1(C(=O)NCC2(C)CC(NC(C(C)N(C)C)=O)C2)csc2c(F)cccc12 Cc1ccc(C(=O)C(=O)NC2CC(NC(C3CC3c3ncccc3F)=O)C2)cc1 C(=O)(C1=CCCCO1)NCC1CC(CNC(c2c(C)cns2)=O)C1 CC(C)C(CC(=O)N1CCC(F)(CNC(C2CC(C)C2)=O)C1)C(C)C C(N=c1cc[nH]c(-c2cccc(C(C)O)c2)c1)c1cc(C(=O)OC)c(OC)cc1 C1(NC(COC(C)C)=O)CN(C(=O)OC(C)(C)C)CC2CCCC12.C12CN(C1)C2=O C(=O)(C(C(C)(C)C)SC1CC1)NCCN(C(=O)Cc1cccc(NS(C)(=O)=O)c1)C C1(C(N2CCC(C)C2CNC(C2CN3CCC2CC3)=O)=O)SC2C=CC1CC2 C1(CNC(C=C2CCC(C)C2)=O)CCCCC1NC(C1CC=CC1)=O c1(C(N(CCNC(C2CCC(C)NC2=O)=O)CC)=O)c(C)nn(C)c1OC C=C(C)CC(=O)N1CC(CNC(c2ccc(C(C)C)s2)=O)(COC)C1 c1(CCC(=O)N(C2CCCN(C(C3CC(F)C3)=O)C2)C)ccc(Br)cc1 N1(C(C(C(C)C)SC)=O)CCCCC2C1CCCN2C(c1ccc(=O)n(C)n1)=O C(=O)(C(C(C)(C)O)NC(=O)Cc1c(C)cnn1C)NCc1ncc(C)nc1 Cc1noc(C)c1CC(=O)N(CC(C)(C)CNC(c1cccc(CCO)c1)=O)C c1(C(N2CCCC(C(=O)NC3C(CCC)C3)C2)=O)ccc(OC(C)C)cc1F c1(C(=O)NC2(CC=C)CCCN(C(c3cscn3)=O)C2)ccc(C)c(F)c1F c1(C(C(=O)NC)N(CCC(=O)ON2CCOCC2)C2CC2)cc(Cl)c(F)cc1F C1(C(=O)NC2C(C)CN(C(=O)CN3CCCCS3(=O)=O)C2)CCC2(CCC2)CC1 C1(NC(CCn2c(CCC)ncc2)=O)CCC(NC(=O)CC2COCCO2)CC1 C1(NC(=O)NCC(c2ccc(Cl)cc2)N(CC)CC)CCCC(N)C1 c1(NCC2(C)CCN(C(C3CC(N=[N+]=[N-])C3)=O)CC2)cc(=O)n(C)c(=O)n1C CCCCC(C)(F)C(=O)N1CCC(CO)(NC(=O)COCC2CCOC2)CC1 C#CCC(C(=O)NC1CC(C)OC1=O)NC(c1ccnn1CCC)=O N1(C(C(N2CCOCC2=O)C)=O)CC2(COC(CNC(=O)C=CBr)C2)C1 CC(CC(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)CC1CC1)CC2)c1ccco1 c1(C(=O)NCC(CN(C(=O)Cc2cncnc2)C(C)C)O)cc(C(F)(F)F)no1 c1(OC)cc(CC(N2CC(NC(c3coc(CO)c3)=O)C(C)C2)=O)ccc1Br C(=O)(CCC(C)(C)F)NC(C(C)C)CNC(C1CCS(=O)(=O)N1)=O N1(C(C(COC)(C)C)=O)CC2CC(NC(C3(C4CC4)CCCO3)=O)CC1C2 N1(C(C(c2ccc(CC)s2)=O)=O)CCC(C)C(NC(=O)Cn2cc[n+](C)c2)C1 Cc1cncc(F)c1C(=O)NC(C)CN(C(=O)Cc1ncoc1C)C CC1CN(C(C2(CC(C)(C)O)CCOC2)=O)CCN1C(c1cnc(C2CC2)[nH]1)=O c1(C(=O)NC2CCN(C(C(CC)O)=O)C2(C)C)sc2cccc(F)c2c1C C1(C)(C(=O)NC2CC(C)(CNC(=O)C(F)=CC3CC3)C2)CCNC(=O)C1 C1(C)(CC)C=C(C(=O)NC(C)(C)CNC(=O)CC2(COC)CCCC2)C1 c1(OC)ccc(CCNC(=O)NCC2(Br)CC2)c2ccccc12 N1(C(c2cccc(F)c2)C(=O)NCC)CCC(O)C(C)(O)C1 c1(OC)cc(C)c(C(=O)NC2COCC2CNC(C2CS(=O)(=O)C2)=O)c(C)c1 N1(C(C2(C#N)CC2)=O)CCC2(CCC2NC(c2ccc(Br)o2)=O)CC1 C(C(C)CCO)NC(C(C)NC(=O)NNC(C1(N(C)C)CCC1)=O)=O c1(C(=O)N(CCC2(CN=c3ccnc(Cl)[nH]3)CCC2)C2CC2)cc2c(s1)CCCCC2 c12cc(ccn1)C(C)(C)S2.C(=O)(CC(C)C)NC1C(NC(C)=O)C1 C1(CC(N2CC(C)C(NC(c3cnc(S)n3C)=O)C2)=O)Cc2cc(F)ccc2O1 c1(OCC(N2CCC(C(c3cn(C)nc3)=O)C2)=O)cccc(CN)c1 Cc1cnnc(C(=O)NCC2CCC(NC(=O)C(c3cccnc3)O)C2)c1 C12(NC(C(CCOC)(C)C)=O)CC(CO)(C1)OC21CCN(C(=O)CSSC)CC1 C1(O)(C(C(N2CC(N(C(C=CC(C)C)=O)CCO)C2)=O)F)CCCC1 C1(CC)CN(C(=O)C(C)(O)COC)CC1C(=O)Nc1cnc(F)nc1 C1(NC(CC2(CNC(C(C)C3CC3)=O)CC2)=O)CC2CCCCN2C1 c1(C(=O)NCC2(C)OCCN(C(CCCOCC)=O)C2)cnn2c1CC(C)CC2 C(CCS(N)(=O)=O)(C(=O)O)NC(C)CC(C(=O)Oc1cccc(C)c1)C CCCC(CNC(C1CCCC1)=O)C(=O)NC(c1ncnn1C)C N1(CC(=O)NCC(C(C)C)NC(c2n(C(C)C)ccn2)=O)CCS(=O)(=O)CC1 C(=O)(CCCCCN(C)C(c1cc(N(C)C)ccn1)=O)NC(C=C)C CC(CN=c1[nH]c(=NC(C)CCO)[nH]c2c1CCCC2)c1cccc(Cl)c1 c1(OC)ccc(SCC(=O)NC2CC2CNC(=O)C(C)CN(C)C)cc1 C1(C(=O)NCC2(CNC(C3(O)CCSC3)=O)CC2(F)F)CCCOCC1 C(C1CN(C(C2CC(CF)C2)=O)CC1C(N1CCOC(CC)C1)=O)=CC c1(OC)cc(Cl)ccc1CNC1CC(F)CN(C(=O)CCc2ccoc2)C1 c1(C(N2CC(C(=O)Nc3cncc(C#N)c3)(SC)C2)=O)cccc(C)c1C#N C1(C)(NC(c2cn(CCOC)nc2)c2nnnn2CC(F)F)CC=CCC1 c1(C2C(C(=O)NCCN(C(c3cc(F)cs3)=O)CC)C2)ccccc1C c1(N2CCCC(C=C)C2)nc(=NC(C)c2cc(Br)ccc2C)[nH]c2cc[nH]c12 C(CCCCCNC(c1nn[nH]c1Cl)=O)N(C)C(c1ccc(C#N)o1)=O c1(C(N2CCC(NC(CSc3n(C)ccn3)=O)C2)=O)ccc(Br)cc1O c1(C(=O)NCC2CC(F)CN2C(=O)CCN2CCC2)coc(=O)c2ccccc12 c1(NC(C(C)NC(C#CC(C)C)=O)C(C)C)ncnc2cnccc12 C(C(C)(C)S(C)(=O)=O)N(C(c1cc(-c2ccc(Cl)cc2)[nH]n1)=O)CC CN1CC(=O)Nc2ccc(NC(c3ncsc3Br)c3nnnn3CC(F)F)cc21 CCC(F)(F)C(=O)NC1CN(C(c2nocc2C)=O)CC1c1ccc(F)cc1 C12(CC(C)(C)C1)C(=O)N2.C(=O)(CCC(C)OC)NC1C(C(=O)OC)OCC1 c1(CC)ncccc1C(=O)NC(CC1CCOCC1)C(=O)NCC[Si](C)(C)C C1(CNC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)C2=C(Cl)CC2)CC1 C(CC(=O)NC1CN(C(c2ccsc2OC)=O)CC1C)(C1=CCCC1)OCC C1(=CCNC(=O)COC(F)F)CCN(C(C2CCS2(=O)=O)=O)CC1 C(=O)(C(C)(C)C(C)(C)C)N1CCN(C(C2(C)CCN(C)CC2)=O)CC1CCO c1(NCC(c2cccc(C)c2)N(C)C)ncnc(N2CCCC(C)C2)c1C C1(C)(C(=O)NC2CCC(CNC(CCC=C(C)C)=O)CC2)CCCNS1(=O)=O c1(C(N2C3CN(C)C(C3)C2)=O)cc2cc(C3=CCC(C)(C)CC3)ccc2oc1=O c1(NC(C(c2cccnc2)C)=O)ccccc1C(=O)N(CCO)Cc1ccccc1 C#CC(C(=O)OC)(C(F)(F)F)OC(=O)CONC(=O)OC(C)(C)C C(=O)(C(CNC(=O)CCC1CC1C)CC(C)C)NC(CCSC)C c1(CC)ncccc1C(N1CCC(NC(=O)C(=O)N(C)C)C1c1ccccc1)=O C(=O)(C(C)C(F)(F)C(F)F)N1C(CN(C(c2ccc(O)cc2F)=O)CC)CCC1 CC(CC(=O)NCC1CN(C(C2CCC(=O)O2)=O)CCC1C)CC(F)(F)F c1(NC(C(=O)NCC2N(C(=O)OC(C)(C)C)CC(F)C2)=O)ccc2ncsc2c1Br C(C)(CNC(c1ncoc1C)=O)(C(C)C)NC(CSCC(=O)OC)=O C1(CC)C(NC(=O)CC(C)(C)C)CCCN1C(=O)CC1CCCC1(F)F C1(C(=O)OC(C#C)C(=O)OC(C)(C)C)CC2(CC(NC(C)=O)CCS2=O)C1 c1(CC(=O)NC2CN(C(C3CC(=C)C3)=O)C(C)C2)c(CC)nn(C)c1CC c1(CC(=O)N(C2CN(C(=O)C(F)CC3CC3)C2)C)cccc(C(N)=O)c1 C1(NC(CN(C)CC)=O)CCCCN(C(c2ccc(CC3CC3)cn2)=O)C1 c1(C(N(C2CCN(C(c3ccc(C)c(F)c3)=O)CC2)C)=O)cc2n(n1)CCCO2 N1(C(=O)CC2CCN2C(c2ncccn2)=O)CCCC12CCCCC2 c1(Cc2c(Br)cc(C(N3C(C)C(=O)NCC3)CN(C)C)s2)ccc2c(c1)CCC2 C(=O)(C(F)CC(C)(C)NC(=O)Cc1ccccc1C)N1C(COC)COCC1 N1(C(C(=Cc2cccnc2)C)=O)CCC(CNC(C2(C)CC2Br)=O)C(F)(F)CC1 CN1CC(C)(C)CC1C(=O)NCC1CN(C(=O)Cn2nnc(C3CC3)n2)CC1(C)C c1(C(N2CC(NC(c3c(C)nn(C)c3C)=O)C(O)C2)=O)ccnc2cc[nH]c12 N1(C(C2(CCCC)CC2)=O)CCCC(C(N)=O)C1 C1(C(=O)NC2CCC(C)N(C(=O)C3=CC(C)C3)C2)CCCC2(CCC2)O1 C1(OC)(OC)CC(C(=O)NOCCOC(C(Cc2ccoc2)C(=O)N(C)C)=O)C1 Cc1c[nH]c2ncnc(N3CC4C(C(=O)Nc5ccc6nnsc6c5)C4C3)c12 C1(NC(C2CC(OC)C2)=O)CCN(C(c2cc(-c3csc(C)n3)cn2C)=O)C1C C(=O)(C(O)C(C)(C)C)NCCn1ccc(CC(=O)NCC(C)=O)c1 CCCCC(CNC(C1CCC2(CC2)C1)=O)NC(=O)C(C)(C)C1CCCC1 C1(C(=O)NCC2(C)N(C(C3CC(C)OC3)=O)CCC2)CCCCCCC1 C1(CCOC)(NC(c2cc(OC)nn2C)=O)CCN(C(C2CCCC2O)=O)C1 c1(NC(=O)NCCC2N(C)CCC2)cnc(Cl)c(Cl)c1 C1(NC(C2COC2)=O)CC2CCCC(C1)N2C(=O)CC1CCCCCO1 C1(C(=O)NCC(CC)N(C)C(c2cn(C)nn2)=O)COC2COCC2O1 C(=O)(CCC(N)=O)NC(C(N1CCC(=C)C1)=O)c1cccs1 c1(C(=O)NC(CNC(CCOC(C)C)=O)C)cccn2[nH]c(=N)nc12 C1(O)(CNC(C(Cc2ncn(C)c2)O)=O)CCN(C(c2nccn2C)=O)C1 c1(OC)ccc(F)cc1S(=O)(=O)N1CCCC(NC(c2cc(C)no2)=O)CC1 N1(C(C2CCN(C(C(C)CC(N)=O)=O)C2(C)C)=O)CCCOC(C)(C)C1 c1(C(=O)NC(C(C)NC(=O)C=CC=C(Cl)Cl)(C)C)ccnc2ccnn12 c1(C(=O)NCC2C(CNC(=O)C3=NOCC3)C2)cc(=O)n2ccccc2n1 N1(CC(C)C)CC(C(=O)ON(C2CCN(CC(C)C)CC2)c2nccs2)CC1=O C(=O)(CCCCC(C)(C)OC)N1CCN(C(C(CC#C)C)=O)CC1C(C)C N1(CCC)CCOC2(CCCN(c3ncncc3I)C2)C1.c12ccc(cc1)o2 N1(C(CN(C)C(N)=O)=O)C2CCC1(CNC(=O)Cc1ccccc1Cl)CC2 Cc1c(C(=O)NC2COCCC2NC(=O)CC2CCOC2(C)C)sc2cncn12 CCCCC(CC)C(=O)NC1(C)CC(C(=O)NCCc2cccnc2)C1 c1(NC(C(CN(C)C)NC(C(c2cnn(C)c2)C)=O)=O)cnc(O)c(F)c1 CCC(CC)(CCNC(=O)c1n[nH]c(=O)[nH]1)NC(c1cc(CC(C)C)[nH]n1)=O C12(NC(C3CC(OC)C3)=O)CCC(CC1)N(C(C1CCC1c1ccccc1)=O)C2 C1(OC)CN(C(c2cc(O)no2)=O)CC1NC(c1ccc(I)cc1)=O n1(C(C)C(=O)N(CC(C)(C)C)Cc2cccs2)cc(C2CC2)nn1 N=c1cc[nH]cc1C(=O)NC12CC1CN(C(=O)CNC(c1ccc(F)cc1)=O)C2 Cc1cc(C(N2CCOC(CCNC(=O)CCCc3cc[nH]n3)C2)=O)ncc1F N1(C(C(=O)NC2C(CC)N(C(=O)OC(C)(C)C)CC2)=O)CCn2ncc(O)c2C1.C C(=O)(C=C1SCC(=O)N1C)N1CCC(CC=C)(C(=O)NC(c2ccco2)C)C1 C12(NC(=O)C3=CCC3)CCCC1CN(C(C1(CC3CC3)CCC1)=O)C2 N1(C(C2(NC(CN(C3CCC3)C)=O)CC(F)C2)=O)CCC2CCCC2C1 N1(C(C2C(C(C)NC(=O)C3=CCSC3)C2)=O)CC2(C1)CC1(CCC1)C2 C1(NC(CC=C(C)C)=O)CCC(C)N(C(=O)C(C)Cc2c(C)noc2C)C1 c1(C(=O)NCC(CCN(C)C(c2ccc(C#N)cc2)=O)O)cnn2ncccc12 C1(C(=O)NCCc2cccs2)CC2CCCCC2N1C(c1ccccc1Cl)=O C1(NC(C(C)CN)=O)CC2CC(C1)CN(C(c1cc(-c3cccs3)on1)=O)C2 CCCS(=O)(=O)C(C)C(=O)NC(CNC(=O)CCSc1n[nH]c(C)n1)CO c1(CNC(CC(C)(C)N(CC(=O)OCC)C2CC2)=O)c[nH]c2c(C)cccc12 c1(OC)cccc(C(C)CC(=O)N2CCC2CNC(c2onc(C)c2C)=O)c1 C1(c2onc(C)n2)CCC(CO)CC1.c1(C=O)ccc(-c2nc(C3CC3)no2)o1 C=CC1COCC1NC(=O)CCN(CCCO)C(=O)Cn1ccc(C)cc1=O C12(CNc3cc(NC(c4ccoc4)COC)nc(C)n3)CC3CC(C1)C(C)CC3C2 c1(N2CCN(c3ccc(C#N)cc3)CC2)ncnc2ncc(Br)cc12 Cc1sc(C)c2sc(C(=O)NC3CC3CNC(=O)Cc3cc[nH]n3)cc12 c1(C(N2C(CNC(=O)C(C)(C)C#N)CC(OC)C2)=O)cc2n(n1)CC(F)C2 c1(CCNC(N2C(CCC#C)CCC2)=O)ccc(C)cc1 c1(CC(=O)NCC(C)NC(c2c(N)cccc2F)=O)cccn(C)c1=O N1(C(C2CC(C)(C)C2)=O)CCN(C(C2CCN2C2CCCC2)=O)CC(O)C1 c1(NC(C(CC)(C)CNC(=O)C(O)COC)=O)cc(C)c(C)cc1C c1(C(N2C3CN(C(C=C4CCN(C)C4)=O)C(CC3)C2)=O)ccc2c(c1)SCCN2 N1(C(COCCOCC#C)=O)CCC(NC(C2CCC2(F)F)=O)C(F)(F)CC1 C1(NC(C2(OCC)CCC2)=O)CCCCN(C(=O)CCC2CC2(F)F)C1 c1(OC)cncc(CCC(=O)NC2CCCC2(C)CSC)c1.C12CN(C1)C2=O CC(C)(CNC(=O)C(C1CCCC1)NC(=O)Cc1cncs1)C1CCCO1 C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(C)N(C(c1oc(C)c(CO)c1)=O)C c1(NC(C2C(NC(C(C(C)C)OC)=O)CC2)=O)ccc2nsnc2c1 c1(CC(=O)NC2C(NC(CCC#C)=O)C2)sc(SCC)nc1C c1(NC(=O)NC(C2CC2n2ccnn2)C2CC2)csc2ccc(Cl)cc12 C12=NC(=NC(=O)NCCc3c(cccc3)O1)ON2.C(C)(=O)O.CC C(=O)(C1=CCCCO1)N1CC(CCNC(c2cc(C)nn2CC(F)F)=O)C(C)C1 n1(CC(=O)NCC(C)NC(c2c(C)cc(C)o2)=O)cc(Br)ccc1=O CC1(C)C2CC(C(N3CCC(C)(NC(=O)C(=Cc4cccnc4)F)C3)=O)CC12 CC1CN(C(c2cccnc2-n2ccnc2)=O)CCN1C(C1CCCSS1)=O N1(CC(=O)NCC#CCNC(C(COC)O)=O)CCN(C2CC2)C1=O C12(CC(=O)NCC(=C3CN(c4ncn(C)c(=O)c4)C3)F)CCCCC1C2(F)F c1(C(N(CC(C)NC(=O)CCOC2CCOC2)C)=O)ccccc1 N1(C(c2ccccc2Br)=O)CCC2C(CCN2C(c2cnn(C(F)F)c2)=O)C1 CC1CCc2nc(C(=O)NCCCCCCN(C)C(c3cncs3)=O)ccc2C1 c1(C(=O)NC2CN(C(c3ccc(O)cc3O)=O)CC2F)cnn2c1CC(F)(F)C2 CC(CC(=O)NCCC1CC2CCC1O2)C(C)(C)NC(=O)C=C1CCC1 CN1CCC(C)(C(=O)NCC2CCN(C(=O)C=Cc3ccccn3)CC2)CC1 C(C(O)C(=O)N=c1ccn(C(C)(C)C)[nH]1)NC(c1nn(CC)c(C)c1)=O C1(NC(CCCOCC)=O)CN(C(C2C3CCC23)=O)C2(CCCCC2)C1 c1(C(N(C2CCCN(C(C3C(COC)C3)=O)CC2)C)=O)cccn2ccnc12 CC1(C)COCCC1C(=O)NCC1(NC(=O)CC23COC(CF)(C2)C3)CCOC1 C1(C(=O)NCCN(C(=O)CCSc2nnsc2Cl)C)CCOCC1 C1(c2nc(C)on2)CCN(C(c2ccc(-c3ccccc3)cc2)C)CC1 C1(CC(=O)NCCC2(NC(CCOC)=O)CCOCC2)OCCOC1(C)C N1(C(c2nc(C34COCC(c5ccccc5)(C3)C4)no2)=O)CC2CC(O)CC(C2)C1 c1(N(C)CC2(OC)CCC2)cc(S(=O)(=O)NCC2CC23CC3(F)F)ccc1C#N C(=O)(CS(=O)(=O)C1CC1)NC1CCC(CNC(C2C(C)(C)C2CN=[N+]=[N-])=O)CC1 O=C(CC(CC1CC1)NC(C(N1CC(F)(CF)C1)=O)c1ccco1)NC1CC1 c1(CCCC)cn(CC(=O)NC)nn1.N(S(=O)(=O)NC)CC(CC(C)SC)=O C1(F)(NC(COCCCOC)=O)CCCN(C(=O)CC(C)F)C1 CC1(F)CCN(C(=NCCCCl)NC2CCC(C(=O)OC(C)(C)C)C2)C1 c1(C(=O)NCC(CC)NC(C2CC(F)C2)=O)cc(S(N)(=O)=O)c(C)cc1C c1(C(C)(F)F)ccc(C(=O)NCCOCCNC(C2CCCN2C=O)=O)cn1 c1(CNC(N2CCOCC2CC2CC2)=O)ccc(CN2C(=O)CNC2=O)cc1 C1(NC(CSC)=O)CCC2CCN(C(c3ccc(Cl)nc3)=O)C1C2 C#Cc1cc(C(=O)NCC(C)N(C(c2cn(C)nc2O)=O)CC)cc(Br)c1 CN=c1[nH]c(=NC(C)c2ccoc2)[nH]c(=NCC(C)CC(F)(F)F)[nH]1 c1(CCC(=O)OCC)ccc(Oc2ccc(NC(=O)C3CC3)cn2)cc1 C(=O)(C(Cn1cncn1)NC(C)=O)N(CCC(=O)OC)C Cc1nc(C(c2ccncc2)N(C(C(=O)OCCN)=O)C)n[nH]1 n1(CC(=O)NCC2C(NC(C(C)SC(F)(F)F)=O)C2)ncc(O)nc1=O C1(C2CCN(C(C3CC3(F)Cl)=O)CC2)(NC(c2cnc3[nH]cncc2-3)=O)CCC1 c1(C2C(CNC(CCNC(C(C)c3cccs3)=O)=O)C2)cn(C)cn1 C(N=c1[nH]c(=N)[nH]c(=NC2CCCN(C)CC2)[nH]1)C1(C)ON=C(C)C1 c1(C(c2nnnn2C2CCCC2)NCC(COCC)(C)C)cc2ccsc2n1C C(=O)(C1=CC2(CCN(C(=O)C=Cc3ccoc3)C2)C1)N(C(C)C(N)=O)C c1(C(C(=O)NCCOC)N(CCF)CC)ccnc(Br)c1 C1(C(=O)NCCC2CN(C(c3c(NC(C)C)nccc3)=O)C2)CCOCC1(C)C C#CCCCCCCCC(=O)N(CCNC(=O)CC(O)CCCC)C1CC1 CC1=C(C)CC(C)(NC(C2CCN(C(c3cc(C#N)cs3)=O)CCO2)=O)CC1 c1(C(=O)NC2C3(CCN(S(CCC)(=O)=O)CC3)C2)cc(O)c(OC)cc1[N+](=O)[O-] N1(C(C=C(C)c2cccs2)=O)CCC2CN(C(=O)C=Cc3nnn(C)n3)CC2C1 CCCCC(O)C(=O)NC(Cc1cn[nH]c1)C(=O)NC(COC)C1CC1 N1(Cc2cc(C)[nH]n2)CC(NC(c2cccc(C(F)(F)F)c2Br)=O)C2(CC2)C1 C1(OCC)CCN(C(c2cc(CNC(=O)CN(C)C(C)=O)[nH]n2)=O)CC1C CC1CCN(C(=O)CC2(n3cccn3)CC2)CCN1C(=O)C(CO)C(F)(F)F c1(C(=O)NC(CC=C)CNC(c2ccc(C)n2C)=O)cc2cccnn2n1 C1(C(=O)NCc2nnc(CC)o2)CCCN(C(c2cnn(C)c2OC)=O)C1 Cc1ccc(CCC(=O)NCCCCN(C(=O)C(O)C2CCCC2)C)c(C)c1 Cc1n[nH]c(C)c1CCC(=O)NC1CCCCC1CNC(c1nc(=N)cc[nH]1)=O c1(C(=O)NCC2C(NC(c3c(C)oc(C#N)c3)=O)CCC2)cnc2c(c1)NCC2 C(CCCCC(=O)NCC(C1CC1)NC(C1CCC(n2cccc2)CC1)=O)=CC C1(C(=O)O)(CC)CCCCN1C(=O)CC1CC1(Cl)Cl.c1(C)cn(CCCC(=O)O)nn1 C(CCC(=O)NC1CC1)N(CCN(CC(=O)NC(C)(C)C)C(C)C)CCO c1(CN(C(=O)Cc2ccsc2)CCNC(C2ON=C(C)C2)=O)ccc(Cl)nc1 c1(C(=O)NCC(C2CCCC2)NC(C2C(OC)C2)=O)cc(Cl)cc2cccnc12 O=S(=O)(CCCF)NC(c1ccsc1)C1CC1 O(NC(=O)C1=CCSC1)CC(=O)N(CCCN(C)C)C Cc1cnc(C(=O)N(C2CCCN(C(c3ccnc(S)c3)=O)C2)CCO)cn1 C(=O)(C(F)C(C)(F)F)NC(C(=O)NC1(C)CCOC1)CO c1(C(=O)NCC(C(C)(C)C)NC(C2C(OCC)C2)=O)cncc(P(C)(C)=O)c1 c1(NC(C2C(NC(c3cncnc3)C)CCC2)=O)ncnc2n[nH]c(I)c12 C1(C(=O)NCC)CSCN1C(c1ccc(CNC(=O)C(CSC)OC)[nH]1)=O Cc1ccc2c(=NCC#CCCO)[nH]c(=NCc3ccc(C#N)cn3)[nH]c2c1 C1(C(=O)NCCC(CNC(c2cncnc2)=O)O)CCC2(CCC2)C1 c1(C(=O)NC2C3CC(NC(C4(P(C)(C)=O)CC4)=O)CC3C2)ccc2sccc2c1 C(N=c1[nH]c2c(F)cccc2o1)C1(CNC(c2cc(F)cc3nc[nH]c23)=O)CC1 c1(C(=O)NCC23CC(NC(CC(CC)(F)F)=O)(C2)C(C)O3)cccc(S(C)=O)c1 c1(N(C)C)ncc(C(=O)NCCC(O)CNC(=O)C(C2CCOCC2)O)o1 CCCCC(C)(F)C(=O)N1CCN(C(c2ccccc2)=O)C(CC(F)F)C1 N1(C(CNS(CC)(=O)=O)=O)CCCC(CNC(C2(C)CSC2)=O)CC1 c1(C(=O)NCC(C2CC2)NC(C(C)n2ccnn2)=O)cccnc1OC(F)(F)F c1(C(=O)OCC)cccc(C(=O)NC2(CNC(c3coc(C)n3)=O)CCC2)n1 CCCC(C)(O)CC(=O)N1CC2CC(NC(c3ncccc3C)=O)CC1C2 C1(C(=O)NC2CC(CNC(C(C3CCCCCC3)OC)=O)C2)CCOC(=O)CC1 C#Cc1cnn(C)c1C(=O)NC(CNC(C1COCC(C)(C)O1)=O)C1CC1 n1(CC(N2C(CNC(C3(C(=O)OC)COC3)=O)CC2)=O)c(=O)oc2ccccc12 c1(C(=O)NCCCNC(c2c(N(C)C)ccnc2)=O)cc(O)nc(Cl)c1 S(=O)(=O)(c1ccc(F)c(C(=O)N(C)C)c1)NCC(c1ccnn1C)N(C)C C1(NC(CCC#CC)=O)C(C)CN(C(=O)CCCc2ccc(Cl)c(Cl)c2)CC1C CC(=O)CC(C)(C)C(=O)NCC1CCCC1NC(=O)CCc1ncc(C)[nH]1 N1(C(C(CC)CC)=O)C2CCC1CC(CNC(c1cc(C(C)(F)F)ccn1)=O)C2 C1(C(=O)NC(C2(CO)CC2)C)(NC(=O)CC2(O)CCOC2)CC(O)C1 CCC(CC(=O)N(C1CC(C#N)(CC)C1)CC1CCCCC1)C1CCC1 N1(C(C(CCCC)O)=O)CCn2ncc(CNC(c3nc(C4CC4)cs3)=O)c2C1 c1(CC)ccc2nc(NC(N3CCC(C)C(CSC)C3)=O)sc2c1 Cc1nc(C)c(C(=O)NC2CC(C(=O)NC3CC=CCC3C)C2)o1 Cc1nc(Cl)ccc1CC(=O)NC1(CCNC(c2ccc(Cl)nn2)=O)CCC1 CC(C)C(CCC(=O)NC1CCOC1C)NC(C1CC(C)(C)CN1C)=O C1(OC)CC2N(C1)C2=O.c1(C(C(=O)NC2(CC(=O)OC)CC2)C)ccn(C)c1 CC(CC(=O)NC(c1cn(-c2cnn(C)c2)nn1)(C)C)P(C)(C)=O C1(C(=O)O)CCC2(C1)CN(C(c1cccc(-c3sccc3[N+](=O)[O-])c1)=O)C2 C1(CNC(CCNC(C)=O)=O)CCCC1C(=O)N(C)CC1(C)CCC1 C1(NC(Cc2nc(COC)sc2)=O)CN(C(C2(C)CC(C)=NO2)=O)CCC1O C1(C(N2CCOCC(NC(C(C)(C)C)=O)C2)=O)CC2(CO1)CC(F)(F)C2 c1(C(N2CCCC(NC(C)=O)CCC2)=O)ccc2c(c1)C=CS2(=O)=O C#CC1CCN(C(=O)CC(COC)NC(c2cccn2C(C)C)=O)CC1 c1(CC(C(=O)OC)NC2CCCC(C)(C)C2)c[nH]c2ccc(F)nc12 C1(C(=O)NC2(C)CC(NC(C(C(C)C)OCC)=O)C2)CCC(C2CCC2)CC1 C1Sc2ccc(Cl)cc2NC1=O.c1(OCC)cccc(OCC)c1COC Cc1ncnc(C)c1CC(=O)NCC1C=CCN1C(c1cc(F)n(C)n1)=O Cn1cnc(CC(O)C(=O)NC2CC2NC(=O)COC2CCCC2)c1 C1(NC(=O)CSCC(F)F)CC2(C1)CN(C(=O)CCc1ccc(F)cc1)C2 CC1CN(C(c2cncc(N)c2)=O)CCCN1C(C12CC1CCC2(F)F)=O C1(C(N(CC(=O)NCc2ccc(CO)cn2)CC)=O)CCOC(C)C1 c1(N2CCCC3(COC)C2C3)nc(N2CCOC(CC(N)=O)C2)nc2c1ncn2C C1(N=[N+]=[N-])(C(=O)NCc2ccn(C(C)C)n2)CCN(C(=O)C=CC(=O)N(C)C)C1 C(CCCC(F)(F)F)NC(CC(CNC(C(C)OC(C)(C)C)=O)O)=O Cc1cncc(C(=O)NC2(C)CN(C(=O)CCCc3n[nH]c(=N)s3)C2)c1C c1(C(=O)NCC(CC=C)NC(=O)CCSCC2CCCO2)cccc(C(C)C)c1 c1(C(N2CCN(C(c3nnn4c3COCC4)=O)CC2)=O)ccc([N+](=O)[O-])cc1O c1(C(=O)NC2(C)CC(NC(c3c(CCC)nco3)=O)C2)ccc(F)cc1C Cc1n[nH]c(C)c1C(C)CC(=O)NC1(C(c2ccccc2)O)CC(F)(F)C1 N1(C(C(CC(C)C)NC(C)=O)=O)CCCN(C(=O)C(N2CCC(C)C2)=O)CCC1 N1(C(C2CCC(C)S2)=O)CCC(O)(CN(C(=O)Cc2csc(S)n2)C)CC1 N#Cc1ccc2c(CNCCC3NC(=O)NC3=O)c[nH]c2c1 N1(CC(=O)N(C2CC(NC(C(c3c(C)noc3C)CC)=O)C2)C)CCCCC1=O c1(NC(C2CCCOCC2)c2n(CCC)nnn2)cc([N+](=O)[O-])ccc1CC N1(Cc2ccc(C(=O)NC(COC)C)cc2)CCC2CCCC12 C1(NC(CCC#C)=O)CN(C(c2cnc(C)s2)=O)CC1n1ccnn1 CCCS(=O)(=O)CC(=O)N1CCC(NC(c2n[nH]c3c2COC3)=O)C1 c1(C(N(CCN(C(c2[nH]cc(CC)c2)=O)C)C)=O)cc2c(cn1)OCCO2 C1(CNC(CC(=O)OCCC(C)C)=O)CC2CCC1N(C(=O)C1=C(Cl)CC1)C2 C1(COC)CC2(CC2)CN1CCc1ncc(C(=O)O)cn1 C1(NC(C=CSC)=O)CCN(C(c2nnn(C(C)C)c2C)=O)CC1C c1(CN2CC(N(C(=O)C(=O)Nc3ccccc3)C)C(O)C2)ccc(Cl)cc1I N1(C(CCC)=O)CCN(C(=O)Cc2ccc(O)nc2)CC1c1ccccc1 CCC(O)C(C)C(=O)N1CCN(C(=O)C=Cc2ccco2)CC1 C(c1cccnc1)=C(C)C(N1CCC(CO)(CNC(C2CN(C(C)C)C2)=O)C1)=O C1(NC(c2cncc(F)c2)c2n(C3(C)CC3)nnn2)CCc2c(nnn2C)C1 N1(C(CCCCC#C)=O)CCC2(CCCN(C(C3CC(C4CC4)=NO3)=O)C2)C1 N1(C(CC2N(CC)CCC2)=O)CC(C2(NC(=O)CC(C)(C)C3CC3)CC2)C1 C(=O)(C(C)C(=O)NCCNC(c1cc(C#N)cs1)=O)OC.C12CN(C1)C2=O c1(OC)cc(CO)ccc1C(=O)N(C1C2CN(C(=O)CCC=CC(C)C)CC12)C N1(C(CCN2CCN(CC)CC2)=O)CC(NC(c2cccs2)=O)CC(O)C1 C(=O)(C(c1ccc(Cl)cc1)=C(O)CON=C1CCCCCCC1)OCC c1(COC)cc(C(=O)NCC2CCCN2C(=O)COCC(=O)OC)n(C)c1 c1(C(=O)NCC(N(OCC)C)=O)ccc(S(=N)(=O)C(F)F)cc1 C(C(C)(O)CC(=O)N1CC(OC)CC1CNC(c1sccc1C(C)(C)C)=O)OC N1(C(C=C(CC)C)=O)CCc2ccccc2C1CNC(=O)CCc1cnc(O)[nH]1 N1(C(C#CC(C)C)=O)CCC(C2(NC(=O)Cc3ccc(Cl)cc3F)CC2)C1 C1(C(=O)OC)CC(=O)NN(C(=O)c2ccc(OCC(N)=O)cc2)C1 C1(C(=O)NC2CN(C(c3ccncc3Cl)=O)CC2O)CCCNS1(=O)=O c1(C(=O)NCC2C(NC(c3cnccn3)=O)C2)cc(C(F)F)ncn1 N1(C(C(CC)C)=O)CC2CN(C(C3CCCS3)=O)CC12 O=C1CCCC(CC(=O)NC23CC(C(=O)NCCC4(C5CC5)CC4)(C2)C3)C1 C1(C(C(=O)NCC2CN(C(=O)C(C)=C3CC3)CC2O)OC)CCC(F)(F)CC1 c1(OC)cc(=O)n(C)cc1C(N1CC(NC(C2(C3CC3)CCC2)=O)CC(O)C1)=O C1(COC)(CNC(=O)C(C)(C)c2nccs2)CCCN1C(=O)Cn1ncn(C)c1=O C(=O)(CCCC(=O)N(CC(O)CF)C(C)C)OC c1(C(=O)NCC(C(C)C)NC(C(CC)(C)OC)=O)c(F)cccc1F C(C(C)(C)CNC(=O)C(c1csc(C)n1)=O)N(C(=O)C(O)CN(C)C)CC c1(C(N2C(CNC(C(F)OC)=O)CC2)=O)cc2c(s1)CCCCCC2 CC1CC(N=c2nc(N(C)Cc3cscc3Br)c3cc(Cl)ccc3[nH]2)CS1 c1(C(=O)NC(C)CC2CCCCC2)ccc(CNC(C2CCNC(=O)C2)=O)nc1 CCC(F)(F)C(C)(C)NC(C1CC2CC1CC2NC(c1cc(C)c(C)[nH]1)=O)=O C(=O)(C1CNC(=O)c2ccccc21)NCC1(C(C)NC(c2cnccn2)=O)CC1 N1(Cc2cc(C)on2)CCCC(C(=O)Nc2ccccc2)C1 N1(C(CC(CC)O)=O)CC(F)(F)CC1C(N1CCC(C)(OC)CC1)=O C1(C(=O)NCc2c(C)nns2)CC(C)(C)CN1C(=O)C(C)N(C)C C1(C(=O)NCC2N(C(c3scc(C(N)=O)c3)=O)CC2)C2CCCCC12 N12CC3CC(C1)C3C(=O)c1ccccc1S2(=O)=O.c1(SC)ccc(N(C)C)cc1 CCC(CNC(=O)C(C(C)C)SC)(CC)C(=O)N(CC(C(C)C)OC)C CC(C(C)(C)C(=O)N1CCC(CC(F)F)C1)NC(c1nn(C)cc1Cl)=O N1(C(C2CN(C(C(CCCCC)F)=O)CC(C)O2)=O)CCc2ccncc2C1 n1(CCCC)cc(C(=O)N(CC(O)CNC(c2[nH]c(O)nc2C)=O)C)c(C)n1 C1(C(N(CCCNC(CCC#CC)=O)C2CC2)=O)CC(=O)c2ccccc2C1 C(c1ccc(Cl)nc1)=CC(N1CCN(C(=O)C2=CCCO2)C(CCO)C1)=O C1(NC(=O)Cc2nnc(O)s2)CN(C(C23CC(F)(C2)C3)=O)CC12CC2 c1(N2CCN(C(CC)C)CC2)ncc(C)cc1S(=O)(=O)NC1CC(C)(C)C1 n1(CC(N2CCC(NC(C3N(CC)CC3)=O)C(F)C2)=O)cc2ncccc2n1 C(C1CCCN1C(C1C=CCS1)=O)=CC(=O)N(CC#CC)CC#C c1(C(=O)NCC(C)CN(C)C)cc(Cl)n[nH]1.N12CCC1C2=O C(=O)(C(CO)C(C)C)N(C)CC1OCCN(C(c2c(C)n[nH]c2)=O)C1 c1(CNC(CCOCC#C)=O)cc2n(n1)CCN(C(=O)Cc1scnc1C)C2 c1(C(N(C)CC2OCCN(C(c3cc(C)sc3)=O)C2)=O)[nH]c(C)c(C)c1C Cc1ccc(CC(N2CC(CF)(NC(=O)C(C)c3ccsc3)C2)=O)c(Cl)c1 c1(OC)ccnc(C(N2CCC(O)(C(C)NC(C3CCN3C(C)=O)=O)C2)=O)c1O C(=O)(C(C)(C)C(=O)NCCCC1(NC(c2sc(N(C)C)nc2C)=O)CC1)OCC N1(CC(=O)NC)CCN(c2nnc(-c3cccn3C)n2CC(C)C)CC1 Cc1ccc(C(=O)N(CCCNC(=O)CN(C)S(N)(=O)=O)CC2CCCC2)cn1 c1(C(=O)NC2CCC(NC(C(C)(CO)OC)=O)C2)cc2sc(C)cc2s1 c1(C(c2n(CC)nnn2)NCc2cn(C)nn2)cccc2c1CCC2 c1(SC)nc(C)cc(=NC(C)CCNC(=O)C(=O)Nc2c(C)cccc2Cl)[nH]1 c1(C(=O)NC(CC)CNC(=O)CCCc2sccc2C)ccc(COC)cc1 CCC(CC(=O)NC1CC(F)CN(C(c2ccncc2OC)=O)C1)C(C)(C)C c1(CC(=O)N(CCC#N)Cc2ccc(C)cc2)cncc(C#N)c1 C1(C(=O)NCC23CC(NC(C4CCC(C(=O)OC)C4)=O)(C2)C3)CCCC1(F)F C1(C(=O)OC)CC2(CCOCC2)CN1C(C1CCC12CCCO2)=O CC1=C(C(=O)N(C)CC=CC(N2CC(C)CC2CO)=O)CC1 c1(N(C2CCNC2=O)C(c2ccccc2)C)cc(C(=O)N(C)C)nn1C N1(CCCn2c(C)ncc2)CC2CCCC(O)C2C1 N1(C(c2occ(C(C)C)c2)=O)CCC2CCC12CNC(c1ccc(=O)n(C)c1)=O c1(C(N2CCC(CC(=O)NCc3c(C)n[nH]c3)CC2)=O)cc2sccn2c1 Nc1cc2c(cc1NCc1c(OC(F)(F)F)cccc1F)CCCC2 c1(C(N2C(CNC(C(F)=CCC)=O)C=CC2)=O)cc(O)cc([N+](=O)[O-])c1 C1(C)(C(=O)NCCCC(=O)NCC(C(=O)OC)C)CC2(CCC2)C1 C12(C(=O)NCCCN(CC)CC)CC(CCO1)N(C(=O)C#CC1CCOC1)C2 C(CCC(=O)NCCC1(O)CC1)NC(c1nc(C(=O)OCC)sc1)=O Cc1ncc(F)c(NC(C2CC3(C2)CN(C(=O)C(O)CC(C)C)C3)=O)n1 C(=O)(CCC(=O)NCC(CO)NC(=O)C(C(C)C)c1cccc(OC)c1)NCC C1(CNC(c2cc(OC)cc(F)c2)=O)CC2(CCN(C(=O)CCC3CC3)CC2)C1 C(C1=CCN(C(c2cnc(N)c(Cl)c2)=O)CC1)NC(C(CC#C)C1CC1)=O c1(-c2nc(CC(=O)OC)c(C)s2)cc(OC)ccc1OCC(C)C N1(C(C(C)=CC)=O)CC(NC(=O)C(C(C)C)n2cc(C)cn2)C(C(F)F)C1 N1(C(C)C(=O)N(C)CCOCCN(C(=O)CCNC(C)(C)C)C)CCOCC1 C(=O)(C#CC1CCOCC1)N1C(C)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CC1 Cc1cccc(C(=O)N(C2CCN(Cc3ccc(O)c(O)c3)C2)C)c1I Cc1onc(C2CC2)c1C(=O)NCCSCc1cn(C2CCCN(C)C2)nn1 N1(C(CC(C(C)OC)NC(=O)CC2(O)CCOC2)=O)CCC2(CCC2)CC1 CC1CC(N=c2ccc3nnnn3[nH]2)CN1C(=O)CCCCCn1cnnn1 Cc1ccn(CC(=O)NC2COCC2CNC(=O)C(C)(C)C(N)=O)c(=O)c1 C(N=c1nc2sccc2c(N2CCc3c(N)cccc3C2)[nH]1)C1CCC(C)(C)O1 C1(NC(c2c(CC)c[nH]c2)=O)CC12CCN(C(C1COCCN1C)=O)CC2 C1(C(=O)N)CCCN(CCc2cccc(F)c2F)CC1.N1CCCC1C(=O)O c1(CN=C(NC2C(C)(C)SC2)NCC2CCCO2)ccc(O)c(Cl)c1 C1(NC(C2CN(C(C(C(C)(F)F)F)=O)C(C)(C)C2)=O)CCCOC12CCC2 CC(C(=O)NCC=CCNC(=O)Cc1cocn1)n1ccnc1.C1CO1 N1(C(=O)OC(C)(C)C)CC(F)(F)CC1C#N.N12CC3C(C3C1)OCCCC2=O c1(C(=O)OCC)nnc(SC)nc1N1CC(NC(C2C=CC(=O)N=N2)=O)C(F)C1 C=C(C)CC(C(=O)NC1CCCN(C(c2scc(Cl)c2Cl)=O)C1)NC(C)=O c1(CC)noc(C(=O)NCC2CCCC2NC(=O)COCCSC)c1C C(=O)(CC1OCCc2ccsc21)N(CCCNC(c1c(CC)occ1)=O)C(C)C c1(C(=O)NCC(F)CNC(C2CC3CC3C2)=O)cnc2ccccc2c1 c1(CC)ccc(C=CC(=O)N(C)CCN(C(C23CC(C)C2C3)=O)C(C)C)o1 c1(OCC(=O)NCC(n2cc(CC=C)nn2)C)ccccc1C C#CC1(C)CCCN(C(C2C(O)CCN2C(c2cc(C(C)C)[nH]n2)=O)=O)C1 C1(NC(C2CCN(C(c3c(O)cccc3F)=O)C2)=O)CCn2cnnc2C1 C1(NC(Cc2cc(C)sc2)=O)CS(=O)(=O)CC1NC(=O)C(C)(C)C1CCCC1 N1(C(C(C)N(C(C)=O)C)=O)CCCCC(NC(c2c(C)coc2C(C)(C)C)=O)C1 C1(C(=O)NC2CN(C(CCSC)=O)CC2(C)C)CCc2ccc(F)cc2O1 CC1(C)C(C)(C)C1(F)C(N1CCC(CF)(NC(=O)CCN2CCCS2(=O)=O)C1)=O Cn1nc(C(=O)NCCC2CN(C(=O)CC3CSC3)CCO2)cc1Cl N1(C(CC(C)(C)O)=O)C2CCC1C(CNC(C1(C)CC1c1ccccc1)=O)C2 C1(OC)CCCN(C(=O)C(c2cccc(Br)c2)O)C1C Cc1ccc2occ(C(=O)NC3CCN(C(c4cnn(C)c4Cl)=O)C34CC4)c2c1 CC1COC(C)(C(=O)NC2CC2NC(=O)CCNC(=O)CO)CO1 c1(CNC(CC2C(NC(C3(C)CC3)=O)CCC2)=O)nc(C#N)cs1 N(C1CCCc2ccc(Br)cc21)C(c1c(OC)ccc(Cl)c1)C C(=O)(C1=C(C)OCCS1)NC1CC(CCC(NOCCC(=C)C)=O)C1 c1(SCCC(=O)NCCC(C)NC(C2(CF)CCOCC2)=O)ccc(Cl)cc1 c1(C(CO)NC(C2C(C)C2)=O)cccc(-n2cc(CCc3ccccc3)nn2)c1 Cc1cc(C(=O)NCc2csc(CNC(=O)C(Cl)=CCl)n2)ncc1CO C=CCCC(C(=O)OC)NC(=O)C(C1(O)CCC1)NC(C1C(C)C1C)=O C(=O)(C1=CC2(CN(C(=O)C=CCO)C2)OC1)NCC(C(C)(F)F)Cl c1(COC)nc(NCC(C2CCCC2)NC(c2cc(C)oc2C)=O)cc(O)n1 C1(CN(C(=O)CCN2CCC(F)C2)C)CCN(C(c2scnc2Cl)=O)C1 c1(C(N(CCNC(C(c2ccc(C)cc2)C)=O)C)=O)cccc2cnnc(O)c12 N1(C(c2c(C(C)C)scn2)=O)CCC(CC(C)NC(=O)C(C)(C)CN(C)C)CC1 N1(C(c2c(C)ncs2)=O)CCC2(CC1)CC2CNC(C1(F)CC1(Cl)Cl)=O C(=O)(C1CCCc2ccnn21)N1CC(c2ccccc2C(F)(F)F)CC(C)C1 N1(CC(=O)NC(CCC)C)CCC(S(=O)(=O)N(C)C)C1 C1(C)(C(=O)NC(CC)CNC(C2CC3(CC3)C2)=O)CCOC(C)C1 CP(C)(=O)c1cnc(C(=O)NCCC(=O)Cc2ccccc2)nc1 CN1CCCC1(C)C(=O)N(CC(CO)(CO)NC(=O)COC1(C)CCCC1)C N1(C(c2n(C)cnc2)=O)CCC2(CC2C(N2CCCN(CCO)CC2)=O)C1 c1(C(=O)NC23CCC(C(=O)OC)(CC2)CO3)c(C)[nH]c2c(OC)cccc12 Cc1cc(C(=O)NCC(C)CNC(=O)CCCc2ncc(C)o2)c(O)nn1 C1(C)(NC(c2n(CC(=C)C)nnn2)C2(CC)CCCC2)C(C)(C)C1(C)C n1(CC(=O)NC2C3CN(C(C4C(COC)C4)=O)CC32)ccc(=O)n(C)c1=O C=CC1CCCCN1C(=O)CC1(NC(=O)CC(O)CN(C)C)CCCCC1 C1(CNC(c2cc(C)c(N)cn2)=O)CC2CCC1N(C(=O)COC1CCOC1)C2 C1(NC(CCC)=O)CCC12CCN(C(c1cnn(C(C)C)c1C(F)(F)F)=O)CC2 Cc1nocc1CC(N1CCCC1C(C)NC(C1(n2cncn2)CC1)=O)=O c1(N(CCC(C(F)(F)F)OC(F)F)C)cnc2c(Cl)cnn2c1 c1(C(=O)NC(C2CCCN2C(=O)CC2CCCC2O)C)cc(C2CC2)ccn1 N1(C(C(n2cc(C3(C)CCCC3)nn2)C)=O)CCC(Cc2ccccc2)C(F)(F)C1 CC1(CNC(c2csc(C(F)(F)F)n2)=O)CCCN1C(=O)C1=CCOC1 C1(C(=O)NC(C2CCN(C(c3cnccn3)=O)CC2)C)CCc2nnn(C)c2C1 C1(NC(c2cc(C3CCCC3)[nH]n2)=O)CC2CCC(C1)N2C(=O)CCCC1CC1 N1(C(C2CCCC2)=O)CC2(CCN2C(C2CCCS2)=O)C1 Cc1ccc(F)c(C(=O)NC2CCC(CNC(=O)CC3(C#N)CC3)C2)c1F CN(CCCC(=O)NCC1C2CN(C(C3CCCC3C3CC3)=O)CC12)N=O N12CCc3cc(cc(OC)c3C1)OC2=O.CC#CCCNC(=O)NC Cn1nc(C(N2CCCC(C(O)C(F)F)C2)C(=O)NC2CCOCC2)c(Br)n1 C1(CC(=O)NC2CCC2CNC(c2ccc(C(N)=O)[nH]2)=O)(OCC)CCCCC1 C(CC(=O)NCC(=O)NCCC1(NC(c2ncc[nH]2)CC)CC1)N(C)CC C1(CNC(c2cnc(-c3cn[nH]c3)s2)=O)CN2CCCC2CO1 C(=O)(C1CCSc2ccccc21)NCCOCCCN(C(C=CCC)=O)C C=CC(C)(O)CC(=O)NC1CN(C(c2cc3c[nH]nc3s2)=O)CC1(C)C C=C(Br)CC(=O)NC(c1ccccc1)C(C)NC(=O)CN(CC(C)(C)C)C CCCC(C)CCCC(=O)N1CCC2(CCCN2C(=O)COC2CC=CC2)C1 N1(C(C2(OC)CC(C)(C)C2)=O)CCC(NC(=O)Cc2ccns2)CC(O)C1 S(=O)(=O)(c1cccc(N(C2(C)CC2)C)c1)NCC(=O)Nc1c(C)cccc1 c12ccc(Br)cc1C(C(=O)OC)N(CC1COC(C)(C)O1)C2.C(CC1CC1)OC n1(CCCC)cc(C(=O)NCC2(F)CC(CNC(c3ccoc3C)=O)C2)c(C)n1 Cn1ccc(C(N2CCCCC2C2CCN(C(c3csc(Cl)c3)=O)C2)=O)cc1=O C1(NC(CC2C(CC)C2)=O)CC2CC1CC2C(N1CCCOC(C)C1)=O C12(CNC(C(C3CC3)OCC)=O)CCC(C1)N(C(C1(C)CC3(CCC3)C1)=O)C2 Cc1cccc2[nH]cc(CCC(N3CCC(C(C)NC(=O)CC4CSC4)C3)=O)c12 N1(C(CCC#CC)=O)CC2CC(NC(=O)C=Cc3cccc(F)c3Cl)CC1C2 C1(CNC(Cn2ncc(C#C)c2)=O)COC(C(F)(F)F)CN1C(=O)C(C)(F)F N1(C(c2nccc(CC)c2)=O)CC(NC(C2CC(=C3CC3)C2)=O)CC2(CCC2)C1 c1(C(N(C(CNC(C(C(C)C)NC(C)=O)=O)C)C2CC2)=O)cc(C)cc(C)c1N c1(C(=O)NC2CCC(NC(c3c(CC)cccn3)=O)C2)cnc2c(c1)CCOC2 c1(CCC(=O)NC(CC(C)NC(CC(=C)Br)=O)C)ccc(OCC)cc1 N1(C(C2CC(N(C)C)C2)=O)CC2CCC1C(NC(=O)CCC1NC(=O)NC1=O)C2 c1(SC)cn(C)nc1C(=O)NC1CC(F)(CNC(C2CC2c2ccccc2)=O)C1 C1(C(N(CC(CNC(c2nccc(OC)c2)=O)(C)C)C)=O)CC2(CCCC2)C1 N1(C(=O)C2=CCCCC2)CC2(CCC2)CC1C(N1CCCC(F)CC1)=O c1(NC(c2ncc[nH]2)CC)nc(N(C)Cc2cc(Br)ccc2F)c2sccc2n1 C1(CCC=C)(C(N2CC3CC3C2)=O)CN(C(=O)COCC(=C)C)C1 C1(C(N2CCC(C)(NC(c3cc(CC)[nH]n3)=O)C2)=O)CCc2nnnn2C1 C=CCCC(C(=O)NCCn1cnnc1CC)NC(=O)C(C)NC(=O)NC C(C1c2ccsc2CCN1C(C1(F)CCCCC1)=O)NC(c1cc(C)ncn1)=O C1(N(C)C(c2nnn(C)c2N)=O)CCCC(NC(C2(N3CCCC3)CC2)=O)C1 CCC(CC)(C(=O)NCCN(C(=O)COCC(F)F)C1CC1)OC N1(C(C(CC)N2CCCC2=O)=O)CCC(N(C)Cc2ccc(C(F)F)cn2)CC1 c1(C(C(=O)NCC(CC)NC(=O)Cc2ccsc2C)O)cc(F)c(F)c(F)c1 c1(CCC(=O)NCC(CC(C)C)NC(c2c(CC)ocn2)=O)cc(C)cc(C)c1 c1(C(=O)NC(c2nc(O)c(C)s2)CCOC)cc(=NCc2ccccc2)[nH]c(Cl)n1 C(=O)(CCCCCS(N)(=O)=O)NCC(C(C)C)(C)NC(c1cnc2n1CCC2)=O C1(CC#C)(C(=O)NC(C)C(C)(C)CN(C)C)CCN(C(c2c[nH]ccc2=O)=O)C1 c1(C(N(CC(C)NC(C(CC)(C)OC)=O)C)=O)cc(C)n(-c2nccs2)c1C CC(C)(F)CCC(=O)NCC1(C)CCCN(C(C2(F)CCCC2)=O)C1 C1(NC(C2(C)CC(=C)C2)=O)CCC(C(=O)NCCC2CCCO2)CC1 N1(C(c2cc(CC)on2)=O)CCN(C(=O)CC(O)CN(C)C)CCC1C c1(CC(=O)N(CCN(C(C(C)SCC)=O)C)C(C)C)ccc2oc(C)nc2c1 N(C1CN(C(c2ncc(OC)cn2)=O)CCc2ccccc21)C(C=C(CC)C)=O C1(CCN(C(=O)C(C)(C)CF)C)CCN(C(c2cccc(Cl)n2)=O)CC1 N1(C(c2cnc(C)[nH]2)=O)CCOC(CN(C(=O)CSCC(F)(F)F)C)C1 N1CCCC(N2CCC(O)C2)C1.N=c1[nH]scc1I CCCCC(F)C(=O)N1CCC(C)(C)C1CC(=O)NCCC1=CCOCC1 C(C(=O)NCC(C)CN(C)C(C1CCSC1)=O)(C1CC1)OC C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)C(N(C)C(C2CC2(C)C)=O)C1 c1(CC)cc(C(=O)NC2CC(F)(CNC(=O)CC(C)OC)C2)cc(F)c1 CC(C)(C)C(C(=O)NCC1CN(C(=O)CCF)CC1(F)CO)C1CCC1 Cc1nccc(C(=O)NC2(C)CC(NC(=O)CCCn3ccccc3=O)C2)c1N N1(CC(=O)NC(C2CCN(C(C3CCCS3)=O)C2)C)CCn2ccnc2C1 Cc1cc(S(C)(=O)=O)cc(C(N2CCCC2c2cn[nH]c2)=O)c1C c1(NC(=O)NC2CCC2C(F)F)cccc2c1OCO2 c1(C(CNC(=O)C=CC2CC2)NC(CNC(C(CC)C)=O)=O)cc(F)cc(Cl)c1 c1(C(N2C(C3(NC(COC)=O)CC3)CCC2)=O)cccc2c1OC(C)C2 N1(C(CCOc2ccc(CC)cc2)=O)CCN(C(=O)C2=NOC(C)C2)CC1CF C1(NC(C2N(C)CC(C)(C)C2)=O)CC12CCN(C(c1ccn(C3CC3)n1)=O)CC2 c1(CN2CCN(C(c3ccc(C(C)(C)C)[nH]3)=O)C3C2C3)cc([N+](=O)[O-])ccc1Cl C1(OC)CC(CNC(c2sccc2C2CC2)=O)N(C(C2CC(C)(C)C2)=O)C1 C(=O)(CC(C)(C)C(F)F)NC(CC(=O)NC1C(SC)CCC1)C(C)C S(=O)(=O)(c1cc2oc(=O)[nH]c2cc1F)N1C(C(=O)OCC)CC(C)CC1 N1(C(C(C)Cc2cnc[nH]2)=O)CC(O)CC1CNC(c1ccnnc1O)=O c1(CNC(C2CC23CCOCC3)=O)cccc2nn[nH]c12 N1(C(C(C)N(c2ccc(Cl)o2)C)=O)CCC(NC(=O)Cn2cnc(=N)[nH]2)CC1 Cc1cc(C(N2CC(NC(=O)C(C)(C)CC3CC3)CC2CO)=O)nc(O)c1 N1(C(C2CC(=C)C2)=O)CCCC(C)(NC(C2CCCCN2S(C)(=O)=O)=O)C1 C=CC(CCC)CC(=O)NCCCCCCNC(c1cc(F)ccc1OCC)=O C1(NC(c2ccon2)=O)CC2CC(NC(C3CCC3c3ccc(F)cc3)=O)C1C2 N1(C(C(C)CC(N)=O)=O)CC2CCC1(CNC(=O)CSCCN(C)C)CC2 c1(C(N2CC3(C(NC(CC(C)(C)OC)=O)CC3)C2)=O)cc(F)c(F)c(O)c1F C1(OC)C(NC(CCC2OCCO2)C(=O)Nc2cc(F)cc(Cl)c2)C2CCCC12 C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(=O)C(CO)N(C)C)CCC1C c1(C(=O)NC(C2OCCN(C(CNC(=O)OC)=O)C2)C)cc(=O)c(OC)c[nH]1 C1(C(N(C)CCNC(=O)C=Cc2ccc(O)cc2)=O)CCc2c(cnn2C)C1 C1(CC)CCC(C(N2CCC(OCCNC(=O)CN3CCNC3=O)CC2)=O)CC1 C(C(O)CC(=O)N1CC(CN=[N+]=[N-])C1)NC(C=CC1(C)COC1)=O C1(C(N2CC(NC(C(CC(C)C)N(C)C)=O)(CSC)C2)=O)CN2CCN1C(C)C2 CCC(=O)CCC(=O)NC(C)(CSCOC)C(=O)N(CC(O)CN(C)C)C c1(C(=O)NC2C(C(=O)NCCCC(=O)OCC)C2)cc(O)c(OC)c(O)c1 N1(C(c2c(C)snc2)=O)CCC(C(=O)NC2CCC(CO)C2)CC1CC c1(C(C(=O)N(C2CCN(C(C3CC34CCOC4)=O)C2)CC)C)ccc(C#N)cc1 c1(C(=O)NC2C(CNC(c3cc(C)nc(O)n3)=O)C2)ccc2oc(C)nc2c1 C(C(C)(C(=O)NC1CC(C)OC1=O)NC(C1C2CC(=O)CC12)=O)SC c1(OCC=C)ccc([N+](=O)[O-])c(C(N2CC(CNC(=O)C(C)(C)C)C(C)C2)=O)c1 c1(C(=O)NCC2C3CN(C(CNC(=O)OC)=O)CC32)ccc2oc(O)nc2c1 c1(CC(=O)NC2(CNC(C3C(OCC)C3)=O)CCC2)ccccc1SCC N1(C(CCC2(C)CN(C(=O)C3=CCSC3)C2)=O)CCOCC1C1CC1 C(=O)(C(F)C(C)CNC(=O)C=Cc1ccco1)N1CC(O)(CCC)C1 C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(=O)CCSCCCC)CC2)C1 c1(C(=O)NCC(CNC(C(C)OCC)=O)C)cccc(NC(C2CCC2)=O)c1 Cc1cc(C(=O)NC2CC(CNC(=O)C(F)(F)CO)C(O)C2)c2ccccc2n1 c1(CC(=O)NC(C2CCN(C(C3CC34CCOC4)=O)C2)C)c(F)cccc1F c1(OCC)ccc(CCC(C)NC(c2cnc(-c3ccccc3C)s2)=O)cc1 C1(N(C(=O)C=CC(F)(F)F)CCC)CCN(C(=O)CCCN2CCCC2)C1 c1(OCC(=O)NC2C(NC(C3(C)CC(F)(F)C3)=O)CCOC2)ccc(F)cc1Cl CC1CCC(O)C(NC(C2(NC(c3cc(O)nn3C)=O)CC(CO)C2)=O)C1 N1(C(c2cc(C)ncc2C)=O)CCN(C(C2(F)C(C)(C)C2(C)C)=O)CC(C)(C)C1 CC1(C(N2CCCC(F)C2)=O)CCCN(C(=O)CCS(C)(=O)=O)C1 C1(CNC(C(CCC2CC2)NC(=O)C(F)c2cc[nH]n2)=O)CC2(CCO1)CC2 c1(C(N2CC(O)(C(C)NC(C3C(=C)C3)=O)C2)=O)c(CNC(=O)OC)cccc1F C1(NC(c2cc(CO)on2)=O)CC2CCC(C1)N2C(C1C=CCS1)=O N1(C(C(NOC)=O)=O)CC2CN(C(=O)CCn3ccnn3)CC(C1)O2 c1(CC)cc(C(=O)NCC2(C(=O)NC3CC4CCC(C3)S4)CC2)ccc1F N1(C(c2ccc(C(C)C)c(Cl)c2)=O)C2CCC1CN(C(C1CC(CF)C1)=O)CC2 C1(NC(c2c(CCC)cccc2)=O)CN(C(=O)CCCN=[N+]=[N-])CC(C)(C)C1 c1(CC)c(C(=O)NCC2C3CN(C(c4cccc(C)c4N)=O)CC23)cccc1F C1(C(=O)NCC2CN(C(Cc3ccc(C)nc3)=O)CC2O)CCCCCCC1 Cc1nc(C)c(C(=O)NCC#CCNC(c2ccc(C(C)(C)C)nc2)=O)o1 C(=O)(CC(O)C(C)(C)C)NCC1CCCN(C(c2c(Br)cn(C)n2)=O)CC1 c1(C(N2CC(CC(CNC(C3C(=C)CC3)=O)(C)C)C2)=O)ccc(CCC)cc1 Cc1[nH]nc2c1CC(C(=O)N(C)CCN(C(=O)CC(=O)OC(C)(C)C)C)CC2 c1(C2(C(=O)NC3CCC(CNC(C4CCC(CC)O4)=O)C3)CC2)ccc(F)cn1 c1(C(=O)NC2CN(C(c3cccc(OC)c3O)=O)C2)cc([N+](=O)[O-])ccc1C C1(C(=O)NCc2cccc(OC)c2)CC2(CC2)CN1C(C1C(C)(C)C1(C)C)=O C1(CCOC)CN(C(C2CCN(C)C2=O)=O)CCN1C(c1c(OC)noc1C)=O Cn1cc(C2=NOC(C(=O)NC3CN4CCC3(C)CC4)C2)cn1 C(CCCCCNC(C1CCN(C2COC2)C1)=O)N(C)C(C1(C)CCCN1C)=O C(C(O)(CNC(=O)CCCC)CO)CC=CC=CC(=O)N(CCC#C)C C1(CNC(c2cn(C(C)C)nn2)=O)(CO)CCN(C(c2ccnc(O)c2)=O)CC1 c1(CCC(=O)NC(C(C)NC(CCCSC)=O)(C)C)ccc(Br)cc1 N1(C(c2c(C)nc(O)[nH]2)=O)CCN(C(c2cnn(C)c2N)=O)C2CC12 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCC2(CC(NC(CC3(OC)CCC3)=O)C2)C1 C1(C(=O)NCC2C(NC(C=CC(CC)=CC)=O)CC2)COc2ccc(O)cc2O1 c1(OC)cc(OC)c(Cl)c(C(N2CCN(C(C3COCCO3)=O)C3CCC23)=O)c1 C#CC1CC2CCC1N(C(C1CCCCC1(C)NC(c1nc(C)oc1C)=O)=O)C2 c1(C(=O)OC(COC2C(C)CCCC2)=O)cc(C(F)(F)F)ccc1Cl S(=O)(=O)(c1cccc(F)c1C(=O)OCc1ccc2ccccc2n1)N(CC)CC N1(C(c2c(C)ncn2C)=O)CCC(NC(=O)CCC2CCCCC2)C(CO)CC1 C1(CC=C)(C(=O)NCC(c2nccn2C)CC)CCN(C(=O)CC2(COC)CC2)C1 c1(OCCCCCC)ccc2cc(C(N3CCCOC(C4CCC4)C3)=O)[nH]c2c1 N1(CC2=NOC(C)C2)CC2C(C(F)(F)F)(CCS2(=O)=O)C1.N1(C=O)CCCC1 N1(C(c2c(NCc3cccc(CC)c3)nccc2)=O)CC2COCC2C1 CCC(CC)(CC)C(=O)N1CC2(C1)CN(C(c1ccc(Br)c(Cl)c1)=O)C2 c1(NC(C=CC(C)NC(C2CC2(C)C)=O)=O)ccc[n+]([O-])c1 C1(CC)CN(C(c2cc(C#N)no2)=O)CCC1NC(c1ncn(C(C)(C)C)n1)=O N1(C(C2C(C(C)C)C2)=O)CC(C2(NC(C3COCCN3CC(F)(F)F)=O)CC2)C1 c1(C(CC)O)ccc(F)cc1.C1(N)CC(CN)C1 C(C(F)(F)CCC(=O)N1CC2OCCOC2C1)n1cc(C(C(C)=O)OC)nn1 C(CS(=O)(=O)CC(=O)N1CCC(N(C(=O)C(C)c2cccs2)CCO)CC1)OC C1(CNC(C2CC23CCCC3)=O)(NC(Cc2c(CC)nco2)=O)CC(C)(C)C1 N1(CC)CC(C(=O)NC2(CNC(C3CC3(C)C3CC3)=O)CCCC2)CCC1=O Cc1cc(CC(=O)NCCCC2CCCC2)n[nH]1.C(=O)(CC(=O)O)NCCOCC c1(C(N2CCN(C(C3C(=C)CC3)=O)CC2C)=O)cn(C)c(=O)nc1O c1(SC(c2nc(-c3ccnnc3)no2)C)ccccc1 C1(CC)CC(C(=O)N(C)Cc2ccoc2)CCN1C(=O)CCCC1CCCO1 N1(C(CN(C)C(=O)NC2CC2)=O)CCC2C(C1)CN2C(=O)Cc1csc(NC)n1 N1(C(c2c(C(C)C)con2)=O)Cc2nccn2CC(NC(=O)Cc2cscn2)C1 CN1N=CC(CC(=O)NCC(O)CC(=O)NC2CCN(CCO)CC2)C1=O CC(C)(O)C(O)CNC(C1COCCC1NC(=O)Cc1ccoc1)=O c1(N2CCCC(OC)CC2)nc(Nc2cc3nc(C)sc3[nH]2)nc2c1SCC2 c1(N2CC(OC3CCN(C(=O)CC4CC(F)C4)CC3)C2)ccccc1[N+](=O)[O-] CCC(C#N)(CC)C(=O)NCC1CC(NC(c2ccsc2Br)=O)C1 c1(-c2c(C(=O)NC(CCC(=O)OCC)C)cccn2)c(F)cccc1F CC(F)(F)CC(=O)N1CC(F)CC1C(=O)NC1CCN(S(C)(=O)=O)C1 C(=O)(C(CNC(=O)Cc1csc(C)n1)CC(C)C)NCCC1(COC)CC1 c1(CC)cc(C(N2C(C(=O)N(C(CC)CC)C)CC2C)=O)c(C)o1 C(=O)(C1=CCC2(COC2)OC1)NC(CCN(C)C(C1(Cl)CC1)=O)C(C)(C)C N1(C(CCCCN(C(C)=O)C)=O)CCC(C)C1CNC(c1cc(C)cs1)=O C(N=c1nc(N2CCC3(CCCO3)CC2)c2cnn(C)c2[nH]1)C1(C)CCN(C)C1 N1(C(c2c(C)nncc2)=O)CCCCCC1C(=O)N(C(C)C(C)(C)O)C CC1CC(NC(=O)C(=O)Nc2cnc3cnn(C)c3c2)CC(C)S1(=O)=O N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(CC(=O)Nc3cnccn3)C2)C1 N1(C(c2cc(C)on2)=O)CC(F)(F)CC1CNC(=O)CCCNC(=O)C(C)(C)C CC1CC(NC(=O)NC2(C(C3(n4cccn4)CC3)=O)CC2)CS1 c1(C(C)C)cnc(O)c(C(N2CCC(c3ccc(Br)cc3)(C(=O)O)C2)=O)c1 N1(C(CN2C(=O)NCC2)=O)CCN(C(=O)CCc2cccs2)C(C2CCCC2)C1 Cc1cc(C(=O)NC(c2ccccc2)CNC(c2ccnnc2)=O)cc(C)c1N c1(C(=O)NCC(C2CC2)NC(C2C(=C)C2)=O)cc(C)ccc1NS(C)(=O)=O c1(N2CC(CN(C)C(C3(F)CCC3)=O)OCC2)nc(Cl)ncc1Br C=CC1CN(C(=O)CC(O)CC)CC1NC(c1cn(C)cc1C(F)(F)F)=O N1(C(Cc2c(C(C)C)con2)=O)C(C(N2CCC2C(N)=O)=O)CCC12CC2 c1(C(=O)NC(C(C)C)CCNC(=O)C(C2CC2)C2CC2)ncccc1S(C)(=O)=O c1(C(N2CCC(NC(CSCCOC)=O)C2)=O)ccc(-c2ccccn2)c(F)c1 c1(C2(Cn3cc(C(C)NC(C(CC)OC)=O)nn3)CCCC2)ccc(C)c(C)c1 CC1COCC(CNC(C(C2(O)CCC2)NC(c2cnns2)=O)=O)O1 C1(C(=O)NCCN(C)C(c2csc(C(F)F)n2)=O)CC2C=CC1C2 N1(C(Cn2ccc(C)n2)=O)CCCN(C(=O)C=C2CCC(C)CC2)CC1C O=C(N=c1ccn(C(F)F)[nH]1)C1c2c[nH]nc2CN1C(=O)C#CC1CCCCC1 CCCC(F)C(=O)NC1CC(NC(c2c(C3CC3)cnn2C)=O)CC1O C1(C(=O)N)CCCCC(=O)N1.CC(C)(CNC(C1(C)CC1)=O)NC1CC1 C(=O)(C(C)CC(=O)Nc1cccc(NC(c2ccc(Br)c(C)n2)=O)c1)OC N1(C(c2ccc(C(C)=O)[nH]2)=O)CCN(C(c2cnn(C3CCC3)c2)=O)CC1CO C123COCC1CN(C2)C3=O.CC(C)CCOC1CC(N2CCCC2)C1 c1(C(N(C)CC2N(C(C(C3CC(F)(F)C3)OC)=O)CCC2)=O)snc(Cl)c1Cl N1(C(C(C)C)=O)CC2CC2(N(C)C(C2CCN(C(C)=O)C2)=O)C1.C(C)(C)(C)CC C(C(CC(=O)N1CCC1CNC(C1CC(O)(C(F)F)C1)=O)C(F)(F)F)N(C)C c1(C(N2CC(N(C)Cc3ncccc3F)C2)=O)ccc2[nH]nc(Br)c2c1 n1(N(C(=O)COCC2CCC2)CCNC(C=C(C)Cl)=O)ccc(C2CC2)n1.CC=C CCC(c1ccc(C)cc1)=CC(=O)NCCCN(C(=O)C(O)CC)CCO c1(C(N2C(C)CC(NC(Cn3c(C)ccc3C)=O)C2)=O)n[nH]c2c1CCCC2 C1(C(=O)NC(C(=O)NCCN2CCC(C)C2)Cn2cncn2)CSCC(=O)N1 c1(OC)nccc(=NC(=O)C2CCCC2NC(=O)CCc2ccc(C)c(C)c2)[nH]1 c1(COC)nc(NCc2cccnc2N)cc(N2CCSCC(C)C2)n1 N1(CC(=O)N(C)CC2(CNC(C(CCCC)F)=O)CC2)C(=O)NC(C)(C)C1=O N1(C(c2cc(C)n(C)n2)=O)CCC2CC2(NC(c2ccc3ncsc3c2)=O)CC1 C(=O)(CCN=C(NCc1ccc(C(C)(F)F)nc1)NCc1cnnn1C)N(C)C c1(C(=O)NCC(CCCC)NC(=O)CN2CC=CC2)[nH]c2ccccc2c1OC CC1CC(CNC(=O)CC2CCC(C)(C)CO2)CN(C(=O)Cc2cncnc2)C1 C=C1CC(C(=O)NCCOCC(=O)NCC(C2CCCO2)O)(C(F)F)C1 N1(C(c2cnc(C3CC3)nc2)C(=O)NCC)CC(C)CSc2ccccc21 O=C(CCCC1CCOCC1)NCC1CN(C(=O)CN2CSCC2=O)C1 c1(CC)ccc(Br)cc1C(=O)N(C)CCN(C)C(C1CCCC(C)C1)=O C1(O)(C(N(CCC(C)c2cn[nH]c2)C)=O)CC2(CCN(C(=O)OC(C)(C)C)C2)C1 C1(C(=O)NCCN(C)C(c2nnc(O)cc2O)=O)CCC(=O)N(c2cnn(C)c2)C1 c1(C(=O)NC(C(C)OC)CC(=O)NC2C3CCCOC23)cccc2ccnn12 CC(C)(CNC(C1CCC(SCCOC2CCOCC2)OC1)=O)C(=O)O N1(C(=O)C=Cc2ncc[nH]2)CCC(CNC(C2(Br)CC2)=O)CC1 c1(C(=O)NC2C(C)N(C(=O)CNC=O)CCC2)cc2cc(Cl)sc2[nH]1 C1(C(N2C(C)(CC)CC2)=O)CCC2(CC2)N1C(=O)C(C)n1cccn1 c1(CCC(=O)NC(CNC(C(C2CC(F)(F)C2)OC)=O)C)ccc(N(C)C)cc1 N1(C(C2C(CC)C2)=O)CCCC2CN(C(=O)CCCN(C)C)CC12 c1(NC(=O)CN2CCN(C(c3cnc[nH]3)=O)CC2=O)ncc(Cl)c(Cl)c1[N+](=O)[O-] CCC(CC(=O)NCC1C2CC2CN1C(=O)C=CCOCC(F)(F)F)SC C(=O)(C1=NOC(C)C1C)NC(C(C)C)(C)CNC(C1CC(C)(C)C1)=O C(=O)(C1=CC2CCCCC12)N1CCCC(CNC(COc2cn(C)nc2)=O)CC1 C1(F)(C(=O)NCC(C)(C2CC2)NC(c2ccc(CCC)[nH]2)=O)CC12CCCCC2 Cc1c(C2(N(C)C)COC2)n[nH]c1C(=O)NC1CC1CNC(=O)CC1CC(CF)C1 C12(CNC(=O)C(=O)NC3CC3c3ccc(C(F)(F)F)cc3)CCC(CO1)C2 c1(CC(=O)NC2CC2CNC(=O)C(F)(F)C(F)F)ccc(O)c(Cl)c1 C1(C(=O)NCC(C(N2C(CO)CC(OC)C2)=O)CC2CC2)CC(C)CC(=O)N1 C(=O)(CC(C(F)F)NC(=O)CCCCN(C)C)C1CC(C#C)NCCCC1 c1(OCC)ccc(C)c(-c2cn(CC(N3CCCOCC3C)=O)nn2)c1 CC1CN(C(=O)C(c2cccc(Cl)c2)O)CC1NC(=O)CO c1(NC2(CO)CN(C(COCCC)=O)C2)ncc(C#N)c2ccsc12 C1(C(C)C)OCCC1C(=O)N(CCC(=O)NCC(O)C1CC1)C Cc1cc(C#N)cc(C)c1CC(=O)NCC(C)CNC(=O)CO CC(C(=O)N1CCC(NC(=O)CNC(=O)CC(C)(C)C(F)F)CC1)P(C)(C)=O Cc1cc(C(=O)NCC2(C)CCCN2C(C2CC2c2ccncc2)=O)nc(C)n1 CC(CC(=O)NCC(C)(CO)NC(C1(Cc2cccc(Cl)c2)CC1)=O)C(F)F C1(CNC(COCCC)=O)CCCN(Cc2nc(Br)c(C)s2)C1 c1(C(N2CC(CCNC(CCc3cc(C)on3)=O)OCC2)=O)ccn2c1CCC2 CC1(C)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C1CNC(=O)C(O)c1ccsc1 c1(OC(C(=O)NCCN(C(=O)C(O)Cc2cnn(C)c2)CC)C)ccc(F)nc1 C12(C(N3CCCC(CC=C)(NC(c4ccc(F)s4)=O)C3)=O)CCC(C)(CC1)CO2 c1(C(C(=O)O)N(C(N)=O)CCO)ccccc1.CC(COC(C)(C)C)CN1CCCC1 Cn1nccc1CC(C(=O)N1CC(CCCC(=O)O)C1)NC(=O)OC(C)(C)C C1(CNC(COCC(C)C)=O)CCCCC1N=c1nc2[nH][nH]cc-2c(O)n1 c1(C(=O)NC2CN(C(c3ccc(F)s3)=O)CCC2CO)cc2ccnn2cn1 n1(CC(=O)Nc2cccc(-n3cccn3)n2)ncc2cc(Br)cnc12 N1(C(CCSCc2nc(C)c(C)o2)=O)CC(C)CC(C)C1 N1(C(C(CCC)OCC)=O)CC(NC(c2ccc(F)cc2O)=O)CC(O)C1 C(C)(C1CCCCC1)=CC(=O)N(CCCNC(C(CC1CC1)OC)=O)CCO c1(OCCOC)ccc(Cl)cc1C(=O)NCC(O)CNC(=O)Cc1cc(C)ns1 N1(C(C2CCCC(O)C2)=O)CC2(C(N3CCC3CO)=O)CC1CO2 C1(C(=O)NC2C(NC(COCCCOC)=O)C2)Cc2cc(OC)ccc2O1 C(=O)(C1=NC2=NC(C)(C(=O)O)CCN12)NCC#C.C12CCN(C1)C(=O)C2 C(=O)(C(N)CCO)NCC(Cn1cc(CC(C)O)nn1)OC.c12ccc(o1)C2 C=C(Cl)CC(C(=O)N(C(CCO)C(F)F)C)NC(=O)C(F)=CC CCCCC(C)(C)NC(=O)CCCn1cc(CN(C)C)nn1 C1(COC)CN(C(=O)CCNC(C2CCCO2)=O)CCN1C(c1cnn[nH]1)=O C1(C2CCCN(C(=O)Cc3cccnc3)C2)(NC(=O)CCCF)CC1 C1(F)(C(N(CCC(C)O)C)=O)CCCN(C(C2CC23CCCC3)=O)C1 N1(C(C(C2CCC2)OC)=O)C2CCC1CC(O)(CNC(c1c[nH]nc1C)=O)C2 c1(CC(N2C3C(NC(C4(Cl)C(C)(C)C4)=O)CC(C3)C2)=O)nsc2ccccc12 c1(COC)cc(C(=O)NCC2(F)CC(NC(=O)C(C)Cc3ccncc3)C2)on1 C1(NC(C2N(CCC)CCC2)=O)CC2CCC1CN(C(C1CC(OC)C1)=O)C2 c1(OC)ccc(-n2nc(-c3ccc(Cl)s3)nc2Cc2cn(C(C)C)nn2)cn1 n1(CC(N2C(CCNC(C3(CC)CC3)=O)CCC2)=O)ncc(C#N)c1N N1(C(C2CC(F)(F)C2)=O)CCCC(NC(C2CCCN2C(c2cccs2)=O)=O)C1 c1(C(N2CCC(O)(C(=O)Nc3ccnc(Cl)c3)C2)=O)ccc(C(F)(F)F)cc1O N1(C(=O)NCCC2CC2(Br)Br)CC=CCC12CCOC2 C(=O)(C1CCCc2nn[nH]c21)NC1CC(F)(CNC(C(CSC)OC)=O)C1 CCC(C)C1CCN=C2C=CNC=C2S(=O)(=O)N1.C(C(C)(C)C(F)F)OC C1(NC(C2CN(C(C(COC)COC)=O)CC2(F)F)=O)CCCCC1N=[N+]=[N-] CC(C)S(=O)(=O)C(C)C(=O)NC1CCCCCC1CNC(=O)CCCS(C)(=O)=O c1(CC(C)C(=O)NCCC2CCCN2C(C2CCC(=O)N2)=O)ccc(C#N)cc1 C1(CNC(C2CC3(C2)CC3F)=O)CN(C(=O)CCc2ncc(F)cn2)CCCO1 C1(C(=O)NCC(C)NC(C2(c3ccccc3)CCC2)=O)CCc2ncnn2C1 c1(C(=O)NCCC2CCC(NC(C3(CC(C)C)COC3)=O)C2)cccc(CC)c1 c1(C(=O)NC(C(C)NC(c2cc(Cl)cnc2O)=O)C)[nH]c2ccccc2c1C#N c1(SCCC)ccccc1.C1(C)C=CCN1C N1(C(C2CCC2)=O)CCCC2(CC(N)CO2)C1.C(c1ccccc1)=C(CC)CC C(C(=O)NC(CC)CO)(C(C)C)NC(c1ccc(CC)s1)=O N1(C(c2cnn(-c3ccccn3)c2)C(=O)NCCCC)CCC(O)(CCC)CC1 c1(C(N(CC(CC)NC(=O)CC2CC(C)(C)CO2)C)=O)ccc2c(c1)CC2 c1(C(CC)NCCC(C)N2CCCC2)ccc(S(=O)(=O)NC2CCC2)cc1C#N S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)N1CC2CN(C(CCC(C)=O)=O)C2C1 c1(CCC)cc(C(=O)NCCC2CC(NC(c3c(C)cnn3C)=O)C2)n(C)n1 Cc1cc2c(NC(C3CCCN3C(=O)CCc3ccccc3F)=O)ncnc2[nH]1 c1(C(N2CC3C(C2)N3C(C2CC2(F)F)=O)=O)ccc(F)cc1Br C(=O)(CC(C)(C)CN(C)C)N1CC2C(C(=O)NC(c3cn(C)cn3)C)(C2)C1 CC(C)S(=O)(=O)CC(=O)NC1CC2CC(NC(c3ccccn4nnc3-4)=O)C2C1 C1(NC(CN(C(C2CCN(CC)C2)=O)CC2CC2)=O)CCCCCCC1 N1(C(C=CC)=O)CCCC(C2CCN(C(c3c(Br)n[nH]c3C)=O)C2)C1 c1(C(=O)NC(CNC(C(C)C(F)(F)F)=O)C(C)(C)C)ccc2cncn2c1 C=C(C)CCCC(=O)N1CCCC1C(C)(C)NC(C1CCS(=O)(=O)N1C)=O N1(C2CN(C(C(COC)C)=O)C2)CCN(C(C2(CN(C)C)CCCCC2)=O)CC1 C1(C(=O)NCc2nnc(C)n2C)N(C(=O)CN2CC3CC3C2)CCCC1(C)C CC1(C)CC=C(C(=O)NCC2CC2CNC(=O)COc2ccc(Cl)cc2Cl)CC1 c1(OC)ccc(CN2CCC(O)(c3ccc(C(F)(F)F)cc3)CC2)cc1I N1(C(c2cc(CC)no2)=O)CCC2(CCCN(C(=O)CCOCC(F)F)C2)C1 c1(CC)ncnc(CC)c1C(N1CC(CCNC(=O)CC2CCCO2)C1)=O N1(C(C2(C)CCSCC2)=O)CCC2CC2(C(=O)NC2CCC3(CCCC3)C2)CC1 N1(Cc2nc(CC(=O)OCC)sc2)Cc2ccccc2C2(CCCC2)C1 C12(C(=O)NC3CN(C(c4ccc(OC(F)F)cn4)=O)C3)CCCC1C2(F)F C1(CC=C)CCCCC1NCc1ccncc1OCC#N C(C(C)C(C)C(=O)NC1CCC(CNC(c2cccc(=O)n2O)=O)C1)OC CC1(O)CCC(C(N2CC(NC(=O)C(N)=O)C3(CC3)C2)=O)CC1 c1(N2C3CN(C(c4cnc(C)[nH]4)=O)CC32)c(Br)cc([N+](=O)[O-])cc1[N+](=O)[O-] c1(C(=O)NC2C(C)CCN(C(C(C(C)C)O)=O)C2)cnn2ccn(C)c12 CCC(C)C(O)C(C)C(=O)NC1(CC(=O)NCC2CC(CO)CO2)CCC1 C1(C(N(CC(COC)O)C)=O)CC2(CCC2)CN1C(C1(O)CCOCC1)=O c1(C(=O)NC(C)(CNC(=O)C(O)C2CCCC2)CO)ccnc2ccc(O)cc12 N1(C(CCOC)=O)CCN(CC2(NC(=O)C(C)(C)CNC(C)=O)CC2)CC1 CC(C)CC(CNC(=NCCF)NCc1nn(C)cc1Cl)CCO c1(NC(N2CCCC(C)C2)CC)nc(=NC)[nH]c(=NCc2ccc(N)cc2Cl)[nH]1 N#Cc1cc(C(C(=O)NC2CCC2)NC2C3COCC23)ccc1F CC(CC(=O)NC1CC2C(C1)C2(F)F)C(C)(C)NC(=O)CSc1cn[nH]c1 c12ccc3nc([nH]c3c1)N2.C(C=CC(=O)N(C1CCOC1)CCC)(CC)=CC N1(C(C23CCC(OC)C2C3)=O)CC2(CO)CC1(C(=O)NC1CCCCCC1O)C2 C1(C(C)(C)NC(c2cc(C)oc2)=O)CCN(C(c2cnsn2)=O)CC1 C(=O)(C1CCCc2c[nH]nc21)NC1C(C)(C)CN(C(c2cnn(C(F)F)c2)=O)C1 c1(C(=O)OCC(=O)N(C(C)N)C)cc(C2CCC2)nn1C.c1(S)nccs1 CCC(C)(C)C(=O)C(=O)NC1CCN(C(c2ccn3c2CCC3)=O)C(C)C1 C1(C(=O)NC2CC(NC(c3cc(Cl)ccc3F)=O)C2)CC2(CO1)CC(F)(F)C2 Cc1cc(C(=O)NC2CN(C(C3C4C(=O)OCC34Br)=O)C2)cnc1O n1(CC)c(CCNC(C2CCCCC2C(=O)O)=O)nnc1O c1(CN2CCC(NC(C(C)Oc3cccc(C#N)c3)=O)C2)cc(Cl)c(O)cc1F c1(C(=O)NCC2CCCN2Cc2ccccc2)c(C2CC2)cccc1F c1(OC)ccc2c(C(N3CCN(C(C4(CO)CCC4)=O)CC3C)=O)cnn2c1 C1(CN(CC(C)C)CC)CCN(C(=O)Nc2ccsc2OC)CC1 C1(C(=O)NCC23OCC(NC(=O)COC4CCCCC4)(C2)C3)Cc2nccn2C1 CC(C)CC(C)CC(=O)N1CCN(C(c2cc(CO)ccc2Cl)=O)C(C)C1 c1(C(=O)OC)ccc2sc(N(CC(C3CCOC3)O)CCO)nc2c1 N1(C(C(CC(F)F)N(C(CC(CC)C2CC2)=O)C)=O)CCC(C2(C)CC2)CC1 N1(C(CC(=C=C)C)=O)CCC2(CC1)CC2(CO)CNC(C1CC1c1ccsc1)=O Cc1cc(C(=O)N2CCNC(=O)C3CC(F)(C3)C2)ccc1F.C1(CF)CC1 c1(C(N2CCCC(NC(c3ccc(C(C)C)o3)=O)C2C)=O)ccc2cc[nH]c2n1 c1(CN2CC(C)CC(NC(CSc3cccc(C)c3)=O)C2)ccc(O)c(Cl)c1 C1(C(CC)CC)CCC(C(N2CCC(CNC(N)=O)C2)=O)CC1.C1(=O)CCCN1 N1(C(c2c(C)nc(C)o2)=O)CCN(C(C2CC2C(F)(F)F)=O)C(CCO)C1 c1(OC)cc(C(C)(C)CNC(c2ccc(=O)n(C3CC3)c2)=O)ccc1C(=O)O c1(C(=O)NC2CC(CNC(C3(C)CC=CCC3)=O)C(O)C2)ccc(P(C)(C)=O)o1 C1(NC(c2c(C)snn2)=O)CC1C1CCCN(C(=O)CSc2nncs2)C1 N1(C(CC(=O)NC)=O)CCC(NC(=O)CC2CCC3(CCC3)O2)C(C)C1 C1(NC(C2C(OC)CC2)=O)CN(C(=O)Cc2cc(Br)cs2)CCC12CCC2 CC(C)CC(CNC(=O)C=CC1CCCN1C)C(=O)NCC1(CO)CCCCC1 c1(NC(=O)CC2(O)CCN(Cc3cnc(Br)s3)CC2)[nH]nc2ncccc12 CC(C)(CS(C)(=O)=O)C(=O)N1C2CCC1CC(CNC(=O)CCc1ccoc1)C2 C1(NC(C=Cc2n(C)ncc2)=O)CN(C(c2sccc2C#N)=O)C2CCCC12 c12cc(cc(F)c1)-n1nnnc1CCC2.C1(c2ccn(C)n2)(N)CCOCC1.C(C)(C)(C)O c1(NC2(C)CC(C)C2)cc(N(C)C)cc(F)c1 c1(C(N(C2CN(C(C3CCCOC3)=O)CC2(C)C)C)=O)c(F)ccc2c1OCO2 c1(OCC(=O)NCCN(C(C)C)C2CC2)ccc2ccccc2c1Br C(CCCCCCO)NC(C(C)N(C(C1N(C(C)C)CCC1)=O)C1CC1)=O N1(C(C(C)Cc2ccccn2)=O)CCCC(CCNC(c2nocc2Cl)=O)C1 C1(CC(=O)NC2(C#C)CCOC2)CN(C(=O)Cn2nnnc2C)CCC1C c1(C(=O)NC(C2CN(C(C3CC(S(C)(=O)=O)C3)=O)C2)C)cc2cc(F)ccc2[nH]1 CC1CN(C(C2CCS(=O)(=O)CC2)=O)CCN1C(C1(C)COC1)=O Cc1c(Cl)cnn1CC(=O)NCC1CN(C(=O)Cc2cccs2)CC1C CC1(C)CCN(C(=O)CC2CSCCO2)C1C(N1CC(C2CC2)=NO1)=O c1(C=O)ccc(C)c(C)c1.C1(N(N2CCC2C(C)C)CC)CCC(C)(C)C1 C1(C)(CC(=O)OC)CC(F)(F)CN1C(=O)NC(C)CCc1ccco1 CC1CN(C(=O)CC(C)(C)C#N)CCC1CNC(=O)CCC1CC(F)(F)C1 N1(C(CCC2CCN(C(c3c(C)[nH]c(C#N)c3)=O)CC2)=O)CCN(C)CC(O)C1 c1(C(=O)NC(CNC(c2ccc(C)s2)=O)(C)CO)sc(N2CCOCC2)nc1C C12(NC(c3c(C)ocn3)=O)CCCN(C(=O)COCC3CCCC3)CCC1C2 c1(-c2ccc(NC(C(C)CC(N)=O)=O)cn2)cccc2c1nnn2C C1(C(=O)Nc2ncc(C)nc2)CC12CCN(C(c1ncccc1Br)=O)C2 N1(C(c2c(C)nc[nH]2)=O)CCC(NC(=O)C(O)Cc2cnc[nH]2)C12CC2 C(=O)(CC(C)CC(C)(C)C)N1CCC(CNC(c2cn(CCOC)nc2C)=O)C1 C(CC(C)C)(C(=O)NC1CCCN(C(=O)C(=O)NCC(F)(F)F)C1)OC N1(C(c2c(C)ccnn2)=O)CCN(C(c2ccc(=O)n(C)n2)=O)C(C(C)C)C1 c1(OC)ccc(CC(=O)NCCC2CCCN(C(c3csc(C)n3)=O)C2)c(C)c1 C1(C(=O)NCCOC2CCN(C(C3C(OCC)C3C)=O)C2)CCN(C)C(=O)C1 c1(-c2nc(C(CC)C)nn2-c2ccc(Cl)nc2)cc2c(Cl)c(Cl)ccc2[nH]1 CC1CC2(CO1)CN(C(C1COCCC1NC(=O)CC1=CCCC1)=O)C2 C1(NC(c2cncc(C)c2)=O)CN(C(=O)Cc2nc(C)sc2C)CCC1F C12CC3(CC3)CN1C(=O)C(C)N2.C1(COC)CN(C(c2ccccn2)=O)CCO1 N1(CC(=O)N(C2CC2)Cc2ccccc2)CCCC1C1CCCC1 C1(NC(C(CC(C)C)(C)C)=O)CC2(CCCN(C(c3nnc(S)n3C)=O)C2)C1 C(=O)(CCCC(C)(F)F)NC1C2N(C(C(CCN(C)C)O)=O)C(CC2)C1 Cc1ccc(C(=O)NC2C=CC(CNC(C3CC(C(F)F)C3)=O)C2)n1C c1(NC(=O)CCn2cncn2)ccc2c(c1)CN(C(=O)Cc1ccc(F)c(Br)c1)C2 C1(C(=O)NC(CC)C(N)=O)CCN(C(=O)C(O)CC2CCCC2)CCO1 C1(OC)CC(NC(C2CC(O)(C(F)(F)F)C2)=O)CN(C(=O)CS(=O)(=O)NCCO)C1 c1(C(=O)NC2(CC=C)CN(C(=O)C(C)C#N)C2)ccc(C(C)C)cc1 C(=O)(C(O)C(F)(F)c1ccccc1)Nc1ccc(CN)cc1 Cc1ccc(C(N2CCC(CO)(NC(c3cc(C#N)[nH]c3C)=O)C2)=O)c(F)c1 c1(C(N2CC(NC(COCC(C)C)=O)CC23CCC3)=O)cn2c(n1)C(C)CCC2 Cc1nn2cc[nH]c(=O)c2c1C(=O)N(CC(O)CNC(=O)CN1CC=CC1)C C1(C(N2CC3(CC(NC(C4(C(N)=O)CC4)=O)C3)C2)=O)COc2ccccc2C1 N1(C(Cc2c(C)n[nH]c2)=O)CCCC(C)(C)C1C(=O)Nc1cnn(C(F)F)c1 c1(CC(=O)NCCN(C(=O)C(C(C)O)N(C)C)CC)ccccc1S(C)=O N1(C(c2c(C#C)cn(C)n2)=O)CCC2CC(C1)CN(C(c1ncsc1C)=O)C2 N1(CC)CCCC(C(=O)NCC(F)CNC(c2ccc(OC(F)(F)F)cn2)=O)C1 C(CCCCCC(=O)N1CCCC1C1CCN(C(C2(C(F)F)CCC2)=O)C1)SC c1(C(=O)NCC(C)NC(=O)COc2cncc(Cl)n2)cc2ccc(O)nc2s1 c1(CC)cc(NC(C2CC3CC3N2C(C2CCCS2)=O)=O)cc(F)c1 c1(OC)ccc2[nH]c(CN3CC(F)CC3C(=O)Nc3cc(C)cc(Cl)c3)cc2c1 C#Cc1cccc(CC(=O)NCC2CCN(C(C3CCS3(=O)=O)=O)CC2C)c1 C1(=O)CS(=O)(=O)N1C1CC1.c1(N(C(C)=O)C2CC2)c[nH]nc1-c1cccnc1 Cc1cc(CC(C2CC2)NS(=O)(=O)C(C)C(=O)N(C)C)ccc1F c1(CC(=O)NCC2OCCCN(C(CCC(C)(C)F)=O)C2)ccc2ccoc2c1 N1(C(CC(C(C)C)O)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccc(F)cc1F N1(C(c2ccn(C(C)C)c2)C(=O)NCCOCC)CC2CS(=O)(=O)CC2C1 c1(-c2n(-c3cccc(SC)c3)nc(CCO)n2)csc2ncnc(O)c12 CC(C)(C)CC(O)C(=O)N1CCCC1C(=O)NCc1cn(C2CC2)cn1 c1(C(C(=O)NCC(=C)C)N2CCC2c2cc(F)ccc2F)ccnc(OC)c1F N1(C(CC(C(C)C)OCC)=O)CC2CN(C(c3ccnc(F)c3O)=O)CCC12 CCCS(=O)(=O)CC(=O)N1CCC(CC)(NC(c2nc(C)c(C)[nH]c2=O)=O)CC1 Cc1cc(CN2CCC(NC(c3nc(C)c(C)nc3C)=O)C(O)C2)cc(C)c1Cl CCC(C)C(O)C(=O)NCCCN(CCCCSC)C.C(=O)(C(C)CN(C)C)N CC(CCNC(=O)CC1CCCCO1)CCNC(c1conc1C1CCC1)=O N1(C(CSCC=C)=O)CCC12CCCN(C(=O)C(c1ccccc1)OC)C2 C1(C(N(C2CCN(C(C3CC34CCOC4)=O)CC2)CCC)=O)CC2(CSC2)C1 C1(=CC(=O)NC(C2CCCN(C(c3ccnnc3)=O)C2)C)CCC(C)(C)CC1 C(=O)(C(O)C(C)(C)C)N1CC(CCC)C(C(=O)NCCC(C)(C)OC)C1 C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CCC(CNC(C(CC)OCC)=O)C1 C1(CC)CN(C(c2ccccc2)=O)CCC1NC(C12CC(C(C)C)(CO1)C2)=O c1(C(=O)NC2C(NC(C(C)O)=O)COC2)ccc2c(c1)CC(C)(C)C2 C1(CC)CCN(C(=O)C(=O)N(C)C)C1C(N1CCOCC1CC1CC1)=O c1(NC2N(CC)CCC2)nc[nH]c(=NCC2(OCC)CCCCC2)c1C CN1CC=CCC1CC(=O)NC1(CNC(=O)C(c2cncn2C)O)CCOC1 c1(CC(=O)NCC(C)N(C(=O)CC23CCC(CC2)OC3)C)ccc2c(c1)OCO2 N1(C(c2cc(SC)oc2)=O)CC(NC(c2ccnc(C3CC3)n2)=O)CC1C CN1CCc2cc(C(=O)NCCC3(NC(=O)C4CC4)CCCC3)ccc21 C(=O)(CC1CCOc2ccccc21)NCC(C)(CO)NC(=O)CCc1cn[nH]c1 c1(NC(CC2CCN(S(CCOC)(=O)=O)CC2)=O)cc2ccc(Cl)cc2nn1 n1(CC(N2CCN(C(CS(CC)=O)=O)CC2CC(F)F)=O)ncc2ccccc12 c1(NCCC2CCC(NC(c3c(OC)nn(C)c3)=O)C2)ncnc(Cl)c1C C1(C(=O)NC2(CN(C(C(C3CCOCC3)OC)=O)C)CCC2)CCC(F)CC1 C1(C(=O)NC(CCN(C(C(C)NC(C)=O)=O)C)C)CC2CS(=O)(=O)CC2C1 CCCCC(C)C(=O)NCCOCCNC(c1cnc(C(C)(C)C)nc1)=O C1(NC(C2CCN(CCC)CC2)=O)CC2CC1CN2C(=O)CC(F)F c1(C(=O)NCCC(C)NC(=O)COCC=Cc2ccccc2)cccnc1S C(C(CNC(=O)CC1CC1(C)C)C(F)(F)F)NC(CCc1cnc(C)s1)=O C1(C(N(CC(C)OC)C)=O)CC(C)(C)CCN1C(=O)Cc1scnc1C N1(C(=O)Cn2nc(-c3cccs3)oc2=O)CC2CCCN2c2ccccc21 CN1CCCC(C(=O)N(CC(O)CN(C)C(c2cc(N(C)C)n[nH]2)=O)C)C1 CON(CCC(=O)NCC(C)C(C)(F)F)C(=O)C1CN(C)C(=O)N1 C(=O)(CCCC(C)Nc1ccc(C)c(NC(C)C)c1)OCC c1(CC)nnsc1C(=O)NC1CCN(C(c2ccc(C3CC3C)o2)=O)C1 n1(CC)ncc(C(N2CC(NC(=O)CC3CCSCC3)CC2C)=O)c1Cl c1(C(=O)NC2(CNC(CC(=C=C)C)=O)CCCC2)cccc2c1NCC(C)C2 c1(C(=O)NC2C3C(C(N(C)C)=O)C4C(C3)C24)cc2ncccn2n1 c1(C(=O)NC2CC(C)CN(C(C3CC(F)(F)C3)=O)C2)nn(C)c2ccccc12 Cc1cc(NC(C2CCC(NC(=O)C=Cc3ccccc3)CO2)=O)nc(Cl)c1 c1(C(N(CCCN2CCN(C(C3(C)CCCC3)=O)CC2)CO)=O)ccnc(Cl)c1Cl C1(C)(CC)CC(NC(C2CC(F)(CO)C2)=O)CN1C(=O)C(C)=C1CC1 C1(C)(COC)CC(NC(=O)Cc2cnc(C)[nH]2)CN1C(=O)C=CCn1cncn1 c1(C(C)=O)ccc(C(=O)NC(c2ccccc2)C(=O)OC(C)(C)C)s1 C(=O)(C(C)(C)C1CCCN1C(=O)C(C1CCOCC1)=O)N(C(C(C)C)C)C c1(C(=O)NCCOCCN(C(C2C(=C)C2)=O)C)cn2cc(C)c(C)cc2n1 C1(C(N(C(C=C)C)CCCC)=O)CC(CNC(C2(COC)CC2)=O)C1 N1(C(c2nccc(C)c2F)=O)C(C)CC2CN(C(C3C4CC(=O)CC34)=O)CC12 CC1CN(C(=O)CC(F)(F)C(F)F)CCCN1C(c1cnc(NC2CC2)s1)=O Cc1cc(C(=O)NCCN(C(=O)CC2CCCCCC2)C(C)C)ncc1C(N)=O c1(C(=O)NCC2C(C)(C)CN(C(c3csnn3)=O)C2)cccc2[nH]ncc12 N12CCc3onc(c3C1)C2=O.N1(C(C(C)NC(C)=O)=O)CCCCC1CCO CCCC(C(=O)NCC(O)CNC(C1CC(F)C1)=O)S(N)(=O)=O c1(C(N2CC(CNC(c3n(C(C)C)ccn3)=O)C3C2C3)=O)cccc2nsnc12 C1(F)(CNC(c2c(=O)ccn(C)c2)=O)COCCN(C(=O)C2=NNC(=O)C2)C1 C(=O)(C(C)(C1CCC1)NC(=O)CN(C)C)NCCSCCCC C(C1c2ccccc2CCN1C(c1cc(O)cs1)=O)NC(C1CCCC2CC12)=O C(=O)(C(C)CC(=O)N1CCN(C(=O)COc2cn[nH]c2)C(CO)C1)OC N1(CC2C(c3c(OC)cccc3)(C)C2)CCS(=O)CC1c1ccccc1 O=C(CCCC(F)(F)F)NC1CN(C(=O)Cc2csc3sc(C(C)C)cc23)C1 c1(C(=O)NCCNC(c2nc(C)sc2)=O)ccccc1-c1nc[nH]n1 c1(NC(C2CCCC(NC(CCC)=O)C2)=O)cccc(O)c1Br C1(C(C)(C)C)CC(CNC(C2CC=CC2)=O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 C1(C2CCN(C(C3CN(CP(C)(C)=O)C3)=O)C2)(NC(Cc2c(C)ocn2)=O)CC1 c1(C(=O)NCC2C(NC(Cc3c(Cl)cn(C)n3)=O)CCC2)ccc(S(C)(=O)=O)[nH]1 CCCCCC(F)C(=O)NC1CCC(CC(=O)Nc2cnc(N(C)C)nc2)C1 CC(CNC(=O)N(CCN=[N+]=[N-])CCO)CC(F)(F)F C#CCC(C(=O)N(C(C)CNC(c1cccnc1N(C)C)=O)C)C1CC1 O=C(NNc1ccc(Cl)nc1)c1cccnc1Br c1(C(CC2CCCC2)NCCC(C)C)nnnn1C1CCCC1 N1(C(CCCCN(C)C)=O)CC2OCCN(C(=O)Cc3ccc(=N)[nH]c3)C2C1 c1(C(N2CC(C)(OCC(=O)N(CC(O)COC)CC)C2)=O)c(C)n[nH]c1C C1(NC(C(CNC(C)=O)(C)C)=O)COC2(C1)CN(C(=O)CC1(C)CC1(Cl)Cl)C2 C1(C(=O)OC)CC2CC1N(C(=O)Nc1c(-c3n[nH]c(OC)c3C#N)cccc1)C2 C1(F)(C(=O)NCCCCCNC(c2cccc(CC)c2F)=O)CC12CCCCC2 N1(C(c2c(O)ncc(CC)c2)=O)CC2CCCC(NC(C3CC3C)=O)(C2)C1 C1(C)(C(=O)NCC(CC)NC(=O)CC=C(C)C)CCc2ccccc21 c1(Oc2ccccc2Cl)nc2ccccc2o1.C(CCO)N(C(C)=O)CCCN c1(C(N2CC(NC(Cc3ccc(OC)nc3)=O)C(O)C2)=O)cnc2ccnn2c1 C12(CCOCC1)C(=O)N1C(C)CC(C1)CNC(=O)CN2.CCS(=O)(=O)CC c1(CC(=O)NC2CN(C(C(C)(O)CC(F)F)=O)C2)csc2ccc(Cl)cc12 N1(C(c2ccnc(F)c2)C(=O)NCCOCC)CCOc2ccc(F)cc21 C1(C(=O)NCC2(O)CCN(C(CCc3cc(C)on3)=O)C2)CCS(=O)(=O)C1(C)C c1(OC)ccccc1C(=O)NCC(C)(F)CNC(=O)C(C)(C)OC(C)C C1(NC(=O)Cc2cccc(Cl)c2)CC2CC1N(C(c1cccc(CN(C)C)c1)=O)C2 N1(C(c2c(CC)nccc2)=O)C2CCC1CN(C(c1cc(C(N)=O)no1)=O)CC2 c1(CSC)ccc2[nH]ccc2c1.C1(=O)N2CC(CO2)NC2CCC1CC2 N1(C(c2c(C)cc(C)s2)=O)CCC2(CCC2)C(CNC(C2CC(C)CCO2)=O)C1 CCC(CC)CC(F)C(=O)NCCCC(C)(C)C(=O)NCCc1ccc(C)s1 Cc1ccc(C(N)=O)cc1C(=O)NCC1(NC(=O)C(C)CC2CCC2)CC1 NC(=O)CCCC(=O)c1cn(C2CCOC2c2cncc(F)c2)nn1 C1(NC(c2ncc(OCC3CC3)cc2F)=O)CCCCN(C(c2cnc[nH]2)=O)C1 C(CNC(=O)CCc1nnc(C(F)F)o1)(CC(C)C)NC(C(CC)O)=O Cc1cccc(Br)c1C(C(=O)NC1CCC1O)NC(C1CCCCS1)=O CC1c2ccc(Cl)n2CCN1C(n1cc(-c2ccc(C3(CN)CC3)cn2)nn1)=O N1(C(CCCS(N)(=O)=O)=O)CC(NC(C2CC3CCC(C2)O3)=O)CC12CCCC2 c1(OC)cccc(CCC(=O)NCC2CCN(C(=O)CC3CCCC(C)O3)C2)c1 c1(C(N(C(c2ccccc2)CNC(C2(C#N)CC2)=O)C)=O)cnn2cccc(Cl)c12 C(=O)(NN=c1cncc(Cl)[nH]1)Nc1c(C(C)O)cccc1 CCCC(C)(O)CC(=O)NCc1cncc(C(N2CCC(C(=O)NC)C2)=O)c1 N1(C(C(C)NS(CC)(=O)=O)=O)CC(NC(c2csnn2)=O)C(O)C1 c1(CC)cc(C(=O)NCC2COC(CNC(c3ccc(OC)s3)=O)C2)on1 c1(C(=O)NCCC(C(C)C)NC(CCC)=O)c(C(=O)OC)sc2ccccc12 N1(C(c2c(CC)n[nH]c2)=O)CCC(NC(C2CCC(C3CC3)CC2)=O)C2(CCC2)C1 C(=O)(C1CCc2c[nH]nc21)NC1CCC(C)(NC(CCC=CC)=O)CC1 C(C)(CNC(=O)Cc1ccc(C(N)=O)cc1)(C(C)C)NC(C(C)OCC(C)C)=O N1(C(C(n2cnc(C#N)n2)C)=O)CCC(CNC(c2ccnnc2)=O)C1(C)C C1(C(=O)NC2CC(NC(c3ccc(Cl)cc3F)=O)CC2O)C(C2CC2)C1(F)F CCCCCCC(=O)NC(CC1CCOCC1)C(=O)NC(C)(C)CCCO CC1(C)COC(=O)C1NC(C1(NC(=O)COc2ccsn2)CC1)=O C=CCC(F)(F)C(=O)N(C)CCNC(c1nc(Br)sc1C1CCOC1)=O C=Cn1nccc1C(N1CCC(CNC(=O)C(C)C(=O)NC)(OC)C1)=O c1(CC(C(=O)NC(CCOC)CO)NC(C2CCOC(C)C2)=O)ccccc1Br CC(C)(C)C1=NOC(C(N2CC(CNC(=O)CCc3cnc[nH]3)C(O)C2)=O)C1 Cc1c[nH]c(C(=O)NCC(C2CCCC2)NC(=O)CC2CN(C)C2)c1 C(C(=O)NC(C1CCCCC1)CNC(C1CCSC(C)C1)=O)(C(C)C)SC c1(CNCC2(C(=O)Nc3cc(=O)cco3)CC2)cccc([N+](=O)[O-])c1 C1(C(=O)NCC(CN(C(=O)CS(N)(=O)=O)CC)(C)C)CCCCC(C)(C)C1 c1(NC(c2c(OC)ccs2)=O)ccc(NC(c2cnc(O)n2C)=O)c(C)c1 c1(CNC(CCc2cc(C)[nH]n2)=O)ccnc(Cl)c1Cl c1(CC(=O)NC2CC(NC(CC=CC(C)(C)C)=O)C2)cnc2cccnn12 CC(CC(=O)N1CC(CC(=O)Nc2cc(OC(C)(C)C)ccc2O)C1)C(F)F c1(OC)cc(C(=O)NC2CCCC2NC(c2ccc(F)cc2O)=O)cc(Cl)c1 C1(NC(C(C)OC)=O)CCOC12CCN(C(c1snc(O)c1Cl)=O)CC2 N1(Cc2ccnc(C)n2)CCC(CCNC(=O)C(C2CCOCC2)C)CC1 c1(C(=O)NC(C(=O)N(C)Cc2ccccc2Br)(C)C)ccn2ccnc2c1 c1(NC(=O)NC(C)(Cc2cccc(Br)c2)CO)ccc2ccccc2c1 C1(C2CCCCO2)(C(=O)NCC(C(C)C)NC(=O)CS(C)(=O)=O)CCOCC1 Cc1cc(NC(=O)CN(C(c2cccnn2)=O)CC2CC2)c(O)cc1F c1(C(c2nnnn2C2CCC2)NCCCC(F)F)ccc2ccncc2c1 Cc1ccc(Br)c(C(=O)NC2CCC23CN(C(=O)C(C#N)C(C)C)C3)c1 Cc1cc(C(=O)NCC(C)NC(c2coc(Cl)n2)=O)ccc1-n1cnnn1 C12(CC3CC3)CCN(C1)Cc1cn(nn1)C2.c1(C(=O)OC)ccn(C(F)F)n1 c1(C(N2CC(CNC(=O)CC3CC=CC3)CC(F)C2)=O)ncc(C2CC2)cc1F CC(C)(O)C(F)(F)C(=O)N1CCC(C)(CNC(=O)CN2CCC(O)CC2)C1 C1(NC(C)(C)COC2CCCOC2)CCS(=O)(=O)C1.N12CCC(C)(C1)NC2=O Cc1nc(C(=O)NCC(C2CC2)NC(=O)Cc2c[nH]nc2O)nn1-c1nc[nH]n1 c1(CC)ccccc1C(C)C.C12CCC(O1)C(=O)N1CCC(C1)CNC(=O)CC2 CC(CC(C)SC1CCC2(CCCCC2)O1)CC(C)(C)C C(=O)(CC(C)P(C)(C)=O)NCCOC1CCN(C(c2nccc(C)n2)=O)C1 c1(NCC(C)SC)nc(N2CCOC(c3nnc(C)o3)C2)nc2sccc12 c1(CCC(=O)NC2CCN(C(CSCC)=O)C2)cccnc1Cl c1(C(=O)NC2CCC(NC(C(C)OCCCC)=O)CC2)ccc(N)c(N)c1 N1(C(C2(CC=C)CN(C(=O)C3=CCSC3)C2)=O)CC2CC1CN2C C1(NC(c2nc(C)oc2)=O)C(C)CN(C(c2ccc(Cl)s2)=O)CC1C CCC(C)(C(=O)N1CC(F)(CNC(c2ccc(OC)c(C)c2)=O)C1)C(N)=O C(C(CC)(CC)C(=O)N1CCCC(C(C)(C)O)C1)NC(CC(CC)SC)=O C1(NC(c2scc(C)c2)=O)(CF)CCN(C(=O)CCn2nc(C)cc2C)C1 N1(C(c2ccc(OC)s2)=O)CCC(NC(=O)C(C2CCOCC2)C)C(F)C1 C1(NC(C2CC(C)(CC)C2)=O)CCN(C(C2CC(=O)NC(=O)N2)=O)CC12CCC2 C(=O)(C1=CCCOCC1)N(C1C2CN(C(C(COC)C)=O)CC21)C CN1CC(F)CC1C(=O)NCc1ccc(C(N2CCC(C)(C(N)=O)C2)=O)o1 c1(C(N2C(CC(N3CCC(C(N)=O)CC3)=O)COCC2)=O)cc(Cl)ccc1I O=C(C1CCCc2sccc21)NCC1=CCN(C(=O)C(F)C2CCOC2)CC1 N1(CCN(c2ncccc2F)CC(C)C)CC(C)OC(C)C1 c1(C(=O)NC2CC(CNC(c3n(C(C)C)ccc3)=O)C2)ccc(N)cc1[N+](=O)[O-] C(C)(CCC(=O)N1CCCCC1NC(C1(NC(C)=O)CC1)=O)SC c1(CC(C)C)cc(C(N2CC(N(C(=O)CC3C=CCC3)C)C(O)C2)=O)cc(O)n1 C(=O)(C(C1=CCC2CC2C1)N1CCc2c(CO)cccc21)NC C(=O)(C1=C(C)OCC1)N(C1CCN(C(=O)CC2COCC2O)CC1)CC#C N#CC1=C(C(=O)NCCOC2CN(C(C3(C(=O)OCCO)CC3)=O)C2)CCC1 Cc1cc(N(CCCC(C)C)C)n2ncc(Br)c2n1 C1(C(=O)NCC(CC(C)C)NC(=O)C=CC2CCOCC2)(OC)CCCCCC1 C(CN=c1[nH]cnc2c(Br)cccc12)(C(C)(C)C)NC(c1ccc(CCC)[nH]1)=O c1(CC(N2C(CNC(c3cc(C)sc3)=O)CC(O)C2)=O)c(C)nn(C(F)F)c1C CCCCC(=O)NCCCOCCN(C(C12CC(O)C1C2)=O)C(C)C c1(N2C(C3(NC(c4ccc(C#C)cc4)=O)CC3)CCC2)ncc([N+](=O)[O-])cc1F C(=O)(CC(F)(F)C(F)(F)F)N(C)CCOCCNC(=O)C(c1ccc(F)cc1)O C(=O)(CCS(=O)(=O)N(C)C)NC(C(C)(C)C)CNC(=O)CC1(O)CCOC1 c1(-c2cn(CC3CN(C(c4c(CC)ccs4)=O)C3)nn2)cccnc1C c1(C(=O)NC2CC(N(C(C3(CC)CCC(O)CC3)=O)C)C2)cc2cc(Cl)sc2[nH]1 c1(CC(=O)NC(C)CCN(C(=O)CC2CCCC2(F)F)C)ccc2c(c1)COC2 N1(C(C=C(C)C)=O)CCN(C(c2ccc(Cl)cc2)=O)CC1c1cn[nH]c1 c1(CC(C)C)nc(C2CC3(CCC3)C2)n(C2CCC2)n1.c1(C)ccccc1 C1(C(C(=O)NCC2N(C(C=NOC)=O)CC2)C)CCC(=O)N1C C12(CCNC(C3(CSC)CC3)=O)CCC(CC1)N(C(=O)CC1(N(C)C)CCC1)C2 C(C1=CCCCC1)(c1n(C(CC)(C)C)nnn1)NCC(=C1CCOCC1)Br Cc1ccccc1COC(C)C(=O)NC1(NC(=O)C#CC2CC2)CCOC1 c1(CNC(C(N2CCNC2=O)C)=O)ccc(C(=O)NCCC(=O)NC2CC2)o1 CCCC(CCC)CC(=O)N(CC(C)(C)C(=O)NCC1CSCCO1)C c1(C(N2C(C(=O)Nc3ccc(CO)cc3)CSCC2)=O)c(Br)ccc2c1OCO2 N1(C(C(C)NC(=O)C(C)(C)C)=O)CCC2(CC1)CN(C(=O)C(C)(F)F)C2 N1(C(C(C)(C)N(C)C)=O)CCN(C(c2cnn(C(C)(C)C)c2)=O)CC1 c1(C(=O)NC2CC(CNC(=O)C=C3CCSCC3)C2)ccccc1C1CCOC1 C(CC(C)C(=O)NCCN1CCN(C(C2CCC(N(C)C)CC2)=O)CC1)OC C#CC1(C(=O)NCCC2CCCN2C)CCN(C(=O)CC2CCCOC2)CC1 C1(C(N2CCCC(OCCC)C2)=O)CCN(C(c2cnncc2O)=O)CCO1 C1(c2n(CC)nnn2)(NCc2cc(C(N)=O)cc(Br)c2)CCC2(CCCOC2)C1 N1(C(C2N(C)CCOC2)=O)CC2(CNC(c3cncc(F)c3)=O)CC1CO2 n1(C(CCC)c2ccsc2)cc(C(C)NC(=O)CC2C=CCC2)nn1 c1(C(N(CCNC(=O)CC2CC=CCC2)CC)=O)nn(CC(C)C)cc1Br C1(C(N2CCCC(CNC(c3cc(C)c(Cl)s3)=O)C2)=O)CCCC12CCOCC2 CCC(CCCC(=O)N1CC(Cc2ccco2)C1)NC(=O)C(C)(C)N(C)C c1(C(=O)NC2(C3N(C(C4C(OCC)C4C)=O)CCC3)CC2)oc(C2CC2)nc1C N1(C(C23CC(C)(C2)C3)=O)CC(NC(C2(n3cnnn3)CC2)=O)CC12CCCCC2 Cc1cc(=NCC2CCN(C(c3c(N(C)C)cccc3F)=O)C2)c(C#N)c[nH]1 N1(C(C2CCN(C(C3=NNC(=O)C3)=O)C2)=O)Cc2ccccc2C1 CONC(=O)C(=O)N1CCC(C(=O)NC2CCCC2C(N)=O)C1C N1(C(C(C=CC)O)=O)C2CCC1C(F)C(NC(c1scc(C)c1OC)=O)C2 N1(C(C(c2ccc(C)s2)C)=O)CC(NC(c2ccc(=O)oc2)=O)CC(C)(C)C1 CCS(=O)(=O)CC(=O)NC1CCC(C(=O)Nc2c(C)ncn2C)C1 C(=O)(C(CC)CCCC)NC(CCCC)CNC(=O)CC(=O)OC c1(C(N(C(CNC(c2cc(C(=O)OCC)no2)=O)C)C)=O)ccc2ccnn2c1 N1(C(c2cn(C)nc2)=O)CCC2(CCOC2)C(CNC(c2n[nH]cc2Br)=O)C1 c1(C(N2CC3C(N(C)C(c4cc(O)cs4)=O)C3C2)=O)cnc2c(c1)COCC2 C1(Cc2cnc(CC)o2)C(C)(C)C(C(=O)Nc2nnnn2C)C1(C)C N1(C(c2n(C)ncc2Cl)=O)CCN(C(C2(C)CCNC2=O)=O)CC12CC2 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCC(C)C(NC(=O)C2CC2)C1 N1(C(CC2CCC(C)CC2)=O)CCCC(C2CCN(C(c3nncs3)=O)C2)C1 N1(C(Cc2nnc(C)s2)=O)CC2CC(NC(c3cn4cc(C)sc4n3)=O)CC1C2 Cc1noc2cc(C(N3CC(O)(CNC(=O)C(C)(O)C(C)C)C3)=O)ccc12 N1(C(C(N2CCN(C)CC2)C)=O)CC(NC(C2CC(=C3CCC3)C2)=O)C2(CC2)C1 N1(C(C2CC(C)(NC)C2)=O)CC2CCN(CC(=O)Nc3ccc(C#C)cc3)C2C1 C1(CN2CCC(N(C)C(c3n[nH]c(C(C)(C)C)n3)=O)C2)CCC(C)CC1 C1(C(=O)OC)CC(C(=O)OCC(C)C2CCC2)N(C(C)=O)C1 C1(NC(c2n(CCOC)nnn2)c2occc2Br)COC2(CCCC2)C1 C1(NC(C2CCC(C(=O)O)C2)=O)C2CC1N(C(c1ccc(OC(F)F)cc1)=O)C2 N1(C(CCCOCC)=O)CCC2(CC1)CC2NC(=O)CCc1ccc(SC)cc1 C1(CNC(=O)CC2(O)CCC2)CCCCCN1C(=O)COC1CC(C(=O)NC)C1 N1(C(c2ncsc2OCC)=O)CC2(CCCC2)C1C(=O)NC C12(C(N(CC(CN(C(=O)C(C)(C)C)C)O)C)=O)CCCCC1OCC2 C1(NC(C2(CO)CCCCC2)=O)CCN(C(=O)CN2CC3CC3C2)CCC1CO Cc1ccc(C(=O)NC(C)C(C)NC(c2cnn(C3CCCC3)c2C)=O)nc1C N1(C(CC2CC(NC(C(CCC)O)=O)C2)=O)CCCCC(C)C1 N1(C(COC2(C)CN(C(C3(C)CCC(C)CC3)=O)C2)=O)CC2(COC(CO)C2)C1 CC(C)(C[Si](C)(C)C)C(=O)Nc1ccc(N2CCNCC2)nc1 C1(CC)CN(C(c2c[nH]cc2-c2ccc(C)s2)=O)CCN1C(=O)CCN(C)CC Cc1ccc(F)c(C(=O)NCC2CN(C(=O)C(c3c(C)n[nH]c3C)C)CC2C)n1 c1(OC)cn(CC(N2CCN(C(C3OCC3(C)C)=O)C(C)C2)=O)c(C)cc1=O C1(NC(CC2(CSC)CC2)=O)CCCC1(C)NC(=O)COCC(F)(F)F c1(C(=O)NC2C(CNC(CCC(=O)NC)=O)CCC2)c(C)nn(C)c1C1CC1 N1(C(C2C(CC)C2)=O)CCC(CNC(c2ccc(Cl)nc2C)=O)C(F)(F)CC1 C1(CC(=O)NCCCNC(c2nccc(CC)c2)=O)CCCC(C)(C)C1 CC(CN1CCCCC1)C(=O)N1CC(CCNC(=O)CC2(C(F)(F)F)CC2)C1 N1(C(CNS(N(C)C)(=O)=O)=O)CC(NC(=O)CNS(N)(=O)=O)C2CCCC2C1 CC1CC(NC(=O)CCn2ccccc2=O)CCN1C(C1CC12CCOCC2)=O c1(C(=O)NC23CN(C(CSCCCC)=O)C(C2)C3)oc2c(OC)cccc2c1C CN1CCN(C(=O)C(F)n2ccnc2)CC1CNC(C1(C(N)=O)CC1)=O c1(C(=O)NC(C2CCCN2C(c2ccncc2)=O)(C)C)csc(-c2ccoc2)n1 C(=O)(C1=CCOCC1)NC1C(NC(CC(C)Oc2ccccc2)=O)CCOC1 C(=O)(C1CCCn2c(C)nnc21)N1CCC(CNC(CCC(C)OCC)=O)CC1 c1(C(N2C(CCNC(CSCCCC)=O)CSCC2)=O)ccc(Cl)c(C)c1 C1(CC=C)(C(=O)NC(C)(C)CN(C)C(c2cnn(CCN(C)C)c2)=O)CCOC1 Cc1ccc(S(N)(=O)=O)cc1C(=O)N(C)CCN(C)C(c1csnc1C)=O c1(C(N2CCSC(C)(C)C2)C(=O)NCC(=C)C)cc(OC)cc(COC)c1 N1(C(C2CC(OC)CN2C(c2nocc2C)=O)=O)CCC12CCN(C)C2 C#CC12CCC(C(=O)NCC(O)CN(C)C(C3C4CCCOC34)=O)(CC1)CC2 C(=O)(CCSC(C)(C)C)N(C1CN(C(=O)CCOC2CCC2)C1)C(C)C c1(C(=O)NC2CN(Cc3cnn(-c4ccccc4)c3)CC2F)cc(F)cnc1Cl C=CC(C)(CCOC)C(=O)N1CC(F)(CNC(=O)Cc2cc(C)no2)C1 N1(C(c2ccc(COC)o2)=O)CCCC(N(C(=O)CCSC)CC2CC2)C1 C(=O)(C(CC)CCCCC)NC1CCC(NC(C(CC=C)(C)CC)=O)CC1 Cc1ccc(C=CCC(=O)NC(C)CNC(c2cc(C(N)=O)cc(F)c2)=O)cc1 Cc1nc(CC(=O)NC2CCC(N(C)C(c3ccc[nH]3)=O)C2)cs1 Cn1nnc2ccc(CNC(Cc3cccnc3)C(=O)O)cc12 c1(C(CC)C)cccc(S(=O)(=O)NC(=O)C(=O)NCc2ccsc2Cl)c1 c1(C(N(CCOC)CCNC(C2(C)CC(F)C2)=O)=O)c(C)cc(C)cc1N C#CCCCCCCCNC(=O)C(C1(O)CN(C(c2cnnc(O)c2)=O)C1)F N1(C(C2CCCC2)=O)CCN(C(=O)C(F)(F)CN2CCCC2)C2(CC2)C1 N1(C(C=CCC)=O)CCN(C(=O)CCc2ccc(O)cc2)CC1C(F)(F)F C12(CC(N3CC(C)C(NC(=O)Cc4ccc(Br)cc4)C3)=O)CCCN1CCC2 C1(NC(c2csc(Cl)c2)=O)COC2(CCN(C(C34CC(CN3C3CC3)C4)=O)C2)C1 CCCC(CCC)=CC(N1CCC(O)C1CC(=O)NCC1(CO)CC(C)(C)C1)=O N1(C(C(C)S(N)(=O)=O)=O)CCCC2(NC(C3(c4cccnc4)CC3)=O)CC2C1 c1(CCNC(C23C(CN(C(CCCSC(C)(C)C)=O)C2)C3)=O)c[nH]c(=N)nc1O C1(NC(CNS(NC)(=O)=O)=O)CCN(C(c2cncnc2C)=O)C(C)C1 Cc1cc(F)sc1C(N1CC2CC1C2NC(C1(CC(F)F)CCC1)=O)=O CC(=O)C(C)CC(C)C(=O)NCCn1cnc(C(N2CCc3ncccc3C2)=O)c1 C=CC(CC)CC(=O)NCC1CC2(CC2)CN1C(=O)C#CC1(CC)CC1 C1(C(=O)NC2CCC(=O)NC2=O)C2Cc3ccccc3C12 C1(O)(CNC(C(C)OCC(C)C)=O)CCCN(C(=O)CCC(N)=O)CC1 C(Cc1cc[nH]n1)(C(=O)NCC1CCSCC1)NC(CCOCCC)=O C1(NC(c2nnc(C)s2)=O)CN(C(=O)C=Cc2ccco2)CCC1C C(C)(C(O)C(F)(F)F)NC(CN1CCCC(c2ccc(OC)cc2)C1)=O N1(C(CN(CCC)C)=O)CCCC(NC(=O)CCc2ccc(N)cn2)CC1 c1(C(N2CCC(N(C)C(C3CCCC(F)(F)C3)=O)C2)=O)cccc2c1COC2 c1(C(N(CCCNC(c2ccc(F)cn2)=O)C)=O)ccc([N+](=O)[O-])n1C Cc1[nH]nc(C(N2CCOC(CNC(=O)C(C)(Cl)Cl)C2)=O)c1F C1(CC)(NC(C2CCC(CCC(N3CCOC(C)C3)=O)C2)=O)CC(C)(C)C1 c1(C(N2CCCN(CC(C)O)CC2)C(=O)NC)cnc2c(C#N)cnn2c1 CC(C)(O)C(C(=O)NCC(C)(C)OCCO)NC(=O)CC1CCSC1 Cc1c(F)ccc(N)c1C(=O)NC1CN(C(c2cccc(C)c2Br)=O)C1 CCCC(CC(=O)N1CCC1C1CCC1)NC(c1ncccc1Cl)=O Cc1c(Cl)ccc(C(N2CC(NC(c3ncccc3C3CC3)=O)CC2C)=O)c1O c1(C(=O)NCCC)cccc(C)c1NCc1ccncc1OC C1(C(=O)NC2(CN(C)C(c3cc(C(C)(C)C)no3)=O)CCC2)COCC1C(N)=O c1(CCCC(=O)NC2CCOC(c3ccc(F)cc3)C2)ccc(F)cc1 CC1(C)CCC(CCNC(=O)C(N2CCCCC2CC2CCCCC2)=O)CC1 N1(C(C(CC#C)C)=O)CCCC12CCCN(C(c1ccc([N+](=O)[O-])o1)=O)C2 Cc1cc(N2CCC(OCC3CCCCC3)CC2)n2nc(C(F)(F)F)nc2n1 c1(COC)cccnc1C(=O)NC1(C2CCCN2C(=O)Cc2ccnn2C)CC1 Cc1cc(C)n(CC(=O)NCCCCC2CN(C(c3[nH]ccc3C)=O)C2)n1 c1(C(=O)NCCC2CN(C(CC3C(OC)CC3)=O)C2)cccc2c1CC(=O)N2 CCCS(=O)(=O)CC(=O)NCc1ccc(C(C)NC(=O)C(C)CNC(C)=O)cc1 c1(OC)cc(-c2cn(C3CCN(C(=O)C(C)n4cnnn4)CC3)nn2)cc(C)c1 N1(C(c2cc(=NC)[nH]cc2)=O)CC2CCC(C1CO)N2C(=O)Cc1coc(C)n1 Cc1nc(NCC2CCNCC2OCc2ccccc2)c(Cl)cc1C#N c1(C(N2CCC(NC(C3C(C)(C)CC3)=O)C2)=O)cc2ccc(F)cc2s1 c1(C(=O)OC)ccc(OC)c(NC(=O)NCC2CC(O)C2)c1 C1(CC#C)(C(=O)N(CCCCN(C(=O)CC2CC2)C)C)CCOC1 C12(NC(c3c(C)ccnc3C)=O)CC(CNc3ncccn3)(C1)OC2(C)C C(=O)(C1=CCCC1(C)C)N1CCC(O)(CN(C(c2c(C)snc2)=O)C)C1 N1(C(C=C(C)I)=O)CC2CCCC(C1)N2C(C1(c2ccc(F)cc2C)CC1)=O N1(C(c2ccc(C)nn2)=O)CCC2CCCC12CNC(c1coc(=O)[nH]1)=O c1(OC)cc(C(=O)NCCN(C(=O)C=CBr)C2CCCC2)cc(Cl)n1 c1(C(N(CC(CN(C(CCCCC=C)=O)C)O)C)=O)cn2cccc(Cl)c2n1 N1(C(CSCC(=O)O)=O)CCN(C(c2cnn(CC(O)CO)c2)=O)CC1 c1(C(N(C2CCCN(c3nccs3)C2)C(C)C)=O)cc2c(Cl)cccc2s1 C(CCC(=O)NN1C(=O)NC(=O)C1C)c1c(S(CC)(=O)=O)c(Cl)ccc1 c1(C(N2CC(C)C(F)C2)C(=O)NCCCC)ccc2cc(F)cc(Br)c2n1 c1(-c2n(C3C(C)OCC3)nc(C(C)(C)C)n2)cc2scc(Cl)c2[nH]1 C(=O)(C#CC1CCC2(CC1)OCCO2)NCC1CC(O)(CNC(CC=C)=O)C1 N1(C(C(CC)SC)=O)CCC(C)(CNC(c2cn(CCN(C)C)nn2)=O)CC1 Cc1cc(F)c(C(=O)NC2(CNC(C3COC(=O)N3)=O)CC2)cc1F c1(CN=C(NCC(c2cn(CC)nc2)O)NC(C)C)cc(F)ccc1C c1(CC)cc(C(N2CCCC(C)(NC(=O)C3=NOCC3)C2)=O)cc(N)c1 c1(C(=O)NCC(CNC(c2ccsc2Cl)=O)CO)n[nH]c2c1CSCC2 C1(C(=O)NCCCC(C)NC(=O)CC2CCCCC2)CCOC1(C)C CCCCCCCCC(O)CCC(=O)OCC1(COC)CCOc2ccccc2S1 C(c1nc2ccccc2s1)=CC(N1CC2CCN(C(CC(C=C)CC)=O)C2C1)=O CCC(CC)C(C(=O)NCC(CNC(C1CC(F)(F)C1)=O)OC)OC C(CNC(=O)COc1cnn(C)c1)(C(C)(C)C)NC(C(C)C1CC1)=O c1(C(N(C(C)CN(C(=O)CCn2ccnn2)C)C)=O)cccc(C(C)(F)F)c1 c1(C(N2CC(C3(NC(C4CCC(=C)CC4)=O)CC3)C2)=O)cc2ncc(C)cn2n1 CCC(CC)(CC)C(=O)N1CC2C(CNC(c3cnc(S)n3C)=O)C2C1 Cc1ccc2c(=NCCCc3cnn[nH]3)[nH]c(=NCc3ccn(C)c3)[nH]c2c1 CCC(CC(F)F)C(=O)NC1CC(CNC(=O)CCNC(=O)CO)C1(C)C C(=O)(C1=CC2(CCN(C(=O)C(O)C3CCC3)C2)C1)N1CCC(C2(C)CC2)C1 c1(OC)ccc(F)cc1C(F)(F)C(=O)NC12CC(NC(=O)CN3CC=CC3)(C1)C2 C=C(C)C(CC(=O)NCCC1COCCN1C(c1cscn1)=O)OCC CC1(C)CN(C(c2ccnc(F)c2F)=O)CC1NC(C1CN2CCC1CC2)=O N#Cc1cc(F)c(NC(=O)CC2CN(Cc3sccc3Br)CCO2)cc1F c1(C(N2CC(C(C)NC(C(C(CC)C)OC)=O)C2)=O)ccc2nc[nH]c2c1 C1(O)(CCNC(=O)CCc2cn[nH]c2)CN(C(=O)CC2(O)CCOC2)C1 C1(C(N2CC(NC(C(CC=CC)C)=O)C2)=O)CC2(COC(=O)N2)C1 c1(C(N2CCN(C(C(OC)OC)=O)C(C)C2C)=O)ccc2c(c1)CC(C)O2 c1(C(N(CCNC(=O)C(C)OCC(F)(F)F)CC)=O)ccc(O)nc1Cl c1(CCC(=O)NCCCC(N2CCC2C(=O)OC)C)csc(Cc2ccccc2)n1 CN1C(=O)CCCC1C(=O)N(C1(Cc2ccccc2)COC1)C CC(C)CC(C)(CNC(c1ccccn1)=O)NC(c1cnc2n1CCC2)=O N1(C(C(C2(O)CCC2)NC(C2C(C)(C)OC(=O)C2)=O)=O)CC(=O)N2CCCC2C1 N1(C(C2CN(C(C)=O)C2)=O)CC(O)C(O)C1CNC(C12CCCC1C2(F)F)=O N1(C(c2nccs2)=O)CCCC(N(C2CCC2)C2CC2)C1 Cc1[nH]c2ccnn2c(=O)c1CC(=O)N(C1CCC(NC(=O)C(C)CO)CC1)C N1(C(c2c(CC)nn(C)c2)=O)CCN(C(c2ccc(C(C)C)s2)=O)CC(C)C1 C12(CNC(COC(C)(C)C(F)(F)F)=O)CCCC1CCN2C(c1cnccn1)=O N1(C(CCSCC)=O)CC(CNC(c2coc(Cc3nc[nH]n3)n2)=O)C(O)C1 N1(C(C2(NC(C)=O)CCCC2)=O)CC2CC(NC(C3CC4(CCC4O)C3)=O)CC1C2 CCC(=O)CCC(=O)N(CCC(=O)NC(C)Cc1cnn(C)c1)CCCO Cc1cc(C(N2CCCC2CCC(N2CCC(CC(F)F)C2)=O)=O)cnn1 N1(C(C2CC(C(F)(F)F)C2)=O)CCCC(C2CCN(c3nncs3)CC2)C1 c1(C(=O)NC2CN(C(C(C)=C(CC)C)=O)CC(O)C2)ccnc2[nH]ncc12 N1(C(CC=C)=O)CC2CCCC2(NC(=O)CN(CC)CC)C1 C1(CNC(c2cc(Cl)no2)=O)CC2(CO1)CN(C(C1C3CCC(=O)C13)=O)C2 c1(C(=O)NCC2(F)CCN(C(=O)COCC3CC3)C2)cc(O)ccc1Cl CCCCC(CC(=O)N(CCC(=O)OC)OC)NC(=O)C=NOC c1(C(=O)NC2CCC(NC(c3n(C)ncc3Cl)=O)C2)ccn2c(O)nnc2c1 C(CC(O)CC(=O)N1CCN(CC(C)(C)N)CC1)SC C1(NC(CC(C)NC(N)=O)=O)CCCN(C(=O)CSc2nc[nH]n2)CC1 N1(C(c2c(Br)cc(C)s2)=O)CCC(C)N(C(=O)Cc2ccsn2)CC1 Nc1cc(Cl)ncc1C(N1CCCC(CO)(NC(C2CC23CCOCC3)=O)C1)=O C(=O)(C(C)(F)CCCC)N1CCC(CCC(N2C(CCCC)CCC2)=O)CC1 N1(C(C(C(C)C)n2ncc(N)n2)=O)CCC2(CCN(C(=O)C=CC(N)=O)CC2)C1 Cc1cc(F)cc(Br)c1NC(=O)C(=O)NC1CC2(CCCC2)C1 c1(CNC(C2(NC(COC)=O)CCCC2)=O)nccc(C)n1 N1(C(C2(C=C)CC2)=O)CC2CCCC(NC(c3ccnc(NC(C)=O)c3)=O)(C2)C1 C1(CNC(c2n(CC)nnc2)=O)C2CCCC1N(C(=O)CC(C)C)C2 CCS(=O)(=O)c1ccc(CN=C(NCc2cccs2)NCC2CNC(=O)O2)cc1 c1(C(=O)OC)c(CNC2CC(CC(=O)NC(C(F)(F)F)C3CC3)C2)cccc1Br C(=O)(CCCC(=O)N(CCC(C(C)(C)C)NC(=O)C(F)C1CCC1)C)OC N1(C(C(C)=CC)=O)CCC2(CCN(C(=O)C(C)CS(C)=O)CC2)C1 C1(C(N(C)CC2CS(=O)(=O)CCN2)=O)CCS(=O)(=O)CC1 CCC(CC(C)C)C(=O)NCC(C)N(C(=O)C(Cl)=CCl)CC C1(S(=O)(=O)NC(C)(C)C)(C(c2n(CCNC3(CF)COC3)nnn2)OC)CC1 N1(C(C(c2cnn(C)c2)NC(C(CCCC)CC)=O)=O)CCN2C(=O)CCC2C1 C(=O)(C(O)CNC(=O)NCc1cnc(C)[nH]1)N1CC(CC)C1 CC1(C)CCCCC1C(N1CC(NC(=O)C(c2ccccc2)n2cccc2)C1)=O CC1(CC(=O)NC2CC(NC(C3(c4ccccc4Cl)CC3)=O)C2)CC(F)(F)C1 N1(C(C2(C)CCN(C)C2)=O)CCCC(F)(C(=O)NCC2CN(C)C(=O)CO2)C1 C(CCCC(=O)NCC1OCCC1(C)C)N(C(=O)CSC(F)(F)F)C N#CC1(C2CCCC2)CCN(C(c2cnc3c(c2)COCC3)=O)CC1 N1(C(c2cnn(C3CCC3)n2)=O)CC2CN(C(C34CCCN3CCC4)=O)CC2C1 c1(C(=O)NC(CC(C)NC(c2cc(C)sn2)=O)C)ccc([N+](=O)[O-])[nH]1 c1(C(=O)NC(CCCC)CNC(=O)CN2CCCC2=O)cc2ccncc2c(O)n1 Cc1c(C(=O)N(C(CNC(C2(n3cnnn3)CC2)=O)C2CC2)C)cnn1C1CC1 N1(C(C(CNC(C2(CC#C)CCOC2)=O)CC2CC2)=O)CCC(F)(F)CC1C c1(C(N2CCN(C(C(C)=CC3CC3)=O)C(C)C2C)=O)cc2nccn2c(O)n1 N1(C(CCc2nnc3n2CC(C(=O)OC)CC3)=O)CCCn2[nH]c(=N)cc2C1 N1(C(C(Br)=C(C)C)=O)CCCC(NC(=O)Cc2cc(F)ccc2C)CC1 N1(C(c2c(CC)nccn2)=O)CCC2(CCN(C(=O)CCCSC)CC2)C(C)C1 C(CN=c1[nH]c(=NCc2ccc(N)cn2)[nH]c2c1CCCCCC2)OCC(=C)C C12(NC(CSCCCC)=O)COC(CNC(C3CC(C)CO3)=O)(C1)C2 c1(C(N2CCC(C3N(C(c4c[nH]c(=N)s4)=O)CCC3)C2)=O)cc2ccsc2s1 Cc1nc(C)c(C(N2CCC(C(C)NC(c3cncc(F)n3)=O)C2)=O)[nH]1 c1(C(N2CC(Cn3cc(-c4cc(=N)[nH]cc4)nn3)C2)=O)cc2c(o1)CCCC2 c1(OC)ccc(CN2CC3CC2CN3C(c2ncsc2C)=O)c(OCC2CCC2)c1 c1(CNC(CC(=O)NCC2N(C(CNC(C)=O)=O)CC=C2)=O)c(C(N)=O)c[nH]c1C c1(N(CC=C)C)nc(=NCCCOCCOC(F)F)[nH]c2c1CSC2.C1(C)CN1 C12(CC)CN(C(c3cccc(N)c3)=O)C(CNC(c3ccc(=O)oc3)=O)(C1)C2 C1(c2nnc(COC)o2)CN(C(c2nnc(C3CNC3)s2)=O)CCO1 N1(C(C(CCSC)O)=O)CCC2(C1)CN(C(=O)CCS(N)(=O)=O)C2 Cn1cnc2c1=NC1=NC(c3ccccc3)CNC=2N1.c1(COC)cnc[nH]1 c1(C(=O)NCC(CC)(C)NC(C2CN(C)C(=O)N2)=O)cc2ccc(F)cc2cn1 C#Cc1nc(C(=O)NCC2CN(C(c3cccc(NC(C)=O)c3)=O)CC2C)cs1 CC1=C(CNC(=O)C(C2(O)CCC2)NC(=O)C2=CCCCO2)COCC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1(NC(CN2CC(C)C2)=O)CCCCC1 CCCC(C)(O)CC(=O)N1CCC(CCOC)(NC(=O)C=CC2CC2)C1 C1(C(C)NC(=O)CSc2nncs2)CCN(C(C2(C(F)(F)F)CC2)=O)C1 C(=O)(C1Cc2ccccc21)NCC(CCC)C(=O)N1CCCC(CC(N)=O)C1 C(=O)(CCC(F)(F)F)NCc1c(C(=O)NC(C)COc2ccccc2)[nH]cc1 C(CN=C(NCC12COCC1C2)NC(C)CC)c1scc(C(=O)OC)n1 C(=O)(C#CC1CCCCO1)NC(CNC(c1n(CCC)ncc1)=O)(C)C(C)C CC(C)CC(CNC(=O)CC1(C)OCCO1)C(=O)NCC(O)C(C)O c1(C(C)OC)nc(C)c(C(=O)NC2CCC(NC(=O)CC3(C)CC3)CC2)s1 c1(CC)ccc(C=CC(=O)NC2CC(c3ccc(F)cc3)C2(C)C)o1 Cc1ccc(CC(=O)NCCC2CCN(C(c3cc(C)c(C)[nH]3)=O)C2)c(F)c1F O=C(C1=NOC2(CCOC2)C1)NCC1(F)CN(C(=O)C=Cc2ccccn2)C1 C(=O)(CC1=NNC(=O)C1)NCCC(C)CCNC(C1C(C)(C)C1(C)C)=O C1(COC)CC2(CCN2C(C2CC(CNC(C34CC(F)(C3)C4)=O)C2)=O)C1 c1(CC(C)SC)cc2ccccc2[nH]1.C1(C)(C)CC(=O)NCc2cn1nn2 C(c1ccc(Cl)c(Cl)c1)=CC(N1CCN(C(c2n(C)ncc2)=O)CC1)=O c1(OC)cccc(C(C)C(=O)NCC2(C)CCCC2NC(=O)C(C)=C(C)C)c1 C(C)(C(C(=O)NCCOC1CCN(C(c2occc2C(C)C)=O)C1)N(C)C)OC C1(CC)(NC(c2cc(C#N)cs2)=O)CCN(C(c2cscn2)=O)CC1 N1(CC)CCCC1C(=O)NCCSCC(=O)Nc1csnc1OC c1(C(=O)OC)ccccc1Cn1cc(CN)nn1.C12CCC(C1)CC(=O)N2.C1CC1 c1(C(=O)NC2CC(CNC(c3c(Cl)cc(C)s3)=O)C2)ccnc2[nH]ncc12 Cn1nc(Br)c2c(NC3CCCC(NC(=O)C(O)Cc4cnc[nH]4)C3)ncnc12 CC1(C)OC(=O)NC1C(=O)NOCc1cn(-c2ccc(Br)nc2)nn1 C(N=c1[nH]nc(O)s1)C1CC(NC(c2cn3cccnc3n2)=O)C12CCC2 C(C(C)(C)C(=O)NC(C1CSCCO1)(C)C)OCC CC1CC(C(=O)NCCCCCNC(=O)CCF)CCC1C C1(C(=O)OC)CC(OCc2ccccc2)CN1C(=O)C(=O)Nc1ccccc1F c1(C(C)NC(=O)CC2OCCOC2(C)C)cc(F)c(Br)cc1F C=CC1CN(C(c2cnc3c[nH]nc3c2)=O)CCC1CC(=O)NC(=O)CSC c1(OC)ccc(CCC(=O)NC2CC(NC(C3CC(O)(C#N)C3)=O)C2)cc1O C(=O)(C(C)C(O)C(C)CC)NC(C(=O)NCCC(CC)(F)F)C1(C)CC1 C1(NC(c2cnc(SC)[nH]2)=O)CCC(C)(CNC(c2cccnc2O)=O)C1 c1(C(N2CCCC(NC(=O)NC3C=CC(CSC)C3)C2)=O)c(F)cccc1F N1(C(c2nn(C)c(Br)c2C)C(=O)NC)CCCC2(C1)NC(=O)NC2=O Cc1cn2nc(C(=O)NC(C)CCCCNC(C3CCCO3)=O)cc(C)c2n1 Cn1nc2ccccc2c1-c1cn(CCCC(=O)NCc2cncc(Cl)c2)nn1 C1(NC(=O)Cc2cn[nH]c2)CCC12CCN(C(=O)CCc1cncc(F)c1)CC2 c1(SCC(=O)NC2CC(CNC(=O)CC3CC(F)(F)C3)C2)cc(F)c(F)c(F)c1 CC(CCCC(=O)NCCCOCCN(C(=O)CCF)C)c1ccon1 c1(C(=O)NCCNC(c2occc2C2CC2)=O)cccnc1C(F)(F)F C1(CNC(C2C(CC)OCC2)=O)CCN(C(=O)C(C)(C)CSC)CC1C1CC1 C1(NC(COCC)=O)CN(C(=O)CNC(c2cccc(F)c2)=O)CC1(C)C Cc1ccccc1C(=O)NC1CCCCC1C(N1CCC(C#N)C1)=O CCC(CCCC(=O)NCC1(Cl)CC1(F)F)NC(C1CCCC(C)(C)C1)=O C1(N=[N+]=[N-])(C(=O)NCc2n(CCC)cnc2)CCN(C(=O)C(C)=C(C)CC)C1 C1(C(=O)NC(CC2(O)CCC2)CO)CCC(Cc2ccccc2Br)CC1 c1(CC(=O)N(CCN(C(C2CCCC(OC)C2)=O)C)C)coc2ccccc12 N1(C(c2c(F)cncc2Br)=O)CCC2(CCN(C(c3cc4ncsc4[nH]3)=O)C2)C1 N1(C(CCC#C)=O)CCC2CN(C(=O)C(c3ccsc3Br)OC)CCC12 N1(C(c2cnc(C(=O)OCC)s2)C(=O)NCCCC)CCC(C2(C)N=N2)CC1 CC1CCCNC1C(=O)NCC1(C)CCN(C(c2cccs2)=O)C1 C1(CNC(c2c(Cl)cccc2Cl)=O)C(C2CC2)CCN1c1ncc([N+](=O)[O-])cn1 CC1(C)CC(C(=O)N2CC3CC(C(=O)NCCCN4CCC4)(C3)C2)=NO1 N1(C(C2CCCN(CC)C2)=O)CCCC2(CC(NC(=O)C(C)(C)OC)C2)C1 N1(CC)CCOCC1C(=O)N(CCCNC(C1(n2ccnn2)CC1)=O)C CCCC(C(=O)NC1CCC1NC(c1csc(C)c1CC)=O)S(N)(=O)=O N1(C(=O)CC2CCSC2)CCN(C(=O)C(c2cccnc2)O)C2(CC2)C1 C(CCCCC(=O)N(C1CC(NC(=O)COCC(F)(F)F)C1)C)SC C12(NC(c3ccc(Cl)c(O)c3)=O)CCN(C(=O)CSc3ccncc3)CC1C2 C1(CNC(c2ccc(C(C)=O)[nH]2)=O)CN(C(=O)C(C)N(C)C)CCC1(C)C C1(NC(c2cc(C)c(C)[nH]2)=O)Cc2ccccc2C1NC(c1ccc(C)n1C)=O C(=O)(CS(=O)(=O)c1ccccc1C)N1CCC(C(C)(C)NC(C(C)SC)=O)C1 N1(c2ncc(C)cn2)CCCC2C1CCN2Cc1cccc(-c2ccco2)n1 O=C1CCC(C(=O)NCC2CCCN2C(=O)CC2(CO)CC2)N1 C=CCC(C(=O)NCc1cnn(C)c1N)NC(=O)C(C)COCC Cc1c(N)ccc(C(N2CC(CNC(c3cc(C#N)c[nH]3)=O)CC2C)=O)c1Cl c1(OC)cc(OC)cc(C(N2CCC3CCC23CNC(=O)C=C(C)C(C)C)=O)c1 C1(NC(c2c(OCC=C)cccc2)=O)CC2CC(C1)CN(C(=O)C(C)OCC)C2 n1(CC=C)nnnc1C(C1(C)COC1)NCCC(O)C1CCC1 N1(C(CSC(C)(C)C)=O)CCC(C)(C)C1CC(=O)NCc1cnccn1 C1(CNC(COCCSC)=O)CN(C(=O)CCc2ccc(C)c(C)c2)C(C)(C)C1 Cc1ccc(C)c(N(C)C(C2CN(C)CCN2C(=O)Cc2ccc(F)cc2)=O)c1 C(=O)(CC(F)(F)C(F)F)NCC1CCC(NC(C2C(C)(C)OCCO2)=O)CC1 c1(CC(=O)NC(CNC(C(CCC(C)C)O)=O)C(C)C)ccc2cnccc2c1 C1(NC(C(C=C)(C)C)=O)CCN(c2ncnc(C)c2Br)CCC1CO C(N=c1cc[nH]c(C(N)=O)n1)C1CN(C(c2c(C)cco2)=O)C(C)C1 N1(C(C(CC)(C)C)=O)CCN(C(C2CC(F)C2)=O)C(c2cccnc2)C1 c1(C(N(C)CCNC(C2(C)CC(F)C2)=O)=O)cc(CO)n(C)n1 C1(NC(C(C2CCCC2)NC(C)=O)=O)CN(C(=O)CCc2ccncc2)CC1C C1(OC)CCC12CC(C(=O)NCC1CN(C(c3ccncc3F)=O)CCO1)C2 C(CC(C)C)(C(=O)NCC1CCNC(=O)C1)NC(C1=C(C)CC1)=O C(=O)(C1=NOC2(CCC2)C1)NCC(C)(CO)NC(c1nccc(COC)c1)=O C1(NC(c2ccc(Br)cc2)=O)COCCN(C(c2cscc2Br)=O)C1 C1(NC(C2(OC)CCCCC2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC(O)C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)NS(C)(=O)=O)ncc(F)cc1F N1(C(C2(CNC(C3CC(C4CC4)=NO3)=O)CC(=C)C2)=O)CC(OC)CC(C)C1 c1(OC)ccc(C(CCO)Nc2nnc(C3CCOC3)o2)cc1 c1(CC(C)C)ccc(NC(=O)Cn2cc(C#N)cn2)cn1 c1(-c2nc(SCC(=O)NCCN(C(C(CC)OC)=O)C)on2)ccc(OC)cc1 c1(CC(=O)NCC2C3CN(C(=O)CCCCCF)CC23)nsc2ccccc12 C12(C(=O)NC3(COC)CC3)CC1CCN2C(=O)CCC1CCC(=O)C1 c1(C(N(C2CCN(c3cc(C(F)(F)F)ncn3)C2)CC)=O)c[nH]c2cccnc12 C(C)(CCN=c1[nH]c(-c2ccccc2)cs1)N(CCCC)CCCC c1(C(C=CC(=O)NCCC(C)NC(CCc2cc(C)on2)=O)=O)ccc(Cl)cc1 N1(CC)CCN(C(c2cnnn2CC)C(=O)NCc2ccco2)CC1=O c1(COC)ccccc1C(=O)NCCNC(=O)CC(=O)OC(C)(C)C C=C(F)C1(CC(=O)NCCC2COCCN2C(=O)CC2CC2CC)CCC1 Cn1ncc(C(N2CCC(OCC(=O)NC(c3cccnc3)CO)C2)=O)c1N Cc1coc(C(=O)NC(C)CC(C)NC(c2nc(Br)sc2C)=O)c1C CC1=C(C(=O)N(C)CCN(C)C(c2c(N3CCCC3)cccc2F)=O)CCO1 C1(C(=O)NCCCOCc2ccccc2)CN(Cc2cc(Br)co2)CCC1O c1(COC)ccc(C(=O)NC(C)(C)CCNC(C2CN(C(C)COC)C2)=O)s1 C1(OCC)CC2CN(C(=O)C(CC3CCC3)NC(=O)Cn3cccn3)CC12 CC(CC(C)(C)C)C(=O)N1CCC(n2cc(C(c3ccccc3)N(C)C)nn2)C1 Cc1ccc(CNC(=O)NC2CCCC(N(C)C)C2)c(Br)n1 C12(C(=O)OC)CC1CN(C(C1CCC(NC(=O)CCn3cncn3)CO1)=O)C2 c1(NC(CCCc2onc(CC)n2)=O)ccc(C(=O)NCCCCCCO)cc1 C1(C(N(CC(CN(C(=O)CC2(CO)CC2)C)O)C)=O)CN2CCN1CC2 C(=O)(C1=CCCCCC1)NC1(c2cn(CC(COC)O)nn2)CCC(C)CC1 CC1CCC(C(N2CCCC2CCNC(=O)CC2COC(=O)C2)=O)CC1 C(=O)(C(=O)CC(C)C)NCc1oc(C(=O)NC(CSC)(C)C)c(C)c1 Cc1cc([N+](=O)[O-])cc(F)c1NC(C1CCN(Cc2nccn2C)CC1)=O c1(C(=O)N)ccnn(C)c1=O.CC(C)C(CCNC(C1(N(C)C)CC1)=O)CCC C(CC(C(C)(C)C)NC(C1CCCN1C)=O)N(C(C1(CC=C)CCOCC1)=O)C c1(CC)nc[nH]c1C(=O)N(CC(C)NC(C1(COC)CC1)=O)C N1(C(C2N(S(C)(=O)=O)CCCC2)=O)CCC(O)(CCNC(C2CC2F)=O)CC1 C12(CC(=O)NCC(C)(C)NC(c3ccc(C4C(C)C4)o3)=O)CCC(CC1)OC2 N1(C(C)=O)CC2CCN(Cc3ccccc3-c3cc(F)c(C)cc3Cl)CC12 N1(C(c2n(C)ncn2)=O)CCC(C2CC2)C1CNC(=O)CCC(C)(F)F C(=O)(C(C)C(F)(F)C(F)F)N1CC(=CC(=O)N(C2CC2(Cl)Cl)CC(C)C)C1 c1(C(N2CC(CNC(c3ccc(SC(C)C)cc3)=O)C2)=O)cccc(F)c1F CC1CCN(C(=O)CCC2CCC2)CC1NC(C1(F)CCCCC1)=O CC1(C)CCN(C(=O)C(F)CC(C)(C)NC(C2CCSC2)=O)CC1CO C(=O)(C(O)CCNC(=O)CC1(NC)CCC1)NCC1(CC)CCCO1 c1(N2CCC(C(C)NC(c3c[nH]c(C(N)=O)c3)=O)C2)ncnc2scnc12 Cn1cc(C(=O)Nc2scnc2C(N)=O)c2cc(C3=CCSCC3)ccc12 C1(C(=O)NC2(CC(=O)OC)CC2)(CO)CCCN(C(c2cc(C)cnc2C)=O)C1 C1(C(=O)NC2(c3cc(C(=O)OC(C)(C)C)on3)CCC2)C2CCC(F)C12 C=CC(C)N=c1[nH]c(=NC(COC)c2ccc(Cl)cc2)[nH]c2c(F)cccc12 Cc1nnccc1C(=O)NC1CC2C(NC(=O)CC(C)c3cccnc3)C2C1 CC1=NOC2(C1)CC(C(=O)NC(c1cn(CC3CNC(=O)CO3)nn1)(C)C)C2 C(=O)(CS(=O)C(F)(F)F)NC1CN(C(c2ccc(OC)c(N)c2)=O)CC1C Cc1c(C(=O)NCC2CCCN2C(C2(C(F)F)CCCO2)=O)oc2ccccc12 c1(C(=O)OCC)nnn(C)c1C(=O)N(CC(=O)Nc1ccccc1)C(C)(C)C c1(C(=O)NCC2C(C)CCN(C(C3(CC#C)CC3)=O)C2)cncc2nnn(C)c12 C(CC1=CCOCC1)NC(C1(NC(c2c(OC)cccn2)=O)CC1(C)C)=O C(=O)(C(O)CCC(C)C)NCc1c(CNC(Cc2c(C)noc2C)=O)cccn1 N1(C(c2c(C)scc2)=O)CCN(C(=O)C(C)Oc2ccccc2)CC1CCO CC1CCSCCN1C(C1(C(F)F)CC1)=O C1(CCNC(C2(SC)CC2)=O)CN(C(=O)C(=Cc2ccccc2)OC)CC(C)O1 C(=O)(CCC(C)(C)F)N1CCC(C(=O)NC(C(=O)OCC)(C)C)C1 N1(C(CC2C(=O)NC(=O)N2)=O)CC2(NC(=O)Oc3cnnc(O)c3Cl)CC1CO2 CC1CCC(CNC(=O)Cc2ccsc2Br)N(C(C2CS(=O)(=O)C2)=O)C1 c1(C(N2CC(C)(NC(C(C)C(F)(F)F)=O)C2)=O)cccc2nc(CO)[nH]c12 C1(CC(=O)N(CCOCCCNC(C(C)NC(N)=O)=O)C)C=CCCC1 C(C)(C(=O)NNC(=O)Cc1ccccc1Cl)NC(C(C)C)=O c1(C(=O)NC(C2CN(C(CCOCCCOC)=O)C2)C)ccc(C)c(O)n1 c1(CN2CC(CNC(c3ccc(N(C)C)cc3F)=O)C2)c(Br)cc(Br)cc1Br C1(NC(C(C)=CC)=O)CN(C(=O)CCCc2cnccn2)C(C)(COC)C1 N1(C(C2(CC)CCC2)=O)CCOCC1C(=O)Nc1c(C)ncn1C C(=O)(C1=CCS(=O)(=O)C1)NC(Cc1cn(CC2CCCC2)nn1)=O.CCS C1(C(N(CC)CC2CCOC2)=O)N(C(c2cocn2)=O)CC12CCCC2 Cc1ccc(Br)cc1CC(=O)N(C1CCN(C(=O)Cc2nonc2C)C1)CCO C(N=c1nc2c(cnn2C)c(NC2CCS(=O)(=O)C2)[nH]1)c1nc(NC(C)=O)sc1 c1(C(CC(=O)NC(C)CNC(c2cc(C3CCC3)[nH]n2)=O)C)ccc(F)cc1.C1CC1 C12(CC(=O)N(CCC(C)NC(C3CC(=C)C3)=O)C)COC(C(F)(F)F)(C1)C2 N1(C(C2C(CCOC)C2)=O)CCC(NC(=O)C(C)CSC)CC1 N1(C(C(N2CCCC(NC(CCC)=O)C2)=O)=O)CCS(=O)(=O)N2CCOCC12 c1(C(N2CCN(C(c3ccc(CCCCCC)s3)=O)CC2)=O)ccc2nonc2c1 C1(C(N2CC(CC(=O)OC)C2)=O)CCCC1CNC(C1(C)COC1)=O C1(CS(=O)(=O)NC(c2c(C)nco2)=O)C(C)(C)C1(C)C C1(C)(CNC(c2ccc(C(C)=O)o2)=O)CCN(C(c2n[nH]c(C3CC3)c2Br)=O)C1 N1(C(CCN(C(c2n(C(C)C)ccn2)=O)C)=O)CCCC2CN(C)CC12 C1(NC(c2ccncc2O)=O)CN(C(C2(F)CC3(CCC3)C2)=O)CC2(CCC2)C1 c1(C(=O)NCC2(c3[nH]cc(C#N)c(=N)n3)CC2)cc2c(s1)CCC2 C1(c2ccc(C)o2)CN(CC2CCCC(C(C)(C)C)C2)CC(=O)N1 N1(C(C#CC)=O)C2CCCC1CC(NC(c1ncc(Br)cc1C)=O)C2 Cn1cnc2cc(C(=O)NCC(F)CNC(C34CCC3C4)=O)ccc12 Cc1nc(C(N2CCC(CNC(c3cnc(OCF)cn3)=O)C2)=O)cn1C CC#CCC(C(=O)NCC1(C)CNC(=O)O1)NC(=O)CCc1cncs1 c1(C(=O)NCC2(COC)CN(C(C3CNC(=O)N3C)=O)C2)c(Cl)cnn1C C1(COC)CC(CNC(c2cnc[nH]2)=O)N(C(=O)C(C)Oc2cccc(N)c2)C1 n1(CCC(=O)NC2(CC=C)CN(C(C3CC(F)C3)=O)C2)cc([N+](=O)[O-])nc1C C(=O)(C(F)(F)CC1CC1)NC1CCC(Cn2cc(CSC)nn2)C1 C1(C(N(CCC#C)C)=O)CCN(C(=O)C2CN(C)CCO2)O1 c1(CC)cc(-c2cnc(C(=O)NCC(c3cccc(O)c3)O)cc2C)ccc1F C=CCCCC(=O)N(C1CCCN(C(c2cc(C(C)CC)no2)=O)C1)CC C1(N(C(C(CC(C)C)O)=O)C)CC2CCC(C1)N2C(c1ccnn1C(C)(C)C)=O C(C1CCCN1C(C1C2(CC2)C12CC2)=O)=CC(=O)NC1CCSCC1 n1(C(C)C)cc(C(=O)NCCN(CC=CC(C)(C)C)C(C)C)c(Br)n1 Nc1ccc2c(c1)CCC2NC(c1ccsn1)=O c1(N2CC(CCO)(NC(=O)CCSc3ccccc3)C2)ncnc2cnccc12 n1(CCC(N2CCC(NC(C=CC=CC)=O)(COC)C2)=O)c(C)c(C)sc1=O CC(O)C(C)(C)C(=O)N(C1CCN(C(C2CCCC23CCC3)=O)CC1)C C1(C)(COC)CC(NC(c2ccnc(O)c2F)=O)CN1C(=O)C(=O)NC1CC1 C1(C(=O)NC2CN(C(c3cc(CC(C)C)[nH]n3)=O)C2)CCSC(C)C1 CCC(C)C(O)CC(=O)N1CC(C(=O)NC2(CO)CCC(C)(C)C2)C(F)(F)C1 c1(OC)cc(F)ccc1CNCC1(Cc2onc(C)c2C#N)CC1 S(=O)(=O)(c1ccccc1Cl)NC1CCN(C(c2cccc(OC)n2)=O)C1 c1(NCC)ccc(C(=O)N(C)CCNC(C23CCC(CC2)O3)=O)cc1[N+](=O)[O-] c1(C(=O)NC2CCN(C(c3c(Cl)ccc(C)c3)=O)CC2C)ncnc2ccsc12 C(=O)(C1=Cc2ccccc2OC1)NC1C(F)CCN(C(C(C=C=C)C)=O)C1 CCC(CCC(=O)NCC1(C)CCCN(C(=O)C(c2ccncc2C)C)C1)OC C(=O)(C(C)(C)C(=O)NCCN(C(=O)C(c1c(F)cccc1F)(C)C)C)NC C=CCCN=C(NCc1ccc(F)c2c1CCCC2)N1CCCC(O)(CO)C1 c1(C(=O)NC2CN(C(c3cnc(CC)nc3C)=O)C(C)C2)cc(C#N)ccc1F C1(CC(=O)NCC(CO)NC(c2ccn(CCOC)n2)=O)CCCCN1C C(C)(C)(C(=O)NCC(O)CNC(=O)C(C)Sc1ccccn1)SC c1(C(=O)NCC2C(C(F)(F)F)CCN(C(COC)=O)C2)ccc(S(N)(=O)=O)cn1 Cc1coc(C(=O)NCc2ccccc2CN(C)C(c2ocnc2CO)=O)c1C C1(NC(C=C(C)C(C)C)=O)CCN(C(c2coc3c2COC3)=O)CCC1(F)F Cc1nc(C)c(CC(=O)NCC(O)CN(C)C(c2oc(CO)cc2C)=O)c(O)n1 c1(CC)ccc(F)cc1C(=O)NCC12CCC(CC1)N2c1ncc(Cl)cn1 C(=O)(C(O)C(F)(F)F)NC1CCN(C(CCN(c2cccc(C)c2)CC)=O)C1 Cc1cc(CC(=O)NC2CCCN(S(N)(=O)=O)C2)cc(F)c1F N1(C(c2cn(CC)nc2)=O)CCOCC(F)(CNC(=O)C(C)OCC2CC2)C1 CC(C)(C)C(O)CC(=O)NC1C2CN(C(c3ccsc3Cl)=O)CC12 C1(CNC(=NCCC)NCCN2CCCOCC2)Cc2ccccc2C1 N1(C(c2c(C)n3c(s2)cnc3)=O)CCC2(CCCCC2NC(c2ccno2)=O)C1 c1(OCC(=O)NCC(CNC(c2cnn(C)n2)=O)CO)cccc(F)c1 c1(C(=O)NC(c2ccc(F)cc2Cl)CC(=O)OCC)ncn2ccc(C)cc12 Cc1ccn(C)c1C(=O)NCCC(O)C(=O)N(C(C)CCC(C)C)C Cc1cn(C)nc1C(=O)NCC(O)CN(C(=O)CCc1cc(Br)cs1)C N1(C(CCCOC)=O)CCCC2C1CCCN2C(c1cc(C(C)C)no1)=O CC1CN(C(c2ncccc2F)=O)CC1NC(=O)CCC1(O)CCC1 CCC(C)CCCC(=O)N1CCCCCC1C(N1CC2(C)CC1CCO2)=O N1(C(CC(C)(C)O)=O)CCN(C(c2cccc(Cl)c2[N+](=O)[O-])=O)C2CCCCC12 Cc1cc(C(N2CCSCC2C(=O)Nc2nnco2)=O)cc(C)c1O N1(CC(=O)NCCCCN(C)C(C2CSCCS2)=O)CCCC1CO C1(C(=O)NCC(C=C)O)CCCCN1C(=O)C(C)NC(=O)C1CC1 N1(C(CCC2N(Cc3scc(C)c3)CCC2)=O)CCN2CCCC2C1 C(=O)(C1Cc2ccccc21)NC1CCC(N(C(=O)CCc2nc[nH]n2)C)CC1 C(c1cccnc1C)=CC(=O)NC1C(OC)CN(C(=O)CCN2CCCC2)C1 CC1CCCc2c(C(=O)NCCOC3CN(C(c4ccccn4)=O)C3)cnn21 c1(CN2C(C(=O)NCc3ncon3)CC3CC32)ccnc(F)c1Cl c1(CC(N2CC(O)(CN(C(=O)CC3CCC(=O)N3)C)C2)=O)ccccc1O N1(Cc2n(CC)ncn2)CCC(CNC(=O)CNC(=O)C2CC2)CC1 c1(OC)cnc(Cl)cc1C(=O)NC1CCC(CNC(=O)C2=CCCC2C)CC1 CCCCC(C(=O)N1CC(CNC(C2(Cl)CC2(F)F)=O)C1)N(C)C C1(C(N2CC(C)SCC2)=O)C2CCC(C2)N1C(=O)C1=CCN(C)C1 N1(C(=O)OC(C)(C)C)CC(C(=O)OCCc2ccccc2Cl)C2CCCC12 C1(C(NNC(C2NCC(C)OC2)=O)=O)CC2(COCCO2)C1 C(=O)(CCCC(C)(C)NC(c1csc(C#N)c1)=O)NC1CN(C(C)C)C(=O)C1 S(=O)(=O)(CC(=O)N1CCC(C(C)Nc2ncc(C)cn2)CC1)NC Cc1ccc(C)c(C(=O)NCCC2CN(C(C3CCC(O)CC3)=O)CCO2)n1 N1(C(C(C=C)(C)CC)=O)CC2CN(C(c3cnc(O)c(OC)c3)=O)CC2(C)C1 c1(OC)cccc(C(n2cc(-c3nccn3C)nn2)C)c1 Cc1cncc(C(N2CCC(C)(NC(C3CC4(CCC4)CO3)=O)C2)=O)c1C C(=O)(CCC(CNC(=O)NC(C1CN(C)CCN1C)C)C(F)(F)F)OC c1(CC)c(OC)ccc(NC(=O)NCC(O)CN2CCN(C)CC2)c1Br C1(CC(=O)NCC(C2OCCOC2(C)C)(C)C)CC(O)CN(C(N)=O)C1 C1(C(=O)NCc2cnc(C)s2)CC2CCCCC2N1C(c1ccc(Cl)cc1I)=O C1(C(N(CCN(C(CCCC(N)=O)=O)C)C(=O)C2CC2)=O)Cc2ccncc2C1 C1(C(F)(F)F)(OC)CCN(C(c2ccn(C(F)F)n2)C(=O)NC2CC2)C1 N1(Cc2nc(C)sc2)CCN2CCOCC2C1.c12c(C)[nH]c(c1C)C(=O)NC2=O c1(-c2cc(CNc3cc(OC)ncc3C(C)=O)ncc2)ncc2ccccn12 C1(CN(C(=O)CC2(CS(C)(=O)=O)CC2)C)COCCN1C(=O)CO c1(N2C(C(=O)Nc3ncc(C)nc3Br)CC(O)CC2)ncnc2cnn(C)c12 C1(CNC(C2C(CC)C2)=O)CC(OC)CN1C(c1ccc(Cn2ccnn2)o1)=O c1(C(N2CC(NC(C(CC=C)CC(C)C)=O)C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 c1(CC(N2C(C)CCC(NC(=O)CN(C)C)C2)=O)cc2cc(Br)ccc2o1 c1(C(N(C(CNC(C=CC(C)C)=O)C)C)=O)ncn(-c2ccccc2)n1 N#CCCC(=O)NC1CCC1CNC(=O)CCC1CCOC1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CS(=O)(=O)CC1NC(c1cccn1C1CC1)=O c1(C(N2CC3CC(NC(c4c(C)oc(Cl)n4)=O)C3C2)=O)ccc(F)c2occc12 C1(CCCC#N)C2(CC2)N1.c1(C(c2nnnn2C2CCCCC2)C)cnccc1C CC(C(F)(F)F)NC(=O)COC(C)(C)CNC(C1COCC1C(N)=O)=O N1(C(c2ccc(SC(F)(F)F)cc2)C(=O)NCC(C)C)CCCCC12CCOC2 Cc1cc(NC(C2CCC2NC(c2n[nH]c3c2CCC3)=O)=O)cc(Cl)c1 C12(C(=O)NCC3(COC)CN(C(=O)Cc4cc(C)n(C)n4)C3)CCC(C1)OC2 S(=O)(=O)(c1ccc(N2CCC3(CC(F)C3)C2)c(Br)c1)NCCOCCC(C)C CC1CCN(C(=O)CCc2nc[nH]n2)CC1CNC(C1OCCCO1)=O c1(C(N2CCC(N(C(COC)=O)C)C2)=O)cc(C(N)=O)ccn1 N1(C(=O)Cc2cc(F)ccc2Br)CCC2(CC1)CCN2C(C1CCCS1)=O CC(C)C(C(=O)N1CCC(C2N(C(c3cc[nH]n3)=O)CC2(C)C)CC1)N(C)C N1(C(c2c(C)coc2)=O)CC2CC1CCC2NC(=O)CCN(c1ccncc1)C c1(CN)cn(CCCC(=O)NCCC2CCNC2)nn1 c1(CNC(C(=O)Nc2scc(C)n2)=O)cnc2cnccn12 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(=O)CC2CC3CCC2CC3)CC1CO N1(C(c2cccc3c2CCC3)=O)CCCC2(CCCN2C(C2CC=CCO2)=O)C1 c1(CN2CCN(CC(=O)NC(C=C)CO)CC2)cccc(C)c1O c1(N(C(C)CNCC)C(c2ccncc2N(C)C)=O)cc([N+](=O)[O-])c[nH]1 C(=O)(C(CNC(=O)CC(O)CN(C)C)C(C)(C)C)NCCCC(C)OC N1(C(C2CCN(C)C2)=O)C2CCC1CC(NC(=O)C#CC1CC1)C2 c1(CC)ccccc1-n1cc(C(N2CC(NC(=O)CCCF)C(C)C2)=O)nn1 Cn1nc(C(=O)NCC(C)(C)OCC(=O)NC2(C)CCC2)cc1F CC(C)C(C(=O)N(C)C)NC(C1CC(C(=O)OCC2CC2CO)C1)=O c1(C(=O)NC2CCN(C(CC=C)=O)C2)nn(C)c2ccc(F)cc12 n12nccc1C=CC2=O.c1(SC(C)C)nnc(C)s1.C(C)(C)(C)N c1(OC)ccnc(C(=O)NCCC2CCCN(C(C3(C(N)=O)CCC3)=O)C2)c1 C1(OCCNC(=O)C=CC2CCC2)CCN(C(=O)CCc2ccccc2)C1 c12cc(ccc1F)CN=C(NCC(=O)OCCCOC)NCCS2.C(F)(F)F c1(C(=O)NC(C(C)NC(CCCC(=C)C)=O)CO)cc(OC)c2c(c1)CC(C)O2 C#Cc1ccccc1CNc1cccnc1C(=O)Nc1cnc(Cl)c(Br)c1 CC(C(=O)NC1(CC=O)CC1)N(C)C1CC1.C(=O)(CCOC1CCOC1)NC C1(C(=O)NC2C(C)C2)CCN(C(=O)COc2ccn(C)n2)O1 c1(C(C(=O)NCC(CC)NC(=O)C(O)C2CC2)C)ccc(C)o1 CC1CC(C(=O)NCCOC2CN(C(c3ccsc3Br)=O)C2)C1(C)C C(=O)(C(C)(F)C(=O)N(CC(C)NC(=O)CCc1ccccc1F)C)OCC Cc1ccc(-c2cc(C(=O)N(CCCNC(=O)CC3(C)CC3F)C)on2)cc1 C(=O)(CC(C)(C)C(C)(F)F)NC1C(CNC(C(CCC)C(C)C)=O)C1 C1(OC)CC(NC(=O)C(=O)NC)CN(C(c2cnc(N3CCC(C)CC3)s2)=O)C1 N1(C(C(C=C=C)C)=O)CCN(C(c2cc(C)nn2CCC)=O)C(c2ncc[nH]2)C1 N1(C(C=Cc2ccc(C)cc2)=O)CCC2C1CCCN2C(C1(C2CC2)CC1)=O c1(C(N2CCC(CCNC(CNC=O)=O)C2)=O)nc[nH]c2ncnc1-2 C1(NC(C(CC2CCCC2)NC(C2C(=C)C2)=O)=O)CCNC(=O)C1 c1(C(=O)OCC2C3CCCCC23)cc(Cl)cc2cc[nH]c12 c1(CNC(C2(F)CCN(C(C3CCC(CC)O3)=O)C2)=O)c(F)cncc1F Cc1ccn2ncc(C(=O)NC3CC(NC(=O)Cc4sccc4Cl)C3)c2c1 C1(OC(NOC(C)C(=O)NCCCCCl)=O)CCCCC1 c1(C(=O)NCC(CC)NC(=O)C(C)CC2CC2)cc(F)c(O)c(Br)c1 C(CC(=O)NC1CC1NC(=O)C(C1(OC)CC1)C1CC1)(OCC)O.C1CC1 N1(C(c2c(C)cccc2)=O)CC(NC(=O)CCCC2CCCO2)CC1(C)C N1(C(C(N2CC(C)OCC2)=O)C)CC(NC(=O)C(C)n2cncn2)C(C)(C)C1 C1(n2cc(CC(OC)OC)nn2)C=CCC(C(=O)NCC(C)(C)C(C)O)C1 N1(C(COC(CC)(C)C)=O)CC(F)(F)CC1CNC(=O)C(F)CC(C)C C1(C(C)NC(=O)CC2CCCCC2)CCN(C(=O)CCN(c2nccs2)C)CC1 C1(O)(C(=O)NCC(C)NC(=O)CCCn2ccnn2)CCCC(C)(C)C1 c1(OC)cc(C(N2CC3CC(C2)C3NC(c2nnc(O)nc2O)=O)=O)c(Cl)cn1 C1(NC(c2cn(C)nn2)=O)C=CCN(C(=O)CCc2ccc(C(N)=O)cc2)C1 C1(CNC(c2c(C)ccn2C)=O)CCN(C(c2cc(C#N)oc2C)=O)C12CC2 c1(C(=O)NCCCC(C)NC(C2CCNC2=O)=O)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NC23CN(C(C(C(C=C)C)C)=O)C(C2)C3)ccc(C)c([N+](=O)[O-])c1 N1(c2cc(CC)ncn2)CCC(NC(c2n[nH]c(-c3ccccc3)c2I)=O)CC1C C12=NC=CC(=NCCCC(=O)N1)N2.C(CCCN(C)C)OC(=O)N(C)CC c1(OC)ccc(CC(CNC(=O)CC(C)C2CCCC2)CO)cc1O N1(C(c2csc(C)c2N)=O)CC2C3CCC(C2C1)N(C(=O)CSCCN(C)C)C3 C1(C(=O)NCC2(OC)CCN(C(=O)C(O)P(C)(C)=O)CC2)OCCOC12CCC2 Cc1cccc(OCC(=O)NCC2CCN2C(=O)COC2C#CCCCCC2)c1C C1(NC(Cc2c(C)nc(Cl)cc2)=O)CC(N=c2nc[nH]s2)C1(C)C CC(CS(C)(=O)=O)C(=O)NC1CCC(NC(=O)Cc2cnn(C)c2C(F)(F)F)C1 Cc1ncsc1C(=O)NCCCC(=O)NCC(C)CNC(C1CC1F)=O c1(C(=O)OCC)cocc1C(=O)NCCC1CC(NC(=O)CC2OCCC2C)C1 C(=O)(C(C)(C)C(C)O)N1CC(NC(c2c(C)sc(-c3ccco3)n2)=O)C1 C1(CNC(=O)C(=O)NC23COC(c4ccccc4)(C2)C3)CC2CC1CC2(F)F C(CCCCC(=O)NC(CC1CCOCC1)C(=O)NC(C)CCOC)OCC C1(NC(C#CC2(C)CC2)=O)CC2CCC1CC2O N1(C(c2c(C)sc(O)n2)=O)CCCN(C(c2ccnc(Cl)c2)=O)CC1C(C)C c1(C(N2C(CNC(c3c(C)nc(CC4CC4)s3)=O)CC2)=O)cc(C#N)cn1C c1(C(=O)NC2(C(=O)NCCOCC)CCCC2)ccn2c(C)ncc2c1 C(c1ccc(C(F)F)o1)=CC(=O)NC(CNC(C(CC)OCC)=O)CC C(C(O)CC(F)(F)F)NC(CCCNC(=O)Cc1cc[nH]n1)=O C1(CC(=O)NC2(CC(=O)NC(N)=O)CC2)CCCCN1C(=O)CCCC(C)C c1(CC)cccc(C(N2CCOCC2CCO)=O)c1O N1(C(c2cnn(CCC)c2C)=O)CCC2(C1)CN(C(=O)CC(CC(=O)O)SC)C2 C1(CNC(C(CC=C)C)=O)CCN(C(c2ccc(F)c(Cl)c2)=O)C12CCC2 c1(C(=O)NC2C(CC)CC2)ccc(SCC(F)F)cc1C(=O)O C1(C(N2CCC(O)C2C2CCOCC2)=O)CCNCC12CCC2 C1(NC(=O)CCC2CCCCC2)CC2CC1N(C(=O)CN1CCCNS1(=O)=O)C2 O=S(=O)(c1ccc(NCCc2ccncc2)c(F)c1)NCC1(C2=CCOCC2)CC1 Cc1ncccc1C(=O)N(C(C)CNC(c1sc(F)cc1C)=O)C C1(CCNC(c2cc(C)ns2)=O)CCCCN1C(=O)C(F)(F)C1(O)CCCC1 CCCCCC(O)C(=O)NC(CC)CCCC(=O)N(C)Cc1occc1C C1(C(N2CC=CC(NC(C3COCCO3)=O)C2)=O)CCC=CCCC1 C(C(CC)CC(C)C)NC(C(Cc1ccccc1Br)NC(C=CC)=O)=O N1(CC2(C(C(N3CCC(c4nccc(C)c4)CC3)=O)=O)CC2)CCc2[nH]ccc2C1 c1(CNCC2(C(C)C)CC2)cccc2c1oc1ccccc21 Cc1noc2ncnc(N3CCCC(CNC(=O)CSc4nncn4C)CC3)c12 c1(C(=O)NC(CNC(C(C)Oc2c(Cl)ccc(C)c2)=O)C)nc2sccn2c1C c1(OC)cccc(C(N2CCC(CC(=O)NCCCN3CCOCC3)C2)=O)c1F c1(CC)ccc(C(=O)NCCC2C(C)CCCN2C(c2n[nH]cc2C)=O)cc1Cl CCC(CC)C(C(=O)N1CC(CNC(C2CC(C(F)(F)F)C2)=O)CCC1C)OC C1(C(=O)NC2C(C(=O)NC3CC(OC)C3)CC2)CC=CCC1C c1(C(=O)NCCCNC(C2CC3CC3C2)=O)cccc2c1oc1ccccc21 C1(C(=O)NCCN2CC(OC)C2)CN(C(C2(OC(C)=O)CC2)=O)CC1C c1(C(N(CCNC(c2ncc(OCC)nc2)=O)CC)=O)c(O)ncc2c1CCC2 C(C)(C)(CC(=O)N1CCC(C(=O)N)CC1)N(C)C.C1CCCCC1n1cccc1 C1(OCC)CCN(C(C2(N(CCOC)CC3CCCO3)CCOC2)=O)CC1 N1(C(Cc2c(C)cnn2C)=O)CC=C(C(=O)NC(C)CS(C)(=O)=O)CC1 c1(C(=O)NCC(CNC(Cc2cn(CC)nn2)=O)O)ccc(CO)c(OC)c1 C1(C(N(C)CC23CCN(C2)S(=O)(=O)C3)=O)COc2ccccc2C1 Cn1nc2c(c1NC(N1CCN(CCNC(=O)NC3CC3)CC1)=O)COCC2 CC(C)C(CCN(C)C(C1CSCCS1)=O)N=c1[nH]c(Cl)ncc1Cl Cc1cc(C(=O)NCC(C)(C)CN(C)C(c2cc(O)cs2)=O)ncc1S(N)(=O)=O c1(C(N2C(CNC(C(C(C)C)(C)O)=O)C(C)(C)CC2)=O)cn(C)c2ncccc12 Cc1c(CNC(=O)Nc2nc(SCC#N)c(C(C)(C)C)s2)nnn1C C1(CNC(c2ncncc2Cl)=O)CCC(F)(CNC(C2CCCS2)=O)CC1 c1(CNC(N2CC3CC(C(F)(F)F)C3C2)=O)cc(=O)c2ccc(Cl)cc2o1 N1(C(Cc2ccc(C)cc2)=O)CC(NC(C2(C)CCCN2C)=O)CC1(C)C c1(C(=O)NC(CN(C(C(C)Cc2ccccc2)=O)C)C)cc[nH]c(=N)c1N c1(C(N2C(CNC(=O)C(C)SC)CC(OC)C2)=O)nccc2ccn(C)c12 N1(CC(N2CCCC(C(=O)OCC)C2CC)=O)C(=O)NC(C)(CC)C1=O c1(CC(=O)NCC2CC(O)CN2C(=O)Cc2n[nH]cc2Br)cc(F)cc(F)c1 N1(C(C(C(C)(C)C)=O)=O)CC2CCCCC2(NC(=O)CC2=NNC(=O)C2)C1 N1(C(C2(C=C)CCC2)=O)CCN(C(=O)CC(C)C)CC2CCCCC12 N1(Cc2nn(C)c(I)c2)CCC2(CCC2)C(NC(=O)OC(C)(C)C)C1 C(=O)(C1CCCn2cc(C)nc21)N1CCN(C(CCC=CC)=O)C(C)C1 C1(CNC(C2(C)COC2)=O)(CNC(c2ncccc2C(F)F)=O)CC12CCC2 CC1CC(C(=O)NC(C)CN(C)C(c2cc3[nH]ccc3s2)=O)CCN1C N1(C(CC)=O)CCC(C2CCCN2C(=O)NCCSCCO)CC1 C1(F)(CNC(c2nc(C(C)C)oc2)=O)CCN(C(C2CCCS2)=O)C1 C1(CNC(C(CC)n2ccnc2)=O)CCN(C(c2cn(CCO)nn2)=O)CC1C C(CC(C(=O)N1CCC1CC1CC1)NC(=O)C(=C1CCCCC1)F)N(C)C c1(C(N2CC(CCC)N(C(=O)CCNC(N)=O)CC2)=O)cc(C)c2[nH]cnc2c1 CN1CCC(C)(C(=O)NCc2ccc(C(=O)NC(CO)CCO)o2)C1 C12CCN(CC1)C(=O)CO2.Cc1ccsc1-c1cn(CCc2cn[nH]c2)nn1 C1(C(=O)NCCCN(C(C=CC(=O)OC)=O)C)CC1(C)C(C)C c1(SC)ccc2cc(C(N3CC(NC(=O)CCn4ccnn4)C4CC34)=O)[nH]c2c1 CC1CC(N=c2[nH]n(C)c(C(F)(F)F)c2S(=O)(=O)NCCN2CCCC2)CCO1 c1(OCC(=O)NC2CC(CS(C)(=O)=O)C2)ccc(Br)cc1C#N S(=O)(=O)(c1[nH]c(=NC(C)CCN2CCCCC2=O)ccc1Br)NC(C)CC1CC1 c1(C(=O)N(C2(C)CC(F)C2)C2CC2)ccc(Br)cc1 Cc1nc(C(=O)NCC2CCN(C(c3scnc3C(F)(F)F)=O)C2)nn1C c1(C(N2CCC(C3N(C(CCC=C)=O)CCC3)C2)=O)cc(OCC)cc(Br)c1C Cc1sncc1C(=O)NC(CO)C(C)NC(C1CC1C(N)=O)=O C1(C(=O)NC2(C)CN(C(CCc3ccn(C)c3)=O)C2)CCn2cnnc2C1 C12(CC)CC1CN(C(C1C(C)OCN1C(c1ccon1)=O)=O)C2 Cn1ncc2c1CCC(C(=O)NCC1CCCN1C(c1nnc(O)nc1O)=O)C2 C1(CNC(c2cccc(C)c2)=O)C(C2CC2)CCN1C(=O)C(c1ccn(C)n1)C CC1(C)OCCC1C(N1CCC2CC12C(=O)NCCC1CC=CCC1)=O CCCCC(O)CC(=O)N1CC(COC)(NC(c2cccc(F)c2OCC)=O)C1 N1(C(c2c(CC)ccs2)=O)CCCC2C1CCCN2C(C1CN(C(=O)OC)C1)=O c1(C(c2nc(F)ccc2Cl)=O)cc2[nH]ccc2cc1-c1cc[nH]n1 Cc1nsc(C)c1C(=O)NCC(C1CCC1)NC(c1cc(C(C)(F)F)n[nH]1)=O Cc1ccc(CCC(=O)NC2CC(CNC(C3CCCN3CCC(C)C)=O)C2)s1 C=CCC(CC)C(=O)NC1(CO)CCN(C(c2cnc(CO)nc2C)=O)C1 C=Cn1nncc1C(=O)N(C(C)C(N1CCCC1C(=O)NC(C)C)=O)C C#CC1(O)CCN(C(C2(CNC(C3CN(C)C(=O)N3)=O)CC(=C)C2)=O)C1 Cc1nc(CC(C)C)c(C(=O)NCC(C)CN(C)C(C2(C)CC2)=O)s1 c1(N(C2CCCN(C(=O)C(c3ccc(F)cc3)F)C2)C)ncccc1[N+](=O)[O-] C1(C(N2CC(C(C)NC(C=C(C)c3cccs3)=O)C2)=O)CNc2ccnn2C1 N1(C(C(CSC)C)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CC1C1CCC1 N1(C(C(CC(C)C)OC)=O)CC2CCCC(C1)N2C(=O)Cn1ncc(Br)n1 C1(CC(=O)NC(C2CCN(C(=O)C(C)=CC)C2)(C)C)(CC=C)CCCC1 N1(C(c2ncc(CC)cn2)=O)CCC(O)CC1C(N1CC(CC2CC2)C1)=O Cc1cc(C(=O)NCCOCCNC(=O)C(CO)N(C)C)cc(C)n1 C1(CC)(NC(=O)C(C)N(C)C)CCCN(C(=O)C(c2ccc(Cl)cc2OC)=O)C1 C12(NC(C(COC)NC(=O)CCc3cn(C)nn3)=O)CC1COC21CCC1 c1(C(=O)NCC(CNC(C(C(C)C)SCC)=O)O)ccc(O)cc1[N+](=O)[O-] N1(C(C(c2ccc(C)o2)C(=O)Oc2ccccc2)=O)CC2CCN(C(=O)CO)C2C1 N1(C(C2CCN(C(CC)=O)C2)=O)CC(C)(C)CC1CNC(=O)CCC1(C)CC1 N1(C(c2ccc(C#N)[nH]2)=O)CC(NC(=O)CSCC(=O)OC(C)(C)C)CC(O)C1 c1(NC(C2N(Cc3ccc(CC)cc3)CC=C2)=O)cnc(C#N)c(C)n1 C12(CNC(c3ccc(Br)nc3)=O)CC1CN(C(=O)CCCC1CCCC1)C2 N1(C(Cc2c3cc(C)sc3sc2)=O)CCC2(CC1)CN(C(=O)Cc1cnoc1)C2 c1(C(N2CC(F)(CNC(C3CC(O)C3)=O)C2)=O)[nH]cc2c1CCC2 c1(CCOCCN(C2CCC(O)CC2)C)ccc(F)cc1F.C=O C(=O)(CCC(F)(F)F)NC(C1CCCN1C(c1ccc(C(N)=O)c(O)c1)=O)C C(=O)(C1=NOC(C(N2CCC(CCNC(=O)CCc3ncc[nH]3)C2)=O)C1)OC C(C(C(=O)N1CC(CC(=O)OC)C1)C(C)(C)C)NC(C1N(CC)CCC1)=O C1(C(CNC(c2c(NC(C)=O)ccs2)=O)=O)CSc2ccccc2O1 C12(C(=O)NC(C)CNC(=O)C(=O)N=S(C)(C)=O)CCC(N=[N+]=[N-])(CC1)C2 C1(C2(O)CCN(C(=O)C(C)(F)CCCC)CC2)(NC(CCC(=C)C)=O)CC1 C1(C(=O)Nc2c(C)nsc2)CCCN(C(C2(C)CC(C)(C)C2)=O)CC1 C1(OCC)CCCC1NC(=O)CN(C(C1CCOC1C)=O)C1CC1 C1(CNC(c2ccc(CCC)[nH]2)=O)COCCN(C(c2c(N)sc(C)c2C)=O)C1 N(C1COCc2ccccc21)C(=O)CC(Cc1cc(I)ccc1F)NCC1CC1 c1(OC)ccc(CCC(=O)NC2CCC2NC(c2ccc(C)nc2)=O)cc1Cl c1(CC)ccc(C(=O)NC(C)(C)CNC(=O)CCC2CC2(Cl)Cl)c(C)n1 C#CC(C(C)(C)C)NC(=O)CCN(C)C(C1(C)CCC(=O)C1)=O c1(C(N2CC(NSC(F)(F)F)C2)=O)cc(Cl)ccc1Oc1ccccc1 C12(C(=O)NCCCN(C(C3(C(F)F)C(C)C3)=O)CCO)CC3CC(C1)CC(C)(C3)C2 c1(OC(C)C)cccc(C(CCCc2ncc(C)s2)OC)c1.C1(C)(C)CC(=O)N1 CCC(CCCC(=O)N1CCC(N(C)C)C1C)NC(C1CC12CCCC2)=O c1(C(=O)NCC2CCN(CCCc3cccc(OC)c3)C2)ccc2c(c1)CCO2 C1(C(=O)NC2(CC(=O)N(CCC#C)CC)CCC2)CC2CC(=O)C1O2 C=CC(C)(O)CC(=O)NC1CCC(NC(c2n[nH]c(C)c2C)=O)C1 C1(NC(CCN(C)CC)=O)CC2CC(C1)CN(C(=O)C1CC1)C2 C1(CCCC)(C(=O)N(C2CC(NC(C3CC3COC)=O)C2)C)CCCCC1 CCCC(C(O)C(=O)NC1(CO)CC1)NC(c1c(CC)noc1C)=O N1(C(C2(CC#C)CC=CCC2)=O)CCCC(NC(c2ccc(N)c(F)c2)=O)CC1 C(=O)(C(CC(N)=O)NC(=O)CN1CCCC1C)NC1(CCC)CCOC1 N1(C(CCSCC)=O)CCCC(C)C1CNC(c1cc(C)nc(C2CC2)n1)=O CC(C)CCCCCNS(=O)(=O)c1cccs1 Cc1nc(NCCn2cncn2)cc(=NCc2ncoc2C(F)(F)F)[nH]1 C(=O)(C(C)(C)C(F)(F)F)NC1CCCC(NC(C(CC)(C)F)=O)C1 c1(C(=O)NC(C2CC(NC(C3C(C)(COC)C3)=O)C2)C)cc2n(n1)CCC2 C(=O)(C1=CC(C)(C)C1)NC(C(=O)OCC)C1CCOC1 N1(C(C(C)N(CCC)C(n2nc(C)cc2C)=O)=O)CCCC(C)(NC(C)=O)C1 c1(C(=O)NCC(C(C)(C)C)NC(C2ON=C(CC)C2)=O)cc(C#N)cn1C N1(C(C2CCCC(=O)C2)=O)CCC(NC(c2ccc(C(F)F)o2)=O)CC(O)C1 c1(OCC)ccnc(C(N2CCCC2CN(C(=O)Cn2cc(C3CC3)nn2)C)=O)n1 C1(C)(C(N(C(CC#C)C)C)=O)CC(NC(=O)C(C)CC2CCCC2)C1 c1(NC(C(CCOCC)NC(C2CC23CCC3)=O)=O)nccc(C)c1F C1(C(N2C(CN(C)C(C3Cc4nncn4C3)=O)CCC2)=O)CCC12CCOCC2 c1(CCC(=O)NCC(C2CCOC2)NC(C(C)=CC)=O)nnc(S)n1C N(C(=NCC(C)C)NCc1cnc(C)s1)C(c1ccc(OC)cc1)C N1(C(C#C)CC2CCC2)CCC(=O)N(CCCOC)C1=O c1(NCCCC)ccc(S(=O)(=O)NC2CCN(C(=O)N(C)C)C2)c(Br)c1 C1(NC(=O)CC2CCCC2)CCN(C(c2cc[nH]c2)=O)CC1F c1(COC(CNCC(Cc2cn(C)nc2)C(F)(F)F)=O)ccc(S(=O)CC#N)cc1 C1(CN)CCCN1C(c1cc(CNC(C)(C)C)cs1)=O.CC1CC1(F)C(=O)C(=O)OC N1(C(C(c2n(C)ccn2)(F)F)=O)CCC(C)(CNC(=O)Cn2nccn2)CC1 C1(CNC(C)=O)CN(C(C)C(=O)Nc2nnc(CC(C)C)s2)CCC1(F)F N1(C(C(CNC(CC(C=C)CC)=O)CCC)=O)CCC2CN(C)CC2C1 CC(C)C(C)CC(=O)N(CC(C1CCCC1)NC(=O)CCF)C1CCC1 N=c1[nH]cc(C(=O)NOC2(C(=O)O)CC2)s1 C1(NC(C2CN(C(C)C)C2)=O)CC2(CCCCN2C(=O)CCc2nncs2)C1 c1(CC(=O)NCC2C(NC(C(C)S(N)(=O)=O)=O)C2)ccc2c(c1)COCC2 N1(C(=O)NC2CCC(CC)CC2)CCN(C(c2cccc(F)c2F)=O)C(C)C1 O=C1CCN(CC2CNC(=O)C2(F)F)C(=O)N1CC1=CCOCC1 C(=O)(C(O)C1=CCCCC1)NCC1N(C(C(c2cncc(F)c2)C)=O)CCCC1 C12(NC(C(C)NC(N)=O)=O)CCCC1N(C(c1cccc(F)c1N)=O)CCC2 c1(C(=O)NC(C2CCCN(C(c3snc(Cl)c3Cl)=O)C2)C)cc(F)cc(Br)c1 C1(NCc2ccn(C(C)C)n2)CCCC2NCCC12 c1(OCCCC)ccc(C(C)NCc2cscc2C#N)cc1 C1(NC(C2(C)CN(C(=O)OC(C)(C)C)C2)=O)CC(C)CN(C(C(CC)CC)=O)C1 N1(C(C2(CC)COC2)=O)CCCC2(CC(NC(=O)C(C)(C)c3cnsc3)C2)C1 C1(NC(CC(C)(C)C(F)F)=O)CC2CCC1CN(C(=O)C1=CCCC1)C2 c1(C(N2CC(C)CC(NC(CCC(C)=O)=O)C2)=O)cc(S(N)(=O)=O)ccc1C c1(OC)cccc(C(=O)NCCC2CCN(C(C3(C)CC(C)=NO3)=O)CC2)c1Cl c1(N2CCN(C(C3C4CCCCCCC34)C)CC2C)nc2c(C)cccc2o1 C(C)(CCCC(=O)NC1CSC1)NC(Cc1cc(C)sc1)=O C1(F)(C(=O)NC(C(=O)N(C)C)CO)CCN(C(=O)CCc2cnn[nH]2)C1 C(=O)(CC(C)C(=O)N1CCC(C=CC(=O)Nc2cc(OC)cc(O)c2)CC1)OC Cc1noc(C(=O)NCC(O)CCNC(C2CC(N(C)C)C2)=O)n1 C1(C(=O)NC2CN(C(c3ncn(C(C)(C)C)c3)=O)C2)CCCC(C(F)(F)F)C1 N1(C(Cc2ncc(C)o2)=O)CC(NC(c2ccc(F)c(F)c2)=O)CC(O)C1 N1(C(C=C(C)C(F)F)=O)CCC(NC(c2ccc(CS(C)(=O)=O)o2)=O)C(C)(C)C1 C1(CNC(C2CN(C(C)=O)C2)=O)C(O)C(O)CN1C(=O)Cc1cccc(Cl)c1 C1(NC(c2sc(C)c(Br)c2)=O)CC2CC1N(C(c1csnn1)=O)C2 c1(C(=O)NCC(C)N(C(C2(CC=C)CC2)=O)C)cc(SC)oc1C CCC(CC(=O)N(C1CCCN(C(c2cnsc2C(F)(F)F)=O)CC1)C)C(F)F c1(C(N2C(CNC(CCC(=C)Br)=O)CC3CC32)=O)cn2c(n1)CCCC2 C1(C=O)CCCCC1C1CC1.Cc1cnc(C)cn1.C12C3CN(CC13)n1nnnc12 C1(CNC2CC(=O)N(CC(F)(F)F)C2)CCCS(=O)(=O)CC1 C1(C(=O)NC2(c3ccccc3)CN(C(C3CC4CCCC34)=O)C2)CC(C2CC2)C1 c1(OC)ccc(CN2CCCC(CNC(c3cnc(Cl)nc3)=O)C2)c(OC)c1 C(=O)(C#CC1(C)CCCO1)NC12C(CN(C(C(C)OCC=C)=O)C1)CCC2 n1(C(CC)C)ccc(=NC(=O)CC2(NC(c3ccnc(OC)c3)=O)CC2)[nH]1 C(=O)(C(CCCC(C)(F)F)N(CC(=O)OC(C)(C)C)C)NCc1c(C)c(Br)ccc1 N1(C(C(CCC)O)=O)CCC(C)(C)C1CNC(=O)C=Cc1ccc(C2CC2C)o1 C(=O)(CC(CC)C(C)C)NC(CC=CC)C(=O)NCC(C)(C)C1=CCCC1 C1(NC(C(CC)=CC)=O)CCC2(CC1)CC2NC(=O)C(=O)NCC N1(C(CC(CCCC)CC)=O)CC2CCN(C(=O)C(CC)CCOC)CCC2C1 c1(C(N2CCC(C)(CNC(=O)CC3COCCOC3)C2)=O)cccn2nccc12 c1(OCCOC(C)=O)nc(OC(c2ccnc(C)n2)C)c2ccccc2n1 N1(C(C(CCSC)O)=O)CC2CCN(C(=O)CC3CCCC(O)C3)CC12 C(=O)(C1CCNc2cc(F)ccc21)NC(C1CN(C(C2CC(C)(F)C2)=O)C1)C Cc1cccc(C(F)(F)C(=O)NC(C2CN(C(=O)CC3CC(O)C3(C)C)C2)C)c1 C1(NC(C(C)Cc2ccccc2Cl)=O)CN(C(=O)Cc2cn[nH]c2)C(C)(C)C1 c1(C(=O)NC2CN(C(C3(C)CCN(C)C3)=O)CC2F)ccc2nnn(C)c2n1 N1(C(C2(OCC)CCCCC2)=O)CCCCC2(CCN(C(=O)C(C)C(C)O)C2)C1 N1(CCC)CCCC(C(=O)NC2CCC(NC(=O)C(CCSC)OC)CC2)C1 C1(C(N2CCC(N(C(=O)COCC3CCCO3)CCC)C2)=O)NC(=O)OC1(C)C C1(N(C(CCCCCCSC)=O)C)CCCC2CN(C(=O)C(C)CC3CC3)CC12 c1(C(=O)NCC(C(C)C)NC(C2(C)CCCO2)=O)cc[n+]([O-])cc1 Cn1ncc2c(O)c(C(=O)NCC#CCNC(=O)Cc3csc(Br)n3)cnc12 c1(NC(C2CC(N(C(c3nc(CC)oc3)=O)C)C2)=O)ccc(C)cc1C N1(C(CC(C)SC)=O)CCOCCC1C(=O)NCCOCC(N)=O CC12CCN(C(C3CCCCC3(F)F)=O)C1CN(C(C1CCCN1C1CC1)=O)C2 c1(CC(N2CC=CC(NC(C3(F)CCOC3)=O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] C1(COC)CN(C(c2coc(C3CC3)n2)=O)CCN1C(C1CC1F)=O.c1nncs1 N(C(=NCCCc1nnc(C)n1C)NCCC(=O)NC)C(CC)C(F)F C1(CNC(C2C(C=C)C2)=O)CN(C(c2csc(S)n2)=O)C(C)(C)C1 C1(C(N2CCCC(OC)C2)=O)C2CCCC1CN(C(c1cc(Cl)nc(Cl)c1)=O)C2 C(=O)(CCC(C)(C)C)N(CC(N1CC(SCC)C1)=O)CC(=O)NC c1(C(N2CCC(CNC(=O)CCn3cnnn3)C2)=O)n[nH]c(C(F)(F)F)c1Cl c1(SCC(=O)N(CC(C)(C)NC(C2CCCS2)=O)C)n[nH]c(O)n1 c12ccc(F)cc1S(=O)(=O)NC2(C)C.c1(COC)ccc(C(=O)O)o1 C(CCCCCN=c1ccc(S(C)(=O)=O)c[nH]1)NC(C(CC)NC(C)=O)=O c1(C(N2CCC(C)C(CNC(c3ccnnc3)=O)C2)=O)cnc(O)n(C)c1=O C#Cc1cc(F)c(C(N2CCC(CN(C)C(C34CCN(CC3)C4)=O)C2)=O)c(F)c1 N1(C(C(CC)N(C)C)=O)CC2(COC(CNC(=O)C(F)=CC3CC3)C2)C1 C(=O)(CN1C(=O)CSc2ccccc21)NC1C(C2CCN(C(CCC)=O)CC2)C1 c1(NC(=O)NC(C)C(C)(C)CN(C)C)cc(O)nc2c1CCCC2 CC1=C(C(=O)N2CCCCC2CCNC(c2nnc3n2CCCC3)=O)CCCO1 c1(OC)cccc(C(=O)NCCN(C(=O)C(C)(C)CC2CC2)C2CC2)c1 C(=O)(C1=CCCCCC1)NC1CCN(C(Cc2c(OC)ccc(F)c2)=O)CC1O N1(Cc2ccc(C(=O)Nc3c(C)ncs3)s2)CCC2CN(C)CCC12 c1(C(C(C)N(C(C)C)C)N)ccccc1.C1C(=O)N1.C1(C(=O)N(C)C)(CCN(C)C)CC1 C1(C(C)NC(C2CCC2)=O)CCN(C(=O)C=C(Cl)Cl)C1 C1(NC(=O)CC2(c3ccon3)CCC2)CC(O)CN(C(=O)C=CCF)C1 N1(C(C2(C(=O)OC)CC2)=O)CC(C(C)(C)NC(C2(C(C)(F)F)CCC2)=O)C2(CC2)C1 N1(C(CSCC=C)=O)CC(NC(c2sccc2NCC)=O)CC1(C)CC CC(C)C(C(=O)NC1CC(F)(CNC(=O)CSc2nnnn2C)C1)n1cnnc1 c1(C(N2C3CN(C(C(COC)N(C)C)=O)CC2CC3)=O)c(S(N)(=O)=O)ncn1C C1(CC)(CC)CCN(C(=NCc2ccc3c(c2)ncn3C)NC)C1.C(C)O c1(CC)nc(C)c(CNC(C2C(O)CCN2C(=O)C(C)(CC)OC)=O)o1 CCCCCCC(=O)N1CCC(NC(=O)CCNC(C)=O)C(F)C1 N1(C(CC2CC(OC)C2)=O)C2CC1CN(C(c1ccc(C)c(C)n1)=O)C2 N1(C(CCC#C)=O)CCCC(C)C1CNC(=O)Cn1nc(C(C)(C)C)cc1N C1(C(=O)NC2(CCNC(C(C)(C)SC)=O)CC2)CN(CP(C)(C)=O)C1 c1(NC(c2c(N)cc(F)cn2)=O)cc(F)cc(Br)c1Cl CC1CC2CN(C(c3ccc(Br)s3)=O)CC2N1C(c1ccc(=N)[nH]n1)=O c1(C(=O)NCC2CCC(NC(C3CC3(F)F)=O)C2)c(Cl)csc1Cl N1(C(c2occ(C)c2)=O)CC(F)(F)CC1C(=O)Nc1cccc(CN(C)C)n1 c1(C(N2C(CNC(c3[nH]cnc3C)=O)CC(OC)C2)=O)cccc2[nH]ncc12 C(C1CCCCC1)=CC(=O)NCCSCC(=O)NC(C)C(C)n1cncn1 CC(C)C(C)CC(=O)N(C1CCC(NC(=O)COC2CCOC2=O)CC1)C N1(C(CC2(CSC)CC2)=O)CCCCCC1CNC(C1OCCC1(C)C)=O N1(C(c2csc(C(F)(F)F)n2)=O)C2CN(Cc3cnc(Cl)nc3)CC12 CN1CCC(NC(c2cccnn2)=O)C12CCCN(C(=O)C1=C(Cl)CCOC1)C2 C1(CCNC(CC(C)NC(C2CCCC2)=O)=O)CSCCN1C(c1cscn1)=O N1(C(C2CC(O)(CC#C)C2)=O)CCC(C)(CNC(=O)CC2(C)CCCO2)C1 CC1(NC(C2CC2F)=O)CCN(C(c2ccc(C(F)(F)F)o2)=O)C1 C1(CC(C)O)CCN(Cc2ccc(Br)o2)CC1.c12cc(ncn1)CN2 N1(C(C2C(C#C)C2)=O)CCOC2(CCN(C(=O)C(C(C)C)NC=O)CC2)C1 c1(CN=C(NC(CC)C)NC2CCC(=O)NC2)nn(C)c2c1COCC2 C1(CNC(C(=O)NC(C)C)=O)(CO)CCN(C(C2CC23CCCC3)=O)CC1 CC(CC(=O)N1CC(CNC(c2cccnc2-n2cncn2)=O)C1)C(F)F N1(C(c2c(C)cncc2F)=O)C2CCC1CC(NC(=O)CCc1cn[nH]c1)C2 c1(C(=O)NCC(C(C)(C)C)NC(C2CC(C)(F)C2)=O)c[nH]c2ccc(Cl)cc12 CC1(O)CCN(C2CCCC2c2ccccc2)CC1(O)c1ccccc1 C1(C(=O)NCCCC)CC(C)CCN1Cc1nc(O)n[nH]1 C1(C#N)(C(=O)NCCN(C(CCc2ccn(C)n2)=O)C2CC2)CCCC1 C(N=c1[nH]c2cc(Cl)ccc2s1)C1N(C(c2n(C)ncc2)=O)CCC1 C(=O)(CCCC(=O)NC1CN(C(C2(C)COC2)=O)CC1C)Nc1c(C)cccc1 n1(CC)nc(C(C)C)cc1C(=O)N(CC(C)(C)NC(=O)Cc1cocn1)C c1(C(=O)Nc2nc3ccccc3o2)cccc2c(I)n[nH]c12 CCC(C)(C)C(=O)C(=O)NC1CCN(C(c2csc3nnsc23)=O)C1C N1(C(C2CC(C)(O)C2)=O)C2CCC1(CNC(=O)Cc1cccc(F)c1Cl)CC2 N1(C(C2N(C)CCC2)=O)CC2CCC(NC(C3CC4(C3)CC3(CC3)C4)=O)(C2)C1 C1(C(=O)NCC2CC(C)N(C(=O)CNS(C)(=O)=O)C2)CCc2nncn2C1 c1(C(N(C(C)CCNC(c2ccoc2Cl)=O)C)=O)cccc(C2CC2(F)F)c1 C(CC)(C(=O)NCCC(C)N(C(=O)CN(C)C(=O)C1CC1)C)=CCCC C1(C)(C(N2CCC(C(C(=O)Nc3ccc(OCC)cc3)C)C2)=O)CCCN(C)C1 C(=O)(C(F)C(C)CNC(c1csnc1OC)=O)NC(CC=C)(C)C Cn1nccc1C(CC#N)Nc1sccc1NC(C1C(C(=O)OC(C)(C)C)C1)=O c1(C(N2CC3C(CNC(c4csc(Cl)c4)=O)(C3)C2)=O)nnc(O)nc1O C1(C(C(=O)N2C3CN(C3)C(=O)C2)C)CCOCC1.C1(SC)CC1 C1(CNC(Cc2cn(C(C)C)nc2)=O)COCCN1C(c1cnc(C2CC2)o1)=O c1(C(=O)NC(C2CCCC2)CNC(C2CC(=C)C2)=O)cnc2n1CCC(C)C2 c1(OC)ccccc1-c1nc(CCCO)nn1Cc1ccc(I)cc1 C(C(C(=O)NC(C1CCCN1C(=O)CCC1CC1)C)c1ccccc1)SC N1(C(=O)NC(c2cccc(Cl)c2)C(F)F)CCOC(C2CCOC2)C1 O=C1NCC2(CCN(C(=O)C(=O)Nc3ccc4sccc4c3)CC2)C1O c1(CC(C)NC(c2cc(CNC(c3coc(CO)c3)=O)[nH]n2)=O)nncn1C N1(C(C(CC=C)C)=O)CC2(CCC2)CCC1CNC(=O)CC1CC1 CC(CCCCN=c1ncc(F)c[nH]1)NC(=O)CCOCC1CCCO1 C(=O)(CC(C)C(F)F)NCC(C(=O)NC(C#C)C1CCC1)CC1CC1 Cc1cc(F)sc1C(=O)N(C(C)CNC(c1cccc(-c2nc(=O)o[nH]2)c1)=O)C C(=O)(CCCC(F)(F)F)N1C(CNC(c2nccc3cc[nH]c23)=O)CC(F)C1 O=C(CC(C(F)(F)F)NC(C1(F)CCOCC1)=O)NCC1CC1[N+](=O)[O-] c1(C(=O)NCCC2(O)CCCN(C(=O)CCCF)C2)ccc2c(c1O)CCCC2 c1(CC)nc(C)c(CC(=O)NCCCCCNC(C2(C)CCCC2O)=O)c(C)n1 C=C(C)CC(C(=O)NCCCN(CC)CC)NC(=O)Cc1cncc(C)c1 C1(OC)CC(NC(C2CC3C=CC2O3)=O)CN(C(=O)CN2CCC(CO)CC2)C1 C1(NC(c2ccc(C(N)=O)cn2)=O)CC2CC(NC(c3sccc3CO)=O)C1C2 C1(C(=O)NCC(C)NC(C2(OCC)CCC2)=O)CC(=O)N(CSCC)C1 C1(C(N2C(CNC(c3c(C)cns3)=O)CC2)=O)CCC(O)CN1C C1(CNC(C2(COC)CC2)=O)CN(C(c2cc(OC)n[nH]2)=O)C(C)(C)C1 c1(OC)ccc(C(=O)NC(C2CCCN2C(c2ncncc2Cl)=O)(C)C)cn1 CC(C)(C)C1=NOC(C(N2CC3CCC2CN3C(C2CC(CC3CC3)C2)=O)=O)C1 c1(C(=O)NCC(CC(=O)N(CCNC(C)=O)C)C2CC2)ccnc(O)c1F C1(F)(CNC(c2c(C)ccnn2)=O)CCC(CNC(C2CCNC(=O)C2)=O)CC1 N(C(=NCCSC)NC1CCOc2ccc(F)cc21)CC(C)N(CC)CC C12(OC)CCC1CN(C(C13CC(CN(C(=O)C(CC(C)C)OC)C1)C3)=O)C2 N1(C(c2c(NC(=O)NC(CC)C)cc(C)cc2)=O)CCCc2cccc(Br)c21 CCC(CCC(=O)NC1CC2CC1CC2C(=O)NCC1CCCC(OC)C1)OC c1(OC)ccc(Br)cc1NC(=O)C(N1CCOC(CCN(C)C)C1)=O Cc1nc[nH]c1CC(=O)NC(C1CCN(C(c2cnsn2)=O)C1)(C)C N1(C(CCC2CCN(C)CC2)=O)CCN(C(C2CC(N(C)C)C2)=O)C2CCC12 C=C(CNC(=O)C(CC(C)C)N(C)C(C1CCCC(=O)N1)=O)C1CCOCC1 c1(-c2cc(C(=O)Nc3cnc4ccccn34)ncc2)cccc(C2=CCOC2)c1 C1(NC(CCC=CCC=C)=O)C2COCC1CN(C(c1cccc(N)c1)=O)C2 CC1(C)CC(CC(=O)NCC(C)(CO)N(C)C)N(C(c2ccc[nH]2)=O)C1 c1(OC)cc(C(=O)NC(C)CN(C(=O)CCC2(C)CCC(=O)N2)C)c(Cl)cn1 C1(C=O)Cc2ccccc2C1.C12CCN(CC1)N2CC.C(=O)(CSCC=O)OCC Cc1ccc(O)c(C(=O)NC(C)(CNC(=O)CC2SC(=N)NC2=O)C2CCC2)n1 CC(C)(CCCNC(c1cccs1)=O)C(=O)N1CC2(CNC(=O)C2)C1 N12CCCC13CCCN(C3)CC2=O.Cc1cc(NS(=O)(=O)CC#N)cc(C)c1Br c1(-c2nc(CC(C)(C3CCC3)OC)n(CC(F)(F)F)n2)ccc2ccccc2c1 CN1CC(O)CCC1C(=O)NC(CC1CC1)CC(N1CCCC(CO)CC1)=O c1(C(N(CC)CC2CCCN2C(c2csnn2)=O)=O)ccc(C)nn1 C(=O)(C(O)(C(C)C)C(F)(F)F)N1CC(C)(NC(Cc2ccc(C)c(C)c2)=O)C1 C(=O)(C1CCCc2ccnn21)N1C(C)CCC(CNC(=O)C2=NNC(=O)CC2)C1 CC1(CNC(C23CCCC2C3(F)F)=O)CCN(c2nc(Cl)ncc2F)CC1 c1(C(=O)NC2(CNC(CC(=O)OC)=O)CCCCC2C)nc2cc(F)ccc2s1 Cc1cc(C(=O)NCC2=CCN(C(C3CCCC(=O)N3C)=O)CC2)cc(Cl)n1 C1(C#N)(C(=O)NCC2(O)CC(C(=O)NCCC(C)CCO)C2)CCCOC1 c1(C(N2CC3C(CNC(C(C)NC(C)=O)=O)(C3)C2)=O)ccc(C(F)(F)F)nc1O C(C(C(=O)NC(C)CCCC1CC1)C(C)C)NC(C(CC=C)OC)=O C12(CNC(c3ccnn3CN)=O)CN(C1)C(=O)N2.C(C)(C)(C)OCC C1(C(=O)NCC2(NC(c3cc(N)c(O)cc3)=O)CCC2)CCCCC12CCC2 Cn1ncc(COc2ccccc2)c1S(=O)(=O)Oc1ccc(N)cc1 c1(NC2C3(CC(NC(CCOCCCOC)=O)C3)C2)ccnc(S(C)(=O)=O)n1 C1(NC(C2CN(C)C2)=O)CC(NC(c2c(O)cccc2Cl)=O)C12CCC2 Cc1cc(C(N2CC3(CNC(C4CC(O)C4)=O)CCC2C3)=O)nc(O)c1 C(CC(=O)NCCOC1CCCC1)(C(C)OC1CC1)NC(C=C(COC)C)=O C(=O)(C1=CC(O)C(NC(C2(O)CCOC2)=O)C1)Nc1cc(C)cc(C)c1 c1(NC(c2[nH]c(=NCc3ccc(OC)cc3)sc2)=O)c(C)ccc2ncccc12 c1(OC)c(C(=O)NC(C2CC=CCC2)C(=O)NC2CN(C)NC2=O)cnn1C c1(CC)ccc(C(=O)NCc2occc2C(=O)N(CC(F)Cl)C)nc1 Nc1cnc(Cl)cc1C(N1CCC1CNC(=O)CC(O)C1CC1)=O C1(CC)CCCC1C(=O)NC1(CCNC(C2CC(F)(CO)C2)=O)CCC1 C(C)(CO)(C(=O)N(CCCCCNC(=O)C(C)N1CCC1)C)OC c1(C(C)C(N2CCC(NC(C3CCC(=O)C3)=O)CC2)=O)ccc(S(N)(=O)=O)cc1 C12(CCOCC1)C(=O)N2.c1(CC)cccc(C(=O)NC2C(O)CC2O)n1 c1(C(=O)NC2(C)CN(C(C3(C=C)CCCCC3)=O)C2)cc(C)c(Cl)c([N+](=O)[O-])c1 N1(C(c2cc(Br)cs2)=O)CCN(C(C2OCCCO2)=O)C(CF)C1 c1(NC(C2CCCN(C(C3CCC(=O)N3)=O)C2)C)cc(C2CC2)ncn1 N1(Cc2c(C(C)(C)C)ocn2)CC2C(NC(=O)C(O)C3CC3)C2C1 CCC(CC(=O)NC(c1ccc(OC)cc1)CNC(C1CNC(=O)C1)=O)SC C(=O)(C(C)(C)CF)N(CC(CN(C(=O)CCc1c[nH]c(=N)[nH]1)C)O)C C(=O)(CC(C)(C)C(C)(F)F)NC1C(C)N(C(=O)COC(F)(F)F)CCC1 N1(C(C=NOC)=O)CC2(C1)SCCC2NC(c1ncc(C)cc1OC)=O Cc1sc(Br)c(C(=O)NC(C)CCCNC(C2(O)CCOC2)=O)c1C N1(CC2N(C(C(C)NC(C3SCCCS3)=O)=O)CCC2)CCCCC1C N1(C(C=Cc2cc(C)on2)=O)CCC(O)C(C(=O)N(C)Cc2cc(C)n(C)n2)C1 N12CC(C3CCCC13)OC2=O.C1(C(=O)OC(CC)(C)C)CCC(CO)CC1 C1(C(N(C(C=C)C2CC2)C)=O)C=CCCN1C(c1cc(=O)cc[nH]1)=O c1(OC)c(C(c2nnnn2C)NC2C3CCC2CC3)cc(Cl)cc1Cl N1(C(c2c(C)ncs2)=O)CCCC1(C)CNC(c1ccc(SC(F)F)cc1)=O C(=O)(CCCCC(N)=O)NCCCC(C)NC(=O)C(C)NC(c1ccoc1)=O N1(C(C(CCCC)F)=O)CC2(C=C(C(=O)NCc3oc(CC)nc3C)CO2)C1 N1(C(C(C(C)C)C2CCC2)=O)CCOCC(C(=O)NC(C(N)=O)C(C)O)C1 N1(C(C(C)OCC#C)=O)CCC(CN(C(=O)C(C)C2CCOC2)CC)C1 C1(CN(C)C(c2cnnn2C2CC2)=O)OCCCC1(C)C Cc1c(C(=O)NCc2nc(CNC(C3(C)CC3C)=O)cs2)cccc1C#N C(=O)(C(C)C(O)C(C)CC)NC(CC=C)CC(=O)N1CCC(CF)CC1 c1(OC(C)C)ccc(N)c(C(=O)N(C(C)CNC(=O)CCN(C)C)C)c1 c1(C(N2C(C(C)C)CN(C(C3CCC4(CC4)C3)=O)CC2)=O)ccn2cnnc2c1 C1(C(F)F)(CN(C(=O)C(C)(C)OCC(F)F)C)CCOCC1 c1(CC)ccccc1C(CNC(=O)Cc1cncs1)NC(=O)C(O)c1ccsc1 Cc1nn(C)c(C)c1OCC(=O)NCC1C=CCN1C(C12CC=CC(C1)OC2)=O N1(C(C(C)C(F)F)=O)CC(NC(c2cc(C3CC3)nc(O)c2)=O)C(C2CC2)C1 N1(C(C2(C=C)CC2)=O)CCCC(C2CN(C(c3cnc(C)cn3)=O)C2)C1 Cc1c(N2CCC(CO)CC2)ncnc1NC1CC1C(O)C(C)C n1(CC(=O)NCC2CCN(C(c3nn(C)nc3Br)=O)C2)cnc([N+](=O)[O-])n1 C=CC(CCC)CC(=O)NCC1(C)CN(C(c2c[nH]nc2CCC)=O)CCO1 CCCCCC=CC=CCC(=O)N1CC(NC(=O)C(C)Cc2cccnc2)C1 N(C(=NCC(C)C)NC1C(C)C1C)CC(CC)(CC)CO C(=O)(CC(C)(C)C#N)NC(C(=O)NCc1cccc(CC)c1)c1ccoc1 C1(NC(C=C(COC)C)=O)CCCCC1CNC(=O)CCC1(C)CC1(F)F c1(C(=O)OCC)ccc(C(=O)CN2CCN(C(=O)Cc3cc(C)no3)CC2)cc1 c1(CC(=O)NC2CN(C(C3(CN(C)C)CC3)=O)CC2C(F)F)cc(O)nnc1O C1(C(=O)NCC(CC(=O)N(C2CCCC2C#N)C)OC)CN2CCN1CC2 C1(NC(c2nnc(O)cc2O)=O)CCN(C(=O)C(F)=CC2CC2)C12CCC2 c1(C(=O)NCCC(CNC(CS(CC)=O)=O)O)nc(-c2ccccc2)ncc1Cl c1(CNC(=O)NCC2C(CC)OCCC2)c(C)nn(C)c1C c1(CCC(CNC(CC)=O)CO)ccc(NC(=O)C(C)CC#N)cc1.S c1(SC)ccc(-c2cccc(F)c2)cc1-c1csc2ncnn12 Cc1cc(C(N2CCCCC2c2cn(-c3cccc(C)n3)nn2)=O)cc(Cl)c1 c1(C(N2CCC(C(=O)NCCCc3n[nH]c(=N)[nH]3)C2)=O)ccn2ccnc2n1 Cn1nnc(C=CC(=O)NCCCNCCCCNC(c2cc(Cl)ns2)=O)n1 c1(N(C(C(CC)n2cncn2)=O)C(C2CCCNC2)C)ncc(C)c(C)n1 c1(CNC(C2CN(C(C34CCCC3OCC4)=O)CCO2)=O)ccc(F)cc1F C(=O)(CC(C)CC(C)C)N1CC(OC)C(NC(c2n[nH]cc2[N+](=O)[O-])=O)C1 c1(CCNC(Cc2cc(C(=O)OC)on2)=O)ccc(OCC(N)=O)cc1 C1(NC(C2C(COC)CCCC2)=O)CCCC1C1CC1.C12(CCCC1)C(=O)N2 C1(NC(C(CC)C)=O)(CO)CCN(C(c2ccnc(-c3ccccc3)n2)=O)CC1 CC(CO)(C(=O)NCC1CCCCO1)NC(C1CC(F)C(=O)N1)=O c1(C(CNC(CC(CC)C)=O)NC(c2[nH]cnc2C)=O)ccc(F)cc1F C1(CC(=O)NCCCN(C(=O)C(C)(O)C2CCOCC2)CC)CCC(O)C1 c1(C(C)C)cc(CC(=O)N(C(C)CCNC(c2ocnc2C2CCC2)=O)C)on1 c1(N2CC(=O)NOCC2)ccc(F)cc1.CCCCC(=O)NCCOC CCCCCC(C)(C)C(=O)N(C)CCN(C(=O)C(C)(O)CCN(C)C)CC N1(C(c2nc(C(C)C)oc2)=O)CCCC2(CNC(=O)CCc3cnccn3)CC12 c1(CC(N2CCC(CN(C)C(c3cc(F)cs3)=O)C2)=O)cnc2cccnn12 N1(C(C2(CC)CC2)=O)CC2CC(C(N3CCN(C)C(C)(C)C3)=O)C(C2)C1 C#CCCC(=O)NC(C)C(c1ccccc1)NC(C1CC(C(F)F)C1)=O C1(C(=O)NC2CC(C(N(CC(=C)C)CC(=C)C)=O)CC2O)Cc2nccn2C1 C#CCCC(O)C(=O)N1CCN(CCCNC(=O)CC(C)NC(=O)C2CC2)CC1 C(=O)(C1=C(C)CCOC1)N1CC(NC(c2ccc(CC)cn2)=O)C(C)(C)C1 C1(CC(N2CCCC(N(C(=O)C(C)(C)c3ncco3)C)C2)=O)CCC(C)(O)CC1 Cc1ccc(C(=O)NC2(C)CCN(C(=O)CC3CCCC(C4CC4)O3)C2)c(O)c1 C12(C(=O)NC(C3CCCN3C(C3CCCCS3)=O)C)CCC(CC1)C2(C)C c1(C(=O)NCC2CCN(C(c3ccon3)=O)C2)ccc(C2=CCOCC2)cc1 C=CCC(CNC(c1nncs1)=O)NC(c1ccn(C2CCC2)n1)=O N1(C(C=C(C)c2cnn(C)c2)=O)CCC2CCN(C(=O)CN(C)C)C2C1 C1(CNC(C(CC)CO)=O)CN(C(C2CN(C(C)=O)C2)=O)CCC1(C)C c1(C(N2C3CN(Cc4cc(OC)c(C#N)cc4)CC32)=O)c[nH]c2ccc([N+](=O)[O-])cc12 c1(C(c2nnnn2C)NC2C(C(C)C)CCC2)cccc2c1COCC2 CC1CCOC1CC(=O)NC(C)(C)CN(C)C(c1cnn(CC(F)F)n1)=O C1(CCC(=O)NCC(CC)(C)O)CCCCN1C(=O)CCc1ccsc1 N1(C(=O)C2CC(=CCCCCCCCO)C2)CCN(Cc2ccccc2F)C2(CC2)C1 Cc1ccccc1C=CC(N1CCC1CNC(c1cnc2n1CCS2)=O)=O C=CC1(C(=O)NC2CCN(C(c3csnc3Cl)=O)CC2F)CCOCC1 c1(C(N2CC3CC(NC(C(C)=C4CCC4)=O)C3C2)=O)cc2c(cn1)CCCC2 c1(NC(C2C(NC(c3cnc(OC)nc3)=O)C2)=O)nccc(Br)c1Cl c1(OC)cc(C(N2CCC(O)(CNC(C3CC(C)(C)C3)=O)CC2)=O)ccc1C C(=O)(CC(C)(C)C(F)F)C(=O)CCC.CC1CN(C(C2CNC2)=O)CCS1 Cc1[nH]c(=N)sc1C(N1CCC(CC(=O)Nc2ccc(C(C)O)cc2)C1)=O Cc1c(F)cc(-c2csc(C(=O)N(C3CCOC3)CCO)n2)cc1F C(=O)(C(CC)C(F)(F)F)NCC(=C)CCNC(=O)C(C)(Cl)Cl c1(C2C(C(N3C(CNC(c4cnn(C)c4N)=O)CCC3)=O)C2)cccc(C#N)c1 c1(C(=O)NCc2nc(=N)[nH][nH]2)n[nH]c2c1CN(C(=O)Cc1ncccc1F)C2 Cn1c(C(=O)NC(C2CCN(c3nnc(C(N)=O)s3)CC2)(C)C)cc(Cl)c1Cl N1(C(c2c(OC)csc2)=O)CC2(CCCC2)C1C(N1CCC(C(C)(C)O)C1)=O C(=O)(CCCCC(=O)N1CCCC1C(C)NC(c1ccncc1F)=O)OC C1(C(C)(C)CNC(c2ccc(CO)o2)=O)CCCCN1C(=O)C=C1CCC1 c1(C(=O)OC)ccnc(Cl)c1NC(C1CN(Cc2cc(C)cc(O)c2)CCS1)=O c1(C(CC)C)ccc(C(=O)NC(C)CNC(=O)C(F)(F)c2nccn2C)c(O)n1 c1(OCC=C)cc(OC)ccc1C(=O)NCCC(C)N(C(=O)CCCCCF)C C12(CNC(=O)C(O)C(F)(F)F)CN(C(c3cncc(O)c3)=O)CC1CCO2 c1(C(N2CCC3CC3C2)C(=O)NCc2ccccc2)sc([N+](=O)[O-])cc1Cl C1(C(=O)NC(C2CCN(c3ccncn3)CC2)C)CCN(C(=O)c2cnsn2)O1 C1(C(N(C(CCNC(C(C)C)=O)C)C)=O)CC2CC(F)(F)CC(C1)C2(F)F N1(C(C(C)N(C)C)=O)CCC(C)(C)C(NC(=O)CC2(n3cccn3)CC2)C1 CC1CN(C(=O)CN(C(C2CC(=O)CC(=O)N2)=O)C2CC2)CC(=O)N1C CCCCC(O)C(C)C(=O)NC(C)CNC(C1(CCN(C)C)CC1)=O CC(C)(C)C(O)CCC(=O)N1CCN(C(c2cc(O)cc(C#N)c2)=O)CC(O)C1 N1(C(c2c(C(C)C)c[nH]c2)=O)C2CCC1CC(C(=O)NCC(C)C#N)C2 C1(C#N)(C(N2CC(CC(C)NC(c3ccn(C)c3)=O)C2)=O)CCCC1 c1(CCC)cc(C(=O)NC(C)(C)CNC(=O)Cc2ccccc2Br)ccn1 c1(NC(C2N(C(CCN(C)CC)=O)CCSC2)=O)cc(OC)c(OC)cc1C C=CCCC(C)(C)C(=O)N1CCN(C(=O)C2=CCCC2C)C(CCO)C1 C1(O)(CN(C(COCC(=O)NC)=O)C)CCN(C(=O)C=CC(=O)N(C)C)CC1 N1(C(=O)Nc2cccc(Cl)c2Cl)CC2CC1(c1cn(CCOC3CC3)nn1)CO2 c1(C(=O)NCC2(F)CC(NC(c3cc(C)ns3)=O)C2)cn(C)nc1C(F)F c1(C(=O)NCCN(C(=O)CC2(C(F)F)CC2)CC)cc(S(N)(=O)=O)ccc1F N1(C(c2cn(C(C)C)nc2)=O)CC(C2CCN(C(C3CCCC(F)C3)=O)CC2)C1 CC(C)(C)CCCCC(=O)N1CC2CC(C(=O)NC(CCO)C(F)(F)F)CC2C1 N1(C(C(c2ccc(F)cc2)(C)F)=O)CCOC(CCNC(c2cnc[nH]2)=O)C1 N1(C(CNC(C2C(C)C2)=O)=O)CCC2(C1)CN(C(c1c[nH]ccc1=N)=O)C2 N1(C(C(C=C)CC)=O)CC2CCCC2(NC(c2[nH]ccc(=O)c2C)=O)C1 C1(NC(C2OCCC(C)(C)C2)=O)CN(C(C2CCC2(F)F)=O)C2(CCCC2)C1 C1(CC(=O)N(CC(C)(C)CNC(C2CCCC2)=O)CC)CCCS(=O)(=O)C1 c1(C(C)OC2CCCCC2C(=O)NC(COCC)CO)cc(C)cc(F)c1 CN1C(=O)Cc2ccc(C(=O)NCC(CNC(C3CC34CCC4)=O)CO)cc21 N1(C(Cc2ccc(NC=O)cc2)=O)CC(C(N2CC(CO)C2)=O)C2(CCC2)C1 C1(NC(C2(CCC)CC2)=O)CCC2CN(C(c3c(C)ccc(F)c3N)=O)CC2C1 CC1CN(C(=O)CCCC(N)=O)C(C)CN1C(c1cc(-c2ccccn2)no1)=O Cc1ncc(C=CC(=O)NCC2CC2NC(C2CCCCN2C(C)C)=O)c(O)n1 C(=O)(CC1=CCCCC1)OC.C(C1C(=O)N1C)N(C)C.C1(=O)C(CN(C)C)N1C CCCCC(F)C(=O)NCC(C)(CO)NC(c1cncc(C2CC2)c1)=O N1(C(c2cncc(OC)c2)C(=O)NC(C)C)CCC2(CNC(=O)O2)C1 S(=O)(=O)(c1ccn(C)n1)N1C2CN(Cc3cccc(C=C)c3)CC1C2 c1(C(N)=O)ccc(C=CC(=O)NCC2(F)CN(C(=O)C(C)C3CCCO3)C2)cc1 C1(CC(N2CCN(C(C#CC(C)C)=O)C(C(C)C)C2)=O)COc2ccccc2O1 c1(SCC(N2CC3C(NC(c4c(CC)occ4)=O)(C3)C2)=O)nnc2ccccn12 c1(NCC(CC)CCO)ccc(S(=O)(=O)N(C)CCc2ccc(Cl)cc2)cc1F c1(C(=O)NCCCC(CCC)NC(C2CCS2(=O)=O)=O)c(F)ccc(F)c1F CCCCCC(C)(CC)C(=O)N1CCC(O)(CNC(=O)CCNC(C)=O)C1 c1(C(N2CCC(O)(CCNC(CC(C)C)=O)CC2)=O)ccn2nccc2n1 N1(C(CCC=C)=O)CCCC2(CCC(NC(c3cncc(C(C)(C)C)c3)=O)C2)C1 C1(CC(=O)NCC2CCN2C(=O)C(O)c2ccco2)CCn2cncc2C1 N1(C(C)C)CC(NC(c2ccc(-n3cc(CC(C)(C)O)nn3)cc2)=O)C(C)C1 C1(NC(C(C(C)C)CCN(C)C)=O)CC2(CCCN(C(C3(C)COC3)=O)C2)C1 c1(C(=O)NCCC(CNC(C=CCOC)=O)O)c(F)cc(F)cc1F C(=O)(CCCCC(C)(C)C)N1CCC(C)C(CNC(C2CC3(CC(=O)N3)C2)=O)C1 Cc1cnc(CC(=O)N(C2CCN(C(=O)CCN(S(C)(=O)=O)C)C2)C)[nH]1 N1(C(CC=C)=O)CC(NC(c2c(C)ccn2C)=O)CC12CCC2 C(=O)(C(F)CCC)NCCCN(C(C1(OCC)CCOC1)=O)CC c1(C(=O)NC(CCCNC(CC=CC)=O)C)cc2ccsc2n1C C1(CN=[N+]=[N-])CCCN1C(=O)CCN(C(=O)Cc1cccs1)C1CC1 c1(N2CCN(C)CC2CNC(c2ccc[n+]([O-])c2)=O)ncnc2c1CCO2 N1(C(C#CC2(C)CC2)=O)C2CCC1CC(NC(c1cc(C(F)(F)F)no1)=O)C2 c1(C(=O)NCC(C(C)(C)C)NC(c2c(C)con2)=O)cc(Cl)c2n[nH]cc2c1 c1(COC(N2C(CN(CC(N)=O)CCOC)C(C)(C)C2)=O)ccc(F)c(F)c1 C(CN(C)C(C1(CCF)CC1)=O)(CO)(CO)NC(CC1(NC(C)=O)CC1)=O C1(C(=O)NCC2=NOC(C)C2)CC(C)(C)CN1C(C1CCCN1C1CC1)=O c1(C(N2C(C)CC(NC(C3CC(C#C)(O)C3)=O)C2)=O)cnc(OC)c(Cl)c1 C1(NC(C(C)(C)C)=O)CN(C(c2cc3ccoc3s2)=O)CC12CC2 N1(C(C)C(=O)N(CCCCNC(=O)C(C)N(CC(F)(F)F)C)C)CCOC1=O CC1CN(C(c2ccc(CNC(c3cccs3)=O)s2)=O)CC(C)(C)C1 C1(NC(CCCN(C(C)C)C(c2ccnn2C(F)F)=O)=O)CCCC1C#N CCC(CC)(CC)C(=O)N1CC(C(N2CCC(C)(COC)C2)=O)CCC1(C)C C1(CC)(NC(=O)C(O)CC(C)C)CCCN(C(=O)C=Cc2ccc(C(F)F)o2)C1 N1(C(c2c(SC)cccc2)=O)CC(NC(c2nn(C)cc2SC)=O)CCC1C C(=O)(CCCCC1CC1)NCC(CNC(=O)C1=CCC1)OC C1(NC(c2scc(C)c2C)=O)CN(C(C2CC2Sc2ccccc2)=O)CC2(CC2)C1 Cc1cn2cc(C(=O)N(C(C)CNC(c3cc[nH]c3C3CC3)=O)C)sc2n1 CN1CCCCC1CCC(=O)NCC(C)(C)NC(=O)Cc1ccsn1 C=C1CC2CCCC(C1)N2C(C1C2CC1N(C(c1ncncc1OC)=O)C2)=O CC1COCC(C(=O)NC2CCC2CNC(c2cn(C)nn2)=O)O1 Cc1ccc(C(C)C)cc1C(=O)NCCCNC(C1CC(C)CCO1)=O c1(NS(=O)(=O)CCCCl)cccc2c1CN(Cc1ccncc1)C2 C(CCC(O)C(=O)NCC1(C)CCCCO1)NC(c1c(CC)n(C)cc1)=O C1(CNC(c2cc(C)on2)=O)CCC2CN(C(=O)C(C)C(C)O)CC12 c1(C(=O)NCC2C(NC(c3c(C(C)(C)C)n[nH]c3)=O)CC2)nc(Cl)c(Cl)s1 N1(NC(=O)C(c2ccco2)N2CCC2C2CCOCC2)CCOCC1 N1(C(CC(=O)NCC#C)=O)CCCC(C)C1CNC(=O)COCc1cc(C)on1 C1(NC(CCN2CCC(CN(C)Cc3ccccc3)CC2)=O)CCCCC1(C)C N1(C(COCCC#C)=O)CCN(C)CC1CNC(=O)CN(c1ccccc1)C c1(C(N(C2CN(C(C(CC=C)CC(C)C)=O)C2)C)=O)ccc2c(=N)[nH]cnc2c1 CN1CC=C(CCNC(=O)CCOCCNC(C2CC2Cl)=O)CC1 N1(CC(=O)NC(C2N(C(Cc3c(C)scc3)=O)CCC2)C)CCS(=O)CC1 O=C(CN=c1cc[nH]cc1)NC1CCCCCN(C(C2CC3(CCC3)C2)=O)C1 C(C(C(=O)N1CCC(CNC(c2ccc(OC)s2)=O)CC1C)C(F)(F)F)OC c1(C(N(CCCNC(C(C)=C(C)C)=O)C)=O)ccc(C(F)F)nc1O c1(C(N2CCN(C(C34COCC3C4(F)F)=O)CC2)=O)cncc2[nH]ccc12 c1(C(N2CCCC(N(C(C3CC3CC(C)C)=O)CC)C2)=O)nccc(N)c1Cl N1(C(C(CC)n2cccn2)=O)CCc2[nH]nc(I)c2C1 C(=O)(C(CC(C)C)NC=O)N(CCOCC(=O)NC(CSC)(C)C)C c1(C(N2C(CNC(C(CSC)O)=O)CC(F)C2)=O)cn(C2CC2)c(C)cc1=O N1(C(CCCN=[N+]=[N-])=O)CCn2c(CNC(C3CCCS(=O)(=O)C3)=O)nnc2C1 CC(O)CCCc1cn(CC2C=CCN2C(C2CC2c2ccc(Br)s2)=O)nn1 CC1CCN(C(C2(Cc3ccccc3)CC2)=O)CCN1C(=O)CC1(C#N)CCC1 Cc1cc(O)ncc1C(=O)N(C(C)C(=O)NCC1(C)CCCC1O)C C#CC(CC(C)(C)C)NC(=O)CC1CCN(C(C2CCCCCN2C)=O)C1(C)C c1(C(=O)NCC2(C)CCCN(C(COC(C)=O)=O)C2)cn2ccncc2n1 C1(C(=O)NCc2c[nH]ccc2=O)CC(F)(F)CN1C(c1ccc(F)c(F)c1)=O c1(N(C)CC2N(C(C3=CC(C)(CC)C3)=O)CCC2)nc2ccc(F)cc2s1 C1(C(N2CCC(COC)C2)=O)CSCCN1S(=O)(=O)C1(c2ccccc2)CC1 c1(NC(C(=O)NCC(CNC(CCC=CC(C)C)=O)(C)C)=O)ccc(C)c(C)c1 C1(CNC(Cc2c(C)non2)=O)CCN(C(=O)CCOCCN(C)C)CC1(F)F CCC1=C(C(=O)NC(C)CNC(=O)Cc2cccc(C(N)=O)c2)SCCO1 c1(OC)ccc(CNC(=O)C(c2ccc(C(F)F)nc2)N2CCOCC2C)cc1 C1(O)(CNC(c2nc(C)[nH]n2)=O)CCN(C(c2nocc2Cl)=O)CC1 N1(CC=C)CCCN(C(=O)C(C2CCC2)NC(C2CC2C(C)(C)C)=O)CC1 CCC(CCC(=O)N1CC(=O)NC(C(C)C)C1)NC(=O)C(C)CSC C(c1ccc(Cl)nc1)=CC(=O)NCC=CCNC(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O N1(C(CC2OCCN(C(C=CCN(C)CC)=O)C2)=O)CC2(C1)CC(C)(O)C2 c1(C(=O)NCC(CN(C(COCC(=O)OC)=O)C)(C)C)ccc2c(c1)CCC=C2 C(=O)(CS(=O)(=O)C1CC1)NC1CCN(C(c2nc(C)nc(O)c2)=O)C(C)C1 CCC(C)C(C(=O)N(CC(c1nn[nH]n1)C)C)NC(=O)C(CN(C)C)CC C(=O)(C1=C(C)S(=O)(=O)CC1)N1C([SH]=C)CN(C(c2nnc(S(C)(=O)=O)s2)C2CC2)CC1 N1(C(CC(C)c2ccccc2)=O)CCOCC(NC(=O)CC2(C)CCCC2)C1 c1(C(=O)NCC2CCN(C(c3c(C)cc(C(F)(F)F)s3)=O)C2)cccn(C)c1=O C1(NC(C2CCCN(C(=O)OC)C2)=O)CC2CCC(C1)N2C(=O)C1CC1 c1(CN(CC(=O)NCC)CC(=O)NC)ccncc1 C1(CNC(CN(CC)CC)=O)CCCC1NC(C1CCCN1)=O c1(CC)cc(CNC(=O)C=CC(C)NC(=O)C(C)NC(N)=O)no1 N(C1CCCn2nccc21)C(C(CC(C)C)ONC(c1nc[nH]n1)=O)=O C#CCC(O)C(=O)N(C)CC1(O)CN(C(c2ccc(C(=O)N(C)C)cc2)=O)C1 n1(CC)c(=O)c(=O)[nH]c2cc(C(=O)NCc3cc(F)ncc3Br)ccc12 N1(C(C(CC)CO)=O)CCN(C(c2nnn(CC3CCCC3)c2C)=O)CC1C C1(C(F)(F)F)(C(N2CC(NC(C3(SC)CC3)=O)C(C)C2)=O)CC2C=CC1CC2 C1(C)(CC(=O)N(C(C(C)C)CO)C)CCN(C(=O)Cc2ccc(O)nc2)C1 C=CC1(CC(N2CCSCC2CO)=O)CN(C(c2ccc(OC)o2)=O)C1 c1(C(C(=O)NC(CN(C(CCCOCC=C)=O)C)C)C)c(C)nn(C)c1C CCC(CC(=O)N(C1CCN(C(c2sc(C)cc2C)=O)C1)C)SC c1(CN2C(C(=O)Nc3cc(F)cnc3Br)CCC2)ccc(O)c2ncccc12 Cc1ccc2c(c1)CC(C(=O)N(C(C)CNC(=O)CCc1cccc(F)c1)C)S2 C=C(C)CCC(=O)N1CCC(NC(c2ccnc(OCCO)c2)=O)C1 C(=O)(C1=CCSC1)NCCC1N(C(CNC(C2CCS(=O)(=O)C2)=O)=O)CCC1 CCCCCCC(C)(C)C(=O)N(C)CC1CC(F)CN1C(C1CC1(C)C)=O C1(N(C(c2ccc(O)cc2)=O)CC)N(C(=O)C(C)N=[N+]=[N-])CCCC1(C)C CCCCCC(=O)NCCCCCn1cc(CCC2CC(OC)C(OC)C2)nn1 C=C1CCC(C(=O)NC2CCOC2C(=O)NC2CCN(C(C)C)C2=O)CC1 c1(CN(C)Cc2cccc(-c3nn[nH]n3)c2)ccc(F)cc1C(=O)O CC1(C)CCCC(CC(=O)NCCC2(O)CCN(C(=O)CSc3nccs3)C2)C1 n1(CC(=O)NC2CCC(NC(C3(SC)CCC3)=O)CC2)cnc([N+](=O)[O-])n1 C(=O)(C1=CNC2=NCCC2=C1)NC1CC(CCNC(=O)CN2CCCCC2=O)C1 C1(CNC(c2c(OC)nn(C)c2)=O)CN(C(=O)C=C2CCN(C)CC2)CCCO1 c1(OC)cc(OC)c(C(=O)CN2CC(S(N)(=O)=O)C2)cc1-c1c(C)cc(C)cc1C C1(=O)C2=CCC(C2)N1.C(CCCN(C)C(C1(c2ccc[nH]2)CC1)=O)N(CC)CC C=CC(C)(O)CC(=O)N1CCCCCC1C(=O)NCc1nccc(OC)n1 C(C)(C(=O)NOCC(N1CCCC1)=O)Cc1ccc(C(C)=O)o1 Cc1oc(CO)cc1C(N1CCC(N(C(=O)CC2(O)CCOC2)CC2CC2)C1)=O c1(C(N2CCCC(CNC(C3(C)C=CCCC3)=O)C2)=O)ccc2cc[nH]c2n1 N1(C(=O)Cc2csc(Cl)n2)CC2OCCN(C(c3ccc4c(c3)NCC4)=O)C2C1 C1(=O)CCC(=O)N2CCCC2CC1.n1(CCC)cc(CCCCCO)nn1 C1(CN(C(=O)C(c2ccc(Cl)cc2)O)C)COCCN1C(C1COC1)=O O(NC(=O)CC1C(C(=O)NC2(CNC(C3(C(C)=O)CC3)=O)CC2)C1)CC C1(NC(=O)NC2CC3COC2C3)CCS(=O)(=O)C2(CCOCC2)C1 C1(OCC)CCCC1N=c1[nH]c(=NC(C)c2ccc(Cl)cc2C)c2sccc2[nH]1 n1(CC)ncc2c(N3CCC(F)(C(=O)Nc4cc(Cl)c(F)cc4C)C3)ncnc12 CC(C1OCCc2ccccc21)N(C)C(C1COCCOC1)=O N1(C(c2ccnn2C2CC2)=O)CC2CCN(C(c3cccnn3)=O)CC2C1 c1(CC)noc(C(N2CCCCC2CN(C(=O)C(C)N(C)C(=O)OC)C)=O)c1C N1(C(c2c[nH]c(=NCC)s2)=O)CC=C(CCNC(C2CC(=O)N(C)C2)=O)CC1 Cc1ccc(-n2cc(NS(=O)(=O)CC3CCC(C)C3)cn2)cc1Cl C(C(C)(C)CC(=O)NCCC1(O)CN(C(=O)CNC(=O)CNC(C)=O)C1)OC c1(CNc2cn(C3CN(Cc4nc(C(C)C)sc4)C3)nc2)ccc(C#N)cc1 N1(C(CCC#N)=O)CC2(CCC2)CC1CNC(c1ccc(C2CCC2)cc1)=O C1(CC(=O)NCC(C)CN(C(=O)C(O)C2CCC2)C)(CC=C)CCCC1 N1(C(CC(C=C)CC)=O)CC(C)CN(C(=O)CCc2ccc(C)o2)C(C)C1 c1(C(C(=O)NC2C(C)N(C(C3CC4C=CC3O4)=O)CC2)(F)F)cccc(F)c1Cl c1(OC)cc(CC2C(C(=O)Nn3cc(-c4cnccc4C)nn3)CCC2)ccn1 C(=O)(C1CCCn2cnnc21)N1CC2C(NC(=O)Cn3cccn3)(CC2)C1 Cn1cc(C(=O)NC2CCCC2NC(c2cn(C(C)(C)C)cn2)=O)nn1 C1(NC(C(COC)O)=O)CCN(C(c2ccc(-c3nnc(C)o3)cc2)=O)C(C)C1 CC(C)C(C(F)(F)F)OC(c1ccccc1Oc1cccc(C(F)(F)F)c1)=O c1(C(N2C(CN(C)C(c3cc(O)nc(O)n3)=O)CCC2)=O)cc(Cl)c(F)cc1F n1(CCOC)nc(-c2ccc(NCC(C)(C)C)nc2)nc1C1CN(C(C)C)C1 C(C(C)(O)C(=O)N1CC=CC(C(=O)NCC(F)(F)C(F)F)C1)OC CC1(C)CC(CC(=O)NCCN2CCC(NC(=O)CCOC3CC3)CC2)CO1 C1(NC(CC2N(CC)C(=O)CC2)=O)CCCCCC1NC(=O)C(C)(C)C1CC1 c1(C(N2C(COC)CN(C(C3CCSC3)=O)CC2)=O)cc(F)cc2cccnc12 CCC(C)C(C(=O)NCC1(C(=O)Nc2cc(C)sc2C)CC2(CC2)C1)N(C)C C1(OC(C)=O)CCN(C(c2[nH]ccc2CNC(c2cn[nH]c2)=O)=O)C1 Cn1ncc2c1CC(Nc1cnc(O)nc1O)C(c1nc(CC3CC3)no1)CC2 C(CC(C(C)(C)C)NC(c1ccnn1C=O)=O)N(C(CSCC=C)=O)C c1(CC)cc(CC(=O)NC(C)CNC(=O)CC(c2c(C)noc2C)C)n(C)n1 c1(CC(=O)NC2(CCNC(=O)C=CC3CCCCC3)CC2)ccc2nc[nH]c2c1 c1(C(N2CC(NC(C3CC(C)(O)C3)=O)CC2(C)C)=O)cccc2nc(Cl)cn12 CCCC(CC(C)C)C(=O)N1CCCC(CC(=O)NCCN2CCC2)CC1 C(CCC(=O)NCC1C=CCN1C(c1c[nH]c(=N)o1)=O)N(C)C c1(C(C)C)cc(NCc2noc(CCC(=O)NCCN3CCCCC3)n2)ncn1 CC1C(CO)CCCN1C(c1ccc(C(F)F)c(F)c1)C(=O)NCCCSC N1(C(CCC(=O)N(C)C)=O)CCCCC(C2CN(C(=O)CC3CCCCO3)C2)C1 CC1CCN(C(C2CCCCN(C)C2=O)=O)CCN1C(c1cc(O)nc(Cl)c1)=O C1(C(=O)NC2CCCC2NC(=O)C=Cc2cncs2)(COC)CC1(F)F N1(C(c2ccc(C)c(C)n2)=O)CCOC2CCN(C(C3CCN(C)C3=O)=O)CC12 C(=O)(C(F)C(CC)CC)N1C(C)CCC(CNC(C2(CC#C)CCOC2)=O)C1 C1(C(=O)NC(C(=O)OCC)COC(C)C)CC(N)CC(C)(C)O1 N1(C(C(=O)NC(c2ccon2)C)=O)CCNCC1CNC(c1ccccc1Cl)=O Oc1nc2ccc(F)cc2cc1CN=c1cc[nH]c(N2CCNCC2)n1 C1(CC(=O)NCCc2n(C)ncn2)CC(NC(c2cccc[n+]2[O-])=O)C1(C)C O=C(CCC(F)F)NCCN(C(c1cnc(N2CCOCC2)s1)=O)C1CC1 N1(CCC)CCC(NC(c2ncoc2CNC(=O)CCc2ccnn2C)=O)C1 C#Cc1cnn(C)c1C(=O)NC1CCC(C)N(C(=O)Cc2cccnc2)C1 CCCCC(O)C(=O)N1CCC(N(C(=O)C(C2CC2)C2CC2)C)CC1 Cc1cc(C(=O)NCCC2(C)CCN(C(C3(C)CC3C)=O)C2)c(C)n1C CCCCCCCCCCCC(O)C(=O)N(CCC(=O)O)CCO c1(CN(C(c2c(O)ccc(C(N)=O)c2)=O)C2CC2)ccc(F)c(F)c1F c1(C(=O)NCC(C)(CO)NC(Cn2nc(C)oc2=O)=O)cc2c(Cl)cccn2n1 CC1CC(CNC(c2ccc(Cl)nc2N)=O)CCN1C(=O)C=Cc1ccco1 CC1CC2CN(C(=O)CC3CCCNC(=O)C3)CC2N1C(c1ccc(Cl)o1)=O C1(N(C(c2c(C)cc(CNC(=O)CC3CCOC3C)o2)=O)CC)CCOC(C)(C)C1 C1(COc2ccc(NC(=O)NCC3CC(C)C3)cn2)(OC(C)(C)C)CCCCC1 CC1(C)CCN(C(C2CCC3(CCC3)CO2)=O)CC1CNC(C1CC(O)C1)=O C12(C(=O)NCC3C(NC(C4(c5cccs5)C(C)C4)=O)CCC3)CC(C)(CCO1)C2 N1(C(CC(CCC)O)=O)CCC2(CCN(C(=O)CC(C)(F)F)C2)C1 C1(C(N(C)CC2(O)CN(C(C3N(CCC)CCC3)=O)C2)=O)(N(C)C)CCCOC1 c1(OCC)ccc(Br)c(C(=O)NCCOCCNC(C2CCC(F)C2)=O)c1 c1(CC(=O)NCC(CCOC)NC(=O)C(C(C)(C)C)OC)c(C)ncnc1C c1(CC)noc(C)c1CNC(c1sccc1CNC(C1COCC1(C)C)=O)=O C1(COC(C)C)CN(C(=O)CN2CCOCC2=O)CCO1 C=C1CCC(C(=O)NCCC(C)N(C(=O)CCCSC(C)(C)C)C)CC1 c1(CC)nncn1CCNC(=O)C(C1(O)CCC1)NC(=O)CN1CCSCC1 c1(-c2nc(-c3cccc(O)c3F)n(C3CCC3)n2)n[nH]c2c1CCCC2 N1(C(c2n(CCC)ncc2)=O)CCCN(C(=O)COCC2CCCC2)CC1C O=C(C1CCCn2cnnc21)NC1(CNC(C23CCCCC2C3(F)F)=O)CC1 C1(C(=O)NC2(CF)CN(C(c3cc[nH]n3)=O)C2)CC2CCC(C1)C2 C1(C(N(C(C)CNC(c2ccc(C(C)C)s2)=O)CC)=O)CCCCCS1(=O)=O N1(C(c2cc(C(=O)OCC)c(C)[nH]2)=O)CCN(C(c2nccn2C)=O)CC(O)C1 c1(OC)nc(Cl)c(C(=O)NCC2CCC2NC(=O)Cc2cccc(OC)c2)s1 c1(C(=O)NCC2(CNC(CC(C=C)CC)=O)CCC2)ccc2c(c1)CCC(C)N2 C1(NC(=O)CCc2cscn2)CN(C(=O)CSCC(F)F)CC12CC2 c1(C(=O)NCC2CC(NC(CCc3onc(C)n3)=O)C2)ccnnc1O c1(CN2CCC(O)(C(=O)NC(c3cccnc3)CC)C2)cc(Cl)cnc1Br N1(C(c2nccnc2C)C(=O)NCCOCC)CC(=O)N(C)CC1CC C1(CNC(C23CC(C)C2C3)=O)CCCC(NC(=O)Cc2ccon2)C1 C(CN=C(NCc1ccc(F)cc1)N1CCC(O)C1)c1nc2scc(C)n2c1 c1(C(N2CCC(CC=C)(NC(=O)C3=CCCO3)CC2)=O)cccc2c1COCC2 C=CCCCCCCCCC(=O)NC(C1CCCN1C(C1(F)CCCC1)=O)C CCC(O)(CC)CCNC(=O)C(C1CC=CCC1)NC(c1csc(C)c1)=O C1(NC(c2sc(CC)c(C)c2)=O)CC2(CCN(C(C3CCC(=O)N3C)=O)C2)C1 Cc1cc(Br)ccc1NC(N1CCN(C(=O)OCCCOC(C)(C)C)CC1)=O c1(-n2c(CC=C)nc(CC(C)OC)n2)cccc2ncccc12 Cc1ccc(-n2nc(-c3ccnn3C)nc2CC2CCCC(O)C2)cc1 Cc1cc(=NC(C)CN2CCCCC2=O)[nH]c(=NCC2(C)CCCC(=O)N2)[nH]1 C(=O)(C(CS(C)(=O)=O)NC(C1CCCCNC1=O)=O)OC c1(CC)ccc(CCCC(N2CCC(NC(=O)C(O)COC(C)=O)CC2)=O)cc1 N1(C(C(=O)Nc2cccc(C(=O)OCC)c2)=O)CC2(CC=CC(C(=O)OC)=N2)C1 c1(C(F)(F)F)cc(C(F)(F)F)cnc1O.C1(N)CCN(c2ccccc2Cl)CC1 N1(C(C(C)CO)=O)CCN(C(=O)C(F)(F)CN2CCCC2)CC(C)(C)C1 c1(C(=O)NCC(CC)NC(=O)CC(F)(F)F)cnc(C2CC2)cc1C C1(C)(C(=O)NCCCCNC(C(=Cc2cccs2)C)=O)CCOCC1 n1(CC)cc(Cl)c(C(=O)NCCC2(NC(C3CC=CCO3)=O)CCC2)n1 c1(C(C(N2CC(NC(C(C)(C3(C)CC3)OC)=O)C2)=O)C)cccc(O)c1 C1(C(N2CC3CN(C(C(C)=CC4CC4)=O)C3CC2)=O)Cc2cc(Cl)ccc2O1 c1(C(=O)NC(C2CCCN2C(c2nnsc2N)=O)C)ccc(C2CC2)cc1 Cc1c(CCC(=O)NC2CC2C)cnn1C.C12(CC1)C(C)NC2=O.CCN(C)C N1(C(c2ncc(N)nc2)=O)CC(NC(c2ccn3c2CCCC3)=O)C(C2CC2)C1 c1(C(=O)NC2CN(C(C3C(C=C)C3)=O)CC2C)ccc(Br)c(C)c1 C(CC(CC)C(=O)N1CCC(C)(NC(c2cnc(C)o2)=O)C1)=CC c1(C(=O)N(C2C=CC(C(NOC)=O)C2)CC2CC2)cccc(F)c1O c1(C(=O)NC(C)CCCNC(=O)C(C)(C)OCC(F)(F)F)cnn(C)c1N C1(C(NOCC(C(C)C)O)=O)CCN(C(c2ccncc2Cl)=O)CCO1 C1(C(N(CC(C)NC(C2(O)CCC2)=O)CC)=O)CCn2ccnc2C1 C1(CN(CCC=O)CC)CC(C(=O)N(CCCNCC)CCO)CC(=O)N1.CCO c1(C(=O)NC2CCC(N(C(CCC#CC)=O)C)CC2)ccc(=NCCOC)[nH]c1 C1(NC(=O)CCCCN2CCCC2)CN(C(C23CCC2C3)=O)CCC12CCC2 CC1CCCCC1C(=O)NCC1(CNC(=O)CCC#N)CC=CC1 N1(C(=O)CC2CCCC23CC3)CCCC2CN(c3nc(C4CC4)ns3)CC12 N(C1CC2(CCC2)Oc2ccc(F)cc21)S(=O)(=O)CCc1ccccn1 C12(C(N3CCC(CNC(C=CCC)=O)C34CC4)=O)CC3CC(C1)CC(F)(C3)C2 CC(CCC(C)(C)C)C(=O)NCC1C(CNC(C2CC3(CCO2)CC3)=O)C1(F)F N1(C(C2C(C)(CC)C2)=O)CCC(NC(c2cnc(C3CCC3)cc2C)=O)C(F)C1 c1(NC(C(=O)OC)(C)c2ccccc2)ccc2oc(Cl)cc2c1 CC1(C)CCN(C(=O)CC2CC(F)(F)C2)C1C(=O)NCc1ncccc1O c1(C(=O)NCCC(C)NC(c2cscc2Cl)=O)ccc(-c2cnn(C)c2)cc1 C1(CNC(c2cc(C)oc2)=O)CCN(C(c2cc(C3CC3)on2)=O)CC1(F)F c1(C=O)c(OC(F)F)cccc1Cl.C(=O)(C(C)(C)C)NCCCN(CC)CC CC1(C)C2CN(Cc3cc(Cl)cc(Br)c3F)C(C(N3CCC(O)C(F)C3)=O)C12 C(=O)(C(F)C(C)C(F)(F)F)N1CCC(C)N(C(=O)Cn2cc(C3CC3)nn2)CC1 c1(C(C)(C)NC(=O)CCCc2ccncc2)cc(F)c(Br)c(F)c1 S(=O)(=O)(c1nnn(C)n1)NC(C(c1ccc(Cl)cc1)OC)=O C1(NC(c2nccc(N)c2Cl)=O)CN(C(=O)COC2CCOCC2)C2(CCC2)C1 C1(C(=O)NCC(C(=O)NCC2OCCN(CC)C2)C)CC(=O)NC(=O)C1 c1(N2CCC(NC(CC(C)(O)C(F)(F)F)=O)C(F)C2)ccc2c(n1)CCCC2=O C1(CNC(C2CCS2(=O)=O)=O)CN(C(=O)Cc2occc2CN(C)C)CC12CC2 C1(CCCC)CN(C(=O)C(CCC)OC)CCN1C(=O)C1=CSCCO1 c1(CC)ncc(C(=O)NCC#CCNC(=O)Cc2nc(C)sc2Cl)c(C)n1 C1(C(=O)NC2C(NC(c3cccnc3SC(F)F)=O)COC2)CC(C2CCC2)C1 c1(COC)ccncc1C(F)(F)F.C12(C(F)(F)F)CN(C1)c1nnc(o1)C2 c1(C(N2CCC(C)C(NC(c3csc(S)n3)=O)C2)=O)cc2n(n1)CCCCO2 C(=O)(C1OCCc2cc(O)ccc21)NC1(CNC(C(C)C(C)(F)F)=O)CC1 C=C1CC(C(=O)NCCCNCC2CC2C(=O)OC(C)C)(COC)C1 C(CC(C(=O)NCC1CC(C)(O)C1)NC(=O)CC1CCN(C)C1=O)OC c1(OC(CC)C)cc(-c2cn(C3CC(C(=O)N(C)C4CC4)C3)nn2)ccn1 c1(NC(C)=O)cccc(C(=O)NC(C)CC(C)NC(=O)C(C(C)O)N(C)C)n1 Cn1cncc1C=CC(=O)NC1CCN(C(=O)C=Cc2ccc(Br)s2)C1 CC(C)C(C(C)NC(=O)Cn1cnnn1)NC(c1cc(C#N)no1)=O C1(C(N2CCCC(CO)(NC(C3CC4CC4C3)=O)C2)=O)(OC)CCS(=O)(=O)C1 c1(N2CCC(CSC)CC2)nc(NCC(C2CCCCC2)C)c2ncn(C)c2n1 C(=O)(C(O)CC[S+](C)C)NCC(C1N(C(CCN(CCC)C)=O)CCC1)(C)C N1(C(C2C(C)(C)C2)=O)CCC(NC(c2c[nH]ccc2=N)=O)C2(CCC2)C1 N1(CC(=O)NC(C)C(N2CC(CO)(CO)C2)=O)CCOCC1 N1(C(c2c(C)[nH]cc2)=O)CC2OCCN(C(=O)CC3CC3(Cl)Cl)C2C1 CC(C)(C#N)CCC(=O)N1CCC2(CC1)CC2CNC(=O)Cc1ccsc1 C12(C(N3C(C)C(O)CC3)=O)CCCC1CCN2C(=O)C(Cl)Cl N1(C(C(C2CCCC2)OC)=O)CC2CC(NC(=O)CC3CCOC3(C)C)C(C2)C1 O=C(CCCc1cncs1)NCCN(C1CC1)CCO.C1(C=O)CC(CF)C1 CCCCCCC(C(=O)N(CC(C)NC(=O)C=Cc1ncco1)C)NC(C)=O C1(C2CCCCC2)(NC(C2N(C(CC3OCC(C)(C)C3)=O)CC=C2)=O)CC1 CCC(C)CCCC(=O)NC1(COCC)CN(C(c2ccnc(C)c2)=O)C1 C(CC(C)C)(C(=O)N1CC2CC2(CNC(c2cc(C)ccc2C)=O)C1)NC(C)=O c1(-c2ccc(CN(c3cccc(C#N)c3)CC)s2)cc(F)cc(N)c1N c1(C(C(=O)NCC2CCN2C(c2nocc2Br)=O)OC)ccc(F)cc1 c1(CC)ncnc(NC(=O)C(=O)NC2(c3ccc(Br)cc3)CC2(C)C)c1F C(=O)(C(CC(C)C)n1cc(C(C)(O)COC)nn1)NCCC(CC)CN(C)C C#Cc1cnc(C(=O)NCC2CCCC2NC(C2NC(=O)OC2C)=O)c(C)c1 CCC(C(=O)OC)C(=O)NCCOc1ccc(Cl)cc1C N1(C(C2(CC)CCCO2)=O)CCN(C(=O)CCCOC(C)C)C(c2ncc[nH]2)C1 C(=O)(CCCCCCNC(=O)C(C(C)C)SC)NCC(CC#C)(C)CO C1(NC(Cc2cccc(OC(C)C)c2)=O)CC(F)CN(C(=O)C(F)=C2CCC2)C1 c1(C(N(C)CC2CCCN2C(c2ccc(F)s2)=O)=O)csc([N+](=O)[O-])c1 N1(C(C2(OC)CCCC2)=O)CC(CCNC(c2ccc(Br)cc2)=O)C(C)C1 C(=O)(C(O)CCC(C)C)NCCCCC(N1CCCC(CCC)CC1)=O C(=O)(CC(O)CC(C)(C)C)NCC1(COC)CN(C(c2cc(C)ncc2C)=O)C1 c1(C(C)C(=O)NC2CCC2CNC(=O)COCc2nc[nH]n2)c(F)cccc1F C1(CC(=O)OCC)NC(=O)N(C(c2ccc(OC)cc2)C(C)(C)C)C1=O n1(CC(N2CC3C(CNC(C(C)O)=O)(CC3)C2)=O)ccc2ccc(F)cc12 C1(c2cn(CCCC)nn2)(N(C)C)CCCN(C(c2cnc(OC)nc2F)=O)C1 C1(NC(CCCCC)=O)CCN(C(c2cc(C(N)=O)n(C)n2)=O)CC1C(C)C c1(CS(=O)(=O)NCc2n(C)nnc2)ccc(F)nc1 Cc1cnc(Cl)[nH]c1=NCC(C1CCCCC1)NC(C1CCN(C)S1(=O)=O)=O C1(C(N(CC(C)NC(c2cnsc2)=O)CC)=O)CN2CCC1CC2 C1(C(C)CNC(=O)OCc2ccccc2)CCN(C(C2(N(C)C)CCCC2)=O)CC1 C1(NC(C2(SCC)CC2)=O)CCN(C(=O)Cn2ccnn2)C(C)C1 O=C(CS(=O)(=O)NC(c1c[nH]nc1-n1cnnn1)=O)NC(C1CCCO1)CO C1(C(=O)NC(C2CCN2C(C2CN(CC(F)(F)F)C2)=O)C)CCOC(C)(C)C1 c1(C(=O)NC(CC=C)CNC(C2CN(C3CCOC3)C2)=O)cc(C)c(Cl)cc1F CCC(CC)C(C(=O)N1CCC2CN(C(=O)C=Cc3ccc(O)cc3)C2C1)OC Cc1ccc(C)n1CC(=O)NC(CCC1CC1)C(=O)N1CCCC(C(N)=O)C1 c1(C(C(=O)OC)N(C2CCC2)CCOC)ccc(-c2ccco2)cc1 C1(NC(c2sccc2C2CC2)=O)CCN(C(=O)CSCc2ccc(F)cc2)CC1 c1(OC(C)C(=O)NCCc2ccccc2)ccc(Br)cn1 C1(COC)CCCCN(C(=O)CCCn2ccnc2)C1.c12csc(n1)CNC2 C1(CNC(CC=C=C)=O)CCN(C(c2cnnn2-c2ccccc2Cl)=O)C1(C)C C1(CC(=O)N(CC(=O)N(C(C#C)C2CCC2)C)CCC)CCSCC1 c1(C(N(CCC2N(C(C(CCC)C)=O)CCCC2)C)=O)cc(OC)nc(OC)c1 CC1=C(C(=O)N2CC(NC(C3CC34CCCC4)=O)C(CC(C)(C)C)C2)CCO1 C(=O)(C1=C(Cl)CCOC1)NCCCCCCN(C(C1C2(CC(OCC)C2)C1)=O)C C1(NC(=O)CSc2ncc[nH]2)CN(C(=O)CCSCC2CC2)CC1O c1(CC)cccc(C(=O)NC(CNC(c2ccco2)=O)C2CC2)n1 n1(CCC(=O)N(C(CNC(C2C(C#C)C2(C)C)=O)C)CC)cnc(C)cc1=O c1(C(=O)NC(C(=O)NC(C=C)(C)C)Cn2cccn2)ccc(F)c(O)c1 c1(C(=O)NCCCN(C)C(C2CCCC23CC3)=O)cc(=O)cc[nH]1 C1(C(N2CC(C(C)NC(C#CC(C)C)=O)C2)=O)CCCC2CCCCC12 N1(c2ccc(C(CC)=O)cc2)C(=O)NC(C)(CCc2noc(CSC)n2)C1=O Cc1ccc(C(CNC(=O)Cn2cnnc2)NC(C2CCC(F)(F)C2)=O)cc1 N1(C(c2c(OC)nn(C)c2)=O)C2CCCC1CC(NC(c1ccc(C)nc1)=O)C2 C1(C)(NC(c2n(CC)cc(Br)c2)=O)CCCN(C(C2COC(=O)C2)=O)C1 c1(C(=O)NC2(CNC(C3CCCN(CC)C3)=O)CC2)cc(C)c(C)nc1O C1(C(=O)NCC(C)CNC(c2c(C(F)(F)F)ncn2O)=O)CN2CCN1C(C)C2 c1(CC(=O)NCC2(CC(=O)NC(CCOC)C)CC2)cncn1C CCCCC(C(=O)NCC(C1CC1)N(C(=O)Cn1nc(C)cc1C)C)C(C)C N1(C(C=CCC)=O)CCN(C(=O)C(CC)N(CC)CC)CC1CC=CC C1(CC)C(=O)NCCN1C(=O)C(N1CCOC(c2cc(C)ccc2C)C1)=O N1(C(CC2(OCC)CCC2)=O)CCOCC1CCNC(=O)CN1CCCNC1=O c1(SC)nc(C(=O)NCC2CC2NC(c2ncccc2SC)=O)c2ccccn12 C(=O)(CC(C)(C)CC)NCC(c1ccc(F)cc1F)NC(C=CCC)=O c1(C(=O)OC)cc(C(=O)NCC#CCNC(C2(Cc3ccccc3)CC2)=O)[nH]n1 C1(NC(C(C)C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)C12CC2 Cc1[nH]nc(C(=O)NCCC2CCCN2C(=O)Cc2ccsc2Cl)c1Cl c1(C(=O)NC2CCC(F)(CNC(=O)C(O)c3ccsc3)C2)csc2nnsc12 C1(C(N2C(C(C)NC(c3ccnn3C3CC3)=O)CCC2)=O)CC(=O)NC(C)C1 CC(C)CC(C)(C)C(=O)N1CCC(CCNC(c2nc(=N)cc[nH]2)=O)C1 C1(C(=O)NC(C2CCCN2C(=O)Cc2cnnn2C)C)C=CC(N(C)C)C1 C1(CC#C)(C(=O)N(CC(O)CNC(=O)CCc2cnc(O)[nH]2)C)CCCCO1 N1(C(CC(C)c2ccco2)=O)CC2CC(C1)CN(C(=O)CN1CCCOC1=O)C2 N1(C(C(C)(C)OC(C)C)=O)CC2C(NC(c3ccc(O)cn3)=O)C2C1 C1(CN(OCC)Cc2cc(O)ccc2C)CC2(CCC2)CN1C(=O)CC(C)O CC(C)(CC(=O)NCC1CCC(NC(C2(C)CC2C(F)(F)F)=O)CC1)C(F)F C1(C)(NC(C=CCC)=O)CCCC1NC(=O)COCC(F)F C1(NC(C2CCC(C)(C)OC2)=O)CN(C(c2csnc2Cl)=O)CCC12CCC2 C(C(C(=O)NCC=CC(=O)NCC(c1ncc[nH]1)C)NC(C)=O)OC C(CCC(C)(C)C(=O)NCC1(CO)CC1(C)C)NC(CC1(NC(C)=O)CC1)=O CC(C)(CCCO)C(=O)NCC1(NC(=O)CCC[N+](=O)[O-])CCCOC1 c1(CC)nn(C)c(C(=O)NC2CCCN(C(=O)Cc3c(C)cccc3F)C2)c1Cl Cc1nc(CC(C)C)c(C(=O)NCCCCC(C)NC(=O)C(O)CN(C)C)s1 C(CCC(C(=O)NCC1=CCCOC1)NC(=O)C=CC1CCC1)OC C(C)(C(=O)N1CCCCCO1)N(C(C(CC)C(C)(C)CC)=O)C C1(O)(C(C)NC(c2ccccn2)=O)CCN(C(c2cccnc2C2CC2)=O)CC1 C(C(CC(=O)N1CCCC1SC1CC1)c1ccccc1)NC(C)=O C(=O)(C(F)C(C)(F)F)N1CCC(C(CNC(C(CC2CC2)OC)=O)C)CC1 N1(C(C=C(CC)C)=O)CCC(C(C)(C)C)CC1CNC(=O)C=C(C)C N1(C(=O)CC2CCCC23CC3)CC2CCCC2(C(N2CCC(CO)C2)=O)C1 c1(C(=O)NCC#CCNC(CS(=O)(=O)NC)=O)ccc2nnn(C)c2n1 C1(NC(C(CC)COC)=O)(CNC(c2[nH]c(=N)ccc2C)=O)CCCCC1C C1(n2ncc(C(=O)OCC)c2)CCN(N(C)C2CCc3ccccc32)CC1 C1(NC(C2(CC)CCCCC2)=O)CCC(C)(CNC(=O)Cc2cccn2C)CC1 c1(C(N2C(C)CC(NC(CCCNC(C)=O)=O)C2)=O)ccc2c(c1)OC(C)(C)O2 N1(C(C(CC)C#N)=O)CCN(C(=O)Cc2ccc(Br)cc2C)C2CCCC12 N1(C(Cc2cc(C)ns2)=O)CC=CC(NC(=O)CC(=O)OC(C)(C)C)C1 CCCC(C#N)C(=O)NC(C)(C(=O)NC1CCCC1OCC)C1CCC1 c1(NCC(CC(C)C)NC(=O)Cc2cc(F)ccc2F)c([N+](=O)[O-])cnn1C CCC(C)(C)C(=O)NCC1CCC(NC(=O)C(c2cccnc2)O)C1 N1(C(c2c(C)nccn2)=O)CCC2C(C1)CN2C(=O)Cc1ncn2c1COCC2 N1(CC(=O)NCCC2CN(C(CCn3c(C)ncc3)=O)C2)CC2C=CC1C2 N1(C(c2c(C(C)C)con2)=O)CC2CC(C1)N2C(C1CC2CCC2C1)=O CC(C)CC(CC(=O)NC1CCC(O)CC1)NC(=O)CN1CC(=O)NC1=O CCCC(CCC)C(=O)N1CCC(C)C1C(=O)NC1CCOCC1F C1(C2CN(C(C3CCNC(=O)C3)=O)C2)(NC(C(C)Cn2ccnc2)=O)CC1 c1(CNC2CCN(C(C3(C(N)=O)CC3)=O)C2)ccc(F)c(C(F)(F)F)c1 CC(C)CCC(C(=O)NCC1CC(=C2CC2)C1)NC(=O)CC1=CCCC1 CS(=O)S(=O)CCN=c1[nH]c(N2CCC(c3cccnc3)C2)nc2ccsc12 c1(SC)ccc(C)c(C(=O)NCCC(C)(C)NC(=O)Cn2cccc(O)c2=O)c1 CCCCCCC(CC)C(=O)NCC(C)NC(c1ccc(-n2cccc2)cc1)=O C1(CC(N2C(CN(C(=O)CN3CCCC3=O)C3CC3)CCC2)=O)(CO)CCOCC1 N1(C(CC(CC)c2ccccc2)=O)CCC2(CCCN2C(=O)CC=C(C)C)C1 c1(-c2cn(CC(C)C)nc2)ccc2c(c1NCc1cnn(C)c1Cl)OCO2 CC1CCOC1C(=O)NCCn1cc(C(=O)NCC(CO)C2CCC2)nn1 c1(CN(C)C(=NCCc2cn(C)nn2)NC2CC2)cc2c(cc1[N+](=O)[O-])OCO2 c1(N(CC(=O)OCC)C)cc2c(s1)CCN(Cc1cccc(O)c1O)C2 Cc1nc(C(=O)NC2CN(C(=O)C(F)=CCCF)CC2C)c(Br)s1 c1(CN(C)C)cc(C(=O)NC2CC(NC(c3cnn[nH]3)=O)C(O)C2)ccn1 N1(c2ccc(CC(=O)OCC)cn2)CCC2(NC(C3CC3F)=O)CCCC12 c1(CCC)nc(C(=O)N(CCCNC(=O)C(F)(F)c2nccs2)CC)cs1 N1(C(C(CC(C)C)O)=O)CCC2(CCC2)C(CNC(=O)C#CC(C)(C)C)C1 C12(CNC(c3nn(CC)nc3C)=O)CC(NC(=O)C=C(Cl)Cl)(C1)C(C)(C)O2 c12cc(C)c(o1)C(=O)NC2.C(=O)(C(F)C(=O)OCC)NCC1CC(O)CN1C(C)=O C(=O)(CCCC(=O)NC(C)C(C)(C)C(=O)NC1CCOC1=O)OCC CCC(CNC(=O)C(O)CNC(=O)C=Cc1cc[nH]n1)C(C)(F)F C(c1cccc(Cl)c1)=C(C)C(=O)NCCCCC(C)NC(C1CC(CF)C1)=O C(=O)(C(O)C1=CCCCC1)NC1(CCC(N2CC(C)(CO)C2)=O)CCCC1 c1(CN(C)CCSC(F)F)ccc2c(c1)OCCO2 CCC(C)(C)CNC(C1(F)CN(C(=O)Cc2cscn2)C1)=O C1(C(=O)NC2C(CNC(C(C)NC=O)=O)COC2)C2CCCCC12 C(=O)(C(C)CC(F)(F)F)N(C(C)C(N1CC(F)C(F)C1)=O)C1CC1 C1(C(=O)NC2C(OC)C(O)C2)CCCCCN1C(c1ncnc(C)c1C)=O C(=O)(CC(F)(F)Br)N(CCCNC(=O)C=C1CCOCC1)CC c1(OC)nc(C(=O)NC(C2CCCC2)CNC(c2cnnc(C)c2)=O)sc1C C1(CC(=O)NC)CN(C(C2CN(C)C2)=O)CCN1C(c1cc(C2CCC2)no1)=O C(=O)(CC(C)(O)COC)N1CC(c2c(C(=O)NCC(CC)CO)con2)C1 CC(C)N=c1[nH]c(=NCC2CC3(CCCC3)CO2)[nH]c2c1CCC2 c1(SC)ccncc1NC(c1cscc1-c1ccnc(-c2ccccc2)c1)=O c1(N2CCC(CC(N3C(C)COCC3)=O)C2)cnc(C#N)nc1 c1(NC(CC)C(O)C(C)C)ncccc1S(=O)(=O)NCc1nc(C(N)=O)co1 C#Cc1cc(C(N2CCC(CO)C(NC(=O)CCOCCOC)C2)=O)cc(F)c1 c1(C(N2CC3C(NC(c4c(SC)snn4)=O)(C3)C2)=O)ccc(C)cc1Cl C1(C(N(CCOCC#C)C)=O)CC2CN(C(=O)C#CC3CCCC3)CC2C1 Cc1ccc(CCC(=O)O)cc1[N+](=O)[O-].n1(C)cc(CC(CO)C2CC2)nn1 c1(NC(=O)C(c2nc(CCO)cs2)N2CCC(CF)C2)ccc2c(c1)OCCO2 C(=O)(CC(C)CC(C)(C)C)N1CCCC(NC(c2ccc(OC)nn2)=O)(CO)C1 C1(CNC(c2cc(C)no2)=O)CN(C(=O)C(C)CN2CCOCC2)CCC1(C)C Cn1nnc2ccc(C(=O)NC3CN(C(c4cc[nH]n4)=O)CCC34CCC4)cc12 N1(CC23C(C)(C)C(CO2)C3)CCn2c(Cc3ccccc3F)nnc2C1 C1(NC(C(C(CC)C)O)=O)CCN(C(c2cc(O)cc(=O)o2)=O)CCC1CO C(N=c1cc(F)nc[nH]1)C1N(C(CN(CCCCCC)C)=O)CCC1 N1(C(c2cnc(C)n2C)=O)CCC(C2CC2)C1Cn1cc(C2(O)CCOC2)nn1 CCCC(C)(CC)NC(C1(CC)CCN(C(=O)CC2CCCO2)C1)=O c1(-n2c(C)cc(C)n2)ccc(NC(C2(C)CN(c3cc(O)ncn3)C2)=O)cc1F C1(CNC(C(C)(C)n2cnnn2)=O)C2CN(C(=O)CCc3n[nH]c(=N)s3)CC12 C1(C(C(=O)OC)(C)C)CCN(S(=O)(=O)CCNc2scc(Cl)c2Cl)CC1 C1(OC)CCCCN(CC(N2CC(NC(=O)C=CC3C(C)C3(Cl)Cl)C2)=O)C1=O C1(NC(C(c2cccc(Cl)c2)C)=O)CC12CCN(C(C1CCCC(=O)O1)=O)CC2 c1(CN)ccc(C(=O)N(C)C)cc1.c1(C(CC)=O)ncc(C)s1 C12(NC(=O)CCc3ccc(F)cc3)CCCC1N(CCC(=O)NC1CC1)CC2 N1(C(CCN(CCCCOC)C)=O)CCC(NC(C2CCOC2(C)C)=O)C(O)C1 C(=O)(C1CCCc2nc(C)[nH]c21)N1C(CN(C(CC2(C=C)CC2)=O)C)COCC1 c1(C(N2CCC(N(C(C3CCCNS3(=O)=O)=O)CC)C2)=O)ccc(N)c(F)c1F N1(C(c2c(O)ccc(N(C)C)c2)=O)CCC2(CC1)CC2CNC(=O)CNC=O O=C(O)CC(CCc1ccccc1)NC(c1cc(-c2cccc(Cl)c2F)no1)=O c1(CNC(C(CC(C)C)NCC=C)=O)c(C)nc2ncnn2c1C C(=O)(CCCCNC(C1CN(Cc2cc(C)ccn2)CCS1)=O)OC c1(C(=O)NCCC2CCN(C(C(CC)(C)C(N)=O)=O)C2)cccc2nc(C)sc12 Cc1cc(C(N2CCOC(CNC(C3CCCC(=O)O3)=O)C2)=O)cc(N)c1 c1(CC(=O)NC2CCC(CNC(C3(C)CSC3)=O)C2)cncc(O)c1 C(=O)(C1CCCc2nnn(C)c21)N1CC(NC(C2(OCC)CCOC2)=O)(CO)C1 N1(C(CCCOCC)=O)CCN(C(C2CC(F)C(=O)N2)=O)C(c2nccn2C)C1 CC1(C)CN(C(c2coc(Br)c2)=O)CC1NC(=O)C=CC1CCOCC1 c1(C(=O)NCCCC#C)cc2cc(-c3cc(F)c(O)cc3F)ccc2cc1O C1(CC)CN(C(=O)CCn2nc(C)nc2C)CCC1NC(c1sc(F)cc1Cl)=O c1(CC(=O)NC(CNC(c2c(C)noc2)=O)(C)CO)ccnc(C(F)(F)F)c1 C1(C(=O)NCC2(C)C(C)CN(C(C34CC(CO3)C4)=O)C2)COc2ccccc2O1 C1(C)(CNC(c2cc(C)c(C)o2)=O)CCN(C(C2SCCC2C)=O)CC1 CCCC(C)(C)CC(=O)NCc1cc(C)c(C(N2CCC(C)(F)C2)=O)o1 Cc1nc(C(=O)NC2CCN(C(C3CCC3)=O)CC2O)cn(C)c1=O CC12CSCC1CN(C(=O)CNC(C1CN3CCN1CC3)=O)C2 c1(C(CNC(C2(SCC)CC2)=O)NC(C2CC(CC)C2)=O)ccccc1 C1(NC(C(C)Cc2cnc[nH]2)=O)CC2CCC1CN2C(=O)C(F)C(C)(C)O N1(C(CSCC)=O)CC(NC(C2CC3CCCC(C2)N3C)=O)CC2(CCC2)C1 C(=O)(CC(C)(O)COC)N1CC(CNC(c2n(CC)ncc2Cl)=O)C(OC)C1 Cc1cccn2nc(C(N3CC(CNC(=O)C(C)n4cccc4)CC3C)=O)cc12 O=C(C(F)(F)CCn1ccnn1)NCC1CCN1C(c1c(F)cccc1F)=O C1(C(=O)NCC2CCN(C(COC)=O)C23CC3)COc2c(OC)cccc2C1 c1(C(=O)Nc2ccc(C)c(Br)c2)cnc(C)c(Cl)c1Cl C1(CNC(C2(CC#C)CCOC2)=O)CCCCN(C(c2cc(O)n(C)n2)=O)C1 C1(CCNC(=O)C(c2ccc(F)cn2)(F)F)CCN(C(=O)CCF)CC1(F)F c1(C(N(C(C)CNC(=O)Cc2nocc2C)CC)=O)ncoc1Br C1(C(N2CC(CCC)C(CO)C2)=O)CNC(=O)CN1C(C1CCS(=O)CC1)=O c1(C(C)O)cn(CC(=O)N(C)CCN(C(=O)CC2CCCC2C)C)nn1 C(=O)(C1CCc2cccc(F)c21)NCCCCCCNC(c1n(C=C)nnc1)=O C1(NC(CCC(=O)NC)=O)CCN(C(=O)C(C(C)C)OC)CC1CN(C)C C(C#CC(F)(F)F)NC(c1c(CNC(CN(S(C)(=O)=O)C)=O)cc[nH]1)=O C1(F)(C(N2CCCC(C(C)C)C2)=O)CCCN(C(=O)CC2CC3(CC3)C2)C1 C#CC1(C(N2C3CSCC2C3)=O)CCN(C(c2ncn3ccccc23)=O)C1 c1(C(N2CC(O)(CNC(CCCC(=O)OCC)=O)C2)=O)cc([N+](=O)[O-])cn1C N1(C(c2cn(CCC=C)nn2)=O)CCCC(C2(NC(=O)C(C)CN(C)C)CC2)C1 c1(OC)ccc(CC(=O)NCC2CCCC(NC(C3C4CC5C(C4)C35)=O)C2)nc1 Cc1cccc(C(N2CCC3C(NC(C4CCOC4C)=O)C3C2)=O)c1O C1(CNC(c2cccc(NS(C)(=O)=O)c2)=O)CC12CCOc1ccccc12 O=C(C(CCCC1CC1)N1CCCC(F)CC1)NCCc1cccc(F)c1 CC(C(=O)NC(CO)CCC1CC1)(C1CCC1)NC(=O)CN(C1CCCC1)C CC1CN(C(c2nnn(C)c2C(F)(F)F)=O)CC1NC(c1cc(C(F)F)[nH]n1)=O N1(C(c2ccc(C(C)=O)s2)=O)CC(C)(C)C(NC(=O)C(Cl)=CCl)C(C)(C)C1 c1(C(N2CCC(C(C(=O)NCC(CC)C#N)C)C2)=O)cc(C)c(C)o1 c1(C(=O)OCC)ccnc(C(N2CCC2CNC(=O)C(Cl)=CCl)=O)c1