SMILES C(=O)(CCCCCOC)NCC1C2CN(C(CC(C=C)C)=O)C1C2 N1(C(C2(C)CC2(Cl)Cl)=O)CCC(CNC(=O)CC2C=CCCC2)CC1 C1(C(N2CCC(OC)(CNC(=O)C=C=C(C)C)C2)=O)CC(=O)C12CCC2 C(=O)(CCCC(=O)N(C)CC1CC(F)CN1C(C1CC2COCC2C1)=O)OC c1(C(=O)NCCC(C)NC(CCc2cnc(C)o2)=O)ccncc1OC(C)C c1(C(=O)NCC2C(CNC(c3c(OC)cc(C)cn3)=O)C2)sccc1S(N)(=O)=O CC(O)CCCCCC(=O)N1CCC(C)(CCNC(=O)C=Cc2ccccn2)C1 C1(NCc2c(CCC)cccc2)CCC(=O)NC12CCC2 c1(C2(C(=O)NC3C(CNC(C(C)C4CC4)=O)CC3)CCC2)ccc(F)cn1 C(=O)(C(CC(C)C)C(C)C)NC1(C(N2C(C#C)CC3(CC3)C2)=O)CC(F)C1 N1(C(CCn2ccc(C)n2)=O)CC2(CCC2CNC(=O)CSc2nnnn2C)C1 N1(C(C)C)CCC(C(=O)NCC(O)CCNC(=O)C(C)(C)O)CC1 C#CC1CCC(C(=O)NC2CCC(NC(C3CC4CC3CC4O)=O)C2)CC1 C12(C(NOCCCC(=O)OC)=O)COCC1CN(C(c1ccnc3cc[nH]c13)=O)C2 c1(C(=O)NCCCC(C)(C)NC(=O)Cn2nccn2)ccn2ccnc2n1 c1(CC)ncncc1C(=O)NC1(C(=O)ON2CC3CC2CO3)CCCC1C c1(C(N2CC(C(C(=O)O)F)C2)=O)ccc(Br)c2c1CCCC2 C1(O)(C(=O)NCC2(C)CCN(C(C)=O)C2)CCCN(C(c2occc2C)=O)C1 C(=O)(N=c1[nH]nc(-c2ccc3c(c2)OCCO3)s1)Nc1c(CC(C)C)cccc1 N1(C(C(=O)NCCSC)=O)C(C)CN(C(c2cccc(C3CC3)c2)=O)CC1C Cc1cc(F)ccc1C(=O)NC(C)C(=O)N1CC(c2nc(=O)o[nH]2)C1 C1(NC(CNC(CN(C(=O)CCc2csnn2)C)=O)=O)CCCO1.C12CC1CS2 N1(C(CCCSC)=O)CC2(CNC(=O)Cc3cc[nH]c3)CCC1CC2 N1(C(C2CCCN(C(C3(Br)CCC3)=O)CC2)=O)CCn2c(Br)nnc2C1 C1(CNC(=O)COCCSC)CCCCN1C(C1(OC(C)C)CCC1)=O C1(C(=O)NC2(C(=O)OC)CC2)CCN(C(=O)Cc2cc(C)on2)CC1 C1(CCC(=O)N(CC(CNC(COCC(=O)NC)=O)O)C)CCCCO1 CCC(C)(CN=c1nc(N(CCC(O)C(C)(C)C)C)c2ncccc2[nH]1)C(N)=O N1(CC=C)CC(C)(n2nc(-c3cccnc3)nc2-c2ccn(C)c(=O)n2)CC1=O C1(C(C)(C)CNC(=O)CCn2ccnc2)CCCN1C(=O)CC(O)C1CCCC1 C1(C(=O)NCc2n(C(C)C)ncn2)CN(C(C2CC(=O)C2)=O)CCO1 c1(C(C(N2CCC(CNC(CNS(NC)(=O)=O)=O)C2)=O)=O)ccc(F)cc1 Cc1ccc(NCC(=O)NCCCC2(NC(C3CC3c3cncs3)=O)CC2)cc1 C1(C#N)(SC)CN(C(=O)C(C)NC(=O)CN2CCCC2)C1 c1(C(=O)NC2C(NC(c3scc(C)c3Cl)=O)C2)c(F)ccc(F)c1O C(=O)(C1=CCC(C)CC1)NC(CNC(C1(OCC)CCOCC1)=O)(C)CO N1(C(C2C(=C)CC2)=O)CCC(CCOC)(NC(c2ncc(OC)cc2F)=O)CC1 C(CC(O)C(=O)NCCCCCC1CC1)NC(Cc1scc(C)c1)=O c1(SCC(=O)N(C2CCN(C(C(CC)O)=O)CC2)CCO)ccc(C#N)cc1 c1(CCNC(c2nnnn2CCC2(C)CC2)CCC)cc(C(C)(C)C)no1 N12CCC(C1CC)C(=O)NCC#CC2=O.C(CCC(=O)OC)OCC O=C(CC(C(F)(F)F)NC(c1cnsc1)=O)NCCN1C(=O)CNC1=O C1(C(=O)NCCC2(CNC(c3nc(C)c(C)s3)=O)CC2)CN(C)CC(C)O1 CCC(C(=O)N1CC2CCC(CNC(c3c(C)ncnc3C)=O)C2C1)C(F)(F)F c1(C(=O)NCCNC(c2ncc(C)cc2Br)=O)oc2c(C)cccc2c1C c1(CC(N2CCN(c3nc(C(F)F)nc(=N)[nH]3)CC2)=O)ccc([N+](=O)[O-])cc1F C1(NC(C2CCC(C)(C)C2)C)CCC2CN(c3nc(C4CCC4)ns3)CC2C1 C1(CC(=O)NCCC(O)CNC(C2C3COCC23)=O)CCCCC1 CCCCCC(O)CC(=O)NC1CC(C)N(C(=O)C(c2ccc(F)cn2)(F)F)C1 c1(C(=O)NC2CCN(C(CCOC)=O)C23CC3)ccc2nc(C)c(=O)n(C)c2c1 c1(OC)ccc(C)cc1C(N1CCC(O)C1C(=O)Nc1ncc(O)cc1Cl)=O c1(C(N2CC(N(C(COCC(=O)OC)=O)C)C(C)CC2)=O)noc2ccccc12 N1(C(C2CN(c3ccc(C)c(F)c3)C(=O)C2)=O)CCC2(CCCN(C)C2=O)C1 C#Cc1cc(C(=O)NC(CNC(=O)C(c2ccccc2)O)(CC)CC)cc(F)c1 C(=O)(C(=O)CCC(C)C)N1C(CNC(C(COC)(C)O)=O)CCC1 Cn1cnc2c1C(C(=O)N1CC(F)CC1CNC(c1cnccn1)=O)CC(=O)N2 C#CC(CNC(C1CNC(=O)CN1C(=O)Cc1ncn(C)c1C)=O)CC(C)(C)C CCC(COC)C(=O)NCC(c1ccccc1OC)NC(c1sc(F)cc1C)=O c1(C(C)(C)C)cc(C(=O)NCCCCCNC(=O)Cn2cc(C(N)=O)nn2)on1 C1(C)(C(=O)NCC2(CNC(c3c(C)nccc3)=O)CCC2)CCCN(C)C1 c1(C(=O)NC2CC(NC(=O)Cc3cc(Cl)cc(Cl)c3O)C2)cc2cccnc2[nH]1 C1(N2CC(NC(C3N(C(C(C)Sc4ccccn4)=O)CC3)=O)C2)CC(F)(F)C1 C1(CNC(COCC(C)C)=O)CCC(C)(C)CN1C(=O)CCCc1ccncc1 C1(C(N2C(C)CC(CNC(=O)C(N)=O)CC2)=O)CN(C)C(=O)CCO1 N1(C(c2c(C)c[nH]n2)=O)CCN(C(c2cn(C)nc2Cl)=O)C2CS(=O)(=O)CC12 CC1=NC(C)(C(=O)N(C)CC2CCCCN2C(C2CC(O)C2)=O)N1C N1(C(C2CCC(=O)NC2)=O)CCC2C(C1)CN2C(=O)Cc1cnoc1 N1(C(c2nc(CCC)sc2)=O)CC2CCN(C(c3noc(CC)c3C)=O)C2C1 C1(C#N)(NC(=O)NC(C2CC(NCc3ccc(C(F)(F)F)cc3)C2)C)CCCO1 C(=O)(CCCCC(C)C)N1C2CC(CNC(CC3(COC)CC3)=O)C1CC2 N1(C(C(CCC)C)=O)CC(C)(C)CC1CNC(C1(CC(=O)OC)CC1)=O C(C(=O)NCC(CNC(=O)CCCn1cncn1)CO)(C(C)C)NC(COC)=O CC1(C)C(NC(=O)C=Cc2ccc(C(N)=O)o2)CCN1C(=O)C1=NNC(=O)C1 c1(C(=O)NC(CNC(C(CC)N2CCCC2=O)=O)C)cc(NC(C)=O)cnc1O c1(-c2ccc(C(N3C(C(N)=O)CCCCC3)=O)o2)c[nH]c2ccccc12 C=CC1CN(C(=O)C2=CCSC2)CC1NC(C1CSCCS1)=O C(CCC(=O)NC1(CC)CC1)SCC.C12(CC(O)C1)C(=O)N2 C1(C(N2CCC(CC=C)(NC(c3nnc(C(C)C)s3)=O)C2)=O)CCCCN1N=O C12(CNC(C3C(CNC(c4c(CC)occ4)=O)CC3)=O)COC(C1)C(O)C2 C1(N(CCC)C(C2CCC2c2ccccc2)=O)Cc2ccccc2C1 c1(C(=O)OC2CCc3ncccc3C2)cccc(S(=O)(=O)N2CCCCC2)c1 N1(C(C(=O)Nc2ccc(OCC)cc2)=O)CCN(C(=O)C(F)(F)F)C(CC)C1 c1(C(N2CC(C)C(C)(CNC(c3ccc(F)o3)=O)C2)=O)cc2cccn2c(O)n1 CC(CC(F)F)C(=O)NCC1(O)CCCN(C(C2(CCN(C)C)CC2)=O)C1 C=CCC(CC(=O)NCC1CC12CCC2)NC(c1cn(CC)nc1C)=O C1(C(N(CCCOCCNC(=O)Cc2ccco2)C)=O)CC2CC1C2 c1(CCC)sc(C(N2CC(CNC(C3(C)CCCC3)=O)CC2C)=O)cc1CC O=C(C1=CCC2CCC1N2C(=O)CCn1cnnn1)NC1C(O)C2CCOC12 c1(C(=O)NC2CCN(C3CCOC3=O)CC2)cnc2sc(Br)cn2c1=O C1(C)(NC(CCc2cn(C)nc2)=O)CCCN(C(c2cc3cscc3s2)=O)C1 c1(C(N2CC(C#C)(C(=O)NC(CC#C)C(=O)OC)C2)=O)c[nH]c2nccc-2c1 N1(C(C2C(c3n(C)ncc3)C2)=O)CCOC(C)(C)C1CO C(c1csc2ccccc12)=CC(=O)N(CCNC(C1(OC)CC1)=O)CC C#CCCCCCC(=O)NCC1(O)CCN(C(=O)Cc2cn3c(n2)CCCC3)C1 c1(CN(CCN)CC)ccc2nonc2c1 N1(C(C2(NC(C3CC(C)(C)CO3)=O)C(C)C2)=O)CCN(CC(N)=O)CC1 c1(CNC2(C(=O)NC)COC(C)(C)OC2)cn(C)c2ccc(OC)cc12 C1(COC)CC(C)(C)CN1C(C1(C(=O)NC2CC2CNC(C)=O)CC(C)(C)C1)=O C(=O)(C1SCCc2sccc21)NC(CCCC)CNC(c1cnn(CC)c1)=O.CC=O C1(NC(c2c(C)nc(C)[nH]2)=O)CCCC(NC(=O)CCN2C(=O)CCC2=O)CC1 c1(N2CC(C(=O)NCCC)OCC2)ncc(Cl)c(N(CCC(F)(F)F)C)n1 C1(CC(=O)NC2(CN(C(CCN(C(C)=O)C)=O)C)CC2)CCC(C2CC2)O1 c1(C(=O)NC(C(NOCCOCC)=O)c2ccco2)cc[nH]c2nccc1-2 c1(CC(N2CC(O)(CN(C(CSCC(=O)OC)=O)C)C2)=O)cccc(C)c1 c1(C(N(CCNC(C(=O)NCC)=O)C)=O)cnn(CC(F)F)c1 C1(C(N2CCC(OCCNC(=O)Cc3csc(S)n3)C2)=O)CCCCOCC1 N1(C(C2C(COC)C2)=O)CC(F)(F)CC1CNC(=O)COC1(C)CCC1 C(=O)(CC1=CCCCC1)N1CCC(C(C)CN(C(C)CCO)C)CC1 C(CCCCC(=O)N1CC(NC(=O)C(c2ccccc2)C)C(O)C1)OCC N12CCCC1C2=O.N1(C(CCC)=O)CC=CC1CNC(=O)Cn1cc(C)cn1 Cn1cc(Cl)c(C(=O)NCC(CO)NC(c2cccn2C)=O)n1 C(C)(C)(CC(=O)N1CC(CCNC(c2sccc2C2CC2)=O)(OC)C1)OC Cc1[nH]c2ccccc2c1C1=CCN(C(C2CC(C(F)(F)F)OC2=O)=O)CC1 N1(C(CNS(C)(=O)=O)=O)CC(CNC(=O)CC2CC(F)(F)C2)N2CCC1C2 C1(C)(CNC(C2C(C)=C2)=O)CCCN1C(C1CC(C)OC1C)=O c1(-c2n(CCCCC)nc(C(C)OC)n2)nn(-c2ccccc2)cc1[N+](=O)[O-] C#CCC(C)C(=O)NC(C)CNC(=O)COc1ccc(C(C)C)cc1 N1(C(c2c(C)oc(Cl)n2)=O)CCC2(C)CN(C(=O)CCC3CC3(C)C)CC12 N1(C(C2(CO)CCN(C(CNC(C(C)(C)C)=O)=O)C2)=O)CC2(CNC(=O)C2)C1 C1(NC(c2cc(C)no2)=O)CCOCC1NC(c1cc(C)c(Br)s1)=O C1(CC=C)(NC(C2CCOCC2)=O)CCN(C(C2CC(=O)N(CC)C2)=O)C1 C(=O)(CCCCC(=O)N1CC2(CCC(NC(C3CCCC3)=O)C2)C1)OC N1(c2nnc(C)c(C)n2)CCC2(NC(=O)C(F)CC3CCCCC3)CCCC12 c1(N2CCCC(N3C(=O)NCC3)C2)nc(=NCCC(F)F)[nH]c2c1CCCCC2 c1(C(=O)NC2C(C(N(CC)Cc3cccc(Cl)c3)=O)C2)ccccc1CO N1(C(C=CC2N(C)CCC2)=O)CCCC(C)(C)C1CNC(c1cccc(N)n1)=O C1(SC)CN(C(=O)C(C(C)C)n2cncn2)CC1NC(c1ccco1)=O c1(C(N2C(CNC(C3CC4C=CC3CC4)=O)CC2)=O)cc(F)ccc1Br C1(C(N2CC(COC)N(C(=O)C(O)P(C)(C)=O)CC2)=O)Cc2ccncc2C1 c1(OC)ccc(C)cc1C(=O)NC1CN(C(=O)C(F)(F)C(C)O)CCC1CO C12(CN(C(c3cc(C)no3)=O)C1)C(=O)NC2.CCC(CSC)OC N1(C(CC(C=C)(C)C)=O)CCC2(CNC(c3coc(SC)c3)=O)CCCCC12 C=CCCC(C)(C)C(=O)N1CCCC(NC(c2ccc(C(F)(F)F)cc2)=O)C1 Cn1ncc2c1CC(C(N1CCCC1CCCNC(=O)CC1CSC1)=O)CC2 S(=O)(=O)(c1nc2c(s1)CC(=O)CC2)NC(C1C(C2C(C)(C)C2(C)C)C1)=O Cc1cc(C(=O)NCC2CCCCN2C(=O)CN2CCC(CO)CC2)ncc1N C1(OC)COCCC1CC(N1CCCC1CN(C)C(c1coc(O)n1)=O)=O C1(C(C)C)C(=O)N1.C1(C)(NC(C)=O)CC(C(=O)NCCC2(COC)CC2)C1 c1(CNC(C(C(C)C)F)=O)nnc2n1CCN(C(=O)Cc1nc(C3CC3)cs1)C2 c1(C(=O)NC2CC3(C2)CC3C(=O)NCC2CC2(F)F)c(F)cccc1F c1(C(N2CC(C=C)C(NC(c3cnc(C)[nH]3)=O)C2)=O)sc2ccccc2c1Cl C1(CC(=O)NCC2(CO)CCCC2)C=CC(NC(c2cncs2)=O)C1 C(=O)(C(C)(C)C1=CCN(C(=O)CCCC2CC2C)C1)NCc1onc(C)n1 CC(C)C(CCN(C(=O)C(C)(C)c1ncco1)C)NC(=O)CO C(=O)(C(CSC)OC)N(CCN(C(=O)C(C)Cc1ccccn1)CC)CC Cc1cc(C)c(C(N2CCCC2C(C)NC(c2ccc(OC(F)F)cn2)=O)=O)s1 C1(C(=O)NCC(CC(C)C)NC(c2c(C)nccc2)=O)CC2CCCCN2C1 c1(C(=O)NC2CCN(C(C(CC(C)C)N(C)C)=O)C2)cccc2c1OCC2(C)C c1(C(N2CCC(CN(C)C)CC2)=O)cc2[nH]ccc2cc1-c1cccn1C CC1(C)CCOC1CC(=O)NCC1CC(NC(=O)C2=CCSC2)C1 c1(C(C)C)ncc(C(=O)N(C)CC2CCN(C(=O)CN3CCCC3CO)C2)[nH]1 c1(C(=O)NC(C2OCCN(C(c3cc(OC)ns3)=O)C2)C)ccc(Cl)nc1Cl Cc1cnc2c(cnn2CC(N2CCCC([Si](C)(C)C)C2)=O)c1 c1(C(N2CC(NC(C3CCSC3)=O)CC3(C2)CC3)=O)cc2cc(Cl)cnc2o1 c1(OC)cc(C)nc(NCC2CC(NC(=O)Cc3cccn3C)C2)n1 N(C1COc2cc(Br)ccc21)C(c1n(CC)nnn1)c1cc(C2(O)COC2)on1 Cc1n[nH]c(C)c1C(C)C(N1CCC(C(C)NC(c2ccc(F)cn2)=O)C1)=O c1(C(=O)NCCC2CCN(C(C(C(C)C)C#N)=O)C2)ccsc1S(N)(=O)=O C1(N(C(=O)C(=O)NC(C)C)CC)CCCN(C(=O)C(c2cn(C)nc2C)C)CC1 Cc1cc(C(=O)N(CC(C)CNC(=O)C(O)C(F)(F)F)C)cc(C)c1F CN(C)N=Nc1ccccc1C(=O)NCC1(O)CS(=O)(=O)C1 C1(c2cccc(OC)c2)CN(C(C2(C)C=CCC2)=O)CCN1C(=O)COC(C)C c1(C(N2C(CNC(CNS(CC)(=O)=O)=O)C=CC2)=O)cc(C(C)(C)C)ccc1O C1(N(C(C2C(CCC)CCC2)=O)C)CCCN(C(c2cnc(F)c(F)c2)=O)CC1 c1(C(=O)NC(C)CNC(C2CC2C2CCC2)=O)c(Br)ccc2n[nH]cc12 c1(C(N(C(C)CN(C)C(C2CC(F)C(=O)N2)=O)C)=O)ncc2c(F)cccn12 C1(CC)(CC)CC(C(=O)OCC(=O)N(C)CC2CCCC2)C1 C1(C(=O)NCCNC(Cc2ccn(C(C)C)n2)=O)COCCN1CC(F)(F)F N1(C(C2(C)CC(=C)C2)=O)CCC(O)(C2CCN(C(C3CN(C)C3)=O)CC2)C1 c1(SC)nccnc1C(=O)NC1CCN(C(=O)CC2CCOC(C(C)C)C2)CC1 C1(C(=O)NCC(C)N(C(=O)Cn2cccc2)C)OCC1(C)C CC(C)CC(C)CC(=O)NC(C1(O)CN(C(=O)C(C(C)C)NS(N)(=O)=O)C1)C c1(CNCC2(C(=O)Nc3cc(O)ccc3I)CC2)ccncc1[N+](=O)[O-] n1(CC(C)C)[nH]c(CC(=O)NC2CC(CCNC(C3CCCO3)=O)C2)cc1=O N1(C(c2c(OC)n(C)nc2)=O)CCC2CCCC(C1)N2C(C1CSCCS1)=O N1(C(CC2C(C)C2)=O)CC2CCC(C1)C2NC(c1cc(Br)cc(Br)c1)=O C=C=CC(C)C(=O)N1CC(F)CC1C(=O)N(C)OC C12(CNC(C3N(C(C4C(C)C4C)=O)CCOC3)=O)CCN(CC1)CC2 C12(NC(=O)OC(C)(C)C)CC1CN(NC(c1c(CSCCCC)ocn1)=O)C2 Cc1cc(=NCC(C(C)C)N2CCC(C)CC2)[nH]c(N2CC(C)C(F)(F)C2)n1 C1(NC(COCCC)=O)CC2CC(NC(=O)C(C3CCC3)OC)C1C2 C(=O)(C(C)(F)C(C)(C)F)NC(c1cccnc1)C(=O)NCc1nc(C)[nH]n1 c1(C(=O)NCC(CO)NC(C2C(C)N(C)CC2)=O)cc(F)c(F)c(Cl)c1F C1(n2cccn2)(C(=O)NC(C2CCOC2)C)CCN(C(=O)COCC2CCC2)CC1 C1(C(=O)NCC(C)(C)CCO)(COC)CCCCCC1 c1(CC)csc(CC(=O)NC2(C3CCCN3C(=O)COC3(C)CCC3)CC2)n1 CCCC(C)(CC)C(=O)N1CC=CC(NC(=O)Cc2ccc(OC(F)F)cc2)C1 C1(C(=O)NCC=C)CC(F)(F)CN1Cc1ccc(C2CC2)cc1 N1(CCCNC(N=c2ccn(CC(=O)NCC)[nH]2)=O)Cc2ccccc2C1=O C1(CC(=O)NCC(CC=C)NC(c2[nH]cc3c2CCC3)=O)CCC(C)(C)CO1 C1(CNC(=O)OC(C(C)C)C(F)(F)F)COc2cccc(Br)c2C1 c1(C(=O)NCC2(C)CCC(NC(=O)CC3CC=CC3)C2)cc(Cl)ncc1O c1(Oc2nccc(C(=O)NCC=CC(C)=O)c2)ccc(C)cc1Br N1(C(=O)OC(C)(C)C)CCC2(CCC2C(=O)NC(CCl)C(=O)O)CC1 N1(C(C2CCC(N=[N+]=[N-])C2)=O)CCC(C2CCN(C(C3CC=CCO3)=O)C2)CC1 C1(C(=O)Nc2nnc(CC(=C)C)s2)CCCC(Nc2ccccc2)C1 N1(C(C(CCCC)(C)F)=O)Cc2n[nH]cc2C1C(=O)N1CCC(O)CC1 N1(C(Cc2cc(C)oc2C)=O)CC2CC1CN2C(c1ncoc1C(C)(C)C)=O N1(C(C(CCF)NC(c2nn(C)c(Cl)c2)=O)=O)CCOCC(C)(C)C1 c1(OC)nc(=NCC2CN(C(c3cnnc(O)c3)=O)CCCO2)[nH]c2[nH]cnc12 c1(C(=O)NC(C(C)C)(C)CNC(=O)CN2CCCC2C)cc2cc(Cl)ccc2[nH]1 N1(C(c2c(CC)nc[nH]2)=O)CC(NC(C2CC3OC2C2CC32)=O)C2CCCC12 C(C1CCC(C)CC1)=C(C)C(N1CC(O)(CNC(c2ncoc2C2CC2)=O)C1)=O CC1CC2CN(CC3C(=O)NCCN3Cc3ccccc3)CCN2C1 c1(-c2scc(NC(C3CCCC3F)=O)n2)cccc(F)c1 c12c(F)cc(cc1F)OC(=O)C2.C1(O)(C(=O)NCCC(=O)O)CCCC1 c1(C(=O)NC(CCCCNC(C(CC)N(C)C)=O)C)nn(C)c(C)c1Br CCCCCC(=O)NCC(N1CC(CNC(=O)COCC(F)F)C(O)C1)=O C(=O)(CS(=O)(=O)N(C)C)NC(C1CCN(C(c2coc(C(F)F)c2)=O)CC1)C c1(CNC(c2ccccc2)C)cc(F)cc2c1OCC2.C1(COC)OCC2CCOC12 C1(C(N2C(CNC(c3n(CC)c(O)nc3)=O)COCC2)=O)CC1C1CCOCC1 CC1C2CN(C(=O)C(C)(C3CCCO3)C3CC3)CC12.C1(CC2CC2)CCC1 N1(C(C2CC(C(C)C)C2)=O)C2CCC1C(F)C(NC(=O)C1=CCOCC1)C2 C1(CNC(c2cnc(C)s2)=O)C2CN(C(=O)CCCNC(N)=O)CC12 c1(C(=O)NCC2C(C)CCCN2C(c2cnc(O)o2)=O)nn(C)c2c1COCC2 C(C(CO)C(F)(F)F)NC(=O)COCc1ccoc1C(N1CC=CC1CF)=O C(=O)(C1CCc2c[nH]nc21)N1C2CC(CN(C(CC(=O)N(C)C)=O)C2)C1 Cc1cc(NC(=O)NCc2cc(C(=O)O)on2)ccc1N1CCCC1 CC1CCN(C(c2cccnc2)=O)CC1NC(C1CNC(=O)N1)=O N1(C(Cn2ncc(C)c2)=O)CCC(NC(C2CC3CCC3C2)=O)CC(C)(C)C1 C1(CCC)(NC(=O)CNC(N)=O)CCN(C(=O)C(C)SC2CC2)CC1 C1(C#N)(C(N2CCC(C)(C(=O)NCC(=O)NC(C)(C)C)C2)=O)CC2CC2C1 N1(c2c(OC)cc(Cl)c(SC)c2)CC2CCCN(C(c3coc(C)n3)=O)C2C1 C=CCC(C(=O)NC1COC(C)(C)C1)NC(C1CC(=O)C1)=O c1(C(=O)NCCC2(O)CN(C(C(C)SCC)=O)C2)cscc1C#N C(=O)(C(C)CCCC(C)C)N1CCC(CNC(C(CC2CCC2)OC)=O)C1(C)C CN1CCN(C)CC(NC(=O)C(Cc2cn[nH]c2)NC(C2CCS2(=O)=O)=O)C1 c1(C(N2CCC(C(C(=O)N(C)CCOCCO)(C)C)C2)=O)cccc2cc[nH]c12 C1(C2CC2)C(=O)N1.C1(C)(OCCNC(C=CC(=O)NC)=O)CCC1 C1(NC(C=CC(C)C)=O)CC2(C1)CN(C(C1CCC(F)(F)CO1)=O)C2 CN1CCOCC1C(N1CC(N(C)C(c2ccc(C3CCCOC3)cc2)=O)C1)=O C(CC1CCC1)(C(=O)N1CC(O)(CCNC(C23CCCC2C3)=O)C1)OC CC(CCl)CS(=O)(=O)NCC1CCCCC1O c1(N2CCCC(CNC(C(C)(C)CF)=O)CC2)nccn2nnnc12 Cc1ccccc1-n1ncc(C(=O)NCC2(CNC(C3CSC3)=O)CCCC2)n1 c1(NC)ccc(C(=O)NCC(C)N(CCCNC(=O)CNC(=O)C(C)C)C)cn1 C(CO)(C(=O)NC(C1CCOC1)CNC(=O)Cn1nnnc1C1CC1)N(C)C c1(NC(=O)C2=CCOC2)ccc(C(=O)NCCNC(C(C)C)=O)cc1 c1(N(C)C)ccc(CN(c2cncnc2Br)CC#N)cc1Br.N12CCC(O)C(C1)C2=O N(C1CCCc2ccccc21)CC1CC(C)C1.C123CCC(CC1)(CC2)C(=O)N3 C(CS(=O)(=O)CC(=O)O)C1CCN(C(Cc2c(C)non2)=O)CC1 Cc1cncc(C(=O)NC2CCCN(C(=O)CCc3ccnn3C)C2C)c1Cl C1(NC(C(COC)OC)=O)CCCN(C(C2CCC2C#N)=O)CC1 CC(CC(=O)NCc1ncccc1NC(=O)CC1CSCCO1)C(C)(C)C Cc1ncc(Br)cc1C(=O)NC(CNC(=O)CC1(C)CCCO1)CO c1(C(N2CC3(CN(Cc4ccc(C(=O)OCC)[nH]4)C3)C2)=O)cc(Br)ncc1Cl c1(C(N(CC(C)(C)CNC(c2cocn2)=O)C)=O)nc2ccc(CO)cn2c1N c1(NC(COCC(=O)NCCN(CCOC)CCO)=O)cccc2c1OCCN2C CC12CN(C1)N2C(C1CCCCN1)=O.c1(CCCC2CCOCC2)cccnc1.CC N1(C(CC(C=C)C)=O)CC2(CC2)CC1C(=O)NCCc1ccncc1C N1(C(C2OCCC(NC(CCCN(C(C)C)C)=O)C2)=O)CC2(CCOC(=O)N2)C1 Cc1ccc2oc(C(N3CCCC(CN(C(=O)C=CC(N)=O)C)C3)=O)cc2c1 c1(C(=O)NCC(C)N(C(C2=NOC(C)C2)=O)C)cc2cc(Br)cn2cn1 c1(C(N2C(C(=O)Nc3c(CC)cccn3)CC3CC32)=O)cccc(C(F)F)c1F C1(C)(CC(N2CC(C(C(=O)N(CC)Cc3ccsc3)O)C2)=O)CCCO1 CC(C)C(C)C(=O)NC1CCC(CCNC(C2(CO)CCOCC2)=O)C1 C(=O)(C(C#N)C(C)(C)C)C1CC2(C(=O)N)C(C1)C2C.CC1CC(=O)N1C Cc1cc(C(=O)NC(C)(CNC(C2CC(C)(C)CN2C)=O)C2CC2)nc(O)n1 CCS(=O)(=O)CCNC(=O)CC1(N(C)C)CC1.C12CCC(O1)CNC2=O C1(C(N(C2CCN(C(=O)C(C)=C(C)C)CC2)CC#C)=O)CC2CC(OC)C2C1 CCC(CC(C)C)C(C(=O)NCC)N1CCC(Oc2ccc([N+](=O)[O-])cc2C)C1 c1(C(N2CC(C3(NC(=O)CC(F)(F)F)CC3)C2)=O)cnc2ccoc2c1 C1(CNC(C(CNC(c2cc(OC)ns2)=O)OC)=O)CC(=O)N(C)C1=O N1(C(C(CCCC)NC(=O)CN(C)CCC)=O)CCOC(C2(C)N=N2)C1 c1(OC)ccc(CN2CCC(O)(C(=O)Nc3cc(Cl)cnc3Br)C2)c(F)n1 N1(C(c2cc(C)oc2)=O)CC(NC(c2ccccc2CC(C)C)=O)CC1C C(N=c1cc(C(F)(F)F)nc[nH]1)C1CC(NC(COC2CCC(C)CC2)=O)C1 N1(C(C2(C#N)CCC2)=O)CC2C=CC1C(C(=O)NCC1CC3(CCC3)C1)C2 C(=O)(CC(C)(C)NC(=O)CSc1ccc(CO)cc1)NC C1(C(N2CC(NC(c3c(C)onc3)=O)C(C(F)F)C2)=O)CCn2ncnc2C1 CN1CCC(O)C2(CCCN(C(NC3CCCOc4ccccc43)=O)C2)C1 C1(N(C(=O)C(C)=CC2CC2)CC)CCCN(C(C23CC(C)(C2)C3)=O)C1 c1(C(=O)NCCCNC(COCC=C)=O)cc(F)cc(C)c1N c1(C(=O)NCC2C(NC(C(CCC)N(C)C)=O)C2)cc(C)c(CC)nc1O c1(C(=O)NC2(C)CN(C(C(n3cc(Cl)cn3)C)=O)C2)cccc(CCO)c1 C(C(CC(=O)OC)C(F)(F)F)NC(c1n(CC=C)nnn1)(C)CCBr N1(C(C(C)NC(CC)=O)=O)C(C(N2CC(C)CC(C)C2)=O)C2CC(F)C1C2 S(=O)(=O)(c1ccc(Br)cc1Cl)Sc1ncnc(-c2c(SCC)cccc2)c1N C(=O)(CC(CN(C)C)C(F)F)N(C1CN(C(CCOCCCOC)=O)CC1O)C CCC(C)C(C(=O)N1CC(CC(=O)N(CC=CCCOC)CC)(OC)C1)N(C)C N1(C(C(CC)Cc2ccc(N)cc2)=O)CC2CC(C1)N(C(=O)CNC(=O)OC)C2 C(Cn1cncn1)(C(=O)N1CCCCO1)NC(C1CN(C)C(=O)C1)=O C(CCCCC(=O)NC(C)(CNC(c1c(C)c[nH]c1CC(N)=O)=O)CO)SC c1(C(N2CCC(COC)(NC(=O)CC(C)F)CC2)=O)ccnc(OC)c1[N+](=O)[O-] CCCC(C(=O)NC1(C(=O)NCC2CC2c2ccsc2)CC1)NC(C)=O c1(C(=O)NC2(CO)CN(C(c3occ(C(N)=O)c3)=O)C2)csc2c1CCCC2 CCCCCC(C)CC(=O)N1CCC(CC(=O)N(CC(C)(C)O)CCC)C1 CCC(C)(C)CC(=O)NC1CCN(c2cc(C3CC3)ncn2)CC1F Cc1cccc2c(CC(=O)NC3CCC(NC(=O)C(C)(C)C(F)F)C3)c[nH]c12 c1(OC)cccc(NC(=O)C(=O)NC2(C)CCC(Cc3ccccc3)CC2)c1Br C12(NC(c3cncc(C(C)=O)c3)=O)CCN(C(C3CCSCC3)=O)CC1C2 C1(CN(C(c2ccc(C#N)s2)=O)CC)CCN(C(C2CCC(F)C2)=O)CC1 C1(NC(CNC(CC)=O)=O)(CO)CCN(C(C2CC=CCO2)=O)C1 C(=O)(CC(C)C)N1CC(C(C)NC(CCOCCOCC)=O)C1.C1(=O)CCN1 Cc1nn(CC(=O)NCC2CCN(C(c3ncncc3Cl)=O)C2)c(=O)n1C N1(C(C(n2ncc(C)c2)C)=O)CCC(NC(c2ccon2)=O)C1C C#Cc1cccc(C(C(=O)NCC2CC2)N(C2CCCCCC2)CC(C)C)n1 Cc1c(C(N2CCC(NC(=O)C=Cc3nnn(C)n3)CC2)=O)ccn1C C#CC1CCN(C(=O)CC2CCN2C(c2ncnc(C)c2C)=O)CC1 c1(C(=O)NC2CN(C(C(CC)C)=O)CC2CC)nnc2ccccc2n1 C1(C(N(CCNC(C(OC)CN2CCOCC2)=O)CCOCCO)=O)CCOC1=O c1(C(=O)C(N2CCN(C(C3CCCO3)=O)C(CO)C2)=O)ccc(F)c(F)c1F Cc1ccc(-n2cc(CC3CCC(NC(c4cnc(Cl)s4)=O)CC3)nn2)nc1 CCCC(C(=O)OC)C(=O)N1CCC(N(C(=O)CCc2scnc2C)CC)C1 c1(C(C(N)=O)N(CC(Cc2ccccc2)OC)C(C)C)ccc(Cl)cc1 CC1(NC(C2CN(C3CCOC3)C2)=O)CCCN(C(=O)C(F)(F)C(F)F)C1 Nc1c(C(=O)NC(CNC(=O)CN2CCCCC2)CC(F)(F)F)cccc1Br c1(CNC(=O)NC(c2cc(Br)ccc2OC)CC)cc2ccccc2s1 N1(C(C(CO)NC(N)=O)=O)CC2CC(NC(C3(O)CCSC3)=O)C2C1 S(=O)(=O)(c1ccc2c(c1)CCC2)Nc1ncc(-c2ccc(C)cc2)cc1C C(CN=c1cc(NCc2nnc(C)o2)nc(C(C)C)[nH]1)NC(=O)OCC c1(CC(=O)NC2CCC(C)SC2)ncnc2c1CCC2 C1(NC(CCn2c(C)nc(C)n2)=O)CCN(C(=O)C(C)S)C(C)C1 CC1CC(C(N2CCC(N(C)C)(CNC(c3ccn(C)n3)=O)C2)=O)CC(=O)N1 c1(C(=O)NC2COCCC2NC(C2CC2F)=O)ccc(C(F)F)nc1O C(=O)(C(C)CS(C)(=O)=O)N1C(CNC(c2ncc(C)c(C)c2)=O)CC1 N1(c2snc(C)n2)CCCC1C1CCCCN1C(C1CCOCC1)=O c1(NC2CC3N(C)C(CC3)C2)ccc(S(=O)(=O)NC(CO)C2(C)CC2)cn1 O=C1CC(C(N2CCC2CNC(C2(F)CCCC2)=O)=O)CC(=O)N1 c1(C(N(CC(C)NC(c2cc(C(F)(F)F)n[nH]2)=O)C)=O)ncn2c1CCCC2 N1(C(C(C)OCCC=C)=O)CC(C)(C(=O)N(CC(C)(C)C)C)CC1(C)C Cc1[nH]c2ccccc2c1CC(N1CCC(N(C)Cc2cncc(Cl)c2Cl)C1)=O C1(OCC(C)C)CC(C(=O)NCCCNC(c2ccc(F)cc2)=O)C1(C)C C1(NC(CC2CCCC(C)O2)=O)CC(F)CN(C(=O)Cn2ncnn2)C1 N1(C(CC2N(C(C3C4CC(=O)CC43)=O)CCC2)=O)CC2(CCC(=O)O2)C1 N1(C(c2c(NC(C)=O)scn2)=O)CC2CN(C(=O)CN(CC(C)(C)C)C)CC2C1 c1(C(N2CC(C)OC(CCNC(=O)Cc3cnc[nH]3)C2)=O)n[nH]c2c1CSCC2 c1(C(=O)NCC(CC)NC(=O)C(C)(F)C(C)(C)F)cc(OC)c(OC)cc1C Fc1c(Cl)ccc(NCCN2CC3(CCOCC3)C2)c1Br c1(C(=O)NC2C3CN(C(=O)CSC(F)F)CC23)ccc2c(c1)CCCCS2 N1(C(C=CC)=O)CCOCC1CNC(=O)Cc1ccc(C2CCC2)cc1 c1(OC)ccc(F)c(C(=O)NCC2C3CCC(C3)N2C(=O)C(C)C(C)(C)O)c1 CC(C)C(F)(CNC(=O)C=C(Cl)Cl)C(=O)N1CCC2(CC(CO)C2)C1 c1(OC)nccnc1C(=O)NCC(O)CN(C(=O)CCN(S(C)(=O)=O)C)C C(CC(C(=O)N(C1(NC(=O)Cn2nnc(-c3ccsc3)n2)CC1)C)OC)OC CC1(CCO)CCN1C(C1CC1CNC(=O)CCn1cncn1)=O c1(C(=O)NCC2CC(COC)CN2C(=O)COC(C)=O)cc(=O)n(C)cn1 c1(C(N2CC(CNC(c3cc[nH]n3)=O)C3C2C3)=O)cc2ccc(Cl)c(F)c2o1 c1(CN2C(C(=O)Nc3nccnc3Cl)CCC2)ccc(O)c2ncccc12 c1(C(=O)NC(CNC(CC(C=C)C)=O)CC)ccc(C)nc1C(C)C c1(C(N2CCC(CN(C)C(c3cnn(C)c3F)=O)C2)=O)c(Cl)cccc1Cl N1(C(CSCC)=O)CC2CCC1C2NC(c1cc(C2(C)CC2)on1)=O N1(C(=O)CCCCC(F)F)CCC2(CCN(C(C3CC(CF)C3)=O)C2)C1 C1(CC2(C(=O)NCCN(C(=O)Cc3coc(C(F)F)n3)C)CC2)CC(O)C(O)C1 c1(NC(C2C(NC(C(CC)NC(N)=O)=O)CCO2)=O)cnc(F)nc1 Cc1c(C(=O)NC23CC(NC(C4CCCO4)=O)(C2)C3)ccc(C(C)(C)C)c1O C#Cc1ccc(C(=O)NCC2(C)CCC(NC(C3CC(CF)C3)=O)C2)c(F)c1 c1(C(=O)NCCCC2CCN(C(c3cnccc3Cl)=O)CC2)ncccc1CO C12(C(=O)NCCC(=O)NC3(c4ccncc4)CC3)CC3CCC(CC(C3)C1)C2 C1(C(=O)NC2CCN(C(C3CC(C)(C)C3)=O)CC2)OC2CCC1CC2 N1(C(C(=O)NCCC#N)C2C(C)C2)CCCC(NC(=O)NC(C)(C)C)C1 C1(C(=O)NC2(CNC(c3c(C)c(N)ccc3)=O)CCCC2)CCCCC(C)(C)C1 C(=O)(C1CC(C)(C)C1)N(C(c1ccccc1)C(=O)NC(CC)(C)C)C1CCCC1 CCCC(C)(C)CC(=O)N1CCC(=CCNC(=O)CC2CC(SC)C2)CC1 CCCC(CC)CC(=O)NCc1cc(C2CCN(C(C3CC3CC)=O)CC2)no1 CC1(C)CCN(C(c2c(N)cccc2Cl)=O)CC1NC(c1cccnc1O)=O CC1CCC(NC(c2cnn3ccsc23)=O)CN1C(=O)CC12CC(C1)C2 c1(OC(CC)CNC(C2(C)CCSCC2)=O)cccc(C)c1 c1(C(=O)NC(CC)CC(=O)NC2COC(C)(C)C2)ccc(O)nc1C C(=O)(C1CCOc2ccccc21)NCC1C(NC(CCCN=[N+]=[N-])=O)CCC1 C(CN(C)C(C1CN(CC(C)C)C1)=O)(CO)(CO)NC(COCCC=C)=O C1(C(N(C2C3CCC23)C)=O)CCCCN(C(=O)CSC(F)F)C1 c1(C(N(CC(CNC(CCCCC)=O)(C)C)CC)=O)cc2c(Cl)cc(F)cc2[nH]1 C1(C(=O)NC2C3CN(C(c4cc[nH]c4C(C)C)=O)CC23)(CC)CC(F)(F)C1 C1(C(=O)NC(CNC(CCCC)=O)CC)COCC(=O)N1C(C)C CCC(C)CC(=O)NC(C)(CNC(=O)C=Cc1cnccn1)C1CC1 C(C(=O)NC(c1cnc[nH]1)C)(C(C)(C)C)NC(c1c(C)cc(F)s1)=O N1(C(c2c(OC)ccs2)=O)CCCC2CN(C(c3cnc(C)cn3)=O)CC12 N1(C(C(C2CC2)SC)=O)CCC(C(F)(F)F)C(CNC(=O)Cc2ccno2)C1 O=C(CC1COc2cc(O)ccc21)N1CCC(N(CCO)C(C2CC(O)C2)=O)C1 N1(C(CCCCCOC)=O)CC2(CCCC(CNC(=O)CCSCC(C)C)O2)C1 c1(C(=O)NCC2(NC(C(C(C)C)c3ccc(Cl)cc3)=O)CC2)ccccc1C#N C(=O)(CC(C)CN(C)C)NCCC1N(C(C(C2CCOC2)OC)=O)CCC1 Cc1ncc(CCNC(C2CCC2NC(C2(C3CC3)CC2)=O)=O)o1 c1(OC)ncc(C(N2CC(O)(CCNC(c3ccns3)=O)C2)=O)cn1 C(=O)(CCCC(C)(F)F)N(C)CC1(NC(C(C)CC=Cc2ccccc2)=O)CC1 C1(NC(c2cnc(C)n2C)=O)CCC(C)N(C(c2cc(C(N)=O)cc(F)c2)=O)C1 N1(C(C2C(C)CCS2)=O)C2CCC1CN(C(C1(c3ccn(C)n3)CC1)=O)C2 C(=O)(CC1CCCNc2ccccc21)NC1CC2(CC(C)(C#N)C2)C1 c1(C(=O)NCCCN(C(C(C=CC)O)=O)Cc2cccnc2)ccncc1O N1(C(CCOCCOCC)=O)C(C(=O)NCCc2ncc(C)o2)CCC1C1CC1 C1(NC(Cc2ccc(C)o2)=O)CCCN(C(c2cn(C3CC3)nc2C2CC2)=O)CC1 N1(C(C(C=C)(C)CCOC)=O)CCCC2(CCCN2C(c2coc(C)c2)=O)C1 c1(C(=O)NCC(=C)CCNC(C2CN(C)CC(C)O2)=O)ccc2cn(C)nc2c1 c1(CN2CCN(c3ccc(-c4c(C)ccnc4F)cn3)CC2)cccc2ccnn12 n1(CCC(N2CC(COC)(NC(=O)CC3CCCOC3)C2)=O)nc(C)nc1C C1(CCCC)CN(C(C2CSCN2C(c2ccc(Cl)nc2C)=O)=O)CCN1CC CC(C)C(F)(F)CC(=O)N1CC2CCC1C2NC(=O)CN1CCCCS1(=O)=O N1(C(C2(CC#C)CCOC2)=O)CCC(CNC(=O)Cn2ccnn2)C(F)(F)CC1 C1(C(=O)NCCN(C(c2c(C)csn2)=O)CC2CC2)CC2CCC2C1 CCC(C)CC(=O)NCC(C1CCN(C(=O)C(C)CC2CCCCC2)CC1)C n1(C(C2CCOCC2)CC)cc(CCNC(=O)C(C)Cn2ccc(C)n2)nn1 CC(C)C(CCNC(=O)CCF)NC(c1cnnn1-c1ccc(F)cc1)=O C1(C(=O)NCC(C)CO)CCCCN1C(=O)CN(C)C(c1ccccc1)=O CN1CCN(C(c2coc(C#N)c2)=O)C(CNC(c2n[nH]cc2Br)=O)C1 c1(C(N2CCC(NC(c3nc(C)c(C)s3)=O)CC2)=O)cnc2n1CCS2 C1(CNC(CCCCNC(C)=O)=O)C(C2CC2)CCN1C(=O)CCn1cccc1 CC(C)CC(=O)C(=O)N1CC(CC(F)C(=O)NC2(C)CCCC2C)C1 N1(C(C(C)SCC)=O)CC(C(=O)N(C)CCN(C)CCO)C(C)(C)C1 c1(C(N2CCN(CC)C3CCCC23)C(=O)NCC)ccc2ccc(Br)cc2c1 C(S(=O)(=O)C(F)F)C1(Cc2cn(C3CN(C(CC#N)=O)C3)nn2)CCC1 n1(CCCC)ncc(C(=O)NCC2CCN2C(=O)CC(C)O)c1CC N1(C(C2C(C)N(C)CC2)=O)CCC2(CC(NC(=O)COCCN(C)C)C2)C1 C(C)(CSC)(C(=O)N(CCCSC)C)NC(c1n(CC#C)ccc1)=O CC(CCCc1ccccc1)C(=O)N1CC(NC(C2CC(F)(CO)C2)=O)C(C)C1 C=C=CCC(=O)N1CCC(NC(=O)CCCNC(c2sccc2C)=O)C1 c1(C(=O)NC2(C)CN(C(C3C(C=C)OCC3)=O)C2)ccc(C2CCC2)cc1C C1(CNC(C(C(C)C)OC)=O)CN(C(=O)CSCc2ccncc2)C(C)(C)C1 CCC(C)(C#N)C(=O)NC(CNC(c1cc(O)cc(F)c1)=O)C(C)(C)C N1(C(C2(CC)COC2)=O)CCC2(CC1)CN(C(=O)CC1CCCN1CC)CCO2 c1(C(N2CCCC(CNC(C3C(C)CC(C)O3)=O)C2)=O)cnn2c1C(=O)NCC2 CCCCCC(O)CC(=O)NCC1C2CC1N(C(c1cccc(O)c1[N+](=O)[O-])=O)C2 CC(=O)CC(C)C(=O)NC1CCCN(C(C2CCOCC2)=O)C1 C(c1cn(C)nn1)=CC(=O)NCC1(NC(Cc2c(C)ocn2)=O)CC1 C1(CNC(CCCSCC)=O)CCCN(C(c2ccc(CC)s2)=O)C1 N#CC1CCCC(C(=O)NCCCCCCNC(=O)Cc2ccc(CO)cc2)C1 C12(C(C)OC(c3c(C)oc(C)c3C)=O)CC3CC(CC(C3)C1)C2 C(CC(F)F)(C(=O)NCCCCCC1CC1)NC(c1c[nH]c(=N)o1)=O C1(C)(CNC(CNC(=O)OCC)=O)CCN(C(=O)C#CC(=O)N(C)C)CC1 C12CN(CC1C)C(=O)C(C)(C)c1cn2nn1.C1(C)(NC(C)C)CC1C(F)(F)F c1(NC(c2n(CCCSCC)nnn2)(C2CCOC2)C)nnc2ccccn12 S(=O)(=O)(c1c(Br)cc(F)c(Cl)c1F)NCc1cc2ccc(C)nc2cc1 c1(CNCc2c(O)c(F)ccc2)cccc2c1OCC2 N1(C(c2n[nH]c(C)c2C)=O)CCC(C2CC2)C1CNC(=O)CNS(=O)(=O)N(C)C C1(NC(=O)C=Cc2ccccc2F)CCCC2CN(c3nc(C4CC4)ns3)CC12 O=C1COc2cccc(C(=O)Nc3cccnc3-c3ccccc3)c2N1 C(=O)(C1CC2(CCN(C(C3(C#N)CC34CCC4)=O)C2)Oc2ccccc21)NC c1(C(=O)NCC(CC)N(C)C(c2cnn(C)n2)=O)c(Cl)n[nH]c1C1CC1 c1(C(=O)Nc2cccc(C)c2Cl)[nH]c2ccccc2c1-c1ccc(C#N)c(O)c1 C1(C(N(CC(=O)N(CC)CC)C)=O)C(C)OCCN1C(C1CC2(C1)CC21CC1)=O C(=O)(C(=O)C(C)(C)CC)N1CC(CCC=C)(C(=O)NC2CCCN(C)C2)C1 N1(C(=O)NCC(c2cccc3ccccc23)CC)Cc2ccccc2CCC1C N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CCCN2C(c2cccc(=O)o2)=O)C1 c1(Nc2ccccn2)nccc(=NCCC(C)N(C)Cc2cc(C)c(Br)cc2)[nH]1 C1(C(C(=O)NCCCCNC(=O)C(C)c2ccco2)OCC)CC(F)(F)C1 C1(C(=O)NCCN(CCCN(C)C)C(c2c[nH]nc2C(F)(F)F)=O)CNC(=O)N1 N1(CCNC(N(C2ON=C(C(C)C)C2)C)=O)CCc2ccccc21 c1(C(N2C(C)COCC2C)=O)cc2oc(Br)cc2[nH]1 c1(C(N2CC(NC(=O)Cc3cnccn3)C3C2C3)=O)c[nH]c2cccnc12 c1(OCC(=O)NC)cccc(C(=O)NC23CCN(C2)C(=O)CCO3)c1.C(C)(C)OC CCCC(C(=O)N(C(C(=O)N1CCOCC1)C(C)CC)C)C(C)C C1(O)(CN(C(=O)CNC(=O)CC(F)(F)F)C)CCN(C(=O)C(O)C(F)F)C1 c1(CCC)sc(C(N2CCC(C(C)(C)NC(C3CC3C)=O)CC2)=O)cc1CC c1(CC(C)CNCC(=O)NC(=O)N(C)C)cccc(Br)c1 c1(C(=O)NCC2OCCN(C(CN3CC(=O)NC3=O)=O)C2)cnn2c1OCC2 CC(C)CC(CNC(c1cn(C2COC2)nn1)=O)NC(C1(N(C)C)CCOCC1)=O C(=O)(C(F)(F)C1=CCOCC1)N1CCC(NC(C(CCC)OC)=O)C(CC)C1 C(C(C(=O)NC(C)(C)C(C)O)C(C)(C)C)NC(CCC(=O)NC)=O C12(C(=O)NCC3(CNC(=O)Cn4cc(Cl)cn4)CCC3)CCCCC1OCC2 CCCC(O)CC(=O)NCC1CCCCCN1C(c1cnn(C(C)C)c1N)=O c1(C(N2CC(NC(c3c(C)cnnc3)=O)C(O)C2)=O)ccc2c(c1)NC(=O)C2 C12(c3ccccc3)CCN(CC1)C2=O.c1(CNC(CCC=C)=O)ccnc(C)c1 C(C1OCCc2sc(F)cc21)NC(=NCC)NCC1CCN1CC N1(C(C(CO)N(C)C)=O)CC(CNC(C2CC(=O)CCO2)=O)C(C)(C)C1 CC(C)C(C(=O)NCc1nnnn1C)C(C)NC(=O)C(=O)C(C)C Cc1cc(C)c(S(=O)(=O)Nc2ncc(CC(=O)Nc3ncco3)s2)c(C)c1 C12(CCCCC1)C(=O)NC2.C1(=O)CC(O)CN1.C1(N(C)C)CC(n2cnnc2)C1 c1(C(=O)NC(C2CC(NC(C(C)OCCCC)=O)C2)C)cccc2c1OCC2 N1(C(C23OCC(C(=O)OC)(C2)C3)=O)CCCC2(CCCN2C(C2CC2(F)F)=O)C1 c1(OC)nc(C)c(C(=O)NC2COCCC2NC(C2CCC(=O)N2C)=O)s1 c1(C(N2CC(CC)C(NC(c3scnc3C)=O)CC2)=O)cc2cnn(C)c2s1 C(=O)(CCCC1CCCO1)NC(CCNC(CC1(C(=O)OCC)CC1)=O)C Cc1ccc(Cl)c(C(=O)N(C2CCCCN(C(=O)C#CC3(C)CC3)C2)C)c1 N1(C(C(c2cccc(C)n2)(F)F)=O)CCCCC(CNC(=O)CCC(C)C)CC1 C1(NC(CN(C(COC)=O)C)=O)CN(C(c2ccc[n+]([O-])c2)=O)CC1COC N1(C(Cc2cc(C)nn2C)=O)CC2CCC1C1CN(C(=O)C=CBr)CC21 N1(C(C(C(=O)OCC)F)=O)CCCCC(CNC(c2cc(Cl)ccc2NC)=O)C1 C(c1ccc(F)cc1F)=CC(=O)NC(C)CCCNC(c1ccnn1C)=O c1(C(=O)OC)cn(C)[nH]c1=NC(=O)N(C)Cc1nc(C2CC2)no1 C1(C(=O)NCC(CO)NC(c2csc(SC(F)(F)F)n2)=O)CCCCS1 c1(CNC(c2cnn(C)c2F)c2n(CC)nnn2)cc2ncccc2s1 C=CCC(C(=O)OCC(C)(C)C)NC(=O)C(O)C1CCC1 N1(C(C=CC(C)C)=O)CCC2(NC(c3cc(Cl)c(N)cn3)=O)CC2C1 c1(-c2c(C)c(F)c(F)cc2)ccc(C(N2CC3CCCCC3C2)=O)c2c1OCO2 C1(C(N(C(CC(C)C)C)C2CC2)=O)CCCC12CCN(C(=O)C=CS(C)(=O)=O)CC2 c1(OC)ccc(C(c2nnnn2C2CCC2)NC23CC(F)(C2)C3)cn1 C1(C(N(CCC(F)(F)F)C)=O)CCC2CCC1N2C(c1ccsn1)=O C1(NC(c2snnc2C2CC2)=O)COCCN(C(C23CCCCC2C3)=O)C1 C1(NC(C2CC(n3cc(CCc4nn[nH]n4)nn3)C2)=O)CC2CC3CC(C2)CC1C3 c1(N2C(C(=O)Nc3ccc(C)nc3I)C=CC2)nc(C)c2cc(Br)ccc2n1 Cc1ccc(C(C)NC(c2c[nH]ccc2=O)=O)nc1 C(=O)(CC1COc2ccccc21)NCC1(NC(c2c(C)cnn2C)=O)CCC1 C=C(C)C(CC(=O)NC1CCCC(NC(=O)C=C2CCCCC2(C)C)C1)OCC C(=O)(C1OCCc2ccccc21)NCCC(C)N(C)C(C1CC2CC1C2)=O C(=O)(C(C)CCOC)NC(C(CO)NC(c1c(CC)ncs1)=O)C c1(C(=O)NCC2(C)CCC(NC(=O)C#CC3CC3)C2)ncc2ccccn12 C1(C(=O)NCCC2CCOC2)(CC)CCCN(C(=O)CC2CCCC2)C1 C(=O)(C(O)(C(C)C)C(F)(F)F)N1CCC(NC(c2csc(C)c2C)=O)C(C)(C)C1 C1(C(N2CC(C(C(=O)O)OC)C2)=O)CCC(=O)N(C)C1 C#CC1CC2CCC1N(C(c1cc(C3CC3)on1)C(=O)NC(C)(C)CC)C2 N1(C(c2c(F)ccc(C#C)c2)=O)CC2CCN(C(C3CC(=C)C3)=O)C2C1 NC1c2ccccc2CC1C(=O)NCc1nnc(-c2ncc(Br)cn2)o1 C=Cn1nccc1C(=O)NCC=CCNC(=O)C=Cc1ccc(Br)s1 C1(C)(CC)CCCN(C(=O)CC=CCNC(=O)Cc2nccn2C)C1 c1(OC)cc(C(=O)NC2CCN(C(C34CCC3CC4)=O)CC2C)c(F)c(Cl)c1 N1(C(c2cc(C)ncn2)=O)CCC2(CC2NC(=O)C(C)Sc2ccccn2)C1 c1(C(=O)Nc2cc(C)no2)cc2ccc(C3=CCOC3)nc2[nH]1 C(=O)(CC(CNC=O)CC(C)C)N1CC(OC)(CNC(c2ccc(Cl)cc2)=O)C1 CC(C)C(O)C(C)C(=O)N1CCCC(C)(C)C1C(=O)NCC(O)C(C)(C)C N1(C(CC2CCCC(C)C2)=O)CCC(F)(C(=O)NC2(C)CCCC2O)CC1 CC(CCC(C)(C)C)C(=O)NCC1CCN1C(c1ccc2c(c1O)CCC2)=O C1(CNC(Cc2cn(C)nc2)=O)CCN(C(c2ccnc(CO)n2)=O)CC1(F)F N1(C(=O)CCCN2CCOC2=O)CC(C2CN(C(=O)CC3COCC3O)C2)C1 c1(CC(=O)NCCN(C(c2csc(Cl)c2)=O)C2CC2)coc2ccccc12 CCC(CC)C(F)C(=O)NCCC1CC(NC(=O)CCc2ccccc2F)C1 c1(C(=O)NC2CCCN(C(=O)Cn3ccnn3)CC2)cc(Cl)cc2c1CCC2 C1(NC(=O)CC2COCC2O)CCOCC1NC(c1cscc1Cl)=O CC1=C(C(=O)N2CCC(C(=O)NC3CCN(C)CC3C)CC2)SCCO1 CC(C)C(C)C(CNC(c1cc(O)n(C)n1)=O)NC(c1cn2c(n1)SCC2)=O CCN=c1[nH]c(C)c(C(=O)N(C2CCC(CNC(C3CCC(F)C3)=O)CC2)C)s1 C(=O)(CCCC(=O)NC(C)CNC(=O)CN1CCCCC1)NCCC c1(OC)ccc(F)c(C(N2CCN(C(=O)CCF)CC2C)=O)c1OC c1(C(=O)OCc2csc(CC3CCCC3)n2)cc(O)cc(Cl)c1Cl N1(C(c2cn(CCOC)nc2)=O)CCOCC(NC(c2cnc(C(F)F)s2)=O)C1 c1(C(N2C(C)(C(=O)Nc3c(NC(C)=O)cccc3)CC2)=O)ccn2cncc2c1 N1(C(c2cc(C(C)C)on2)=O)CCC2(C1)CN(C(c1cnncc1O)=O)CCO2 C1(NC(C2C(C#N)C2)=O)CCCOC1C1CCN(C(=O)COC2CCCC2)CC1 N1(c2c(C)cncn2)CC2CC(NC(=O)C3=NOCC3)CC1C2 c1(CC(=O)N(CC(C)NC(C2CC2(C)C(C)C)=O)CC)ccc(OC)cn1 c1(CNC(C2ON=C(C)C2)=O)c(C)noc1C1CC1 n1(CC)ncc(C(N2CCCC(CCNC(=O)Cc3cncnc3O)C2)=O)c1Cl CC1CCC(CC(=O)NCC2(CNC(c3cnc(C4CC4)s3)=O)CCCC2)O1 CC(C)(C)CC(O)C(=O)NC1CCC1C(N1CCCC(O)(C(N)=O)C1)=O CCC(CC)C(C(=O)NC1CC(F)CN(C(c2coc(C)n2)=O)C1)OC C1(C(=O)NC2C(OC)CN(C(CN(CCC)C)=O)C2)CCc2nn(C)cc2C1 c1(OC)cc(O)ncc1C(N1CCC(CO)(NC(=O)CSc2nc[nH]n2)C1)=O C=CCC(CC)C(=O)NCc1cc(C)c(C(N2CCCC2C(O)CC)=O)o1 c1(C(N(CC(CN(C(CC2C(C)CCC2)=O)C)O)C)=O)cc(C2CC2)ccn1 c1(C(=O)NCC2CN(C(CC(C=C)C)=O)CC23CC3)occ2c1CCOC2 CCC(CCCC(=O)N(CC(C)(F)F)C)NC(c1cc(CO)n(C)n1)=O CC1(C)OC(C)(C)C1C(=O)NCCNC(c1cnoc1C1CC1)=O c1(SCC)ccc(Cl)cc1C(=O)NCCCNC(c1cc(C#N)no1)=O C1(C(N2CC(C)(NC(c3coc(C4CC4)n3)=O)C2)=O)CC(C2CC2)C1 C1(F)(C(=O)NC(C)CC2CN(C(c3csc(S)n3)=O)C2)CCC(F)(F)CC1 C1(C)(C(=O)NCC(C(C)(C)C)NC(c2cn(C3CC3)nn2)=O)CCCNS1(=O)=O C1(C(=O)NCCC(C)NC(C2(COC)CCC2)=O)CCC(N=[N+]=[N-])C1 Cc1ccc(Br)c(CC(=O)NCC2CCC(=O)NC2)c1 C(=O)(CC(=O)N1CCCC1C(C)(C)NC(C1CNC(=O)N1)=O)NC C1(C(N(CC(C(=O)NC)C)C)=O)CC12CCN(C(C1CCCC(O)C1)=O)C2 C(=O)(CCCC(C)(C)C#N)NC1(C(N(CCCCC=C)C)=O)CC1C c1(C(=O)NCC2(F)CC(NC(CC=C)=O)C2)cc2cc(C)ccc2nc1C CCC(O)(CC)CCNC(=O)NC1CCC(C(=O)OC)O1 C1(C(N(CCCOCCN(C(c2nc(C)oc2C)=O)C)C)=O)CCCC(C)CC1 c1(N2CCC(NC(c3c(CC)csc3)=O)C(C)C2)ccc([N+](=O)[O-])cc1C(C)=O C1(NC(C2CCCCC2(F)F)=O)CC2CCC(C1)N2S(=O)(=O)c1cccs1 N1(C(c2c(N)nccn2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C(C2CCC2)C1 N1(c2c(C)c(O)ncn2)CCC2CCC(C1)N2C(=O)CCCCN(C)C C12(CC(=O)NC3CN(c4n(C)nnn4)CC3(C)C)CC3CC(CC(C3)C1)C2 C1(NC(Cc2cc(C)no2)=O)CC1C1CCCN(C(C2CC3(C2)CC3F)=O)C1 c1(C(CNC(CC2(C#N)CC2)=O)NC(C2CC2(F)F)=O)cc(F)cc(Cl)c1 S(=O)(=O)(c1ccc(F)cc1Cl)NC1CCC(NC(c2ccc(C)c(Br)c2)=O)C1 c1(C(=O)NCCC(C)N(C(=O)C(C)C#N)C)cccc2scnc12 Cc1c(CC(=O)NOCCCCC(=O)NC2CCC2C)cnn1C C(=O)(CCN1C(=O)CCc2ccccc21)N(CCC)CCNC(C1CC(O)C1)=O Cc1ncc2ccccc2c1C(=O)NC1CC(C)CN(C(C2(C#N)CCC2)=O)C1 Cc1ccc(C)c2c(C)c(C(N3CCCN(C(=O)C=CS(C)=O)C(C)C3)=O)oc12 c1(-c2cc(CN3CCCC(N(C(C)=O)CC)C3)sc2)ccc(O)c(OCC)c1 c1(C(=O)NCC2C(NC(CN(CCCCCC)C)=O)C2)c(Cl)ccc(F)c1C N1(C(C(C#C)(C)C)=O)CC2(C1)OC1(C)CC2(NC(c2ccn3ncnc3c2)=O)C1 c1(C(=O)NC(C)(C)CCCNC(=O)Cc2ccc(O)cn2)cnc2[nH]cnc2c1 Cc1cc(C(N2CCN(C(c3ncccc3C)=O)CC23CC3)=O)cc(C)c1O C#CCC(CC)NC(=O)C(C1(O)CN(C(=O)C(C)c2cccs2)C1)F c1(C(=O)NC(CCNC(C(CC)F)=O)C(C)C)ccc2nc(N(C)C)sc2c1 C(=O)(CC(C)NC(c1c[nH]nc1OC)=O)N(CC(C)C#N)CC Cc1cn(CC(=O)NC2(C)CC(NC(C3CCS(=O)(=O)C3)=O)C2)c(=O)nc1O C(=O)(CC(C)(O)C(F)(F)F)N(C1CN(C(c2cnc(C(C)(C)CF)o2)=O)C1)C CC1CCC(C2CCC2)CN1C(=O)C(=O)Nc1ccc(S(C)=O)cc1 C1(CNC(C(C)C2CC2)=O)CCN(C(=O)C=Cc2cccc(F)c2)C12CCC2 C1(C(=O)NCC(C(C)O)(C)C)CC2(CCN(C(C3CN(C(C)C)C3)=O)C2)C1 N1(C(CC(=C)C)=O)CCC(CO)C(NC(c2cnc(CC)s2)=O)C1 N1(C(CN2C(C(=O)OC(C)(C)C)CCC2)=O)CCC(C)(C2CC2)C1 c1(OCC)cccc2c1OCC(C(=O)NC1CCCC(NC(=O)C=CSC)C1)C2 C1(CC#C)CCNCC1.c1(OCCN(C=O)C)ccccc1C(C)C c1(C(N2C(CNC(c3c(C)nc[nH]3)=O)CC2)=O)cnn(CC(C)(C)O)c1C N1(C(C(c2ccc(Cl)s2)C)=O)CCN(CC2CN(C(C3CC3(C)C)=O)C2)CC1 CCS(=O)c1ccccc1C(=O)NCC1CC(F)CN1C(=O)CN1CC2CC2C1 c1(C(N2CCCC(F)(CNC(CC(C)OC)=O)C2)=O)cc2cc(F)ccc2cn1 C1(C)(C(=O)NCC(CC=C)NC(CC2(CSC)CC2)=O)CCC(=O)N(C)C1 C(CCCCCNC(=O)COC1CCCCC1C)N(C(c1c(C)occ1)=O)C c1(C(N2C(CN(C(c3c(C)nc(C)o3)=O)C)CCC2)=O)cc(Cl)n[nH]c1=N CC(CNC(C1CCC(C)C(C)C1)=O)N=c1[nH]nc(C(C)(C)C)o1 C1(CNS(CC(=O)OC)(=O)=O)CN(C(C2(c3cc(C)no3)CC2)=O)CC1(C)C N1(C(COC2CN(C(C)=O)C2)=O)CC2CC(C1)N(C(C1CC1F)=O)C2 CC#CCCC(=O)NC(CC(C)C)C(=O)NC(C)C(C)(C1CC1)OC Cc1[nH]c2c(C(=O)N(c3ncncc3I)CC3CCCN3)cccc2c1C N1(C(C(C)OCCOCC)=O)CC2(CC(NC(=O)Cc3coc(C)n3)C2)C1 CC(O)CC(C)(C)CNC(c1ccc(CNC(C2COCC2C(N)=O)=O)s1)=O C1(O)(CNC(CN(CC)CC)=O)CCN(C(=O)Cn2cccc(N)c2=O)CC1 C(=O)(CCS(C)=O)NCC(C(C)C)NC(c1n(C(C)C)ncn1)=O Cc1coc(C(=O)NC(C)CC(C)NC(c2ccc(N(C)C(C)C)cc2)=O)c1C N1(C(c2cc(F)c[nH]2)=O)CC2OCCN(C(c3cc4cccc(F)c4o3)=O)C2C1 Cc1cc(C(N2CC(NC(c3cnnn3C)=O)CC(C)C2)=O)c(F)cc1Cl c1(NC(C2(CNC(C(C(COC)C)C)=O)CC(C)(C)C2)=O)cncc([N+](=O)[O-])c1 c1(CNC(CC2(C(=O)OCC)CCC2)=O)ccccc1CNC(c1cc[nH]n1)=O N1(C(c2cc(C)nc(O)c2)=O)CC2(CCN(C(c3ccoc3Br)=O)CC2)C1 N1(C(CC2CC(=C)C2)=O)CC=CC1(C(=O)NCCn1cnc(CO)c1)COC C12(NC(CCCCOC)=O)CCN(C(=O)C(=Cc3cscn3)F)CC1C2 c1(C(=O)NCC23CC(NC(CCOCCOC)=O)(C2)C3)cc(C(C)C)ccc1O N1(C(C2(F)C(C)C2)=O)CCC(c2cccc(C(F)(F)F)c2)CC1 CC1=NOC2(C1)CC(C(=O)NC1CCN(C(C3CCC(=O)O3)=O)C1C)C2 C1(NC(c2c(N)n(CCO)nc2)=O)CS(=O)(=O)CC1NC(C1CCCC1O)=O c1(COC)nc(NCc2ccoc2C)cc(N(C)Cc2ncc[nH]2)n1 c1(CCC(=O)N(C(CNC(C2CCCC2)=O)C2CC2)C)cc(F)ccc1C(F)(F)F C(CC(CC)(CC)NC(C1CC1C(F)(F)F)=O)NC(COCCN(C)C)=O C1(F)(CNC(=O)CC2(c3ccon3)CC2)CC(CNC(=O)Cn2cnnn2)C1 C#Cc1cc(C(=O)N(C2CCN(C(=O)C=COCC)C2)C)ccc1C Cc1ccc(Cl)c(S(=O)(=O)Nc2ccc(C3CCC(=O)N3)cc2)c1Cl C(C(CC(=O)NCC(CNC(c1cc(N)ccc1O)=O)CO)C(F)(F)F)N(C)C C1(C(C(=O)N2CC(Cn3cc(CCC=C)nn3)C2)(C)C)CCC(C(C)(C)C)CC1 C1(NC(C2CC(C3CCC3)C2)=O)CC(F)CN(C(=O)CC2CC(F)(F)C2)C1 C1(NC(CC(=O)NC2CC2)=O)CC(=O)N(C2CN(C(=O)C(=O)NC3CC3)C2)C1 C(=O)(C(C)CCCC(C)C)NC1CCN(C(c2ccc(C)o2)=O)C(C)C1 C1(NC(CN(C)C(C2CC(=O)OC2(C)C)=O)=O)CCC(=O)NC1=O C1(C(N2CC(NC(CCCN(C(C)=O)C)=O)C2)=O)CCC2(CC1)OCCO2 CS(=O)(=O)C1CCCCN(C(=NCC2CC2)NCc2ccn(CCF)n2)C1 c1(N2CCC(CCC)C2)nc(N2CC3CC(C2)N(C)C3)c2ncn(C)c2n1 N1(C(C2CCCN2C(=O)CSc2ccccc2)=O)CCC(O)C1CO C1(CNC(COC2(C)CCCC2)=O)(CO)CCN(C(=O)CCc2cccnc2)C1 C1(N(C(CSCCOC)=O)CCO)CCN(C(C2(C)CC=CC2)=O)C1 c1(COC(C2C(CC)CC2)=O)c2cc(Br)ccc2nn1C c1(CC(N2CC(CNC(C3(CC#C)CC3)=O)OCC2)=O)c(Cl)cccc1Cl C1(C)(C(=O)NC(C)CN(C(=O)CNC(=O)OC(C)(C)C)C)CCC(=O)C1 c1(N(C)C)ccc(NC(=O)NC2(CO)COC(C)(C)C2)cc1Cl C1(CC)C(C(N2CCC(NC(N)=O)CC2)=O)CCN1C(=O)Cn1nccc1C c1(CC)cccc(C(=O)NC2CCC(N(C(=O)CC3C4(CC4)C34CC4)C)CC2)c1 c1(C(=O)NC2CC(C(=O)NC(C)C(N)=O)C2)ccccc1Cl C(C(CNC(=O)CC1CC1(Cl)Cl)C(F)(F)F)NC(Cc1cc(C)nn1C)=O c1(COC2CCN(C)CC2)cnn2c1CN(C(=O)C(Cl)=CCl)CC2 C1(NC(C)=O)CC(CNC(=O)C2=CSCS2)C1(C)C CCC(C)C(CC(=O)N(C(C)CC(=O)OC)C)NC(=O)Cn1ncn(C)c1=O c1(CC(=O)N(C2CSC2)CC#C)c(C)ncnc1C N1(C(c2cccc(N(C)C)n2)=O)CCOCC(NC(=O)CC2CCCCCC2)C1 C1(NC(CCCC2C(C)C2)=O)CCC(C)N(C(=O)CCOCC(F)(F)C(F)F)C1 C1(C)(C(=O)NCCn2cc(CNC(C(C)=CC)=O)nn2)COC(=O)C1 N1(C(c2c(C)c[nH]n2)=O)CCS(=O)(=O)C(CCNC(=O)CCOC2CC2)C1 c1(OC)c(C)ccc(C(=O)NC(C)(CNC(=O)Cc2cnc[nH]2)C(C)C)c1F Cc1c(F)ccc(CN2CC3CC3(C(=O)Nc3cc(Br)cnc3O)C2)c1F c1(OC)cccc(C(N2CC3CC(NC(c4ccoc4Cl)=O)C2C3)=O)c1N C(=O)(CC(O)CC(C)C)N1CCC(C(=O)NC(c2nn[nH]n2)CC)(CC)C1 C1(CCNC(=O)C(=O)NC(=O)OCC)NC(=O)N(c2cccc(CO)c2)C1=O C(=O)(C1CCCc2nn[nH]c21)NC1C2CN(Cc3cnn4ccn(C)c43)CC21 C1(O)(CCNC(c2c(CC)con2)=O)CCN(C(=O)Cn2nnc(C)n2)C1 N1(C(Cc2cc(=N)[nH]cc2)=O)CCC(NC(=O)COC2CCCCC2)C(F)C1 C(=O)(C(CC(C)(C)C)NC(=O)CC1CCCC2CC12)NCC(N(OC)C)=O C1(NC(N2CC(c3c(C)nccn3)C2)=O)CC2CC(CC3CC3)C1C2 Cc1ccc2c(C(=O)NCC3(C)CCN(C(C4CNC(=O)C4)=O)C3)coc2c1 CC(CC(=O)N1CC(CCNC(c2n[nH]c3c2CC(C)CC3)=O)C1)CC(F)(F)F C(C(C)(C)CC(=O)NCC(N1CCN(C)CC1)(C)C)N(C)C(=O)OC(C)(C)C N1(C(C2N(C)CCN(C(=O)CCC3CCCCC3)C2)=O)CCC2(CCCN2C)C1 C1(NC(=O)Cc2nc3c([nH]2)CCCC3)CCN(C(C2(Cl)CC2)=O)CCC1CO C(C(N=[N+]=[N-])C(=O)NCC1(NC(C2CNC(=O)CC2C)=O)CC1)OCC c1(C(N2CC(CNC(c3cccc(C#C)c3F)=O)C2)=O)c(F)c(F)cc(F)c1F CC(=O)C(C)(C)CC(=O)NC1CCOCC1C(N1CCC(F)(F)CC1)=O c1(NC(C2(NC(c3ccccc3F)=O)CC(O)C2)=O)ccc2c(c1)OCC2 Nc1cc(C(=O)NC2CCN(C(C3(C4CC4)CCC3)=O)C2)cc(Cl)n1 Cc1cc(C(=O)NCC2(C3CC3)CC2)ccc1C#N.C12CCCC1NC2=O C(C(CC(=O)N1CCCCC1CNC(=O)CC(C)(C)C#N)C(F)F)N(C)C1CC1 C(C(=O)NC(C)(CNC(C1CN(S(C)(=O)=O)C1)=O)C1CC1)(C(C)C)SC Cc1nc2ccccc2nc1NC(=O)CC1COCCN1C(C1CCSCC1)=O N1(C(c2ncc(C)c(Cl)c2)=O)CCCC2(CCCN2C(C2CC(=O)N(O)C2)=O)C1 n1(CC(=O)NCCN(C(=O)CC23CC(C2)C3)CC)c(O)nnc1O [N-]=[N+]=NC1CC(C(=O)OCc2ccccc2)N(CC2CCCC23CC3)C1 N1(C(=O)NCC2C(OCC)COC2)CCCC(OCc2ccccc2)C1CC Cc1cnn(CC(N2CC(NC(=O)C(F)(F)C3(O)CCCC3)C2)=O)c1 N1(C(c2n(C)cc(C#N)c2)=O)CCC(C2(NC(=O)CC=C(Cl)Cl)CC2)C1 C12(NC(Cc3cn(CC)nn3)=O)CCCC1(F)CN(C(C1(SC)CCC1)=O)C2 c1(C(N2CC(CCCNC(=O)C(=O)C3CCCC3)OCC2)=O)ccc(F)cc1F c1(OC)cc(NC(C2(F)CCN(Cc3c(Br)ccnc3Br)C2)=O)c(C)cc1Br c1(NC(C2CC(O)CN2S(=O)(=O)CC2CC2)=O)cc(Cl)c(Br)c(Cl)c1 c1(N2CCC(CCOC)(NC(=O)CNC(C)=O)CC2)ncnc(C)c1C#N CCC1=NOC(CC(=O)NC(C)(C)C(C)NC(c2ccncc2OC)=O)C1 CCCC(CC)C(=O)NC1(CNC(c2cnoc2C)=O)CCCCC1 N1(C(C2C3(CC(NC(C(C)NC(C)=O)=O)C3)C2)=O)CCCCC(F)(F)C1 Cc1cc(F)c(CC(=O)Nc2cccc(NC(=O)C3=CCSC3)c2)cc1F c1(C(N(C(C)C)CCN(C(=O)C(c2cncn2C)O)C)=O)cn2ccncc2n1 C=CCC(C)(C(=O)NCC1CCN1C(=O)CCCc1ccc(C)s1)N(C)C N1(C(c2cc(OCC)n[nH]2)=O)CC(=O)CCC1C(N1CCCCC1CF)=O c1(-n2cc(CCN(C(C3(O)CCC3)=O)CC)nn2)c(NC)n(C)c(=O)n(C)c1=O C1(NC(CN2CCC(C)CC2)=O)CCC12CCN(C(C1CCS(=O)CC1)=O)CC2 CCCCC(O)C(=O)N1CCC1CNC(c1ccc(Cn2ccnc2)o1)=O C(c1cncn1C)=CC(=O)NCCN(C(c1ccc(CCCCC)o1)=O)C CCCCCC(F)C(=O)NCc1cc(C(=O)NC2(CC(=O)OCC)CC2)n[nH]1 n1(CC)ncc(Br)c1C(=O)NC(C)CN(C(=O)COC1CCCC(C)C1)C C1(C(=O)NCCC(C)(O)C2CC2)C2CN(C(=O)CC3CCOC3=O)CC12 O=C(N=c1ccc(SCc2ccccc2)n[nH]1)NC1CC2COCC12 c1(C(=O)NCCC2(O)CN(c3nnc(C(C)C)s3)C2)ccc2nsnc2c1 Cc1cc(C(N2CC(NC(c3ccncn3)=O)C(C(F)(F)F)C2)=O)sc1C c1(NC(C)C(=O)NC2CC(CNC(=O)CCn3ccnn3)C2)ccc(C#N)cc1 Cn1cc(C(=O)NCC23CC2CN(C(=O)COc2ccc(Cl)cc2)C3)ncc1=O N1(C(CCNC(=O)OCC)=O)CCC2(CNC(c3cnn[nH]3)=O)CCCCC12 c1(C(C)OCC)ccccc1-c1nc(-c2ccc(C(F)F)nc2)no1 C(=O)(CCCC(C)(C)C)N(CC(=O)NCC1CC1Cl)C CCCC(C)(C)C(=O)NCC1CCCCC1C(N1CCC2(CC1)N=N2)=O c1(CSC2C(CC)COC2)ccc(N)cc1.C1CCCCO1 c1(C(C)=O)ccccc1C(N1CCC(N(C)C(C2(C)C=CCCC2)=O)C1)=O Cn1nc(C(=O)NCC2(CCNC(C34CCC3CC4)=O)CC2)c2c1CCC2 C1(C(N2C(C(=O)NCCC(C)N(CCC)C)CC=CC2)=O)CC2CC(=O)C1O2 C1(C(C(=O)N(CCC(C)(C)C)CC=C)=O)CCOCC1OCC Cc1nc2cccc(C(N3CC(C(F)Cn4cc(C5CCCO5)nn4)C3)=O)n2n1 C1(F)(CNC(C2(C)C(C(=O)OC)C2)=O)CCN(C(C2CCCC2O)=O)CC1 c1(C(N2CC3=C(CN(C(Cc4cc(CC)no4)=O)C3)C2)=O)cnc2n1CCC(C)C2 c1(C(=O)NC2C(OCC)CN(C(COC(CC)C)=O)C2)cnn2c1NCC(C)C2 CC1CC(=O)NC1C(N1CCC(NC(c2cc(-c3ccn(C)n3)on2)=O)CC1)=O c1(C(=O)NCCC(=O)OC)ccc2[nH]ccc2c1.C1=CC(=O)N2C1CCC2 N1(C(C(C)Cc2ccnn2C)=O)CCC2CN(C(C3(Cl)CC3)=O)CC2CC1 c1(CNC(N(C(c2cccnc2)C(C)C)CC)=O)cc2c(nc1O)CCCC2 c1(C(=O)Nc2cccc(-n3ncc4ncccc34)c2)cc([N+](=O)[O-])cc(C)c1Cl C(=O)(CC(C)C(F)(F)F)N1CCC(CCOC)(NC(C2CCC2C)=O)C1 N1(C(c2c(C#C)cnn2C)=O)CCCC(C2(NC(C3CCS3(=O)=O)=O)CC2)C1 c1(C(=O)NC(CCCCNC(C(CC)CCOC)=O)C)cnc2c(c1)COCC2 c1(OC)cc(C)cnc1C(N1CCCN(C(C2CC(C)CC(C)C2)=O)CC1)=O N1(CC2(CC(=C)C)N=N2)CCCC(C(F)(F)F)(CC2CC2)C1 C1(CC)CC(C(=O)NCC(C)CN(C(=O)CCn2ncn(C)c2=O)C)CC(=O)N1 C1(CC)CCN(C(c2coc(CNC(c3scc(C)c3C)=O)n2)=O)C1C C1(NC(=O)C=CC2CCC2)CCCCN(C(c2scnc2C2CC2)=O)C1 N1(C(c2cc(C)[nH]c2C)=O)CCOC(C)C1C(N1CC(Cn2ccnn2)C1)=O N1(CC=CC(=O)NC(C2CCN(C(C(COC)C)=O)C2)(C)C)CCN(C)CC1 O=C1CCC(S(=O)(=O)N2CCCCC2C(N2C3CCC2CC(O)C3)=O)CC1 N1(C(c2ccc(C#C)o2)=O)CCCC(C(=O)NCC2CCCCO2)CC1 O=C1CC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)CN2CCSCC2)CN1 c1(CC)cc(C(=O)N(CC(O)CN(C)C(c2cncnc2)=O)C)cc(Cl)c1 c1(C(=O)OC)n[nH]c2c1CCN(C(c1ccc(-c3coc(O)n3)cc1)=O)C2 C1(N(C=O)CC2(c3cccs3)CCCCC2)CCC2(CCOCC2)CO1 c1(CCNC(c2n(C(C)(C)C)nnn2)C2(CS(C)(=O)=O)CC2)ccc(Cl)c(F)c1 C1(CNC(C(N2CCC(C(=O)NC)CC2)=O)=O)CC(c2ccc(C)cc2)=NO1 C1(C(=O)NC(CNC(Cc2cc(OC)no2)=O)CO)Cc2ccccc2C(=O)O1 C(=O)(C1=CC2(CCN(C(=O)CN3CCN(C)CC3)C2)C1)NC(CCCC)C C1(CC(=O)NC2(CCC=C)CC2)CN(C(=O)C(C)C2CCCO2)CCO1 N1(C(c2n(CC)nnc2C)=O)CCCN(C(=O)CP(C)(C)=O)CC1C C1(CC(=O)NC(C(C)NC(=O)CCCNC(N)=O)CO)CCC(C)(C)O1 CC(C(O)C(=O)NCCCN(C(=O)Cn1nccn1)CCO)c1ccccc1 C1(CC(NOCCC)=O)CC(NC(=O)C(O)C2CC2)C1(C)C N1(C(C2CC(C(C)C)C2)=O)CCN(C(C2CN(C(N)=O)C2)=O)C(C(C)(C)C)C1 C1(C(=O)NCCSCC(=O)NC(C2CCCCO2)(C)C)CC(=O)NC1=O C(=O)(C1=CS(=O)CCC1)N1CCC(NC(c2occ(OC)c(=O)c2)=O)C(F)C1 S(=O)(=O)(c1ccc(N2CCC(c3nc(C)no3)C2)c(Cl)c1)NCC(C)SC CCC(Cc1cccc(C)c1)C(=O)NC1CC1NC(c1ccc(SC)cc1)=O C1(C(=O)NC(CNC(C2(CC)COC2)=O)C)COCCN1CC1CCCC1 N1(C(CN(C2CCC2)C)=O)CCC(F)(CNC(c2coc(Cl)n2)=O)C1 C1(CC(=O)N(CC(C)(C)CNC(CCc2cnc(C)s2)=O)CCO)CCCC12CC2 Cc1nc(C)n(CC2CCCCN2C(=O)CC2CCCN(C(C)C)C2)n1 C1(c2cccnc2)(C(=O)NC2CC(NC(C3C4COCC34)=O)C2)CC(F)(F)C1 C1(NC(C(COC)OC)=O)CCC2(CC1)CN(C(c1ccccc1C)=O)CCO2 N1(C(CN(CC)CC)=O)CCC(C(=O)NC(C)CCCCO)(CC)C1 c1(C(=O)NC2C3CN(C(CCC(C)(C)OC)=O)CC32)c(F)ccc(Cl)c1N c1(OC(C)C)ncc(C(C)Nc2cc(-c3cccnc3F)ccc2C)cc1Cl C1(C(=O)Nc2cccc(CO)c2)(OC)CCN(C(=O)C=Cc2nc(C)co2)C1 N1(C(C2C(C)CCOC2)=O)CCC(C)(C(N2CCC2CC2CC2)=O)CC1 N1(C(C2CC(=C)C2)=O)CCCC1(C(=O)N(CCS(C)(=O)=O)C)CC Cc1ocnc1C(c1nnnn1Cc1cccs1)NCCc1ccc(Cl)s1 c1(C(N2CC(NC(C=C(C)C(C)C)=O)C(O)C2)=O)cn2cc(Cl)cc(Cl)c2n1 n1(CC(N)=O)ccc(=NC(=O)C2(CCNC(=O)Cn3nccn3)CCCCC2)[nH]1 C1(C(=O)NCC2CC(CF)C2)C=CCN(C(c2ncc[nH]2)=O)C1 C1(C(N2CCCC(NC(=O)CCSc3ncccn3)C2)=O)CCCC12OCCO2 C#CC1CN(C(=O)C(CC=C)C(C)C)CCN1C(c1ccnn1CCF)=O c1(OC)cc(C(=O)NC2CC(C)N(C(=O)CCn3cncn3)C2)cnc1C C1(C(N2CC(=C)C2)=O)CC(O)CN1C(=O)COCC1CCCO1 C1(NC(CN(C)CCNC(=O)C=CS(C)=O)=O)CCCCC1Cc1ccccc1 C(=O)(C1=C(Cl)CCC(C)C1)N1C(CCNC(CNS(CC)(=O)=O)=O)CCC1 N1(C(C2OCCN(C)C2)=O)CC(NC(=O)Cc2cccc(O)c2F)CC12CCC2 C1(C(=O)Nc2c(C)cccc2)CC2(CC2)CN1C(=O)CC1CCCOC1 Cc1n[nH]c(C)c1C(=O)NCC(C)CC(=O)NC1(C)CC(C)(C)C1 c1(C(N(C2CC(NC(C3(C)CCCO3)=O)C2)C)=O)cn(C)c(C(F)F)n1 C(=O)(CCC(=O)NN(C)C)NC1CC2(C(C(N(C(C(C)SC)C)C)=O)C2)C1 C1(CNC(C2CCS(=O)(=O)C2)=O)CCC2(CCC2)CN1C(=O)COCCF C1(CC)CCCN(C(=O)C(C)OCCC(C)C)C1C(=O)NCc1ccncc1C c1(C(C(=O)NC(C(C)NC(c2c(CCC)nns2)=O)C)(F)F)ccc(F)cc1 Cc1coc2ccc(C(N3CC(NC(=O)C(O)CC(N)=O)CC3CO)=O)cc12 C(=O)(CC(O)C(C)C)NC(C(=O)NC1C(SC)COC1)c1ccoc1 N1(C(C(CSC)C)=O)C(C(=O)NCc2ccc(Cl)cc2)CC2CCCC12 C1(C(=O)NC2CN(C)C2)C2CC1N(C(c1cccnc1Br)=O)C2 c1(C(=O)NCCN(C(C2CCN(C)CC2)=O)CC)ccc(OC2CCCC2)cn1 C1(CC(=O)NCCCCN(C(c2c(C(C)C)nn(C)c2)=O)C)CCC2(CCC2)O1 N1(C(c2ccc(=N)[nH]n2)=O)CCN(C(=O)C(=O)NCC(F)F)C2CCCCC12 C1(N(C(=O)CC2CC(F)C2)CC)CCCN(C(=O)COC(C)(C)C(F)(F)F)CC1 CCC(C)(C)CCCC(=O)N1CCC(=CCNC(C2CC2F)=O)CC1 Cc1c(O)ccc(C(=O)Nc2ccc(NC(C3CCCC(O)C3)=O)cc2)c1C C1(CNC(C(c2cccc(Cl)c2)OC)=O)CC2CC2N1C(=O)C(C)(F)F C#Cc1ccc(Cl)cc1NC(=O)C(C)(C)CN(CCCCC)C Cc1ccc(C)c(CNC(c2n[nH]cc2NC(c2ccccc2C2CC2)=O)=O)c1 C1(c2cccc(CC=C)c2)NC(=O)N(CCF)C(C)=C1C(=O)N(C)C C(C(C(=O)OC)N(C)C)OC.C1(CC)C(=O)NCC(=O)N1C Cc1cccc([N+](=O)[O-])c1C(N1CCN(C(C2CC2C(F)(F)F)=O)C(CO)C1)=O S(=O)(=O)(c1ccc(C(=O)NC23CC(C2)N(C(=O)CC(C)COC)C3)cc1)NC C1(C(=O)NCc2nc(CNC(C3CC(OC)C3)=O)sc2)CC(C2CCC2)C1 c1(C(C)C)c(N2CCCCC(NC(C3(c4cccnc4)CC3)=O)C2)ncnc1Cl C1(CCNC(CCCNC(c2cnccn2)=O)=O)CSCCN1C(=O)CSCC N1(C(C(C2CCN(C(C(C(=O)OCC)(C)F)=O)CC2)C)=O)CC2CC(C1)C2(C)C N1(C(CCC=CC)=O)CCC(C)C(CNC(C2(CO)CCOCC2)=O)C1 CC(C)CCC(F)C(=O)N1CCC(C(=O)NCC2CC3C=CC2O3)C12CC2 C1(C(=O)NCCN(C(c2cnc(C)n2C)=O)CC)CCC(=O)CC1C N1(C(CC=CC)=O)CC(NC(C2CC(=O)N(CCOC)C2)=O)C(O)C1 C(c1ccc(SC)cc1)=CC(=O)NC1CN(C(c2cnc(OCC)s2)=O)CC1O c1(NS(N)(=O)=O)ccc(CC(N2CCN(C(C3CCC3F)=O)CC2)=O)cc1 c1(C(=O)NC2CCC(N(C)C(c3ccc(=O)oc3)=O)C2)cc2ncccc2o1 CCN=C(NCCC1CCCN1C)N1CCC(OC(=O)Nc2cnccn2)CC1 c1(OC)cc(Cl)c(C(=O)NCC2CC2NC(c2ncncc2F)=O)cc1Cl c1(C(N2CC(NC(c3cnc(OC)s3)=O)CC2(C)C)=O)cc(F)cc2nc[nH]c12 c1(CC)cnsc1C(N1CC=CC1C(=O)NC(c1snnc1C)C)=O c1(CONC(Cc2cc(OC)c(Br)cc2)=O)cc(OC)c(OC)c(I)c1 C1(C(=O)OCC)CC(O)(C(F)(F)F)CN1Cc1cc(C)[nH]n1 Cn1nnc2cc(NC(C3(CNC(c4cc(Cl)cnc4F)=O)CC3)=O)ccc12 C1(NC(c2ccsc2)=O)CS(=O)(=O)CC1NC(c1cc(C2CC2)nc(O)c1)=O Cc1ccc(CC(N2CCOC(C(C)NC(=O)CC3CCOC3)C2)=O)cc1F Cc1ccc(C(=O)NC2CC(CNC(=O)C(C(C)C)n3cnc(C)c3)C2)c(C)n1 CCC(C)(CNC(=O)C=CC(=O)OC(C)(C)C)C(=O)NCc1nc(C(C)C)n[nH]1 S(=O)(=O)(c1[nH]c(=NCC2CC3(CC3)CO2)ccc1Br)NC1(CC)CCCC1 N1(C(C(=O)Nc2ncc[nH]2)=O)CC2CC(C1)N(C(C1CCOC1C1CC1)=O)C2 N1(C(c2nc(CC)oc2)=O)CCC(F)C(NC(c2ccccc2CC)=O)C1 N1(C(CN(C(C2CN(C(C)C)C2)=O)CC2CC2)=O)CCCC(F)(F)C1 N1(C(C)=O)CCC2(CCCCC2NC(c2cc(C(C)C)[nH]n2)=O)C1 c1(OC)ccccc1C(C)CC(=O)NCCCCCNC(=O)CSC c1(C(=O)NCCOCCCNC(CC(C=C)CC)=O)cscc1S(C)(=O)=O C(=O)(C(C)CC(C)C(C)=O)N(CCOC)CCNC(C1(CCOC)CCC1)=O C1(CS(=O)(=O)NCC(c2ccc(F)cc2F)(C)O)CC2C(C1)C2(F)F C1(CNC(c2cccc(C)c2F)=O)CN(C(c2cnc(O)s2)=O)C2(CCC2)C1 c1(C(=O)NC(C2N(C(CC(C)NC(N)=O)=O)CCC2)(C)C)cc2c(s1)CCSC2 CCC(C)(C)COCCN.C(C(CC)ON)S c1(C(=O)NCC2CN(C(CC(C)F)=O)C3(C2)CCC3)cc2ccccc2cc1F C=CCCCC(C)(C)C(=O)NCC1C(O)C(O)CN1C(=O)CN(C)C(C)C c1(C(=O)NCC(N(C(C(C(CC)CC)C)=O)C)C2CC2)cc2c(=O)[nH]ccn2c1 C(=O)(CC1COc2cc(O)ccc21)NCC(C)NC(c1cnc2nccn2c1)=O C1(CC(C)(C)C)(CC)c2nnnn2-c2nn(C)cc2N1.c1(CC)c(C)ccnc1C c1(C(=O)NC2CCN(C(C3C4COCC34)=O)CC2F)ccc(F)c(Cl)c1F Cc1ccc(C(CNC(=O)C(Cl)=CCl)NC(c2ccncc2F)=O)cc1 c1(C(=O)NCCN(C(COCC)=O)C)ccc(N2CCN(C)CC2)c(F)c1 N1(C(C(c2c(C(=O)OC)cccc2)(F)F)=O)CCC(O)(CNC(=O)C(C)C)CC1 c1(C(=O)NCC2OCC(CNC(C3C(=C)C3)=O)C2)cc(N)cnc1Cl c1(C(=O)NC(c2occ(C(=O)NCCCCCC#C)n2)C)cccn2cncc12 C(=O)(CC(F)(F)C(F)(F)F)N1CC2C(CNC(c3c(SC)nccn3)=O)C2C1 c1(OC)cnccc1C(N1CCC(N(C(=O)CC(C)(F)F)CC2CC2)C1)=O N1(C(c2ncn(CC)n2)=O)CC2(C)CC1(C(=O)NC1CCC(=O)NC1=O)C2 c1(C(N2CCC(c3ccon3)C2)C(=O)NCCC)cccc(NS(C)(=O)=O)c1 C1(C2CCN(C(c3n[nH]cc3C(F)(F)F)=O)C2)(NC(c2ccc(Cl)cc2)=O)CC1 C12(CNC(C(CC)(C)C#N)=O)CCCC(CN1C(c1ccc3nc[nH]c3c1)=O)C2 c1(C(=O)NC2(CCCCNC(C3CCCO3)=O)CC2)cc(C(F)F)[nH]n1 CC1CC(NC(C2(N3CCOC3=O)CC2)=O)CN1C(c1coc(O)n1)=O N1(C(C2(CNC(c3cnc(Cl)s3)=O)CCCO2)=O)CCOC(CC2CC2)C1 N1(C(C(C)NC(c2ccc(C)s2)=O)=O)CCc2ccncc21 c1(C(=O)OC)nsc(=NC(CNC(c2ccc(F)o2)=O)C(C)C(C)C)[nH]1 Cc1ccc2c(C(N3CCC(C(C)NC(c4occc4F)=O)CC3)=O)csc2c1 c1(C(N2CC(NC(C(C)n3cccc3)=O)(CO)C2)=O)cc2c(cn1)CCCC2 C#CCC(CC(F)F)NC(=O)CNC(=O)CNC(=O)CC=C Cc1c(C(=O)NCC2CC2NC(C2(CCO)CC2)=O)noc1-c1ccccc1 c1(CC(=O)NC(CNC(COCc2onc(C)n2)=O)(C)C2CC2)cc(Cl)n(C)n1 C(=O)(CCN(OC)C(=O)C(C)C(O)C(C)C)NCCC1(OCC)CCCC1 c1(C(N2CC(CN(C(C(C)OCCCC)=O)C)C2)=O)cc(O)c(F)cc1N C(=O)(C1=CC2CCC(C1)C2)NCC1C(C)(C)CCCN1C(C1CC2CC2C1)=O c1(-c2ccc(CN(C)C(C3CCOC3c3cnn(C)c3)=O)o2)ccc(Cl)cc1 c1(C(N(CC(C)N(C)C(C2(F)CCCC2)=O)C)=O)cnn2c(=N)[nH]cnc12 c1(C(N(CC)CC2CCN(C(C3(CO)CC3)=O)CC2)=O)cc2sc(Cl)cc2s1 c1(CN(C)C(=O)NCc2cncc(C(F)(F)F)c2)cn2ccccc2n1 c1(CC)ncnc(CC)c1C(=O)NCCCNC(=O)C(C(C)C)c1cc(C)no1 CC1(C)CCN(C(C2CCS(=O)(=O)C2)=O)C1CNC(=O)CC(=O)Nc1nccs1 c1(-c2cn(CCN(C(CNS(NC)(=O)=O)=O)C)nn2)cccc(-c2cc[nH]n2)c1 c1(C(N(C2CN(C(c3c(C)nns3)=O)C2)C)=O)cncc2ccccc12 c1(CNS(C)(=O)=O)cn(CC(F)CCNC(=O)C(N2CCOC2=O)C)nn1 O=C(C#CC1CC1)NC(C(=O)NCCCF)C1(O)CCC1 N1(C(C(C)SCC)=O)CCC(C)(C)C1CNC(c1c[nH]nc1-c1ccncc1)=O c1(C(N(CCCCCC)CCNC(=O)C=C2CC2)=O)ccc(F)cc1OC c1(C(=O)NCCC2CCC(NC(c3cnco3)=O)C2)c(Cl)cncc1Cl C1(CNC(c2ccc(C)cn2)=O)CCN(C(C2C=CCC2)=O)C1(C)C c1(-n2c(NCC3C(c4onc(C)n4)C3)ncc2)ncccc1Br C1(NC(C(C)O)=O)CCC2CN(C(=O)CN3CC=CC3)CC2C1 c1(N(C(=O)C(F)(F)CC2CC2)C(C2CCCN2)=O)cccc(NC2CC2)c1[N+](=O)[O-] C1(CC=C)(NC(=O)C(C2CC2)OCC)CCN(c2ncc(Br)c(C)n2)CC1 N1(C(c2ccc(C)cc2N)=O)CCC2C(CCCN2C(c2c[nH]nc2F)=O)C1 N1(c2nc(C)nc(C(F)(F)F)c2)CCN(C(=O)Nc2cccc(Br)c2)C(C#N)C1 N1(C(=O)NCCC(COC)O)CCc2n[nH]c(C)c2C1 C(=O)(C1=CCCCC1)NC1(C)CN(C(C2CCC23CCCO3)=O)C1 c1(OC)ncc(Cl)cc1C(=O)N(CCCN(C(=O)Cc1ccco1)C)C C1(N(C(Cc2cc(C)no2)=O)C)CCCN(C(=O)C(C)(C)n2cnnn2)CC1 N1(C(C2ON=C(C(=O)OC)C2)=O)CCCC2CN(C(C3CC(C(C)C)C3)=O)CC12 C1(NC(CCCCOCC)=O)CN(C(=O)C(C)n2cncn2)CC(F)(F)C1 C(CC(=O)NC12CCC(CC1)C2)(C(F)(F)F)NC(CSC(C)C)=O N1(C(c2c(C)c[nH]c2CC(N)=O)=O)CCC(C)C(CNC(C2CC(CF)C2)=O)C1 N1(C(c2c(COC)noc2)=O)CC(C)CCC1CNC(=O)C(F)(F)C1CCCC1 CC1(C)OC(C(=O)NCC(C)(O)CNC(c2csc(Br)n2)=O)C(C)(C)O1 C1(C)(CNC(CC2C(CC)C2(F)F)=O)CCCN(C(c2c(C)nsc2C)=O)C1 N#CC1CCC(C(=O)NCC2CCCN2C(=O)C(C2CCCCC2)O)C1 N1(C(=O)CC2CCCCCO2)CC2(C1)CN(C(C1CC13CCOCC3)=O)CCO2 N1(C(COCCOCC#C)=O)CCC2OCCN(C(c3ccsc3C#N)=O)C2C1 C1(NC(C(C)=C(C)C)=O)CC2CC(C1)CN(C(=O)Cc1ncc(F)cc1F)C2 N1(C(c2cc(OC)ncc2)=O)CC(CNC(C2CC(=O)NC(=O)C2)=O)C(C)(C)C1 C1(CNC(C2(NC(C3C(C)=CCS3)=O)CCCC2)=O)CCCC(F)C1 c1(C(N2C(CNC(c3c(C)ccs3)=O)CC2)=O)c2c(nn1C)CCC2 c1(OC)c(C(N2CCOCC2CCNC(c2cocn2)=O)=O)ccc(Cl)c1Cl C1(CNC(=O)NC(c2c(F)cccc2I)CO)CCc2c(O)cccc2C1 c12ccccc1NC(=O)CC1CCN(C1)C2.c1(C(=O)OC)ccc(Br)cc1 N1(C(CCN(C(=O)CCc2ccncn2)C(C)C)=O)CCC2(C1)CC2(F)F S(=O)(=O)(CCC(=O)N1CCC(O)(CCNC(=O)CCC=CC(C)C)C1)NC c1(C(=O)NCCCN(C(c2ccnnc2O)=O)CC)cncc(OC)n1 N1(C(C)=O)CCC2(CC1)CN(C(=O)C1CC1)C2.C(=O)(C(C)CC=Cc1ccccc1)O Cc1[nH]nc2ccc(C(N3CCCC(F)(CNC(=O)CSC(C)C)C3)=O)c(Cl)c12 c1(C(=O)NCC2(F)CCC(NC(C(CC)O)=O)C2)c(OC)cccc1Cl C1(N(C)C(c2ccn(CC#N)n2)=O)CN(C(c2c[nH]nc2F)=O)CC1F N1(C(C=CC2(C)CCOCC2)=O)CCC2CN(C(=O)CC3CC(=O)NC3=O)CC12 c1(C(=O)NCCC2CCCN(C(c3cnc(C)[nH]3)=O)C2)cc(C)c(C)cn1 CCC(CCC(=O)N1CCC(OCCNC(C2CCC2)=O)CC1)OC O=CN1CCCC1C(=O)NCC1(F)CC(CNC(=O)C(C2CCOCC2)O)C1 c1(NCC(C)CO)ccc(S(=O)(=O)NCc2cc(Cl)n(C)n2)cc1C#N CC1CC(NC(c2ccc(C(N)=O)cc2)=O)CN1CCCCOc1ccc(F)cc1 C1(CC)(NC(C2CCCN2N=O)=O)CCCN(C(C2CCC(C)=C(C)C2)=O)C1 c1(OCC(=O)NCC2CC(F)(CNC(C(C)C)=O)C2)cc(F)ccc1F CCC(C(=O)NCC#CC(N1CCC(C2CCC2)C1)=O)C(C)(C)CC C(=O)(C#CC(=O)NCC1CC1CNC(c1ccc(C2CC2)cc1)=O)N(C)C c1(CN2CC(C3N(C(C=CCCCCC)=O)CCC3)(O)C2)ccnc(OC)c1 c1(CCC(=O)NC2CC(NC(CCC3CCCN(C)C3)=O)C2)c(O)cccc1F C#Cc1ccc(C)c(NC(=O)C(C2CC2)N(C)C(c2cnc(O)n2CC)=O)c1 c1(C(=O)NCC2CC(NC(C3OCCCO3)=O)C2)ccc(-c2ccccn2)o1 CCC(N=c1nc2sccc2c(NCC2COc3cc(CO)ccc3O2)[nH]1)C(C)C N1(CC2CC(CCOC)C2)CCCN(C)CC1C N1(C(CN2CC(C)(OC)C2)=O)CCC2CCN(C(=O)CCC(C)N(C)C)C2C1 C(C)(CC(=O)NCc1cc(C)on1)NC(C(C1CCC1)OCC)=O C1(C(=O)NC(C(=O)NCCC2CCCCCC2)C2CCC2)C2CCC(F)C12 N1(C(c2c(CCC)occ2)=O)CCC(CNC(=O)CCc2scnc2C)C(C)C1 CC(=O)CCCC(=O)NCC1CN(C(=O)CCOC2CCCC2)CC1C CCCCCC(CC)C(=O)N1CCC(CC(C)NC(c2csc(C)c2N)=O)CC1 Cc1ccc(C(N2CCN(Cc3ccn(CCF)n3)C(C(F)(F)F)C2)=O)cc1Br N1(C(CC2(OC)CC2)=O)CCC2(CCC2)C(NC(=O)CN2CC(=O)NC2=O)C1 c1(C(N2C(C)CN(C(CC)=O)C(C)C2)=O)cc2c(s1)C(C)(C)CCC2 c1(C(N2CC(CC=C)(NC(=O)COC3CCOC3)C2)=O)ncnc2sccc12 N1(C(CCC(=O)NC)=O)CCCC12CCCN(C(=O)C(C)S(N)(=O)=O)C2 Cc1cc(C(N2CCC(N(C)C(c3ocnc3C)=O)C2)=O)c(C(F)(F)F)o1 CC(CO)C(=O)N(CC=CC(N1CC(SC(F)F)C1)=O)C1CC1 c1(OC)ccc(C=CC(=O)NCCC2CCCN(C(c3csc(=N)[nH]3)=O)C2)cc1 c1(C(N2CCC(N(C(C3(C(C)C)CCCO3)=O)C)CC2)=O)cnc2[nH]ccc2n1 c1(C(=O)NCc2scc(CNC(c3c(CC)nn[nH]3)=O)n2)cc(Cl)ccc1C C(CC1CC1)(C(=O)N1CCC(CCC2CCC2)C1)NC(=O)Cn1ccnn1 CC1(NCC2(C(N)=O)CC(F)(F)C2)CCOC12CC2(F)F C(C)(Cc1ccco1)(C(=O)NC(CNC(c1csc(C2CCC2)n1)=O)CO)OC c1(SCCNC(C2CN(C(COCCOC(C)(C)C)=O)C2)=O)ccc(F)cc1 N1(c2nccc(C#N)n2)CC(NC(=O)Cn2ccc(C(F)F)n2)C2CCCCC12 c1(C(N2CCC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)c[nH]c2nccc(Br)c12 CCCCC(CNC(=O)C=Cc1ccc[nH]1)NC(=O)C(CN(C)C)N(C)C N1(C(CNC(c2cc(Cl)ccc2Cl)=O)=O)CCc2ncnc(O)c2C1 c1(C(N(C2CCCN(C(=O)CCc3ccccc3O)C2)CC)=O)cc[nH]c(=N)c1 c1(C(N2CCCC(NC(CCC#CC)=O)C2C)=O)oc2ccccc2c1COC C(=O)(C(C)(C)C(F)F)N1CC=CC(NC(COCc2n(C)ncn2)=O)C1 C1(CNC(C=CCN(C)C)=O)CCC2(CN(C(c3noc4ccccc34)=O)C2)O1 c1(CC(=O)NC(CC=C)CNC(C2CC(O)C2)=O)csc2nc(C)cn12 c1(NC(N(C)CC2(O)CCC(C)CC2)=O)cc(Br)cc([N+](=O)[O-])c1 c1(C(=O)NCC2(CO)CCN(C(c3c(C#C)c[nH]n3)=O)CC2)cc(Cl)cc(C#C)c1 N1(C(C(CC)CC2CCCC2)=O)CCCN(C(C2CCN(C)C2C)=O)CC1 c1(Cc2ccc(C(=O)NC(CC)(C)C)cc2)cccc(F)c1F C1(C(=O)NCCN(CCC)C(C2CCCN2N=O)=O)CCc2cc(C)ccc2O1 Cc1c(C(N2CCC(F)(CNC(C3(CCO)CC3)=O)C2)=O)ccc2ccccc12 N1(C(c2c(C)cn(C)n2)=O)CCN(C(c2ccc(Cl)cc2N)=O)C(C)C1C CCCCC(=O)C(=O)NCC=CCC(=O)NCC1(C(C)C)CCC1 Cc1[nH]nc(C(N2CC3C(C(N4CCCC4C4CCCC4)=O)C3C2)=O)c1Cl C1(C(=O)NC(C)CN(C)C(c2cnnn2C)=O)CC2OC(=O)OC2C1 CC1(C)C(c2ccccc2)CN1C(c1ccc(C(=O)O)s1)=O CC(c1ccsc1)=CC(=O)NC1COCCC1NC(=O)C(C)(C)c1ncco1 C1(C(CC)C(c2nnnn2-c2ccccc2)NC2(CCOC)CC2)CCOCC1 C1(CC(N2CCC(NC(C(C(C)C)(C)C)=O)CC2)=O)Oc2ccccc2NC1=O C1(C(=O)OC)(C(N2CC(CO)(NC(=O)C(C(C)C)N(C)C)C2)=O)CC2(CCC2)C1 c1(C(=O)NCc2n[nH]cc2NCc2cnc(Cl)cn2)ccc(C(F)(F)F)cc1F Cc1cc(C2CCN(C(c3cnc(C(C)C)s3)C(=O)NC(C)C)CC2)cnc1C C1(C(=O)NC2CCSC23CN(C(C2CCOC2)=O)C3)CC(c2cccnc2)=NO1 N1(C(Cc2cnc(C)[nH]2)=O)CCOC(C(=O)NCC(=O)NCCO)C1 CC(c1ccccc1)=CC(=O)N(C(C)C(=O)NCC1CCC(C)C1)C1CC1 CC(C(=O)NCC(C1CCC1)NC(C1CC(C#N)C1)=O)C(C)(C)C C#CCC(C)C(=O)NCC(C1CC1)NC(c1ccc(Cn2ccnc2)cc1)=O c1(N(CCNC(C2CCCN2c2ncccn2)=O)CC)ccncc1C#N c1(C(=O)NCCC(C)NC(C(CC)c2ccccc2)=O)cc(F)ccc1N c1(OC)ccc(C(=O)NC2CCCCC2NC(=O)C(C)OCCC(C)C)nc1 C1(CNC(CCC(=O)N(CC)CC)=O)CN(C(c2ccnnc2O)=O)C(C)(C)C1 c1(C(N2CCC3(C(C(=O)NCC4C(C)(C)COC4)C3)C2)=O)ccn2ccnc2c1 C(=O)(C1=CCOCC1)N1C2(C(N3CCC(NC(=O)NC)C3)=O)CC2CC1 C=CCC(C(=O)N1CC(CNC(=O)C=C(C2CC2)C2CC2)C(O)C1)C(C)C CCC(CCC(=O)NCC1(C(C)(C)C)CCN(C(=O)OC(C)(C)C)C1)OC c1(N2CCC(N(C)C(C3CCOCC3)=O)C2)nc(C(F)(F)F)ns1 N1(C(c2n(C)ncc2-c2cnc(=N)[nH]c2)=O)CCC(O)C(F)(F)C1 c1(OC)nc(C)ncc1C(=O)NCCC(C(C)C)NC(c1cc(C)cc(Cl)c1)=O C1(C(=O)NCC(C)(C)NC(C(c2ccc(F)c(Cl)c2)C)=O)CCc2ncnn2C1 C1(C(=O)NCc2nccc(C)c2)CC12CCN(C(=O)Nc1ccccc1)C2 c1(OC)cc(C)ccc1COCC(=O)NCC(C)NC(C1CC(F)C(=O)N1)=O N1(C(c2c(C)coc2C2CC2)=O)CCC(C)C(NC(C2C3(CC3)C23CC3)=O)C1 C(=O)(CC(C)(C)c1cccc(Br)c1)NC(C(CO)NC(C(F)=CC)=O)C C(C(=O)NC1CN(C(=O)Cc2conc2C)CC1O)(C(C)C)(C(C)C)NC(C)=O N1(C(CCCSC)=O)CCCC12CCN(C(C1CCc3ncccc3C1)=O)CC2 C1(C(N(CCCC)CCO)=O)CCOC1CNC(=O)CCc1nccn1C C1(NC(c2c(C)c[nH]n2)=O)CN(C(=O)C2=CCSC2)CC12CCOCC2 CC(=O)CCCC(=O)NC(CNC(=O)COc1cccnc1)C(C)C C1(NC(C(c2ccccc2F)(C)OC)=O)CCC(C)N(C(=O)C2=COCC2)C1 S(=O)(=O)(c1nccs1)N1C(C(=O)NCCF)CC1 C12(C(=O)NCCC(C)N(C(c3cnn(C(C)C)n3)=O)C)CCC(CC1)C(C)(C)O2 c1(NC(CN2C(C(=O)Nc3ncc(C)cc3O)CC2)=O)ncc([N+](=O)[O-])cc1Br C1(C(=O)NCCCCC=C)CCCN(C(c2ccncc2Cl)=O)C1 CC(F)(F)CCCC(=O)NC1C2COCC1CC(NC(=O)CCNC(=O)CO)C2 c1(C(N2CC(N(C(c3cnc(C)s3)=O)C)C(F)C2)=O)cnn2ccncc12 c1(C(=O)NC(C)C(=O)NC(c2ccccc2)C)ccc(Br)o1 C1(C(N(C2CC(C#N)C2)CC(=O)N(C)CC2CC(F)C2)=O)CCNC1=O c1(C(=O)NNc2ccncn2)ccc2c(c1)CNCCN2 C1(NC(c2cnc3[nH]cncc2-3)=O)CCN(C(C23CCN(CC2)C3)=O)C12CCC2 c1(C(=O)NCC2(F)CC(NC(C(C)OCOC)=O)C2)cncc(-c2ccoc2)c1 c1(C(N2C(C)CC(c3ccoc3)C2)=O)cc2c(n1C)CCNC2 CC(=O)CCN=C(NCCCC(F)(F)F)NCC1CC(=O)N(C(C)C)C1 N1(C(c2n(C)cnc2)=O)CCCC(CNC(=O)CCc2ccc(Br)cn2)C1 Cn1ccc2ccnc(C(N3CCC3CNC(C3CC4CCC(C3)S4)=O)=O)c12 CC(CC(=O)NC12CCC(CC1)N(C(=O)C(C)(C)CC(F)F)C2)CC(F)(F)F C(=O)(CCCCCCC(=O)OC)N1C(CNC(CCC=CC)=O)CCCC1 N1(C(C(C)NC(C2CCCC2)=O)=O)CC=CC(NC(C2(S(N)(=O)=O)CC2)=O)C1 N1(C(C2CC(C)(F)C2)=O)CCCC2(C1)CN(C(=O)CSCc1ccccc1)C2 C1(C(=O)NCC(=O)OC)(NC(c2cnc(SC)nc2)=O)CCCC1C CC(CCCC(=O)NC1(C)CCCN(C(c2ccncc2O)=O)C1)c1ccccc1 c1(CNC(=O)NC2CS(=O)(=O)CC2O)ccc(NC(=O)C(F)(F)F)c(F)c1 c1(C(=O)NCC2(NC(Cn3cc(CSC)nn3)=O)CC2)cc(C2CC2)oc1C C1(NC(C(F)=CC)=O)CC2CCC(C1C)N2C(c1ccc(-n2ccnc2)cc1)=O C(=O)(C(CNC(=O)COCCCN=[N+]=[N-])N(C)C)NC1(CC=C)CC1 c1(C(=O)NC2CCCN(C(C(C)NC(=O)NC)=O)CC2)cc2cc(Cl)ncc2[nH]1 c1(C(=O)Oc2ccccc2)cc(C(N)=O)cn1C.CCC(C)(Cl)C CCCCCCC(CC)C(=O)N1CC2CN(S(C)(=O)=O)CC2C1 c1(C(=O)NC2CC(NC(Cc3c(C)ncs3)=O)C(O)C2)cccc2[nH]ncc12 N1(C2CCC(NC(=O)NC(C(C)N(C)C)=O)C2)CCN(Cc2ccccn2)CC1 CCCC(O)CC(=O)NC(C)CNC(c1cn(-c2cccc(F)c2)nc1C)=O c1(C)ccc(F)cc1N.c1(CCN(C2c3c(cccc3)SC2)C)c(C)nn(C)c1C.CO N(C1CCc2cccn21)C(C1(C)N(Cc2ccc(C)o2)CC1)=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC1CCCN(C(Cn2nc(C)n(C)c2=O)=O)C1 C1(F)(C(=O)NCC(CN(C(c2c(C(C)C)[nH]cc2)=O)C)C)CCN(C)CC1 CCCCC(C(=O)NCCC(C(C)(C)C)NC(=O)C=CCCC(C)C)ON=C(C)C S(=O)(=O)(C(C(F)(F)F)NC(=O)CCn1ccc2ccccc12)NC(C)(C)C C1(C2CN(C(=O)CCCNC(c3ccsc3)=O)C2)(NC(CN(C(C)C)C)=O)CC1 C#CCCC(C(=O)OC)NC(=O)C(C)N(C(C1(C)CNC(=O)C1)=O)C1CC1 CC1Cc2sc(C(=O)N(C)CC3(NC(c4cnc(O)o4)=O)CC3)cc2C(C)C1 CC1=CC(C(=O)NCC(=O)NCC(=O)NCc2nc(C(C)C)n[nH]2)SC1 c1(CC)ccc(C(=O)NC(C)CC(C)NC(=O)C=CSC)c(F)c1 c1(CSCC)ccc(C(=O)NCC2(O)CN(C(=O)C(n3cc(C)cn3)C)C2)cc1 Cc1cc(C(=O)NC(CNC(=O)C(C)n2cccn2)CO)nc(C(F)(F)F)n1 C(=O)(C(F)(F)C(F)F)N1CCC(C(=O)NCC(O)CC2CCCC2)CC1 S(=O)(=O)(c1cccc(=NC(C)c2ccccc2Br)[nH]1)NCc1cc(OC)no1 c1(C(=O)NCC(CC)NC(C2(COC)CC=CC2)=O)cnc2cccnn12 Cc1ccc(F)cc1C(N1CCC(O)(C(=O)NC(C2CCOC2)C)C1)=O C1(C(=O)NCC(CC)(CC)NC(=O)CCCN(C)N=O)CCC2(CCCO2)CC1 C1(CNC(c2nc(-c3ccc(C)s3)sc2)=O)C(C)CCCN1C(=O)C=C1CC1 C1(NC(C(CC)OC)=O)CC(N=c2cc(Cl)nc(S(C)(=O)=O)[nH]2)C12CCC2 C1(CC)CN(C(=O)C(C)(C)CN(C(=O)C(C)SC(C)C)CC)C(C)CO1 CC(C)C(C)(C)C(=O)NC(CNC(=O)C(C)OCC1CC1)CO c1(NCC)cncc(C(=O)NC(C2CN(C(C3CCC(C(N)=O)O3)=O)C2)C)c1 C(=O)(C(C)(C)CF)NC1CCC(CCC(=O)NCCCCCN(C)C)C1 c1(C(=O)NCCC(CNC(c2ccc(F)c(F)c2)=O)O)cccc2nc(S)oc12 C(=O)(C(C)(C)C(=O)N(CC(C)N(C)C(c1cc(SC)oc1C)=O)C)NC C1(NC(COc2cccc(C#C)c2)=O)CC2CN(C(C3(C)CC3)=O)CC2C1 c1(C(C)NC(CCC2(NC(CC(C)C3CC3)=O)CCCC2)=O)cccc(F)c1 C1(C(N(CCCNC(=O)C(C)(F)F)CC)=O)CCCCC12CCC2 c1(OC)ccc(C(=O)NC(Cc2ccoc2)C(=O)N2CC(CN=[N+]=[N-])C2)o1 C1(CC(=O)NCCC2N(C(c3c(COC)scc3)=O)CCC2)CCCCC1F C(CN=c1cncc[nH]1)NC(C(=O)NCCCC1CCCC1F)=O C1(NC(c2cnccc2Cl)=O)CN(C(=O)CCCCC2CC2)C2(CCCCC2)C1 CC1c2cc(Cl)c(Cl)cc2CCN1C(c1cncc(CN)c1)=O C(=O)(C(F)CC(CC)CC)N1C(C)CCC(C(=O)NCCC(C)N(CCC)C)C1 C1(NC)CC(C)(C)OC1(C)C.C(=O)(CN=S(C)(C)=O)N1CCC(C)CC1 C=CC(C)(O)CC(=O)N(C(C(=O)O)C(C)C)C(C1(O)CCCCCC1)C1CC1 C1(NC(c2cc(C)nc(C)c2)=O)CCC12CCN(C(c1cc(C)oc1C)=O)CC2 Cc1c(Cl)ccc2[nH]c(C(=O)NCC(C)N(C(=O)C(C)c3ncco3)C)cc12 c1(NCC(c2ccc(C)cc2)NC(C2C(C(=O)OC)C2)=O)nccc2occc12 C1(CC)CN(C(=O)C(c2cccc(Br)c2)O)CCN1C(c1cncnc1C)=O Cc1cccnc1CC(=O)NC(C)C(CO)NC(c1cc(C(C)(C)C)c[nH]1)=O c1(C(C)C)nc(=NC2CN(C(=O)C=Cc3cnc[nH]3)CC3(CCCC3)C2)s[nH]1 c1(C(C)C(N2CCC(N(C(=O)C=CCOC(C)(C)C)C)C2)=O)cccc(F)c1 C(=O)(C(C)C(C)C(C)(C)C)N(CCN(C(c1c(CC)n[nH]c1)=O)C)C(C)C Cc1cccc2[nH]c(C(N3CC(O)CC3C(=O)NCCc3nn[nH]n3)=O)cc12 c1(NC)ccc(C(=O)NCC2CC(CNC(=O)C(=O)C(C)C)CO2)nc1 C#CCC(CC#C)C(=O)N(C1CC2CCC(C1)N2C(C12COCC1C2)=O)C N1(C(C(C)CF)=O)CC2CC(C)N(C(c3cc(-c4ccncc4)no3)=O)C2C1 Cc1c(C(=O)NC2CC(C)N(C(=O)CCS(C)=O)C2)cnn1-c1ccccc1 CCC(C(=O)NCC(C)NC(c1n[nH]c2cccnc12)=O)C(C)(F)F CN(C1CCCC1n1cccn1)N1CCN(c2ccccc2F)CC1 N1(C(CCCCN(C(C)=O)C)=O)CCN(C(C2CCCC(O)C2)=O)CC12CC2 C1(CNC(C2OCC(C)(C)C2)=O)CCN(C(c2cnsc2)=O)C12CCC2 c1(NC(C(C)OCCC=C)=O)ccc(NC(N)=O)cc1 C1(NC(C(CC)C)=O)(CNC(c2cc(OC)ncc2F)=O)Cc2ccccc2C1 c1(C(=O)NC(CC)CNC(=O)C(CC)C(F)(F)F)cnc(P(C)(C)=O)cn1 c1(C(=O)NCC(C)N(C(c2csc(C(C)OC)n2)=O)CC)ccnnc1O c1(C(=O)NCC2(F)CN(C(c3ccc(Cl)nc3O)=O)C2)c[nH]c2ccc(F)cc12 N1(C(CN(CC(C)NC(C2CC2c2cccs2)=O)C)=O)CCC(CO)CC1 c1(NC(C(=O)N(C)CCNC(=O)C=CSc2ccccc2)=O)ccc(CO)cc1 Cc1cc(CC(=O)N(CCCCN(C(=O)C(C)Cn2cccn2)C)C)n[nH]1 CCC(CC(=O)NCC1CC2(CC(NC(=O)C(O)CC(C)C)C2)C1)C(F)F CCC(CC)C(=O)NCC1(F)CCN(C(C2CC(=O)C2)=O)C1 C#CCC(C(=O)N(C)CCOC(C)=O)NC(=O)C(C)CC=CCC c1(OC)ccc(F)c(C(=O)NCC(F)CNC(C2CCSCC2)=O)c1F c1(C(N2C(CNC(CC(C)c3cccnc3)=O)C=CC2)=O)ccn2ccnc2c1 Cc1ncc(Br)c(C(=O)NC2CC(CCNC(C3(O)CCC3)=O)C2)n1 CC1(C)CCCC1CNC(C1OCCC1CNC(=O)Cn1cnnc1O)=O C(CC(C)CC)(C(=O)NCCc1cccs1)NC(c1c(CC)nns1)=O O=C(CCCC(F)(F)CO)NCCC1CCCN(C(=O)CC2CCCC2)C1 c1(C(C)NC(=O)CC=CCNC(C2(F)CCC2)=O)cn(C)nn1 C1(C)(CNC(C=COCC)=O)CCN(C(=O)CC2CC(F)(F)C2)C1 C1(NC(CCC#CC)=O)CN(C(c2ccc(CO)c(Cl)c2)=O)CC2(CCC2)C1 C1(CCC)CN(C(C2CCCSC2C)=O)CC1C(=O)Nc1ccccc1F C(=O)(C(C)(C)C(=O)NC1CCN(C(=O)C(NC(C)=O)=Cc2cccs2)C1)NC N1(CN2CCN(C(=O)C(c3ccc(F)cc3)N3CCCCC3)CC2)C(=O)CNC1=O c1(C(=O)NC2C(F)CCN(C(c3cn(CC)nn3)=O)C2)cscc1S(C)(=O)=O C1(C(=O)NCc2cn(CC=C)nn2)C=CCN(C(=O)CCn2ccnn2)C1 c1(C(=O)NC(CC)CCOC)cccnc1CNC(=O)CC1CC2CC2C1 c1(C(N(C=O)CC2(c3ccccc3)CCC2)C)ncc(Cl)cc1F C(C(CC(=O)NC1CCCNC1=O)C1CCC1)NC(c1cc(C2CC2)on1)=O N1(C2CCN(C(CC3(C)CCC3)=O)C2)CCC(NC(C2CC2(Cl)Cl)=O)CC1 c1(CC(=O)NCCC2(NC(CN(C)C(=O)OC(C)(C)C)=O)CC2)ccn(C(F)F)n1 n1(CC)nc(C)c(C(=O)NCC2(F)CC(CNC(=O)Cn3nnc(=O)[nH]3)C2)c1C c1(C(N2CCCS2(=O)=O)=O)cc2c(s1)-c1ccccc1OC2 C1(NC(C(COC)(F)F)=O)CCN(C(c2c(F)cncc2Br)=O)CC1C N1(C(C=CCN(C)CC)=O)CCC2CC2(NC(=O)CCCCCF)CC1 N1(C(C(C)N(C(C)=O)C)=O)C2CC=C(C(=O)N(CCCN=[N+]=[N-])C)C1CC2 C=CC1(CC(=O)NCC(C)(CO)NC(=O)CC2COC(C)(C)C2)CCCCC1 C1(NC(CCNS(CC)(=O)=O)=O)CC2CC1CN2C(c1cccn2cnnc12)=O C(C(=O)NC1CC(C(C)C)C1)(C(C)(C)C)NC(CC(C)(C)SC)=O c1(C(=O)NC2C(C(=O)NCc3c(OC)cccc3)C2)cccc(Cl)c1OC c1(CNC2CC(C(=O)NCC(O)CO)C2)ccc(Br)c2nsnc12 c1(OC)cc(C(N2CC(NC(=O)Cc3cc(C)no3)CC2C)=O)cc(C)c1 c1(C(=O)NCC2C3CC2N(C(=O)CCCc2ccncc2)C3)cc(F)cnc1O C=CCC(CNC(C1(C)CC(C)C1)=O)NC(c1ccncc1)=O C(Cc1cn[nH]c1)(C(=O)NCCCOC)NC(CCN(CCC)C)=O.c1cn[nH]c1 c1(C(=O)NC(CC)(CNC(c2ccnc(OC)n2)=O)CC)cc(Cl)c(C)cn1 C1(C(=O)NCC(CN(C(=O)Cn2ccc(Br)n2)C)O)CCc2nn[nH]c2C1 c1(CC)cnn(C)c1C(C(=O)NC1CCOC1)N(CCOCC)C1CC1 C1(c2nnnn2C(C)(C)CC)(NCC(=C)Br)CCC(P(C)(C)=O)C1 c1(C(N(CCC(C)NC(CS(CC)=O)=O)C)=O)nc2ccccn2c1F CC1CN(C(=O)CCc2cnn[nH]2)CC(C)N(C(=O)CC23CCC(CC2)CC3)C1 c1(CC)c(C(=O)NCC23CC(NC(=O)C(C)C(F)F)(C2)C3)[nH]c2ccccc12 c1(OC)nc(C(=O)NCC2CCCCN2C(=O)C=Cc2nnn(C)n2)sc1C N1(C(C2(CC=C)CC=CC2)=O)CC2CCCC(C1)N2C(C1CCCN(CC)C1)=O C(CC(O)C(F)(F)F)NC(C1CN(C(C2CCN(C(=O)OC(C)(C)C)CC2)=O)C1)=O CCC(C)CC(C)C(=O)NCc1ccc(C(=O)NCC(=O)NC2CCCC2)o1 C(=O)(C1=NNC(C(F)(F)F)C1)N(CCC(C)NC(C1CC(CCC)C1)=O)C N1(C(C(c2c(C)cccc2C)O)=O)CCOCC(F)(CNC(=O)C2CC2)C1 C1(NC(CN(CCC)C)=O)C(CNC(=O)CCOCC)C1(C)C C1(NC(CC)=O)CN(C(c2ccc(C)c(C)n2)=O)C2(CCCOC2)C1 c1(C(N2CCC(O)(C(C)NC(c3ccnn3C)=O)CC2)=O)ccc(F)c(Cl)c1N CC(CCC(C)(C)C)C(=O)N1CCCCCC1C(N1CCC(N=[N+]=[N-])CC1)=O Cc1cnc(C(=O)NCC(CO)NC(c2csc(C)c2C)=O)cc1Br N1(C(C(F)=C(C)C)=O)CCN(C(=O)CCC(N)=O)C(CF)C1 C12(C(N(C)CC3(CNC(C(C)NC(N)=O)=O)CC3)=O)CCC(C)(CO1)C2 c1(C(=O)NCCCCCCN(C(=O)CC2COCCO2)C)cncc(C(F)F)c1 C1(C(N2CCC(NC(c3c(CC)con3)=O)(CF)C2)=O)CCC(C2CC2)CC1 Cc1cc(C(=O)NC(C2CCCN2C(C23CCC2CC3)=O)C)c(C(F)(F)F)o1 C1(NC(c2c(C)occ2)=O)COC2(CNC(=O)C(C)C3CC3)CC1C2 c1(CC2CCN(C(NOC(CC)CC)=O)C2)cccc(Cl)c1 CC1(CNC(c2cc[nH]c(=N)c2)=O)CCCN1C(=O)COc1cccc(F)n1 C12(CNC(CCOCC#C)=O)CC(NC(c3cnc(CC)[nH]3)=O)(C1)C(C)(C)O2 c1(CCCC(=O)NCC2CCC(NC(COCC=C)=O)CC2)ccc(CC)cc1 C1(CC2c3cccc(c3)N2)CCC2(CNC2)OC1.c1(OC)ccccc1 C12(CNC(CCCOC)=O)COC(CNC(=O)C(c3cccs3)N(C)C)(C1)C2 Cc1cc(C(=O)NC2CCCC2CN(C)C(C2CC(C3CC3)C2)=O)nc(O)c1 Cc1c(CC(N2CC=CC(NC(c3cc(Br)no3)=O)C2)=O)ncn1C Cc1cc(F)ccc1CC(=O)N(CCCNC(C1CC1C(F)(F)F)=O)C c1(C(N2C(C)(C)C(NC(=O)CSCCC#N)CC2)=O)ccc(F)c(F)c1F CC1CC(NC(c2ccc(F)o2)=O)CCN1C(C1CC2CC2CC1C)=O c1(C(=O)NCCC2CCCN(C(=O)C=Cc3cc[nH]n3)C2)cc(O)nc(O)c1 C(=O)C(O)C(C)(C)C.N1(CC(C2(O)CN(C(C34CC3C4)=O)C2)(C)C)CCOCC1 CCCC(C)CC(=O)N1CCCC(N(C)C(c2c[nH]nc2OC)=O)C1 Cc1ccc(C(N2CCCC2C2CCN(C(C3(F)CCS(=O)(=O)C3)=O)C2)=O)nc1O C1(NC(c2cncc(N)n2)=O)CCCCN(C(c2cncc(C(F)(F)F)n2)=O)C1 O=C(C#CC1CCCO1)NC(c1cccc(Cl)c1)CNC(c1cnc(O)o1)=O c1(CC(=O)NCCN(C(C2CC2C2CCC2)=O)CC)cccc(OC)c1Cl N1(C(CCCNC(C2CC(C)(C)C2)=O)=O)CCCN(C2CC2)CC1 c1(C(=O)NCCCN(C(=O)Cc2ccn(C)n2)C)cncc(OCC(F)F)c1 c1(C(N2CCC(NC(C3CC4C=CC3CC4)=O)(CF)C2)=O)cnc2ccccn12 O=C(C1OCCn2ccnc21)NC12CC1CN(C(=O)CCn1ccnc1)C2 C1(C(=O)NC(c2csnn2)C)CC2(CCN(C(=O)CN3CCNC3=O)C2)C1 N1(C(C2C(C(C)C)CCO2)=O)CC2(CCC2)C1 c1(C(=O)NCC2CN(C(c3c(C)nc(C)o3)=O)CC2O)ccccc1S(C)=O CC1CCC(CNC(=O)C=CC(C)(C)C)CN1C(=O)Cc1nnc(O)s1 C1(CNC(C(CCOC)O)=O)(NC(=O)Cc2ccc(C)s2)CCCCC1C n1(CC(=O)NCC(CC)NC(C2Cc3nccnc3C2)=O)c(C)cc(O)cc1=O C(=O)(C(O)C1=CCCCC1)NC1(CNC(c2cc(F)c[nH]2)=O)CC(OC)C1 c1(C(C)OC(=O)CC(C)(O)C2CC2)nc(N(C(C)CCNCC)C)cc(Cl)n1 c1(OC)cccc(C(F)F)c1C(=O)NCC1(NC(=O)C(CC(C)C)N(C)C)CC1 C(=O)(C(CCC1CCCO1)Nc1cccnn1)OCCC(N)=O C1(C(=O)NCC(C(C)C)(C)NC(c2cn[nH]c2)=O)CCC2(CCC2)O1 C1(C(=O)NC2CCC(NC(=O)CN3C(=O)CCC3=O)C2)CC2CC(=O)C1C2 c1(OCC)ccc(C(=O)NCC2(N(C(=O)C=CCO)C3CC3)CCOC2)cc1 N1(C(Cc2c(C)cc(Cl)cc2)=O)CC2CCN(C(C3SCCS3)=O)CC12 C(CC(C)C)(C(=O)N1CCCC(O)(CN(C(=O)CC2CC2)C)C1)NC(C)=O N1(C(c2c(CC)cnn2C)C(=O)NCC2CCCO2)CCN(C)CC1CC(C)C c1(OC)ccc(CCC(N2CCC(C)(CC(=O)Nc3cc(O)ccn3)C2)=O)cn1 c1(OC)cncc(CCC(=O)NC2CC(NC(=O)C=C(C3CC3)C3CC3)C2)c1 CCCCCCC(CC)C(=O)N1CCC(O)(CNC(=O)CSC(F)(F)F)C1 N1(C(CC=C=C)=O)CCC2(CC(NC(=O)C(C)CN(C)C)C2)C1 c1(SC)ccc(N)cc1C(=O)NCCC1(O)CCN(C(C2CCC2(C)C)=O)CC1 c1(C(=O)OC)cc(C(N2CC(N3CCOCC3)CC2C)=O)ccc1OC c1(C(N2CC(CN(C(=O)CCCC3CC3C)CC)C2)=O)cc(O)ncn1 CC1CCN(C(C2CCC(=CF)CC2)=O)CC1NC(c1ccccn1)=O c1(CSC(C(C)O)C)nc2cc(Cl)ccc2n1C C(=O)(N=S(C)(=O)C1CC1)C1(c2cc(C(=O)OC)cc(OC)c2)CC1 Cc1cc(N)c(C)nc1C(N1CC=CC(NC(=O)COC2CCOC2)C1)=O c1(CC)c(C(=O)NCC(CO)NC(=O)C=CC2CC2)cnc2cc(O)nn12 C1(C(N(CCCC#C)C)=O)(NC(c2[nH]cc(C)c2C)=O)CCC(C)(C)C1 C#Cc1ccc(F)c(C(=O)NCC2CCN2C(=O)C(F)C2CCOC2)c1 C=CCCC(F)(F)C(=O)N1CCC(NC(c2n[nH]cc2C(F)(F)F)=O)C1 S(=O)(=O)(c1cccc(N2CCC(N)C2)c1Br)N(CC(N)=O)C C12(NC(C34CC(CC(C)C)(C3)C4)=O)CCC(CC1NC(=O)C=CC(=O)N(C)C)C2 Cc1ccc(C(N2CC(CO)CC(C)C2)C(=O)NC2CCCCC2)c(F)c1C c1(C(=O)Nc2cccc(C(=O)Nc3nc(C)c(C)s3)c2)cccc(F)c1Br C(=O)(C(CCC(C)C)NC(c1ccc(C)cn1)=O)NCC(CC)O N1(CCNC(C2C3CN(Cc4cn(C)nc4)CC32)=O)C(=O)CCCC1=O c1(C(=O)NC(C2CN(C(=O)C(F)(F)c3nccs3)C2)C)ccc2oncc2c1 CC(c1cnn(C)c1)=CC(=O)NCC1CCCCN1C(=O)Cc1cn(C)nc1Cl C12C=CCCC1c1nc(no1)CC(=O)N2.Cc1nscc1CC#N Cn1cc(C(=O)NCCNC(c2ccccn2)=O)c(C(C)(C)C)n1 C1(NC(Cc2ccc(C)cc2)=O)CN(C(c2cnc(C)cn2)=O)C2(CCC2)C1 N1(C(c2c(=O)cc(C)n(C3CC3)c2)=O)CCC2(CCC(NC(C3(Cl)CC3)=O)C2)C1 C(=O)(CC(C)CCCCCC)N1CC(CC)N(C(c2ccn(CC#N)n2)=O)CC1 c1(C(=O)NC(CNC(CC(C(C)C)OCC)=O)C)ccc(=O)n2c1CCCCC2 C12(NC(C3(C=C)CCN(C(c4nccc(C)c4N)=O)C3)=O)CC3CC(CC1C3)C2 CCC(CC1CCCCC1)C(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)C(F)C1 c1(CN(C)C(C2(CCF)CNC2)=O)cc(F)ccc1F N1(C(c2c(C)[nH]cc2)=O)CCC2CN(C(c3cc(F)cc(F)c3)=O)CCC2C1 C1(NC(C(C(CC)C)N(C)C)=O)CC2CC1CN(C(c1ccnc(S)c1)=O)C2 C1(CNC(C(N2CCCCC2=O)C)=O)CN(C(C2COCCO2)=O)CCC1C c1(OC)nc(N2CCC(C)(NC(=O)CC3CC(F)(F)C3)CC2)cc(C)n1 c1(C(N2C(C(=O)Nc3nnc(C)o3)CSCC2)=O)ccc(Br)cc1CO C(=O)(CCCCN1CCCC1)N1CCC(CNC(C(C)c2cc[nH]n2)=O)C1 C1(CC(=O)NCCOC2CCOC2)CCCN1C(C1(CO)CC1)=O N#Cc1ncc(C(=O)NCCN(C2CCCCCC2)C(=O)Cc2cscn2)s1 CC1(NC(c2ncsc2Br)=O)CCN(C(=O)Cn2cnc(C#N)n2)C1 c1(NC(c2c(-c3c(C)cccc3)cncn2)=O)nc2ccc(Br)c(C)n2n1 CC1CN(C(=O)C=Cc2ccc[nH]2)CCN1C(C1CC(=C2CCC2)C1)=O CCCCC(CC)CC(c1nnnn1C)NCCc1nnc(C)s1 C1(C(N2CCC(N(C(C(CC)n3cncn3)=O)C)C2)=O)(OC)CCC(C)(C)CC1 c1nc2ccccc2s1.C(=O)(C(C)C(C)(C)C)NC.C1(=O)CCCN1C(C)C C1(NC(COc2cn(C)nc2)=O)CCC(C)(CNC(=O)C2=CCCCO2)CC1 c1(C(N2CCC(C(F)F)(CNC(C3CCCC3)=O)C2)=O)ccc2ccncc2c1 c1(CC(=O)NC2CC(NC(c3ccsc3Br)=O)C2)cnc2[nH]ccc2c1 C1(NC(Cn2c(C)cnc2)=O)CCN(C(C2(CO)CCCCO2)=O)CCC1CO C1(C(N2CC3C(NC(=O)C(O)C4CCC4)(C3)C2)=O)CC2(CCCCC2)C1 C1(C(N2CC3(CN(C(CCCOCC=C)=O)C3)C2)=O)CC2COCCN2C1 c1(OC)ccncc1C(=O)NC1CC1NC(=O)CC(C)c1cccnc1 N1(C(COC2(C)CCCC2)=O)CC2(NC(=O)CCc3cncc(F)c3)CC1C2 N1(C(CC(C)F)=O)CCC2(CC1)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C2 c1(CCSC)n[nH]c(=NC(=O)C2(C#N)CC3C=CC2C3)s1 c1(C(=O)NC(CNC(CC(C)CF)=O)(C)C2CCC2)cccc2ncccc12 C(=O)(CCCC(F)F)N(C)CC1CCN(C(C(C)O)=O)C1 C(CC(F)CN=[N+]=[N-])NC(C(C1CCN(C(C=CC(C)(C)C)=O)C1)F)=O c1(C(=O)NCCNC(C2CC2[N+](=O)[O-])=O)nn2c(c1I)CCCC2 c1(CC)ccc(OCC(=O)NC2(CNC(=O)CCNC(N)=O)CCCCC2)cc1 C1(C(N2CCC(CC)C2)=O)(CC)CCN(C(c2csc(CO)n2)=O)C1 N1(C(C(C)CN(C)C)=O)Cc2[nH]nc(C(=O)N(C3CCCC(C)C3)C)c2C1 c1(-c2c(C(=O)NCC3CN(C(CCC)=O)C(C)C3)cccn2)ccc(F)c(F)c1 c1(C(C(N2CCC(CCNC(c3ccnnc3)=O)C2)=O)(F)F)cccc(Cl)c1Cl C12(C(N3CCCC(C(=O)NC4CN(C)C4)C3)=O)CCC(CC1)CO2 CC(C)CC(CNC(=O)CC(C)n1ccnc1)NC(=O)C(c1ccccc1F)O CN=c1[nH]c(=NCc2ccc(Br)cn2)[nH]c(=NC2CCCC(C(=O)NC)C2)[nH]1 c1(C(N2C(C)CCC(NC(CC(=O)NC)=O)C2)=O)cccc2c(C)c(C)[nH]c12 c1(CC)cc(C(N2CCCCC2CNC(=O)C(C)C(O)CC)=O)cc(C)c1 C1(C(N2C(C3(NC(CCOC)=O)CC3)CCC2)=O)CC(c2ccccc2F)=NO1 C1(c2nnnn2C2CC(F)(F)C2)(CN(C)C)CCCC(CC2(N)CC2)C1.C1CC1 Cc1cc(C)n(CC(N2CC(CNC(c3cnn(CC(C)C)c3C)=O)C2)=O)n1 CCC(CC(=O)N1CCCCC1c1cn(Cc2[nH]nnc2C)nn1)C(C)C N1(C(N2CCOC2=O)=O)CCC2(CCCN2c2nc(-c3ccc(F)cc3)cs2)C1 c1(OC)cc(OC)cc(CN2CC3CC3(C(N3CCCCC3CCCO)=O)C2)c1 c1(OC)cc(CNC2C=CC(NC(=O)Cc3ccccc3)C2)ccc1F Cc1cccc(OC(=O)Cc2noc(Cc3ncc(C(F)(F)F)n3C)n2)c1 C1(CNC(C2(C)CC2)=O)CC(CNC(c2cnoc2C2CCOCC2)=O)CO1 C(C1=NOC(C)C1)NC(C(CC1CN(C(CCSCCC)=O)C1)F)=O c1(C(=O)NCC2CC2NC(C2CCOCC2)=O)cccc(F)c1F c1(NC(C2N(C(C3C(C)CCC3)=O)CCC2O)=O)cc(Cl)nc(Cl)c1 c1(CC)oc(C(N2CCC(CNC(C3(C)CCCS3)=O)C2)=O)cc1C(=O)OC N1(C(C=C(COC)C)=O)CCOC2(C1)CN(C(c1cncc3c[nH]nc13)=O)C2 S(=O)(=O)(c1ccc(N2CCN(C=O)CC2)c(Cl)c1)NCc1c(C)cc(Br)cc1C c1(CC)ncc(C(N2CCCC(N3CCN(C(C4CCC4)=O)CC3)C2)=O)c(O)n1 c1(C(=O)NCCN(C)C(c2cccc(F)c2)=O)ccccc1OC(C)(C)C Cn1ncc2c1CC(CCC(=O)NCCC1CC(NC(=O)C(F)F)C1)CC2 c1(SCC)cccc(CC(=O)NC(C)CCNC(C2(CC3CC3)CCC2)=O)c1 Cc1ccc(C(=O)NC2(C)CC(NC(c3cnc[nH]c3=N)=O)C2)cc1Cl N1(C(CCSC)=O)CCC2(NC(C3CN(C4CCOC4)C3)=O)CCCCCC12 N1(C(C2(C)CC2)=O)CC2(CC(NC(C3COC4(CCCC4)O3)=O)c3nccn32)C1 N1(C(C(CC)NC(C)=O)=O)CC2CCC1CN2c1nccc(C(F)F)n1 C1(C(=O)O)(CNCCc2ccc(C)nc2)CCCCCCC1 Cc1cnc(C(=O)NCC#CCNC(=O)C(C(C)(C)C)n2ccnn2)cc1C#N C1(NC(CCC(=C)Br)=O)CC2(C1)CC(NC(=O)C(C)NC(=O)C(C)(C)C)C2 c1(CCOCC(=O)NCCC2CCCN(C(=O)C(F)(F)CO)C2)ccc(O)cc1 c1(C(N2CC3C(C(N4C(CC)CCCC4)=O)C3C2)=O)cc(Br)c(O)c(Br)c1 C1(C(=O)NC(C2(CNC(=O)C(c3ccc(F)cc3)(F)F)CC2)C)CCS(=O)(=O)C1 N1(C(c2nccc(CC)c2)=O)CCC2C(CCCN2C(=O)CC2CNC(=O)C2)C1 N1(C(C(c2cccnc2)OC)=O)CCC(CNC(=O)C(=O)C(C)C)C1(C)C CC(CC(=O)N1CC(O)(CNC(c2cnn(CCF)c2)=O)C1)c1ccncc1 c1(NC23CC(C(=O)Nc4c(OC)cccc4Cl)(C2)C3)ncc2c(n1)CCC2 C1(NC(c2nc(COCC)[nH]n2)=O)CCCN(C(c2ccccc2)C(=O)O)C1=O N1(C(CCNS(C)(=O)=O)=O)CCCC(C2CCCCN2C(=O)Cn2ccnn2)C1 c1(N2CC=C(C)C2)nc(N(C)Cc2cc(Br)cn2C)c2c(n1)CSC2 c1(NC(C2N(C(c3c(CC)noc3)=O)CCCC2)=O)ccc(C)c(Cl)c1 Cc1nc(C(=O)N(C)C)ccc1C(N1CCC(NC(=O)C2=CCC2)C1C)=O C1(C)(CNC(c2cc(CCOC)on2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C N1(C(Cc2c(SC)cccc2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(F)C1 c1(C(N2CC(C)(C)C(c3ccccc3)C2)=O)cc(Cl)c2ccccc2n1 c1(C(N(C(C)CNC(c2c(Cl)cccc2Cl)=O)C)=O)cc(F)cc2ccncc12 C(=O)(CC(C(F)(F)F)c1c(C)nn(C)c1C)NCCNC(COCCC)=O C1(C(N2CCC(N(C(C3=C(C)OCCC3)=O)C)C2)=O)CCOCC12CCCCC2 Cc1ncccc1CN1CCOCC1C(=O)Nc1cnn(-c2cccc(Br)c2)c1 C1(NC(C(COC)C)=O)CN(C(C2(Cc3ccc(F)cc3)CCC2)=O)CC1O N1(C(CC2CN(C(=O)Cc3ccccc3Cl)C2)=O)CCc2c(F)cccc21 C1(C)(CC)CCN(N(C)Cc2ccc(C)cn2)CC1 C(=O)(C(C)C(CC)CC)NC1(C2CN(C(c3cc(CC)c(C)cc3)=O)C2)CC1 N1(C(CNC=O)=O)CCC(N)CC1.C1(CCF)CCCN1C(=O)Cc1ccsc1Cl c1(CC)ccc(N)c(C(=O)NCC2CN(C(c3ncncc3Br)=O)C2)c1 C1(NC(=O)CCOCC(F)(F)F)CN(C(C2CCCNS2(=O)=O)=O)CC1C1CC1 c1(CN(C(c2c(F)ccc(C)c2)=O)C)cnn2c1CN(C(C1CC1(F)F)=O)CC2 N1(C(=O)Nc2cn(C)nc2-c2ccoc2)CCOC2COCCC12 C1(NC(C(C(C)O)C)=O)CCCC12CCN(c1nccnc1C#N)CC2 N1(C(CCC(C)NC(CC2(CSC)CC2)=O)=O)CCn2c(cnc2C)C1 N1(C(C(CC)C)=O)CC(OC)CC1CCNC(C1(C(N)=O)CC1)=O CC(C)C(C(=O)N(C)C)NS(=O)(=O)CC1(C(F)(F)F)CCC1 C(=O)(CCCCC(=O)N1CC2(COC(CNC(=O)CSCC(N)=O)C2)C1)NC N1(C(C2CC(C#N)(O)C2)=O)CCc2ccccc2C1CNC(C1CC=CCC1)=O N1(C(C)=O)CCC2NCCCC2C1.C1(Nc2nn[nH]n2)CCC2CC12CC(F)F C(C1CCCCCC1)=CC(=O)NCC(CC(C)C)NC(=O)C(C)(C)OC(C)C c1(CC)ccnc(C(N2CCOCC2CNC(=O)CCN(C)CC)=O)c1 C1(C(=O)NCC(C#C)CC)CCN(C(=O)C2=CCCCC2)CC1C N1(C(Cc2c(OC)cccc2)=O)CCN(C(=O)C(O)CC(C)C)CC1C1CCC1 C1(C(=O)NCCCCCCC)CCCN1NC(=O)c1ccc(C(C)C)o1 N1(N2CCC(C)C(CC=O)C2)CCC(C)(C#N)CC1.C1(C=O)(C(=O)C2CC2)CC1 C(CC(CC)C(=O)N(C)CC1(NC(c2oc(C3CC3)nc2C)=O)CC1)=CC C1(CC(=O)NCC=Cc2ccc(Br)cc2)(OC)CC2NCCC12 c1(C(C)=O)[nH]c2ccccc2c1C(N1CCN(C(=O)C(C)C(C)C)C(C)C1)=O C(=O)(CCCCCOC)NC.C1(C(=O)NC)(OCCCNCCCO)CCOCC1 N1(C(C2C(C)(C)C2(C)C)=O)C(C(=O)NCCc2ccsc2)CCC12CC2 C1(NC(C(CC2CN(C(c3c(C)n[nH]c3)=O)C2)F)=O)CC2CC1CC21CC1 Cc1c(C(=O)NCC2CC2NC(=O)C2=COCCO2)nc2sccn12 C1(NC(c2scc(C)c2)=O)CCCCC1C(=O)NCCC1CCCCC1O C(C(=O)NC(C)(C)CCNC(C1CCCN1C)=O)(C(F)(F)F)OC(C)=O C12(CCC(F)(F)CC1)C(=O)OCC2.c1(CC(=O)NC)coc(CN)n1.OC N1(C(C2N(C)CC(O)CC2)=O)C(CNC(=O)Cc2cnnn2C)CC2CCCC12 C12(O)CCN(C1)C2.C1(C)(C(=O)OC)CC(C(=O)NC(c2cn(C(C)C)nn2)=O)C1 N1(C(c2cc(OC)ns2)=O)CC2CC(NC(=O)C(C)(C)CNC3CCCC3)C1C2 C1(NC(C(C)CN(C)C)=O)CCCCC12CCN(C(=O)CC13COCC(C1)C3)C2 Cc1ncnc(C)c1OCC(=O)NC1(CCCNC(c2ccoc2C)=O)CC1 c1(C(=O)NCCN(C(C2CCCC2)=O)CC)ccoc1C(F)(F)F N1(C(Cc2ccc(CCCC)cc2)=O)CC2(CCC2)CC1CNC(=O)CNC=O c1(C(=O)NC(C2CCCC2)CNC(CN(CCC#C)C)=O)c(N)sc2c1CCC2 C1(NC(C(C)SC)=O)CN(C(=O)CCc2ccc(F)cc2F)CC12CCC2 c1(N2CCCC(OC)CC2)nc(NC2CCN(CC)C2)nc2c1cnn2C C1(C(N(CCN(C(=O)CCCc2ccc(Cl)cc2)CC)CC)=O)COCCN1C Cn1cc(C(=O)N(C2CCCC2)CCNC(C2C3CC3C3CC23)=O)c(O)nc1=O C1(NC(C(C)(C)CO)=O)CN(C(=O)CCn2cncn2)CC2CCCC12 C(CSC)(C(=O)N1CC(=C(F)CNC(=O)Cc2cc(C)cs2)C1)OC C1(CC)CCOC2(CCN(C(=O)CCC(=O)N(CC)CC)CC2)C1.C1(C)C(=O)N1 c1(C(N(CCCNC(c2n(CC)ccc2)=O)CC)=O)cc(C)c(F)cn1 c1(CNC(C2C(OC)CCC2)=O)cccc(C(=O)NCCCC2CC(C)C2)n1 c1(C(=O)NC2(CNC(c3c(C)cc(Br)s3)=O)COC2)ccc2n[nH]cc2c1 C(=O)(C(=O)N1CC(OCC)C1)NCCN(CCCOCC)C(C)(C)C c1(C(=O)OC)c(Br)ccc(CN2CCCC2c2ccc(Br)c(Cl)c2)c1F C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(=O)C(C)OC)C2 C1(CNC(c2cnc[nH]2)=O)C2CCC(C2)N1C(=O)C=CC1CCCCC1 C1(C(=O)NCCCOCCNC(CC2CC(OC)C2)=O)CCCC2CC12 O=[N+]([O-])c1cc(C(F)(F)F)ccc1CN(C1CC1)Cc1cccnc1Cl CN1C(=O)COc2ccc(C3(C(=O)NCC(C4(O)CCSCC4)C)CC3)cc21 CC(C)S(=O)(=O)CC(=O)N1CCCC1CCNC(=O)COc1cccnc1 C1(C(=O)NCCN(C(C(CC)NC(N)=O)=O)CCOC)CCCC1(C)C c1(C(N2CC(NC(C3C(=C)C3C(=O)OC)=O)C2)=O)ccc(F)c(C(C)C)c1 C1(C)(C(N2CCC(N(CCC)C(c3ncoc3COC)=O)C2)=O)CCC(=O)N1 C1(CC(=O)NC2C(C)CN(C(C3(C)CCOC3)=O)C2)CCCNC(=O)C1 c1(CC(N2CC(C3N(C(C(CC)SC)=O)CCC3)(O)C2)=O)cc(F)ccc1Cl C1(NC(CCc2ncc(C)[nH]2)=O)CN(C(=O)CSc2ncccn2)C2CC12 C1(C(=O)NCC2CCCN(C(C=COCC)=O)C2)Cc2ccc(F)cc2C1 C1(SC)CN(C(=O)C2=CCC(NC(=O)Cn3ccccc3=O)C2)C2(CCC2)C1 c1(C(=O)NC2CC(F)(CNC(C(C)NC(=O)NC)=O)C2)nn(C)cc1[N+](=O)[O-] C1(C(=O)OC)CC(C)CN(C(c2cccc(-c3ccc(C(=O)O)cc3)c2)=O)C1 N1(C(C2=CC(C)(CC)C2)=O)CCC(C2CC2)C1C(=O)N(C1CCC(O)CC1)C CCC(O)CC(=O)NC1(C(N2CCN(C(C)=O)CC2)=O)CC1 C1(CC)CN(C(c2cccc(N)c2O)=O)CCN1C(=O)CC(C)c1cccnc1 N1(CC(N2C(CNC(C(CC=CC)C)=O)CCCC2)=O)CCCC2(CC2)S1(=O)=O c1(OCCC(=O)NC2CC(CCNC(=O)CC3CC=CCC3)C2)cccc(F)c1 C[Si]1(C)CCC(C(=O)NC2CCOCC2O)CC1 C12(NC(CS(=O)(=O)N(C)C)=O)CCCC1CN(C(C1(F)CC3(CCC3)C1)=O)C2 CCC(C(=O)N1CCCC1(C(N1CCCC(O)CC1)=O)CC)C(C)(C)CC N1(C(c2c(CNC(CC3(N(C)C)CC3)=O)cco2)=O)CC(C)(CO)CC1(C)C N1(C(CNC(CC)=O)=O)CCN(C(=O)C(=Cc2cccc(F)c2)F)CCC1C c1(NCC(C)(C)CCN2C(C)COCC2)ccc(S(=O)(=O)NCCO)cc1C#N c1(C(N2C(CN(C(CC(CC)SC)=O)C)CCC2)=O)ccc(S(=O)(=O)NC)o1 CCC(C)(C)C(C(=O)N1CCC(NC(c2cnc(C)n2C)=O)C1)OC c1(C(=O)OC)ccc(C(=O)NC2CCC(C)N(C(=O)C(CSC)OC)C2)c(Cl)c1 c1(CCC)cnnc(C(=O)NC(C)C(CO)NC(=O)COCC(C)C)c1 CCC(C(=O)N1CCC(NC(c2ccccc2C(C)(F)F)=O)CC1)C(C)O C#CCCCC(C)C(=O)NC(CN(C)C)C(=O)N(CC)Cc1ccccc1 Cc1cc(N(C)CCN(C(c2cn(C3CCOC3)nn2)=O)C(C)C)nc(Cl)n1 C1(C(N2CCC(CCN(C)C(C3CC(=O)N(O)C3)=O)CC2)=O)C(F)(F)C12CCC2 c1(CNC(c2sc(Nc3cccc(F)c3)nc2Cl)=O)cccc(OC(F)(F)F)c1 Cn1nc(C(F)(F)F)c(CN2CCC3(CC3C(N3CCC(C)(C#N)C3)=O)C2)c1Cl C(=O)(CCC(c1nnnn1CCCSCC)NC(C)Cc1ccc(C)nc1)NC c1(C(N2CC(NC(C3(CC)CCC3)=O)C(C)CC2)=O)oc2ccccc2c1Cl C(CC(=O)NCC(C)N(C(=O)CN(C)C(N)=O)C)N(CCN)C.CO N1(C(C(=O)NCCC)C2CC2(C)Br)CCC(C2CC2)CC1 N1(C(CCC(C)NC(CN(C(=O)OCC)C)=O)=O)CC2(CC(C)CO2)C1 C(=O)(NCC)NCCSCCN(C)C1CC1 c1(OC)cccc(OC)c1C(N1CC(CNC(=O)C(F)=C(C)C)C(C)C1)=O C(C(=O)NC1CN(C(c2ccncc2NC(F)F)=O)CC1O)(C(C)(C)C)N(C)C Cc1cc(C(=O)N(C2CCCN(C(=O)CCN3CCNC(=O)C3)C2)CCO)n(C)n1 C1(CNC(NCC(C)(C)C)=NCC2CC3(CC3)CO2)CC2(C1)C(F)(F)C21CC1 C1(C)(C(N(CCCCN(C(=O)CCc2cnn(C)n2)C)C)=O)COC(=O)C1 c1(COC)ncc(C(=O)NC2CCCC2CNC(=O)CCc2ccn(C)n2)s1 N1(C(C2(c3cc(C(=O)OC)[nH]c3)CCC2)=O)CCN(C(C)=O)C(C2CCC2)C1 N1(C(CC=C=C)=O)CCC(O)(CNC(=O)COc2ccc(C)cc2C)CC1 c1(OC)ccnc(OC)c1C(=O)NC1CCN(C(=O)C(C)C2CC2)CC1CO C(=O)(CC(C)(O)C(F)(F)F)NCC(C)N(C(c1nc(C)sc1Br)=O)C C12(NC(C3N=C(C)SC3)=O)CCCN(C(c3ccncc3OC(C)C)=O)CC1C2 C1(C#N)(CNC(C(Cn2ccnn2)NC(C(C)SC(C)C)=O)=O)CCCCC1 C(=O)(C(C)C(O)C(C)C)NC1CCCC(CN(C(c2cc(C)ncc2C)=O)C)C1 c1(C(=O)NC2CN(C(C3CC(C)(O)C3)=O)C2)ccc2c(c1)C(=O)OCC2 c1(CNC(C2CN(Cc3cnc(OC)nc3)CC(F)C2)=O)ccc(Cl)c(F)c1Cl N1(C(CCOCCC)=O)CCC(CCNC(C2CCC(c3cc[nH]n3)O2)=O)C1 c1(C(=O)NCCC(=O)NC(C)(C)C=CC(=O)NCCC2CC2)ccc(O)cc1 C(C(CC(=O)N1CC=CC(O)C1)C1CCC1)N.CCC(C(=O)C(COC)=O)OC N1(C(C=CS(C)=O)=O)CC(NC(=O)CSc2cccs2)CC(C)(C)C1 C1(NC(c2ccccn2)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1 N1(C(Cc2nc(CC)sc2)=O)CCC(NC(c2n[nH]cc2Cl)=O)C1(C)C c1(CC(=O)NC(C)CCNC(C2CC2(Cl)Cl)=O)cccc2ccccc12 C(=O)(C1=CC2(CN(C(c3cn(CCO)nn3)=O)C2)OC1)N1C(CO)CCC(C)C1 c1(NC2CCN(CCNC(CC(C)OC)=O)CC2)ncnc2c1nnn2C CCC(C(=O)N(C1CCN(C(=O)CC2(N(C)C)CC2)CC1)CC)C(F)(F)F n1(CCOCC)cc(C(N2CC(O)(CNC(=O)CCc3nccn3C)C2)=O)nn1 CN1N=C(CC(=O)NC2CC3CC(NC(C4CCC(C)(F)CC4)=O)CC23)CC1=O C1(C(N(C)Cc2cn[nH]c2)=O)COCCN(C(=O)C2=CCCOC2)C1 c1(C(=O)NCC(C)N(C(c2c(CC)nns2)=O)C)cnc2c(c1)N(C)CCO2 Cc1cc(C(=O)NC(c2ccccc2)CC2(O)CCCCC2)nc(S(C)(=O)=O)n1 c1(N(C2CNCCC2(F)F)C(C2CC2F)=O)ncnc2c(Br)c[nH]c12 C1(C)(CC)C=C(C(=O)NCC(CCOC)NC(c2ccc(C(C)=O)c(C)c2)=O)C1 CC(C)CC(CNC(c1ccoc1)=O)NC(=O)C(C)OC1COC1 Cc1nn(CNCc2cccc(C)c2)c(C)c1Br.c1(C(=O)N)ccc(C(N)=O)nc1 c1(CNC(c2cscn2)=O)cccc(C(=O)NC2CCC(F)CC2)n1 c1(C(=O)NCCOC(CNC(C(C)=C(C)C)=O)(C)C)csc(C)c1C n1(CC)nccc1C=CC(=O)NC(C)C(C(C)C)NC(=O)COC(F)F CC1(C#CC(=O)NC2CN(C(=O)C(O)c3ccsc3)C2)CCCO1 C(=O)(C1=CC2CCC(C1)C2)NC1(CNC(CSc2n(C)ccn2)=O)CC1 C1(C(=O)NCC2C(CNC(=O)Cc3cn[nH]c3)C2)CCC2(CCOCC2)C1 c1(C(=O)NC2CC3(CN(C(CC(=O)NCC)=O)C3)OC2)cnc2snc(C)c2c1 C(C(O)CC(=O)N(CCCN(C)C(C1CC(c2cccc(Cl)c2)C1)=O)C)N(C)C C=C=CC(C)C(=O)N1CCCC1CC(=O)NCCC(C)CO C1(C(N(CCOCC)C)=O)C2CCN(C(c3cc(OC)cnn3)=O)CC12 CC1(C(F)(F)F)CN(C(=O)CC2CNCCN2)CC1C(=O)O N1(C(c2c(C)csn2)=O)CC(C(=O)NCC(c2ccncc2)C)C2(CC2)C1 CCC(CC(=O)NC1CC(NC(=O)C=C2CCN(C)C2)C(O)C1)C1CC1 C(c1ccnc(Cl)c1)=Cc1ccc(CNC(C(C)(C)C)=O)o1 CCC(C)(C)C(=O)Nc1ccsc1C(N1CCCC1COC)=O CC1C2CCC(C2)C1C(=O)NCCCN(C(=O)C=Cc1ccc[nH]1)C CC1CCCN1CC(=O)NCCNC(CC(C1(CCC(N)=O)CC1)C1CC1)=O c1(C(N(C(CNC(c2cc(C)sn2)=O)C2CC2)C)=O)cc2nccnc2cc1F c1(OC)cc(C(=O)NC2COCC2NC(=O)CCC(C)(F)F)ccc1C#N N1(C(C(C)N(C(C)=O)C)=O)CC2(COC(CNC(C34CCCN3CCC4)=O)C2)C1 C(=O)(C1=CC2(CN(C(=O)C(C(C)CC)N(C)C)C2)OC1)NCc1c(CC)n[nH]c1 c1(OC)ncc(C(=O)NCC(C2CCCN2C(C2(CN(C)C)CC2)=O)(C)C)s1 c1(C(=O)NC(C2(O)CN(c3cnc(C#N)cn3)C2)C)cc(F)c(F)cc1Cl C1(NC(C=CCOCCOC)=O)(CNC(=O)C(N2CCOCC2)C)CCCCC1 N1(C(c2ccc(CC)cc2F)=O)CCCN(C(C2CC2C(F)F)=O)CCC1 n1(CC)cc(NC(=O)CCC2CCCN2C(=O)CCc2ccsc2)c(C)n1 N1(C(c2cn(CC=C)nc2)=O)CC2CN(C(c3ccnc(CC)n3)=O)CCC12 CON(C(=O)C(CNC(=O)C(C)CC(C)C)CC(F)(F)F)C1CCOCC1 c1(C(N2C(C(=O)NCC3(CCOC)CC3)CSC2)=O)cn(C)c(=O)n1C c1(SC)cc(C)c(C(=O)NC(C2CCCN2C(=O)CC2CC(C)=NO2)C)o1 c1(COC(=O)Cc2cccc3occc23)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 c1(C(=O)NCC2N(C(c3scc(C)c3)=O)CCC2C)ccc2ccccc2c1 n1(CC(=O)NC2C(NC(c3c(C)oc(Cl)n3)=O)CCC2)ccc(=O)n(C)c1=O C1(O)(CNC(c2c(C)snc2)=O)CC2CCC(C1)N2C(C1(O)CCCCCC1)=O c1(C(=O)N(C2CCCC2)CCNC(C2CCOC2)=O)ocnc1C1CC1 C1(CC(N2CCC(N(C(COCC)=O)C)C3(C2)CC3)=O)Cn2ccnc2NC1=O CCCC(O)CC(=O)NCC1CC(O)CN1C(c1cc(Cl)cnn1)=O C(=O)(CC1=NNC(=O)C1)NC(CC)CN(C(=O)CCn1c(C)csc1=O)C N1(CC)CCC(c2nc(CC)no2)(CF)C1.C(=O)(C(C)(O)CCO)OC1(C)CCCC1 C(=O)(C1=NOCC1)N1CCC(C(C(=O)NCCN(CCC)C(C)C)F)C1 Cn1cc(CN2CCC3(CC3C(=O)NCCCC(F)(F)F)C2)c2ccccc12 c1(CN(C(=O)CCn2ccnc2)C)ccc(CNC(c2cccn2C)=O)cc1 C12(CCNC(Cc3cccc(COC)c3)=O)CCC1CN(C(C1(C#N)CC1)=O)C2 C1(OC)CCC2(C(=O)NC3CCCCC3NC(C3C4COCC34)=O)CC12 C1(C(C(=O)OC)O)CCN(C(=O)Nc2cccc(-n3cncn3)c2)CC1 C(CNC(c1ncoc1C(C)C)=O)(C(C)(C)C)NC(C1C(CC(C)C)C1)=O Cc1cc2nc(N(CC(C)CNC(=O)C(C)CC(C)(C)C)C)cc(=O)n2o1 O=S(=O)(c1cccnc1NCCc1cc(Cl)ccc1F)NC(CO)CCF n1(CC(=O)NCc2cn[nH]c2)ccc2ccc(-c3c(O)cccc3F)cc12 c1(OC)ccc(CN2CCC(F)(C(N3CCC(C(C)(C)O)CC3)=O)C2)c(F)c1F N1(C(c2nccc(C)n2)=O)CCCC(N(C)C(c2cc(Cl)c(Cl)n2C)=O)CC1 N1(C(c2n(C)cc(C(N)=O)c2)=O)CC(NC(=O)CCC(C)(C)C)C2(CCC2)C1 c1(C(=O)NC(CNC(c2cccc(N)c2)=O)CO)cc(F)cc(F)c1 C1(C(N2CCC(N(C(CC(=C)C)=O)CC)C2)=O)CN(C)CCO1 C1(C(N(C)CC2CCN(C(=O)C=Cc3ccsc3)CC2)=O)CCC2(CCC2)C1 C1(N(C(=O)Cc2cc[nH]n2)CC)CCCN(C(c2ocnc2C2CC2)=O)C1 c1(CNC(C(C2CC2(C)Br)N(C2CC2)CC)=O)ccc(-c2cc(C)[nH]n2)cc1 O=C(CCCCCn1cc(C2CC3(CCC3)C2)nn1)N1CC(C2C3CCCCCC23)C1 CC1CCN(C(C2C3(CC3)C23CC3)=O)CC1NC(=O)CCC(N)=O c1(C(N2CCOC(c3n[nH]c(C)n3)C2)C(=O)NC)ncc(Br)cc1C C=CC(C)(CC)C(=O)N1CC(C(=O)O)C(CNC(=O)COCC2CC2)C1 C1(NC(c2n(CCC)ccc2)=O)CCN(C(C2C=C2C)=O)C12CCCC2 N1(C(CC(CC=C)NC(=O)CCn2cncn2)=O)CCC2(CC1)CN(C)C2 c1(-c2cc(C(=O)NCC34C(CN(C(C(C=C)O)=O)C3)C4)no2)ccc(Cl)cc1Cl c1(C(=O)NC2CN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)cc(F)c(Cl)c([N+](=O)[O-])c1Cl c1(CC)nc2ccccc2cc1NC(=O)C(N1CCC2CCCCC2C1)=O Cc1ccc(S(=O)(=O)N2CC(CC(=O)ON3CC4(CC(N(C)C)CO4)C3)C2)cc1 N1(C(c2cc(OC)no2)=O)CCC(CC(C)NC(C23CSCC2C3)=O)CC1 C1(F)(CNC(C2C(CC)C2)=O)CN(C(C2CCN2S(C)(=O)=O)=O)C1 c1(CN(C2CCN(C)CC2)Cc2c(C)nn[nH]2)cccc(Cl)c1 C(C(C)(O)C(C)(C)C)OC.C(=O)(C1=NOC(C)C1)N1C2(C=CC1)C(=O)NC2 C1(C(=O)NC(CNC(CCCC#C)=O)C(C)C)CC2C(C1)C2(C)C Cc1cccc2c1CC(C(=O)Nc1cc(F)cc(F)c1CO)N2 C1(C(N(CCC)CCNC(C2(C)CC3(CC3)C2)=O)=O)CCN2CCOCC12 C1(N(C(C(C)C)=O)C)CN(C(c2cccn2-c2ncccc2F)=O)CC1F N1(C(C(C)OCCC=C)=O)C(C(N2CC(C(=O)OC)C2)=O)CCC12CC2 N1(C(CSC(C)C)=O)CCC2(CCN(C(C3CCc4n[nH]cc4C3)=O)CC2)C1 C1(C(=O)NCC(C)NC(c2cc(Br)cnc2O)=O)CCCNS1(=O)=O CC(CC(=O)NCC12COC(CNC(=O)CCCCCF)(C1)C2)C(C)(C)C Cc1ncc(CC(=O)NC2(CCCNC(C3COC(=O)N3)=O)CC2)[nH]1 c1(C(=O)NC2(CC(=O)NCC(CC(=O)NC)C)CCC2)cncc(F)c1C C1(CNC(c2cc(Cl)cs2)=O)CN(C(C23CCCC2C3)=O)CCO1 c1(C=O)c[nH]c2ccc(OC)cc2c1=O.N1(C(C=CC=CC)=O)CC(NC)C1 c1(C(N2CCC(C(C(=O)NC(C(=O)NC)C)C)CC2)=O)cc([N+](=O)[O-])ccc1C N1(C(c2cc(C(C)C)on2)=O)CCC(CNC(=O)Cn2cc(CO)nn2)C12CC2 N1(C(C2OCCC(C)C2)=O)CC2(CC2)CC1C(=O)NC1CC1CN(C)C c1(C(=O)NC(CC)CN(C)C(c2cnsc2C)=O)cc(Cl)cn1C C(=O)(CC(C1CC1)NC(=O)CC=CCNC(=O)CC1(N(C)C)CC1)OC C1(CN(CCC)CCC)CCN(c2nc(C)ns2)CC1 c1(C(=O)NCCCCNC(=O)COC2CCS(=O)(=O)C2)ccc(Cl)c(F)c1F CCCC(C#N)C(=O)NCCOC1CN(C(c2cnn(C3CC3(F)F)c2)=O)C1 CC(CN=C(NC1CCC1)N(C)CCc1ccc2c(c1)OCCO2)C(C)(C)C c1(C(N(CCCNC(c2ncc[nH]2)=O)CCO)=O)cc2n(n1)CC(F)C2 Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)N2CC3CC2C3)cnn1 S(=O)(=O)(c1ccn(C)n1)N1C(C)C(c2ccccc2)CC1 C1(C(=O)NCC2C(C)CN(C(=O)C=CBr)C2)C2C3CC4C1C1C2CC3C41 C(=O)(C(O)(CN(C)C)C(F)(F)F)N1CC(CNC(c2c(OC)scc2)=O)C1 N1(C(C=C(C)Cl)=O)CCC2CN(C(=O)CCn3cncn3)CCC2C1 C(c1ccncc1)=CC(=O)NCCC(CNC(C1(CO)CCCCO1)=O)OC C1(CSC)CCN(C(c2csc(Cl)c2)C(=O)NC(C)(C)CC)C1 C(=O)(C(C)(C)N=[N+]=[N-])NCC(CN(C(C1OCCN(CC)C1)=O)C)(C)C C(CC(=O)NC(c1cncnc1)C)(C(C)(C)C)NC(c1ncnc(C)c1C)=O N1(C(C(C2CC2)OC)=O)CC(C(=O)NCc2ccnc(C#N)c2)CC1(C)C C1(C(=O)NC(CC)C(N)=O)CN(C(c2ccc(O)cc2)=O)CC1F C#CC1CN(C(c2nccn2C)=O)CCN1C(c1csc(C(C)=O)n1)=O Cc1c(C(=O)CN2CCOC(c3cccc(F)c3)C2)[nH]c2ccccc12 C(=O)(C(C)(C)C(C)C)NCC(C1CC1)NC(C1CN(CC(C)C)C(=O)C1)=O C1(C(=O)NC(C)C=CC(=O)NCC(=O)N(C)O)CCCC(=O)CC1 CC(C(C)(C)NC(c1cnn(CCO)c1)=O)NC(=O)CCOC1CCC1 C1(NC(=O)C2=CCCCC2)CCN(C(=O)C=C2CCC2)CC(O)C1 c1(NC(N(C2CCN(C(C3CC(=C)C3)=O)C2)CCO)=O)ccc(F)cc1O CCCC(C)(CC)C(=O)NC(CNC(=O)C(C)(C)OC(C)C)CC(F)(F)F Cc1ccncc1C(=O)NC1CC1CNC(=O)CCc1cn(C)nc1C c1(CC(=O)NCCC(C)NC(C2CC(C(=O)OCC)C2)=O)ccncc1 N1(C(C(C)n2ccnc2)=O)CCC2C(CCCN2C(c2cc[nH]c(=N)c2N)=O)C1 C1(C)(CC)CC(C(=O)NCC(C2CCCN2C(=O)CSC(F)(F)F)(C)C)C1 C(=O)(C(=O)CCC(C)C)N(CCN(C(CCc1c(C)nn(C)c1)=O)C(C)C)C n1(CCOC)nc(CS(C)(=O)=O)nc1CCN1CCCCC1 c1(C(N2C(C3CCN(C(COCC)=O)CC3)CCC2)=O)cccn(C2CC2)c1=O N1(C(C=Cc2n(C)cnc2)=O)CCC(C)(C)C1C(=O)NC1CC2CCCC2C1 C1(NC(C(CC=C)NC(=O)CC2CCOC2=O)=O)CCCCCC1C(N)=O C1(C(N(CCNC(C(C(C)C)C)=O)C2CC2)=O)CCN(C)S1(=O)=O C1(NC(c2cccc(NC)n2)=O)CCN(C(=O)CC(C)C2CC2)CC1O Cc1ccc(O)c(C(N2CCC(CNC(=O)CC(C)c3ccncc3)C2(C)C)=O)c1 C1(NC(c2c(CC)c[nH]c2)=O)CC2CCC(C1)N2C(C1CCC(=O)N1C)=O C1(C(N2CCC(C)(NC(C3CCC(F)C3)=O)C2)=O)(COC)CCCCC1 C#Cc1cc(C(=O)NC2CCC2NC(C2CCCCN2C(=O)CC)=O)cc(F)c1 Cn1c(=O)ccn(CC(=O)NC2C=CCN(C(C3CCNC3=O)=O)C2)c1=O C1(CCNC(C2(C)CC2(F)Cl)=O)CCN(C(C2(CC=CC)CC2)=O)CC1.C(N)=O C(=O)(CCCCCNC(c1cnn(C)c1)=O)NC(CC(=O)NC)C N1(C(CN(C)C)=O)CCC1CNC(C1(CCO)CC1)=O c1(CC)c(C(=O)N(C2CC(NC(=O)CC(C)C3CC3)C2)C)cccc1C CC(C(=O)N(CC(C)CNC(=O)COCC1CCOC1)C)OCCN(C)C C1(CCC2N(C(C(C)c3ccsc3)=O)CCC2)CCCCN1C(=O)CNC=O c1(C(C(=O)NCCN(CCC)C(C2CC2C#N)=O)(C)C)c(F)cccc1F N1(C(C2C(=C)C2)=O)CCCCC(C2CN(C(=O)C(O)C(C)CC)C2)C1 c1(C(=O)NCCCCC=C)ccc2c(c1)CN(C(=O)C=CCC)CC2 c1(OC)cccc(C(C)CC(=O)N(CC(C)CNC(c2ncccc2F)=O)C)c1 C1(CC(=O)NCCC(C)NC(c2cn3c(n2)SCC3)=O)CC2C=CC1CC2 C(=O)(C1CCCc2ccnn21)NC1C(NC(C(C(C(C)C)O)C)=O)CCCC1 C1(C(=O)NCC(CCOC)NC(=O)C=CCN2CCOCC2)CC2(CCCO2)C1 C1(C(=O)NCCC(C)NC(C(CC)NC(C)=O)=O)CCC2(CC2)C1 N(C1CCCc2ccc(Cl)cc21)Cc1n(CCc2c(O)cccc2)nnn1 S(=O)(=O)(c1cc(C(F)(F)F)co1)N1CCN(C(=O)C(O)CC(F)F)CC1 C1(NC(c2c(C)ccc(C)c2O)=O)CCN(C(C2C=CCC2)=O)CC(C)(C)C1 CCCC(O)C(=O)NC1CN(C(=O)CCN2CCCCC2)CC1c1ccccc1 c1(NCC(CNC(C2CCC(C(C)C)CC2)=O)C)ncc([N+](=O)[O-])cc1F CC1(NC(c2ccnc(N3CCCC3=O)c2)=O)CC2CCC1CC2=O C1(C2CCC2)(C(=O)NC2(CCCCNC(c3n(CCC)ncc3)=O)CC2)CC1 N1(C(C2N(C(c3cnc(SCC)o3)=O)CC2)=O)CC2C(C)C2C1 CN=c1nc(N(CC(C)OC)C)[nH]c(=NCCOc2c(C)cccc2C)[nH]1 C1(CNC(C(CSC)OC)=O)(CNC(C2(C(C)C)CCOCC2)=O)CC12CCC2 c1(C(C)C)cc(=NCC2CCN(C(c3ccn4ccnc4n3)=O)C2C)[nH]cn1 N1(C(C(CC)(C)OC)=O)CC(S(=O)(=O)N2CCN(CC(C)(C)O)CC2)C1 c1(C(=O)NC2CCN(C(CC(C)OC)=O)C2C(C)C)ccc(Br)c(F)c1C C#CCCCC(C)C(=O)NCc1ocnc1C(=O)N(C)CC1CCOC1 c1(C(=O)Nc2cnc(O)nc2O)nnn2c1CN(C(c1sccc1Cl)=O)CC2 C1(Nc2cnc3cc(C)nn3c2)C2Cc3cc(F)ccc3C12 C(=O)(C(C)(C)C(N)=O)NC(C)CN1CCN(C(C2CC2c2ccccc2)=O)CC1 c1(NCNC(=O)NC(CC)C(=O)O)cnc(O)nc1O N1(C(C2(CC=C)CCC2)=O)CCC2CN(C(=O)C(C(=O)OC(C)(C)C)OC)C2C1 CCC(C(C)C)C(C(=O)Nc1cccc(OC)c1)N1CCSC(C)C1 C(CC(C(C)C)NC(C1CCOC1CNC(C1CC(C2CC2)C1)=O)=O)OC C1(O)(CCNC(CCCCN(C)C)=O)CCN(C(C23CCC(CC2)O3)=O)CC1 Cc1[nH]c(=N)ccc1C=CC(N1CCC1CNC(c1cc2c([nH]1)CCCC2)=O)=O N1(C(C2(CCC=C)CCCCCC2)=O)CC2(CCCC(CO)O2)C1.C(=O)(C1CC1)N C=C=CC1CCCCN1C(=O)Nc1cnc(Br)cn1 CCCCC(F)C(=O)NCCCC(O)C(=O)NCC1CC2(CCC2)CO1 C(C(C)C(C)C(=O)NC1COCCN(C(=O)C(c2c(C)noc2C)C)C1)OC c1(OC(C(=O)NCCCC(C)NC(c2cc(C3CC3)[nH]n2)=O)C)cccc(F)c1 c1(C(N2C(CNC(C(CCC)C)=O)C=CC2)=O)ccc([N+](=O)[O-])c(NC)c1 S(=O)(=O)(c1cnccc1N1CCN(c2nnnn2C)CC1)NCCCCN(C)C Cc1ccc(-c2ncco2)cc1C(=O)NCc1cc(C(N)=O)co1 Cc1cc2cc(NC(c3sccc3NS(=O)(=O)CCCl)=O)ccc2[nH]1 N1(C(C2(C)CCCC2)=O)CC2CC(NC(C3CCC4(C3)CC4(F)F)=O)C(C2)C1 C1(C)(C(N2C(CNC(C3N(C(C)C)C(=O)CC3)=O)CCCC2)=O)CCN(C)CC1 c1(CNC(c2ccc[nH]2)=O)nc2c(s1)CCN(C(C1CC3C=CC1C3)=O)C2 Cc1cncc(C(=O)NCc2ccccc2CN(C(=O)Cn2nnnc2C)C)n1 N1(C(=O)Cc2ccc(-c3nn[nH]n3)cc2)CC2CCCC(C1)N2C1CC1 N1(C(CCCC(C)C)=O)CC(NC(C2CCCS2(=O)=O)=O)C(N=[N+]=[N-])C1 N1(C(CCC)=O)CC2C(CNC(c3cnoc3-c3c[nH]c(C(=O)OC)c3)=O)C2C1 CC1CCC(C(=O)NCC2CCCC2NC(=O)CCc2ncc(C(C)(C)C)o2)O1 N(C1c2ccccc2CC1NC(=O)COc1ccccc1)C(CCS(C)(=O)=O)=O c1(C(=O)NCC2CN(Cc3cccc(O)c3)C2)cc(Cl)c(Cl)cn1 N1(C(CCCC)C)CCC(C2CC(=O)N(C(c3ccoc3)=O)C2)CC1 CCC(C)(CNC(c1csc(C#N)c1)=O)C(=O)NCCCC(=O)NC1CC1 C1(NC(c2c(C)ccs2)=O)CN(C(=O)Cc2ccc3nc[nH]c3c2)CC1C1CC1 c1(N(C)C)ccc(C(CNC(c2cnc(O)o2)=O)NC(=O)CCC2CC2(F)F)cc1 C1(CC(N2CC(C)C(CCNC(=O)C(N)=O)C2)=O)CCOC(C)(C)C1 C12(CNC(C(N3CC(C)C3(C)C)=O)=O)CC3CC(C1)CC(O)(C3)C2 O(N(C)C(=O)CN=C(NCC1CC1)N1CCC(CC2CC2)C1)CC c1(CC(=O)NCc2ccc(C(NOC)=O)o2)nnc(C)n1C CCC(CO)C(=O)NC(CNC(C1(CS(N)(=O)=O)COC1)=O)C(C)C C(C(CN=c1[nH]cc([N+](=O)[O-])c(=N)[nH]1)C(F)(F)F)NC(C=Cc1n(C)cnc1)=O C1(C(=O)NCCNC(C2C(C)C2)=O)CCCN(C(=O)CC2COC(=O)N2)C1 C12(C(=O)NCC=C(C(=O)NCCC(C)OC)C)CC(C#N)(C1)C2 N#Cc1nc(NC2CCC(C3CC3)C2)[nH]c1C#N c1(OC)cc(N)c(C(=O)NCC2CCCCN2C(C2CC3C=CC2C3)=O)cc1F c1(C(=O)NC(CN(C(Cc2cccc(SCC)c2)=O)C)C)cccc(F)c1O c1(C(N2CC3(F)C(NC(C=CC)=O)(CCC3)C2)=O)ccc2c(c1)C(=O)N(C)C2=O C(=O)(C1CCc2nccn21)NCC1(F)CCN(C(CCC(CC)CC)=O)CC1 C1(NC(=NCC)NCC(c2ccc(F)cc2)(F)F)CC1C1CCCC1 C(=O)(CC(C)CC(=O)N1CCN(C(c2[nH]cc(C)c2C)=O)CC1C(F)F)OC C#Cc1ccccc1C(N1CCC(C)(C)C1C(=O)NCC1(C#C)CCCCC1)=O c1(C(=O)NCC(c2ccccc2)NC(CC=CC)=O)nn[nH]c1Cl c1(OC)cc(C(=O)NCCC2CN(C(c3cc(CN(C)C)n(C)n3)=O)C2)ncn1 C1(NC(CC2N(C)CC=CC2)=O)CCCCCC1NC(c1ccc(Cl)cc1)=O c1(C(=O)NCC(C2CCCC2)NC(c2c(C)ocn2)=O)c(F)ccc2c1OCC2 CC1(C)CCCN(C(=O)CC2C=CCCC2)C1C(=O)NCc1ccc(C#N)cn1 Cc1cc(C(N2CC3CC2CN3C(c2cn3ccnc3s2)=O)=O)cnc1C Cc1nc(C(=O)N(CC(C)NC(=O)C(C)(O)C2CC2)C)sc1C c1(C(=O)NCC(CNC(=O)COc2cccc(C)c2)OC)ccc(C)c([N+](=O)[O-])c1 c1(C(=O)NC(C)C(C)(C)C(=O)N(CCN=[N+]=[N-])C)cc2cccnc2[nH]1 C1(CC)CCN(C(c2cnns2)=O)C(C(=O)NCC(C)(C)C2(O)CCC2)C1 N1(C(CC2(C)N(C(c3c(C)c(F)ccc3)=O)CC2)=O)CCC2(CCCO2)C1 C1(CCNC(C(CSc2ccccn2)NC(CC(C)C)=O)=O)CCCC1(C)C c1(C(=O)NCCN(C(CNC(C)=O)=O)CC(C)O)cscc1C#N Cc1nn(C)cc1CN(CCC(=O)N(C)Cc1ccc(OC(F)F)cc1)C C1(C(=O)NC2CC(CNC(CCc3ccc(NC)cc3)=O)C2)CC(=O)NC(=O)N1 Cc1cc(C(=O)NCCC(C)NC(=O)C2=CCOCC2)cnc1OC(F)F c1(C(=O)NC2C(CNC(c3c(C)noc3C)=O)CCC2)cnn2c1NCC(C)C2 c1(CC)cc2c(N3CC4C(CNC(C5CCCO5)=O)C4C3)nc(C)nc2s1 C1(CNC(C=CCC)=O)CCC12CN(C(=O)CCNc1ccc(F)cc1)C2 CC1(C)CC(C(N2CCCC(CCF)C2)=O)CCN1C(c1ccc(N)c(F)c1)=O C1(C(=O)NC(CN(C(=O)COc2ccccc2)CC)C)CCCN2CCCC12 C1(CNC(C2CC(N(C(C(C3CC3)SC)=O)C)C2)=O)COCCO1 c1(N)ccc2[nH]ccc2c1.N1(C(c2c(C(=O)O)cco2)=O)CC2(C1)CC2(F)Br c1(CNC(=O)NC2CC(c3cc(C)[nH]n3)CC2O)cc(C)c(C)c(C)c1 c1(C(=O)NC(C2C(c3cccc(C)c3)C2)C)sc2c(Br)cccc2c1C C1(NC(Cn2ncc(C#N)c2)=O)CN(C(=O)Cc2ccsn2)CC2CC12 C12(C(=O)Nc3cnn(CC)c3C)CCCC1CCN2C(=O)Cc1ccn(CC)n1 c1(CN2CC(NC(c3c(C(C)C)cccc3)=O)C(F)(F)C2)c(F)cc(Cl)cc1Cl C12(C(N3C(C)CN(C(=O)C(=O)c4ccco4)CC3)=O)C3C4C1C1C2C3C41CO c1(NC2CCCCN(C(C3(C)CCCOC3)=O)C2)ncc2c(n1)CCCCC2 O=C(N=c1ccc2nnc(C(F)(F)F)n2[nH]1)c1ccc(Cl)o1 C1(C(=O)NCC(C(CC)C)CO)CC2(CCN1C(C1COCCC1C)=O)CC2 C#CCCCC(C)C(=O)NC1(C)CN(C(=O)CCNC(=O)CCC(C)C)C1 N1(C(c2c(C)cccn2)=O)CC2(C1)CN(C(c1cc(Br)cn1C)=O)CCO2 C(=O)(N=c1cc(C)n(C(C)C)[nH]1)C1C(CNC(c2c(F)ncc(C)c2)=O)CCC1 C12(C(N(C)CC3CCCN3C(C3CC4CC(=O)C3C4)=O)=O)CCCC1CS(=O)(=O)C2 C1(NC(c2ccc(C#C)o2)=O)CC2CC1N(C(c1c(Cl)cnn1C(C)C)=O)C2 c1(-c2cc(F)c(OC)c(F)c2)cc2c(s1)CCN(Cc1cn[nH]c1)C2 C1(NC(CCC(C)OCCOC)=O)CCN(C(=O)CSCc2nc[nH]n2)CC1O C1(C(=O)Nc2cnc(OC)nc2)N(C(=O)C(O)Cn2cncn2)CCCC1(C)C c1(C(=O)NC2C(NC(C(N3C(=O)CCC3=O)C)=O)CC2)c(N)sc2c1CCC2 C(=O)(C1OC(=O)c2ccccc21)N1C(CNC(CCC(=O)NC)=O)CC(C)(C)C1 C1(O)(CC(=O)NCC2C(C)CCN2C(c2cc(C(N)=O)[nH]n2)=O)COC(C)(C)C1 N1(C(C(C(C)(C)C)SC)=O)CCN(C(c2csc(C)c2C)=O)CC(C)C1 N1(C(=O)NC2CC23CC3(F)F)CCC(C2CCOCC2)C1 CC1(C)COC(C(=O)NC2CCC(NC(=O)C3=CCOC3)CC2)CO1 C(C)(C(CC(=O)N1CCSCC(C)C1)NC(=O)CC1CNC(=O)O1)OC C(Cc1cnc[nH]1)(C(=O)N(CCC(=O)N)OC)C(C(CCCC#C)C)=O C1(C(N2CC3N(C(C=COCC)=O)CC(C3)C2)=O)CCc2c(nnn2CC)C1 C#CC1(C(=O)NC(CO)CCC)CCN(C(c2ccc[nH]2)=O)C1 c1(C(=O)NC2CC(CNC(C3(C)CCN(C)C3=O)=O)C2)ccn2[nH]c(=N)nc2c1 c1(C(N2CCC(NC(C(CC(=C)C)C)=O)C2(C)C)=O)cc2c(s1)CCC(C)(C)C2 c1(C(c2cc(-c3nc(C4CC4)no3)nn2CC(C)C)OC)ccc2c(c1)C(=O)OC2 N1(c2n(CC(C)C)c(-c3cc(C4CC4)[nH]n3)nn2)CCOC(C)(C2CC2)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)NCC1N(C(C(CC)F)=O)CC(O)C1O c1(C(=O)NC2(C)CC(NC(c3n(CC)nnc3)=O)C2)cc(Cl)ccc1Br c1(C(=O)NCC(=C)CCNC(C2COC(C)C2)=O)cc(Cl)cc(Cl)c1Cl N1(C(Cc2c(C)occ2)=O)CCC(NC(C23CC(CN2C2CC2)C3)=O)CC1C C(N=c1nc(O)c2c(ncn2C)[nH]1)C1(NC(C2CCC(=O)NC2)=O)C(C)CCC1 N1(C(CC2C(C)(C)CC2)=O)CCC(C)(CNC(=O)C(O)C2CCCC2)C1 CN1CCN(C(c2ccsc2C#N)=O)CC1C(=O)N(CC(O)C1CC1)C1CCC1 C1(OC)CC2(CCC(Nc3ccccc3Cl)CC2)C1.N12CCN(CC1)CC2=O C1(C(N2C(NC(Cc3c(C)nsc3)=O)CC2)=O)CCCN(c2cc(O)ncn2)C1 C(C(C)(F)C(C)(C)F)n1cc(N2CCCC(NCc3n(C)c(Br)nn3)C2=O)nn1 c1(C(=O)NCC2CC(C)N(C(C3CCCS(=O)(=O)C3)=O)C2)nc(=O)cc(N)[nH]1 c1(OC)ccc(C)c(C(=O)N(CCNC(c2ccc([N+](=O)[O-])s2)=O)CC2CC2)c1 c1(C(=O)NC(C2(O)CN(C(c3nc(COC)[nH]n3)=O)C2)C)ccccc1Cl C1(NC(CNC(=O)OC)=O)CN(C(C2(n3cccc3)CCCC2)=O)CC12CC2 S(=O)(=O)(c1ccc(Cl)c2nonc12)N1C(CC(=O)OC)COC(C(F)(F)F)C1 CC1(NC(=O)C(F)=CC2CC2)CCCN(C(c2cnc(N(C)C)cn2)=O)C1 N1(C(C2(CC)CCC2)=O)CCOC(C(=O)NCCc2ncccc2F)C1 N1(CCC)CCCCC1C(=O)NC(CNC(=O)CSCc1ncc[nH]1)CCOC N1(C(C(C)SC)=O)C2CCCC1CC(NC(C1(C(F)F)CCC1)=O)C2 N1(C(C2CN(C(=O)OC)C2)=O)C(=O)NC(c2cncn2C)C2=C1C(C)N(C)C2=O Cc1ccc(C=CCCCSCC(=O)OC(C2CC3C=CC2C3)=O)s1 c1(C(N(CC(N2CCC2CC(=O)NC)=O)CC)=O)ccc(F)cc1F c1(-c2nc(C(CCC)C)nn2C2CSC2)cc2ccc(Br)cc2s1 CCC(CC(F)F)C(=O)NC(c1ccccc1)CNC(=O)Cc1cn[nH]c1 Cn1nc(CN2CCCC2)c2c1CCN(C(=O)NC(C1(C#N)CCC(=O)N1)=O)C2 C1(CNC(=NCc2cc(C)on2)NC(CO)CCF)CCC2(CCC2)O1 c1(Cc2c(C)cc(C(=O)Nc3cccc(C(=O)OC)c3)s2)cc(Cl)c(Cl)nc1Cl C1(NC(c2n[nH]c3c2CCSC3)=O)CC2CC(C1)N(C(C1CCCCO1)=O)C2 CC1CCCC(C(=O)NCC2CN(C(c3cccc(F)c3)=O)C2)CC1 CC1CN(C(c2nccnc2Cl)=O)CCC1CNC(c1c(Cl)cnn1C)=O C1(NC(c2nc(CCC)oc2)=O)CC2CCC(C1F)N2C(C1CC(C)(O)C1)=O CC(C)CC(C(=O)NC12CC(CN(C(=O)C(C(C)C)NS(C)(=O)=O)C1)C2)C(C)C c1(C(=O)NC2CN(C(C(C(C)C)(C)O)=O)CC2F)noc2c1CC(C)(C)CC2 N1(C(c2cnn[nH]2)=O)CC2C(NC(=O)C(F)(F)c3nccs3)C2C1 c1(N(C)CCO)ccc(F)cc1NC1CCN(C(=O)CN=[N+]=[N-])C1 c1(-n2ncc(NC3(C(=O)OC)CCN(C(=O)C(F)(F)CO)C3)c2)c(F)cccc1F n1(CC(=O)NCCCNC(=O)CC2CCCCC2F)c(=O)cnc2ccccc12 S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1CCN(C(C2CCC(Br)CC2)=O)CC1 Cc1ccsc1C=CC(=O)NCC(F)CNC(=O)CCNc1nnnn1C N1(CC)CCOCC1CC(=O)NC1CCCC1NC(c1ccn(C(F)F)n1)=O N1(C(c2cc(C)cc(C)n2)=O)CCC2CN(C(=O)C(C)(O)CC(C)C)CC12 c1(C(N2CCC(CN(C(C(C)CN(C)C)=O)C)C2)=O)ccc2c(c1)N(C)CC2 c1(OC)ccc(CN(C2CS(=O)(=O)CC2O)Cc2nc(C(C)C)no2)cc1Br CCC(C)(CNC(c1sccc1C)=O)C(=O)N(CC(C)COC)C N1(C(CC(C(F)F)NC(c2c(OC)csc2)=O)=O)CCc2cccnc2C1 CCCCC(CCCC)C(=O)NCCC(O)CNC(c1cnc(C2CC2)[nH]1)=O n1(C(C)C)cccc1C(=O)N(CC(C)NC(=O)CC1CC12CC2)C C(CCCC(=O)NCC(c1ccc(C)cc1)NC(=O)C=C(C)C(F)F)(OC)OC c1(OCC)cccnc1C(=O)NCC1CCCN(C(C2(O)CCOC2)=O)C1 c1(OCC(N2C(CNC(C(CC=CCC)C)=O)CC(F)C2)=O)c(F)cccc1F CCCCCC(O)CC(=O)NC(C)C(C)(C)C(=O)N1CC2(CCC2O)C1 N1(C(c2cccc(N)c2Br)=O)CCC2(CCN(C(c3cc[nH]n3)=O)CC2)C1 c1(C(=O)NCC(CCNC(C(COCC)C)=O)O)cc2ccc(C)cc2[nH]1 N1(C(=O)Nc2ccc(C)c(I)c2)CCCC2(CCCO2)C1 C1(C(=O)NCCNC(=O)OC)CN(C(c2ccc(C#N)cn2)=O)CCN1C C1(C(=O)NCC2CC(C)N(C(C3CC=CC3)=O)C2)CCS(=O)(=O)C(C)C1 C(=O)(C1Cc2c(Cl)cccc21)NCC1C(C)CN(C(=O)CCOCC2CC2)CC1 C1(CNC(C(C2CC2)SC)=O)CCC2CN(C(=O)C(C#N)CC)CC12 c1(C(=O)NCC#CC)ccc(CNC(=O)C(C)c2cccs2)cn1 CC(CC(=O)NC(C(N1CCC(CCCO)CC1)=O)c1ccoc1)CC(C)(C)C c1(NCCC(C)OC)cc(C)c(S(=O)(=O)N2CCCC(CO)CC2)cn1 C(C(C)CC(=O)NCc1cnnn1C)NC(CC1C(CC)C1)=O c1(C(C)C)ccccc1OCC(C)COC1CC(N2CCOC(C)C2)C1 C1(NC(c2nc(COC)sc2)=O)CCCC(N(C(=O)CN2CCN(C)CC2)C)C1 c1(C(N2CCC(NC(C(CN(C)C)N(C)C)=O)C2)=O)cc(F)c2[nH]nnc2c1 C1(CNC(Cc2cc(C)n(C)n2)=O)CN(C(c2c[nH]nc2C(F)F)=O)C(C)(C)C1 n1(CC)ncc2c1CC(C(N1CCC(CN(C(=O)CN(C)C)C)C1)=O)CC2 c1(OC)ccc(C(=O)NC(CNC(c2coc3c2COC3)=O)C2CCC2)cc1O c1(C(=O)NCCC2CCN(C(=O)C=CBr)CC2)cc2c(=O)[nH]ccn2n1 C1(N(C(CC)=O)C)CCCN(C(=O)C=Cc2ccc(I)o2)CC1 CCC(C)(COC)C(=O)N1CCCC(CO)(NC(c2ccc(N)cc2OC)=O)C1 c1(NC(C)=O)ccc(C(N2CCN(C(=O)CC3=CCCC3)CC2CF)=O)cc1F C(C)(C(C)(C)C(=O)NC1CCN(C(=O)CSC(C)C)CC1)NC(C)=O c1(NC(NCC(CC)(C)CO)=NC)cc(C)c(Br)cn1 C1(N(CC(CC)OC)C)CCCN(C(c2cc(C)c(Cl)s2)=O)C1 c1(C(N(C2CN(C(c3ccc4ccoc4c3)=O)C2)C)=O)nn(C)cc1[N+](=O)[O-] c1(C(N2CCN(C(CN(C)C)=O)CC(C)(F)C2)=O)cccc2c1OC(C)(C)C2 c1(-c2nc(C(c3c(F)ccc(C)c3)C(C)C)on2)cc2c(s1)CCCC2 c1(C(=O)NC2C(NC(C(=O)NC(C)C)=O)CC2)cocc1Br c1(OC(c2ccc(CCC)cc2)C)ccnc(O)c1C=O C1(CNC(c2ocnc2C2CC2)=O)CC2(CCN(c3nnc(O)s3)C2)CO1 Cc1cc(Br)c(C(=O)NCC2C3CN(C(c4coc(C#N)c4)=O)CC23)s1 CC(C)S(=O)(=O)CC(=O)NCC1CSCC(CO)C1 C1(N=[N+]=[N-])(C(=O)NCc2c(C)cccc2F)CCN(C(C2CC2C(F)(F)F)=O)C1 C(=O)(C(C)C(C)(F)F)N(C1CCN(C(CCn2c(C)ccc2C)=O)CC1)C C(C(C)C(F)C(=O)NCC1(C)CCCC1)NC(C(CC)C#N)=O C=Cn1nncc1C(=O)NCCN(CCOCCO)C(C1C(F)(F)C12CC2)=O C(N=c1nc2scnc2c(N2CCSC(C)CC2)[nH]1)c1cc(C)oc1C N1(CC2(NC(Cc3nnc(C)o3)=O)CC2)CCN(C(=O)C(C)(Cl)Cl)CC1 Cc1ccc(C(N2CC(O)(CNC(=O)C(C(C)C)c3ccccc3)C2)=O)cc1C Cn1ncc2c(NCc3cn4c(n3)SCC4)[nH]c(=NCCC3CCOC3)nc12 C(CC(C)(C)C(F)F)NC(CC1CCN(C(c2ccc(OC(C)C)cc2)=O)C1)=O c1(OC)ccc(S(=O)(=O)NC(C(=O)O)C2(CC(C)C)CC2)c(C(F)F)c1 c1(CC)ccccc1NN1CCN(C(N2CC(COC(C)(C)C)C2)=O)CC1.O S(=O)(=O)(c1cc(Nc2sc(-c3ncnc4c3CCCC4)nc2C)n(C)c1)NC Cc1ncc(C(N2CCCC2CCNC(=O)CC(O)C(C)C)=O)cc1N C=CC1CCN(C(=O)C(CCC2CC2)NC(c2cnc(C)nc2)=O)C1 C123CCC(CC1)(CO2)C(=O)NC3.C1(C(=O)NC2C(COC)C2)CC(C(F)(F)F)C1 C1(NC(c2nc(C(=O)OC)oc2)=O)CCN(C(c2ccoc2C2CC2)=O)CC1(C)C C(N=c1nc(OC)c(F)c(C)[nH]1)C1C2CN(C(c3c(CC)cncc3)=O)CC21 C1(NC(=O)N(CCCCCCC2CC2)c2ccccc2)C2C3CCC(C3)C12 N1(C(C(CSC)O)=O)CCCC(C(=O)N(CC(C)O)C)C1 N1(C(CCn2cnc(=N)[nH]2)=O)CCCCCC1Cc1cn(CCCO)nn1 c1(C(N(CCCC2(N3CCCC3)CCCC2)CC)=O)cnc(C)c(C)n1 Cc1nn(CCO)c(C)c1-c1cccc(C(F)(F)F)c1.N12CCC(C1)C2=O c1(CCCC(=O)NC2CN(C(C3C(C)C3)=O)C2)ccc2c(c1)Cc1ccccc1-2 c1(OCCNC(c2n(CC)nnc2)c2nnnn2C)cc(F)ccc1C CC(C)C1=CCC(C(=O)NCC2(NC(=O)COCc3nc[nH]n3)CCOC2)CC1 c1(NC(C2CCN2C(c2cnccc2Cl)=O)=O)cccc(Br)c1Cl C1(C(N2CC(NC(CC3(CC)CCC3)=O)C(OC)C2)=O)CCC(C2CCC2)CC1 c1(OC)ccc(F)c(F)c1CN1CCC(CC(=O)NCCCCCCO)CC1 C1(C(N2CCC(O)(CNC(C3CCN(C(=O)NC)C3)=O)C2)=O)(CC)CCCCC1 c1(CC(N2C(C3(NC(CN(CC)CC)=O)CC3)CCCC2)=O)ccc(F)cc1C N1(C(C2(C)CCC2)=O)CCN(C(c2ncccc2Br)C(=O)NC2CCOC2)CC1 CC#CC1CCN(C(=O)CCC2CCC(NC(=O)C3=CCCC3C)C2)C1 c1(C(=O)NC2CC(C)(C)CN(C(=O)C(C)(C)CC#N)C2)c(Cl)oc2ccccc12 C(=O)(NNc1cc(I)ccn1)NC(CC(=O)O)Cc1ccc(F)cc1 C(=O)(C1=COCCO1)N1C(C2CCN(C(CN(C(COC)=O)C)=O)CC2)CCC1 c1(OC)ccc(Cl)cc1CC(=O)N(C)Cc1c(C)nn(C)c1C N1(CC2CN(C(C3C(CC)C3)=O)C2)CCN(C(=O)COC)CC1 N1(C(C(C)(C)c2ccno2)=O)CC(NC(C2(CCO)CC2)=O)C(N=[N+]=[N-])C1 C=CCC(CC(=O)NC1CN(CC)C1)NC(=O)C(C)COC c1(C(N2C(C3CCN(C(C(C)C)=O)C3)CCC2)=O)cnc2ncnn2c1N CC(C)(C)C(CNC(=O)CCN1CCCCC1)NC(C12CCCC1(C(N)=O)C2)=O C(CC(F)CN=[N+]=[N-])NC(C(C)(CO)NC(CC1ON=C(C)C1)=O)=O c1(C(=O)NC2(COC)CCN(C(C(CCC)OCC)=O)C2)cccc2c1COC2 c1(OC)cc(C)c(C(N2CC3CC2CN(C(C2(C)CC2Br)=O)C3)=O)cc1OC c1(C2(C(=O)NCC(C)CN(C(=O)CN3CCCC3C)C)CC2)ccccc1Cl N1(C(c2c(C)nns2)=O)CCC(F)(C(=O)NCCN(C)CCO)C1 C1(C(=O)NC(C#C)C)CC12CCN(Cc1ncc(Cl)cc1Cl)CC2 C1(CNC(CC(CC)C)=O)CC2CN(C(c3ccc(C)nc3)=O)CC12 c1(C(N2C(C#N)CC(F)C2)=O)csc2c1CCN(C(c1ccc(Br)cc1O)=O)C2 C1(CC(=O)NCc2occ(C(N(C)Cc3cnn(C)c3)=O)c2)CC2(CCO1)CC2 c1(C(N2C3C(C(=O)Nc4ncc(C)c(Cl)n4)C(C3)C2)=O)ccc2c(c1)NC(=O)C2 N1(C(C(c2cccc(C)c2)NCC(F)(F)F)=O)C2C=CCC1CC2 C(CCCCCC(=O)NC1CCCCC1O)NC(CCC(C)(C)OC)=O C1(CNC(c2c(CC)con2)=O)CCN(C(C2CC(OC3CC3)C2)=O)C12CCC2 Cc1cccc(N2CCC(CNC(=O)CCC(C)N(C)C)C2)c1C C(CCCC(=O)NCCC(C)(C)CNC(=O)C(c1ccc(F)cc1)=O)N(C)C C(C)(C)(C(=O)NCCN(C)C(C1(O)CC(c2ccccc2)C1)=O)OC(C)C C1(C(=O)OC)CCCCC1C(=O)NC1CCCC1CNC(=O)CCCNC(N)=O c1(C(N2CCC(NC(CCC(=O)NC)=O)CC2C2CC2)=O)ccc([N+](=O)[O-])cn1 C1(N(C(=O)C=Cc2cscn2)C)CCCCN(C(C2CCC23CCC3)=O)C1 C12(CNC(C=CCC)=O)CCC(CC1)N(C(=O)C(C)(Cl)Cl)C2 c1(CNC(COCCOCC#C)=O)ccccc1CNC(=O)C=C1CCC1 CC1CCN(C(=O)CC2CCSC2)C1CNC(c1nccc(C(F)(F)F)n1)=O c1(OC)ncnc(C(=O)NC23COC(CNC(=O)COC4CCCC4)(C2)C3)c1F C(c1c(C)noc1C)=CC(=O)NC(CCOC)CNC(c1cc(C(F)F)[nH]n1)=O C1(C(N(C)CCNC(c2ccc(C(F)(F)F)cc2)=O)=O)CC2CCCCC2O1 CCC(CC(=O)N1CC(C2CC2)C(F)(C(=O)NC)C1)C(C)(C)C C(=O)(C(CC(C)C)C(N)=O)N1C(CNC(C2CC(C#N)(OC)C2)=O)CC1 Cc1ccc(F)c(C(=O)NC2(CNC(=O)Cc3cc(Cl)cs3)CCC2)n1 CCCCCCCCOCC(=O)NCC#CCNC(C1(O)CCN(C(C)=O)C1)=O c1(C(=O)Nc2cc(C(=O)O)ccc2C(F)(F)F)c[nH]c(=O)c2ccnn12 c1(C(C(=O)N(C2CN(C(C(C)OCCC#C)=O)C2)C)N2CCCC2)ccccc1 c1(OC)cncc(C=CC(N2CCCC2CCCNC(C23CC(C)C2C3)=O)=O)c1 c1(OC)c(C(N2CCC(O)C(NC(c3csc(C(C)C)n3)=O)C2)=O)c(C)nn1C N1(C(C2C(OCC)C2)=O)CCOCC(C)(CNC(c2nc(C)sc2C)=O)C1 c1(C(C(=O)NC(CC)C)N(CC(C)C(C)C)CC)cc(Br)cs1 C1(C(N2CCC(c3nc[nH]n3)CC2)=O)CC2CC1CC2(F)F c1(C(=O)NCC2CN(C(CCn3c(C)cc(C)n3)=O)CC2C)cc([N+](=O)[O-])no1 Cc1cn2cc(CC(=O)NCCCNC(=O)C(C)(C)c3cnsc3)nc2s1 CC1CCCc2nc(C(=O)OCC3NC(=O)NC3=O)cn21 C1(CC(N2CC(C#C)C2)=O)CC(C)(C)CN1C(=O)C(CC=C)CCl Cc1[nH]nc(C(C)C)c1C(=O)NCC(C)(CO)NC(C1CCCS1)=O C1(N(C(C)Cc2ccccc2)C(c2cc(C)no2)=O)C2CCC1CNC2 Cc1nnccc1C(=O)NC1COCCC1NC(c1cc[nH]c1C1CCCC1)=O c1(OC)cc(C(=O)NC(C)CC2CN(C(C3(CF)CCC3)=O)C2)ccn1 Cc1ccnc(O)c1C(=O)NCC1CCCCC1NC(c1csc(C2CC2)n1)=O CC1(C(=O)NCCN(C2CCCCC2)C(C2(C(F)F)CCCO2)=O)CCNC1=O C(=O)(CCC(=O)NC1CC(CNC(c2coc(Cl)n2)=O)C1)OC(C)(C)C C(CN=C(NCc1c(F)cccc1Cl)NCC1(C)CCCCC1O)OCC N1(C(CN(C)C2CC2)=O)CCC(CNC(=O)COCC2CCCO2)C12CC2 C123CC1CN(C2)C3=O.c1(C(=O)OC)cccc(C2CC2)n1.C123CC(C1)(C2)CNC3=O C(=O)(C1CCCc2ccnn21)N(CCN(C(CC(C)P(C)(C)=O)=O)C)C(C)C n1(C2(C)CC2)nnnc1C(C1CCCSC1)NCCC1CC1 c1(N(CCNC(C=CCC)=O)CC2CC2)cc(C(=O)OC)ncn1 c1(CCCC)ccc(C(C(=O)NCC2CCCO2)N(CCC(N)=O)C)cc1 C(C(C(=O)NC1CC(F)(F)C1)C(C)C)NC(COCCSC)=O Cc1scc(C(=O)NC(C)CNC(=O)C(c2ccc(Cl)cc2)C)c1N CCC(CN(C)C(C1CC(NC(C)=O)C1)=O)N(C)C.C12(CC1)C(=O)N2 c1(CC(N2CC(C(C)NC(=O)CCc3cscn3)C2)=O)c(F)cccc1Br CCCC(O)(CCC)CC(=O)N1CCCC1CNC(=O)CCc1cccc(C)c1 CC1(NC(c2cccnc2O)c2nnnn2CCCF)CCOC1C1CC1 c1(C(=O)NCC2CC(F)(CNC(=O)Cc3ccoc3)C2)cc2cccnn2c1 c1(C(C(=O)NCC(F)F)N(CCCn2ccnc2)CC)ncc(C(C)(C)C)o1 c1(C(=O)NCCC(CNC(CC(C)SC)=O)O)ccc(C2CC2)c(Cl)c1 C1(CNC(C2CC(C#C)(O)C2)=O)CC2CCCC2N1C(c1ccn(C)c(=O)c1)=O c1(C(=O)NCC2(F)CC(CNC(=O)NC3C(CC(C)C)C3)C2)cc(Cl)cnn1 c1(C(N(C)CC2CCS(=O)CC2)=O)nc2ccccc2[nH]1 Cc1ccc(OCCC(N2CCOCC2c2ccccc2Br)=O)cc1 C1(C(N2CCN(C(c3nc(C)n(C)c3)=O)CC2)=O)CC(O)c2ccccc2O1 O=C(CCCCC(F)F)NC1CCC12CN(C(c1cc3c(s1)CCC3)=O)C2 C12(C(=O)NC3C(NC(CN(C)C(N)=O)=O)COC3)CCN(CC1)CC2 C1(CNC(C(C)(C)CO)=O)COCCN(C(=O)CCc2ccc(N)cn2)C1 c1(NC(=O)CCC2CCCO2)cccc(CNC(c2cc[nH]n2)=O)c1 CC1CC(C(=O)N2CC3(CC(CC(=O)NC4(C)CCCCC4)C3)C2)=NO1 Cn1ncc(C(N2CC(NC(=O)Cn3cccn3)C(CO)C2)=O)c1N c1(C(=O)NCC2(NC(c3ccc(CC(N)=O)cc3)=O)CCOC2)cncc(O)c1 N1(C(C=C)=O)CCCC1(C)CNC(c1cc(C(F)(F)F)nn1CC)=O C1(C(C)NC(=O)Cn2ncnn2)CCCN1C(=O)Cc1ccns1 N1(C(c2cccc(CC)n2)=O)CC2C3CCC(C(NC(c4cc[nH]n4)=O)C3)C2C1 c1(NCCC2(C)CC2(Cl)Cl)cc(S(=O)(=O)N(CCCCO)CC2CC2)ccc1C#N N1(C(C(C)SC)=O)CCC(NC(=O)CC(c2cccc(F)c2)C)C1(C)C C(CCN=C(NCc1ccnc(C2CC2)n1)N1CCC(c2cccnc2)C1)SC C1(C)(NC(C2C(C)(C)OCC2)=O)CCCCC1C(=O)NOC1CC1 CC1(C)CC1S(=O)(=O)N(CCO)Cc1ccc(Br)cc1 CCCCCC(O)C(=O)N1CC(F)CC1CN(C)C(c1sccc1Cl)=O c1(C(N2CCCCC(NC(=O)C(F)CC3CC3)C2)=O)cc(O)nc2c1CCCN2 CC(C)(F)C(C)(F)C(=O)N1CC(NC(c2ccon2)=O)C(C)(C)C1 Cc1cccc(C(N2CCC(NC(c3cnn(C(C)(C)C)c3)=O)C(O)C2)=O)c1I C1(O)(CC(=O)N(CCCCNC(C(C)CO)=O)C)CCCOC1 CC1(F)CCC(NC(=O)CN2CC(Oc3ccc(F)cc3)C2)CC1 c1(OC)cc(CC(=O)NCC2CCN(C(=O)Nc3nnn(C)c3C)C2)ccc1C c1(C(=O)NCC2CCC(CNC(COCC)=O)CC2)[nH]c2cc(C)ccc2c1C c1(NC2C3N(C(c4ccc(C)cc4)=O)CC(CC3)C2)nc(C)c([N+](=O)[O-])cc1Cl C1(NC(=O)C2=CCS(=O)(=O)C2)CCC2CN(C(C34CC(C3)C4)=O)CCC2C1 CCCC(C)(CCC)C(=O)N1CCN(C(=O)C(O)CCN(C)C)C(CCOC)C1 CCS(=O)CC(=O)N(C1CCCC1)CCNC(c1ccc(Cl)cc1)=O CCC(CC(=O)N(C1CCOC1)CCF)NC(c1cc(C)on1)=O N1(C(C2CCC=CO2)=O)CCCC(O)(Cn2cc(-c3cccnn3)nn2)CC1 N1(C(C(CC)N(C)C)=O)CCC(CO)C(NC(C2(OC)CCOCC2)=O)C1 N1(C(CC2CCC(NC(C(C)C#N)=O)C2)=O)CC2C=CC1CC2 C1(CC(=O)NC2CCN(C(CCCC=C)=O)CC2)SC2=NCCN2C1=O CC1=NOC(C)(C(=O)N(CCCNC(=O)C(c2ccncc2C)C)C)C1 C(=O)(C1Cc2ccccc21)N1CCN(C(C2(F)C(C)(C)C2(C)C)=O)CC1C1CC1 C(=O)(CCCCC(N)=O)NC(CN(C(c1ccc(OC)c(Br)c1)=O)C)C C1(OC)CN(C(=O)CCCCN(C)C)CC1NC(=O)CC1COCCOC1 Cc1sc(Cl)nc1C(=O)NC1CC1NC(=O)CC(O)c1cnc(Cl)s1 N1(C(c2cnc(CC)[nH]2)=O)CC2CCN(C(=O)CC(c3ccccc3F)C)C2C1 Cc1cn(C)nc1C(=O)NC(C1CCN(C(=O)CCc2nc(C)c(C)[nH]2)CC1)C C12(C)CCN(C1)C(C1CC1C)C(=O)OCCNC2=O.n1(CCC)cc(CC)nn1 c1(NC2CC(CNC(c3c(C(C)(C)C)ncnc3)=O)C2)c(Cl)cncc1[N+](=O)[O-] C(C(C)(C)C#CC(=O)NC(C)Cc1ccccn1)NC(c1cc(COC)on1)=O C1(F)(CNC(C(CC)(C)O)=O)CCCN(C(=O)C(c2cncn2C)O)CC1 C1(NC(CSCC)=O)CCCN(C(=O)C(c2cnc(Cl)c(C)c2)(F)F)C1C c1(C(=O)NC(CC(C)NC(CSCCCC)=O)C)cc(C)c(C)c2ncccc12 C1(C(N2CCN(CCNC(C3C(C)C3C)=O)CC2)=O)CC2(C1)CC(C)(C)C2 c1(C(=O)NC2CCC(F)(CNC(C(CSC)C)=O)C2)cnc2c(ccn2C)c1 c1(CC)ocnc1C(=O)N(CC(=O)NC(C)C(C)n1cncn1)CC N(C(=NCCc1ncccc1F)Nc1cccc(F)c1)CC(COC)(C)C CC(C)C(C)CCNC(C1CCCN1C(c1cnc(C2CC2)o1)=O)=O N1(C(CC2(OC)CCC2)=O)CCCC2C1CCN2c1nc(SC)ncc1Br Clc1cccnc1CCNC1CCC2CC12 CC1CCC(C)(C(=O)NCC2CN(C(=O)CCC=CC(C)C)CC2C)C1 CCC(C)(C)C(=O)NC1(C(=O)N(CC(O)CN(C)C)C)CSC1 Cc1cnc(C(N2CCN(C(c3cccnc3C)=O)C(C3CCC3)C2)=O)c(F)c1 C1(CC(=O)NCCN2CC(c3cn(C(C(=O)OC)C)nn3)C2)CC2CCC1CC2 C1(C(N2C3(CNC(CCN(CC(F)(F)F)C)=O)CC(C2)C3)=O)CCC2(CCC2)O1 c1(NC)cnncc1C(=O)NC(C)CCNC(c1sc(CO)nc1C)=O c1(C(N2CCCC(CNC(N)=O)C2)C(=O)NC)ccc(OC)c2oc(C)cc12 c1(NC(C2CN(C(c3cc(Br)ncc3F)=O)CCC2O)=O)ccc(Br)c(Cl)c1Cl c1(CCC)nc(C)c(C(=O)NCC2CC3CC3N2C(=O)C=CC2CCCO2)s1 c1(C(N2CCN(C(C3C(=C)CC3)=O)CC2CCO)=O)ccc2c(c1)B(O)OC2 c1(OC)cc(OC)c(C(N2CCCCCC2CNC(C2CCC(=O)N2)=O)=O)cn1 c1(C(N2CCC(CO)C(NC(=O)C(F)(F)C3CC3)C2)=O)cc2c(Cl)nccc2o1 c1(C(=O)NCCCNC(C(C(=O)OCC)OC)=O)cncc(Cl)c1C C1(NCc2cc(CC(=O)OCC)on2)CCC2(CC1)CNCCO2 C1(C(N(C2CCN(C(C3CN(C(C)C)C3)=O)CC2)CC)=O)C2CCCCC12 Cc1cc(C(=O)N(CC(N2CCCCCC2)=O)CCN(C)C)ccc1O CC1C(C(=O)N2CC(C)CCC2C(=O)NC2CCC(CO)C2)=NOC1C Cc1cnccc1C(=O)NCC1CCC(N(C(=O)C(O)CN(C)C)C)CC1 c1(C(=O)NC2CCCC(N(C(c3c(C(C)C)occ3)=O)C)C2)cnc(O)c(Cl)c1 Cc1cncc(-c2ccc(C3(C(N4CCCCCC4)=O)CCC3)cn2)c1 C1(C(=O)NC2CC(NC(c3n[nH]c4c3CSCC4)=O)C2)CCc2[nH]nc(O)c2C1 c1(OC)ccc(CC(=O)NC(CCc2ccc(F)cc2)C(C)(C)C)c(C)c1 CCS(=O)(=O)C=CC(=O)N1CCC(C(C)(C)CNC(C2CCNC2=O)=O)CC1 C1(C(=O)NC2CN(C(c3ccc(C)cc3F)=O)CC3C2C3)CCc2c[nH]nc2C1 c1(C(N2CC(C3CN(C(c4cc(Br)cs4)=O)C3)OCC2)=O)ccc(F)c(Cl)c1 C1(C#N)(C(N2CCCC(O)(CNC(CCC(C)OC)=O)C2)=O)CCN(C)CC1 c1(C(=O)NCC2CCC2NC(=O)C(c2cccc(Cl)c2)O)ccc(Cl)c(F)c1 Nc1c(Cl)c(C(=O)NCC2CCC2NC(=O)C=Cc2ccco2)cc(F)c1Cl c1(C(N2C(CNC(C3CC3CF)=O)CCCC2)=O)ccc(F)cc1OC(F)F C1(NC(C=CC)=O)CCN(C(C2CCCC3(C2)CC3(F)F)=O)CC(C)(C)C1 C1(C(=O)NCC2C(C)CN(C(=O)C(c3cccc(Cl)c3)O)C2)CC2(C1)CC(O)C2 c1(C(N(CCN(C(=O)CSc2ccccn2)C)C)=O)cc(O)cc(O)n1 S(=O)(=O)(c1[nH]c(=NC(Cc2ccncc2)CO)ccc1Br)NCC1(C)CC1 C1(C(N2CCC(C)CC2)=O)CCN(C(=O)C(c2cncc(O)c2)=O)CCC1CO c1(C(N(CCN(C)C)C)=O)cccn2c(-c3cc(F)c(F)c(F)c3)cnc12 N1(C(C(C=C)(C)CC)=O)CCC(C2(O)CC(NC(=O)C(C)=C3CC3)C2)CC1 C1(CNC(c2c(C)ccnn2)=O)CCCC2(CN(C(C3(O)CC(F)(F)C3)=O)C2)O1 C1(CCOC)CN(C(C2C3CCCCCC23)=O)CCN1C(C12CC(F)(C1)C2)=O C(=O)(C(C(C)(C)O)NC(C1CC1F)=O)NCc1nnn(C)n1 C(CCNC(C1C2CCCC12)=O)(C(=O)N1CCC(C(C)(C)O)CC1)OC N1(C(c2c(CC)nco2)=O)CCN2C(=O)C(NC(C3CCN(C)CC3)=O)CC2C1 CC1(C)C(NC(=O)C(=O)NCC2CC3C=CC2CC3)CS1(=O)=O Cc1cc(S)nc(N2CCCCC2)n1.C1(C#N)(C=O)CN(Cc2ccccc2)C1 C1(C(N(CC(=O)N(C)CC2C(C)C2)CC2CC2)=O)CC2CCC2C1 N1(C(C=CC(C)C)=O)CCN(C(c2cc(Cl)cn2C)=O)CC(CO)C1 c1(C(=O)NC2C=CC(CNC(C3C=CCC3)=O)C2)cc(F)cnc1O C(=O)(C1OCCc2ccccc21)N1CC(CN(C(COC(CC)C)=O)C)C1 c1(C(=O)NC2CCN(C(CC=C)=O)C2c2ccccc2)nn(C)c(=O)cc1C C(C1CCNc2ccccc21)NC(C12CC(C(=O)OC)C(C1)C2)=O N1(C(CC2CCCC(NC(C3C(C)CC3)=O)C2)=O)CCC2(CSC2)C1 C1(C(=O)Nc2c(C)ccc(-c3cccc(Cl)c3)c2)CCN(C)C12CCCNC2 CN=c1cc(C(=O)NC2CCC(CCNC(=O)CCC3CCCCC3)C2)cc[nH]1 C12(C(=O)NC3(C#C)CCCOC3)CCC(CC1)N(C(C1(OC)CCSC1)=O)C2 CC(C)(C)C(CNC(=O)C=Cc1cnc[nH]1)NC(=O)CSCc1csc(=N)[nH]1 C12(CNC(C3CCN(CC)C3)=O)CCC(CC1)N2C(C1CC(N(C)C)C1)=O N1(C(C(N2C(COC)CCC2)=O)=O)CC2(C1)CN(C(c1c(OC)cccc1C)=O)C2 c1(N2CCC(CCC(C3N(C(CC)=O)CCCC3)=O)CC2)ncnc(Cl)c1C#N C1(CNC(CC2C(NC(c3c(CC)nsc3)=O)CCC2)=O)CCCC(OC)C1 N1(C(C(CCOC)OC)=O)CC(NC(=O)CC(C)(O)C2CC2)CCC1C C(CCCC(=O)N1CC(OC)C(NC(c2ccc(=O)n(C)c2)=O)C1)(OC)OC N1(C(N(CC(C)C)Cc2n(CC)cnn2)=O)CC(C)CCC1C C1(NC(c2c(CNC(=O)CC3CCOC3)cco2)=O)CCCC2(CC2)C1 n1(CC(N2CCC(NC(C3C(C(=O)OC)CCC3)=O)C2)=O)ccccc1=O c1(C(C)Nc2ccc(N3CCOCC3)nc2)cc(F)cc(Cl)c1 C1(NC(C(=C)Cc2ccccc2)=O)CCN(C(=O)CCc2c(C)c[nH]c2C)CC1 c1(CC(=O)NC2C(CNC(CCSC)=O)CC2)ccc(OC(C)C#N)cc1 c1(OC)nc(C)cc(=NCC2CCCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2)[nH]1 n1(CC(=O)NC(C)Cn2cc(Cn3cccn3)nn2)ncc2ccccc12 c1(-c2cn(Cc3c(OC)ccc(C)n3)nn2)ccc2nc[nH]c2c1 C12(C(=O)NCCCN(C(=O)CC(=O)OC(C)(C)C)C)CCCN1S(=O)(=O)CC2 C12(C(=O)NCC3(CNC(C4C(C)COCC4)=O)CCCC3)CCCN(CC1)C2 C1(C)(C(=O)NCC(CNC(CCc2c(C)nccc2)=O)CO)CCN(C)CC1 Cc1ccnc2c(C(=O)NC3CN(C(C4Cc5ccc(F)cc5O4)=O)C3)cnn12 c1(C(=O)OC)ccc(N)c(SCCNC(=O)CC(O)C(C)C)c1 NS(=O)(=O)CCCCCCC(=O)NCCN(C(C1CCC(O)C1)=O)C1CC1 C1(C)(C(=O)NC(C2CCN(C(CNC(C(CC)C)=O)=O)C2)C)CC(C2CC2)=NO1 C1(C)(C(=O)NC2C(N(C(c3nc(C)n(C)c3)=O)C)CCCC2)CC(=O)N(C)C1 N1(C(c2ccc3oc(O)nc3c2)=O)CCc2sc(-c3ccc4c(c3)CC4)cc2C1 c1(C(=O)NCC2CCCN(C(C3C=CCC3)=O)C2)c(Cl)ccc2ncccc12 N1(CCOCCCC)CCC2(CC1)CN(C(=O)C(C)CCOC)CCO2 C1(C(=O)NC2CCCC(NC(c3c(OC)ccs3)=O)C2)CCCCC(F)(F)C1 c1(C(c2nnnn2CCCC2CC2)NCCCCC=C)nn(C)c(Cl)c1Br CCC(C)CCC(=O)NC1(C)CCCN(C(=O)C(C)(C)n2ccnn2)C1 C1(CC=C)(NC(=O)CC2(CN(C)C)CCC2)CN(C(=O)CCC2CC2(C)C)C1 N1(C(CCCOC(C)C)=O)Cc2ccccc2C(C(=O)O)C1 C(=O)(C(CC)C(C)C)NC1(CC=C)CCN(C(c2cnc(Cl)[nH]2)=O)C1 N1(C(c2c(CC)n(CCC(C)C)nc2)=O)CC(NC(C2CC(O)C2)=O)C(C)(C)C1 c1(C(C)(C)C)ccc([N+](=O)[O-])cc1NC(=O)CCCCCF CCCCCCC(C)C(=O)NC1CC2(C1)CC(C(N1CCC3(CCC3)CC1)=O)C2 Cc1ccn(CC(=O)NCCN(C(=O)CC2(C)CCS(=O)(=O)N2)C)c(=O)c1 C(=O)(C1=CNC2=NCCC2=C1)NC1(CN(C(=O)Cc2cnns2)C)CC1 c1(C(CC)NC(C2CCN(C(C)(C)CC(=O)NC)C2)=O)cc(Br)ccc1C c1(C(=O)NCC=CCC(N2CC(C(C=C)C)C2)=O)cc(C)co1 C=C(C)CCCC(=O)NC1CCCC1NC(=O)Cn1nc(C)n(C)c1=O CC(C)(C)C(CNC(=O)CCc1n[nH]c(=N)s1)NC(=O)CC1CC2(CC2)CO1 C1(NC(CCCCNC(C)=O)=O)COC2(C1)CN(CCOc1ccccc1C)C2 c1(OC(C)C)cccc(C(=O)NCc2cccc(C(=O)OCCC(C)(C)C)c2)c1 CN1C2CCC1CC(C(=O)NCC(O)CCNC(C13CCC(CC1)CO3)=O)C2 C1(NC(Cc2cc(C)sc2C)=O)CCN(C(C2(CO)CCC2)=O)CC1F C1(C(=O)Nc2c(C)scc2)CN(C(=O)CNC(N)=O)CC1C C=CCC(C)(CC)C(=O)NC(c1ccccc1CC)CNC(=O)CCC(C)(F)F Cc1ccccc1C(C)CC(=O)NCC1(NC(c2cnc(SC)s2)=O)CC1 C(CCC(=O)N(C)CCN(C(=O)CNC(=O)CC1CCCCC1)C(C)C)OCCC C1(NC(c2c(C)n(C)cc2)=O)CC=C(C(=O)NC2COCCN(C)C2)C1 N1(C(Cc2c(C)ccs2)=O)CC2CC1CC2NC(=O)Cn1ncccc1=O C12CC3CC(C1)N(C3)C2.c1(C(C)(C)OC)cccc(CCNc2ccccc2)c1 c1(C(=O)NC2C=CCN(C(=O)C(F)OC(F)(F)F)C2)cccc2oc(O)nc12 C1(C(=O)NC(C)Cn2cnc3ccccc23)CN(C(=O)OC(C)(C)C)C2(CCC2)C1 C1(NC(C2CCCN2c2ncccn2)=O)CCC(N=c2[nH]nco2)CC1 c1(CC)c(C(=O)NC2CCC2C(=O)Nc2cnn(C(C)(C)C)c2)ccn1C C1(CNC(c2c(C)nncc2)=O)CC2CCC1N2C(c1cccc(C)c1O)=O C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(C)(C2CC2)OC)CC1c1cnn(C)c1 c1(NCC23C(O)CCC2C3)nc2ccccc2nc1NC1(CCO)CCCCC1 C1(C(=O)NCC#CCNC(=O)CCCc2ccsc2)CN2CCN1CC2 c1(C(N(CCCNC(=O)C#CC2CC2)CC)=O)ccc(F)c(C)c1C#N c1(OC)cc(CN2CCC(C)(C(=O)NCc3ccccn3)C2)c(Br)cn1 O=C(CC(F)(F)F)NC1CCCCC1C(=O)NC(c1ncc(F)cn1)C N1(C(C=CC=CCC)=O)CCC(CF)(NC(=O)CC2CCOCC2OC)C1 N1(C(CCSC)=O)CCC2CCN(C(=O)CC=Cc3ccc(F)cc3)C2C1 c1(OCC)cnc(C(N2CCC3(NC(=O)CC4CCCCC4)CC3C2)=O)c(Cl)c1 N1(C(C(CCC)N(C)C)=O)CC2CCC2(NC(=O)C=CCOCCOC)C1 C1(C(=O)NCC2C(NC(c3cn(CC)nc3OC)=O)CC2)CC(C2CC2)=NO1 CCCCCCC(C)C(=O)N1CC2CCCN(C(=O)C3=CCC(C)OC3)C2C1.C=O C1(C(=O)NC2(C(N(C)CC3(C)CCCO3)=O)CC2(C)C)C2CCCC(=O)C12 c1(C(=O)NC(CC(C)NC(c2cccc(CC)n2)=O)C)ccc(C)c(Cl)c1N c1(C(=O)NC(CC)CNC(c2cnnc(O)c2)=O)ccc2oc(O)nc2n1 C1(NC(C(c2scc(C)n2)C)=O)CCCC(NC(c2ccnc(C(N)=O)c2)=O)C1 C(=O)(C(C)N=c1cncc[nH]1)N1CCC(F)(C(=O)Nc2cccc(OC)n2)CC1 N1(C(C=CC=CC)=O)CCCCC1C1CCCN1C(c1cc(OC)ccc1N)=O c1(C(=O)NCCN(C(=O)C(c2ccccc2Cl)OC)CC)cn(C(F)F)c(C)n1 C=Cc1cncc(C(=O)N(C2CCCN(C(=O)CSCCC(C)C)C2)CC)c1 C(=O)(CN1C(=O)COc2ccc(Cl)cc21)NC(C(C)(C)C)CNC(=O)CCCF C1(SC(C)(C)C)CC(NC(=O)CC2(NC(=O)C(F)C3CCCC3)CC2)C1 c1(SC)ncc(N)c(C(=O)NC(C)CC(C)NC(=O)CN2CC3CC3C2)n1 c1(C(N2CCCC(NC(C(C(CC)(C)C)O)=O)C2C)=O)sc2ccccc2c1C c1(-c2nc(C)sc2)cccc(C(=O)NCCCN(C)C(C2CCCOCC2)=O)c1 C12(CNCC(c3ccc(F)cc3)CO)CC1CCC2(F)F N1(C(C=CC(C2CCCC2)=O)=O)CCC2C(C1)CN2C(=O)CC(C1CC1)C1CC1 c1(CC(N2CCC(CNC(CCCC#C)=O)C(O)C2)=O)ccc(O)c([N+](=O)[O-])c1 c1(CNC(c2n(CC)ccn2)=O)cccc(CNC(=O)CC2CN(C)CC2O)c1 N1(C(CC(C)C)=O)CCOC(CCCNC(C2CCCC(O)C2)=O)C1 CN1CC(N=c2[nH]c(N3CC(C)(C)OC(C)(C)C3)nc3ccsc23)CC12CCC2 c1(C(=O)NC(C2CCN(C(C(C)SC)=O)C2)(C)C)nnn(C)c1C(F)(F)F C1(CNC(C2C3(CC(NC(=O)CC4CC=CCC4)C3)C2)=O)CC2(C1)CC(O)C2 C(CC(C)(C)C(=O)NC1CCC(CCNC(c2nn(C)cc2SC)=O)C1)SC C(=O)(C1=NN2CCCN=C2N1)NC1CC2CN(C(CCCC(C)C)=O)C(C1)C2 C1(C(=O)Nc2ccc(-c3n[nH]c(C)n3)cc2)(CC)CCNC1=O c1(C(=O)NCC(CNC(c2c(C)n(C)nc2Cl)=O)C)cc2cc(Cl)sc2[nH]1 C(C(CNC(=O)CC(C)N(C)C(c1nnccc1C)=O)C(C)C)OC O=C(NNc1ccc2c(c1)CCO2)C1CCC(c2nc[nH]n2)O1 c1(OCC)cccc(C(=O)NC2(CNC(C3OC(C)CC3C)=O)CC2)c1N C(C(C)(C)CC(=O)N1CCCC(F)C1)NC(CCc1ccn(C)n1)=O C1(CNC(c2cccn(C)c2=O)=O)CC2(CC2)CN1C(c1cc(CO)[nH]n1)=O N1(C(C2(F)CCCN(C(c3n(C)cnc3)=O)C2)=O)CCN2CC(F)CC2C1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(NC(C2CC(F)(F)C2)=O)C12CC2 C1(C(N2C(C)(C(N3CCC(OC)C3)=O)CC2)=O)C2CCC(C2)C1C Nc1cnc(Cl)cc1C(N1CC(CNC(c2ccc(F)cc2Cl)=O)C(F)(F)C1)=O C12(C(C)NC(c3nnnn3C)CC)CCC(CC1)C2 C=CC(O)C(=O)N1CC(=C(F)CNC(C2CCCN2C(=O)OCC=C)=O)C1 c1(CC)noc(C)c1CNC(=O)CN(C1CC(C#N)C1)C(C1C2CCC(F)C12)=O n12ncc(n1)CN2CC.C1(CN2CCC2)CCOC1 c1(C(=O)NCC(C)(C)OCCNC(C(C)OCCC#C)=O)ccccc1Cl c1(C(=O)NCC(CNC(C2C(CC)C2)=O)OC)cccc(C2OCCO2)c1 c1(C(=O)NCCC(C)N(C(C=C(C)C)=O)C)cc(C(F)(F)F)nn1C c1(C(N2C3CN(C(C(C)(C)SC)=O)CC2CC3)=O)ccnc(S(N)(=O)=O)c1 CCCC(C)(O)CC(=O)N1CCC(NC(c2ccnn2CC(F)(F)F)=O)C(O)C1 Cc1cc(O)ccc1C(N1CC(NC(c2cnn(CCF)c2)=O)C(C)C1)=O Cc1c(C(N2CCCC(C(C)NC(=O)CCc3cccn3C)C2)=O)cnn1C c1(-c2c(C(=O)NC)nccc2)ccc(S(=O)(=O)N2CCC23CCCCC3)cc1 CC1CC2CN(C(=O)Cc3cscn3)CC2N1C(C12CCC(CC1)C2(C)C)=O C1(C(=O)NCC(N(OC)C)=O)CCC2CCC1N2C(=O)CN1CCCNC1=O C1(n2cc(C3CN(C(CN4C(C)CC4)=O)C3)nn2)CCCN(S(C)(=O)=O)CC1 CC(C)C(F)(CNC(=O)C(C)S(C)(=O)=O)C(=O)N1CC(c2nncs2)C1 c1(C(=O)OC)ncccc1C(=O)NC1CCN(C(=O)C(c2ccccc2Cl)O)C1 N1(C(c2c(C)nc[nH]2)=O)CCCOC(CNC(=O)CC2CCC(=O)NC2)C1 CC(C)C(C)C(CNC(c1cccc(F)c1)=O)NC(c1coc(Cl)c1)=O c1(-c2cn(C)nc2)ccccc1CNC(c1ccsc1-c1nn[nH]n1)=O Cc1nc(-c2ccsc2)ccc1C(=O)OC1Cc2cscc2C1 Cc1cc(C(=O)NC2CN(C(=O)COC3CC=CC3)CC2(C)C)cc([N+](=O)[O-])c1 c1(CC)cc(C(=O)NCC2CCCCC2NC(C2C=C(C)CS2)=O)n(C)n1 c1(C(=O)NC2CC(C)(NC(C(C)=C3CC3)=O)C2)cc(N(C)C)c2ccccc2n1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1C2C(CNC(=O)Cc3cncnc3)CC(C2)C1 c1(C(=O)NC(C(CO)NC(C(C2CC2)OC)=O)C)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C(=O)NC(c2onc(C)n2)CO)C1 C12(CCNC(C(=O)NC(C)C)=O)CCC1CN(C(=O)C(F)(F)C1CC1)C2 N1(C(C)=O)CCCCC1CC(=O)NC(C)(C)CCNC(C1CC=CC1)=O C1(NC(C2CCN(CC(=O)O)C2)C)CCCN(C2CCN(C)CC2)C1 c1(-c2cc(C)cc(C)c2)ccc2c(c1)CCN(C(=O)CNC(N)=O)C2 C#CCCCCCC(=O)N1CCC2CN(C(=O)CC3CCCCC3)C2C1 N1(C(CCn2c(C)cc(C)n2)=O)CCC(CO)C(NC(c2cnc(S)n2C)=O)C1 N12CCc3c(OC)c(O)cc(c3C1)C2=O.C1(C(C#C)OC)CCCCO1 C12(NC(C(CC#C)O)=O)CCC(CC1)N(C(c1cc(O)ncc1Br)=O)C2 c1(CC(=O)NCC(CNC(c2cccc(C)c2O)=O)O)oc2ccccc2c1C Cc1nn(C)c(Cl)c1C(N1CC(CO)C(C)(C)C1)C(=O)Nc1cccc(Cl)c1C C(CCCC(OC(C(C)NCC)=O)OC)(C(=O)OC)CC(=O)NC Cc1cnn2ccc(C(=O)N(CC(C)NC(=O)C(C)(C)c3cnn(C)c3)C)nc12 N1(C(C(C)C#N)=O)CCC2(C1)CN(C(=O)NC1(c3ccc(F)cn3)CC1)C2 C(CCCN=c1[nH]c(=NCC23CCC(CO2)C3)c2ccccc2[nH]1)OC C1(OC)CC(NC(C2CSC2)=O)C12CCN(C(c1c(C)[nH]c(C)c1C)=O)CC2 C(CN=C(NCC(c1ccc(C#N)cc1)C)NC1CC1)=CC=CC C1(N(C)C(C2CCCCC2)=O)CC2CCC(C1)N2C(=O)C(=O)Cc1ccccc1 c1(C(N2CCC(CNC(C3CCCN(C(CC)=O)C3)=O)C2)=O)cc(=O)c(OC)co1 c1(C(NOCCOCC)=O)coc2c1CN(C(=O)CN1CCCC1C)C2 c1(C(N(CCCCN(C(=O)CCCC2CCC2)C)C)=O)cnn2ccn(C)c12 N1(C(c2cc(C)c(C)s2)C(=O)NCC=C)CCNC(=O)CC12CCOCC2 C12(C(CNC(=O)COc3ccccc3)NC(C3CCCO3)=O)CCC(CC1)C2 c1(C(C(=O)NCc2nnn(C)n2)N(C(CCOC)C)C)cc(Cl)ncc1Br N1(C(c2c(CC)onc2)=O)CCC(C2(O)CCN(C(=O)C(C)O)CC2)CC1 CCC(C(=O)NCC1CC2(C1)CN(C(=O)CC(C)=C(C)C)C2)C(C)O C(=O)(CCCC(=O)NC1CCC(N(C(=O)Cn2nnc(C(C)C)n2)C)C1)OCC C1(NCc2ccc(-c3c(C)n[nH]c3C)cc2F)CCNC2(CCC2)C1 c1(C(=O)NC(CCCC)CNC(=O)CCCC(C)O)cc(F)c(N(C)C)c(F)c1 N1(C(CN2C(C)CC2)=O)CC2C(CN(C(=O)C=Cc3ccc(C(N)=O)o3)C)C2C1 Cc1nc2cc(C(=O)NC3CCN(C(c4ncccc4C)=O)C(C)C3)cnc2[nH]1 CCS(=O)(=O)C=CC(=O)NCCCCC1CN(c2ncc(C#N)cc2F)C1 c1(C(=O)OCCOCC)ccnc(OC2CC(C(N3CCC(OC)CC3)=O)C2)n1 n1(CCOCC)nnnc1C(c1cnc(C)s1)NC(C)CC1CC1 c1(C(N2CCC(CC(=O)NC(COCC)C)C2)=O)cc(NC)ccc1Cl N1(C(c2cc(C(C)=O)on2)=O)CCC(C(C)NC(C2(F)CCOC2C)=O)CC1 c1(C(=O)NCC2N(C(C(C)=CC)=O)CCCC2)cc2c(C)cccn2c1 c1(N2CCC(CCOC)(NC(c3cnc(O)n3C)=O)C2)nc2cccnc2s1 c1(C(CCOC)SC)nnnn1CC(N1CC=CC1)=O Cc1nc2c(C(=O)OCC3c4ccccc4CC3)ccnc2[nH]1 CC(C)C(O)C(=O)NCCCC(C)NC(=O)CC1CC2(CC2)CO1 Cc1cc(C(=O)NCCCCNC(=O)C(C)(C)CF)c(N)c([N+](=O)[O-])c1 C(CCCCC(=O)NC1C2CC1N(C(c1cnc(C)cn1)=O)C2)NC(C)=O C(=O)(C(F)Cc1ccccc1)NC(C(=O)N1CCCC1)C1CCOC1 N1(C(c2c(C)nsc2Br)=O)CCC2(C1)CN(C(=O)CSCCC#N)C2 c1(C(N2CCC(NC(C3(CCF)CC3)=O)C2C)=O)cc(C(F)(F)F)ncn1 C1(CNC(C(CCOC)C)=O)CCCN(C(c2ncn(CC(C)C)n2)=O)CC1 c1(CC)onc(C(N2CC3C(CC(=O)N(CC(O)CN(C)C)C)C3C2)=O)c1C C(=O)(C#CC1CCCCC1)N1CC(NC(CCCCCCC)=O)C2(C1)COC2 N1(C(c2c(C)nc(C)o2)=O)CCC(C(=O)NCC2CCN(C(N)=O)C2)CC1(C)C C1(NC(CSCC=C)=O)CCCC12CCN(C(c1ccc(F)cc1O)=O)C2 N1(C(CCN(C)CCO)=O)CC2(C1)C(NC(C1CC3CC3C1)=O)CCS2(=O)=O c1(C(=O)NCC(CC)(C)NC(c2ccc(CN(C)C)o2)=O)cnccc1Cl N1(C(C2CC2Br)=O)CC2CCN(C(=O)CCc3ccccc3F)C2C1 c1(C(C(=O)NC(CC)C)N(C2C3CCCC23)C)ccnc(-c2ccccc2)n1 N1(C(=O)NC(C)(C)C)CCCN(CC2CN(CC)C(=O)O2)C(CCOC)C1 c1(OCC(=O)N(CCCCCNC(=O)CNS(C)(=O)=O)C)cccc(F)n1 C1(C(C)OC)CCN(C(=O)C(C2CCCCC2)NC(C2CC(C)=NO2)=O)CC1 C1(CC)CN(C(C23COC(CCO2)C3)=O)CCN1C(=O)Cc1ccoc1C N1(C(CCc2n(C)cnc2)=O)CC(O)CC1C(=O)NCCc1cccc(F)c1 N1(CCCOCC)CCC(C(C)NC(=O)C(C2CCCC2)OC)CC1 c1(OCC)cccc(C(=O)NC2CC(O)CN(C(=O)CCCF)C2)c1N c1(C(=O)NC2C(CNC(c3c(Br)cn(CC)n3)=O)C2)cccc2[nH]ncc12 N1(c2cc(NCC(C)CC(C)O)nc(C)n2)CCN2CCCC2C1 c1(C(N2CCC(CC(=O)NC3C(CN(C)C)CCC3)CC2)=O)ccc(N)c(F)n1 C1(C(C)C)CN(C(c2cnn(C)c2)=O)CCCN1C(c1cnc(O)c(F)c1)=O C1(CC)CCN(C(c2cc(C(=O)OC)ns2)C(=O)NCCCCCC)CCO1 c1(C(=O)NC2C(c3c(C)ccs3)C2)ccnc(C(F)(F)F)c1[N+](=O)[O-] C1(NC(C(C(C)C)C)=O)CN(C(C2(c3ccccc3F)CCC2)=O)CC1(C)C C1(OC)CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(c1coc(C)n1)=O c1(C(=O)NC2CN(C(C(CC)(C)F)=O)CC(O)C2)ccnc2ccc(O)cc12 C1(NC(c2cncc(OC)c2)=O)CC1C1CCN(C(C2(CC(F)F)CC2)=O)CC1 C(=O)(C(C(=O)NC1(CO)CCN(C(c2ncc[nH]c2=O)=O)C1)OC)OCC C1(CNC(C(C(C)(C)C)OC)=O)CC2CCC(C1)N2C(=O)C(C)(C)SC N1(C(c2cccc(CC)c2)=O)CCC(CNC(=O)Cn2ccccc2=O)C(C)C1 CCC(CC(=O)NC1CCN(Cc2ncccn2)CC1)CC(F)(F)F C12(NC(C(c3ccccc3F)C)=O)CCCC1N(C(=O)CCC(N)=O)CC2 N1(C(C)=O)CCc2c(NC(c3cc(C(N)=O)cc(F)c3)=O)cccc2C1 N1(C(=O)NCc2ccc(O)nc2)CCC(O)C(O)C1 c1(NC(c2c(NC(c3n(CC)ccc3)=O)nc(Cl)cc2)=O)cc(C)cc([N+](=O)[O-])c1 C(=O)(C(CO)N(C)C)NC(CN(C(=O)COCC1CCCOC1)CC)C c1(OCC)cc(Cl)ccc1C(=O)NC1(CCCNC(=O)Cc2ccon2)CC1 c1(C(N2C(C)CSCCC2)=O)ccc(S(=O)(=O)N2CCC3(CC(F)C3)C2)cc1 C1(CNC(C23CC(CCC)(C2)C3)=O)(COC)CCN(C(=O)CC)CC1 Cc1ccc(-n2cc(CNC3CCC4(CC3)CC4)nn2)c(C)c1 CCCCCC(O)CC(=O)N1CC(C(F)C(N2CCOC(CC)CC2)=O)C1 C1(C)(C(=O)NCC2CC(NC(C3(SCC)CC3)=O)C2)CCCC1(F)F CCC(C)CCCCC(=O)NC(CC(=O)NCC=CC(C)(C)C)C(C)OC c1(CC)cc(N2CCCC(C(F)(F)F)CC2)nc(CNC(C2(C(N)=O)CC2)=O)n1 c1(C(=O)NC(C)CCCNC(c2ccoc2)=O)ccnc2ccccc12 C1(C(=O)NC2C(C)(C(F)F)C2)(NC(c2ccc(CCF)cc2)=O)CC(F)(F)C1 c1(-c2onc(-c3cc(C)cc(C)c3)n2)cnn2c1CCCC2 Cc1ccc(C(N2CC(NC(=O)C(C)(C)c3cnc[nH]3)CC(C)C2)=O)c(O)c1C Cc1nc(=NCCNC(C2(CC#N)CCN(Cc3ccccc3)C2)=O)[nH]cc1Br C1(C(=O)NCCN(CC(C)O)C(c2ccc(Cl)[nH]2)=O)CCCCC1 N1(C(C(C=C)C)=O)CC(NC(=O)Cc2cc(F)ccc2C)CC1(C)C c1(CC(=O)N(C)CC2N(C(c3c(C)onc3)=O)CCOC2)cccc(C)c1Cl C1(NC(C2C(C(C)=O)C2(C)C)=O)CC(C)CN(C(C2CC3CCC(C2)O3)=O)C1 c1(COC)cc(C(=O)N(CC(C)NC(=O)C(n2ccc(Br)n2)C)C)no1 c1(CC(=O)NCC(CC=C)NC(=O)CC2CCC(C)CO2)ccc(Br)cc1 C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NCCNC(c1c(C)cc(OC)c(Cl)c1)=O c1(C(N(CC(C)NC(C2CCC(=O)O2)=O)CC)=O)c(C2CC2)nn2ccccc12 c1(C(=O)NCC(c2ccccc2)CNC(C=C(C)C2CC2)=O)ccnnc1O CC1CN(C(C23CC(C4CC4)C2C3)=O)CCCN1C(c1nc2cccnc2s1)=O N1(C(C(=O)Nc2ncc[nH]2)=O)CCC2(CCN(C(c3ccc4c(c3)CC4)=O)C2)C1 N1(C(c2cnn(-c3ccc(Br)cc3)n2)=O)CC2CCCC(C1)C2(F)F C1(N(C(C(CC)N(C)C)=O)CC2CC2)CCN(C(=O)CNC(N)=O)CC1 c1(C(=O)NC2CC3CC2N(C(=O)CC2CCOC2=O)C3)cnc2c(c1)CCCO2 N1(C(C2C(C(=O)OC)C2)=O)CC(C2CCCN(C(=O)C(C)N(C)C)C2)C1 C(N=c1nn[nH]n1C)C1(F)CC(NC(C(C)C2CCCO2)=O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CCC(C)(C)CC1C(=O)NC12CC(F)(C1)C2 N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1c1nccn1C c1(C(N2C(C)(C)C(CNC(C3CC4CCC3C4)=O)CC2)=O)ccc2oncc2c1 N1(C(CCCCCOC)=O)CC2CC(NC(=O)C(n3nc(C)cc3C)C)C(C2)C1 c1(C(=O)NCC(CO)NC(C2(OCC)CCCC2)=O)cccc2c1NCC2 C(CC(C)C(=O)N1CC(C(C)(C)O)(CNC(=O)CC2CCCO2)C1)=CCC N1(CC)CC(C(=O)NCCOCCNC(c2sccc2C#N)=O)CC1=O C1(C(=O)NCC2C(NC(c3cc(C4CC4)[nH]n3)=O)CC2)COc2ccccc2O1 c1(C(=O)NC(CNC(C2(C)C(C)C2)=O)CO)cc(C(F)(F)F)ncc1N c1(C(N2CC(CNC(C3(OC)CCCOC3)=O)C2)=O)ccc(C)c(F)c1N C(=O)(CCC(=O)NCC1COCCN1C(C1CCC2CC12)=O)NCCC C(=O)(C1=CCS(=O)(=O)C1)N1CC(NC(c2n(CC)ncc2Br)=O)C(C)C1 C(CC)(C(=O)NC(C)C(CO)NC(c1ccc(C2CC2)s1)=O)=CC C(=O)(C(O)C(F)(F)F)N1CCN(CC(=O)NCC(C)(C)O)CC1.C1(C(N)=O)(N)CC1 C1(CCNC(Cc2cnc(C)s2)=O)CSCCN1C(c1cc(CO)c(C)o1)=O c1(N(CCCCOC(C)C)C)nc2c(c(=NCC3COC(=O)O3)[nH]1)CCC2 CC(C)C(C(=O)NC(CCF)C(=O)N(C1CC2CCC1O2)C)C1CCC1 Cc1cc(C(=O)NC2CCN(C(=O)Cc3ccc(Cl)cc3)C2)c2c(n1)CCCC2 c1(CC)ncc(Br)cc1NC(C1CN(C(c2ccc(O)cn2)=O)C1)=O c1(C(N2CC(NC(c3ccnc(OC)n3)=O)CC2(C)C)=O)cc(F)c(F)c(F)c1 c1(C(C)NC2CCCC2N2CCCC2)ccc2[nH]ccc2c1 C(=O)(C(C)(C)CC(=O)Nc1cccc(NC(c2sccc2F)=O)c1)OC c1(C(C)=O)cn(C)nc1C(=O)NC1COCCC1NC(=O)CCc1ccncc1 N1(C(c2cc(SC)oc2C)=O)CCC(C)(NC(=O)CCC2CCCC(=O)N2)CC1 CC1CCCCC1(C(=O)O)NC(=O)COC1CCCCCC1 C(CC(C)c1ccccc1)(C(=O)NC1CCCC1C#N)N(C)C c1(C(=O)NCC(CO)NC(c2cn(C)nn2)=O)cccc2c1CCCC2=O c1(C(N2CCC(O)C(C)C2)C(=O)NC(CC)C)sc(S(N)(=O)=O)c(OC)c1OC C1(NC(Cc2nc(C(C)C)sc2)=O)CC2(C1)CN(C(=O)C(F)CC1CCOC1)C2 C(CC(=O)N1CC(C)CC(O)C1)(C(F)(F)F)NC(C(CCC)C)=O CC(CNC(=O)CN1CCNC(=O)C1)CN=c1cc(C(N)=O)nc[nH]1 C=C=CC(C)C(=O)N1CCN(C2CCC(NC(=O)C3=C(C)CC3)CC2)CC1 N1(C(c2occ(C(N)=O)c2)=O)CCC(O)(C2(NC(=O)Cc3ccsc3)CC2)CC1 CCC(CC)(C(=O)N(C)CCOCCNC(C1CC2CCCC2C1)=O)OC c1(N2C(CN(C)C(C3CN(S(C)(=O)=O)C3)=O)COCC2)nccn2nnnc12 Cc1cccc(C)c1C(N1CSCC1C(c1ccccc1)=O)=O.N1CS1 CCC(F)C(=O)NCC(C1CC1)NC(=O)C(C)(C)C1CCCCC1 CCC(CCC(=O)NC1CCCC1N(C)C)NC(=O)CCc1cnn[nH]1 c1(CC(=O)NCCCN(C(=O)Cc2ccsn2)CCO)ccc(O)c(F)c1 N1(CCCC=C)CCC2(CC1)CC2(C)C(N1CCNC(=O)C1)=O N1(C(c2c(C)ncs2)=O)CC2CC1CCN2C(c1cc(CO)on1)=O c1(C(N2CC(N(C)C(c3cnc(Cl)s3)=O)C(C)(C)C2)=O)ccc(S(N)(=O)=O)o1 C(C)(C)(C(=O)NCC1(F)CN(C(C2CCCO2)=O)C1)OC(C)=O C(=O)(CCCCCC(=O)NCCCC(C)NC(=O)CC1CCSC1)OCC c1(C(=O)NCc2cc(C(=O)NCc3c(C)nn[nH]3)on2)c[nH]c2cnccc12 N1(C(=O)C#CC2CC2)CC(CO)C2(CCN(C(C3CCC=CCC3)=O)CC2)C1 N1(C(C(C#C)(C)C)=O)CCC2CN(C(c3c(C(F)(F)F)cccc3F)=O)CC2C1 Cc1ccn(CC(=O)N(CC(C)N(C(=O)Cc2ccc(Cl)c(C)c2)C)C)c(=O)c1 C12(NC(C(CCC#C)O)=O)CC(C)(C1)OC21CN(C(=O)C(CC)N(C)C)C1 OC1CCN(C(=NCCCC2C=CCC2)NCCF)CC1 Cc1ccc(CC(=O)NCC(=O)N)cc1C.c1(OCC2CCCC2)ccccc1 C(C1COCc2ccccc21)NC(=NCC=C)NCC1CCS(=O)(=O)C1 c1(C(N(CC(CNC(C(C)(C2CC2)OC)=O)C)C)=O)cc2cc(N)ccc2s1 N1(C(C=CCOC)=O)CCCC2(CC(NC(c3ccnc(C4CC4)n3)=O)CO2)C1 C(=O)(C(C)(F)C(=O)NC1CCC(C(=O)NCc2cnsc2)C1)OC c1(C(=O)NCC(CO)NC(=O)Cc2c[nH]nc2O)nn(CC(F)(F)F)cc1Cl N1(C(C=CCC)=O)CCC2(COCC(CNC(=O)CCC3CC(F)(F)C3)O2)C1 C(=O)(C(CCC(C)C)NC(=O)CC(C)C(C)C)NCc1c(C)nns1 C1(C(=O)NC2(CNC(=O)C(C)Cn3ccnc3)CC(OC)C2)CCCCCCC1 c1(OCC(=O)NC2COCC2NC(C2CC(C)(C(=O)OC)C2)=O)ccccc1C c1(CC)nc(C)c(CC(N2CC(C)N(C(=O)COC3CC3)CC2C)=O)c(C)n1 N1(C(COCCOCC#C)=O)CCC(C)(CNC(C2CC3CC2CC3O)=O)CC1 C(CC(C)C(F)F)NC(C1C(CNC(c2c(C)snn2)=O)OCC1)=O c1(C(=O)NCC2(NC(CC=C)=O)CC2)nnn(C2CC2)c1C(F)(F)F C(C(C)(C(=O)NCC(O)(CO)CO)NC(=O)Cn1cnnc1)SC N1(C(c2cc(CC)[nH]n2)=O)CCC(CC(=O)NCC2CC2(C)C)CC1 c1(C(=O)NCCC(C(C)C)NC(C(N(C)C)C2CC2)=O)cc2c(s1)CCCCC2 C(=O)(C(C)(C)CSC)NCC(CCC)NC(c1cnn(C(C)C)c1F)=O n1(CC(N2C(CNC(C3CN(CC)C(=O)C3)=O)CC(F)C2)=O)ncc(C)cc1=O Fc1c(CSCCCn2ccnc2)cccc1Cl C1(C)(CNC(CNC(=O)OCC=C)=O)CCN(C(=O)C=C2CCSCC2)C1 CCCCCCC(=O)NC(c1ccc(F)cc1)CNC(=O)C(C)(C)OC(C)C C1(CC(N2CC(NC(c3n(CC)ncc3)=O)C2)=O)CCCC2(CC2)C1 c1(C(NNC(CCC)=O)=O)c(-c2cnn(C3CCCCCC3O)c2)nn2c1CCC2 N1(C(C(C(C)O)N(C)C)=O)CC2CN(C(c3cn[nH]c3)=O)C2C1 c1(C(N2CC(OCC)C(CNC(C3CC3(F)F)=O)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(CNC(C2(CCCC)CC2)=O)CCCCC1NC(C1(SC)CC1)=O c1(C(C)=O)cncc(C(N2C(CNC(=O)Cc3cn[nH]c3)CC3CC23)=O)c1 c1(Oc2cccc3c2OC(C(=O)O)C3)ccc2nc(Cl)sc2c1 c12ccc(c(C)c1)s2.C(CC(=O)NCCCCC1CN(C(=O)CC2CC2)C1)=CC c1(C(N(CC(C)NC(C2(O)CCSC2)=O)C)=O)ncc2[nH]ncc2n1 c1(C(=O)NCC(CC)(CC)NC(=O)C(C)n2ccnn2)cn2c(n1)C(C)CCC2 C1(CNC(C2C(OCC)C2)=O)CCCN(C(=O)CN(C2CCSC2)C)CC1 c1(C(=O)NCCCCC(C)NC(c2nc(OC)c(C)s2)=O)cc(N)c(O)c(F)c1 c1(C(=O)NC2CCN(C(C3CCNC3=O)=O)CC2F)nc2ccccc2[nH]1 C(=O)(C(C)CCCC(C)C)NCCC1(OC)CN(C(=O)CCc2cnco2)C1 C(CNC(C1CCCN(C)C1)=O)(CC(=O)NCc1c[nH]nc1C(C)C)OC N1(C(c2c(C(C)C)nns2)=O)CCC2(CC1)CC2NC(c1cccc(=O)o1)=O O=C1CN(C(c2ccccc2F)=O)C(C(=O)NC2CCCC2(F)F)CN1 c1(-c2cn(SCCOC)nn2)ccnnc1C CCC(C)CCC(=O)N1CC2CC(NC(c3cnn(C)c3C(C)(F)F)=O)C1C2 c1(C(=O)NC2C(CNC(C=Cc3ccc(C)s3)=O)CC2)cnc2[nH]cnc2c1 c1(C(C(N2CC(CCNC(CCCCOC)=O)C(C)C2)=O)=O)ccc(F)c(Cl)c1 c1(CN(C(C2CCCN(C(c3cnc(OC)nc3)=O)C2)=O)CC)cncnc1C C1(CNC(c2n(C)nc(C(F)F)c2)c2nnnn2CCF)CCCC(F)(F)CC1 C1(C)(CC)CC(NC(C)=O)CN1C(=O)CCc1ccncc1 c1(C(N2CCC(CN(C)C(c3cnsn3)=O)C2)=O)cnnc(C2CC2)c1 c1(Cc2c(C)nc(NC(N3CCC4(CCOC4)C3)=O)s2)cc(N)c(Br)c(F)c1 n1(CCC(=O)NC2CN(C(C3CCC3)=O)CC2C(F)F)sc2ccccc2c1=O C1(C(N2C3(CNC(c4cc(C(F)(F)F)no4)=O)CC(C2)C3)=O)CCCNS1(=O)=O CC1CN(C(c2ccc(CN(C)C)[nH]2)=O)CCC1NC(=O)C(O)C1CC1 C1(C(=O)Nc2ncc(C#N)s2)CN(Cc2cccc(-c3ccco3)n2)CCC1O c1(C(=O)NCCOC2CN(C(C3(CC)COC3)=O)C2)cc2ccccc2n1C Cc1c(C(=O)NCC2CCC2NC(=O)C(C)(F)F)sc(Cl)c1Cl C=CCCC(C(=O)NCC1(OC)CN(C(c2ncn(C)n2)=O)C1)c1ccccc1 c1(OC)cccc(-n2c(SCC3CC(F)C(=O)N3)nnc2-c2ccco2)c1 CC1CC(=O)NCC1C(=O)NCCCCCNC(c1cscc1C(N)=O)=O C1(CC(=O)NC2CCN(C)C2=O)CC(C)(C)CN1C(=O)Cc1csnn1 N1(C(c2c(CCC)[nH]cc2)=O)C(C(=O)NCC(C(C)CC)OC)CC2CC12 CCC(C)CC(=O)N(CC(CC(=O)N1CCC(F)C1)Nc1cccnc1)CC c1(OC)cc(C(c2nnnn2C2COC2)NC2(CCC3CCC3)CC2)ccn1 c1(OC)ccc2cc(CN3CCCC(NC(=O)CCCCCBr)C3)c(Cl)nc2c1 C1(C(=O)NCCC2CCCC2)CC12CCN(C(=O)CN1CCNC1=O)C2 C1(CNC(c2c(C)nccn2)=O)CCC(C)(C)CN1C(C1C(C)C1(F)F)=O CC1(C)Cc2cc(Br)ccc2C1NC(C1CCC2(CC1)CSC2)=O N1(C(=O)NCCC2CCN(CC(F)(F)F)CC2)CC2(CCSCC2)C1 Cc1cc(C)c(NC(C2CCCCC2NC(=O)OC(C)(C)C)=O)cn1 N1(C(C2N(CC)CCOC2)=O)CC2CCCC(C1)N2C(=O)Cn1cnnn1 c1(CNC(c2cnc(C)s2)=O)ncc(C(=O)NC2CC3CCC2C3)cn1 Cc1cc(C(=O)NCC(C2CCCC2)NC(C23CCCC2C3)=O)no1 Cc1cc(NCc2ncoc2-c2ccccc2)c(F)cc1[N+](=O)[O-] C=C1CCN(C(=O)CCCOCC)C(C(=O)NCCC(F)(F)CC)C1 c1(C(=O)NCC2CC(C)SCC2)cnc2sc(Br)cn12 c1(C(N2CC(CC(=O)NCC(CCC)NC(C)=O)C2)=O)ccc2c(c1)OCC2 Cc1ncc(N)cc1C(=O)NCC(C)(C)NC(c1csc(S)n1)=O CCCCC(F)C(=O)NCCC(C)(C)C(=O)NCCC(=O)N(CC)CC C1(CN(C(CN(C)C(=O)OC(C)(C)C)=O)C2CC2)CCCN1C(=O)Cn1cccn1 C(=O)(CCN=[N+]=[N-])NC(C)C(=O)NCCN1CCCNC1=O N1(C(c2cnn(CCOC)c2C)=O)CCCCC(NC(C2OCCOC2C)=O)C1 S(=O)(=O)(CCc1ccccc1)N(C(C1C=CCC1)=O)C1CC1 Cn1cnn(CC(=O)NCCCNC(C2CC2C(F)F)=O)c1=O c1(C(=O)NC2CN(C(c3scc(C(N)=O)c3)=O)C(CO)C2)cc(O)nc(O)n1 N1(C(C(C(C)C)CNC(C2CC2(C)C(F)F)=O)=O)CCC2CC1C(=O)O2 CC1CCOCCN1N1CCCC(Oc2ccc(F)cc2)C1 C12(C(CNC(=O)C(C)C#N)NC(CCc3cc(C)[nH]n3)=O)CCC(CC1)C2 C1(C(=O)NC(C2CCCC2O)C)C(C)CCN1C(=O)CC1CNC(=O)O1 C1(C(=O)Nc2cc(O)nc(C3CC3)n2)CC12CCN(Cc1cccnc1O)CC2 C(C(=O)N1OC2C=CC1CC2)C1(O)CN(C(=O)Cc2ccc(F)c(F)c2)C1 C1(COCC(=O)NC2CC(OCC(c3ccccc3)C)C2)CCC2(CCC2)O1 c1(CCCC(N2CCC(c3cn(CC4CC(=O)OC4)nn3)C2)=O)cccc(Cl)n1 Cc1ccc(Cl)cc1C(=O)NC(C)CN(C)C(C1CC1(C)C)=O N1(C(=O)CCC2CCCO2)CC(CNC(C2C3C4CCC(C4)C23)=O)C2(CC2)C1 C(=O)(CC(C(C)C)C(C)C)NCCC(C(C)(C)C)NC(C(C)SC)=O c1(OC)ccc(N)c(C(N2CCC(CNC(=O)COC(F)(F)F)(OC)CC2)=O)c1 c1(CCn2cc(CSCC(N3CCOCC3)=O)nn2)cnn2c1CCC2 c1(N2CC(C3N(C(c4cncc(C(F)F)c4)=O)CCCC3)C2)ncnc(O)c1Br C(CC(C)C)(C(=O)NCCc1ccoc1)NC(C(CC)OCC)=O N1(C(c2ccn(C(F)F)n2)=O)CC2CN(C(c3ncccc3Br)=O)CC2C1 CC1(C)CCC=C(C(=O)NCCCCNC(=O)C(O)c2cnc[nH]2)C1 CC1CC2(CCN(C(=O)CCCN3CCCC3)CC2)CN1C(C12CCC1C2)=O C1(C(=O)Nc2cccc(NC(c3n(CCC)ccc3)=O)c2)CC12CC(C)(C)C2 Cc1cc2[nH]c(C(=O)NCC3CC(C)(C)CN3C(=O)CSCC#N)cc2o1 C(CN=c1[nH]c(=NCC(C2CCCO2)OC)c2sccc2[nH]1)c1cn(CC)nn1 c1(C(N(C2CC2)CC2N(C(C3C(=C)C3C(=O)OC)=O)CCC2)=O)cc(Cl)cn1C N1(C(C(C)SCCCC)=O)CCC(CNC(=O)CCn2ccnn2)(COC)C1 Cc1nc(=NCC(CC(C)C)NC(=O)CCC2CCOC2)s[nH]1 CC1CC(F)(F)CN1C(=O)COC1CCN(C(C2CC2c2cccnc2)=O)C1 CCC(C)C(O)C(=O)N1CC(F)(F)CC1c1ccccc1C(F)(F)F c1(C(=O)NCC2CN(C(C(C)(C)OC)=O)CC2C)cc2cnccc2cc1F CC1CN(N2CCCCC2c2cncnc2)CCC1(F)F c1(CC(=O)NCCOCC2OCCCN(C(C)C)C2)cc(F)c(F)c(F)c1F Cc1cc(COC(F)F)nc(NC(C2CC(F)C2)=O)n1 Cc1nc(CO)ccc1C(=O)NCC12CCC1CN(C(c1cccc(N)n1)=O)C2 c1(C(=O)NC(C2N(C(C(C)c3ncco3)=O)CCC2)C)ccc(Br)cn1 CN1CCN(C(=O)CC2(C)OCCO2)C(C(=O)NCCC2CCC(C)(C)O2)C1 C=C(Br)CCC(=O)NCC1(n2ccnn2)CC1.c12cn(nn1)C1CN(C1)C2=O Cn1cc(CC(N2CCC2CNC(c2cncnc2O)=O)=O)c(Cl)n1 N1(C(c2cccc(OC(C)C)c2)=O)CC2CN(S(=O)(=O)CCCCl)C2C1 C1(NC(C(C)(C)OC(C)=O)=O)COCCC1NC(c1cnc(C(F)(F)F)nc1)=O N1(C(C2CCN(C)C(=O)C2)=O)CC2(CCCC2)C1C(=O)Nc1cncc(Cl)c1 N1(C(c2c(C)ccc(OC)n2)=O)CCC2CCN(C(=O)C(O)CN(C)C)CC12 c1(C(N2CC(NC(C(CC)(C)C)=O)C(OC)C2)=O)ccc(OC)cc1O c1(OC)cccc(F)c1C(C)OC(c1cc(OC(F)(F)F)cc(Br)c1)=O C1(C(=O)NCCC(CCNC(c2n(CC)cnn2)=O)C)CCCC(C)(C)CC1 c1(OC)cccc(C2CC(N3CC4(CCC4)C3)C2)c1 c1(C(N2CCN(C(CC(C=C)C)=O)CC2C)=O)cc(C)c(C)cc1C c1(OC)cc(C(=O)NC23CCN(C(=O)Cc4cnoc4)CC2C3)ccc1OC C1(NC(C2(COC)CN(C(=O)Cc3cnsc3)C2)=O)CC2CCC1N(C)C2 Cc1nc(C)n(CCN(C(C)CNC(=O)Cc2cnco2)C)n1 C12(C(=O)NCC3CCCN(C(CC4(C#N)CC4)=O)C3)CC3CC1(CO)CC3C2 C1(C(N2CC3C(CNC(c4cc(Cl)ccn4)=O)(C3)C2)=O)CC2CCC(C1)C2 C1(C(=O)NC2CC(NC(c3c(C(=O)OC)c[nH]c3)=O)C2)COCCN1C(C)=O N1(CCC(=O)NCC(=O)NCC(=O)NCc2ccoc2)CCCCC1 CN1CCCC1CNC(C1CC(CNC(c2cnn(CCO)c2)=O)C1)=O C1(C(N(CCN(C)C(C2CC(NS(C)(=O)=O)C2)=O)C)=O)CC(C2CC2)=NO1 C1(CC(=O)NC2CC(CNC(C(C)CN(C)C)=O)C2)OCCCC1(C)C C1(C(=O)NC(c2ccc(Br)cn2)C)C(O)CCN1C(c1ccc(F)cc1)=O c1(NCC(CNC(C2C(NC)COC2)=O)OC)ncccc1S(=O)(=O)NC1CC1 N1(C(c2c(CC#N)ccs2)=O)CCC2(CCC2)C(NC(=O)C=CC2CCCO2)C1 CC(C)C(=O)C(=O)NC1CCOCC1C(=O)NC(C1CCCC1)C CON=C(C(=O)NCC1CCN(C(=O)CC(C)(C)O)C(C)C1)c1ccco1 N1(CC=C)C(=S)NC(c2cc(C)c(F)cc2O)C(C(=O)N(C)C)=C1C C=CC(C)(CC)NC(=O)C(C)(C)NC(c1ccnn1C(C)C)=O c1(CCC(=O)N(C)CC2(NC(C=C(C)Cl)=O)CC2)c[nH]c2ccccc12 c1(C(CC2CC2)NC(c2nnc(C)s2)=O)ccc(C(F)C(F)(F)F)cc1 n1(CCCOC)nc(-c2cccc(OC(C)C)c2)nc1C1CC1CF N1(C(Cc2c(C)nc(O)nc2C)=O)CC(C)CN(C(c2ccns2)=O)CC1C c1(CC(=O)N(CC(C)NC(C(c2c(C)noc2C)C)=O)C)ccc(S(N)(=O)=O)s1 C(CC(C(C)(C)C)NC(=O)C(c1ccc(C)cc1)F)N(C(CCCSC)=O)C C1(C(=O)NCc2nc(CNC(CC=CC(C)(C)C)=O)sc2)CC(=O)NC(=O)C1 C1(NC(c2cccc(OC)c2O)=O)CC2CC(NC(C3(Cl)CC3)=O)CC2C1 O=C(NNc1ccnc(Cl)c1)Nc1cnn(C(F)(F)F)c1 C1(C(=O)NS(c2c(C)oc(C(=O)O)c2)(=O)=O)CCC(=O)N2CCCCC12 N1(C(C(=O)NCSc2ccccc2)C2(CCCCC)CC2)CCC2CCCC2C1 C1(NC(C(CCOCC)NC(C2CCC(=O)CC2)=O)=O)CCOCC1(C)C C(C(N=[N+]=[N-])C(=O)N1CCC(O)(Nc2ncc(C)cn2)C1)OCC C(CC(=O)NCC(=O)N(c1ccc(C)cc1)C)(C(F)(F)F)OC C(CN=c1ccnc(N2CC=CC2)[nH]1)OCC(N1CCC(OC(C)=O)C1)=O CN1CCCC1(C)C(=O)NCC1CCN(C(c2ccnn2-c2ccncc2)=O)C1 C1(C(N(C(C)C)CCN(C)C(c2cc(Cl)n(C)n2)=O)=O)CCN(C)C(=O)C1 C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(CCCC#C)=O C1(C(N(C)Cc2nnc(CC)o2)=O)CCCN1NC(=O)COCCC(C)C n1(CCC)ccc(CN(C=O)C(c2csc(Br)c2)C)n1 CCC(C)(C)C(C)CC(=O)N(C(C)CN(C(=O)COC(C)C)C)C C(CC(=O)NC1(CF)CC1)OCCN(C)C(C)=O C1(CC(=O)NC(CCC=C)C)CCCC(NC(c2cccnc2O)=O)C1 CC(C)(C)C(C(=O)NCc1cc[nH]n1)NC(c1cn[nH]c1)=O C1(C(CNC(C)CCC2CCCO2)(C)C)CCN(C(=O)OC(C)(C)C)CC1 C1(NC(c2ccc(CC)o2)=O)CCCCC1C(=O)NCCCSC(F)F c1(OCCC)ccc(CCC(=O)NCC(C(C)C)NC(C2CN(C)C2)=O)cc1 c1(C(C(=O)N(C)Cc2cc(N3CCOCC3)ncn2)O)ccc(Cl)cc1Br C1(CNC(C2CCC(C)(C)CC2)=O)CN(C(=O)CCN2CCCC2)CCC1(F)F c1(C(=O)NC(C(C)C)CNC(C2CC(N(C)C)C2)=O)c(F)c(F)c(F)c(F)c1F C1(NC(CSc2n(C)nnn2)=O)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CC1O C1(CNC(C2N(C)C(=O)CC2)=O)CCN(C(=O)C=Cc2ccsc2)CCC1(F)F N1(C(CC=CC=C)=O)CCCC(N(C(=O)CCOCC(C)(C)C)C)CC1 Cc1nn(C)cc1CN(C(=O)CCCNC(=O)CCCF)C Cn1nccc1CCNC(=O)CCC1CC(NC(C2CCC2C#N)=O)C1 C12(NC(C3CC(=O)N3)=O)CCCN(C(=O)C=CCCc3ccccc3)CC1C2 C(CC(C(=O)N(C1(C)CC1)C)NC(C1CCS1(=O)=O)=O)OC c1(NC)ccc(C(=O)NC2CCC2NC(=O)C(c2c(C)cccc2C)O)cc1F C12(CNC(CC(C)(C)OC)=O)CN(C(=O)C=C3CCOCC3)CC1(C(F)(F)F)C2 Cc1cc[nH]c1C(=O)NCC1CCC(NC(=O)CSc2n[nH]c(O)n2)C1 N1(C(C=CC(C)(C)NC(c2cnsn2)=O)=O)CC2CCC2C1 C1(C2CCC2)(CNC2CCN(C(C(C)C)=O)C2)CCNCC1 N1(C(C(CC)N(C)C(c2cccnc2N)=O)=O)CCOC(CN(C)CC)C1 c1(C(=O)NCC2N(C(Cc3nnc(C)o3)=O)CC2)ccc2c(c1)CN(C)CC2 C1(C(N2CCC(NC(C(C(CC)C)OC)=O)C(CC)C2)=O)CCn2ccnc2C1 N1(C(c2ncn(C(C)C)n2)=O)CC(C2CN(C(c3coc(C4CC4)n3)=O)C2)C1 c1(CC(N2CC(C(C)NC(C3CC(C)(SC)C3)=O)C2)=O)nc2ncccn2n1 S(=O)(=O)(c1ccc2c(c1)C(=O)NC2=O)Nc1ncc(C)[nH]1 c1(C(N2CCC(CNC(c3cnc(CCCC)s3)=O)C2)=O)cccc2c1OCC2 C=C1CN2C(=O)CCC2(C(=O)NC2CC2NC(C2OCCO2)=O)C1 C(C(C)(C(C)C)NC(c1cnn(C)n1)=O)NC(C(Cc1ccccc1)OC)=O c1(C(=O)NC(c2ccsc2)C)nc2ccccn2c1-c1cccc2c1ccn2C C1(CNC(C=CCC)=O)N(C(C23CC4CC2C3C4)=O)CCCC1(C)C C=C(C)CC(C(=O)NCC(c1ccco1)O)NC(c1sccc1C)=O C12(CNC(c3cc(C)sc3)=O)CCCN(C(=O)COc3cccc(C)c3F)C1C2 C1(C(N2CC3(CN(C(C4C(C)(Br)C4)=O)C3)C2)=O)Cc2ccccc2N1 CCC(CNC(c1ccc(C(C)(C)O)cc1)c1nnnn1C1CCCC1)CCO C1(C(N(CC(CN(C)C)O)C)=O)COCCN(C(c2ccc(C#N)cn2)=O)C1 C1(NC(=O)CCn2ccnn2)CCC2(CC1)CN(C(c1cnco1)=O)CCO2 c1(N2C3CC(NC(C(CCCNC(=O)OC)O)=O)C(C3)C2)cc([N+](=O)[O-])ccc1C N1(C(CCC2CCCN(C(c3c(C)noc3C)=O)C2)=O)CCCN2CCCC2C1 c1(CC(N2CC(n3cc(CCCC)nn3)C(C)C2)=O)ccc(OC)c(Cl)c1 C1(CC)CN(C(C2CCC2(C)C)=O)CCC1NC(=O)CCCn1ccnc1 c1(NCC(c2ccccc2)NC(c2ccc(C)[nH]2)=O)cc(O)ncn1 CC1CN2CCN1C(C(=O)NCC#CCNC(=O)CC1CCOC(C)(C)C1)C2 N1(C(c2cc(C)oc2C)=O)C2CCCC1CC(NC(c1ccnc(C)c1N)=O)C2 c1(C(=O)NCC2(C)CCC(NC(COCCOC)=O)C2)nc(C)ncc1Br N1(C(c2nc(C)[nH]n2)C(=O)NCC2CCC2)CCCC(C)(CN(C)C)CC1 c1(SC)ccc(C(=O)NC(C)C(C)NC(c2ncnc(O)c2F)=O)cc1[N+](=O)[O-] c1(C(=O)NCC23N(C(=O)CO)CC(COC)(C2)C3)ccc2oc(S)nc2c1 c1(C(=O)NC2CCCC(NC(c3ccc(F)s3)=O)C2)csc2ncnc(O)c12 N1(C(c2ccc(CC)[nH]2)=O)CCC2CC12C(=O)NOCCOCCF C(C)(C)(CC(F)(F)CC)NC(C(OC)OC)=O C1(NC(c2ccc(C(=O)OC)c(O)n2)=O)COC2CCCCC12 N1(C(Cc2ccc(OC)cn2)=O)CC(C)CCC1CNC(=O)CC(C)(C)C N(C(=NCCc1nc2c(s1)CCCC2)N1CCCC2(CCOC2)C1)C(COC)C C(C(=O)Nc1ccc(-n2cnnn2)cc1)(C(C)C)OCC(C)C c1(C(N(C(C)(CC2CC2)NC(=O)OC(C)(C)C)C)=O)ccc(C(F)(F)F)c(Cl)c1 C1(NC(C2C(c3n(C)ncc3)C2)=O)Cc2nc3ccccc3n2C1 c1(C(=O)NC2C(CNC(CCCOCC=C)=O)CCC2)cncc(N(C)C)c1 Cc1cccc(C)c1CC(=O)NC(C12CCC(CC1)C2)CNC(=O)C(C)S(C)(=O)=O c1(N2CCC(c3c(OC)cccn3)C2)nc(N2CCC(C#N)C2)c2sccc2n1 C1(C(N(CC(C)NC(C2CSCN2C(=O)OC(C)(C)C)=O)C)=O)COCCO1 c1(OC)cc(OC)cc(C(=O)NC(C)CN(C)C(c2c(C)ccnc2Cl)=O)c1 c1(C(N2C(CN(C(=O)CC(C)(C)O)C)CCCC2)=O)cccc2[nH]cc(Cl)c12 c1(CC(=O)NC(C(=O)NCCCN2CCCCC2)c2ccco2)ccc(O)cc1 c1(C(N2C(CNC(c3cc4n(n3)CC(F)C4)=O)CC2)=O)cc2nc[nH]c2cc1F C1(OC)CC2CCC(C1)N2C(c1coc(C(C)NC(c2ccc(C)o2)=O)n1)=O O(NC(=O)CC1CC1NC(c1c[nH]cc1C1CC1)=O)CC(C)C C(=O)(C#CC1CCOCC1)NCC1N(C(c2ccc(OC)c(N)c2)=O)CCC1 CCC(CC)(CCNC(=O)C(SC)SC)NC(=O)CCSc1ccccn1 N1(CC(=O)NCC(=C)CCNC(C2(C)CC2(F)F)=O)CCC(OCCOC)CC1 C1(=O)C(NC(C2(c3ccsc3)CC2)=O)C(=O)NCC12CC2.CCOCC c1(C(=O)NC2C(F)CCN(C(CCCC(C)C)=O)C2)cc2ccccc2nc1O c1(OC)cnc(C(=O)N(C(C)(C)CCNC(C2(CF)CC2(F)F)=O)C)nc1 N1(C(C)=O)CCC(c2nnnn2C)(NC2CC(=O)N(C)C2)CC1 CC1CN(C(C2CC3(C2)CC(F)C3)=O)CCC1NC(C1Cc2cscc2C1)=O C1(C(=O)NCc2cc(OC)ns2)CN(C(C2CCCC2)=O)CC12CC2 C(C1(O)CCc2cc(F)ccc21)NC(N1CC(C)(C)C(CC(N)=O)CC1)=O Cc1cc(C(N2CCOCC2CN(C)C(C2CC2CF)=O)=O)c2c(O)n[nH]c2n1 Cc1cc(=O)n(C)cc1C(N1CC2(CCC2)CC1CNC(=O)C(C)S(C)(=O)=O)=O CCC(C)(CC)C(=O)N1CCN(C2CN(C(=O)COCCF)C2)CC1 N1(C(c2ccc(C)nc2)C(=O)NCCOCC)CCOCC12CCC2 C#CC1CN(C(c2nnn(C)c2C)=O)CCN1C(=O)C(COC)OC C#CC1(O)CN(C(=O)CCC2(NC(=O)C(O)CC)CCC2)C1 N1(C(c2cccc(C(=O)Nc3cccc(OC)n3)c2)=O)CCCC(C)(F)C1 CCCCC(C(=O)NCC12CC1CN(C(=O)C(CO)N(C)C)C2)N(C)C Cn1ccc2cc(C(=O)NC3CCCCN(C(C4(CF)CC4)=O)CC3)ccc12 c1(N2CCC(NC(c3ccc(C)c(OC)c3F)=O)C2)nc(C)nc2[nH]ccc12 CN1CCN(C(c2cc(C3CC3)[nH]n2)=O)C(C(=O)NC2CCCN(C)C2)C1 N1(C(C=CC(C)NC(C(C)C2CCC2)=O)=O)CCOCC12CC2 C1(C)COC(C)(C)CN1C(=O)C(CCC)C=O.n1(CC=C)cc(C=CC(C)C)nn1 c1(C(N2CCCC(O)(CNC(CS(CC)=O)=O)C2)=O)cc(Br)c(C)nc1O C(=O)(C(CNC(c1sncc1C)=O)CC(C)C)NC1C(OC)C(C)(C)C1 C1(NC(c2ccnc(C(F)(F)F)c2)=O)CCN(C(c2nc(Cl)cs2)=O)CC1O C1(CNC(C(C)(C)c2cc[nH]n2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C2(CCC2)C1 CN1N=C(CC(=O)NC2CC3COCC(C2)N3C(=O)CSC(F)(F)F)CC1=O C12(C(N3C(CNC(=O)CSc4ccncc4)CC(OC)C3)=O)CCCC1C2(F)F c1(C(=O)NC2(C)CC(NC(C3(C(=O)NC)CC3)=O)C2)c[nH]c2nc(Cl)ccc12 N1(C(=O)CC2CCCN(C(c3ccc(O)cn3)=O)C2)CCC2(CCCO2)CC1 N1(C(C2CC(=O)NC2)=O)CC(NC(c2c(Br)cncc2Br)=O)C(F)(F)C1 C(CC(C)C)(C(=O)NC1CCN(C(=O)C(C)CC(N)=O)CC1C)NC(C)=O C(=O)(C1=CCCSC1)N1CCC(CNC(CCc2ccc(=N)[nH]c2)=O)CC1 N1(C(CCCC(C)=O)=O)CCCC2(CCCCC2NC(=O)CCCN(C)N=O)C1 CC1=NN(C)C(=O)C1CC(=O)NC(C)CCN(C)C(c1cc(Cl)cs1)=O N1(C(Cc2n(C(C)C)cnn2)=O)CC(NC(=O)CN2CCS(=O)CC2)C(C)(C)C1 C1(CC)CN(C(=O)C(O)C2CC2)CCN1C(c1ccc(C(C)(F)F)cn1)=O c1(C(N2C(C(=O)NCCN(CC)CC)C(C)CC2)=O)ccc(F)c(C)c1F C1(NC(c2c(C)ncn2O)=O)CC2CC(C1)N(C(c1scnc1Cl)=O)C2 N1(C(CCC=C)=O)CC(=O)N(C)CC1C(=O)OC.c12cn(nn1)c1ccsc21 C1(C)(CNC(c2c(C)n(C)nn2)=O)COCCN(C(=O)C2=NOC(C)C2)C1 C1(C(N2CC3C(CNC(=O)CCc4ccoc4)(C3)C2)=O)CCC(F)(F)CC1 c1(CC(=O)NC(CC2CN(C(C3C(CC)OCC3)=O)C2)C)ccc(CC)cc1F C(=O)(CC(CC(C)C)NC(=O)Cc1sccc1C)Nc1c(C)ccc(C)c1 C(CC(=O)N1CCC(N(C(c2nccnc2C)=O)CC)C1)(C(C)C)OCC c1(C(C(=O)NC(CNC(C(C=C)O)=O)C(C)C)(F)F)ccc(F)cn1 C(=O)(C1=NN(C)C(=O)CC1)NCC(C(=O)NCC#CC)CC(C)C c1(CCC(NC2C3C(CNC(C)=O)C(CC3)C2)=O)nc2cc(C)cc(C)c2[nH]1 O=C1CCC(C(=O)N2CC3CC3(C(=O)Nc3nccc(C(F)F)c3F)C2)=NN1 CN1CCN(C(c2cccc(N3CCCC3)n2)=O)CC1CNC(C1CCO1)=O c1(C(=O)NC2CC(NC(C34OCC(C(C)C)(C3)C4)=O)C2)ncc(Cl)cc1Cl C1(NC(C(C)(C)OC)=O)Cc2ccccc2C1Nc1ncnn2c(Br)ccc12 C(CCc1ccccc1)(C(F)(F)F)NC1(c2n(CC)nnn2)CCSC1 c1(C(CC)(C)C)ccccc1C(=O)NCC1CCN(C(C2C3CCCC23)=O)C1 N1(C(C2N(C(Cc3cc(C)on3)=O)CCCCCC2)=O)CCC(C2=NOCC2)C1 C(N=c1[nH]c(Cl)ncc1C(=O)OC)C1CN(C(CN(CCC)C)=O)CC1(C)C CC(C)C(O)CC(=O)N(CC(C)(C)NC(c1ccc(C(F)(F)F)[nH]1)=O)C N1(c2nnc(C3C(CC)C3)n2Cc2ccccc2)CC(OC)CC2CCCCC12 CCC(C)C(O)C(C)C(=O)N1CCC(NC(c2c[nH]nc2C2CC2)=O)CC1C C(C)(CCC(=O)N1CCCC1(C)CNC(=O)CCc1cnco1)OCC C1(C(N2CC(NC(C3C(C=C)C3)=O)CC2(C)C)=O)CCC(=C(F)F)CC1 CN1CCc2cc(C(=O)NCCC3CC(NC(c4cnn(C)c4N)=O)C3)sc2C1 C(=O)(CC(C)C(F)(F)F)NCCCN(C(C)C)C(C12CCCC1CCC2)=O C1(C(N2CC(O)(CN(C(=O)CCc3ccncc3)C)C2)=O)CC2(CC2)CN1C N1(C(CC(C)c2cnn(C)c2)=O)CCN(C(=O)CC2(O)CCC2)C(CCO)C1 C12CCCC(N=CNN=C(CCOC)S1)CC(CC)CCC(CC)C(=O)N2 c1(C(N2CC(F)(CNC(C3=CCCCC3C)=O)C2)=O)cnc2c(ncn2C)c1 C(=O)(C(CC(C)C)C(N)=O)NCCCCCCNC(c1cncc(NCC)c1)=O C#CCC(C(=O)N(C1CCN(C(C2(C3CC3)CC2)=O)CC1)CC(C)C)C1CC1 c1(C(=O)OC)cc2c(s1)CN(C(=O)CC1CCCCCC1)CC2 C1(C(=O)Nc2ccc(C)c(NC3CC3)c2)CC2CSCC(C1)C2 N1(C(c2snc(Cl)c2Cl)=O)CCC(N(CCO)C(c2[nH]nnc2C2CC2)=O)CC1 C1(CC(=O)OC)CC(C)(C)CN1C(=O)CCc1ccc(Br)cc1Cl c1(C(=O)NCCOCCNC(C(CC#C)CC#C)=O)ccc2[nH]ccc2c1F C(=O)(C(F)(CNC(C1(O)CCC1)=O)C(C)C)NC1C(SC)CCC1 C1(CNC(C(=O)NCC)=O)CN(C(=O)COc2cccc(C)c2)CCC1C C=CC(CCC)CC(=O)NC1(C)CCCC1NC(c1cc(Cl)cs1)=O CC1CCC(CCOCC2(NC(=O)Cn3cccn3)CC2)O1 C1(CNC(C(CC)OC)=O)CCCN(C(c2cn(Cc3nc(C)cs3)cn2)=O)C1 C(=O)(CC(C)(O)C1CC1)N(CCC1CN(C(C(CC)Nc2ccccc2)=O)C1)CC CON(C)C1CN(C(C2CCCC2NC(=O)C(C)N2CCCC2)=O)C1 Cc1nc(C(=O)N(C2CCC(NC(=O)C(C)(C)n3ccnn3)C2)C)c(C)o1 C1(C(=O)NC(CN(C(C(C)=C(C)C)=O)C)C)(CF)CC1(F)F C1(NC(C2(CF)CCNC2=O)=O)COC2(CNC(c3cc(Cl)ccn3)=O)CC1C2 c1(OC)ccc(C(=O)NC(C)(CNC(c2ccc(Cl)cc2OC)=O)CO)c(Cl)c1 Cn1ccc2cnc(N3CC(NC(c4ccc5cnn(C)c5c4)=O)C(N)C3)nc12 CCC1=NOC(C(=O)NC(CO)C(=O)NCCc2ccon2)C1 c1(C(=O)NCC2N(C(C3(C)CCC(=O)NC3)=O)CCC2)cnc2[nH]nnc2c1 c1(CC)cc(C(=O)NCC(C2CCCC2)NC(=O)C(C)CC)n(C)n1 S(=O)(=O)(c1cccc(=NCC(=O)NC2CCCC2)[nH]1)NCC1C(C)(C)CCC1 N1(C(Cn2c(C)ncc2)=O)CCC2(CCCN(C(=O)CC3CCCOCC3)C2)C1 c1(OC)ccc(CN2CCCC(C(=O)NC3CCC(F)(F)C3)CC2)c(Br)c1 c1(CCCC(=O)NC(c2cnc(C)s2)C)nc(-c2ccccc2)nn1C C1(C(N(C)CC2(NC(=O)Cc3ccccc3O)CC2)=O)CCC12CCOCC2 c1(C(N(C2CCN(C(C3CCOC3=O)=O)C2)CC)=O)cc2n(n1)CC1(CC1)C2 C=CCCC(C(=O)N1CC(N(C)C)C(C)C1)NC(c1cc(C2CC2)on1)=O N1(C(c2ccn(C)n2)=O)CCC(F)CC1C(=O)NCC1(C)CCC(=O)N1C C1(NC(COC)=O)CN(C(c2cccc(C#N)c2)=O)Cc2ccnn2C1 C1(C(N2CC(NC(=O)C(F)F)C3(CC3)C2)=O)(OCC)CCC(F)(F)CC1 C1(CNC(CCCOCCOC)=O)CC(NC(=O)C(C)O)C(O)C1 C(CS(=O)(=O)CC(=O)NC(C1(C(=O)NC2CCC(=O)N2)CC1)C)OC C1(CC=C)(NC(c2cc[nH]c2C)=O)CCN(C(c2c(C)nn(CC)c2Cl)=O)CC1 C1(CNC(c2cc(C)oc2)=O)CC(F)(F)CN1C(c1coc(C)n1)=O N1(C(CC2(OC)CC2)=O)CC(F)(F)CC1CNC(c1cnc(-c2cccs2)s1)=O C1(CC=O)CC=CCC1.C(=O)(CNC)N(CCOCC)CC.C1(=O)CN1 N1(C(C(C2CN(C(=O)CCCc3ncco3)C2)OC)=O)CC2CCC(C1)C2C#N c1(C(N2CCC3(CCN(c4ncccn4)C3)C2)=O)cc(Br)cc2cn[nH]c12 C1(C(C)C)(C(=O)NCCCOCCO)CCN(C(=O)Cc2ccccn2)C1 N1(C(C2CCC(CC)O2)=O)CCC(NC(=O)CSCCN(C)C)C1CC C1(CCC(=O)N2CC(N3CCC3)C2)CCN(C(=O)CC2(O)CCCC2)C1 CC(C)C(O)C(F)(F)C(=O)N1CCC(=CCNC(C2CCC(=O)N(C)C2)=O)CC1 N1(C(C(=O)NC(COCC)(C)C)=O)CC(OC)CC(C(=O)OC)C1 C1(NC(C2C(C)C2)=O)CC(N=c2[nH]ccc(C#N)c2[N+](=O)[O-])C12CCC2 C1(C(F)(F)F)(CNC(c2n(CC=C)nnn2)c2csc(Br)n2)CCCCC1 c1(CC(=O)NCCN(CCC)C(c2ccccc2OC)=O)ccc(Cl)cc1 C1(C#N)(C(N2CCC(N(N3CC(O)C3)C)CC2)=O)CC2CC2C1.C1(C=O)CCCSS1 C12(C(=O)NCCCCCN(C(CC(=O)NCC#C)=O)C)CCC(CC)(C1)OC2 c1(C(N(C2CCN(C(Cc3c(OC)nccc3)=O)C2)C)=O)cccc(F)c1Cl C(CC(C)C)(C(=O)NCC1CCN(C2CC2)CC1)NC(CC=C)=O c1(C(N2CCCC(C(C)NC(=O)C(F)OC(F)(F)F)C2)=O)cc(N)cc(O)c1 c1(CC(N2CC3CC(CNC(COCCOC)=O)C3C2)=O)c(C)nc(O)nc1C c1(CC)ccc(Br)cc1C(=O)NCCC1CCCCN1C(=O)C=CCO C(=O)(C1COc2cc(C)c(C)cc21)N(C(c1ncccn1)(CC)C)CCO c1(C(=O)NCC2COC(=O)O2)ccc(Cn2cc(C3CC3)nn2)cc1 c12nocc1C(=O)NC2.C(C(C)(C)CSC)NC(C1(OC)CCC1)=O N1(C(c2cc(C(=O)OCC)n[nH]2)=O)CC(NC(=O)C(CC)SC)CC1C(=O)OC Cc1cc2cc(C(=O)N(C(C)CNC(=O)Cn3ccnc3C(C)C)C)ccc2[nH]1 C(N=c1[nH]c(C(F)F)nc2ccccc12)C1C(OCC=C)CCC1 CC(C)CCC(=O)NCCC1CCN(C(C2(CC(F)F)CCOCC2)=O)C1 CC1C2CCC(C2)C1C(=O)NC1CC2(C1)CC2NC(=O)CC1CCC(C)(C)C1 C(CCCC(C)(C)C(=O)NNC(=O)CCCC1CCC1)NC(c1c(C)occ1)=O C1(NC(=O)NCC(=O)N(CCN(C)C)Cc2nccs2)CCSCC1 c1(C(=O)NCC2C(NC(C3CCC(CC)O3)=O)C2)cc2c(cc1Br)OCO2 C(=O)(C1=C(Cl)CCCC1)N(C1CCN(C(=O)CC2CC(O)C23CCC3)CC1)C C(=O)(C1=CC2C=CC1C2)NCC1CCN(C(CCc2c(C)cccn2)=O)C1(C)C c1(C(N2CC(CN(C(CCCC(=C)C)=O)C)OCC2)=O)ccc(F)c(F)c1F C1(NC(C2(OC)CC2)=O)CCC(C)(C)CC1CNC(=O)CN1CSCCSC1 N1(C(c2cncc(C)n2)=O)CCN(C(c2ccc(C(C)(C)C)nc2)=O)C2CC12 C1(CNC(=O)NC(COCCCC)C)CCC(C(=O)OC(C)(C)C)CC1 CN1CCOC(C(=O)NC2C3CC2N(C(=O)CSCc2cccnc2)C3)C1 CN1CCC(CC(=O)N(CC(C)(C)NC(c2cc(-c3cnn(C)c3)[nH]n2)=O)C)C1 N1(C(C=C2CCC(C)CC2)=O)CCC2CN(C(C3CCCCCC3)=O)C2C1 C(C1(C)CCOCC1)=CC(N1CCOCC(NC(CCSCCCC)=O)C1)=O C12(NC(C=CC)=O)CC3CC(C1)CC(NC(=O)C(C)CSc1ccccc1)(C3)C2 c1(NCc2cn(C3C(C(=O)OCC)CCC3)nn2)ccc(-c2n[nH]c(C)n2)cc1 C12(CNC(c3c(OC)cnnn3)=O)CCC(CC1)N2C(C1(C)CCC2CC2C1)=O C(CNC(Cc1ccc(C(=O)NC)c(C)c1)=O)(C(C)C(C)C)NS(CC)(=O)=O C=CCC(CNC(=O)C(C)(C)C(O)C(C)C)C(=O)NOCC(N)=O Cc1ccc(F)cc1C(=O)NCC1CC(NC(=O)CN2CCCCS2(=O)=O)C1 c1(NC(C(CCSC)NC(=O)CC2CCCC23CC3)=O)ccc(O)c(Cl)c1 N1(C(c2c(C)nn(C3CC3)c2)=O)CC(CNC(C2CS(=O)(=O)C2)=O)C(F)(F)C1 CC1OC(=O)NC1C(=O)NCC1CC(F)(CNC(=O)OC(C)(C)C)C1 CC1CC(C(=O)N(C2(C(=O)Nc3ccc(C(C)C)cc3)CC2)C)CCC1=O C#Cc1ccc(C(=O)OCC)nc1.C12(CNC(=O)C1)C(=O)O2 C(=O)(CCC(=O)C(C)(C)C)N1C2(C(=O)Nc3c(OC)ccc(C)c3)CC2CC1 c1(C(=O)NC2CCC(CNC(=O)C=Cc3cc[nH]c3)C2)cnnc(O)c1 N1(CCC=O)C2=CC=CSC(CC)C(C1)N(C)C(=O)C2(C)N(C)C C1(NC(c2cn(CC)nc2C)=O)CCCC12CN(C(c1sccc1COC)=O)C2 CC1CCCN(C(C2C3CCC2CC3)=O)C1CNC(=O)CN(C1CCC1)C C1(CNC(c2cn(C)c(O)n2)=O)CC2CCC1N2C(c1cccc(C2CC2)n1)=O N1(C(CC2CCC(C)(C)CO2)=O)CC2(CC(NC(C3(O)CCOCC3)=O)CO2)C1 c1(C(N(CCN(C(=O)CCC2CCC(=O)N2)C)C)=O)nc2ccccc2s1 C1(C(=O)NCC(CCCCC)O)CC2(CCC2)CN1C(=O)CCCNC(=O)OC N1(C(C2(C)CC2Br)=O)CCC2(COC(CNC(c3c(F)cccc3F)=O)C2)C1 C1(C(N2CCC(NC(C(C)OCCCC)=O)C(O)C2)=O)CC(F)(F)C12CCC2 c1(NC(C(C)N(C(c2c(C)n[nH]c2)=O)C)=O)ncccc1C(C)C c1(C(=O)Nc2ccc(N(C)C)nc2)ccc(F)c2occc12 C1(NC(=O)Cc2ccncc2)CCC2(CC1)CCN(C(=O)CC1CC1)CC2 c12ccc(cc1)CNC2=O.c1(OCC2(O)CN(S(C)(=O)=O)C2)ccccc1Cl c1(C(N2CCC(NC(C3CC4(C3)CC4(F)F)=O)C(F)C2)=O)cc[nH]c2nccc1-2 C1(NC(=O)CCc2ccccc2)(CNC(c2ccco2)=O)CC2CCC1CC2 C(=O)(C1=CC(O)CCC1)N1CCC(CCNC(CNC(=O)OC(C)(C)C)=O)C1 C(=O)(C(CC=CC)NC(c1c[nH]c(=S)cn1)=O)N(CCOCC=C)C CCC(O)C(=O)NCC(C1CCC1)NC(=O)Cc1ncc(Cl)s1 C1(CNC(Cc2ccc(CCC)cc2)=O)COCCN(C(c2cnc(C)s2)=O)C1 c1(CC)nc(CN(C)CC2CN(C(=O)C(C)NC(c3ccccn3)=O)C2)n[nH]1 C1(CNC(CCSCC)=O)CCCCC1NC(=O)C(C1CC1)SC CCCC(C(=O)NCC(CC(C)C)NC(C1(OC)CCC1)=O)NC(C)=O N1(C(c2ccncc2Cl)=O)CCC2OCCN(C(C3CC4C=CC3C4)=O)C2C1 Cc1cc(C(=O)NC(C)CN(C(=O)Cn2nccn2)C)n(C(F)F)n1 C1(N(C(=O)C=CC(C)SC)CC)CC(NC(=O)C(C2CCC2)OC)C1 C(=O)(C#CC1CCCCC1)N1CCC(=CCNC(C(=Cc2cn[nH]c2)C)=O)CC1 C(C1c2ccsc2CCN1Cc1cccc2ccncc12)NC(=O)OC(C)(C)C c1(OCC(=C)C)ccccc1C(=O)NC1CC(NC(c2n[nH]cc2Cl)=O)C1 C(C1CN(C(=O)C(N2CCNC2=O)C)CC1C(=O)NC(C)CCCCCO)=CC C1(NC(CC=CC)=O)CCCCCN(C(=O)C(=Cc2cnc[nH]2)C)C1 c1(CNC(c2c(C(=O)OC)c(C)[nH]n2)=O)ccc(I)c(Cl)c1 C1(C(N(C(C)CO)CCC)=O)COC2(CCN(C(c3ccno3)=O)CC2)C1 C12(C(N3C(C)(CCO)CC3)=O)CCC(CN(C(C3(C)CCCC3O)=O)C1)C2 C(c1nnn(C)n1)=CC(=O)N(CCCCN(C(=O)CCCN1CCCC1)C)C c1(OC)cc(C)c(C(=O)NC2(C)CC(NC(=O)C(C3CCOCC3)C)C2)cc1Cl C1(CNC(CC2CCN(C(C)=O)C2)=O)CC(F)(F)CN1C(c1cc(C(C)=O)c[nH]1)=O N1(C(C(C)n2ccnc2)=O)CCC2CN(C(=O)C(=O)NCC(F)(F)F)CC12 N1(C(c2cc(C(=O)NC3CCCCO3)c(F)cc2)=O)CCC2(CCNC2=O)CC1 C(=O)(C(C)(CC)CCC)N1CCC(C(C(=O)NCC2CCN(CCC)C2)F)C1 C1(C(=O)NC(CCCOC)(C)C)CC(C)CN(C(c2sccc2C#N)=O)C1 C1(NC(c2ccnc(Cl)c2Cl)c2n(CC)nnn2)CC2CC(OC)C2C1 c1(CCNC(C(C)C2CCCO2)=O)ccc(CNC(=O)Cn2ccnn2)cc1 C(C(C)C(C)C(=O)NCC(COC)(C)C)NC(=O)CCCNC(C)=O Nc1ccc(C(=O)NC(CNC(C2CCC2)=O)Cc2ccccc2)nc1 O(NC(=O)C(CC(C)(C)C)NC(=O)Cc1ncccc1C)CC#C C12(C(=O)NC(C)CN(C)C(c3cc(C#N)cn3C)=O)CCCC(C1)C(=O)NC2 C1(CCC(=O)NCC(=C2CN(C(C=CC(C)(C)SC)=O)C2)F)CCCCN1C C1(OC)CC(NC(=O)OC)CN(C(C23CCCC2(C(=O)O)C3)=O)C1 Cc1cc(C(N2CCCCC2CCNC(=O)CCSC(=N)N)=O)ccn1 c1(C(=O)NCC(CC)NC(C2CC(C3CC3)C2)=O)cc(C)c(CO)cn1 C(C(NC(=O)NCCOCC1CCC1)NC1CC1)OC C1(CC=C)CCN(c2cc(N(C)CC3(OCC)CCOCC3)ncn2)CC1 C1(CC(N2CCC(CC(C)C)C2)=O)C2CCCC2N1C(c1cccc(F)c1)=O c1(C(C(N2CC(C(C)NC(=O)CCC3CCCN3C)C2)=O)O)ccc(F)cc1 C1(CC)(CC)C(OC)CC1N=c1cc[nH]cc1S(=O)(=O)NCCc1ccn(C)n1 C1(CNC(C(C(C)(F)F)F)=O)CC12CCN(C(c1cnn[nH]1)=O)CC2 CCCCCCC(C(=O)N1CCC2C(NC(c3ccco3)=O)CC12)NC(C)=O c1(C(N2CC3(CCCC3Nc3cc4nncn4cn3)C2)=O)cnc2cc[nH]c2c1 N1(C(=O)NC)CCC(C(=O)NC2(CO)CCN(C(c3ccc(CO)o3)=O)C2)CC1 C(=O)(C(C)(C)CC(=O)N1CC(F)CC1CC(=O)N(C(C)CC(C)C)C)OC C1(NC(C(C#C)(C)C)=O)CC2(C1)CC(CNC(c1ncccc1N)=O)C2 c1(C(=O)NCCC2CC(NC(c3c(C)ccs3)=O)C2)cnc2nccn2c1 CCCC(C)(CC)C(=O)NOCC(=O)NC1CN(C(=O)C2CC2)C1 C1(C(N2C(C(=O)NCCc3ncc(C)o3)C=CC2)=O)CCCC1C1CC1 CCCCN=C(NCCC1(O)CCCOC1)NC(C)CC C1(C(C(=O)NCCC(C)NC(c2cc(C)nn2C2CC2)=O)C)CCC(C)(C)CC1 C1(C)(C(=O)NCC=CC(N2CC(OC(=O)NC)C2)=O)CCC(=O)NC1 C1(NC(C2(C)C=CCC2)=O)CN(C(=O)CC2OCCO2)CC2(CCOCC2)C1 CCCC(C)(CCC)C(=O)NC1CN(C(C2CC2CC(C)C)=O)CC1CC1CC1 C1(NC(C(COC)OC)=O)CCN(C(=O)CCCNC(C)=O)C12CCC2 Cc1cc(NC(C2CCCS2(=O)=O)=O)ccc1NC(=O)CCN1CCN(C)CC1 N1(C(C(C)C#N)=O)CC2CCCC(C1)N2C(C1CCn2cnnc2C1)=O C1(CCC=C)(C(=O)NC(C2CCOC2)CC)CN(C(=O)C(C)=C(C)CC)C1 C1(NC(=O)CC2COCCO2)CN(C(=O)C=CC2CC2)CC12CCCC2 c1(OC)cc(C)c(C(=O)NCC23CCN(C2)C(=O)C3)cn1.c1(OC)cccnc1 Cc1cccc(C(N2CCCC2CN(CCCc2cc(Cl)sc2Cl)C)=O)n1 C(=O)(C1CCCc2sc(C)nc21)N1C2CC(NC(c3cc(C)oc3C)=O)(C2)C1 Cc1nn(C)c(Cl)c1C(=O)NC1CC(CO)N(C(C2CC23CC3)=O)C1 c1(CC(N2CCCC(Cn3cc(C4(C)CCCC4)nn3)C2)=O)cc(F)cc(F)c1 C1(OC)C(NC(=O)CNC(=O)C(C)(C)n2cccn2)CC1O C(CC(C)C)(C(=O)NCC1(NC(C2CCCC(C)(C)C2)=O)CCOCC1)OC N1(C(C2(c3cccnc3)CCC2)=O)CCCC(NC(C23COCC(C2)C3)=O)CC1 C1(NC(c2cc(OC)nn2C)=O)C(C)(C)CN(C(=O)CP(C)(C)=O)CC1(C)C S(=O)(=O)(c1cccc(=NCCC(C)N2CCCCC2)[nH]1)NC1(CC=C)CCOC1 C(CC(=O)N1CCC(NC(=O)Cc2cc(F)cc(F)c2)C1(C)C)(C(C)C)OCC N1(CC#CCOCC)C(=O)c2ccccc2C1=O.C1(C(F)(F)F)CN1 N1(C(c2c(COC)cco2)=O)CCCC(C)C1CCNC(c1cc[n+]([O-])cc1)=O CC(C)S(=O)(=O)C(C)C(=O)N1CC(CC(=O)C(C)C(F)(F)C(F)F)C1.N C(=O)(CCCCCC(C)O)NCCC1(O)CCN(C(CC(CC(C)C)C)=O)CC1 C1(N(C(=O)CCCC2CCCC2)C)C2CN(C(=O)COCC3CCC3)CC12 N1(C(CN(CCC)C)=O)CC(C)OC2(CCN(C(C3CC4C=CC3C4)=O)CC2)C1 c1(CNC(C(CC)=CC)=O)cc(O)nc(CNC(=O)C(F)CC2CCOC2)n1 CC1CCCCC1CCNC(=O)NCCc1csc(Br)c1 C(=O)(C(F)(F)C(F)F)NCC1(CNC(C(C)(F)F)=O)CCCCC1 S(=O)(=O)(c1c(C)ccc2ncccc12)N1CC(CC)N(C(C(C)(C)C)=O)CC1 C1(CNC(CNS(CCCC)(=O)=O)=O)CN(C)CCN1C(c1cccnc1Cl)=O c1(C(N2C3CC(CC(NC(C4CCC4CF)=O)C3)C2)=O)cc2c(F)cccc2s1 c1(C(=O)NCC(C)N(C(CNC(C(CC)C)=O)=O)C)cccc(OC(C)C)c1F c1(OC)cscc1C(C(=O)Nc1ccccc1)N(CC(=O)NC1CC1)C Cc1cc(C(N2CCCC2CNC(=O)CSc2cnn(C)c2)=O)on1 C(=O)(C(C(C)C)N1CCCC1=O)NCC(CNC(C(C)C)=O)F C#CCCCCC(=O)NCC(C)(C1CCC1)NC(=O)Cc1ccc(F)c(C)c1 C1(COC)(NC(=O)CCCF)CCN(C(c2cnn(CC3CCC3)c2)=O)C1 c1(C(N(C2CN(C(c3c(C)n[nH]c3)=O)C2)C)=O)ccc2c(n1)CCC(C)C2 N1(C(C(n2cc(-c3c(OC)nsc3)nn2)C)=O)CCCN(C(C)C(=O)O)CC1 Cc1cocc1C(=O)NC1CC(CCNC(=O)CSCc2cccs2)C1 Cc1cccc(CC(=O)NCC(C2CC2)NC(c2conc2C)=O)c1Br Cc1cnc(CNC(C2CC(CSc3ccc(C(C)C)cc3)OC2)=O)cc1C c1(N(C)Cc2cc(Cl)cc(Cl)c2F)nc(N2Cc3cncnc3C2)nc2c1CSC2 c1(NCc2ccc(OC(C)C)cc2Cl)[nH]c(=NC(C)C2CC2)nc2ncn(C)c12 Cc1noc(C)c1C(C)C(=O)NC1CN(C(c2conc2C2CCC2)=O)CC1C Nc1c(C(=O)NCCNC(c2cc(Cl)ncc2O)=O)cc(Cl)cc1Br Cc1ccnc(NC(C2CC(F)CN(C(=O)Cc3cc(Br)cc(Br)c3)C2)=O)c1Br CCC(C(=O)NC1CN(C(c2ccc3snnc3c2)=O)CC1CC)C(F)(F)F Cc1cc(F)cc(Cl)c1Cn1nnnc1N(C)CC1CCS(=O)(=O)N1C C(=O)(C(C)C(=O)OC)NCCN(C(C1CCC(c2ccccc2)CC1)=O)CC c1(NC(C(C)C)=O)cc(Cl)c(C(=O)NC(c2ccc(C(F)(F)F)cc2)C)c(Cl)c1 Cc1ccnc(C)c1CNC(=O)CC1CCCCN1C(=O)CCP(C)(C)=O C(=O)(C(C)(C)C)NCC1CN(C(CN(C)C(c2ccns2)=O)=O)C1 C12(NC(=O)Cc3cnccc3Cl)CCCC1N(C(C1(N3CCCC3=O)CC1)=O)CC2 N1(C(CC=C)=O)CCC2(CC1)CC(NC(=O)C(C)C(O)CCCC)C2 c1(OC)cccc(C(C)C(=O)N(CCCNC(=O)C(C)N2CC(C)C2)C)c1 c1(C(=O)NCC2(OC)CN(C(C3Cc4nncn4C3)=O)C2)cc2sccc2n1C C(=O)(C(F)(F)CN(C)C)N1C(CN(C(C(c2nc(C)sc2)=O)=O)C)CCC1 c1(OC)ccc(CC(=O)NCC2C=CCN2C(=O)CN2CC(C)C2)c(Cl)c1 C1(CC(=O)NCCCNC(c2cncc(Br)c2)=O)Cc2ccccc2NC1=O c1(CC(=O)NC23CCCC2N(C(=O)C(F)C2CCC2)CC3)cccc2c1OCCO2 c1(C(=O)NCC(CC(N2CCCC(O)CC2)=O)OC)cc(F)ccc1F C1(NC(c2ccc(Cl)o2)=O)CN(C(C2CCC2)=O)CCC12CCC2 N1(C2CCCN(C(C3C(=C)C3)=O)C2)CCN(C(=O)COCC(=O)OC)CC1=O C1(NC(c2cncc(C#C)c2)=O)CCN(C(=O)C(C)OC(C)(C)C)C12CCC2 c1(C(N(C(CNC(C)=O)C2CC2)C)=O)ccc([N+](=O)[O-])cc1O c1(CC)cc(C(=O)NCCC2CN(C(=O)CCc3cnn[nH]3)CCO2)cc(O)n1 c1(SCCNc2c(C(=O)OC)cccc2)c(Cl)cc(OC)cc1Cl c1(C(=O)NCC23C(CN(C(c4c(C)nccc4)=O)C2)C3)cccc(C(N)=O)c1C C1(CC(=O)NC2C(CNC(Cc3ccn(C(C)C)n3)=O)C2)COCCOC1 C1(C(=O)NCC2CCN(C(c3cnc(O)n3C(C)C)=O)C2)(OC)CCSCC1 C#CC1(C(=O)NC2CC(O)(CNC(c3nccnc3C)=O)C2)CCOCC1 C12(C(N(CC(C)(O)C3CC3)C)=O)CC(CCO1)N(C(c1sccc1C#N)=O)C2 CC(CNC(=O)C=Cc1cnccn1)CC(=O)N1CCC1C1CCCOC1 C1(C(=O)NCC(C)(Cn2cccn2)NC(C2(CO)CCCC2)=O)CC12CC(O)C2 N1(C(C(CCN(C)C)O)=O)CC(C(N2CC3(CCC(=O)N3)C2)=O)CC12CCC2 C(N=c1[nH]c(=NCC(C(C)(C)C)SC)[nH]c2ccsc12)C1(SCC)CC1 C(=O)(C(C)N(OC)C(=O)C1CCC(NC(=O)C2Cc3ccccc32)CC1)OC C1(CNC(C(C2CCC2)OCC)=O)CCOC1C(=O)NCc1nn[nH]n1 c1(C(=O)NCC(CC=C)NC(c2c(Cl)n[nH]c2CC)=O)cnc(C(F)(F)F)cn1 N1(C(c2cccc(C#C)c2Cl)=O)CCC2CN(C(C3CCCS3(=O)=O)=O)CCC12 c1(OC)ccc(C(C(C)C)NC(C2CC(F)(F)C2)=O)c(F)c1 N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCC12CN(C(=O)CCc1cccc(C)c1)C2 c1(C(N(C2CN(C(c3c(F)ccc(Cl)c3F)=O)C2)C)=O)cc(F)c(Br)cc1F N1(Cc2c(C)noc2C)CCC2CN(C(=O)CNCCCC(C)C)CC12 CCCCC(C(=O)NCC1CCCC(=O)N1)NC(=O)Cc1cc(C)nn1C C12(C(=O)Nc3ncccn3)CCC(NC(=O)Cc3ccc(F)cn3)(CC1)CC2 C1(NC(Cc2c(OC)ccnc2)=O)CCCN(C(c2cc(Cl)cs2)=O)C1C C(=O)(C1CCCc2nncn21)N1CCCC(N(C(=O)C2=COCC2)CCOC)C1 CC1(C(=O)NC2CCCCC2C(N2CC(OC(=N)O)C2)=O)CCC(=O)NC1 c1(CC)ccccc1CC(=O)NCC(C1CC1)NC(c1cnc(C(C)C)n1C)=O C(=O)(C(CC)C(=O)NC1(C)CCCN(C(c2ccn(C(F)(F)F)n2)=O)C1)OCC CCCCC(CC(=O)N1CC(C(=O)N(C)C)C1)NC(=O)CCc1cnccn1 CCC(CC(=O)NCC(C)CN(C(=O)C(C)Cc1ccc(OC)cc1)C)C1CC1 N1(CC)CCC(C2CC2)C1CCC(=O)O.C12(CCCC1)C(=O)NC2=O C(=O)(C1=CCC2(COC2)OC1)N1CC(O)CCC(NC(=O)C=CC2CCCC2)C1 CC1CCC(NC(=O)NCC(C)CN2CCCCC2=O)C(C)C1 C1(NC(C(CC)CO)=O)CCCCC12CCN(C(=O)C=CI)C2 CC(C(=O)OC(C)(C)C)C(=O)NCCC(C)N(C(=O)CCCn1ccnn1)C CC(C(=O)NC(C1CCCC1)CNC(c1ccc(-n2cnnn2)cn1)=O)C(F)F C1(CNC(C(C(C)C)n2ccc(C)c2)=O)CN(C(c2cc(F)n[nH]2)=O)CC12CC2 c1(C(N(C(CN(C(CNC(CC)=O)=O)C)C)C)=O)ccc2c(c1)CCCC2 C1(C(=O)NCCC2CCCN(C(c3ccc(C#C)o3)=O)C2)CCC2(CCC2)OC1 c1(SC)cc(C)ccc1C(=O)NCC1(O)CCN(C(C2C3(CC3)C23CC3)=O)CC1 C1(C(=O)NCC(C2CC(C)(C)C2)O)CCCN(C(C2CC23CCC3)=O)C1 N1(C(C(C)Oc2ccc(Cl)cc2)=O)CCC2(CC2NC(C2CCCO2)=O)C1 Cc1c(C(=O)NCC2CC(C)N(C(=O)CC(C)(C)N(C)C)C2)cccc1Br C1(F)(NC(C(C)OCCOCC)=O)CCN(C(=O)Cc2cnn(C)c2C(F)F)C1 Cc1cc(C(C)C)nc(N2CCN(CCNC(c3c[nH]nc3[N+](=O)[O-])=O)CC2)n1 c1(NC(c2n(C)ncc2CNC(=O)Cc2cc[nH]c2)=O)cnc2[nH]cnc2c1 CCCCC(C)CCC(=O)NC(C)(CSC)C(N1CC2CC(O)CC1C2)=O c1(OC)ccc(C(=O)NC2CCOCC2NC(c2cnc(C(C)C)[nH]2)=O)cc1O c1(C23N(CC4CCCN(CC(=O)OC)C4)CC(C2)C3)cccc(OC)c1Br c1(C(=O)NC(C)CNC(=O)Cc2cnn(C)c2)ccc2nc(O)[nH]c2n1 C1(NC(c2ccc(SC)s2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(F)F CC(C)(C)S(=O)(=O)CCNC(=O)C(=O)Nc1cccc(CNC(=O)OC(C)(C)C)c1 N1(C(C)C(=O)Nc2cc(F)c([N+](=O)[O-])cc2F)CCC(C)C2(CCCCC2)C1 N1(CC)CC(C(=O)NCCC2CCCN2C(C2CC=C(C)CC2)=O)CC1=O c1(-c2cc(C(=O)Nc3scc(CN=[N+]=[N-])n3)n[nH]2)cc(O)c(F)c(F)c1 N1(C(Cc2cccc(OC)c2)=O)CC(NC(=O)C(F)C2CC2)CC12CCC2 C1(C(=O)NC(CC=C)CNC(=O)CN2CC3CC3C2)CC2(CC(=C)C2)C1 CCCC(F)C(=O)N1CCSCC1CCNC(c1ncsc1C(C)C)=O Fc1ccc2ncnc(N3CCCC(n4ccnn4)CC3)c2c1 N1(C(C2C(CC)CN(C(C3CC=CC3)=O)C2)=O)CC2(CCC2)OCC1C CCC(C#N)C(=O)N1CCC(CNC(c2nc(C)oc2C)=O)C1 c1(C(=O)NCc2ncc(OC)nc2)c(C)ccc(C)c1O N1(C(C2C(=C)C2)=O)CCC(CC)(NC(c2cc(C)cnc2F)=O)CC1 CCC(C)C(CN(C)C)NC(=O)C(C)N(C(C1(C)CC(=O)C1)=O)C1CC1 Cc1cc(NC(c2csc(C(=O)Nc3ccc(C(C)C)nc3)n2)=O)ncc1Cl C1(CC(C)(C)C)CCCN(Cc2ccccc2)C1.C12CCN(C1)C(=O)C(=O)N2 N1(C(COCCOCCOC)=O)CC2CCC1C2NC(c1nn(C)cc1N)=O c1(NC(C(=O)NCCC(c2cccc(OC)c2)C)C)ccc(C#N)cc1 N1(C(C(=O)Nc2cc(C)c(Br)cc2)C)CCc2oc(C(C)C)nc2C1 c1(OC)c(C(N2CCC2CNC(=O)C(CC)C(C)C)=O)ncnc1C c1(C(=O)NC(CNC(CSC(C)C)=O)CO)cc(F)c(Br)c(F)c1N c1(C(=O)NC2(C)CCN(C(C34CC(F)(C3)C4)=O)C2)cccc(Br)c1Cl c1(N2CCC(CNC(CCC(C)OC)=O)C(C)C2)cnc(C#N)c(C#N)n1 C1(C(C)C)(C(N2CC(O)(CCNC(c3ccns3)=O)C2)=O)CNC(=O)C1 C1(C(=O)NCC2=NOC(C)C2)CN(C(=O)Cn2c(O)nnc2O)CCC1(C)C C1(NC(C2(CCN(C)C)CCCC2)=O)CCCC(CNC(=O)Cn2ncnn2)C1 CCCC(C)C(=O)NC1CCN(C(c2ccccc2COC)=O)C1C c1(C(=O)NC2CCC(NC(=O)CCc3cncs3)CC2)cc2ccncc2o1 N(C1c2ccccc2OCC1O)C(=O)NCCC(CC)CO c1(-n2c(-c3n[nH]c(C4CC4)c3Br)nc(CCC)n2)ccnc2c(CC)cccc12 C1(C(=O)OC)COCCN1NC(=O)CCC(O)C1CC1 N1(C(C2N(C(c3nc(OCC)oc3)=O)CC(OC)C2)=O)CCCC(C)(C)C1C C1(O)(C(C(=O)NC(c2ccccc2)CCC)NC)CCCCC1 C1(C(=O)NCC(C)CC(C)O)(CONC(c2ccc(CC)o2)=O)CCCCC1 COn1cnc(C)c1C(=O)N(CCCCNC(=O)Cc1ccoc1)C C12(C(=O)NC(C(=O)OCC)CC)CC1CN(C(C1CC13CCCC3)=O)C2 C1(NC(C2(C)CC2c2ccccc2)=O)CN(C(=O)CCC(=O)c2ccc[nH]2)CC1O c1(C(=O)NC(CNC(=O)COc2cccnc2)CO)cn(C(F)F)nc1C(F)F Cc1c(C)c(C)c(C(=O)NCC(C)(O)CN2CCOCC2)c(C)c1C C(C)(CCC(=O)NCC(CC(C)C)NC(=O)C(O)Cc1ccccc1)OCC C1(CCCNC(c2ccccc2)=O)CCCN1C(c1csc(CO)n1)=O C(=O)(C1=NN(C)C(=O)CC1)N(C(C)C)CCN(C)C(C1COCC1(C)C)=O CC(CC(=O)N1C2CCC1CN(C(c1cnn(C)c1Cl)=O)C2)CC(F)(F)F C1(C(N(CCCNC(CCC=C=C)=O)CCO)=O)CCC2CCCCN12 C1(NC(c2c(C(C)NC(=O)CN3CCNC(=O)C3)noc2)=O)CCC12CCCC2 C#CCC(O)C(=O)N(CC(C)C(=O)NC(CC)CCO)C c1(C(=O)NCCCCNC(C=C(CCC)C)=O)c[nH]nc1-c1ccsc1 c1(SCCC(=O)N(C2CCC(NC(=O)Cc3nccn3C)C2)C)ccccn1 C(CC(=O)NC1CC(F)CN(C(c2cccc(F)c2F)=O)C1)(C(F)(F)F)OC C1(CC)(NC(=O)CC(C)(C)O)CCN(C(=O)COC2CCOC2)CC1 CC(C)CC(CC(=O)NC1CCCC1O)NC(=O)CC(O)C(C)C CC(O)C(C)C(=O)NCCCC(C)(C)NC(=O)CCNC(c1ccccc1)=O N1(Cc2ccc(C#C)s2)CCC2(CC1)CC2C(=O)Nc1cccc(I)c1 C12(C)CCC(CC1)N2C(=O)O.C1(c2cn(COC)nn2)(NC(C)(C)C)CCCCC1 c1(C(C)C(=O)NC2CC(NC(=O)C(F)(F)c3cncs3)C2)ccc(F)cc1F C1(NC(C2(CC)CC2)=O)CN(C(C2CC2c2cccc(Cl)c2F)=O)CC1C1CC1 C(=O)(C(F)(F)C(C(C)C)NC(C1CCCCC1CC(F)(F)F)=O)OC C=CC(CC)CC(=O)N1CC(CNC(=O)CC(=O)NCC(F)(F)F)C(C)C1 N1(C(c2c(C)csc2)=O)CCC(C(=O)NCCc2cnnn2C)C(C)(C)C1 N1(Cc2ncc(CC)o2)CCC2CCC(C1)N2C(c1cc2ncccc2s1)=O C1(C(N(CC(N2CCC(C#C)C2)=O)CCOC)=O)CCCCCN1C CC1(C(=O)NCCCOCCCNC(C23CCCC2C3)=O)COC(=O)C1 C1(NC(c2c(CC)n(C)cc2)=O)CCN(C(C2CC(C(C)C)=NO2)=O)C1(C)C C(=O)(CC(C(F)(F)F)NC(c1c[nH]c(=NC)o1)=O)N(CC(C)OC)CC CC1(NC(c2cc(C(N)=O)co2)=O)CCN(C(c2cnc(C(C)(F)F)s2)=O)CC1 c1(COCC)c(N2CCN(C(C3CCC(F)(COC)C3)=O)CC2)nc(=N)[nH]c1C c1(C(=O)NCC2CCCCN(C(C(C)SC)=O)C2)c(C)cccc1[N+](=O)[O-] C1(NC(CCC(C)SC)=O)CCOC12CCN(C(c1cc(C(N)=O)[nH]n1)=O)CC2 CCC(O)C(C)C(=O)NC1(CCNC(c2c(C)coc2C2CC2)=O)CCCC1 C1(CC2(O)CCN(CC(=O)NCC3CCC(C)CC3)CC2)Cc2ccccc2O1 N1(C(C2(COC)CC2)=O)CC(NC(c2cnn(C(C)C)c2N)=O)C(SC)C1 c1(CNC(C)(CCC#N)c2n(CCCSC)nnn2)ccc(F)cc1Br c1(NC)cc(C(N2CCCC2CNC(=O)C(C)(C)CNC(C)=O)=O)ccc1OC C1(CC)CN(C(C2(C(F)(F)F)CC2)=O)CCC1CNC(=O)Cc1ncc[nH]c1=O c1(C(C(=O)NC2(CN(C(C3C(OCC)CCC3)=O)C)CC2)C)c(F)cccc1F N1(C(C(CCSC)OC)=O)CCCC(CC(=O)NCc2ccc(F)c(C)c2)CC1 c1(C(N2CCCC(C(N3CCCC(CC)C3)=O)C2)=O)cc(C)c(O)nn1 c1(C(N(C)CC2OCCN(C(CC(C)O)=O)C2)=O)ccc(F)cc1C1CC1 C(CCCCCC(=O)NC1CC12CCN(C(c1cc(C)ns1)=O)C2)SC n1(CC(N2CCC(C(=O)OC)(CO)C2)=O)c2ccccc2c(=O)c2ccccc12 N1(C(=O)OC(C)(C)C)CC(C(=O)NCC(C)(C)CO)C(C2CC2)C1 N1(C(c2nc(OCC)sn2)=O)CCN(C(c2cc3occc3s2)=O)CC1C C1(C(=O)NC2CCN(c3n(C)nnn3)C2)CCN(C(N2CCOCC2)=O)CC1 Cc1nc2cccc(C(=O)NC3CN(C(C4CCCSC4C)=O)C3)c2[nH]1 C(CCCCS(=O)(=O)CC)N1C(CNC(CCCC(=C)C)=O)CN(C)CC1 C1(NC(c2c(OC)scc2)=O)(CNC(C2(C#N)CC3(CC3)C2)=O)CCCCC1C c1(CCCC(=O)NCCCN(C(=O)CCCNC(C)=O)CC)ccc(C#N)cc1 c1(NC(C2(F)CN(C(C3CC3(F)Cl)=O)C2)=O)ccc2nn[nH]c2c1 C1(CCNC(CCC2(C)CC2)=O)CN(C(C2(O)CC(F)(F)C2)=O)CCO1 C1(C)(CC)CC(NC(C2(CCCC)CCCC2)=O)CN1C(c1ccc(C)o1)=O c1(CNC(C(N2CCCC(CC=CC)C2)=O)=O)cnc(O)c2ccccc12 C1(CCNC(CCC=C)=O)CN(C(=O)CCCn2cncn2)CCS1(=O)=O c1(C(=O)OC)ccc(C(O)C(n2cc(-c3noc(CC(C)C)n3)nn2)C)cc1 c1(C(CNC(=O)C(F)=CCCF)NC(c2ccc(CO)s2)=O)ccccc1 C1(CC)(NC(c2cc[nH]c(=N)c2)=O)CCN(C(=O)Cc2nnc(C)s2)CC1 n1(CC(=O)N2C(CC)C2)nc(C)c(Cl)c1C.C1(C)(OCC(=O)OCC)CCOCC1 C1(NC(Cc2c(C)ccnc2)=O)CC1C1CCN(C(C2CCCC23CC3)=O)CC1 CCC(C)C(=O)C(=O)NC(CCC1CCC1)C(=O)NC(c1nc(C)cs1)C N1(C(c2n(C)cc(Cl)c2)=O)CCCN(C(=O)C(C#N)CC2CC2)CC1 N1(CC(N2CC(C(C(=O)NC34CCC(CC3)C4)OC)C2)=O)C(C)CCC1C c1(SC)ccc(C(N2CCC(C)C2CNC(=O)CCc2ccccc2Cl)=O)cn1 C(CCCCC(=O)NCc1ccc(CNC(c2cc(C#N)c[nH]2)=O)cc1)OC c1(-c2cc(CNC(N(CC(C)C#N)C)=O)no2)cccc(F)c1 C1(C(N2C(C)(CNC(c3ccc(CCC)s3)=O)CCC2)=O)CCCCC12CCC2 c1(OCC)cccnc1CC(N1CC(CNC(C2CCCC2(C)C)=O)C1)=O C(=O)(CC1OCc2ccccc21)N1CC=C(CNC(Cc2c(C)ocn2)=O)CC1 C1(C(C)NC(c2n(CC)ncc2)=O)CN(C(=O)CCn2c(C)ccc2C)CCO1 C(=O)(C(C)CC(=O)N1C(CNC(c2ccc(F)cc2F)=O)CC2CC12)OC c1(C(=O)NC(CC)CNC(=O)C(C)c2ncco2)cc(C)ccc1Br C1(CNC(C(C(C)C)NC(N)=O)=O)CN(C(C2C3(CC3)C23CC3)=O)C(C)(C)C1 C1(O)(CNC(=O)C(C2CCCCC2)F)CCN(C(C2CCC(C(F)(F)F)C2)=O)C1 Cc1cc(C(=O)N(C)CC2(CNC(c3nc(C4CC4)cs3)=O)CC2)n(C(F)F)n1 C#CC1(C(=O)NCc2cc(C(=O)NCC(C)(O)C(F)F)n(C)n2)CC(=O)C1 C1(CC=C)(NC(c2cc3n(n2)CCO3)=O)CCCN(C(=O)CN(C2CCC2)C)C1 CC(C)C(O)CC(=O)NC1CN(C(=O)CN2CCCCCC2)CC1C N1(C(CCC(C)OCC)=O)CCC(C)CC1C(=O)NCC=Cc1ccccc1 CCC(CC)C(C(=O)N1CCCC1CNC(=O)C(=Cc1ccccc1Cl)C)OC c1(C(=O)NC2(CO)CN(C(C3CC3c3ccc(Cl)s3)=O)C2)ccc(F)cc1Cl C1(CNC(C(C)(C)C2CCCCO2)=O)NCCC1C1CC1 C1(CC(=O)N(CC(C)NC(C(C)C(C)(C)C)=O)C)CCCCCC1(F)F c1(OC)cccc(CCC(=O)NCC=CCNC(=O)CCOCC(C)C)c1F c1(COCCCOCC)ccc(NC(=O)C(F)(F)CN(C)C)cc1Cl c1(C(=O)NC(CCCNC(C2CC(=O)NC2)=O)CO)cnc2ccncc2c1 C1(C(=O)NCCN(C(=O)CN(c2ccncc2)C)CC)CC2CCCC2C1 c1(C(N2CCN(C)CC2)C(N2CCC(O)(C(=O)OC)C2)=O)cccc([N+](=O)[O-])c1 CC1CCCC(C(=O)Nc2n[nH]cc2CN)C1 c1(CC(=O)N(CC(C)(C)CNC(=O)C(C)=C2CC2)CC)cccc(C#N)c1OC C(=O)(CC(CC)N(C)C(c1cncc(CO)c1)=O)N(CCCO)CC#C C=CCC(CC(C)C)C(=O)NC1(C(=O)NC(CC)C(C)(F)F)CC1 C(C(CC)N=c1nc(COC)[nH]s1)NC(CC(CCC)CC)=O c1(-c2ccc(C(=O)OCC)s2)c(Cl)ccc(NC(=O)CCCCCSC)c1F C(=O)(C(C(C)CCC(=O)OC)N1CC(C)C(N=[N+]=[N-])C1)NCCCCCC C(c1ccccc1C#N)=CC(N1CCCN(C(C2(C)CCCOC2)=O)CC1)=O C(=O)(C1CCCc2cncn21)NC1CN(C(C(F)=CCC)=O)C2C1CCC2 c1(OC(COC)OC)cc(CC(=O)O)cc(F)c1 C12(CNC(c3occ(C(=O)O)c3)=O)CCCC1N(C(=O)CC13CCCC1C3)CC2 N1(C(c2c(C)nsc2)=O)CCCCC1C1(CNC(C2(CF)CC2)=O)CCOCC1 C1(CC)(NC(=O)C(C)COC)CCCN(C(=O)CN2CCC(=O)NC2=O)C1 c1(OC)cncnc1C(=O)NCC(CC1CC1)C(=O)N1CC2(CC2)C1 N1(C(C2N(C(CC3C(C)OCC3)=O)CCOCC2)=O)CCCC(N=[N+]=[N-])C1 c1(OC)ccc2cc(C(=O)NCCN(C)C(C)=O)ccc2n1 C1(OC)CCN(C(C2CSCN2C(c2ncc[nH]2)=O)=O)CC1(C)C c1(C(=O)NCC2N(C(C(CSC)(C)C)=O)CCCC2)cc(C)cnc1C C#CCCN=C(NCc1ccc(CN2CCCC2)cc1)NC(c1ccccn1)C Cn1ncc2ncc(C(N3CCC(NC(c4nccs4)=O)C(C)(C)C3)=O)cc12 N1(C(c2occ3c2CCC3)=O)CCC2(NC(=O)COC3CCC3)CCCCCC12 N1(C(c2c(OC)cccc2F)C(=O)NCCC2CC2)CCCOCC1(C)C C(=O)(C=C1SCC(=O)N1C)NC1CCN(C2CCN(C(C(C=C)O)=O)C2)CC1 Cc1cccc(C)c1NC(=O)C(c1ccoc1)NC(=O)CN(C)C(N)=O N1(C(CC(C)(C)NC(N)=O)=O)CCC2(CCCN2C(=O)COC2CCOCC2)C1 c1(C(N(C2CC(NC(=O)CCc3csc(Br)c3)C2)C)=O)cnccn1 N1(C(C=C(CC)CC)=O)CC2CCCC(CNC(=O)COC)C2C1 N1(C(C(C)n2ccnc2)=O)CC(NC(=O)COCCCF)C(F)C1 N1(C(CC(=O)OC)=O)CCc2ccc(C(=O)NC3CC3)cc2CC1 C1(CN(C(=O)CSC(C)(C)C)C)CN(C(=O)C2=NOCC2)CCO1 Fc1c(CNC(=NCCC2CC(F)C2)NCC2CC2)ccnc1Br Cc1cnc2n1CC(C(=O)NCC(C1CCC1)NC(=O)C(F)(F)C(F)(F)F)CC2 CC1(C)CC(NC(c2ccon2)=O)CN1C(c1c[nH]c(C2CC2)n1)=O c1(CCC(=O)NC2(CF)CCN(c3ccnc(C4CC4)n3)C2)nnc(O)nc1O Cc1nc(C2CC2)ccc1C(=O)NC1CC(NC(c2ocnc2C(F)(F)F)=O)C1 Cc1cc(C(=O)NC2CC(F)CN(C(C3CC3C)=O)C2)n2ncnc2n1 c1(C(N2CC(N(C(c3c(C)nncc3)=O)C)C(C)(C)C2)=O)cnc2ccnn2c1 Cc1cc(C)n2nc(C(N3CCCC3C3(O)CN(C(=O)CN(C)C)C3)=O)cc2n1 c1(C(N(CC(C)(C)NC(C)=O)C2CC2)=O)cc(C2CC2C)on1 C(=O)(C1=C(Cl)CCCC1)N1CCN(C)CC1C(=O)NC1COCC1C(N)=O n1(CCC)ncnc1CN(C1CCN(C)C1)CCOCCNC C#Cc1cc(C(N2CCC(NC(=O)C(=O)Nc3ccc(C)cc3)C2)=O)cc(F)c1 c1(NC)ncc(C(=O)NCCCC(C)NC(c2ccncn2)=O)cc1Cl c1(C(C(=O)NCCC(Cl)Cl)NC=O)cccc(C(F)(F)F)c1.CC(C)C=O N1(C(C2(CC(=O)OC)CC2)=O)CCOC(C)C1C(N1CC(F)(F)CC1C)=O C1(C(=O)NC(c2csnn2)C)CCC2CCC1N2C(c1ccncc1)=O C(C(=O)NCC(C1CC1)NC(=O)COc1ccccc1C#N)(C(C)(C)C)SCC C1(NC(c2c(C)nc(CNC(C3CCN(C)C3C)=O)o2)=O)CCC2CC2CC1 C1(N(C(c2cnc(Cl)[nH]2)=O)CC)CCCN(C(=O)Cc2c(Cl)cnn2C)C1 c1(C(=O)NC2(CCOC)CCN(C(=O)C(C)CO)C2)cncc2ncn(C)c12 n1(C2CC(C(N(CCN(CC=C)C)C(C)C)=O)C2)cc(Cc2cccs2)nn1 CS(C)(=O)=NCCNC(=O)N(C(c1ccccc1)C(F)F)CCO N1(c2ccnc(OC)n2)CC2CCC(NC(=O)CO)CC2C1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(n2cc(-c3cccc(C)c3)nn2)CC1 CN(OCC(F)(F)F)C(=O)C(c1ccoc1)NC(=O)CC(C)(C)CN(C)C C1(NC(C2C(CC)C2)=O)CN(C(c2ccc3ncnn3c2)=O)CC(C)(C)C1 Cc1nn(C)c(C)c1C(=O)C(=O)NCC(CO)NC(=O)C(O)CC1CCCCC1 c1(C(CNC(C2(C)CCN(C)C2)=O)NC(C2(C)CC2)=O)cc(F)cc(Cl)c1.C1CC1 Cc1cc(O)c(C(=O)NC2CCCC(CNC(=O)Cc3cnc[nH]3)C2)nn1 C1(CNC(CC=CC=C)=O)CCCN(C(C2CCCCS2(=O)=O)=O)CC1 Cc1ccc2nsnc2c1C(=O)NCCCCN(C(=O)CCCC(C)C)C CN1CCCCC1NC(c1cccc(C(=O)NC2CN(C(N)=O)CC2CO)c1)=O C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCC(C)NC(c1cccc(C(=O)NC)c1)=O CC(C)C#CC(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cccnc1)C c1(C(=O)NCC(C)NC(C2CC=CCC2)=O)cc(C(N)=O)[nH]n1 N1(Cc2c(C)c(Br)cnc2)CC2OCCN(Cc3cccc(OCCO)c3)C2C1 C#CC1(C(=O)NCC(O)CCNC(=O)C(F)OC(F)(F)F)CCCCC1 C1(CNC(C(C)CO)=O)CN(C(c2cccc(Br)c2Cl)=O)CC12CC2 C(=O)(CC1=CCN(C(=O)C(C)(C)OCC2CCCC2)CC1)N(CCCSC)C N1(C(CN(C(=O)OC)C)=O)CCC(C(N2CCCC2c2ccon2)=O)C1 C1(NC(c2c(OC)n(C)nc2)=O)CC2CCC1C(NC(=O)C1=COCCO1)C2 N1(C(CCN(C)Cc2ccc(Cl)nc2)=O)CC2CCC(C1)C2NC(=O)CCC(N)=O N1(C(C(C(C)C)(C)O)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC12CCC2 C1(CC(N2CC(c3onc(C)n3)C2)=O)CC2(CC2)CN1C(=O)C=Cc1cncn1C CC1COC2(CCC2)CN1C(=O)C(Cc1ccoc1)NC(=O)C(N)=O CCC(C)(CC(=O)N(CC(C)CNC(=O)Cc1cncnc1)C)C(=O)OC Cc1cc(=NC(=O)C(=O)N2CC(O)(C(C)NC(=O)CC(C)C3CCCC3)C2)[nH]o1 c1(C(C2C(C(=O)N(C(C3CCOC3)CO)CCO)C2)=O)ccc(Br)cc1 CC(C)(CCC(=O)NCC1(O)CCN(C(c2ccc(Cl)nc2N)=O)C1)[N+](=O)[O-] C(=O)(C1CCCc2sc(C)nc21)NC1C2C(NC(C(F)=CC)=O)CC(CC2)C1 c1(OC)ccc(-c2cccc(OC)c2F)c(CC2N(SC)CCC(CO)C2)c1 c1(C(N2C3(CN(C(CC(=O)NCC)=O)C3)CC2)=O)ccc(S(C)=O)cc1 CCCC(C(=O)NC1CCCC(CNC(=O)CCC2CC2)C1)S(N)(=O)=O c1(C(=O)OC(c2ccc(Cl)cc2)C#C)coc2ccc(Cl)cc12 C(CC(C)(C)C)(C(=O)NCCC1CC1C)NC(C(CC)CCOC)=O Cc1nc2cncc(C(N3CC=CC3CNC(=O)COCC3CCCC3)=O)c2[nH]1 c1(C(=O)NC2C(NC(C(C)(C)OC)=O)CC2)ccn2ccnc2c1 CC1CN(C(=O)C(C(C)O)NC(c2ccsc2C#N)=O)CC1F N1(C(=O)N(C(=O)C2CC2)CCC2CCC2)CCCCC1CN1CCOCC1 C1(C)(CNC(Cn2ncc(CC)c2)=O)CN(C(c2c[nH]c(=O)cn2)=O)CCO1 C(c1ccc(Cl)nc1)=CC(=O)NCCNC(c1ccn(-c2ccncc2)n1)=O c1(NC(CNC(CC2CCCC(C)(C)O2)=O)=O)ccc2c(c1)OCO2 C12C(C(=O)O)C3CC1C2C3.N1(C(CN2CC(=O)NC2=O)=O)CCC(C=CC(=O)O)CC1 C1(NC(c2ncc(CC)s2)=O)(COC)CCN(C(c2cnc(C(C)C)[nH]2)=O)CC1 C=C(Cl)CC(C(=O)N(CC1=CCSC1)C)NC(c1ccn(C)n1)=O S(=O)(=O)(c1cccnc1)NCCC(=O)NC(c1ccc(F)cc1F)(C(=O)OC)C C(=O)(C1=CC2(CCN(C(c3c(F)cccc3F)=O)C2)C1)N(CC(C)C)C N1(C(Cc2nc(C(C)C)sc2)=O)CCC(CC#N)C(F)(F)CC1 c1(C(=O)NC)[nH]c(=NCc2ccccc2C2CCC2)nc2scnc12 C1(CCOC)(NC(=O)Cn2ncccc2=O)CCN(C(c2ccnn2C)=O)CC1 CC1(C2CN(C(=O)NCC3CCCN(C(=O)NC(C)(C)C)CC3)C2)CC1 Cc1ccc2c(c1)CC(C(=O)NC1CCC(CNC(=O)C3=COCC3)C1)S2(=O)=O C1(CNC(C(CC)OCC)=O)C(C2CC2)CCN1C(=O)CC1(COC)CC1 C=C(C)CC(C(=O)NCC(O)(C)CC)NC(c1cc(C2CC2)[nH]n1)=O C(C(C)(C(=O)OC(C(=O)NC(C)(C)C)C(=O)O)Nc1ccc(I)cn1)OC c1(C(N(C)CC2CCN(C(=O)CNC=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 Cc1cc(C(=O)NCC2CCCN(C(c3cc(C#N)on3)=O)C2)nc(Cl)c1 N1(C(C(C)(C)c2cscn2)=O)CCC(F)(F)C(CNC(C2CC23CCC3)=O)C1 CC1CC=C(C(=O)N2CCC(CC(=O)NCC3OC(=O)CC3(C)C)C(O)C2)CC1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(=O)COCCCN=[N+]=[N-])CC(C)C1 C(=O)(C(C(C)CC(C)(C)C)N(CCC(c1ccccc1)O)CC)NCCSCC c1(OC)cc2c(c(OC)c1OC)CN(C(CC(C)CO)C(=O)OC)CC2 c1(C(N2CCC(CNC(C34CCC(C3)C4)=O)C23CC3)=O)cc2ncccc2o1 Cc1ccc2c(C(N3CC(N(C)C(C4(O)CCOC4)=O)C3)=O)csc2c1 c1(C(N2CC(NC(C(=C)Cc3ccccc3)=O)(CO)C2)=O)c[nH]c(C)c1Cl C1(C(C)NC(c2cscc2Br)=O)CC(F)CN1C(C12CCC(C1)C2)=O c1(C(N2CCC(F)(CNC(C=CCC)=O)C2)=O)c(OC)ncc(Cl)c1C CN1CCN(C)C2(CCCN(C(C(=O)NC3CC3)C3=CCCCCC3)C2)C1 C1(C)(C(=O)NCC(CNC(C2(CC)CC2)=O)(C)O)CCCC12CC2 c1(C(=O)NCC(CNC(CCSCCC)=O)C)coc2cc(OC)ccc12 N1(S(C)(=O)=O)CCN(C(c2cc(Cl)cs2)C(=O)NC2CC2)CC1.c12noc(n1)C2 C1(CC(=O)NCC2C(C(N(CC(C(=O)NC)C)C)=O)C2)CC(C)(C)CO1 N1(C(C(c2ccccc2)C)=O)CC(F)CC1CN(C(=O)C=CSc1nc[nH]n1)C c1(C(N2C(CN(C(=O)CCC(C)(C)O)C)CCCC2)=O)cc(F)cc(Cl)c1N CC1CC2(CCN(C(=O)CC3(O)CCOC3)CC2)CN1C(=O)CCc1nc[nH]n1 c1(CNC(C2C(NC(c3cc(C)sn3)=O)CCO2)=O)ccc(CN(C)C)cc1 c1(CNC(C(c2ccn(C)c2)C)=O)ccc(C(=O)N(CCCC(O)CO)C)nc1 c1(NC(CC2N(C(C=NOC)=O)CCC2)=O)cn(CC)nc1C#N c1(C(=O)NC(C2CCN(C(C3(O)CCSC3)=O)CC2)C)cc(O)nc(C2CC2)n1 C(=O)(CCC(=O)NCC1CCCCN1C(=O)C=Cc1cnc(C)s1)OCC c1(C(N(C2CCCCCC2)C(C)C)=O)cnc(O)c([N+](=O)[O-])c1 N1(C(CCCSC)=O)CCC2CCN(C(C3CC34CCC4)=O)C2C1 c1(C(N2CCN(C(C3CCN(CC#C)CC3)=O)C(C)C2)=O)ccc(Cl)c(C)c1O C(=O)(CCCCCN(C)C)N(CCN(C(C(CC#C)O)=O)C)C c1(C(N2CC(NC(c3cc(CC)cc(Cl)c3)=O)C2)=O)c(C)ccc2nsnc12 Cc1cnc2c(C(=O)NC(C)CC3CN(C(C4CCC(C)(C)C4)=O)C3)cccn12 c1(C(=O)NC2CC(NC(c3c(Cl)cn(C)n3)=O)C2)nc2cnccc2s1 C1(CC)CN(C(=O)CN(CC(=O)NC(C)C)C)CCN1C(=O)C1=CC(C)CC1 N1(C(=O)CC2CCCOCC2)CCN(C(c2cnc3n2CCS3)=O)C(CF)C1 C1(CCC)(NC(=O)C(C)CC(C)C)CCCN(C(=O)C=Cc2ccc(SC)s2)C1 c1(C(=O)OC)sc(C(N2CCS(=O)(=O)CC2)=O)c2c1CCCC2 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC2C(CCN2C(C2CCC2)=O)C1 C1(Nc2ccccc2)CC(OC)C1(CCC)COC(CC)CCOC c1(CNC(C23CC(NC(=O)CCc4ccoc4)(C2)C3)=O)c(F)cncc1F N1(C(C(C(C)C)OCC)=O)CCC2CN(C(=O)C(C)(C)COC)CC12 C1(CCC(=O)N(C2COCC2O)C)CCN(C(=O)CCC2(C#N)CCC2)C1 c1(CNC(C(C)O)=O)ccc2c(c1)CCCC2NC(c1ccc(N=[N+]=[N-])cc1)=O n1(CC)c(C)c(C(=O)NC2CN(C(=O)C(C)C)C3CC23)c2cc(OC)ccc12 C1(NC(c2n(CC)c(O)nc2)=O)CCC12CN(C(c1cccc(F)c1SC)=O)C2 Nc1cc(F)c(Cl)cc1C(=O)NC1CCC(CCNC(=O)CC(=O)NC2CC2)C1 N1(C(C2OCCN(C(c3ccc(C)c(C)n3)=O)CC2)=O)CCCC(C)(C)C1C CCC(CC(C)O)C1CC1NC(=O)C(=O)Nc1ccccc1CC(=O)N(C)C C1(C(=O)NC2C3(CC(NC(C4CN(C(C)C)C4)=O)C3)C2)CC(=O)NC(=O)N1 CCC(CC(=O)N1CCN(C(C2CC(CCO)C2)=O)CC1C(C)C)C(F)F CCCC(CNC(=O)C(C)c1ccco1)NC(c1cnc(C)[nH]1)=O c1(C(N(c2c(F)cccc2F)C)=O)ccc2c(S(N)(=O)=O)cccc2c1 C1(C)(CC(=O)NC(CCNC(c2ccn(CCC)n2)=O)(C)C)CCCCC1 c1(CC(=O)NCC(C)N(C)C(c2cccn2C)=O)ccnn1-c1ccccc1 N1(C(C(C)NC(CC)=O)=O)CCC(N(CC(C)C)C(C2(F)CC=CC2)=O)CC1 C1(Cc2nc(COC)on2)CC(O)CN1C(=O)NCc1ccc(N(C)C)cc1 C1(C(=O)NCCC2CCCC2O)CCCCN1C(c1c[nH]nc1Cl)=O C1(N(C)C(c2c(C)occ2)=O)CCN(C(=O)C2(n3cccn3)CC2)O1 C1(C(C)NC(c2c(CC)scc2)=O)CCN(C(=O)CCOC)CC1 C(=O)(C(CC(C)C)n1ccnc1)OC(C(=O)NCCc1ccc(OC)c(Br)c1)C C(=O)(CC(O)CC(C)(C)C)N1CCC(CN(C(c2cc(C)n(C(C)C)n2)=O)C)C1 c1(C(N2CC(CCNC(c3ccc(CC)s3)=O)C(C)C2)=O)ccc(OC)cc1C C1(C(N(CCOC)CCF)=O)CN(C(c2cnsc2)=O)CC1F C1(NC(C(C)(C)c2cc[nH]n2)=O)CCCC2CN(C(=O)Cc3ccsc3Cl)CC12 C1(C(=O)NCCCN(C(c2c(OC)nsc2)=O)C)CCC(=O)N(C2CC2)C1 O=C1CC(C(=O)NCc2ccccc2CNC(C2(Cl)CC2)=O)CN1O Cc1cc(Cl)cc(C(=O)NC2(CNC(=O)CN(C)C(C3CCOC3)=O)CC2)c1O c1(CC(=O)NC(CC2CN(C(C(C)NS(CCC)(=O)=O)=O)C2)C)cccc(C)c1 c1(C(N2CC(C(=O)NC(COCC)C)C(C(F)(F)F)C2)=O)ccccc1OC C(=O)(C(CNC(C1CC1C(C)C)=O)N(C)C)NC(c1nc[nH]n1)CC C12(C(N(CCCNC(C3CCCN3c3ncccn3)=O)C)=O)CCCN(CC1)C2 N1(C(CCC2CC(C)C2)=O)CCC2CCN(C(=O)C=CCF)CC12 c1(C(N2CC(CC=C)(NC(c3csc(C)n3)=O)C2)=O)csc2ccccc12 Cc1cc(C(=O)Nc2cc(C(F)(F)F)cc(Br)c2O)c2c(C3CC3)noc2n1 C(=O)(C1=CCCC(C)(C)C1)NC1C(CC)CN(C(=O)CCc2nc[nH]n2)CC1 C1(NC(CC2OCC(C)(C)C2)=O)CCN(c2nnc(CO)s2)C12CCC2 N1(C(c2ncn(CC)c2)=O)CCC(CNC(C2CCCN2C)=O)C(O)C1 C1(C#N)(CNC(CN(C(C(C)n2cncn2)=O)CCO)=O)CCCC1 C1(NC(CCc2ccc(C)s2)=O)CCOC1(C)C C1(NC(CNC(C(CC)C)=O)=O)C2CC1CN(C(c1cc(C)nc(C)n1)=O)C2 C(=O)(CC1=CCN(C)CC1)NCC(C(=O)NC(CC)(C)CN(C)C)C Cc1n[nH]c(C)c1SCC(=O)NC(C12CCC(CC1)C2)CNCc1ncccn1 N1(C(C(N(C)C)C2CC2)=O)CC(CNC(c2c(N)cccc2Cl)=O)C(C)(C)C1 C1(C(=O)NC(C2N(C(Cc3c(C)n[nH]c3C)=O)CCC2)C)CCC=CCCC1 C1(C(=O)NC(C(=O)NCCCC(F)F)Cc2cc[nH]n2)CC2C=CC1O2 CCCC(C)CC(=O)NC(Cc1ccco1)C(=O)NCc1csnn1 CC1CC(NC(c2csc3nccn23)=O)CCN1C(c1ccncc1)=O CC(C)(C(=O)NCCOC1CCN(C(c2coc(CO)c2)=O)C1)N1CCCC1 c1(C(=O)NCCN(C(C2CCCC2COC)=O)CC)cncn1C c1(OC)cccc(Cl)c1NC(C1CCCC1NC(c1ccc(C)c(F)c1)=O)=O c1(CNC(N2CCC(CO)C(c3ccccc3)C2)=O)noc2c1CCCCC2 C1(CC(=O)NC(C2CN(C(=O)Cn3ncc(O)nc3=O)C2)C)CCOC(C)(C)C1 c1(C(=O)Nc2nccc(CC)c2)cc(C)nc2ccnn12 c1(C(N2C(C(CNC(C=CC(C)C)=O)(C)C)CCC2)=O)cc(F)c(F)cc1O C1(CC)C(C(=O)N(C)CC2CC3CCCC23)CCN1Cc1ccccc1 N1(C(c2c(C)[nH]cc2)C(=O)NCSc2ccccc2)CC2CC1CN2C C1(CN(C(=O)C(C)Sc2nncn2C)CC)CCCCN1C(C1(CC)CCC1)=O C1(C)(C(N(CCCCNC(C2CC(C(F)F)C2)=O)C)=O)COc2ccccc2O1 C1(NC(C2C(c3n(C)ncc3)C2)=O)COCCN(C(C2CC3CCC3C2)=O)C1 c1(C(N2C(CCNC(C(C)C(C)(C)C)=O)COCC2)=O)ncn2c1CCCC2 C(CNC(=O)C(C)(C)C1CCN(C(c2cnn(CCO)c2)=O)C1)(C(C)(C)C)OC C(=O)(CCCCCC#N)NC(C(C)O)C(=O)NCc1ccc(Cl)cn1 CCCC(C(=O)NC(C(=O)NCCSCC)C(C)OCC)N(C)C CCCCC(CC(=O)N1CCOCC(CO)C1)NC(=O)CN1CC2CC2C1 N1(C(CCCC(C)O)=O)CC2CCCC(NC(=O)CCc3ccn(C)n3)C2C1 CCC(N=c1ccnc(NCC(CC)(CC)SC)[nH]1)c1cccnc1 c1(OC)ncc(C(N2CCC(NC(=O)CSCC3CC3)C(C)C2)=O)cc1Cl C1(C(=O)NCCC(C)c2cn[nH]c2)(OC(C)C)CCC1.C1C(=O)N1.C1C(=O)N1 N1(C(C(C=C)O)=O)C(CNC(=O)Cc2ccc(OC)c(F)c2)CC2CCCCC12 N1(C(CSc2n(C(C)C)cnn2)=O)CC(NC(=O)Cc2ccn(C)n2)CC1C N1(C(C=C)=O)CCN(c2ncc(C(F)F)cn2)CC12CCC2 C1(C(C)C)C(C(=O)N(C)Cc2cccnc2)CCN1C(=O)C(O)C1CCC1 C1(NC(C2(C)CC2(Cl)Cl)=O)CC(NCc2cnsn2)C12CCC2 N1(C(C(C(C)C)NC(=O)OC(C)(C)C)C)CC2CN(CC(F)(F)F)CC2C1 CC(O)C(C)(C)C(=O)N1CCC(N(C)C(C2CCC(C)CC2)=O)CC1 c1(C(N2CC(NC(C(CC=C)NC(C)=O)=O)C(C)C2)=O)cc(N)ccc1SC c1(OC)c(C(=O)NCCN(C(C2CCOCC2C)=O)C2CC2)cc(F)cc1F c1(C(N(CCCNC(Cc2nc(C)oc2)=O)C2CC2)=O)snc(O)c1Cl Cc1cc(F)cnc1C(=O)NC(c1cn(CC2(CC(=O)O)CC2)nn1)C c1(OC)ccc(C)cc1-n1cc(CNC(=O)C(C)SC)nn1 C(C(=O)N1CCC(=CNC(=O)COc2nc(O)nc(O)n2)CC1)(C(C)C)NC(C)=O C(=O)(C1CCC(=O)c2cccn21)N1CCCC(NC(c2cncc(C)c2C)=O)C1 C1(SCC)CCC(C(N2CCC(C)(CNC(C3(F)CC3)=O)C2)=O)CC1 N1(C(C23CN(C(C(CCSC)N(C)C)=O)C(C2)CO3)=O)CC2(COC(C)(C)C2)C1 c1(C(=O)NC(C2CN(C(c3cc(C)no3)=O)C2)C)c(O)cc(F)cc1F c1(NC(=O)NC2CN3CCC2C3)cc(Cl)ccc1Cn1cc(-c2nccs2)nn1 N1(C(C(n2c(C)ccn2)C)=O)CC2(CC2)CC1CNC(c1cc(Cl)cs1)=O Cc1cc(Br)cc(C)c1COc1ccccc1C(=O)NC1CCCCC(F)(F)C1 N1(C(C2CC(CC)C2)=O)CCCC(C)C1CCNC(c1cnc(O)cc1OC)=O C1(F)(C(=O)NC(C(C)OC)C)CCN(C(c2cc(C)ccc2C)=O)CC1 C#CCCC(O)C(=O)NCC1CCC1NC(c1cccc(C(F)(F)F)c1)=O n1(CCCc2ccccc2)nc(CCCC2CCCCO2)nc1C1CCCCS1.S c1(CC)cc(C(=O)N(C(C)CNC(C2CC(CF)C2)=O)C)c(Br)s1 c1(OC)ccc(O)c(C(N2CCCCCC2CNC(C2CC2C(F)F)=O)=O)c1 C1(C(=O)NC(c2cccc(C)c2)CNC(=O)CP(C)(C)=O)CCCC2(CC2)C1 CCCCC(C)CCC(=O)NCCC(C)N(C(=O)CC1CC(F)C1)C c1(SC)ncc(N)c(C(N2CC3C(NC(C4(C)CC4)=O)C3C2)=O)n1 c1(N2CCC(NC(c3cccc(=O)o3)=O)C(F)C2)ncnc2[nH]ccc12 C1(C(=O)NC2CCC(NC(c3n(CC)ccc3)=O)C2)CCCS1(=O)=O N1(C(c2ccc(C)o2)=O)CCCCC1C1(NC(c2cnn(C(C)C)c2)=O)CC1 CCCCCCC(=O)NC1CN(C(C2(CC(C)C)CCC2)=O)CCC1C C(=O)(C1CCCc2c[nH]nc21)NCCC1CCCN(C(c2c(C)nccc2)=O)C1 N1(C(N2OCC(=C)C2)=O)CCC2(CC1)CC2C(=O)OC(C)(C)C N1(C(c2cncc(OC)n2)=O)CC2CCCC1(CNC(=O)C(C)(O)C(C)C)C2 C1(CN=[N+]=[N-])CCCN(C(c2cc(CNC(=O)Cn3ccnn3)no2)=O)C1 Cc1cnc(Cl)c(C(=O)NCC2(O)CCCN(C(=O)CNC=O)C2)c1 Cc1nc(C2CCC2)oc1C(=O)NC(C1CCCN1C(c1ccc(CO)s1)=O)C C1(OC)CN(C(=O)C2=CCCCO2)C(C)(CNC(=O)Cc2sccc2C)C1 c1(NC2C(C)SCC2)ccc(S(=O)(=O)NCc2cc3c(s2)CCSC3)cc1Cl C1(C(N2CCC(n3cc(CN4CCCC4)nn3)C2)=O)(CO)CCCO1 Cc1ccc(C(=O)NCC2(C(=O)NC3CCN(C)C3=O)CC23CCC3)nc1 c1(N(C(c2scc(C)c2)=O)CC2CCNCC2(F)F)ncnc2cc[nH]c12 Cn1cnc2cc(C(=O)NCCCOCCNC(c3ccsn3)=O)ccc12 C1(CNC(=O)CCc2nccn2C)CCN(CC2N(C)CC(O)C2)C1(C)C C1(CNC(c2n[nH]c(C)c2C)=O)CC2(CC2)CN1C(=O)CCc1nc(O)n[nH]1 C1(c2n(C)ccn2)CN(C(=O)CC#N)CCN1C(c1cnc(C2CCOC2)s1)=O c1(OC)ccc(NC(=O)C(C)NC(C2CC2C(=O)NCCO)=O)cn1 c1(OCC(=O)N(C2CN(C(CCSCC)=O)CC2F)C)ccc(Cl)cc1F C(=O)(C1c2ccccc2C2CC1C2)NC1(CN(C(=O)C(C2CC2)N(C)C)C)CC1 c1(C(N2CCC(NC(C3CC(CF)C3)=O)C2)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 C1(CNC(C(C)OCCOC)=O)CC(=O)N(C)C1.C12(CC1)CCNC2=O c1(C(=O)O)ccc(S(=O)(=O)N2CC(NCc3cnc(Cl)cc3Cl)C(C#N)C2)cc1 CCCC(CC(=O)NC(c1cnc[nH]1)C)NC(=O)CC1CC1 N1(C(=O)OC(C)(C)C)CCC(C(=O)O)(CCOC(=O)CCCCN(C)C)C1 N1(C(CCC(=O)NC)=O)CCC2(CC1)COC(CNC(=O)C(C)(C)C)C2 Nc1ccc(F)c(C(N2CCC3C(NC(c4cnsc4)=O)C3CC2)=O)c1F c1(N(C2CCN(C(C3CCCS3)=O)CC2)CC2CC2)cc2nncn2cn1 N1(C(c2c(CC)cns2)=O)CC2CC(C1)CN(C(c1conc1C(C)C)=O)C2 C(CCCCC(=O)NCC(O)CN(C)C(c1cn2ccsc2n1)=O)=CCCC c1(OC)ccc2nc(C)c(C(=O)NC3CC3NC(c3cc(Cl)nn3C)=O)n2n1 CCCS(=O)(=O)CC(=O)NCC1(NC(c2cn(C)c(C(F)F)n2)=O)CCCCC1 CCCCCC(F)C(=O)N1CCC(C(=O)N(CCCC(CC)CC)C)(CC)CC1 C(C(C)C(=O)NC1CC(C)(CNC(c2cncnc2)=O)C1)OC c1(-c2scc(C(=O)NCCCOC)n2)ccc(F)c(N(C)C)c1 c1(C(=O)OCC)ccc(C=CC(=O)NCC2CC2NC(=O)C(C)S(N)(=O)=O)cc1 C1(C(=O)NCCOCCCNC(CC(C)(C)O)=O)Cc2c[nH]cc2S1(=O)=O CCCC(C)CC(=O)NOCc1cc(N2CCCC2)ncn1 C1(C(N(CCN(C(c2nc(C)oc2)=O)C(C)C)C)=O)CCOCC12CCCC2 C1(C)(C(=O)NCCC2(NC(CC=C=C)=O)CCOCC2)CCC(=O)NC1 C1(C(N2C(CNC(=O)C(O)C3CC3)CC2)=O)CCCC12CCOCC2 CCC(CNC(=O)C(C)NC(c1ccc(CO)s1)=O)C(C)(F)F N1(C(=O)NC(c2ccsc2Br)C)CCC(C2CCN(C)C2)C1 C1(C(=O)O)CN(C(c2ccc(CCF)cc2)=O)CC12CCOCC2 N1(C(C2CC(C)=C(C)CC2)=O)CC2CCC1CN(C(c1ccc(CO)cn1)=O)C2 N1(C(C2(C(=O)OCC)CC2)=O)CCC(O)(CNC(c2cc(Cl)c(C)cn2)=O)CC1 c1(CC)cc(C(N2CCCCC2CNC(=O)CC(=O)N(C)C)=O)c2c(c1)CCO2 c1(C(CNC(COCC=C)=O)NC(c2cc(CC)[nH]n2)=O)cccc(Cl)c1 N1(C(C(C)(C)CNC(c2ccncc2Cl)=O)=O)CC2(C)CC1CCO2 c1(C(N(CCN(C(C2C(CC)C2)=O)C)C(C)C)=O)cnc2cc[nH]c2c1 CC(C)CC(=O)C(=O)N1CCC(C)(C(N2CCOC(C3CC3)CC2)=O)C1 N1(C(c2ccc(NC(C)C)nc2)=O)CCN(C(=O)C(C)c2ccon2)CC(O)C1 Cn1cc(NC(=O)C(c2ccccc2)=O)nc1C(=O)Nc1ccc(O)cn1 CC(O)CC(=O)NC1CC(C(=O)NCC(C)Oc2ccccc2)C1 c1(OCC)cnc(C(N2CCCC(N(C(=O)CC3CCCC3(F)F)C)C2)=O)cn1 O=C(C1=CC2CCC=CCCC12)NCC1CC(O)CN1C(=O)C=Cc1nccs1 C(=O)(CCN=c1[nH]ccs1)NC1CN(C(C(c2c(C)n[nH]c2C)C)=O)CC2C1C2 c1(OC)cc(C(N)=O)cc(C(N2CCC3(NC(=O)C4=NOCC4)CC3C2)=O)c1 N1(C(C=CC=CC)=O)CCC2CC1CN(C(=O)C1=CCCOC1)C2 c1(N(CCCNC(COCC)=O)CC)snc(Cl)c1C#N C1(C)(NC(C2CCC(CNC(c3ncn(CC)n3)=O)O2)=O)CC2(CCC2)C1 C=C(Br)CCC(=O)N1CC(NC(=O)CN2CCCCC2=O)C(SC)C1 N#CC1(C(=O)NCCCCCNC(=O)CSCc2cccc(Cl)c2)CCCO1 c1(OCC(=O)NC2C(NC(=O)CCCc3cnccn3)CCC2)ncccc1O C1(CNC(C=C(C)Cl)=O)CC(F)(CNC(c2ccnnc2)=O)C1 C(=O)(C#CC1(C)COC1)NC(C(=O)NCC(C#C)CC)C1(C)CC1 c1(NC(C(C(C)OC)NC(c2ccsc2C)=O)=O)ccc(C)nc1O N1(C(CCN(C(CN2C(C)CCC2)=O)C)=O)CCC2CC12CO C1(C(C)(C)NC(c2cnc(C)[nH]2)=O)CCCCN1C(c1nnsc1C)=O c1(C(N2CC(C)C(NC(c3ccccc3Cl)=O)CC2)=O)ccc2nnn(O)c2c1 CC1c2nncn2CCN1C(c1ccc(Cl)c(F)c1)C(=O)NC1CC(F)(F)C1 c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(C)C)C(=O)C1)CC2 c1(CC)cc(C#N)ccc1NC(=O)NC(Cc1c[nH]c2cnccc12)C1CC1 C1(O)(C(N2CCC(N(C(=O)CC3CC4CCC3O4)CCC)C2)=O)CCCCCC1 C(N=c1[nH]c(=NC2CCCC(C)C2)[nH]c2cccnc12)c1ccc(C(C)C)cc1 c1(CC(=O)NC(CC=C)CNC(c2ncncc2Br)=O)cc(F)ccc1F CC1COC2(C1)CN(Cc1ccc(-n3cccc3)cn1)C2 N1(C(C2CCCOCC2)C(=O)NCCC#N)CCC(C2CC2)CC1 CC1Cc2ccccc2N(C(c2ccnn2C2CCCC2)=O)C1C c1(C(N(CCCNC(COCCC)=O)C(C)C)=O)cnc2ccccc2c1OC C1(CNC(C=CC=CCC)=O)CCC2(CN(C(=O)CN3CC(C)(C)C3)C2)O1 c1(CCNC(C)=O)cccc(CC(=O)NCC2CN(C(=O)CNC=O)CCO2)c1 C1(NC(CC(C)C)=O)CC(=O)N(c2ccccc2F)C1.C123CC(C1)(C2)CNC3=O Cc1ncccc1C(=O)NC(CNC(=O)Cc1cc(C(F)(F)F)co1)C(C)(C)C N1(CCC2CC(C)(C)OC2)C2CCC1CC(F)(CN)C2 C1(NC(=O)C(O)CC2CCCC2)CCC(NC(=O)CCCC2CCCCC2)CC1 N1(C(C2(CC)CCC2)=O)CCC2OCCN(C(=O)COCc3nc(C)no3)C2C1 C1(C(=O)NCC(C(C)O)C)CCC(C)(C)N(C(C2CC2(C)C)=O)C1 Cc1ccc([N+](=O)[O-])cc1C(=O)NC(Cn1cc(CC(C)(C)C)nn1)CC(C)C C1(NC(c2c(C(C)C)cccc2)=O)CCCCN(Cc2nc(=O)n(C)[nH]2)C1 c1(C(N(C)CC2CCCN(C(C(=O)NC)=O)C2)=O)cc2ccc(Cl)nc2s1 CN(C)NC(=O)CCC(=O)NC1CN(C(C2C(F)(F)C23CC3)=O)C1 c1(CNC(C(CC)C)CO)ccc(-c2sc(C(F)(F)F)nc2C)cc1[N+](=O)[O-] c1(NC2(CCNC(=O)CC3CCC(O)C3)CCC2)ncc([N+](=O)[O-])cc1Br C(=O)(CC(C)CC(C)(C)C)N1C(C(N2C(C)(C(=O)NC)CC2)=O)CSC1 Cc1cc(C(=O)NCC2CCC2NC(c2nc(Cl)ccc2N)=O)cc(C)c1Cl C(C(CCNC(C1CCCN1C(=O)CCN1CCCCC1)=O)OC)OC C(N=c1[nH]c(=NCc2cnsc2)c2c(F)cccc2[nH]1)C12C(F)(F)C1CCCC2 CS(=O)(=O)c1cccc(OCCCOC(=O)NC2CC2)c1 c1(N2CC(C)C(F)(F)C2)nc(=NCc2cnccc2Cl)[nH]c2c1CCCCCC2 CC#CCCC(=O)N(CC(C)CNC(c1ccccc1CC(=O)OC)=O)C N1(C(COCCN(C)C)=O)CC2(CCCN(C(c3cc[nH]c3)=O)C2)C1 c1(CC)cnn2ccc(C(=O)NC(CNC(=O)C(F)(F)C(C)O)C3CC3)nc12 c1(N2CCC(NC(=O)NC(c3ccccc3F)(C#C)C)C2)cc(F)ncc1F C(=O)(CCCC(C)(F)F)N(CC(O)CN(C(=O)Cc1n[nH]c(=N)s1)C)C C12(OCC)CCC(C(=O)NC(C)(C)COCCCNC(=O)CC=C(Cl)Cl)(CC1)C2 C#CC1(C(=O)NCC(C)(O)CC)CCN(C(c2ccsc2)=O)C1 c1(C(N2C(C)CCC(N(C(=O)OC(C)(C)C)CC)C2)=O)cc2cn[nH]c2cc1O C1(C(C)NC(c2c(-c3cn(C(C)C)nc3)n[nH]c2)=O)CN(C(=O)C(N)=O)CCO1 c1(SC)cc(C)c(C(=O)NC2CC(F)(CNC(C3CC3C3CC3)=O)C2)s1 c1(C(N2CCC(C(=O)NCCCCC#C)(CO)C2)=O)nccc(C)c1N C1(NC(C(OC)OC)=O)CC2(C1)CN(C(c1cc(F)ccc1C(F)F)=O)C2 Cc1cc(C(=O)NCCCC(C)NC(=O)CC(C)CN(C)C)ccc1O N1(C(C2CCN(C(c3cnns3)=O)C23CC3)=O)CCc2ccccc2C1 c1(C(C)=O)cc(C(=O)NC2CN(C(=O)C(C)(C)C(F)(F)F)C2)c(C)nc1C n1(CC)cc(Br)cc1NC(=O)NC(c1noc(C2CC2)n1)(C)C N1(C(C(c2ccc(C)o2)C)=O)CCN(C)CC1CNC(c1nscc1C)=O C(=O)(C(C(C)(C)C)N(C)C)NCC1CN(C(CSc2nc(C)[nH]n2)=O)CC1O N1(C(c2c(CC)nn(C)c2)=O)CCCCC(NC(C2CC(=C3CCC3)C2)=O)C1 N1(C(C(CCCC)NC(N)=O)=O)CCOC2(C1)CN(C(c1cnco1)=O)C2 N1(C(Cc2nc(C)[nH]n2)=O)C2CCC1CC(NC(=O)Cn1[nH]cnc1=N)C2 C1(CNC(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(=O)C=C(C)C(F)F)CC1C C(CN=c1[nH]c(N2CCNC(=O)CC2)nc2c1CSC2)(c1cccc(C)c1)OC C12(C(=O)NCC3CCN(C(C4C(C)(C)C4(F)F)=O)CC3)CC=CCN1CCC2 c1(NCC2CC(NC(=O)C=Cc3ccncn3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl C(=O)(C(C)(C)C(N)=O)NC(CC)CN(C(=O)CCc1ncccc1C)C C(=O)(C(CCC1(C#N)CC1)N(C)C(=O)OC(C)(C)C)Nc1ccc(C(C)C)s1 C12(C(=O)NCC(C)(O)CNC(=O)CCc3ccc(Cl)nc3)CCCCC1C2(F)F c1(N2CC3CN(C(c4c(C)cc(Br)cn4)=O)C3C2)[nH]cnc2nc(Br)cc1-2 c1(C(=O)NC2(C)CN(C(C3CC3F)=O)C2)cccc(Cl)c1C(F)(F)F CC1(C)CC(C(N2CCCC2CC(N)=O)=O)CN1C(=O)CC1CCCCC1 C1(n2c(CNCC(COCC)(C)C)ccc2)CCC(C)CC1 C1(C(=O)NC(C2CCN(C(C(C(CC)C)O)=O)CC2)C)CCC(C2CCC2)CC1 n1(CC(=O)O)nc(-c2ccc(Cl)c(Cl)c2)c2ccccc12 c1(CC)ncnc(N2CC3(CC3)CC2CNC(=O)CCCc2nncn2C)c1F c1(CCC)[nH]ccc1C(N1CC(CNC(c2cncnc2)=O)(COC)C1)=O N1(C(C(CC)OCC)=O)CCC2(CC1)CCN(C(=O)COC1CC1)CC2C C1(O)(C(=O)NC2CC(OCC(=O)N(C3CC4(CC4)C3)C)C2)CCCCC1 c1(CC(=O)NC2CC3(NC(=O)CC=C(Cl)Cl)COC2C3)n[nH]c2c1CCCC2 N(C1CCCc2c[nH]nc21)C(c1ccc(CNC(C(C)CC(F)F)=O)cn1)=O C1(C(=O)NCC2C3CN(C(c4nonc4N)=O)CC23)(CC)CCCCC1 c1(C(N2CCC(NC(C3(C(=O)NC)CCC3)=O)C2)=O)ncccc1Br Cc1cc(Br)cc(C)c1CC(=O)OC1C=CC(C(=O)N(C)C)C1 C1(CNC(=O)CC2CCSC2)CN(C(C2(c3ccno3)CC2)=O)CCC1(F)F C1(Cc2cn(CC(CC)C)nn2)CCCCN1C(C1(C(F)F)CC(=O)C1)=O C1(C(N2CC(C)N(C(=O)CCC=CBr)CC2)=O)CCC2(CCOCC2)O1 c1(C(=O)NCC2C(NC(CCC3N(C)CCC3)=O)CCCC2)ccc(C#N)cn1 c1(CN2CC3C(C(=O)Nc4c(N(C)C)ccnc4)(C3)C2)cc(O)cc(O)c1 C1(CNC(CCC#C)=O)C2CCCC1N(C(C1CNC(=O)O1)=O)C2 c1(OC)cc(C(N2CCN(C(=O)C(C)(C)C3(C)CC3(F)F)CC2C)=O)nc(C)c1 Cc1cccc([N+](=O)[O-])c1C(=O)NC1CC2CC(C1)N(C(C1(C(N)=O)CC1)=O)C2 N1(C(c2cncc(C)c2Cl)=O)CCCC2(CNC(c3cccs3)=O)CCCC12 c1(C(=O)NC(C)CNC(C2(C)CCCC2C)=O)ccc2c(O)n[nH]c2c1 N1(C(c2cnc(OC)nc2C)=O)CCC2C(C1)NC(=O)CCN2C(=O)C(C)SC C(=O)(CCCCC(=O)NCc1ccoc1C(N1CCC(C)(O)CC1)=O)OC CC(C)(C)C(O)C(=O)N1CCCC(CNC(=O)CCNC2(C)CCC(O)CC2)C1 c1(C(CC)O)cn(C2CC(Cc3ncoc3-c3ccccc3)C2)nn1 c1(NC2CCC(CCCC)C2)ncc(C)cc1S(=O)(=O)N1CC(CO)(OC)C1 N1(C(C2CCC(C)N2C(c2ccnc3c2OCO3)=O)=O)CCNC2(CCC2)C1 c1(SC)cncc(C(=O)NC(C)CCNC(c2ccncc2)=O)c1 C1(F)(C(N2CC3C(NC(=O)CC4CN5CCN4CC5)C3C2)=O)CC12CCCCC2 c1(CNC(C2N(C(C(=O)NCCC)CSC)CCC2)(C)C)ccc(F)cc1 N1(C(CNC(C)=O)=O)CCCC(CCN(C2CCC2)C(C2(C(F)(F)F)CC2)=O)C1 c1(SC(c2scc(CNC(CNC(=O)OC)=O)n2)CC)ccc(Br)cc1 C=CCCC(C)(C)C(=O)N(CC(C)N(C(=O)C(c1ccccc1F)C)C)C C1(C(N(C(C)C)CCNC(C23CC(CO)(C2)C3)=O)=O)CCCN1C=O CC1CCCC1C(=O)NCc1n[nH]cc1CNC(=O)CCCN1CCCC1 C1(CNC(=O)NC23CC(c4ccccc4)(C2)C3F)CC2(C1)CC2(F)F CC1CC(C(=O)NCC2(C(=O)NC3(CF)CC3)CC2)=NO1 N1(C(C2C(C)CCS2)=O)CCN(C2CCN(C(=O)CSc3nncs3)C2)CC1 C1(CNC(C2(C)CC2Br)=O)CN(C(=O)CCCc2ccccc2)CCC12CCC2 Nc1c(F)ccc(F)c1C(N1CCC2C(NC(c3cscn3)=O)C2C1)=O CC(O)CCCCCC(=O)NCC1CCN(C(c2cnc3[nH]c(=N)sc3c2)=O)C1 C12(CNC(C3CC(NC(CCc4ccn(C)n4)=O)C3)=O)CCC(CC1)CC2 c1(C(=O)NCC(CNC(c2cc(CCC)oc2C)=O)O)ccc(Cl)c(Cl)c1OC N1(C(CC=CC=C)=O)CCN(C(=O)CCC(=C)C)C(C(F)(F)F)C1 C=CC(C)(C)C(=O)NC(C)CCNC(=O)CC1CCC(C2CC2)O1 C12(CNC(C3CCCN(C(C(CC)C)=O)C3)=O)CCC(CC1)CN2C(C)=O N1(C(C(CSC)(C)C)=O)CCCC2(CCN(C(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)C1 N1(C(c2ccncc2)C(=O)NC)CCN(CC(C)O)CC1 C(C(COC)CC(=O)N1CCC(C(N2CC3(CCC3O)C2)=O)CC1C(C)C)OC c1(CC(C(=O)NC(c2c(F)ccc(C)c2Br)=O)N)ccc(S(N)(=O)=O)cc1 C(N=c1[nH]c(Cl)ncc1F)C1C(NC(C2CCC(CN(C)C)O2)=O)CCC1 C=CC(C)CCS(=O)(=O)NC(CC)COC.OCC C1(N(C(=O)CCC2CC2(C)C)C)CCN(C(c2nn[nH]c2Cl)=O)C1 N1(C(C(C2CCCCC2)OC)=O)CCC(NC(=O)C(C)N2CCC2)C(C)(C)C1 N1(C(C(=O)NCCC2CC(C)(C)C2)=O)CCCSCC1C1CCC1 c1(OC)c(C(=O)NCC(C2CC2)N(C(=O)CCC2CC2C)C)ccc(Cl)c1Cl c1(N2CCC3(CN(C(C4(C)CC4(F)F)=O)C3)C2)ccc([N+](=O)[O-])cc1S(C)(=O)=O CC1CC(NC(C2(CCF)CC2)=O)CCN1C(=O)CCN1CCCS1(=O)=O CC1=NNC(=O)C1Cc1cn(CCCCCNC(=O)COCC2CCCO2)nn1 c1(C(N(C2CCN(C(=O)CC3CC(C)OC3C)C2)CC)=O)cncc(O)c1 C(=O)(C(CC(F)F)NC(=O)CCC(N)=O)NCCC=CC=C C(=O)(CC(C)CNC(=O)C=C(C)c1ccco1)NCC1(CC=C)CCCC1 c1(CC)noc(CC)c1CC(=O)NCC1C2CN(C(=O)CN3CCOC3=O)CC12 N1(C(C2(NC(CC3CC(CC=C)C3)=O)CC(F)(F)C2)=O)CCCC(C=C)C1 C=CC1OCCCC1C(=O)NCCC(C)(C)NC(C1CCC(F)(F)C1)=O N1(C(c2cnn(C)c2Cl)=O)CC(C2CC2)(C(=O)NCCc2ccncc2)C1 CC1CCN(C(=O)CC2C=CC(NC(=O)C(=O)C(C)(C)C)C2)CC1(C)C C#CCCC(=O)N(CCCN(C)C)CCNC(=O)C(C)OCOC C1(NC(c2nn(C)c(O)c2)=O)CN(C(c2cccc(O)n2)=O)CC1C#N c1(NC(CCCN(C)C(C2CC2F)=O)=O)cccc2c1CCC2 c1(N2CC3(CN(C(C(N4C(=O)CCC4=O)C)=O)C3)C2)ncnc2c1cnn2C(C)C C(=O)(CCCC(=O)OC(C1CC(O)(c2ccccc2)C1)=O)NCCN(CC)CC C(CCCCCNC(c1ccnc(O)c1)=O)N(C(=O)C(F)(F)C1(O)CCCC1)C CCC(C(C)C)C(C(=O)NCC1CCOCC1)N1CCCC(NC(=O)C(N)=O)C1 CC1(C(=O)NCc2ncoc2C2CN(C(=O)C=CCF)C2)CCC(=O)NC1 C1(C(=O)OC)CN(C)CCN1C(C1CC(O)CN1C(=O)C(C1CCCCC1)=O)=O C1(C(=O)NC(CC#C)CO)CN(C(C2(Cl)CC2(F)F)=O)CCO1 c1(C(N2CCC(C)SCC2)=O)cc(O)nc2c1CN(C(=O)CCCF)CC2 N1(C(c2n(C)cnc2)=O)CC(CNC(=O)C(O)CC(F)F)CC12CCC2 N1(C(Cc2ccc(C#C)cc2)=O)C2CCC1C(C)C(NC(C1(CCO)CC1)=O)C2 C1(NC(c2n(C)nnn2)C2CC3CC3C2)CCCCCCCCC1 Cc1ncc2n1CCN(C(=O)CC1CCN(C(C3CNC(=O)C3)=O)C1)C2 CCCC(CCCNC(C1(O)CCC1)=O)Nc1cc(Cl)nc(C2CC2)n1 c1(CC)c(C(=O)NC(C2CCCC3CC23)=O)cnn1CC.C12(O)CC(C1)OC2=O C1(C)(COC)CC(NC(c2csc(Cl)n2)=O)CN1C(c1cn(C)nc1OC)=O N1(C(C=CCN(C)C(C2CC3C(C2)C3(F)F)=O)=O)CC(S(N)(=O)=O)C1 Cc1ccc(C(=O)N(CCCN(C(=O)C(O)C2CCC2)C)C)o1 C12(CC(N3C(C)CC(CNC(=O)CN(CC(C)(C)C)C)C3)=O)CCCN1CCC2 c1(C(=O)NC2CC(NC(c3c(O)cccc3O)=O)C2)ccc([N+](=O)[O-])s1 Cc1cc(CN=C(NCC(=O)NC2CC(C3CC3)=NO2)NC(C)C)n2ncc(I)c2n1 C=CCC(CC=C)NC(C12CC(NC(=O)CCC(C)N(C)C)(C1)C2)=O C1(N(C(C(C)=C(CC)C)=O)C)CN(C(c2occc2C(C)C)=O)CC1F N1(C(c2c(C)coc2)=O)CCC(CO)(CNC(=O)CC2CCSC2)C1 c1(C(=O)NCCNC(C(C2CC(F)(F)C2)OCC)=O)n[nH]c(C(C)C)n1 O=S(=O)(c1ccc(Br)nc1)N1CCCC1N1CCC(Cl)=C(Cl)C1 c1(N(C(c2cc(F)ccn2)C(=O)NC2(C)CC2)C)cc(Br)cc([N+](=O)[O-])c1 N1(C(CC(C)CNC(=O)C(F)F)=O)CCC2(CC1)CC2C#N C(=O)(C(N)Cc1cnn(NC)c1)N1CCC1c1ccccc1.CCO Cc1ncc(N)cc1C(=O)NCC(C)(O)CNC(=O)CC(C)n1cccn1 Cc1nc2ccc(C(=O)NC(C)CNC(C3CCC(C)CC3)=O)cc2[nH]1 N1(C(C2CC(C)(C)OC2)=O)CCCC(C2(NC(=O)C#CC3CCCCO3)CC2)C1 C(C)(N=c1[nH]c(=NCC2COCC2O)[nH]c2c1COC2)c1ccc(C)s1 Cc1cc(CC(N2CCC(C)(CNC(C3(Br)CC3)=O)C2)=O)ccc1CO c1(C(N(CC(C)N(C(c2c(SC)csc2)=O)C)C)=O)cnn2ccc(C)cc12 C(=O)(CS(=O)(=O)C12CC(C1)C2)NCC(CNC(CC(CC(C)C)C)=O)C CCCC(C)CCCC(=O)NCC(C)CNC(=O)CCn1nc(C)cc1C C1(CCC)C(=O)NCCN1C(c1cn(CCNC(=O)CS(=O)CC)nn1)=O C1(C)(CNC(CC(CC)OC)=O)CCC(NC(=O)C(C)(C)N2CCCC2)CC1 C1(N(C)C)CCC(C(=O)NCC(CNC(=O)C(c2cccc(Cl)c2)O)CO)CC1 c1(C(=O)NC23C(CN(C(C4N(S(C)(=O)=O)CC4)=O)C2)C3)cc(N)ccc1Cl c1(CC(=O)NCC(CC(C)C)NC(C=CC(CC)C)=O)ccc2c(c1)NC(=O)C2 c1(-c2n(Cc3cccc(OC(F)(F)F)c3)nc(C3CC3)n2)[nH]nc2c1COC2 N1(C(C(C(=O)Nc2n(CC)nc(C)c2)C2CC2)=O)CC2CCCCC2(OC)C1 C(C(C)(C(F)(F)F)NC(=O)NCC1(C(=O)OC(C)(C)C)CC1C)OC c1(CNC(c2n[nH]cc2C(=O)NC2CC(NC(N)=O)C2)=O)ncc[nH]c1=O C1(CC)CCCCC1C(=O)N(C)CC1CN(C(c2ncc(F)cn2)=O)C1 CC1(CNC(C2CC3CCC2C3)=O)CCCN(C(C2CCC=CCCC2)=O)C1 C=C(C)CCCC(=O)N1CC2(CC2)CC1C(N1CC(C)CC(O)C1)=O Cc1ncc(C(=O)NCC(C)CN(C)C(C2(CCN(C)C)CC2)=O)o1 C(=O)(CC(C)(O)C(F)(F)F)NC1C2(CN(C(c3cccc(C)c3N)=O)C2)CC1 C1(C(=O)NC(CC)C(N)=O)CC(C)CCN1C(=O)CC1OCCO1 C1(C(=O)NCC2CN(C(C3=C(C)CCC3)=O)C(C)(C)C2)COc2ccccc2O1 c1(CC(=O)NC2CN(C(=O)CC3CCC3)CC2F)cc2ccccc2s1 N1(C(C(COCC)C)=O)CCN(C(=O)CC(C)(F)F)CC1c1ccccc1Cl N1(C(CCCCNC(N)=O)=O)CC2ON=C(CNC(c3coc(Cl)n3)=O)C2C1 C1(NC(C2(C)CCNC2=O)=O)CC(C(N2CCC3(CC2)N=N3)=O)C12CCC2 c1(C(=O)NC2C(NC(=O)Cc3ccccc3)COC2)c(F)ccc(F)c1Br Cc1nn(C)c2sc(C(N3CCC(NC(=O)C(C)C(F)(F)F)C3)=O)cc12 N1(C(c2cccc(CNC(C3CCN(CC)C3)=O)n2)=O)CCNC(=O)C1C C(CN=c1nc(C(C)(C)C)[nH]s1)C1(OC)CN(C(c2nc(OCC)oc2)=O)C1 C1(NC(C2CCC(C)(C)C2)=O)C2CC3CN(C(=O)CCP(C)(C)=O)C1C3C2 n1(C(CC)CC)nc(C)cc1C(=O)NC1CCCCC1NC(=O)CC1CCCO1 c1(CN(C)CC2CN(C(CC=CCC)=O)C2)ccc(Br)cc1OC(F)(F)F c1(OCCC(=O)NC2CN(C(C3(C=C)CC3)=O)C3C2C3)cc(F)cc(F)c1 N1(CCC(C)F)CCC2(CC1)COC(CNC(C1CC3CCCC13)=O)C2 CC1CN(C(=O)CN2CCCC2C)CC1NC(C1CC1C#N)=O CC1CN(C(=O)C(O)c2ccco2)CCN1C(=O)C(F)C(C)(C)O N1(C(=O)Cc2csc(Br)c2)CCN(C(=O)CC2(O)CCCOC2)CC(O)C1 c1(C(=O)NC2CCCN(Cc3cc(C)c(Cl)c(C)c3)C2)oc2ccccc2c1C N1(C(C2=NOC(C(C)(C)C)C2)=O)CC2OCCN(C(C3CC3C(C)(C)C)=O)C2C1 C1(OC)(CNC(=O)C=CSn2cncn2)CCN(C(=O)Cn2nccn2)C1 S(=O)(=O)(CCC(=O)NCCOCCNC(=O)Cc1ccn(C(F)F)n1)NC Cc1n[nH]cc1C(=O)NC1CCN(Cc2ncnn2C)C1 C(C)(C)(CCC(=O)NC1COCCN(C(c2conc2C2CCC2)=O)C1)OC C1(C(N(C2CCC3(CC3)C2)C)=O)CCC(CNC(C2CC2C(F)F)=O)CC1 C1(NC(CSCC)=O)CCN(CCCSC2CC2)C1.C1(C=O)CC(C(N)=O)CO1 c1(C(=O)NC)ccc(-n2nc(C(CC(C)C)OC)nc2-c2n[nH]cc2Br)cc1 C1(CN(C)C)CN(C(c2cocc2Br)C(=O)NCC2CCCO2)CCO1 c1(CN(C(=O)NC2CCC(C)=C(C)C2)CC2C(C)=NOC2=O)cnc(O)c(Cl)c1 CN1CCCC(C(=O)NC(C2CCCCC2)CNC(C2CCCC2O)=O)C1 N1(C(CCN(CC)CC)=O)CC2CC(NC(C3CC4CCC3C4)=O)C2C1 Cn1cc(S(=O)(=O)NC(c2ccccc2)c2cnccn2)cc1C(=O)O N1(C(C2(CC)CCC2)=O)CCC2(CCC(NC(=O)CN(CC(=O)NC(C)C)C)C2)C1 C(=O)(C(N=[N+]=[N-])C(C)C)NC1(C(=O)NCCCn2c(C)nnc2)CCOCC1 Cc1[nH]nc2c1CN(C(C13CC1CN(C(c1cccc(Br)c1CBr)=O)C3)=O)CC2 N1(C(CS(=O)(=O)NCC)=O)CC2COCCC2(NC(=O)C(CC(C)C)OC)C1 C1(C(=O)NCc2ccc(C(N)=O)cn2)(CC)CCN(C(C2CC3(CC3)C2)=O)CC1 c1(N2CCC(NC(C3CC3F)=O)(CF)C2)nc(C(F)F)nc2ccccc12 c1(C(=O)OC(C)(C)C)c(C)nn2c1CCCC2C.C(CC1CC(=O)N1)OC Cc1c(O)c(=O)ccn1CC(=O)NCCOCCN(C)C(C1CC=CCC1)=O CC1CN(C(=O)CSCCN(C)C)CC1NC(C1CC(O)(c2cccnc2)C1)=O Cc1ccc(C(=O)NCCC2(C)CCN(C(=O)C(C)C(F)(F)F)C2)n(C)c1=O c1(C(=O)NC(C(C(C)C)NC(c2c(CC)nn[nH]2)=O)C)coc2ccccc12 N1(C(COC(CC)C)=O)CC(C)N(C(=O)CC2CC3C=CC2C3)CC1C CC(C)C(C(=O)N(C(C)CNC(=O)CCCn1ccnn1)C)NS(N)(=O)=O N(C(=NCC#CC1CCCCO1)NCC1CCC1)C1C(C)CC1 C1(NC(c2cncc(C3CC3)c2)=O)CC(N=c2nc[nH]c3[nH]c(Br)cc23)C1 CC1CN(C(=O)C(C)(C)N=[N+]=[N-])CC(C(=O)N(C2CCCN(C)C2)C)O1 N1(C(Cc2cccc(C)c2F)=O)CC2CCN(C(c3ncccc3C)=O)C2C1 N1(C(C(C)OCC(C)C)=O)CC2(CC(NC(C3CCCC34CC4)=O)C2)C1 c1(C(=O)NC2CC(F)(CNC(c3sccc3CO)=O)C2)cc(Br)ccn1 c1(C(N(C2CN(C(c3ccc(C(N)=O)s3)=O)C2)C)=O)cc(C(N)=O)cc(F)c1 N1(C(c2ccc(N3CCCCC3)s2)C(=O)NCC)CC2(CSC)CCC2(CO)C1 c1(SC(C)C)cc(C(N2CCC(CN(C(=O)C(F)(F)C(C)O)C)C2)=O)ccc1F C(CNC(=O)Cn1cc(Cl)cn1)(CCC)NC(C=CCC)=O c1(OC)ccc(CNCCS(=O)(=O)NC)c(C)c1.C1(N)CC(SC)C1 c1(C(N2CCC(C(C)NC(COCC=C)=O)C2)=O)cccnc1N(C)C N1(C(C2C(=C)C2)=O)CC(NC(c2cc(-c3ccc(Cl)cc3)[nH]n2)=O)CC(C)(C)C1 N1(C(C(N(C)C)C2CC2)=O)CC(NC(=O)COC2(C)CCC2)CC12CCOCC2 CCCC(CC)CCC(=O)N1CCC(NC(C2(CNC(C)=O)CCC2)=O)C1 N1(CC2CC(OC(C)C)C2)CCN(CCCNC(c2coc(C(C)C)n2)=O)CC1 c1(C(=O)NC2CC(CNC(COC)=O)C2(C)C)ccnc2ncnn12 C#Cc1ccc(C(=O)N(CC(CC)NC(=O)COc2c(F)cccc2F)C)nc1 c1(NS(C)(=O)=O)ccc(F)cc1OCC(F)F.C1CC(c2nn[nH]n2)N1C Cc1cc(=NC(=O)C2CCN(C(=O)C(C)S(C)(=O)=O)CC2C)[nH]n1C c1(CNC(=O)CC2C=CCC2)ccccc1CNC(c1cnccn1)=O C1(NC(CSc2cn(C)nc2)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1O N1(C(c2cscc2Cl)=O)CCC(F)(F)C(C(n2cc(CCCO)nn2)OCCO)C1 C1(CNC(CSCC)=O)CC2CC2N1C(=O)C(C)Cc1cnc[nH]1 Cc1nc(C)c(C(=O)NCC2COCC2NC(C2CCCN(C)C2)=O)o1 N1(C(c2cn(CCCC)nc2C)=O)CCC(NC(c2cc[nH]c2)=O)C(CC)C1 C(=O)(C(F)(CNC(=O)C(C)CC(N)=O)C(C)C)N(C)Cc1c(C)cccc1 c1(C(N2CCN(C(CNC=O)=O)CC2CO)=O)ccc2ncccc2c1Cl c1(C(=O)NC2C(NC(c3c(C)c(O)ccc3)=O)CC2)nc(C)n2ccccc12 CCC(C(=O)NC1CCC(NC(c2cc(C3(C)CC3)on2)=O)C1)C1CCC(=O)N1 c1(C(C(N2C(CNC(c3c(C)c[nH]n3)=O)CCCC2)=O)=O)cc(F)c(F)cc1F C1(C(=O)NC(c2nnc(C)o2)(C)C)CC(C)(C)CCN1C(=O)C(C)NC=O N(C1CCc2cccc(Br)c21)C(C(=O)NC(c1c(C)cc(C)c(Cl)c1)C)=O c1(NC(c2c(C)c(Cl)ccc2)=O)nc2ccc(O)nc2s1 C1(C(=O)NCC2CCN(C(c3n(C=C)nnc3)=O)C2)CC2(C1)CC(C(=O)OC)C2 C(CCN=C(NCCc1cnc(C)s1)N1CCOC(C2CCCO2)C1)OCC Cc1nn(C)c(C)c1C(C)C(=O)NCCC1CCN(C(C2(C3CC3)CC2)=O)C1 C1(NC(c2cncs2)=O)CN(C(c2ncccn2)=O)CC12COC2 C1(C)(C(N2CC3C(NC(C(=Cc4ccco4)C)=O)(C3)C2)=O)CCCCC1(F)F C#Cc1cc(C(=O)N(CCCOCCNC(=O)CC2CCCO2)C)cc(F)c1 Cc1nn(C(C)C)c(C)c1CC(=O)NC1CCN(C(C23CC(C)C2C3)=O)C1(C)C C(=O)(C1CCc2ccccc21)NC1CCCN(C(C2CN(C)C(=O)C2)=O)CCC1 S(=O)(=O)(c1cccc(F)c1)N(Cc1c(C2CCN(C)CC2)nc2n1CCCC2)CCl c1(C(=O)NC2C(CNC(C3CN(C(N)=O)C3)=O)CCC2)c(F)cc(Cl)cc1F N1(C(C=CC(C)(C)NC(c2n[nH]cc2Cl)=O)=O)CCCNC(=O)CC1 C(=O)(C1=NOC(C)(C)C1)NCCC1(NC(CC2CCCC(C)C2)=O)CCCC1 N1(CC=C)CCC(NC(=O)Cc2nsc3ccccc23)C(C)(C)C1 n1(CC)nc(C(N2CCC(C(C)NC(c3cc(CO)[nH]n3)=O)C2)=O)cc1C N1(C(C(C2CCCC2)OC)=O)CC(C(N2CC([N+](=O)[O-])C2)=O)C2(CCC2)C1 c1(C(=O)NC2C3CN(C(CCCC=C)=O)C(C3)C2)ccc2ncnn2c1 c1(OC)cc(C(F)(F)F)[nH]c(=NCCCN(C(=O)C(CC2CCCC2)OC)C)n1 C(N=c1cc(Cl)nc[nH]1)C1N(C(C2CCS2(=O)=O)=O)CCC1 C1(C(=O)NCC2C3CN(C(CC=C(C)C)=O)C2C3)CCc2[nH]nc(O)c2C1 c1(OC)cccc(C(=O)NC2CN(C(=O)CC3CC(C)=NO3)CC2O)c1C c1(C(N2CCN(C(=O)Cc3cncs3)CC2C2CCC2)=O)cc2ccncc2o1 C1(C(=O)NC2C(NC(CC(CC)c3ccccc3)=O)COC2)CCS(=O)(=O)CC1 N1(c2c(C)c(NCc3ccnc(Cl)c3)ncn2)CC2CCC1CN2CC(F)F Cn1cc(C(=O)NCC(CO)NC(c2ccccc2C2(C)CC2)=O)c(O)nc1=O c1(C(N2C(C)(C(=O)NCCOC#N)CC2)=O)ccc(Cl)c2cc[nH]c12 S(=O)(=O)(c1cc(C)c(Cl)cc1C)N(C1CN(C(c2cnc(OC)c(Cl)c2)=O)C1)C Cc1csc(C(C(F)(F)F)NCC2(C3CCCN3)CCCC2)n1 c1(CNC(c2n(CC)nnn2)(C)CCSC)ccc(Cl)cc1OC C1(N(C(=O)C(Cl)=CCl)C)CCCCN(C(C2(CO)CC2(F)F)=O)C1 C(=O)(CC1=NNC(=O)C1)N1CC(C(C)NC(c2cnccn2)=O)OCC1 CCCCC(CNC(=O)Cc1c[nH]nc1C)NC(C1CCC(=O)N1C1CC1)=O C(=O)(CC(C)CN(C)C)NCC(CCOC)NC(c1cnc[nH]c1=N)=O C1(F)(C(=O)NCCc2cnc(C)[nH]2)CCN(C(c2sncc2C)=O)CC1 C1(C(N(CCNC(=O)C=CCF)CC)=O)CC(c2cccc(Br)c2)=NO1 c1(CC(=O)NCC(C)NC(c2scc(C(=O)OC)c2)=O)ccc(C(C)(C)C)cc1 N1(C(C)=O)CCC(C(=O)NC2(c3nc(C)no3)CCC2)C(c2ccccc2)CC1 C1(C(F)F)(CNC(c2cc(C)[nH]n2)=O)CCN(C(=O)Cc2ccccn2)C1 C1(C(=O)NC2CCC(C(N(CCN(C)C)CC)=O)C2)C2(CC2)C12CC2 C(=O)(C(N)CCC(=O)O)N1CC(C)C(NC(c2ccc3nonc3c2)=O)CC1 CC1CCNC(=O)C1NC(c1cc(CNC(c2cc(Cl)ns2)=O)ccn1)=O N1(C(Cn2cc(-c3cccc(CC(=O)O)c3)nn2)=O)CCCC2(CCSC2)C1 c1(C(c2nnnn2C2CCC2)Nc2ncn(C)n2)c(Br)ccc2c1OCO2 c1(C(=O)NCC(C)(C)NC(C(COCC)C)=O)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(CCN1C(=O)COc2ccccc21)N(C1CCCC1(C)O)C C1(COC)CC(O)CN1C(c1cc(CNC(C2CCC(=O)NC2)=O)no1)=O CCC(C)CC(=O)C(=O)NC(C(N1CCCCC(C)(F)C1)=O)C1CCOC1 C(=O)(CC(CC(C)C)NC(c1cccn(C)c1=O)=O)NCC(C(C)C)O C1(C(=O)NCCSCCCO)CC12CCN(C(c1cc(CO)co1)=O)C2 Cc1coc2c(C(=O)N(C)CCN(C)C(c3cnn(C(C)(C)C)c3)=O)cccc12 C#CC1CC2CCC1N(C(=O)CC1CC1CNC(=O)Cc1cc(C)[nH]n1)C2 C1(NC(Cc2cccc(C)c2F)=O)CC2CC(C1)N(C(=O)CCC(C)O)C2 c1(CC(=O)NC2C(CNC(C(C)c3ccsc3)=O)CCC2)ccc(F)c(Cl)c1 C(=O)(CCCCCCCCCO)N(CCCNC(C1(C)COC(=O)C1)=O)CC C(C(C)(C)CCC#N)(c1nnnn1CCCSC)NCCC(=O)N(CC)CC N1(C(CCC(=C)C)=O)CCN(C(c2ccc(Cl)c(OC)c2F)=O)C2COCC12 c1(C(N2CC(NC(=O)C(F)CC3CC3)C3C(C2)C3)=O)cc2c(Cl)cccc2s1 C(=O)(C(F)(CC)C(=O)OC)N1CCC(C)(CNC(c2c(CC)cco2)=O)C1 c1(C(=O)NC2CC(NC(c3cn(CCOC)nn3)=O)C2)cncc(C(=O)OC)c1 N1(C(C(C)(CO)OC)=O)CCN(C(=O)CC2OCCCO2)C(c2ccncc2)C1 N1(C(CCSCCCC)=O)CCC(C(=O)NC(C)CNC(=O)OC)C1 C1(CCC)CCC(C(=O)NCC=CCNC(=O)C(n2nccc2C)C)CC1 C(=O)(C1=CSCCO1)NCC1N(C(c2cc(C3(C)CC3)on2)=O)CC1 C(N=c1[nH]cnc2ccsc12)C1(C)CCN(C(c2ccc(-n3ccnc3)nn2)=O)C1 c1(C(=O)NC2CCC(NC(C(C)SCCCC)=O)C2)oc2c(C)cccc2c1C CC1(C(N2CCC(CS(=O)(=O)F)C2)=O)CC(c2ccccc2)=NO1 Cc1cc(N2CCC(c3cc(NC(=O)CCCC4CCC4)on3)CC2)nc(C)n1 c1(CSC)ccc(C(=O)NC(C)(CNC(C2(C)CC(C)=NO2)=O)CO)cc1 N1(C(C2C3CCCC23)=O)CCCN(C(c2ccoc2C2CC2)=O)C(CO)C1 C1(C(=O)NC(Cc2cc(C)no2)C)CC(F)CN(C(=O)Cn2cccn2)C1 N1(C(C2N(C(CC(C)C(F)(F)F)=O)CCCC2)=O)CCOC2(CCCC2)C1 c1(OC)cccc(C(N2CC3CCC(C2)N3C(=O)CP(C)(C)=O)=O)c1[N+](=O)[O-] c1(OCC(=O)N(CC(CNC(C)=O)O)C)cccc(CC2CC2)c1F c1(C(N2CCC(O)(C(C)NC(COCC#C)=O)C2)=O)cc(CC)nnc1C C=C(Cl)CCC(=O)NC1CCOCC1C(=O)NCCCn1ccnc1C c1(CC)ccc(F)cc1C(N1CC(OC)CC1CNC(c1nocc1C)=O)=O CON1CC(C(N2CCN(CC(N3CCOC(CF)C3)=O)CC2)=O)CC1=O c1(CCC(=O)OC)ccc(C(=O)NC2(C)CCN(C(=O)C(C)O)C2)cc1 C1(C#N)(C(N2CC(N(C)C(c3cn(C4CCOC4)cn3)=O)C2)=O)CCCO1 C(=O)(C1=CC(O)C(NC(=O)C2=NOC(C)C2)C1)NC(c1nc(C)[nH]n1)CO c1(NC(c2cnc(N3CCNCC3)cn2)=O)cccc2ccccc12 c1(C(=O)NC2C(NC(c3c(C)coc3)=O)C2)sc2ccc(C)cc2c1C Cc1cc(C)c2c(c1)C(NC(=O)C(=O)NCC1COCC(C)(C)O1)CCO2 C=CC1CN(C(=O)CCCSC)CC1NC(C1CC(CC)=NO1)=O C1(NC(C(C)=C(C)C)=O)CN(C(=O)CCC(F)F)CC1C1CC1 C(=O)(C(C)(C)C(O)C(C)C)NC1CCCN(C(c2c(OCC=C)cccn2)=O)C1 N1(C(c2ccc(-n3ccnc3)c(C)c2)C(=O)NCC=C)CCC2(CCC(O)C2)C1 C(=O)(CCCCCC(C)O)N1CC(C2CN(C(c3c(CC)nc(C)n3C)=O)C2)C1 C(C(N=c1[nH]nc(-c2ccccc2)o1)C1CC1)NC(C(=O)Nc1ccc(C)[nH]1)=O c1(OC)ncc(CN2CCCC2CCC(=O)NCCCc2cccnc2)cc1Cl C1(NC(C(C)OCc2ccccn2)=O)C=CCN(C(=O)C=CC=C(Cl)Cl)C1 C1(C(=O)NC2(CC#C)CCOC2)CC(N=[N+]=[N-])CN1C(=O)C(c1ccn(C)n1)C n1(CC(=O)NCC2(COC)CN(C(=O)C=CC3CCOC3)C2)ccccc1=O CCC(C)(C)CC(=O)NCC1CC(F)CN1C(C12CCC(CC1)OC2)=O C(N=c1ccc(Br)c(S(=O)(=O)N2CCCC(C)(C)C2)[nH]1)C1CCCN(C(C)C)C1 N1(C(C(C=C)O)=O)CC2(CCC2NC(c2cc(SC)oc2C)=O)C1 C1(C(N2CC(CNC(c3c(=N)cc[nH]c3)=O)OCC2)=O)CCC12CCOCC2 C=CCC(C)(C)CC(=O)NCC1CCC(CNC(c2cc(F)ccc2F)=O)CC1 N1(C(c2ccn(CCC)n2)=O)CC2CC(C(N3CCN(C)C(=O)C3C)=O)C(C2)C1 c1(C(=O)NC2CCN(C(Cc3c(C)n(C)nc3)=O)C2)cc(Cl)c(Cl)c(Cl)c1 C1(NC(c2c(C(C)NC(c3ccon3)=O)noc2)=O)CC(CO)CC1O Cn1nc2ccccc2c1CN=C(NCC1C(F)(F)C12CC2)NC(C)(C)COC C(=O)(C1=NOC(C(C)(C)C)C1)NCC(CC)NC(=O)C(c1cccc(C)c1)(C)C N1(C(C=COCC)=O)CCC2CN(c3ncnc4cc(Br)sc34)CCC12 CCC(CC(=O)N(C1CN(C(=O)CC2C(C)(C)C2(C)C)CCC1O)C)C(F)F N1(CCCNC(C(C)c2cncs2)=O)CCC(NC(=O)CCc2cnccn2)C1 c1(C(=O)NCCCCCNC(C2CC3CCCC3C2)=O)ccc2ncccc2n1 c1(CC)ccc(C(=O)NC(CSC)C(=O)N(C(C)C(C)C)C2CC2)[nH]1 N1(C(C2(C=C)CCCCC2)=O)CCC2CCCN(C(=O)COCC(F)(F)F)C2C1 C(=O)(CC(=O)N1CCC(C(F)C(=O)N(CC(O)C2CC2)C)C1)NCC N1(C(C(C)N(CCC)C(C)=O)=O)CCCCCCC1C(=O)NCc1csc(CC)n1 C1(C#N)(C(N2CC3C(CNC(C(=O)NC(C)C)=O)(C3)C2)=O)CCN(C)CC1 C1(C)(CNC(c2nccc(C)n2)=O)CCN(C(c2coc(Br)n2)=O)CC1 CC1(C)CCCC(C(N2CC(NC(=O)CCNC(N)=O)C(F)C2)=O)O1 c1(C(N2C(CO)CC(NC(C3CN(C(C)=O)C3)=O)C2)=O)cnc2ncccn12 N1(C(c2n[nH]c(=N)s2)=O)CCCC(NC(c2conc2C2CCCC2)=O)C1 N1(C(c2c3ccn(C)c3ccc2)=O)CCC2CN(C(c3cnc[nH]3)=O)CCC2C1 N1(C(C(C)N(C2CC2)Cc2ccc(C(=O)O)o2)=O)CC(C)CC(C)C1 Cc1ccc2nsnc2c1C(N1CC(NC(=O)Cc2c(F)cccc2Cl)C1)=O CN1CCN(C(=O)C(O)C(F)(F)F)CC1CNC(c1scnc1Cl)=O c1(C(=O)NC(CNC(C2(CCOCC)CCC2)=O)CO)c(C(F)F)cccc1F c1(C(C)NC(CC2CC(OC)CN2C(=O)C(C)C)=O)ccc(F)c(Cl)c1 c1(C(N2CC(C(C)NC(Cc3c(C)noc3)=O)C2)=O)n[nH]c2nccc(Cl)c12 Cc1cc2c(C(=O)N(CCCN(C)C(c3ccnc(Cl)c3N)=O)C)cccc2o1 CCC(C)(CCNC(=O)CC1CC2(CC2)CO1)NC(=O)CCc1cnoc1 N1(C(C(C=C)(C)CC)=O)CC2(NC(C3CCC3(F)F)=O)CCC1CC2 c1(C(=O)NC(CC)(C)CNC(=O)C(Cc2ccccc2)OC)ccc(C)c(N)c1 N1(C(c2ccc(C(C)C)s2)=O)CC2CCC1C(NC(C1(Br)CC1)=O)C2 C1(C(N(CC=C)C)=O)CCCN1NC(=O)CC1CC1 Cc1c(F)ccc(C(=O)NCC2CC(O)CN2C(c2ccc(Cl)c(Br)c2)=O)c1F C1(OC)CN(C(=O)CC(F)(F)CC)C(C)(CNC(c2cc[n+]([O-])cc2)=O)C1 N1(C(CC(=C)C)=O)CC(CNC(c2noc(C3CC3)c2C)=O)OC2(CCC2)C1 c1(C(=O)NCC(CC)N(C)C(c2nncn2C2CC2)=O)n[nH]c(C)c1C N1(CC=C)CCN(C(C2CC(=C)C2)=O)CC1Cc1ccccc1 c1(CN2CC(Cn3ccc(NC(CC(C)C)=O)n3)C2)cc2ccc(C#N)cc2[nH]1 n1(CC(N2CCN(C(=O)Cn3nccn3)C(CCO)C2)=O)ccc2ccccc12 c1(Nc2c(OC)cc(F)c(C)c2)c(-c2ccccc2SC)ccc2c1OCO2 N1(C(C(C)O)=O)CCOCC(F)(CNC(C2(c3nc(S)n[nH]3)CCC2)=O)C1 C(=O)(CS(=O)CCC(F)(F)F)N1CC(C(C)NC(CSCC)=O)C1 N1(C(COCCCOC)=O)CCOC(C)(CNC(c2cnc(C)[nH]2)=O)C1 c12ccccc1CC2.CC(CC1CCC1)C(=O)NN(C(=O)C(C)OC1CC1)C N1(C(CCC#C)=O)CCCC(C(=O)NCCNC(=O)C(N2CCCCCC2)C)C1 C1(CC=C)(CC=C)CCCN1C(=O)C(C(C)C)NC(=O)OC.N1S(=O)(=O)NCC1 C(=O)(CCCCCN(C)C)N1C(CC)CCC1.N1(CCC(=O)N)CCCCC1=O N12CCN(CC1)CC2=O.N1(C(C2(CC)CCC2)=O)CCCC1CCCC(=O)NC Cc1cc(Cc2nc(-c3ccn(C)n3)nn2-c2cccnc2)ccc1Br C(=O)(C#CC1(C)CC1)NCCCN(C(=O)C(C1CCC(C(C)(C)C)CC1)O)C CC1C2CCC(C2)C1C(=O)NCC1CC(C(=O)NCC2(O)CCCCC2)C1 N1(C(CCC)=O)CCC(NC(c2cc(C)ccc2OC)=O)C(CC)C1 C1(C(N2CC(F)(CNC(C3CC=C(C)CC3)=O)C2)=O)Cc2ccncc2N1 N1(C(Cc2cccc(SC)c2)=O)CCC2(CC2NC(c2csnn2)=O)C1 c1(OC)cn(C)c(C(=O)N(CCC(C)NC(c2c(C)[nH]c(C)c2C)=O)C)cc1=O C(=O)(C(F)(F)C(F)(F)F)N1CCCC(n2cc(-c3c(C(=O)O)cc[nH]3)nn2)CC1 N1(C(=O)OCC(C)C)CCN(C(c2nc(Br)cs2)=O)C(C)C1 C(=O)(C1CCCc2ccccc21)NC1C(C)N(C(=O)CC2COC(=O)C2)CC1 c1(C(=O)NCC2CN(C(c3c(C)nn[nH]3)=O)C(C)C2)cc(Cl)ccc1[N+](=O)[O-] CC1(C)CC(C)(CNC(C2CCCC2C(F)F)=O)CN1C(C1C(C)(C)C1(C)C)=O N(C1CCCn2nccc21)C(C(CNC(=O)CCC(C)(C)C#N)N(C)C)=O Cc1cn2c(n1)CCC(C(=O)N(C1CCCN(C(C3OCCO3)=O)CC1)C)C2 C1(C(C)C)CC2CCC1(CC1CCCCN1C(N)=O)C2.N12CCCC1CC2=O c1(C(NOCC(=O)NC2C(C(C)(C)C)CC2)=O)ccc([N+](=O)[O-])[nH]1 c1(CNC(COCC)=O)ccc2c(c1)CCN(C(=O)C(C)NC(=O)NC)C2 C1(C)(C(N2CC(C(C(=O)OCC)O)C2)=O)CCCN(C(=O)C(C)C(F)F)C1 C(CC(C(=O)NCC(C)N(C(=O)C(C)(C)CN1CCN(C)CC1)C)NC=O)SC n1(C2(C(=O)NC3CCC(NC(c4c(C)[nH]cc4)=O)C3)CC2)cc(C#N)cn1 CC(C)C(O)C(F)(F)C(=O)N1CCC(NC(=O)CC2CCC2)C(O)C1 N1(C(C(CC#C)O)=O)CCC2CN(C(=O)CCc3nc(C)cs3)CCC12 c1(OCC(=O)NCc2cn(CC3COC(=O)C3)nn2)cccc(-n2cnnc2)c1 N1(C(CC2(OCC)CCC2)=O)CCC(CCNC(=O)COCC)CC1C C1(C(=O)NCCCN(C(CC(CC)SC)=O)C)CN2CC3CC2(CO1)C3 C(=O)(CCC(=O)NCC(C)CNC(=O)CCN1CCCCC1C)OC O=C(C1=CC2(CCOC2)C1)N1CCN(C(c2ccccc2CO)=O)C2(CC2)C1 CCCCCS(=O)(=O)CC(=O)NC1CCN(C(c2cc3cc(F)ccc3[nH]2)=O)C1 N1(C(C2CCN(CC)C2)=O)CC(C)(C)C(NC(C2CCC(C)CC2)=O)C(C)(C)C1 C(=O)(C1CCc2ccccc21)NC1CCN(C(c2cnc(CCC)s2)=O)C12CC2 N1(C(C(CC)(C)CNC(c2cscn2)=O)=O)CCCC(O)(C2CC2)C1 c1(SC)c(CNCC(C)(C)NC(=O)C=Cc2cocn2)cccc1C c1(NC(c2c(OC)cccc2)CO)ncccc1S(=O)(=O)NC1(CC2CCC2)CC1 c1(C(=O)NCC2C(NC(c3cc(COC)on3)=O)CCCC2)ccc(C)c(C)c1 Nc1c(Cl)ccc(F)c1C(=O)NC1CC(CNC(c2ccn3nnnc3c2)=O)C1 N1(C(C(=O)NCC(CC)C)C)CCCC(C(c2ccncc2)=O)C1 c1(N(C)Cc2cc(C)on2)nc(NC2CCC(C#N)CC2)nc2c1CCC2 CC(C)C(O)C(C)(C)C(=O)N1CCOC(CNC(c2ccc(C(F)(F)F)s2)=O)C1 C(=O)(CCCS(C)(=O)=O)N1C(CNC(c2cn(C)c(Br)c2)=O)CC2CC21 N1(CC(=O)NC2(OCCN3CCOC3=O)CC2)CCCCC1CO c1(CNC(COc2ccc(C)nc2C(C)C)=O)ccc(F)c2cnccc12.CC(C)(C)O c1(C(=O)NCC2(NC(C(C)O)=O)CCCC2)cc(F)c(C(F)(F)F)c(F)c1 c1(C(=O)NCC2C(NC(C3CCC(N(C)C)C3)=O)CCC2)ccc([N+](=O)[O-])[nH]1 C1(CNC(C(C)c2cc[nH]n2)=O)CN(C(c2cc(C3CC3)ncn2)=O)CC1(F)F C=C1CCN(C(=O)CCN(C(c2cnn(C(F)F)c2)=O)CC)C1 c1(OCC=C)ccccc1C(N1CC(NC(=O)C(C(C)C)OCOC)C1)=O N1(C(C(C)(F)F)=O)CC2CC3CC2C1C3NC(c1noc2cc(F)ccc12)=O C1(OC)CCC(C(=O)NCCC2(C(N3CC(c4ncc[nH]4)C3)=O)CC2)CC1 N1(C(=O)C(F)CC2CCOC2)CCC(F)(CO)C1.C(C=O)NCCOC C1(CNC(C(CC2CC2)NC(C(N2CCOCC2)C)=O)=O)CC2(CC2)C(=O)O1 CC1CN(C(=O)CC(C2CC2)C2CC2)CC1(C)C(=O)NCC1CNC(=O)C1 CCC(C)CCN=c1[nH]c(N2CCC(C)(C(C)=O)CC2)nc2c1COCC2 C12(NC(CNC(CCC)=O)=O)CCOC(CNC(=O)C=Cc3sccc3C)(C1)C2 c1(CCCC)ccc(C(=O)N(CCCN(C)C(C2COCC(C)O2)=O)C)cc1 N1(C(N2CCC(C3C(OCC)C3)C2)=O)Cc2c(CC)cccc2C(C(=O)OC)C1 c1(C(C(=O)NC2(C(NOCC(C)C)=O)CCC2)C)ccn(C)c1 C123CCCC1N(CC2)C3=O.c1(NC(CNC=O)=O)cccc(Cn2cccn2)c1 c1(C(=O)NCC(C(C)C)(C)NC(=O)CCF)cnc2c(c1)NCC2 c1(CC(=O)NC(CCN(C(C2(CC#C)CCCC2)=O)C)C)c(F)cccc1Cl c1(C(N2C(NC(CCOCC)=O)CC(OC)C2)=O)ccc2cc(OC)ccc2c1 c1(OC)nsc(C(=O)N(C2CCN(c3cnn(C)c3)C2)C)c1Br c1(C(N2CC3C(NC(c4ccc(CCC)s4)=O)(C3)C2)=O)ccc(S(N)(=O)=O)o1 C=CCCCC(C)(C)C(=O)NCC(C(=O)NC1CC2CC1CC21CC1)C(C)C c1(SC)c(C(=O)NCCCN(C)C(c2cncn2C2CC2)=O)cccc1F c1(CC)cc(C(N2CC(C(C(=O)NC(c3nncn3C)C)OC)C2)=O)no1 c1(C(N2CCN(CC(=O)Nc3ccc(O)cc3)CC2)=O)cc(O)nc(O)n1 CCC(C)C(CNC(=O)C(C)N(C(=O)CCC=CC(C)C)C)CO C1(C(N2CCN(C(C=C(C)C)=O)C(C3CCC3)C2)=O)CC(C)CC(C)(C)C1 c1(C(C)NC(=O)NC2NCCCC2c2ccccc2)ccc(C(F)(F)F)nc1C C1(CNC(C2C(CCC)C2)=O)CC(F)CN1C(=O)C(Cc1ccccc1)OC c1(C(N2CC(CN(NC(c3c(CC)scn3)=O)CC)C2)=O)cc(C)nn1C1CC1 C(C(=O)N(C1CN(C)C1)C)(C(C)C)NC(c1cc(C)no1)=O C1(NC(C(C(C)C)SC(C)C)=O)CCCC2CN(CC=Cc3ccccc3)CC12 c1(NC2CN(C(C=Cc3n(C)cnc3)=O)CC23CCC3)ncc2c(n1)CCOC2 N1(C(COCC=C)=O)CCC(CO)C(NC(=O)CNC(=O)C(CC)CC)C1 C1(NC(C2(OC)CCN(C(c3cc(SC)n(C)n3)=O)C2)=O)CCC(C)(C)CC1 c1(C(=O)NCCOCCNC(CNC(C(CC)C)=O)=O)cc(C)ccc1Cl c1(C(=O)NC(C)C(=O)NC2C(C(=O)NCc3ccccc3)CC2)coc(O)n1 C(C(C)(CC(C)C)NC(C1CN(C)CCN1C)=O)NC(C(C)(C)OC(C)C)=O c1(OC)coc(C(=O)N(CCCN(C)C(c2cc(C)cnc2Cl)=O)C)cc1=O C#Cc1cccc(NC(=O)CC2(CNC(c3ncccc3F)=O)CC2)c1 Cc1cc(Cl)ccc1OCC(=O)NCC=CCNC(=O)C(n1cnc(C#N)n1)C C1(NC(C2N(CCC)CCCC2)=O)CC1C1CCCN(C(=O)CCC2CC2)C1 CCCC(CCCNC(C1CC12CC(O)C2)=O)NC(=O)CCC(=O)OCC C1(CCC(=O)NC(CO)C(=O)NCC(O)CCC2CC2)CCCCC1 c1(C(=O)NC2CN(C(C3CCN(C4CCCCC4)C3)=O)C2)ccnc(C2CC2)n1 Cc1cccc2c(C(=O)NCC3CN(C(c4cnn5c4CCC5)=O)C3)c[nH]c12 CC1(C)CN(C(C2CC23CC(NC(=O)CCc2nncs2)C3)=O)CCO1 C1(C(=O)NCCC(CNC(CC=CC=C)=O)O)CCC(C(C)(C)O)CC1 c1(C(C(=O)NCCCOC2CC2)N(C(C(=O)OC)C)C2COC2)ccc(Br)s1 c1(C(=O)NCCC2CCN(C)C2=O)cc2cccnc2nc1O C1(NC(CCCOCC=C)=O)CN(C(c2cn(CC)cn2)=O)C2CCCCC12 Cc1cnc(NCc2cnc(F)cc2C)c(S(=O)(=O)NCCN2CCCOC2)c1 C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCC(C)(C)CNC(c1ccccc1)=O c1(C(C(=O)NC(C)CCCNC(c2ccsc2C)=O)OCC)cccc(Cl)c1 C(C)(N=c1[nH]c2c(c(=NC(C)C3CCCC3)[nH]1)CSC2)c1cccc(C)n1 CC1=NOC(C(=O)NC(C2CN(C(c3coc(C(F)F)n3)=O)C2)C)C1C C1(CC(N2C(CNC(c3cc(OC)ncn3)=O)CC2)=O)COCC2(CCC2)O1 C(=O)(NNC(=O)C(N)=O)N(CCCn1cc(Br)cn1)C N1(C(c2c(CC)ccs2)c2nnnn2NCc2ccccc2)CCCC(C)CC1 c1(NC(=O)NC(Cc2cnc[nH]2)CO)cccc(NC(C2CCC(F)C2)=O)c1 N1(C(CCC(C)OC)=O)CC(F)(F)CC1CNC(C1(C)CCNC(=O)C1)=O c1(C(N2C(CNC(=O)CC3CCCOCC3)CCCC2)=O)nccc2c[nH]nc12 CCCS(=O)(=O)c1ccccc1C(N1CC(O)(C(C)NC(=O)CC(C)(F)F)C1)=O N1(CC(=O)N(CC(=O)NCC2C=CCN2C)CC)CCCCC1C C1(NC(C(C(CC)C)O)=O)COC2(C1)CN(C(=O)C(C)O)C2 C1(C)(C(=O)NCC(CC)(C)Cl)CCCN(C(=O)Cc2cnn(C)c2C)C1 C1(C(=O)NCCN(C(c2cccc(C)c2C)=O)CC)CCc2ncccc2C1 C(CN=c1cc(C)c(S(=O)(=O)NCC2CCN2C)c[nH]1)=CCCC CC(C)S(=O)c1ccc(C(N2CC3CC2C3NC(C2CCC(=O)N2C)=O)=O)cc1 n1(CCOC)cccc(C(=O)NC(C)CNC(=O)C(C2CCCO2)OC)c1=O C(CC(O)CC(=O)NCC1CCCN(C(c2scnc2Cl)=O)C1)SC N1(C(CC2CCC(=O)NC2=O)=O)CCCCC(NC(=O)COCCF)CC1 CC1CN(C(=O)CS(=O)(=O)CCO)CCCN1C(=O)C=C1CC1 C1(C)(CNC(c2onc(C)n2)=O)CCCN1C(=O)CC(C)(C)C C(=O)(C(C(C)(C)C)NC(C1CC1(C)C)=O)N(C1CC(CC2CC2)C1)C c1(CC)cc(C(=O)NCC2CCCCN2C(=O)Cc2cnsc2)ccc1F C1(C(=O)NCC(CNC(c2c(C)c[nH]n2)=O)F)CCCN(c2ncccn2)C1 N1(C(C(C=C)C)=O)CCN(C2CN(C(c3conc3COC)=O)C2)CC1 c1(C(=O)Nc2ccc(-n3ccc(O)n3)cc2)cc(S(=O)(=O)Nc2nccs2)c(Cl)s1 CC(C)CC(CNC(C1CC1(C)C(F)F)=O)NC(c1cc(Cl)no1)=O Cc1ccc(C(C)CC(N2CCC(O)(CNC(c3ccc(Cl)o3)=O)C2)=O)cc1 C(=O)(C1OC2(CCN(C(c3cc4sccc4s3)=O)C2)C1)NC1(C)CC1 c1(C(=O)NC2C(NC(Cc3cc(C)ns3)=O)COC2)cccc2nccn12 C1(C(=O)NCCC2(O)CN(C(C(N)=O)=O)C2)CCc2nnc(O)n2C1 CCC1C(=O)Nc2ccc(C(=O)NC3CC[Si](C)(C)C3)cc21 c1(C(=O)NC(CNC(C(CC)N(C)C)=O)C2CCC2)c(C)oc(C)c1C c1(C(N(CC(=O)NCC2CC3CCCC3C2)CCOC)=O)ccc2ccoc2c1 c1(CC)ccc(F)cc1C(=O)NC1CCN(C(c2cnc(N)c(Cl)c2)=O)CC1O CC(C)CC(C)C(=O)NCC(C)=CC(=O)N(CC(C)(C)O)C n1(CC)cc(C(=O)N(CC(C)NC(c2coc(C(C)C)n2)=O)CC)c(C)n1 c1(C2OC(=O)N(C3CC3)C2)ccccc1S(=O)(=O)N1CC23CCCC2(CO)C13 c1(C(=O)NC2C3CCN(C(c4cccc(OC)c4C)=O)C32)nccc2cc[nH]c12 c1(C(=O)NCC(CN(C)C(C2(Br)CC2(C)C)=O)O)ccc2c(c1)COCO2 Cn1cc(C=C(F)C(=O)NC2CCC(F)(CNC(=O)Cc3cccs3)C2)nn1 c1(C(=O)NCCC23C(CN(C(CC(=O)OC)=O)C2)CC3)cnc2n1C(C)CCC2 c1(C(=O)NCC(CC)NC(=O)C=CS(C)=O)c(Br)sc2nnsc12 C1(C(=O)NCCCNC(CC23CC(C)(OC2)C3)=O)CC1C1CC(F)(F)C1 C(=O)(CCCN(C)N=O)NCC1CCN(C(c2cnc(CC(C)C)s2)=O)CC1C CC1CN(C(=O)C(c2ccccc2)NC(=O)CCP(C)(C)=O)CCN1C1CC1 c1(-c2cc(C(=O)O)n[nH]2)cc(Cl)nc(Cl)c1.S(=O)(=O)(c1cn[nH]c1)N C#CCC(C(=O)N1CCC(OCCF)C1)NC(=O)Cc1csnc1C N1(C(Cn2cc(C(C)=O)nc2)=O)CCN(C(C2CC(O)(C(F)(F)F)C2)=O)CC1C CP(C)(=O)C(O)C(=O)NCC1(O)CCN(C(c2cnc(N3CCOCC3)s2)=O)C1 N1(C(C2N(C(C(CC)N(CC)CC)=O)CSC2)=O)CCOC(C2CC2)CC1 N1(C(C#CC(=O)O)=O)CCc2cccc(C(=O)N(CCO)Cc3cccnc3)c2C1 CC1CN(C(C2(Cl)CC2)=O)CCC1NC(=O)C=Cc1cn[nH]c1 C#CCCCCC(=O)NCC1(F)CC(CNC(=O)C(C)O)C1 c1(C(=O)NC2CC(CC(=O)NCc3c(OC)nsc3)C2(C)C)cc[nH]c2nccc1-2 c1(SCC2N(C(C3CCC3)C)CCC2)ccccc1F N1(C(C(COCC)c2ccccc2)=O)CCC(O)C(NC(=O)C(C)(C)CSC)C1 c1(C(N2C(C(=O)NC(Cc3cc(C)no3)C)CCCC2)=O)coc2ccccc12 c1(NC(C2C3CC2N(Cc2ccc(N4CCOCC4)cc2Br)C3)=O)cnc(O)nc1O C(=O)(C(C)(C(C)C)OC)N(CCCNC(c1cccc(CC)n1)=O)C(C)C c1(OC)cccc(Cl)c1CC(N1CCN(c2cc(F)ncn2)C(CCO)C1)=O C1(NC(C2(CCCC)CC2)=O)CC2CC1N(C(c1nn(C)c(C)c1Cl)=O)C2 C12(C(=O)NC(C=C)C)CC1CN(C(=O)CN1CCC(C)CC1)C2 c1(C(=O)NCCN(CCC)C(C2CN(C)CC2C)=O)ccnc2ccsc12 N1(C(C=CSC)=O)CC2CCN(C(c3cn(C)c4ncccc34)=O)C(C2)C1 N1(C(c2cc(C)c(F)cc2)C(=O)NCC(C)C)CC=CCC12CCOCC2 n1(CC(=O)NC(C)C(C)NC(=O)CNC=O)cc(CO)nn1 CC(C)C(C)(CNC(C1CC2CCC1C2)=O)NC(=O)Cn1cc(C(F)(F)F)nn1 C1(C2CC2)(C(=O)NC(C2COCCN2C(=O)CC2(O)CCCCC2)C)CCC1 C=C1COc2c(C(=O)NCC(C3CCCC3)NC(c3sccc3C)=O)cnn2C1 C1(C(=O)OCC)CCc2nc(NC(C3(C)CC(COC)C3)=O)sc2C1 CC1CC=C(C(=O)NCC(Cc2ccccc2)NC(C2CCOC(C)C2)=O)CC1 Cc1ccccc1C(C(C)(C)C)NC(c1ccccc1OCC(N)=O)=O c1(NCC(C)(C)CC2CCOCC2)ncc(C(=O)OC(COC)C2CC2)[nH]1 C(=O)(C(C)(C)C(=O)NC(CCN(C)C(C1Cc2nccn2C1)=O)C(C)C)OC CCCCC(CNC(=O)Cc1nncn1C)NC(c1cn(CC2CCC2)nn1)=O CCCC(C)(O)CC(=O)NC1CC2(C1)CC(C(N1CCOC(C)CC1)=O)C2 N1(C(C2C(NC(C3N(C)CC(O)C3)=O)COC2)=O)CCn2ncnc2C1 C(=O)(C(C)(O)CCC)N1CC(CCC)C(NC(c2c(C)nsc2C)=O)C1 c1(OCc2cn(C3CC4(C(=O)NC5C(OC)C(O)C5)C3C4)nn2)cnn(C)c1C#N C1(C)(CNC(CCCC)=O)CCN(C(=O)C(N2CCC(O)CC2)C)C1 C1(NC(C(C=C)C)=O)CC2CC(C1)CN(C(=O)CCc1cccc(C)c1)C2 Cc1ccc(C)c(C(=O)NC2CCC(NC(c3[nH]c(=N)sc3C(F)F)=O)CC2)n1 CC1CCN(C(c2nc(C3CC3)cs2)=O)CC1NC(c1ccc(C(C)(C)C)[nH]1)=O c1(C(=O)NC2C(NC(C(C(CC)C)O)=O)CC(F)(F)C2)cc(F)cc(Cl)c1O Cc1nn(C)c(=O)c(C(N2CC3(C2)C(NC(=O)CCCF)CCS3(=O)=O)=O)c1C C(=O)(C(O)C(C)(C)C)NCc1c(CNC(C(C)c2cc[nH]n2)=O)cccn1 CC(C)CC(C(=O)NC(C)(C(=O)NCc1cc(=O)cc[nH]1)C1CCCO1)C(C)C C1(OC)CC2CC(C(N3CC(NC(=O)C(F)(F)CN4CCCC4)C3)=O)CC12 N1(C(CC2CN(C(C)=O)C2)=O)CCCC(C(C)C(=O)NCCN=[N+]=[N-])C1 CC(C)C(O)CC(=O)N(C(C)(C(=O)N1CCC(CC(F)F)C1)C1CC1)C c1(C(N2C(C(=O)N=c3[nH]onc3C3CC3)CC(F)C2)=O)c[nH]c2cccc(F)c12 C1(C(=O)N(C2CC=CCO2)C2CCCC2)C2CN(C(=O)C=CCO)CC12 C12(NC(c3cc(OCC)cc(F)c3)=O)CCN(C(=O)COC)CCC1C2 C1(C(N2CC(CNC(C(CC)(C)OC)=O)(OC)C2)=O)CC2(C1)CC2(F)F Cc1cnc2n1C(C(=O)N(CC(O)CNC(=O)CSCC(C)C)C)CCC2 c1(C(=O)NCC2(O)CN(C(C3CC34CCOCC4)=O)C2)c[nH]c2ncccc12 C(CCC(=C)Br)SCC(=O)C(=O)OC.C#CCOCCN(C)CCN c1(N(C)Cc2cc(F)c(Cl)cc2F)ncc(S(=O)(=O)NCC(O)CF)cc1Cl C12(NC(CCNS(CC)(=O)=O)=O)CCCN(C(c3cc(O)ccc3F)=O)CC1C2 C(CCN=c1nc(SC)cc(SC)[nH]1)N(C(C(C(CC)CC)C)=O)CC C1(C(N(C)CCNC(c2cccs2)=O)=O)CCN2CCOCC12 N#CC1CCC(CC(=O)NCC2(F)CNOC2)C1 C(=O)(C(C)(C)CN1CCOCC1)NCC(CC)(C)NC(c1ccn(C)c1C)=O C=CCC(C(=O)N1CCC(CCC(N2CCC3CCC23)=O)C1)NC(C)=O C1(C(=O)NC2CC(CCNC(c3cc(CSC)c(C)o3)=O)C2)(CC)CCNC1=O C(=O)(C1=NOCC1)N(CC(C)CNC(C1CC(n2cnnc2)C1)=O)CC c1(C(N(CC(=O)NCCN(CCCC)C)CCC)=O)sccc1Cl C=CC1CN(C(=O)C(c2cc(Cl)cc(Cl)c2)=O)CC1NC(=O)C1=CCOCC1 c1(C(=O)NC2(C)CC(NC(C3CC(=C)C3)=O)C2)ccc(C)c(S(=O)(=O)N(C)C)c1 C#CCC(CC(=O)NC(c1cnsc1)C)NC(=O)C(C)=C(C)CC N1(C(=O)NC(c2cc(C)[nH]n2)CC)C2CCC1CC(F)C2 C1(CNC(CN(C2CCC2)C)=O)CC(C)(C)CN1C(C1CS(=O)(=O)C1)=O C1(NC(C2CCN(C(C)=O)C2)=O)COCCN(C(=O)CCS(C)(=O)=O)C1 Cc1ccc2n[nH]cc2c1C(=O)NC(CNC(=O)CC1CCCC1(F)F)CO N1(C(C(=O)NC2C(COC)C2)=O)CCCc2sccc2C1 N1(c2nccc(-c3onc(C)n3)c2)CCCC(C(=O)NC(C)CO)CC1 C1(NC(c2cc(C)cc(O)n2)=O)CCCCCN(C(=O)CN2CCS(=O)CC2)C1 Cc1cc(C(=O)NCC2CCC(C)CN2C(c2cc(Cl)no2)=O)ccc1F N1(C(N2CC(c3ccccc3Br)(C)C2)=O)CCCNCC1.C1CC1 C1(C(N2C(CCNC(C3CC3(Cl)Cl)=O)CSCC2)=O)COC2COCC12 c1(C(=O)NC(C)CCN(C(=O)CC2(C(F)(F)F)CC2)C)ccsc1Cl c1(CC(=O)NCC2(C(C)NC(=O)CCc3cnccn3)CC2)cnnn1C CC1CCCC1(C(=O)N(C)C1CC1)NC(=O)CC1(NC2(N(C)C)CC2)CC1 C1(O)(CCNC(c2cc(CF)on2)=O)CCCN(C(C2COCCC2(F)F)=O)C1 c1(C(N2CCC(CC#N)C2)=O)csc2c(F)cccc12 N1(C(=O)Cc2ccc(C#N)s2)CCC2(C=Cc3ccccc32)CC1.C1(=O)CO1 C(C1CCOC1)=CC(=O)NC1C(NC(C(C2CC2)OCC)=O)C1 S(=O)(=O)(c1cn(C)nc1C)Nc1ccc(C(=O)Nc2c(C)ccc(Br)c2)nc1 C(=O)(CC(C)(C)CCOC)N1CC(CCNC(c2c(CC)[nH]c(=N)s2)=O)C1 C1(CCC(N2CCCC2Cn2cc(C3C4CCC34C3CC3)nn2)=O)CCCCC1 C#CCCCCCC(C(=O)NC1CCOCC1)N1CC2CCC1C(O)C2O N1(C(C2CC(CCC)C2)=O)CC=CC(NC(c2cc(-c3cnn(C)c3)no2)=O)C1 c1(Oc2cc(O)ccc2O)c(-c2ccc(OC)c([N+](=O)[O-])c2)ccc2c1OCO2 c1(CC(=O)NC(CC)(C)CNC(C2CC(COC)C2(C)C)=O)ccc(Cl)cc1Cl C1(C(N2CCC(CCNC(CC(C)(C)F)=O)CC2)=O)Cc2nncn2C1 C#CCC(CC(=O)NCc1coc(COC)n1)NC(=O)CC1(C)CCOC1 C1(COC)CN(C(=O)CC2(C)CCC2)CCN1C(c1cc(C(F)F)cc(Cl)c1)=O C1(CC(C)C)(C(=O)NC2C=CC(C(N3CCC(C(C)(C)C)C3)=O)C2)CC(=O)C1 Cc1cc(F)c(CN2CCC(C(=O)NCc3cnc(Br)c(F)c3)C(O)C2)c(F)c1 Cc1ccc2sc(C(N3CCCC3CNC(C3CCCSS3)=O)=O)c(C)c2c1 c1(SC)cccc(C(=O)NCC2CCC(C(=O)Nc3ncccc3O)CC2)c1O CCC(CCC(=O)N1CCC(C)(C(=O)NCc2cc(C)cc(C)c2)CC1)OC C1(C(=O)NCC=CCNC(CCN(CCCCC)C)=O)CNC(=O)N1 C1(C2CCC2)(CNC(CC(C)C)c2nnnn2-c2ccccc2)CCC1 N1(C(COCC)=O)C2CCC1CC(CNC(=O)CC1(C)CCOC1)C2 c1(C(C2CC2)NC(=O)NCC2CN(C(C)(C)C)C(=O)C2)cc(F)ncc1Br O=S1(=O)CCCN1c1ccc(-n2cc(C3CCCCC3)nn2)cc1 C1(CC)(NC(c2cc(O)cc(=O)o2)=O)CCN(C(=O)C(CC)n2cncn2)CC1 C(=O)(CCCCCc1cccs1)NCC1C2CN(C(C(C(C)SC)O)=O)C1C2 CC(CCNC(=O)NCC=C1CCSCC1)C(C)(C)C c1(CCC(=O)N2CC(C(C)NC(=O)CCOC3CCC3CF)C2)ccncc1 CCC(C)CC(C)SCc1cnn(-c2ccccc2F)c1 C1(NC(CN(C)C(=O)C2CC2)=O)CCCCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1 C(C(CO)(CO)NC(c1cc(OC)cs1)=O)N(C(C1(C(=O)OC)CC1C)=O)C N1(C(CN2CCC(C)C2)=O)CCC(O)CC1C(=O)NCC1(O)CCCCCC1 CCCCC(CC)CC(CNC(=O)OCC)CC.C1CCOC1.CC O=C1CN(C(=O)C2=C(F)CNC2)c2ccccc2N1.N1CCc2ncccc2C1=O C1(C(N2C(C3(NC(C4C(=O)NCC4)=O)CC3)CCC2)=O)Cc2cccnc2C1 CN1N=C(C(=O)N2CCC(C(=O)NCCn3ncnn3)C2C2CC2)CCC1=O c1(NC(C)=O)cccc(C(C)NC2CCOC(c3ccccn3)C2)c1 c1(N(C)C)ccc(Br)cc1CNC1CCC(CNC(=O)C(C)OC(C)(C)C)C1 N1(C(c2cccc(OC)c2)=O)CCC(C)(Nc2cnc(C)c(F)c2)CC1 C1(C(N2CC(c3ccco3)C2)=O)CCC2CCC1N2C(C1CC1Cl)=O C1(N(C)Cc2csc(-c3ccccc3)n2)C2CN(C(=O)OC(C)(C)C)CC12 Cc1[nH]nc(C(N2CCC(C(C)NC(=O)COC3CC3(F)F)C2)=O)c1O C1(CC(=O)NCC2C(NC(=O)COCC3CCOC3)C2)C=CS(=O)(=O)C1 N1(C(C2C(C)C2)=O)CCC(F)C(NC(c2ccc(CCF)cc2)=O)C1 C1(C(=O)NCC(CNC(C(C)(C)F)=O)CO)CCC2(CCC2)CC1 N1(C(Cc2c(C)cccc2)=O)CC(F)(F)CC1CNC(=O)C(O)CC(N)=O CC1(C)CC(CNC(=O)CCCC2CCC2)CN1C(c1c[nH]cc(Cl)c1=O)=O c1(C(N2CC3C(C2)N3C(C2CCC(F)(F)C2)=O)=O)cccc([N+](=O)[O-])c1O CC1COCCCN1C(C1(F)CCCN(C(C2COC(=O)N2C)=O)C1)=O Cc1cc(Cl)c(C(N2CC3CC(NC(c4ccc(F)o4)=O)C3C2)=O)cc1N C(=O)(C(C)(C)CCS(C)(=O)=O)NCC1N(C(c2nc(CC)[nH]n2)=O)CC(O)C1O c1(C(C)NCC2CC2c2ncccc2Br)ccc2nn[nH]c2c1 N1(C(C2NC(=O)OCC2)=O)CC(NC(c2cc3ccncc3[nH]2)=O)CCC(O)C1 CCCCC(O)CNC(=O)C(Cn1cccn1)NC(=O)CSC(C)C CCC(C)(C(=O)N1CC2CCC(C1)N2C(c1nccc2c[nH]nc12)=O)C(F)F N1(S(CCC)(=O)=O)Cc2[nH][nH]c(=NC(=O)c3cnnc(O)c3)c2C1 C12(C(=O)NCC(C)CN(C(=O)C(c3ccc(C#N)cc3)O)C)CCC(C)(CO1)C2 c1(C(=O)NCC2C(NC(C3CC(C)(C)OCC3)=O)COC2)cc(F)cc(N)c1F N1(C(c2cc(OC)ncc2)=O)CC2CCC(C1)C(NC(C1CC13CCCC3)=O)C2 C(=O)(C(Cc1ccccc1)C(F)(F)F)NC1C(NC(CCSC)=O)C1 c1(C(=O)NCCC2CC(NC(c3nc(COC)oc3)=O)C2)cccc(Br)c1 c1(C(=O)OCCSC)cc(Br)c(F)cc1F.C(=O)(N1CCNCC1)NCC C(=O)(C1CCc2nnc(C)n21)N1CCC(NC(c2ccc(SC)cc2)=O)C1(C)C Cc1cc(-c2cn(CCC3CN(C(=O)CCN4CCC4)C3)nn2)ccn1 c1(-c2cccc(C)n2)cc(C(N2CC(OC)C(NC(=O)CS(C)(=O)=O)C2)=O)sc1C C=C(C)CCCC(=O)N(CC(C)NC(=O)C=Cc1ccc(Br)cc1)C CC(CNC(C1CCC1(F)F)=O)CC(=O)NC(C)(C)C(=O)N(C)C Cc1cn2c(n1)CCC(CN=c1[nH]c(C)c(-c3ccccc3)o1)C2 N1(C(C(c2c(OC)cccc2)=O)=O)CC2CC1CN2Cc1ccns1 C12(CC(=O)NCCC(C)CCNC(C3(C)CC(F)(F)C3)=O)CCC(CC1)C2(C)C n1(CC(N2CC3C(CNC(c4ncn(C)n4)=O)(C3)C2)=O)ccc(O)nc1=O c1(OC)ccccc1C(=O)NC(C1CCN(C(=O)Nc2ccc(CO)cc2)C1)C Cc1ccc(Br)c(-n2cc(CONC(c3cc(Cl)cnn3)=O)nn2)c1 N1(C(c2nc(C)nc(O)c2)=O)CCCC(C2CCN(C(c3ncsc3Cl)=O)C2)C1 C#CC1CN(C(=O)C(C)C(C)O)CCN1C(=O)Cc1cc(F)ccc1Cl C(N=c1[nH]c(Cl)nc2ccccc12)C1C(NC(c2cncs2)=O)CCCC1 C(CN=c1[nH]c2c(c(=NCc3cscc3C)[nH]1)SCC2)(S(C)=O)OC c1(C(=O)NCCNC(COC(CC)(C)C)=O)cncc(NC(C)C)n1 N1(C(C(c2scc(C)n2)(F)F)=O)CCC2C(NC(c3coc(C)n3)=O)C2CC1 N(C(=NCC1CCC1)N(C)CC1CCOC1)CC1(C#C)CCC1 C(=O)(C1CCc2c[nH]nc21)N(C)CC1COCCN1C(C1CCC1C(C)(C)C)=O c1(C(=O)NC(C)CN(C)C(c2nccc(Cl)c2F)=O)ccn2c1CS(=O)(=O)CC2 N1(C(C2(F)CCN(C(Cc3c(C)nn(C)c3C)=O)C2)=O)CCc2cccc(C)c21 C1(C(N2C3(C(=O)NC(C#C)CC)CC(C2)C3)=O)CC2CCCC2C1 C(=O)(C(F)(F)CC(C)C)NCC(CC)(CC)NC(=O)Cc1cnco1 N1(C(C(C)OCCOC)=O)CCN(CCCCCNC(C2(COC)CC2)=O)CC1 C(C(O)C(F)(F)F)NC(c1nc(C(=O)Nc2nccs2)sc1)=O C1(C(N(CC(=O)OC)CC)=O)CCC(O)CN1C(c1ccccc1F)=O CCC(CC(=O)NCC1CN(C(=O)CC2(C)NC(=O)NC2=O)CC1(F)F)C(C)C c1(CCC)nc(C(=O)NC2COCC2NC(=O)C(C)CN(C)C)co1 C1(C(=O)NC2CC(CNC(C(C)(F)c3ccccc3)=O)C2)Cc2ccccc2S1 C1(C(=O)NCCCN(C)C(C2CCN(CCO)C(=O)C2)=O)CC(=C(F)F)C1 CCCC(F)(F)C(=O)NCCC(N1CCC(C)C1C)=O CC(=O)CC(C)(C)C(=O)N1CC2C(C(=O)NCC(C)OCCO)C2C1 c1(C(=O)NCCCN(C(=O)CC2(O)CCOC2)CC)cccc(C(F)F)c1 C1(C(=O)NC2CC(CCNC(=O)CCc3cc(C)[nH]n3)C2)(CC)CC(F)(F)C1 O=C(CCS(=O)(=O)c1ccc(Br)cc1)NC1COCC1O c1(C(N(CC(CNC(CCCN(C(C)=O)C)=O)O)C)=O)ccc2oc(S)nc2c1 CCCCCC(CC)C(=O)N1CC(C(=O)Nc2ccc(Cl)c(F)c2)CC(C)(C)C1 c1(CCC(=O)N(CCNC(c2cncc(O)c2)=O)CC)c(F)c(F)cc(F)c1F Cc1c(C(=O)NC(C)C(C(C)C)NC(=O)C=Cc2ccc(Cl)s2)cnn1C CCCC(C(=O)N1CC(C(C(=O)N(C)CCN2CCN(C)CC2)OC)C1)OC c1(CCOCC(=O)N(C(CNC(C(C)NC(=O)NC)=O)C)C)nccn1C CC(C)CC(=O)C(=O)NCc1ccc(SC(F)F)cc1 CCCC(C)(C)CC(=O)N1CC(C)(NC(c2cc(N)nc(Cl)c2)=O)C1 c1(C(N2C(C(C)(F)F)CCC2)=O)cc(Br)c(I)s1 c1(C(=O)NC(CC(C)C)CNC(=O)C=C2CCCCC2)ccc(N)cc1Cl N1(C(C2C(OC)CN(C(c3cc(C)nc(C)c3)=O)C2)=O)CCC(C)(C2CC2)C1 c1(C(=O)NC2CC3CN(C(c4ccc(CC)cc4)=O)CC32)cc2ccccn2c1 CC(C)(C(O)CO)NC(=O)CC1CCN(C(=O)CCNC(N)=O)C1 C1(NC(C2(N(C)C(c3ccc[n+]([O-])c3)=O)CC2)=O)CCn2cncc2C1 Cc1cc(F)cnc1C(N1C2CCC(C2)C1CNC(=O)C(F)C(C)(C)O)=O c1(NC(=O)NC(CC)C(O)c2ccccc2)c2c(nn1C)CCC2 c1(SC)ccc(NNC(=O)C2CCN(c3cccc(OCC(F)F)n3)CC2)cc1 c1(CC)ncnc(CC)c1C(=O)NC(CCN(C(=O)COCCF)C)C(C)(C)C c1(C(=O)NCC(C(N2C(C(=O)NC)CCCC2)=O)OC)ccc(C)nc1C N1(C(C(c2cnn(C)c2)OC)=O)C2CCC(C2)C1CNC(c1nn[nH]c1Cl)=O N1(C(c2n(C(CC)C)ncc2)=O)CCC2(C1)CN(C(=O)C(F)=CCCF)C2 C1(C(=O)NCC2(CNC(c3ccc(Cl)o3)=O)CC2(F)F)CCC2(CC1)CC2 Cc1nn(C)c(CNc2cccc(SCc3ccccc3)c2)c1Cl c1(-c2c(C(N3Cc4n(C)cnc4CC3)=O)c(F)cnc2)c(F)ccc2[nH]ccc12 C1(C(=O)NCC2C(C(=O)NCC(C)CN3CCCC3)CC2)COCC1(C)C C1(C(N2CCC(NC(c3cc(O)ncn3)=O)C(F)C2)=O)CC1C1CCOCC1 C1(CC)CN(C(c2cnnc(-c3ccccc3)c2)=O)CCC1NC(=O)C(C)(C)C C(=O)(C(C)(C)O)NC1CC(CC(=O)N(CCC(N)=O)CC)C1 CC1CC(NC(=O)C(c2ccccc2)C)CN(C(c2ccc([N+](=O)[O-])s2)=O)C1 c1(CC(=O)NCc2cccc(NC(C(C=C)(C)C)=O)c2)ccc2c(c1)CC(=O)N2 C1(CC(=O)NCC(C)CNC(=O)CN(C)C(=O)C2CC2)CCC(F)C1 C1(O)(CC)CCCN(C(C(=O)NCCCF)C(C2CCC2)OC)C1 C(=O)(C1=NNC(=O)CC1)NC(CNC(c1c(C)nn(C)c1C(F)F)=O)(C)CO C1(CNC(COCC(=C)C)=O)CC2CCC1N2C(=O)CC1CCN(C)C1 c1(CC)nc2sc(C)cn2c1C(=O)NC1CC2CCC1(CNC(=O)COC)C2 C=CCC(CC(=O)N1CC(N(C)CC)C1)NC(CC(=O)OCC)=O.C(C)(C)O CCC(C(C)C(=O)OC)NC1(n2cnnn2)CC1 C(=O)(C1=NOC(CNC(c2occc2C(C)C)=O)C1)N1CC(C)(OCC)C1 c1(OC)nscc1C(=O)NC1CC(F)(CNC(C2CC2(C)C(F)(F)F)=O)C1 c1(OCC(=O)OCC(c2ccc(Cl)cc2)CC)ccc(C)cc1C N1(C(c2cc(NCC(F)(F)F)n(C)n2)C(=O)OCC)CCCC(O)(C(N)=O)C1 C(=O)(C(O)CC(C)(C)C)NCCC(CCNC(CC=Cc1ccc(C)cc1)=O)C N1(C(CCC(N)=O)=O)CC2CCN(C(=O)C(O)CN3CCOCC3)CC12 c1(C(=O)NCC2(NC(CCC#CC)=O)CC2)cc2c(C)ccc(Br)c2[nH]1 c1(OC)cccc2cc(C(=O)NC3CC3NC(=O)C(C)=C3CC3)c(=O)oc12 C1(CCNC(CCSCC)=O)CCN(C(C2CC2C(F)F)=O)CCC1(F)F C1(C(=O)NCC2N(C(c3ccc(C)cc3F)=O)CCC2C)CN(C)CCN(C)C1 c1(CC(N2C(CNC(C3N(CC)CC3)=O)CC3CC32)=O)cccc2ccsc12 c1(C(N2CCC(CNC(Cn3c(C)ccn3)=O)(CO)C2)=O)cnc2cc[nH]c2c1 N1(C(C(=O)NC(c2onc(COC)n2)C)=O)CCc2nn[nH]c2C1 c1(C(N2CC(N(C(C(F)OC)=O)C)C(C)(C)C2)=O)cc(O)nc2[nH]c(=N)ccc12 C1(CC(N2CC(NC(c3cnc(CC)[nH]3)=O)C(F)C2)=O)CCC2(CCC2)O1 N1(C(c2ccc([N+](=O)[O-])o2)=O)CCN(C(c2ccnc(O)c2)=O)C2CCC12 C=CC(CC)CC(=O)N1CCOC(CCNC(=O)C(F)(F)CC2CC2)C1 C1(C(=O)NCC(C2CC2)NC(C2(COC)CCCO2)=O)CN2CCCN1CC2 C(C)(C)(CC(=O)NCC(C)(C)NC(=O)C(CC#N)c1ccccc1)N(C)C C(=O)(CC(C)CNC(C1(C)CC(C)=NO1)=O)N(CC#C)C c1(SCC(=O)NCC2CN(C(CC=CC=C)=O)C3C2C3)ccc(F)c(F)c1 Cc1ccnc(O)c1C(=O)NCC(C)(C)NC(=O)C(c1cccc(Cl)c1)C C1(CO)CC(CC(=O)NC(C2CC(=C3CCC3)C2)C)C1(C)C N1(C(c2n(C)ccn2)=O)CCOCC1CCNC(=O)COCCc1cccs1 C(=O)(C(C)(C)C(F)(F)F)N1CC(C)(C)C(CNC(=O)C(F)=C2CCC2)C1 CN1CCN(C(C2CCC2C(N)=O)=O)CC1CNC(c1scnc1C(F)F)=O N1(C(CNC(CC)=O)=O)CC(NC(=O)C(=O)NC(C)C)C1 C1(C(=O)OC)CC2CN(C(=O)NC(c3ccc(C(C)C)cc3)C)CC2C1 C(=O)(C(CC(F)F)C1CCCO1)NCC1CCC(CNC(C2CN(C)C2)=O)CC1 C1(CC(=O)NCCCCCN(C(c2cc(COC)sc2)=O)C)CCCNC(=O)C1 C(c1ccc(Cl)cc1F)=CC(N1CCC(NC(C2CCC(=C)CC2)=O)C(F)C1)=O C1(C(=O)Nc2c(C(C)C)noc2)CN(C(=O)COCCC(C)C)CCO1 c1(N(CC(CC)(C)OC)C)ccc(S(=O)(=O)NCC2CCCC(F)(F)C2)cc1F c1(C(N2CCC(NC(C3ON=C(CC)C3)=O)C2(C)C)=O)cccc2c1CCC2 N1(C(Cc2ccc(C)nc2)=O)CCC(NC(c2ccc(Br)c(C)n2)=O)C(F)C1 c1(SCCn2ccc(C)n2)ncccc1C(=O)NC(CC(C)C)c1cccs1 C1(NC(c2cncc(F)n2)=O)CCCCN(C(c2sncc2Br)=O)C1 c1(C(N2CC3CC(NC(C4(C5CC5)CC4)=O)C(C3)C2)=O)cnn2c1OCCC2 C1(C#C)(C(=O)NC(C2CCCC2)C#C)CCN(C(=O)C(CC(C)(C)C)OC)CC1 C1(CC(N2C(CN(C3C4CCN3CC4)C)CCC2)=O)SC(=N)NC1=O N1(C(C(C(C)O)N(C)C)=O)CC2CC(C1)CN(C(c1cc(O)cs1)=O)C2 N1(C(Cn2c(C)nc(C)n2)=O)CCCCC(NC(=O)CN2CCS(=O)CC2)CC1 c1(CNC(C2(CC)CC=CC2)=O)ccc(C(N2CC(C#N)(SC)C2)=O)cc1 C(N=c1[nH]cnc(Cl)c1Br)C1OCCC1.c1(CN)ccc(C(=O)OC(C)(C)C)[nH]1 N1(C(C2(OC)CCCC2)=O)CCC(=CCNC(=O)C(n2cnc(C#N)n2)C)CC1 C1(C(N2CCC(C(C(=O)N(C3(CO)CCOCC3)C)F)C2)=O)CCC(F)(F)CC1 C12(C(N(CC(C)(C)CNC(C3(COC)CC3(F)F)=O)CC)=O)CCCC1C2(F)F O=C1CC(CC(=O)NC2CN(C(=O)CSc3ccccc3)C2)CCCN1 c1(CCC)ccc(C(=O)NC(C)CCCNC(=O)CC(C)C(C)C)cc1[N+](=O)[O-] C1(C)(C(=O)NCC2C(C)(C)C2C(=O)NCCSC(C)(C)C)CCCC1O C12(NC(C=CCCC)=O)CCC(CNC(c3cc(C)c(C(N)=O)o3)=O)(CC1)OC2 C1(CNC(C2C(OC)CCC2)=O)CCC(C(N2CCSC(C)C2)=O)CC1 c1(C(=O)NCCC(Cc2ccccc2)NC(C2ON=C(C)C2)=O)ccc(F)cc1 c1(C(=O)NC2CN(C(C3CCN(C)C3=O)=O)C2)cc(C(F)F)cc(C(F)(F)F)c1 C1(N(C(c2c(CC)csc2)=O)C)CN(C(C2CCCOCC2)=O)CC12CC2 N1(C(C)C)CCCC(C(=O)NCC2CC(NC(=O)C(C)(O)C3CCC3)C2)C1 Cc1cc(F)ccc1-n1cc(CONC(C2CCn3nccc3C2)=O)nn1 c1(CC(N2CCOC(CNC(=O)C(F)(F)CO)C2)=O)c(F)cccc1F Cc1cnccc1C(=O)NCCCC1CCCN1C(=O)C(C)Cc1cnn(C)c1 c1(COC)noc(C(=O)NC2CCN(C(CC)C(=O)OC(C)(C)C)CC2)c1C CC1CN(C(=O)C2=C(Cl)CC2)CCN1C(=O)CN(CC(C)(C)C)C c1(CNC(c2c(C)ncnc2)=O)cnn2c1CN(C(C13CC(CO)(C1)C3)=O)CC2 c1(C(N2C(C)CC(NC(c3ccoc3)=O)C2)=O)cc2c(nn1)CCCC2 Cc1nc(C)c(C(=O)N(C2CCN(C(C3CCOC3)=O)C2)C)o1 C1(C(=O)NC2C3CN(C(c4c(CC)con4)=O)C2C3)CC2CCC1CC2 C1(CC)C(C(=O)NCCCn2cccn2)CCCN1C(C1COCC(C)O1)=O N1(C(C(n2ncc(C)c2)C)=O)CCC(NC(C2CC3CCCC23)=O)CC1C c1(CC)cnn(CC(=O)COC2CCN(C(=O)CSCc3ccco3)C2)c1.C(C)N C(CC(O)CNC(C1(c2ccsc2)CC1)=O)NC(C1C(C(C)(F)F)C1)=O c1(C(=O)NCCCC(C)NC(C2(Cl)CC23CCC3)=O)cnc2ccoc2c1 Cc1cc(C(=O)NC2CCCC(C(=O)NC3CC4C=CC3C4)CC2)cc(C)c1 Cc1ccn2cc(C(=O)NC(C3CCN(C(=O)C(F)CC4CCC4)C3)C)nc2c1 Cc1cc(P(C)(C)=O)oc1C(=O)NC(C1CCN(C(C2(F)CC=CC2)=O)C1)C n1(CC)ncnc1CSc1cccs1.o1[nH]c(=O)o1 c1(N2CCCC(NC(C(C)(C)O)=O)C2)ncc2c(n1)NC(=O)C2 c1(CC)ncccc1C(=O)N(CC(=O)Nc1ccc(OC)cc1)CCN(C)C C1(O)(C(C)NC(C2N(C(C)=O)CSC2)=O)CCN(C(=O)C(C)(O)C2CCC2)CC1 [N-]=[N+]=NC1CC(C(=O)NCC2CCCSC2)N(C(c2ccnnc2)=O)C1 Cc1cn2cc(C(=O)NCC3(C)CCCN3c3ncc(Cl)c(O)n3)sc2n1 C1(C(=O)NCC=CCNC(C(C2CCC(C)(C)CC2)C)=O)CC(C(C)(C)C)=NO1 C(C)(C(F)(F)C(F)(F)F)NC(C(C)Oc1ccc(Cl)cc1)=O Cc1cnc(N(C)CC2CC=CCC2)c(S(=O)(=O)N2CC3CCOC3(CO)C2)c1 N1(C(c2ccco2)=O)CCC2C(CCCN2C(c2cccc3[nH]ccc23)=O)C1 c1(CNC2C(C(=O)O)CCC2)ccc2c(c1)S(=O)(=O)NC=C2 C1(N(C(c2c(SC)ccs2)=O)C)CCCN(C(=O)C(C2CC(F)(F)C2)O)C1 Cc1nc2ccc(C(N3CC4CC(C3)N4C(C3CCC(C)C3)=O)=O)cc2[nH]1 C(CC(C)C(=O)NCC(CC(C)C)NC(c1c(Cl)n[nH]c1C)=O)OC C=CCC(CCC=C)N(C(=O)C(C=C)CC)c1ccccc1 C1(CC(=O)NCC2(C)N=C(C)SC2)CC2(C1)CN(C(=O)C(F)F)C2 C1(C)(C(N(CCCCCC=C)C)=O)CCCN(C(=O)C(C(C)C)NC(C)=O)C1 c1(C(=O)NC(C2N(C(C(C(=O)OC)C)=O)CCC2)C)nn(C)c(Br)c1C CS(=O)(=O)c1ccc(C2CCC(C(=O)OCCCCCCCCCCO)C2)cc1 Cc1coc(C)c1NC(C1(NC(=O)COCCF)CC(O)C1)=O CC1CN(C(C2(O)CCCC2)=O)CC(C)CN1c1cc(O)ncn1 N1(C(C(CCOCCO)NC(Cc2c(C)n[nH]c2)=O)=O)CCOC(C)(C)CC1 N1(c2nccc(=N)[nH]2)CCC2(CC1)CC2C(N1CC2C(C(=O)O)C2C1)=O c1(CC)cc(C)ccc1C(=O)NC(CNC(=O)C=CCN1CCOCC1)(CC)CC C(CNC(=O)CCC1CCCO1)(C(=O)N(C)Cc1ncco1)OC N1(C(CCN(CC)CC)=O)CCC2CCN(C(c3cnc(C(C)C)[nH]3)=O)CC12 c1(C(=O)NCCOC2CN(C(c3ccn(C)c3)=O)C2)cncc(P(C)(C)=O)c1 C12(NC(C(C(C)C)OC)=O)CCC(C(=O)N(CCCCCCO)C)(CC1)C2 c1(C(=O)NCC(CC=C)NC(=O)C(C)CCOC)ccc(Cc2nc[nH]n2)cc1 C1(O)(C(=O)NC2C(NC(C(C)(C)SC)=O)CCOC2)CCc2ccccc2C1 c1(C(=O)NCCCCCNC(C(C)C(F)F)=O)cc(N)c2ncccc2c1 C=C(C)C1OCCC1C(=O)NCC1CCCCCN1C(=O)CC(=O)NCC Cc1cc(C(c2nnnn2C2CCOCC2)N(CC(C)(C)C2CC2)C)cc(C)c1 C1(OC)CCC2(C(=O)NCC(C)C(=O)NCCC(C)N3CCC3)CC12 C1(CNC(C(C)OCCOC)=O)CN(C(c2ccc(C3(C)CC3)cc2)=O)CCO1 C1(NC(Cc2c(C)con2)=O)CCN(C(c2nnsc2C)=O)C(C)C1 c1(C(=O)NC2CCCN(C(CCCN=[N+]=[N-])=O)C2)n[nH]c2ccc(Cl)cc12 N1(C(C(C)(N(C(CCC(C)OCC)=O)C)C2CC2)=O)Cc2nncn2C(C)C1 S(=O)(=O)(c1ccc2c(c1)OCCO2)C(CC(=O)N(C1CCC2(OC)CC12)C)N(C)C C1(=O)C2=CC(O)C(C2)C2CCN12.C(=O)(C1=C(C#N)CCC1)NC1CCCN(C)C1 CC1CC(NC(c2cccc(=O)n2C)=O)CCN1C(c1cc(F)c[nH]1)=O N1(C(C(F)=CCC)=O)CCC(C(=O)OC)(CO)C1.c12oc(cc1C)c(=O)[nH]2 C1(C(=O)NCC2C(NC(c3c(C)nco3)=O)COC2)CC(O)CN1C c1(CC(=O)NC2CCCC(NC(C3(O)CC(C)(C)C3)=O)C2)cc(O)nc(O)n1 Cc1nn2ncccc2c1C(N1CC2CCC(C1)N2C(=O)CN1CCC(C)C1)=O C1(CNC(c2n(C(C)C)ncc2Cl)=O)COC(C)(C)CN1C(=O)Cc1cscn1 C1(C(N(C)Cc2nnc(C)s2)=O)CC(C)N(C(c2nccn2C)=O)C1 N1(C(CC2CCC(C)C2)=O)CCC2(CCCN(C(c3cnc[nH]c3=N)=O)C2)C1 O=C1CN(C(c2ccc(CO)s2)=O)C(C(=O)NCCCc2ncc[nH]2)CN1 Cc1cccc(Cl)c1CC(=O)Nc1cccc(CNC(=O)C(C)CF)c1 c1(C(N(C2CC(NC(=O)Cn3cnnc3O)C2)C)=O)c(OC(F)F)cccc1Br C(=O)(C(F)C(F)(F)F)N(C(C(=O)N(C1CN(C)C1)C)C1CC1)C c1(C2(C)CC2C(=O)NCCNC(C2CCC(CN3CCOCC3)O2)=O)ccccc1 C1(NC(C2CCC(=O)N2)=O)CC2CN(C(=O)CCc3nc[nH]n3)CC12 N1(C(C)C)CC(NC(=O)CN(CCCC(=O)Nc2cc[nH]n2)C)CC1=O C1(C(=O)NCC(CNC(CCN(c2ccncc2)C)=O)F)COC2(CCC2)CO1 c1(C(=O)NC2CC(C(=O)Nc3cccc(OC)c3)C2)ccc(C)cc1Cl c1(OC)ccc(CC(=O)NC(C2CCN(C(C3CC(=C(F)F)C3)=O)C2)C)c(Cl)c1 C1(C(=O)NCC(C2CCC2)Nc2ncc(C#C)cn2)CCC2(CCC2)CC1 C(=O)(C(CC1CC1)OC(C1(COC=O)CCCC1)=O)OC(C)(C)C.C(C)(C)(C)O c1(OC(C)C)ccc(Cl)cc1C(=O)NCC1CCN(C(c2cn[nH]c2)=O)C1(C)C n1(CCC)ccc(=NC(=O)C2CC3CCC(C2)N3C(=O)CC2CCCOC2)[nH]1 c1(NC(C2CC2CNC(c2ccc(N(C)C)cc2)=O)=O)ccc2ncsc2c1Br c1(CC(=O)NCC2(C(C)(C)O)CN(C(C3C(C)OCC3)=O)C2)ccc(N)cc1 c1(C(N(CCOCCNC(C2C(OCC)CC2)=O)C)=O)c[nH]ccc1=O C1(C(=O)NC2(C(N(C)C)=O)CC2)CC2(CCN1C(=O)C#CC1CCC1)CC2 C1(N(C(=O)CC2CC2(Cl)Cl)CC)CCCN(C(=O)C=C(C)CCc2ccccc2)C1 Cn1cc2c(n1)CCC(C(=O)NC1(CF)CCN(C(=O)CCc3cncs3)C1)C2 N1(C(c2c(C)ocn2)=O)CCC2(CC1)CC2CNC(C1(O)CCOC1)=O CON(CCC(=O)N1CCOC(C)(C)C1)C(=O)c1cccn(C)c1=O c1(C(N2CCC(COC(C34CCC(OC)C3C4)=O)C23CC3)=O)ccccc1[N+](=O)[O-] c1(OCC(=O)NC(c2c(C)cc(Br)cc2)C)cc(Cl)c(Cl)cc1Cl C1(C(=O)OCC)CC2(C(=O)NC3CC(CCS(C)(=O)=O)C3)CC1C2 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CC(C1)N(C(=O)CN1CCS(=O)CC1)C2 O=C1CCC(CNC(=O)CC2CC(O)CN2C(=O)Cc2ccoc2)CN1 C(=O)(C(F)(F)C(F)F)NC1CC(N(C(C(c2cccc(O)n2)C)=O)C)C1 CCC(CC(C)C)C(=O)N1CCC2C(C1)CN2C(c1cncc(C)c1)=O c1(CN(C(=O)CC(C)C(=O)OC)CC(=O)OC)ccc(-c2cncnc2)cc1F c1(C(N(CC(C)N(C(CCNC(COC)=O)=O)C)C)=O)nccc(Cl)c1O C12CCC(CC1)C(=O)N2.c1(CCN(C(=O)OC(C)(C)C)CC)ccc(O)cc1 C1(CNC(C2(CCOC)CCC2)=O)CC2(CC2)CN1C(=O)CCc1cc(C)no1 Cc1nc2c(s1)C(N(C)C(C(C)(C)C)=O)CCC2.C(CC(O)C(=O)OC)NC1CC1 Cn1ncc2nc[nH]c(=NC3CCCN(C(C4(c5cccs5)CC4(C)C)=O)C3)c12 C(=O)(C(=O)C(C)CC)NC1CC(SCCn2cc(C(C)OC)nn2)C1 c1(CC(=O)NC2CC(N(C(=O)CN3CCC(O)CC3)C)C2)cn2ccccc2n1 CCCC(CC)CC(=O)N(C1CN(C(=O)COC2CCC(F)(F)CC2)C1)C C1(N(c2cn[nH]c2)C(C2CCCO2)=O)CCCC12CCNCC2 c1(C(=O)NC2CN(C(C3(OCC)CCS(=O)(=O)C3)=O)C2)cc2nn[nH]c2cc1F c1(C(N2CCC(N(C(=O)CC3CC4(COC4)C3)CCO)C2)=O)cccc2cnnn12 C(CC(C)C)(C(=O)NCc1nc(CNC(C2CCCC3CC23)=O)cs1)OC C=C1CC(N=c2[nH]c(=NC(CCC)CCO)[nH]c3ncn(C(C)C)c23)C1 C1(NC(=O)CN2CC3CC3C2)C=CCN(C(C2(c3ccccc3)CC2)=O)C1 N1(C(C(CC)n2cccn2)=O)CCC(C(O)CNC(C2CCC23CCC3)=O)CC1 C1(CNC(NCC(C(F)(F)F)OCC)=NCC2CCC2)CCCOC1(C)C c1(C(=O)NC(CNC(CC2CC(OC)C2)=O)C)ccc(CF)cc1 C1(C(N(CCCC(F)(F)F)C)=O)CC(F)CCN1C(=O)CCCCCF C1(CC(=O)N(CCOC(C)(C)CNC(=O)CCOC2CC2)C)CC(F)(F)C1 C1(CCNC(C=CCC)=O)CN(C(c2cc(N)ccc2Cl)=O)CCS1(=O)=O c1(C(=O)NCCCN(C)C(c2cnc(-c3cccs3)o2)=O)ccc(C#N)cn1 Cc1cc(=NC(C)c2nncs2)[nH]c(=NCc2cnc(C(F)(F)F)s2)[nH]1 CC1(C)CCC(CC(=O)NCC2(F)CC(CNC(C3(C)CCC(=O)N3)=O)C2)CC1 c1(OC)ccc(OC)c(CC(N2CCN(C(=O)C(O)C(C)C)CC2C(F)F)=O)c1 Cc1cc(F)cc(C(N2CCC(CNC(=O)CCCc3nccs3)C2)=O)c1C N1(C(C=C(C)C(F)F)=O)CCC(F)C(NC(=O)C2=COCC2)C1 S(=O)(=O)(c1ccc(F)cc1)N1C(C(N2CCCN(C(=O)C(F)(F)F)CC2)=O)CCC1 c1(CC(=O)NCC2C=CCN2C(C2CCCSC2)=O)ccc(F)cc1Br c1(-n2cc(CCN(C(C(C(=C)Cl)(C)C)=O)C)nn2)ccc(S(N)(=O)=O)cc1 c1(C(=O)NC(CC)CN(C(=O)Cc2cnns2)CC)coc2c(C)cccc12 C1(F)(C(N(CCN(C(C(C)CSCc2cccnc2)=O)C)C)=O)CC2(CCC2)C1 CC1CCn2ncc(C(=O)NCC3CC(F)CN3C(=O)C#CC3CCCO3)c2C1 c1(C(N(CCC)CCNC(c2nc(C3CC3)cs2)=O)=O)ccc(O)c([N+](=O)[O-])c1 c1(C(=O)NC2C(OCC)CN(C(=O)COCCSC)C2)ccc2[nH]ccc2c1F N1(C(c2cc(-n3ccnc3)no2)=O)CCOCC1c1cn(CC2CCCO2)nn1 N1(C(C(C)C(C)O)=O)CCC(F)(F)C(CNC(=O)CC2CCCCN2C)C1 CCC(CC)(CCNC(=O)CC(C)(C)C)NC(=O)C(O)Cc1cnc[nH]1 c1(C(=O)NC2C(C)CN(C(c3ccc(Cl)c(F)c3)=O)C2)ccc2c(c1)NC(=O)C2 c1(CN2CCCC(C(C)NC(c3c(C)cccc3C)=O)C2)ccc(Cl)c(C#N)n1 S(=O)(=O)(CCC(=O)NCC1C(C)CCCN1C(=O)C(C1CCC(=O)N1)C)NC Cc1ncc2c(n1)CCC(C(N1CCCC(O)(c3ccccc3)CC1)=O)C2 C(c1ccc(C)nc1)=CC(=O)NC(COC)C1(C)CC1 Cc1cc(C(N2CCC(CNC(C34CCC3C4)=O)CC2)=O)cn(C)c1=O c1(CC)c[nH]cc1C(N1CC(N(C)C(c2cc(C(C)C)[nH]n2)=O)C1)=O N1(C(CC=C)=O)CC2CCC(C(=O)NCC(C(C)C)C(C)C)(C2)C1 C1(C#N)(C(=O)NCC(=O)NC(C(C)SC)C)CCOC1 CC(C)C(C)CC(=O)NCc1ccc(C(=O)NC2CC(=O)N(C3CC3)C2)cc1 N1(Cc2cn(CCC(=O)NCC(C(C)c3cnccn3)O)nn2)CC(NC)C(C)C1 c1(CC)cncc(C(=O)NC2CC(OCC(=O)NC(C)(CC)C(N)=O)C2)c1 N1(C(C(C)SCC)=O)CCC2CCN(C(C3CCOC4(CCCC4)C3)=O)CC12 c1(CN2CCC(CNC(c3nn(C)c(O)c3)=O)C2)ccc(F)c(S(C)(=O)=O)c1 C1(NC(C2(O)CCC2)=O)CN(C(=O)C=CCN2CCC2)CC1F c1(CC(N2CC(NC(C3C(C)(C(F)F)C3)=O)C2)=O)cc(C(F)(F)F)co1 C(C(C(=O)NCC(C(=O)N1CCC(OCC(N)=O)C1)N(C)C)N(C)C)N(C)C c1(C(N2C(CC)CN(C(=O)CCC(C)C)CC2)=O)cnc2ncn(C)c2c1 S1(=O)(=O)c2cccc(c2)N1C.c1(NC(=O)C(=O)NCCO)ccc(C#N)nc1Br C1(C(=O)NC(C(N2CC(COC)C2)=O)c2ccco2)CC(C)(C)CCO1 c1(N(C)C)ccncc1-c1nc(-c2cnn(C)c2)nn1CCF c1(C(N(C2CCCN(C(=O)C(C)(C)C3CCCO3)C2)CC)=O)cn(C)nc1O c1(CNC(=NCCF)NC2CCN(CC3CCCC3)C2)cccc2c1OCC2 C(=O)(C1=CCC(NC(c2cccc(=O)o2)=O)C1)NC1CC(C(=O)OC)OCC1 c12ncc(Br)nc1O2.c1(CNC(=O)NC)ccc(OC2CCC2)nc1 S(=O)(=O)(c1ccc(NC2CC(C(=O)NC)C2)c(F)c1)N(CC)Cc1ccncc1 C1(C(=O)NC2CCN(C(C(C(C)OC)N(C)C)=O)CC2)C2CCC(F)(F)C12 N1(C(CN(C)C(C2(CC(C)=O)CCCC2)=O)=O)CCN(C(c2cnccn2)=O)CC1 Cc1cccc(F)c1C(=O)NCC1CC(C)N(C(=O)Cn2ccnn2)C1 CCCS(=O)(=O)NC1CCC1(c1nnnn1C)NCCS(=O)(=O)NC N(C(=NCCC1(C)OCCO1)NC1CC(c2ccc(C)cc2C)C1)CC(O)SC C(=O)(C1=C(C)N(C)c2ncnn2C1)N1CCCC(NC(C(C)(C)OCC)=O)C1 c1(CN2CC3N(C(c4cncc(C(F)(F)F)c4)=O)C3C2)cc(O)nc(C2CC2)n1 C1(C(N(C(c2cn(-c3cccc(C)c3N)nn2)C)C)=O)CN(C)C(=O)CCO1 C1(C)(C(=O)NCc2ccc(C)nc2)CCCN(C(=O)CN2CCCC2)C1 c1(C(=O)OCC)ccc(C2CC2)cc1.C1(=O)C(CN(C)C)N(C)C(C)CCCN1 c1(CN(C(=O)OCCOC)C)cccc(OC)c1.c12ccccc1CS2 C(=O)(C(CC(C)C)N(C)C(C1CC(OC(F)(F)F)C1)=O)N(CCOC)C(C)C C(=O)(C(C)(C)C(O)C(C)C)NC1CCN(C(c2n(C)nc(C)c2Br)=O)C1 Cc1cc(C(=O)NC(C2CCOC2)CNC(c2ccnnc2O)=O)cc(C)c1F N1(C(C(C)c2ccco2)=O)CC(C)(NC(=O)C(F)Cc2ccccc2)C1 c1(CC)ccc(C(=O)N(C)Cc2ccccc2Sc2n[nH]c(C)n2)nc1 c1(C(=O)OCC)ccc(NCC(C)CNC(=O)Cc2ccoc2)nc1 [N-]=[N+]=NCCCCNC(c1csc(CNC(=O)C(O)C2CC2)c1)=O N1(C(c2ccn(CC)c2C)=O)CCCC(C2CC2NC(c2ccc(F)s2)=O)C1 c1(N2CC3(C(NC(C4N(C)C(=O)CC4)=O)CCS3)C2)nc(Cl)nc2ccccc12 C1(N2CCN(c3cc(C)[nH]c(=N)n3)CC2)CCC2(CCOCC2)N1 c1(C(N2C(CNC(c3[nH]cc(CC)c3)=O)CCC2)=O)nccc(C(F)(F)F)n1 N1(C(CCC(C)N)=O)CC2OCCN(Cc3ccccc3)C2C1 N1(c2nccc(SC)n2)CC2CCCC(NC(C3CCC(O)CC3)=O)C2C1 CC1(C(=O)NC(CNC(c2ncc(F)cc2N)=O)C2CC2)CCCCC1(F)F C1(CNC(c2c(F)ccc(C)c2)=O)CN(C(C23CC(C#N)(C2)C3)=O)C2(CCC2)C1 C12(NC(CC(C)(C)O)=O)CCOCC1CN(C(c1ccnc(F)c1O)=O)C2 c1(OC)csc(C(=O)NC(C)CC2CN(C(c3cc[nH]c3)=O)C2)c1OC C1(NC(c2c(OC)n[nH]c2)=O)CN(C(c2ccnn2C(C)C)=O)C(C)(C)C1 N1(C(CCCNC(=O)OC)=O)CCCCC1C(C)(C)CN.C(=O)(C(F)F)N n1(CC)c(N2CCC(c3ccnc(O)c3)CC2)nnc1C1(O)CCOC1 N1(C(C2C(CCOC)C2)=O)CCC(C)(C(=O)N(C)Cc2ccsc2)C1 c1(C(N(C2CCCN(C(C3C(C)C3C)=O)C2)CC)=O)ccncc1Br c1(C(N2C(CNC(CCNC(COC)=O)=O)CCC2)=O)cc(F)c(O)c(F)c1 CC1CN(C(C2(NC(=O)Cc3nc(=N)[nH][nH]3)CCC(C)(C)C2)=O)CC2(CCC2)O1 C(=O)(C(C)(C)C(=O)OC)NC(CN(C(CCCC=C)=O)CC)C c1(C(N(C(C)CNC(=O)C(O)CC2CCCCC2)C)=O)ccc2c(c1)OCO2 S(=O)(=O)(c1ccccc1C1(C)Nc2ccccc21)NC1CCN(C)C1 c1(OC)cncc(C(=O)NC2CCCC2(C)NC(=O)CSCC(=O)OC)c1C C1(OCCNC(=O)Cc2cscn2)CCN(C(c2cnc(-c3ccsc3)s2)=O)C1 CC1(C)C(C)(C(N2CCOC(CNC(=O)CC3CCC(=O)N3)C2)=O)C1(C)C C1(NC(C2C(C)C2C)=O)CN(C(c2cc(F)c(Cl)cc2Cl)=O)Cc2nccn2C1 CCCC(CC)CCC(=O)NC1(CNC(c2ncoc2COC)=O)CCC1 CC(C)C(F)(CNC(=O)C(C)(C)C(C)(C)C)C(=O)NC(C)CS(N)(=O)=O N1(CCC(N2CCC(N(C(=O)CCC3CCCCC3)C)C2)=O)CCCCC1=O C1(OC)CCCCC1.C12(CCC1)CC(=O)OCC(=O)N(CC)CCC(C)NC2=O C(=O)(C1Cc2ccccc21)N1CC(=O)NCC1C(=O)NCc1ccnc(Cl)c1 N1(C(COCCC)=O)CCN(CC(C)(C)NC(C2CC2C)=O)CC1 c1(C(=O)NCC(C)CNC(c2coc(C3CCC3)n2)=O)ncccc1Cl CC1(CNC(c2cc(C3CCC3)on2)=O)CCCN1C(c1sccc1F)=O N1(C(C2C(CC)C2)=O)CCCC1CN(C(=O)C(c1cnn(C)c1)C)C c1(C(CNC(N(C)Cc2ccnn2C)=O)(C)O)cccc(Cl)c1 N1(C(C23CC(CC)(C2)C3)=O)CCC(O)(CNC(c2nc(C)sc2C)=O)CC1 c1(NC(C2CCN(C(c3c(C)scc3)=O)C2)=O)ccc(Br)cc1O c1(C(N2CCCC(N(C(CC(=O)OC)=O)C)C2)=O)cc(C)nc2c1cnn2C CC1C(NC(=O)COC2CCOCC2)CCN1C(c1cnc(C(C)(C)C)s1)=O C1(O)(CNC(C(C)=CC2CC2)=O)CCCN(C(c2ccc(O)nn2)=O)CC1 c1(OC)cnc(C(=O)NCCC2(O)CCN(C(C3CC3F)=O)C2)nc1 c1(C(=O)NC2CC(NC(CCN(C)CC)=O)C2)csc(-c2ccsc2)n1 C(=O)(C1=NOC2(CCN(C(c3cc[nH]c3)=O)CC2)C1)Nc1c(OC)ccc(C)c1 c1(-c2cc(C(C)OCC)sc2)cccc(Cl)c1O n1(CC)c(C(=O)NCc2csc(C(N3CCCC3C(C)C)=O)c2)cnc1O c1(C(=O)NCCC(C)NC(c2cnccn2)=O)cc(C2CC2C)on1 c1(CC)cc(C(=O)N(CCCNC(=O)C(C)C=Cc2ccccc2)C)cc(Cl)c1 Cc1nsc(N)c1C(=O)NCC1(CNC(=O)C(C2CCCCC2)O)CC12CCC2 C12=CNC(=NCCS1)C=C2.c1(C(=O)NCCN2CC(COC)C2)ccccc1 Cc1cc(-c2cn(CC3CCN(C(C4C5CCCCCC45)=O)C3)nn2)ccc1F Cc1c(C(N2CCC(F)C(NC(=O)C=Cc3ccc[nH]3)C2)=O)sc(Cl)c1Cl C(C(C)(C)CCO)NC(c1cccc(Cl)c1)c1n(CCC(=O)OCC)nnn1 N1(C(CCCOC)=O)CC2(CCN2C(c2nccc(OC)c2O)=O)C1 N1(C(C(c2cn(C)nn2)NC(C(CC=C)C)=O)=O)CC2(CCOC2)C1 C(=O)(C1CC(C)Nc2ccccc21)N(CC(C)NC(=O)CCOC(C)C)CC N1(C(c2ncc(C)s2)=O)CCC(O)C(C(=O)NC(c2ccccc2C)C)C1 N1(C(C(=O)NCCCOC)CC2(C#N)CC2)Cc2ccccc2N2CCCC2C1 c1(C(C)=O)cc(NC(C2CC3CC3N2C(=O)CCc2cn(C)cn2)=O)ccc1F c1(NC(N2CC(CO)CC(C(C)(C)C)C2)=O)cc(Cl)nc2ccccc12 CCC(C)(O)C(=O)N(C)CCC1CCN(C(C23COCC2C3)=O)CC1 C#CCC(CC(=O)NC(COC)C1CC1)NC(=O)CC1(N(C)C)CCC1 N1(C(c2c(C)n[nH]c2)=O)CCC(NC(C2(N(C)C)CCCOC2)=O)C(F)C1 C(c1c(C)cc(C)cc1C)=CC(=O)NCC1CN(C(CC(C)SC)=O)C1 c1(C(=O)NC(CNC(C(C)(C)SC)=O)C(C)C)cccnc1O c1(CCCSCC(=O)NC(c2ccccc2)CNCCC2C(C(N)=O)C2)ccccc1 c1(C(=O)NCC2C(NC(c3cc(N(C)C)n[nH]3)=O)C2)cc(F)cc([N+](=O)[O-])c1 CCCC(CCC)=CC(=O)NCCOCCNC(=O)C(c1ccc(Cl)s1)C N1(C(C=CSC)=O)CCN(C(=O)CC(O)C(C)C)C2(CCC2)C1 Cc1nc(C(=O)C(=O)NC(C2CCOC2)CNC(c2ccsc2Cl)=O)cs1 C1(C(N(CC(CNC(C(C)OCC)=O)C)C)=O)Cc2cc(C)ccc2S1 C(=O)(CC(O)COC(C1CC(N(C(COCCCOC)=O)C)C1)=O)NC(C)(C)C Cc1cc(CCC(=O)NC2CC2NC(=O)CCc2ncc(F)cn2)cc(C)n1 CC1=CCSC1C(=O)NCC(CO)NC(=O)CCn1ccnn1 CCCCCC(CC)C(=O)NC1CC1NC(c1cn(C)c(C)cc1=O)=O Cc1cccc(OCC(N2CC(C)(NC(c3cnsc3C)=O)C2)=O)c1 C(=O)(C1CCCc2nc[nH]c21)N(CCC(C(C)(C)C)NC(c1cncs1)=O)C C1(C(=O)OCC)CCN(S(=O)(=O)NC2CCC3CCCCC3C2)C1 c1(CC(=O)NC)ccccc1O.C(CCC(=O)O)N(C)C C(=O)(CCCCCN(C)C)NC1(C(NOCC(CC)O)=O)CCOC1 N1(C(C(CC=CC)NC(C2CC2OC(C)=O)=O)=O)CCCN(C=O)CC1 C(=O)(C(C)(C)C(O)c1cc(Cl)cc(Cl)c1)NCCC1CN(C(CSC)=O)C1 C#Cc1ccc(C(=O)NC23CCC(C2)N(C(c2cc(O)nc(OC)n2)=O)C3)nc1 c1(C(=O)NCC(CNC(C(C)(C)OCC)=O)(C)O)cnn(CCC(C)C)c1C c1(C2(COC(C3CCCC(=O)N3)=O)CC2)ccc2c(c1)OCO2 c1(CC2CCC(C)C2)nc(CC2CC2)nn1-c1cncc(Br)c1 c1(C(=O)NCC(CC=C)NC(C2C(C=C)C2)=O)cc(S(=O)(=O)N2CCC2)c[nH]1 c1(CC)cc(C(N2CCCOC(CNC(C3SCCS3)=O)C2)=O)c2c(c1)CCO2 Cc1c(CC(=O)N(CCCn2cc(C(O)C3CC3)nn2)C2CC2)cnn1C c1(CC(N2CCN(C(C(CC)CO)=O)CC2)=O)cccc2cccnc12 C1(CCCN2CCC(N(C(c3sccc3F)=O)CC)C2)CCS(=O)(=O)C1 CC1=CCC(CN(C(=O)CC2CCN(C(=O)C(c3ccccc3)C)C2)C(C)C)CC1 c1(CC)ccc(S(=O)(=O)N2CCOCC(Cc3c(SCC)ccc(F)c3)C2)cc1 C1(C)(NC(CC(C)SC)=O)CCN(C(C2(F)CCOC2C)=O)CC1 C(CCF)(C(=O)NOCC(C)O)NC(CC(CC)SC)=O c1(C(N(C2CCN(C(C(C(C)(C)C)N(C)C)=O)C2)CCO)=O)cc(Cl)c(F)cc1F C(=O)(C1=CC2CCCCCC12)NC1N(C(CCc2nnc(C)o2)=O)CC(C)(C)C1 C1(C(N2CC3C(CNC(c4cnn(CC(F)F)n4)=O)(C3)C2)=O)CC12CCSCC2 c1(C(N(CC(C)NC(=O)Cn2cccnc2=O)CC)=O)ncn2ccccc12 c1(OC)ccc(F)cc1S(=O)(=O)NC1CC(NCc2cccc(C#N)c2F)C1 c1(N2C(CC)CCCCC2)ncnc2c1ncn2C(CC1CCCCO1)CO C1(C(=O)NC2(CN(C(=O)Cc3cccnc3)C)CC2)CCCC12OCCO2 c1(C(=O)NC(C2CCN(C(=O)CCC#N)C2)C)cccc(NC(N)=O)c1 C(C(C)(C)CN=c1nc2sccc2c(NC(C)Cc2ccc(C)cc2)[nH]1)OCC c1(CC(=O)NCC(CC)NC(c2cncc(C)c2C)=O)cnc(C(N)=O)c(Cl)c1 c1(C(C(=O)NC2COC2)N(C(C(=O)OC)C)C)ccoc1C C1(NC(C=C(C)Cl)=O)CC2CCC(C1C)N2C(C1CCCCCC1)=O N1(C(C(N2CCC(O)CC2)C)=O)CC2(CCCC2NC(=O)CCC(C)(C)C)C1 Cc1cn2cc(C(=O)NCCC(c3cnn(C)c3)C)nc2s1 c1(NC(CC=C)C)nccc(=NC(CCO)c2ccccc2)[nH]1 C(CCCC)N.c1(CCC(=O)O)cn(CC(C(=O)C(F)(F)c2cccnc2)=O)nn1 CC1(C)CN(C(=O)C2=CCCSC2)CCC1NC(c1[nH]nc2ncccc12)=O c1(N(C)C)ccc(N)c(C(=O)NC2CCCC2NC(=O)CC2CCCOC2)c1 Cc1cnc2nccc(C(=O)NC3CC(C)N(C(=O)Cc4sccc4C)C3)c2c1 C1(C)(CNC(c2c(OC(C)C)cccc2)=O)COCCN(C(C2(C)CC2)=O)C1 CCC(CC1CC1)CC(=O)NCCC1CN(C(=O)C(c2cccc(OC)c2)C)C1 C1(CCC2(C(CC)(C)C)N=N2)CCCN1C(C1CC(=O)NC1)=O C=CC1CCN(C(C2CN(C(=O)CCCCSC)CC2CCC)=O)C1 C1(C)(CNC(C(CCC)C)=O)CCCN(C(=O)CC2(C3CC3)CC2)C1 C1(C(=O)NCC2CC(NC(C3C(C)CC3)=O)C2)CC2(COC(=O)N2)C1 CCC(C)C(=O)NCC(=O)NCC(C(=O)NOCCn1cc(C)cn1)C c1(COCC)cccnc1C(=O)NC(C(C)NC(C1CCCCO1)=O)c1ccco1 C12(NC(c3cc(CC)c(CC)o3)=O)CCC(C1)N(C(=O)COC(C)CC)C2 C1(C(=O)NC(CNC(c2oc(CC)c(C)c2)=O)CC(C)C)CC2C(C1)C2(F)F CC(C(F)(F)F)NC(=O)C(F)CC1CN(C(c2cc(C(N)=O)[nH]n2)=O)C1 CCCC(CCC)CC(=O)NC(C)(C)CNC(=O)C(C)(C)COCC N1(C(CC2(N(C)C)COC2)=O)CCC2(CCCN2C(=O)Cc2cncc(O)c2)C1 Cc1c(NC(=O)CC2CN(Cc3ccccc3N(C)C)C2)[nH]c2ccccc12 N1(C(CCC=C=C)=O)CC23CCCC2(C1)CN(C(C1CNC(=O)C1)=O)C3 c1(CC)ncccc1C(=O)N(CC(O)CN(C)C(c1ccn(C(C)(C)C)n1)=O)C N1(C(CCC)=O)Cc2ccccc2CC1CNC(c1nnn(C)c1C(F)(F)F)=O c1(C(C)=O)cc(CN2CCC(SC)C2)n(C)c1.c1(C(CCC)O)cccc(Cl)c1 N1(C(C(CCC)CC)=O)CCC2CCN(C(=O)C=CC(=O)N(C)C)C2C1 N1(C(c2ccn(C(C)C)n2)=O)CCCC(C)(CNC(=O)C(C)(C)CF)C1 CCCCC(C)(F)C(=O)N1Cc2[nH]nc(C(=O)NCC3(O)CC(CO)C3)c2C1 N1(C(CCC(C)OCC)=O)CCCC2(C1)CN(C(C1CCOC1)=O)C2 C1(C(=O)NCC(n2cccn2)C)(CO)CCCN(C(C2CC3CC3C2)=O)C1 CC1CCSC1C(=O)NC1CN(C(=O)Cc2csc(NC(=O)OC(C)(C)C)n2)C1 C(=O)(CCCCC(F)F)NC(C)CNC(=O)C(c1ccccc1)O C=CCC(C)(C)C(=O)N1CCC(C(=O)N(CCCC)CCCO)C(C)C1 N1(C(C(CC)SC)=O)CC(NC(c2ncc(C)cc2C)=O)C(S(C)(=O)=O)C1 c1(CNC(c2cc(C3CCCCC3)n[nH]2)=O)cccc(C(F)(F)F)c1.c1csc(C)c1 C1(NC(C(CC)n2ccnc2)=O)CC2(CCN(C(=O)CC3CSCCS3)CC2)C1 Cc1ccc(CC(=O)NC23CC(C2)N(C(=O)CNC(=O)CCCCO)C3)c(F)c1 c1(C(=O)NC(CCCNC(C2CCC(C)C2)=O)(C)C)cc2ncccc2[nH]1 C(CC(=O)C(c1cc(NCC)cc(C)c1)=O)(C(F)(F)F)OC.C1(C(=O)OC)(O)CC1 c1(Cc2oc(=O)n(-c3cccc4c3CCCC4)n2)ccc(Cl)c2cccnc12 C12CCCCC1CN(C1CC1)C(=O)C(=O)N2.c1(CCC(=O)OCC)nn[nH]c1OC C1(NC(C(COC(C)C)NC(C)=O)=O)CN(C(=O)C(F)(F)CO)CC1C Cc1ncc(NC(C2CCN(C(=O)CCc3ccccn3)C2(C)C)=O)c(C)c1C CN=c1[nH]c(C(N2CCCC(CCNC(C3ON=C(C)C3C)=O)C2)=O)cs1 c1(C(C)OCN(CS(C)=O)C(C)=O)ncc(-c2ccccc2)o1 N1(C(CC(CC)C)=O)CCCN(C(=O)NC(c2ccccc2)C)CC1C N1(C(C2(C(C)(C)O)CCOC2)=O)CCN(c2ncncc2Cl)CC1 CCCCCCC(C)C(=O)N(CCC(=O)NCCc1ccccc1)C1CC1 C1(NC(C2(c3cccc(F)c3)CCN(C3CC3)C2)=O)CCC(=C(F)F)CC1 c1(CC(Cn2cc(C3(OCC)CCOC3)nn2)O)ccc(Cl)cc1 CN1CC=C(CC(=O)N2CC3CCC(CNC(C4(CN(C)C)CC4)=O)(C3)C2)CC1 c1(C(=O)NCCC(CNC(CC)=O)O)ccc(NCCNC(C)=O)cc1 C(=O)(C(C(C)(C)C)OC(C)(C)C)NC1CN(CC(=O)NC(C)C)CC1C S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)N1C(CC)CN(C(c2scnc2C)=O)CC1 c1(C(CN(CC(C)O)C)NC(C2(Br)C(C)C2C)=O)ccccc1 N1(C(C2CCSCC2)=O)CCCC2C1CCN2Cc1cccc(O)c1Cl c1(CC(=O)NC2CN(C(c3c(C(C)C)cccc3)=O)C2)cc2c(cc1Br)OCO2 n1(C(CC)C)ccc2ccc(OC(C3CCCCN3C)=O)cc12.n12cc(nn1)C2 N1(CCC(C)NCC23CCC(C(=O)OCC)(CC2)C3)C(=O)c2ccccc2C1=O C1(C(=O)N)CC2(CCC2)C1.C1(C(CCCC)(C)O)CCN(C(c2ccns2)=O)CC1 c1(C(N(CCOC)CCNC(C2C3CCC2CC3)=O)=O)cccc(C)c1Br N1(C(CN(C)C(=O)C2CC2)=O)CCC2(C1)CN(C(C1CCCC3CC13)=O)C2 c1(NC(c2c(NC(c3c(C)nn(C)c3C)=O)cn(C)n2)=O)ccc(C#N)c(Cl)c1 c1(OC)ccccc1NC(c1ccc(-n2ccnc2)nc1)c1nnnn1C N1(C(Cc2c(C)ncs2)=O)CC(O)CC1C(=O)NC1CN(C)CC1C N1(C(CNS(CCOCC)(=O)=O)=O)CCN(C(=O)C(C2CC2)OC)CC1C(C)C C1(C)(C(N(CCN(C(c2cc(CCC)on2)=O)C(C)C)C)=O)CCNC1=O C12(C(=O)NCC3(O)CC(CNC(C4CS(=O)(=O)C4)=O)C3)CCC(CC1)CO2 C(=O)(C(CC(C)C)C(N)=O)NC1C(CNC(c2cc(C)c(O)nn2)=O)CC1 CC1CC(C(=O)NC2COC(C)(C)C2)CCN1C(C1CC2(C1)CC(O)C2)=O c1c[nH]cc(F)c1=O.O=C1CN(CCC(=O)Nc2cccc(N)c2)CCN1 CC1(C)CC(O)(CC(N2CCC(O)(CCNC(C3(CO)CCCC3)=O)C2)=O)CO1 N1(C(CN(CC)CC)=O)CC2CCN(C(C3CC(=O)N(CC(F)(F)F)C3)=O)C2C1 Cc1cc(C(=O)N(C)CCN(C(c2c[nH]nc2C)=O)C(C)C)ccc1Cl c1(NC(c2cccc(NCc3c(OC)c[nH]n3)c2)=O)c(C)ccc(C)c1O N1(C(c2c(C)oc(C#N)c2)=O)CC2CN(C(=O)C=Cc3cncc(F)c3)CC2C1 C(=O)(C(O)CC(F)(F)F)NC1C(CC(=O)Nc2cccc(OC)c2O)CCC1 N1(C(C(CC=C)(C)C)=O)CCC2(CCCC2CNC(=O)CCNC(C)=O)CC1 Brc1ccccc1C1(NCc2noc(Cc3ccco3)n2)CC1 C1(C(N2CC(CN=[N+]=[N-])OCC2)=O)CCN(C(=O)CC2CNC(=O)O2)O1 c1(CC)ccc(OC)cc1C(N1CC(NC(=O)CN=S(C)(C)=O)CCC1C)=O C1(NC(CC2(OC)CCC2)=O)CCN(C(=O)C(C)N(C)C(C)=O)CC1F N1(c2nnc(C(C)(C)C)s2)CC2(COC(CNC(C3(CF)CCC3)=O)C2)C1 n1(Cc2ccc(C(C)C)cc2Cl)c(=O)c2c(C)cccc2n(C)c1=O N1(C(CCCCCC)=O)CCOC2(C1)CN(C(C1CCC1n1cccn1)=O)C2 C(C)(C(CC)CC)NC(c1ccc(CNC(c2ccc(CC)s2)=O)o1)=O N1(C(C2CCCN(C(N)=O)C2)=O)CC2C3CCC(C2C1)N(C(=O)CCC(F)F)C3 CC(CNC(=O)CCc1cnn[nH]1)C(=O)NCc1nc(C2CC2)n[nH]1 C1(NC(c2cncs2)=O)CN(C(=O)Cc2cnsc2)CC1C1CC1 c1(CCC(=O)N(CCNC(C2CCCCN2C)=O)CC)cccc(F)c1Cl N1(C(CN(C2CCC2)C)=O)CC2(CC(NC(C3(C)COCCO3)=O)C2)C1 C12CN(C(=O)C(CC)n3ccnc3)CC1CC(=O)N2.C1(CCCC)(CF)CCC1 CC1CCCC(NC(=O)C=CCN(C)C(c2cnn(C)c2N)=O)C1 Cc1ccc(F)c(N)c1C(=O)NCCC(C)NC(=O)C=Cc1ncc[nH]1 N#Cc1ccc(C(=O)NCC2(F)CCN(C(c3ccc(Cl)s3)=O)CC2)cc1Cl CCC(CCC(=O)Nc1cnccc1CO)NC(=O)C=Cc1cc[nH]n1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(CN(C)C(c2c(Cl)n[nH]c2C)=O)CC1 C(=O)(C(C#N)C(C)(C)C)NC(C1(c2ccccc2)CCCC1)CNC(CC=C)=O c1(OC)ccc(N=c2scc(CC3(CO)CCCC3)n2-c2cncnc2)c(F)c1 C(=O)(C(F)(F)CCn1cccn1)NCCCCNC(CCCCOCC)=O C=CC(C)(O)C(=O)NCC1CC(F)CN1C(=O)C(C)OC(C)=O c1(C(=O)NC2(C)CC(NC(C=C(CCC)C)=O)C2)cc(S(C)(=O)=O)ccc1C C1(n2c(C(c3cn(CC)cn3)NCC(CC)CO)nnn2)CCC(F)(F)CC1 C1(O)(CC(=O)NC2CC(C(C(=O)NC(C(CC)C)C)F)C2)CCOCC1 C1(NC(=O)CCCC2CCCCC2)CN(C(C2CC(O)C2)=O)CCC1C(F)(F)F c1(NC2CC(C(C)(C)OC)N(C(=O)OC(C)(C)C)C2)ccc2cccnc2n1 C(=O)(C#CCNC(=O)CN(C)C)NC(C#C)(C)C1CC1 c1(C(C)(C)C)ccc(NC(=O)NCC2CCCN2CCCc2ccccc2)cc1 C1(NC(CNC(C)=O)=O)CCN(C(c2ccc3cn(C)nc3c2)=O)CC(C)(C)C1 C1(=CC(=O)NCC(CN(C(c2c(C)nsc2N)=O)C)C)CCCCC1(C)C CC(C)C(CNC(=O)C=Cc1ccncn1)C(=O)N1CC2CC2C2CC12 c1(NC(C2(C=C)CCN(C(C3COCCO3)=O)C2)=O)cccn2ncnc12 C(=O)(C1Cc2c(Cl)cccc21)N1CCC(NC(c2ccc(O)nc2Cl)=O)C1 N1(C(CC2C=NN(C)C2=O)=O)CC2(CO)CC1(C(=O)NCC1CCCC1)C2 c1(NC(C2(OC)CCN(C(COCCCC#C)=O)C2)=O)cnc(F)cc1C O(NC(=O)C(C)CSC)CC(=O)N.CCCCC(CN1CCCC1)N N1(C(CS(CC)=O)=O)CCC2CCN(C(c3ccc(C(F)(F)F)cc3)=O)CC2C1 c1(CC(=O)NCCN(C(=O)C(F)(F)C(C)(C)O)C)c[nH]c2ccccc12 CC1(C)CC(=O)OC1CNC(=O)CN(C(=O)CC1CC2CC2C1)CC1CCCC1 c1(OC)ccccc1CCNC(c1cncc(-c2ccncc2)n1)=O C1(C(C(=O)NCC2(CNC(COC)=O)CC2)O)CCOCC1 N1(C(CCC(CC)NC(c2c[nH]c(C#N)c2)=O)=O)CCCNC(=O)C1C Nc1sc2c(c1C(=O)NCC1CC1CNC(c1ccc(=O)oc1)=O)CCC2 C=C(C)C(C)(C)C(=O)NCC1CN(C(=O)C(C2CCC2)OCC)CC1C C1(NC(C(C)Oc2cccc(F)c2)=O)CC(N=c2[nH]c(Cl)ncc2OC(F)(F)F)C1 c1(C(C)=O)cc(C(=O)NCCn2ccc(C(=O)NCCS(C)(=N)=O)c2)no1 N1(C(c2cccc(C)c2N)=O)CC2CC1CCC2NC(=O)CC(C)C n1(CC)nc(C(=O)NCC(C2CC2)NC(=O)C(CC)OC2CCCC2)c(C)n1 CC12CC(NC(=O)C3CC3)(C1)C1(CN(C(=O)Cc3cccc(C#N)c3)C1)O2 c1(OC)cc(C)ccc1C(N1CC(F)(C(=O)NCC2C=CCC2)C1)=O N1(C(C(C)n2ccnc2)=O)CC2CCC(NC(c3ncc4ccccn34)=O)C2C1 Cn1ccc2ccc(CNC3CC(C(=O)Nc4ccc(CC#N)cc4F)C3)cc12 c1(C(N2CC(NC(C(CC)(C)CC)=O)C(N=[N+]=[N-])C2)=O)ccc(F)c2c1CCC2 C1(NC(C(CSC)O)=O)C2CN(C(=O)CC(=O)NCC(F)(F)F)CC12 C1(O)(C(C)NC(C)=O)CCN(C(c2cccnc2-c2ccncc2)=O)C1 C1(CC(=O)NCC2(O)CN(C(C3CCC(N(C)C)C3)=O)C2)(CC=C)CCCC1 N1(C(C(C)NC(=O)NCC)=O)CCC2(C1)CN(C(c1scc(C)c1C)=O)C2 Cc1nc(C(N2CC(CCc3cn(C(C)C)nn3)C2)=O)n(C)n1 N1(C(CC=CC=C)=O)CCC2CCCN(C(c3nc4ncc(C)cn4n3)=O)C2C1 N1(C(C(CC2CCOCC2)NC(C2CC=CCC2)=O)=O)CCCC2(CCCC2)C1 C(=O)(CC(C(C)OC)NC(c1ccc(O)cc1F)=O)N(CCCCCC=C)C c1(C(=O)NCC2C(C)CCN2C(c2occ3c2CCC3)=O)cccc2ncnn12 c1(CNC(C2CN(Cc3c(F)cccc3F)CCO2)=O)ccc2c(c1)C(=O)CC2 N1(C(C2C(OC)CCC2)=O)CCN(CCNC(c2cncc(C(F)F)c2)=O)CC1 CCCC(O)(CCC)CC(=O)NC(C)(C)CCCNC(c1nn(C)cc1C)=O C1(CC(=O)NC2(NC(C)(C)C)CCC2)(OCC)CN(C(C)=O)C1 C1(CC)CC(c2nnnn2C2COC2)(NCCC2(C)CC2)CCS1 C1(NC(Cn2ccc(C)n2)=O)CC2CC(NC(=O)CN3CSCCSC3)C2C1 c1(OCC(=O)NCCNC(C(n2cc(Br)cn2)C)=O)ccc(O)cc1 c1(C(=O)NC23CCC(C(=O)NCC4CCC(O)CC4)(CC2)C3)c(F)cccc1Cl C(=O)(CC(C(F)F)NCC(=O)NC1NCCCC1c1ccccc1)OC N1(C(C(CCOC)OC)=O)CCCCCC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C1 Cc1noc(C)c1C=CC(=O)NC(CNC(=O)C(C)Sc1ccc(F)cc1)CO C(CC(=O)NC1C(CC(C)(C)C)C1)(C(F)(F)F)NC(=O)CC1COC(C)(C)C1 C1(CCC)(NC(=O)CS(=O)(=O)NC)CCCN(C(C2CCCC3(CC3)C2)=O)C1 CC(CN(C)C(C1CC2(CC2)C1)=O)C(=O)NC(C)C(C)(C)O CCS(=O)CC(=O)N(C)CC1(O)CN(C(=O)COc2cccc(OC)c2)C1 C(=O)(C(=O)Nc1ccco1)N(CCN(CCCN(C)C)C)CC1CC1 N1(C(C2CC(CC)C2)=O)CC2C(CNC(=O)CC(C)Sc3cccc(Cl)c3)C2C1 CC1(C)CC1(C(=O)NCC1CC1CC(=O)NC1CC(C)(O)C1)OC Cc1ccc2[nH]c(C(=O)NCCNC(c3ncnc(O)c3F)=O)c(Cl)c2c1 c1(OC)ccnc(O)c1C(=O)NC1CC2(C1)CN(C(=O)CC1(C3CC3)CC1)C2 c1(-c2ccc(N(C)C)nc2)cccn2ncc(C(=O)NCCC(N)=O)c12 n1(CC)nnc(C)c1C(=O)NCCC1COCCN1C(c1cn(C)[nH]c1=N)=O C(=O)(CC(F)(F)C(C)C)NCC(C(C)C)(C)NC(c1cncc2c1CCC2)=O C1(OC)CCOCC1NC(=O)CCCCN(C(=O)C(F)CC1CCOC1)C N1(C(CCN(C(CC(CC)C2CC2)=O)CCO)=O)CCC(O)C(C)C1 c1(OC)ccc(C)cc1C(=O)NC1CCN(C(=O)CC2C=CCC2)C(C)C1 N1(C(C2SCCS2)=O)CCN(C(c2cccc(F)c2O)=O)C(CC(F)F)C1 C=CCCCCC(=O)NCC1CC2(CC(NC(C3CC3F)=O)C2)C1 C(C)CCC(=O)NCC(CO)NC(c1cnnn1C(=O)OC)=O.CCOC c1(C(=O)NC2(CCNC(C3CCC(N(C)C)C3)=O)CC2)cccnc1S C1(CC=C)(C(=O)NC(c2cnc(F)cn2)C)CNCCO1 CCC(CC(=O)NCCCCc1ncc[nH]1)NC(C1CCCSC1)=O C(=O)(CC1CC(=O)Nc2ccccc21)N(CCNC(C1CC=CCO1)=O)CC N1(C(C(C)(C2CC2)OC)=O)CCC2C(C1)CN2C(c1cc(C)c(C)[nH]1)=O N1(CC(CCCC)C)CC2CCCN(C(=O)Cc3ccccc3OC)C2C1 C12(C(N3CCCC(NC(Cc4nnn(C(C)(C)C)n4)=O)C3)=O)COCC(C1)OC2 C1(C(N(CCOCCN(C)Cc2cn(CC(CC)C)nn2)C)=O)CCCC2(CC2)C1 N1(C(CCC)=O)CCC2C(NC(c3ccc(C4(C)CC4)cc3)=O)C12 C=CCC(C(=O)N1CC(CNC(c2scc(C)c2OC)=O)C1)C(C)C c1(CS(=O)CF)nc(-c2cncc(F)c2)nn1-c1cccc(Cl)c1 n1(CCC)nccc1C(N1CCCC1CC(=O)NC1CC(F)C1)=O C1(CNC(C2C=C(C)CS2)=O)CC(C)N(c2nnc(CC(F)(F)F)s2)C1 C(=O)(C(CCC1CCC1)NC(C1CC2(CC2)CO1)=O)NCC1CCC(C)C1 N1(C(CSCC(=O)OC)=O)CCC(NC(c2cnn(CCCOC)c2)=O)C1(C)C N12CCN(C(C#N)C1)C2=O.c1(NCCCOCC#C)ccnc(OC)n1 N12CC3CCCC1C3CNC2=O.c1(OCCC(C)C)ccc(C(F)(F)F)cn1 c1(OCC)ccc(CN2CC(NC(C3CCCC3C)=O)C(F)C2)cc1Br Cc1nc2ccnn2c(C)c1C(N1CCN(C(=O)C(F)CC2CC2)CC1C)=O N1(C(C(C)NC(C)=O)=O)CCCC(O)(CO)C1.N12CCC(C1)C(C)C2=O Cc1cc(Cl)c(C(N2CCCC2CN(C)C(C2CCC(=O)N2C)=O)=O)s1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(C=C)(C(N2CCOC3CCCC23)=O)C1 C1(C(=O)NCC(CNC(C(C)C2CCC2)=O)F)CCn2c(O)nnc2C1 C(=O)(C(C)C(C)NC(C1CC(OC2CC2)C1)=O)NCCSC(C)C C(CCCC(=O)NCC1CC1)OC.c12nc(co1)C(=O)NOCCO2 c1(C(=O)NC(C)C(C)NC(=O)CN2C(=O)NC(C)(C)C2=O)ccnc2cc[nH]c12 C1(C(N(C2CC(F)(F)C2)C)=O)CCCCN(C(=O)CCc2cnn(C)c2)C1 C1(CNC(c2c(C)coc2)=O)CCN(C(c2cn(C)ccc2=O)=O)CC1C CC1(C)CCC(CNC(=O)C2=CCCCC2)(NC(=O)Cn2ccnn2)CC1 c1(C(C(=O)NCC(=C)C)N(C)Cc2ccc(C)cc2)cn2ccc(Br)cc2n1 N1(C(C(CC(C)C)OC)=O)CC2CC(NC(c3cn(CCO)nn3)=O)CC(C2)C1 c1(OC)cccc(CCC(=O)NC(CNC(c2ccc(Br)o2)=O)CO)c1F C1(c2cccc(OC)c2)CN(C(=O)CCCCCF)CCN1C(C1CC1C)=O c1(OC)ccc(C(=O)NC(C)CCNC(c2c(C(C)C)cccc2F)=O)c(F)c1 c1(OCOC)ccc(C)c(-c2cc(C(=O)NCc3ccc(Cl)nc3)ccn2)c1 N1(CCC(=O)NCC2(CCNC(C=CCCC(C)C)=O)CC2)CCSC(C)(C)C1 N1(C(C2CC(N(C)CC)C2)=O)CCN(C(C2(C(=O)OC)CC2)=O)C(CCO)C1 C1(c2n(CCCSCC)nnn2)(NCCC2CC23CCC3)CSCCSC1 C(=O)(C#CC1CC1)NCC(CNC(c1oc(Br)cc1C)=O)OC Cc1[nH]nc(C(=O)NC(C)C(C)NC(=O)Cc2ccccc2O)c1C c1(OCC)cccc(CC(=O)NCCC(C)NC(=O)CCc2ccoc2)n1 c1(C(N2CCC(F)(CNC(c3csc(F)c3)=O)C2)=O)cnc2c(n1)CCCC2 C(=O)(CCCC(=O)NCCOCCCNC(c1sc(C)nc1C)=O)N(CC)CC c1(C(N2CC(NC(Cn3c(C)cc(C)n3)=O)C(F)C2)=O)c(Cl)cccc1Cl Cc1nc(C)c(CC(=O)NC2(c3ccccc3)CC(NC(=O)C=C3CC3)C2)s1 N1(C(C(=O)NCC(F)F)=O)CCCC2(CNC(=O)C3=CCCS3)CCCC12 N1(C(C(CCC)(C)C)=O)CC2CCOC2(CNC(c2snc(Cl)c2Cl)=O)C1 c1(C(=O)NC(CNC(Cc2cccc(C#C)c2)=O)C)nc2ccccc2[nH]c1=O N1(C(c2c(C)cc(F)nc2)=O)CCCC2CN(C(=O)CC3(O)CCCOC3)CC12 C1(OC)CN(C(=O)Cc2cc(C)cs2)CCC1NC(C1CCN(C)C1C)=O C(=O)(N=c1nc(Cl)nc2[nH][nH]cc1-2)C1(c2cccc(C)c2)CCN1C(=O)Nc1cccs1 c1(C(=O)NCC2(C)CCN(C(C3(C)CCC(=O)C3)=O)C2)cc2n(c1)CCCC2 CCC(O)C(C)C(=O)N1CCC(NC(=O)CNc2ccc(C#N)cc2)C(C)C1 C1(CN(C(COC)=O)C)C2CN(C(C3CC(C(F)(F)F)CO3)=O)CC12 N1(C(CCOC)=O)CCC(CO)C(NC(=O)CC2CCSCC2)C1 c1(NC(C)=O)cccnc1C(N1CC(C(C)NC(C2COC(C)C2)=O)C1)=O Nc1c(C(N2CCN(C(c3cnc(S)[nH]3)=O)C3CC23)=O)cccc1F C(C(=O)NOCC=CCl)(C1(CC)CC1)NC(C1CCCO1)=O C1(NC(CS(=O)(=O)NCC)=O)COCCN(C(=O)C(N2CCCCC2=O)C)C1 c1(CC(=O)NC2CC(CNC(C(CC#C)C)=O)C2)c(C)nn(C(C)C)c1C C1(C(N(C(CNC(c2c(CC)scn2)=O)C2CC2)C)=O)CC2(CCCC2)CO1 c1(C(=O)NCCCN(C(=O)CCC(C)OC)CC)ccc2c(C)noc2n1 c1(C(C(N2CC(CNC(c3c(C)cccn3)=O)C2)=O)C)c(F)cccc1F Cc1cc(C)c(C)c(C(=O)NC2CN(C(=O)C(O)C(C)C)CCC2O)c1C C(=O)(C(C)(C)CN(C)C)N(C(C)C(N1CCC(CSC2CCCO2)C1)=O)CC C1(C)(C(=O)NCCN(C2CCCCC2)C(c2ncn(C)n2)=O)CC2(CC2)C1 C1(C2CCC2)(C(N(CCOC)CCNC(C2(C)CC(C)(C)C2)=O)=O)CC1(F)F C(=O)(N=c1ccn(-c2nc(C)cc(C)n2)[nH]1)C1(OC)CCN(c2ncccc2Br)C1 C1(NC(c2cc(CC)oc2C)=O)CCCCCC1NC(C1C=CCS1)=O C=CC1(C(=O)NCCc2nc(CC)no2)CCN(C(=O)CCn2ccnc2C)C1 C(=O)(C(F)(F)C(C)O)N1CCC(NC(C=CCCC)=O)(CO)C1 Cn1ccc(=O)c(C(N2CCN(C3CCN(c4nnc(O)s4)C3)CC2)=O)c1 C1(C(=O)NCC(C)CNC(c2nnc(C(F)(F)F)s2)=O)CCCC(C)CC1 CCCCCC(C)(C)C(=O)N(C)CCNC(c1c(C)sc(Br)c1C)=O N1(C(C2CC(C)C2)=O)C2CCC1CN(C(c1ccnc(N3CCCC3)n1)=O)CC2 c1(C(=O)NCCN(C(=O)C(C2CCCC2)OCC)CCC)cccs1 c1(C(=O)NC(C)CCNC(C2CC3(C2)CC3(F)F)=O)ccc2n[nH]cc2c1Cl C(CCCCCCC(=O)NC1COCC1C(=O)CCCF)SC c1(C(=O)NCc2ccc(CN(C(C(C)SC)=O)C)cc2)ccc(C)c(O)n1 c1(NC(C2(CO)CCN(C(C3CC(OCC)C3)=O)C2)=O)nc(OC)ccc1C CN1CC(F)CC1C(=O)NCCC1CSCCN1C(=O)C(O)C1CCCC1 c1(C(C(=O)NC2CCN(C(Cc3ncc(C)s3)=O)C2)O)ccc(F)cc1 N1(C(CCNC(N)=O)=O)CCOC2CN(C(c3ccc4nc[nH]c4n3)=O)CC12 c1(C(=O)NCC2CC(NC(C(=O)NC(C)C)=O)C2)cnn(CC2CCOCC2)c1 C1(CC(=O)NC(C)CCNC(c2cscc2Br)=O)CCCC2(CC2)C1 N1(C(C2=CCCC2C)=O)CCC(C2(O)CN(C(c3cc[nH]c3)=O)C2)CC1 c1(C(=O)NC2C(C(=O)NC3CC(C)C3)CC2)ccoc1Br C(=O)(CC(C)CC(C)(C)C)NC1CN(C(c2nc(CC)sc2N)=O)CC1O c1(NCCC=CC=C)ccc(S(=O)(=O)N2CCC(C3CCCCO3)C2)cc1F C12CCCN(CC1)CC(=O)NC(=O)C(C)C(=O)N2C.C(=O)(N)NC(C)C.C1(N)CC1 N1(C(CCC2(NC(C(=Cc3ccco3)C)=O)CCC2)=O)CCc2ncncc2C1 C1(C(N(CC)CC2CCCN2C(c2cocc2C)=O)=O)CCCN(C(=O)OC)C1 C1(C)(CC)CC(NC(C2(C)CC2)=O)CN1C(=O)CCc1cccc(O)c1 C1(NC(c2c(CC)oc(C)c2)=O)CC(F)CN(C(c2ccc(C(C)O)cc2)=O)C1 c1(CC(N2CCC2CNC(C23C=CC(CC2)C3)=O)=O)cc(Cl)ccc1[N+](=O)[O-] CC(C#N)C(=O)N(CC(C)C(=O)NCc1nnnn1C1CC1)C C1(CNC(CCCN(C(C)=O)C)=O)CN(C(=O)CCCCC(F)F)C2(CCC2)C1 c1(C(c2n(CC)nnn2)(C)NC(c2ccncc2)COC)ccnc(C2CC2)n1 CC1(N(CC(O)Cc2cccc(Br)c2)Cc2ccccn2)CCC(N)CC1 C1(C(N2CCC(OCC#C)C2)=O)CNC(=O)CN1C(=O)C(CC)CC c1(C(=O)OCC2C(C(=O)OC(C)(C)C)C2)c(Cl)nc2cc(Br)ccn2c1=O c1(Cn2cc(CNC(C3CCn4ccnc4C3)=O)nn2)nc2cc(Br)ccc2s1 N1(C(c2cc(C)nc(O)c2)=O)C2CCC1CC(NC(c1cn(C)nc1O)=O)C2 N1(C(c2c(C)cc(F)s2)=O)CC2CCC(C1)N2C(=O)CCC1CC(C)C1 c1(N)ccc(-n2cccn2)cc1.C(CCC(=O)OCC(=O)NC(C)C1CC1)SC CCC(CNC(c1cnc(CC(C)C)[nH]1)=O)(CC)NC(=O)C(C)SC C1(C(N(CC(C)CNC(=O)CN(CC(C)(C)C)C)C)=O)CCS(=O)(=O)C(C)C1 Cc1cnc(C(=O)NC(CCC2CCC2)C(=O)Nc2cc(Cl)cnc2C)c(F)c1 c1(C(N2CCN(CC(C)(C)NC(CC(C)SC)=O)CC2)=O)ccc2sccc2c1 C1(O)(CCNC(C2C(C(N)=O)C2)=O)CCN(C(c2c(Cl)cccc2Cl)=O)CC1 N1(C(Cc2cnc(C)o2)=O)CCCC2(CC(NC(=O)CCc3nc[nH]n3)C2)C1 C1(NC(CC(C)CNC(C2CC(=O)N(C)C2)=O)=O)CC2(C1)CN(C)C2 Cc1oc2ccccc2c1CNC(=S)NNC(=O)c1ccc(C(=O)N(C)C)cc1 CCS(=O)CC(=O)N1CC(COC)(NC(=O)Cc2cccc(Br)c2)C1 C(=O)(C1=CCN(C(=O)COC2(C)CCC2)C1)N(CCC=C)CC C(=O)(C(CNC(=O)Cc1cccnc1)CC(C)C)NC1CCN(CC)CC1C N(C1c2ccccc2CC1NC(c1ccc(C(F)F)cc1)=O)C(C(CC#C)C)=O N1(C(c2c(C)nn(C)c2)=O)CCCC(C2CN(c3ccnc(C(F)(F)F)n3)C2)C1 c1(C(=O)NCCOCCN(C(C(CC)(C)C#N)=O)C)cc2ccncc2cc1F Cc1nc(C(=O)NC2(C)CC(NC(=O)CC3CCCN3C(C)C)C2)n[nH]1 C1(N(C(c2c(CC)cco2)=O)C)CCCN(C(=O)CCc2nccs2)CC1 C1(C)(NC(C2CC(CNC(C(C=C)(C)O)=O)OC2)=O)CCC(C)(C)C1 c1(C(N2CCC(O)(C(=O)Nc3n(C)nnc3)C2)=O)coc2ccccc12 CC1(C)CCCN(C(=O)Cc2ccco2)C1CNC(C1CCCCCCC1)=O c1(CCC(=O)N(CC(C)O)CCNC(C(C(C)C)SC)=O)cnc(C)nc1O C=CCC(C)(C)CC(=O)N(C)CC1CCCN1C(C1(C)CC=C(C)CC1)=O N1(C(C(=O)NCC2CCN(C(c3c(COC)noc3)=O)C2)C)C(=O)CCC1=O S(=O)(=O)(c1cnccc1N1CCC(S(N)(=O)=O)C1)NCCSCC(OC)SC c1(C(=O)NCCC(C)NC(c2cocc2C(N)=O)=O)csc(C(C)(C)C)n1 c1(CC)ccoc1C(=O)NC(CC1CCCC1)C(=O)NCC=CCl C(=O)(C1=CCCO1)N(CC(C)O)CCNC(COC1(C#C)COC1)=O C1(COC)(NC(c2c[nH]c(=NC)s2)=O)CCN(C(c2cnncc2C)=O)CC1 c1(SCC(=O)NCC(CO)NC(C2C(C)(Br)C2)=O)nnnn1C1CC1 C1(CNC(C(c2ccccc2)C)=O)CC(C)(C)CN1C(C1(CF)CC1)=O C(=O)(CC(CN)C(F)(F)F)Nc1c(C)c(F)c(F)cc1 N1(C(C(C)n2cncn2)=O)CCC(NC(=O)C(C)SC(F)(F)F)C(C)(C)C1 CC1OC2(C(=O)NC3CN(C(c4cccc[n+]4[O-])=O)CC4(CC4)C3)CCC1CC2 c1(OC)ncccc1CC(=O)NCC1CCN(C(c2n[nH]c(C)c2C)=O)CC1 CCCCC(CC(=O)N(C1CCN(OC)CC1)C)NC(C1CCC(=O)CC1C)=O n1(C(C)C)ncc(C(=O)NCCCNC(c2nn[nH]c2C(F)(F)F)=O)c1F c1(NC(=O)CN2CCC(O)CC2)ccn2nccc2n1.C12CN(CCO1)C2C Cc1c(C(=O)NC2CCCC(C(N3CCC(C4(C)N=N4)C3)=O)C2)c[nH]c1C#N Cc1c(C(N2CCOC(c3cccnc3Br)C2)=O)nnn1-c1cnn(C)c1 CCCCC(CNC(C1CCCC1CCC)=O)NC(c1ccnc(OC)c1)=O C(C(C)(C)n1ccnc1)NC(CNC(C1C(CC(C)C)C1)=O)=O N1(C(CC2C(C)CCC2)=O)CCC2(CC2)CC1C(=O)NCc1ccnc(CO)c1 N1(C(CCNC(COC)=O)=O)CCN(C(c2cnc(O)n2CC)=O)C(C)C1C C(=O)(C#CC(C)(C)CNC(c1ncoc1C1CC1)=O)NCC1(OC)CC1 Cc1sc(C)c2sc(C(=O)NC3CN(C(C45CCC(CO4)C5)=O)C3)cc12 N1(C(CCC2(C)CC2)=O)CC(NC(c2sc(C#N)cc2Cl)=O)C(C)(C)C1 n1(CC(N2C(CN(C(=O)C(C)CCO)C)CCC2)=O)ncc(C#N)c1N C(=O)(CC(C=C)CCC)NCCSCCOCCCN(C(=O)OCC)C N1(NC(C(N2CCC(C)C2)=O)=O)CCN(C(C2C3CCC23)=O)CC1 c1(C(=O)Nc2scc(-c3cc(C)oc3C)n2)c[nH]c2ncc(Br)cc12 C1(CC(=O)N(C)Cc2ccn(C)n2)C2CCCC2N1C(c1cn(C)cn1)=O c1(C(=O)NC2CC3CN(C(COCCC)=O)C(C2)C3)ccc2c(c1)C(=O)NCC2 CCC(C)CC(=O)N(C1CCCN(C(=O)Cc2cnn(CC)c2)C1)C C1=NC(NCCS(=O)C(F)(F)F)c2ncnn2C1 c1(C(N2CC(n3cc(-c4c(C(=O)OCC)n[nH]c4)nn3)C2)=O)c(C)cccc1Cl C1(C(N2CC(CNC(=O)CNC(=O)NC3CC3)C2)=O)C(Cl)(Cl)C12CC2 N1(C(c2cc(C)[nH]n2)=O)C(C)C2CC1C2NC(=O)C(C)(F)CC1CCCC1 C1(C(=O)NCCCCC(C)NC(CCc2nc(C)c(C)o2)=O)CC1C1CCCC1 C1(NC(C=C(C)C)=O)CS(=O)(=O)C12CCN(C(C1C(C#N)C1(C)C)=O)CC2 C1(CCNC(c2cnc(C(C)C)[nH]2)=O)CSCCN1C(c1cc(Cl)ccn1)=O CC1(C)COCCC1NC(=O)C=CC1CCCN1C(=O)CNC=O C(=O)(C1CCCc2ccc(O)cc21)N1CCN(C(c2nc(C)oc2)=O)CC(O)C1 c1(C(=O)NCC2CC(COC)CN2C(C2CCOC2)=O)ccc2c(n1)OCCO2 N1(C(CCCCOCC)=O)CCC=C(C(=O)N(CC(C)C)CCO)C1 C(=O)(N=c1ccnc2[nH][nH]cc1-2)C1C(C(NC2CCc3ccccc32)=O)C1 C(=O)(C(C)C(C)NC(c1cnnc(C)c1)=O)Nc1occ(C)c1 N1(C(C=C(C)Cl)=O)CCC(n2cc(CNC(C34CSCC3C4)=O)nn2)CC1 c1(CN(C(=O)C(C)NC=O)C)cnn2c1CN(C(=O)CCCc1nccs1)CC2 C(=O)(C1CCCn2cc(C)nc21)NC(CC)CNC(C1(O)CCCCCC1)=O N1(C(C2(NC(C)=O)CC2)=O)CC(NC(=O)C(C(C)C)NC=O)CC1C c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC2C)cnc(Cl)cc1N N1(C(c2ccc(C)s2)=O)CCN(C(=O)C(C)c2ncco2)CC1C(F)F c1(N2CCC(C(C)C)C2)nc(NCC(C)Cc2ccc(Cl)cc2)nc2c1CCC2 c1(C(=O)NCC(CNC(=O)CCOc2ccccc2O)OC)coc2c1CSC2 c1(OC)ccc(C(=O)NC2(CCNC(=O)C3=NOC(C)C3C)CC2)c(F)c1Cl CC(C)C(CO)C(=O)NC(CNC(c1cc(F)cnc1Cl)=O)CC(F)(F)F N1(CC)CC(C(N2CCC(N(C(=O)CC3(OC)CCCCC3)C)C2)=O)CCC1=O C1(C(=O)NCC2C(NC(=O)CCc3ccc(F)cc3F)C2)CCC2(CCC2)CC1 C(=O)(CCC(C)(C)F)NC(CNC(c1ccc(NC(=O)OC)cc1)=O)CO CC1=C(C(=O)N2CCN(C(=O)CCCOc3ccccc3)C3CCC23)CCCC1 C12(CNC(=O)CSC(F)(F)F)CCCC1CCN2C(=O)Cn1ccc(O)nc1=O N1(C(CCC=CC)=O)CCC2(CCC2NC(c2ccn(CC(F)(F)F)n2)=O)CC1 Cc1nc2ccccc2cc1C(=O)N(C)CCNC(C1CCC(O)C1)=O O=C(C1=NOC(C2(O)CO2)C1)NN1CC(c2ccc(F)cc2F)C1 C1(SCC(=O)NCC2C(NC(C3CC(CN(C)C)C3)=O)C2)CCOC1=O c1(OC(C2CCCC2)CN(C)CC)ccc([N+](=O)[O-])cc1C c1(CC(=O)NC2CN(C(C3(COC)CC=CCC3)=O)C2)ccc(S(C)=O)cc1 Cc1nc(CC(=O)NCCC2CCC(NC(c3cc(F)cs3)=O)C2)cs1 N(C(=NCCC(C)(C)C)NC1CCC2(CC2)C1)CCSC c1(C(=O)NCCN(CC(C)O)C(=O)Cn2ncnn2)c[nH]nc1-c1cnn(C)c1 N1(C(c2[nH]cc(C)c2)=O)CCC(NC(c2cc3n(n2)CCC3)=O)C(F)C1 C1(NC(c2cc(CCC)on2)=O)CCN(C(=O)Cc2cc(F)ccc2C)C(C)C1 S(=O)(=O)(c1cccc2c1NCCC2)N1C(C)C(C)N(C)CC1 C1(C(=O)NC2CC(CCNC(c3c(SC)cn(C)n3)=O)C2)CC2(C1)CS(=O)(=O)C2 n1(CC(=O)NCCCCNC(CC2C(C)CCCC2)=O)cnc([N+](=O)[O-])n1 CC(CN(C)C)CC(=O)NC1CC(CC(=O)NCCc2cccs2)C1(C)C Cc1cccc(N(C(c2cc(Br)ccn2)C(=O)NCCCC2CC2)C)c1 C(=O)(CCCC(C)(C)NC(=O)CCc1cncs1)NCC1(CC)CCOC1 C1(CNC(c2c(C)nccc2)=O)CCC2CN(C(C3CC(=O)C3C)=O)CC12 n1(C2CN(C(=O)OCC3N(CCC#C)CCC3)C2)ncc([N+](=O)[O-])n1 CC1(O)CCC(C(=O)NCCCNC(c2cc[n+]([O-])cc2)=O)CC1 C1(NC(C2CCN(C)C2)=O)CN(C(c2ccncc2N)=O)CCC1O C(=O)(CC(CC)C(C)C)NC(CCN(C(c1ccc(OCC)nc1)=O)C)C(C)C N1(c2n(Cc3ccccc3)c(C3CCCCO3)nn2)CCCC(O)CC1 C1(CCCC)CN(C(c2cc(C(F)(F)F)n[nH]2)=O)CCN1C(=O)C(O)CCSC c1(CC(c2cnn(C)c2)C)nccc(=NCC(O)CN2CCC(COC)CC2)[nH]1 C12(NC(c3cc(C)n(C)c3)=O)CCCC1N(C(C1CCc3nn[nH]c3C1)=O)CC2 C1(OC)CC(C(N2CCC(N(C(=O)Cc3ccns3)C)C2)=O)N(S(C)(=O)=O)C1 c1(OC)coc(C(=O)NCC2CC2CNC(=O)Cc2ccccc2O)cc1=O C(C)(C(=O)N=c1ccn(CC(=O)NC2CCCC(C3CC3)C2)[nH]1)OC(C)=O c1(-c2cn(CCC3(C)CCN3C(=O)C(F)(F)CF)nn2)cccc(C#N)n1 c1(OC)ccc(C(N2CCOCC(CNC(c3sccc3C)=O)C2)=O)c(OC)c1 C1(C(=O)NC(CCC)C)CCCN(C(c2cnn(C)c2N)=O)C1C N1(C(c2onc(COC)n2)=O)CC(NC(=O)C(O)C(F)(F)F)CC2(CCC2)C1 CC(C)C(O)C(C)C(=O)NCCOCCC(N1CCCC1C)=O C1(S(=O)(=O)NC23CNCC(CC)(C2)C3)(C(=O)OCC)CC1C CC1CC2CN1C2=O.c1(CNC(C2CCCC2)=O)cnccc1Cl N1(C(C(C2CCN(C(CN(C3CC3)CC)=O)C2)C)=O)CC(C)(C#N)C1 Cc1cnc(NCC2C3CCCC23)[nH]c1=N N1(C(CCC#C)=O)CCCC2(C1)C(NC(=O)CCC1CCCCC1)CCN2C c1(N2CCN(Cc3c(C)nc(C)[nH]3)CC2C)ncnc2cnn(C)c12 C(C(C)(C)CNC(=O)OC(C=C(COC)C)=O)NC(=O)CC(C)SC N1(C(C(CCC)CCC)=O)CCC(C2CCCN(C(c3cncn3C)=O)C2)CC1 C1(C(=O)NCCCNC(CCSCCC)=O)CCCN1C1CCCC1 c1(OC)cc(Cl)c(C)cc1C(=O)NCC1CC1NC(=O)C=C1CC1 CN1CCN(CC(=O)NCCC2CN(C(C3(C(F)F)CCCO3)=O)CCO2)CC1 C1(NC(=O)Cc2cccs2)CN(C(c2ccn(-c3ccc(F)cc3)n2)=O)C2CC12 c1(C(=O)NCC(n2cc(CC(C)(O)CC)nn2)CC)cccc2c1oc(=O)n2C C(CC(C)C(=O)NCC(CO)NC(c1cccn1Cc1ccccn1)=O)OC C=CC1(CN(C)CC2CN(C(C3(NC(C)=O)CC(F)(F)C3)=O)C2)CCCCC1 CC1C2CCC(C2)C1C(=O)NCc1nc(C(=O)N(c2ccccc2)C)co1 N12CCC(C3CN(C3)C(=O)C3C(C3)C1=O)CC2.C1(C(=O)OCC)CN(C(C)=O)C1 N1(C(CCC=CC)=O)CCC2(CCN(C(=O)COC(F)F)CC2)C(C)C1 c1(CC)ncoc1C(=O)N(CC(=O)N(CC(O)CO)C)CC(C)C c1(C(=O)NC2CCCC(NC(CNC(C)=O)=O)C2)cc(OC)c2nc(C)cn2c1 C(c1cc2ccccc2o1)=CC(=O)NC1CCCCN(C(=O)C2=COCC2)CC1 C1(C(=O)NCCC2CCN(C(c3cc(OC)no3)=O)C2)CCC2(CCCCC2)C1 c1(C(=O)NCCCCCn2cc(COC(C(=O)OC)C)nn2)ccc(Cl)cc1Br c1(CC)nc(=N)[nH]cc1C(=O)NC(CCNC(c1cc(Cl)cnn1)=O)C(C)C C(=O)(CC(C)CC(C)(C)C)NCC(C)(C1CCC1)NC(C#CC(C)C)=O CCC(C)CC(=O)C(=O)NC(COC(C)C)C(=O)NC1CCC2CC1CO2 C1(C(=O)Oc2n(OC)nc(C3CC3)c2)CCC2C(N1C(=O)OC(C)(C)C)C2(F)F c1(NC(C)=O)ccc(Cl)c(C(=O)NC2C=CCN(C(c3cnc(C)[nH]3)=O)C2)c1 CC(C)(CNC(=O)C(CCF)NC(=O)CC1OCCCO1)C(F)F CC1CN(C(c2nccc(N)c2Cl)=O)CCC1NC(C1CC(=O)N(C)C1)=O C=CCC(C(=O)NCC(C(C)C)NC(C1CCCC1CC)=O)N(C)C C(C1CCN(C(C2(F)CCCOC2)=O)CC1)=CC(=O)NC(c1cccnc1)CO c1(C(N2CC3(CCN(C(C4CC=CCO4)=O)CC3)C2)=O)ccc2ccccc2c1 C=C(Br)CCC(=O)NCC1(COC)CCN(C(c2cn(C)c(O)n2)=O)C1 N1(C(C2C(C)(C)C2(F)F)=O)CC2CCCC2C1C(=O)Nc1conc1C(C)(C)C c1(C(=O)OC)c(C(=O)NCCN(C(C2CCCCC2)=O)CC2CCCC2)csc1C C1(C(=O)NCC)CCCCCC1NC(C1CC1C(C)(F)F)=O CC(CC(=O)N(C(C)CCNC(c1[nH]ccc1C1CC1)=O)C)c1ccco1 C1(C(=O)NCCC(=C)CNC(=O)CC2CCC(C)(C)CC2)CC2CCC1CC2 Cc1c(N)ccc(C(=O)NC2CCCC2NC(C2CCS2(=O)=O)=O)c1C C1(C(=O)NCC=C)CC(F)CN(C(=O)CC2CCCC3CC23)C1 C1(NC(CC(N2CCCCC2=O)C)=O)CN(C(=O)Cn2cnnc2)CC1N=[N+]=[N-] c1(-n2cc(C(C)O)nn2)ccc(CCNC(=O)CCc2ncc(F)cn2)cc1 CC(C)CC(C(=O)NCC1COCCN1C(C1CCCOCC1)=O)n1ccnc1 c1(C(=O)OC)ccc(CNC(C2CCN2Cc2ccc(SC)o2)=O)cc1 CCC(CC(F)(F)F)C(=O)NC12CC(NC(c3cnn4c3N(C)CC4)=O)(C1)C2 Cc1ccc(N2CCCCC(CNC(C3C4CCCC34)=O)C2)c([N+](=O)[O-])c1 C(=O)(CC(F)(F)C(C)C)N1CCCC(CNC(c2nc(C)sc2)=O)C1 Cc1cc(C(F)F)nn1CC(=O)NC1(CNC(C2(C)CCC(=O)C2)=O)CC1 c1(-c2cncc(C)c2)cccc2c1CN(C(c1ccc(Br)cc1I)=O)CC2 N1(C(C2ON=C(C(C)C)C2)=O)CCCC2CN(C(C3CCCS3)=O)CCC12 C1(NC(CCCC(C)=O)=O)CCN(C(=O)C=Cc2ccc(C(F)F)o2)CC1(C)C C1(C(C)NCC2CCCCN2S(C)(=O)=O)COC(C)(C)O1 c1(NC(c2cc(Br)ccc2F)=O)cc2ccccc2nn1 c1(C(=O)NCCCC(C)(C)NC(c2cncc(C)n2)=O)cc(C)c(C)nc1O c1(C(C)C)ccnc(NC(=O)CCc2cc(Br)cnc2Br)c1F c1(C(C(=O)NCC(CO)NC(C=CCCC)=O)C)ccc2ccccc2c1 N1(C(CCCOC(C)C)=O)CCC(NC(=O)C(C)CC2CC2)CC(C)(C)C1 C1(C)(C(N(C2CC3CCC2CC3)C)=O)CC12CCN(Cc1ccccc1)CC2 C1(N(C(C(C2CCC2)OC)=O)Cc2ccccc2)CCN(CC2CCOC2)CC1 C12(CNC(C(CO)N(C)C)=O)CC(C1)C(NC(c1ccsn1)=O)CO2 N1(C(C2(C)CCCS2(=O)=O)=O)CCCCC(NC(=O)CCSCC(N)=O)CC1 c1(C(N2CC(CCCCNC(C(C=C)(F)F)=O)C2)=O)ccc([N+](=O)[O-])c(C#N)c1 c1(SC)ncc(C#N)c(N2CC(NC(c3ccoc3)=O)C3(CC3)C2)n1 C(C1=CN(C(=O)OC(C)(C)C)CC1)=CC(=O)N(C(CCNC(C=NOC)=O)C)C C(=O)(C#Cc1ccccc1)N1C(C)(C(N2C(CNC(C)=O)CC(O)C2)=O)CCC1 C1(NC(c2cc(C)no2)=O)CC2CN(C(=O)Cc3c(F)cccc3Cl)CC2C1 CC1CN(C(c2c(Cl)cnn2C)=O)CCC1CNC(=O)CN(S(C)(=O)=O)C N1(C(C2(CCNC(C(CCCC)O)=O)CCCC2)=O)CCN2CC(C)CC2C1 N1(C(C2N(C(CCc3ccc(C(=O)OC)[nH]3)=O)CC(F)C2)=O)CCOC(C)(C)C1 C(C(CNC(c1cnsn1)=O)C(F)(F)F)NC(c1ccc(-c2ccco2)s1)=O c1(C(=O)NCC2CCN(C(c3c(CC)cno3)=O)CC2O)ccc2oncc2c1 CC(F)(F)CCC(=O)NC1CCCC1NC(c1cnsn1)=O S(=O)(=O)(c1c[nH]c2ccc([N+](=O)[O-])cc12)N1CCN(c2cc(C)[nH]c(=N)n2)CC1 c1(C(=O)NC(CC(C)NC(c2cnnc(O)c2)=O)C)ccnc(CO)c1 CC(C)C(O)C(F)(F)C(=O)NCC1(C)CCCN(C(=O)CSCc2cccs2)C1 n1(C(C2CCC2)C)nc(-c2ccoc2)nc1-c1ccc(-c2ccccc2F)n1C C(=O)(C(CO)C(C)(C)C)N(C)CC1CCCCN1C(c1cnc(O)o1)=O CCCC(C)(O)CC(=O)N(C)CC=CC(N1CCOCC(C)C1)=O c1(NC(CCC)CO)ccc(S(=O)(=O)NCCC2(C)CC2(F)F)c(Cl)c1 c1(NC)ccc(C(F)(F)F)cc1C(=O)NCC1CCCN(C(C2CCCO2)=O)C1 C(=O)(C(COC)C(F)(F)F)NCC1CC(NC(C2C(CCC)CCC2)=O)C1 c1(OC)cccc(C(=O)NC(C2CCCCN2C(=O)CNc2ccccc2)C)c1 c1(N(CC(N2CCCCC2)C2CCC2)C)nccc(=NCCN(C)C)[nH]1 C1(CC(=O)NC2CCN(C(=O)CCCC3CC3)C2C2CC2)CC2(CCC2)CO1 c1(C(=O)NCC(CNC(CC(C)N2CCCC2=O)=O)C)ccc2sccc2c1 C(=O)(C(C)(CC#C)NC(=O)CC1C=CCCC1)NCC1(C(=O)OCC)CC1 C1(COC)(NC(c2cc(OC)ns2)=O)CCCN(C(c2ccc(C)n2C)=O)C1 C(CC(C)(C)C(=O)N1CC2(NC(=O)C(C)OC3CCCCC3)CC1C2)SC N1(C(c2cc(CC)c(F)cc2)=O)CCC2(CC1)CC2NC(=O)C=Cc1cn[nH]c1 c1(NC)ccccc1C(N1CCC(C(C)CNC(c2cnc(C3CC3)[nH]2)=O)C1)=O N1(C(C(=O)NC(c2cc(O)cc(Br)c2)C)=O)CCC(=C(F)F)CC1 Cc1cc(NC(=O)CN(C)C(c2ncnn2C)=O)ccc1O c1(CC(=O)NCCN(C(c2c(F)cc(C)cc2F)=O)C)cn2cccc(C)c2n1 N1(C(CCCN(C)C(C2CCCN2C(N)=O)=O)=O)CC(C(N)=O)C2(CCC2)C1 CC1(CC(N2CCCC2CCC(N2CCCC2CC(N)=O)=O)=O)CCCC1 C1(CNC(C(COC(C)C)(C)C)=O)CCN(C(C2CC2C(N)=O)=O)C12CC2 S(=O)(=O)(C1(CSc2cccc(Cn3cncn3)c2)CC1)NC C12(C(N(C)CC3CCN(C(c4ccc(C#N)[nH]4)=O)CC3)=O)CCC(C)(C1)OC2 N1(C(C2C(CNC(C=C(CC)CC)=O)OCC2)=O)CCOCC1CCC CCS(=O)(=O)CC(=O)N1C2CN(Cc3cccc(C)c3O)CC12 N1(C(c2cc(C(C)=O)[nH]n2)=O)CCC2(CC1)CC2NC(=O)CC1CCC1 n1(CC(N2CCOCC2)=O)cnc([N+](=O)[O-])n1.n1(C)cc(CCC)nn1 c1(C(C)C)noc2ncc(C(=O)NC(C)CCNc3ncnc(O)c3Br)cc12 C1(NC(Cc2c(C)occ2)=O)CCCN(C(=O)Cn2cccnc2=O)CCC1 N1(C(CSCC)=O)CCOC(C(C)NC(c2csc(CCCOC)n2)=O)C1 c1(C(N2CCCC(N(C(C(=O)NCC)=O)C)C2)=O)cc2c(C)cc(OC)cc2[nH]1 CC1CN(C(c2sc(Br)c(Br)c2F)=O)CCN1C1CC1 c1(OC)ccc2c(=NC(C)c3cnsc3)[nH]c(=NCC3CC4CCC4C3)[nH]c2c1 c1(C(=O)NC2C(CNC(c3ccnnc3)=O)C2)csc2nccn12 c1(C(N2CC(NC(C3C(CC)CCO3)=O)C(C)C2)=O)c(N)cc(Cl)cc1F C(C)(C)(CCNC(=O)CSCC(C)C)NC(C(C1CCC1)OC)=O c1(CC)nc2cnc(NCC(C)CC(C)CC)nc2[nH]1 C(CN=c1[nH]c2c(c(=NCC3COCC(C)O3)[nH]1)CCC2)c1nc(C)oc1C Cn1c(C(=O)NCC2CN(C(C3CS(=O)(=O)C3)=O)CCO2)cnc1Cl c1(OC)cc2[nH]c(C(N3CC(C)CCCC3CO)=O)nc2cc1OC CC1CCN(C(=O)CC2CC(F)(F)C2)CC1CC(N1CCCN(CCO)CC1)=O c1(C(=O)NC(C(=O)N(CC=C)CC=C)c2ccoc2)ccnnc1O c1(C(=O)NC(C)(CNC(=O)Cc2c[nH]ccc2=O)C2CC2)ccc2snnc2c1 C1(C)(CNC(C2C(OCC)CCC2)=O)CCCN(C(c2conc2CC)=O)C1 c1(OC)ccc2c(=NCc3ccc[nH]3)[nH]c(=NCc3csc(O)n3)[nH]c2c1 Cc1cc(CN2CC3CN(C(c4cc(C(C)C)[nH]n4)=O)CC23)ccc1O CC(=O)CCCC(=O)N1CCCC(C(C)NC(=O)C(O)Cc2cnc[nH]2)C1 C12(NC(C(=O)N(CCNC(C)=O)F)C)CC(CO)(C1)OC2(C)C.S(C)(=O)(=O)N N1(C(C(CCC)NC(N)=O)=O)CCN(C(C2CN(C)C(=O)N2)=O)CC1CO c1(C(N2C(C)(C(=O)NC(C3(CO)CC3)C)CCC2)=O)ccc2cncn2c1 c1(C(=O)NC2CC(O)CN(C(=O)Cn3cnnc3O)C2)cccc2cc[nH]c12 CC(N=c1ccc(C#N)n[nH]1)C1CCCN(C(=O)C=CCN(C)C)C1 N1(C(c2cc(C)c(F)nc2)=O)CCC(C2CC2)C1CNC(c1c(C)noc1C)=O c1(N(c2ccccc2)C(=O)CCc2cnoc2)ccc(C(=O)CF)cc1 C1(CC(=O)N(CCC)CCNC(c2cc(C(F)(F)F)no2)=O)CN(C)CC1O c1(OC)cc(C)c(CN2CC(C(=O)Nc3nc(Br)c(Br)cc3Br)C2)cc1OC c1(C(=O)NCC2(C)C(C)CN(C(c3cc(C)sn3)=O)C2)cc(Cl)c(N)c(Cl)c1 c1(OCC)nccc(C)c1C(N1CCC(NC(c2csnc2Cl)=O)C(O)C1)=O C1(C(=O)NCC2(C)CC(=O)C2(C)C)CC2(C1)C(C(=O)OC(C)(C)C)C21CCC1 C1(C(=O)NCc2nc(-c3ccc(C)s3)sc2)CCCN(C(=O)C2=NOC(C)C2)CC1 N1(C(c2ccn(C)n2)=O)CCN(Cc2cnco2)CC1Cc1ccccc1 CCCN=C(NCC(C)Oc1ccccc1)NCC1CCCSC1 c1(C(=O)NC2(C)CCN(C(=O)C(Cl)=CCl)C2)cc2c(Cl)cncc2s1 CC1(C(=O)NCC2CCCC2NC(=O)CNc2ccc(Cl)cn2)CCC(=O)N1 N1(C(CC=C(C)C)=O)CCC2CN(C(c3cc(S(C)(=O)=O)cs3)=O)CC2C1 N1(C(c2c(CC)scc2)=O)CCN2CCOCC2(CNC(=O)CC2CC23CC3)C1 c1(CSCCOCC(=O)OC)cn(C2c3c(Br)cccc3OC2C)nn1 N1(C(CC(=C=C)C)=O)CCC(O)(C2(NC(c3cn(C4CC4)cn3)=O)CC2)CC1 C(c1ccncc1)=CC(=O)N(C1CCC(NC(c2cncn2C(F)(F)F)=O)C1)C c1(C(C)C)ccc(S(=O)(=O)N2CCC3CCCCC3C2)cc1 C(=O)(C(F)(F)CC(C)C)NCC1CCC(NC(C(C)=C2CCC2)=O)C1 C#CCCC(O)CCNC(=O)C(C)(C)CNC(C1CC=CCC1)=O C1(OC)COCCC1C(N1CCC1CNC(=O)CCCNC(N)=O)=O C1(CCC)(NC(=O)COC(C)CC)CCN(C(C2CCOC(=O)N2)=O)CC1 Cc1n[nH]cc1CC(N1CCC(N(C(C2CCOC2C2CC2)=O)CC2CC2)C1)=O C1(C#N)(CNC(C(C2CCN(C(C3C(C)CC3)=O)C2)F)=O)CC(C)(C)C1 C1(C(=O)NCC2OCC(CNC(c3ccc(OC)s3)=O)C2)COCCC1(F)F N1(C(C2C(=C)CC2)=O)CCC(CO)C(NC(=O)CSCC(c2ccccc2)=O)C1 C(CN=C(NCc1ncc(C)s1)NC1CC(c2cc(F)ccc2F)C1)OC Cc1cc(=NC(=O)C(=O)N2CCC(NC(=O)Cc3nn(C)cc3Cl)C2)[nH]o1 c1(CN2CC(C(=O)Nc3c(OCC)cc(Cl)cc3)C2)ccc(OC)c(C#N)c1 n1(CC)ccc(C(N2CCOC(CCNC(c3ccc(Cl)[nH]3)=O)C2)=O)c1C c1(C(=O)OC)cn(C)nc1C(=O)NCC1(NC(C2CCCC2(C)C)=O)CC1 c1(C(=O)NCC2(CNC(C3C(CN(C)C)C3)=O)CC2)cc(Cl)no1 N1(C(c2cc(CC)no2)=O)CCC(O)(CNC(C23CCC(CC2)O3)=O)C1 CC(C(C(=O)NC1CCOCC1)N(C1CC(=O)NC1=O)C1CC1)C(C)(C)C N1(C(c2c(C)nsc2)=O)CCC(O)(CN(C)C(c2cc(C(C)(C)C)n[nH]2)=O)C1 c1(OC)cc(N)ccc1C(=O)NCC1(CO)CCN(C(C2C=CCS2)=O)C1 Cc1nn(C)c(C)c1CC(=O)NCc1ncccc1CNC(=O)CC1CCCO1 CC(C(=O)NC1CC1CNC(c1cc2c(s1)CCC2)=O)C(C)(C)C C12(NC(=O)CCC34CCC(CC3)C4)CCOCC1CN(C(=O)C(F)(F)C(F)F)C2 Cc1cc(F)cnc1C(=O)NC12COC(C1)C(NC(c1ccncc1F)=O)C2 c1(C(=O)NC2(C)CC(NC(C3CC4CC4C3)=O)C2)cc([N+](=O)[O-])c(Cl)cc1Cl CC1=NC(C(=O)NCCCOCCNC(c2ocnc2C(F)F)=O)CS1 c1(CC)cnc(O)c(C(=O)NC2CCN(C(=O)CNS(C)(=O)=O)C2C)c1 N1(C(c2ccc3nc(C4CC4)sc3c2)C)CCCC2CCCN(C)C12 N1(C(C2(C(=O)OCC)CCC2)=O)CC(NC(=O)C(C)C(F)(F)F)CC(F)C1 C1(C(N2C(C(=O)NC3CCC(O)C3)CC3CC32)=O)CCc2ccccc2C1 N1(C(c2cc(CNC(C(=Cc3cccnc3)C)=O)sc2)=O)CCC2CN(C)CC2C1 c1(COC)cncc(C(=O)NC2CCCC2NC(=O)CCC=CC(C)C)c1 C=CCCCC(C(=O)NCCCc1cnn[nH]1)NC(c1noc(CC)c1C)=O N1(C(C(c2n(C)ccc2)=O)=O)CC2CC2(C(N2CCOCC2CN(C)C)=O)C1 C(=O)(C1CCCc2nn[nH]c21)NCCOCCNC(Cc1cc(C)c(O)cc1)=O C1(NC(CC2C(Cl)(C(=O)OC)C2)=O)CCC(NC(=O)CSCC(N)=O)CC1 C1(NC(C(CSC)C)=O)CCCN(C(c2cc(C3CCOCC3)no2)=O)C1 N1(C(C(=O)NCCOC)c2cc[nH]n2)CC(C)C12CCOCC2 N1(C(CCCC2C(C)C2)=O)CCC(C)(CNC(=O)Cn2nnc(C3CC3)n2)C1 c1(C(N2CCC(CN(C)C(C3CCC(=O)N3C)=O)C2)=O)ccnc2[nH]c(O)nc12 C(CCC(F)(F)F)N(C)CC1CCCN(C2CCC(N)CC2)C1 Cc1cccn2cc(CC(=O)NCC(C(C)C)NC(C3CC(C#N)C3)=O)nc12 N1(C(C2CC2c2ccc(Cl)cc2)=O)CCC2(CCCN2C(C2CCCCS2)=O)C1 N1(C(C(CC)O)=O)CCc2c(CNC(=O)CC3COC(C)(C)C3)cccc2C1 C(CC(O)C(=O)N1CCC(C=O)(CF)C1)SC.N12CCC(C1)C2.C(C)(=O)OCC C1(CC(=O)NCC2CC(NC(=O)CCN3CCC3)C2)(OC)CCC1 c1(C(N(C2CCN(C(C3(CCCC)CC3)=O)C2)C)=O)ccc(Cl)cc1C c1(C(=O)NC2CC(C)(NC(c3n(CC)ccc3)=O)C2)cc(C)c(C)nn1 c1(C(=O)NC2CC3CC(NC(C4CC(C)C4)=O)C3C2)cnc2c(F)cccc2c1 c1(NC(C=CC(N2CC(NC(c3ccccc3)=O)C2)=O)=O)n[nH]cc1C(F)F N1(C(CCSC)=O)CC2CC1CN(C(C1OCCC1C(C)C)=O)C2 c1(C(=O)NCC2(CNC(C(CO)OC)=O)CC2)[nH]c(C)nc1C CC1OC2(C(=O)NCC3(NC(C4CC(C5CC5)C4)=O)CC3)CC1C2 c1(C(C)C)cc([N+](=O)[O-])ccc1C(=O)NC1CCC(CNC(c2cscn2)=O)C1 C(=O)(CC1=NNC(=O)C1)N1C(CCCC)CN(C(C2(C)CCCS2(=O)=O)=O)CC1 C1(N(C(C(C)(N(C(=O)CCC2CCCCO2)C)C2CC2)=O)C)CCC2(CC1)CC2 C(CCN=C(NCCC1CC1OC)N1CC(C)N(C)C(C)C1)SC c1(C(C)NC(C2(C3(C4CCCO4)CC3)CC2)=O)ncc(Cl)cc1Cl c1(C(N2CC(C(C(=O)NCC(c3ccccn3)O)N3CCC3)C2)=O)cccnc1S C(=O)(CCC(C)(F)F)N(C1CCN(C(CC(C)O)=O)CC1)Cc1ccccc1 N1(C(CS(C)(=O)=O)=O)CC2CC(O)C1C2NC(=O)CNC(C1CCC1)=O C(=O)(CCC(C)SC)NCCNC(C(n1cc(CSC)nn1)C)=O N1(C(C2(F)CCN(C(CC(CC)C)=O)C2)=O)CCC(CO)C(C)(C)C1 c1(C(N2CC(Cn3cc(CSC)nn3)C2)=O)ccc(OCCO)nc1 c1(CC(=O)NC(CNC)C)cc(Cl)cc(Cl)c1F CCCCC(C)C(=O)N(C1CC2CCC(C1)N2)C(C)(C)C(N)=O C1(NCC(=O)NC(C#C)C(C)C)CCN(C2CCCC2O)CC1 CC(C)CC(CNC(=O)C=CCN1CCCC1)C(=O)NCC1(C2CC2)CC1 C1(CNC(c2c(C)noc2N)=O)OCC2CCN(C(c3ccon3)=O)CC12 C12(CNC(CCCCC=CC)=O)CCC(CC1)N(C(=O)C(C)OC)C2 c1(CCC2CCC(C)C2)[nH]c(=NCC2(C)CCC(C)(C)CC2)nc2c1ncn2C C1(CNC2CC2)CN2CC3CC2(CO1)C3.Cc1cc2ccc1N1CCN2CC1 C1(NCCNC(c2[nH]cc(C#N)c2)=O)CCS(=O)(=O)CC1 N1(C(C2CNC(=O)N2)=O)CCC(CO)(CNC(c2cnc(Cl)s2)=O)C1 c1(C(=O)NCCc2cccc(C)c2)cc(Br)c(C)c([N+](=O)[O-])c1 C1(NC(c2ccc(CNC(c3cccc(C)c3)=O)cn2)=O)C(C)CCCC1C C1(CNC(C2(CCC=C)CC2)=O)CCN(C(=O)CCCCC=CC)CC1C c1(CC(=O)NC2C(NC(C(CC#C)O)=O)CC2)cccc2ccsc12 C1(CN(CCC)Cc2csc(C(F)(F)F)c2)CC(C2CCCCC2)CN1C c1(C(=O)NCCOC2CCN(C(c3c(C)snn3)=O)C2)ccc2c(c1)NCCC2 N1(C(c2c(OC)ccc(I)c2)=O)CCC2(CC1)CC(NC(c1nc(Br)cs1)=O)C2 N1(C(c2n(C)nc(O)c2)=O)CCC2C(C1)CN2C(c1nc(Br)c[nH]1)=O CC1CCC(C2CCC2)CN1c1ncnc2c1ncn2C1CCCCCCC1O CCCC(C)(CC)C(=O)N1CCC(=O)C(OCC(C)C)C1 N#Cc1ncc(C(=O)NC2CN(C(c3cncc(-n4ccnn4)c3)=O)C2)s1 N1(C(C2C=CC(NC(CSS(C)(=O)=O)=O)C2)=O)CC2COC(=O)C2C1 C1(C(=O)NCc2cc(C)sc2)CCN(C(=O)CCc2cccnc2)C12CC2 c1(OCCNC)ccc(C(=O)C(N)Cc2c(C)cccc2C)cc1Br N1(C(c2scc(C)c2)=O)CC2CCC2(CCNC(c2cc3ccsc3s2)=O)C1 C1(C(=O)NCC2(CS(C)(=O)=O)CCCCC2)CC2CCCCC2N1 N1(C(c2n[nH]c(C)c2O)=O)CCN(C(=O)C(C)CCN(C)C)CC(O)C1 c1(C(=O)NC2CN(C(c3n(CC)ccn3)=O)C(C)CC2)cnn2cnnc2c1 Cc1cccc(C(CNC(c2ccccc2O)=O)NC(c2cnn(C)c2F)=O)c1 Cc1cc(NC2(C)CCN(C(c3ccnnc3C)=O)CC2)c(F)cc1[N+](=O)[O-] C(=O)(C(C)C1=CCCC1)N(C1CC2CN(C(c3n(CC(C)C)ncc3)=O)C1C2)C c1(C(N(CC(C)C#N)C2CC2)=O)cncc(CNC(C2CC2C#N)=O)c1 C1(C)(C(=O)NCCC(CCNC(c2ncn(CC)c2)=O)C)CCC(C)=C(C)C1 CCCCC(C)CCC(=O)NCC1OCCC1C(=O)NC(C)C(=O)OCC c1(C(=O)OCc2c(C)noc2C)ccc(S(N)(=O)=O)cc1.c12ccccc1CO2 CC(C)(O)CC(=O)N1CCCC(NC(=O)Nc2cc(-c3ccnc(O)c3)on2)C1 N1(C(C(N2CCCCCC2)C)=O)CCCC(NC(c2cc(F)ccc2N)=O)CC1 C1(NC(COC(C)C)=O)CC2CN(C(c3cc(C4CC4)[nH]n3)=O)CC12 Nc1cnc(C(=O)NC23CCC(CC2NC(=O)CC2CCCCC2)C3)c(Cl)c1 C1(C(N(C)Cc2c(OCC)nccc2)=O)COc2cc(O)ccc2C1 C1(C(N2CC=CC(NC(C(CCC)NC(N)=O)=O)C2)=O)CC2(CCOCC2)CO1 C(=O)(CC(C(F)F)NC(=O)C(C)CC#N)NC(CCSCC)C N1(C(C=CCC)=O)CC(C(F)(F)F)OCC1CNC(c1occc1C1CC1)=O Cc1[nH]cc(C(=O)NC2CC3CCC2(NC(c2ccsc2)=O)C3)c(=O)c1Cl CN1CC2CCN(C(c3ccoc3CNC(c3sccc3CO)=O)=O)C2C1 C1(NC(c2cc(Cl)cs2)=O)CN(C(=O)C(F)(F)c2ccncc2)CC12CC2 Cc1ccn(C(C)C(=O)NC(C)C(CO)NC(=O)CN2CCOCC2)n1 c1(C(C)OC(=O)C(C2CCCO2)NC(=O)OCC(F)(F)F)ccccc1 CCC(CC(=O)NC12CC1CN(C(=O)CCc1ccc(F)nc1)C2)CC(C)C Cc1cc(O)c(C(=O)NC(c2ccccc2)CNC(=O)CCc2cn[nH]c2)nn1 C(CCC(C)(C)C(=O)NCC1CC(C(=O)NCC2CCCC2)=NO1)OC N1(C(CC(=C)C)=O)CC2(CCN(C(c3cnn(CC(F)(F)F)c3N)=O)CC2)C1 c1(C(C)=O)ccc(C(=O)NCC(C2CC2)NC(=O)CCn2ccc(=N)[nH]2)nc1 c1(C(N2CCC(O)(C(C)NC(C3(C)CCCN3C)=O)C2)=O)ccn(C)c(=O)c1 C1(C(=O)NCc2cc(C(=O)NCC(C)F)no2)COCC1(C)C N1(C(C(=O)Nc2c(C)c(Cl)ccn2)=O)CCc2ccsc2C1 C1(C(N(CCCCn2ccnc2)C)=O)(NC(=O)CC2CC3CC3C2)CCN(C)C1 N(C1CCCn2ccnc21)C(C1CCC(NC(=O)CCCn2cncn2)CC1)=O N1(C(C(N2CCC(c3c(OC)cccc3)CC2)=O)=O)CCCC2(CNC(=O)C2)C1 c1(CC(N2CC3C(CN(C(C(C)NC(CC)=O)=O)C)C3C2)=O)cccc(F)c1O CCC(C)(CNC(=O)C(Cc1cnc[nH]1)NC(c1ccc(=N)[nH]n1)=O)C(N)=O N1(C(C=C(C)c2cccs2)=O)CCC(C)C(NC(C2CCCS(=O)(=O)C2)=O)C1C C1(C(CCCOC)C(=O)N(C)C)CCCN(C(=O)C(=O)OC(C)=O)C1 C1(C(=O)NC2(CN(C(C(C=C)O)=O)C)CC2)CCc2nncn2CC1 C1(NC(=O)CC2CSCCO2)C=CCC(C(=O)Nc2ccc(O)nc2)C1 N1(C(c2cccc(OC)c2C)=O)CCC2C1CCCN2C(c1cnncc1C)=O CCC(CN(C)C)C(=O)NC(C(=O)N(CC(O)C1CC1)C)C1(C)CC1 C1(NC(C=C(COC)C)=O)CC2CCC1C(NC(c1csc(C)c1C1CC1)=O)C2 c1(C(C(=O)N(CCN(C(=O)C=Cc2cncn2C)C)C)O)cccc(F)c1 N1(C(Cc2nc(C)on2)C)CCC(O)C(C(=O)N(C(C)(C)CC(C)C)CCO)C1 C(c1ccccc1)=CC(C(=O)NC1CC(C)(NC(c2cc(C)on2)=O)C1)C c1(C(N2CCC(O)(CCNC(C3CC(O)C3)=O)CC2)=O)ccc2oc(S)nc2c1 c1(OC)cc(F)ccc1CN1CCC(C(F)(F)F)C1.C12C=CC(C1)C(=O)NC2 C=C(C)C1OCCC1CNC(=O)CN(CCOC)C(c1ncoc1C1CC1)=O CN1CC(C(=O)N(CCCCN(C)C(c2ccc(F)cc2)=O)C)OCCC1=O c1(C(N2CCC(C)(CNC(c3ccc(C(C)C)cc3)=O)C2)=O)cc2sccc2s1 N1(C(C2ON=C(CC)C2)=O)CC2CCCC1(CNC(=O)Cn1cccnc1=O)C2 C1(CC2CCC3(C(C)C)CC23)(OC)CCCOC1.c12nnnn1NC2(COC)C CCCCCC(=O)NCC(=O)NC(C)CNC(c1ccsc1Cc1nc[nH]n1)=O C(=O)(CCCC(F)(F)CO)N1CC(N(C(Cc2cccc(C)c2F)=O)C)C(O)C1 C(CC(O)C(=O)NCC1(F)CC(NC(c2cc(C(F)(F)F)ncn2)=O)C1)N(C)C c1(OC)cc(C(=O)NCC2CC3(C2)CN(C(=O)C(F)(F)C2CC2)C3)c(F)cn1 c1(C(=O)NC(C)CCCNC(C2COCCC2(F)F)=O)ccn2ncccc12 C(=O)(CCC(=O)Nc1nnc(CC)s1)NC1(NC(=O)CSC2CC2)CCCCC1 Cc1ccc(Cl)c(S(=O)(=O)N2CCC(Oc3ccccc3F)C2)c1 c1(C(=O)NC2CN(C(c3cc(Cl)ncc3F)=O)CC23CC3)cc(Br)cc(Br)c1O Nc1c(F)cc(F)c(F)c1C(=O)NC1CCN(C(C2(C3CCC3)CC2(F)F)=O)C1 CC1CCC(CNC(c2ccc(O)cc2)=O)N(C(=O)Cn2cc(C(C)O)nn2)C1 Cc1cnc2cc(C(=O)NC(CNC(=O)C(C(C)C)N(C)C)C(C)C)ccn12 c1(CC(=O)N(c2ccc(Cl)cc2)CCNC(C=CC)=O)ccc(F)cc1COC c1(C(C(=O)NCC(CNC(C)=O)C)C)ccc(Cl)c(Cl)c1.C(=O)(CC1CC1)OC Cc1cc([N+](=O)[O-])cnc1C(=O)NCC(C)NC(c1ccc2[nH]c(=N)oc2c1)=O C1(CNC(C=CC=CC)=O)CCC2(CN(C(=O)CC3CCCCN3C)C2)O1 C1(NC(CC2(OC)CCCC2)=O)CCN(C(=O)C=C(Cl)Cl)CCC1CO c1(NCCNS(=O)(=O)C(Cl)Cl)ccc(S(=O)(=O)C(F)(F)F)cc1 C1(CNC(CC(CC)C)=O)CCN(C(c2ccnc(C)c2)=O)C1(C)C c1(N2CCC(CCNC(CCCC#CC)=O)C2)ccc([N+](=O)[O-])cc1Cl CN(CCCC(=O)N1CC(CCNC(=O)CCc2cccnc2Cl)C1)N=O c1(C(N2C(C(=O)Nc3ncc(C(F)(F)F)cn3)C(O)CC2)=O)c(Cl)cncc1Cl c1(C(=O)NC(c2cccnc2)C(=O)N(CC)Cc2ccccn2)ccnnc1O C(=O)(C(C)(C)C1CCCCO1)N1CC(CNC(C=C(C)C(C)C)=O)C1 c1(CC(=O)NC2CCCN(C(C(C=C)O)=O)C2C)nc(F)c(F)cc1F Cc1cc(N)c(C)nc1N(CCNC(C1CC2CCC1C21CC1)=O)C(C)C n1(CC(N2C(CCN(C(C=CSC)=O)C)CCCC2)=O)cc(Cl)c(O)nc1=O c1(C(=O)NC2CC(CNC(C3(C)CC3(F)Cl)=O)C2)ccc(F)c2[nH]ccc12 c1(CNC(C2CCCN(C(C(CNC(=O)OC)(C)C)=O)C2)=O)cccc(F)c1O O=S(=O)(c1ccc(Br)cc1NCCCN1CCCOCC1)N1CC(CO)C(F)C1 c1(C(N2C(CN(C)C(C3CN4CCN3CC4)=O)CCC2)=O)cc(F)ccc1F S(=O)(=O)(c1ccc(NCc2cccc(Cl)c2)cc1Br)N(CCC#N)Cc1cnsc1 CCCCC(C)C(=O)NCC(O)CCNC(c1cccc(C(=O)NCCC)c1)=O C1(C(N2CCC=C(CNC(C3CC(=O)NC3)=O)C2)=O)CCC([N+](=O)[O-])CC1 N1(C(Cc2c(C)nc[nH]2)=O)CC2CCC1CN2C(c1cc(C(F)(F)F)nn1C)=O N1(C(Cn2c(CCC)ncc2)=O)CC2CC1CN2C(c1csc(C(C)OC)c1)=O c1(OC)cc(C)c(Cl)cc1C(=O)NCC(C)(C)NC(=O)Cc1ccsc1C CC(=NOCC#N)C(=O)NCC(C)C(=O)N(C)Cc1cocn1 C=C1Cn2c(C(N3CCC(CF)(NC(=O)C=CC4CCOCC4)C3)=O)nnc2S1 C(=O)(CC(C(F)F)C(C)(C)C)NC1C(C)(C)CN(C(=O)CCCC2CC2)C1 c1(CC(N2CCC(C)(C(=O)NCC(=O)N(C)C)C2)=O)ccc(Cl)cc1F c1(-c2nc(-c3cc(CC(C)C)on3)on2)ccc(S(C)(=O)=O)nc1 C1(NC(C2C(C)C2C)=O)CN(C(c2c[nH]c(-c3ccncc3)n2)=O)CC12CCC2 CCCC(C)CC(=O)NCc1cc(C)c(C(=O)N(CC(CC)OC)C)o1 C1(CNC(C(CC)N2CCCC2=O)=O)CC(C)(C)CN1C(=O)Cc1nnc(S)n1C c1(CC)ccc(CN(C(C(=O)NCc2sc(C3CCCCC3)nc2C)C)C)cc1 C#CC1(C(=O)NC2CCC(O)CC2)CCN(C(=O)CC2CC=CC2)C1 c1(NC(c2cncc(-c3ccc(OC)cc3F)n2)=O)cc(Cl)c(Br)cc1F Cc1ccc(C(N2CCC(C3CCCN3C(c3cnc(C)[nH]3)=O)C2)=O)o1 C(CC(C(=O)NCC(O)CN(C)C)NC(=O)CC1CCCCC1)=CC O=C(C1CCCc2scnc21)NC1CN(C(C2CCC3CC23)=O)C1 CN1CCCC1CCNC(=O)CC=CCNC(=O)C=CC1CCCC1 C1(CO)C2CCCC1N(c1ncc(I)cn1)C2.c1(OC)ccc2cc1CC(=O)N2 c1(C(=O)NCC2CC(NC(Cc3nc(=N)[nH][nH]3)=O)C2)cnn2ccc(O)nc12 c1(C(=O)NC)cc(CCC(=O)N(C(CCNC(C=CCC)=O)C)CC)oc1C c1(C(N(C2CN(C(c3ccc(C4CCCO4)[nH]3)=O)C2)C)=O)cc(N)cc(O)n1 c1(NCc2c(CSC)nccc2)nc2c(cc1C#N)CC(C)CC2 C1(CNC(c2c(C)nn(C)c2)=O)N(C(=O)CSc2nncn2C(C)C)CCC1(C)C CCCCCS(=O)(=O)CC(=O)N1CCCC(N(C(c2ccc[nH]2)=O)CC)CC1 C1(NC(C(CC)N(C)C)=O)CC(F)CN(C(=O)CCc2cn(C)cn2)C1 S(=O)(=O)(c1cnn(CC(F)(F)F)c1)NC(C(=O)NC)CC(C)C C1(C(N(CC(C)SC)C)=O)CCCN(C(=O)CC2COCC2O)CC1 N1(C(CC=C=C)=O)CCN(C(c2ccc(Br)c(C)c2N)=O)C(C)C1C C1(C(N2C(CNC(c3cnco3)=O)CC2)=O)COCC1n1cccn1 N1(C(C2CCC(CC)CC2)=O)CCOC(C(=O)NCCCCCCO)CC1 CC(C)(C)CCCCC(=O)N(CC(C)O)CCNC(C1(C)CC2CC2C1)=O C(=O)(C1CCc2c[nH]nc21)NCCC1(C(=O)NC(C)Cc2ccco2)CC1 C(=O)(CC(C)(C)CN(C)C)NC1(C)CCN(C(CC(C)c2ccncc2)=O)C1 C1(C)(C(=O)NCC2C(CC(=O)NC3(CN(C)C)CC3)C2)CC(O)CN1C c1(CC(=O)NC2CN(C(CC(=O)OC)=O)C2)cn2c(n1)CCCC2 C1(CC(=O)N(C)CCN2CC(C)(O)C2)C2CCC(C2)N1C(C12CC(CO)(C1)C2)=O c1(C(=O)OCCOC2(c3ccc(OC)cc3)CC2)nc(F)ccc1Cl C1(C(=O)Nc2cccc(-c3nc(COC(F)(F)F)on3)c2)CC2C=CC1CCC2 c1(C(=O)NCc2cnc[nH]2)cn2c(n1)CCN(C1CCS(=O)(=O)CC1)CC2 N1(S(CCc2c(OC)cccc2)(=O)=O)C2CCC1CC(N(C)C[Si](C)(C)C)C2 Cc1cn(C)nc1NC(c1ncccc1Cl)=O.C12(CCC1)CCC(=O)N2 C12(C(N3CCC(N(C(C(CC=C)C(C)C)=O)C)C3)=O)C3CCC(CC13)C2(F)F N1(C(c2c(N(C(CC)=O)C)cccc2)=O)CCCC(N=c2[nH]nc(O)s2)CC1 C1(NC(c2cn(CC)nn2)=O)CCCN(C(c2ccnc(CC(C)C)c2)=O)C1C Cc1cc(C(=O)NCCC(C)NC(C2CC2(Cl)Cl)=O)cs1 N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(=O)CC2CN3CCC2CC3)C(CF)C1 CCC(CC)OCC(=O)NCC1(C(=O)NCC(F)F)CC1 C12(CC(=O)NCCOCCCC)CCC1CN(C(c1ccc(F)cc1Cl)=O)C2 Cc1nc(Cl)ccc1NC(c1nc(C(=O)Nc2csc(-c3ccccc3)c2)cs1)=O c1(C(N2CCC(C)(C(N3CCC(C#N)C3)=O)C2)=O)cccc2[nH]ccc12 C1(NC(c2cc[n+]([O-])cc2)=O)CCC2(CC1)CN(C(=O)C1CCc3c[nH]nc31)C2 C(=O)(C(CNC(=O)CN1CCC(O)CC1)C(C)(C)C)NCC1C(C)COCC1 c1(C(=O)NCCNC(C=C(CC)c2ccccc2)=O)cn2ccc(OC)cc2n1 N1(C(=O)NC(CC=C)Cc2ccccc2)CC(C)(C)C(O)C(C)(C)C1 C1(C(=O)NC2(C(=O)NC(CC(=O)NC)C3CC3)CC2C)CCCCCC1 N1(C(c2ccn(C3CC3(F)F)n2)C(=O)NC2(C)CC2)CC2CC1CO2 N1(CC)CC2(CC(CNCCc3n[nH]c(C4CC4C(=O)OC)n3)CO2)C1 CC(C)CC(C(=O)N1CC(NC(C2CC23CCCCC3)=O)C2(CC2)C1)NC(N)=O c1(NC(c2cnc3n2CCC3)c2n(C(C)C)nnn2)cc(Cl)cc2c1OCC2 C1(NC(CCCC#C)=O)CC2CC1CN(C(c1cccc(F)c1Br)=O)C2 C1(C(=O)OC)C(C)CCN1C(C1(CCNC(=O)Cc2ccc(F)cn2)CC1)=O Nc1ccc(C(N2CCN(C(=O)Cc3cccs3)CC2)=O)nc1N c1(C(=O)NC2CCCN(C(=O)C=C(Cl)Cl)CC2)cnc2[nH]nc(O)c2c1 c1(CC(=O)OC)ccc2c(c1)CN(C(=O)C(=O)NCCN)C2 N1(C(=O)CCCC(F)(F)F)CCC2(COCCN2C(c2cc[nH]n2)=O)C1 c1(CC)c(C(N2CCOC(CN(C)C(c3[nH]cnc3C#N)=O)C2)=O)cnn1CC c1(C(N2CCCC(N(C(CCC(=O)NCC)=O)C)C2)=O)cn2c(C)cccc2n1 c1(C(=O)NCCc2c(C(N(CCC3CC3)CC)=O)c[nH]n2)[nH]ccc(=O)c1C Cc1ccc(C(=O)NCC2CCC(C(=O)N(C)C)O2)c(F)c1F CC1(C)CCC(C(N2CC(NC(C3CCC3)=O)C(CC3CC3)C2)=O)CO1 c1(CNC(=O)Cc2ncc(-c3ccccc3)o2)ccc(OC(F)(F)F)cc1 C1(CC(=O)N(C2(C(=O)NC3CCC4(CC4)C3)CC2)C)CC2CCC1O2 C1(NC(=O)NCCc2ncc(CC)s2)CCN(c2cc(C)nn2C)C1=O N1(C(c2c(C)[nH]cc2)=O)CC(N(C)C(c2ccc(-c3ccco3)s2)=O)C2(CC2)C1 c1(-n2cc(CCCCNC(C3CCC3c3ccncc3)=O)nn2)ccccc1 O(NC(=O)C(Cc1cn[nH]c1)NC(C1CC(=O)NC(C)C1)=O)CCCC#C N1(C(c2ccc(CO)s2)=O)CCN(C(c2ccc(-c3nncs3)cc2)=O)C2CC12 S(=O)(=O)(c1ccc(F)c(C(N2CCC(CNC(C)=O)(OC)CC2)=O)c1F)NC C(C)(CC#CC)NC(CCN(CC=C)C(C1CCNC1=O)=O)=O c1(OC)ncc(C)c(C(=O)NCC2CN(C(C3CC(=O)N(C(C)C)C3)=O)C2)c1Cl c1(NC(CCC(CC)NC(C2(C#C)CC(=O)C2)=O)=O)ccc2c(c1)OCC2 c1(C(N(C2CN(C(CCCN(CC)CC)=O)C2)C)=O)ccc(CC2CCC2)cc1 c1(C(=O)NC2CCCN(C(C(C)=C3CC3)=O)C2)cccc2[nH]c(=N)oc12 C(=O)(C(C(C)CC)N(C)C(C1CCCC(CF)C1)=O)NCCCCCC#C c1(C(=O)NC2CCN(C(c3ccnc(C)n3)=O)C(C)C2)cc2ccccc2o1 C1(CNC(c2ccon2)=O)CC(F)CN1C(c1ccc(O)nc1)=O C(CC(F)F)(C(=O)NC(c1nn[nH]n1)C1CC1)N(C(C1C(=C)C1)=O)C CC1(C(=O)NCC2CC2NC(=O)C(=O)Nc2ccc(Cl)cc2)CC(F)(F)C1 C(=O)(C1=NOC(c2ccccc2)C1)NCC(C)NC(C=C(CC)C)=O N1(C(C2N(C(=O)Cn3nccc3C)CCC(CC)C2)=O)CC2(CNC(=O)OC2)C1 Cc1cc(NC(C23CCC2C3)=O)ccc1NC(c1cc2n(n1)CCC2)=O C1(CC)C(=O)NCCN1C(=O)CCN(C(=O)CC=C(Cl)Cl)CCO c1(C(N2CC(C(=O)NCc3cc(Cl)ccc3Cl)OCC2)=O)c(F)ccc(Cl)c1Cl C1(C(=O)NCCCCCCNC(c2c(C)cccc2F)=O)CC2COCCN2C1 C1(CCC(C)(C)NC(=O)C(C)(F)F)CCCCN1C(=O)C=CC1CCCC1 c1(OC)ccc2occ(C(=O)NC(C3CCN(C(c4ncsc4C)=O)C3)C)c2c1 N1(C(CN(S(N(C)C)(=O)=O)C)=O)CCC=C(C(=O)NCC2(C3CC3)CCCO2)C1 c1(OCCC(=O)NCCCNC(c2c(N)nccn2)=O)ccc(F)cc1Cl N1(C(c2[nH]c(=NCC)sc2)=O)CCCC2(CC(NC(=O)CP(C)(C)=O)CO2)C1 Cc1cc(NC(C)(C)CNC(c2nnn(C)c2C(F)F)=O)nc(CC2CC2)n1 C12(NC(C3CSC3)=O)CCC(CC1n1cc(-c3ccsc3)nn1)C2 C1(C(N(CCCC)CCO)=O)CC12CN(Cc1ccc(C(F)(F)F)nc1)C2 C(C(CC)(CC)NC(=O)CN(C(=O)COC)C)NC(C1C(OCC)C1)=O C=C(C)CCCC(=O)NCC1CN(C(c2sccc2C)=O)C2CC12 N1(C(c2c(CC)occ2)=O)CC(O)(C2CCN(C(=O)CC3CC(CC)C3)CC2)C1 N1(C(CC(C)SC)=O)CC2(C=C(C(=O)N3CC4(CC(F)C4)C3)CO2)C1 C(C(=O)NCc1ccnc(C(=O)NCC(c2cccnc2)O)c1)(C(C)C)OC C1(NC(CC(CCC=C(C)C)C)=O)CS(=O)(=O)C2CN(C(=O)C3CC3)CC12 C1(C(N2C(C)(COC)CCC2)=O)CC(NC(=O)Cn2nc(C)cc2C)C12CCC2 CC(C)(O)C#CC(=O)N1CCC(N2CC(NC(=O)C=CC3CCC3)CC2=O)C1 Cc1nc(C(N2CCCC(C(N3CC(F)C(F)C3)=O)C2)=O)ccc1Br CC1CCN(C(=O)CN(C)C(c2cncn(C)c2=O)=O)C(C)C1 C1(CNC(COCc2cc(C)on2)=O)C(C)CCN1C(c1ccc(C#N)s1)=O C(CC)(CCC(=O)N1CCC(CC(C)C)C1)NC(C(CC)=CC)=O c1(OCC)ccc2cc1NC(=O)c1ccc(s1)CNC2=O.C1(COC)CC1(C)C C1(C(=O)NC(C2CCCCC2)C(=O)NCC2(SC)CCC2)CC(O)C(F)C1 C1(C2(O)CCC2)(CNC(CC2CCN(C(CCC(C)O)=O)C2)=O)CC1 N1(Cc2nccc(OC)c2)CCC2(CCCN2C(c2ccc(I)cc2F)=O)C1 C1(NC(C2(C)CS(=O)(=O)C2)=O)CN(C(c2cc3c(s2)CCC3)=O)C(C)(C)C1 N12CCC(C=CC1=O)CC2.C1(CC2(C3CC3)CCC(C)C2)CN2CCC1CC2 CC1(C)CCn2cc(C(=O)NC3CN(C(C45CC(F)(C4)C5)=O)CCC3F)nc2C1 c1(C(=O)NC(C2CCN(C(=O)CCOCC(F)(F)F)C2)C)ccn(C)c(=O)c1 N1(C(Cn2c(=N)nc[nH]2)=O)CCC2(NC(=O)CN3CCCCCC3)CCCCCC12 c1(N2C(COC)CC(O)C2)cc(Cl)nc(CCS(N)(=O)=O)n1.n12cc(nn1)C2 C1(C(=O)NC2CC(C(=O)NCCOCC(N)=O)C2)C2COCC12 c1(C(N(C2CCN(C(C3(CO)CCC3)=O)C2)CCC)=O)ccc(C)nc1 C1(NC(=O)C(F)F)C=CC(C(N2CCC(C(F)(F)F)C2)=O)C1 c1(NC(=O)CC2CN(C(C3CC3F)=O)C2)cccnc1I N1(C(C2CC(CNC(C3(CC)CC(C)(C)C3)=O)OC2)=O)CC(C)CC(C)(C)C1 Cc1cnn(C)c1CC(N1CCCC1C(C)NC(C1CCN1C)=O)=O C1(CNC(C(C#C)(C)C)=O)COCCN(C(c2cccnc2OCC)=O)C1 CC1(C)CC(CN)N(C(c2ccc(F)cc2F)=O)C1 c1(C(C2CN(CCc3ccccc3)C2)NC(c2ncn(C)c2)=O)nccc(OC)n1 C1(NC(C)=O)CCN(C(C2(COc3ccccc3C(C)C)CCCCO2)=O)CC1 c1(C(N(CC(C)N(C)C(c2ccc(Cl)cc2)=O)C)=O)ccc(Cl)nc1N CC(C(=O)NC1CCC1C(=O)NCC(F)Cl)=C1CC1 c1(C(N(C2CCN(C(C)=O)C2)CC)=O)cc2ccc(OC)cc2[nH]1 C1(NC(C2CCC(C)O2)=O)CC2CCC(C1F)N2C(C1COCCOC1)=O C1(CC=C)(NC(=O)CC(C)C2CC2)CCN(C(C2(C)CCCC2C)=O)C1 N1(C(C2CC(=O)N2)=O)CCC(O)(C(=O)N(c2cccc(Cl)n2)Cc2cccs2)C1 N1(C(CCNC(COC)=O)=O)CCC2CCCC(C1)N2C(=O)CCC(F)(F)F C1(C(=O)NC(CNC(c2scc(C)c2)=O)C2CCC2)CC(C)CC(=O)N1 c1(CC)[nH]nc(C(=O)NCCCCN(C(=O)CC2C(C)(C)C2(C)C)C)c1Br N1(C(C2(F)C(C)C2)=O)CC2OCC(NC(c3ccsc3-n3cnnn3)=O)C2C1 N1(C(C=CC)=O)CCN(C)CC1CNC(c1cncc(C#N)c1)=O C1(N(C)C)CCCN(CCC(=O)NCC=CCNC(=O)Cc2cncn2C)C1 CC(C)CC(CNC(=O)CCc1ccccn1)C(=O)NCCN1CCCCC1 N1(C(=O)NCCCc2nc3c(s2)CCCC3)CCC(C2(O)CC2)C1 C1(C(N2CCC(CCNC(=O)Cc3ccon3)C2)=O)CCC(C)(C)C1.CO c1(NCC2CCN(C(c3c(C(C)(C)C)n[nH]c3)=O)C2)ncc(Br)cn1 CCN=c1nc(C(N2CCCC2CN(C(=O)CC(C)F)C)=O)cc(C)[nH]1 C1(CC)CN(C(C2CCCCC2F)=O)CC1C(=O)NCCNC(c1ccoc1)=O c1(C(N2CCC(C)(NC(CCOCC#C)=O)C2)=O)cc2c(s1)CCC(C)C2 CCCCCCCCC(C)C(=O)NCC1CC(NC(=O)C(O)CCn2cncn2)C1 c1(CCC(=O)NC(C(C)NC(=O)CSc2ccccn2)(C)C)cc(F)ccc1F C1(C(=O)NC(C)C(C)NC(c2cncc(N)c2)=O)(OC)CCCCCCC1 C1(CNC(c2ccc(CC)nc2)=O)COC(C)(C)CN1C(=O)C=C(C)C(C)(C)C c1(OC)ccc(Br)nc1NC(C1(C)CCCN1C(c1occc1Br)=O)=O C1(C(=O)NCCN(C(C(C)Cc2ccccn2)=O)C)(NS(C)(=O)=O)CCOCC1 CC(C)CS(=O)(=O)CCC(=O)N1CCC1CNC(=O)Cc1cccc(F)c1O C1(COC)CN(C(=O)Cc2cnn(C)c2)CCN1Cc1cc(F)ccc1I C(=O)(C(S(C)(=O)=O)C1CC1)NC1C(C)CN(C(C2(C(F)F)CCCCC2)=O)C1 c1(NC(CC2OCCN(Cc3ccc(C)cc3F)C2)=O)cccc2nc(O)oc12 S(=O)(=O)(c1cc2sc(=NC(CCO)C3CCC3)[nH]c2cc1Cl)N(CCCCC)C N1(C(C(CCC)(C)C)=O)CCC(NC(C2(C)CCCS2(=O)=O)=O)CC(O)C1 N1(C(C(CC)OCC)=O)CC(C(=O)Nc2cccnc2OC)C(C)(C)C1 c1(OCC(=O)O)ccc(CC(=O)NC2CCC(CNc3ccc(Cl)cn3)C2)cc1 c1(C(=O)NC(C2CN(C(c3ncoc3Br)=O)C2)C)sccc1C1CC1 c1(OC)ccc(-c2nc(CC3(C)CC3)nn2-c2ccncc2C)nc1OC N1(C(CN(CC)CC)=O)CCN(C(=O)C(c2ccccc2)OC)C2(CC2)C1 c1(C(=O)NCCCC(C)NC(C(CSC)C)=O)ncnc2cc[nH]c12 c1(C(N2CC(O)CC(NC(CN(CC)CC)=O)C2)=O)ccc(OC)c(OC)c1Cl c1(C(=O)NC2CN(C(C(CCC)OC)=O)C2)cc(OC)c(OC)c(Br)c1 c1(C(=O)NCC(C)NC(c2ncc(Cl)n2C)=O)c(C#N)cnn1C C1(NC(C2CC(F)(F)C2)=O)CC2CCC1N(C(=O)C(c1ccc(F)cn1)(F)F)C2 c1(OC)c(C)cc(CN(C)C(c2ccccc2OC(F)(F)F)=O)cc1C C1(C(=O)NCC(CC)NC(=O)C(C)Cc2ccccc2F)CCCC(C)(C)C1 C1(NC(C(CNC(C2(CC(C)C)CC2)=O)O)=O)CCN2CCC1C2 N(C(=NCCc1ccn(C2CCC2)n1)NC1CCOC(C2CC2)C1)C(COC)C C(C)(C)(CC(=O)NC1CC(C)OC1=O)N(C(COCCN(C)C)=O)C c1(CC(=O)NCC(CN(C(C(C)=C(CC)C)=O)C)O)ccc2nn[nH]c2c1 c1(CC(=O)N(CCCNC(=O)C(C)C(C)C)CC)ccc(O)c(Cl)c1 c1(CN2CCC(Oc3cnccc3)C2)cc(C2CC2)on1 CC1CN(C(c2cc(O)cc(O)n2)=O)CCC1NC(c1ccc(C(N)=O)nc1)=O c1(NC(CC)CNC(=O)Cn2cc(Cl)cn2)nc(Cl)nc2c1COCC2 C1(CCNC(=O)CC(F)(F)F)CN(C(=O)COC2CCCOC2)CCCO1 Cc1cc(O)cc(=O)n1C(C)C(=O)NCCC1CN(C(C2(CF)CC2)=O)CCO1 C(=O)(CCCCN1CCCC1)NC(CC(C)NC(C1C2CCC(=O)C12)=O)C c1(OCC)ncccc1CC(=O)NCCC(C)NC(C1CC(=O)N(CC)C1)=O CN1CCOC(C(=O)NC2CCN(C(=O)Cc3cnnn3C)C23CC3)C1=O Cc1csc2nc(CNC(C(C)c3ccccc3)C(F)(F)F)cc(=O)n12 c1(CN2C(C(N(C)Cc3cc(C)nn3C)=O)CNCC2)cc2ccccc2o1 N1(C(c2c(C)coc2)=O)CC2CCN(C(C3CCC(=O)N3)=O)CCC2C1 c1(CC)cccc(CC)c1C(=O)N(C)CC1CN(C(c2cncc(O)c2)=O)C1 CCC(CC)CC(=O)NCc1nc(CNC(=O)Cc2ccc(O)c(C)c2)cs1 CCCC(C)(C)CC(=O)NCC(CC(F)(F)F)NC(c1cnn(CC2CC2)c1)=O C=CC1OCCC1N=c1nc2c(ncn2CC)c(N(C)CC2CCCS2)[nH]1 C1(CNC(C2(OCC)CCOC2)=O)CC2CCC1N2C(c1cnc(C(C)C)o1)=O CC(C)C(CCN(C)C(c1occc1C1CC1)=O)NC(=O)C=CCF C1(=CC(C)NC(=O)CC2CC2NC(=O)CCc2cccs2)CCCO1 C(=O)(CC(C(F)F)C(C)(C)C)NC1CC2CN(c3snc(C)c3C#N)CC21 C1(CNC(C2(OC)CC2)=O)CN(C(C2CCC3(CC3)C2)=O)C2CCCCC12 C1(C(=O)NC(C(C)C)C(C)C)CN(C(c2cccc(CO)c2)=O)CCN1C N1(C(C(c2cncnc2)C)=O)CCC2CC12C(=O)NCCC(C)C(F)F C(C)(CCC(=O)N(C)CC1CCOCC1)NC(C(C)SC)=O N1(C(C(C)(O)C2CC2)=O)CCCCC(CNC(c2ncsc2Br)=O)C1 C12(C(=O)NCC3(COC)CCN(C(CCC(=C)C)=O)C3)CCCC1CCC2 CC(CC(=O)NCCC1(C)CCN(c2nnn(C)n2)C1)CC(C)(C)C C=CCC(C)(C(F)F)NC(=O)COCCNC(C1C2CCCOC12)=O Cc1nonc1CC(=O)NCc1cn(CCNC(=O)CN2CCCC2C)nn1 C=CCC(C)C(=O)NCc1cc(C(=O)NC(C2(OC)CCC2)C)n[nH]1 C1(C(=O)NCCC(CO)NC(=O)NC(C)(C)C)(CC)CCOC1 N1(Cc2ccc(CC(=O)OC)[nH]2)CCNC(=O)C1C C1(NC(C2CCCC2O)=O)CC2(C1)CC(NC(C1CC1(F)F)=O)C2 C#CC1(C(N2CCCC(NC(C)=O)C2)=O)CCN(C(=O)C=CC(C)C)C1 C1(C)(C(=O)NCCC(C)CCNC(=O)CCCn2ccnc2)CCCC(F)(F)C1 c1(CNC(CCCC=C)=O)nc2c(s1)CCN(C(c1ccco1)=O)C2 c1(NC(C2N(Cc3c(C)noc3C)CCC2)=O)ncc(Br)nc1CO CC(C(C)(C)CN(C)C)NC(C1(CNC(=O)Cc2cccn2C)CCC1)=O N1(C(c2cc(CC)sn2)=O)CCCC(C)(C)C1CNC(C1(CC2CC2)CCC1)=O c1(C(=O)NC(C)CNC(=O)CCNC(c2ccco2)=O)cccc(Br)c1O c1(CC(=O)NCC2(C(=O)NOCCc3cccnc3)CC2)ccnc(O)c1 c1(CC)ccc(C(N2CC(CO)(NC(=O)CN3CCCC3C)C2)=O)cc1 Cc1c(C(N2CCC2CC(=O)NCCC2(C)CC2(F)F)=O)cccc1O CC(CC(N)=O)C(=O)N(C)CC1CCN(C(=O)Cc2cc(F)ccc2O)C1 C1(NC(CC(CCC)NC(c2ncn3ccccc23)=O)=O)CCc2n[nH]cc2C1 N1(C(C=C(C)C(C)C)=O)CC=CCC1C(=O)NC(CO)C(C)(C)C C12(C(N3CC4(N(C(CNC(N)=O)=O)CC4)C3)=O)CCCCC1OCC2 c1(OC)ccc(Cl)cc1CC(N1CC2CC(NC(C3CC(O)C3)=O)C1C2)=O c1(C(C(=O)OC)NC(N2CCC(C(c3ccccc3)=O)C2)=O)ccc(Cl)s1 C(CCS(C)(=O)=O)(C(=O)NCc1cc(C)[nH]n1)n1cc(CCC(CC)O)nn1 n1(CCC)ccc(=NC(=O)CC2CCC(C(=O)NC3(CC)CCCO3)C2)[nH]1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCC1CN(C(C(F)OC)=O)CC12CC2 CC1(C)CC(CO)CN(C(=O)C(C2(C)CC2)NC(c2ccc(C#N)cn2)=O)C1 C1(C(=O)NC(c2cnn(C)c2)C)C(O)CCN1C(C1CCCSC1C)=O c1(CC(C(=O)OC)NS(=O)(=O)CCC2CNCCO2)nc(C)c(C)nc1C Cc1cc(Cl)c(C(=O)NC2CCC2NC(C2CC2C(c2ccccc2)=O)=O)cc1N c1(OC)c(C(=O)NC(CNC(C2CC2F)=O)C(C)C)ccc(Br)c1F c1(C(N(CC(C)N(C(CCOCC)=O)C)C)=O)cn(C(F)F)cn1 c1(C(N(CCCNC(c2cc(CO)[nH]n2)=O)CC)=O)ccc(SCC(C)C)cc1 N1(C(CCOCCNC(c2cc(CC)on2)=O)=O)CC2CCCC2(COC)C1 C(CNC(c1c[nH]nc1-c1cccs1)=O)(N=c1nc[nH]s1)c1c(OC)cccc1 C(=O)(C(C(C)C)c1ccc(F)cc1)OC(c1c(C(C)=O)ccs1)=O CCCC(C(=O)NCC12CC1CN(C(=O)C=Cc1cccnc1)C2)OCC c1(CC)cccnc1NC(=O)NC(CNC(C1CCCC1)=O)CC(C)C N1(C(CC2CC(NC(C=CC(C)(C)N(C)C)=O)C2)=O)CC2C3C=CC(O3)C2C1 n1(CC(=O)NCC2N(C(CCC=C=C)=O)CCOC2)cc2ccccc2n1 C1(CC)CN(C(c2coc(SC)n2)=O)CCC1NC(c1nc(=O)n(C)[nH]1)=O C1(C)(CC)CCC(C(=O)NCc2cc[nH]c2C(=O)NC2(C)CC(O)(CO)C2)O1 C1(CNC(c2c(C)c(N)ccc2)=O)(NC(=O)C=C2CCC2)CCC(F)(F)CC1 C(=O)(CCCCCNC(=O)NCC(F)(CC)CC)OCC CC(C#N)CCC(=O)NC1(C)CN(C(=O)CCc2ccc(Cl)c(F)c2)C1 C1(NC(C2(CC)CC=CC2)=O)CCCC(CNC(=O)CNC(c2cccs2)=O)C1 c1(C(N2CC=C(CO)CC2)C(=O)NC)ccc2c(c1)OCC(=O)N2 C(=O)(C(Cc1cnc[nH]1)NC(C1CC(C)=NO1)=O)NCC(C1CC1)SC Cc1cc(N)c(C(=O)NCCCN(C(=O)COCC2CCCO2)CCO)nc1C c1(SC)nc(N2CC3CCC(C(=O)OC(C)(C)C)(C3)C2)cc(C#N)n1 c1(C(N2C(C(=O)Nc3c(C(C)C)ccnc3)CC(F)C2)=O)csc2ccccc12 N1(C(CC2C(OC)C2)=O)CCN(C(=O)C(C)(C)OC(C)=O)CC1CC1CC1 C(=O)(C1=CCCC1)N(C1CN(C(=O)CCc2cccnc2)CC1F)C CCC(CC)CCC(=O)NC1(C)CC(C(=O)NCc2cnccc2Cl)C1 CC1Cc2c[nH]nc2C(C(=O)NC2(CCNC(c3c(Cl)nn(C)c3Cl)=O)CC2)C1 c1(C(=O)NC2CC(CCNC(C3CC(O)C3)=O)C2)cn2cc[nH]c(=O)c2n1 C1(C(N2CC(C)C(NC(=O)COCC3CC3)C2)=O)CCC(=C(F)F)CC1 C1(NC(C2(C#C)CCN(C(=O)CCC(=O)OC)C2)=O)CC1C1CCCCC1 C1(NC(CCc2c(C)nn(C)c2)=O)CCN(C(c2ccoc2C)=O)C12CC2 c1(C(N(C2CCN(C(=O)CO)CC2)CCOC)=O)ccc2cc(C)ccc2n1 n1(CC)c(CNC(=O)C(CNC(=O)CCC2(C)CCC(=O)N2)N(C)C)cnc1C c1(NC(C2CCCN(C(c3n[nH]c(C)c3C)=O)C2)=O)cccc(Cl)c1O c1(OC)cc(C(=O)NCC(C2CCCC2)NC(=O)C(C)n2ccnn2)cc(F)c1 C1(NC(C(C)(C)OC)=O)CN(C(C2CCN(C)C(=O)C2)=O)CC2(CC2)C1 CC1(C(=O)NCC2=CCN(C(c3cnccc3C(F)F)=O)CC2)CCCCCC1 C=CCC(C(=O)NC1CN(C(=O)CC23CCC(CC2)OC3)C(C)(C)C1)C(C)C C=Cc1cnn(C)c1C(=O)NCC1CCC(C)CN1C(=O)CC1CC(C)(C)C1 N1(C(C(C)OC2CCOC2)=O)CCC2C(NC(c3ccc(N(C)C)nc3)=O)C2C1 C(CCNC(=O)OCc1ccc(OC(C)C)cc1)(C(C)C)OCC CC(C)CC(F)C(=O)N1CCCCC1C1CCN(C(c2ccc(O)nn2)=O)CC1 C1(CNC(c2[nH]cc(C)c2)=O)CCCCC1NC(=O)C(O)CC1CC1 C1(NC(C2C=CCC2)=O)CCN(C(=O)CC23CC(C2)C3)CC1 CCC(CNC(=O)NC1C2CC3C(C2)C13C(=O)OC(C)(C)C)(CC)C(N)=O C1(NC(c2cnco2)=O)CN(C(C23CCCC2C3(F)F)=O)C2CCCC12 C(=O)(CC(C)P(C)(C)=O)NCCCNC(C1ON=C(CC)C1)=O.C1(=O)CO1 C1(NC(COCCNC(Cc2cc(C)sc2)=O)=O)CC2C=CC1C2 C1(CNC(=O)C=Cc2cnc[nH]2)COCCN1C(c1cc(=O)cc[nH]1)=O Cc1ncsc1C(=O)NCCC(C)NC(c1ncoc1-c1cccs1)=O Cc1cn2cc(C(=O)N(CC(C)(C)CNC(=O)Cn3ncnn3)C)nc2s1 C1(NC(CCCOCC)=O)COC2CN(C(=O)Cc3ccc(C)nc3)CC12 c1(C(=O)NC(CC)CN(C(=O)C(O)CC(C)C)C)cc2c(s1)CCCCC2 Cc1c(F)c(C(N2CC3OCCC23)C2CC2)cc(Br)c1F C#CC1CC2CCC1N(C(=O)CC1C3CN(C(=O)CC(O)C(C)C)CC13)C2 C1(OC)CC(NC(=O)CCC(=O)N(C)C)CN(C(c2cn(CCF)nn2)=O)C1 N1(C(c2cn(C)nc2)=O)CC2CC1CC2NC(c1cccn(C2CCC2)c1=O)=O CC(C)(C)C(C(=O)NCCc1ccc(F)c(F)c1)n1cc(-c2ccccc2)nn1 Fc1ccccc1C(C(F)F)Nc1ccc(OC2CCCC2)o1 N1(C(C)=O)CC2CC1CN2C(=O)C(C(C)O)NC(=O)CC(C)C(F)F C(=O)(CCCCC(N)=O)NCC(CCOC)NC(C1(c2ccccc2F)CC1)=O c1(C(N2C(CNC(c3c(Br)sc(C)c3C)=O)CC2)=O)cc2ccsc2s1 N1(CCC(N2CCC(N(C(=O)CCc3ccc(C)s3)CC)C2)=O)CCOCC1=O C1(C(=O)OC)CCC2(CC1)CC(S(=O)(=O)N1CC(C)CCC(C)C1)C2 C12(NC(CCCCCN(C(C(C(C)(C)C)OC)=O)C)=O)CCC(CC1)C2(C)C N1(C(c2scc(C(=O)OC)c2)=O)CCCCC(NC(c2conc2C)=O)C1 C(=O)(CCC(F)(F)F)NC(C(=O)NCCN(C(CC)C)C)CN(C)C N1(C(c2ccn(CC)n2)=O)CC2CCC(C1CO)N2CC.C12(CC)CCN1C2=O C1(CCC)CC(C(=O)NCC2C3CN(Cc4ccc(F)cc4)CC23)CCO1 C1(CNC(c2n(CCOC)ncc2)=O)C2CC2CN1C(c1nccnc1N)=O C1(NC(C2N(C=O)CCC2)=O)CCN(C(=O)CSc2cn[nH]c2)CCC1(F)F Cc1ccnc2sc(C(=O)NC(CNC(=O)C(F)n3cccn3)C3CC3)c(C)c12 c1(SCC(c2cc(C)n(C3CCS(=O)(=O)C3)c2C)=O)cc2ccccc2n1C C(C(CC(C)C)C(=O)NCC1CCCCC1(C)C)NC(c1c(CC)n[nH]c1)=O c1(C(=O)OCC)noc2c1CN(C(=O)NC1CCCC13CCCO3)CC2 N(C1CS(=O)(=O)Cc2ccccc21)C(c1c2nc(C)sc2ccc1)C1CC1 Cc1nn(C)c(Cl)c1C(=O)NC1CCCC1CNC(=O)C(N1C(=O)CCC1=O)C N1(C(c2c(CC(C)C)onc2)=O)CC(C)N(C(C2C3CCC2CC3)=O)CC1C N1(C(c2cc(Cl)ncn2)=O)CCC2(CCC(C(N3CCC3CO)=O)C2)CC1 N1(C(CSCC)=O)CCCC1(CNC(c1ccccc1CO)=O)CC O=C(CC(C(F)F)NC(c1ccccc1F)=O)NCCCC1CCCCO1 Fc1ccc(CNC(=NCCN2CCCC2)NCC2CCC23CCC3)c(F)c1 C(=O)(N=c1[nH][nH]c(C)c1C)C1C=CC(NCc2ccc(OC)c(C)c2)C1 N1(C(C(=O)NCCCOC)CCc2nc(C)c(C)n2C)C2CCC1CC(CO)C2 N#Cc1nccc2cc(NC(c3ccc(Cl)c(C(F)(F)F)c3)C(N)=O)ccc12 C(=O)(C1=CCC(NC(=O)CC2CCCOC2)C1)NCCOCC CCCCC(=O)C(=O)NCc1nnn(C)c1C(=O)NC1CCOC1C C(=O)(CCCC(C)(C)C)N(CC(C)(C)C(=O)NCCC1CCCC1O)C C=CCC(CC(C)C)C(=O)N1CCC(CNC(=O)C(CC)(CC)CC)C12CC2 N1(C(Cn2cnc(C#N)n2)=O)CCOC2(CCN(C(c3csnc3Cl)=O)CC2)C1 c1(OC)cccc(Br)c1C(N1CCN(C(=O)Cc2ccc(O)cn2)C(CO)C1)=O n1(CC(=O)NC(C)CCNC(=O)CC23COC(C)(C2)C3)ccc(Br)cc1=O C(C(C)(O)CC(=O)N1CCOC(C(N2CCC(C)=C(C)C2)=O)C1)OC C1(CCC(=O)NCCCCC#C)CCCCN(C(=O)C(CC(C)C)N(C)C)C1 C1(C(N2CCC(CN(C)C(c3cccc4cncn34)=O)C2)=O)CC2C(C1)C2(C)C N1(C(CCOCC#C)=O)CCC(=CCNC(=O)C(F)=CCC)CC1 CCCCC(C(=O)NCC(C1CCCC1)NC(=O)C(F)(F)CC)NC(N)=O C1(C)(C(N2CC(NC(CC3C=NN(C)C3=O)=O)C3(C2)CC3)=O)CCS(=O)(=O)CC1 C1(CNC(c2ncc(CC)s2)=O)CCN(C(=O)CC2=CCCCC2)C12CCC2 C1(C(=O)OC)CCc2ccccc2C1.C=CCCN=C1NC2CC(N1)C2 C1(NC(CC(C)OC)=O)CCCCC1C(=O)NCC1SCCS1 C(=O)(C1CCCc2scnc21)N1CC2C(C(=O)Nc3cc4c(s3)CCC4)C2C1 N1(C(C(CC)N(CC)CC)=O)CCC2(CC1)CC2C(N1CCCC1C1(C)CC1)=O C1(C(=O)NC(C(=O)NC2CN(CC)CC2C)Cn2ccnn2)CC(C)(C)CCO1 C1(NC(CCN(C)C)=O)CN(C(C2C=CC(C(=O)OC(C)(C)C)C2)=O)C2(CCC2)C1 c1(C(N(CC(CC)NC(=O)C#CC2(C)CC2)C)=O)cccc(Br)c1Cl C1(CC=C)(NC(=O)CCCOCC)CCCN(C(C2(NC(C)=O)CCOC2)=O)C1 C(=O)(C(C#N)C(C)(C)C)N(C(C(N1C2(CC(COC)C2)CC1)=O)C1CC1)C N1(C(C=CC)=O)CC(F)(F)CC1C(=O)NC(C)C N1(C(C2CCC(CNC(C(C=C=C)C)=O)C2)=O)CC2C3CCC(C3)C2C1 C(C(C)(O)C(F)F)NC(COC1CN(C(C(CC)OC(C)=O)=O)C1)=O C(=O)(C(CNC(=O)Cc1cnccc1C)C(C)(C)C)N1CCC(N(C)CC)C1 c1(C(N2CC(NC(CCSCC)=O)CC2(C)C)=O)cnn2cccnc12 c1(C(C)=O)cc(C(=O)N(CC(C)NC(c2ccc(C(F)(F)F)cc2)=O)C)oc1C Cc1cc(C(N2CCCC2(C)CNC(=O)Cn2ncnn2)=O)cc2ccoc12 C1(C(=O)NC(CCN(C(=O)CC2CCCOC2)C)(C)C)CCc2ncncc2C1 O=C(C1=C(Cl)CCC1)NC1CCC(CNC(c2ccsc2)=O)C1 N1(C(CC2(C)CC2(Cl)Cl)=O)CCN(C(=O)Cc2c[nH]nc2O)C(CO)C1 c1(C(=O)NCC(CCNC(C=CCCC)=O)O)cc(CCC)c(C)s1 CC(N=[N+]=[N-])C(=O)N(C)CC1CCCCN1C(=O)CCCC1CC1 CCC(O)C(C)C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CN1CC=CC1 C1(NC(CCCOCC=C)=O)CC(OC)CN(C(=O)C(C)CC)C1 Cc1cc(CC(=O)NC(Cc2cn[nH]c2)C(=O)NC2CC(OC(F)F)C2)nn1C N1(CCCC(=O)NC(CNC(C(F)=CCC)=O)(CC)CC)CCc2ccccc21 C1(NC2CCN(c3cc(C)nn3C)C2=O)CCCCCCC1 C1(O)(CNC(C(C)OCC=C)=O)CCN(C(=O)CNc2ccc(CC#N)cc2)C1 C1(NC(c2cc(C)c(C)s2)=O)CCCN(C(c2ccccc2F)=O)CC1F c1(OC)cc2ccccc2cc1C(=O)NCCN(C(C1CCNC1=O)=O)C1CC1 O=C(C1COc2ccccc21)NC1CN(C(c2cc3c(s2)CCCC3)=O)C2CC12 C(=O)(C(C)C(C)NC(c1oc(CNC(C2CC(=O)C2)=O)nc1C)=O)OC Cc1cc[nH]c(=N)c1C(=O)NC1CC(NC(=O)CS(C)(=O)=O)C12CCC2 C(c1ccc(Cl)s1)=C(C#N)C(=O)NCCCC(c1ccccc1)NC(=O)CCF c1(CNC(C2CCS(=O)CC2)c2n(C3(C)CC3)nnn2)ccnc(F)c1F C1(NC(C(CCC)O)=O)Cc2ccccc2C1NC(=O)CC(C)(C)C1CC1 c1(N(C(C)(C)CN2CCOCC2)C(=O)NC2CC(=O)N(C3CC3)C2)ccc(Cl)cc1 C1(CNC(c2cnc3nccn3c2)=O)CN(C(c2ccco2)=O)C2COCC2O1 C(CC(=O)N1CC(OC(=N)O)C1)N(C(=O)C(C)C1CCC1)CC N1(C(c2ncn(C)c2)=O)CCCC(CCO)CC1.N12CCCC(C)(C1)C2=O C1(NC(C2COCOC2)=O)CC2CC(C1)N(C(c1ccn3nncc3c1)=O)C2 c1(OC)cc(F)c(F)cc1NC(=O)NCc1cnc(O)c(F)c1 N1(C(C2=C(C)CCC2)=O)CC2CC(CNc3nccc(C(C)(C)C)n3)CC1C2 C1(NC(C(N2CC(C)C2)C)=O)CC(C)CN(C(C2(F)C(C)(C)C2(C)C)=O)C1 C(=O)(C(F)CCC(C)(C)C)NC1(CCNC(CCc2n(C)ncc2)=O)CCOC1 C(CO)(C(C)(C)CO)NC(C1(C(C)NC(=O)CC2CNC(=O)O2)CC1)=O c1(C(N)=O)cc([N+](=O)[O-])cnc1N1CCCCC(NC(=O)C(C)n2cccc2)C1 C1(NC(CCN(C)CCO)=O)COC2(C1)CN(C(c1ccns1)=O)C2 C=CC1(C(=O)NC2CC(NC(C3(C)CC4CC4C3)=O)C(O)C2)CCOCC1 CCC(C(=O)N1CC(CNC(=O)CN2CCCC2=O)C2(CCC2)C1)C(F)(F)F C=CC(C)(CCOC)C(=O)NC1C2CN(C(c3cncc([N+](=O)[O-])c3)=O)CC12 C1(CN(C)C)CCC(C(N2CCC(CNC(=O)Cc3coc(C(F)F)n3)C2)=O)O1 CC1=NN(C)C(=O)C1CC(N1CCC(NC(C2COCCOC2)=O)C12CC2)=O C1(C(N(C2CCN(C(=O)Cc3cccc(SC)c3)C2)CC)=O)(CC)CCOCC1 CCCC(O)C(=O)NCC1(C(=O)NC(C)CN(C)C(C)C)CC=CC1 C(=O)(N=c1ccn(CCCO)[nH]1)C1C2(CC(NC(CCOC(C)C)=O)C2)C1 c1(C(N2CC(C(C(=O)NCC3CCC3CO)OC)C2)=O)csc(Cl)n1 N1(C(C=CCN(CC)CC)=O)CCC(NC(=O)CN2CCN(C)C(=O)C2)C(C)C1 C1(CCCNC(c2c(CC)nco2)=O)CCCCN1C(=O)CC1CCC(=O)N1 N1(C(CCC=CCC=C)=O)CC(O)CC1(C)C(N1CC(O)(C(F)F)C1)=O Cc1cc(NCC(=O)O)ccc1C(=O)NC12CC(F)C1C2 CC1(C)OC(=O)NC1CNC(C1(CO)CCN(C(=O)C(C2CCOCC2)=O)C1)=O C(CCC(C)CC(=O)NC(C)C(C)(C)NC(c1cnc(O)n1C)=O)=C(C)C c1(CNC(C(CC)C#N)=O)ccc2c(c1)CCC2NC(c1cc(COC)cs1)=O CC1OC2CCC1(NC(=O)CN(C1CC(C#N)C1)C(c1cccc(=O)n1C)=O)C2 Nc1cccc(C(N2C3CCC2C(NC(=O)CCc2ccccc2Cl)C3)=O)c1O N1(C(C=CCC)=O)CCCC1C1CCCN1C(c1ccc(CC)s1)=O C(=O)(C(C(C)C)C(C)C)N1C(CC)C(NC(c2cccc(C)c2O)=O)CCC1 C(N=c1[nH]c2c(c(=NC3CCC4CC34)[nH]1)SCC2)c1c(Cl)ccs1 c1(CSCC)cc(C(=O)NC2(COc3cnn(-c4ccccc4)c3)CC2)no1 C(N=c1[nH]c(=NC2CC(S(C)(=O)=O)C2)[nH]c2cc[nH]c12)C1C(C)(C)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C2CCCCC2)F)cccc2cnnn12 c1(CC)nc(C)c(C(=O)NCC(c2ccccc2F)NC(=O)C(C#N)CCC)s1 C(C#Cc1cn(CC2CC(F)(F)C2)nn1)NC(C1C(C)CC(=O)N1)=O c1(C(C)(C)C)ncc2c(n1)CCN(C(c1c(F)cc(Br)cc1Cl)=O)C2 N1(C(Cn2ccc(C)n2)=O)CCC(F)(CNC(=O)CN(C2CCSC2)C)C1 N1(Cc2c(-c3c(Br)nccc3)nn3c2CCC3)CC(S)CC12CCOCC2 c1(SCCCC(=O)NC(CNC(c2nc(CC)oc2)=O)CC)ccc(OC)cc1 C1(CNC(C(C)(C2CCC2)NC(CCC2C(C)C2)=O)=O)C2CCCCCC12 CN1CCCC(O)(CNC(C2CCCN(CC3COCCO3)CC2)=O)C1=O c1(C(=O)NC2(CCNC(C(C(C)(C)C)NC(N)=O)=O)CC2)cc2c(s1)CCC2=O Cc1cc(Br)cc2c(C(=O)N(C(C)CCNC(C3CCC3C)=O)C)n[nH]c12 N1(C(C(C)C2CCC2)=O)CC(F)(F)CC1C(=O)NCC=CC1CC1 Cc1cc(C(=O)NC2CCCC23CN(C(C2CCN(C)C2=O)=O)C3)c(O)nc1C Cc1ccc2snc(C(=O)NCCC(O)CNC(=O)CCc3nc[nH]n3)c2c1 C1(CNC(CC2CC(=C)C2)=O)CCCCC1NC(=O)CNS(=O)(=O)NC c1(CC(=O)NCCN(C(CCOCCOC)=O)C)nc(C)sc1Cl c1(CC(=O)N(CCC(C)NC(C2(CF)CC2(F)F)=O)C)ccccn1 N1(C(=O)NC(C)C)CCCCC(N(C(=O)CC2OCCCC2(C)C)C)C1 C1(NC(=O)Cc2ccccc2)CCN(C(=O)CCCF)CCC1CO C1(C(=O)C2CC2)CN(C=O)CCO1.c1(C(=O)NCCCOCCCN)cc[nH]n1 N1(C(CS(=O)(=O)NC)=O)CC(NC(c2cc[nH]c2C2CC2)=O)C(C)(C)C1 c1(C(=O)NC2C(NC(C=Cc3n(CC)ccn3)=O)C2)ncc(Cl)cc1Cl N1(C(C2CCC(C(N)=O)C2)=O)CCCN(C(c2sccc2N(C)C)=O)CC1CO C(=O)(C(=O)CC(C)C)N1CCC(OCCNC(C2(CC#C)CCOCC2)=O)C1 N1(C(c2c(OC)nsc2)=O)CC(C)(C(=O)NCC(n2cccn2)C)CC1(C)C CC1CN(C(=O)CN(C)CCO)CC(NC(=O)Cc2nc(C3CC3)nn2C)O1 C1(CNC(c2c(C(C)(C)C)ncs2)=O)C2CN(C(c3cc(Br)n[nH]3)=O)CC12 c1(N(CC(=O)NC2(C)CN(C(C(CN(C)C)O)=O)C2)C)ccccc1[N+](=O)[O-] c1(CC)cccc(OCC(=O)NCC(C)(C2CC2)NC(C2CC2F)=O)c1 CN1CCCCC(CNC(=O)CCCNC(=O)CCCn2cccc2)C1 Cc1cc(C(=O)NCCN(CCOCCO)C(C2CC3CC2C2CC32)=O)cc(C)n1 C(=O)(C(C)(CC)C(C)O)N1CC(CNC(CC(=O)NCC)=O)C(C(F)(F)F)C1 N1(C(c2n(CC=C)ccc2)=O)CC(NC(c2cc(Br)c(C)cn2)=O)CC(C)C1 CCCCCC(=O)NCC(N1CC(CNC(=O)C(C)CC2CCC2)C(C)C1)=O C1(C(N(CCCNC(=O)Cc2csc(S)n2)CC)=O)COCCN1C C=CCC(C(=O)NC1COCC1NC(=O)CCc1ccc(Br)cc1F)C(C)C c1(OC)ccnc(C(=O)NCCC(C(C)C)NC(c2cccc(N)n2)=O)c1OC Cc1cnc(C(=O)NC(C2CCN(C(=O)CCF)C2)(C)C)cc1C N1(C(CN(C2CCSC2)C)=O)CC2CC(C1)N(c1ncc3ncnc-3[nH]1)C2 C1(C(=O)NCCOCC)CCN(C(=O)C(c2cccs2)OC)O1 C(=O)(C(C)(C)CC(=O)N1CCCC(N(C(=O)CC2(C)CCCO2)C)C1)OC N1(C(c2ccsc2Cl)=O)CCCC2(CCCN(C(c3ccnc(Br)c3Cl)=O)C2)C1 C1(C2(O)CCN(C(=O)Cc3cccc(C(F)F)c3)CC2)(NC(=O)C=CCO)CC1 N1(C(=O)Cn2ccnn2)CCC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])(CO)CC1 C1(C(=O)NCC2(CSC)CCC2)CCN(C(=O)C2(C)CC2(C)C)O1 c1(C(N2C(C(N3CCC(C(=O)OC)C3)=O)CC3CC32)=O)cc(Br)c(O)c(Br)c1 c1(C(=O)NC2CCN(C(CCCSC)=O)C2)cc2cc(C#N)ncc2[nH]1 C(=O)(CC(F)(F)C(F)F)N1C(CNC(C2CC2C(F)(F)F)=O)CC1 n1(CC(=O)NCC(Cn2cc(CC(C=C)O)nn2)(C)C)cc(S(C)(=O)=O)cn1 C1(C(N2CC(CC(C(=O)N(CCCC(C)O)C)F)C2)=O)NC(=O)OC1(C)C Cc1cc2c(C(N3CCC(C)(CNC(=O)C(C)O)C3)=O)nccn2n1 N1(C(CNC(=O)OCC)=O)CC(NC(c2csc(C(C)(F)F)n2)=O)C2(CCC2)C1 C1(C(N(CC(C)C#N)CC)=O)CCCC1CNC(C1(CC2CC2)CCC1)=O C1(CC(=O)Nc2ccc(CCO)cc2)CCCN(C(=O)CC2NC(=O)NC2=O)C1 C12(C(=O)NC3CCC(N(C)C(c4nc(Cl)cs4)=O)C3)CCN(CC1)S(=O)(=O)C2 C1(C(=O)NCCC2CCN(C(C(C)NC(C)=O)=O)C2)C(=O)ON=C1C CC(CC(N)=O)C(=O)N1CCN(C(C2CC(=C3CC3)C2)=O)C(CCO)C1 CC(CS(C)(=O)=O)C(=O)NCc1cccc(NC(=O)CCC2CCCN2C)c1 C1(c2cn(C(C)C(=O)N3CCCC3)nn2)(N(C)C)CCN(C(=O)C(F)F)CC1 N1(C(C(C)(C(F)(F)F)OC)=O)CCC2(COCCO2)C1 N1(C(CC2C(C)OCC2)=O)CCCC(C(=O)NC2CC(Cl)C2)CC1 C1(NC(C=Cc2cc(OC)ns2)=O)COC2(CCN(C(C3(C#N)CCC3)=O)C2)C1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCCC(CN(C(CCCCSC)=O)C)C1 CC(CCN(C)C)C(=O)NC1CC(C(=O)Nc2ccccc2)CC1O N1(C(CN(CCOC)C)=O)CCCC(C(N2CCC(C)(C)C2C)=O)CC1 C=CC1CN(C(=O)CC(CNC(C2CCC2COC)=O)OC)CC1O c1(C(=O)NC(CN(C)C(C2CC(C)(F)C2)=O)(C)C)ccn(C2CCCC2)n1 c1(CNC(=O)C2CC2)ccc(NC(Cc2ccc(Br)cc2)C(=O)O)cc1F C1(NC(C2(OCC)CCOCC2)=O)CC2CC1N(C(=O)CC1CC(F)C1)C2 Cc1cc(C(=O)NC2CC3(C2)CC3C(N2CCOC(C)(C3CC3)C2)=O)cc(C)n1 N1(C(c2c(C)ccs2)=O)CCCC(O)(CNC(C2(C)CC=CCC2)=O)C1 c1(C(=O)NC(C)C(CO)NC(c2ccc(Cl)o2)=O)ccccc1Br CC1CCN(C(C2(n3ccnn3)CC2)=O)CC1NC(c1ccc(Br)s1)=O c1(C(=O)NC(C)CCCNC(=O)C=Cc2cc[nH]n2)cccc(-n2cnnn2)c1 N1(C(Cc2n(C)c(S)nn2)=O)CCC2CCCC(C1)N2C(C1CCOCC1)=O c1(CC(=O)NCCNC(c2cn(C3CCC3)nn2)=O)cccnc1OC(F)F C1(C)(CC(=O)NCCCC(C)NC(=O)CCn2cc(Cl)cn2)CC(F)(F)C1 Cn1cc(Br)c(C(N2C3CCC2CC(NC(=O)CCC#N)C3)=O)cc1=O N1(C(=O)C=CC2CCOC2)CCN(C(c2cc(C3CC3)no2)=O)C(CO)C1 C(=O)(C(C(C1CC1)OC)N1CCC(OC(C2CCCC2)C2CC2)CC1)NCCCC C1(CC)CN(C(C23CCC(OC)C2C3)=O)CC1C(=O)Nc1ccccc1CCO C1(NC(C2CC(C(F)F)(OC)C2)=O)CN(C(C2CC(C)(O)C2)=O)CC1O c1(N2CCC(CNC(C(C)SCC)=O)C2)nc(C)ncc1F c1(C2(C(=O)NCC(c3cncc(F)c3)C)CC2(Cl)Cl)ccc(Cl)cc1 N1(C(c2c(C)cn(C)n2)=O)CCCC2C1CCN2C(C1CN2CCN1C(C)C2)=O C1(C(=O)NC(CNC(=O)NC)C2CC2)CCCCC1Nc1ccccc1 C1(C(N2CCC(CC)(CC)C2)=O)CN(C(c2cc(C#N)cs2)=O)C(C)(C)C1 c1(C(=O)OC)cnc(O)c2ccsc12.C12CC13CCN(CC3)C2=O C1(CNC(c2ncn(CC)n2)=O)CCCC1(C)NC(C1CN(C(=O)N(C)C)C1)=O C(=O)(CC(COC)COC)N(C1CCN(C(=O)CCC2CC(C)C2)CC1)CC O=C1CC(C(=O)N(CCCN=[N+]=[N-])CCO)N(C(C2C=CCS2)=O)C1 C=C1CCC(C(=O)NCCC(C)(C)CNC(=O)CC(C)c2cnn(C)c2)CC1 c1(CC(=O)N(CCCN(C(CCCC)=O)C)C)cccc2c1CCC2 N1(C(C=Cc2c(C)ccnc2)=O)CCC(NC(c2ncn(C)n2)=O)CC(C)(C)C1 C(C1=C(C)CCOC1)NC(C(C1CN(C(C(C=C)(C)C)=O)C1)O)=O C(=O)(CCCC(C)(C)C#N)NC(CNC(c1nc(C)c(C(F)F)cc1)=O)C C(=O)(C(C)(F)C(F)(F)F)NCCC1CCN(C(c2ccc(C(C)(C)C)cc2)=O)C1 C1(N(C)C(c2ccncc2C2CC2)=O)CCCCC1NC(C1CC1C(C)(C)C)=O c1(NC(C(CCC)OC)c2nnnn2C)ccc(NC(C)=O)cc1C N1(C(CCC(c2ccc(CC)cc2)=O)=O)c2ccccc2N(C)CCC1C N1(C(c2ccc(C(C)(F)F)cc2)=O)CC(NC(=O)Cn2cnnn2)CC(O)C1 c1(OC)ccc(CC(C)C(N2CCC(O)(CNC(=O)C(C)=CC3CC3)C2)=O)cc1 N1(c2ccc(C(=O)OC)cn2)CCC(C2CC2)(CNC(c2cnccn2)=O)C1 c1(C(=O)NCCO)ccccc1OC.C1(F)(N)CC1(F)F.C1COCCO1 c1(-c2cccc(C(N(c3ccccn3)CCCC)=O)c2)nnc2n1CCC2 c1(OC)ncc(Cl)cc1C(C(=O)NC1CCCC1)N(CCC#N)C c1(CC)oc2ccccc2c1C(C)C(=O)NC1CCC(Cc2ccncc2)C1 C(=O)(C1CNC(=O)c2ccnn21)NC(C)(C)Cc1ccc(Br)cc1 C1(CNOC)C2CN(C(=O)C(c3ccc(F)cn3)(F)F)CC12.C1(C2CC2)C(=O)N1C C1(CNC(c2c(C(C)C)nns2)=O)COCCN(C(c2nncn2C2CC2)=O)C1 C1(C(N(C)CC2(NC(C(c3ccccc3)SC)=O)CC2)=O)CSCCS1 c1(C(=O)NC2C(CC)CN(C(C3CC3C)=O)CC2)ccc2c(c1)nc(O)n2CC C(=O)(C(C(C)O)NC(=O)C(F)CC1CCOC1)N1CC(c2nc(C)[nH]n2)C1 C1(CC)CN(C(c2cc(C3CC3)n(C)n2)=O)CCC1NC(=O)C(F)(F)C1CCCC1 Cc1cc(Br)c(C(=O)NCC2CN(C(=O)CCC#N)C3CC23)s1 C1(CCOC)CC(N=c2cc(NCCc3ccccc3C)nc(C(C)C)[nH]2)C1 Cc1ccn(C(C)(C)C(=O)NCC(O)CN(C)C(c2c[nH]cc2C)=O)n1 c1(C(=O)NC(CNC(c2cc(O)nc(O)n2)=O)C2CC2)nc2cc(O)ccc2[nH]1 c1(OC)cc(NCC2CC(C(=O)Nc3cccc(C(C)(F)F)c3)C2)nc(OC)n1 C12(NC(C3CCCC3)=O)CC(CNC(c3cnc(C4CCCO4)s3)=O)(C1)C2 c1(C(=O)NCC2(O)CC(NC(CCNC(=O)NC)=O)C2)c(Cl)c([N+](=O)[O-])nn1C c1(-n2cc(C3(C)N(C(CC4N(C)CCC4)=O)CCC3)nn2)cccc2cncn12 CCC(C(=O)N1CC(CNC(=O)C#CC2(C(F)(F)F)CC2)C(O)C1)C(C)C Cc1cc(C)c([N+](=O)[O-])c(C)c1C(N1CC(NC(=O)C(O)C2CCC2)C(C)C1)=O N1(C(C(C=C)(C)C)=O)CCC2C(NC(c3ccccc3OCC)=O)C2C1 N1(C(C(CCC)NC(C)=O)=O)CCC(NC(=O)C(C)=C(C)CC)C(C)C1 C(C(O)CN=c1[nH]cc(C#N)cc1C)NC(CCc1n2cc(C)nc2sc1)=O n1(CC)ncc2cc(C(=O)NC3CCC3NC(=O)CC(=O)NCC3CC3)c(C)nc12 c1(CC(N2C(CCNC(CN3CC(C)(C)C3)=O)COCC2)=O)ccc(F)cc1F C(=O)(N=c1nc2c(I)cccn2[nH]1)NCC1(OCC)CCCCCC1 c1(C(N(C2CCN(C(=O)C(C)(C)c3cncs3)C2)C)=O)cc2n(c1)CCC2 C(C)(C(C(C)C)NC(=O)CCc1cccc(O)c1)NC(CCOCCC)=O N1(C(c2c(Cl)cn(C(C)(C)C)n2)=O)CC(NC(C2CCCC2)=O)C(S(C)(=O)=O)C1 C1(CC)C(NC(=O)C(C2CCC2)OCC)CCCN1C(=O)CC1CCCCCC1 N1(C(C(c2ccc(O)cc2)(C)C)=O)CCC(=C(F)F)CC1 c1(C(=O)NCC(c2ccccc2)NC(C(=C(C)C2CC2)F)=O)cc(C)ncc1C N1(C(CCc2ccc(C)cc2)=O)CC2CC1CCC2NC(C1CC2C=CC1C2)=O CC(C)C(C)(O)C(=O)NC1CN(C(c2cc(C#N)cs2)=O)CC1n1ccnn1 c1(C(N(C2(CO)COC2)C)=O)sc(F)cc1Br N1(C(C=C(C)C(F)F)=O)CCC2CC12C(=O)N(CCCCC(C)C)C c1(CNC(C2CC(C)(NC(c3cccc(Cl)c3)=O)C2)=O)ccc(F)nc1F C1(C(=O)OC)C2CCCC2CN1C(c1coc(C#N)c1)=O C(C(CC)(CC)NC(C1CC(O)C1)=O)NC(CN(CC)CC)=O CCC(COC)C(=O)NC1CCC1NC(=O)Cc1sc(S)nc1C CC(O)CCCC(=O)NCC1(NC(c2ccc(CN(C)C)o2)=O)CCOCC1 n1(CC(N)=O)cc(NC(C2CCN2C(=O)CC2CC2)=O)cn1 CN1CCC(CCNC(c2c[nH]nc2CNC(=O)C=CC2CCCC2)=O)C1 c1(CC=C)ccccc1C(=O)N(C)CCNC(=O)C(c1cccc(C)c1)=O N1(C(CC(C)CNC(=O)C(C)(C)CF)=O)CCC2(CC1)CSC2 C1(C(=O)NC2CC(C)(NC(C(C(C)C)n3ccnc3)=O)C2)CN2CCCC2CO1 C(=O)(CC(O)CC(C)(C)C)NCCC1(O)CCN(C(C(CCC#C)O)=O)CC1 CC1CN(C(C2(NC(=O)C#CC(=O)N(C)C)CCC2)=O)CC1N(C)C.C1CC1 c1(C(=O)NCC(CNC(C(c2cccnc2)C)=O)C)ccc2c(c1)N(C)CCO2 C1(c2ccc(F)cc2)(C(=O)NCCCNC(=O)CN2CC3CC3C2)CCCCC1 C1(C#N)(C(N(CCC)CCNC(=O)CC2CC3(CC3)C2)=O)CC12CCC2 N1(C(CCCN(C)C(C2CCCN2C2CC2)=O)=O)CCN(CC(N)=O)CC1 C1(CNC(=O)COc2ccsc2)COCCC1NC(=O)Cc1ccc(O)nc1 C1(NC(C(CC)NC(c2ccco2)=O)=O)CC2C1CCN2C(=O)CCF N1(C(C(CC#C)(C)NC(c2cnn(C)n2)=O)=O)CC2CC(C1)N(C)C2 N1(CC)CC(NC(=O)CCC2CC(NC(=O)Cc3ccoc3)C2)CCC1=O c1(CC)nc(C)[nH]c1C(=O)NCC1CCCN1C(c1cc(O)n(C)n1)=O N1(C(C2C(C)(C)C2)=O)CCCC(C)(NC(c2ccc[nH]2)=O)C1 c1(NC(C2(CC)CCCN2C(=O)Cn2ccnc2C)=O)cccc(F)c1F c1(C(N2CCC(C(=O)NCc3cc(C)cc(F)c3)C2)=O)cc(F)c(Cl)cc1C C1(C(=O)NC(c2cccnc2)C(=O)NCC(=O)NCC2CC2)(OC)CCOC1 C=CCCC(C(=O)N(C)C)NC(=O)NC(C(=O)OCC)C c1(C(=O)NCCCCC(C)NC(C2CC(C)OC2C)=O)nnc2ccccc2n1 C=CC(C(=O)NC(C(=O)NC1CCC(O)C1)C1(O)CCC1)OC N1(C(C(C=C)(C)O)=O)CCCN(C(c2cc(C)c(C)c(Br)c2)=O)C(C)C1 c1(C(=O)NC2C(NC(=O)Cn3cccc3)CC2)cc(Br)cc2scnc12 C1(CC(C)C)C(=O)N(C)CCN1CC(=O)N(C1CCOC1C)C1CC1 C1(CC=C)(C(=O)N(CCCCC)CCO)CCN(C(=O)C=Cc2ccoc2)C1 c1(NC(=O)NCC(c2ccc(OC)cc2)O)ccc2c(c1)CCN2 CC1(C)CCC(C(=O)NCCOCC(=O)NCCC(Cl)Cl)CO1 N1(C(C(CC(CC)CC)F)=O)Cc2n[nH]cc2C1C(=O)N1CCCC1CC(N)=O CCC(C)C(O)C(C)C(=O)N1CCCC1CCC(=O)NC1(C)CSC1 c1(C(C)NCc2csc(C#N)c2)ccc2c(c1)CCCO2 c1(CN(C(=O)NC2CCN(CC)CC2)C)cc(C)cc(Br)c1 Nc1ccc2nccnc2c1C(=O)NCCC1CCN(C(C2(O)CC2)=O)CC1 C1(CNC(c2c(C)cc(Br)cn2)=O)CN(C(=O)COCCF)CC(C)(C)O1 C(=O)(C(CC(C)C)C(C)C)NCC1(OC)CCN(C(c2occc2C)=O)C1 c1(NC(=O)NCc2c(OC(C)C)n[nH]c2)cnn(C)c1-c1ccccc1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)NCC(CO)NC(CN(CCC)C)=O c1(C(=O)NCCOCCN(C(c2c(CC)con2)=O)C)cc(Br)ccc1C C(=O)(CCCCCC#N)N1CC(C)OC(CCNC(=O)C(C)(C)C2CCC2)C1 C=CCC(C)(C(=O)N1CC(OCCNC(=O)C(C)CO)C1)N(C)C CC1=C(C)CC(C)(NC(=O)C(CO)NC(=O)CCc2ccccn2)CC1 Cc1[nH]c2ncnc(NCc3nncn3-c3ccccc3)c2c1C C=C1CCN(C(c2c[nH]nc2OC)=O)C(C(=O)NCC(C)C(F)F)C1 C(C(C)(CC(C)C)NC(=O)CCc1cncn1C)NC(COCCCC(C)C)=O C1(NC(c2cc(SC)oc2C)=O)CCN(C(c2ccn(C(C)(C)C)c2)=O)C(C)C1 C(=O)(CCCCCS(N)(=O)=O)N1CC2=C(CN(C(C=Cc3n(C)ccc3)=O)C2)C1 C(C(=O)N1CCN(C2CN(C(=O)C(CO)N(C)C)C2)CC1)(C(C)C)n1ncc(C)c1 CCCS(=O)(=O)CC(=O)N1CCN(C)CC1CNC(=O)CSCC(F)F C1(N(C(CC(=O)NCC#C)=O)CC)CCCN(C(C2CC(c3ccccc3)O2)=O)C1 c1(NC(=O)Nc2nc(COC)nc(N3CCCCCC3)c2)cc(C#N)ccc1Br N1(C(C(C=C)OC)=O)CC2(C1)CN(C(c1cc(C)c(F)cc1O)=O)CCO2 CC1CN(C(=O)C(N)=O)CCC1CNC(=O)Cc1cc(N2CCCC2=O)ccc1F N1(C(c2c(COC)cco2)=O)CCC(NC(C2(CO)COC2)=O)C(C)C1 N1(C(c2c(C)ccc(O)c2)=O)C2CCC1CN(C(c1cnn(C)n1)=O)CC2 N1(C(C(c2cn(C)nc2)=O)=O)CC2(C1)CN(C(C1CCCCC1F)=O)C2 C1(C(=O)NCC(O)CCC2CC2)(COC)CN(C(=O)CC(C)C)C1 n1(C2CCN(C(=O)NCC3C(C)COCC3)C2)cnc2ccccc2c1=O c1(N(C(C)C)CC2(C)CCN(C(C)=O)C2)ccc(F)cc1Cl C1(C(=O)NC2C=CCN(C(C3(CO)CCOCC3)=O)C2)CC2CCCCC12 c1(NC(c2c(NC(C(C)NC=O)=O)cnc(Cl)c2)=O)ncc([N+](=O)[O-])cc1I c1(C(N2CCC(O)(CNC(=O)C3=CCCCC3)C2)=O)cc(Cl)cc2ccccc12 C1(c2cn(C3C(c4c(C)nn[nH]4)C3)nn2)CN(C(C2(C#N)CCCO2)=O)CC1O CCCC(C(=O)NCCC1CCCN1C)NC(=O)C(C)OC(C)(C)C CC1(CCNC(c2cc(C3CCC3)[nH]n2)=O)CCN(C(C2CCO2)=O)C1 c1(CN2CC(NC(CNS(CC)(=O)=O)=O)C2)ccc(F)cc1OC N1(C(CC2(N(C(=O)CC=CC(C)(C)C)C)CC2)=O)CC2CC2(C(N)=O)C1 c1(C(N2CCN(C(CCC(C)OC)=O)C(CF)C2)=O)ccc(Cl)c(C)c1Cl c1(N(C)CC2CCCN(C(C(COC)O)=O)C2)nc(C(F)F)nc(=N)[nH]1 c1(C(=O)NCCC(CNC(C2CCC(C)(C)OC2)=O)O)cc2cccnc2[nH]1 C(CNC(c1cc(F)ccc1OC)=O)(C(C)C(C)C)NC(c1ccn(CC)n1)=O C1(CC)C(NC(=O)CCSC)CCN1C(C1CC(C)CCO1)=O c1(C(=O)NC2CCC(CNC(C3CCC(CC)O3)=O)C2)cc2cc[nH]c(=O)c2s1 N1(C(c2c(C)cno2)=O)CCC(NC(=O)CC2CCCCC2C)C(C)C1 c1(NC(C(CC)OC)=O)ccc2c(C(=O)NC3CCCCC3)ncn2c1 C(=O)(C#CC1(C)CC1)N(C(CNC(CC(C)SC)=O)C1CC1)C c1(C(N(C(C)CN(C(=O)CCCF)C)C)=O)ccc(Br)cn1 c1(N2CC(CC=C)(NC(c3cc(C(=O)OCC)no3)=O)C2)nccc(CC)n1 N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CC2CC(NC(c3cc(O)cc(Cl)c3)=O)CC1C2 N1(C(c2cc(C)nn2C)=O)CCN(C(c2cc(CO)oc2C)=O)C(CO)C1 N1(C(c2ccc(CC(=O)OC)cc2)=O)CCN(C(=O)C(C)CCN(C)C)C(C)C1 C1(C)(C(=O)NCCN(C(c2cnc(C3CCOC3)s2)=O)CC)CC(C(C)C)=NO1 N1(CC(N2CCC(N(C(=O)CCSC)CCC)C2)=O)CCC(=O)CC1 N1(C(C(C)(C)C(F)F)=O)CCC2(CCC(NC(=O)C3=CCOC3)CC2)CC1 c1(C(=O)NCC2N(C(C(C(CC)O)(F)F)=O)CC2)cc([N+](=O)[O-])ccc1SC CC1(C)C(CC(=O)NC2CCC(NC(=O)CNC(=O)Cn3cncn3)C2)C1(C)C C1(CNC(c2cc(CNC(C3(SC)CC(=O)C3)=O)ncc2)=O)CCCC(C)(C)O1 CC(C)(C)C(C)(C)C(=O)N1CCCC2(NC(=O)C3=CCCC3)CC2C1 C1(CC(N2C(CC)COCC2)=O)C2CCCC2N1C(=O)CC(Cl)Cl c1(CN(C(CCC2(C)CC2)=O)CCNC(C2CC2Cl)=O)cccc(Cl)c1 CC(CCC(=O)NCC(C1CC1)N(C)C(c1ccncc1C1CC1)=O)S(C)(=O)=O c1(CC(C)NC(CNC2(C(=O)OC)COC2)=O)cccnc1 Cc1cc(C#N)sc1C(N1CCC(N(C)C(C2CCC(C)(C)OC2)=O)C1)=O N1(C(c2c(C)nc[nH]2)=O)CCOCC1C(N1CCOC(C(N)=O)C1)=O C1(CCN(C)C(c2csc(=N)[nH]2)=O)CCCCN1C(c1ccc(C(C)(C)C)[nH]1)=O CCC(CC(=O)N(CC(O)CNC(=O)COC(F)(F)F)C)CC(F)(F)F C(=O)(C1CCCn2ccnc21)N1C(CN(C(CC(CCC)C)=O)C)CCC1 c1(C(c2nnnn2C(C)C)NC(COC)COC)cnn(C)c1C(C)C N1(C(C(=O)N(CCC(C)O)C)=O)CCCCCCC1c1ccccc1 c1(C(=O)NC2CCN(C(C3(c4ccn(C)n4)CC3)=O)CC2)occ2c1CCOC2 CCC(C(C)(F)F)NC(=O)CC1CCCC1NC(c1cc(OC)nn1C)=O N1(C(CC=CC)=O)CCC(CO)C(NC(c2ccnc(Cl)c2N)=O)C1 N#Cc1cc(=NCC2CCCCN2C(c2cccc(F)c2)=O)[nH]cn1 c1(C(=O)NCC2(NC(c3ccc(O)cc3O)=O)COC2)n[nH]c2cccc(F)c12 C=CC1(CC(=O)NC2CCCC(NC(=O)Cc3ccc(C)cc3)C2)CCCCC1 C=C=C(C)CC(=O)NCCN(C(=O)CCCc1ccc(Cl)cc1)C Cc1cc(S(=O)(=O)N2CCOC(CC(=O)NCCCCCO)C2)c(C)cc1Cl C=CCCCCCC(=O)NCC1(F)CC2CCC(C1)N2C(=O)Cc1ccco1 c1(C(=O)OCC)ccc(NCc2n[nH]cc2C)cc1O c1(C(N2CC(O)CC(NC(c3scnc3Cl)=O)C2)=O)ccc2ccsc2c1 c1(C(=O)NC2CCC(CNC(CCCS(N)(=O)=O)=O)C2)cnc2ccccc2c1 c1(CC(=O)NCCC2CCC(NC(C3(N(C)C)CCCC3)=O)C2)cnccc1Cl c1(CC)cnn(CNC(=O)C(C)(C)C2CCN(C(=O)CCOC3CCCC3)C2)c1 C12(CNC(C3=NOC(C)C3)=O)CCCC1N(C(=O)CC1(C(F)(F)F)CC1)CCC2 c1(CC(=O)NCC(CN(C(c2cnn(CCC)c2C)=O)C)O)noc(C)c1C#N c1(CONC(C2C(C)CN2C(=O)CC(C)O)=O)ccc(OCF)c(F)c1 C1(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)CC(F)F)C2(CCOC2)C1 C1(C2(O)CCOC2)(C(=O)OCC2CCN(c3c(C)cccn3)C2)CCC1 Brc1cn2c(CCNCC3COC3)cnc2s1 c1(OCCCC)ccc(C(=O)NCCN(C(=O)C(O)c2ccsc2)CCOC)cc1 N1(c2[nH]c(=NCCc3c(C)nn(C)c3C)[nH]c(=N)n2)CC(C)(C)C12CCOCC2 C#Cc1ccc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2CC(OC(C)C)C2)nc1 N1(C(CCc2n(C)c(S)nn2)=O)CC2CCCCC2(CNC(=O)C(N)=O)C1 C1(NC(C(C)(F)F)=O)CN(C(c2cccc(NS(N)(=O)=O)n2)=O)C2(CCOC2)C1 C1(C(C2CCN(C(=O)CCC=CC(C)C)C2C)CC)CCC2(CC1)OCCO2 c1(CN2CC(CC(=O)NC3CCC(CC)CC3)C2)cc(C)c(F)c(F)c1 c1(C(=O)NCC2OCCCN(C(C3C(OC)CC3)=O)C2)ccc2cnc(C)n2c1 N1(C(c2c(C)oc(Br)c2)=O)CC2CC(NC(c3ncncc3Cl)=O)CC2C1 C=C(CC1CC1)C(=O)N1CCC(C(C)OC)C1 c1(C(N(CC(CNC(C(C)OCCC=C)=O)(C)C)C)=O)cccn(C)c1=O c1(CNC2CCN(CCC(=O)OCC)CC2C)cnc2ccnn2c1N C(=O)(C1CC(C)Nc2ccccc21)NC(c1ccc(Br)cn1)C(=O)OC Cc1cc([N+](=O)[O-])cnc1C(=O)N(CC(C)N(C)C(c1cncc(CO)c1)=O)C C(=O)(CC(C)C(C)C)NC(CN(C(c1c(C(=O)OC)nccn1)=O)C)C C1(CN=[N+]=[N-])COCCN1C(c1ccc(CNC(c2ccc(O)cn2)=O)cc1)=O N1(C(CC(=O)OCC)=O)CCC(NC(c2cccn2C)=O)C(O)C1 Cc1ccc(CC(N2C(CNCC3CC(n4cnnc4)C3)CC3CC23)=O)cc1O C(C(C)(C(=O)NC1CC12CC(OC)C2)NC(=O)Cc1cncc(C)c1)SC CC1CN(C(=O)NCCCC2CCOC2=O)c2ccc(Br)cc2O1 CCCCC(C(=O)NCCCN1CCC1)NC(=O)CC1C(=O)NN=C1C c1(OC(C)C)ccc(C(N)=O)cc1CO.C1(C(N(CCNC=O)C2CC2)=O)CC1Cl c1(C(=O)NCCC(C)N(C(=O)C2=CCCC2(C)C)C)cc2sccc2n1C c1(OC)cc(C(=O)NC2CCOCC2NC(c2ccc(=N)[nH]c2Cl)=O)ccc1Cl c1(C(N(CC(O)CN(C)C(c2c(C(F)F)cccc2N)=O)C)=O)c(O)cccc1O Cc1ccc(S(N)(=O)=O)cc1CN1CC(O)C(F)C1 C(C(CNC(N1CCC(O)C1c1ccccc1)=O)C(F)(F)C(F)(F)F)OC C(=O)(C1CN(C(=O)N(C)CC2COC2)Cc2n[nH]cc21)OC O=S(=O)(c1ccc(NCC2CCOC2C(F)(F)F)c(F)c1)N1CCCC(F)(F)CC1 C1(NC(Cc2nnn(C(C)(C)C)n2)=O)(CO)CCCN(c2ccncn2)C1 CC(C)CC(C)(CN(C(C1C2CC1N(C(=O)OC(C)(C)C)C2)=O)C1CC1)CC c1(C(=O)NC2CC(C)(NC(Cc3c(C)scc3)=O)C2)cc(C(F)(F)F)cc(Cl)c1 Cc1ccc(CC(=O)NC2CC(C)(C(=O)NOCc3ccc(F)cc3)C2)cc1 C(CCCCC(=O)N(C)CC1CCCN1C(C1CC2CC1CO2)=O)SC c1(C2C(C(N(CCNC(CCCC#C)=O)CCC)=O)C2)ccc2ccccc2c1 N1(C(C(C)C)=O)CCC(C)(C)C(CNC(=O)CC(C)c2cnn(C)c2)C1 C1(CNC(c2c(Cl)cnc(C)n2)=O)CC2(CO1)CN(C(=O)CCC1CC1(C)C)C2 C1(CC(=O)NC(c2cn(Cc3ccc(Cl)cc3)nn2)CCC)CC2C=CC1C2 C(CC(C)CCNC(c1c[nH]cc1Cc1ccccc1)=O)NC(C(C)C)=O Cc1cc(CNC(C2SCCS2)=O)oc1C(=O)N(CC(C)O)CCF C(=O)(CCCCCN(C)C)NCC(C1CCN(C(=O)CSCC(F)(F)F)CC1)C N1(C(C2N(C(C)C)CCCC2)=O)CC(NC(c2ccncc2Cl)=O)C(C2CC2)C1 N1(C(=O)NCN2CCC2c2ncon2)CCCC(NC2(C)CCC2)C1 c1(CC(=O)N(CCC(C(C)C)NC(C(C)SCC)=O)C)ccc(F)cc1Cl c1(OC)cc(NC(=O)CSCc2ccc(C(=O)O)cc2)ccc1C c1(C(=O)NCC2(C)CCN(C(C(C=C)O)=O)C2)cc(S(N)(=O)=O)c(C)cc1C Cc1cc(C(=O)NC(C)(CNC(=O)CC2CC3C=CC2CC3)CO)cc(N)c1 N1(C(CSC)=O)CCCC2(CNC(C3CCC(C(N)=O)CC3)=O)CCCC12 C(C(=O)N=c1ccc2cc(Br)ccc2[nH]1)NCCCCSC N1(C(=O)NCCc2cccc(Br)c2F)CCC2CS(=O)(=O)CC2C1 C(=O)(C1=CCCN(C(C2C3CCC(F)C23)=O)C1)NC(C)C(C)n1cccn1 c1(OC)nc(C(=O)NCC2(C)CCC(NC(c3cc(Br)no3)=O)C2)ncc1F CCC(CC(=O)NCC1(C(C)(C)O)CCC1)NC(C1CC1(F)F)=O C(=O)(C(C)(C)CC(C)(C)C)N1C2C(NC(c3cncc(OCC)c3)=O)C(C2)C1 c1(OC)c(C(N2CCCC2(C)C(=O)NC(C2CCCC2)C)=O)cccc1F c1(C(=O)NC(C2N(C(C3C(C)C3C)=O)CCC2)(C)C)ccnc(F)c1 c1(CC(=O)N(C2CCCN(C(C(C)OCCC#C)=O)C2)C)ncc(F)cc1F c1(-c2c(NC(N3C(C)CN(C)CC3)=O)nccc2)cccc2nc(O)ccc12 N1(c2nc(C(C)C)nc(N3CCC(c4ccco4)CC3)c2)CC2CC(O)CC2C1 C1(CS(N2CCCC(C(F)F)C2)(=O)=O)CCn2cnnc2C1 C12(OCC)CCC(C(N3CCCC(CN(C)C(c4nncn4C)=O)C3)=O)(CC1)C2 N1(C(CCS(=O)(=O)NC)=O)CCC2C(C1)CN2C(=O)C(C1CCCCC1)O N1(C(c2cnc(N(C)C)nc2)=O)CCC2(CC1)CN(C(=O)C1=CCCCO1)C2.CN C(N=c1[nH]c(N(C)CC2CCCC2O)nc2c1SCC2)c1c(C)cn(C)n1 CCCCCC(O)C(=O)N1CCN(C(c2ccn(CC)n2)=O)CC1CCCC c1(C(N2CCC(OC)(CNC(C3CCCC3C(C)C)=O)C2)=O)cc(F)ccc1F c1(C(=O)NCC(CCNC(=O)Cc2cncs2)O)nccc2ncccc12 C1(NC(C(=O)N(CCC(=O)N(C)C)CCCO)=O)CC2CCCCCC2C1 c1(C(N2CCC(NC(C3CCC4CC34)=O)CC2)=O)c(F)cc(Cl)cc1F C1(CC)CCC(C(=O)NCCC2(NC(c3cc(C4(O)COC4)on3)=O)CCC2)C1 C1(CC(=O)NCCC(=O)NC(C)(C)C)C2CN(C(C3CCSC3)=O)CC12 c1(C(N2CC(NC(C3CC3F)=O)CC23CCC3)=O)cncc2cc(Cl)ccc12 c1(C(=O)NCC(Cn2cc(COC)nn2)(C)C)cc2sc(C)cc2s1 c1(CC(=O)N(C(C)=O)C(C2CC(O)C2)C2CCCO2)nc(Cl)cs1 C1(C(N(C(C2CCCC2)(C)C)C)=O)CCC(n2cc(CC3CCOCC3)nn2)C1 C=CC(C)(CC)OC.C(=O)(C(C)NCC(F)(F)F)OCC(C)(C)O C(c1ccccc1)(C(F)(F)F)=CC(=O)NCC1CC(NC(C2CC2(F)Cl)=O)C1 C1(C(=O)NC(COCC)C)CC(NC(c2cc(NC)ncn2)=O)C(O)C1 C#CCCCCCCCC(=O)N1CCN(C(c2cnc[nH]2)=O)CC(O)C1 CC1CCN(C(c2cnc(Cl)n2C)=O)C1C(=O)N(CC(O)CO)C N1(C(C(C)SC)=O)CC(F)CC1CC(=O)NC12CC(F)(C1)C2 C1(CC(=O)NC(CN(C(=O)CCCOC(C)(C)C)CC)C)C=CCCC1 CC1=CCN(c2cccc(NC(=O)C(C)COCCO)n2)CC1 N1(C(CS(CC)=O)=O)CCC2CCCC(C1)N2C(=O)C(F)(F)c1nccn1C Cc1cc(NC(=O)NC2CCC(c3ccccc3)C2)n(C2CCOCC2)n1 N1(C(=O)CN2CCOCC2)CC2CCC1CN2C(c1cc(Cl)ncc1Cl)=O C(=O)(CCCC(=O)NC1CCOC1C(=O)NCc1ncc[nH]1)N(C)C Cc1ncccc1C(N1CCC(C)C1C(=O)NC(CCO)C(C)C)=O c1(CNc2c(OCCOC)ccc(Br)c2)ccc(N)c(C)c1Cl c1(CC)ccc(C(=O)NCCC2CCCN(CCOC)C2)cc1[N+](=O)[O-] N1(CC)C2CCC1CC(N(C1(c3cn(-c4sc(C)cc4Cl)nn3)CCSC1)C)C2 c1(NC(C2CC2F)=O)cccc(NS(=O)(=O)Cc2cccc(Br)c2)c1 C(=O)(CCC(CF)CF)NC1CCCC(C(N2CC3C(C)C2C3)=O)CC1 N1(C(C2(NC(c3csc(=N)[nH]3)=O)C(C)C2)=O)CCC2(CC2)C1 S(CS(C)(=O)=O)CC(=O)N(CC(=O)N(C)C)CCOC c1(C(N(CCN(C(C(COCC)(C)C)=O)C(C)C)C)=O)cnc2cc[nH]c2c1 C(c1ccc(C)cn1)=CC(=O)N(C1CCCC(N(C(CC=C(C)C)=O)C)C1)C c1(N2C3C(NC(C=CCCC)=O)(CCC3)CC2)c(F)cc(C#N)cc1[N+](=O)[O-] Cc1nc(NCCSc2ccccc2)cc(=NCCN2CCCC2)[nH]1 C1(NC(C(c2cccc(C)c2)F)=O)CC2CC1N(C(c1[nH]nnc1C)=O)C2 Cc1cc(Cl)ccc1CC(=O)NCC1(CNC(C2CNC(=O)C2)=O)CC1 c1(NC(C23C(CN(C(C=CC)=O)C2)C3)=O)cc(C)c(O)cc1C C(=O)(C1=CCC(F)(F)CC1)N1CCC(OC)(CNC(C2(C)CCCS2)=O)C1 n1(CC)nc(C)cc1C(=O)NC1(CC(=O)NC2CCCC2(C)CO)CCC1 c1(OC)cc(C(N2CCC(NC(=O)COCP(C)(C)=O)C2C)=O)c(F)cc1N C=CCCCCCCCC(=O)NCC(CC=C)NC(=O)CC12CC(C1)C2 c1(C(C)C)ccc(NC(C2CN(C(=O)CSc3nnnn3C)CCO2)=O)c(Br)c1 N1(C(c2c3n(nc2)CC(C)CO3)=O)CCOC2(CCN(Cc3cnon3)CC2)C1 CCC(C)(CO)C(=O)NCC(C)CN(C)C(c1cnc(=N)[nH]c1)=O c1(C(N2CC=C(CNC(c3c(C)nccc3)=O)CC2)=O)cccc2cc[nH]c12 C1(NC(C(C2CCOC2)OC)=O)CCN(C(c2cc(N)c(F)cn2)=O)C(C)C1 C1(CC)CN(C(c2cnc(CC(C)C)s2)=O)CCN1C(c1cncn(C)c1=O)=O CCCC(CCCNC(=O)CNC(C)=O)NC(c1sc(NC(C)=O)cc1C)=O N1(C(CC(OCC)OCC)=O)C2CC1CN(C(c1ccc(O)cc1C)=O)C2 c1(SCC)ccc(C=CC(=O)NCC2(NC(=O)C(C3CCCCC3)OC)CC2)cc1 Cc1cc(C(=O)NCCc2n[nH]cc2C(=O)NC2(C)CCOC2)no1 CCCC(CCC)C(=O)N(C)CCN(C(=O)C(c1ccncc1)C1CCCC1)C c1(NC(c2cnn(CC(F)(F)F)c2C2CC2)=O)cc2cccc(O)c2[nH]1 C(C(CC(F)(F)F)NC(c1cncc(N)c1C)=O)NC(C(CC)C)=O CCCCCCC(=O)N1CCCCC(N(C)C(c2cnc(OCC)cn2)=O)C1 N1(C(c2c(C)nco2)=O)CCN(C(C2CCC(=O)N2C)=O)C(CC(F)(F)F)C1 c1(OCC(=O)NC2CCN(Cc3cnc(COC)s3)C2)ccc2c(c1)OCO2 C1(C(N(C)Cc2cccc(CNC(C3CC(F)C3)=O)c2)=O)CC2C(C1)C2(F)F CC1CCCCC1(CNC(C1(C)CCCCC1)=O)NC(=O)COc1ccccc1 C(=O)(CS(=O)(=O)C(C)C)N1CC(SC)C(NC(=O)C=Cc2ccccn2)C1 C1(C)(C(N(CC(CN(C)C)(C)C)C)=O)CCN(C(C2CCN2C2CCCC2)=O)C1 C(=O)(C1CCc2nccn21)NC(C(=O)NC(c1ccc(C)cc1)C)c1cccs1 C1(CCC)(NC(c2cn(CCCC)nn2)=O)CCN(C(=O)C(COC)OC)CC1 C(=O)(C1=CC(O)C(NC(=O)C(C2(O)CCCC2)F)C1)NCc1cc(C)on1 c1(SC)ccc(Cl)c(C(N2CCC(CNC(=O)C(CO)NC(=O)C(C)C)C2)=O)c1 N1(C(CCN(C(c2cc[nH]n2)=O)CC)=O)CC2CC1C2N(C)C Cc1cc(C(=O)NC2CN(C(c3c[nH]c(=N)c(C)c3)=O)CC2F)c(C)cc1F c1(C(=O)NCC(=C)C)ccc2c(c1)C1CN(C(=O)C(C)=O)CC1NC2=O C1(NC(C(C)=C(CC)C)=O)C(CNC(=O)CCc2ccn(C)n2)CCC12CCC2 C1(C(=O)NCC2(COC)CN(C(=O)C=CC3CCCO3)C2)CC(=O)NC(=O)N1 CN1CCC(N=c2cnc(C(N)=O)c[nH]2)(C(F)(F)F)C1 C1(C(N2CC(OCCNC(C3C(C#N)C3)=O)C2)=O)CC2CCC1C2 N1(C(=O)NCc2nccc(OC)c2)CC2CCCCN2CC1C c1(NC)cnc(C(N2CC(F)(CNC(=O)C=Cc3ccc(C(N)=O)o3)C2)=O)cn1 C(=O)(C1=COCCO1)N1CC(CNC(c2c(C)nc(CCCC)s2)=O)C(O)C1 Cc1n[nH]c(C)c1S(=O)(=O)NC1CN(Cc2cc(Br)cc(Cl)c2O)CCC1F O(NC(=O)C(Cc1cc[nH]n1)NC(=O)Cc1scnc1C)CC(COC(C)=O)O c1(OC)c(C(=O)O)cccc1C(C)NC(C1(c2ccccc2)CCCCO1)=O N1(C(c2cc(S(N)(=O)=O)cs2)C(=O)NCCSC)CCCC2(CCNC2=O)C1 c1(C(N2CC3C(CNC(c4ncn(C)n4)=O)(C3)C2)=O)cc2cccc(F)c2o1 N1(C(C2C(C=C)C2)=O)CC2(CC(NC(c3cc(-c4cn(C)nn4)on3)=O)CO2)C1 c1(C(N(C)CCNC(=O)C=Cc2ccccn2)=O)ccc(Cl)c2c1OCCO2 c1(C(=O)NC2CCN(C(C=C(C)C(C)C)=O)CC2C(C)C)cc2c(nn1)CCC2 CCCC(C)CC(=O)N1CC2(CC2)CC1CNC(=O)CCn1ccnc1 c12cc(cc3ccccc13)NC2=O.c1(OC)nc(-c2nn[nH]n2)c(C)o1 N1(C(C2(C(C)C)CC2)=O)CCCC(N(C)C(c2cnn(C)c2F)=O)C1 C1(CNC(CCCCNC(C)=O)=O)CN(C(c2cnc(N(C)C)s2)=O)CC1(C)C c1(-c2cc(CCC(=O)N(C3CCOCC3)CC)no2)ccc(F)cc1F N1(C(CCCOCC)=O)CCC2(C1)CN(C(c1nccc3occc13)=O)C2 C1(CNC(Cn2c(C)ncc2)=O)CC(NC(C2CC(CF)C2)=O)CC1O c1(CNC(N(CCCF)CC)=O)ccc(OC(F)(F)F)cc1C CC1(C)C(NC(c2cc(Cl)no2)=O)CC1CNC(c1ccccc1SCCO)=O N1(C(c2ccc(C)cc2O)=O)CCC2CCC(NC(=O)C(C)C3CCCO3)C1C2 Cc1nc2ccnn2c(C)c1C(=O)NC1CC1NC(=O)CC(C(C)C)C(C)C C1(c2n(CCCOC)nnn2)(NCc2ccc(F)c(F)c2)CCCN(C)C1 C1(NC(c2c(C)nc(C(C)C)s2)=O)CC(F)CN(C(=O)CCN2CCCC2=O)C1 C(CC(C(=O)N1CC(NC(c2nc(C)nn2C)=O)C(O)C1)NC(N)=O)SC c1(C2(CN=C(NC(CC)CC)NCc3nc(C)c(C)s3)CC2)cc(C)cnc1F N1(C(c2ccc(F)c(C(F)(F)F)c2)=O)CCC(C2CCN(C(C3CCC3)=O)C2)C1 C1(CC(=O)NCCOCCNC(Cc2cn(CC)nn2)=O)CCCC(=O)C1 C1(C(=O)NC(C(=O)OC)C(C)C)CC(C)CN(C(=O)CC2C=CCCC2)C1 c1(C(C(=O)NCc2nnn(C)n2)N(CCOCC=C)C)ccc2c(n1)OCCO2 C12(NC(c3c(Cl)ccc(CC)c3)=O)CCCC1N(C(=O)CCCC1CCC1)CC2 N1(C(CCC)=O)CCCC(N(C(=O)C(F)=CC2CC2)CC2(COC)CC2)C1 C1(C(=O)NC2CC(OCC)C2)C2CCCC1N(C(=O)CC(C)(C)SC)C2 C1(C(=O)NC(CNC(c2coc(Cl)n2)=O)CO)CCCC2(CCCCC2)C1 CC1(C)CCC=C(C(=O)NC2(CNC(c3sc(C#N)cc3Cl)=O)CCC2)C1 CC1Cc2c[nH]nc2CC1NC(c1ccc(NC(=O)C(=O)N(C)C)c(F)c1)=O C1(C)(CNC(c2ccnc(C)n2)=O)CCN(C(=O)CCC2CCCCN2C)CC1 N1(C(C(COC)(C)C)=O)CCC2CN(C(=O)Cc3cn[nH]c3)CC2C1 c1(N2CCC(OC)C2)nnc(CCN2CCCC2)n1CCc1cccs1 CC1(C)CN(C(=O)CC2=CCN(C(C3CCCC4(CC4)C3)=O)CC2)CCCO1 CCC(CC(=O)N1CC2(CCN(C(C3CCC3c3nc[nH]n3)=O)C2)C1)C(F)F N1(C(C(C)=CC2CC2)=O)CCC2C(NC(c3ccc(OC(F)F)nc3)=O)CC12 C1(C(=O)OC)CC(n2ccnn2)CN1C(C1CN(CC2CNC2)C1)=O N1(C(c2cnc(CC)nc2O)=O)C2CCCC1CN(C(C1CCCOC1)=O)C2 c1(C(N2CCC(C(C)(C)NC(C(C)NC(CC)=O)=O)C2)=O)cc(O)nc(O)n1 c1(CC(=O)NC2CN(C(CN(C3CC3)CC)=O)CC(O)C2)n[nH]c2c1CCCC2 O(NC(=O)CCOCCCO)CC(=O)N(CC(F)OC)CCO C1(CNC(C(C)CO)=O)(NC(=O)C=CC=C(Cl)Cl)CC(F)(F)C1 N1(C(C2CCC(C)O2)=O)CCCC2(C1)CN(C(=O)CN1CCOC1=O)C2 C1(C(=O)OC)C(C2CC2)CCN1C(=O)NCCCSC(F)F C=CC(C)(CCOC)C(=O)NCC(C1CC1)NC(C1(C2CCCO2)CC1)=O C1(NC(c2cc(C)cc(Cl)c2)=O)CCN(C(=O)C(C)O)C12CCCC2 C#Cc1ccc(OC)c(C(N2CCC(C)C(NC(=O)Cn3ccc(C)n3)C2)=O)c1 CC(C)CCCCCC(=O)NCC(C1CCCCC1)NC(c1coc(C(N)=O)c1)=O c1(CCC(N2C(CN(C(C(F)=CC)=O)CC)CCC2)=O)ccc(O)nn1 c1(OC2CN(C(C(c3c(C)cncc3)C)=O)CC2C)ccc(Br)cc1F C1(C(N(CC(C)O)CCO)=O)CC(NC(=O)CN2CSCC2=O)CCO1 c1(C(=O)NCCCN(C(c2sccc2SC)=O)CC)ncc(C)nc1OC N1(C(C(CC(C)C)C)=O)CC(C(=O)NC2(CN(C)C)CCC2)C2(CCC2)C1 N1(C(c2cn(CC)nc2)=O)CC2(C=C(C(=O)N3CC(O)C(O)C3(C)C)CO2)C1 C1(NC(COCC#C)=O)CC2CC(NC(c3ccc(C(F)F)cc3F)=O)CC12 C1(C(N2CCC(CC=C)(NC(=O)CNS(N)(=O)=O)C2)=O)COC(C)(C)CO1 c1(CC)ccc(C(N2C3CCC2CN(C(=O)C(C)NC(N)=O)C3)=O)cc1C#N N1(C(CCn2ncc(C)c2)=O)CCC(C)(C)C1CC(=O)NCC1=NOC(C)C1 CC1(CNC(=O)COCCN(C)C)CCCN1C(=O)Cn1nccn1 c1(C(C)C)ccc(C(=O)N(C)CC2CCN(C(=O)C(O)CC(F)F)C2)cc1F Cc1nc(N(CCCNC(c2ncccc2Cl)=O)C(C)C)cc(O)n1 c1(N2CCCC(NC(C(CCSC)O)=O)C2C)cc(C#N)nc(C)n1 N1(C(CC2CCN(Cc3ncc(C)cc3F)CC2)=O)CCc2cc(F)ccc2C1 C1(CNC(c2cnn(CC)n2)=O)CCC(NC(=O)CCCc2n[nH]c(=N)s2)CC1 N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCC(CNC(=O)CC(F)F)C(O)C1 CC1CN(C(=O)C=Cc2cc[nH]n2)CCC1NC(=O)C(c1ccccc1)C c1(N(C(C(=O)NC(C)CNC(=O)CC2CC2C2CC2)C)C)nccn2cnnc12 C1(C(C(=O)NC(CNC(=O)Cc2ccoc2)CO)OC)CCCCC1 N1(C(c2cc(F)cc(F)c2)=O)CC2CCCCC2(CNC(C2CC(O)C2)=O)C1 c1(-c2cc(C)c(=N)[nH]c2)cccc2c(C(=O)NCc3noc(C)n3)[nH]nc12 N1(C(CC2CCN(C)CC2)=O)CCN(C(=O)Cc2c(O)ncnc2O)C(CF)C1 c1(C(=O)NCCCCN(C2CCC(F)(F)CC2)C)nc(F)ccc1Br c1(C(N2C3C(NC(CCC#C)=O)C(C3)C2C)=O)ccnc2[nH]c(C)nc12 Cc1cc(NC(=O)CC2C=CC(NC(=O)C(N3CCCCC3)C)C2)ccc1Cl c1(C(C(=O)NCC=C)N(C2(CCNc3ccccc3)CC2)C)ncc(CC)o1 c1(C(N2CCN(C(=O)CSc3ccccc3)C3C2C3)=O)ccc2c(c1)OCCN2 C1(C#N)(C(=O)NC(C2CC2NC(c2cc(F)ccc2F)=O)C)CC12CCCC2 CC(CC(=O)NCCCN(C)C(c1csc(C(F)(F)F)n1)=O)c1cccnc1 c1(NC(C2N(CC)CCSC2)=O)cc(Cl)cc(Br)n1.c12ccc(cc1)CNC2=O c1(OC)cscc1C(=O)NCCC1CN(C(c2cnc(S)[nH]2)=O)C1 c1(C(=O)NCC(CC)NC(=O)CC2CCOCC2)ccc(OC)c(S(N)(=O)=O)c1 C1(NC(c2ccc3c(c2)CCC3)=O)CN(C(c2ccsc2)=O)C2(CCCOC2)C1 O=S(=O)(c1ccc(Nc2ccnc3ncnn23)cc1)NCC1CC1 C1(CN(C2COCC2O)CCCC)CCCN(C(C)=O)C1 Cc1cc(C#N)sc1C(=O)NC1CCCCC1NC(C1CC12CCCC2)=O c1(N2CC(NS(CCC)(=O)=O)C2)nccc(=NCCCCCN2CCCC2)[nH]1 C(=O)(CC(C)CC(C)C)NCC(CCCC)NC(c1cc2ncccn2n1)=O c1(C(N2CCN(C(C3CCCC(=O)O3)=O)C(C3CC3)C2)=O)cncc2nc[nH]c12 c1(OC)cccc2c1OCCC2NC(c1ccoc1C)c1nnnn1C1(C)CC1 c1(CC)cn2c(n1)CCC(C(=O)NCCC(C)NC(c1c(C)cnn1C)=O)C2 c1(OC)ccc2c(C)c(C(=O)NCC3CCCN3C(C3CCC(=O)O3)=O)[nH]c2c1 c1(OC)cc(F)ccc1CNC1CC1C(=O)Nc1cc(F)ccc1C Cc1cccc(C)c1C(=O)NC(C)Cn1cc(-c2cc(F)ccc2N)nn1 C=C(C)CC(Cc1ccccc1)NC(C1CC1C1CC1C(c1ccccc1)=O)=O N1(C(c2ccc(C#C)cc2)=O)C(C)CC2CN(C(C3CC4C(C3)C4(F)F)=O)CC12 C(c1cocn1)=CC(=O)NCC(CNC(=O)C(C)C#N)OC C(CCCCN=[N+]=[N-])NC(CCC1CC(NC(C(C)n2cccn2)=O)C1)=O C1(O)(C(=O)NC2CC3CN(C(CCC(=O)NC)=O)CC32)CCC(C)(C)CC1 c1(C(=O)NC(C2CCN(C(C3CCOCC3)=O)C2)C)cc2cccnc2[nH]1 S(=O)(=O)(c1ccc(C)cc1)CC(=O)NC(CC(C)NC(c1scc(C)c1)=O)C c1(C(N2CCC(N(C)C(C3CC=CCO3)=O)C2)=O)coc2c1NC(=O)CCC2 C1(C(=O)NCC(n2ccnc2)C)COCCN(C(=O)CC2CCC(=O)NC2)C1 CCCC(C)(C)CC(=O)N1CCC(CNC(C2CC3CCC3C2)=O)(OC)C1 Cc1cc(C)c(C(=O)NCCCCCN(C)C(C2CN3CCC2C3)=O)cn1 c1(CCC)ccc(C(=O)NCC2CC2NC(=O)CNC(=O)CC(C)(C)C)cc1 C1(N(C(CN(CCOC)C)=O)C)C2CN(C(=O)C(CC3CC3)CC3CC3)CC12 N1(C(C2(F)CN(C(c3nccc(CC)c3)=O)C2)=O)CC(C#N)C2(CCC2)C1 Cc1nc(C2CC2)ncc1C(=O)NC(C)CNC(c1cnn(C(C)(C)C)c1)=O C1(C(=O)OCC)CCCC(C(=O)NC23CC(NCc4ncccc4C)(C2)C3)C1 C1(OC(c2ccc(OC)cc2)=O)CCN(N2Cc3ccccc3CC2C(N)=O)C1 N1(C(C2CC(C)(O)C2)=O)CCC2(NC(C3(n4cnnn4)CC3)=O)CCCCCC12 N1(C(c2c(C)cccn2)=O)CC2(CCN(C(=O)CC3CC(C)CC(C)(C)C3)C2)C1 c1(C(=O)NC2C3CN(C(C4C(C(=O)OC)C4)=O)C2CC3)cc2nccc(Cl)c2s1 c1(C(=O)NCC(CNC(C2(C)N(C(C)=O)CCC2)=O)(C)O)ccc2nnnn2c1 C1(NC(C2CC(N3CC(F)C3)C2)=O)CCN(Cc2cnn(-c3ccccc3)c2)C1 C1(N(CCC)C(c2c[nH]c(Br)c2)=O)CCN(c2ncns2)CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(CN(C(C2C=C(C)CS2)=O)C)COCC1 c1(C(=O)NCCNC(C23CCC2C3)=O)cccc(-n2cnnn2)c1.C1(C)CCCC1 c1(NC(c2scnc2-c2ccc(C(F)(F)F)nc2)=O)cc(F)ncc1F C(=O)(C(C(C)(C)C)n1cc(C2CCCCC2O)nn1)NCC1(C)CNC(=O)O1 N1(C(c2c(C)nn(C3CCCC3)c2)=O)CC2CC1CN2C(C1CC1c1cnc[nH]1)=O C1(NC(CCOCCOC)=O)CC2(C1)CC2NC(=O)C(c1ccccc1F)(F)F C(=O)(CS(=O)(=O)CC(=O)NC1CN(C(C2CCCC2(F)F)=O)CC1(C)C)OC N1(C(C(CC)OC)=O)CCC(F)CC1C(=O)NC(C)(C)COC(C)C c1(-c2nc(C3(C(C)C)CC(=O)C3)on2)ccc(C(=O)NC2CC23CCOC3)nc1 C1(c2nnnn2CCCSC)(Nc2cc(CC)nn2C)CC2(COC(C)C2)C1 N1(C(C2CCC(C)(C)CC2)=O)Cc2nccn2CC(NC(=O)C=C2CCCC2)C1 c1(C(N2CCC(C(CO)NC(c3cc(Cl)no3)=O)CC2)=O)cc2n(n1)CCOC2 CCC(CCC(=O)NOC(COC)COC)NC(=O)CCN(C)C c1(C(=O)NC2CCC(CNC(c3cc(C)n(C)n3)=O)C2)ccc2ocnc2c1 C1(OC)CC(NC(=O)CN2CCCS2(=O)=O)C12CCN(C(c1cn[nH]c1)=O)CC2 c1(OC)ccc(F)c(CN2CCN(S(=O)(=O)CCCCCl)C(C(C)C)C2)c1OC N1(C(c2c(OCC)ccs2)=O)CC(NC(c2nc(C)nn2C)=O)C(O)C1 N1(C(CCN(CCN=[N+]=[N-])CC(N2CC(OC)C2)=O)=O)CCC2CC3C(C2)C13 C1(CC)CCCCC1C(=O)NC(c1ccnn1C)C(=O)N(C)CCOCCO c1(CC(C)C(=O)NCC(CO)NC(=O)CCOCC(F)(F)F)ccc(Cl)cc1 C1(O)(CCNC(C2CC(OCC)C2)=O)CCN(C(C2OCCC2C)=O)CC1 c1(C(=O)NCC(CN(C)C(c2cc[nH]c2)=O)(C)C)cn(C)nc1-n1cncn1 c1(C(N(C(CNC(=O)C(O)C(C)(C)C)C2CC2)C)=O)ccc(=O)n(C)n1 N1(C(CCC(C)SC)=O)CC(C(=O)O)CC(O)(C(F)(F)F)C1 N1(C(c2c(C)nccn2)=O)CC(C)(C)OCC1CNC(C1CSCCS1)=O c1(OC)ccnc(C(=O)NCC2CCCC2NC(C2(C)CCCO2)=O)c1 C1(OCCOCC)CCCN(C(C2(C)CNC(=O)N2)=O)CC1 C1(CC)(CC)CC(C(=O)NC2CC(C(F)C(=O)Nc3cnsc3)C2)C1 c1(CN(C)C(C2CCCCCC2)=O)ccc(C2(c3nn[nH]n3)CCOCC2)cn1 N1(C(CN2CCC(C)C2)=O)CCN(C(CNC(C2(CCO)CC2)=O)C(F)F)CC1 C1(C)(C(N(CCC#C)C)=O)CCN(C(=O)C=CC2(C)COC2)C1 C1(C(N2CC(C(N(CCOCCO)CC)=O)OCC2)=O)CC2CCCC2C1 c1(C(=O)NCC2CCC(NC(C3ON=C(C)C3)=O)C2)c(C)csc1Cl C=CCCCCC(=O)NCC1(NC(=O)CC2(O)CCOC2)CC1 CC1CN(C(c2ncc(Br)cn2)=O)CCCN1C(c1cnc(O)s1)=O C1(CC(=O)N(c2ccc(-c3nc(C)on3)cc2)C)CCNCCC1C.C(=O)C(C)=O C(=O)(CCCC(C)(F)F)NC(CNC(C(COC(C)=O)C)=O)C(C)C C1(CC(NOCC2(C)CCC2)=O)CN(C(C2CNC(=O)C2)=O)C(C)(C)C1 c1(OC)ccc2c(C(=O)NC3(C)CCCN(C(C4(O)CC4(C)C)=O)C3)n[nH]c2c1 C1(NC(CCCCC#C)=O)CCCC12CCN(C(c1cnc(CC)s1)=O)CC2 C=C(Cl)CC(C(=O)NC1CCCCC1C#N)NC(=O)C=CC(=O)OCC C1(C(=O)NCC2(C)CCCN2C(c2cc(Cl)cnn2)=O)CCS(=O)(=O)C1(C)C C1(CC)CN(C(=O)C=CCNC(=O)Cn2ccc(CC)n2)C(CC)CO1 c1(C(=O)NC2CC(CCNC(C3(N(C)C)CC3)=O)C2)ccc(S(N)(=O)=O)cc1Cl c1(C(N2CC(NC(C(CC)N(CC)CC)=O)(CF)C2)=O)cc(F)c(F)cc1O N1(C(C2(CSC)CCC2)=O)CCCC(NC(=O)CCc2cnc[nH]2)C1C C1(CC)CCCC(NC(C2CCN(C(c3ccc(SC)o3)=O)C23CC3)=O)CC1 C1(NC(CCN(C)CC)=O)CCC(O)CN(C(C2(C)CCN(C)C2)=O)C1 C1(CNC(=NCC)NCC(=O)NC2CCCCC2)CCC2(CCCCC2)O1 Cc1sc(CNC(=O)NC2CCC(C(F)(F)F)CC2)nc1C1CCCOC1 C(=O)(C(=O)CC(C)C)NCC(C1CCOC1)NC(C1(COC)CC(=C)C1)=O c1(OC)ccc2nc(C(=O)NCC3CC(OC)CN3C(=O)C=C3CCC3)cn2n1 C1(NC(C2(C)CCSCC2)=O)CN(C(=O)Cc2cn[nH]c2)CC2(CCOCC2)C1 c1(OC)cc(OC)cc(CCNC(c2ccccc2N2CCOCC2)=O)c1 C1(C(N2CC(CC(C)NC(c3c(C)nns3)=O)C2)=O)CCc2nnnn2CC1 C1(CC)CCC(C(=O)NCC2COCC2NC(=O)CCNC(=O)CC(C)C)O1 C1(NC(C2CC(N(C)C)C2)=O)CC1C1CCN(C(=O)C=Cc2cn(C)nn2)CC1 C1(CCC)(NC(c2cn(CCCC)nn2)=O)CCCN(C(=O)C(C)(CC)CC)C1 N1(C(CCCCOC)=O)CC2CCC1C(NC(c1ncccc1Cl)=O)C2 c1(NCC2(OC)CC2C2CCOCC2)ccc2[nH]c3c(c2c1)CCCC3C#N C1(CNC(c2ccsc2C(F)F)=O)CN(C(C2(CO)CCCC2)=O)CCCO1 N1(C(c2ccc(COC)cc2)=O)CCCC2CN(C(c3cn(C)nc3Cl)=O)CC12 C1(CNC(=O)CCc2ccccc2)C2CC2CN1C(=O)Cn1cc(Br)cn1 c1(C(=O)NCCCC(C)NC(C2C(F)(C(=O)OC)C2)=O)cc(C(F)(F)F)cn1C c1(CC(=O)NC(CCCCNC(c2ccc(OC)s2)=O)C)cccc(F)c1Cl N(C(=NCCCc1ncn(C)n1)N1CCN2C(=O)OCC2C1)CC(CSC)(C)C C(c1ccncc1)=CC(=O)NCC1(F)CC(NC(c2ccoc2C(F)(F)F)=O)C1 C1(C(=O)Nc2c(C)nccc2)CC2CCCCC2N1Cc1cc(F)ccc1Br c1(C(=O)NC2CCC(CNC(CCC)=O)CC2)cc2scnc2[nH]1 c1(C(=O)NCC(C)N(C(=O)C=Cc2cncn2C)CC)ccc(Cl)cc1F Cc1ncc(C(N2CCCC2C2(NC(c3cccc(O)n3)=O)CC2)=O)cn1 CC1(C)CN(CC(=O)NN2CCCC2)C1.C1(CCCCO)(N2CC2=O)CCC1 C(C(C)C(C)(C)C)NC(C(CC)N(C)C(c1ccc(COC)o1)=O)=O c1(C(=O)NC(C(C)NC(c2cn(CCC)nc2)=O)C)ccc(OC(C)C)cc1 N1(CC(=O)NC2(CC=C)CN(C(c3ocnc3C)=O)C2)CCN(CC)C(=O)C1=O N1(C(C2CC=CC2)=O)CCC(C2CCN(C(C3CC4CCC3C4)=O)C2)CC1 c1(C(=O)NCCCNC(C(c2ccc(Cl)cc2)OC)=O)cccc(Cl)c1N CC1CC=C(C(=O)NCC(=O)N(CC(C)C(F)(F)F)C)CC1 C1(CNC(C(COC)NC(C)=O)=O)CC2CCCC2N1C(c1cccc(=O)o1)=O CCCCC(C)C(=O)N1CC(n2cc(C(C3CCCC3)OC(C)=O)nn2)C(C)C1 C(=O)(CCC(=O)N(CCCCCCNC(=O)C(F)(F)C1CCC1)C)N(C)C C1(NC(c2cnc(C)[nH]c2=N)=O)CN(C(C2CCC(C)O2)=O)Cc2nccn2C1 c1(C(=O)NCC(C2CC2)NC(C2(CO)CCC2)=O)ccnnc1NCC1CCC1 C1(CNC(C2(CC)CCC2)=O)CN(C(c2cc[nH]n2)=O)C2CC12 C(=O)(C#CC1(CC)COC1)NC(c1nncn1C)C(=O)N(CC(CC)OC)C C(=O)(C(C)S(N)(=O)=O)NCC(N(C(CCn1c(C)ncc1)=O)C)C1CC1 C1(CNC(c2c(C(C)C)cco2)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C12CC2 C12(CNC(c3n(CCC)ccc3)=O)CC1CN(C(=O)Cc1cc(COC)on1)C2 CC1C(=O)CC1C(N1CC(C)(NC(=O)CN2CC3CC3C2)C1)=O O=C(CCS(=O)(=O)C(F)(F)F)NC1CCC(CCNC(=O)Cn2cccn2)C1 c1(C(=O)NCC2(C(N(C)Cc3cnn[nH]3)=O)CCC2)ccc(Cl)cn1 C(C(CNC(C1(C)CCCCO1)=O)C(F)(F)F)NC(CC(=O)OCCC(C)C)=O C12(CNC(c3cc(C)no3)=O)CCCC1N(C(=O)CN1CC3C=CC1C3)CCC2 c1(C(=O)NCC2CC(C)N(C(c3cnn(C)c3Cl)=O)C2)n[nH]c2ccc(Cl)cc12 C1(C(=O)NC(C2CCCO2)(C)C)CC2CCCC2N1C(=O)CC1NC(=O)NC1=O Cc1sc(C(=O)NC2CC(NC(=O)C(C)Cn3ccnc3)CC2O)nc1O C1(C(N(CC(C)NC(=O)CC2CNC(=O)O2)CC)=O)CCC2(CCCC2)C1 c1(C(=O)NC(CNC(c2nc(C)sc2)=O)C(C)C(C)C)cc(Cl)cc2c1CCC2 O=C1CNc2ncc(C(N3CC4CC3CN4C(c3ccc(F)cc3)=O)=O)cc2N1 C1(NC(CC2C(CNC(C3CC(C)(C)C3)=O)C2)=O)CCC2CCCC1O2 c1(C(=O)NC2CCN(C(c3c(SCC)cncc3)=O)C2)ccnc2ncsc12 N1(C(C(c2c(C)cc(F)cc2)O)=O)C2CCC1CN(C(c1cccc(=O)o1)=O)C2 C=CCC(C(=O)NC(C1CCCN1C(c1cnc(O)n1C)=O)(C)C)C(C)C C(CCCC(=O)N1CC(F)(F)CC1C(N1CC(=O)NCC1C(N)=O)=O)(OC)OC C1(OC)CC2(CCC(NC(=O)NC3CS(=O)(=O)CC3NC)CC2)C1 C=CC(C)CCNC(=O)C(C)N(C(C1(CCF)CCC1)=O)C1CC1 CC1CN(C(c2cc(F)ccc2Br)=O)CCN1C(=O)CC1CC=CC1 C1(CNC(C=CC=CCC)=O)C2CN(C(c3cnn(C)c3C)=O)CC12 n1(C(C)C)cc(-c2cn(CCCCNC(C3CCC3C#N)=O)nn2)cn1 c1(C(N2C(C(=O)Nc3c(OC)ccc(C)n3)CC(O)C2)=O)ccc(Br)c(F)c1F N1(C(CC2CCN(C(C(C=C)C)=O)C2)=O)CCC(C)C(O)C1 Cc1nc(N2CC(C(C)NC(=O)CCC3CCC(C)O3)C2)cc(C#N)n1 CC(C(=O)NCCN(C(=O)CCc1nnc(C2CC2)o1)CCOCCO)C(C)(C)C c1(COC(=N)O)cn(C2CC(NC(c3cc(Cl)on3)=O)C2)nn1 C1(NC(=O)C2=CCCC2)CN(C(c2ccn3ccnc3c2)=O)CC1C1CC1 O=C1CC(c2cn(CC(c3ccc(Cl)cc3O)N3CCOCC3)nn2)NC(=O)N1 C1(NC(Cc2c(C)noc2C)=O)CC(O)CN(C(c2ccnc(N(C)C)c2)=O)C1 C(CCCC(=O)NCC1CC(O)CN1C(=O)CC1NC(=O)NC1=O)OCC C(CCC(c1ccccc1)NC(CCCC1CCCC1)=O)N(CC)CC Nc1cc(CC(=O)NCC2CCC2NC(=O)COC2CC2)c(Br)cc1[N+](=O)[O-] N1(C(c2cc(C)ncn2)=O)CC(C2CCCN(C(=O)CCC3CCC(=O)N3)C2)C1 N1(C(CC(=O)N(C)C)=O)CCCN(C(c2cccc3c2CCO3)=O)C(CO)C1 CC(C)CC(F)C(=O)N(C1CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)CC1)C C1(C(N2CCN(C(c3cnc(S)[nH]3)=O)CC2CF)=O)CCc2cncn2C1 c1(-c2cn(CCN(C(c3cc(CC)sc3)=O)C)nn2)c(C)nsc1N c1(C(N2CCC3(C(C(=O)Nc4c(Cl)ccnc4Br)C3)C2)=O)cc(Br)c(O)cc1O c1(OC)cnc(C(=O)NCC2CCN2C(=O)CSc2ccccc2O)c(F)c1 C1(NC(C(C)SCC)=O)CC2(C1)CC2NC(c1coc(C(F)F)n1)=O C1(C(=O)NC(CN(C(c2nc(CC)oc2)=O)CC)C)CC(O)CN1C C1(O)(CNC(=O)COC2COC2)CN(C(C2CC(O)C2)=O)C1 c1(CC)nccnc1C(=O)NCC(O)CCNC(=O)C(C(C)C)n1cnnc1 C1(C(C)(C)C)C(NC(=O)C(N)=O)CCN1C(C1(CN(C)C)CCCO1)=O N1(C(c2ncc(C)c(Br)c2)=O)CCOC2(CCCN(C(=O)CCCCBr)C2)C1 C1(CC)CN(C(=O)CCOCC(F)(F)C(F)F)CCC1N(CC)CC c1(OCC)ccccc1C(=O)NCc1cn[nH]c1.C12(CC1)C(=O)N2 C1(CC)CN(C(=O)C(F)(F)CO)CCC1CNC(C1CC1C1CCCO1)=O C1(CNC(CSC(C)C)=O)CN(C(=O)CCCCN2CCCC2)CCCO1 C(=O)(C1CCCc2ncc(C)n21)N1CCC2(CN(C(c3c(C)nco3)=O)C2)C1 N1(S(CC(C)C)(=O)=O)CC2CC1CN2Cc1c(Cl)cncc1Cl C(=O)(C1=CCS(=O)(=O)C1)NC1(C2CN(C(c3cc(C)ns3)=O)C2)CC1 C1(C)(C(=O)NC2CC(CNC(C3CCN(C)CC3)=O)CC2O)CCCCC1(F)F N1(C(C(c2ccc(C)o2)C)=O)CCOCC(CNC(c2ncoc2C)=O)C1 N1(C(C2(OC)CCCC2)=O)CCC2(CC1)CN(C(C1CC1C#N)=O)C2C(C)C CC1(C)CCCC(C(=O)NCC#CCNC(=O)CCNC(c2ccsc2)=O)C1 C1(CNC(C(C)NC(N)=O)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 C1(NC(C(c2ccc(OC)cc2)O)=O)CN(C(c2cnccn2)=O)CC2(CC2)C1 C1(NC(CC2CCN(C(CCCCCC)=O)C2)=O)C2CCC(C2)C1(C)C c1(C(=O)OC)c[nH]c(C(=O)C(c2cc(OC)no2)=O)c1.C1CC(O)(CN)C1.CN Cc1c(CCN2CCCC(CCNC(C3CCC(=O)N3)=O)C2)cnn1C c1(CC(=O)NC2C(NC(c3cc(C)cc(F)c3N)=O)C2)cccc2ncccc12 N1(C(C=CC2N(C)CCC2)=O)CC2CC1CN2C(c1cc2[nH]ccc2s1)=O c1(C(N(CC(CNC(C2CCCC(OC)C2)=O)C)C)=O)cnc2[nH]cnc2c1 C1(C(N2CC(OCCCCC)C2)=O)CC(F)(CNC(=O)OC(C)(C)C)C1 C12(CNC(C(C(C)C)F)=O)COCCN1C(=O)CN(C(=O)Cc1cnc[nH]1)C2 C1(CC)CCN(C(C2(C)CN(C(C3CCC3(F)F)=O)C2)=O)C1 c1(C(C)NC(C2CCCN2C(=O)C(O)CN(C)C)=O)cn(C)nn1 C1(=CC(=O)NC(C)CNC(c2cn(CCC(C)C)nn2)=O)CCN(C)CC1 C(=O)(C(C)(O)C(C)(O)C(=O)N1CC2C=CC2C1)OC C1(NC(C2(C#N)CC2)=O)CC2(C1)CC(NC(c1n[nH]cc1C1CCC1)=O)C2 C1(NC(c2n(C)c(S)nn2)=O)CCC2(CCN(C(C3CC3(C)C(F)F)=O)C2)C1 Cc1cc([N+](=O)[O-])cc(C(=O)N(C2CCN(C(=O)C(O)C(C)C)C2)C)n1 c1(C(=O)NCC2C(NC(c3ccc(C)c(C)n3)=O)CCCC2)cc(N)c(Cl)c(O)c1 N1(CC(N2CCN(C(C(CC)(C)C#N)=O)CC2)=O)CC(=O)Nc2ccccc21 CC1(C)CN(C(C23CSCC2C3)=O)CC1NC(c1cc(N)ccn1)=O Cc1c[nH]c(=NCCCC2CCN(C(=O)CC3C(=O)N(C)N=C3C)C2)nc1O CC1CCC(C)(C)CC1(c1nnnn1C)NCC1CCN(CC(F)F)CC1 c1(C(=O)NCCC2CCN(C(C3N(C)C(=O)CC3)=O)C2)nc2c(s1)COCC2 N1(C(C2OCC(C)C2)=O)CCC2(CCN(C(c3cnsc3)=O)CC2)C1 C(=O)(CC(C(C)C)NC(=O)CCCC(C)=O)NC(C#C)CNC(N)=O c1(C2C(C(=O)NCC(CCNC(CCCN(C(C)C)C)=O)O)C2)ccccc1Cl C=C1CC2(C1)CC(C(N1CCC1CNC(c1c(C)nn(C)c1SC)=O)=O)C2 C1(OC)CC2(C1)CC2C(N1CC2CC1(Cc1cn(CC(O)CO)nn1)C2)=O C1(C(N2CCC(NC(=O)Cn3cnnn3)(CF)C2)=O)Cc2cc(F)ccc2O1 C(CN=c1cc(C)nc(CC)[nH]1)N(C(C1(CC#C)CCCCC1)=O)C N1(C(CCCOCC=C)=O)CC(CNC(C2(CC3CC3)CCC2)=O)C2(CC2)C1 c1(NC(CC(C)C)=O)ccccc1C(=O)NCC1CCCN1C(C1CC(O)C1)=O C(C)(CC(=O)N1CCC(NC(=O)C(O)c2ccco2)CC1)(C1CCC1)N(C)C S(=O)(=O)(c1cccc(Cl)c1)NCCC(=O)NC(CN(C(=O)CCOC)CC)C c1(NC2(COC)CCOCC2)[nH]c(=NCCSC(C)C)nc2c1ncn2C C1(CNC(CCOC(C)C)=O)CCC2(CCC2)CN1C(C1CCCCN1N=O)=O c1(C(N2CCCC(N(C(C(C=C)(C)O)=O)C)C2)=O)[nH]c2ncnc(N)c2c1C N1(C(C2(F)C(C)C2)=O)CCCCC(CNC(=O)Cc2ccc(F)cc2F)C1 C#Cc1ccc(C(N2CCCC2CNC(c2occc2C(C)C)=O)=O)c(OC)c1 Cc1cc(C(N2CCC(NC(C3CC3C(F)F)=O)C(O)C2)=O)c(C)n1CC1CC1 c1(C(=O)NC(C)CCN(C)C(C2CC(=C3CC3)C2)=O)cc2cc(Cl)cnc2[nH]1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CC(C)NC(C(c1cc(C)c(Cl)nc1)(F)F)=O)C C1(N(C(CN(C)CC)=O)C)CCCN(C(=O)C(c2ccc(F)c(F)c2)=O)CC1 Cc1ccc(C(C(C)C)NC(C2CCCN2C(=O)CCC#N)=O)cc1 N#CCCCC(=O)N1CCC(OCCNC(c2cnn(CCO)c2)=O)C1 C1(N(C(=O)Nc2cccc(C(=O)O)c2)CC2CCOC2)CC2CCC(C1)S2 N1(CC)C(=O)CCC1C(=O)NC1CC(NC(c2ccnn2C2CCOCC2)=O)C1 Cc1n[nH]c(=NC(=O)c2ccnn2CCC(F)(F)F)n1C N1(C(C2CC=CCO2)=O)CCC2C(CCCN2C(=O)CCOc2cccnc2)C1 C1(N(C(=O)Cc2cccs2)CC)CCCN(C(C2CC(C)(C)O2)=O)C1 Cc1cc(N)cc(C(N2CCN(C(=O)CCC3OCCO3)CC2C(C)C)=O)c1F C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CN(C(C2N(CCC)CCCC2)=O)CC1C c1(C(=O)NCC(C)(C)NC(=O)C(CO)c2ccccc2)cnc(C#N)s1 c1(C(=O)NC(CC(C)C)CNC(C2CN(C(N)=O)C2)=O)ccc2sncc2c1 C(CCCCC(=O)NCC1CN(C)CC(C)O1)n1cc(-c2c(C)nsc2)nn1 c1(C(N(C)CCOCCNC(=O)CC2CCCO2)=O)c[nH]nc1Cl C(CC(=O)NC1CCOC1C1CC1)(CC(C)C)NC(C1(CC#C)CCCO1)=O C1(O)(C(C(N2CCOC(CNC(C3CC4C=CC3C4)=O)C2)=O)F)CCCCCC1 C1(c2onc(CC(=O)Nc3ccccc3)n2)CC2(CCCC2)CO1 c1(CCC)cc(C(=O)NC2CC(NC(c3cc(C#N)c[nH]3)=O)CC2O)ccc1Cl C1(CNC(CN2CCN(C)C(=O)C2)=O)CCCC2CN(C(=O)C(=O)N(C)C)CC12 C(=O)(C(C)C(C)C(C)(C)C)NC(CNC(c1ccc(C(=O)OC)nc1)=O)C1CC1 Cc1ccc(NC(N2CC3C(C(N4CCC(F)(C(=O)N(C)C)C4)=O)C3C2)=O)cc1C C1(C(c2n(CCCSC)nnn2)(C)NCC2CSC2)CCS(=O)(=O)CC1 Cc1noc(CCC(=O)NCC=CC(=O)NCCc2ncc(C)o2)n1 C1(NC(c2c(CC)c[nH]c2)=O)(CO)CCCN(C(=O)CCCOC(C)=O)C1 C(CCCCC(=O)N(CCCNC(=O)C(C)c1ccco1)C(C)C)NC(=O)OC c1(C(N(C2CCC(NC(C3(C(C)(C)C)CCCC3)=O)C2)C)=O)ccc(C2CC2)o1 C1(C(=O)NC(C)(C)CN2CCOCC2)CCC(NC(c2ccsc2Cl)=O)C1 C(N=c1[nH]c(=NCCC#N)[nH]c2cc(OC)ccc12)c1ncc(CC)o1 N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CC(C1)CN(C(=O)C1=CCC1)C2 C1(OC)CN(C(=O)C(c2ccccc2)O)CC1CCN1CCCC1.C1(=O)CO1 c1(NCCn2c(C)cnn2)cc2c(cc1F)NCCC2 C1(C(=O)NCC(C(C)(C)C)NC(CCSCCC)=O)CC(C(C)(C)C)=NO1 C12(C(=O)NC)CCCC1CN(C(=O)C(C)(F)C(C)(C)F)C2 Cc1cc(Cl)c(C(=O)N(CCC(C)NC(=O)C(C)(C)N2CCCC2)C)cn1 CCCCCCC(CC)C(=O)NC(C)CC(C)NC(=O)C(C(C)C)SC C1(CC(=O)N(C(C)C(=O)N2CC(n3cccn3)C2)CC)CCCCC1 N1(C(C(C(C)(C)C)C2CC2)=O)CCC2CN(C(c3cc(Cl)cs3)=O)CC2C1 c1(C(=O)NCC2(NC(C(CO)N(C)C)=O)CCC2)cccc2nonc12 C1(CC(=O)NC(c2ccco2)COC)CCCC(NC(c2sccc2C#N)=O)C1 N1(C(C(C(CC)C)O)=O)CCC(C2(NC(=O)CCN(C)CC)CCC2)CC1 N1(Cc2cc(C)sc2C)CCC2(CCN(C(=O)CC(C)(C)c3ccccc3)C2)C1 c1(OCC)cc(C(=O)NC(C2CCCC2)CNC(C2CC2(F)Cl)=O)ccn1 C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCN(C(=O)CN2CC=CC2)CC1 c1(-c2ccc(OC)c(O)c2)n[nH]c(=NC(=O)NC(c2ccccc2Cl)C)s1 N1(C(C2CC(=O)NCC2)=O)CCC2(CC(C(=O)N3Cc4cccnc4C3)=NO2)C1 C12(C(N(CCN(C(C3(O)COC3)=O)CC)CC)=O)CCN(CC1)CC2 n1(CCN(C)C)nccc1C(=O)NCC1(O)CN(C(c2cc(Br)no2)=O)C1 C1(CNC(c2ccc(C3CC3)cc2)=O)CC(O)CN1C(c1ncc(Br)cn1)=O C(=O)(C(C)(C)C1=CCSCC1)NCCN(C(=O)C(C(C)C)NC(C)=O)CCC c1(C(=O)NCC(CCNC(CC=C)=O)O)cnc2c(c1)NCC2 C(N=c1[nH]c2c(c(=NC(C)c3c[nH]ccc3=O)[nH]1)CCC2)c1nc(C)[nH]n1 Cc1cccnc1-c1cn(Cc2ncoc2CNC(C2CC2(F)Cl)=O)nn1 C12(CNC(=O)C=C3CCC3)CCC(CC1)N(C(=O)C(F)C1CCCC1)C2 c1(OC)ccc(F)c(CC(N2CC(CNC(=O)CCN(CC(F)(F)F)C)C2)=O)c1 C(=O)(C1=CC2C=CC(C1)C2)NCC(COC)(C)NC(=O)CC(C)(C)CCOC Cc1ccc(Cl)c(C(N2CC(=C(F)CNC(C3(C)CC=CCC3)=O)C2)=O)c1 C1(O)(CNC(C2C(C(=O)OC)C2)=O)CCCN(C(=O)CCOCC(F)F)C1 c1(C(=O)NCCC2CCN(C(CC=C=C)=O)C2)nc2c(Br)cncc2[nH]1 N1(C(Cn2c(CCC)ncc2)=O)CC2C(CNC(c3conc3C3CC3)=O)C2C1 C(=O)(CC(C)(O)C(F)(F)F)N1CC2C(CNS(C)(=O)=O)C2C1 O(N(C(=O)C1CC(Nc2ccc(C(C)C)cn2)C1(C)C)C(C)C)CC N1(C(c2cc(Br)nn2C)C(=O)NC)c2ccccc2CC1Cc1ccccc1 Cc1oc([N+](=O)[O-])cc1C(=O)NCCCOCCNC(c1ccc(N)cc1Cl)=O Cc1nn(CC(C)C)c(Cl)c1C(=O)NC(C)CCCNC(=O)COC1CCC1 C12(C(N(CCOCCN(C)C(c3cccc(N)n3)=O)C)=O)CCN(C1)S(=O)(=O)C2 Cc1ccc2c(C(=O)NC(C)CNC(=O)CCC3CC3C)ccnc2c1 c1(N2CCN(CC3CC(C)(C)OC3(C)C)CC2)nc2c(F)cc(Cl)cc2s1 N1(C(C23CC(C)C2C3)=O)CC(NC(=O)CN(C2CCCC2)C)CC(C)C1 c1(CNc2c(F)ccc(Br)n2)cc2cc(Br)ccc2s1 N1(C(C(C)(Cl)Cl)=O)CC(CNC(c2sccc2-n2cnnn2)=O)C(O)C1 CCCCC(C)CC(=O)N1CCN(C(=O)CCc2cncc(C)c2)C(COC)C1 CC(C)CC(=O)NC(C1CN(C(=O)CCN2CCC2)C1)C N1(C(C2C(C)(C)CO2)=O)CC2CCC1CN2C(=O)CCC(=O)N1CCOCC1 c1(CC)cc(C(=O)NC2(CCNC(=O)C(C)(C)c3cnn(C)c3)CCC2)ncn1 C(=O)(CC(C)(C)C(=O)N1CC(C(C(=O)NCc2cnccc2Cl)OC)C1)OC c1(OC)ccc(S(=O)(=O)NC(C)(C)CCN2CCCC2)c(F)n1 C1(NC(c2c(C)nc(C)s2)=O)CCCCCC1C(=O)N(C1CC(O)C1OC)CCOC C=CCCC(F)(F)C(=O)N1CC(COC)(NC(=O)Cc2ccn(C(C)C)n2)C1 c1(C(N2CC3CC(NC(c4nc(Cl)cs4)=O)C3C2)=O)cccc2ncoc12 c1(CC(N2C(CCCNC(c3cc(C)ncc3)=O)CCC2)=O)ccc(O)c(Cl)c1 c1(C(=O)NC23CCC(CNC(CCCC)=O)(OC2)C3)csc(S(N)(=O)=O)c1 N1(C(c2c(OC)scc2)=O)CC(NC(=O)Cc2c(F)cccc2Cl)C(C2CC2)C1 CC12CC(C(=O)NCC3CCC(NC(c4cc(O)ncn4)=O)C3)(C1)C1(CCC1)O2 c1(CC(=O)NCC(CNC(C(c2ccccc2)OC)=O)F)cc2ccccc2s1 Cc1ncc(CCC(N2CCOCC(NC(C3CCC(=O)O3)=O)C2)=O)c(O)n1 c1(C(C(=O)NCCC)N(C)Cc2nnc(C3CC3)o2)cccc2c1nnn2C C1(C(C(=O)OCC)C)CCN(C(C2CCN(CC(CC)CC)CC2)=O)CC1 c1(NCC(=O)N(CCCNC(=O)Cc2ccnn2C)CC)ccc(Cl)cc1 C1(NC(Cn2nnc(C)n2)=O)COC2(CCCN(C(c3cccnc3O)=O)C2)C1 N1(C(C(CC=C)(F)F)=O)CCC2(CC1)CN(C(=O)CCC(C)OCC)CC(C)O2 c1(C(=O)NC(C(C)NC(=O)CC2CCOC2=O)CO)cc(Cl)cn1C N1(C(C2COCCC2n2ccnc2)=O)CCN(CCN(CC(F)(F)F)CCO)CC1 c1(C(C)=O)ccc(Br)cc1NC(=O)C(C1CCN(C(c2ccc(F)nc2)=O)CC1)C C(=O)(CCCCSC)N1CC(C(N)=O)(CNC(c2ccc(CSC)o2)=O)C1 CC(CC(=O)N(CC(C)CO)C)C(C)(C)NC(c1cnccn1)=O c1(C(C)NC(C)C)cn(C)[nH]c1=NC(=O)C12CCC(C(F)(F)F)(CC1)C2 CC(C)CC(C)(O)C(=O)Nc1cccc(NC(C2CC(=O)N(O)C2)=O)c1 c1(C(=O)NCC(CNC(c2nccnc2C)=O)OC)ccc(C(C)C)c(C)c1 c1(NC)ccccc1C(=O)NC1CC(CCC(=O)N(CC(C)CC)C)C1 C1(NC(c2ccc(C)nn2)=O)CCC(C)N(C(C2CCC(C)(C)O2)=O)C1 C(C(C(C)C(C)C)NC(c1cc(O)nn1C)=O)NC(CC1(OC)CCCC1)=O C=C1CCC(C(=O)NC(C)(C)CN(C)C(c2ncccc2NCC)=O)CC1 C(=O)(C(CNC(c1cc2occc2[nH]1)=O)CCC)NC(C=C)CO c1(C(=O)NCC2(c3ccno3)CC2)coc(C2CCCN2c2ccncn2)n1 CS(=O)(=O)c1ccccc1CNC(=O)NC12CCCC1NCC2 c1(OC)cc(C)c(C(N2CCC(O)C(NC(=O)CC(C)NC(N)=O)C2)=O)c(F)c1 C(C(C)(C)CC(=O)N(C1CCCN(C(=O)C(C)c2ccsc2)C1)CCO)OC CCCC(C)CC(=O)N1CCN(C(c2cnncc2C(F)(F)F)=O)CC1C1CC1 Cc1nc2cnn(C)c2cc1C(N1CCC(N(C)C(c2cscn2)=O)C(C)C1)=O N1(C(CC(CC)CC)=O)CCN(C(c2cccc(SC)c2)=O)C2CCCCC12 C(N=c1[nH]c2c(c(=NCc3ncc(C)[nH]3)[nH]1)COC2)c1c(CCC)nns1 C1(CNC(C(C=C)(C)C)=O)CC2(CCC2)CN1C(C1CCC(=O)NC1)=O Cc1c(Cl)c(C(=O)NCC(C)(CC(C)C)NC(=O)C=CC(=O)N(C)C)nn1C N1(C(CC=CCNC(C2(C)CCC(=O)NC2)=O)=O)CC2CCC(O)C2C1 c1(C(=O)NCCC2(NC(Cc3ccc(C)o3)=O)CCC2)cnc2n1CC(C)CC2 c1(C(N2C3CN(C(CC(C(=O)OC)(C)C)=O)CC2C3)=O)cc(C)c2cc[nH]c2c1 C(=O)(C1CCCc2c[nH]nc21)N1C2CC(NC(c3cc(C)nn3C)=O)C(CC2)C1 C1(NC(=O)C=Cc2ccncn2)CC(O)CN(C(c2cscc2C(F)F)=O)C1 CCC(CCOC)C(=O)N1CC(O)CC(C(=O)Nc2cnn(C(C)C)c2C)C1 N1(C(C(CC)C)=O)CCN(C2CCC(NC(=O)Cc3c[nH]nc3O)CC2)CC1 N1(C(CCCCC)=O)CC2CCCC(C1)N2C(=O)CSCc1csc(=N)[nH]1 N1(C(C=NOC)=O)CC2CC(C)C(C1)N2C(C1CC1OC(C)(C)C)=O c1(CC)cccc(C(=O)N(CC(O)CNC(=O)C(F)n2cccn2)C)n1 CC1(CS(=O)(=O)NC(c2cccnc2)C(=O)O)CCCO1 C1(C(=O)NC(CC(=O)NC)C)CCN(C(c2cccc(CO)c2)=O)C12CCC2 C1(C(=O)NC23CC(NC(=O)C(F)F)(C2)C3)CCC2C1C2(F)F Cc1ccc(-c2csc(CNC(=O)C(c3ccccc3)C)n2)cc1 Cc1ncccc1CCC(N1CCCC(N(C(=O)CSc2cn[nH]c2)C)C1)=O c1(NCC(Cc2ccco2)CO)ccc(N(CC(F)(F)F)C(C)C)cc1 N1(C(C2C(=C)C2)=O)CCC2CCC(C1)N2C(=O)C=C1CCCCC1(C)C c1(CCC(=O)N(C2CCN(C(c3cnccc3Cl)=O)C2)CC)ccc(C)cc1C C1(N(C(C(C)S(N)(=O)=O)=O)C)CCN(C(c2cc(C3CC3)ccn2)=O)CC12CC2 C#CC1(C(=O)NCC2CCC(=O)N2)CCN(C(=O)CCCn2ccnn2)C1 c1(NC(C)=O)c(C(=O)N(CCCNC(=O)Cc2cnc(C)[nH]2)C)cccc1C c1(C(=O)NC2C(CC)CN(C(=O)C(C)C(C)O)CC2)cccc2c1CNC2=O C1(CN(C(COC(C2CC(=C)C2)=O)=O)Cc2ccccc2)CC(C)CO1 N(C1CCc2c(Br)ccc(Cl)c21)Cc1ccc(F)c(N2CCCC2)c1 N1(C(c2c(CC)occ2)=O)CCCC(NC(C2CCN(c3ccncc3)C2)=O)C1 c1(NC(c2c(OC)nccc2Br)=O)nc2nc(C)c(C)c(C)c2s1 c1(CC(CO)NC(C(N2CCCCC2)C)=O)ccnn1C C1(NC(C2CCC(C(=O)OC)O2)=O)CCN(C(C2CC3CCC2C3)=O)CC1(C)C c1(C(N2CCC(OC)(CNC(=O)CSC)CC2)=O)sc2[nH]cnc(=O)c2c1C N1(C(=O)C=Cc2cn3c(n2)CCCC3)CCc2nc[nH]c2C1c1ccncc1 C1(C(N(C2C(C)C2)C)=O)C(c2ccncc2)C1(C)C c1(CC)cc(C)ccc1NC(=O)C(F)C1CC(NC(c2c[nH]nc2C)=O)C1 N1(C(C(CCC)N(C)C)=O)CCCC(CCNC(c2c(C)n[nH]c2C)=O)CC1 N1(C(C=Cc2c(C)ncs2)=O)CC(CNC(=O)C=C2CCC2)CC12CCC2 CC1CN(C(=O)C(C)(C)C2CCCO2)CCN1C(=O)CSCC(N1CCOCC1)=O C(=O)(C(C)(C)CC(F)(F)F)N1C(CO)CC(NC(c2cc(C)n(C(C)C)n2)=O)C1 C1(N(C(C(C)=C2CC2)=O)C)CCC(NC(=O)Cc2cc(C)cs2)C1 CS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CCC(CNC=O)CC2)n1 c1(OC)cc(Br)ccc1CNC(c1cncc(NC2CN(C(C)=O)C2)c1)=O.OCC c1(OCCn2c(C(C)(C3CC3)NC3(CC)CC3)nnn2)ccncc1 C12CCC(CC1)CN(C)C2.C(C(O)C(=O)NC(C1(CCN(C)C)CC1)=O)SC C1(C)(OC)CC(NC(C2CCCCC2(C)NC(=O)CCc2nc[nH]n2)=O)C1(C)C c1(C(N(C2CCN(CC(=O)N(C)Cc3nccs3)C2)C)=O)nc(Cl)sc1Cl N1(C(CCCC)=O)CC(OC)C(NC(=O)CSCc2cccc(F)c2)C1 C1(NC(c2c(C)nsc2)=O)CC(C2CCN(C(=O)Cc3cccc(Cl)c3)C2)C1 n1(CCC=C)cc(C(=O)NCCC2(O)CN(C(c3cnc(C4CC4)o3)=O)C2)nn1 CCCC(CCC)CC(=O)N1CCC(NC(C2CN(C(=O)N(C)C)C2)=O)C1CC CC1CCCCN1CC(N1CC(NC(=O)C(N2CCCCC2=O)C)C1)=O C1(CNC(c2cn[nH]c2)=O)CCCCCN1C(=O)Cc1ccsc1Br Cc1cncc(NC(C2(CNC(C3(C)CCSCC3)=O)CC2)=O)c1 C(C)(C)(CC(F)C(=O)N(C1CCN(C)C1)C)NC(c1c(CC)cncc1)=O C1(CNC(=O)NC2CC(C#N)(COC)C2)CC2CCCCC2N1Cc1ccccc1 C12(NC(c3c(C)nc(N(C)C)s3)=O)CCCC1N(C(=O)NC1CC1)CCC2 C(=O)(C#CC1CCCO1)NC1CCN(C(c2ccnc(C)c2C)=O)CC1 C=CCC(C)(CNC(C1CC(O)CN1C(=O)CCOCCCOC)=O)CO C1(NC(C(Cc2ccc(C)cc2)C)=O)CCSC12CN(C(=O)C(C)CN(C)C)C2 CCCC(C(=O)NCC1CCC(CN(C)C(C23CC(F)C2C3)=O)CC1)OC c1(C(=O)NCCC(CNC(c2c(SCC)cccn2)=O)O)cnn2c1N(C)CC2 C(=O)(CC(C)(C)C(=O)c1ccc(F)cc1)N1CCN(S(CC)(=O)=O)CC1.C1CN1 C1(C)(CNC(=O)Nc2sc(C(=O)OC)c(C)n2)CCC(C)C1(C)C C(C(=O)NCCCF)(C(C)CC1CCOCC1)N1CCC(c2c(C)ncs2)CC1 CCCCCC(O)C(=O)N1CCCC(CN(C)C(c2c(C3CC3)cnn2C)=O)C1 CCC(CC)CC(=O)N(CCSC)C(C)C.C12CCN(CC1O)C2=O N1(C(CC(C)OC)=O)CCC2CC12C(=O)Nc1cccc(OCF)c1 C#CCCC(=O)NC(CNC(=O)C(C)(C)NC(=O)NC)Cc1ccccc1 c1(C(C)C)cc(C(=O)NCC2CC(NC(c3sc(C#N)cc3Cl)=O)C2)cc(O)n1 C(=O)(CCCCCC1CCCO1)NCC(C1CC1)NC(C1(C)C=CCCC1)=O N1(C(c2[nH]c(=N)sc2)=O)CCCC(NC(=O)C(O)Cc2cnc[nH]2)CC1 C1(CNC(C(C=C)(C)C)=O)CN(C(C2CCCCN2CC)=O)C2(CCC2)C1 c1(C(C(N2CCC(N(CC)CC)C2)=O)NC(C2CCC2)=O)ccc(F)cc1 C12(COCCCNC(CNC(C)=O)=O)CC(C1)C(C)(C)O2.C(CC=O)OCC C#CCC(C)C(=O)NC1CC1CNC(=O)CSCC(=O)Nc1ccncc1 C1(C(=O)NC(C2CCCCC2)C(=O)NCCC(C)CO)CCCN1C=O c1(C(=O)OC)cnc(Cl)cc1NC(c1cc(-c2c(OC)cccc2F)cs1)=O C1(NC(C(CC(=C)C)C)=O)CC2CC(C1)CN(C(=O)CC13CCCN1CCC3)C2 N#Cc1ccccc1N1CCCC(C(=O)NCC2CSCCO2)C1 Cc1cc(NC(C23COC(Cc4ncc(OC(C)C)cn4)(C2)C3)=O)oc1Br C1(=CC(=O)NCC2CCCC2NC(C2CCC(=O)N2)=O)CCOc2ccccc21 C1(NC(c2nc(C(CCCC)(C)C)sc2)=O)CC12CCN(C(=O)CC(C)F)C2 c1(SCC(=O)NC2CCc3cnoc3C2)ccc(Cl)cc1[N+](=O)[O-] C1(CNC(C2CC(=O)N2)=O)CCCCN1C(c1conc1C(F)(F)F)=O c1(CN2CC3CN(C(=O)COc4ccccc4F)CC32)ccc2n[nH]cc2c1 N1(C(c2n(C)cnc2)=O)CC2(CCCN(C(C3CC3c3ccccc3Cl)=O)C2)C1 N1(C(c2n(C)nnc2)=O)CC2COCC2(C(=O)NC2CCCC(C(N)=O)C2)C1 N1(C(c2nc(C(C)=O)sc2)=O)CCC(NC(c2cc(C)n(C)n2)=O)C1(C)C c1(C(=O)NCCC2(CNC(C3CCC(CC)C3)=O)CC2)cnc(OC)c(C)n1 C1(NC(=O)COCCN(C)C)CCCN(C(=O)CN2CC3CC3C2)C1 c1(NC(C2C(CNC(C3CC3c3ccccc3)=O)C2)=O)cc(Cl)cc(Cl)n1 C(CC(C)C(=O)NC1CC1NC(=O)CSCc1nnc(C)n1C)=CC N1(C(CCc2n(C)cnn2)=O)C(CC(=O)NCCn2cnccc2=O)C2CCCC12 Cc1ccncc1CC(=O)NC(C)CC1CCN(C(c2cccc(Cl)c2)=O)CC1 CC(C)CCC(O)C(=O)NC(C1CCCN1C(=O)Cc1ccc(F)cc1F)(C)C c1(CNC(C2CCC(Cn3cc(C(C)OC)nn3)CC2)=O)ccc2c(c1)CCO2 C1(C2CCCN(C(c3nccn3C)=O)C2)(NC(CCc2n(C)c(S)nn2)=O)CC1 c1(C(N2CCC(CNC(C3(O)CC(C)(C)C3)=O)C2)=O)ncc(Cl)cc1Cl CC(CS(C)(=O)=O)C(=O)N1CCC(CCNC(c2cncc(C(N)=O)c2)=O)CC1 N1(C(C(C)N(C)C)=O)CCN(C(c2ccc3cc(F)ccc3n2)=O)CC12CCC2 c1(C(C(=O)NCCCF)N(CCCC)C)ccc(OCCOC)cc1 C12(C(N(CC)CC3CCCN3C(=O)CSC(C)C)=O)CCCC1C2(F)F C(=O)(C(C)C(O)CC)N1CC(CNC(c2ccc(C(=O)OCC)cc2)=O)OCC1 c1(CC(=O)NC2(C)CN(C(=O)CCC(F)(F)F)C2)cc(C(F)(F)F)cc(F)c1 C12(C(N3C(C(=O)NC)CC3)=O)CCCC1CCN2C(=O)C(n1cc(C)cn1)C N1(C(c2cc(C#N)[nH]c2)=O)CC2CCN(C(=O)CCc3cccc(F)c3F)CC12 N1(C(c2c(C)oc(Br)c2)=O)CCC(O)(CNC(=O)C=C2CCC(C)C2)CC1 C1(O)(C(=O)NC2C(NC(C(=O)NCC)=O)CCC2)CCCC(C)(C)C1 C1(C(=O)NC(C)CCCNC(=O)CCN2CCOCC2)NC(=O)OC1C C(C(C(=O)NC1CC=CC1)NC(C1CSC1)=O)OCC C1(NC(c2cc(OC)ncc2)=O)CCN(C(c2ncc(C)cc2OC)=O)CC1C C=CCCCCCC(=O)NN1CCCC1C(=O)NCC1C(C)(C)C1(F)F C1(C2=CCOCC2)(CNC(N2CCCC(C(=O)OCC)C2)=O)CC1 N1(C(C(Cc2ccc(Cl)cc2Cl)NC(C2C(C)C2)=O)=O)CC(O)C2(CCCC2)C1 c1(NC(CN2CC(C)C2)=O)csc2c1CCOC2 CC1(N(C(=O)C(=O)NC2CCCCC2)C)CCCC1C(=O)Cc1ccccc1 C(CC(C(=O)N1CCOCC1CCC)NC(C1C=CC=CC=C1)=O)=CC N1(C(c2c(C)con2)=O)CCN(C(c2cc(Br)cnc2N)=O)C2CC12 C(=O)(C(F)C(=O)N(C1C=CC(C(=O)OC)C1)CC)OCC.C1(C)C(=O)N1 c1(N2CCC(OC)(OC)C2)ccc(S(=O)(=O)NCc2ccn(C(F)F)n2)cc1Cl C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)C(NC(=O)CCc2cnccn2)C1C C1(C(N2C(C)(C(=O)OC)CC2)=O)CCCC(NC(=O)CC(C)c2ccco2)CC1 C#CC1(N(C2CCCC2)CCC#N)CCN(CCCc2cc(Br)ccc2F)CC1 C1(C(C)C)CN(C(C2CC2C)=O)CCN1C(c1cc(Cl)no1)=O N1(C(=O)CN2CCCCC2=O)CCC2CC(C(N3CCCCC(CO)C3)=O)C2C1 Cn1ncc2c1CN(C(c1csc(NC(c3ccc(O)cc3)=O)n1)=O)CC2 C1(C(=O)OCC2N(C(=O)OC(C)(C)C)CCCC2)C2CC(F)(F)CC12 C(=O)(C(C)(C)c1cnsc1)N(CC(O)CNC(=O)C1CC1)C N1(C(c2nc(C#C)sc2)=O)CCCC2(C1)CN(C(=O)CNC(=O)CC)CCO2 N1(C(C2CC(C#C)(O)C2)=O)CCC(CCNC(C2(COC)CC2)=O)C(F)(F)CC1 C1(NC(C2CCC(O)CC2)=O)CC12CCN(C(c1cc(Cl)ccc1O)=O)CC2 C1(NC(CCC#C)=O)CCCCCC1NC(=O)COc1ccc(F)cc1Br C1(C(F)F)(CNC(c2ccccn2)=O)CCN(C(=O)C(c2ccccc2)O)C1 c1(C(=O)OC)cc(NC(=O)C(=O)NC2CC(CS(C)(=O)=O)C2)ccc1F C(N=c1nc2c(ncn2C)c(NCC2CCSC(C)C2)[nH]1)c1cc(C)cc(C)n1 CN1CCOC(CNC(C2OCCC2NC(c2cnn[nH]2)=O)=O)C1 CCCCCCCC(=O)NCc1cc[nH]c1C(=O)NCc1cc(C)ncn1 CCC(C(=O)NC(C(=O)N1CCC1C(C)(C)O)c1ccco1)C(C)C CCCCC(CCC)NC(C1(NC(=O)CN(C)C(=O)OC)CCN(C)C1)=O C(=O)(C(C)(C)CCCF)N1CC(C(NOC)=O)C(CCO)C1.C(C(F)F)N C(CC(C(C)(C)C)NC(=O)Cc1ccc(Cl)cc1)N(C)C(C1CCNC1=O)=O c1(C(=O)NCC2CCN(C(C(C(C)C)OCC(C)C)=O)C2)sc([N+](=O)[O-])cc1Cl CC(C)(C)CC(CNC(=O)CCNC(=O)NC1CC1)CO N1(C(C(CC)O)=O)CC2CCOC2(CNC(c2c(C(F)(F)F)cccc2F)=O)C1 c12cc-1ccc2F.C(C(=O)N(CCOC)CC)=CCC C1(NC(c2n(CCOCC)nnn2)C(C)C)CCN(c2cnn(C)c2)C1=O C1(NC(Cc2nc(NC(C)=O)sc2)=O)CN(C(C2CCCN2C)=O)CC12CCC2 CC1(C)COCC1CNC(=O)Cn1cc(CCc2ccc(C(F)(F)F)cc2)nn1 C(C)(C1=NOC2COCC12)N.c1(C2CNC(=O)N2CCC)ccc(Cl)cc1.SC C(=O)(C(CC)(CC)CC)N1CC(CCC)C(C(=O)NC2CCOC2CC)C1 n1(CCC)ncc(C(=O)N(CCNC(=O)C(=O)NC2CC2)CC)c1Cl C1(CC(=O)NC(CCCCC)C)CCCCN(C(=O)CCN2CCCC2=O)C1 C1(C(N2CCN(CCOC)CC2)=O)CC2(C1)CN(Cc1cccc(Br)c1Br)C2 C#CCCCC(=O)NCC(C)(C1CCC1)NC(=O)CCc1conc1C C1(NC(C2CCC(O)CC2)=O)CC2CC(C1)N(C(c1ccc3sncc3c1)=O)C2 c1(C(N2CCC(NC(C(C(C)C)CO)=O)(CO)CC2)=O)cccc2cncn12 c1(C(=O)NCCCN(C(=O)Cc2cc(Br)cs2)C)ccc(Cl)cc1N C12(NC(C3CC(C)(C)C3)=O)CC(C1)N(C(=O)C(=O)NCc1ccc(F)cc1)C2 S(=O)(=O)(c1cnccc1N1CCC(O)CC1(C)C)NCc1cnc(OC)c(C)c1 C1(NC(C(C)OCC)=O)CCCN(C(c2ccc(C3CC3)o2)=O)C1CC C1(NC(C2(OC)CCSC2)=O)CN(C(C2SCC=C2C)=O)CC1(C)C n1(CC)cnc2c(NC(C)=O)[nH]c(=NCCSC(C)(C)COC)nc12 c1(C(N2CCC(CC=C)(NC(=O)C(C)NC(=O)C3CC3)C2)=O)cc(C)cnc1C CC(C1CCCc2ccccc21)NC(c1ccnc(Cl)n1)=O c1(C(CC(=O)Nc2c(C)ncn2C)O)nc2ccccc2[nH]1 N1(C(C2CN(C)C(=O)C2)=O)CC(NC(c2cnc(C3CC3)nc2)=O)C(C)(C)C1 C1(C(=O)NC(C)(C)CNC(N)=O)C2CCCC2CN1C(=O)C=CC1CCOC1 C(C)(C(=O)N1CCC(C(=O)NC2CC(OC)C2)O1)OCC N1(C(c2cc(CC)c(C)s2)=O)CC(C)N(C(c2nc(OC)cc(C)n2)=O)CC1C c1(CC(C)C)nnc(NC(=O)CC2CC(C)(C)C2)s1 c1(NS(C(C)C#N)(=O)=O)ccnc(N=c2nc[nH]cc2C#N)c1 C1(OC)(CNC(=O)CCC=C(C)C)CCN(C(=O)CCCF)C1 C1(NC(C2C(c3c(Cl)ccc(OC)c3)C2)=O)Cc2cccnc2NC1=O C(C1CCCN1C)=CC(=O)NC(C1CN(C(c2coc(C(F)F)c2)=O)CCO1)C Cc1cc(C(F)(F)F)nc(NC2(CNC(=O)C(C)C3CCCO3)CCC2)n1 c1(C(=O)OC)ccc(Br)c(C(=O)NCC(c2cccc(Cl)n2)(C)C)c1 C1(NC(c2occ(C)c2)=O)CC2(C1)CC(CNC(C1COCCN1C)=O)C2 Cc1oc(COc2ccc(C(n3cc(CN)nn3)C)cc2)cc1Br Cc1ccc(C(=O)NCC2CC(C)N(C(=O)CCC(N)=O)C2)c2c1CCC2 CC(F)(F)CCCC(=O)N1CC(c2ocnc2CNC(c2ccc(Cl)o2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(CCCC(C)=O)=O)C2)c(Cl)nc2sc(C)cn12 c1nnc2ccccn12.c1(N2CC(C)OC(C)C2)nccc(=NCC2CCCC2)[nH]1 CC1C(NC(C2CCCC3(CC3)C2)=O)C(C)CCN1C(=O)CCc1cn(C)nn1 C1(NC(c2nccc(OC)n2)=O)CCC12CN(C(=O)CN1CCN(C)C(=O)C1)C2 N1(C(CN(C)C(C2CCCC(F)C2)=O)=O)Cc2ccc(O)cc2C1 C(c1ccc(F)cc1)=C(C)C(=O)N(CC(C)NC(C1(F)CCOC1)=O)C CCC(C)C(O)CC(=O)C1CCCC(=O)N(CC(F)(F)CC)CC1 C1(C)(CNC(=NCCC)NCC(CC)Oc2ccc(Cl)cc2)CCC(F)(F)CC1 c1(OC)cc(F)c(C(=O)NC2CCC(NC(=O)CC34COCC(C3)C4)C2)c(F)c1 n1(C(C(=O)NCC2N(C(C3C(C)(C)OCC3)=O)CC2)(C)C)cc([N+](=O)[O-])cn1 c1(C(C#C)NC(C2CCCO2)=O)cc(-c2cc(OC)ccc2OC)ccc1F C1(NC(c2cncc(CC)c2)=O)CCN(C(c2cocn2)=O)CC12CCC2 O=C1NCC2(CN(C(=O)CC=CCNC(c3cc[n+]([O-])cc3)=O)C2)N1 c1(CNC(C2CC(O)CN2C(C23CCN(CC2)C3)=O)=O)ccccc1[N+](=O)[O-] c1(C(N2CC3(CCN3C(c3cc[nH]c3C3CC3)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 C1(C(=O)NCc2c(C)c[nH]n2)CCC(C2CC2)N1C(c1ccnc(O)c1)=O c1(C(=O)NC(CNC(CC(CC)C)=O)(C)CO)cc(C)cc2c1OCC2 Cc1ccnc2nc(C(=O)NC(C)C(C)NC(C3(C#N)CCSCC3)=O)nn12 C1(CNC(=O)C(O)C2CC2)CCN(C(C2(n3cnnn3)CC2)=O)C12CCC2 C1(NCc2c(=NC)cc[nH]c2)CNc2ccnn2C1 C(=O)(CCCCC(C)=O)NC1CN(C(C(CC)CC)=O)CC1(F)F N1(C(CC2(N(C)C)CCC2)=O)CCC2(C=C(C(=O)NC3CCOC3=O)C2)C1 n1(CCC(=O)NCC2CCCN(C(=O)CC3CC3)C2)ncc(=O)c2ccccc12 c1(C(=O)NC2CCC2C(=O)NC2CCCN2CC2CC2)cnc(O)c2ccccc12 C(=O)(C1CCCc2ccccc21)N1CC(NC(c2nn[nH]c2Cl)=O)CC2(C1)CC2 CC1C(NC(=O)Cn2ccccc2=O)CCCN1C(=O)C(O)CN(C)C c1(C(C)C)cccc(CC(=O)NC2(CO)CN(C(=O)COCC3CC3)C2)c1 c1(C(C)=O)ccc(C(=O)NC(C)C(C)NC(=O)CC2CC(N(C)C)C2)cc1F CC1CN(C(=O)C=Cc2ncc[nH]2)CCCN1C(C1CCCCN1N=O)=O c1(COC(C2CCCC(N(C)C)C2)=O)cccnc1C#N c1(CC(N2CCC(CNC(=O)Cc3ccnc(O)c3)C2)=O)nc2c([nH]1)CCCC2 Cc1cc(=NC(=O)C(c2ccc(Cl)cc2)OC(=O)CNc2ccccc2)[nH]o1 CC1C(Nc2ccc(C(=O)ON)cc2)CCN1C(=O)OC(C)(C)C c1(C(=O)NC2C(OC)CN(C(c3cc(C(N)=O)no3)=O)C2)nccn2nccc12 c12[nH]c3ccc(cc3c1C)NS(=O)(=O)C2.c1(NC(CCCC)=O)cn(C)nc1C c1(C(=O)NC2CN(C(CN(CCOC)C)=O)C(C)C2)ncc(OC)nc1OC c1(C(=O)NCC2N(C(C(C)N3CCC3)=O)CCCC2C)ccnc2nccnc12 c1(OC)c(C(N2CC3C(NC(=O)C(F)C4CC4)C3C2)=O)csc1Cl N1(C(C2CCCO2)=O)CCN(CCCNC(C2C(c3ccccc3)C2F)=O)CC1 c1(C(C(=O)NCC2C3CN(C(C(C)OC)=O)CC32)(C)C)ccc(Cl)cc1F C(CCC(=O)N(C(C)C(=O)N(C)CCc1ncccn1)C)OC(C)C C1(COCCOCCOC)CCN(C(c2ncccc2C(F)F)=O)CC1C Cc1cc(C)c(C(=O)NC2CC(NC(C3CCC(C(F)F)CC3)=O)C2)cn1 n1(CC(N2CCC(CC=C)(NC(=O)CC=C(C)C)C2)=O)nc(C2CC2)n(C)c1=O C1(C(N2C(CCC(=O)NC(c3ccncc3)CC)CCC2)=O)CCCN1C=O C1(NC(CC(C)(C)OC)=O)C(C)(C)C(NC(=O)C(CCO)N(C)C)C1(C)C CN(C)S(=O)(=O)N(C)CC(=O)NCC1CCCCN1C(=O)C(F)Cc1ccccc1 Cc1ccc2c(c1)CC(C(=O)NCC1(NC(=O)C#CC3CCCC3)CCC1)S2 C(=O)(CCS(=O)(=O)CC(C)C)NCC(CCCC)NC(C1CC1(C)C(C)C)=O CCC(C)C(O)C(=O)NC1CC2CC1N(C(=O)Cc1ccc(F)c(C)c1)C2 C1(CC)C(NC(=O)C(C)CC(N)=O)CCCN1C(=O)CC1CC(C)(C)CO1 C(CCCOC)(C(=O)N1CCOCC(O)C1)NC(C(C)OCC=C)=O C1(C(=O)OC2CN(CCNS(C)(=O)=O)C2)CCN(C(c2cccnc2)=O)CC1 c1(C(=O)NCC(C2CCOC2)NC(CSCCCC)=O)cncc2nnn(C)c12 c1(C(=O)NC2(C)CC(NC(C3CCC(C)(CC)O3)=O)C2)cc([N+](=O)[O-])cn1C c1(C(=O)NC2CC3(C2)CC(NC(=O)C(O)C2CCC2)C3)ccc2ncncc2c1 C1(C(=O)NCC2C(CNC(c3ccc(C(C)=O)cn3)=O)C2)CC(=O)CC(=O)N1 N1(c2nc(C)nc3c2cc[nH]3)CCC2(CCCN(C(C34CCCCC3C4)=O)C2)CC1 N1(C(C2=CC(O)C(NC(C3(C)CCSCC3)=O)C2)=O)CCC(O)(C2CC2)CC1 C=C(C)C(CC(=O)NCC(C)NC(=O)COc1ccccc1C#N)OCC CC1(NC(c2ccccc2NC(N)=O)=O)CCN(Cc2cccc(F)n2)C1 c1(C(N2CC(C(C)NC(=O)CC3CC=CCC3)OCC2)=O)ccc2ncsc2c1 C(C(=O)NC(C)(C)CCCO)(C(C)O)NC(C1CC(CCC)C1)=O c1(C(=O)NC2CC(C)N(C(c3cnsn3)=O)C2)cc(=O)cc(Cl)[nH]1 CC(N=c1[nH]c2c(c(=NCCN(c3cccnc3)C)[nH]1)COC2)C1CCCCC1 C1(CNC(c2ccc(OC)cc2Cl)=O)CCC2(CCOCC2)CN1 C1(c2noc(-c3cc(C#N)c[nH]3)n2)CCN(C2CC2)CC1.C1(C(C)C)CC1C1CC1 c1(CCC(=O)N(CCCNC(CC=C)=O)C(C)C)cccc(C(=O)OC)c1 C1(C(=O)NC2CCCC(C(=O)NC(CCO)C3CC3)C2)(CF)CCOCC1 N1(C(CC2C(C)CCC2)=O)CC2CCCN(C(C34CCOC(C)(C3)C4)=O)C2C1 c1(COCC)nc(C)c(C(=O)NCC2CN(C(=O)C(C)Sc3ccccc3)C2)s1 C12(CC=O)CC3CC(CC(C3)C1)C2.C1(C(N(CC(CC)N)C)=O)CC=C(C)CC1 CC(C)CC(O)C(=O)NCC1CC(CNC(=O)Cc2cccc(C(C)C)c2)C1 C1(C(=O)NC2CCC(C)CC2)CCN(C(C2C3CCCC23)=O)CCC1CO C1(C(=O)NC(C)(CO)C2CC2)C2CCN(C(C3CN(C)C3)=O)CC12 N1(C(CC=CC)=O)CCC(CNC(C2CC2c2ccc(C(C)C)cc2)=O)CC1C c1(N(C)C(=O)NCC2OCCC2F)ccccc1F c1(CN2C(CC(N3CCC(C(=O)OC)CC3)=O)COCC2)ccc(Br)c(OC)n1 c1(C(N2CCN(C(C(CCCCC)O)=O)C(CF)C2)=O)ccc([N+](=O)[O-])c(C)c1 C(=O)(C1=NNC(C(F)(F)F)C1)NCC(CNC(C1(OC)CCSCC1)=O)OC c1(C(=O)NC23CC(CNC(c4ccoc4)=O)(C2)C3)cc2c(F)cc(F)cc2o1 n1(CC)nc(C(=O)NC2CC2NC(=O)COCC2CCC2)cc1C(F)(F)F C1(CC(=O)NC(CC)CNC(=O)CCC2CC2(C)C)COC(C)(C)C1 C(=O)(CCC(C)(C)NC(=O)CC1COC(=O)C1)NCC(C)CC1CCCC1 C#CC1(C(=O)N(C)Cc2ccc(F)cc2)CCN(C(=O)C(C)Cn2cccn2)C1 c12ccc(c(F)c1)s2.CC1(NC(=O)CC2CC2)CC(C(=O)Sc2ccccc2)C1 N1(C(C2C(C3C(C)C3)C2)=O)CC2CC1CN(C(=O)CN(C)C(c1cccs1)=O)C2 C1(C(C)C)COCCN(C(c2ccc(C(N)=O)o2)=O)C1.C12CN(CCO1)C2 N1(NC(=O)CCc2cn(CCCn3cccn3)nn2)CCCS(=O)(=O)CC1 N1(C(c2cc(CC)on2)=O)CC(C)C(NC(c2cnn(CCO)c2N)=O)C(C)C1 CN1C(=O)C(c2nnc(-c3ccncn3)o2)Cc2ccccc21 c1(CC)nc(COc2ccccc2)n[nH]1.C1(=O)C(C)N1 C(=O)(CCS(=O)(=O)c1ccccc1)N1C(CNC(C(C(C)C)F)=O)CCCCC1 CC(C)CC(CN(C)C)N=c1[nH]c(=NC(C)c2nc(=N)[nH][nH]2)[nH]c2cc[nH]c12 c1(C(=O)NC2CC3CN(C(COCC(=O)NC)=O)C2C3)ccc2nonc2c1 c1(NC(C2CC3(CN(C(c4c(C)nco4)=O)C3)OC2)=O)ccc2ncccc2c1 C12(C(=O)NCC3N(C(C4CCOC4)=O)CCC3)COCC1CS(=O)(=O)C2 CCCCC(C)CCC(=O)N1CC=CC1(C)C(N1CCCC1)=O C(C(C)C(F)C(=O)NOCC1(C)CCC1)NC(c1cccc(CC)c1)=O N1(C(CC2N(C(CC(C)C(F)F)=O)CC2)=O)CCC(F)(F)C(O)C1 N1(C(CC2=NNC(=O)C2)=O)CCC(C2CN(C(=O)CS(=O)(=O)C3CC3)C2)CC1 C1(CNC(C(C)=C(C)C)=O)CN(C(C2CCCCN2C(N)=O)=O)CC1C(F)(F)F N1(C(CCC2N(C)CCC2)=O)CC(O)CC1C(N1CCC(C)(C(=O)OCC)C1)=O C(C(=O)NOCC(=O)N(CC(C)(O)C1CC1)C)OCCCCC c1(C(=O)OCC)cc(C(=O)NC2CN(Cc3ccc(Br)[nH]3)CC2F)n(C)c1 c1(N2CCCCC(CNC(C(CCC)C)=O)C2)ncnc2cccc(C)c12 n1(C2CCN(C(C3C(c4ccc(C)c(Br)c4)C3)=O)CC2)c(=O)oc2ccccc12 Cc1noc(C)c1CC(C)NCC(CCBr)C(=O)O.C1CCOC1=O C1(NC(C(C)OCCC(C)C)=O)CC2CCC1CN2C(=O)C(C)CC(F)(F)F N1(C(=O)NC(=O)OC(C)C)CCCC(Nc2ccccc2OCC#N)C1 c1(NC(C(CNC(CC2C(C)(C)CCO2)=O)CC2CC2)=O)cccc2c1CCC2 CN(C)S(=O)(=O)N(C)CC(=O)NC1CC(C)(NC(=O)CC2(O)COC(C)(C)C2)C1 C1(CCOC)CN(C(=O)C=C=C(C)C)CCN1C(=O)C(C1CCOCC1)F Brc1ccc2[nH]nc(COCC3(CCCCCC)CCCCCCC3)c2c1.OC c1(C(C)C(N2CC3CC2C3NC(=O)CCc2cnccn2)=O)ccc(Cl)c(Cl)c1 C1(CNC(C2C(C)OCCC2)=O)CN(C(=O)CC(Cl)Cl)CC12CCC2 c1(N2CCC(C(C)NC(=O)C=CSc3ccccc3)C2)cncc(C#N)n1 C=CCC(CNC(=O)CCCN(C)C)C(=O)N1CC=CC1(C)COC N1(C(CC2(OC)CC2)=O)CCCC(NC(C2(c3cc[nH]n3)CCC2)=O)CC1 c1(C(N2CCC(CC)C2CNC(C2CCCCC2O)=O)=O)cccc(F)c1C c1(C(=O)NC2(CNC(c3ccn(C)c3)=O)CCCC2)cn2ccsc2n1 C1(NC(CCC(=O)NC)=O)COCCN(C(C2CC(C)=NO2)=O)C1 C1(C(=O)NCCN(C(C2(C(=O)OC(C)(C)C)CCC2)=O)CC)CC2COCC2C1 c1(CC(=O)NC2CC3(C(NC(c4c(N)nccn4)=O)C3)C2)cc(F)cc(F)c1 c1(C(N2C(C3(NC(C(CC#C)(C)C)=O)CC3)CCCC2)=O)cc(F)c(C)cc1F CC(CC(C)(F)F)C(=O)NCC1(C)CCN(C(=O)Cc2csc(Cl)n2)CC1 C1(NC(C=C(CCN(C)C)Cl)=O)(CO)CCN(C(=O)C(O)CC2CCCC2)C1 C12(C(N(CCN(C(=O)C(F)C(C)(C)O)C)C)=O)CC(C)(C1)OC2(C)C CN1CCCCC1C(=O)NC1C=CC(C(=O)NCCN2CC3CC3C2)C1 c1(C(N(C2CCCOC2)C(CN(CCCC)CC)=O)=O)ccc(OC)nc1F c1(OC)nccnc1C(=O)NCC(C)CC(=O)NC1(c2cc[nH]n2)CC1 C1(CNC(c2c(C)nn(C(C)C)c2)=O)CCN(C(=O)CC2CC(F)C2)C1(C)C C(=O)(CCCCCO)NC1CCC(CNC(CCNC(COC)=O)=O)C1 c1(N(CCC(C)O)C)nccc(=NC(C)c2c(F)cccc2Br)[nH]1 N#Cc1ccc(C(N2CC3CC2CN3C(c2cc(Br)c(O)cc2F)=O)=O)c(Br)c1 c1(OCC)ccc(-c2nc(C(=O)Nc3nc(C)cs3)ccc2F)cc1[N+](=O)[O-] C12(NCC(C)(C)SC)CC3CC1CC3ON(CCOCC)N=NN=C2 N1(C(Cc2ccn(C)n2)=O)CCC(C2CCCN(C(=O)C(C)(C)C)CC2)CC1 c1(NC(=O)NCC2CCC(F)(CC#N)C2)cc(F)cc2cccnc12 CS(=O)(=O)C1CCCN(Cc2cc(=NCc3cc(F)ccc3F)[nH]cn2)C1 N1(C(c2cnc(C3CC3)s2)C(=O)NC2CC2)CCOc2cc([N+](=O)[O-])ccc2C1 C1(F)(C(N(C)C)=O)CCN(C(c2cccc(-c3cccc(CO)c3)c2)=O)C1 c1(C(N2CC(OC)(CNC(C3CCOC(C)C3)=O)C2)=O)cccc2c1COC2 CCC(CN(C)C)C(=O)NCC1CC1CC(=O)NC1CCNC(=O)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NC1C2CCN(C(C(c3cn(C)nc3)(C)C)=O)C21 N1(C(C(C(C)OC)NC(c2cnn(C3CC3)c2)=O)=O)CCCC(CCF)C1 CCCCC(CO)NC(=O)CCOCCNC(=O)C(C)C1CCCO1 N1(CC)CCOCC1C(=O)NCCC(O)C(=O)NCCn1cnccc1=O c1(C(N2CC(CNC(c3cc(C)sc3Br)=O)C2)=O)cnc2[nH]nnc2c1 c1(C(C)C)nc(=NC2CC(NC(c3ccc4sncc4c3)=O)C2(C)C)s[nH]1 C1(CCOC)(NC(=O)Cn2cnnn2)CCN(C(=O)CC2(CO)CC2)CC1 c1(CC)nccnc1C(=O)NCC(c1ccccc1)N(C(=O)C(F)CC)C N1(C(C2OCCN(C)C2)=O)CCC2CN(C(c3ccc(CC4CC4)s3)=O)CC2C1 Cc1cccc(N2CCC(OC(=O)CC3CC(C)OC3C)C2=O)c1 N1(CC(C)C)CCC(NC(C2CC(CSC3CCCCC3)C2)=O)C1 C1(CN=[N+]=[N-])CCCN(C(C2CCCCN2C(=O)C=CC2CCCC2)=O)C1 CN1CC(C(=O)NCCCCC2CN(C(c3cccn3C)=O)C2)NC1=O CON(CCCO)C(=O)C1(NC(C2CCC3CC23)=O)CC1(C)C c1(C(N2C(C)(C(=O)NC)CC2)=O)[nH]c(C)c(C(=O)N(C)CCn2ccnc2)c1C N1(C(c2c(CC)con2)=O)CCC(C)N(C(=O)CCc2conc2C)CC1 Cc1cncc(C(=O)NCC2CC(NC(=O)Cn3ncn(C)c3=O)C2(C)C)c1C N1(C(Cn2c(C)cc(C)n2)=O)CCCC12CCN(C(C1CCCN1C(C)C)=O)C2 C1(C(=O)OC)CC2COCC(C1)C2NC(=O)NC(=O)C(F)(F)c1csc(Br)n1 Cc1ccc(C)c(C(N2CC3(NC(C4CCCOC4)=O)CCC2C3)=O)c1O N1(C(C(c2cccnc2)OC)=O)CC(NC(c2ccoc2Br)=O)CC(O)C1 NC(=O)CCCC(=O)NC1CCCN(CCC2CC2C2CC2)C1 N1(C(C(CCCC=C)NC(=O)C(C)CC(=O)OC)=O)CCc2oc(C)nc2C1 Cn1cc(C(=O)NCC(CNC(c2cccn2C2CCCCC2)=O)CO)nn1 c1(C(=O)NC(C(=O)O)C2CC2)ccc2cccc([N+](=O)[O-])c2n1 N1(C(c2n(C=C)nnc2)=O)CCCC(C)(C)C1CNC(c1cn(C)nc1C)=O C(=O)(CCCCCC#N)NCC1(Cn2cc(C(CC)N(C)C)nn2)CCOCC1 C1(CC(=O)NCCCCSC)N(C(=O)CC2CCC(F)(F)C2)CCC1(C)C C(=O)(C(C)(C)C1=CCN(C(=O)CCC=CC(C)C)C1)Nc1c(COC)n(C)nc1 N1(C(c2cn(CC=C)nn2)=O)CCOC(C(=O)Nc2ccsc2CO)CC1 N1(C(C(CC(=O)OC)NC(C)=O)=O)CC(NC(=O)CN(C)C)C2CCCC12 C(=O)(CCC(=O)NC1CC(CNC(c2n[nH]cc2Cl)=O)C1)Nc1nnc(C)s1 c1(CC)cc(C(=O)NC2CC(CNC(C3CCCC(C)CC3)=O)C2)cc(Cl)c1 c1(C(=O)NCC(CC)NC(C2(C#N)CC3CC3C2)=O)c(F)ccc(C)c1F c1(C(N2CC3C(CNC(C4CC4C(F)(F)F)=O)(C3)C2)=O)c(F)cccc1F c1(C(=O)OCC)nnc(S(=O)(=O)N2CCN(C(=O)Nc3nc(C)c(C)[nH]3)CC2)s1 CCC(CC)C(C(=O)N1CC(C(=O)NC)Cc2ccsc21)N1CCOCC1 c1(C(ONC(CNC(C(CC)O)=O)=O)C)cccc(Br)c1 c1(OCC)ccc(C)cc1C(=O)N(CCC1CN(C(C23CC(C)(CO2)C3)=O)C1)C1CC1 C(C(C(C)(C)C)NC(=O)CC1NC(=O)NC1=O)NC(C(c1ccccc1)C)=O CCCCC(CC)CCCN(C)C(c1c(-c2ccccc2)nn2c1CCCC2)=O N1(C(C2CCCN(C(C)CC3CC3)C2)=O)CCCN(Cc2ccc(F)nc2F)CC1 c1(CC)ccc(C(N2CC(NC(c3cc(C)ccc3F)=O)CC(C)C2)=O)cc1Br c1(OC)cccc(C(N2CCC(C)(NC(=O)CC3(O)CCC3)C2)=O)c1 N1(C(C(C)(CO)OC)=O)CCOCC(C)(CNC(=O)C=Cc2ccnn2C)C1 c1(C(N2CC3C(CNC(C4C(C)C4C)=O)(C3)C2)=O)occ2c1CCC2 c1(C(N2CC(NC(=O)CCc3nc(O)n[nH]3)C2)=O)cc2c(o1)CCCNC2=O c1(C(=O)NCCOCCNC(CC(=O)NCC#C)=O)ccc(C(F)F)cc1 N1(C(C2CC(CC)(CC)C2)=O)CCC(CNC(c2cc(Cl)ccc2N)=O)CC1C c12cccc(c1)C1(CC1)N2.c1(C(C(C2CC2)SC)OC)nnnn1C1CCC1 c1(C2(C(=O)NCC(C)N(C(=O)COC3CC3)C)CCCC2)ccc([N+](=O)[O-])cc1 C1(C(N(CC(C)NC(c2cnc(S)[nH]2)=O)C)=O)CC2(C1)CC(O)C2 C1(CC(=O)N(C)CC2CCCN(C(=O)CCS(C)=O)C2)CC2CCC(C1)C2 C(CC(=O)NN1CCCC1C(=O)NCC1CCN(CCF)C1)OC(C)(C)C C(=O)(C(CC(C)C)NC(=O)CC(C)N(C)C(c1cc(F)n(C)n1)=O)NC c1(C(N2CCN(C(=O)CCc3ccon3)C(C3CC3)C2)=O)cccn2cncc12 C(=O)(CC(CC)CCC)NCC(CN(C(c1cnc(CCCC)s1)=O)C)C N(CCCN(CCNC=O)C(=O)COCC(C)C)C(C(CCCCC)CC)=O CCC(CC1CCCC1)C(=O)NCC1CC1NC(c1ccnc(OC(C)C)c1)=O c1(C(=O)NC2CN(C(c3[nH]cc(OC)c(=O)c3)=O)C2)cnc2n1CCCC2C CCC(CC)C(C(=O)NC(C1CCCN1C(c1sccc1C#N)=O)(C)C)OC N1(C(C(CN(C(CCCCC=CC)=O)C)C)=O)CCC2(CCN(C)C2)C1 C1(CC)CCCCC1C(N1CCC(CO)(CNC(=O)C(C)SC(F)(F)F)C1)=O C(CC(CNC(=O)CC1COCC1O)NC(c1ccoc1C(F)(F)F)=O)OC N1(C(C2N(c3c(Br)cnc(C)n3)CCC(O)C2)=O)CCC2COCC2C1 N1(C(C2C(C)CC2)=O)CCC2(CC1)CCN(C(c1cncc(N)c1)=O)C2 C1(F)(CNC(CCSCC(C)C)=O)CCCN(C(C2CC(C)(C)CO2)=O)C1 CCCCCCCC(=O)N(C)CC1CCCCN1C(C1CC(=O)CCO1)=O c1(C(=O)NCC(C(C)C)NC(=O)C2=CCCO2)ccc2c(c1)CC(C)(C)O2 C1(C(N(C)CCc2nn[nH]n2)=O)CCC(Cc2ccccc2)C1 N1(C(c2nc(Cl)cs2)=O)CCC2(CCCN(c3cc(C(F)(F)F)ncn3)C2)C1 C1(C(N2CCC(CCF)C2)=O)(CC)CCCN(C(=O)CSCCC(C)C)C1 C(=O)(C#CC1CCCOC1)N1C(CNC(C2(CCCC)CC2)=O)COCC1 N1(C(CCc2n(C)ccc2)=O)CC(O)CCC1C(=O)NCC1OC(=O)CC1(C)C CC(c1cccnc1)=CC(N1CCC(CF)(NC(=O)CNc2ccccn2)C1)=O C1(C(=O)NC(C2CN(C(=O)Cc3ccc(CO)cc3)C2)C)CCCC(C(N)=O)C1 CC1(C)CC1(C#N)CNC(C1(n2cc(Br)nn2)CC1)=O C1(C(N2CCC(F)(CNC(CP(C)(C)=O)=O)C2)=O)CCCCC12OCCO2 c1(CCC)cc(C(=O)NC(C2CCCN2C(C2C=CCCC2)=O)C)n(C)n1 O=C1NC(C(=O)NCC#CCNC(c2sccc2-n2cccc2)=O)CO1 CCC(CCO)C(C)NC(=O)NC1C2CCOC2C1(C)C O=C(C1=CCCCCC1)N1CC(C(=O)NCCc2ccon2)C2(CCC2)C1 N1(C(C2C(C)CCCC2)=O)CCC(C)C(CNC(C2CCC3CC3C2)=O)C1 c1(CN2C(C(N3C(C)(C(=O)OC)CCC3)=O)CC(O)C2)cccc(Br)c1O c1(C(N(CCNC(C2CC(C)(F)C2)=O)CC)=O)ccc(NC)c(F)c1 c1(OC)ccc(Br)c(C(=O)NC2CCC(NCc3cnc(Cl)cc3Br)C2)c1F c1(C(=O)[NH+](CC2(F)CC(NC(C(CN(CC)CC)F)=O)C2)[O-])cnc(C)cn1 O=C(CC1CCOc2ccccc21)NCCC1(CC(=O)O)CC1(F)F C1(CC)CCC(C(=O)NC(C)C=CC(=O)NCC2(C3CC3)CC2)O1 CN1C2CCCC1CN(C(C1CC3CC1C1CC31)C(=O)NC1CCCC1)CC2 CC1=CCN(C(C2(NC(=O)CC3CCCC3C)CC(F)(F)C2)=O)CC1 C1(C(N(C(C)CC(c2ccc(Cl)cc2)=O)C)=O)CCOC(C)(C)C1 c1(CC)cc(OC)ccc1CNC(=NCc1cccs1)NC(C)COC N1(C(=O)Cc2cnsc2)CC2=C(C1)CN(C(=O)C(c1ccc(Cl)cc1F)O)C2 N1(C(c2cn(CCC(C)C)nn2)=O)CCC(NC(c2sccc2F)=O)C12CC2 c1(C(=O)NCC23C(CN(C(CSCC)=O)C2)C3)cnc(Cl)cc1I c1(N(CC(S(=O)(=O)NC)C)C)ncccc1S(=O)(=O)NCc1csc(COC)n1 C1(CC)CCCN(C(C2CC(C)(C)CO2)=O)C1C(=O)NCCC(C)O N1(C(C(CC)O)=O)CCN(C(c2cccc(C(F)F)c2OCC)=O)CC1C1CC1 C(=O)(C1CCCc2c1ncn2C)N1CC(CNC(C(C)=C(C)C)=O)CC12CCC2 c1(CNC(C23CC(NC(C(C)OCCOC)=O)(C2)C3)=O)cnc(O)c(F)c1 O=C1NC2(CCN(Cc3cc(F)c(Cl)cc3F)CC2)c2ccc(O)cc21 c1(OC)ccc2[nH]c(=O)c(C(=O)NCCc3cc(C)sc3C)cc2c1 c1(CNC(c2ccc(F)c(Cl)c2F)=O)ncnc2c1OCCO2 C1(CN)CCC2(CCC2)C1NC(=O)CC1(CC(=O)Nc2ccc(Cl)cn2)CC1 C1(NC(CN(C)C(N)=O)=O)C=CCC(C(=O)N(CCCC(O)CO)C)C1 CC(CCCNC(=O)CCN(C)CCO)NC(=O)CC1CCSC1 N(C1CCOc2c(Cl)cc(Cl)cc21)C(C(=O)N1CCC1c1cccc(Br)c1)=O N1(C(C(CC)C(C)C)=O)CCC2(CC1)CC(NC(C1CC1(C)Br)=O)C2 C1(C#N)(C(=O)NC(C(C)NC(Cc2c(C)cnn2C)=O)C)CCOCC1 c1(CC)ccc(C(=O)NCC(CC)NC(c2nc(C)ncc2OC)=O)c(OC)c1 O=C(C(Cc1cccc(Cl)c1)CCCCCO)OCc1noc(-c2ccsc2)n1 Cc1cc([N+](=O)[O-])nn1C(C)C(=O)N(CC(O)C1(C)CC1)C N1(C(c2oc(C3CC3)nc2C)C#C)CCOCC(C(=O)NCC2CCC(CC)O2)C1 C(=O)(C(C)C(C)NC(=O)CCOC)N(CC=C)C c1(C(=O)NCC2C(C(=O)NC(CCC)C)OCC2)cc(CC)nn1C C1(OC)(CNC(=O)C(C)SC(C)C)CN(C(C2CCN2S(C)(=O)=O)=O)C1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(c2cccc(F)c2)(NC(C(N)=O)=O)C1 C1(NC(C(C)OC2CCOC2)=O)CC(NC(=O)C(C)Cc2ccncc2)CC1O c1(N(C(=O)OC(CC=C)=O)C)ccc(C2(F)COC2)cc1 c1(C(=O)NCCC2N(C(C(CCCC)O)=O)CCOC2)c(F)ccc(C)c1Cl N1(C(C(CC(=C)Cl)NC(C2CCC(C)CC2)=O)=O)CCC2(CCC(O)C2)C1 C1(c2cn(CCCC(N3CCSCC3C3CC3)=O)nn2)CC12CCCCCC2 N1(C(CC2(OC)CCC2)=O)CCOCC(CNC(C2CC(C(C)C)=NO2)=O)C1 Cc1nc(C)c(CNC(C2CCCC2CNC(=O)CC2CCOC2C)=O)[nH]1 c1(SC)ccc(Br)cc1C(=O)NCC1C=CCN1C(c1cccnc1)=O Cc1nc(O)ccc1C(=O)NC(C)(C)CN(C(=O)CC1C=NN(C)C1=O)C c1(N2CC(CCOC)OCC2)nc(=NC(C)CCO)[nH]c2c1ncn2C(C)C Cc1cc(C(=O)NC2(C3CCN(C(=O)C(CO)N(C)C)C3)CC2)c(Cl)cc1Cl C(N=C(NC(C)CC)NC1CCN(CC(F)(F)F)C1)c1nc(CC)oc1 CCC(C)CCCCC(=O)N1CCCC(Cc2cn(Cc3cnn[nH]3)nn2)C1 CCC(CCOC)C(=O)N1CCC(C(N2CCC(OC(C)=O)C2)=O)O1 c1(N(CC(=O)NCC=CCOc2cn(CCCF)nn2)C)ccc(Cl)cn1 C1(C(N(CCCOC(C)C)C)=O)CC(C)(C)CCN1C(=O)CC1CCOCC1 CC1CN(C(c2cccc(Cn3cc(COCCO)nn3)c2)=O)CC(C)(C)C1 C1(C(=O)NCC23CCCC2C3)CN(C(C2CC3(CC3)CO2)=O)C2(CCC2)C1 c1(C(=O)NCC2CCC(NC(C3(n4ccnn4)CC3)=O)C2)ncc(F)cc1F c1(C(C(=O)N(CC(=O)OC)C(C)C)N(C2CCCC2)CC=C)ncccc1Br c1(C(N2C3CC(CNC(c4c[nH]c(=O)cn4)=O)C(C3)C2)=O)n[nH]c2ccc(F)cc12 N1(C(COc2cccc(CC)c2)=O)CCN(C(c2ccnnc2C)=O)C(C)C1 c1(C(=O)NCC(C2CCCCC2)NC(=O)CCF)sccc1Cl N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(=O)CN2CCCCC2=O)C2CCCC12 Cc1nccn1CC(=O)NC(CNC(=O)CCc1nccn1C)C1CCC1 C(=O)(C(CN(C)C)NC(=O)CCc1ccsc1)NC(C1CCOCC1)C N#Cc1ccccc1C=CC(=O)NC1CC1CNC(=O)CCc1cnc(O)[nH]1 c1(C(=O)NC2CC(C)(NC(c3nc(CCC)oc3)=O)C2)ncc(Br)cc1N Cc1cc(C)n2nc(C(=O)OCC34CC=CCN3CCC4)nc2n1 c1(C(=O)NC2CCCN(C(c3cccc(Cl)n3)=O)C2)n[nH]c2cccnc12 c1(C(=O)NC2CC(CNC(=O)CC3CC3(Cl)Cl)C2)cccc2c1CCO2 c1(C(N2CCCC(NC(CC(C(C)C)O)=O)CC2)=O)cnc2ccnn2c1 C(=O)(CCCCCC(c1nnnn1C1CCC1)Nc1cccc(Cl)c1C)OCC N1(C(Cc2c(CC)noc2CC)=O)CC2CC(NC(=O)C(Cl)=CC3CC3)CC1C2 C#Cc1ccnc(SC)c1.C(=O)(C(CC1(C)CC1)c1ccccc1)N Cc1cc(CNC(=O)CNC(N)=O)oc1C(N1CCC(F)CC1)=O C12(C(N(CCNC(c3csc(COC)n3)=O)CC)=O)CCCC(C1)OC2 C1(CNC(C(CC)NC(C)=O)=O)CN(C(c2ccc(N)c(O)c2)=O)CCC1(C)C CCCC(C)(O)C(=O)N1CCC(C)(CNC(c2cc(F)ccc2C(C)C)=O)C1 C=Cc1cc(C(=O)N(C2CCCCN(C(=O)C3=CCCCC3C)C2)C)cc(F)c1 CC(C)CC(C(=O)C(=O)C(C)S)NC(N)=O.C1(CC(=O)NCC(C)N)CC2(CC2)C1 CC(C)C(O)CC(=O)NC(C)CC(=O)NC(c1ncccn1)(C)C C1(OC)C(C)OCCN1C(=O)CCCC1CCC1.c1(-n2cc(COC)nn2)cccc(Cl)n1 C12(CNC(=O)CSCC3CCCCO3)CCC(CC1)N2C(C1CC1F)=O CCC(C)(F)C(=O)N(CCCCCCNC(=O)C(O)c1ccsc1)C C1(CC(C)NC(CC(=C)C)=O)CC2CCC(C1)N2C(=O)CSc1ccc(C)cc1 Cc1[nH]c2cccnc2c1CNC1CCN(CCC(C)C)CC1 N1(C(c2ccc(C)s2)=O)C(C)CC2CN(C(=O)C(C)(O)CC(C)C)CC12 N1(C(C(C2CCCOC2)OC)=O)CC(F)(F)CC1Cn1cc(Cc2cccs2)nn1 C(=O)(CCCCCN(C(=O)CC1(OCC)CC1)C)N1C(CCC)CCC1 Cc1cc(CC(C)NC(=O)C(C)CNC(c2scnc2Cl)=O)n[nH]1 C1(NC(C2C(CN(C)C)C2)=O)COCCC1NC(c1ccc(F)cc1)=O N1(C(CCCCCSC)=O)C2CCC1CC(C(=O)N(C)Cc1cncc(F)c1)C2 c1(C(=O)Nc2ccc(-c3cccc(O)c3)cn2)c[nH]c2cc(Cl)ccc12 c1(OC)ccc2c(c1)CCC(C(=O)NC13CC(NC(C4CCCC4O)=O)(C1)C3)C2 c1(OC(c2[nH]nnc2COC)=O)ccc(C(=O)CSc2ccc(Br)cc2)cc1Cl C1(NC(C(C(CC)(C)C)=O)=O)CN(C(=O)CCn2cc(Cl)cn2)CC2(CCC2)C1 C=CC(C)C(=O)N(C(C)CC(=O)NCC(C)(C)COC)C C1(C)(C(=O)NCC(CNC(=O)C(c2cnccc2C)(C)C)OC)CC2CC2C1 N1(C(C2C(O)CCN(C(C3CC(=C)C3)=O)C2)=O)c2ccccc2CC1C(N)=O C(C(C)(C)C(=O)NCC=CCNC(c1ccnc(-n2cncn2)c1)=O)SC C(CC(C)(C)C(=O)N(CCCNC(c1cccc(-c2nc(O)n[nH]2)c1)=O)C)OC N1(C(C2C(CC)OCC2)=O)CC(=O)N2CCCCC2C1 c1(C2C(C(N(C3CCN(C(c4nn[nH]c4Cl)=O)C3)C)=O)C2)ccc(F)c(F)c1 N(C1C(=O)NCCCc2ccccc21)C(=O)CC1Cc2ccccc2O1 S1(=O)(=O)c2ccc(s2)CN(C)C(=O)C2CN1CCC2O.c1(C)noc(C)n1.CN C(=O)(N(C)OCC(=O)NC(Cc1ccccc1)C1CC1)C1C(C)(COC)C1 CC1CC(C(=O)NCC2(F)CC(NC(c3ccnc(C4CC4)c3)=O)C2)CC(C)(C)C1 N1(C(c2c(CC=C)cccc2)=O)CCC(F)CC1C(=O)NCCCP(C)(C)=O C1(C(N(C)CC2(O)CN(C(CNS(NC)(=O)=O)=O)C2)=O)CCCC1(F)F N1(C(c2c(F)ccc(C)n2)=O)CCC2(CCCC2NC(=O)CCc2ccoc2)C1 C12(CCO)CN(C1)C2=O.c1(C(C(=O)C=CC2CC2)=O)cnccn1.N c1(C(=O)NC(C)Cc2cc(Cl)ccc2Cl)ccc(-c2ccncc2)nc1O N1(C(c2n(CCC)ccc2)=O)CCCOC(CNC(=O)C(N)=O)C1 c1(C(=O)NCCCC(F)F)cccc2cc(F)ccc12 C(=O)(C(C)CC(C)C(C)=O)NC(COCC)C(=O)NCc1coc(C)c1 c1(C(N(CC(C)NC(=O)C(O)C(C)(C)C)C)=O)cccc2c1NCCC2 C1(NC(c2ccc(CC)[nH]2)=O)CCN(C(=O)CC2COCC(C)(C)O2)C1(C)C c1(CC)cc(Cl)c(NC(C2CCNC(C(=O)NC)C2)=O)cc1Cl C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(=O)CC2CNC(=O)C2)CC1(C)C N1(C(C)=O)C2CCC1CC(N(C(c1ccccc1S(C)=O)=O)C(C1CCCC1)=O)C2 C1(C(=O)Nc2cc(CC)cc(O)c2)CCN(C(=O)C(C(C)CC)NC(C)=O)O1 C(=O)(C(F)C(F)(F)F)N1C(C(CNC(C(C=C)C)=O)(C)C)CCC1 C(=O)(C(COC)CC(C)C)N1CCC(O)(CCNC(CC(C=C)(C)C)=O)C1 N1(C(=O)NCCOC(C)(C)C)CCC(F)(F)C(NCc2cnc(O)c(C#N)c2)C1 N(C1CCCc2ccoc21)C(C(CN(C)C)NC(c1ccc(C#C)cc1)=O)=O O=C(C1=CCCOCC1)NC1CC(NC(c2ccc3c[nH]nc3c2)=O)C12CCC2 c1(C(=O)NCC2C(CNC(c3cc(CCCCC)[nH]n3)=O)C2)nc(C)oc1CC N1(C(C2CCC(C)NC2)=O)CCCCc2c(O)cccc21 Cc1nnc2n1CCC(C(=O)NCC(C)NC(=O)CCN1CCCC1)C2 c1(C(=O)NC2CN(C(=O)Nc3ccc(C)cc3)CC2F)ccc([N+](=O)[O-])cc1F c1(NC(C)=O)c(C(N2CC(NC(c3cccc(Br)c3F)=O)C2)=O)cccc1C Cc1ccccc1C(C)CC(=O)NC(C)(C)C(C)NC(c1nn[nH]c1Cl)=O N1(C(COCCC=C)=O)CCOC2CCN(C(c3cccc(=O)o3)=O)CC12 c1(OC2CCN(C(c3cn(CC)nc3)C(=O)NCCC#N)C2)c(F)cccc1F Cc1cn2c(CC(N3C(CNC(C4(CO)COC4)=O)CC4COCC34)=O)csc2n1 C(=O)(C(C)(C)CNc1cc(C)sc1C)NC(C(CO)SC)C C(C1=CCCSC1)(c1nnnn1C)N(C)Cc1cccc(Oc2ccccc2)c1 CCC(CC)CCCC(=O)NCC1CCCN1C(C1(c2ccncc2F)CC1)=O C1(C#N)(C(=O)OC)CCN(C(C2N(C(=O)OC(C)(C)C)CC2(C)C)=O)CC1 c1(C(=O)NC(C)CCNC(=O)CCC#N)ccc(C2CCCCC2)cc1 C1(NC(C(CO)OC)=O)CC2(CCN(C(c3c(C)coc3C3CC3)=O)C2)C1 c1(C(N(C2CCN(C(C3CC34CC4)=O)C2)C)=O)nnn(C2CC2)c1C(F)F C1(C(N(CCC(=O)NC(c2cnn(C)c2)CO)CC)=O)CC=C(C)CC1 c1(C(=O)NC2CC(C)(CNC(c3ccsc3Cl)=O)C2)coc(C#N)c1 c1(C(=O)NC(C2N(C(CCC(=C)Cl)=O)CCCC2)C)ccc2c(c1)CC(=O)N2 CC1CCC(CNC(=O)Cc2ccon2)N(C(C2CN(C)C(=O)N2)=O)C1 c1(C(N2C(C)(CNC(CNC(C(CC)C)=O)=O)CCC2)=O)cnc2ncccn12 CC1CN(C(=O)CCc2csnn2)CC1CNC(c1cccc(C2CC2)c1)=O CC(CC(=O)NCC1(Nc2ccccc2)CC1)CC(F)(F)F c1(N2CCCC(N(C)C)C2)nc(=N)[nH]c(=NC2CC2c2ccsc2)[nH]1 c1(COC)cncc(C(=O)NC(C(=O)NCC2(C(C)(F)F)CC2)C2CC2)c1 C1(NC(C2N(C)CCCC2)=O)CN(C(=O)C(C)(C)O)Cc2ccnn2C1 C1(NC(C2C(c3c(C)c(Br)ccc3)C2)=O)CCC2(CC1)CNC(=O)C2 N1(C(c2ccoc2)=O)CCCC2(CCCN2C(c2cc(Cl)cc(Cl)c2)=O)C1 N1(C(CC2C(CC)C2)=O)CCC(NC(C2CCN(C(=O)OC)CC2)=O)C(C)(C)C1 C1(C(=O)NCCC2CC(C(N(CC(CC)O)C)=O)C2)CC(C2CC2)C1 c1(-c2cccc(OC)c2C)ccc2cc(C(N3CCC(C)C3)=O)cn2c1 C1(C(N2CC3C(CNC(c4c(COC)cco4)=O)(C3)C2)=O)CS(=O)(=O)CCO1 C1(NC(CSCC#C)=O)CN(C(=O)CCSc2ccccn2)C2CCCC12 c1(CC)ccc2ccccc2c1COC(=O)Cc1ccc(O)cn1 N1(Cc2c(C)cccn2)CCC2(CC2C(N2CCCC2CO)=O)C1 CCCC(O)(CCC)CC(=O)NC1(C)CCN(C(c2conc2COC)=O)C1 Cc1nc(O)ccc1C(N1CCCC(N(C)C(C2CC3(CCC3O)C2)=O)C1)=O C1(C(N2C(CCNC(c3c(C(C)(C)C)ocn3)=O)CCC2)=O)CC2(C1)CC2(F)F C1(NC(C2C3CCCC23)=O)CCN(C(c2ccsn2)=O)C12CCC2 c1(OC)c(NC(=O)C(C)NC(C2(C)CCC2)=O)cccc1F n1(CC)cnc2c(NCC3(Cl)CC3(F)F)[nH]c(=NCCCc3cccnc3)nc12 O(P(C)(=O)CNC(C1CC(C)CN1C(=O)CCC1CCOC1)=O)CC N1(C(C(C(C)C)(C)O)=O)CCC2(CC1)CC2CNC(=O)CC1CC(OC(C)(C)C)C1 N1(c2nccc(OC3CCN(N(C)C)CC3)n2)CCc2ncncc2C1.C(=O)O n1(CC)nncc1C(=O)N(C)CC1CCN(C(=O)C(C)Cn2cccn2)C1 C(=O)(CC(O)CC(C)(C)C)N1CC(COC)(NC(c2[nH]nc3ncccc23)=O)C1 C1(C(=O)Nc2c(CC)cccc2)CCN(C(=O)CCCCCNC(C)=O)C(C)C1 N1(C(C(COC)C)=O)CCN(C(=O)COc2ccc(F)cn2)C2COCC12 CCC(C)(C)C(O)C(=O)N1CCC(F)(n2cc(CC3CC4(COC)C3C4)nn2)CC1 CC1CN=C2NC=CC1=CC(Cl)=CC=C2N(C)C CC1CN(C(C2CN3CCN2CC3)=O)CC(C(=O)NCC=CC(C)(C)C)O1 N1(C(C2CC(OC)C2)=O)CCCCC1CN(C(=O)CCCOC)C C(CC(C)C(=O)NCc1ccc(C(N2CCC(n3ccnc3)C2)=O)s1)=CC c1(C(C)OC(C(CCC)CC2CCCC2)=O)cc(F)c(N(C)C)c(F)c1 C(CNC(C1CCN(C(=O)C(C)C)CC1)=O)(C(C)C(C)C)NC(CCOCC)=O c1(N(C(C(COC)NC(C2CC(CC3CC3)C2)=O)=O)C)ccc(O)cc1F C(=O)(CCCCCN(C(=O)C=CC1CCOCC1)C)NC(C=C)C(F)(F)F c1(C(N2C(CNC(C=CC(=O)OCCCC)=O)CCC2)=O)cccc(C#N)c1 S(=O)(=O)(c1cccc(Cl)c1F)N1CC(OC)C(NC(C2CCCC(C)C2)=O)CC1 N1(CC)CCC(NC(=O)CC2CCN(C(c3coc(C(F)F)c3)=O)CC2)C1=O C1(NC(CN2CC(CC)C2)=O)CCCC1CNC(C1CCSC1)=O Cc1c(CC(=O)NC(C)C(C)NC(c2ncn(C)n2)=O)ncn1C N1(C(c2c(C)scn2)=O)CCCCC(CNC(c2ccc(=N)[nH]n2)=O)C1 C1(C(=O)NC(C2CCCCC2)CNC(CC=C(C)C)=O)CCCC(=O)N1C C(=O)(C1=C(C#N)CCC1)NCCC(CNC(=O)CC1CC2CCC1C2)OC c1(COCC)cccc(OCCOCc2[nH]cnc2C)c1 CCC(CC)C(F)C(=O)N(C1(CC(=O)N(C2COCC2(C)C)C)CC1)C N1(C(C2C(NCc3c(Br)ccc(C#N)c3)C2)=O)CCc2ccc(Cl)cc2C1 CC(CC(=O)NCC1(CNC(c2ocnc2C(F)F)=O)CCCC1)P(C)(C)=O CN1CC2CCC(C1)N2C1CN(Cc2c(O)ccc(F)c2F)C1 C1(CC=C)(NC(C2CCCOCC2)=O)CCN(C(=O)CCCn2ccnc2)C1 N1(C(c2cc(C)ns2)=O)CC(NC(c2ccc3scnc3c2)=O)CC12CCOC2 N1(C(C2C(C)(C)CCN2C(=O)CC2CNC(=O)O2)=O)CCC(C)(O)C(O)C1 C12(C=O)CC3CCC(C1C2)N3C(C1CC1(C)C)=O.c1(OCC)ccc2nn[nH]c2n1 N1(C(C(C)(C)C2CC2)=O)CCC2(CC1)CN(C(c1cc(Cl)ccc1Br)=O)C2CO C12(C(N3CCC(=CCNC(c4c(C)nco4)=O)CC3)=O)CCC(C)(CC1)OC2 N12CCOC(C1)C(=O)N1CC3C(C3C1)CC2=O.C12(CC)CC(C1)C2 c1(C(=O)NC(C(=O)NCCOCCC)Cn2cccn2)cncnc1C C1(C(N2CC(O)(CNC(c3c(C)cccc3F)=O)C2)=O)CCN2CCCC2C1 N1(C(COCC)=O)CC2CCC1C(NC(c1ccc(OC(C)C)cc1Cl)=O)C2 C(N=c1[nH]cnc(Cl)c1C#N)C1CN(C(CCC2CCC(C)O2)=O)CC1(C)C CP(C)(=O)c1cccc(NC(=O)C(=O)NC2CC3CCC2CC3)c1 N1(C(C(C)CC(F)(F)F)=O)CCC2CN(C(c3cc(O)cc(O)n3)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)CC2COCCO2)C)cc(Cl)c(F)c(Cl)c1 C1(C(=O)NC2CC3N(C(CC(=O)OC)=O)C(CC3)C2)CC(F)(F)CCC1(C)C N1(CC(=O)NC2(C)CC(NC(C3N(N=O)CCCC3)=O)C2)CCCCCCC1=O N1(C(CC(c2ccc(OC)cc2)N)=O)CCC(O)C(NC(=O)CCCC(N)=O)C1 N1(c2cccc(C)n2)CCCC(C(=O)NCc2cc3c[nH]nc3s2)CC1 Cc1nc2sc1C(=O)NCC(C1CCC1)OC2.C1(CC(=O)N)CCOC1.C1(C)CC1 N1(C(CC2C(CC)CC2)=O)CCCC(C(=O)Nc2nccc(OC)c2N)CC1 CC(CC(=O)N1CC(CNC(c2ccc(C3CC3)nc2O)=O)CC1C)C(F)(F)F C(=O)(C(C(C)(C)C)OC)N(C)Cc1c(CNC(C2C(CCC)C2)=O)cccc1 c1(NC(C2C(CNC(C(C=C)C)=O)CCCC2)=O)cn(CC)nc1C#N C(=O)(CCCCCOC)N1C(CN(C(C23CCN(CC2)CC3)=O)CC)CCC1 C1(NC(c2c(C)nn(C)c2C)=O)CC2(CCCN(C(=O)C(O)C3CCC3)C2)C1 c1(SCC)ccccc1C(N1CC2C(N(C(=O)C(C(C)C)OCC)C)C2C1)=O C1(O)(C(=O)NCC(=O)NCC(=O)NCC2CNC(=O)CO2)CCCCC1 c1(C(N2CC3N(C(=O)Nc4c(CC)cccc4CC)C3C2)=O)cc(O)ccc1Cl Cc1ccc(OCC(=O)NCC23CCC(C2)N(C(C2OCCO2)=O)C3)cc1C C(=O)(C(CC(C)C)N(C(=O)C=Cc1ccco1)C1CC1)N1C(CC)CCCC1 N1(C(CC2C=NN(C)C2=O)=O)CCCC(C(=O)NC2CCC(C)(O)CC2)CC1 c1(NC(C(C(C)C)C2CC2)=O)cnc2[nH]c(O)nc2c1.C12C3CN(CC13)C(=O)C2 N1(C(COC)=O)CCC(C2(O)CCN(C(=O)CC3COC4(CCC4)CO3)C2)CC1 N1(C(C(C(=O)N(C)C)(C)C)=O)CC2(C1)CN(C(c1cnc(S)n1C)=O)CC2CO C1(OC)COCCC1N(C)C(C1CCC(NC(=O)OC(C)(C)C)C1)=O C1(NC(c2c(C)cccn2)=O)CCN(C(c2ccc(C)c(CO)c2)=O)CC1(C)C C(CC(C)(C)CC(=O)NC1CN(C(C2CC(OC)C2)=O)CC12CC2)OC C1(CCOC)(NC(=O)CC(=O)N(C)C)CCN(C(C2CCCSC2)=O)CC1 C1(CC(N2C(COC)COCC2)=O)CCCN(C(C2CCOC2C2CC2)=O)CC1 N1(C(CCCCC)=O)CCN(C(c2c(C)nsc2NC(C)C)=O)CC1C1CC1 Cc1nn2c3sc(cc13)C(=O)N1CC(C1)C2.C(=O)(C1=CCCC1)Sc1ccc(F)cc1 c1(C(=O)OC)ccc(C(=O)NC(C)CCCNC(c2cc(Br)no2)=O)[nH]1 Cc1nsc2cc(C(N3CCOC(CN=c4[nH]nc(O)s4)C3)=O)cnc12 C1(NC(C2(COC)CC2)=O)CCCN(C(c2cnn(CCO)c2N)=O)CC1 CCC(C(=O)N(C)CC1CC(F)CN1C(c1cc(C)on1)=O)C(C)(F)F N1(C(C(C2CC2)OCC)=O)CC2CC(C(N3CCCC(C(C)C)C3)=O)(C2)C1 C(=O)(C(F)CCC(C)(C)C)NC1CC2(CN(C(C(CC)COC)=O)C2)OC1 c1(C(=O)NCC(C)N(c2snc(CCC)n2)C)ccc2scnc2c1 C(=O)(CCC(C)(C)C#N)NCc1c(C(N2CC(C)S(=O)CC2)=O)n[nH]c1 N1(C(c2c(C)coc2C)=O)CC2(CCCC(CNC(C3CC(F)C(=O)N3)=O)O2)C1 c1(C(N2CCCC(F)(CNC(C=NOC)=O)C2)=O)c(OC)cc(OC)cc1N C1(C(C)C)CN(C(=O)C(C)c2ccsc2)CC1C(N1C(C)CC1(C)C)=O C1(c2cn(CC)nc2)CN(C(=O)CN2CCC(n3cccc3)C2)CCO1 C(c1ccc([N+](=O)[O-])cc1)=CC(C1(F)C(C(=O)OC)C1)=O.C(=O)O NS(=O)(=O)c1ccc(F)c(C(N2CC3CC3(CNC(=O)C(O)C3CCC3)C2)=O)c1 C1(C)(C(=O)NC(C)CCNC(=O)CC2CSC2)CCCCC1 c1(C(=O)NCC2CCCC2NC(C2CCCS2)=O)ccnnc1S c1(OC)ccc(C(=O)NCCC(O)CNC(c2nocc2Cl)=O)nn1 C(=O)(C#CC1CC1)N(C)CC1CCC(C(N2C(C(N3CCCC3)=O)CCC2)=O)O1 N1(C(C(CC)n2ccnc2)=O)CCN(C(C2CCC(=O)N2)=O)C(COC)C1 C#CC1(C(=O)N(C2CCC2C)C)CCN(C(=O)CCc2cc(C)[nH]n2)CC1 N(C(=NCC1CCCN(C(C)=O)C1)N1CC=C(F)C1)C(CC)CC Cc1csc2ncnc(N3CCC(O)CC3C(=O)Nc3ccccc3)c12 O=C1CCOC(COC(=O)CCc2ccc(C(F)(F)F)cc2)C1 c1(C(=O)OC)cccc(Cl)c1S(=O)(=O)NC1CN(C(c2cn[nH]c2)=O)CC1OC Cc1cccc(Cl)c1CC(=O)NC1CN(C(C23CC(C)(CO2)C3)=O)CCC1C c1(C(=O)NCC(CNC(CCCCOCC)=O)O)nc(Cl)ccc1F c1(C(=O)NC2CCN(C(c3cnc(Cl)nc3)=O)CC2F)c(O)cc(O)cc1O CCCCC(C)(F)C(=O)N1CCN(C(=O)CC(C(N)=O)NC(C)=O)CC1C N1(C(c2ncn(C(C)(C)C)n2)=O)CCC2(CC(NC(C3CC34CCC4)=O)C2)C1 c1(NS(CCN(C)CC2CCCC2)(=O)=O)ccc(F)c(N2CCC(=O)NC2=O)c1 c1(CC)cc(CC(N2CC(C(N3CC=C(C)C3)=O)(CO)C2)=O)on1.C(C)(C)N n1(CC(N2C(CNC(C3C(C)C3(F)F)=O)CCC2)=O)nnc2ccccc2c1=O c1(C(=O)NC(CNC(C(C)=C(C)C)=O)C)cnc(N(C)C)cn1 C(=O)(C(C)CC(C)(F)F)NCC1(C(F)F)CCN(C(c2c(C)nsc2C)=O)C1 NC(CSCCCN=[N+]=[N-])C(=O)N1CCCC1 C(=O)(C(CCC1CCC1)NC(=O)CCC=C(C)C)NC(CC)CSC N1(C(CN(C)C(N)=O)=O)CC2CC(NC(C3CNC(=O)N3)=O)CC(C2)C1 c1(C2C(C(N(CCCNC(=O)CCc3ccco3)C)=O)C2)ccncc1 c1(CCC(=O)NC2(CNC(C3CC(CC)OCC3)=O)CC2)cccc(F)c1Cl Cc1cnccc1C(C)C(=O)NC(C)CN(C(=O)CCC1CC1)C CCC1=C(C(=O)NC(C)C(c2ccccc2)NC(=O)CN(C)C(C)C)CCCO1 c1(C(N2CC(C(=O)NCc3nn[nH]n3)(SC)C2)=O)cc[nH]c(=N)n1 Cc1c(C(N2CCN(C(C34CC(C3)C4)=O)CC2)=O)cccc1F C1(C(CNC(C2CC=CC2)=O)NC(c2ccn(C3CC3)n2)=O)CCCCCC1 N1(C(c2cc(C)ns2)=O)CCC2CCN(C(c3cc4c[nH]cnc-4n3)=O)C2C1 CN1CC(O)CC1(C)C(N1CC(C)(NC(c2cc(C(C)(C)C)c[nH]2)=O)C1)=O N1(C(c2c(C)c[nH]n2)=O)C2CCC1CC(NC(c1ccc(CN(C)C)cc1)=O)C2 c1(CC)nn(C)cc1C(=O)NCC(O)CNC(=O)COc1ccccc1O c1(CC(=O)NCC=CCNCCC(C)O)cncc(Br)c1 c1(CNC(C2C(C)C2)=O)nc(CNC(=O)CCc2cc(F)cc(F)c2)cc(O)n1 N1(C(CCOCCOCC)=O)CCC(C(=O)NC2(C#N)CC2)C1 C1(CCCC)CN(C(=O)CSC)CCN1C(=O)CCCCSC c1(C(=O)OC)ccc(F)c(F)c1-c1noc(N2CC3CCN(C)C3C2)n1 C#CCCCCCCC(=O)NC(C)(C(=O)NCCc1ccn(C)n1)C1CCC1 c1(OC)ccc2ncccc2c1C(N1CCCC(CN(C(=O)CC(C)O)C)C1)=O C1(NC(C2C3COCC23)=O)CCCCCN(C(=O)C=Cc2cn[nH]c2)C1 C1(NC(C=CC)=O)CC(CNC(C2CN(C(=O)NC3CC3)C2)=O)C1(C)C.O c1(N2C(C(=O)Nc3cc(C(=O)OC)sc3C)CNCC2)ncnc2ccsc12 c1(NC2CC(=O)NCC2)ccc(S(=O)(=O)NCc2ccsc2)cc1F c12conc1NC(=O)CNCCN(CC(F)F)C2=O.N1(C2CCC2)CCOC1=O c1(C(N2CC3CCCN(C(CCCC#C)=O)C3C2)=O)c(F)ccc([N+](=O)[O-])c1C c1(-c2cn(CCOC)nc2)ccc(C(=O)Nc2cc(C(C)(C)C)no2)c2[nH]ccc12 c1(C(N2CCC(C(C)NC(=O)C(F)=C3CCC3)C2)=O)cc(C(F)(F)F)cc(N)c1 c1(C(=O)NC(CNC(C2N(C(C)=O)CCOC2)=O)CO)c(C(C)C)nn(C)c1C(F)F C(c1cnn(C)c1)=C(C(=O)NC1C(CNC(C(C)=C2CCC2)=O)C1)C C(=O)(C1=NN(C)C(=O)CC1)NC1C(C)CN(C(=O)CCNC(=O)CO)CC1C c1(C(=O)NCC2(CNC(C3(C)CC3(F)F)=O)CCCC2)cc2cnccc2[nH]1 C1(C(=O)NC(C)C(F)(F)F)CC12CN(C(=O)Cc1ncsc1Br)C2 C1(C(N2CC(CNC(c3cn(CCN(C)C)nc3)=O)C2)=O)CC1C1CCCC1 N1(C(c2cn(CCC)nn2)=O)CC(NC(c2csnc2Cl)=O)CC1(C)CC c1(C(=O)NCC2OCCN(C(CSCCN(C)C)=O)C2)ccc2nc(S)oc2c1 C1(CC)CC(C(=O)NCC(C)N(C(=O)Cc2c(C)noc2Cl)C)CCC1=O Cc1[nH]nc(C(N2CCCC2C(C)(C)NC(=O)CC2CCCO2)=O)c1C C1(O)(CN(C(C(C)NC(C2CCCC2)=O)=O)C)CN(C(C2CC(F)(F)C2)=O)C1 O=C(C1=CCC(F)(F)CC1)NC1CCCC1NC(c1cc(O)nc(C2CC2)n1)=O C1(C(N(CCNC(C(CC)F)=O)CCOC)=O)OCC2CCCC12 c1(C(=O)OC)cc(C(=O)NC2CCCCC2NC(C2CCC(C)(C)O2)=O)c(C)o1 N1(C(COC(CC)(C)C)=O)CC=C(CC(=O)NCC(C)CC2CC2)CC1 CC1(C)CN(C(C2CC=CCO2)=O)C1C1CCN(C(C2CCS(=O)(=O)N2)=O)CC1 C1(CNC(CSCCOC)=O)CCC(N(C(=O)C(C)CO)C)CC1 C1(CC(C)NC(=O)CC2(CNC(C3CCCS3)=O)CC2)CCOC1 C1(C(=O)NCC2(C(=O)NC3(C)CCSC3)CCCC2)Cc2nccn2C1 CC(C)(C)C(C)(C)C(=O)NCCNc1ccc(Cl)cc1C#N c1(CN2C(C(=O)NCc3ccc(COC)o3)C=CC2)ccc(OC(F)(F)F)cc1Br C1(CCOC)(C(=O)NCC2(CNC(=O)C=CC(=O)N(C)C)CC2)CCC1 C1(C(N2CC(=C(CNC(C(=O)NCC)=O)F)C2)=O)CC2COCC(C1)C2=O N1(c2cc(NS(C(CCC)C)(=O)=O)ncn2)CCC(F)(F)C(C#N)C1 Cc1c(C(N2CC(F)(CNC(C3CCOC3)=O)C2)=O)sc2cc(F)ccc12 C1(N(C(=O)C(C2(C)CC2)NC(c2cnn[nH]2)=O)C)CCC2(CC1)CC2 C1(C(=O)NCC2C(NC(c3ccc(C)cc3O)=O)C2)CC(C)(C)OC(C)(C)C1 C1(C(N2CC=CC(NC(Cc3cc(C)cc(F)c3)=O)C2)=O)Cc2ccccc2N1 CC(C)(C(=O)N(CCCNC(C1(F)C(C)(C)C1(C)C)=O)C1CC1)C(N)=O N1(c2n(C(N3CCOCC3)=O)c(-c3ccon3)nn2)CCc2ccc(CO)cc2C1 C(=O)(C1=CCC2CCC1N2C(=O)C(C)CC(C)C(C)=O)NCc1c(CC)noc1 C1(CNC(C(CNC(=O)Cc2cn[nH]c2)N(C)C)=O)NC(=O)CC1(C)C Cn1ccc2ccnc(C(=O)NC3CCN(C(c4snc(O)c4Cl)=O)C3(C)C)c12 c1(OC)ccc(C)cc1CC(=O)NC1CC(O)CN(C(c2csc(C)c2)=O)C1 C(=O)(C(CCCCNCCCCOC)N(C(CCC)C(N)=O)C)OC C1(C(=O)NCC(CNC(c2n(CCCC)ncc2)=O)CO)CN(C(C)C)CCO1 c1(OC)cc(C)cc(C(=O)NC(C2CCN(C(c3nc(O)sc3C)=O)C2)C)c1O N(C1CCc2cccnc21)C(C(C(C)NC(CC(C=C)CCC)=O)(C)C)=O Cc1cccc(F)c1C(N1CCC(NC(C2CCC2(F)F)=O)CC1)=O C1(C(=O)O)C=CCCN1C(=O)CCC1CCCN1C(=O)CC=Cc1ccccc1 c1(C(=O)NCCOCCCNC(CC(C)CF)=O)c([N+](=O)[O-])cnn1CC(F)F c1(C(=O)NCCOC2CCN(C(C3(O)CC(O)C3)=O)C2)cc(F)c(F)cc1F N1(c2nc(SC)nc(C)c2)CC(C2CCCN(C(c3cc(O)cs3)=O)C2)C1 Cn1nc(Br)nc1C(=O)NC(c1cn(CC2(F)CCOC2)nn1)(C)C N1(C(CCOCCC)=O)CCCN(C(=O)CC2CNC(=O)C2)CCC1 N1(C(C(CC)SC)=O)CC(NC(C2CC(C(C)C)=NO2)=O)C(C)(C)C1 C1(C2CCC2)(C(N(C)CC2CCN(C(c3cncs3)=O)C2)=O)CC1(F)F C(=O)(C(CC)CC(C)C)NCC(CNC(COCC)=O)OC c1(C(=O)O)cc(CN2CCCC(c3ccc(F)cc3F)C2)cnc1O c1(CC(=O)NC(C(C)(C)C)CNC(c2cc(C3CC3)no2)=O)cc(O)nnc1O N1(C(C(C)OCC)=O)CCC2(CCN(C(c3cnns3)=O)C2)C1 CCC(CC)CCCC(=O)N1CCC(C(=O)NCC(C)(F)C(C)(C)F)(CO)C1 c1(C(=O)NCC(C(C)C)NC(C2CC2c2cnc[nH]2)=O)cnc2[nH]cnc2c1 C1(NC(C(CC)C#N)=O)CC2(CCCCN2C(=O)C(c2ccccc2)F)C1 C1(NC(C2CCC(=O)N2)=O)CCC2CN(c3nnn(CCCO)n3)CCC2C1 C1(NC(C2CC2F)=O)CC2CC1N(C(c1ccncc1-n1cccn1)=O)C2 C1(CNC(CCC(=O)NCC)=O)CC2CCC1N2C(C1(O)CN2CCC1CC2)=O c1(-c2n(-c3c(C)noc3C)nc(C3CCCC3)n2)ncccc1S(C)(=O)=O N1(C(C)=O)CCCC(O)(CNC(=O)C2=NOC(CNC(=O)OC(C)(C)C)C2)C1 N#Cc1ccc2cc(C(N3CCN(C(c4csnn4)=O)C4CCC34)=O)ccc2c1 C1(NC(C(=O)NCCCc2ccc(C#N)cc2)=O)Cc2cccnc2C1 c1(N2C(C)CCC(NC(c3ccn(CC)n3)=O)C2)ccc([N+](=O)[O-])cc1Br N1(C(C(C)NC(c2ccccn2)=O)=O)CC2(CCCN(C(=O)CS(=O)(=O)CCl)C2)C1 Cc1cccnc1C=CC(N1CCCC(N(C(=O)C2=CCCCC2)C)CC1)=O Cc1ccc(CNC(=O)C(CCN(C)C)NC(C2CC(O)C2)=O)nc1 N1(C(c2cc(C)c(Br)s2)=O)CC(NC(c2n[nH]c(C)c2F)=O)CC(F)C1 C12(CNC(c3scc(C)c3C)=O)CCC(C1)N(C(=O)C(C1CCC1)C1CCC1)C2 C=CC1(CC(=O)NC2CCCC(CN(C(=O)C=CBr)C)C2)CCOCC1 C1(C(N2CCN(C(c3cnn(C)n3)=O)C(CO)C2)=O)CCCCCC1(F)F C1(C)(NC(Cc2nc(C3C(C)C3)sc2)=O)CCN(C(=O)CO)CC1 Cc1cc(C)c(C(=O)NCCCC2CCCN2C(=O)CNS(N)(=O)=O)c(=O)o1 c1(CN(C2CN(C(=O)C=Cc3cccnc3)C2)C)ccc2c(c1)CCO2 c1(NC(C2SCCN(C(C(CC)O)=O)C2)=O)ccc(C(F)(F)F)c(C#N)c1 C1(SCC(=O)NC2C(NC(c3c(CC)c[nH]n3)=O)CCC2)CCS(=O)(=O)C1 N1(CC(=O)N(CCC(=O)N(C)CCc2cccs2)CC)CCCNC1=O CCCC(CNCC(C)C(=O)OC)C(=O)N1CC(=Cc2cc[nH]n2)C1 c1(NC(c2ncccc2NCc2scc3c2OCCO3)=O)c(Cl)cc(C#N)cc1Cl C=CC1(C(=O)NCC#CCNC(c2ccncc2Br)=O)CCOCC1 CCCCC(CC)CC(=O)NCc1ccc(C(C)NC(c2ccncn2)=O)cc1 c1(C(N2CCC(N(C)CC)C2)=O)ccc2c(c1)n(C)c(=O)n2C c1(SC)ccc(O)c(C(=O)NCCCCC(C)NC(c2ocnc2C2CC2)=O)c1 N1(C(CSCC=C)=O)CC(NC(=O)CN=S(C)(C)=O)CC12CCCOC2 c1(C(N2CC(N(C(C3CCC(OC)C3)=O)C)C2)=O)nc(C)c(C)[nH]c1=O CCN=C(NCc1cccs1)NCCc1ccc(Cc2ccccc2F)cc1 c1(C(=O)NCC(CN(C(=O)CCCS(C)(=O)=O)C)O)nnc(O)c2c1CCCC2 C1(C)(COC2CN(C(C(CC)N(C)C)=O)CC2CNC(N)=O)CC2(CCC2)C1 Cc1ccc(O)c(CNC(=O)C(CO)NC(c2ccc(C(C)C)o2)=O)n1 n1(CCC(=O)NCC2(O)CC(NC(CC3ON=C(C)C3)=O)C2)ccc(O)nc1=O C1(OC)CN(C(C2CC2C2(C)COC2)=O)CCC1NC(C1CCC1(F)F)=O c1(CNC(C2(C(=O)OCC)CCNC2)=O)cncc2c1CCC2 C(CN=c1[nH]nc(C(C)(C)CC)s1)C1N(C(CCC(=C)Cl)=O)CCCC1C CC(C)C1=NOC(C(N2CCC(CF)(NC(=O)CCCc3cccnc3)C2)=O)C1 C(=O)(C#CC1CCCO1)NCC1N(C(c2cccc(C(C)C)c2F)=O)C2C(C1)C2 N#Cc1ncc(CC2CC2)nc1N1CCC(C(N)=O)CC1 C1(NC(C2CC(=C)C2)=O)CN(C(c2cn(CC(F)F)nc2C)=O)CCC1C C1(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC12CCN(C(=O)CO)CC2 Cc1[nH]nc(C(N2CC(NC(c3cc(Cl)c[nH]3)=O)CC2C)=O)c1O c1(OC)ccc(C(C)=CC(N2CCCC(NC(=O)COC3CC=CC3)C2)=O)cc1 CCCCC(CC(=O)NC1(C(N)=O)CCCOC1)NC(C1CCC1C(C)(C)C)=O N1(C(Cc2c(C)n[nH]c2)=O)CC(N(C)C(C2CCCS(=O)(=O)C2)=O)C(C)(C)C1 c1(CCC)cc(Oc2nnc(C(F)(F)C(=O)OC)n2C)ccn1 C1(CNC(=O)Cc2cc[nH]c2)COCCN1C(=O)CC1CC=CC1 Cc1cc(CO)oc1C(=O)NC(CNC(=O)C(O)CCc1ccccc1)CO C=C1Cn2c(C(=O)NCC(CNC(c3cc(C4CC4)on3)=O)CO)nnc2S1 CC1(C)C=NN1C(=O)C(C(F)(F)F)NC(C1CC(OC(F)F)C1)=O c1(C2(C(=O)Nc3sccc3Br)CC2)ccc(-n2ccnc2)cc1 C1(C(N2CCN(C(c3c(C(C)(C)C)cccn3)=O)CC2)=O)CC2C(C1)C2(F)F C#Cc1ccc(C(C)(COC(=O)C(N)COC)OCC)cc1 C(CC(C(C)(C)C)NC(c1cnc(Br)s1)=O)N(C(=O)C1=CC(C)(C)C1)C c1(CC)ncc(Cl)c(C(=O)NC2CN(C(=O)C(CC)n3cncn3)CC2(C)C)n1 Cc1cn2nc(C(=O)NCC(O)Cn3ccnc3)cc(C)c2n1 N1(C(c2cc(C)oc2)=O)C2CCCC1CC(NC(=O)Cc1c[nH]c(=N)nc1O)C2 C1(NC(c2ncn(CCNC(CC(C)C#N)=O)c2)=O)CC2CCC(C1)N2C CCC(C)(CCCNC(N1CCC(Oc2cc(Cl)ccc2Cl)CC1)=O)C1OCCO1 N1(C(CNS(C)(=O)=O)=O)CC2CC1CC2NC(c1cc(Cl)ccc1O)=O C(=O)(C(=O)C(C)(C)C)NC(C)CCCCNC(c1cccc(C2(O)COC2)c1)=O CC1(C)C(CNC(=O)C=CCN2CCC2)CCN1C(c1cc(O)nc(O)c1)=O n1(CC(=O)NC2C(CNC(c3c(CCC)n[nH]c3)=O)C2)nc(C)n(C)c1=O N1(C(C(Cc2ccccc2Br)NC(CC(CC)OC)=O)=O)CCC(C)(F)CC1 c1(OC(C(N2CCC(NC(CCC=C)=O)C2)=O)C)ccccc1OC CN1CC(CNC(C2(N(C(=O)Cn3cnc(C#N)n3)C)CC2)=O)CC1=O C1(C(=O)NC(C2CSC2)C)CCOCCN1C(=O)Cc1nc(=N)[nH][nH]1 Nc1c(C(N2CCC=C(CNC(=O)CC3CCCC3)C2)=O)cnc2ccnn12 c1(C(N(CC(C)N(C(CCSCC(C)C)=O)C)C)=O)cc2c(nc1N)CCCC2 Cc1cccc2nc(NC3CC(NC(C4(CO)CCCC4)=O)C3(C)C)sc12 C(=O)(C(F)(CNC(c1ccn(COC)n1)=O)C(C)C)NC(C1CCOCC1)CC c1(C(=O)NCC2C(NC(CCCC=C)=O)C2)ccc(C(F)(F)F)c(O)c1 C1(CCCC)CN(C(=O)C(C2CCC2)OC)CCN1C(C1CCC1)=O c1(C(=O)NCC2N(C(c3ccc(OC)o3)=O)CC2)c(OC)cncc1Br C1(C(N2CC(N(C(=O)C3=NOCC3)C)C2)=O)CCc2nncn2CC1 N1(C(c2cc(F)ccc2F)C(=O)NCCCSCC)CCC2(CC1)CNC(=O)C2 N1(C(c2nccc(C)c2)=O)CCCC(O)(CN(C(=O)CCC(C)(F)F)C)C1 c1(C(=O)NCC(C)NC(CC2CCC(C)O2)=O)cc2c(=O)[nH]ccn2n1 c1(OC(C)C)ccc(=NC(=O)CCCc2ccc(Br)cc2)[nH]n1 c1(C(=O)NCC2C(C)CN(C(C3CC4(C3)CC(O)C4)=O)C2)c(F)ccc(O)c1F c1(C(=O)NCC(C(C)(C)C)NC(=O)C(O)P(C)(C)=O)c(N)cccc1[N+](=O)[O-] c1(C(=O)NC2CC(CC(=O)NCC3CC(c4ccccc4)C3)C2)[nH]ccc1CO C#CCCCCC(=O)NCC(C1CCCCC1)NC(C1CC(C)=NO1)=O c1(CCC(=O)NCCC(C)N(C)C(c2cc(C(F)F)n(C)n2)=O)cncc(F)c1 c1(C(=O)NCC2C(C)(C)C(=O)C2)ccc(F)c(F)c1F C#CC1CN(C(C2CC(O)C(F)C2)=O)CCN1C(=O)CCCOC(C)(C)C c1(C(C(=O)NC(C)(C)CC)N(C(c2ccc(C)cc2)CC)C)ccc(F)c(I)c1 N12CC(C(C)(C)C1)C2=O.c1(CC)conc1C(=O)NCCC1CC(CO)C1 N(C1CC2(CCCC2)Oc2ccccc21)C(=O)C=Cc1c(Cl)nc2sccn12 N1(C(C(C)(CC2CCC2)OC)=O)CC2CC(NC(=O)CC3C=CCCC3)C(C2)C1 Cc1cc(Cl)cc(Cl)c1OCC(=O)NC1CCC1CNC(=O)CN1CCN(C)CC1 c1(CC)nc(C#N)cc(=NCCN2CCC(NC(C3NC(=O)CC3C)=O)C2)[nH]1 CCC(C(=O)N1CCCC1CC(=O)NCc1ocnc1C1CC1)C(F)(F)F C(=O)(CC1C(=O)Nc2cc(OC)ccc21)NC1C(NC(COCC)=O)CC1 N1(C(CCC(C)OC)=O)CC(NC(c2cnn(C)c2C(C)C)=O)CC12CCCC2 CCCCC(C(=O)NC1CC1NC(=O)COc1cccc(F)c1F)C(C)C C1(C(=O)NC(C2CC(NC(COCCCC#C)=O)C2)C)CCCC(SCC)C1 N1(C(C)=O)CC(O)CC1C(=O)N(C1CCN(C(c2coc(C(F)F)c2)=O)C1)C c1(C(N(CCN(C(=O)CCN2CCCCC2=O)CC)CC)=O)nn(C)c(N)c1C n1(CCC(C)C)nc(-c2ccc(F)cc2)nc1CC1COC(C)(C)C1 C(CC(O)C(C)(C)C)N(N1CCCC(CC(F)(F)F)C1)C.C(=O)NC c1(C(C(C)C)N(CC)CC)ccc(Br)c(F)c1.c1(=O)c(=O)o1 CCC(CCCC(=O)O)NC(c1cnc2ccccc2n1)C C1(NC(c2scc(OC)c2)=O)CCN(C(=O)CC2(O)CCC2)CCC1(F)F c1(CN2CCC(NC(=O)C(c3ccccc3)C3CC3)CC2)cc(Cl)nc(Cl)c1 C1(C(=O)NC(COC)(C)C)CC2C(C1)C2(F)F.c12ccc-1o2 C1(NC(C(CC)SC)=O)CCCCN(C(=O)C(c2ccc(F)cc2C)(F)F)C1 C1(C(C)N)(CCC=C2CCC(C)C2)CCCN(C(=O)CCCCN2CCCC2)C1 c1(C(=O)NCCCN(C(CCNC(N)=O)=O)C2CC2)onc2ccccc12 c1(CCC)cnc(N(C2CCC(NC(C)=O)C2)C2CCN(C)C2)nc1 N1(CCC(C)CNC(=O)OC(C)(C)C)CCCCC1C N1(CC(=O)NC2C=CCN(C(COC(CC)C)=O)C2)CCSC(C)(C)C1 c1(C(N2C(C3(NC(CCSCCC)=O)CC3)CCCC2)=O)cnc2ccoc2c1 c1(C(=O)NCCC(C)N(C(c2ccn(CC(C)C)n2)=O)C)ccccc1S(C)=O C1(=CC(=O)NCC2CCC(NC(=O)C(F)(F)C3CCCC3)C2)CN2CCC1CC2 Cc1ccc(N(C(=O)CNC(=O)C(O)CNC(C2CCCC(O)C2)=O)C)cc1 C(=O)(C(F)C(C)(F)F)NC1CC(C(=O)NC(C2CNC(=O)N2)C)C1 N1(C(C2(CC=C)CCC2)=O)CC2CCC2(CNC(=O)CN2CC(C)(C)C2)C1 N1(C(C2(CCOC)CCCC2)=O)CCN(C(C2CCCC(C)C2)=O)CC(C)(F)C1 C1(CC)C(CO)CCN1C(=O)NC(c1ccc(F)cc1)C(F)(F)F CC1CCN(C(=O)Cc2ccc3n[nH]cc3c2)CCN1C(=O)CC(C)NC(N)=O C(=O)(C1=CS(=O)(=O)CCC1)N1CCCC(O)(CN(C(=O)C(C)(C)CCC#N)C)C1 CC1(CNC(C23CCC(CC2)CC3)=O)CCCN(C(C2CCCN2C2CC2)=O)C1 c1(C(N2CC(C(C)NC(c3csc(C4CC4)n3)=O)C2)=O)ccsc1S(N)(=O)=O O=C(CC(C(F)(F)F)NC(C1CCC2(CCC2)C1)=O)NC1CC(O)C1O c1(-c2nc(CC=C(C)C)nn2CCCCO)cc(C)c(OC(C)C)c(C)c1 C1(CC(N2C(CC(=O)N(C3CC4CC4C3)C)CC2)=O)CC=CCN1C C(=O)(CCCC(C)(C)CC)NCC1CCC(C(=O)NC2C(OCC)C2C)C1 C(=O)(C(C)(C)CCCNC(=O)CC1CCC(C)(C)O1)N(CC(F)(F)CO)C c1(C(=O)NC(CCOC)CNC(=O)COc2cnc(Cl)cn2)ccnc(Cl)c1O C1(CC(=O)NCC2(C)CCN(C(c3ncc(Cl)cc3F)=O)C2)CN2CCN1CC2 C(=O)(C(F)(F)C(C)(C)O)N1CC(O)CC(NC(c2cn(C)c(=O)n2C)=O)C1 c1(CNC(=O)C(C)NC(C2CC(NC(CCCC#C)=O)C2)=O)cc(O)ccc1C N1(C(CC2N(C(c3cc(C)nc(C)n3)=O)CCCC2)=O)CCn2ncc(O)c2C1 c1(C(=O)NC2CC(O)CN(C(=O)Cc3csnn3)C2)ccc2ccccc2c1 C12(NC(CN(CCC)C)=O)CCCN(C(=O)CSc3ccc(OC)cc3)CC1C2 C(=O)(C(C)CN1CCOCC1)NCCN(C(=O)CC1(CC(=O)OC)CC1)CC C1(NC(c2[n+]([O-])ccc(OC)c2)=O)CN(C(C2(F)CCCCC2)=O)CC1N=[N+]=[N-] c1(C(N2CCC(NC(c3cccc(C)n3)=O)C(CO)C2)=O)sccc1S(C)(=O)=O C1(O)(CN(C)C(C2CCCCC2O)=O)CCN(C(=O)CSc2nncn2C)C1 CC1=C(C(=O)N(C)CC2CCN(C(c3n[nH]c(C)n3)=O)C2)CCCC1 C1(c2n(CCOC)nnn2)(Nc2ccc(O)cc2)CCC(C(N)=O)C1 N1(c2nc(N3CCC(c4ncc[nH]4)CC3)cc(C)n2)Cc2nn(C)c(N)c2C1 C1(C(=O)NC(c2nc(C(=O)N(C3(C4CC4)CC3)C)co2)C)CCOC1=O CC1CC(C(=O)NC2C3CCN(C(c4ccnn4C)=O)C23)=NO1 c1(C(N2CC(COC)(CNC(=O)CC3CCC4CC34)C2)=O)ccc(C)n(C)c1=O C(CCC(C)CC(=O)N1CC(NC(=O)C(C)(C)C(C)C)C(C2CC2)C1)=C(C)C C(=O)(N1CCCc2nccn21)C1N(C(C2(C3(O)CCOC3)CC2)=O)CCCC1 c1(C(=O)NCC(C(C)C)NC(c2scc(C)c2Cl)=O)cc2cnccc2[nH]1 C(CC(C(=O)NCOC)SC)OC.C(CN)(C(=O)CSC)OC.C1(C=O)(O)CCC1=O.C.N(C)C.N.N N1(C(c2nc(C)oc2)=O)C2CCC1CN(C(=O)CN1CCCCCCC1=O)CC2 c1(C(N2CC(N3CCN(C(CCC)=O)CC3)C2)=O)ccc(N)cc1Br Cc1nccc(C(=O)NC(C(=O)NCCCc2c[nH]nc2C)C2(C)CC2)n1 Cc1nc2sccn2c1C(N1CC2CCC1CC2NC(=O)CC1CC2(CC2)C1)=O Cn1cc(C(N2CCC3(C2)CN(C(=O)CC(F)(F)F)C3)=O)c2c(c1=O)CCCC2 C1(C(N2CCC(N(C(=O)Cc3cn(C)nc3C)CC)C2)=O)CC(C)CC(C)(C)C1 C(=O)(N=c1nc(O)c2cnn(C)c2[nH]1)c1ccc(-c2nncc(C)c2)cc1 c1(C(=O)NCC2N(C(c3cc(C)ncn3)=O)CCCC2C)cc(F)c(F)cc1F CCC(CC)(C(C)C)NC(C1CC(O)(CNC(=O)C(=O)C(C)(C)C)C1)=O c1(NC(C2CC(OC)CN2C(c2[nH]cnc2C)=O)=O)cnc(O)c(Br)c1 N1(C(Cc2c(C)ccs2)=O)CC2CCC2(CNC(C2CCS2(=O)=O)=O)C1 C(=O)(CC(=O)N(CCCNC(=O)CCC1CC1)Cc1nccs1)NCC#C N1(C(CCCN(C)C)=O)C2CCC1CC(NC(=O)CCCc1ccsc1)C2 C1(NC(c2cc(=N)[nH]cc2)=O)CCN(C(=O)CC2CCCCC2)CC1CO N1(C(C(C(C)C)N2CC(C)C2)=O)CCCC(F)(C(=O)N(C)C)C1 N1(C(CCC=C)=O)CC(NC(c2cnc(C)cn2)=O)C(C#N)C1 Cc1cc(C(=O)N(CCNC(=O)C(O)Cc2cc(Cl)sc2Cl)C(C)C)c(C)o1 Cc1ccc(OCC(=O)NCCC23CCC(C2)C3)cc1C.C12CC(C)N(C1)C2=O C(c1cccc(Cl)c1Cl)=CC(=O)NCC1(C)CCN(C(C(C)CC(N)=O)=O)C1 c1(C(N2CCOCC2COCCO)C(=O)NCC=C)cc(Cl)c(F)c(Cl)c1 C1(C2(O)CCN(C)CC2)(C(=O)NC2CCN(C(C(CC)(C)CC)=O)CC2F)CC1 CCC(C(=O)NC1CCC(NC(c2cc(C3CC3)[nH]n2)=O)C1)N(C)C CCCC(CNC(=O)C1=CCCC1)C(=O)NCc1[nH]ccc(=O)c1O N1(C(C=C(CCC)C)=O)CCN(C(=O)CC2(OCC)CCCC2)C(C(C)C)C1 S(=O)(=O)(c1ccc(N2CC(C)OC3(CCCC3)C2)c(Br)c1)NCC(C)C CCCC(C)(O)C(=O)NC(Cc1ccccc1)C(N1CC2CCC(C2)C1)=O CCC(CC(=O)NC1CCN(C(=O)CN2CCCNC2=O)CC1F)C(F)F C1(NC(C2CSC2)=O)CCN(C(=O)CC2CCS(=O)(=O)CC2)CC1F C1(C(=O)NC(C)Cc2ncn(C)n2)CC(N=[N+]=[N-])CN1C(=O)C1=CCCCC1 c1(OC)ccc(OC(C)C(=O)NC2CCCN(C(C3CCCC(=O)N3)=O)C2)cc1 O=C(C(O)CC(F)(F)F)NC1CCN(C(=O)Cc2ccnnc2O)C1 c1(OC)ncc(CONC(C(=O)NCc2ccccc2F)=O)cn1 C1(CNC(C2C(C)CC(=O)NC2)=O)CC2(CCC2)CN1C(C1(NC(N)=O)CC1)=O N1(Cc2ccc(C)c(C)c2)Cc2ccccc2C1C(=O)Nc1cc(Br)cnc1Cl N1(C(c2cnc(CC)[nH]2)=O)CCC(=O)NC2CN(C(=O)CC=C(Cl)Cl)CCC12 C=CC(C)N=C(NC1CC1C1CCOCC1)N1CCc2cc(Cl)cc(Cl)c2C1 c1(NCCC2(O)CCN(C(C3(C(C)C)CCC3)=O)CC2)ccc(Br)cc1[N+](=O)[O-] CC1CCC=C1C(=O)N1CCC(CN(C(=O)C(O)Cc2ccccc2Cl)C)CC1 c1(C(N2CCC(C(C)NC(c3cn4c(n3)SCC4)=O)C2)=O)ccc2nccn2c1 C1(NC(C=C(C)Cl)=O)CCCOC12CCN(C(C1CC(C)(F)C1)=O)CC2 C(CN=c1ccc(C)c[nH]1)NC(=O)NCC=CCCOC N1(C(c2cncnc2C2CC2)=O)CCC(c2cn(CC3CCCO3)nn2)C12CC2 c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)cc(Cl)c(N)c([N+](=O)[O-])c1 c1(C(N2CCCN(C(C3CCOC(CF)C3)=O)CCC2)=O)cc(=O)n2nccc2[nH]1 c1(C(C(F)(F)F)OC(C2(C)CC(=C)C2)=O)c[nH]c2ccccc12 c1(C(=O)NC2C3OCC(NC(c4c(CC)ncs4)=O)(C3)C2)cc2c(s1)CCCCC2 Cc1c(C(=O)NC2CCCCC2NC(=O)CC2CC(C)(C)CO2)cccc1C#N CC1CN(C(=O)C(N)=O)CCC1CNC(=O)COc1cccc(O)c1 N1(C(C2C(C#C)C2)=O)CCCC2(C1)CN(C(c1cc(C(=O)O)cc(Br)c1)=O)C2 c1(-n2cc(CONC(C3(C)CCCCO3)=O)nn2)cc(F)cnc1Br c1(OC)ccc(NC(=O)C(c2c(C)cnn2C)N(C2CSC2)C)cc1 CN1CCN(C(c2cncc(Cl)c2)=O)C(CNC(=O)C2=CCOC2)C1 c1(CC)cc(C(N2CC(C)(NC(c3noc(C)c3Br)=O)C2)=O)c(C)o1 C(=O)(C(F)(F)c1nccs1)NCC1(CNC(C=CC(C)(C)SC)=O)CCC1 c1(CC(=O)NC(C)CNC(C2(C(=O)N(C)C)CC2)=O)cc(F)ccc1Cl C1(Cc2cn(CC(C)NC(=O)CCCc3cccs3)nn2)CCCCN1C C(CC(Cc1ccccc1)NC(=O)C(C)C#N)NC(C=C(CC)C)=O c1(CC)nc(C(=O)NC2(C(=O)NC(C)Cn3cncn3)CCSC2)co1 c1(C(C)OC(C2C(C)CN2C(=O)OC(C)(C)C)=O)ccc2cccnc2c1 CC(CC(=O)N1CC(NC(C2(C#N)CC3CCC2CC3)=O)C(C)C1)CC(C)(C)C C(C)(C)(CCCC(=O)NCc1nncn1C)NC(c1cc(OCC)n[nH]1)=O CN=c1cc(CNC(c2ccccc2CCC(C)C)=O)cc[nH]1 c1(C(=O)NC2CC(CNC(=O)Cc3ccsn3)C2)cnn2c1OCC(F)C2 c1(C(=O)NC(C)CCCCNC(C2CC3CCC2CC3)=O)ccnc2[nH]cnc12 C1(N2C(C3CCN(C(CNC(CCC)=O)=O)C3)CCC2)CCN(C(=O)C(C)O)CC1 c1(C(=O)NC(C2(CNC(c3cc(COC)oc3C)=O)CC2)C)cn(C)ccc1=O C1(N(C)C(c2cccc(CF)c2)=O)CCCCN(C(C2(C)CCCCO2)=O)C1 CC1(C(=O)NC(C2CCCC2)CNC(=O)CCc2csc(=N)[nH]2)COCCO1 C=CC(C)(CCOC)C(=O)NCC1CC(O)CN1C(c1ccc(C)c(C)c1)=O N1(C(CN(C2CCSC2)C)=O)CCC(OCCN(C(C2CCCO2)=O)C2CC2)CC1 c1(OC)cc(CC(N2CC(N(C(=O)C(F)F)C)C2)=O)ccn1 c1(C(=O)NC(C(C)NC(=O)CC(C)C2CC2)C)ccccc1OCCN(C)C.C=O C12(C(=O)NC3CCC(OCCC(C)C)CC3)CCC(C1)C(=O)NC2 CC(C)CC(C(=O)NCC1(CNC(=O)CN2CCCCCC2=O)CCC1)C(N)=O C1(NC(C(F)=CCC)=O)CN(C(=O)CCn2c(C)n[nH]c2=O)CCC1C N1(C(CCSC)=O)CCN(C(c2ccnc(OC3CC3)c2)=O)CC1C(C)C Cc1ccnnc1C(=O)NC(C)CCCCNC(C1CC(=O)N(C(C)C)C1)=O N1(C(C(C)C(F)F)=O)CC2CCN(C(=O)CCCc3ccc(F)c(F)c3)C2C1 CC(CC(C)(C)C)C(F)C(=O)NC1(NC(=O)C2=CC3C=CC(C2)C3)CCC1 C(=O)(CC(C(C)OC)NC(=O)CCC(N)=O)NCCC(=O)NCC c1(OC)cc(F)c(C(=O)NC(C)CN(C)C(C2Cc3nncn3C2)=O)c(F)c1 CC(C)CC(C)CC(=O)N1CCOCCC1C(=O)NCc1cn(C)nn1 N1(C(C(OCC)O)=O)CCC2CN(C(c3ccnc4c3CCO4)=O)CC12.CC C(=O)(C(CC(F)F)c1ccccc1)NC(CC=C)CNC(=O)Cc1occc1C c1(N2CCC(N(C)C(c3cc(Cl)c(Cl)cn3)=O)C2)ncnc2c1CCCC2 C=CCC(C)C(=O)NC(c1ccccc1)CNC(c1sccc1C1CC1)=O N1(C(C(OC)OC)=O)CCN(C(C2(O)CC2(C)C)=O)CC1 CC1CC2(CC(C(N3CCN(C(c4cnsc4)=O)C(CC(C)(C)C)C3)=O)C2)C1 c1(C(=O)NC(c2cccc(-c3c(C)cc(C(=O)O)s3)c2)C)c[nH]cc(Br)c1=O c1(C(CC)C)cc(NC(=O)NCC2(c3sccc3OC)CC2)on1 c1(OC)csc(C(=O)NC2CC(N(C(=O)CC3CCSCC3)C)C2)c1OC C(C(C)(O)C(=O)NCC1(CNC(C2CCN(C(C)=O)CC2)=O)CC12CCC2)OC c1(N2CC(O)(CCNC(C3C(C)CC(=O)NC3)=O)C2)cccc(F)c1[N+](=O)[O-] N1(C(CCSC)=O)CCN(C(=O)C(F)CC2CCOCC2)CC1CCC(F)(F)F N1(C(c2c(C)ocn2)=O)CCCN(C(C2CCC3C2C3(F)F)=O)CCC1 C1(NC(C(CC)=CC)=O)CN(C(c2cc3ncccc3o2)=O)Cc2ccnn2C1 CCC(CC(=O)NC(CNC(=O)Cc1csc(NC=O)n1)CCOC)C1CCC1 c1(CN(CC(F)F)C(C2C(=C)C2C(=O)OC)=O)ccncc1.C1C(=O)N1 C1(CNC(c2cc(CC)oc2)=O)CC(C)N(C(=O)Cn2cc(CO)nn2)C1 N1(C(CS(CC)(=O)=O)=O)CC2CCC1CC2NC(C1CCC(C)C1)=O C(=O)(C1CCCc2nnn(C)c21)N1C(CCNC(CCCC#C)=O)CCCC1 c1(NCC2ON=C(CC)C2)cc(N2CCC(C)(CO)C2)nc(C(C)C)n1 C(C(CN=c1cc(C)nc(OCCOC)[nH]1)C(F)(F)F)NC(CSCCCC)=O C1(CNC(C(CNC(CSCCCC)=O)O)=O)CNC(=O)CO1 C=CC(C)CC(=O)NC1CCCN(C(c2ccc(CCC(F)(F)F)cc2)=O)C1 C1(NC(C(C)(C)NC(C=COC)=O)=O)CC2CC(NC(=O)CC3CSC3)C1C2 c1(C(=O)NCC#CCNC(C(c2cccc(OC)c2)C)=O)ccc2c(c1)CCN2 N1(C(COCC(=C)C)=O)CC(NC(c2ccc(N(C)C)cc2)=O)CC(C)C1 C(=O)(C1=CCc2ccccc21)NC1CCCN(C(C(C(C)(F)F)(C)C)=O)C1 Cc1ncc(Br)c(C(=O)NC(C)CCNC(=O)CCOCC2CCCO2)n1 N1(C(C)=O)CCCCC1COCc1ccc(CSC)cc1 C1(C(=O)NCCc2cnc(C)s2)C2CCC(C2)N1C(=O)C(O)CC(N)=O CC1(C)CCCN(C(C2CCCC(O)C2)=O)C1C(=O)NCCCOC1CCCC1 c1(CC(=O)N(C)CC2CCCN2C(=O)C(C2CCCCC2)=O)ccnnc1O CCCCCC(O)CC(=O)NOCC(N1CCC2(CCSCC2)CC1)=O CC1CN(C(C2(C(C)(F)F)CC2)=O)CC2(CCN(C(=O)C(C)(C)CF)CC2)O1 C=CCN=c1[nH]cc(C(=O)N(C(C)CNC(=O)CC2CN(C)C2)C)s1 C1(CNC(CC=C)=O)CN(C(c2cnn[nH]2)=O)CCC1C(F)(F)F C1(C(=O)NC2CCN(c3ncn(C)c(=O)c3)CC2F)CC2(CCCC2)CO1 CC(CNC(=O)CC1(C)CC1)C(F)C(=O)N(C)Cc1cocn1 C(=O)(C(C(CC)CC)OC)N1CCCC(CC)(NC(=O)CCCc2cc[nH]n2)C1 C=CC(CC)CC(=O)N1CC(C(N2CCC3C(C(N)=O)C3C2)=O)(CC)C1 c1(C(CC(=O)OCC)OC)cc(C)ccc1ON1CCCC(C)C1C c1(C(=O)NC(C)(C)CNC(c2ccccc2CC#N)=O)cncc2sccc12 N1(C(c2c(OC)c[nH]n2)=O)CCCC(CCCCNC(C2(Cl)CC23CCC3)=O)C1 c1(C(=O)NCC(C2CC2)NC(Cn2cc(C(C)=O)nn2)=O)c(C)nsc1C c1(C(N2CCC(NC(=O)C(O)CF)CC2)=O)cnc2nc(O)nc(O)c2c1 C(=O)(C(C)(C)CCC(=O)N1CCC(NC(C2C3COCC23)=O)CC1)OC CCC(CC(=O)NC1COCC1NC(=O)C(c1ccncc1)C1CCCC1)C(F)F c1(C(N(C2CCN(C(CC3CC(C)C3)=O)C2)C)=O)cc(=O)c2ccncc2o1 CC(CC(N)=O)C(=O)N1CCCN(C(C2CCCCC2C(C)(C)C)=O)CC1 c1(C(=O)NCCNC(C2(Cc3ccccc3)CCCO2)=O)cc(O)cc(O)n1 c1(CCC)onc(C)c1C(=O)NCCC(C)NC(C1CCOC1=O)=O c1(C(=O)OC)c[nH]c2ncnc(N3CCOC(CN4C(=O)C4CC)C3)c12.OC Cc1ccc(CNC(C2CCC(NC(C3(F)CCOCC3)=O)CC2)=O)nc1 c1(C(N2CC(NC(CCOC)=O)C(F)C2)=O)cc2cc(Cl)sc2[nH]1 Cc1cc(C(N2CCC(O)(CNC(=O)Cc3cc[nH]c3)C2)=O)ccc1Cl C1(CC)CN(C(C2CSCCS2)=O)CCN1C(c1cnc(C(C)(C)C)s1)=O CCC(CNC(=O)CN1CCCS1(=O)=O)(CC)NC(=O)C(=Cc1cnc[nH]1)C C(=O)(CS(=O)(=O)CC(F)(F)F)N(C)CC1CCCN(C(C(CCC)OC)=O)C1 Cc1cc(OC2CN(C(c3ccc(I)cc3F)=O)C2)cc(C)c1 N1(C(CSC)=O)CCC(C2CCN(C(C3(n4ccnn4)CC3)=O)CC2)C1 c1(OC)ccc2[nH]c(C(=O)NCCN(C(=O)CC3CC3(C)C)C3CC3)cc2n1 N1(CC(=O)NCc2c(Cn3cc(C4(CC)CC4)nn3)nco2)CCCCCC1=O C1(CNC(c2scc(C#N)c2)=O)CN(C(C2(CF)CCC2)=O)CC12CC2 C1(CC(NOC(CC)CC)=O)CCCCN1C(=O)CC1CC1CC C1(CC=C)(NC(=O)CCCn2cccc2)CCN(C(=O)C(O)CCSC)C1 c1(C(N(C)CC2(NC(C(C(C)O)C)=O)CC2)=O)c(F)cncc1Br C1(OCC)CC(NC(=O)Nc2ccnn2CCO)C12CCCCC2 C(=O)(CCC(C)(C)C(=O)N1CC(NC(=O)CC(C)(C(F)F)N(C)C)C(C)C1)OC Cc1coc(C)c1C=CC(=O)NCC1CN(C(c2cnc(Cl)[nH]2)=O)C(C)(C)C1 C1(C(N(CC(CNC(c2nccc(C)c2N)=O)(C)C)C)=O)CCn2nnnc2C1 C1(CC(=O)OCC2N(C(C34CC(C3)C4)=O)CC2)SC(=Nc2ccccc2)NC1=O C(C(O)CCCCCCCCCC)N(C(c1ccccc1)CCC)CC Cc1nn(-c2ccccc2)cc1-c1nc(CC2CC2)nn1CC1CCCO1 C12(C(=O)NC(C)Cc3ccccn3)CCCC1CCN2C(C1CCC(=O)O1)=O O=C(C1CCc2c[nH]nc21)NCC1(O)CCCN(C(=O)C2=CCCC2)CC1 C1(C)(CC)CCN(C(=NCCN2CCC(C)CC2)NC(C)COC)C1 N1(c2ccccc2)CCC2(C1)C(=O)OCCSCCCOC2.CCC.C(C)(=O)NC CCC(=O)CCC(=O)NOCC(N1CCCC12CCOC2)=O N1(C(C2(CC#C)CC2)=O)CC(NC(C2CC(O)C2)=O)C(C2CC2)C1 c1(COC)nc(C(C)NC(C2CC2C(C)NC(=O)C(=O)N(C)C)=O)cs1 CC1(C(=O)NCC2CC2NC(=O)CSC2CC2)CCNC1=O CCC(C(=O)N1CCN(C(c2ccccc2N2CCCCC2)=O)CC1)C(C)O C12(CNC(C(C)SC)=O)CCCCC1N(C(c1cc[nH]c1C)=O)CC2 C1(C#N)(C(=O)OC)CCN(C(=O)C(n2cc(C(C)COC(C)C)nn2)C)C1 c1(C(=O)NCC(C)CNC(C2(C)CCCNC2=O)=O)cccc(Cl)c1Cl N1(C(C2(C=C)CC2)=O)CCC(NC(=O)C(C2CCCN(C)C2)(C)C)C(F)C1 c1(C(N2CCN(C(CCOCC)=O)C(CC(F)(F)F)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 Cc1nc(NC(c2ccc(F)cc2Cl)C)cc(N2CCCC(OCC3CC3)C2)n1 C(=O)(C1=NNC(=O)CC1)N(C(C)CNC(=O)Cc1csc(-c2nc[nH]n2)n1)C c1(C(=O)NCC(C2(O)CCN(C(C3CC(O)C3)=O)C2)C)cccnc1N1CCCC1 c1(C(=O)NCCC(C)N(C(=O)C#CC2CCCO2)C)ccc2cnnc(O)c2c1 Cc1cccc(C(N2CC(NC(C3CC(C)(C)C3)=O)C3(CCC3)C2)=O)c1C#N C1(C(=O)NCC(CC)(C)O)CC2(CC2)CN1C(c1ccc(F)c(C(C)C)c1)=O C12(CC)CC1CN(C(c1cc(CNC(=O)C=CCN3CCCC3)on1)=O)C2 C(CC(C)C(=O)NCCN(CC(C)O)C(=O)Cc1cnsc1)=CC c1(CNC)ccc(OCC(=O)NC2CCC2c2ccc(F)cc2)cc1 C12(O)CCN(C1)C(=O)CCCNC(=O)C(=O)NCC2.C=CCCOC(C)(C)C N1(C(C(c2ccc(CC)s2)=O)=O)CCC2CN(C(C3CCCC(=O)N3)=O)CC12 C1(C(=O)NC(C(=O)NC(CCC=C)C)Cc2ccoc2)CC2CC(=O)C1C2 C=C1CC(NC(c2ccnc(F)c2)=O)N(Cc2ccc(N(C)C)s2)C1 CC(C)(C#N)CC(C)(c1nnnn1C1CCCC1)NC1C2COCC12 C1(C(=O)Nc2n(CC)nnn2)C2CC1N(C(C1CC1C)=O)C2.c1(N)ccc(C(F)F)cc1 Cc1nc2cccc(C(=O)N(C3CN(C(=O)C=Cc4ccsc4)C3)C)c2s1 c1(OCC)ccc(Cl)cc1NC(c1cscc1CC)c1nnnn1C1COC1 C(=O)(C1CCCc2nccn21)NC1CC(C)(NC(C(C(C)C)C)=O)C1 N1(C(n2ccc(CCNCC)c2)=O)CCC=C(c2ccco2)C1 N1(C(C(CC)c2ccccc2)=O)CCN(C(=O)C(C)CO)CC1CCO CCC(C)(C)CCNC(=O)CC=CCNC(C1COCC1C(N)=O)=O CCC1=C(C(=O)N2CCCCC(CNC(c3conc3C)=O)C2)SCCO1 C(CCC)(C(C)(C)C)N(C(CS)=O)CC.C=CC(C)C(=O)C(CC(CN)CCN)=O C1(C)(CC)C=C(C(=O)N2CCC(C)C(N(C(=O)CCc3cncc(F)c3)C)C2)C1 CN1CC(C)(C(=O)NC2CCC(NC(=O)CCc3ccc(Cl)s3)CC2)CC1=O Cc1c(C(N2CCCC(NC(c3cnc(C#N)s3)=O)C2)=O)cncc1Br C1(NC(C2CC(=C)C2)=O)CC2CC(NC(C3CC(C(F)(F)F)(OCC)C3)=O)C2C1 C(=O)(CCC(=O)c1ccc(Cl)cc1)N(CC(CN(C(CC(C)C1CC1)=O)C)O)C CCCCCCC(C)NC(=O)CCN(C(=O)C(O)CCC)CCCO c1(CC(C)NC(C(C)C)=O)ccc(CNC(c2scnc2C(C)(C)C)=O)cc1 C1(CNC(C(CN(C)C)(C)O)=O)CN(C(=O)C(C)(C)N(C)C)CC12CCC2 N1(C(C2C(C=C)C2)=O)CCC2(C1)CN(C(C1CC13CCCC3)=O)C2 CC1(NC(=O)C(O)CC(N)=O)CCCCC1C(=O)NCCC(O)CO CCC(C)(C)CCN=c1[nH]c(=NC)[nH]c(=NCCc2cccc(Cl)c2)[nH]1 C=CCCC(C(=O)NCC(C)(C)C1CCCO1)NC(C1CC2(CCC2O)C1)=O N1(C(C2CC=CC2)=O)CCC(C2CCN(C(=O)C3=C(Cl)CCOC3)C2)C1 CC(C)(C)C(O)CNC(C1CC1CNC(=O)CNC(N)=O)=O CCC(C)(CO)C(=O)N1CCC(CCNC(c2cnc(-c3ccccc3)[nH]2)=O)C1 C(=O)(C1Cc2ccccc21)NCC(Cn1cc(C(=O)OC)nn1)OC C(=O)(C1CCCc2cccnc21)NCC1N(C(CCc2nc(C)c(C)[nH]2)=O)CC1 C(C)(C(=O)NCCCCN(C(=O)COC1CCOC1)C)OCC=C c1(NC(CC2N(C(C3N(CCC)CCC3)=O)CC2)=O)cn(C)nc1C#N C12CC(F)CN(C1)C(C(C)C)CNC(=O)N2.c1ccc(Cl)cc1.OC(F)F C(=O)(C(F)CC1CCCCC1)N(CC(C)NC(=O)CCNC(=O)C1CC1)CC C1(CNC(C2CCCC(F)C2)=O)C2CN(C(c3ccc(Cl)s3)=O)CC12 C1(CCC(=O)O)CCCCCN1C(=O)C(c1nc(Cl)sc1Cl)F C1(CNC(C2CC(CC)C2)=O)CC(F)(F)CN1C(c1cc(OC)no1)=O c1(C(=O)NCC2(NC(C3CCC(CC)O3)=O)CC2)c(Cl)cccc1[N+](=O)[O-] N#CCCCC(=O)N1CCC(N2CCC(n3cc(COC(=N)O)nn3)C2=O)CC1 C1(O)(CNC(C2C(COC)C2)=O)CCN(C(=O)C(C)(C)C#N)C1 c1(C(=O)NC2(CC)CN(C(=O)CC(C)N(C)C)C2)ccc(C(C)C)c(C)c1 Cn1nnc(C(=O)NC2COCCC2NC(c2csnc2Cl)=O)c1N C1(C(N(CCCO)CC#C)=O)OCCC1NC(=O)CN(C)CCOC.OC CCCCCC(O)CC(=O)N1CCN(C)C(CNC(c2occ(C)c2C)=O)C1 C1(C(N(CCCNC(C2CCCC23CCC3)=O)CCO)=O)CC2(CCO1)CC2 N1(C(=O)CNc2cnc3cc(F)c(F)cc3n2)CCC2(CCOCC2CO)CC1 N1(C(c2cccc(CC)c2)=O)CCC(C)(C)C1CNC(c1cnc(CC)o1)=O c1(CC)ccnc(C(=O)N(CCCNC(c2cnn(C)c2COC)=O)C(C)C)c1 N1(C(C(C=C)C)=O)CCN(CC(=O)NCCn2cc(CO)nn2)C(=O)C1 C1(CCOC)(NC(c2c(C)csc2Cl)=O)CCN(C(c2nc(O)c(C)s2)=O)C1 c1(C(=O)OCC)cc(C(=O)N(CCCNC(=O)COCC)CC=CCSC)on1 Cc1nn(C)c(Cl)c1C(=O)NCCC1CCCN(c2ccnc(C3CC3)n2)C1 c1(OC)ccc(OCC(O)CNC(=O)CSCC2CCCC(C)C2)cc1 CC1OCCC1C(=O)NC(Cc1ccoc1)C(=O)NC(CC1CCCC1)CO c1(C(N2C(CCNC(C(CCC)CCC)=O)CCC2)=O)nccn2nc(C)cc12 c1(NC(C2C(C(N3CC(NC(COC)=O)C3)=O)C2)=O)onc(C)c1SCCO c1(C(=O)NC2CC(NC(c3cnc(OCC4CC4)s3)=O)C2)ccc2c(n1)NCC2 C12(C(N3C(CF)CC(OC)C3)=O)CCC(CC1NC(c1cn(C)c(=O)n1C)=O)C2 N#Cc1cc(F)c(C(N2CCSC(C(=O)NCC3CCC(O)CC3)C2)=O)c(Cl)c1 CCCCC(O)C(=O)NCCC1CN(C(=O)Cn2ccc(Br)cc2=O)C1 CCC1=NOC(C(=O)NC(C)CN(C(c2cnn(C(C)C)c2)=O)CC)C1 n1(CC(=O)NCC(CO)NC(c2nnc(C3CC3)s2)=O)nnc(=O)[nH]1 n1(CC=C)ncc2c(O)nc(=NCC3(C)CCN(C(=O)C=CBr)C3)[nH]c12 C1(C(N2CCCC(NC(C(CC)CC)=O)C2)=O)CC(F)(F)CN1C(=O)C1CC1 N1(C(COCC)=O)CC(C(=O)NCc2cocn2)C(C2CC2)C1 c1(C(=O)NC(C)C(C)(C)NC(C2CCC(=O)O2)=O)ncnc2c1OCCO2 c1(OC)ncc(C(N2C(C(=O)NCCn3cc(C)cn3)CC3CC23)=O)cn1 C12(NC(c3c(C)nc(C)[nH]3)=O)CCC1CN(C(=O)CN1CCC(C)(O)C1)C2 c1(NC(N2C(c3onc(-c4c(OC)cccc4)n3)CCC2)=O)c(F)cccc1Cl c1(C(N(C)CC2CCCN2C(c2cnccn2)=O)=O)cccc(NS(C)(=O)=O)c1 N1(C(CC(=O)NC)=O)CCCC(N2CCC2)C1 O=C1COC(c2ccc(NC3CC4CCCC(C3)C4N)cc2)=NN1 C1(NC(C2CCCC(C(C)C)C2)=O)CCC(P(C)(C)=O)C1 CCC(CC)CCCC(=O)NC(CCC1CC1)C(=O)N(CC(C)C#N)C C(=O)(CCCCCCCC1CC1)NC(CCCNC(C1(CC)CCCC1)=O)C c1(-n2c(Cc3cc(C)no3)nc(-c3ccn(C)n3)n2)ccc(F)cc1C C(CC(C)C)(C(=O)N1CC(OC)CC1CNC(c1nnc(Cl)cc1N)=O)OC N1(C(C2CCC(NC(C(C)OC(C)=O)=O)C2)=O)CCc2ncncc2C1 c1(CN(C2C(CNC(N(c3sccc3C)CCC)=O)CCC2)C)ccccc1 Cc1cc(=NCCC2CC(OC(C)(C)C)C2)[nH]c(=NCC2CSC2)[nH]1 c1(OC)cc[n+]([O-])c(C(=O)NC2CC(N(C)C(C3CCCCC(=O)N3)=O)C2)c1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCCCOCCNC(CCS(C)(=O)=O)=O CCC(CC)CCC(=O)NCC(C)C(F)C(=O)N(CCOC)CCOC N1(C(Cc2c(C)nc(S)s2)=O)CCCC(C)C1CNC(c1coc(C(N)=O)c1)=O CC1(C)CN(c2cc(=O)c(C#N)c[nH]2)CCC1NC(=O)CC1CC=CCC1 CC(CN(C)C)CC(=O)N1CCC(C(F)CNC(=O)Cc2cnn(C)c2)CC1 c1(CN=[N+]=[N-])ccc(C=NOC2CCOC(C(F)(F)F)C2)cc1F CC1Oc2ccc(C(=O)NC3CCCN(C(=O)CCc4ncc[nH]4)C3)cc2C1C C1(NC(Cc2c(OC)ccc(Br)c2)=O)CCCC2CN(C(C3CCCO3)=O)CC12 N1(C(C(C(C)O)N(C)C)=O)CCCC(N(C)C(c2cc(C3CCC3)[nH]n2)=O)CC1 N1(C(c2cccc(CSCC#C)c2)=O)CCC(NC(=O)Cc2cscn2)C(C)C1 C1(C(=O)NCc2c(C(=O)NCC3CCC(C)C3)c[nH]n2)CC2(CC(=O)C2)C1 [N-]=[N+]=NC1CCN(C(=O)C(=O)Nc2ccc(OCC(N)=O)cc2)CC1F Cc1cnc(C(=O)NCCCC2(NC(C3CCOC3C(F)(F)F)=O)CC2)c(C)c1 c1(C(=O)NCCN(C(CC(C)C2CC2)=O)C2CCCC2)cc2ncccc2o1 c1(C(=O)NCC2CC(O)CN2C(C2CCCC2)=O)ccn2ncnc2c1 c1(NC(C(CC)Oc2cccc(F)c2F)=O)nc2c(s1)CC1(CCCCC1)CC2 C1(NC(CN2C(C)CCC2)=O)CN(C(=O)CCc2cc(Cl)sc2Cl)CCC1F C1(C(=O)NCCC(C(=O)OC)O)C2CC3C(C2NC(=O)Cc2cn[nH]c2)C13 N1(C(C2=CC(C)(CC)C2)=O)CC2(CCN(C(c3nnn(C(C)C)c3C)=O)CC2)C1 C1(C(=O)NC(C=C)CO)C(C2CC2)CCN1C(c1ccc(OC)nc1)=O c1(C(N(C)CC2CCN(C(=O)COCC(C)(C)C)C2)=O)cnc(N)cn1 c1(C(N(CCC(C)NC(CCCCCC)=O)C)=O)cccc2sncc12 CC(C)CC(F)C(=O)N(CCCOCCN(C)C(c1c[nH]c(=O)cn1)=O)C Cc1oc(N)c(C(N2CC(OCCNC(c3ccnc(S)c3)=O)C2)=O)c1C N1(C(C(CCNC(=O)C=Cc2ccoc2)OC)=O)CCC2(CCC2)CC1 C=CCC(CC=C)C(=O)NC(C)C=CC(=O)NCC#CCCC CCC(C)C(C(=O)N1CC(NC(C2CC2c2ccccc2Cl)=O)C(C)C1)N(C)C C1(COC)CC(CNC(c2c[nH]c(=N)s2)=O)N(C(=O)C(C)n2cccn2)C1 CC(CCCNC(C12COCC1C2)=O)NC(=O)CSS(C)(=O)=O N1(C(COCC#C)=O)CCC(NC(=O)CCCC2CC2C)C1 C1(C(=O)NC(C)C(C)(C)NC(C2CCCC2)=O)Cc2ccc(Br)cc2C(=O)O1 c1(CC)c(C(=O)NCC2CC2NC(c2ccoc2C)=O)cnn1-c1ccc(C)cc1 CCC(CC(=O)NCCC(C)NC(C1(C)CCCO1)=O)C1CCC1 C(=O)(N=c1cc[nH]c2ccc(Br)cc12)C1N(Cc2cc(C#N)c(Br)cc2)CC1 C(C(C)(C)CNC(=O)CN(C)S(N)(=O)=O)NC(C(c1ccccc1)OCC)=O CCCCC(=O)NCC1CCC1C(=O)NC(CCC)c1ccco1 C(=O)(C1CCCc2cncn21)NC(CCCNC(c1c(C)cncc1)=O)C C1(C(C)NC(=O)CCC2CCC2)CCN(C(=O)CC(C)C2CCCCC2)CC1 c1(CCC(=O)NCC=C)cn(CC2CCC(C(=O)O)C2)nn1 Cc1ccnnc1C(=O)NC(C)C(C)NC(=O)C(c1ccccc1)N1CCCC1 CN1CCCCC1CCC(=O)NC1CCOCC1NC(c1cnsn1)=O C1(C)(C)CCC(C2CC(F)(C(c3ccccn3)N(C3CC3)OC(C)(C)C)C2)O1.CO C1(NC(Cc2cc(OC)ncc2)=O)CN(C(c2ccc(C)s2)=O)CCC12CCC2 c1(CNC(C(C2CC(NC(c3cnc(CC)s3)=O)C2)F)=O)[nH]c(C)nc1C Cc1c(NCCCOC2CCCCCC2)ncnc1NCC1CC(C)OC(C)C1 c1(SCC)nccnc1C(N1CCC(O)(C(C)NC(C23CC(C)(C2)C3)=O)C1)=O C1(NC(C2CC(C#C)(O)C2)=O)CN(C(c2ccc(OC)nc2OC)=O)CC1(C)C c1(C(N(C2CCN(C(C3CC(C#C)(O)C3)=O)CC2)C)=O)cc(F)c(O)c(F)c1 CCCC(CCC)CC(=O)N1CCOCC1CCNC(c1c[nH]cc(F)c1=O)=O Cc1nsc(N)c1C(=O)NC1CCCC(NC(=O)COCCOCCO)C1 c1(C(=O)NC(CNC(C(C)SC)=O)(C)C2CC2)ccc2nc(C(C)(C)C)[nH]c2c1 CCC(CCC(=O)NC(CNC(c1ccc(C2CCCC2)cc1)=O)C(C)C)OC C(CCC)(C(=O)N1CCC(NCC2CC(O)C(O)C2)C1)=CCC CC1CN(C(=O)C(C2CCCO2)NC(c2cn(C)nn2)=O)CC1N(C)C C1(NC(C)=O)CCN(Cc2cn(CCc3csc(-c4ccco4)n3)nn2)CC1 c1(CC(=O)N(CC(C)NC(C2ON=C(CC)C2)=O)CC)csc2ccc(C)cc12 C1(C(=O)NCC2C(NC(C(C(C)C)F)=O)CCCC2)CCC2CC(C)CN2C1 c1(C(=O)NC(C)C=CC(=O)NC2CC(C(N)=O)C2)ccc(N)c(F)n1 c1(CC)cc(C(=O)N(CC(C)(C)NC(C2CC(SC)C2)=O)C)cc(O)n1 c1(C(=O)NC(C2CN(C(C3(C)CC3C)=O)C2)C)cn2cc(Cl)cnc2n1 c1(NC(CC2CC(=O)OC2)=O)nc2c(s1)CC(C(=O)O)CC2 Cc1ccc2cc(C(=O)NCC3CC3CNC(c3[nH]c(O)nc3C)=O)[nH]c2c1 CC(C)CCC(=O)NCCCCCNC(c1cnn(C)c1Br)=O C1(C(=O)Nc2ncc(CC3(C=C)CCCCC3)s2)CC2(CCCCC2)C1 C(=O)(CCCCCCSC)N(CC(C(=O)NCCN(C(CC)C)C)C)C C1(OC)CN(C(=O)C=CC=Cc2ccccc2)CC1NC(=O)C(C)(F)F Cc1c(C(N2CC3C(CNC(=O)CC4CCOC4=O)C3C2)=O)cccc1N N1(C(CN(CC)CC)=O)CCOC(C(C)NC(c2cc(C#N)on2)=O)C1 C(=O)(C(C(C)C)Sc1cccs1)NC1(CCNC(c2c(C)cco2)=O)CC1 N1CCCC(F)C1.C#CC1(CNC(=O)CN(C(=O)C(C)C)C)CCCC1 c1(C(N(C)CCOCCCNC(c2cnc(S)nc2)=O)=O)cc(F)cc(N)c1F Cc1ccnc(C(=O)NCC2(F)CCCN(C(C3(C)CCCS3)=O)C2)c1F C(=O)(C#CC1CCCCC1)N1CCC(CC=C)(NC(=O)CCC2CCCO2)CC1 C#CCCCCCC(=O)NC.C1(C(=O)OC)CC2COCC2N1C(=O)CCCNCC N1(C(c2cc(C)c(Br)s2)=O)CCc2c(ccc(Cl)c2F)C1 c1(OCCOC)ccc(-c2nc(C(C)C(C)O)n(-c3ccc(SC)cc3)n2)cc1 N1(C(c2c(NC(=O)Cc3ccccc3F)cccn2)=O)CCCC12CCCC2 C1(NC(c2ccc(I)cc2O)=O)CN(C(c2ccc(Br)c(F)c2)=O)CC1(F)F C=CC(C)(C)CCNC(=O)C(C)(CSC)NC(=O)C=C1CCC1 Cc1ccc(CCNC(=O)NC(CCO)C(C)C)cc1O Cc1noc(C(F)F)c1C(=O)NC1CCCN(C(=O)CC2CCCN2C)C1 c1(C(N2CC3(CN(C(C4CC4C4CCCC4)=O)C3)C2)=O)sc2sccc2c1Cl c1(NC)cc(F)ccc1NC(C1CCN(OCc2ccccc2)CC1)=O c1(C(N(CCCCNC(Cc2c(C)occ2)=O)C)=O)cc(C)c(Cl)s1.C1C(=O)N1 Cc1nn(CC(N2CC=CC(NC(C3CCC(F)CC3)=O)C2)=O)cc1Cl C(=O)(C(C)(O)COC)N1CC(CC(=O)NCc2sccc2Cl)(OC)C1 C(N=c1ccnc(NC2CCCC2CO)[nH]1)c1ccc(NC(C)C)cc1 C1(C(N(CC(COC)C)C)=O)(OC)CCN(C(=O)CC2(C#N)CC2)C1 c1(OC)ccc(C(=O)NCCOCCn2cc(-c3n[nH]c4c3CCC4)nn2)c(O)c1 c1(OCC)ncc(C(=O)NC2(CNC(=O)CCc3cc[nH]n3)CCCC2)cn1 C(C)(N=c1[nH]c2cc(F)ccc2o1)C1N(C(CC(=O)NC)=O)CCCC1 C(=O)(C(CCC)S(N)(=O)=O)NCCC(=C)CNC(C1CCC(C)(C)C1)=O N1(C(C(COC)OC)=O)CCCCC1CNC(=O)CCCCN(C)C C(CC(=O)C1=C(c2ccccc2)OCCC1)N(C)Cc1ccc(C#N)cc1O C#Cc1ccc(C)c(NC(C2C(C)CCN2C(C2CC3(CCC3)C2)=O)=O)c1 c1(C(CNS(N(CCCOC)C(C)C)(=O)=O)O)cc(F)c(F)c(F)c1 Cc1nc2cccc(C(N3CCCC3C(C)NC(C3COCCO3)=O)=O)c2[nH]1 N1(C(CCC=CCC=C)=O)CC(NC(=O)CCc2cnc[nH]2)C2CCCC12 N1(C(C=C=C(C)C)=O)CC2(CCC2)CC1CNC(=O)CCCn1ccnc1C N1(C(Cc2c(C)c[nH]n2)=O)CCN(C(=O)C(=O)c2cccs2)CC(O)C1 C#Cc1ccc(C)c(NC(=O)C(CCOC)NC(=O)C(CC=C)OC)c1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C(N2CC(C3(C)N=N3)C2)=O)CC1(C)C N1(C(C23CC(OC)C2C3)=O)C2CCC1CN(C(=O)Cc1cc(Cl)cnc1C)C2 Cc1cnc(C=CC(N2CC(CNC(=O)C=C3CCC(C)C3)C2)=O)[nH]1 Cc1c(C(=O)NCCCNC(=O)C(C)CC(N)=O)sc2[nH]cnc(=S)c12 C1(C(=O)NCC(CNC(c2c(CCC)[nH]cc2)=O)CO)C2CC3C(C2)C13 CCC(C)C(C)C(=O)NC(C)CCNC(=O)CC1(O)CCCC1 c1(C(CC2CC2)N(C)C(C2C(F)(F)C23CC3)=O)cccc(F)c1F Cc1cc(C(N2CC(c3ocnc3CNC(c3[nH]cnc3C)=O)C2)=O)c(C)o1 CC1(C)CN(C(=O)CCC2CCCCN2C(=O)C#CC2CCC2)CCS1 c1(C(=O)NC2CC(CNC(C3(CC#C)CCOC3)=O)C2)cccc(N(C)C)c1 c1(C(C(=O)NC2C(CNC(C(C)=C(C)C)=O)C2)(F)F)ccc(C)cc1 N1(C(CNS(N)(=O)=O)=O)CCN(C(=O)Cc2ccns2)C2(CCC2)C1 N#CC1(C(N2CC(CC(F)C(=O)NCC3(C4CCC4)CC3)C2)=O)CC2CC2C1 CC1(CNC(C2(C)CCCO2)=O)CCN(C(C2(C3CCCCO3)CC2)=O)C1 N1(C(CC2CCCN(C)C2)=O)CCC2C1CCN2C(c1cc[n+]([O-])cc1)=O CC1(C)CC(CNC(=O)Cc2c(F)cccc2Cl)N(C(=O)Cc2cnc[nH]2)C1 c1(C(=O)NC2(CO)CN(C(c3ccsc3C(F)F)=O)C2)n[nH]c2c1CCSC2 N(C(=NCCn1cccn1)NCCc1nccs1)CC(n1cncn1)C N1(C(c2c(CC)nc[nH]2)=O)CCCN(C(C2CS(=O)(=O)CC(=O)N2)=O)C(CO)C1 C12(C(N3C4CC(NC(Cc5c(C)cccc5)=O)C(C4)C3)=O)CC(C)(C1)OC2(C)C c1(OCC(=O)OC)ccc(NC(=O)C(C)C2CCCO2)c2ccccc12 C1(=CCNC(C2C3COCC23)=O)CCN(C(=O)C2=CCCS2)CC1 CCS(=O)(=O)C=CC(=O)NCC1CC(NC(C2(C#N)CC2C)=O)C1 CCCC(C#N)C(=O)NCC1CC2(C1)CN(C(c1cn(C)ccc1=O)=O)C2 C(CCC(O)C(=O)Nc1cccc(CC)c1)NC(CCSCCCC)=O c1(CCC)cc(NC(=O)COCC(F)F)ccc1Cl.N12CCCC(C1CC)C2=O N1(Cc2cn(C3C(C(=O)O)C3)nn2)CC(C)CCC1CO.N12CCC(CC1)C2=O c1(C(=O)NCC2CN(C(C3CC3C(F)F)=O)C2)ccc(Br)cc1OC(F)F c1(CN(CC(C)NC(c2cnc(OCC)nc2)=O)C)ccc2ccccc2c1 N1(C(=O)CCc2c(Cl)cncc2Cl)CC2CCCC(C1)N2C(C1CCCO1)=O N1(C(CCOC)=O)CCC(CNC(=O)C(C)CC2CCCC2)C1(C)C c1(C(N2CCCC(C)(CNC(C(CC)(C)CO)=O)C2)=O)cc2c(cn1)OCCC2 C1(NC(C(C(C)C)NC(=O)C#CC(C)(C)C)=O)CC2CCC(C1)C2O N1(C(C23CCC(OC)C2C3)=O)CC2(CC2)CC1C(=O)NC1COCC1SC C#Cc1ccccc1CN1CCC(C(=O)Nc2ccnc(-c3cc[nH]n3)c2)CC1 CCCCCCSCCC(C)(C)F Cc1nc(Oc2[nH]cnc2C#N)ccc1NC(C1CC1C(=O)N(C)C)=O N1(C(=O)OC(C)(C)C)CC2(CCCC(CSc3nc(-c4ccsc4)no3)O2)C1 Cc1cc(C(N2CC(N3CC(NC(c4occc4C)=O)CC3=O)C2)=O)ccc1Cl c1(C(N2CC3C(CNC(=O)CC4CCCO4)(C3)C2)=O)cc(Cl)cc(Cl)c1O C(CN=c1ccnc(N2CCC(C3CCC3)C2)[nH]1)OCC(c1ccccc1)C Cc1cc(NCC(=O)NCCCc2ccncc2Cl)ccc1F N1(C(c2ccnn2CCF)=O)CC2CCC1CN2C(C1CCn2nncc2C1)=O c1(-c2n(CCOCC)nc(CSc3cccc(Cl)c3Cl)n2)cccc2scnc12 CCC(CCC(=O)NC(c1cscn1)CO)NC(c1ccc([N+](=O)[O-])o1)=O c1(C(=O)NC(CC)CNC(c2ccc(OC(C)(C)C)cc2)=O)ccc(F)cc1C N12CC(CC1(C)C)C2=O.C(CCCCCC1CC1)c1n(C(C(=O)OC)C)nnn1 C=CC(C)(O)CC(=O)NCC1CC(NC(=O)CCNS(C)(=O)=O)C1 CC1CC(CNC(C2CCC23CCC3)=O)CCN1C(c1ccco1)=O C1(C(C)NC(=O)C=CC(=O)N(C)C)CN(C(=O)CSC2CCOC2=O)CCO1 c1(C(N2CCC(N(C(=O)Cc3cnccc3Cl)C)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 N1(C(C(CC)c2ccccc2)=O)CC2CCOC2(CNC(=O)CC2CCCC2)C1 CC1CC2(CCN(C(c3ccc(Cl)[nH]3)=O)CC2)CN1C(=O)Cc1cocn1 C1(NC(CC(OCC)OCC)=O)CCCCC12CCN(C(C1CCCCS1)=O)C2 N1(C(CC(CC)(F)F)=O)CC2CCN(C(C3Cc4nc(C)cn4C3)=O)CCC2C1 CCC(O)C(C)C(=O)NCCCCC1CN(C(c2cc(O)ccc2Cl)=O)C1 c1(C(=O)NC(C)CCNC(c2cnn(C)c2F)=O)ccc(N)cc1[N+](=O)[O-] CC(C1COc2ccccc21)NC(=O)C(CN)C1CCOC1 CCCC(CCC)=CC(=O)NCCCC1CCCN1C(c1cnoc1C1CC1)=O N1(C(C(C=CC)O)=O)CCN(C)CC1c1cn(CCCC(=O)OC)nn1 c1(OC)ccc(C(F)(F)C(=O)NCC2CCN(C(c3cc(C)co3)=O)C2)nc1 CCCCCC(O)C(=O)N1CCCC1C(C)NC(c1cccc2ccoc12)=O N1(C(c2nccc(OC)c2)=O)CCOCC(NC(=O)CC23CCCC2C3)C1 c1(C(N(C(c2ccc(C#N)cc2)C(=O)OC)C2CC2)C)ccc2ccccc2c1 c1(C(=O)NC2CC(O)C2)cc2[nH]ccc2cc1-c1cc(CO)ccn1 O=C(CCOCC1CCCO1)NOC1CCCCC1.C1C(=O)O1 CCN=C(NCc1nncn1-c1ccccc1)N1CCC(NC(=O)NC)C1 C1(N(C)C(c2cccc(Cl)c2)=O)CC2CCC(C1)N2C(=O)CCn1cncn1 CCCCC(CNC(C1CC(C)(C)CO1)=O)NC(=O)Cn1cc(CO)nn1 c1(OCC)cccnc1C(=O)N(C)CCN1CCCC1 C1(CC(=O)N(CCCN(C(COCCOCC)=O)C)C)CCCCO1 C(c1ccc(Cl)cc1F)=CC(=O)N(CCNC(C1Cc2nncn2C1)=O)C1CC1 C1(N(C(c2scc(CC)c2)=O)CC)CCCN(C(C2C(C)C2C)=O)CC1 C1(C(=O)NC2CC2CNC(=O)Cc2cncc(F)c2)(OC)CCSCC1 c1(CC(=O)NCC2(NC(C3CCC3n3ccnc3)=O)CCC2)ccoc1 c1(C(=O)NCCC2N(C(C(CO)NC(N)=O)=O)CCCC2)nccc2n[nH]cc12 c1(C(N(C)CC2(CNC(C(CC=C)C)=O)CC2)=O)cc2c(s1)CCC(CC)C2 N1(C(C(C(C)C)(C)O)=O)CCC2(CC1)CN(c1ncc3ccsc3n1)CCO2 c1(CC)n[nH]c(CC)c1CC(=O)N(C1CCN(C(=O)COC2CCCCC2)C1)C c1(C(=O)NCCC2CC(=O)C2)cc([N+](=O)[O-])ccc1Oc1ccccc1 c1(N2CCCC(=CCC)C2)nc(=NCCN(C)C2CC2)[nH]c2cc[nH]c12 N1(CC(c2c(Cl)ccc(OC)c2F)C)C(=O)NC2(CC(CO)C2)C1=O O=S(=O)(c1c[nH]ccc1=NC1CCn2cnnc2C1)N1CC2CC1CO2 C1(NC(C2C(CCOC)C2)=O)CCN(C(c2cnn3c2OCCC3)=O)CC(O)C1 C1(NC(Cc2cccc(C(C)=O)c2)=O)CCN(C(c2ocnc2C)=O)CC1C CC1=C(C(=O)NC2CN(C(C3C(C)C3C)=O)CC2O)CCS1(=O)=O C1(C2CC2)(C(=O)NCc2c(C)cccn2)CN(C(c2cc(=N)[nH][nH]2)=O)C1 Cc1cc(C(=O)NCCNC2CCCC(F)C2)c2c(c1)CCCN2 N1(C(CCCCCOCC)=O)CC(N=c2[nH]ccn3nnnc23)C(C)(C)C1 c1(CC)nc(C)ncc1C(=O)NC1CN(C(=O)CC2CCCO2)CC1(C)C C1(NC(c2cc(C)nc(O)c2)=O)CCCOC12CCN(c1nnco1)CC2 CCCC(C)(C)CC(=O)NC1CC(NC(C2(F)CCCN(C)C2)=O)C(O)C1 c1(C(=O)NCC(CC(C)C)NC(C2CCC(C)(C)OC2)=O)cc(Cl)c(Cl)cc1N c1(OC)ccc2c(=NCCC(N)=O)[nH]c(=NC3CC(OC)C3)[nH]c2c1 CCCC(C)(O)C(=O)NCC1CCN(C(c2ncncc2OC)=O)C1 C#CC1(O)CCN(C(C2CCN(C(=O)Cc3sccc3C)C2C)=O)C1 c1(C2(C(=O)NC3CCN(C(C(COC)O)=O)C3)CC2)nn(-c2ccccc2)cc1C C1(C(N(C(C)C(N)=O)C)=O)(CNC(=O)C=CC(F)F)CC12CCC2 Cc1ccc(C(N2CC(F)(F)CC2CNC(C2CCN(C)C2=O)=O)=O)c(N)n1 c1(C(=O)NC(CCCC)CNC(=O)CCC(N)=O)ccc2ccc(O)nc2n1 c1(COC)nnc(CNC(c2csc(Cl)c2)c2nnnn2CCCSC2CC2)o1 CC(C(=O)N1CC(CNC(=O)CCn2cnc([N+](=O)[O-])c2)C1)C(F)(F)C(F)F Cc1nn(C)c(-n2cncn2)c1C(=O)NC(CNC(C1(CO)CC1)=O)CC(C)C C1(C(=O)NCC2C(C)CN(C(=O)Cn3ccnn3)CC2)CCC2CCCCC2C1 c1(C(N2CCC(NC(COCCCC)=O)C(C)C2)=O)c(F)cc(C)cc1Cl C1(CNC(C2(C=C)CCC2)=O)C(C2CC2)CCN1C(=O)C(O)C(C)(C)CC C1(C(=O)OCC(=O)Nc2cc(Br)ccc2F)CC2(CCOC2)C1 Cc1sc2ncn(CCC(=O)NCCC(C)NC(C3C(C)C3C)=O)c(=O)c2c1C c1(C(=O)NC(CCN(C(C(C)OCCC=C)=O)C)C)cc(C(C)C)nc(O)c1 N1(C(C(CCSC)NC(C)=O)=O)CC(NC(c2ccc(F)c(C)n2)=O)C2(CC2)C1 Cc1cc(CN2CCOCC2C(=O)Nc2ccc(Cl)cc2I)cc(C#N)c1 CCCC(C#N)C(=O)N(C)CC1CCCC1NC(C1OCCCC1(C)C)=O c1(C(=O)NC2C(NC(C3(SC)CCC3)=O)CCC2)cc(C#N)ccc1Br C(=O)(C(C)S(C)(=O)=O)N(C(=O)CCCc1cn(C2CCCNC2=O)nn1)CC c1(C(=O)NCCC(CNC(c2cc3ccccn3n2)=O)O)ccc2nc[nH]c2c1 C1(C(N(C)CC2CN(C(C3CC(C)SCC3)=O)C2)=O)CCCC12CCOCC2 Cc1ccoc1C(=O)NC1CCC1NC(=O)C(C1CCC1)C1CCC1 O=CN1CCCC1C(=O)NC(Cc1cc[nH]n1)C(=O)NC1CC(CF)C1 C(CCCC(C)(C)C(=O)NNC(=O)C1CC1F)NC(C1=NN(C)C(=O)CC1)=O N1(C(C2C(CC(C)(C)C)C2)=O)CC2CCC(C1)N2C(C1(C)CSC1)=O Cn1c(C2CCC2C(=O)NCC(O)CNC(=O)CCC2CCCC2)nnc1S CC(C)C(C(=O)NC(CC(=O)OC(C)(C)C)(C)C(F)F)C(=O)Nc1ccccc1 Cc1cc(=O)c(C(=O)NCC23CC(CN2C(C2CC2(C)C(C)C)=O)C3)cn1C c1(OC)nc(C(=O)N(C2CCCCC2NC(c2ccc(F)s2)=O)C)cc(O)n1 c1(COC)nc(CC(=O)NC2CC(CNC(=O)Cc3ccnn3C(C)C)C2)cs1 N1(C(CC2CN(C(C(CC)C)=O)CC2O)=O)CC2CC1CN2CC C1(F)(CNC(C(C2CC(F)(F)C2)OC)=O)CCCN(C(c2ccn(C)c2)=O)C1 C#CC1(C(=O)NCCC2(C)CCN(C(c3ccc(CC)[nH]3)=O)C2)CCCC1 N1(C(C(C)CSC(F)(F)F)=O)CCC(NC(=O)C(=O)Nc2ncc[nH]2)C1C1CC1 c1(CCc2n(CC=C)c(N3CC(OCC)CC(F)C3)nn2)ccc2c(c1)COC2 C1(C(=O)N(C2(CO)CC2)C)(CC)CCCN(C(=O)CCN=[N+]=[N-])C1 c1(CC(=O)N(C2CCC(NC(C=NOC)=O)CC2)C)ccc2ccccc2c1 Cc1ccc(CNC(N2CC3CC2CC3O)=O)c(F)c1F N1(C(c2c(NC)cncc2)=O)CCCN(C(c2ccc(F)cc2F)=O)C(CO)C1 C1(C(=O)NC(CCCC)(C)CO)CCN(C(=O)C(C)C(CC)CC)O1 C1(NC(C2(C#N)CC=CC2)=O)CCCCC1NC(N)=O.C12(CC1)CC(=O)N2C Cc1cn2c(CCC(N3CC4CC4(NC(=O)COC4CCOC4)C3)=O)csc2n1 N1(c2nc(N3CC4CC3CS4=O)cc(C)n2)CC2(CCOCC2)CC1CO N1(C(CC2CCC(C)C2)=O)CCC2(CC1)CN(C(c1cc[nH]c(=N)c1)=O)C2 c1(C(=O)NC(C2N(C(c3cc(C)oc3)=O)CCCC2)C)c(C)nn(C)c1F N1(C(c2c(OC)ccs2)=O)CCC(C2CC2NC(=O)CN2CCCCC2=O)CC1 N1(C(C2C(C)(C)C2)=O)CCC(N(C(=O)Cn2nccn2)CCO)C1 C1(NC(c2ccc(CC)o2)=O)CN(C(=O)Cn2cc(F)ccc2=O)CCC1F C12(C(=O)NC(CNC(c3c(C)cccc3)=O)CO)OCCCC1C2(F)F c1(OC)cc(N)ccc1C(=O)NC1CCC(CNC(C2CC=CCC2)=O)CC1 c1(-c2c(NC(N3CCN(CCF)CC3)=O)cccc2)nccc(C(F)(F)F)n1 c1(C(N(C(C)CCNC(=O)C(F)=CC2CC2)C)=O)ccc(N2CCC2)nc1 c1(C(N2C(C)CNC(=O)C2)=O)cc(O)nc2c1CN(C(C1CC1C(F)F)=O)CC2 Cn1cc(C(N2CCC(Oc3ccccn3)C2)(C2CCCC2)C)cn1 c1(N2CC(CC=C)(NC(c3ccncc3OCC)=O)C2)ccc2nccnc2n1 CC1NC(=O)OC12CN(C(=O)CC(C(F)(F)F)NC(=O)CC(Cl)Cl)C2 c1(C(N(C(CNC(COCCC#C)=O)C2CC2)C)=O)cc(Cl)c(Cl)s1 C1(CC)CC(C(N2CCCNC(=O)C2)=O)CCN1C(C1OC2CCC1C2)=O Cc1c(N)cc(C(N2CC3CC(NC(c4ncn(C)n4)=O)C3C2)=O)cc1N Cc1nn2c(C(=O)NC(c3cccc(Cl)c3Cl)CNC(=O)C(C)C)c(C)nc2s1 c1(C(=O)NCC2(NC(C(C3CCC(=O)N3)C)=O)CC2)ccc(Br)c(O)n1 C(C(CCC)C(=O)N1CC=CC1CN(C)C)NC(C1C(=C)C1)=O c1(C(=O)NC(CN(C(C(Cc2c(C)nc[nH]2)O)=O)C)(C)C)cc(F)cc(Cl)c1N c1(C(=O)NC)cc(Cl)ccc1N(C1CCCN(c2ccccc2)C1)C N1(C(C2(C)CNC(=O)C2)=O)CCC(O)C(NC(c2cccc(C3CC3)c2)=O)C1 N1(CC(=O)N(CC(=O)NC(c2ccco2)CC)CCOC)CC(=O)N(C)C1=O N1(C(C2CN(CC(C)C)C(=O)C2)=O)CCN(C(=O)C(c2cncn2C)O)C(C)C1 C#CC1(C(N2CCCC(CCCO)C2)=O)CCN(C(=O)C=CC2CCOCC2)C1 C1(NC(c2ccc(C#C)cc2)=O)CN(C(C2(NC(N)=O)CC2)=O)CC2(CCC2)C1 Cc1ccc(C(N2CCC(NC(=O)Cc3nonc3C)CC2)=O)nc1 c1(COC)nc(C)cc(=NC2CN(C(=O)CCn3cccnc3=O)CC2C)[nH]1 C1(C(=O)NC2C(C(=O)NCCc3c(C)cncc3)CCCC2)CC2(C1)CC(C)C2 N1(C(c2scc(C)c2)=O)CCOC(CNC(C2CNC(=O)N2C)=O)C1 N1(C(C(CC)=O)=O)CCC2(CC1)CC2C(=O)NCCCc1ccccc1O N1(C(C2(C=C)CCCCC2)=O)CCCCC2(CCN(C(=O)C(O)C3CCC3)C2)C1 C(C(CO)(CO)NC(=O)C(C1CC1)OCC)N(C(CCCOCC)=O)C N1(C(C(C)SCC)=O)CC2(C1)C(NC(C13CC(C)(CCO1)C3)=O)CCS2(=O)=O C12(C(=O)NC(C3CCN(C(=O)CCc4cncn4C)C3)C)CCCC1C2(F)F N1(C(CCCC(=O)NC(C)C)=O)CCC(NC(c2cn[nH]c2)=O)C(CO)CC1 c1(C(=O)NCC(C)(C)NC(c2cn(CCOC)nc2C)=O)cc(O)nc(O)n1 N1(C(C2(CCOCC)CCC2)=O)CC(NC(=O)C(F)(F)COC)CC(O)C1 CC(O)CCN=c1[nH]c(=NCCn2cc(Br)nn2)[nH]c2c1SCC2 C12(C(=O)NCC(CNC(c3cncc4nc[nH]c34)=O)O)C(=O)C3CCC1C2C3 N1(C(C=C(C)c2ccsc2)=O)CCC(NC(=O)CCc2cnoc2)C12CC2 C(=O)(CCC(C)(F)F)N1CCC(C(N(CC(C)C)C)=O)(CF)C1 c1(CN(CCOC)CCNC(C2CCC(C)O2)=O)cnn2c1CCCC2 n1(CC)nc(C)cc1C(=O)OC(c1nc(-c2ccccc2C)no1)COC N1(C(C2C(COC)C2)=O)CCN(C(c2cccc(C)c2Cl)=O)C(c2cn[nH]c2)C1 c1(C(=O)NC(C2CCCC2)CNC(c2cc(Cl)on2)=O)sccc1C1CC1 C1(F)(C(=O)NCC2(OC)CCC2)CCCN(C(C2(C)CCCCO2)=O)C1 c1(-c2cn(CC3CCN(C(CC4N(CC)CCC4)=O)C3)nn2)cc(Cl)ccc1F c1(C(C(=O)NCC2(C)CCN(C(CC3CC(C)C3)=O)C2)C)ccc2c(c1)OCO2 C(=O)(CC1=CCOCC1)N(C)CC1(CNC(c2ccn(C3CCC3)n2)=O)CC1 C(=O)(CCCCC(C)(C)C)N1CC(C)(CNC(CC(C=C)C)=O)CC1(C)C CC1CCN(C(=O)CCN=[N+]=[N-])C(C)C1NS(=O)(=O)Cc1nnc(-c2ccccc2)o1 N1(C(C=CCCC)=O)CC(NC(=O)Cc2cnn(C)c2)CC12CCCC2 CCCC(O)C(=O)NCC(C1CCCC1)NC(=O)CCC(C)O c1(CC)nc(C(N2CC=CC2CNC(C2CCN(C)C2)=O)=O)c2ccccn12 c1(OC)cc(I)c(Cl)cc1COC(C1(c2ccc(C(F)(F)F)cc2)CCC1)=O N1(C(c2c(C)cc(Br)cc2)=O)CCc2c(C(N3CCCCC3C)=O)cccc2C1 c12ccc(cc1)S(=O)(=O)NC(=O)C2C.c1(C(=O)OC)cc(C(=O)O)c(Br)c(C)c1 Cc1cc(=NC(=O)C2CC(C)CN2C(c2cccc(Br)n2)=O)[nH]c(C)c1C#N N1(C(C(C)N2CCCC2)=O)CC=C(CC(=O)N2CCC(C)C(CO)C2)CC1 C12(CNC(=O)C3=CCCC3)CCC(Nc3ncc(O)cn3)(CC1)CO2 c1(OC)ccc(-n2nnnc2C2(NC(C)CCSC)CCSC2)c(C)c1 C1(CCNC(CC(C=C)C)=O)CN(C(=O)CC2CCCCCCC2)CCCO1 N1(C(=O)NCC(C)(C2CC2)NC(=O)OC(C)(C)C)C2CCC(C2)C1c1ccccc1 c1(CN2CC(C(=O)Nc3cc(OC)cc(C)c3)C(O)CC2)cc(Cl)c(O)cc1F c1(C(CC)N(C)C)cn(CC2CC2)nn1.C1CCCN1C(C1C=CCS1)=O Cc1ccc2c(=NCCc3cccnc3C)[nH]c(=NC(C)C3CCC3)[nH]c2c1 CC(c1ccccc1F)=CC(=O)NCCCCNC(c1cccnc1N)=O N1(C(C2N(C)CC2)=O)C2CCC(C2)C1CC(=O)NCCC(O)CO c1(OCC)cc(-c2nc(-c3cncs3)nn2C2CCS(=O)(=O)CC2)oc(=O)c1Br CN1CC2OCCN(C(=O)CCCNC(c3ncn4ccccc34)=O)C2C1 c1(C(=O)NC(CNC(C2(C=C)CC2)=O)CCOC)c(OC)ccc(Cl)c1C C1(NC(C(COC)C)=O)CCN(C2CCN(C(c3cscc3F)=O)CC2)CC1 CC1=C(C(=O)NC2CCN(C(C3CCCN3C)=O)C2)CCC1 N1(C(C)=O)CCCC1C(=O)NC1(C2CCCN2C(=O)C=CC(C)(C)C)CC1 C(=O)(C1=CCC(C)CC1)NCC(C(C)C)NC(c1cnc(C(C)OCC)s1)=O c1(C(C)C)c(NC(C2(NC(=O)C(C)N3CCCC3)CCCC2)=O)cnn1C CCCCCC(CC)C(=O)N1CCCCC(NC(=O)CCc2c(C)n[nH]c2C)C1 C=CC(CC)C(=O)NCC(CC1CCCC1)C(=O)N(C)CCC1CCOCC1 C(C1=CCN(C(=O)CCC2(C)CC2)CC1)NC(C(c1ccccc1)NC(C)=O)=O N1(C(c2cn(CCOC)nc2)=O)CCOCC1CCNC(C1CCCC1(F)F)=O Cc1cnc(C=CC(=O)NC2COCC2CNC(=O)CC2CSCCS2)[nH]1 CC(C)CC(C(=O)N1CCC(C)(F)CC1)NC(c1ccc(C(N)=O)o1)=O c1(C(N2CCC(C(N(CCCC(=O)OC)C)=O)CC2C)=O)cccn2nccc12 N1(C(c2n(CC)nnc2)=O)CCCC(C)(NC(=O)CCc2cnco2)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCN(C(c2cncc(OC)n2)=O)C(C2CC2)C1 c1(CC(=O)NC(C)C(C)NC(c2conc2C(C)(C)C)=O)cn2ccccc2n1 N1(C(C2C(CC)OCC2)=O)CCCC2(CCN(C(c3n[nH]c(C)c3F)=O)C2)C1 C(CC(C)C)(C(=O)NCC1CC(O)CN1C(c1ccccc1Cl)=O)OC C(c1c(F)ccc(Cl)c1F)=CC(=O)NC1C(NC(C(C)c2cccs2)=O)CC1 Cc1nn(C)c2c(NCc3ccc(Cl)nc3)nc(=NCCCOC(C)(C)C)[nH]c12 c1(C(=O)NCCN(C2CCCCC2)C(=O)C2CC2)cccc2c1NCCC2 N1(C(C(F)OC)=O)CCC(CNC(c2ccccc2O)=O)C12CC2 N1(C(C(C)Cc2ccnn2C)=O)CCSCC1CCNC(c1cnsc1)=O C(=O)(C(C)(C)CCC#N)N1CC(CCNC(C=CC(CC)C)=O)OCC1 C1(CCN(C(=O)CSC(F)F)C)CCCCN1C(c1cc[nH]n1)=O C(CCO)(CC(C)C)NC(C1(NC(c2c(OC)nn(C)c2)=O)CC(O)C1)=O C1(C2CCCN(C(=O)CSc3cccs3)C2)(NC(C(CC)C(C)O)=O)CC1 CCC(O)C(C)(C)C(=O)NCCCC1CCN(C(=O)CN2CC(=O)NC2=O)CC1 C1(NC(C(C)c2ncco2)=O)CCCC1NC(=O)C=Cc1ccco1 N1(C(CNC(C2C(C)C2)=O)=O)CC=CC(NC(c2ccc(CC(N)=O)cc2)=O)C1 C1(C(N(C(C(=O)OCC)C)C)=O)CC2CC2N1C(=O)CCOCC(C)C c1(C(N2C(CNC(C(C(C)C)OCC)=O)CCCC2)=O)cc(=O)n2ccsc2n1 C1(C(=O)NCC2(NC(=O)CCN3CCOCC3)CCOC2)(OC)CCCOC1 c1(-c2cccc(SCCCC)c2)ccc(C(=O)NC2CC(C)(COC)C2)nc1C C(C)(CCCC(=O)N1CC(C)(O)CO1)NC(C(CC)CCOC)=O N1(C(=O)OC(C)(C)C)CCCC(CC(=O)NCC(C(F)(F)F)n2cccn2)CC1 C(=O)(CCC(C)CN(C)C)N(C(C)CC(=O)NCC1CC2(CC2)CO1)C c1(CNC(C2CSC3(CNC3)C2)=O)cn2c(Br)cccc2n1 N1(C(c2n(COC)ncc2)=O)CCCCC1CNC(=O)C(C)c1ccsn1 C1(CC(N2CC=CC(NC(=O)Cc3cnn(C)c3)C2)=O)(OC)CCCCC1 c1(CNC(=NCC)NCc2cnn(CC(C)C)c2)cn2cc(Cl)cc(Cl)c2n1 c1(C(=O)NCC2(F)CC(NC(C(CSC)C)=O)C2)ccc2ncnc(O)c2c1 C(CCC(N)=O)(C(=O)NCc1cc(F)c(Br)cc1O)n1cc(CCC(C)O)nn1 c1(C(=O)NC(C2(C(=O)NC(C#C)C(C)OC)CC2)C)nc(C)c(C)s1 c1(C(=O)NCC(CCCC)NC(C2(C)COCCO2)=O)cncc([N+](=O)[O-])c1 c1(CC)cn2c(n1)CCC(C(=O)NCC1(NC(C3CCCC(=O)O3)=O)CC1)C2 c1(C(C(=O)NCC(=C)C)N(c2ccccc2)CCCO)cncc2ccccc12 c1(C(=O)NC2C(OC)CN(C(c3ccc(C#N)o3)=O)C2)cc(F)c(F)cc1Cl N1(C(C2CCC(=O)N2)=O)CC2CCCC1C2CNC(C1CCC(F)C1)=O n1(CC(C)C)ccc(=NC(c2csc(Cl)c2)c2nnnn2CC2CCOC2)[nH]1 Cn1ccc2ccnc(C(=O)NCC3CCCN(C(C4(C)CC=CC4)=O)C3)c12 N1(C(c2ccc(OCC)cc2)=O)CCN(C(=O)CNC(C)=O)C2CCCCC12 N1(C(c2c(C)snn2)=O)CC(CC(=O)N2CC2CN(C)C)C2(CC2)C1 N1(CC)CCOC(C(=O)NCC=CCNC(=O)CCn2cccc2)C1 C(CNC(C1CCN(c2ccccc2F)C1)=O)(C(F)(F)F)OC C1(F)(CNC(C2CCSC2)=O)CN(C(=O)CCc2nc(-c3ccccc3)no2)C1 c1(CNC2CC(NC(=O)Nc3c(C)cccc3C(N)=O)C2)c(Br)cc(F)cc1Br CC1CN(C(=O)CSc2nncn2C)CC(C)C1NC(c1ccn(CC#N)n1)=O C1(NC(c2scnc2C2CC2)=O)CCOCC1NC(c1ncccc1F)=O c1(C(=O)NCC(C)(O)CNC(=O)C=CC(=O)N(C)C)ccc(Cl)c([N+](=O)[O-])c1 C1(CC(=O)NC(CC)CN(C)C(C2(N(C)C)CCCC2)=O)CCCC12CC2 Cc1ccc2ncc(C(N3CCCOC(CN=c4[nH]cncc4I)C3)=O)n2c1 c1(CC(=O)NCCCOCCNC(C2COC(=O)O2)=O)ccsc1Br C12(NC(COCCC=C)=O)CCC(CC1)N(C(c1cc(F)cc(C)c1N)=O)C2 c1(CC)c(NC(=O)NC2(CC3CCC3)CCCC2)cnn1CCO C1(C(=O)NCCN(C(=O)CC2C=CCCC2)C)Cc2ccccc2O1 C1(NC(C2(n3cccc3)CC2)=O)COCC1NC(C1CCC1)=O c1(C(=O)NC(C2(CNC(C3CC3(C)C)=O)CC2)C)cnc(C(F)(F)F)s1 c1(CC(C)NCC(C2CCC3(CC2)CC3)=O)nc2ccccc2s1 N(C(=NCCSC1CCOCC1)NCC1(C#N)CC1)C(CC)C C(=O)(C1=C(CC)OCCC1)NC(CCC)C(O)C(=O)NC1CCC(C(C)O)CC1 c1(C(N2CCC(C(C)(C)OC)C2)=O)[nH]c(Cl)c(Cl)c1Br C1(NC(C(C)(C)CF)=O)COC2(CCN(C(=O)CCc3cccnc3)CC2)C1 Cc1nc(S)sc1CC(=O)NC(C)CNC(=O)CCNC(=O)C=Cc1ccoc1 c1(C(N2CC(C)N(C(=O)C(=Cc3cccn3C)F)CC2)=O)cnc2cc[nH]c2c1 C1(C(N2CC(NC(CCc3ccc(C)s3)=O)C(O)C2)=O)CC12CCCCCC2 C1(NC(CNC(CNC(C=C(C)C(C)C)=O)=O)=O)CN(C)C2(CCC2)C1 c1(C(N2C(C(=O)Nc3c(C)cc(F)nc3)C3CCC2C3)=O)cc2cccnc2[nH]1 c1(NC(=O)C(C)(O)C2CC2)ccc(Cl)cc1.C(=O)(C(C)O)N(CC(=O)OC)C n1(CCCCC)nc(-c2ccnn2C)nc1CCc1cncnc1 C1(NC(C2CN(C(C)C)C2)=O)C2CCC1N(C(=O)C(c1ccc(F)cc1)(F)F)C2 c1(CC(C(=O)OC)NC(CCOC)C(C)C)csc2nccn12 C12(CNC(C3(OC)CCC3)=O)CCCN(C(=O)CCOCC(C)C)C1C2 N(C1CCCc2c[nH]nc21)C(CC1(NC(C(CC=CC)CC)=O)CCC1)=O C1(NC(C(C)NC(CC)=O)=O)CN(C(c2cc3ncccc3s2)=O)CC12CCC2 C=CC1COCCN1C(C12CC1CCN2C(c1cc[nH]c1)=O)=O c1(CN2C(C(=O)NCC3CCN(C(C)=O)CC3)CC2)c(F)ccc(F)c1N N1(C(c2ccn(C)c2)=O)CCCN(C(C2CC3C=CC2C3)=O)CCC1 C1(O)(CNC(c2cc(Br)ncc2Br)=O)CCCN(C(c2cnnc(O)c2)=O)C1 Cc1ccc(CNC(c2cc(CNC(=O)CCOC3CCOC3)cs2)=O)cc1C n1(CCCC(=O)N(CC)CC2CCCN2C(=O)CCCSC)nc(C)cc1C CC1CCC(C2CCC2)CN1C(=O)C(N1CC(C)(Cc2ccccc2)C1)=O C1(C(=O)NC(COC)C(=O)N(C)Cc2nncs2)C2CC3C(C2=O)C13 C(=O)(C(=O)N=S(C)(C)=O)NCC1CCCN(C(C(C)N(C)C)=O)CC1 c1(CN2CCCC(NC(c3cccc(Cl)c3Cl)=O)C2)cc(F)c(Br)cc1[N+](=O)[O-] CCC(C)(C)C(=O)N1CC(NC(=O)CCc2ncc[nH]2)C(c2cncn2C)C1 c1(N2CC(C(N(CC(=O)NCc3ccccc3)C3CC3)=O)C2)cc(F)cc(F)c1 CC1C(C(=O)OC(C2CC2(Cl)C(=O)O)=O)CCN1.c1ccccc1 C(=O)(C(C)CCCC(C)=O)NCC1N(C(CC(C)SC)=O)CC1 c1(CCNC(c2cc(OC)ncc2-c2ccn(C)n2)=O)cc(F)c2cc[nH]c2c1 c1(C(N2CC(C(C)NC(c3cnc(N(C)C)cn3)=O)OCC2)=O)nc(Cl)ccc1Cl CC(F)(F)CCC(=O)NCCCOCCNC(c1ncnn1C1CCOCC1)=O N1(SCCCOCCCCCC)CCC(=O)N(CCc2csnn2)C1=O c1(C(C)C)ccc(C(=O)NCC2CC(O)CN2C(=O)CC2CCCCC2O)nc1 CCCCC(CCCC)C(=O)NC1CCCC1NC(=O)CSc1n[nH]c(=N)s1 Cc1cc2c(cn1)CN(C(C1CC(=O)C3CC13)=O)C2 N1(C(c2c(O)cccc2Cl)=O)CCCC2C1CCN2Cc1cc(O)cc(F)c1 C1(CC(N2CCC(CC=C)C2)=O)CN(C(=O)C(C2(O)CCCCC2)CC)CCO1 c1(NCC2(C)CC2Br)[nH]c(=NCCN2CCNC2=O)nc2sccc12 C1(NC(c2ccc(OC)c(OC)c2)=O)CC2CC1CN(C(=O)CC1CC(F)C1)C2 N1(C(c2nc(NC(C)=O)sc2)=O)CC(CNC(C2(N(C)C)CCC2)=O)CC1C C(=O)(CS(=O)(=O)Cc1ccc(Cl)s1)NC1CN(C(c2cc(C)no2)=O)CC1O O=C(CCCC(=O)NCCC1CN(C(C2CCCO2)=O)C1)c1ccccc1 C1(NC(C(=O)N(C)Cc2ccc(OC)cc2)=O)CC2(CCCCO2)C1 C1(NC(C(C)SC(C)C)=O)CN(C(c2ccc(CN(C)C)o2)=O)C2CCCCC12 C1(NC(C2CC(C)(C)OCC2)=O)CN(C(=O)CCC(N)=O)CC12CCCC2 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(CNC(=O)CCC(F)F)COCC1 C1(CNc2nccc(C(=O)OC)n2)CN(C(=O)CN2CCC(O)CC2)CCC1C C1(C(F)F)CC(N=c2nc3sccc3c(NC3CC3c3ccc(F)c(Br)c3)[nH]2)C1 c1(NC2(C3CN(C(C4C=CCCC4)=O)C3)CC2)nc(Cl)nc2ccccc12 Cc1cc(C(=O)NC2CCC(NC(=O)CCCOC(C)C)CC2)cnc1O N1(C(=O)CCC2CCN(C(=O)C(F)C3CCC3)C2)CCc2ncccc21 CS(=O)(=O)c1cccc(C(N2CCC(NC(C3CCSC3)=O)C(O)C2)=O)c1 N1(C(c2c(CCC)nns2)=O)CCC2CN(C(c3ccc(OC)nc3)=O)C2C1 C#CCCCC(C)C(=O)NCC(C)N(C(=O)CCCN1C(=O)CN(C)C1=O)C Cc1cc(C(=O)NC(CNC(=O)COCc2nnc(S)n2C)C2CC2)c(C)s1 N1(CCC)C(=O)CCC1C(N1CC(NC(c2cnn(CC)c2CC)=O)C(C)C1)=O CN1CC(C(=O)NCCCC2CCN(C(C3CC(O)(C(F)F)C3)=O)CC2)CC1=O Cc1ccc(F)c(C(=O)NC2CCC(CNC(c3nnc(O)nc3O)=O)CC2)n1 c1(OC)cccn2ncc(C(N3CCN(C(=O)CC(F)(F)F)C4(CC4)C3)=O)c12 C1(C2(O)CN(C(=O)CC(F)(F)C(F)F)C2)(CNC(C23CC(C)(OCC2)C3)=O)CC1 c1(C(=O)NC(CC)CN(C)C(C2CCCCN2C(C)=O)=O)cc(Cl)c(Cl)cc1N CC1CCCC(CCNC(c2ccc(=N)[nH]c2)=O)C1 C1(C(=O)NCC(CNC(C2(C(=O)NC)CCC2)=O)C)CCCCN1C(N)=O N1(C(c2ccc(SC)cc2)=O)CCC2CCN(C(=O)C=CC3CCCN3C)C2C1 C=CCC(C(=O)NC(c1cn(C)nn1)C(N1CCC(N(C)C)C(C)C1)=O)C(C)C C1(CNC(C2(CC)CC=CCC2)=O)C(C)CCCN1C(=O)C(F)CC1CCCC1 N1(C(CC)C)CCCC1C1CCCCN1C(=O)C(C1(OC(C)=O)CCCCC1)C CC1(F)CCC(NC(C2CCC(O)CC2)=O)CC1 C1(NC(=O)CC2(CNC(C3CC=CC3)=O)CC2)CC(Cl)(Cl)C1 c1(NC(C2(SC)CN(C(C3CC4(C3)CC43CC3)=O)C2)=O)cc2cc[nH]c2cn1 C=CCCCCCN=c1[nH]c(=NCC2(CN(C)C)CC=CC2)[nH]c2c1CCCC2 c1(C(=O)NCC2C(C)CN(C(C3CCNC3=O)=O)C2)cc(Br)c(C#N)s1 c1(C(=O)NCC2(F)CC(NC(CS(CC)(=O)=O)=O)C2)cc2ccc(F)cc2o1 c1(CC)oncc1C(=O)NCC1(CNC(c2ccc(C)s2)=O)CC1(F)F N1(C(c2cnc(C)s2)=O)CCOC(CCNC(C2CCCC2(C)C)=O)C1 C12(NC(c3sc4cccnc4c3Cl)=O)CCCCC1CN(C(=O)C=CCO)C2 C(CCCCCS(N)(=O)=O)c1nc(-c2nn(C(c3ccccc3)C)nc2Br)on1 C1(c2n(CC=C)nnn2)(NC(CCOCC)C(C)C)CCOC(C(F)(F)F)C1 C12(C(=O)Nc3cc(C)c(NC(C4CC(CO)CO4)=O)cc3)CCC(CC1)C2(C)C C(=O)(C1=NOC2(CCOC2)C1)N1CCC(NC(c2c(Cl)cccc2[N+](=O)[O-])=O)C1 C1(NC(c2cscn2)=O)CCN(C(c2ccns2)=O)CC1O N1(C(c2c(C)cc(F)cn2)=O)CCC(C(=O)NCC(CO)C2CC2)C(C)(C)C1 C1(C(N(CCC(=O)NCC2(C)CC3CC3C2)CC2CC2)=O)CC2(CCC2)CO1 N1(C(C2CN(C(CN(C)C(N)=O)=O)CC2F)=O)CCC12CCC(O)CC2 C1(C(=O)NCCNC(=O)CO)C2CC1N(C(=O)CC1CCCSC1)C2 C1(CCC(C)C)C(=O)N1.C(C)(C)(CCC(=O)N1CCCC(OC2CC2)C1)OC C1(NC(c2cn(CCC)nn2)=O)(CNC(=O)COC(C)=O)CC2CCC1C2 c1(C(=O)NCC2C3CN(Cc4c(OC)ccnc4)CC32)nccc2ccccc12 c1(CC(=O)NC(CNC(C2CCC(C)(C)O2)=O)(C)C2CC2)cnc2n1CCOC2 C(C)(N=c1cc[nH]c(=NCCc2cncc(OC)c2)[nH]1)c1cccc(COC)c1 N1(C(c2cc(C)nn2C)=O)CC2CC(CNC(=O)Cc3ccc(Cl)c(F)c3)C2C1 C(=O)(C1CCCc2nncn21)N1CCN(C(CNC(C(C)CC(N)=O)=O)=O)CC1 c1(C(N2CCC(CN(CCC)C)C2)=O)c(C)nn(CC(F)F)c1C Cc1cc(F)c(CC(=O)NCC(O)CCNC(=O)CCS(C)=O)cc1F C1(NC(C2(CC(C)C)CCCC2)=O)C=CCN(C(C2CCCC(=O)O2)=O)C1 c1(C(=O)NC2(C)CN(C(c3n(C(CC)C)ncc3)=O)C2)ccnnc1O CC1CCN(C(=O)CC2CCC(=O)N2)CC1NC(=O)CCc1cc[nH]n1 C1(CNC(CCS(=O)(=O)N(C)C)=O)CCC2(CN(C(C3CCOCC3)=O)C2)O1 Cc1cnc(Cl)[nH]c1=NCCCCNC(C1CCC(NC(=O)N(C)C)CC1)=O C1(NC(C(C)CC#N)=O)CN(C(=O)CC2CCC2)C2(CCC2)C1 Cc1cc(C(N2CC3CC3(CNC(c3nnn(C)c3N)=O)C2)=O)cc(F)c1 C=CCCC(F)(F)C(=O)NC1CCC(CNC(c2ncc(Cl)cc2Cl)=O)C1 c1(C(=O)NC(CN(C(=O)CC2CCC2)CC)C)ccc2c(n1)OCC(=O)N2 c1(C(=O)NCC2C(NC(C(c3ccc(OC)cc3)O)=O)C2)cc2c(ncn2C)[nH]1 C1(CC)(CC)CC(NC(=O)C(C)=CC(C)(C)C)CN1C(=O)Sc1ccc(F)cc1 C1(C(N2CC(CC(=O)OCC)C2)=O)(CNC(c2cccnc2O)=O)CC12CCC2 C(C)(CC1=CCCCC1)NC(C(CC)NC(=O)CCc1nccs1)=O C1(C(NOCC=CC)=O)CC(C)CN(C(c2cc(CC=CCOC)[nH]n2)=O)C1 N1(C(CC=CC=C)=O)CC2(C1)CN(C(=O)Cn1ccc(C3CC3)n1)CCO2 N1(C(C(CCC)F)=O)CCC(NC(c2ccc(OC)cc2F)=O)C(CO)C1 c1(OC)cc(C)cc(C(=O)NC2CCCCCN(C(=O)C(F)=CC3CC3)C2)c1C C1(C(=O)OC)CCN(C(C2(CNC(c3cc[nH]n3)=O)CC=CC2)=O)C1C N(C1CN(C(=O)COCCSC)Cc2ccccc21)C(CC(C=C)CC)=O C1(=O)C(=O)NC2(CCCN1)CC2.CC1CC1.C(=O)(CC1(N(C)C)CC1)NC(C)(C)C c1(CN(C)CC2CN(c3nc(SC)nc(C)c3)C2)cc(Cl)cc(Br)c1O c12c(C)nn(c1C)COC2=O.c1(C(=O)NCC)cc(C2CCCCN2C)nn1C C1(CNC(C=CCOC)=O)CCC2(CN(C(c3ccc(C(C)=O)cc3)=O)C2)O1 c1(C(C)(C)C)nn(Cc2ccccc2)cc1NC(=O)NCCC1CCNC1=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)(CC)CCNC(=O)C(C#N)CC N1(C(C(=Cc2ccco2)C)=O)CCN(C(=O)Cc2csnn2)C2CCCC2(C)C1 C1(NC(CNC(=O)OCC=C)=O)CCCC(C(C)NC(c2csc(C)n2)=O)C1 C1(CNC(C2CC3CCCC23)=O)CC2CCC1N2C(C1CC1(F)F)=O c1(-c2c(C(C)C3CC3)cccc2)ccc(=O)n(CC(F)(F)F)c1 Cc1ccc(C(=O)NCC2CC3CN(C(C4CC4(C)C)=O)CC23)cc1F C1(O)(C(=O)NCC2C(CNC(C(COC(C)=O)C)=O)C2)CN2CCC1CC2 CCC(C)(C)C(O)C(=O)N1CC2CN(C(=O)COC(C)(C)CC)CC2C1 C(=O)(C1CCc2c(Cl)cccc21)N1CCC(NC(C=Cc2cncc(C)c2)=O)C1 C1(CNC(CCCC#C)=O)COCC2(CCN(C(=O)C=CC3CC3)CC2)O1 C12(NC(c3cc(C)[nH]n3)=O)CCCN(C(c3c(C)cc(F)cc3C)=O)CC1C2 N1(C(c2on(C)c(=O)c2)=O)CC2CCN(C(=O)C=Cc3cccc(F)c3)CC2C1 c1(OC)ncccc1CC(=O)NCC(C)NC(c1nocc1-c1ccccc1)=O Cc1nc(N2CCC3(C(N4CC(CO)C(CO)C4)=O)CC3C2)ncc1Br c1(CN2CCCC(C(=O)Nc3nnc(Br)s3)CC2)ccc(F)c(Br)c1F N1(C(C2(C=C)CC2)=O)CCC(NC(=O)Cc2ncoc2C)C(CO)C1 Cc1cc(C)c(-c2nc(Cc3ccccc3F)no2)cn1 c1(CC)cc(C(=O)NC2CC(NC(c3ncc(F)cc3N)=O)CC2O)cc(F)c1 O=C1CC(CC(=O)NCC2CCC(NC(=O)CC34CCCC3C4)CC2)=NN1 C=C1CC2CC1CN2C(=O)C(C)(CSC)NC(=O)C(C)C(C)C c1(OC(c2cn(CC)nc2C)=O)ccccc1C#N.c12cc(cc(Cl)c1)N2 C(=O)(C1=NOC2(CCC2)C1)N1CC(NC(C(C)OCCC#C)=O)(COC)C1 C(=O)(C(C)CC(N)=O)N(C1CN(C(CC2(CC=C)CCCC2)=O)CC1O)C C(C(N=c1[nH]nc(C)o1)c1ccccc1)NC(CCc1c(OC)cccc1)=O c1(C(N2CCC(C(C(=O)NCC(C)OCC#C)(C)C)C2)=O)ccc(CC)cc1 Cn1cc(C#CCNC(=O)NC2(c3cccc(Br)c3)CCC2)cn1 c1(C(=O)NC(CNC(c2ccc(CCC)[nH]2)=O)C(C)C)ccc(C#N)c(F)c1 c1(C(N2CCC(C(=O)OCC)(C(C)C)C2)C(=O)OC)ccc(S(C)=O)cc1 c1(C(N2C(C)(C(N3C(C)CCC3)=O)CCC2)=O)c[nH]c2cnccc12 N1(C(C2CCC(=O)N2)=O)CCOC(CCNC(c2cccc(C(F)(F)F)n2)=O)C1 c1(CC(=O)N(C(C(=O)NCCC(CC)O)C)C2CC2)ccnc(O)c1 Cc1nc(NCC2CC(=C3CC3)C2)cc(NC(c2ccccc2Cl)CC(N)=O)n1 C12(CNC(c3c(C)cccn3)=O)CC(NC(=O)CCSC(F)(F)F)(CCO1)C2 N1(C(CC(C(C)C)C)=O)CCC(CNC(c2cncc(C(F)F)c2)=O)C(F)(F)C1 c1(C(=O)NCCn2ncc(C(=O)NCCC3ON=C(C)C3)c2)ncc(C)cc1C C1(C(N(C)CC2CCCN(C(COCC#C)=O)C2)=O)CN2CCN1CC2 C1(Cn2ncc(Cl)c2)CN(N2CCC(CN3CCCCC3)CC2)C1 c1(C(=O)NC2(CNC(C(CC)CCOC)=O)CC2)cc(OC)c(OC)c(N)c1 S(=O)(=O)(c1cc(C(=O)NCC2CC3(CC3)CN2C(=O)C2=CCSC2)c(C)o1)NC C1(NC(Cn2c(C)ncc2)=O)CCCN(C(c2scnc2C(F)(F)F)=O)CC1F Cc1ccc(N)cc1C(=O)NCC(F)CNC(c1coc(C(F)F)c1)=O C12(C(=O)NC(CC)CNC(c3ncc(N(C)C)cn3)=O)CC1COC2(C)C N1(C(CCC(C)(C)NC(c2cnn(C)c2N)=O)=O)Cc2n[nH]cc2C1CO C1(C(=O)NC2(CCNC(=O)CCCn3cncn3)CC2)COC2(CCC2)C1 CC1CC(C(=O)NCC2CCCCC2NC(C2CCOC(C(C)C)C2)=O)=NO1 C1(NC(C(C)S(N)(=O)=O)=O)CCN(C(c2n[nH]cc2Br)=O)CC1(C)C CCCCC(O)CC(=O)NC1(C)CCCN(C(c2ccc(C)c(C)c2N)=O)C1 c1(-n2c(C(c3c(CC)ocn3)NC(C)(C)COC)nnn2)c(C)cccc1C N1(C(CC(CC=C)(C)C)=O)CC2CC(C)N(C(C3CCCN3C3CC3)=O)C2C1 CCCC(CCCNC(C1(Cl)CC1C(C)=O)=O)NC(=O)CN1C(=O)CCC1=O N1(C(CCOCC)=O)CCN(C(=O)CC2OC(C)(C)OC2=O)CC1C1CCCC1 CC1CN(C(=O)CCCOc2cccnc2)CC1NC(C1CSCCS1)=O c1(N(CCC)CCc2ccccc2)nnc(-c2cnc(C3CC3)[nH]2)n1CC(C)C N1(C(C(C(C)C)O)=O)CCN(C(c2ccnnc2S)=O)C(CS(C)(=O)=O)C1 C1(C(N2CC(N(C(=O)CSC3CCOCC3)C)C2)=O)CCC2(CCC2)O1 CON1CCC(C(=O)NC2CC(O)C2CC(=O)NCC2CC=CC2)CC1 C1(O)(C(N(CCN(C(=O)C(O)CF)C)C)=O)CCC(NC(=O)OC(C)(C)C)CC1 CC(C)C(C)C(C)CC(=O)N(c1ccc(Cn2ccnn2)cc1)CCC#N CN1CCCN(C(=O)C(C(C)(C)C)NC(c2ccc[nH]2)=O)CC1 C1(CC)(CC)CC(NC(=O)CN(C)CCO)CN1C(c1cc(O)nc(O)n1)=O C1(C(=O)NCCCCC(CO)NC(CC=CC=C)=O)CCc2ncccc2C1 C(C(=O)N1CC(O)CCO1)(N(C(C(CC=C)CC)=O)C)C1CC1 CC(C)C(O)CC(=O)N1CCOC(C)(CNC(c2cocn2)=O)C1 C=CCCC(F)(F)C(=O)N(CCCCCNC(c1cc(Cl)cs1)=O)C N1(C(c2csc(C(C)C)n2)C(=O)NC(CC)C)CCc2c(ccnc2C)C1 Cn1cnc2nc(N3CC(CCNC(=O)C(c4ccc(F)cc4)(F)F)C3)ncc12 N1(C(C(CC)NC(c2ccccc2)=O)=O)CC2CC(C)N(C(=O)CSC(F)F)C2C1 c1(C(N2CC(NC(=O)C=CC3CCCC3)C(F)C2)=O)cc(Cl)c(Cl)cn1 N1(C(C2CCC(C)(C)OC2)=O)CC2(CCCC2NC(=O)C2=CCCOC2)C1 C(=O)(CC(C(C)CC)NC(=O)CCc1ccnn1C)N1CC(C#C)C1 C(c1ccc(Cl)cc1F)=CC(=O)NC(C(C)C)C(=O)N1CCCC1 c1(C(=O)NCC2CC(OC)CN2C(c2cccs2)=O)csc(=NC2CC2)[nH]1 N1(C(C2N(S(C)(=O)=O)CC2)=O)CC(C)(c2cn(C)nn2)C1.C1(CC=O)CC2CC2C1 C12(C(=O)NC(C)(CNC(=O)Cc3sccc3Cl)CO)CCCC1CC(=O)C2 c1(OC)ccc2c(n1)NC(C(=O)NC1CC1NC(=O)CCCCC(N)=O)C2 c1(SC)ccc([N+](=O)[O-])cc1CNC1CN(C(c2ccoc2)=O)CC1C Cc1ccc(NC2CCC(NC(C3(NC(c4cccc(O)n4)=O)CC3)=O)C2)cc1 CC1CCCC(C(=O)NCc2ncccc2C(F)(F)F)O1 CCC(CC(=O)NC1(CO)CCCCC1)NC(=O)C(C)C(C)NC(C)=O c1(C(=O)OC(C)(C)C)cc2n(n1)CCCN(C(=O)CN1CC(=O)NC1=O)C2 C(=O)(C(C(C)C)SC(=O)N(C)C)NCCN(C(c1nc(C2CC2)no1)=O)CC N1(C(CCC(=O)NC)=O)CCCC(O)(CNC(=O)CN(C)S(=O)(=O)N(C)C)C1 C12(NC(C(c3cccc(O)c3)C)=O)CCCC1CN(C(=O)COc1ccsn1)C2 c1(C(N2C3CN(C(c4c(C)ccc(O)c4)=O)CC32)=O)cccc2c1OCO2 C1(N(CC(=O)NC2CCCNC2)C)CCN(CC(F)F)CC1 c1(C(N2C(C)C(NC(=O)Cc3ccoc3)CC2)=O)coc2c1NC(=O)CCC2 Cc1nc2ccnn2c(N2CCC(OC(C3CCCNC3)=O)CC2)c1C C1(CC)CN(C(c2ccccc2Br)C(=O)NC2CCC2)CC(C)O1 N1(C(COCC(C)C)=O)CC(N(C)C(C23CC(CO)(C2)C3)=O)C(F)C1 N1(C(c2c(CNC(C3CC4(CC4)CO3)=O)noc2)=O)C2COCC1C2 c1(SCCC(=O)NC2CN(C(c3nc(C(C)C)oc3)=O)C2)nc2ccccc2[nH]1 c1(OC)ccc(Br)cc1CC(N1CC(CN=c2[nH]nc(C3CC3)o2)CC1C)=O C1(c2cn(C)nc2)CN(C(=O)C(N)=O)CC1NC(=O)CC(C)(C)NS(C)(=O)=O c1(OC)ccc(Cl)cc1C(F)(F)C(=O)NCC(CO)NC(C1CCSC1)=O C(=O)(N1CCCc2nncn21)C1C(NC(=O)OC(C)(C)C)CCO1 N1(C(c2ccn(CCCC)n2)=O)CCN(C(=O)CCC=C2CCCC2)CC1 N#Cc1nccc2cc(NC(C3CN(c4ccccn4)C3)=O)ccc12 C(=O)(CC(F)(F)C(C)C)NC1CCCN(CC(=O)NC(CN(CC)CC)C)C1 C(C(C)(C)CC(=O)NC1CC(CNC(=O)CCc2cccc(C#N)c2)C1)OC C1(C(=O)NCC(C2CCCCC2)C)CC2(CCN1C(=O)C(C)CO)CC2 N1(C(C2NCCC23CC3)=O)Cc2ccccc2CC12CCC2 N1(C(C(CC=C)OC)=O)CC(C)(C)OCC1C(=O)Nc1csnc1OC N1(C(c2cccc(CC)c2)=O)CCCN(C(c2cnc(N)c(Cl)c2)=O)C(C)C1 C=CC(C)(CCOC)C(=O)NCC(CCNC(c1cc(C(C)(C)C)no1)=O)OC C(CCN=C(NC(C)C1CC1)NC1CC(=O)N(C(C)(C)C)C1)=CC=C c1(C(N(C)CCNC(C2CCC3CC3CC2)=O)=O)ccc2sc(=N)[nH]c2c1 Nc1cc(C(=O)NC2CCC2C(=O)NC2CC(CO)(CO)C2)cc(F)c1 Cc1ncncc1NC1(c2nnnn2C2CCOCC2)CC2CC2C1 N1(C(C(CCC=C)(C)C)=O)CC2COCCC2(NC(C2CCCN(C)C2)=O)C1 C1(C)(NC(c2nc(C(C)NC(CC=CC)=O)oc2)=O)CC=CCC1 C1(C2CCN(CC(=O)CC3CCOCC3)C2)NC(=O)NC1=O C1(C2CCCC2)(C(=O)NC2C(CNC(=O)CCC3CCC3)CCC2)CCNC1=O N1(C(C(NOC)=O)=O)CCN(C(C2CN3CCN2CC3)=O)CC1C1CCC1 Cc1nc(C(=O)N(C(C)(C)CC(=O)N2CC(F)(C#N)C2)C)sc1C C1(S(N)(=O)=O)(C(=O)NC2C(CNC(C3(C)COC3)=O)COC2)CC1 N1(c2n(CC(C)C)c(-c3csnn3)nn2)CC2CN(C)CCC2(CO)C1 c1(CC)cc(C(=O)NCC(C)(C)OCCNC(c2cscc2F)=O)ccc1C c1(C(N2C(CO)CC(NC(C(CC)CC3CCCC3)=O)C2)=O)c[nH]c(=N)cc1C C1(NC(C2C(CCC)C2)=O)CC2(C1)CC(C(=O)NOCC1CC1)C2 c1(C(C(=O)NC(C)C(C)N2CCCC2)O)ccccc1Br Cc1cc(Cl)ccc1C(N1CC(NC(=O)C2=COCCO2)C(O)C1)=O C1(OCC)CC2(C1)CC2C(N1CC(CC(C)NC(=O)C(C)(F)F)C1)=O Cc1ccc2c(c1)SC(C(=O)NC(C)(CNC(c1occc1F)=O)C1CC1)C2 c1(CN2CCC(NC(c3c(C)nc(Br)cc3)=O)C(F)C2)ccc(Br)c2nsnc12 c1(SCC(=O)NCC2CN(C(c3cc(C4CCC4)on3)=O)C2)ccncc1Cl c1(C(N2CCCCC(C(N3CCC(C(F)(F)F)C3)=O)C2)=O)ccc(Br)c(Cl)c1F N1(C(C(C)OCOC)=O)CC2CCN(C(C3CCN(C)CC3)=O)C2C1C C#CC(CNC(=O)C(CCSC)NC(=O)C=C(C)COC)CC(C)(C)C C12(C)CCCN(C1)C2=O.C1(NC(C2(COC)CCC2)=O)CCCC1C#N CC(CCCNC(=O)C(C)Cc1cccnc1)NC(c1cn(CCO)nn1)=O CCC(C)CCCCC(=O)NC1CCCCN(C(=O)C(C)(C)C)CC1 N1(C(C)C(=O)NCCc2cnccn2)C2CCC1CN(C(=O)Cn1cnnn1)C2 c1(C(=O)NC(C)CNC(=O)CC2CCCC2C)cn2c(n1)CCC2 C(N=c1cc(NCCCn2cnnc2)nc[nH]1)c1c(C)sc(Br)n1 c1(C(=O)NCCNC(=O)C=CCC(=O)NC2CC2)ccnc(OCC(F)F)c1 N1(C(c2ccc(C#N)[nH]2)=O)CCC2CC1CN(C(=O)CC1CCC3(CC1)CC3)C2 C1(N(C(C(C)SC(C)C)=O)C)CCN(C(C2CC(O)C(O)C2)=O)CC1 CC1CC2(CC2)CN1C(c1cc(CNC(c2cncs2)=O)on1)=O c1(C(N2CC(CCNC(C(C)C3CC3)=O)OCC2)=O)cc2n(n1)CCC2 C(C)(CCC(=O)NCC(C)NC(=O)C(C)Cc1ccncc1)OCC C(C(C)(O)CCO)NC(C1CCC(CNC(C(C2CC2)SC)=O)C1)=O C(=O)(C1=C(Cl)CCC1)NCCC1(C(N2CC(C)SCC2)=O)CCCC1 N1(C(CN2CCC(OC)C2)=O)CCCCC(CNC(=O)CCC2OCCO2)C1 Cc1c(N)cc(C(N2CCC(NC(C3CCS(=O)(=O)N3)=O)C(C)C2)=O)cc1N C1(NC(C2(CSC)CCC2)=O)CC2CC(NC(c3cnccc3Cl)=O)C2C1 c1(C(N(C2CCCC(NC(c3c(C#C)c[nH]n3)=O)C2)C)=O)cccn2nccc12 Cc1sccc1CC(=O)NCC(C(C)C)NC(c1c[nH]cc1Br)=O c1(C(=O)NCCOCCNC(C(CSC)O)=O)cc(C2CCCCC2)ccc1O C1(NC(CCCCC)=O)C2CC3CC(C2)CC1(CNC(=O)C(F)(F)CC)C3 C1(NC(c2c(CC)cco2)=O)CN(C(c2ccc3oncc3c2)=O)C2(CCC2)C1 N1(C(C(COC)O)=O)CCC2(CCCN2C(=O)C(C)c2ccco2)CC1 N1(C(C(C2(O)CCC2)NC(c2cc(CC)n(C)n2)=O)=O)CCC2(CNC(=O)N2)C1 C1(C)(CNC(c2ncc(C)nc2)=O)CCCN(C(C2CCCS2)=O)C1 C1(OCC)CC2(C1)CC2C(=O)NCC(O)CNC(=O)Cc1cnccc1C c1(SCC)ccc(C(=O)NCC2CC2NC(C2CCCN2C(C)C)=O)cn1 CC1CN(C(=O)C=Cc2ncco2)CC1NC(=O)C(c1ccc(Br)cc1)C C(C(CC(F)(F)F)NC(C1CCCOCC1)=O)NC(C(C)NC(N)=O)=O C1(CNC(C2(SC)CC2)=O)COCCN1C(=O)Cc1ccc(C(F)(F)F)o1 N#CC1CCCCC1NC(=O)Nc1ccc(OCC(F)F)cc1 C(CNC(C1CC2CC2N1C(=O)CCC(C)N(C)C)=O)(C(C)(C)C)OC C(=O)(CCC1=NNC(=O)CC1)N1CC(NC(c2nc(OCC)sn2)=O)C2C1C2 Cn1ncc2c1CCC(C(=O)NC1CCCCC1NC(=O)CCc1ccsc1)C2 N1(C(c2cc(CC)nnc2C)=O)CC(C2CN(C(C3(C(C)(C)O)CC3)=O)C2)C1 CC(C)C(C(=O)NCC1CC1CNC(=O)CN(C)C(C)C)C(F)(F)F C1(N(C)C)CN(C(C2CC(NC(=O)CCC(N)=O)C2(C)C)=O)CC1O C1(COC)(CNC(=O)C(C)CF)CCCN1C(c1c(C)cnn1C)=O c1(CNC(c2cc(CNC(C3N(C(=O)OC(C)(C)C)CC3)=O)n[nH]2)=O)c[nH]nc1F c1(C(N2CC3N(C(c4cccc(=O)n4O)=O)C(C3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] C(CCCC(=O)N(CCC(=O)NC12CC(CC3CC3)(C1)C2)CC1CC1)N(C)C C(=O)(CC(C)CCC(=O)NC(C)(C)CN(C(=O)CCCc1nc(C)cs1)C)OC C=CC1(C(=O)NCCCCCNC(=O)Cc2cccn2C)CCC1 Cc1cc(C(=O)NCC2CCCC2NC(=O)CC2CCCOC2)ns1 C1(NC(=O)CC2C=CCC2)CC2CC(NC(c3csc4nnsc34)=O)C1C2 c1(CN2C(C(=O)NCC3CCCOC3)CCC2)c(F)ccc(Cl)c1Br c1(C(=O)NCC=CCOC)cccc(C(=O)Nc2ncccc2C(C)C)c1 C(=O)(C(CCC1CC1)NC(=O)CCn1cnc(=N)[nH]1)N(C)CC1CC(C(N)=O)C1 C(=O)(CCC(CC)OC)NCCN(CCOC)C(C1CCC(N(C)C)CC1)=O N1(CCC#C)CC2CCN(C(c3csc(C(F)(F)F)n3)=O)C2C1 CC1(C)CCCCC1NC(=O)CC(N)C1CCCCC1 c1(C(=O)NC(C(=O)Nc2cc(C)cc(C)c2)CS(C)=O)ccnc2cc[nH]c12 N1(C(c2c(C)n(C(C)C)nc2)=O)CCC2C(NC(=O)CC(O)C3CCCC3)CC12 CC(C)CC(O)C(=O)N1CCN(C(c2ccc(-c3nc(O)n[nH]3)cc2)=O)C(CO)C1 C(=O)(C(CCCC)C(C)C)NCC1(C(N2C(CC#C)CCCC2)=O)CC1 c1(C(=O)NCc2cccnc2N2CCCCC2)cc2c(cn1)OCCC2 CC1CCN(C(c2cnccn2)=O)CCN1C(C1CC2(C1)CC(C)(C)C2)=O c1(C(=O)NC(C(=O)N2CCC(COCC#C)C2)CCC)ccn2ccccc12 c1(CC(N2CCC(CCNC(COC(C)(C)C)=O)C2)=O)cccc(S(C)(=O)=O)c1 C1(C(=O)Nc2cc(C(=O)OC)[nH]c2)CN(Cc2cccc(C)c2N)CCC1(F)F CC1(C(=O)NCC2(CNC(c3cc(C#N)no3)=O)CC23CCC3)CCOCC1 CC1CCN(C(C2CCC2C(N)=O)=O)CC1N(C(=O)C(=O)NC1CC1)C N1(C(c2c(C)nc(CO)nc2)=O)CCC2CCN(C(c3cccnc3S)=O)CC12 N1(C(CSCCC(C)C)=O)CCC2C(C(=O)NCC3CCC(C)(C)CO3)C2C1 C(=O)(C=C1SCC(=O)N1C)NC(C(C)C)CNC(C1CN(S(N)(=O)=O)C1)=O CC1C(NC(c2cc(Cl)ccc2Cl)=O)CC2CCC1N2C(C1(CO)COC1)=O c1(C(N2CC(C)(NC(c3ccc(C)[nH]3)=O)C2)=O)cccc2c1OCC2C CON1CCC(CC(=O)NC2CC(CNC(C3CC3F)=O)C(O)C2)CC1 N1(C(Cc2n(C)cnc2)=O)CC(C(=O)NC(c2cscn2)CO)C(F)(F)C1 c1(C(=O)NC(CC)CN(C)C(C2(C)CCCO2)=O)cc2c(cc1C)OCO2 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(C(C)NC(C2CC2C(F)F)=O)CCC1 C(=O)(C(O)CC(N)=O)NC1(C(=O)Nc2c(OC)cccc2)CCN(C)C1 c1(-c2ccc(N(C)C)nc2)cccc2ccc(C(N3CC(O)CC3(C)C)=O)nc12 S(=O)(=O)(c1cccc(CC(=O)NCCc2nc3c(s2)COCC3)c1)NC C1(C(=O)NCC2(C(N)=O)CN(C(=O)CNC(c3cscn3)=O)C2)CCS(=O)(=O)N1 C1(C(=O)NCC2(C=C)CCC2)(C(C)C)CCCN1C(=O)Cn1cc(CO)nn1 c1(C(=O)NC(CC)CNC(c2c[nH]cc(Cl)c2=O)=O)ccc2c(c1)C(C)CN2 n1(C(C)(C)C)ncnc1CSc1nc(C(F)(F)F)cs1 CC(C)S(=O)(=O)C(C)C(=O)NCC(C)N(C(c1ncsc1Br)=O)C1CC1 N1(C(c2cc(C#N)sc2)=O)CCC(NC(=O)COCC2CCCO2)C(F)(F)CC1 c1(C(=O)NC2C3CN(C(c4cnn(C)c4Cl)=O)C2CC3)cc2c(s1)CC(C)(C)C2 C1(C(=O)OCC)CCCCN1CCc1nnc(C(F)F)o1 c1(C(N2CCC(N(C(Cc3c(C)con3)=O)C)C(C)C2)=O)ccc2cncn2c1 c1(C(N2CCC(N(C(c3csc(SC)n3)=O)CC)C2)=O)nccc2occc12 N1(C(C(C)Cn2ccnc2)=O)CC2=C(C1)CN(C(=O)CN1CCOCC1=O)C2 c1(OC)cnc(F)c(C(N2CC(C)(C)CC2CNC(=O)CC2CCCC2C)=O)c1 c1(C(N(CCCN(CC(=O)NCc2cccnc2)C)C)=O)onc2c1CCCC2 Cc1c(F)ccc(Cl)c1C(N1CC2OCC(NC(C3CC3F)=O)C2C1)=O c1(C(=O)NCC2CC(CNC(c3cscn3)=O)C2)cccnn1 N1(C(C2C3(CN(C(c4ccc(CC(C)C)cc4)=O)C3)C2)=O)CCn2cccc2C1 c1(C(=O)NC(C)CCCCNC(C2CCSC2)=O)cnc2c(F)cccc2c1 c1(C(=O)OC)nccc2c1CCCN2C(=O)C(CC(F)F)C1CCC1 c1(C(=O)NC2CC(C)(NC(CCOC)=O)C2)cnc(O)nc1O c1(C(=O)NCCCN(C(=O)C(F)(F)C2CC2)C2CC2)cc(C(F)(F)F)ncn1 C1(C(N(CC)OC)=O)CN(C(C2CC(=O)CS2)=O)CC12CCC2 C1(NC(C2(C(C)C)CC2)=O)CCC(CNC(C2CC2C)=O)CC1 CC1CCCC1(C)NC(c1[nH]ccc1CNC(C1(F)CCCCC1)=O)=O C1(C(N2CC(CC(=O)Nc3ccno3)OCC2)=O)Cc2nccn2C1 c1(CN(C(=O)NC2C(C(=O)NCCC)C2)CC)cc(F)cc(F)c1Br Cc1ccc(C2CC2C(=O)N(CCCNC(C2CCO2)=O)C)cc1C N1(C(C(C2(OC)CCCC2)(F)F)=O)CCCN(C(c2cnc3n2CCC3)=O)CC1 c1(C(=O)NC2C(CNC(=O)CCc3cnn[nH]3)CCCC2)cc2cscc2s1 c1(C(=O)NC2CC(CNC(C(CSC)O)=O)CC2O)cncc2c1CCC2 C=CCC(C(=O)N1CCCCC1CNC(c1cc(SCC)nc(O)c1)=O)C(C)C c1(OC)ccc(NC(C2CC3CC2CN3C(C2C3C=CSC23)=O)=O)cc1C#N CC#CCCCCNC(=O)C(C)N(C(c1cc(CCC)on1)=O)C1CC1 N1(C(C2CCCC(NC(c3c(C#C)cnn3C)=O)C2)=O)CCCC(C)(OC)CC1 C1(OC(C)(C)C)CCOC12CCCC2.N12CC(F)(F)CC1(CO)C2=O C1(CCC)CN(C(c2c(C(F)(F)F)ncn2O)=O)CCN1C(C1CC12CC2)=O C12(NC(C(C)NS(CC)(=O)=O)=O)CCCN(C(c3c[nH]c(=O)cn3)=O)CC1C2 c1(CNC(c2cc(C)on2)=O)cc(C(=O)N(CCCO)C(C)C)ccn1 Cc1ccccc1S(=O)(=O)CC(=O)NC1CCCN(C(c2cncnc2)=O)CC1 c1(OCC(=O)NCCC2CSCCN2C(=O)CCF)ccc(Cl)nc1 c1(C(C(=O)NCC2N(C(CC(C)(C)OC)=O)CC(OC)C2)O)ccc(F)c(F)c1 N1(C(CCc2cc(C)no2)=O)CC(NC(c2cc(C(C)=O)oc2C)=O)C2CC12 c1(CNC(C(CC)(C)O)=O)nn(C)c2c1CN(C(c1cc(=O)cc(Cl)[nH]1)=O)CC2 C1(NC(C2(CN(C)C)CC2)=O)CN(C(C2CCCC23CC3)=O)C2(CCCC2)C1 c1(C(=O)NCC2N(C(C(CCC)CC)=O)CC=C2)ccc(F)c2c1OCC2 C1(CC)(CC)CC(NC(c2cc(Cl)ccc2N)=O)CN1C(C1CC1(C)C)=O N1(c2nnc(C(C)C)n2CCC(=O)N(C)C)CCC(F)(F)C(O)C1 C(=O)(C1=CC(O)C(NC(=O)C(c2ccn(C)c2)C)C1)NC(CC)CCOC c1(C(N(C(C)CN(C)C(C2CCCN2C=O)=O)C)=O)cc(F)ccc1O c1(OC)cccc(N(C(=O)CSC(C)C(N2CC(CN)C2(C)C)=O)C)c1 N1(C(C2CCN(C(CC(C)F)=O)C2(C)C)=O)Cc2cccc(F)c2C1 C1(C(=O)NC2(CNC(C(C)n3cncn3)=O)CC2)CNC(=O)C(C)(C)C1 C(C(C)C(=O)NCCCN(C(=O)CC12CC(C(C)=O)(C1)C2)CC)OCC c1(C(=O)NC(CCSC)C(=O)N(C)CCN2CCCCC2)cn(C)c(=O)n1C c1(C(=O)NC2(CF)CCN(C(C3(C#N)CC34CCC4)=O)C2)cccc2c1CCO2 CC(C)C(CC(=O)NC1(CCO)CCC1)NC(C1CC(F)C(=O)N1)=O C(=O)(CCCCCc1cccs1)N1CCC(N(C(CCC=C=C)=O)CC(C)C)CC1 N1(C(COCC(C)C)=O)CC(F)CC1CNC(c1csc(-c2cnc[nH]2)n1)=O c1(NC(c2ccc(NC(=O)OC(C)(C)C)o2)=O)cnn(S(C)(=O)=O)c1 C(=O)(C1CCCc2sc(=N)[nH]c21)NCCOCCCN(C(=O)C(O)CC(N)=O)C S(=O)(=O)(c1ccc2c(c1)CCCC2)N1C2CCCN(C(c3nccs3)=O)C2CC1 C1(NC(CC(c2c(C)noc2C)C)=O)CCN(C(=O)CN=S(C)(C)=O)CC1F N1(CC(=O)NC(CNC(c2ncccn2)=O)CO)CCSCC1 C(C)(C)(CCC(=O)NC1CC1CC(C)C)OC.C12CC1CNC2=O Cc1cc(C(N2CCC(O)(C(C)NC(C3CCC(=O)C3)=O)C2)=O)cc([N+](=O)[O-])c1 C1(CNC(C2(C(N)=O)CC2)=O)CCCC(CNC(=O)CC2CC3(CCC3)C2)C1 c1(C(=O)NC(C(=O)OCC)Cn2cc(C)cn2)ccc(CO)cc1F N1(C(c2cc(OCC)ns2)=O)CCN(C(=O)C(C)OC)C(c2cn[nH]c2)C1 C1(C(N2CC3(CC(NC(COCC(=O)OC)=O)C3)C2)=O)CC2CC(O)CC(C1)C2 c1(-c2ccc(CCCC)s2)cccnc1OCCSc1ccc(C(F)(F)F)nc1 C1(CC(N2CC(O)(C3CCC3)C2)=O)C2CCCC2N1C(C1(CO)CC1)=O c1(NS(CCOC)(=O)=O)ccc(O)c(NC(C2CCOC(C)(C)C2)=O)c1 N1(CC(=O)NCC(CNC(C2C(CC)C2)=O)CO)CC(=O)NC1=O C1(C(=O)NC2C(c3cn(CC)nc3)OCC2)CCS(=O)(=O)CN1 N1(C(C(CC)(C)C)=O)CCC2(CC1)CC2c1cn(CC2(OC)CC=CC2)nn1 N1(C(C(C2CCC(NC(=O)CCCn3ccnc3)C2)C)=O)CC2(CC2)C1 C1(O)(CN(C)C(C2CC(O)CN2C)=O)CCCN(C(=O)C(C)CSC(F)(F)F)C1 N1(C(Cn2c(=N)[nH]nc2)=O)CCCC2(NC(=O)Cn3cnnn3)CC2C1 Cc1cc(CNC(C2(C(C)NC(=O)CCOCC(C)C)CC2)=O)cc(F)c1 C(C(CC1CC1)CO)NC(CN(C(=O)Cc1ccnn1C)CCC)=O C(N=c1[nH]c(=NCCN(C)C(C)C)[nH]c2c1SCC2)C1CCCC(CC)C1 CCCCC(CC)CC(=O)NC(C1(NC(=O)CC2(C)CC2)CC1)C S(=O)(=O)(c1cccc(NC(=O)CN2CCC(C3CC3)C2)c1)NCC c1(C(N(CCNC(c2cc(C)c[nH]2)=O)CC)=O)cc2ccccc2cc1C C12(NC(CCCC=C)=O)CCOCC1CN(C(C1(C#N)CCN(C)CC1)=O)C2 CC(CCC(=O)NC1COCCC1NC(=O)C(C)(C)O)c1ccc(Br)cc1 N1(C(C2CN(CC)C(=O)C2)=O)CCCC2C1CCN2C(c1ccncc1)=O c1(C(N2C(CNC(c3c(O)ncc(CC)c3)=O)CC2)=O)cccc2c1CC(=O)N2 Cc1cccc2c1CC(C(=O)NC1COCC1NC(c1cc(CO)[nH]n1)=O)O2 C1(CCNC(c2n(CC#C)ccc2)c2nnnn2CCCF)CC(C)(C)NC1=O O=C(N=c1nc[nH]s1)C1CCCC(NCc2ccc(-c3cnccn3)cc2)C1 C(CC(C(F)(F)F)N1CCOCC1)NC(c1cccc(-c2ccc(O)nn2)c1)=O C1(C)(NC(C2(C=C)CC2)=O)CCN(C(=O)Cc2csc(C(=O)OC(C)(C)C)n2)C1 c1(C(=O)NC(CC)CNC(C2CSCN2C)=O)c(C)ccnc1C N1(C(CCC#C)=O)C2CCC1C(CNC(c1cncc(OC(F)F)c1)=O)C2 C(=O)(C1CCc2c[nH]nc21)N1CCC2C(C(=O)N=c3ccn(CCF)[nH]3)C2C1 CCCC(O)C(CO)NC(=O)CCC1CCCN(C(=O)Cc2ncccc2F)C1 Cc1nc(N2CCCC(CN(C(=O)CC3CCCCO3)C)C2)c2c(C)csc2n1 N1(C(C(C2CC(NC(=O)COCC3CCC3)C2)F)=O)CCCC2(CC2)C1 CC1(C)CC(NC(c2ccc(F)cc2)c2ccccc2)CS1 N1(C(CC2(C(=O)OC)CC2)=O)CC(C)(NC(=O)C=CC2(C)COC2)C1 C(c1cc(Cl)ccc1OC)=CC(=O)NCC(CCNC(C=C(COC)C)=O)(C)C C1(NC(CSCC=C)=O)CC2CC(NC(c3cnn(CC(F)F)n3)=O)C1C2 C1(NC(C2(C)CN(C(=O)Cn3ccnn3)C2)=O)CCOCC12CCC2 c1(CC(=O)N(C(C)C(=O)NCC(c2ccco2)O)CC)cc(C)on1 N1(C(C(CCC)CNC(c2c[nH]c3cccnc23)=O)=O)C2CCC1CC(CO)C2 c1(C(N(CCC(C(C)C)NC(C(CCC)(C)O)=O)C)=O)cc(S(C)(=O)=O)oc1C c1(CC(C(=O)NCCC(=C)CNC(C2(n3cncn3)CC2)=O)C)cccc(F)c1 N1(C(CNC(CCC)=O)=O)CC2ON=C(CNC(=O)CCn3ccc(C)n3)C2C1 C(=O)(C(C)(C)CC(C)(C)C)N1CCC(NC(COc2ccc(C)cc2C)=O)CC1 C1(CN(C(=O)Cc2cc[nH]c2)C)CCCN(C(=O)CC2C=CCCC2)C1 c1(C(N(CC(C)NC(c2nnc(C(C)C)s2)=O)C)=O)cc(C#N)c[nH]1 C1(CNC(CCC2(C)CC2)=O)CN(C(=O)C(C)C(C)(F)F)CCC12CCOCC2 C(CO)(CCCCNC(=O)CCC1CCC(O)CC1)NC(CC(C)F)=O c1(CC(=O)NC(CCN(C(C=C(C)C)=O)C)C)cn(C)c2ccccc12 C1(C(N2CCC(CNC(C(N3CCC(O)CC3)C)=O)C2)=O)CCC2(CCC2)CC1 C1(CC)CN(C(C23CCC(CO)(CC2)C3)=O)CCN1C(c1ccncc1)=O c1(C(=O)NC2CCN(c3nc(CC)cc(CC)n3)C2)ccc([N+](=O)[O-])cc1C C1(C(=O)OC)CN(C(=O)NCc2cccc(NC(C)C)c2)CCS(=O)(=O)C1 N1(C(c2n(C=C)nnc2)=O)CCOCC1(C)C CC1=C(C)CN(C(C2(CNC(C34CCCC3C4)=O)CC2)=O)CC1 c1(C2(CN3CCC(C)(c4onc(C)n4)C3)CC2)ccc(Cl)c(Cl)c1 CC(C)(C)C#CCCNC(C1CC(O)CN1C(=O)Cc1cnns1)=O C1(NC(c2cnn(C)n2)=O)CCC(F)(CNC(=O)COC2CCCOC2)C1 c1(C(=O)NCC=CC)cc2c(cnn2C)nc1C Cc1cnc(N2CC(=C(F)CNC(C3CC(CC(F)F)C3)=O)C2)nc1 c1(CNC(=O)NC2CCN(CC(=O)OCC)CC2)cnc(C#N)c(Cl)c1 n1(CCC)ncc(C(=O)NCC2CCCC(NC(C3(SC)CC3)=O)C2)c1Cl c1(NC(N(C2CCN(C)C2=O)C2CC2)=O)ccnc2c(C(F)(F)F)cccc12 c1(CN2CCC(NC(c3cc(C)nn3C(F)F)=O)C2)ccc(F)c(C#N)c1 c1(C(N2CCC(CNC(CCCNC(=O)OC)=O)C2)=O)nnccc1C c1(C(=O)NC(C(C)C)C(=O)NC2CC=CC2)ccc(=O)n(C)c1 c1(C(CNC(C2C3CCC23)=O)NC(CC2(OC)CCC2)=O)ccc(C)cc1 C(=O)(CC(=O)NCC(C)(C)OCC(=O)NCCCC1CCOC1)N(C)C N1(C(c2ccn(CC)n2)=O)CCC2(CNC(=O)CNC(=O)C3CC3)CCCCC12 c1(SCCSC)ccnc(Cl)c1.C(=O)(C(F)(F)N1CC(N)C1)C(c1ccccc1)=O c1(C(=O)NC(CNC(C23CCCC2C3(F)F)=O)C2CC2)ccc2cc[nH]c2c1 C1(C(=O)NCCC2(NC(C3CC(CC(=O)OC)C3)=O)CC2)CCCOCC1 N1(C(C(=O)NCC(=C)C)C(C(C)CC)OC)CCC(C(C)(C)C)c2ccccc21 N1(C(C)=O)CC2(CCC2)CCC1CNC(c1csnn1)=O CCC(C)CC(C(=O)NCC12CCC(CC1O)C2)NC(=O)CC1CC(N(C)C)C1 CCCC(C(=O)NCC1CC1CC(=O)NCC1C(C)(C)C1(F)F)N(C)C CCCCC(CNC(=O)C(c1cnn(C)c1)O)NC(=O)C(COC)COC C(CC(C)P(C)(C)=O)NC(C1(C=C)CCC1)=O C(CCCCCC1CC1)NC(C1(NC(C2N(CCC)CCC2)=O)CC1(C)C)=O CC(C(C)(C)O)N(C)C(C1(NC(=O)CCOC2COC2)CC(CO)C1)=O c1(C2(C(=O)OCC(c3cccc(Br)c3F)C)CCC2)cc(Cl)ccc1F N1(C(CC(=O)NCC#C)=O)CC2CCCC(NC(=O)C(C#N)C(C)C)C2C1 N1(CC(C)C)CCc2nc[nH]c(=N)c2C1.N12CC(Cc3ccccc3)(C1)C2=O N1(CC(COc2cccc(C)c2)O)C2CCC1CC(C(C)(C)O)C2 C(=O)(C(C(C)NC(c1cc2cccnc2[nH]1)=O)C(C)C)NCC(CSC)OC c1(C(N2CCCC(N3CCCCC3)C2)C(=O)NC(C)C)ccc2c(c1)CCCO2 Cc1ccc(C(N2CC(NC(=O)CN(c3ncccn3)C)C3CC23)=O)cc1F O(NC(=O)C(C1CC1)N(C(=O)CCC=C(C)C)C)C(C(=O)OCC)C c1(C(=O)NCC(C)CNC(C2CSCCS2)=O)cc(CC2CCC2)c[nH]1 CC(=O)C(C)(C)CC(=O)NC(C(=O)Nc1ccc(C)c(CO)c1)c1ccco1 N1(C(C=CC(CC)C)=O)CCC2CCC(NC(c3cnn(C)c3C(C)C)=O)C1C2 c1(C(=O)NC(CNC(COCC#C)=O)CC=C)cc(OC)cc2c1NC(=O)CO2 CC1CN(C(c2cc(CCNC(C3(C#N)CCC3)=O)on2)=O)CCN(C)C1 C(=O)(C(COC)COC)NCCC1(C(N(CC#C)CCF)=O)CCCC1 C1(OC)CCCC(CC(=O)N(C)CCN2CCN(C(=O)CCCC#N)CC2)C1 c1(OC)ccc(C(=O)NC2CCN(C(=O)CN3CCS(=O)CC3)C23CC3)c(Cl)c1 c1(C(=O)NCC(CNC(C(C(C=C)C)C)=O)(C)C)ccc(OC)c2occc12 c1(C(=O)NC(C2CC(NC(C3CC4CCC4C3)=O)C2)C)ncccc1CO c1(C(N(CCCNC(C2(C)CCOC(C)C2)=O)CC)=O)ccc2cnc(C)n2c1 C1(C(=O)N(CCC(C)NC(=O)Cc2cncs2)C)(OC)CCC(C)(C)CC1 C(CCCC(C)NC(C1(c2cccc(F)c2)CC1)=O)NC(C(C)SCCCC)=O C1(CC(=O)NCCn2cc(CNC(C(COC)C)=O)nn2)Cc2ccccc2O1 C1(NC(COCC(=O)NC)=O)CC2(C1)CN(C(c1[nH]c(C3CC3)nc1C)=O)C2 O=C1NC(C(=O)NC2CC(CCNC(=O)CCNC(c3ccncc3)=O)C2)CO1 C1(C(=O)NC(C(C2CC2)OC)C)CN(C(=O)C(C)NC(C)(C)CC)CCO1 c1(SCOC)ccc(NC(C2CC2C(=O)Nc2sccc2C(N)=O)=O)c(Cl)n1 N1(C(C(c2ccccc2Cl)N(C)C)=O)CC(NC(=O)C2CC2)C2(CCC2)C1 c1(C(N2CC3C(NC(CCC=CCC=C)=O)(C3)C2)=O)cccc2[nH]cc(Cl)c12 S(=O)(=O)(c1cccc(Cl)c1C)N(C)C(c1c(Cl)cc(F)cc1Cl)=O.C12CN(C1)C2 N1(C(C(c2cc(F)cc(F)c2)C)=O)CCC(F)C(NC(C2(NC(N)=O)CC2)=O)C1 N1(C(CN(C(=O)C(F)C2CCC2)C)=O)CCN(C(c2ccc(O)cn2)=O)CC1 c1(OCC(=O)NCC2(C)CCN(C(C(CCC)OC)=O)C2)cc(C)c(Cl)c(C)c1 c1(C(C)C)cc(C(=O)N(C(C(=O)NCc2ccccn2)C2CC2)C)n[nH]1 c1(SC)onc(C)c1CC1C(=O)O1.C1(C)(C(=O)OC(C)(C)C)CCOC1 N1(C(C(CC#C)CC#C)=O)CCC2(CCC2)C(CNC(C2C3CNC(=O)C23)=O)C1 C(CCC)(c1nnnn1CCC1CC1)C1CC1.c1(C2C(CNCCC)C2)ccccc1 Cc1nsc(C(=O)NC2CCC(N(C(=O)C=Cc3ccc(C(N)=O)o3)C)C2)c1N c1(C(N2CC(C)N(C(=O)C=Cc3ncco3)CC2)=O)cncc2[nH]ccc12 C(=O)(C(F)(F)C(O)C(C)C)NCCCCCCN(C(CCc1cc(C)[nH]n1)=O)C C1(OC)CC(NC(c2sccc2C#N)=O)CN(C(c2c(C)[nH]c(C)c2C)=O)C1 Cc1cn2nc(C(N3CC(NC(=O)CCC4(C)CC4)C4(CC4)C3)=O)cc2c(=O)[nH]1 c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)CC2C)cccc2c1COCC2 C1(C(=O)NC(c2nccs2)CC)CCN(C(=O)CC23CCCC2C3)CCO1 N1(C(c2snc(C)c2N)=O)CC2CC(C1)N(C(=O)C(C)Cc1cnn(C)c1)C2 N1(CC)CCOCC1CC(=O)NC1CN(C(C23CC(CCO2)C3)=O)CC1SC N1(C(C(CC)C)=O)CC2CC(O)C1C2NC(c1sc(C2CCC2)nc1C)=O N1(C(C(=O)NCC)=O)CC(C)(C)CCC1C(=O)NC1C2CCC(C2)C1COC C1(NC(C(C)NC(N)=O)=O)CN(C(c2csc3cccnc23)=O)C2(CCCC2)C1 N1(C(C(C)C#N)=O)CCCC(NC(c2cc(C(F)(F)F)ccn2)=O)C1C C(=O)(C(C)CC(C)(F)F)N(C1CCN(C(c2nccc(C)c2O)=O)CC1)C c1(NC(C)=O)cccc(N(C)C(=O)NCC23CCCCC2C3)n1 CC(N=[N+]=[N-])C(=O)N(CC(=O)NOC(CCCF)c1nn[nH]n1)C1CC(C#N)C1 c1(C(=O)OC)c(C)cc(C)nc1NC1CCN(C(=O)C(C)C2CC2)CCC1CO C(=O)(C1=NNC(=O)C1)NCC(C)N(C)C(C1CCOC1)=O n1(CC(=O)NCCNC(CCN(C)CC)=O)nc(C)cc1C N1(C(C(COCC)N=[N+]=[N-])=O)CC2(CCC2)CC1C(=O)NCC1CCC(=O)N1C N1(C(c2ncc(OC)cn2)=O)CCC(NC(=O)C=CCN2CCCC2)C(C)C1 c1(CC)noc(C)c1C(=O)NC1CCC(N(C(=O)Cc2ccc(Cl)cc2)C)C1 c1(C(c2nnnn2C2CC2)NC(c2cc(Cl)cc(Cl)c2F)C)ccccc1[N+](=O)[O-] N1(C(c2c(CC)nn[nH]2)=O)C2COCC1CC(NC(c1cc(C)[nH]n1)=O)C2 N1(C(C2(CC#C)CCC2)=O)CCC(NC(=O)CCC2CCCN2C)C(C)C1 C=CCC(CC)C(=O)NC(CNC(C1CC2CCC(C1)S2)=O)(CC)CC c1(-c2nnc(NC(N3CCC(CC(=O)OC)CC3)=O)o2)c(F)cc(F)c(Br)c1F C1(C(=O)NCC2(NC(c3ccc(C)cc3F)=O)CC(OC)C2)CC2(C1)CC(C)C2 C(N=c1[nH]c(=N)[nH]c(=NC2CCN(C3CCCCC3)C2)[nH]1)c1nc(C)oc1C C=C(C)C(O)CC(=O)NC1CCCN(C(=O)CCCc2ccc(CC)cc2)C1 C1(C(=O)NC2CC(C(=O)NCC(C)C(F)F)C2)CC(=O)C12CCC2 c1(C(=O)NCCN(C(C2CC2c2ccccc2F)=O)C2CC2)cc2[nH]ccc2s1 C(=O)(C(O)CC(C)C)NC(CC)CN(C(=O)C(CN(C)C)c1ccccc1)CC c1(OC)ccc(F)c(C(N2CCC(NC(c3sccc3OC)=O)C(F)C2)=O)c1 CCS(=O)CCC(=O)N1CCC(NC(C2(O)CCCSC2)=O)C1 C1(NC(C=CC(CC)C)=O)CCN(C(c2cccc(Cl)c2N)=O)C1(C)C N1(C(CC(=C=C)C)=O)CCN(C)CC1C(=O)NCC(=O)NCCc1ccc(C)s1 C1(CC=C)(C(=O)NC2CCC2(C)C)CCCN1C(=O)C(n1ccnc1C)C N(C1c2ccccc2CCC1c1ccsc1)C(C(=O)Nc1ccc(N)cc1)=O N1(C(C(CC)(C)O)=O)CCOC2(CCN(C(c3ccc(N(C)C)cn3)=O)C2)C1 c1(C(=O)NC2C3CN(C(CC(CC)C4CC4)=O)C2C3)cccc2nc[nH]c12 N1(C(Cc2ccc(OC)cc2)=O)CCC(C2CCCN(CC(O)COC)C2)C1 Cc1ccc(C(C)C(=O)N(C(C)CCNC(=O)C=C2CCOCC2)C)s1 N1(C(C2(C(C)C)COC2)=O)CC2CCCC2(C(=O)NC2CNC(=O)C2)C1 C1(C(=O)NC2(CC)CCCC2)(CC)CCCN1C(=O)COCc1nnc(CC)o1 c1(OC)ncccc1C(=O)NC1CCN(C(C23CC(CO)(C2)C3)=O)CC1 CCCCC(C(=O)NCC1CCN(CC)C1)NC(=O)CC(CC)C1CCC1 C(=O)(C1Cc2ccc(F)cc21)NCC(C(C)C)NC(=O)CN(CCO)C1CC1 C(c1c(C)coc1C)=CC(=O)NC(CNC(c1c(CC)ncs1)=O)(CC)CC c1(C(C(=O)NC(CC(=O)OCC)Cc2ccccc2)C)cn(C)nc1CC c1(OCC)ccc(CNC(C2CC(NCc3ccc(Br)cc3Cl)C2)=O)cc1Br c1(NC(C(C2CC(NC(CC(C)O)=O)C2)F)=O)cccc2c1OCC2 CC1(C)CN(C(=O)CN2C(=O)CNC2=O)CC(CNC(C2CCCO2)=O)O1 c1(CN(C(=O)CC(c2ccccc2)OCC)CC=C)ccncc1 CCC(CC(=O)NCC1(CCO)CN(C)C1)NC(c1cn(C)nc1C)=O N1(C(=O)NC(c2c(O)cc(C)c(Cl)c2)C)CCc2ccc(C#N)cc2C1 c1(OC)ncc(F)cc1C(=O)N(CC(C)CNC(=O)COc1ccc(F)cn1)C C1(NC(C=C(C)C(C)C)=O)CCC(C)(CNC(c2ccc(F)cc2)=O)C1 CCC(C)(C)CC(=O)NC1CCC1CNC(c1cc(C(F)F)cs1)=O CC1CN(C2CCOCC2)CCN1N1CCCC1CC1CC(c2ccccc2)C1 N1(C(c2cccc(CC)n2)=O)CC2CCN(C(c3cccc4nccn34)=O)C2C1 C1(CNC(COC(CNC(C2(CC=C)CC=CC2)=O)(C)C)=O)CCOC1(C)C C1(C(=O)OC)(OC)CCCN(C(=O)C(c2cccc(Cl)c2F)NC(C)=O)C1 N1(C(CC2(C#N)CCCCC2)=O)CCC2(CCC(NC(c3cn[nH]c3)=O)CC2)CC1 c1(NC(C2OCCN(C(c3n(CC)ccc3)=O)C2)=O)ccc2c(c1)CCO2 N1(C(C(CC)C(F)(F)F)=O)CCN(C(c2cc3n(n2)CCCO3)=O)C2(CCC2)C1 C=CC(C)(CCOC)C(=O)NCCN(CCC)C(c1cc(C(F)F)cs1)=O C1(NC(Cc2n(C)nnc2)=O)CN(C(=O)CS(C)(=O)=O)CCC1O C1(NC(CC(C)(C)OC)=O)CCc2nc(=N)[nH]cc2C1 c1(NC(C(N2CCCC(C(=O)NCCCC)C2)=O)=O)cc(O)nc(C2CC2)n1 CC1CN(C(=O)CSCC2CCCO2)CCC1CNC(c1ccnc(Cl)c1)=O C1(NC(C2CC(OC)C2)=O)(CNC(c2csc(C)c2)=O)CCCCC1C N(C(=NCC1CCCOC1)NCC1(C(N)=O)CCC1)C(CC)C CC1C(NC(c2cccc(SC)n2)=O)CCCN1C(=O)CCCOC(=O)C(C)C c1(CC(=O)NCC2(NC(CCCOC)=O)CCCCC2C)csc2sc(C)cc12 C1(CNC(C=CC(=O)OCC)=O)CC(C)(C)CN1C(=O)CC1CC(C)C1 n1(CC(N2CCC(C(C)(C)NC(C3(F)CC=CC3)=O)C2)=O)ncc2ccccc12 C12(C(=O)NC(C(CCC)C)C)CCC(CC1)N(C(c1cc(C)n(C)c1)=O)C2 C(=O)(CC(C)n1cc(Br)cn1)NCC(C)NC(CCN(C)CC)=O C1(C(=O)NCCC(C)N(C)C(C2COCCN2C)=O)CC2C=CC1C2 c1(C(=O)NCC=C)cccc(-c2cnc(N3CCCC3C(=O)N(C)C)nc2)c1 c1(-c2c(C(=O)Nc3c(C)ncc(C#N)c3)ncnc2)cccc([N+](=O)[O-])c1O Cc1ccc(C2(C(=O)NCCCC(C)NC(c3nc(C)oc3C)=O)CC2)cn1 O=S(=O)(c1cccc(=NC2CCSC3(CCC3)C2)[nH]1)N1CCC(O)C1 c1(C(=O)NCCN(C(C(COC)C)=O)C)ccc(OC2CCCC2)cc1 c1(CCCC)nc(C)c(C(=O)NC(C2(CNC(=O)C(O)CCc3ccccc3)CC2)C)s1 C(=O)(CCCC(F)(F)CO)NC(CCNC(C1CCN(C(CCC)=O)C1)=O)C C(=O)(C(O)C(F)(F)F)NC(C(=O)NCC1(C)CCOCC1)CCC1CCC1 c1(OC)c(NC(=O)C=C2CCN(Cc3c(F)cc(O)cc3F)CC2)cc(Cl)cc1Cl Cc1nc2cc(C(N3CC(Nc4ccccc4)C3)=O)[nH]c2s1 c1(C(N2C(CC(=O)Nc3nccc(Cl)c3Cl)CCC2)=O)c(Br)cncc1F Cc1nc(O)[nH]c1C(=O)NC1(CNC(C2CCCC2n2cccc2)=O)CCOC1 c1(CC)c[nH]nc1C(=O)NC1CC(NC(C2CCC(NC(=O)OC)C2)=O)C1 CC1CCC(CNC(=O)CCc2cscn2)N(C(=O)C(C2CCC2)C2CCC2)C1 C(C(C)(C)C(F)(F)F)NC(C(c1ccnn1C)NC(C=CC(C)N(C)C)=O)=O S(=O)(=O)(c1ccc(NC2CCC(O)CC2)cc1Cl)N(CC(C1CCCC1)OC)C C12(CN=C(NC3C(OCC)C3)NC(C)C)CCCC1C2(F)F C1(NC(CNC(CC)=O)=O)CCCC(C(N2CCCC2(C)C(=O)NC)=O)CC1 c1(C(=O)NC2(CNC(C(C)C#N)=O)CCOCC2)cccc(F)c1F Cn1cc(C(=O)NCCC2CCCN2C(=O)COC2CC=CC2)c(O)n1 C1(NC(C2C(OC)CC2)=O)CCN(C(C2CN3CCN2C(C)C3)=O)CC12CCC2 C1(CCC(=O)NCCC#CCC)CCCCN1C(c1cc(C)nn1C)=O N1(C(C(C)NS(CC)(=O)=O)=O)CCC(c2cn(C3CCCCC3)nn2)C12CC2 N1(C(CC2(OC)CCC2)=O)C2CCCC1CC(NC(c1ccnn1C(C)C)=O)C2 C1(CC)(NC(c2nnn3c2CCC3)=O)CCCN(C(=O)CCOC2CC2)C1 N1(c2c(C#N)c(O)cs2)CCCC2(CNC(=O)CSc3ccccc3)CCCC12 N1(C(COCCCC)=O)CCCC(F)(C(=O)NCC2CCCS2(=O)=O)C1 c1(OC)ccccc1-c1csc(-c2nc(-c3cccc(NC(C)=O)c3)no2)n1 C1(C(=O)NCCC2C(C)C2)CNC(=O)CN1C(c1ccncc1N)=O c1(C(=O)NC(c2cccs2)C)c[nH]c2ccc(-c3scc4c3OCCO4)cc12 N1(C(C(C)C#N)=O)CC(CNC(=O)C=Cc2cc[nH]n2)CC(C)(C)C1 CC(C)C(O)C(c1ccccc1)NC(c1ccc(CC(C)(C)O)s1)=O C12(C(=O)NCc3cc(OC)ns3)CC1CCN2C(C1CC(O)C(F)C1)=O CS(=O)c1ccccc1C(N1CCC2(NC(c3cc(C#N)c[nH]3)=O)CCCC12)=O c1(CC)ccccc1CC(N1CCC(C(C)NC(c2ccc(CO)nc2)=O)C1)=O C1(C(=O)NCc2ccc(C(N)=O)o2)COCCC1NC(C1(O)CCSCC1)=O C1(NC(c2c(C)ccs2)=O)CN(C(=O)C(N)=O)C2(CCOC2)C1 CCC(C(=O)NCCCCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O)NC(C)=O CCC(C)C(O)C(=O)NCC1(NC(=O)CC2COC(C)(C)CO2)CCCCC1 c1(CN2CC(C(=O)Nc3c(OC)cc(O)cc3)OCC2)n[nH]c2ccc(Cl)cc12 C1(O)(CNC(=O)CC2(O)CCC2)CCN(C(c2cnnc(Cl)c2)=O)C1 N1(C(c2ccc(Cl)cc2Cl)=O)CCC2CN(c3cc4ncnn4cn3)CCC12 C(N=c1[nH]cnc(Cl)c1F)C1CCC(NC(c2c(C)nc(CC)o2)=O)CC1 C=C(Cl)C(C)(C)C(=O)NCC1CN(C)CCN1C(c1nncn1CC)=O c1(CC(=O)N(C(C)C)CCN(C(=O)COC2CCCC2)C)cc(F)cc(F)c1 C1(CC(=O)Nc2c(OCCOC)cc(O)cc2)Cc2cc(F)ccc2O1 C#CC1(O)CC(C(=O)NC2CCN(C(=O)C(C(C)C)c3cccc(Cl)c3)C2C)C1 c1(C(C(=O)NCCOCCCN(C(C2C(C=C)C2)=O)C)CC)c(C)noc1C C1(CCC)(NC(=O)C(C2CC2)OC)CCCN(C(C2CC(F)(F)C2)=O)C1 C1(CC)CC(CC(=O)NCCC(C)(C)CNC(=O)Cc2ccsc2)CCO1 C1(CNC(C2=C(C)OCC2)=O)CCC2(CN(C(C3CCCN3C=O)=O)C2)O1 N1(Cc2c(F)ccc(C)c2Cl)CC(C)Cc2cccc(F)c21 CCCCC(CNC(C1(C)CCCOC1)=O)NC(=O)C(C)CCc1ccccc1 c1(N(C2CCC2)C(N(c2ccccc2)C)=O)cccc(C(F)(F)F)c1Cl c1(C(=O)OCC)cc2cc(NC(c3ccc(I)cc3O)=O)cnc2[nH]1.C12(CC1)CN2 CC1CCC(C(N2CC(F)(CNC(C34CC(F)(C3)C4)=O)C2)=O)C1 c1(C(=O)NC2CCC(CNC(Cc3scc(C)c3)=O)C2)cnc(O)cc1C C(C(C)(C)S(C)(=O)=O)NC(=O)NC1(c2ccc(Cl)c(Cl)c2)C(C)C1 C1(CCNC(COC(C)(C)C)=O)CN(C(C2(C)CC=CCC2)=O)CCS1(=O)=O N1(C(C2(C3N(C(C)=O)CCC3)CC2)=O)CCC(NC(=O)Cc2cncs2)CC1 c1(CNC(=NCC(C)C)NC2CC2NC(C)(C)C)ccc2c(c1)C(=O)NCC2 c1(C(=O)NC2CC(C)(NC(C(CC)N3CCCC3=O)=O)C2)nnn(CC)c1C c1(-c2nc(C3CCC(=O)NC3)nn2CCF)ccc2c(n1)CCCC2 N1(C(CC2C(C)(C)C2)=O)CCCC1Cn1cc(C(C2CC(F)(F)C2)O)nn1 N1(CC)CCCC1C1CCCN1Cc1ccc(N)c(C)c1 CC1CCN(C(=O)CCc2nncn2C)C(C(=O)NCC2CC2(C)C)C1 Cc1cc(CN2CC3C(C(=O)NCCCN4CCOCC4)C3C2)c2cc[nH]c2c1 c1(C(=O)NC(C(=O)NC2C(C)CCC2C)Cc2ccoc2)cn(C)ccc1=O C(C(C(=O)NCC#CC1CC1)NC(c1cc[nH]c1)=O)OCC C1(C(=O)NC(CCN(C(CC(CCC)O)=O)C)C(C)C)CCC2CC(C)CN2C1 C1(C(C)C(N2CC=CC2n2cccn2)=O)CCCN(C(C2COCC2(C)C)=O)C1 C(=O)(CCCCC#N)N1CCC(C2N(C(Cc3cnc(C)s3)=O)CCCC2)C1 N#Cc1cscc1C(=O)NC1(CNC(=O)CCOc2ccccc2Cl)CC1 C(=O)(C#CC1(C)COC1)NC(CCCOC)C(=O)NCP(C)(C)=O C1(C(=O)OC)CCCCCCN1C(C12CC(CN(C(=O)C(=O)C(C)(C)C)C1)C2)=O CC(COC1CCCO1)C(=O)NC(=O)NC1CC=CCC1 CCC(CC(=O)N1CCCC1C(=O)NCc1cc(OC)ncn1)C1CCC1 CC1(C(=O)NC(C2CCOC2)CNC(=O)C2=NNC(=O)C2)CCS(=O)(=O)CC1 c1(C(N2CC(CC(C)NC(c3cn4c(n3)SCC4)=O)C2)=O)ccc(F)cc1O CCCCC(C)C(=O)N(CC(=O)Nc1cncc(F)c1)C(C)C c1(C(=O)NCC(C2CCOC2)NC(Cc2nc(C)oc2)=O)nsc2ccccc12 C1(CNC(C(C(C)C)NC(C)=O)=O)CCC2(CCNCC2)CO1 Cc1cc(CNC(=O)CCN(CCO)C(C2COCC(C)O2)=O)oc1C C1(C(N2CCCC(CC=C)C2)=O)CCC2CCC1N2C(c1cn2c(n1)CCC2)=O Cc1oc(C)c(C(=O)NCC(C2CC2)NC(C2CCCN2C(N)=O)=O)c1C N1(C(c2c(C)nn[nH]2)=O)CC(NC(C2CC2OC(C)(C)C)=O)CC2(CC2)C1 c1(CC(=O)NC2(n3ccnn3)CCOCC2)ccc(Oc2ccccc2)c(Cl)c1 C1(C(=O)NCc2ccc(O)cc2C)(CC)CCCN(C(C2CC(C)=NO2)=O)C1 C1(COC)(NC(C2CC(C(=O)NCCc3ccsc3)C2)=O)CCCC1 Cc1cc(N2CC(C)OC(C)C2)ncc1S(=O)(=O)N(C)Cc1ccc(Cl)cc1Cl C1(NC(c2scc(C)c2)=O)CN(C(C2COCCC2(F)F)=O)C2CCCC12 CC(C)(CCNC(=O)CC1CCC(=O)C1)C(=O)NCCCN=[N+]=[N-] c1(C(=O)NC2CC3CC(NC(=O)CC4CC=CCC4)C2C3)cc2sccc2cn1 CC1CCCN(C(c2ncc(F)cn2)=O)C1CNC(=O)Cn1ccccc1=O C1(C(N2CCCC(C)C2)=O)CN(C(c2ccnc(CO)c2)=O)CC(C)(C)C1 CC1CN(C(=O)Cn2cccn2)CC(C)N(C(=O)Cn2ccnc2CCC#N)C1 CCC(C)CCCCC(=O)NC(C)CN(C(c1ccc(P(C)(C)=O)cn1)=O)CC Cc1nn(CC(=O)NCC2CC(NC(C3C(C)(C)C3(F)F)=O)CCO2)c(C)c1C N1(C(C(c2cnn(C)c2)OC)=O)CC(NC(c2cnc(O)cc2C)=O)CC(O)C1 Cn1c(CCNC(c2cc([N+](=O)[O-])c[nH]2)=O)nc2cc(Cl)ccc12 N1(C(C2(C(=O)NC)CCC2)=O)CCC(F)(F)C(CNC(C2CC23CCC3)=O)C1 C1(NC(C(COC)OC)=O)CCCCC1NC(=O)COCC1CCOC1 c1(C(N2CCC(C(=O)NCc3c(CC)c[nH]n3)(C(C)C)C2)=O)cnc2n1CCC2 c1(-c2cn(CC3N(C(C4C=CCC4)=O)CC=C3)nn2)ccc2ccccc2c1 C#CCCC(=O)NCC(O)CNC(=O)CC1CC(F)C1 c1(CC)nn(C)c(C(=O)NCC(C)NC(c2ccn(C)c(=O)c2)=O)c1Cl N1(C(Cc2nccc(OCC)n2)=O)CCC(NC(=O)C(CCO)N(C)C)C1(C)C Cc1nc(C(=O)NCCC(O)CNC(C2(O)CCSCC2)=O)c(C)o1 c1(COC)nn(C)cc1C(=O)NC1CCC1NC(c1cccc(C(F)F)c1)=O C1(C(N2CCC(CNC(C3CC(SC)C3)=O)C2)=O)CCCC(C)(C)C1 C(=O)(C1CCc2cc(Br)ccc21)N(CCCNC(C1C(C)OCCC1)=O)C c1(CC(N2C(CN(C)C(C3CCC(=O)N3)=O)CCCC2)=O)cc(F)c(F)cc1F c1(CCC(N2CCC(C(C)NC(CCOCCC)=O)C2)=O)ccc(N)nc1 N1(C(C(C)OCCCC)=O)CC2(CC(NC(=O)CCNC(=O)NC)C2)C1 C(=O)(C(C)(CC)CCC)NCC(CCNC(CC=C=C)=O)O c1(C(N2C(C(=O)NC(c3c(OC)cccc3)C)CCC2)=O)ncc(F)cc1C C1(C)(NC(C2(OC(C)=O)CC2)=O)CCN(C(=O)CC2CCOC(C(C)C)C2)C1 N1(C(C(CC)N(C)C(C)=O)=O)CCC2(CC1)CC(Nc1ccc(Cl)cc1C)CO2 Cn1cc(Cl)cc1CC(=O)NC1C2CC(NC(C3CC(C)(F)C3)=O)CC12 C1(CC)(CO)CCCN(CC(=O)N(C)C)C1.C(C)(C)(C)N(C)C(=O)O Cc1c(C(N2CC(NC(C34CC(CCO3)C4)=O)C2)=O)sc2ccc(Cl)cc12 c1(C(N2CCC(OCCNC(CCC)=O)C2)=O)cn(C)cc1C N1(C(c2c(C)scn2)=O)CCC2CN(C(=O)CCC3CCCCN3C)CCC12 C12(CCNC(CC(C)(C)OC)=O)CCC(CC1)N(C(C1CCOC1C(C)C)=O)C2 C1(C(N2CCOCC(NC(c3c(C)ocn3)=O)C2)=O)CCC(S(N)(=O)=O)CC1 CC1CCc2nc(N(CC(=O)N(C)C)C)[nH]c(=NC3CN(c4ncco4)C3)c2C1 c1(C(=O)NCC2OCCN(Cc3scc(C)n3)C2)cc2n[nH]cc2cc1Cl CC(C)C(C(=O)N(CC(C)(C)C#N)C)C(C)NC(=O)CCCn1cccc1 C(=O)(C1CCCc2ncccc21)N1CCC(CNC(C2CCOC2)=O)C1 C1(CNC(Cc2nc(C)oc2)=O)CCC(F)(NC(c2nn(C(F)F)cc2Cl)=O)C1 c1(OCCOC)cccc(CC(=O)N(C(C)CNC(=O)C=C(Cl)Cl)C)c1 N1(C=O)CC(S(C)=O)C1.C1(CNC(=O)OC(C)(C)C)(CF)CC1(F)F C(=O)(CCC(C)OC)N1CC(C(N2C(C(=O)NC)C=CC2)=O)(CC)C1 CC(C)CC(CNC(=O)CC1CCCOC1)NC(=O)C(C)CO c1(CC(=O)NC2CCN(C(C3CC3F)=O)CC2)ccc(Cl)cn1 CC12CCC(C(=O)NCC3(CN=c4nc[nH]s4)CC(F)(F)C3)(CC1)CO2 CC1(C)C(CNC(=O)C(F)F)CCN1C(C1Cc2nncn2C1)=O c1(C(=O)NCC2C(CNC(C(CC)C(C)(F)F)=O)C2)ccc([N+](=O)[O-])cc1C CCC(C)CCC(O)CC(=O)N(CCCCCCNC(=O)C1=CCCS1)C C1(CNC(C2(OC)CCC2)=O)CCCCN(C(C23CCC2C3)=O)C1 c1(C(=O)NCC2(O)CC(NC(C(C)=C3CC3)=O)C2)cnc(OCC(F)F)c(Cl)c1 Cc1cc(F)ccc1C(O)C(=O)NCCCC1(NC(c2cnc(S)[nH]2)=O)CC1 c1(C(=O)NCC2CN(C(C)=O)C(C)(C)C2)ccc2c(c1)C=CS2(=O)=O CC1(C(=O)NC2CC(NC(=O)C(O)Cc3ccccn3)CC2O)CCCCO1 C(=O)(CC(C)(C)CNC(C1OCCCC1(C)C)=O)NC(CC=C)CO C=C(Cl)CCC(=O)N1CCC(N(C(=O)C(C2CC2)OCC)C)CC1 C1(C(N2CCCC(N(C)C(c3cc[nH]n3)=O)C2)=O)CCC2(CC1)CC(O)C2 c1(OC)ccc(Cl)cc1S(=O)(=O)NC(=O)C(C1CCC(=O)N1)C CC(C)CC(CN=c1cc(C(F)(F)F)nc[nH]1)NC(C1CC1C1CCCCC1)=O CC1CCN(CC(=O)NC(CC2CCC2)C(=O)NCCCSC(F)F)C1 C1(C(=O)NC(CCNC(Cc2ccc(SC)cc2)=O)C)CCC(N=[N+]=[N-])C1 N1(C(C(C=C)CC)=O)CCC2(CC2NC(c2ccc(F)c(C)c2)=O)C1 C#CCCC(=O)N(C1CC1)Cc1cn(CC(C)NC(=O)C(C)(C)C)nn1 Cc1c(C(N2C3CCC2C(NC(=O)C(C)(C)CO)C3)=O)cc(O)cc1N Cc1cc(C)c(C(=O)NC(c2ccc(F)cc2)CNC(=O)CNC(N)=O)cn1 N1(C(CCNS(C)(=O)=O)=O)CCC(NC(=O)CC2CCCC2)C(C(N)=O)C1 C(=O)(CCCCCCC(C)C)NCCOC(CNC(C(CC(=C)C)C)=O)(C)C c1(CCN2CC(CNC(C(CN(C)C)O)=O)OCC2)nnc2ccccn12 n1(CC(=O)NC2CCC2CNC(c2ccsc2)=O)ncc2c1CCCC2 N12CCC(CC1C)NC(=O)CCOC2=O.C1CN(CCCC)O1.N(C)(C)CC C(C)(C(=O)NC1CC(NC(=O)CC2(O)CCC2)C1)NC(C)=O c1(C(=O)NCCCC(CCC)NC(c2cnsc2C)=O)ccn2ccnc2n1 CCCCCC(C)(C)C(=O)NC(CC)CC(=O)NC1(C)CCC(=O)NC1=O C1(C(=O)NC(CN)CO)(C)CC=CC1.C(C(C)=CC(=O)C1CC1)OC S(=O)(=O)(c1cc(F)ccc1C#N)NC1CCN(C(CC)CC)C1 c1(C(=O)NCCC(C)N(C(C(C)NC(C)=O)=O)C)cccc2nccn12 C1(NC(COCc2nnc(C)s2)=O)CCN(C(C2(CO)CCCCC2)=O)CC1(C)C C1(C(=O)NC(CCNC(c2ccc(C(CC)(C)C)cc2)=O)C)CCCCS1(=O)=O c1(OC)cccc2oc(NC(C3CCCCC3C)=O)cc(=O)c12 CCC(CC(=O)Nn1ccccc1=O)N(C(=O)CC1CCOC1(C)C)C CN1C(=NC(=O)c2cc3n(n2)CC(O)CO3)Sc2ccccc2S1(=O)=O CCCC(CNC(=O)Cc1ccns1)C(=O)NC(C)(C)CC(N)=O C1(CNC(C2(OC)CCC2)=O)CCCCN(C(c2cccc(CSC)c2)=O)C1 N1(C(C(c2ccnn2C)C)=O)C2CCC1CC(NC(=O)C(C1CCCCC1)=O)C2 C1(NC(C(c2ccccc2)SC)=O)CN(C(=O)CC2CC(F)C2)C2(CCC2)C1 c1(CN(CC(C)NC(CC2(C(=O)OC)CCC2)=O)C(C)C)cc2cnccc2[nH]1 CCC(C)C(C(=O)NCC(C)(C)OCC(=O)NCc1ccc(OC)nc1)OC Cc1cc(C2CC2)ncc1C(N1CCCN(C(=O)C(C)OCCN(C)C)CC1)=O C1(C)(NC(C(C)Cn2ccnc2)=O)CCCC1NC(c1cc[nH]c1C1CCC1)=O c1(C(N2CCN(C(C3=C(C)OCCS3)=O)C(C)C2)=O)cc2ccccc2cn1 N(C1CCCc2ccoc21)C(C1(NC(c2ncn(C(C)C)n2)=O)CC(CO)C1)=O c1(C(C(=O)NC2CCN(C(COCCOC)=O)C2)OC)cc(F)cc(F)c1 c1(CC)ncc(Cl)c(C(N2CCC(C3CCCN3C(C3(C4CC4)CCC3)=O)C2)=O)n1 S(=O)(=O)(CC(=O)NC1C=CC(CC(=O)NC(C)CCCO)C1)NC Cc1nc(Cl)ccc1CC(=O)NC1CCN(C(c2cc(O)no2)=O)CC1C CC(F)(F)C(C)(C)C(=O)NCC1CCC1NC(c1ccc(-c2cc[nH]n2)cc1)=O N1(C(C(CC)N(C)C)=O)CCC(NC(=O)COCCN(C)C)C(C(F)(F)F)C1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)N1CC(C)CN(C(C=C(C)Cl)=O)CC1C N1(C(c2c(C)nc(C3CCCO3)s2)=O)CCN(C(C2(CO)CCC2)=O)CCC1C CC(C)(C)C(CO)C(=O)NCC1CC(NC(=O)Cc2ccc(F)c(Cl)c2F)C1 C(CS(=O)(=O)CC(=O)N1CCC1CNC(=O)C(N1CCCCCC1)C)OC N1(C(=O)C)C(C)(C)CCCC1(C)C.Cc1ccc(-c2cn(CCC)nn2)cc1Cl C1(NC(CC=CC=C)=O)CCCC(C(N2CCC3(CSC3)C2)=O)CC1 O=C1CCCCC1Cc1cn(CCCCNC(=O)CC2CC3CCC3C2)nn1 N1(C(c2cc(C)ncn2)=O)CCC(C)C(CC(N2CC=CCC2)=O)C1 C(c1c(F)ccc(Cl)c1F)=CC(=O)NCCNC(c1cn(C(C)C)nn1)=O c1(OC)ccncc1CN1CCOCC1.C12CCCN1C(=O)CCCn1cc2nn1 CC12CCC(NC(=O)C(=Cc3cnc[nH]3)F)(CC1)O2 c1(OC)ccc(OC(=O)C(C2CC=CCC2)NC(C2CC(=O)CCO2)=O)cc1 C1(C(N(CCCNC(C2C(C=C)C2)=O)CCO)=O)CCCN1Cc1ccccc1 C(CC(C)(C)C(=O)N1CCN(C(c2ccc(C(C)(C)C)[nH]2)=O)C(CCO)C1)OC C1(C(=O)NCCN(C)C(C2CCOC2C(F)(F)F)=O)CC2OC(=O)OC2C1 C1(CS(=O)(=O)NC)CCN(CC2CC(=C)C2)CC1C c1(NC(C2(OC)CCN(C(CC3ON=C(C)C3)=O)C2)=O)cnc2[nH]ncc2c1 C1(C(C)NC(C2(C)CC=CC2)=O)CN(C(c2nn(C)cc2N)=O)CCO1 CC(C(=O)NCC1(O)CC(C(=O)NCC2SCCS2)C1)S(C)(=O)=O C1(NC(c2c(C(C)C)ncs2)=O)CC(NC(C2CCCC(C)C2)=O)C(O)C1 Cc1cccc(Br)c1CN1CC(CNC(=O)OC(c2nccn2C)=O)C1 c1(NC(=O)C2=CCC2)cccc(NC(C2C3CCCOC23)=O)c1 C1(O)(CNC(COCC(C)C)=O)CCN(C)CC1 N1(C(CSCC)=O)CCC2(CCC(CNC(c3ocnc3C(F)F)=O)OC2)CC1 C=CC1(C(N2CCC(OC3CC3)C2)=O)CCN(C(C2CC23CCC3)=O)CC1 c1(C(=O)NC2CC3CN(C(C4C(C)N(C)CC4)=O)C2C3)ncc(P(C)(C)=O)cn1 C=CCC(C(=O)NCCC1(NC(=O)C(O)C(C)C)CC1)C(C)C C(=O)(CC1OCc2ccccc21)N(C1CC(NC(CCC=C)=O)C1)C C1(NC(CCN(C(=O)CC2CCOC2)CC)=O)CCC2CC12 N1(C(C2(C)N(C(c3c(C)cc(C)o3)=O)CC(O)C2)=O)CCc2nc[nH]c2C1 Cc1cnn(C(C)C(=O)NCC2CC2NC(C2CC2c2ccc(Cl)s2)=O)c1 c1(C(N(CCCNC(=O)CC2CC(C(N)=O)C2)C)=O)cccc(=O)n1C c1(CNC(CC=CC)=O)cc2n(n1)CCN(C(c1cnc(CC3CC3)nc1O)=O)C2 c1(C(=O)NCCCCC2CN(C(C(C3CC3)SC)=O)C2)ncc2ccccn12 Clc1ccc(-c2cc(CSC3CC=CCC3)on2)cc1 C(=O)(C1=NOC2COCC12)N1CCOCC(CNC(CC(C=C)(C)C)=O)C1 C1(NC(C2(C)CCCOC2)=O)CC2CC1N(C(c1c[nH]nc1C1CC1)=O)C2 C1(NC(C(C(CC)O)C)=O)CC2CCCC(C1)N2C(=O)CCSc1ccccn1 C(=O)(C1=CCC2CCC1N2C(c1cncc(Cl)c1)=O)N(CC(CC)O)C C1(C)(CC(=O)NCC(CC=C)NC(=O)Cc2cnccn2)CCCCC1 C(=O)(NNC(=O)CCCCCCC(=O)OCc1ccc(OC)c(OC)c1)OCC c1(C(N2CC(O)(CNC(c3nc(CC)oc3)=O)C2)=O)n[nH]c2cc(OC)ccc12 C1(C(N(C)Cc2ccc(CC)o2)=O)CN(C(c2cnn(C)c2N)=O)C(C)(C)C1 C(C)(C(C(=O)N(CC(=O)NCC1COCC(C)O1)CC1CC1)N(C)C)OC n1(CCCC(=O)NC(CC)CNC(=O)CC2(C3CC3)CCCO2)c(O)nnc1O C1(C(=O)NCC2CCN(C(c3cncc(OCC)c3)=O)C2)CCc2cnnn2C1 C1(NC(C(C2CCOC2)OC)=O)CCCN(C(=O)CC2OC(C)(C)OC2=O)CC1 C1(OC)CC(CCNC(c2csc(O)n2)=O)N(C(=O)CCOCC2CCCO2)C1 C=C(C)CC(C(=O)N(CC(C)(C)CNC(C1CCC1C(=O)OC)=O)C)NC(C)=O C1(NC(c2c(CNC(c3nsnc3O)=O)occ2)=O)(CO)CC(F)(F)C1 N1(C(=O)NC2CCn3ncnc3C2)CC2(CC2)c2ccncc21 CN1C(=O)CCCC1C(N1CCCC(n2cc(-c3ccc(Cl)cc3)nn2)CC1)=O N1(C(=O)CN2CCN(C(c3cccs3)=O)CC2)CC2CCC(C1)C2O CC1(NC(c2ccc(C3CCOC3)cc2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)C1 N1(C(C(C)(C)C2CCOCC2)=O)CCCC(CNC(=O)CN2CC3C=CC2C3)C1 C1(CNC(=O)CN2CC3CC3C2)CCC(C(N2CCC3CC23)=O)CC1 C(=O)(C(Cc1cnc[nH]1)NC(=O)CC12CCCC1C2)NCC(C)OC(F)F N1(C(C(CC)SC)=O)CCN(C(C)CNC(C2CCCN2C=O)=O)CC1 C1(CC)(CC)CC(O)CN1C(=O)C(O)CNC(c1ccn(CC)c1C)=O C1(C(=O)NC2CC(CNC(COCC(=C)C)=O)C2)CCCCC(C)(C)C1 c1(C(=O)NCCC(F)Cn2cc(C3(C(=O)O)CC3)nn2)cnc(O)c2ccsc12 N1(C(CC(CCC)(C)C)=O)CCC2(CC1)CCN(C(C1(O)CCCC1)=O)C2 C1(C(=O)NCCCC2N(C(COCCCC#C)=O)CCC2)C(F)(F)C12CC2 c1(C(=O)NC(CNC(C2(CC=C)CC=CC2)=O)C)cc2ccc(F)cc2nc1O Cc1cc(C(=O)NS(=O)(=O)CC2CCCCCC2)ccc1N1CCCC1 C1(C(=O)NC2C(C)CCC2)CC2OCCC2N(C(=O)Cc2ccsc2Br)C1 c1(C(N2CC(NC(C(C(=C)Cl)(C)C)=O)CC3(C2)CC3)=O)ccc2c(cnn2C)c1 CC1CC(NC(c2ccc(F)c(F)c2)=O)CN(C(C2C(C3CC3)C2(F)F)=O)C1 c1(C(=O)NCC2C(NC(C3CC(N=[N+]=[N-])C3)=O)CCC2)cnn2c1OCCC2 CC1CC(C(=O)NCC(F)(F)CO)CN(C(=O)CC=CC(C)(C)C)C1 N1(C(c2c(OC)cc(=O)n(C)c2)=O)CCC2OCCN(C(=O)CSC3CC3)C2C1 N1(C(c2ccnnc2S)=O)CCC2C(C1)CN2C(=O)CC(c1cccc(F)c1)O C(c1ccoc1)=CCO.C12(C(C)NCCO)CC(CO1)C2 C12(NC(c3c(OC)nc(C)s3)=O)CCC(CN(C(=O)CC(C)n3ccnc3)C1)C2 c1(C(N2CCC(NC(=O)CCCn3ccnc3)C(F)C2)=O)cccc2[nH]ncc12 C1(CNC(c2cc(SC)oc2C)=O)CC2(CC2)CN1C(=O)CC1OCCC1(C)C N1(C(C(CSC)(C)C)=O)CC2(CC(CNC(=O)Cc3cc(F)ccc3C)C2)C1 C(CC(C(=O)NCC(C)C1CCC1)NC(c1ccc(OC)o1)=O)OCC C(CCN(C(=O)CCSCC)C)(C(C)(C)C)NC(C(c1ccc(CC)cc1)C)=O N1(C(COC(C)(C)C)=O)CCC2(C(=O)Nc3cc(F)c(F)c(F)c3)CCCC12 c1(C(N(C2CCCN(C(=O)Cc3[nH]cnc3C)C2)CC)=O)ccc(C(C)=O)cc1 c1(C2(F)C(C(N3CC(F)(c4ccccc4)C3)=O)C2)cccc(C(F)(F)F)c1 Cc1cccc(CC(=O)NCC2(O)CC(NC(=O)C(c3ccccc3)F)C2)c1 O=S(=O)(c1c[nH]ccc1=NCC1CC2(C1)OCCO2)N1CCCCC1CCCO c1(C(C)(C)C)ccc(Oc2ccc(N(CCO)Cc3ncco3)cc2)cc1 c1(CC(=O)N(C2CN(C(C3CC3F)=O)CC23CC3)C)cc(Br)cnc1F C1(C)(OC(=O)CNc2cn(C)nc2C)CCN(OC)CC1 C1(C(N2C(C(N(C(CC(C)C)C)C)=O)C(C)C2)=O)COCCN1C C1(NC(C2C(C(=O)OC)CCC2)=O)CCC(O)CN(C(c2nccc(C)n2)=O)C1 c1(C(CNC(c2cc(C)[nH]n2)=O)NC(C2(NC(N)=O)CC2)=O)cccc(Cl)c1 c1(C(CC(=O)OC)NC(=O)NCC(C)(C)OC(C)C)ccccc1F Cc1cc(Cl)ccc1C(=O)NCCC1CCCN1C(c1cnc(S)n1C)=O C1(CNC(CC(CC)CC)=O)CCC2C(CC1)C2(F)F n1(CC(C)C)[nH]c(CC(=O)NCC(C)(C)CNC(C2CC2(C)Br)=O)cc1=O N1(C(c2cc(C)nn2C2CC2)=O)CC2(C1)CN(C(=O)Cc1cnco1)C2 CC(C)(C)CC(C)(C)C(=O)NCCCCC(N1CCc2c(O)noc2C1)=O c1(OCCNCN(C(=O)CCOC(C)(C)C)CC)ccc(Cl)cc1F.C1(=O)CN1 CC(C)(O)C(F)C(=O)N1CC2CC1C2NC(=O)CC1=CCCC1 N1(C(c2cc(C)nc(C)n2)=O)CC(NC(C2(C(F)F)CCCC2)=O)CC(C)(C)C1 c1(OC)c(C(N2CC(F)CC2C(=O)Nc2cc(C)c(F)cn2)=O)cccc1Br N1(C(CC2CC(=C)C2)=O)CC2CC3CC2C1C3NC(=O)C=C1CCCC1 C1(CCC)(NC(=O)C(C)CO)CCN(C(c2cccc(F)c2SC)=O)CC1 C12(NC(CC(=O)OC)=O)CCCC1CN(C(c1nccc3occc13)=O)C2 C1(NC(C(C)(C2CCCCC2)NC(C)=O)=O)CCC(NC(=O)CNC(N)=O)CC1 c1(C(=O)NC2CC(C(C(=O)NCCC=CC)F)C2)cc(OC)n[nH]1 C(=O)(CS(=O)Cc1cccc(Br)c1)N(CC=C)CCOC N1(C(c2ncc(C)cc2C)=O)CCC(NC(c2cnn3c2OCC3)=O)C12CCC2 N1(C(C2CCC(NC(CCOC)=O)C2)=O)CCCC(C)(CO)C1 c1(NC(C23C(CN(Cc4c(O)ccc(OC)c4)C2)C3)=O)cccc(C#N)c1F C(C(C)(C(=O)N(C)Cc1ccncn1)NC(=O)Cc1cc(C)n(C)n1)SC C1(COC)(NC(=O)C(C#N)C2CC2)CCN(C(=O)Cc2ccc(Cl)cc2C)CC1 N1(C(c2cc3c(Cl)cccn3n2)=O)CCC2OCCN(C(C3C=CCC3)=O)C2C1 C1(C(=O)NCC(c2ccccc2)CNC(CCCOC)=O)(OC)CS(=O)(=O)C1 C1(CCC(=O)NCC2(C(N)=O)CN(C(CC(C)SC)=O)C2)CCCCN1C c1(C(=O)NC2(COC)CN(C(C3CCCCC3(C)C)=O)C2)ccc(C#N)cc1C CC1(NC(c2cc(=O)cc(Cl)[nH]2)=O)CCN(C(C2OC3CCC2CC3)=O)CC1 C(=O)(CC(C)NC(N)=O)NCCC(C)N(C(=O)C=CC(=O)OC)CC CCC(CC(=O)N1CCC2(C1)CN(C(c1cc(C)c(F)cc1O)=O)C2)C(F)F c1(NC(C(=O)NCC(C(C)(C)C)(C)C)=O)cccc2c1C(=O)NC2 C1(C)(C(=O)NCCN(C(CC(C)C)=O)Cc2ccc(N(C)C)cc2)CCCN1C c1(CNC(C2(CCC=C)CN(C(=O)C(C)CCC)C2)=O)cncc(C#N)c1 C1(C(N2CCCC(CNC(C(C(=O)OCC)F)=O)C2)=O)CCOCC1(C)C N1(C(c2c(C)nc(C)o2)=O)CC2C=CC1C(C(=O)NC1CN(C(N)=O)C1)C2 C(=O)(CC(C)C(F)(F)F)NC(C1N2C(C)C2C1)C(Cc1c(OC)cccc1)=O CCC(C)C(O)C(C)C(=O)N1CC(CC(NCP(C)(C)=O)=O)(OC)C1 c1(NC(C2CCOCC2)C=C)nccc(N(C)CC2CCN(C)CC2)n1 N1(C(CC(=O)N(C)C)=O)CCCC(C2CN(C(C3CCO3)=O)C2)C1 CC1(C)CC(NC(=O)Cc2cc[nH]c(=N)c2)CN(C(c2ccc(Cl)nn2)=O)C1 c1(C(=O)NC2CN(C(C3(C=C)CCCC3)=O)C2)cc(N(C)C)ccc1F c1(OC)c(C(N2CC(NC(=O)CCc3nccs3)C3CC3C2)=O)c(C)nn1C Cc1cc(=NC2CCN(C(c3noc4c3CCCC4)=O)CC2C)[nH]cc1C#N c1(Cc2c(C)ccs2)nc(-c2ccnc(F)c2)nn1C1COC(C)(C)C1 c1(C(=O)NC(C)(CNC(=O)Cn2cccn2)C2CC2)cccc(C2(C#N)CC2)c1 N1(C(C(C)CO)=O)CCC(CNC(=O)CC2CC(F)(F)C2)C(F)(F)CC1 c1(C(=O)NCC(CC(F)(F)F)NC(C(CCOC)C)=O)c(C)cc(C)oc1=O Fc1cc(-c2cccc(CC3COCCC3O)c2)ccc1-c1nccn1C(F)F C1(C(=O)NC2(C#C)CC2)CC12CCN(C(=O)CCOCC(F)F)CC2 CC1(C)CN(C(=O)C(CNC(C2(C)CNC(=O)N2)=O)CC2CC2)CCS1 N1(C(C2C(C=C)C2)=O)CCCC12CCC(NC(=O)C=C(C)CCC)CC2 Cc1cccc(F)c1C(N1CCCC(CCCCNC(c2cnn[nH]2)=O)C1)=O C1(CNC(C(COC)NC(C)=O)=O)CCC2(CN(C(C3CCCC3)=O)C2)O1 Cc1ccc(CCC(N2CC3CN(C(c4cnon4)=O)C3C2)=O)c(C)c1 C1(NC(C(C)N(C)C)=O)CCCC12CN(C(=O)C(n1cc3ccccc3n1)C)C2 n1(COC)nccc1NC(C)(C(=O)NCCCF)c1cccs1 N1(C(c2c(C(=O)OC)[nH]cc2)=O)CCC(O)(C(C)CNC(=O)CCN(C)CC)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)CNC(C1(COC)CC=CC1)=O C(=O)(C(C)(C)NC(=O)CC(O)c1ccccc1)N(CC(O)CO)C n1(CCSC)nnnc1C(c1ncoc1C(F)F)NCCC1CCOC1 N1(C(CCCCN(C)C)=O)CC(O)CCC1C(=O)NCCN1CCOCC1 c1(C(N(C(C)CNC(c2ncnc(C)c2C)=O)CC)=O)cc(N)cc([N+](=O)[O-])c1 C(=O)(C1CCCc2cccnc21)NCCCCNC(c1nc(CCC)sc1)=O c1(NC(N2CCCC2c2cccc(O)c2)=O)nc2c(s1)CCCC2 c1(-c2cc(C(=O)NC(C(C)NC(=O)C3=CCC3)CO)no2)cc(F)ccc1F c1(C(C(N2CCC(NC(C3C4C=CC3CC4)=O)CC2)=O)=O)ccc(Cl)cc1O Cc1cnc(C(=O)NCCCN(C(C23CC(C#N)(C2)C3)=O)C2CC2)cc1Cl c1(CCC(=O)NC2CCCC23CC3)ccccc1-n1cc(CCO)nn1 c1(CCCNC(C(C=C)O)=O)cccc(OC2CCCC2)c1.C1CCCNC1=O C1(NC(C2(CNC(C3C(=O)NCC3)=O)CCC2)=O)(CO)CCCCC1 CC1CN(C(C2CCCCC2NC(=O)CCC(F)(F)F)=O)c2ccccc21 c1(CN(C2COCC2O)C)ccc(-c2cnoc2)nc1 c1(NC(=O)CC)nc2c(s1)COCC2.C1(CCC)CN2CCN1C(=O)NCC2=O c1(-n2cc(C3CCN(C(C4(OC)CC4)=O)C3C3CC3)nn2)ccc(Cl)cc1 c1(C(c2nnnn2-c2ccccc2)NC2(CCOC)CC2)cccc(C)c1CCl CCCC(CCC)=CC(=O)NCC1(OC)CCN(C(=O)C(O)C2CCC2)C1 C(=O)(CCCCCCC)NCC1(C(=O)NC(CCC)C)CCCO1 C(=O)(CCC(C)C)N1CCC(n2cc(-c3n(CC4ON=C(C)C4)ccn3)nn2)C1 Cc1cc(C(N2CC(C(O)C(=O)NC3CCC4(CCC4)C3)C2)=O)cnc1O Cc1ccc2c(c1)C(NC(=O)C(Cc1cc[nH]n1)NC(=O)OCC)CO2.C(C)(C)(C)O C(=O)(CCCNS(C)(=O)=O)N(C1CC(Cl)(Cl)C1)CCC C1(CNC(C2(NC(C3N(CC)CC3)=O)CC(F)C2)=O)CC[Si](C)(C)C1 Cc1noc2cc(C(=O)NC3CCC34CN(C(=O)CN3CCCC3=O)C4)ccc12 Cc1cc(C(=O)NC2CN(Cc3c(F)cccc3Cl)C2)ncc1C(N)=O c1(C(=O)NC(CCCC)CNC(C2(C(F)(F)F)CC(O)C2)=O)sc(C)c(C)c1C N1(C(CCOCC#C)=O)CCC(CNC(=O)C(C)N2CCCC2)C(C)C1 N1(C(CC(C)O)=O)CC(C)(C)CC1CNC(=O)CCCCN(C)C c1(NC2C(c3ccc(C)cc3)CCC2)ccncc1S(=O)(=O)NCc1cncs1 C1(C(N(C2CCCNC2=O)C)=O)CC2(CCN(C(C3CC34CC4)=O)C2)C1 C1(NC(CSCC(C)C)=O)(CO)CCCN(C(C2CC3(CCOC3)C2)=O)C1 C(=O)(CS(=O)(=O)CCO)NC(CNC(C(C(C)(C)C)NC(N(C)C)=O)=O)CO C(=O)(CCCC(F)(F)C(F)(F)F)NC1CC(C)(CC)C1.C1C(C)=CC(=O)N1 C(=O)(C1=CC2(CCN(C(c3csc(=N)[nH]3)=O)C2)C1)N1CC2C(C)(CSC2)C1 n1(C(N(CCN(C(=O)CCOC2CCCC2)CC)CC)=O)nc(C)c(C)c1C N1(C(CC2(CC=C)CCCC2)=O)CC(CNC(=O)C(C)CC)C(C)C1 CC1CCC2(CC2)N(C(c2nc(Sc3cn(C4CCC(C)(F)CC4)nn3)cs2)=O)C1 C12(CNC(=O)Cc3cnc[nH]3)CCC1CN(C(c1ccc(C3CCC3)nc1)=O)C2 Cc1cc(C(=O)NCC2CC2CNC(C2(C)CC2Br)=O)nn1-c1ccccc1Cl N1(C(c2c(CC)c[nH]c2)=O)CCN(C(c2nc(C)ccc2F)=O)C(C)CC1C N1(C(C2CC(=C)C2)=O)CC(CNC(c2cc(O)nc(OC(C)C)n2)=O)C(F)(F)C1 c1(C(=O)NC(CNC(C(CCCC)O)=O)(C)C)ccc2c(c1)NC(=O)CCC2 N1(C(CN(C(=O)OC)C)=O)CC2CCN(C(=O)C=Cc3ccc(F)cc3)CC2C1 c1(CC(N2CCN(Cc3cc(O)ncc3Br)C3CC23)=O)ccc(Br)cc1I C1(NC(=O)CC2CCOCC2)CC2CCC(C1)N2C(C1CNC(=O)N1)=O c1(C(N2CC(N(C(=O)Cc3cn(CCO)nn3)C)C(O)C2)=O)ccc(Cl)nc1N C#Cc1ccc(OC)c(C(=O)NC(C)(CNC(=O)Cc2ccc(F)cc2)CC)c1 Cc1ccc(C2(C(=O)NC3CCN(c4nc(C)ns4)CC3)CC2)c(Cl)c1 Cc1cccc(C)c1C(N1CC(F)(F)CC1C(=O)NCc1cccnc1Br)=O C=C(C)CCCC(=O)NCC1CCC(NC(=O)CCCC2CCCO2)C1 C1(CNC(Cc2c(C)con2)=O)CC(C(=O)NCCC2(C)CCCO2)=NO1 C1(O)(C(C)NC(C2CCC(=O)N2)=O)CCN(C(=O)CC2CCCO2)CC1 C=CCCCCCCCC(=O)N(CCCNC(=O)C(c1ccccc1OC)C)C CCC(CCC(=O)NCCCCn1ccnc1)NC(=O)CC1CCC(=O)N1 CC1(C(=O)NCCOCCC(=O)NC(N)=O)CC2C=CC1C2.C1(N)CC2(CCC2)C1 C1(C(=O)O)(CC)CCCN(Cc2ccc(C(N)=O)cc2)C1 C(C(C)N=c1[nH]c2ccccc2cc1C#N)(C1CCCC1)NC(C(C=C)(C)C)=O O=C(CCCC(=O)NC1(CC(N2C3CSCC2C3)=O)CCC1)C1CC1 C(=O)(C(C)CC1CCC1)N(CCC(=O)NCC1CC12CC2)CC=C c1(CC(=O)NC2C(NC(CNS(N)(=O)=O)=O)CCCCC2)cn2ccccc2n1 c1(C(N2C(CNC(CCC3N(C)CCC3)=O)CC2)=O)cnc2cccnc2c1 C(C)(N=c1[nH]c2ccccc2cc1C#N)CNC(CNC(CNC(=O)OC)=O)=O c1(C(=O)NCC2N(C(c3ccc(C)o3)=O)CC=C2)cc(C)c(F)c(C)c1 C1(C(=O)NC(C2CCCCN2C(c2cccc(F)c2O)=O)C)CN(C)CC(C)O1 c1(C(=O)NC(CN(C(CCCC(CC)C)=O)C)C)cc(F)c2ncccc2c1 c1(CCC(=O)NC2CCN(C(CCC#C)=O)C2)cncc(F)c1 CC1(C)CC(NC(c2conc2-c2ccccc2)=O)CN1C(=O)CNC(N)=O C1(CNC(CN2CC(CC)C2)=O)CN(C(=O)C2=COCC2)CC1c1cncn1C C(=O)(C1=CCC2(CC1)CC2)N1CCC(CN(C)C(C2CC(CF)C2)=O)C1 N(C(=NCc1ccncc1Cl)N1CCC(CN2CCCCC2)C1)C(C)C N1(C(CC2N(C)CCC2)=O)CCCC(NC(=O)Cc2cc[nH]c2)CC1 c1(OC)cccc2[nH]c(-c3cccnc3C(=O)NC3CCNC3=O)cc12 Cc1cc(C)cc(C=CC(N2CCN(C(=O)CCC(F)(F)F)CC2C2CC2)=O)c1 Cc1c(C(=O)OCc2nn(C)c(C)c2Br)cccc1CO N1(C(C=CCC)=O)C2CCC1CN(C(c1cnc(C3CC3)nc1O)=O)CC2.C1CC1 N1(C(c2c(C)nccn2)=O)CC(NC(=O)C(c2ccc(Cl)c(F)c2)=O)C(C)(C)C1 C(=O)(CC1=CCCC1)NC1C(NC(CCC=CCC=C)=O)CCC1 N1(C(C2(CC)CC2)=O)CCC(CNC(=O)C=CCNC(C2COCCO2)=O)C1 c1(NC(N2CC(NC(C3CC(C)C3)=O)C2)=O)ccccc1OC1CCCCC1C CC12CN(Cc3snc(Cl)c3Cl)CC1(C)CN(CC1(Cc3ccccc3)CC1)C2 C1(NC(c2n(CCOC)ncc2)=O)CCCN(C(=O)Cn2nc(C)cc2C)C1 c1(CC(C)NC(=O)NC(c2ccccc2)C2CC2)cn(C)c2ccc(F)cc12 C(=O)(CCCCC#N)NC(c1ccc(C)cc1)CNC(C1(Cl)CC12CCC2)=O C=CC(C)(O)C(=O)NC1CC(O)C1CC(=O)NC1CCNC(=O)C1 C1(C)(N(C(C2C(C)CN2C(c2ncccc2Cl)=O)=O)CCO)CCC(=O)N(C)C1 CC(C)CC(C)(O)C(=O)N1CCC(F)(C(=O)NCCCCCCC2CC2)C1 c1(C(=O)NC2CC3(CC(NC(CC(CC)SC)=O)C3)C2)cnn2c1CN(C)CC2 N1(C(C(CNC(C)=O)(C)C)=O)CC2(CCC(CNC(=O)C(C)(C)O)O2)C1 Cc1cnncc1C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CCc1cnoc1 CN(C)S(=O)(=O)N1CC2(CC(C(=O)NC3C=CCCC3C(N)=O)C2)C1 CCC(CC)C(C(=O)NCCC1(NC(C2CC(OC)C2)=O)CCCC1)OC CC1=C(C(=O)NC2CN(C(=O)Cc3csnn3)C3CCCCC23)CCS1(=O)=O N1(C(C(C)OCC)=O)CC(CNC(c2csc(C(F)F)n2)=O)C(O)C1 CC(O)C(C(=O)NC1CC(CCC(=O)NCC2COCCC2O)C1)N(C)C C(=O)(C(C)(C)C(C)(C)C)OC.C12CCC3(CCC13)C(=O)NC1CC(C1)CN2 c1(C(N2CC(NC(CCC(=O)NC)=O)C2)=O)nc(Br)n2c1COCC2 C(C)(C)(CCC(=O)NC1CCCC(OC)C1)NC(C(COC)COC)=O C1(COc2ccc(C(=O)OC)cc2C)CN2CCCN1CC2 N1(C(C2(C)C(C)(C)C2)=O)CC2CC(C1)CN(C(=O)CN1CCC(C(N)=O)CC1)C2 C=CCC(CC=C)C(=O)NCC(c1cccc(C)c1)NC(c1csnc1OC)=O Cc1ccnc(O)c1C(=O)NC1CCCC(N(C(=O)CC2CSC2)C)C1 C1(C)(CN(C)C(c2ccc(CC#N)cc2)=O)CCCC1NC(c1ccoc1Cl)=O C1(NC(=O)C(=Cc2c[nH]cn2)F)CCOCC1NC(=O)CC1CCCC12CC2 c1(C(N(CC(=O)N(C2CC(F)(F)C2)C)CC)=O)ccc(=O)n2c1CCC2 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCCCCCNC(C(CNC(C)=O)(C)C)=O Cc1cnc(Cl)c(C(N2CCSC(C(=O)Nc3ccccc3C(C)O)C2)=O)c1 C1(COC)CC(CNC(c2cc(C3CCC3)no2)=O)N(C(C2COC(=O)C2)=O)C1 CCC(C)(C#N)C(=O)NCCC1CN(C(c2nccn2C)=O)CCCO1 C1(C(C)=O)CC(CC(=O)NCCN(C)C(c2ccnnc2)=O)C1(C)C c1(C(N2CC(F)CC(C(=O)Nc3cc(O)n[nH]3)C2)=O)ccc(F)c(F)c1O C1(NC(c2cc(OC)nc(Cl)c2)=O)CN(C(C2(CO)CC2)=O)CC2(CC2)C1 c1(OC)ccc(C(CNC(=O)C=C(C)C)NC(C2OCCCO2)=O)cc1 N1(C(CCC(C)N(C)C)=O)CCn2nc(CNC(=O)CC=C(Cl)Cl)cc2C1 N1(C(C(C(CC)(C)C)=O)=O)CC2CCCC(NC(c3ccno3)=O)C2C1 C1(CC)(CC)CN(C(C2(NC(c3ccncc3F)=O)CCCC2)=O)CCO1 C1(C(=O)NC2CCC(NC(C(C)=C3CC3)=O)CC2)CCN(CCO)C(=O)C1 c1(OC)cc(C(=O)NCCCCNC(=O)C(C2CCC(C)(C)CC2)C)cc(Cl)c1 N1(C(CC2CC(=O)NC2=O)=O)CCC2(CC1)CC(NC(c1ccns1)=O)C2 C(N=c1[nH]nc(C(C)(C)C)o1)C1C(NC(c2cc(CC)no2)=O)CCCC1 C1(NC(c2n(C)nnc2)=O)C2CCN(C(c3cccc(O)n3)=O)CC12 c1(OC)cccc2c(C(=O)NC3CCN(C(=O)CS(C)(=O)=O)C3C)c(C)[nH]c12 C1(NC(c2c(CC)oc(C)c2)=O)CN(C(c2cc(COC)no2)=O)C2(CCC2)C1 C1(C(N(C2CCN(C(=O)CC(C)C)C2)CCC)=O)CCc2c(nnn2C)C1 c1(C(=O)NCCC(CNC(Cc2c(C)scc2)=O)O)cnn2c1CCC2 CC(O)CCCCCC(=O)NC1CCC1NC(c1ccnc(S(N)(=O)=O)c1)=O C(=O)(C(O)C(CCC)NC(=O)C(C)C(O)C(C)C)N(CC#C)CCF C1(NC(=O)CC(C2CCC2)C2CCC2)Cc2cc(F)ccc2NC1=O N1(C(COCC=C)=O)CCC2(CC1)CC(NC(c1cccc(C)c1)=O)CCO2 C(C#CC(=O)NC(C1CCCN(C(c2cccnn2)=O)C1)C)(OCC)OCC C1(CC(=O)N(CCc2cn(CC)nn2)CC)CCCN(c2ccc(OC)cc2)C1 c1(C(=O)NC2CCCC(NC(c3ccns3)=O)CC2)cccc2c1CCC2 N1(C(C2N(C(c3c(C)nsc3)=O)CC(=O)NC2)=O)CCCN(C)C(=O)C1 c1(C(N2CCC(OC)C23CC3)=O)nn(C)c2ccc(F)cc12 N1(CCCNC(=O)CC2C=CCC2)CCN(C(=O)C2=CSCS2)CC1 C1(CNC(c2cnc(C(C)C)[nH]2)=O)CCCCC1NC(=O)C1=CCCC1 c1(C(=O)NC(C2CN(C(c3c(C)snc3)=O)C2)C)nc2sccn2c1C c1(OC)cc(F)c(C(=O)NCC(Cc2ccccc2)NC(=O)CO)cc1Br c1(COC)ncsc1C(=O)N(CCCNC(=O)C(N)=O)C1CC1 C1(CC)C(C(N2CC(CNC(C3(OC)CCOCC3)=O)C2)=O)CCN1C C1(NC(C(CC(C)C)C)=O)CN(C(=O)Cc2ccnc(O)c2)CC2(CCC2)C1 N1(C(CC2C(C(=O)OCC)C2)=O)CCC2(C1)CN(C(=O)CCN1CCCC1=O)C2 Cc1cc2c(C(N3CC(CNC(c4ccc(C)s4)=O)CCC3C)=O)cccc2o1 c1(CNC(CCCCC)=O)nnc2n1CCN(C(C1(n3cccn3)CC1)=O)C2 C1(C)(CNC(CSc2ccc(C)cc2)=O)CCCN(C(=O)C#CC2CC2)C1 c1(C(=O)NC(CNC(C(=O)NCCOC)=O)C(C)C)ccn2c1CCC2 C=CCCC(C(=O)NC(c1cnn[nH]1)(C)C)NC(c1ccc(C)c(C)c1)=O C1(C)(NC(c2cc(CC)[nH]n2)=O)CCN(C(=O)CCc2ccc(Cl)s2)CC1 CC1(CCNC(=O)CCF)CCN(C(=O)C(O)C2CC2)CC1 C1(C(=O)OCCC(C)C)(CN(CC)CC)CCCC1 c1(CC(=O)NCC(CNC(CSCCOC)=O)F)cnn2c1OCCC2 C1(NC(C2CCCC(C)C2)=O)(CO)CCCN(C(=O)COC(F)F)C1 c1(C(C)C)ncc(C(=O)NC(C2CCCCO2)C)[nH]1 n1(CC(=O)NC2CC(C)N(c3ncc(C#N)cc3Br)C2)cc2ncccc2n1 c1(C(CNC(=O)CP(C)(C)=O)NC(C(CC)C#N)=O)ccc(Cl)cc1Cl N1(C(C(CC)OCC)=O)CC(NC(c2cccnc2C(F)F)=O)CC2(CC2)C1 Cc1nc(-c2ncc[nH]2)sc1C(=O)NC(C)CC(C)NC(C12COCC1C2)=O C(C1CN(C(C2(CC)COC2)=O)CC1C(N1CC(F)(CF)C1)=O)=CC N1(C(CCc2ccc(C)s2)=O)CCC(NC(=O)CN2CCCC2)C(O)C1 C(CCC(C)C)(C(=O)N1CCC(C(C)OC)CC1)NC(C(CCCOC)C)=O N1(C(c2c(C)cccc2F)=O)CCOC2(CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C1 c1(OC)cc(CNC2CCCC2C(=O)NC2CCCOC2)cc([N+](=O)[O-])c1 Cc1ccc(C2CCN(C(c3nc(C(C)C)n[nH]3)C(=O)NC3(C)CC3)C2)c(C)c1 C1(C)(NC(C=C(C)C(F)F)=O)CCC(NC(c2cccc(C3(C)CC3)c2)=O)CC1 CC1CN(C(C2(C)CCCCC2)=O)CCN1C(c1cscc1Br)=O C1(CC#C)(C(=O)NCC(C)(C2CC2)NC(=O)Cc2c(C)noc2Cl)CCOCC1 CC1CN(C(=O)C(N2CC3CCC2(C(F)(F)F)C3)=O)CC(C)(C)C1 C12(NC(C=CC=CCC)=O)CC3CCC(C1C2)N3C(=O)Cn1nc(C)cc1C C(=O)(C#CC1CCOCC1)N1CC(C(=O)NC2CCC(CCO)C2)C1 c1(C(=O)NC(CCNC(C2C(CCOC)C2)=O)(C)C)c[nH]c2ccc(Cl)cc12 c1(C(C(=O)NCC2CN(C(c3c(C)nns3)=O)C2)C)ccc(Br)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(C)CCN(C(=O)CCc2ncccn2)CC1 C1(C(N2CCC(N(C(=O)CN(C)S(N)(=O)=O)CCC)C2)=O)CCC(=O)N1CC N1(C(c2cn(C)nc2)=O)CCC(C(C)(C)CNC(c2ncoc2C2CC2)=O)CC1 c1(SCC(=O)NCCCNC(c2cc3scnc3[nH]2)=O)ccc2c(c1)CCC2 C1(C(=O)NCC2C(NC(CCCNC(=O)OCC)=O)CC2)CC(=O)N(C)C1 c1(C(N(CC(CNC(c2ccc(C)c(Cl)c2)=O)C)C)=O)c(C)sc2ccccc12 C1(c2n(CCOCC)nnn2)(NC2CC(=O)NC(=O)C2)CC2CCC(C1)O2 N1(C(C(C)CO)=O)CC(CNC(=O)C=C2CCOCC2)CC1(C)C c1(OC)cccc(F)c1C(=O)NCCCCNC(=O)C=Cc1ncc(C)[nH]1 CN1CCc2cc(C(N3CCC3C(N3CCC4(CCC4)C3)=O)=O)ccc21 c1(SC(=O)NCC(=O)C2CC2C2(O)CCC(SCC)CC2)cc(N)cc([N+](=O)[O-])c1.NC N1(C(c2c(C)n(C)nc2)=O)CCN(C(=O)Cc2nn(C)cc2Cl)C(CC(F)F)C1 C1(C(=O)NCCCN(C(=O)C(C)=C2CC2)CC)CCCN1c1nccs1 S(=O)(=O)(c1ccc(NCCCCCN=[N+]=[N-])c(F)c1)N1CC(C)OC(C)C1 c1(C(N2CC(NC(CCC=C)=O)C(CC)C2)=O)cnc(OC)c(F)c1 Cn1ccnc1C(=O)NCC1CCC1.C1(C)(C2CC2)CNC(=O)N1 N1(CC)CCN(N(Cc2ccccc2)C(C)C(C)C)CC1=O.c1ccc(Cl)cc1F c1(CC)oc(C)cc1C(=O)NC(C)C(C)NC(=O)C(C)CSC c1(C(=O)NC2(C)CN(C(c3ccc4n[nH]cc4c3)=O)C2)nccc2ccn(C)c12 c1(C(=O)NCC2CN(C(C(CCC)(C)O)=O)CC2C)ccc2c[nH]nc2c1 C(=O)(CCS(=O)(=O)c1ccccc1)OCc1ccc(CC)c(CO)c1 c1(C(=O)NC2(C)CCN(C(=O)C(O)CC(N)=O)C2)cccc2c1NCCC2 CC1ON=C(C(=O)NCC(CO)NC(C2(C(=O)N(C)C)CC2)=O)C1C c1(NC(C(C)C)CNC(=O)C(C)(C)C2CCCO2)cc(-c2ccccc2)ncn1 C(=O)(C1COc2ccccc21)N(C1CCN(C(C2CC2CCOC)=O)C1)CC N1(C(CCSc2ccc(C)cc2)=O)CCN(C(=O)C(O)C(C)(C)C)CC12CCC2 N1(C(CCCOCC)=O)CCN(C(C2CCCCN2C(C)=O)=O)C(CC(F)F)C1 c1(C(N2CCC(N(C(C=CC(C)C)=O)CCO)C2)=O)cc(N)ccc1Br N1(C(C(CC(C)C)O)=O)CCC(C(=O)NCC2CC[Si](C)(C)C2)C12CCC2 N1(C(C2CC(NC(C(C)=CC=C)=O)C2(C)C)=O)CCCC(C2CC2)CC1 CCN=c1[nH]cnc2cc(C(NC3=NC4C5CCC(C5)C4C3)=O)ccc12 C#CCCC(C(=O)N(C1COC(C)(C)C1)C)NC(c1cc(O)cc(F)c1)=O C(=O)(CC1C(=O)Nc2ccccc21)NCC1CC(OC)CN1C(C1CCC1)=O C1(NC(CC2(C)CC2)=O)CCCN(C(=O)CCN2CCC(F)C2)C1 N1(C(C(C(C)C)O)=O)CC(CNC(c2cc(C(F)F)ccc2F)=O)C(C)(C)C1 c1(C(=O)NCC2CCCN(C(C3CC(=C)C3)=O)C2)ccc(Cl)c(C)c1 CS(=O)CCC(=O)NCC1CCCCC1NC(=O)CC1(CO)CCCC1 c1(SC)cc(C(N2CC(CNN(C(C=CC)O)C3CC3)C2)=O)no1 C1(NC(C2N(C)CCCC2)=O)CC2(CCCCN2C(c2cnccn2)=O)C1 Cc1ccc(CC(=O)NC(C)CCCNC(c2ccc(Cl)nc2O)=O)cc1Cl C1(CNC(C2(C)CNC(=O)C2)=O)CN(C(=O)CC2(CO)CC2)CC2(CCC2)O1 C1(C(=O)NC2CCN(C(=O)CSc3ccncc3)C2)CC2C=CC1CCC2 C12(NC(=O)COC3CC3)CC1CN(C(=O)CCc1cncs1)C2 C1(NC(c2sccc2F)=O)CCN(C(=O)C(F)n2ccnc2)CC12CCC2 C1(NC(C=CC)=O)C(C)(C)C(NC(c2ccc(-c3nc(C)cs3)cc2)=O)C1(C)C N1(CCN(C(c2ncc(Br)s2)C(=O)NCCC#N)C)CC(=O)Nc2ccccc21 C1(NC(CCCCSC)=O)CN(C(C2SCCCS2)=O)C2CCCCC12 N1(C(C2(C)CCCN2)=O)CCOCC(C)(CNC(=O)C(c2ccccc2)O)C1 N1(C(C(CCC(C)C)NC(Cc2c(C)occ2)=O)=O)C2CCCC1CN(C)C2 Cc1nccc(C)c1C.N12CC(C(C)(C)C1)C2=O.c1(OCC(=O)NC)ccsn1 CC1CC(C)(C(=O)NC2CC(CNC(c3nc(Cl)c(=O)[nH]c3N)=O)C2)CC(C)O1 C1(C(=O)NCC)CCN(C(c2ccncc2F)C(=O)NCCCF)CC1 c1(C(=O)NC2CCCC(C(=O)OC)C2)c(C)n(C)c2ccccc12 Cc1cccc2c1CCOC2C(=O)NCC(CNC(=O)C1CC1)C(F)(F)F c1(OC(C)C)cnc(F)c(-c2ccccc2C(=O)N(C)Cc2ccccc2O)c1 c1(C(=O)NCCC2(C(F)(F)F)CC2)ccccc1C(F)(F)C(F)(F)F C#CC1(O)CCCN(C(=O)CCC2(NC(C3CC3C3CCCC3)=O)CCCC2)C1 C(=O)(C(C)(C)CC(F)F)NCCC1CCN(C(c2scc(C)c2C)=O)C1 c1(OC)cc(F)ccc1CN1CC=CC1C(=O)Nc1ccc(SC)cc1 C1(NC(C(N(C(=O)CC2OCCCO2)C)C2CC2)=O)COC2(CCC2)C1 C1(NC(=O)NCc2c(OC)cccc2OC)CCC2C(CCN2C)C1 c1(C(=O)NC2C(C(=O)NCCCCC3C(C)C3)COC2)ncccc1F N1(C(C(C)Cc2ccco2)=O)CC2(C1)CN(C(=O)CCC1CC(F)(F)C1)C2 O(NC(=O)C(C1CN(C(=O)C(F)F)C1)OC)CC#C c1(CC(=O)NCCCC2N(C(C(CC)(C)C)=O)CCC2)ccc(F)c(F)c1C N1(C(C=C(C)C(C)C)=O)CC(CNC(c2cc(=O)cc[nH]2)=O)CC(C)(C)C1 CC(C)(CC(=O)NCC1(NC(c2cc(C3(C)CC3)n[nH]2)=O)CC(F)(F)C1)C1CC1 N1(C(c2c(CC)c[nH]c2)=O)CC(CNC(C2CS(=O)(=O)C2)=O)C(O)C1 C1(C(F)(F)F)(C(=O)NCCCCN(C(C(CC)n2cncn2)=O)C)CCCCC1 N1(C(c2ccn(CC)c2C)=O)CC2(CNC(C3CC3(C)C(C)C)=O)CCC1CC2 C(=O)(Nn1cnnc1CC)C1N(C)CCN(C(C(C=C)OC)=O)C1 N1(C(C2(CCOC)CCC2)=O)CC(C2(NC(=O)CCCc3ccc(C)s3)CC2)C1 C1(N(C(CSCCCC)=O)CC2CC2)CCN(C(=O)C(C)C=C=C)CC1 S(=O)(=O)(c1ccc(NC(c2nncs2)C)c(Br)c1)NCC(COC)(C)C C1(NC(C=CC=CC)=O)CC(CNC(=O)Cc2ccc(O)cc2C)C12CCC2 Cc1ccnnc1C(=O)NC1CN(C(c2cc[n+]([O-])cc2)=O)CC1CC1CC1 C12(CNC(CCC=C)=O)CC1CN(C(=O)C(C1CCOCC1)OC)C2 c1(OC)cc(Cl)ccc1C(=O)N(CC(C)(C)CNC(c1cnc2n1CCS2)=O)C c1(CCC(=O)NC2CCC(N(C)C(c3ccnnc3)=O)C2)ccc(C(F)F)cc1 C1(C(N2CCC(C)(CCNC(C(c3ccnn3C)C)=O)C2)=O)CCS(=O)(=O)CC1 c1(C(=O)NC(C2CCCC2)CNC(c2ccnc(S)c2)=O)ccc2cnoc2c1 C1(C(=O)NCC(N(C(c2c(C)nc[nH]2)=O)C)C2CC2)Nc2ccccc2C1(C)C CC(O)C(C)C(=O)N1CC(CNC(=O)C=Cc2cccnc2)C1 CC(Cn1ccnc1)C(=O)NCc1nc(C(N2CC(O)(c3nn[nH]n3)C2)=O)co1 CC1=C(C(=O)NC(CNC(C2CCCCN2C(C)C)=O)C2CCC2)CC1 N(S(=O)(=O)N(C)C)CC(=O)NC(C1CN(C(CC2CCN(C(C)=O)C2)=O)C1)C C(=O)(C(C)(Cc1ccccc1)C(C)C)NCC(CNC(CN(C1CC1)CC)=O)O C(CCCCC(=O)Nc1ccc(F)cc1OC(F)F)N1CCCC(NC(C)=O)C1 c1(C(=O)NCC(C)OC)ccc2c(n1)CN(C(=O)C1=NOC(C)C1)CC2 c1(C(=O)NCC(CNC(CC2C(C)(C)C2)=O)O)cc(Cl)cc(Cl)c1O C1(N(C(C=CC(C)NC(=O)C(c2cnn(C)c2)O)=O)CCO)CCCCC1 C1(NC(CSCCC)=O)CCC(NC(C2(COC)C=CCC2)=O)C1 N1(C(C2(F)C(C)(C)C2(C)C)=O)CCCC(C2CN(C(=O)COCP(C)(C)=O)C2)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCCC(C)(C(=O)NC(c2nncn2C(C)C)C)C1 CC1CCN(C(=O)C2=COCCC2)CC1CNC(c1ccccc1C(C)(F)F)=O C(C(CC(C)C)NC(c1cnnc(O)c1)=O)NC(Cc1cnc(C)[nH]1)=O C(=O)(C(C)(C1CC1)OC)NC(C(=O)N(CCC(=O)OCC)C)C1CCOC1 c1(COC)ccc(C(=O)NCC(C)(F)CNC(c2n[nH]cc2C)=O)o1 S(=O)(=O)(c1ccc(NCC=C2CCOCC2)c(Cl)c1)NCC=CCCOC c1(OC)cc(C(=O)N(CCC(=O)NCc2cc(C(C)C)[nH]n2)CCCO)ncn1 c1(C(N2CCOCC(NC(CCC=C)=O)C2)=O)cc(O)cc([N+](=O)[O-])c1 CS(=O)(=O)CCC(=O)NCCOC1CCN(C(C2OCC3CCCC23)=O)C1 c1(CC(=O)N(CCCCCCNC(=O)Cn2nnc(=N)[nH]2)C)ncn2c1CCC2 c1(NC(C(CCOCC)NC(c2c[nH]c(=NCC)s2)=O)=O)cccc2c1CCC2 C12(NC(c3c(CC)nccc3)=O)CCC1CN(C(c1cn3ccnc3s1)=O)C2 N1(C(CNC(CCCCC)=O)=O)CCC(NC(c2scnc2C)=O)CC1C N1(C(C2(C)CC2c2ccccc2)=O)CCCCCC(NC(=O)Cn2ncnn2)C1 C1(C(N(C)Cc2cn(CC)nn2)=O)CC(O)CCN1C(C1CCCO1)=O N1(C(=O)NC(C)C(C)N(C)C)CC(C(=O)OC)C(C)(C)C1.N(C)C C=CC1(CC(=O)NCC2C(C)CCCN2C(c2ccc(SC)o2)=O)CCOCC1 C1(C2CCC2)(C(N2CC(O)(C(C)NC(C3CCC(F)C3)=O)C2)=O)CC1(F)F N1(C(C(C)OC)=O)Cc2ccccc2C1CNC(=O)CN1C(=O)CCCC1=O C1(OC)CCC(CC(=O)NCCC2CC(NC(=O)CC(O)CN(C)C)C2)CC1 Cc1ccc(N)c(C)c1C(=O)NC1CC(NC(c2sc(Br)nc2C)=O)C1 c1(CN2CCC(N(C(c3c(C)ncc(Br)c3)=O)C)C2)ccnc2ccccc12 c1(OC)ccc(F)c(C(=O)NCCC2CCCCN2C(=O)CN(C)C)c1OC C(C(C)(C)CCNC(=O)Cc1ccco1)NC(C(C)OCCC#C)=O Cc1c(CNC(=O)CC23CCC2CN(C(c2cc(Cl)no2)=O)C3)cccc1F Cc1ccc(C(CO)NC(=O)NC(C2CCC3(CCC3)O2)C2CC2)c(F)c1 c1(C(=O)NCCC(C)NC(C2CCCOCC2)=O)cncc(F)c1C(F)(F)F c1(N2CCN(C(=O)C(N3CCCC4C(O)CC34)=O)CC2)ncnc2ccccc12 N1(C(CC(COC)C)=O)CCC(N(C(=O)CCc2cccc(O)n2)C)C2(CC2)C1 c1(C(N2CC(CCNC(C(CC)=CC)=O)OC(C)C2)=O)cc(CC)c(=O)n(C)c1 N1(C(C=C(C)C(C)C)=O)CC(O)(CCNC(C2(Cc3cnn[nH]3)CCC2)=O)C1 C1(C(=O)NCC(C)CNC(c2ccnc(C(F)(F)F)c2)=O)CCc2nncn2C1 CCCCC(O)C(=O)NCC(C)(Cn1cccn1)NC(=O)CCC(=O)N(C)C CCC(C)(CCO)NC(=O)C(CO)NC(=O)CC1CC(F)(F)C1 n1(C(COC)C)nc(-c2ccncc2)nc1-c1ccnn1Cc1ccccc1 c1(CC)n[nH]c(=NC(CNC(C2CCCOC2)=O)C(C)C(C)C)o1 N#CC1CN(Cc2ccccc2)CCN1C(c1cc(Br)c(Br)cc1O)=O c1(CCC)c(C(=O)NCC(C2CCS(=O)(=O)C2)(C)O)nnn1CC c1(C(N2CCC(C#N)(NC(c3cncc(Br)c3)=O)C2)=O)c(O)cccc1[N+](=O)[O-] C1(NC(CC2(C)CCN(C(CC3CCN(C)C3=O)=O)C2)=O)CCn2cnnc2C1 C12(C(=O)OCCC3(C)CCN3)CCOCC1C2(F)F C1(C(=O)NCCN2CCN(C(C(C(=C)C)(C)C)=O)CC2)C2CCCCCCC12 c1(C(=O)NC2CN(C(C(c3cc(C)sc3)(F)F)=O)CC2C)c(C)cc[nH]c1=N C1(C(=O)N(CCCCN(C(=O)COCCCOC)C)C)(OC)CCCCC1.C(C)=O Cc1cncc(C(N2CCCC(N(C(=O)C=CC3CCCO3)C)C2)=O)c1 C(=O)(C(C(=O)N1CCC(CCNC(=O)C(F)CC2CCC2)CC1)OC)OC C1(C(=O)NCC2(C(=O)NCC(C#C)OC)CCC2)CCC(=O)C1 n1(CC)nc(C(=O)NCC(C)(F)CNC(=O)C(C(C)C)n2cnnn2)c(C)n1 N1(C(c2nc(COC)sc2)=O)CCC2CCC12CNC(C1CCCC1)=O C1(C(=O)NC2C(NC(c3c(C)nsc3)=O)COC2)C2CCCCC12 C(C(C(=O)NC(c1ncc(C)[nH]1)CC)NC(=O)C(C)N1CCCC1)OCC CCC(CN=c1cc(NC(c2ccoc2)C)nc[nH]1)N1CCCC1 Cc1ccc(C(N2CCC(c3c(Cl)cccc3Cl)C2)C(=O)NC2CC2)c(F)c1C N#CC1(N(S(=O)(=O)Cc2ccccc2N2CCCC2)CC(=O)O)CCOC1 CC1CN(C(C2(n3cc(C)nn3)CCOCC2)=O)CC2(CC2)C1.C1CCCSC1 C1(CC)CC(C)CN1C(=O)CC1CCC(NC(=O)C(C2CCCCC2)C)CC1 C1(NC(C2(NC(c3cnnc(O)c3)=O)CCSC2)=O)CC2CCCC2C1 O=C(C1Cc2ccccc21)NC1CC2CN(C(=O)C=Cc3ccccn3)CC2C1 CC1CCC(CNC(=O)CC=CC(C)(C)C)CN1C(=O)C(=O)C(C)(C)C c1(NC(=O)Nc2cc(C(C)C)nn2C)ccc2c(cnn2C(C)C2CC2)c1 c1(COC)nc(N2CCCC(CNC(=O)CC3CC(F)C3)CC2)cc(C)n1 O=S(=O)(c1cnc(C2CCOCC2)o1)N1CC(C(=O)O)CC(C(F)(F)F)C1 CN1CC(NC(=O)C(Cn2cccn2)NC(=O)CNC=O)C(C)(C)C1 c1(CCC(N2CCN(C(CN(C(C)=O)C)=O)CC2)=O)c[nH]c2ncccc12 Cc1cc(C(=O)NC2CCC(NC(=O)CC3CC=CCN3C)C2)c(C)n1C(C)C Cc1cc(C(=O)NC2CCC(C)N(C(c3oc(Br)nc3C)=O)C2)cc(O)c1 c1(C(N2CCC(N(C(=O)CSC(C)C)CC)CC2C)=O)ccc2n[nH]c(C)c2c1 C(=O)(C(N)CCC1CCCCC1)NCCCC(=O)NC C1(NC(Cn2c(C)nnn2)=O)CN(C(C2CC2Br)=O)CC1(C)C Cc1ccc(C(=O)Nc2ccc(NC(c3cccc(=O)n3C)=O)cc2F)c(C)c1 N1(C(C2CCN(C(C)=O)CC2)=O)CCN(C(c2csc(C)c2)=O)C(C(C)C)C1 C1(C)(NC(C2CCN(C(CCCCCOC)=O)C2)=O)CN2CCC1CC2 C1(NC(c2cn(CC)nn2)=O)CC(C(=O)NC(COC)CO)C1(C)C CC1(C)Cc2cc(C(=O)NC3CN(C(c4cscn4)=O)CC34CC4)sc2C1 c1(C(=O)NC2(CCOC)CCN(C(=O)C(F)=C(C)C)C2)nn2c(c1C)OCCC2 n1(C(CC)NC(c2nc(-c3ccc(C)c(F)c3)cs2)=O)cc(Br)ccc1=O c1(C(N2C(CNC(C(c3n(C)cnc3)O)=O)CC2)=O)occ2c1CCCC2 C=C(C)CCN=c1cc[nH]cc1S(=O)(=O)N1CC(C)SC(C)C1 c1(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)OC)c(F)cncc1Cl c1(C(=O)NC(c2ccccc2)C(C)C)cccnc1OC(=O)C1CC1 N(C1CCc2ccc(Cl)cc21)C(C1CC2(C1)CN(C(c1coc(Cl)n1)=O)C2)=O Cc1nnc(CNC(=O)CN(C2CC(C#N)C2)C(=O)C(F)C2CCCC2)o1 c1(C2C(C(=O)NC3C(CC)CCC3)C2)ccc(F)cc1F CC1=CCC(C(N2CC3CC2(CNC(=O)C(O)C(C)C)C3)=O)CC1 c1(C(=O)NCCN2CCN(C(C3(C)CC(=C)C3)=O)CC2=O)cccc2nonc12 CC1CN(C(=O)Cn2cc(P(C)(C)=O)cn2)CCCN1C(=O)CC1CC(F)C1 c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)CO)cccc(S(=O)(=O)N(C)C)c1 C1(CNC(Cc2cc(C)no2)=O)CCCCN1C(c1ccnnc1)=O CCCC(C)CC(=O)N1CCCCC1CN(C(=O)C(=O)C(C)(C)C)C CCC(C)(O)C(=O)N(CCCN(C)C(C1CC1C#N)=O)C CCS(=O)(=O)c1ccccc1C(=O)NCC12CC1CN(C(C1CCN(C)C1)=O)C2 N1(C(=O)CN2CCOCC2)CCC2CN(C(=O)CCC3CCCCO3)C2C1 C1(CN(C(=O)CC(=O)OC(C)(C)C)C)CC(O)CN1C(c1cncs1)=O c1(C(N2CCC3(NC(CCCCNC(C)=O)=O)C(C2)C3)=O)cc(C#N)ccc1O C(CC(C(=O)N(CC(C)O)C)NC(=O)C(C)=C1CC1)OC CCCC(C)CC(=O)N(CC(O)CN(C(=O)C(F)CC1CC1)C)C n1(CCC(=O)OC)cc(Cl)c(C(=O)NC(CO)C(C)NC(=O)CCCOC)n1 N1(C(c2cnn(CCCl)c2)C(=O)NCCOCC)CC(C)CCC1CC#N C1(OC)CN(C(=O)C(=O)Nc2ccccc2CC2CCOC2)CC2CC12 N12CCC(CC1)n1ccc(n1)NC2=O.Cc1nc(C(C)NC2CCCC2)n[nH]1 c1(C(=O)NC2CC(n3cc(-c4n(CC)ncc4)nn3)C2)cc(Cl)c(Cl)c(Cl)c1 C(=O)(C(C)CC(F)(F)F)N1CCN(CC(N2C(C(=O)OC)CC2C)=O)CC1 C1(C(=O)NC2CCC(NC(C3(C4CC4)CC3)=O)C2)(OC)CS(=O)(=O)C1 C1(CC(N2C(CNC(C3(CF)CC3)=O)CC(OC)C2)=O)SC2=NCCN2C1=O N1(C(CCC)=O)CCC2(CC1)CC2NC(c1ccnc(C2CCNCC2)n1)=O C1(N(CC)C(=O)OC(C)(C)C)(CC)CCCCO1.C(=O)(C(C)OCC1CC1)N c1(CC)ccccc1C(N1CCC(OCC(=O)NOC2CC2)C1)=O C(=O)(C(Cc1cccnn1)NC(=O)NC(C)COC(C)(C)C)OCC N1(C(CC=CCC)=O)CCN(C(=O)C(C(C)(C)C)S(=O)(=O)CCCC)CC1CC O=C(C1=NOCC1)N1CCC(NC(C2CC(c3ccccc3)C2)=O)C1 c1(OC)cc(C(=O)N(C)CC2CCCCN2C(=O)C(n2ccnc2C)C)n(C)n1 N1(C(C2C(C)CCO2)=O)CC=C(CC(=O)N2CC3CC(C2)CN(C)C3)CC1 c1(CCC(=O)NC2CC(C(=O)NCCC3CC(CN(C)C)C3)C2)nnc(S)n1C CN1CCC2CCC(C1)N2C(c1coc(CNC(=O)CNC(=O)CN(C)C)n1)=O c1(C(=O)NC2CCCN(C(C(C)(O)C3CC3)=O)C2)c(F)cc(N)cc1F C1(NC(CC(CC)CC)=O)CCN(C(c2cnc(C)c(N)c2)=O)CCC1CO c1(CNC2N(Cc3c(C)nco3)CCC2)ccc(F)cc1.n12nnnc1N2C N1(C(C2CC2(F)F)=O)CC2C(NC(C3(c4ccco4)CC3)=O)C2C1 N1(C(CC2CC(C(C)C)OCC2)=O)CCNC(=O)CCCC1 N1(C(C=CCCC)=O)CCCC(NC(=O)CC2CCCC2)C(F)C1 c1(C(N2CCN(C(=O)C=CCl)CC2)C(=O)NCCOCC)ccnc(Cl)c1F C#CCCCCCCC(=O)N1CCCCC1CNC(C1CCC2CC12)=O C(C)(C)(CCCC(=O)NC1CC1c1cncs1)NC(C1C(C)(CC)C1)=O C1(CNC(C(CC)N2CCCC2=O)=O)CN(C(=O)CC23COCC(C2)C3)CC1N Cc1cc(C(=O)N(C)CCOCCNC(=O)C(O)C(F)(F)F)c(N)c([N+](=O)[O-])c1 CSC=CC(=O)NCCCN(C(C1COCC1c1ccccc1)=O)C1CC1 Clc1ccc2nc(CN(C(c3ccccc3)C3CCCO3)CC3CC3)sc2c1 CN1CCC(C)(C(=O)NCC2C(C(N3CCC(C)(C#N)C3)=O)C2(C)C)CC1 N1(CC)CCN(C(=O)C(Cn2cncn2)NC(=O)CN2CC(=O)NC2=O)CC1 Cc1ccc2c(C)c(NC(=O)C(=O)NC(c3ccn(CC(C)C)n3)C)ccc2c1 CCCCCC(C)(C)C(=O)NCc1cc(C)c(C(=O)NCCCn2nccn2)o1 C1(C(=O)NCC2CC3CCC3C2)(CNC(=O)Cc2cc[nH]n2)CC12CCC2 C(=O)(CCC(C)(C)CN1CCCC1CS(=O)(=O)C(F)F)OCC N1(C(c2cc(C(F)F)no2)=O)CCC2CC12C(=O)NCc1ccncc1Cl Cc1ncncc1C(=O)N(CCCN(C(=O)C(CO)c1ccccc1)C)C c1(C(C2CC=CCC2)(CC)NC(COC)C2(C)CC2)nnnn1-c1ccccc1 c1(C(=O)NCC2OCCN(c3nccc(CC#N)n3)C2)ccc2cnsc2c1 CCC(CC(=O)NC(C)CN(C(=O)CN1CCCCC1=O)C)CC(F)(F)F N1(C(C(C)OC)=O)CCN(CCCCCNC(C2C=CCCC2)=O)CC1 CC(C)CC(C)(C)C(=O)N(CC(=O)NCCC1CCN(C)C1=O)C N1(C(C2C(=C)C2)=O)CCCN(C(=O)CC2CC2C2CC2)CC1C Clc1cccc(CCNC2(c3cc(Br)cc(Br)c3)CC2)c1Cl CCCC(C(=O)N1CCC(C(=O)NCc2ccco2)(OC)C1)C(C)C C1(NC2CCC2)CCC(C(=O)NC(CNC(C(C)NC(C)=O)=O)=O)CC1 N1(C(C2C(CCC)C2)=O)CCC(CNC(=O)Cc2cc(C(=O)OC)no2)C12CC2 C1(NC(c2ncn(CC)c2)=O)(COC)CCN(C(=O)C(n2nccc2C)C)C1 CCCCC(CNC(c1nnc(C(=O)OC)s1)=O)NC(=O)C(C(C)C)SC c1(NC(C2N(C(c3ccn(C)c3)=O)CC=C2)=O)cc(F)c(Cl)nc1Cl c1(-c2ncc(C)[nH]2)ccccc1NC(=O)C(=O)NCC1CCC(C(F)(F)F)O1 Cn1ncc2cc(C(N3CCSCC3CNC(c3ccc(F)c(F)c3)=O)=O)sc12 CCC(C)C(O)C(C)C(=O)N1CC(C)(C(=O)NCC2(C3CC3)CC2)CC1(C)C CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(CC(C)C)NC(c1cscn1)=O c1(C(N(CCCNC(C2CC=CCO2)=O)CC)=O)cc2c(s1)CCC2=O C1(CN=C(NC(C=C)C)NCc2ccc(C(F)(F)F)o2)CCc2cnn(C)c2C1 c1(CCCCSC)nc(-c2cccc(C(F)(F)F)c2)nn1C(C)C(C)C c1(C(=O)OC)cc(N2CCCC2CCCNC(C2CC23CCCC3)=O)ncn1 c1(C(=O)NCC(CC)NC(C2CC2C)=O)nn(C)nc1Br Cc1cc(C(=O)NC(C2CCCN2C(=O)Cc2cccc(Br)c2)C)c(C)cn1 Cc1cc(Br)sc1C(N1CCC(NC(=O)CSCC(N)=O)C1)=O C(=O)(CCCC#CC)N1CC2C(CNC(C(CC=C)OC)=O)(C2)C1 N1(c2ccc(COCCN(CCOC)CCN(C)C)cc2)CCCN2CCCC2C1 CC(C)CC(C)C(=O)NCC(C(C)C)NC(c1cc(N(C)C)ccn1)=O c1(C(N2CC(NC(=O)CCOCC3CC3)C(C(F)F)C2)=O)cc2c(s1)CCSC2 N1(C(=O)COC2CCCNC2)CCC12CCCOC2 c1(C(=O)NC2(COC)CCN(C(=O)C(C)OCCC(C)C)C2)cnc(O)cc1C C1(CC(=O)NC2(C)CN(C(=O)CCc3ccccc3F)C2)CCn2cncc2C1 C1(CNC(c2sc(CC)c(C)c2)=O)CCN(C(=O)C2=C(Cl)CC2)CCC1(F)F Cc1cc(C(=O)NCC(CO)NC(=O)C=Cc2cn[nH]c2)c2nccn2c1 C1(NC(C2ON=C(CC)C2)=O)CC(NC(c2[nH]cnc2C)=O)C12CCC2 CCC(CC)(CCNC(c1cccc(C(C)(F)F)n1)=O)NC(C1(N(C)C)CC1)=O Cc1ccc(Br)c(S(=O)(=O)NC2CN(C(=O)NC3CCN(C4CCCC4)C3)C2)c1 N1(C(C(c2ccoc2)NC(CCOCCCOC)=O)=O)CC2CCC(C1)C2C#N CC1CC(C(=O)NCCc2cccc(Cl)c2)CN(C(=O)Cc2ccc(O)cc2)C1 C=CCC(CC(=O)Nc1cc(CC)ccc1C)NC(=O)C(COC)OC C(=O)(CN=c1ccc(Cl)n[nH]1)NC(C)CCCCNC(C12CC(C1)C(C)(C)O2)=O c1(C(N(CC(CC)NC(CC2CC(=C)C2)=O)C)=O)cc(C(C)(C)C)[nH]c1C c1(CNC(C(C#C)(C)C)=O)ccc2c(c1)CCCC2NC(c1n[nH]cc1F)=O CCC(C)CC(=O)C(=O)N1CCC(CNC(C2CCCS(=O)(=O)C2)=O)C(O)C1 c1(CNC(C2CCCN2C(=O)Nc2ccncc2)=O)cc(C2CCC2)ccc1F c1(CC(N2CC3C(CNC(C4CC5CCCC5C4)=O)C3C2)=O)c(Cl)cncc1Cl CC(O)CCCC(=O)N1CCC(C)(CNC(C2CC(C(C)C)C2)=O)CC1 C12(C(=O)NCCCN(C)C3CC3)CC(CN(C(=O)CC3CCCCN3C)C1)C2 C1(NC(=O)C=CCCCCC)(CCC(N2CCC(=C)CC2)=O)CCC(C)(C)C1 c1(C(=O)NCC2CC(NC(C(C(C)O)(F)F)=O)C2)cc2cc([N+](=O)[O-])ccc2o1 C(=O)(C(C)(CC#C)NC(=O)CC1CCCC(C)O1)NCCCCCC#C O(NC(=O)C(Cc1cnc[nH]1)NC(C1CCOC1C)=O)CCOC C1(CCC)CC(C(=O)NCc2cc(C3CCN(C(C)C)CC3)no2)CCO1 FCCC(N=c1ccn2ncc(I)c2[nH]1)C1CCC(N2CCOCC2)CC1 CC12CN(C(c3ccc4oc(O)nc4n3)=O)CC1(C)CN(C(C1(C#N)CC1)=O)C2 CS(=O)(=O)c1ccsc1C(=O)NCC1COCCN1C(C1CCCCNC1=O)=O C(=O)(CC(C)CC(=O)N1CCC(C(N2CCc3n[nH]cc3C2)=O)O1)OC c1(C(=O)NCC(C)(O)CNC(C2CC(F)C2)=O)ccc2c(c1)NC(=O)CCS2 O=C1COc2ccc(-c3cscc3C(F)(F)F)cc2N1.c1(CC)ccc(Cl)cc1Br C(=O)(CCCC(=O)NC(C)(CSC)C(=O)NC(c1ncc[nH]1)CO)OC N1(C(CNC(C(CC)CC)=O)=O)CCN(C(=O)C2=COCCO2)C(COC)C1 c1(OC)ccc(OCCC(=O)NC2(CN=c3[nH]nco3)CCCC2)cc1 c1(CNC(C2N(CC)CCC2)=O)ccccc1CNC(=O)CCCc1ccsc1 C1(C#N)(C(=O)NCCN(C(c2n(CCC)nc(C)c2)=O)CC)CC12CCCC2 Cc1cc(Br)ccc1CC(=O)NCC1CN(C(C2CC=CCC2)=O)C(C)(C)C1 Cc1cccc(CN(C)C(c2ccn(CCNC(=O)C(C)n3cncn3)c2)=O)n1 c1(OC)cccc(C(=O)NCC2CC2CNC(=O)CC=C(C)C)c1O C1(O)(CCNC(=O)CC2CCOC2)CCCN(C(C2CCC3(CC2)CC3)=O)C1 CC1CC2(CC(C(=O)NC3(CCNC(=O)CCCF)CCOCC3)C2)C1 CC1CC=C(C(=O)NC2CC=CCC2C(=O)NCCCc2nnnn2C)CC1 c1(OC)cccc(Cl)c1C(=O)NC1CCC1NC(C1(C)CCC(OC)CC1)=O c1(CCC)ccc(C(=O)NCC2CC(CNC(=O)C=CCO)CO2)[nH]1 C(=O)(C#CC1CCOCC1)N1CC2=C(CN(C(CNS(N(C)C)(=O)=O)=O)C2)C1 C1(CNC(c2ncc(NC(C)C)nc2)=O)C(C)CCCN1C(C1CC1C)=O.CC C(=O)(CC(C)C(=O)NCC)OCC.C1(=O)C(C)(C)CN1 c1(C(=O)NC2(C)CN(C(c3cc(C(F)(F)F)ns3)=O)C2)cnc2ccccn12 C1(NC(C(CC)C)=O)CCN(C(c2nc(-c3ccccc3C)oc2C)=O)C1C N1(C(C2CCC(C)O2)=O)CCC2(NC(c3cncc(-n4cccn4)n3)=O)CCCC12 C12(NC(C=Cc3c(C)ccs3)=O)CCN(C(=O)C(c3ccccc3)F)CC1C2 c1(CC)ncc(C(=O)NC2CC3(C2)CN(C)C3)c(C)n1.C1(C)(C)CNC(=O)CO1 Nc1ccc(F)c(F)c1C(N1CCN(C(C2CCCS2)=O)C(C2CC2)C1)=O N1(C(c2c(C)n(C)cn2)=O)CCC2(CC2)CC1C(=O)NCCC(C)(C)C N1(C(C2(C#N)CC2)=O)CCC2(CCC(CC(N3CCOCC34CC4)=O)CC2)CC1 N1(C(Cc2c(Br)cn(CC)n2)=O)CCN(C(=O)C(C)(C)F)C(COC)C1 CN1CCC(C(=O)Nc2cccc(NC=O)c2)(NC(C2CC2(C)C)=O)C1 C(CC(C(C)C)NC(=O)CCc1ncnn1C)NC(C(CC)n1cccn1)=O CON(CCC(=O)N1CCSC(C)(C)C1)C(=O)c1ccc2c(c1)CC2 N1(C(CC2CCC(=O)O2)=O)CC2CCC1C(CNC(c1snnc1C1CC1)=O)C2 C12(NC(CC#N)=O)COCCC1CN(C(c1cc(C(F)(F)F)ncn1)=O)C2 C1(C(=O)NC2(C(C)O)CC2)CN(C)CCN1C(=O)Cn1cnc(=N)[nH]1 C1(NC(C2(CC)CN(C(c3cc4ccccn4n3)=O)C2)=O)CN(C)CCN(C)C1 C(CC(C(=O)N(CCCC(F)(F)F)C)NC(=O)C=Cc1cc(C)no1)OC N1(C(C2CC(=C)C2)=O)CC(NC(=O)Cc2cc(F)ccc2O)CC(O)C1 c1(C(N2CCC(O)(C(CNC(COC)=O)C)C2)=O)n[nH]c2c1COC2 C1(N(C(CCC2(NC(CCC=C=C)=O)CCC2)=O)C)CCC2(CC1)CC2 Cc1ncnc(O)c1C(N1CCC(NC(=O)C(N2CCSCC2)C)C1)=O CC(C)(CC(=O)N1CCCC(C)(NC(=O)COCCO)C1)C(F)F N1(C(CC(CNC(c2ncn(CC)c2)=O)(C)C)=O)CCC2CCN(C)CC12 CCC(C)CC(C(=O)NCCCCC(=O)NCC)NC(=O)C1=C(Cl)CCC1 N1(C(c2ccc(C(F)(F)F)cc2)=O)CCC12CN(Cc1c(Cl)cccc1I)C2 CCC(CC(=O)N1CC(NC(=O)Cc2ccn(C(C)C)n2)C2(CC2)C1)C(C)(C)C C1(NC(CN(CCC)C)=O)CCS(=O)(=O)C12CN(C(C1CC(C#N)C1)=O)C2 Cc1ncc2ccccc2c1C(=O)NCC1CC(C)N(C(=O)CCC(C)(C)C)C1 c1(C(=O)NC2CN(C(CC(C)(F)F)=O)CC2O)nc2ccccc2[nH]1 N1(C(CN(C(C)C)C)=O)CC(NC(=O)CNS(C)(=O)=O)C(S(C)(=O)=O)C1 c1(CNC(Cc2cc(CC)no2)=O)nc(C(=O)NCc2cncc(Cl)c2)c(C)o1 C(CC(C)C)(C(=O)NCC(F)CNC(c1cccc(F)c1Cl)=O)NC(C)=O C(C)(C)(C(C)NC(c1cn(CCO)nn1)=O)NC(C(F)OC)=O c1(N)ccc(O)cc1.C1(C(C)C)CC(C(=O)NC2CC(NC(C3CC3C)=O)C2)C1 c1(C(N(C2CCC2)C)=O)ccc(CNC(=O)CC2CCCOC2)o1 C1(NC2(c3n(CC(=C)C)nnn3)COC2)CC(C(=O)OC)C12CCC2 C1(Cc2cn(CCC=C)nn2)CN(C(=O)C(C)CC2CCC2)CCO1 c1(OC)ccc(OC)c(C(N2CCC(CCNC(c3n[nH]c(C)n3)=O)C2)=O)c1N c1(C(=O)NC2CCCC(CC(=O)NCc3ccnc(F)c3)C2)c(O)cccc1F C(CN=c1[nH]cnc2c(Br)cccc12)OCCNC(C1(CC#C)CCCCO1)=O c1(N2CCc3c(nc(C)o3)C2)nc2c(cc1C#N)C1CCC2C1 Cc1cc(C(N2CCC2C(N2CCC(Oc3ccccc3)CC2)=O)=O)cc(Br)c1 N1(CCC(=C)C)CCC2(CCN(C(c3n[nH]c4c(C)cccc34)=O)C2)C1 N(C1CCCn2ncnc21)C(c1c(CNC(C(CO)OC)=O)nccc1)=O CC1CCS(=O)(=O)CCN1C(c1csc(Br)n1)C(=O)NCc1cccc(Cl)c1 c1(C(=O)NCC2(NC(C(C=CCCC)O)=O)CC2)c(F)cc(F)c(O)c1F c1(CNC(c2c(OC)csc2)=O)ccnc(Br)c1 C1(C(=O)NC(c2ccc(Br)o2)C)C2CN(C(c3ccc[nH]3)=O)CC12 C(=O)(CC(C)(C)CC(=O)OC)NC(CN(C(c1ccc(C#C)cc1F)=O)C)C CC(F)(F)CCC(=O)NC1CS(=O)(=O)CC1NC(=O)COC1CCC1 c1(OCC)ncc(C(=O)NCC2CC(NC(C3CC3[N+](=O)[O-])=O)C2)cn1 Cc1cc(C(=O)NCC(C)NC(C2CC2c2ccccc2)=O)nnc1C C(CC(C)(C)CC(=O)N1CCC(C)(NC(=O)C(C)(C)C(F)(F)F)C1)OC CC1(CNC(C2CCCCC2CNC(C2COC(=O)N2)=O)=O)CC2(CCC2)C1 CC(C)C(C(=O)N1CCC1CNC(c1cncc(Cl)c1)=O)NC(c1cccs1)=O CCCCC(O)C(=O)NC1CCC(F)(CNC(C2(C)SCCCS2)=O)C1 C1(NC(=O)CCC2CC(F)(F)C2)CC2CC(C1)N(C(C13CCCC(C1)OC3)=O)C2 CN1CCN(c2cccc(C(=O)NCC3(CNC4CC4)CC3)n2)CC1 Cc1c(C(N2CCCC(C)(CNC(=O)C(C)OC3CCOC3)C2)=O)nn(C)c1N N1(C(c2ccc(C)n2C)=O)CCCC1C1CCCN1C(=O)CNC(N)=O c1(C(=O)NC(C)C(C)NC(c2cnc(C(F)F)s2)=O)coc(Cl)c1 Cc1noc(Cl)c1CCC(=O)NC(C)CC1CN(C(c2cnn(C(C)C)c2)=O)C1 C(C1=CCCN(C(=O)CC2CCCC3CC23)C1)NC(C1CC(OC)C1)=O.C1(C)CC1 c1(OCC)ccc(-c2nc(C(C(C)CC)OCC)n(-c3ccc(C)cc3)n2)cc1 Cn1cc(Cl)cc1C(N1CCN(C2CN(C(c3cc(CO)[nH]n3)=O)C2)CC1)=O c1(-c2cccc(C#C)c2)ccc2[nH]cc(C(=O)Nc3ccc(OC)c(F)c3)c2c1 Cc1cc(C(=O)N(C)CCNC(=O)CCN2CCC(F)C2)cn(C)c1=O c1(C(=O)NCCC(C(=O)N(CCCCC)CCO)O)ccc2cc[nH]c2c1 CC1CN2CCN1CC2C(=O)NCC(CNC(c1ccccn1)=O)C(F)(F)F C1(NC(C2C(c3ccc(C)o3)C2)=O)CCCC(NC(c2cnn(C)n2)=O)C1 c1(C(=O)NC2C(NC(=O)Cc3cscn3)CCCC2)cc2cccnn2c1 CCC1C(=O)Nc2ccc(C(=O)NCC3CC(NC(=O)CCS(N)(=O)=O)C3)cc21 N1(C(C(C)C(C)(C)C)=O)CC(C)(C)OCC1CNC(=O)CCC1CCCCCC1 C1(C(=O)NC2CN(C(=O)C(C)(C)COC(C)C)CC2C)(SC)CCC(F)(F)CC1 Cc1cnn(C)c1C(=O)NCCC1CCCCN1C(=O)CNC(=O)C1CC1 C1(CCNC(C(C2CCOC2)OCC)=O)CCN(C(=O)Cc2ncc(C)[nH]2)CC1 N1(C(c2cc(C(CC)C)no2)=O)CC(CNC(=O)CO)C(F)(F)C1 CC1CC(CNC(c2nn(C(F)F)cc2Cl)=O)CN1C(C1CSC1)=O c1(C(N2CCCC(CNC(C3ON=C(C)C3)=O)CC2)=O)nc2ccccn2c1F Cc1nc(O)[nH]c1C(=O)NCCCCNC(c1ccc(C2CC2)cn1)=O c1(C(N2CC3C(NC)C3C2)=O)cccnc1OC(C)C(F)(F)F C1(C(=O)NCC(CNC(C2CC(C)(CC)C2)=O)(C)OC)CC2CC(=O)C1O2 CC1CCN(C(c2ccsc2)=O)C1CNC(=O)CCc1cc(Br)n(C)n1 c1(C(C)C(=O)N(CCO)Cc2nc(C(F)(F)F)n[nH]2)cccc(C#N)c1 CC1CN(C(C2CCC(N(C)C)CC2)=O)CCN1C(C1CCS1(=O)=O)=O C=CC1OCCC1C(N1CCC1CC(=O)NC(CC)CCOC)=O C(C(C)(C)CC(=O)NC1CCC(C)(CNC(=O)C2=NOCC2)C1)N(C)C C12(NC(=O)Cc3cccc(C4CC4)c3)CCN(C(c3cocn3)=O)CC1C2 c1(C(=O)NC2CCCN(C(C3CC(=O)NC3)=O)C2)ccnc(O)c1F c1(C(N2C(CNC(C(C)OCCN(C)C)=O)CCC2)=O)cc(N)cc(O)n1 c1(C(C)C)cc(C(=O)NC2CCC(C)N(C(=O)C(=O)NC3CCCC3)C2)ccc1O CCC(CC(=O)NCCCC(C)NC(C1NC(=O)CC1C)=O)C(C)C C1(C2CCN(C(c3cn(C(F)(F)CO)nn3)=O)CC2)(NC(CC(CC)O)=O)CC1 C1(C#N)(C(=O)NCC(CNC(c2n(CC(C)C)ncc2)=O)O)CC2(CC2)C1 C1(NC(C(C)NC(CC)(C)C)=O)CCN(C(c2cncc(Cl)c2)=O)C1C(C)C c1(C(C)C(=O)NCC2CC3CC2CN3C(=O)CSC(F)F)ccc2c(c1)OCO2 CC(C)C(O)CC(=O)NCC(CNC(=O)CSCC(N)=O)CO c1(-c2n(C(C)CC3CC3)ccn2)ccc(F)cc1-c1cccc(C2CC2)c1F C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1(C)CCC(NC(C(C=C=C)C)=O)CC1 N1(C(c2c(C)ccc(OC)n2)=O)CC2CCN(C(c3nc(C)nn3C)=O)CC2C1 c1(C(N2CCN(C(=O)COCC3CC3)CC2CC2CC2)=O)ccc2occc2c1 C1(CC=C)(NC(C2CCCCN2CCC)=O)CCN(C(=O)C(CCC)N(C)C)C1 C1(C)(CC)CC(NC(C23CC(F)(C2)C3)=O)CN1C(c1ccc(C#N)cc1)=O c1(C2C(Cc3onc(CC(C(C)C)=O)n3)C2)ccncc1OC(F)F Cc1cc(Br)cc(CNCC2(OC(C)C)CCOC2)c1O c1(C(N2CCC(CC(N3CCCC(C(=O)OC)C3)=O)CC2)=O)c(I)ccnc1Cl CC1(C)CCCCC(C(=O)NC2CCCN(C(c3csc4nnsc34)=O)CC2)C1 C(CCC(F)(F)F)N(C(C1(NC(c2c(CC)con2)=O)CCCC1C)=O)C Cc1ccc(CC(=O)NC(C2CCN(C(=O)C(c3ccccc3)=O)C2)C)c(Cl)c1 Cc1ccc(F)c(O)c1C(=O)NCc1cn(-c2nc3ccccc3s2)nn1 CC(C)CCC(=O)NC.C1(C)CC1C1CCC1.C12(CCC1)CCC(=O)N2 C1(CNC(Cc2cccc(C(N)=O)c2)=O)CC12CCN(C(=O)CNS(N)(=O)=O)CC2 CC1CN(CCOC(c2nnc(-c3ccco3)n2C2CC2)=O)C=C1C C1(OC)CC2CC(CNC(=O)C#CCNC(=O)CC(C)(C)OC)CC12 n1(ONC(c2c(C#N)ccs2)=O)ccc(=NC(=O)CC(Cl)(Cl)Cl)[nH]1 C1(C(=O)NCCCC(C)NC(=O)CCOc2ccccc2)CCC(N(C)C)CC1 CCC(CC(=O)NCCc1ccsc1)N(C(=O)CC1CCCC2CC12)C N1(C(c2ccnc(OC)c2Br)C(=O)NCCSC)CC(C)OC2CCCCC12 C=C(F)C1(CC(=O)NCC(C)NC(c2ccc(NC3CCC3)cc2)=O)CCC1 C1(C(=O)NCC2N(C(c3c(C)nc(C(C)C)o3)=O)CC(F)C2)CCCC(F)(F)C1 N1(C(CC(C)(C)OC)=O)CCOCC(NC(=O)C(C2CCCO2)C2(COC)CC2)C1 c1(C(=O)NCC2(C)CCN(C(CC(CC)OC)=O)C2)cc2c(Cl)cncc2o1 C1(CC(=O)NC2(C)CCC2)C(NC(=O)NC2CC2C2CCCOC2)CC1O c1(NC(c2ccc(C)c(C)c2)C)ncnc2c1CCCC2 CS(=O)(=O)c1sccc1C(=O)NCC1(NC(=O)CC2CCOC2=O)CCC1 Nc1c(Cl)cnc(C(N2CC3CC2CN3C(=O)CC2=NNC(=O)C2)=O)c1Cl N1(Cc2ccc(OCC)nc2)CCC(O)C(C(=O)NC2CCCC(O)C2)C1 c1(C(N2CCC(NC(c3c(C)nc(CO)s3)=O)C(F)C2)=O)cnc2cc[nH]c2c1 N1(C(c2ccccn2)=O)CCCC2(C1)CN(C(=O)C(F)(F)Oc1ccccc1)C2 CCCCCC(=O)NC1CCOCC1OCC.c1(C23CC2NC3=O)ccccc1 c1(C(=O)NC2CC(NC(c3cn(-c4nccs4)nn3)=O)C2)cc(Cl)sc1Cl Cc1ccc(C=CC(=O)NCC(C)(Cn2cccn2)NC(=O)C(C)O)c(C)c1 CC(C)(CS(N)(=O)=O)C(=O)NC1CCCN(C(c2ccc(C(=O)O)cc2)=O)CC1 CCCC(CNC(c1ccnc(C)c1)=O)C(=O)N(CCN=[N+]=[N-])CC c1(CCC(=O)NC2(C)CC(C(=O)NC3(CC#C)CCOC3)C2)ccc(NC)cc1 CC1CN(C(=O)Cn2nnc(-c3ccco3)n2)CC1Nc1ccncn1 C(=O)(C1=CCCCO1)NCc1occ(C(=O)NC2CC(CC(N)=O)C2)n1 Cc1ncnc(O)c1C(N1CCCN(Cc2ccccc2)CC1)C1COC(C)C1 C(=O)(CCC(N)=O)NC(CNC(CNC(CN(C(C)=O)C)=O)=O)C C1(NC(=O)CC2CCCC2NC(=O)Cc2ccc(O)nc2)CC2CC3C(C2)C13 CCCC(C#N)C(=O)NCCCC(CO)NC(=O)CCc1cnoc1 N1(C(c2ncc(C)nc2)C(=O)NCc2cccs2)Cc2cccc([N+](=O)[O-])c2C1 C1(Cn2cc(C(C)OC)nn2)COCCN1C(=O)Cc1ccccc1C(N)=O C12(NC(c3c(C)scc3)=O)CCC(CC1)N(C(C1CNc3ccnn3C1)=O)C2 C(CN=c1[nH]c(=NCCCn2cncn2)[nH]c2c1CCC2)(C(C)(C)C)OC Cc1c(CCNC(C2CCN(C(c3ccoc3)=O)C2C)=O)cnn1C N1(C(C2C(C)C2)=O)CCOCC1CNCc1ccc(F)nc1 C#CCC(C)(C)C(=O)N1CC(C(=O)N(C2C3CCCC23)C)C(C)C1 N1(Cc2c(C)noc2C)CCC2CCCC12C(=O)OC(C)(C)C C1(NC(COCCOCC)=O)CCCC(NC(c2cccc(F)c2)=O)C1 c1(C(C)C)ccc(F)c(C(=O)NC(C)CCCNC(C2(CO)CCOC2)=O)c1 c1(OC(C)C)cncc(C(=O)N(C2CCCCC2N(C(=O)C(C)CO)C)C)c1 c1(C(C(=O)NC2CC(C(=O)OC)C2)N(CC(CC)C)C)nn(C)cc1CC1CC1 C=CCCC(F)(F)C(=O)NCC(CC(C)C)C(=O)NCC1(n2ccnn2)CC1 C1(CNC(C(C)NC(=O)NC)=O)CN(C)CCN1C(C1CC1C(C)O)=O N1(C(c2cnc(OC)c(C)n2)=O)CC(NC(=O)Cc2nccn2C)C(N=[N+]=[N-])C1 C1(NC(c2cc(CC)[nH]n2)=O)CN(C(=O)Cc2ccc(F)c(CC)c2)CC2CC12 C1(NC(c2ccc(C)s2)=O)CCC(C)N(Cc2snnc2C)C1 N1(C(CCOCCCOC)=O)CCC(C)N(C(C2CC(C)(F)C2)=O)CC1 N1(C(c2n[nH]c(C)c2C)=O)CCC2(NC(C3CC3C3CCCC3)=O)CCCC12 C1(NC(CC(C)(C)C2CC2)=O)CCCN(C(c2cc[nH]c2C2CC2)=O)CC1 N1(C(c2ccc(OC)c(F)c2)=O)CC2(CC1CNC(=O)CCC(N)=O)CC2(F)F c1(C(=O)NC2(C)CCN(CC#C)CC2)cccc2ccsc12 c1(C(=O)NCC2C(C)CCN2C(c2ccoc2Cl)=O)cc2ccnn2cn1 c1(NC(=O)CC2CCCN2C(c2cnncc2O)=O)cc(Br)cc(Cl)c1O C#Cc1cnn(C)c1C(=O)NCC(C1(Cc2ccc(F)cc2F)CCC1)N(C)C C1(NC(C(C)OC)=O)CC(C)N(C(c2cccnc2Cl)=O)C1 CCC(C)C(C)C(=O)N(C)CCNC(C1(c2cccc(Cl)c2F)CCCC1)=O C1(NC(c2cn(CC(C)C)nc2)=O)CC2CC(NC(=O)Cn3ccnn3)C2C1 N1(C(C=C(C)C)=O)CCC(n2nccc2Nc2cncc(Br)c2)CC1 CON1CCC(C(=O)NC2CCCCC2N(C(=O)CC2CC(SC)C2)C)CC1 N(C1c2cccc(F)c2OC1C)C(N1C(c2ccc(OC)cc2F)CCC1)=O N1(C(c2n[nH]c(C)n2)C(=O)Nc2ccc(OC)cc2)CCCN(C(C)CO)CC1 N1(C(Cc2c(C)nsc2)=O)CC(C(=O)NCC(C)(O)C(C)(C)C)CCC1(C)C CS(=O)(=O)C1CCCC1C(=O)NCC1CN(C(=O)CCc2ccc(F)cc2)C1 c1(C(=O)NCC(CC)NC(c2c(C(F)(F)F)n[nH]c2C)=O)cncc(SC)c1 c1(C(=O)NCCC2N(C(C(C)c3ccsc3)=O)CCC2)ncccc1C(F)F C(C1CN(C(c2ccncc2Cl)=O)CC1C(=O)NC(c1ncc[nH]1)(C)C)=CC Cc1cc(C(=O)NCCCN(CCCCNC(C2(C#N)CCCC2)=O)C)ccc1F C1(C(=O)NC2(CC(=O)NC(C(C)C)c3cncs3)CCC2)CCCC2CCCCC12 CCCC(C#N)C(=O)NC1(CNC(c2ccc(-c3sccc3C)s2)=O)CC1 C12(C(N3CCCC(F)(CNC(C4C=CCCC4)=O)C3)=O)CCC(CO)(CC1)CC2 c1(C(=O)NC(C2CN(C(CC)=O)C2)C)cnn(-c2cccc(C(C)C)c2)c1C C(C)(CC(=O)NCCCCCC(=O)N1CCCC1)C1(C2(CC(C)C)CCC2)N=N1 c1(NC(C(=O)C(=O)N2CCCC2)C(F)(F)F)cccc(S(=O)(=O)C(F)(F)F)c1 c1(C(=O)NCC2C(C)CCN(C(=O)C(C)(Cl)Cl)C2)cnn2c(N)ccnc12 c1(CN(C(c2cnn(C)c2C)C(=O)NCC=C)C)ccc(Cl)c(Cl)c1Cl C1(CC(=O)NCCN(CCOC)C(c2ccnc(NC)c2)=O)CC2CCC1CC2 C=CCC(C(=O)NCC1CN(CC(=O)OC(C)(C)C)C(=O)O1)OC CC(C)C(C(=O)NC1CC(=O)N(C(C)C)C1)NC(c1ccncc1Cl)=O c1(NC(C=CC(C)NC(C2(SC)CC2)=O)=O)cc(C#N)ccc1O c1(C(=O)NCC2C(CNC(CC3ON=C(CC)C3)=O)C2)cc2cc(F)ccc2o1 c1(C(=O)NCC(CN(C(c2cc(C)sn2)=O)C)(C)C)cc(C)n(C2CC2)n1 C1(NCc2scc(C(=O)NC(COC)C)n2)CCCC(C)C1 c1(NC(C2CC(O)CN2c2ccncn2)=O)n[nH]c2ccccc12 Fc1cccnc1N1CCN(c2cnnc(Br)n2)CC1.c1(N)ccccc1C(F)(F)F N1(C(CCCOC(C(C)C)=O)=O)CCC2C1CCCN2C(C1C=CCCC1)=O c1(OC)cc(C(=O)NC2CCCN(C(=O)C=C3CCC(C)C3)C2)cc(F)c1C#N N1(CC(=O)NCC2C3CCC(C3)N2C(=O)CC2CC23CC3)CCCCCC1=O c1(C(=O)NCC2N(C(c3cncc(C)c3)=O)CCC2)ccc(N)c2ccncc12 c1(OC)ccnc(C(N2CC(NC(=O)CC3CCS(=O)(=O)C3)CC2C)=O)c1 Cc1ccc(C)c(CN2CCC(NC(c3c(Cl)cncc3Cl)=O)C(O)C2)c1O C1(NC(C2SCCS2)=O)CCCC(C(=O)NCCCc2cccs2)CC1 N1(C(c2c(C)nsc2N)=O)CCC(C2CC2)(NC(=O)CN2CCCC2C)C1 C(=O)(CCN=c1[nH]ccs1)N1CC(C)(C)C(CNC(=O)CCc2cnoc2)C1 CC1(C)CN(C(=O)CC23COCC(C2)C3)CC1NC(c1ccc(Cl)c(O)c1)=O N1(C(Cc2cn(C)nn2)=O)CC2(CCC2)CC1C(=O)NCC1NC(=O)NC1=O c1(CC(=O)NCC2CN(C(c3ccnc(OC)n3)=O)CC2O)ccnc(Cl)c1F O(S(=O)(=O)c1ccc(Cl)c(Br)c1)c1c(C)ccc(NC(=O)C(C)C)c1 C1(C(N2CCC(CN(C)C(c3cscc3Cl)=O)CC2)=O)CC(=O)C12CCCC2 Cc1nnc(CCCC(=O)NC2CCN(C(C3CN(C(C)C)CCO3)=O)C2)n1C c1(NC2CC(C)SCC2)cc(Br)ccc1S(=O)(=O)N1CC2CSCC(C2)C1 c1(N(CC(C)C)C(C2CC2C2CCCC2)=O)ncnc2c1CCC2 C=CC(C)(C)CC(=O)N(C1CCN(C(c2cn(C)nc2Cl)=O)CC1)CC c1(N(C2CCOCC2)C(CN2CCC(CC)C2)=O)ccc(C)c(OC(F)F)c1 c1(C(=O)NC(CCOC)CNC(=O)C(C)n2ccnc2)ccc(C#N)c(F)c1 C1(NC(C(=O)OC)=O)(Cc2ccccc2Cl)CCCN(C(=O)NC(C)(C)C)C1 CC(C)CC(C)(O)C(=O)N1CC2(C1)CN(C(c1ccc(C3CCCC3)cc1)=O)C2 CC1CC(C)N(C(=O)CCNC(=O)CCS(C)(=O)=O)CCN1C(C1CCC1)=O C1(NC(c2c(Br)cn(CC)n2)=O)COC2(CCN(C(=O)CC3CC3)CC2)C1 CC1CCCCC1(CNC(c1cnc(S)n1C)=O)NC(c1cscc1C(N)=O)=O S(=O)(=O)(c1ccccc1F)NCc1ccc(N2CC(C)CS2(=O)=O)cc1 c1(N2CCC(NC(c3c(CCC)n[nH]c3)=O)C(F)C2)ncnc2ccc(Cl)cc12 c1(C(=O)NC(CCC)C(=O)NCC2CCC(CO)CC2)cc([N+](=O)[O-])c[nH]1 c1(CN2C3CN(CC(=O)Nc4ccccn4)C(C3)C2)cn2ccc(CO)cc2n1 CC1(C(=O)Nc2cc(CO)ccc2O)CCN(Cc2c[nH]c(Br)c2)CC1 c1(OC(F)F)ccc(C=CC(N2CC3CC2CN3C(=O)C=CCO)=O)c(OC)c1 CC(C)(C)CC(O)CC(=O)NCCC(O)C(=O)Nc1ccc(F)c(CO)c1 C1(n2cc(-c3n(C)c(S)nn3)nn2)CC2(CCCCC2)CO1 CC(C)C(C)CN(CCC(=O)NCCCN(C(=O)CC1(O)CCC1)C)C C1(C(=O)NCC(CNC(CN(c2ccccc2)C)=O)(C)C)CCC2(CCC2)O1 Cn1nc(-c2ccco2)cc1NC(c1sc(Br)cc1Cl)=O C(=O)(C1=COCCO1)NCC=CCNC(Cc1c(C)cccn1)=O N1(C(c2ccc(OCC(N)=O)cc2)=O)CC(CNC(=O)CC2CC2)C2(CC2)C1 CC1CCc2ccccc2N1CCC(=O)NC(CNC(=O)Cc1cnc[nH]1)CO C1(NC(C2(CNC(CN(C3CCC3)C)=O)CC(C)(C)C2)=O)C=CC(C)(C)CC1 C(CCC)(C(=O)NC1(C)CC(C(=O)NCCc2ncon2)C1)=CCC C#CCC(CC#C)C(=O)NC(CN(C(=O)C=C1CCOCC1)CC)CC Cn1ccc(C(=O)NCCOCCNC(c2csc(CO)n2)=O)c1 CCC(C)N(OC)C(=O)C1C2CCN(C(C3CC(=O)NC(=O)N3)=O)CC12 CCC(CNC(C1CC(CCSC)C1)=O)NC(=O)CCc1ccsc1 CC1CCCC(C(N2CC(O)(CCNC(=O)CC3(C)CCCC3)C2)=O)CC1 C1(NC(Cc2c(C)scc2)=O)C2CCC1N(C(=O)C(C1CCCCC1)N(C)C)C2 c1(NC(c2cnn(CCO)c2)=O)cnc(C2CCNCC2)o1 CCCC(C)(O)CC(=O)NCC1(NC(C23CCCC2C3(F)F)=O)CCCCC1 S(=O)(=O)(c1ccc(C(=O)NC2CC2CNC(=O)CCn2ccc(C)n2)o1)NC CC(CCC(=O)NC12CCN(CC1)C2)NC(C1CC(=C2CC2)C1)=O c1(NCC(=O)NC)nc(NCC(CC(C)O)c2ccccc2)c2ncn(C)c2n1 C(C)(CCN=c1[nH]cc(C#N)cc1C)NC(c1ccc(C)c(F)c1)=O N1(C(c2c(CC)cno2)=O)CCCC(C)(C)C1CNC(c1ccc(O)cn1)=O Cc1cc(C(=O)NCC(C)CN(C)C(C2CC(N(C)C)C2)=O)ccc1C(C)C N1(C(CC(C)OC)=O)CCC(c2ccccc2)(NC(c2cc(C)cnn2)=O)C1 C1(NC(=O)CCOCC2CC2)CCN(C(C2(C3CCC3)CC2)=O)CC12CCC2 c1(OC)cnnc(C(N2CCC(NC(=O)C(=O)NC(C)C)C2C2CC2)=O)c1 c1(C(N2C(C)CC(NC(C3CCCN3CC(F)(F)F)=O)C2)=O)ccn2ccccc12 N1(C(C2CCC(N(C)C)C2)=O)CCCC(C2OCCO2)C1 c1(OC)cc(C)c2cc(C(N3CCCC3c3ccccc3OC)=O)[nH]c2c1 C(=O)(CC(C(F)(F)F)N(C)C1CC1)N(C)CC1(C)CC(C(=O)NC(C)(C)C)C1 C1(NC(c2scc(C)c2Cl)=O)CCC2CC1CN2C(c1ccc(C#N)[nH]1)=O c1(C(=O)NCCN(C(=O)CCS(=O)(=O)NC)CCC)cn(CC)c2ccccc12 CCC(C)N(OC)C(=O)CC1CCCN(C(=O)C=Cc2cn(C)nn2)C1 c1(C(=O)NCCCCCN(C)C(C2CCOC2(C)C)=O)ccc2cnn(C)c2c1 C=CCC(CC)C(=O)N1CCC(C(=O)NCCCCOC)(C(C)C)C1 C1(C(=O)NC2(CO)CN(C(C3(CCO)CC3)=O)C2)CCCC(F)(F)CC1 c1(OC)c(C(N2CCC(O)C(NC(=O)C=C3CC3)C2)=O)oc2ccccc2c1=O CCCCC(F)C(=O)NCC(C)(CC)NC(=O)CC1CN(C)CC1O c1(C2C(N)C2)ccc(C)cc1.c1(C2CN(C(c3c(C)c[nH]c3)=O)C2)ccc(O)cc1 c1(C(N2C(C)CC(NC(c3c(CC)n[nH]c3)=O)C2)=O)cc(C)cc(Br)c1F c1(C(=O)NC2CC(NC(C3(C(N(C)C)=O)CC3)=O)C2)cc(O)nc2cnccc12 N1(C(C2C(C)CCOC2)=O)CCC(C(=O)NCCC2CCCC3CC23)C(C)(C)C1 C1(C(N(CCCC)CCO)=O)(OC)CCN(Cc2cnc(N3CCCC3)nc2)CC1 C1(NC(C(CCC2CC2)NC(C(CC)n2cncn2)=O)=O)CCn2nccc2C1 c1(OC)ccc(O)cc1C(N1CCC(NC(=O)CCSC(F)(F)F)C12CC2)=O C1(CCNC(CCSCCC)=O)CCCN1C(=O)C(CO)N(c1ccccc1)C N1(C(C(CC)C#N)=O)CC(OC)CC(NC(C2(c3ccn(C)n3)CC2)=O)C1 C1(CNC(CC(CC)SC)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CC12CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CCCC(CNC(=O)C(c2cn(C)nn2)OC)C1 c1(C(=O)NCC2N(Cc3cnc(CC(C)C)o3)CCC2)cccc(F)c1 c1(C(N2CCN(C(=O)CS(=O)(=O)CCO)C(CO)C2)=O)cc2cccnc2[nH]1 Cc1ccc(C(N2CC=CCC2C(N2CCCC(CC3CC3)C2)=O)=O)cc1F C(=O)(C(O)CC(F)(F)F)N(C1CCN(C(=O)C=Cc2ccccc2OC)C1)CC c1(SCC(N2CC3C(NC(C=NOC)=O)C3C2)=O)nnc2ccccn12 c1(OC)ccc(C(=O)NCCCN(C)C(c2cocc2C)=O)nn1 c1(CCNC(C(C)(C)C)CCC2(O)CCCCC2)c(F)c(F)c(F)c(F)c1F C1(C(=O)NCC(CC(F)(F)F)NC(c2cn(C)nc2)=O)CCC(N=[N+]=[N-])CC1 N1(C(=O)OCC)CSCC1C(=O)NC1CCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(C(N(CC(C)O)CC(C)O)=O)CCN(C(=O)CC2C=CCCC2)C1C C1(NC(c2c(C)[nH]nc2Cl)=O)CC2CC1N(C(c1cc(Cl)ccn1)=O)C2 N1(C(CCNS(CC)(=O)=O)=O)CC(CNC(=O)C=Cc2ccc(C)o2)CC1(C)C N1(C(C2C(NC(C3CCCO3)=O)C2)=O)CCOC(C2CC2)C1 Cn1ccc2nc(N3CC(c4cccs4)(NC(c4ccno4)=O)C3)ncc12 CC1COCC(C(=O)NCc2n[nH]cc2C(=O)N(c2ccccc2)C)O1 CC(C)CC(C)CC(=O)NCC=CC(N1CCN(C)CC1)=O N1(C(C(C=C)(C)CC)=O)CCC(C(=O)NCCCn2cncn2)C(C)(C)C1 C(=O)(C(Cc1ccnn1C)C(N)=O)OCC.C(C)(C)(C)OC(=O)O c1(C(CO)NC(C2NCC(=O)NC2)=O)c(F)cccc1Cl c1(C(N2CCC(OC)(CNC(=O)CN3CCC3C)CC2)=O)noc2c1COCC2 CCC(CC(=O)N(C)CCN(C(=O)C(C)COC)C(C)C)C(C)C c1(C(=O)NC2CCC(NC(c3ccc(CC)s3)=O)CC2)cc2n(c1)CCCC2 CCC(C)(CNC(c1cnnn1C)=O)C(=O)N1CC2C=CC1CC2 c1(C(N2CCC3C(NC(C(C)OCC=C)=O)C32)=O)ccnc2c1cnn2C c1(CN2CC3C(CN(C(c4cnn(C)c4C4CC4)=O)CC)C3C2)cccc(F)c1F c1(SC)ccc(C(=O)N(CC(C)NC(c2nocc2Cl)=O)C)cc1[N+](=O)[O-] n1(CC(=O)NC(CC)CN(C)C(C2CCSC2)=O)nnc(C)n1 C(CC(=O)N1CCCC1C(O)CO)(C(F)F)NC(CCc1ccc(C)o1)=O c1(C(=O)NCCCCNC(CCC2CCC(C)O2)=O)cnc2ccccn2c1=O Cc1nnc(C(=O)N(C(C)CNC(=O)C=CI)C)s1 C1(CNC(C=C(C)C(C)C)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)CC1C CCC(CC(=O)NC(Cc1ccc(OCC(F)(F)F)cc1)CO)c1ccccc1 c1(C(=O)NC(c2ccccc2F)C(=C)C)cc(C(F)F)cc(C(C)C)c1 CC1CC2CN(C(=O)CC3CC3)CC2N1C(C1CC2CC2C1)=O N1(C(C=Cc2n(CC)ncc2)=O)CCCC1C1CCCN1C(c1nonc1N)=O Cc1cc(C(N2CCSCC2CCNC(C2CC2C(F)F)=O)=O)sc1C C(C)(CO)(CN=c1ccc(Br)c(S(=O)(=O)NC2(c3ccccc3)CC2)[nH]1)OC C(=O)(CC1CCOc2ccccc21)NC(CCCC)CNC(=O)C(Cl)=CCl N1(C(c2c(CC)n[nH]c2)=O)CC2(CC(NC(=O)C(c3ccccc3)F)CO2)C1 N1(C(C2(OCC)CCCC2)=O)CCOC(C(C)NC(c2cncc(F)c2)=O)C1 C1(C(=O)OCC)CCCCN1C(C1CCCN1Cc1ncco1)=O C1(C(=O)O)CC2C(CC1C(=O)NCCCOc1ccccc1O)C2(F)F CC1=NN(C)C(=O)C1CC(N1CCN(C(c2[nH]cnc2C)=O)C(C2CCC2)C1)=O N1(C(CC(=O)NCC#C)=O)CCCC(NC(c2cncc(C)n2)=O)C1CC c1(C(=O)OC)ccc(S(=O)(=O)NC2CC2C(=O)Nc2cc(O)nc(C)c2)cc1 C1(C(=O)NCC=CCC(=O)N(CC(C)OC)C)CCCC(=O)C1 c1(C(N(CC(CO)(CO)NC(=O)C=Cc2cnc[nH]2)C)=O)csc([N+](=O)[O-])c1 CC1(CNC(c2ccncn2)=O)CC(F)(F)CN1C(c1cscc1Cl)=O N1(C(CCC=CC(C)C)=O)CCN(C)C(C(=O)NCC(c2cccs2)O)C1 c1(CC(=O)N(c2ccc(O)cc2)CC(=O)OCC)cccc(F)n1 C1(C2CCCNC2)(C(N(CCC(=O)O)C2CC2)=O)CC1 C1(C)(CNC(CCN(C(CCOC)=O)C2CC2)=O)C=CCCC1 C1(NC(C(C(C)C)OC)=O)CC2(CCCCN2C(=O)C(CSC)OC)C1 c1(C(=O)NC2CCC(N(C)C(c3cccs3)=O)C2)cccc(NS(C)(=O)=O)c1 C1(C(N2C(CO)CC(NC(C(CCCC)NC(N)=O)=O)C2)=O)Cc2nnc(C)n2C1 Cc1ccc(F)cc1N(C)Cc1cccnc1.c12coc(n1)CS(=O)C2 Cc1cc(C(=O)NC2(C(=O)NC(c3ccns3)C)CCCC2)ncn1 C(=O)(CC(C(=O)N1CCC(NC(=O)CC(C)OC)C1C)N(C)C)OC c1(OCC)cccc(Br)c1C(=O)NC1CCN(C(=O)CN(C)C(=O)OC)CC1F C1(CNC(c2ccc(C(CC)C)cc2)=O)CCCCN(C(=O)CC(F)F)C1 CCC(C)(C#N)C(=O)NCC(C)CNC(c1nc(C)ccc1Br)=O c1(C(=O)NC(CNC(C(Cc2c(C)noc2C)C)=O)C)ccc(F)c2occc12 CN=c1[nH]c(=NCc2cncnc2)[nH]c(=NCCCN2CCCN(C)CC2)[nH]1 c1(C(=O)OC)cc(NC(=O)C(=O)NC2CCC2CF)on1 N1(C(CCNC(CC(C)C)=O)=O)CCCN(C(c2ncccc2Cl)=O)CC1C c1(CC(=O)N(C)CC2(CNC(C(C(CC)O)C)=O)CC2)c(C)nc2ccccn12 CC(C)CCCC(=O)N1CCC(NC(c2cn(C(C)C)nn2)=O)C1 CCC1=NOC(C(=O)NC(CNC(=O)C(c2cncn2C)=O)CC(C)C)C1 Cc1nn(CCO)c(C)c1C(=O)NCC(C)CN(C)C(C1COC(=O)C1)=O Cc1cc(C(=O)NC2CC(F)(CNC(c3cc(C(C)C)on3)=O)C2)c(N)cc1F N1(C(C=C(COC)C)=O)CC(C2CN(C(=O)Cc3ccc(Cl)c(OC)c3)C2)C1 C1(C(N2CCC(NC(c3sccc3-n3cnnn3)=O)C2)=O)CCCCC12CCC2 C1(C(=O)NC23CC(CNC(c4cnccc4Cl)=O)(C2)C3)CCCC1C1CC1 c1(NC(N(CC(c2ccccc2)CC)CC)=O)nc2ccc(I)cc2s1 C=CCN=C(NCc1cc(Cl)n(C)n1)N1CCC(CC(=O)OC)CC1 c1(CC(CNC(c2cc(C3CC3)ns2)=O)CO)ccccc1F C(=O)(CC1=CCCCC1)NCC(N(C(C(C(COC)C)C)=O)C)C1CC1 N1(C(CCOCC#C)=O)CC(C)C(C)(CNC(c2cc[nH]n2)=O)C1 c1(N(CCOc2c(C)cccc2)C)ccc(S(=O)(=O)N(C)CC2CC2)c(Cl)c1 c1(C(=O)NC(C)CC#N)cc(N2CCCC2)ccn1.C12CCCC1C(=O)N2 N1(C(c2n(C=C)ncc2)=O)CCC2(NC(=O)C=C3CCSCC3)CCCC12 c1(CCC(=O)NCC(C)N(C(c2n[nH]c(C)n2)=O)CC)cncc(F)c1 c1(C(=O)NC2C3N(C(C(C)C#N)=O)C(CC3)C2)cc(Br)cc([N+](=O)[O-])c1 N1(Cc2c(C)nc(Cl)cc2)CCc2ncc(NC(C3CCCCO3)=O)cc2C1 c1(C(N2CCC(OCCNC(=O)Cc3cncs3)C2)=O)cncc(C(F)F)c1 c1(C(N2C(C)(CC)CC(NC(c3csnn3)=O)C2)=O)cc(O)c2cnn(C)c2c1 N1(C(C2(CC#C)CCCCO2)=O)CCC(C)N(C(C2CC3CCC2CC3)=O)CC1 Cc1ccc(O)c(NC(=O)CC2CN(C(=O)C(O)CNC(N)=O)CC2C)c1 c1(OCC)cncc(NC(C2CCCN2C(=O)CCc2ncccc2Cl)=O)c1 C(=O)(C(CN(C)C)C(C)C)NC(CC=C)C(=O)N1CCCC(CSC)C1 C1(C(N2CCC(NC(=O)NC)CC2)=O)CCC2CCC1N2C(C1CNC(=O)O1)=O C1(C)(C(N2CCCC(CNC(C(=O)NCCOC)=O)C2)=O)CC2(CCC2)C1 Cc1nc(CCNC(C2(NC(=O)CCc3ccsc3)CCOCC2)=O)c(C)o1 C(=O)(C1=C(c2ccccc2)SCCO1)N1C2CC(NC(=O)CC(F)(F)F)C(C2)C1 CC(C)(CC#N)C(=O)NCC1(F)CCC(CNC(=O)CSc2ccccc2)C1 N1(CC(=O)NC2CCC2N2CCOCC2)CCN(CC(N2CCCC2)=O)CC(O)C1 C12(C(N3CC(N(C(=O)Cc4ccsc4)C)C3)=O)CCCC1CS(=O)(=O)C2 CCCCCCC(C)(CC)C(=O)NC(CNC(C1(C(N)=O)CCC1)=O)CC CC1Cc2cccc(C(=O)Nc3cccc4c3OCC4C)c2O1 N1(C(C2(C)COC(=O)C2)=O)CCCC(C)(C)C1CNC(=O)CCCC1CC1 c1(C(C(=O)NCCCN(CCCC)CCCC)N)cccnc1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(C=COCC)=O)(CO)C1 c1(CNC(C2(C#C)CC2)=O)ccc(C(=O)NCC(C2CCOCC2)C)cc1 N1(C(C(C=C)CC)=O)CCC(C)(C)C1CC(=O)NC(C(C)(C)O)C1CC1 C(=O)(C#CC1CCCOC1)NC(C)(C)CNC(=O)C(C)(C)C(C)(C)C C1(C2CC2)(C(N(C(COC)COC)C)=O)CCN(C(=O)OC(C)(C)C)C1 N1(C(C2CC(=O)N(C)C2)=O)CCC(CN(C(=O)CC)CC2C(=C)CC2)CC1 Nc1ccnc(C(N2CCC(F)(CNC(c3cncn3C3CC3)=O)C2)=O)c1 c1(CC(C)NCc2cn(CCCCCO)nn2)ccc(O)cc1 C1(C(N2CCC(C)(NC(c3sc(C)c(O)n3)=O)C2)=O)CC1C1CCCCC1 c1(CC)nc(=N)[nH]cc1C(=O)NC(CNC(=O)C1=CCCC1)CC(F)(F)F c1(C(=O)NC2CC(CNC(=O)CC3CCC4CC34)C2)cc2c(=O)[nH]ccn2n1 N1(C(C2CC=CCC2)C(=O)NCCCF)CCCC2(CC(O)C2)C1 N1(C(C2CCCC(C)(C)C2)=O)CCC2(CC1)CN(C(=O)Cc1ccccc1Cl)C2 CC1(C)CN(C(C2CC(NC(=O)C=Cc3cc[nH]n3)C2)=O)CCO1 CCCC(CC)CC(=O)NC(C)CCNC(=O)CCSc1ccccc1F c1(CNC(c2cc3ncccc3[nH]2)=O)cccc2ccccc12 C1(C(N(C2CN(CC(=O)Nc3cccc(F)c3)C2)C)=O)C2CC3C(C2)C13 C1(C(=O)NCCCCCNC(CSCC#C)=O)CCC(C2CC2)C1 CCC(CC(=O)NCCOCC(=O)NCC1CCCC12CC2)C(C)(C)C Cc1c(NC(=O)C(CCC2(C#N)CC2)N(C2CC(F)(F)C2)C2CC2)cccc1Cl C(=O)(C(O)CC(C)(C)C)NC(CNC(c1n(CC)nc(C2CC2)c1)=O)CC(C)C C(=O)(C1=NN2CCCN=C2N1)N1C(CCNC(C=CC2C(C)C2(Cl)Cl)=O)CCC1 c1(C(=O)NCCC(C)NC(=O)C(C)(C)c2ccnn2C)cc(Cl)c(Br)[nH]1 C1(NC(CN2CCN(CC)CC2)=O)CC(F)CN(C(c2cncs2)=O)C1 N1(C(C=C(CC)C)=O)CC2(CC(NC(=O)CCNC(=O)C=CCl)C2)C1 C1(NC(C(c2ccco2)NC(C2CC3(CCC3=O)C2)=O)=O)CCCCCCC1O c1(C(=O)NCC(CO)NC(c2ccn(C)n2)=O)ccc2cc(O)ccc2c1 c1(CN2CCN(C(C3C(C4CCC4)C3)=O)CC2)cc(-c2nn[nH]n2)cc(F)c1 C(=O)(C(CC)C(=O)OC)N(C)Cc1ccc(CNC(C2CC(CCC)C2)=O)cc1 c1(C(N2CCC(CC(=O)NCC3(C)OCCO3)C2)=O)ccnc(Br)c1F CCC(CC(=O)NC(C)(C)CN(C(=O)CCCCN(C)C(C)=O)C)C1CC1 C(c1ccc(SC)s1)=CC(=O)NCC(CC=C)NC(=O)C(C)CC1CCCC1 c1(C(C)(F)F)ccc(C(=O)NCCOC2CN(C(C3CC3Cl)=O)C2)nc1 c1(C(=O)NCC(C2CCCC(C)C2)=O)cc(S(N)(=O)=O)cc(F)c1Cl c1(C(N2C3(CN(C(c4c(C)ncn4O)=O)C3)CC2)=O)cc(C#N)c(N)cc1O CC(C)CC(O)C(=O)NC1(C)CCN(C(=O)C(C)C(F)F)CC1 N1(C(C2OCCC(=O)C2)=O)CCC(NC(=O)C=Cc2ccco2)C(F)C1 c1(N(C(C)C)C)cc(N2CC3C(C(N4CCN(C)CC4)=O)C3C2)nc(=N)[nH]1 CC1(CNC(C2CC2F)=O)CN(C(=O)C(c2ccc(F)cn2)(F)F)CCO1 c1(C(N2CC(O)(CNC(C3C4COCC34)=O)C2)=O)ccccc1Br c1(CC(C)C(=O)NCC2C=CCN2C(=O)C2=COCC2)cccc(F)c1 C(=O)(CCCC(=O)NC)NCC1N(C(C(CCC)F)=O)CC(O)C1 N12CCOCC1CC2=O.c1(OCC)nc(C(=O)NCCc2ncoc2C)co1 Cc1cc(C(=O)NCC2COCCN2C(c2cc(Br)ccc2Cl)=O)ncc1F C1(CNC(C(c2ccc(C(F)F)cc2)C)=O)CCC(NC(=O)C(F)(F)CO)CC1 N1(C(C(CC)SC)=O)CCCCC12CN(C(=O)CN(c1c(C)noc1C)CC)C2 N1(C(C(CC(C)C)ONC(CC2ON=C(C)C2)=O)=O)CCCC(C)(C#N)C1 C(C(C)(C)C1=CCCC1)NC(C(C1CN(C(CC2CC(SC)C2)=O)C1)OC)=O Cc1sc(C(=O)NC2CCN(C(c3ccoc3Cl)=O)C2C)nc1Br CCC(C)(C(=O)N1CCN(C(C)CNC(C2(C3CC3)CCC2)=O)CC1)C(F)F CC(CN=c1[nH]c(N(CC(C)(C)CO)C)nc2c1COC2)Oc1ccccc1F C1(C(N2CCC(N(C)C(c3nccnc3Cl)=O)C2)=O)CC2CCC(C1)S2 c1(CN2CCC(F)(C(N3C(C#N)C4CC4C3)=O)CC2)cccc2c(Cl)ccnc12 c1(CC(=O)NCC(C)NC(C2CNC(=O)N2C)=O)c[nH]c2cc(F)ccc12 Cc1cc(NC(=O)C(N2CCC23CCSCC3)=O)ccc1S(N)(=O)=O C(CCC(C)C(=O)N1CCN(C(c2nc(C)ccc2OC)=O)C(C)C1)OC CN1CCC(C)(C(N2CC(NC(=O)C(Cl)=CCl)C(F)C2)=O)C1 N1(C(C)C(=O)OCCc2csc(O)n2)CCC(CC(c2ccccc2)=O)CC1 c1(OC)ncc(Br)cc1NC(C1CC1C(=O)Nc1cccc(SC)n1)=O N1(C(C(C(=O)OCC)OC)=O)CCOCC(NC(=O)CCC2CC(F)(F)C2)C1 c1(C(=O)NC(C)(CNC(C2CCC(O)C2)=O)CO)nnc(Cl)cc1N CCCCCCCC(=O)NC(CN(C(=O)Cc1ccnc(Cl)c1F)C)CC C=C(C)CCCC(=O)NC1(C)CN(C(c2ccc(OC)cc2C(F)F)=O)C1 N1(C(=O)NC2CC(C)C2)CCCC2CN(CC(=O)Nc3ncnn3C)CC12 c1(-c2nnn(C3(OCC(C)(C)C)CC(O)(c4n(C)nnn4)C3)n2)nc2ccccc2s1 c1(C(=O)NC(C)CNC(C2C=CCCC2)=O)cc(C(F)(F)F)cnc1O N1(C(C2=CC(C)(CC)C2)=O)CC2(CCN(C(c3occ(C)c3C)=O)C2)C1 C(C)(C)(CC(=O)NC(C1CCN(c2ccc(C(C)=O)cn2)C1)C)OC c1(CC)c(C(=O)NCC2(F)CC(NC(c3c(C)coc3SC)=O)C2)cccc1C c1(C(N2CCC(NC(c3c(C)nccc3)=O)CC2C)=O)cc2ccccc2cn1 CN1CC(O)CC1C(N1CC(CCCCNC(=O)C(c2cccnc2)O)C1)=O CC(C)CCCCC(=O)NC1C2CN(C(=O)C(=CC3CCCCC3)F)CC12 C1(C(C)CNC(=O)Cc2csc(NC=O)n2)CCN(C(=O)CC(C)(C)C)CC1 N12CCOCC(C)(C1)C2=O.c1(SCC(C2CC2)OCC)ccc([N+](=O)[O-])cc1 N1(C(C2(COCC)CCC2)=O)CC2OCCN(C(=O)C(C)CSC)C2C1 NS(=O)(=O)c1ccsc1C(=O)NC1CC(NC(C2CCCO2)=O)C1 c1(C(=O)OC)ccc(C(=O)N(CC(O)CN(C(=O)CN2CCC2C)C)C)c(F)c1 c1(CC(N2CCC(CC=C)(NC(=O)CC34CCCC3C4)C2)=O)cccc(F)c1Cl C1(N(C(CC(C(C)C)O)=O)C)CC2CCC(C1)N2C(=O)C(F)C(C)(F)F Cc1ccc(C(C)C)cc1OCC(=O)NCC1CCC1NC(c1cccnn1)=O N1(C(C(CC)C(=O)OC)=O)CCC2(CCC2)C(NC(c2nc(C)oc2C)=O)C1 N1(C(C2C(=C)CC2)=O)CCC2(CC1)CN(C(=O)CC1CCC(F)(F)C1)CC2CO N1(C(c2cncc(OC)c2)=O)CC2CN(Cc3cc(F)ccc3Br)CC12 C=CC(CC)CC(=O)N1CCC2C(C(=O)NCC3CCCC(OC)C3)C2C1 C(=O)(C1=CSCCO1)N(CCCCCNC(C1C2COCC12)=O)C c1(C(=O)NC(CNC(c2n(CC)ccc2)=O)C2CCC2)cccc(N)c1O Cc1ncc(C(=O)N(C)C)cc1Cl.N12CCCC1(CC(C)C)NC2=O c1(C(C(=O)N(C(C)C)CCNC(=O)CNC(=O)C(F)(F)F)C)cccc(Cl)c1 S(=O)(=O)(c1c[nH]ccc1=NCC(C)(C)C(C)(F)F)N1CCN(c2n(C)cnn2)CC1 n1(CCc2cccc(-c3ccc(C#N)cc3)n2)cc(CO)cc(C(F)(F)F)c1=O N1(C(c2cc(OCC)no2)=O)CCN(C(=O)C(C)N2CCCC2)C2(CCC2)C1 c1(CC)cc(C(=O)NCC(C(C)(C)C)NC(=O)CCNC(=O)C(C)(C)C)sc1C C(=O)(CCCCN1CCCC1)N1CC(C)(N(C)C(=O)OC(c2ccccc2)=O)C1 c1(OC)c(Cl)ccc(C(N2CCC(F)C(NC(=O)CSC(C)=O)C2)=O)c1F N1(C(c2cc(-c3ccc(OC)cc3)nn2C)=O)CC(N2CCOCC2)CC1(C)C c1(CC)ncnc(NC2CCCC(NC(c3c(C)nsc3NC)=O)C2)c1F c1(OC)cccc2c(C(N3CCC(N(C(=O)C(C)C4CC4)CCO)C3)=O)coc12 C1(C(=O)NC2CC(C)C2)CCN(C(=O)C2=COCC2)CC1(C)C c1(C(=O)NC(C)C(=O)N(C2CCCC2O)C)ccc(N)cn1 C1(C(C)C(=O)NC2(CF)CN(C(=O)CCC3CCC3)C2)CCC(=O)N1C CC1(C)C2CCC1(CC(=O)NC1CCCC(NC(c3cc(F)n[nH]3)=O)C1)CC2 N1(C(c2cc(OC)ncc2)=O)CCN(C(C2CCN2C2CCCC2)=O)CC1C C1(C(C)C)(C(N2CC(NC(=O)CC(C)CF)C(C)C2)=O)CCOCC1 C(CC(C)C(=O)N1CCC(CN(C(=O)CC(C)CF)C)CC1)=CCC N1(C(c2ncc(OCC)nc2)=O)CCN(C(=O)C=CSC)CC1CC C1(OC)(CNC(C2C(C)C2C)=O)CCN(C(c2sccc2C(C)C)=O)CC1 N1(C(c2sc(CC)c(C)c2)=O)CCC(NC(c2cncc(C(C)C)c2)=O)C(C)C1 O=C(C(F)C(F)(F)F)N1CC2(C(N3CC4(CC4)CC3CO)=O)CCC1C2 c1(NC(C2(F)CCN(C(=O)Cn3cc(Br)cn3)C2)=O)cc(Br)cnc1[N+](=O)[O-] C1(CC=C)(NC(c2coc(Cl)n2)=O)CCN(C(=O)C(N2CCNC2=O)C)C1 C1(NC(CCCC(=O)NC)=O)CCC2CN(C(C34CC(CC3OC)C4)=O)CC2C1 C1(NC(c2cc3ccccn3c2)=O)CCCCC12CCN(C(=O)CCCF)C2 N1(C(CC2C(C)=NNC2=O)=O)CC2(CCN(C(C3CS(=O)(=O)C3)=O)C2)C1 c1(C(N2CCC(NC(C(C)OCCN(C)C)=O)C2(C)C)=O)cc2ccccc2o1 Cc1cc(C2CC2)ccc1C(=O)NC1(C)CCN(C(=O)CCc2csc(=N)[nH]2)C1 c1(C(=O)NC(CC)CN(C)C(c2coc(COC)n2)=O)cc(OC)cnn1 C(=O)(C1=C(F)CN(C(=O)CC(C)F)CC1)N(C1CCCC1)CCC C1(CNC(C2(C)CC2F)=O)(NC(=O)CC2CC3(CCC3)C2)CCOCC1 C1(CNC(C(COCC)C)=O)CC(OC)CN1C(=O)C(C)Oc1cccnc1 c1(C(C(N2C(C(=O)NC)CCC2)=O)NCc2cn(CC)cn2)c(C)cccc1Br CC(C)(C(=O)NC1CCC(NC(=O)CC2CCOC2)C1)C1CC1 c1(OC)cccc(C(C)=CC(N2CCN(C(=O)CC#N)C(C)C2)=O)c1 c1(CC)nn(C)c(CC)c1CC(N1CC(N(C(=O)CCC(C)SC)C)C(F)C1)=O c1(C(=O)NC(C)(C)CNC(c2coc(Cl)c2)=O)ccc2c(c1)CC(C)(C)C2 C12C3CCC(C3)N1C2=O.O=C(CCN1CCCCN=C1)NC(C(F)(F)F)C1CC1 C1(OC)CN(C(c2nn(C)nc2Br)=O)CC1NC(c1ccc(C)cn1)=O C1(C2CN(C(C3CCC(F)(F)CO3)=O)C2)(NC(c2n(C)ncc2)=O)CC1 C1(CN(C(=O)C(F)(F)CO)C)C2CN(C(=O)CCc3cccn3C)CC12 c1(OCC)cc(Cl)ccc1C(N1CCC(CNC(C2(C)CC3CCC2O3)=O)C1)=O n1(CCC(=O)NCCC(=C)CNC(=O)CSC)sc2ccccc2c1=O c1(N2C3(CN(C(C4CCc5c[nH]nc5C4)=O)C3)CC2)nc2ncc(Cl)cc2s1 C1(C)(CC)CC(C(=O)NC(C2(O)CN(C(c3cnccc3C)=O)C2)C)CCO1 CC12CCCCC1CN2c1ncc(I)cn1.C(CCCO)N1CCCC1 c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC2)=O)ccc(F)c(Cl)c1F C(=O)(C#CC(=O)N(C1CN(C(c2ccc(C(F)(F)F)o2)=O)CC1F)C)N(C)C C1(c2n(C)ccn2)CN(C(c2ccc[nH]2)=O)CC1NC(C1CC1[N+](=O)[O-])=O CC(C)CCC(O)C(=O)N1CCCC1C(C)(C)NC(=O)C=Cc1cccc(F)c1 C(=O)(C(=O)C(C)(C)C)N1CCC(C(=O)NCCC(C)O)(OC)C1 Cc1cccc(CC(=O)NCC2(C(N3CC(CSC4CC4)C(C)C3)=O)CC2)c1Cl c1(C(=O)NCC(C)CNC(=O)CCC(C)N2CCCC2)cc(C#N)ccc1Cl N1(C(c2c(Cl)ccc(C)c2)=O)CCN(C(C2CC(C)(O)C2)=O)C2CS(=O)(=O)CC12 C1(NC(c2cccc(OC(C)(C)C)c2)CCO)CC2CCC(C1)O2 C1(C(N(CCOC)CCO)=O)CCC(CNC(C2CCCCC2C)=O)CC1 c1(C(=O)NCC(CN(C(CNC(c2c(C)occ2)=O)=O)C)(C)C)c[nH]ccc1=N C1(C(=O)NCC(C)F)CN(C(=O)CCC2CCCC2)CC1F Cc1ccnc(C(N2CCCCC(CN(C)Cc3ccccc3)C2)=O)c1Br c1(CCC(=O)N(CC(=O)NC)CC)cncnc1.C12(CC1)C(=O)OC2 Cc1[nH]cc(C(=O)NC2CN(C(c3cc(C#N)c[nH]3)=O)CC2C)c(=O)c1Br C1(C(N2CC(C)(NC(C(CCCC)O)=O)C2)=O)CC(=O)CC12CCC2 N1(C(C2CC23CCCC3)=O)CC2CCN(C(=O)Cc3ccc(C(F)F)cc3)C2C1 C1(C(=O)NC(C(C)NC(c2n(CC)cnn2)=O)(C)C)CN(C(C)=O)CCO1 CC(C)(CCNC(=O)CCn1cnnn1)C(=O)NCC1CC1Cl c1(CN(C)C(C2CCCSC2)=O)ccccc1CNC(=O)C(CO)N(C)C n1(CCCOC)nnnc1C(c1ccn(CC(F)(F)F)n1)NCC1CC1(C)C c1(C(=O)Sc2n[nH]cc2-c2nccs2)cccc(OC2CCCC2)c1 CCC(O)C(C)C(=O)N1CCCC1C=CC(=O)Nc1cccc(Cl)c1 CC(C)CC(C(=O)NC1CCCC(O)CC1)N(C)C(C1CN2CCC1C2)=O c1(C(=O)NCC(CC=C)NC(=O)CC(C)C2CC2)c([N+](=O)[O-])cnn1CC(F)F c1(C(=O)NC2CN(C(c3nc(C)oc3)=O)CC2C)c(Cl)cncc1Cl C1(C(=O)NC2CC(O)C2CC(=O)NCCC2C=CCC2)(CC)CCCC1O N1(C(C(CC)Sc2ccccc2)=O)CCC(C)(NC(c2nn(C)cc2N)=O)C1 c1(CCNC(N2CCCC2C2CCOCC2)=O)ccnc(Cl)c1 c1(OC)cc(C(C(=O)NC2(C)CC2)N(C2CCS(=O)(=O)C2)C2CC2)ccc1Cl C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(CCOC)N(C(=O)CC2(O)CC2)CC1 N1(CC)CC(NC(C2CC(C)CN2C(c2cc[nH]c(=N)n2)=O)=O)C(C)(C)C1 C12(CC)COC(C(N3CCCC3CN(C(=O)CN(C)C(C)C)C)=O)(C1)C2 C(=O)(C(CC(F)F)N(C)C(c1nc(Cl)cs1)=O)NC(c1scc(C)n1)C C1(N(C(=O)C(c2cccnc2)NC2CCC(=O)NC2)OCC)CCCCC1(C)C c1(-c2nnc(COC3CCN(CCC(=C)C)C3)o2)cccc(Cl)c1 C12(NC(c3n[nH]c4ccccc34)=O)CCCN(C(C3CC(OCF)C3)=O)CC1C2 C(=O)(C#CC1CCCC1)NCC1N(C(C2CNC(=O)C2)=O)CCN(C)C1 c1(CN2C(C)(C(=O)NCC(=O)Nc3ccccc3)CC2)cc(Cl)cc(Br)c1O C1(CNC(c2c(C(C)C)cccn2)=O)CCN(C(C2CC3(C2)CC3F)=O)C1(C)C C1(NC(c2c(C(C)=O)cccc2)=O)CC2CN(C(C3CSC(C)=N3)=O)CC2C1 Cc1ccnc(C)c1C(=O)NCC1(F)CCC(NC(=O)C(C)Cc2cnc[nH]2)C1 C1(NC(CCC#C)=O)CCCCN(C(c2ccc(N3CCC(O)C3)cc2)=O)C1 N1(Cc2cc(C(=O)O)c(O)cc2)CC2CCN(C(=O)Cc3ccc(Br)cc3)C2C1 C(=O)(CCCC(C)(C)C)NCC1(F)CCCN(C(C(C)OCC2CC2)=O)C1 C1(OC(c2ccc(C(c3n(CCC)nnn3)NC(C)C)nc2)=O)CCOC1(C)C N1(C(CCOCC)=O)CCCC(C(C)NC(c2onc(OC(C)=O)c2Br)=O)C1 c1(CNC(c2nc(C(N3CCN(CC)CC3)=O)cs2)=O)c[nH]c2ncc(Cl)cc12 Cc1nc2c(s1)CN(C(c1c(F)cccc1Cl)C(=O)NC1CCOC1)C2 C1(C(=O)Oc2ccc(C3(C(=O)NCC)CC3)cc2)CN(C(C)=O)CC1(C)C S(=O)(=O)(CC(C)c1ccccc1)NC(NOCC=C)=O c1(OCC(N2CC(CCNC(C(C)(C)n3ccnn3)=O)C2)=O)nc(O)nc(O)n1 C=C1CCN(C(c2ccc(C3CCCC3)cc2)C(=O)NCCOCC)CC1 N1(C(c2c(C)coc2)=O)CC2CCC(C1)N(C(c1csnc1Cl)=O)C2 CCCC(O)CC(=O)N1CCOC(c2cn(C(c3ccc(C)cc3Cl)C)nn2)C1 CC1CC=C(C(=O)N2CCC(NC(c3cccc(F)c3C(F)F)=O)C2C)CC1 c1(C(=O)NCC2(NC(C(C)C(F)F)=O)CCOC2)ncc(C(F)(F)F)cc1N C1(NC(C(C)=C2CCC2)=O)CC2(C1)CC2NC(c1cc(C(C)(C)C)on1)=O C(c1ccccc1Cl)=CC(N1CCCC(CNC(C(n2c(C)ccn2)C)=O)C1)=O c1(NC(COCC)=O)ccc2c(c1)CN(C(=O)CCc1ccc(C)nc1)CC2 C1(C(=O)NCCC)N(C(=O)CN2CSCC2=O)CCC1(C)C c1(C(=O)NC2C(CNC(c3cn(C4CC4)nn3)=O)C2)cc(F)cc(Br)c1O Cc1ccnn1CC(=O)N(CCC(=O)NCCCn1cncn1)C1CC1 CCC1=NOC(C(=O)NCC2CN(C(=O)CC(C)CN(C)C)C2)C1 CON1CC(C(=O)NCCN(CCOCCO)C(c2ccccc2C)=O)CC1=O c1(OC)cccc(C(N2CCOCC(NC(=O)C3=C(Cl)CC3)C2)=O)c1O N1(C(C=C(C)C(C)C)=O)CC2(CCC2)CC1CNC(c1nc(=O)n(C)[nH]1)=O c1(CC)cnccc1CN(C(C)COCC)CCOc1ccccc1C c1(CCC(=O)N(CC(C)N(C(C(CC)O)=O)C)C)ccc(O)c(OC)c1 c1(C(=O)NCCCNC(=O)C=Cc2ccc(Cl)nc2)cc2cccn2c(O)n1 C1(NC(CC2C(C)CCO2)=O)CN(C(=O)CCCCN2CCOCC2)CC1F c1(C(N(CC(C)NC(c2cnn(C)c2)=O)CC)=O)cc(C(C)(C)C)n(C)c1C N1(C(CC=CC)=O)CC2C(CNC(=O)Cc3csc(Cl)n3)C2C1 C(=O)(CCCCCSC)NCC(CN(C(CCCOCC)=O)C)C C1(C(N2CC(NC(c3cccnc3C)=O)C(O)C2)=O)(CC)CCCCC1 c1(N2CC(C(C)NC(c3cc(C)cc(C)n3)=O)OCC2)c(Br)cncc1[N+](=O)[O-] Cc1ccncc1NC(c1ccc(CNC(=O)C(O)CC2CCCC2)s1)=O c1(OC)cc(C(N2CCCC(NC(=O)C(C)C(C)C)C2)=O)cc(Cl)n1 C1(NC(C(C)C2CC2)=O)CCC2(CC1)CN(C(c1ccnnc1S)=O)CCO2 c1(N(C)Cc2ccc(F)nc2)nc(N2CCC=C(Cl)C2)nc2scnc12 Cc1cccc(C=CC(=O)NC2CCN(C(=O)Cn3cc(C(F)(F)F)cn3)C2)c1 c1(OC)ccc2c(c1)CC(NC(=O)NC1(CF)COC1)CCC2 c1(OC)ccc(NC(=O)CC2C(N)CC2O)c(OC(C)C)c1 CCC(COC)C(=O)N1CCCC1(C)C(=O)NCc1ncn(C2CC2)n1 Cc1[nH]c(C)c(C(=O)NC(C)CCNC(=O)CC2NC(=O)NC2=O)c1C O=C1CCC(C(=O)N2CC(CNC(=O)COCc3ccncc3)C3CC23)=NN1 N1(C(C(C(C)(C)C)O)=O)CC=C(CC(=O)NC2CC3(COCCO3)C2)CC1 C(=O)(N=c1nc[nH]n2cc(Br)cc12)c1c(C)nc(CN)nc1C N1(C(C=Cc2c(C)nsc2)=O)CC2CC1CN(C(c1cc(O)n(C)n1)=O)C2 C1(CNC(=O)CCCc2cccs2)CC2COCC2N1C(C1CCC(=O)N1)=O N1(C(C(N2CC(NC(C(C(CC)(C)C)O)=O)C2)=O)C)C(=O)c2ccccc2C1=O Cc1csc(C)c1C(=O)NC1C2CN(C(=O)CCCc3cnn[nH]3)CC12 C1(O)(CN(C)C(c2cccs2)=O)CN(C(c2cn(C3CC3)nn2)=O)C1 Cc1c(C(=O)N=c2nn[nH]n2C)cc(-c2ccc(CBr)cc2)cc1[N+](=O)[O-] O=C(CC1CCc2ccc(O)cc21)NCC1(CCNC(=O)C(O)C(F)(F)F)CC1 CC1(O)CC(CNC(C2CCN(C(=O)CCC3CCOC3=O)C2)=O)C1 Cc1cc(C(=O)N(C)CC2(O)CCN(C(C34CC(C)(C3)C4)=O)C2)cc(Cl)c1 C(=O)(C(O)P(C)(C)=O)N1CCCC(N(C(=O)CC2(OC)CC2)CC)C1 N1(C(C2CC2(Cl)Cl)=O)CCCC(n2cc(CC(c3cccnc3)O)nn2)C1 N1(C(C(COC)C)=O)CC(OC)CC1CNC(C1CCC(=O)N1C)=O C1(C(N(C)Cc2nnnn2C)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C(C)(C)C1 CC1CCCN(C(=O)C(=O)NC(C)CCN(C(=O)COc2ccsn2)C)C1 c1(C(C)C)ocnc1C(=O)NC1CC1CNC(=O)CC1CC2(CC2)C1 C(=O)(C(F)C(C)(F)F)NC(CC(=O)N(CC=C)CC1CC1)CC1CC1 CC1(C)CC(CN2CCC(O)(C(=O)NCCC3CC3(F)F)CC2)CCO1 CC1=C(CNC(=O)C(N2CCC3CSCC3C2)=O)C(C)S(=O)(=O)c2ccccc21 N1(C(c2cc(COC)sc2)=O)CC(C)(C)CC1CNC(c1cccc(OC)n1)=O N1(CC(=O)NCCCCC(C)NC(c2nc(=O)n(C)[nH]2)=O)CCn2nccc21 Cn1nc(C(=O)NCC(C2CCN(C(=O)COCC(C)(C)C)CC2)F)cc1O CC1(C)CC(NC(c2coc(C(N)=O)c2)=O)CN(C(=O)C(C)(C)C(F)(F)F)C1 C(=O)(C(C)CC(=O)c1cccc(F)c1)NCC(CNC(=O)CCC(N)=O)OC c1(NC(C2CCC(C)N2C(c2cnc(Cl)s2)=O)=O)cccc2c1C(=O)CC2 C12(NC(c3c(COC)scc3)=O)CCOCC1CN(C(=O)C(C)=C1CC1)C2 c1(CC)cccnc1C(=O)NCCCC1(NC(C2CCC(C#N)C2)=O)CC1 Cc1sc(S(=O)(=O)Nc2ccc(OC3CCCCC3)nc2)cc1[N+](=O)[O-] C=CCC(CO)NC(C1(NC(c2cc(C)co2)=O)CCC1)=O c1(CN2CC(NC(c3cc(Cl)cnc3Cl)=O)C(F)C2)ccc(C(F)(F)F)cc1I c1(C(=O)NCCOCCC(=O)N(C)CC2(C)CCC2)cccc(=O)o1 CC(C)CC(C(=O)N1CCCC(N(C)C(c2coc(C(F)F)c2)=O)CC1)N(C)C C=CCCC(C(=O)NC1CCCC(CO)C1)NC(C1(NC(C)=O)CC1)=O c1(CN=C(NC2CCCN(C(C(C)C)=O)C2)NC2CC2)cc(Cl)ccc1Cl c1(CC(N2CC(NC(C3(O)CCCCC3)=O)C(O)C2)=O)noc2ccccc12 C1(C)(C(=O)NCC2(OC)CN(C(C3(O)CCOC3)=O)C2)CC(C2CC2)=NO1 N1(C(Cc2c(C)nc(SCC)s2)=O)CCN(C(=O)COc2cnn(C)c2)C(C)C1 C1(C(=O)NCC(CC)NC(=O)CCc2cc(C)sc2C)CCCC2(CC2)C1 N1(C(C2C(C)(C)OCC2)=O)CCOCC(NC(=O)C(c2cc(F)cc(Cl)c2)=O)C1 C(=O)(C1CNc2ccccc21)NCC1CCC(NC(=O)Cc2csnn2)CC1 c1(OCCC(=O)NC(C)CNC(=O)Cc2ccc(C(C)(C)C)s2)ccc(Cl)cc1 C1(C(=O)NC(C)CC2CN(C(=O)CN(C)C(N)=O)C2)C=CC=CC=C1 N1(c2ncnc(NCCN(CCC)CC)c2C)Cc2ccc(C)cc2C1 O(NC(=O)C(C1(C)CC1)NC(=O)CC1OCCO1)CC(CC)O C#Cc1cccc(CN(C2CN(C(=O)OC(C)(C)C)CCC2F)C=O)c1 N1(C(c2c(OC)c[nH]n2)=O)CC2CCN(C(=O)C(C)=C(C)C)CC12 C(=O)(CC(C)(C)CNC(C1CCNC1=O)=O)N1CCN(C(C#C)C)CC1 Cc1nn(C)cc1-c1cn(CC(O)CCC2CCC(=O)NC2)nn1 C1(C(N(C(CC)C(=O)OC)C)=O)C=CCN(C(=O)CCc2nc(C)no2)C1 Cc1nc(C(=O)NC2CC(NC(=O)C=CC3(C)COC3)C2)c(C)o1 Cc1cnc2n1CCC(C(=O)NCC13CC(NC(=O)CSCCC4CC4)(CCO1)C3)C2 C=CC1(C(=O)NCCC(=O)N(C)CC)CCN(C(C2CC(N(C)C)C2)=O)C1 S(=O)(=O)(c1ccc(NC2CC(Cl)=NO2)cc1Cl)N(C)C Cc1cccc(NC(C2CC23CCN(C(c2ccccc2Br)=O)C3)=O)c1[N+](=O)[O-] Cc1cc(C(=O)N(C)CC2(NC(C3CNC(=O)CC3C)=O)CC2)c2c(c1)CCO2 c1(C(N2CC(NC(C34CCCC3C4)=O)C2)=O)ccc(Cl)c(C(F)(F)F)c1 CC1CCN(C(=O)C(O)Cc2cnc[nH]2)CC1NC(c1n[nH]cc1Cl)=O CC(C)(F)C(C)(F)C(=O)N1CC2CC(C(=O)Nc3cccc(C(F)F)c3)(C2)C1 c1(C(N(CCCNC(=O)C(C)(F)CC2CCCC2)C)=O)cc(Cl)c(F)cc1F c1(CC(CNC(=O)C(C)c2ccsc2)NC(C2(C(=O)OCC)CC2)=O)ccccc1 c1(SCC(=O)NCC(CC)(C)NC(C2CC23CCCC3)=O)ccccc1O c1(C(N(CC)CC2CCN(C(c3ncoc3C)=O)CC2)=O)cccc(=S)n1O c1(CNC(C)=O)noc(-c2ccn(CCC(=O)OC(C)(C)C)n2)n1 N1(C(C(CC)(C)OC)=O)CCC12CN(C(c1cn(C(F)F)c(C)n1)=O)C2 CC(CC(Cl)Cl)NC(C1CCC1C(F)(F)F)=O C(=O)(C(F)(F)CCn1cccn1)NC(CC(C)NC(C(C1CC1)OC)=O)C n1(CC(=O)N(CC(C)NC(c2cc(C)nc(Cl)c2)=O)C)cnc2ccccc12 C#CCCCCCC(=O)NCC(C1CCCC1)NC(=O)CC1COCC(C)(C)O1 CC(C)(O)CC(=O)NCC1(C)CCCN1C(=O)CC1CC(=O)NC1=O c1(C(C)C(=O)NC2CCCC(NC(C34CC(CO3)C4)=O)C2)c(F)cccc1F Nc1ccc(C(=O)N(CC(N2CCS(=O)(=O)CC2)=O)CC2CCCO2)nc1N Cc1ccc2c(C(=O)NC3CCCN(C(c4cnsn4)=O)C3)coc2c1 N1(C(CCN(c2ccccc2)C)=O)CCC(NC(C2(F)CCCCC2)=O)C(F)C1 CC1=CCC(C)(C(=O)NC(C2CN(C(=O)C(C)N3CCCC3)C2)C)CC1 CC1COCC(CC(N2CC(=O)CC2C(=O)NOCCOCCO)=O)O1 C(c1cnn(-c2ccccc2)c1)=CC(=O)NCCCN(C)C(C1CC1[N+](=O)[O-])=O CC1(CNC(C2(F)CCC2)=O)CCC(NC(c2ccc(C3CCCC3)cc2)=O)C1 C(C1=NOC2CN(C(=O)C3=CCCCCC3)CC12)NC(c1cc(C)c(Cl)cc1)=O n1(CC(=O)NC(C(=O)NCC(F)(F)Cl)C2CC2)cccn1 N1(C(c2ccc(Cl)o2)C(=O)NCCCC)CCCC(C2CCCC2)C1 C(N=c1ccnc(N(C)CCn2cncn2)[nH]1)c1c(C)cc(Cl)nc1 N1(C(C(CC)Cc2ccccc2)=O)CCCN(C(C2(C(=O)NC)CC2)=O)CCC1 N1(C(c2cc(Br)co2)C(=O)NC2CCOCC2)CCc2ccc(C3CC3)cc21 C#CCC(O)C(=O)N(C1CN(C(=O)CC2CCC(=O)N2)C1)C C(=O)(C(C)(O)C(C)(C)C)NC1CCN(C(c2cnc(CCCC)s2)=O)CC1 CCCCC(O)C(C)C(=O)NCc1ccc(C(=O)N(C)Cc2cnccn2)cn1 c1(C(N(CC(CNC(c2cnc(C)s2)=O)C)C)=O)c[nH]c(=N)c(C)c1 C=C(Cl)CCC(=O)NCc1ncccc1CNC(c1cccnn1)=O c1(CNC(c2ccc3cccnn23)=O)cnn2c1CN(c1ncc(Cl)cn1)CC2 c1(CN(C(C)Cn2cccc2)C(=O)CSCC(=O)O)cn(C)c2ccccc12 c1(C(N(CCOCCNC(CS(C(C)C)(=O)=O)=O)C)=O)ccc2oc(=O)oc2c1 C1(CNC(C2C(CCC)CCC2)=O)CC(F)CN1C(c1[nH]cnc1C)=O C1(CCCC)CCCN(C(C2C(C)CN2C(=O)CCC)=O)C1 CC(C)(CNC(c1ccc(Br)cc1)=O)CCNC(=O)Cc1cocn1 Cc1nn(C)c2c(N(CCC(N)=O)C)nc(N3CC(C)(C)OC(C)(C)C3)nc12 N(C(=NCCF)NCc1cc(C)nc(C)n1)CC(CC)(C)Nc1cccs1 C(=O)(C(=O)C(C)(C)C)NC(C1CCN(C(c2ncsc2C2CC2)=O)C1)C c1(CN(C(C)=O)C(c2ccncc2)C)nc(C(C)(C)C)nn1-c1ccnc(F)c1 C1(C(=O)Nc2cn(CC)nc2)CCCN(C(=O)OC(C)=O)C1 C(=O)(C1=C(C)OCCC1)NC(CC(=O)N1CC(C)(OC)C1)C(F)F c1(C(=O)NCCOCCNC(C2CC3CC3C2)=O)ccc(-c2cnn[nH]2)cc1 CC(C(=O)NCc1cc(C(N2CC(C)OCC2C)=O)co1)C(C)(C)C c1(OC)c(CNc2csc(-c3cc(OC)cc(O)c3)n2)cccc1C#N N1(C(C(CC)(C)C)=O)CC2CCC1CN2C(=O)C(=O)NC1CCCC1 N1(C(c2c(C)snc2)=O)CCCCC1C(C)NC(c1csc(-c2nc[nH]n2)n1)=O C12(NC(CCC#CC)=O)CCC(CNC(=O)CC3OCCO3)(CC1)OC2 CCCN=C(NCc1nnc(CO)s1)NCC(c1ccncc1)O C(CC(=O)NNc1ncccc1[N+](=O)[O-])(c1ccc(F)cc1)OCOC(C)(C)C c1(-c2n(-c3cccc(CC)c3)nc(CCN(C)C)n2)n[nH]c2c1COCC2 N1(C(CCn2cc(C3(C(=O)OC)CCCC3)nn2)=O)CCC(O)CC1 CC1CN(C(c2ccnc(F)c2)=O)CCN1Cc1ccc(-c2nn[nH]n2)cc1 C=CCCCCCC(=O)NCCCN(C(c1ncc(C(=O)OC)s1)=O)CC Cn1nnc(C(=O)NC(CNC(=O)CCc2nccs2)CO)c1C(F)(F)F N1(C(C(=O)Nc2n(CC)ncc2)=O)CCC(C(=O)OC)c2cc(Br)ccc21 C(N=c1[nH]cnc2[nH]ccc12)c1ccc(NC(=O)C2=CCS(=O)(=O)C2)cc1 Cc1ccc(C(N2CC(NC(C3CNC(=O)C3)=O)C3(CCC3)C2)=O)c(N)c1Cl C1(C(=O)NC(C)C(C)(C)NC(c2ccc(O)c(CO)c2)=O)CC2(CCC2O)C1.C(N)=O c1(C(=O)NCC(CC)NC(c2cccc(CO)n2)=O)cc(NS(C)=O)ccc1F C(=O)(C1CCCc2scnc21)NC1C(CC)CN(C(=O)Cn2nccn2)CC1 N1(C(C(=O)Nc2ccc(OC)cc2)c2ccco2)CCS(=O)CC(C)C1 N1(C(C23C(CN(C(C(C4CC4)OCC)=O)C2)C3)=O)CCn2nc(C)cc2C1 C(C(C(=O)Nc1cccn2ncnc12)C(C)(C)C)NC(CCC#C)=O N1(C(C(Cc2ccc(C)cc2)C)=O)CCC2CCC(NC(=O)CC3CC3)C12 C=CCC(CC(C)C)C(=O)NCC1CN(C)C2(CCCC2)C1 Cc1cc2cccc(NC(C3CCCC(C4CC4)O3)=O)c2cn1 C(=O)(CCCn1ccnn1)NC(C1CCN(C(=O)CC(C)c2ccncc2)C1)C N1(C(C(C)(C)C#N)=O)CC2CCC1C(NC(=O)CC1CC(=O)NC1=O)C2 C(=O)(C1CC(=O)Nc2ccccc21)NCCNC(C1(c2c(C)cnn2C)CC1)=O c1(C(=O)NCC(N(C(C(C)=CCC)=O)C)C2CC2)cc2ccccn2c1CC CCC(C(=O)N(CCNC(C1CCCC1O)=O)CCOC1CCCOC1)N(C)C C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCN(C(C2CC(C)OC2C)=O)C1 c1(OC)cccc(C(=O)NCCNC(=O)Cc2ccc(Br)c(F)c2)c1C Cc1nc(SCC(=O)NCCCc2ccc[n+]([O-])c2)c(C#N)c(C)c1C N1(C(C2C(C)C2)=O)CCCC2(C1)CN(C(=O)Cc1cccc3c1CCC3)C2 c1(C(=O)NCC(CC)NC(c2csc(C3CCCO3)n2)=O)cccc([N+](=O)[O-])c1 c1(N(C(Cc2c(C)nc(C)s2)=O)C)nccn(C2CC2)c1=O.C(C)(C)(C)O C1(NC(CCC(=O)OCC)=O)CN(C(=O)CCc2nc(C)no2)C(C)(C)C1 CCC(CCCC(=O)NCC=CC(C)(C)C)NC(=O)C(F)C(C)(F)F N1(C(c2c(OC)scc2)=O)CC(CNC(=O)C(C)(O)Cc2ccccc2)C(C)C1 c1(NC(c2nccc(C)n2)C)ccc(C(F)(F)F)cc1S(=O)(=O)N(C)CCO C(=O)(CCCOC)N(C1(C(=O)NC(C(=O)N(CC)CC)C)CC1)C c1(C(N2C(C(=O)NCCOCCC)CCC2)=O)cccc2c(Cl)cccc12 c1(C(=O)NC(CN(C(=O)C(c2cnccn2)C)CC)C)c[nH]c2c(F)cccc12 CC#CCCCC(=O)N1CCCC1CC1CCN(C(=O)C(C)(C(C)C)OC)CC1 CCCC(O)CC(=O)N1CCC(CN(C)C(C2(C#N)CC3CC3C2)=O)CC1 C1(CC(=O)N(CC(CC)NC(c2c(CC)con2)=O)CC)COCC1(C)C N1(C(Cn2ccc(C)n2)=O)CC2C(CNC(=O)CC(O)C3CCCC3)C2C1 C(=O)(C(O)CC(C)(C)C)N.CN1CC(NC(=O)CCCCN2CCOCC2)C(C)(C)C1 c1(C(=O)OC)cnc(C2CN(C(=O)NC(c3cn[nH]c3)C)C2)nc1 c1(C(=O)NC(CC2CN(C(c3c(C)nns3)=O)C2)C)nnn(C2CC2)c1C(F)F N1(C(c2c(C(C)(C)C)ccnc2)=O)CC(C2CN(C(=O)C=CSc3nc[nH]n3)C2)C1 c1(NCC2C(C)C2)cc(Br)ccc1S(=O)(=O)NC12CCC(CC1)OC2 C1(CNC(=O)CCn2cncn2)CCCCCN1C(=O)Cc1ccc(F)cc1Cl c1(C(=O)NC(c2ccc(Br)cc2)C#C)ccnc2ccc(Cl)cc12 C(=O)(C(CCC1CC1)NC(C1CC12CC2)=O)NCC1CC(C(N)=O)C1 c1(SC)cn(-c2ncc(C(N3CCCC3)=O)s2)nn1.N12CCC1C2=O N1(C(C2CCC(=O)N2)=O)CCC(C2CC2)(CN)C1.C1(=O)C2=NOC(C2)C1=O.CO C1(CCNC(c2c(C)nsc2)=O)CN(C(C2CC3CC2C3)=O)CCO1 N1(C(C(c2scc(C)n2)C)=O)CC(NC(=O)Cc2sc(C)cc2C)C2(CCC2)C1 c1(C(=O)NCC(CNC(C(COC)(C)OC)=O)(C)F)cccc2cn(C)nc12 N1(C(C2CS(=O)(=O)C2)=O)CCC2CC12C(=O)Nc1cccc(O)c1 C1(C(=O)NC(C(CC)C)CN(C)C)CCN(C(=O)Cn2ncnn2)C(C)(C)C1 Cc1ncc(C(=O)NCC(C2CCC2)NC(=O)Cc2cccc(O)c2)n1C(F)F c1(C(N(C(CNC(C(C)OCCC=C)=O)C)CC)=O)cn(-c2ccccc2)cn1 C(=O)(C1CCCc2nncn21)NCCCCCNC(=O)C(F)C(F)(F)F c1(C(N2C3C(NC(C4CCC(=C(F)F)CC4)=O)C(C3)C2)=O)n[nH]c2cccnc12 C(=O)(CCC(C)(C)F)N1CC(OC2CCN(C(C3C(C=C)C3)=O)CC2)C1 C(C(=O)NCc1cnco1)(C(C)(C)O)NC(CNC(CC)=O)=O C(=O)(C(CNC(=O)CNC(=O)CC1CCCC1)N(C)C)N(CCCF)C c1(C(=O)NCC(C)NC(C(CC)N(C)C)=O)cnn(-c2ccccc2)c1F N1(C(c2c(C)nco2)=O)CCC(CNC(C2(O)CC(C)(C)C2)=O)C(F)(F)C1 N1(C(CN(C)C)=O)CCCC1(C)CNC(c1ncoc1-c1ccc(F)cc1)=O C1(NC(CCN(CC)CC)=O)CC(O)CN(C(c2nc(OC)cc(OC)n2)=O)C1 C1(C(N(C2CCN(C(=O)Cn3cnc(C(N)=O)n3)CC2)C)=O)CC(C2CC2)=NO1 c1(CN(C(C2CC2)C)CC)cc(OC)c(Br)cn1 n1(C(c2ccccn2)CC)ncc2c(O)cc(-c3cccc(C)n3)nc2c1=O CCC(CC(=O)NCCOCCCN(C(=O)CCNc1ccccn1)C)C1CC1 CN1CCN(C(C2CC(=O)N2)=O)C(CNCc2ccc(Cl)nn2)C1 n1(CC)nc(CNCC(C(C)C)OCC)c(Br)n1.C(C)(C)O C1(NC(c2nc(C)oc2)=O)CC(F)CN(C(c2cnn(C3CCC3)c2C)=O)C1 N1(C(C(C)N(C(=O)CC(C)O)CC)=O)CCN(C)CC(C)C1 N1(C(C2CCCN(CC)C2)=O)CCC(C2(NC(c3ncc[nH]c3=O)=O)CC2)CC1 C1(C(=O)NCCNS(CC)(=O)=O)CCCCCC1NC(C12CCCC1C2(F)F)=O N1(C(C2CC(OCC)C2)=O)CCCN(C(c2ccc([N+](=O)[O-])cc2)=O)CC1C c1(C(=O)NC(C2CCCC2)CSC)n[nH]c2ccccc12.C1CC(=O)N1 c1(C(=O)NCC(N(C(CC=C)=O)C)C2CC2)c[nH]c2nccc(Cl)c12 N1(C(C(C=C=C)C)=O)CCN(C(c2ccnc(C)c2N)=O)CC(C)C1 CC1(CNC(=O)CC(O)CNC(c2nc[nH]n2)=O)CCCC(=O)N1 Cc1cc(C)c(C(=O)NCC2CCN2C(c2csc(Br)n2)=O)c(=O)o1 N1(C(C2=C(C)CCC2)=O)CC2OCC(NC(=O)C(CCO)N(C)C)C2C1 CC1(C(N2CCCCC2CNC(=O)CCN2CCNC(=O)C2)=O)CC=CCC1 C1(C(=O)NCC=C(CC)C)CCCCCC1N C1(CC)COCCN(C(=O)CCC2CCN(C(C3CC4CCC(C3)O4)=O)C2)C1 c1(C(N2C(C)CC(CNC(c3cncc(N)n3)=O)C2)=O)coc2ccc(Cl)cc12 C1(CNC(C(C)OCC(C)C)=O)CN(C)CCN1C(c1cn2c(n1)CCC2)=O C(=O)(CCC(C)(C)C#N)N1CC(C(C)NC(c2c(CC)scc2)=O)OCC1 c1(C(=O)NC2(C)CCN(C(C3(OC)CCC3)=O)C2)cnc(O)n(C)c1=O C1(CN(c2ccccn2)C(C(C)C2CCCC2)=O)CCN(C(=O)C(C)(C)C)CC1 O=C(CCCCCF)NC1CCCC(C(N2CCC3(CSC3)C2)=O)CC1 N1(C(C=NOC)=O)CC2CCN(C(c3cccc(F)c3Cl)=O)C2C1 C#CCCCC(C)C(=O)N1CC=CCC1C(N1CCC(CO)(OC)C1)=O C(=O)(C(O)Cc1ccccn1)N(CC(C)NC(CCN(CC)CC)=O)CC C1(NC(c2c(OCC)c(F)ccc2)=O)CN(C(c2cnoc2C)=O)CC12CCC2 C(CCC(C)(C)C(=O)NCC1(C)CC2(CC2)C1)NC(CC1C(C)CCO1)=O C=CC(C(=O)NCC1(O)CC(NC(c2cnn(CC)n2)=O)C1)OC CC(C)CCCCCC(=O)N1CCC(C)C(NC(=O)CCSc2ccccn2)C1 C1(NC(c2cccc(CC=C)c2)=O)CCCC(C(=O)NCC)CC1 C1(C#N)(CNC(C2C(NC(C(C3CCC3)OCC)=O)CCCC2)=O)CC(C)(C)C1 c1(C(N(C)CC2CCCN(C(CSCCC)=O)C2)=O)ccc(S(N)(=O)=O)cc1Cl c1(C(N2C(CNC(c3cc(COC)cn3C)=O)CCC2)=O)cn2cccnc2n1 c1(OC)ccc2cc(C(N3CC(F)(CNC(C4CC5CC5C4)=O)C3)=O)[nH]c2n1 N1(C(C2C(C(=O)OC)C=C2)=O)CCC(C)(NC(c2sc(COC)nc2C)=O)CC1 Cn1ccc(C(C)(C)C(=O)NCC(C)(C)CNC(c2ccc(Cl)o2)=O)n1 C=C(C)C(CC(=O)NC(C)CC(=O)NCC1CCCCC1(C)C)OCC c1(C(=O)NCc2n(CC(C)C)ncn2)ccnc2c1CNCC2 C1(CNC(c2cc(CNCC3N(C(=O)OC)CCC3)on2)=O)CCC2(CC1)CC2 Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccc(F)s3)=O)C2)nc1C C1(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)CCN(C(=O)CCCCCF)CC1O c1(C(=O)NCC(CNC(c2cccc(OC(C)C)n2)=O)C)nc2c(s1)CCCC2 C(=O)(CCP(C)(C)=O)N1CC(C)C(CCNC(c2sccc2CO)=O)C1 N1(C(CSCC)=O)CC(CNC(c2cn(CC(C)(C)C)nn2)=O)CC1C N1(C(C2C(CC)N(C(C3CCCC4CC34)=O)CC2)=O)CC(N(C)C)C2(CC2)C1 CC1=C(C(=O)N2CCCCC2CCNC(=O)Cc2cn[nH]c2)CCC1 c1(C(=O)OCC)c(CNC(=O)NC(C)Cn2ccnn2)nn2c1CCC2 c1(C(=O)NCCCOC2CCN(C(CC(C)F)=O)CC2)cnc2sccn12 C(C(CC(C)C)NC(C1(C)CCN(C)C1)=O)NC(CCCOC(C)=O)=O C1(=O)CC(C)N(C)N1CCCC(C)CC(=O)N(C)C.CO CCCC(C#N)C(=O)NC12CC(C(=O)N(C3CS(=O)(=O)C3(C)C)C)(C1)C2 C1(CC=C)(C(=O)OCC)CCN(C(c2c[nH]c(C)c2)=O)CC1 c1(C(N2CC3C(NC(CC(CCC)(C)O)=O)C3C2)=O)cc([N+](=O)[O-])ccc1NC CC(C)S(=O)(=O)C(C)C(=O)NC1COC2C(NC(=O)C(O)C(F)(F)F)COC12 C1(CNC(=O)COCCF)CCN(C(=O)CC2(O)CCC2)CC1O N1(C(C2CN(C(C)=O)C2)=O)CCCC(F)(C(=O)NC(C)(C)CCCF)C1 C#Cc1ccnc(C(=O)NCC2(NC(=O)C=CC3CCCC3)CCCCC2C)c1 C#CCCCC(C)C(=O)N1CCC1C(=O)NCC(CO)OC c1(C(=O)NC2(C)CCN(C(C(CCCC)C)=O)CC2)cc(F)cc(C)c1N N1(C(C2(CC)CCN(C(=O)CCc3ccncc3)C2)=O)CC2CSCC2(C)C1 N1(C(=O)OC(C)(C)C)CCC(C)(C)C1CNC(C1CNC(=O)CC1C(F)(F)F)=O N1(CCCC)CCOCC1C(=O)NCCCC(C)NC(c1cnoc1C(C)C)=O c1(CCNC(C)=O)cn(CC(N2CCCC2CN)=O)nn1.C1(CC(=O)N)CC=CCC1 C1(CCNC(C2CCCO2)=O)CCCN(C(c2ccc(C(F)(F)F)o2)=O)CC1 c1(C(N2CCC(C)(N)C2)=O)ccc(F)c(F)c1.Cc1ccccc1CC1(C)CC1 Cc1nccc(CNC(C2(CNC(=O)CCCF)CC(C)(C)C2)=O)n1 N1(c2nnc(-c3c(O)ccc(C)n3)n2CCN(C)C)CC2CCCC(C1)N2C C1(C(=O)NC2CCCN(C(c3cc(C)c(Cl)s3)=O)C2)CCC(C)(F)CC1 C(=O)(C(C)CC(C)C(C)=O)NCc1c(C(=O)NCC(CCCC)O)n(C)nn1 C1(NC(C(C)=CC)=O)CCCC(CNC(=O)COc2ccsc2)C1 c1(CC)oc(C(N2CCCC2CN(C(=O)C(O)C2CCC2)C)=O)cc1C N#Cc1c(F)c(NC(C2CCCN2CC2CCCCC2)=O)nc(F)c1F CC(O)CCCC(=O)N1CC(N(C(=O)Cc2cccc(O)c2F)C)C1 C1(COC)(CNC(C2CC3(CC3)CO2)=O)CCCN1C(=O)C=Cc1cc(C)no1 C#CCCCC(C)C(=O)NC1(C(=O)NC(CO)CCC2CC2)CCCC1 N1(C(c2n(C(C)C)ccc2)=O)CCCN(C(c2cccn3ccnc23)=O)C(C)C1 N1(C(C(CC(C)C)OC)=O)CCC2CCCC(C1)N2C(c1cncnc1C)=O N1(C(C2CCCC(C)C2)=O)CCC2(CC1)CN(C(c1n[nH]cc1Br)=O)C2 c1(OC)cc(C)nc(NNC(=O)NCc2ccc3cc(F)ccc3n2)n1 c1(Nc2cncc(C)c2C)nncc2ccccc12 N#Cc1ccnnc1N1CCC(Cc2ccc(Cl)nc2)C1 C12(C(=O)NCc3cn(C)nc3)CCCC1N(C(C1CCC(F)CC1)=O)CC2 C=C(C)C(C)(C)C(=O)NCC1CC(COC)CN1C(=O)CC1CS(=O)(=O)C1 Cc1cc(Br)ccc1CN1CCN(CC(=O)Nc2ccnc(Cl)c2C)CC1 N1(C(CCS(C)=O)=O)CCC(NC(=O)Cn2ncc3ncccc23)C12CCC2 C(=O)(CCCCN(C)C)NCC(CO)NC(C(c1ccccc1Cl)OC)=O C(CC(C)(C)C)(C(=O)NCCCCCC(=O)NC1(CCF)CCC1)OC C(=O)(CC(C)(C)CN(C)C)N1CC(COC)(CNC(=O)C(C)CCOC)C1 C(=O)(C(F)CC(C)(C)NC(C1CCC(=O)CC1)=O)Nc1c(OC)ccc(C)c1 CCCCCC(O)C(=O)NC(CNC(=O)C(c1cnn(C)c1)C)(CC)CC N1(C(CCC(C)C#N)=O)CCC2C(C1)CN2C(=O)CCc1ccc(Cl)c(Cl)c1 Cc1cc2occ(C(=O)N(C3CN(C(C4CCNC(=O)C4)=O)C3)C)c2cc1C N1(C(CC2(C)CC2)=O)CC2CN(C(=O)CC3(O)CCOCC3)CCC2(CO)C1 N1(C(C(C)(O)c2ccccc2)=O)CCCC(NC(c2cccs2)=O)C1.CS C1(C(=O)NC(C(=O)NCCc2cn[nH]c2)C2(C)CC2)CCCC1 C1(CNC(c2ccc(C)o2)=O)(NC(c2ccc(OCF)cc2)=O)CCCCCC1 c1(CC2(NC(c3cc4c(cc3)C(=O)NC4)=O)COC2)ncnc2ncc(Br)cc12 Cc1c(C(N2CCC(NC(=O)CC3CCC3)C(CO)CC2)=O)nn2ccccc12 C1(C(=O)NC2(CCC)CCN(C(C3CCCO3)=O)CC2)CC2(CCOCC2)CO1 C(C(C)(CC(C)C)NC(=O)Cc1cccc(Cl)c1)NC(C(CC)=CC)=O C1(C)(C(=O)NC(C)CCCNC(c2c[nH]ccc2=N)=O)Cc2ccccc2C1 N1(C(CC=CCCCCC)=O)CC2CCC(CNC(c3cscc3C)=O)C2C1 C1(C(=O)NC2CCC(N(C(CC3CCN(C)C3)=O)C)CC2)CN(CP(C)(C)=O)C1 CC(C)CC(C(=O)NCC1CN(C)CCO1)NC(=O)C1=CCCC1 c1(C(=O)NC(C(C)(C)C)c2cccs2)ccc(-n2cccn2)c(F)c1 CC1CC1C1CC1NC(=O)CC(C)(C)NC(=O)C(F)n1ccnc1 c1(C(=O)NCC2CC(NC(C(C)OCOC)=O)C2)coc2cc(F)cc(F)c12 CN1CC(C)(C(=O)NCC(C)(C)NC(C2C(C(F)F)C2(C)C)=O)CCC1=O C(=O)(CC(C(C)C)NC(=O)Cc1ccoc1)NC(CCC)CCC C1(C(N(CCCC)CCN(C)C)=O)COCC1NC(=O)CN(C)C(C)=O C1(C2CCN(C(C3CNc4ccnn4C3)=O)C2)(NC(c2c(C)cn(C)n2)=O)CC1 c1(C(=O)NCC(C)N(C(=O)C(F)C(C)(C)O)CC)[nH]c2c(C)cccc2c1C c1(CC)[nH]ccc1C(N1CC(CNC(=O)C(C)c2ccco2)(OC)C1)=O C1(NC(Cc2ccc(CC)c(F)c2)=O)CCN(C(=O)C(C)(C)CO)CCC1(F)F c1(C(=O)NC2C(NC(C(COC)C)=O)CCOC2)cc(C)cc([N+](=O)[O-])c1N c1(CNC(CCN(CC#C)C(C2CCCS2)=O)=O)nn(C)cc1CO c1(C(=O)NCC2C(CNC(CCC=CC)=O)C2)cn(C)nc1COC n1(CC)cc(C(=O)OC2CCC(N(C)C)C2)c(C)n1 CC#CCC(C(=O)Nc1cnc(COC)nc1)NC(=O)Cc1cn(C)nc1C Cc1cc(C)c(C(N2C3CC2CN(C(=O)CC2CCC(F)(F)CO2)C3)=O)cc1C N1(C(Cn2ncc(CC)c2)=O)CCCN(C(c2coc3c2COC3)=O)CC1C C1(NC(Cc2c(C)n[nH]c2)=O)CC2CCC1N2C(c1ccc(N)cc1F)=O c1(-c2cn(C(COCC)C(=O)NC3(C)COCCC3CC)nn2)cc(O)nc(O)n1 C1(NC(C2C(C(C)C)CCC2)=O)CN(C(=O)C=CCOC(C)(C)C)CC(C)(C)C1 N1(C(CC2(CC)CCOCC2)=O)CC(NC(=O)C2=CCCS2)CC(C)C1 CC(C)C(C(=O)NCCOCCNC(=O)C(C)n1ccnc1)c1cccc(Cl)c1 C1(CNC(C(=Cc2cccnc2)C)=O)CCCCCN1C(C1(F)CCOC1)=O N1(C(CCC(C)O)=O)CCCC12CCN(C(c1cc3ncccc3s1)=O)C2 CCC(C)CCCC(=O)NCC1(C(=O)NCC(O)C(C)C)CCC1 C12(NC(CCC)=O)CCN(C(c3cnn(C(C)(C)C)c3N)=O)CC1C2 N1(C(C=C=C(C)C)=O)C2CCC(C2)C1CNC(C1CC(C)(O)C1)=O C1(C(N(C)CC2N(C(c3n(C(C)C)nnc3)=O)CCCC2)=O)CCC(C)(C)OC1 c1(C(=O)NCC2C(NC(=O)Cn3cccn3)CCC2)c[nH]nc1[N+](=O)[O-] c1(C(N2CCN(C(C(C)c3cccs3)=O)CC2)=O)ccc2cc(C#N)ccc2c1 CC1(C2CN(C(C3CCC4CCC3N4C(=O)CCCC3CC3)=O)CCO2)N=N1 c1(C(=O)NCCC2(O)CCN(C(c3ccc(OC)nc3)=O)C2)c[nH]cc(C)c1=O c1(C(N2CC(C)(NC(c3ccc(=NC)[nH]c3)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 Cc1cccn2nc(C(N3CCCC(C)(NC(c4ncncc4Cl)=O)C3)=O)cc12 c1(CNN2CC(C)(C(N3CCOCC3CO)=O)C2)cn2ccccc2n1 c1(CC)cc(F)ccc1C(N1CCC(O)C(NC(c2cscc2OC)=O)C1)=O CC1Cn2nc(C(N3CCCC(N(C)C(C4CC=CC4)=O)CC3)=O)cc2C(=O)N1 CN1CCN(C(=O)CC#N)CC1C(=O)NOCCCC1CC1 c1(C(N2CC(O)(C(C)NC(C3CCNC3=O)=O)C2)=O)ccc2c(n1)CCC2=O c1(CCC)nnc(N2CCC(CC3(CO)CCOCC3)C2)n1CC c1(C(N2C(C)CCC2C(=O)NCC(F)(F)C(F)F)=O)cncn(C)c1=O C(=O)(C1CCCc2scnc21)NCCCNC(C1N(C)S(=O)(=O)CC1)=O CCC(CC(=O)NCCCOCCC(=O)NCC(=O)NCC(F)F)SC c1(CC)c(C(=O)NCC2CC(C)CCN2C(c2cc[nH]c2)=O)sc2ccccc12 N1(C(CC2C(C)C(=O)CC2)=O)CC=C(CNC(C2CCC3CC3C2)=O)CC1 N1(C(c2n(C)cc(Cl)c2)=O)CCC(NC(c2ccn(C(F)F)n2)=O)C(C(N)=O)C1 C(=O)(C1=CCCCO1)C(CC1C2CNCC21)=O.O=C1CC2C(N)C2C1 c1(-n2c(CNC(c3cncs3)C)nnn2)ccccc1OC(F)(F)F CC(c1ccccc1)=CC(=O)NC1CCC1CNC(=O)C(C)(C)C O(N1CCC(NC(=O)CC2CN(C(C3CC3(Cl)Cl)=O)CCO2)CC1)CC N1(C(c2nc(CC)oc2)=O)CC(CC(=O)NCC2CCCC23CCC3)C2(CC2)C1 C1(NC(C(C=C)(C)CC)=O)CN(c2ccnc(C(=O)OC)n2)C2CCCCC12 N1(C(C(=O)N(C(C)C)Cc2nc(C)on2)=O)CCS(=O)CC1C C1(C(N(CC(C)O)CCNC(C2(F)CCOCC2)=O)=O)CCCCCCC1 n1(C(C)C)ncc(C(=O)NCC2(NC(=O)C(c3ccc(Cl)s3)C)CCOC2)c1N N(C(=NCCC(C(F)(F)F)N1CCOCC1)NCC1CCC1)CCC(CC)C c1(C(N2CCC(C)(NC(CN3C(=O)CC(C)(C)O3)=O)C2)=O)cn2ncccc2n1 C1(NC(C2CCCC(F)C2)=O)(CNC(C2Cc3nccn3C2)=O)CCCCCC1 N1(C(c2cc(COC)on2)=O)CC2(CC2)CC1CNC(c1c(F)cccc1F)=O C1(CCNC(C(=O)NCC)=O)CCCN(C(=O)CCCOc2cccc(Cl)c2)C1 C(=O)(C1CCCc2ccnn21)N1CC2C(CNC(c3c(C)[nH]c(C#N)c3)=O)C2C1 C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C1CCC1)NC(c1cc(C)n(C2CC2)n1)=O N1(C(C=CC(C)(C)SC)=O)CC(C)C(NC(C2OCCCC2(C)C)=O)C(C)C1 C12CCCC1C2.C1(CC(=O)N(CCCNC(C2(O)CCC2)=O)C2CC2)CC12CC2 c1(OC)ccc(F)cc1S(=O)(=O)N1CC(CC(=O)Nc2c(Br)c(C)nn2C)C1 c1(C(=O)NC2(CC)CCCN(C(C(CC=C)C)=O)C2)cc(F)c(CC)cc1F Cc1csc(C)c1C(N1CCOC(CCC(=O)NCc2nc(N(C)C)no2)C1)=O CN1CC(C(=O)NC(Cc2ccccc2)CCNC(=O)C(C)(C)F)CCC1=O N1(C(C2(CC)CCCC2)=O)CC(OC)CC(NC(=O)C(C(C)(C)C)SC)C1 C1(OC)CC2CC(NC(C3(CO)CCN(C(=O)CCCN(C)C)C3)=O)CC12 C1(O)(CCNC(c2cnnc(O)c2)=O)CCCN(C2CCc3c(F)cccc32)C1 c1(C(=O)NC2CN(C(C(C)(C)CC#N)=O)CC2(C)C)nc2ccccn2c1F C(C1CC(C)(C)Oc2ccccc21)NC(=NCC)NCC(CC)C(C)C CN1CC(O)CC1C(N1CCC(C)(CC(=O)NCCCOCCCO)C1)=O C1(OCCCCOCC)CCN(C(=O)CN(C(=O)CCOCC)C(C)C)CC1 CC(C)C(C(=O)N1CC(CNC(c2ccoc2)=O)C(O)C1)c1ccccc1 c1(C(=O)NC2CC(CNC(=O)C3=CCOC3)C2)cn2c(n1)COCC2 CCC(CC)CC(=O)NCC1CC(NC(c2nocc2Cl)=O)C12CCC2 N1(C(C(C)=CC=C)=O)CC=CC(C(=O)NC(C2CCC2)C2CC2)C1 c1(C(=O)NC(CN(C(C2CN(S(CC)(=O)=O)C2)=O)C)CC)cccnc1 N1(C(C(C2CC2)NC(C(CC=C)NC(C)=O)=O)=O)CC(CO)C2(CC2)C1 CC(C)C(CO)CCNC(=O)C(C1CCCC1)NC(C1OCC2CCCC12)=O Cc1cccc(C)c1C(=O)NCC1CCCCN1C(c1cc(O)nn1C)=O C(C(=O)N1CCC(C)(NC(c2cnn(CCO)c2)=O)CC1)(C(C)(C)C)N(C)C C1(NC(c2cc[nH]n2)=O)(CO)CCCN(C(c2ccc(-c3ccco3)s2)=O)C1 C#CCCCCCCC(=O)N1CCN(C(=O)C#CC2CCCOC2)C(C(C)C)C1 Cc1c(C(N2CC=CC2C(=O)NC(C2CCC2)C2CC2)=O)ccn1C c1(C(=O)NCCCN(C(=O)CC2CC=CCC2)C)ccsc1Br c1(C(=O)NCC2CN(C(C3CC3(F)F)=O)CCCO2)cc2n(n1)CCCO2 c1(C(N2CC(CC(C(=O)NCCC3(C)CCCO3)F)C2)=O)ccc2c(c1)CCC2 N1(C(C(CC)CC)=O)CC2OCCN(C(C3COC(C)C3)=O)C2C1 c1(C(=O)NC(C2(O)CN(C(C(C)O)=O)C2)C)cccc(C(F)F)c1 C1(CC)CCN(C(=O)CC#N)C1CNC(=O)Cc1cc(C)[nH]n1 N#Cc1cccc(NC(C2CCN(C(c3c(I)ccnc3Cl)=O)C2)=O)c1Cl c1(C(=O)OC(C)(C)C)sccc1NC1CCC1C(=O)NS(C)(=O)=O c1(NC(C2CCN(Cc3cccc(C)c3)C2)=O)cccc2nccn12 O=C(C1c2ccccc2CN1C(c1nc[nH]n1)=O)Nc1ccc(-c2nncs2)cc1 CC(c1ccco1)=CC(=O)NC(C(=O)NOC1CC1)C1(C)CC1 C(=O)(C(C)CC(C)C(C)=O)N1CCC(CCNC(CCC(=O)NC)=O)CC1C C1(C(C(=O)NCC)N(C)CC2CCSCC2)C(C)(C)C1(C)C CCCC(C)C(=O)NCCCN(C(=O)CC1CCCCC1C)C(C)C C=CC(C)C(=O)N(C)CCN(C(=O)CC1CC(F)C1)C c1(C(N2C(CN(C(=O)C(C)(C)C(C)(C)C)C)COCC2)=O)ncn2ccccc12 S(=O)(=O)(c1ccc(F)cc1CCl)NCc1c(C(=O)OC)nccn1 N1(C(C2N(C(C=C(COC)C)=O)CC3(CC3)C2)=O)CCC(CO)C(C)(C)C1 n1(CCC)cc(C(=O)N(C)CCN(C)C(c2coc(C)c2)=O)c(C)n1 c1(CC)cc(C(=O)NCC(=O)NCC(=O)NCc2ccncc2)no1 N1(C(c2ccc(SC)o2)=O)CC2(CCCCN2C(c2nccn2C)=O)C1 C1(O)(CN(C(C(C=CCCC)O)=O)C)CCN(C(=O)CCc2cn[nH]c2)C1 c1(CC)ccnc(C(=O)NCC2CCCC(CNC(c3nn(C)cc3N)=O)C2)c1 CCCCC(O)CC(=O)NC(C)C(C)(C)C(=O)NCC1(C)CCOC1 C1(C(=O)NC2C=CC(CNC(c3c(C)csc3)=O)C2)CCCC(=O)N1 c1(C(N2CCC(C3(NC(=O)C(F)(F)CO)CC3)CC2)=O)ncn2cc(Cl)ccc12 c1(NC(C2CC(=C)CN2C(c2c(O)ccc(F)c2F)=O)=O)c(Cl)nc(C)nc1Cl C=CCCCC(C(=O)NCCC(C)(O)CC)NC(c1cc(C)c(C)s1)=O C12(C(N(CCNC(C(C(C)C)O)=O)C)=O)CCC(=O)N1CCS2 C1(NC(C2(CC)CCOCC2)=O)CCN(c2nc(C3CC3)ns2)C(C)C1 N1(C(C2(C)CC2(F)F)=O)CC(CNC(=O)C=CCN2CCC2)C2(CC2)C1 C1(CNC(CCOCCCOC)=O)CN(C(c2cc(C)nn2C)=O)CCO1 c1(C(=O)OCC2CC=CC2)sc(Br)cc1F C1(CCC)CN(C(C2CCC3(CC2)CC3)=O)CCN1C(=O)C(F)=C(C)C C12(NC(c3cnn(CC)n3)=O)CCCC1N(C(=O)C=Cc1ccccn1)CC2 C1(O)(C(C)NC(C2CCSC2)=O)CN(C(=O)Cc2ccnn2-c2ccccc2)C1 C=C(C)CCCC(=O)N(C)Cc1cn(CC2(F)CCOC2)nn1 CC(CC(=O)NC1(C)CC(N(C)C)C1)c1ccccc1.C12CCC(O1)C(=O)NC2 c1(SC)c(C(=O)NCC(c2ccccc2)NC(=O)Cc2csc(Cl)c2)cnn1C C1(CNC(C2CC(C(=O)OC)C2)=O)CN(C)CCN1C(=O)CC1CCC(=O)NC1 C(=O)(CC(C)CC(=O)NC1CCCC1NC(=O)CC(F)(F)Cl)OC c1(C(=O)NCCCC(C)NC(=O)C=Cc2nc[nH]n2)cnc(C(C)C)nc1 Cc1c(Cl)ccnc1C(=O)NCC(C(C)(C)C)NC(C1CC1(C)C)=O N1(C2CC(c3ccc(OC(F)F)cc3)C2)CCNC(=O)C1CC(F)(F)F c1(C(=O)NCC(C(C)(C)C)NC(C2CCC3CC2CO3)=O)ncn2c1CCC2 N1(C(C(CNC(C2OCCC(C)C2)=O)CC2CC2)=O)CC2(CCC(=O)N2)C1 c1(C(N2CCC(NC(=O)CCCCC3CC3)C2)=O)ccc2c(=O)ccoc2c1 N1(C(C=CCCC(C)C)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C(C2CCC2)C1 Cc1cc(C(=O)NC2CCCN(C(C3CCC3(C)C)=O)C2)cc(=O)n1C c1(NCCC2CCN(C)CC2)ccc(S(=O)(=O)NCCCCC(F)F)cc1C#N N1(C(COC(C)=O)=O)CCCC(C(C)NC(c2sc(F)cc2Br)=O)C1 c1(N2CCC(F)(C(=O)OC)C2)ncnc2c1cnn2C(C)(C)C Cc1cc2ncn(CC(=O)NCC3CCN3C(=O)CC3OCCO3)c2cc1C C#CCCCC(=O)N1CC(CNC(c2ccc(-c3cnco3)cc2)=O)C(O)C1 C(=O)(C(CO)NC(=O)CC(C)C)N(CC(C)N(C(COCCOC)=O)C)C C(=O)(NNC(=O)C1OCCC1F)NCc1nc(CCC(C)C)sc1 C1(C(C)C)CCC(C)CC1NC(=O)Cn1cnc(-c2ccccn2)n1 C1(CC(=O)NCCc2onc(CC)n2)CC(F)CN1C(=O)CC(C)n1cccc1 C1(CC=C)(NC(c2cnc(C)[nH]2)=O)CCN(C(C2CCCC2C(F)F)=O)C1 N1(C(Cc2nc(C(C)C)sc2)=O)CC(C)C(C)(CN(C)C)C1 N1(CC(=O)N(CC(CNC(c2cnc(C)[nH]2)=O)C)C)C(=O)NC(C)(C2CC2)C1=O C(=O)(CCCCC(=O)NCC1(O)CCCN(C(=O)C(C)NC(C)=O)C1)OC C1(CCC)C(=O)NCCN1C(=O)C=CCC(C)(C)NC(c1coc(CO)c1)=O c1(NC(C2CC=CCC2)C)ccc(S(=O)(=O)NCCn2cnnn2)cc1Br C1(CCCNC(COCC=C)=O)CCN(C(C2CCC3CCC23)=O)CC1 C#CCCC(C(=O)NCCn1cc(C)cn1)NC(C1CC2(CC2)CO1)=O c1(C(N2C(C(C)NC(C(N3CC(C)C3)C)=O)CCC2)=O)ccc(SC(F)F)cc1 C(CCNC(=O)CC(C)F)(C(=O)NC1COCC1CN(C)C)OC Cc1cc(C(c2nnnn2C2COC2)NCCc2ccnn2C)ccc1Cl N1(C(C(C=C)(F)F)=O)CC(O)(C2(CNC(=O)COCC3CCOC3)CC2)C1 C1(C(=O)NC2(CO)CN(C(C(C)(O)C3CCC3)=O)C2)CCCC2(CCCCC2)C1 Cc1scnc1C(=O)N(C)CCOCCN(C)Cc1cnn(-c2ccccc2)c1 N1(C(CCCSC)=O)CC(CNC(=O)CN2CC3C=CC2C3)C(C)C1 CC(C)C(C#N)C(=O)N1CCOCC(NC(=O)CCCOc2cccnc2)C1 c1(OC)ncc(C(=O)NC2CC3(C2)CC3NC(=O)C2CC2)cc1C(F)(F)F c1(C(=O)NCC(CCCC)NC(=O)COC2CCC2)cc2c(cnn2C)nc1C N1(C(C=CC(=O)OCC)=O)CCN(C(C2CN(CC(F)(F)F)C2)=O)CC(C)(F)C1 C1(CNC(c2c(C)cc(F)s2)=O)CC(C)(C)CN1C(C1CCC(F)(F)CC1)=O c1(OCC)nc(C(=O)NC(C2CCN(C(=O)C(C)=C3CCC3)C2)C)ns1 C1(C(F)(F)F)(C(N(C2CN(C(CP(C)(C)=O)=O)C2)CCO)=O)CC2CCC1C2 C1(CNC(C2C(CNC(c3c(C)ocn3)=O)CCC2)=O)CCC(CO)CC1 N1(C(C#CC(C)C)=O)CC(CO)C2(C1)CN(C(=O)CCCc1cccnc1)C2 CC(C)C(O)C(C)C(=O)NCCN(C(C1(F)CCCN(C)C1)=O)C1CC1 c1(NCC2CCC(=O)NC2)nccc(=NCC2CCN(Cc3ccsc3)CC2)[nH]1 c1(C(C(=O)NC2CCOCC2)N(CCCF)CC)cnc(-c2ccccc2)s1 c1(CCCCO)nnc(C(c2onc(CCC)n2)(C)C)o1.OC(F)F C123CCC1CN(C2)C(=O)C(O)CNC(=O)C3.c1(C(=O)OCC)ccoc1C(C)C c1(CSC)cc(C(N2CC(NC(C3(C#N)CC4CC4C3)=O)C(C)C2)=O)ccc1F c1(C(=O)NCC(C2CCC2)NC(c2cc(F)cc(F)c2)=O)ccccc1[N+](=O)[O-] N1(C(C2CCN2C(C2CCOC2C2CC2)=O)=O)CCc2sccc2C1 N1(C(CC2CC(=C)C2)=O)CC2(C1)CN(C(c1cc(C)ncc1C)=O)CC2CO N1(C(C)=O)CCCC(C2CN(C(c3cc(C)c(Br)cc3Cl)=O)C2)C1 C1(C(=O)NCC(=O)N(C)CC)(OC)CCN(C(C2CN(C)CCO2)=O)C1 S(=O)(=O)(c1cccc(S(C)(=O)=O)c1)NC1CN(Cc2cc(C)[nH]c2C)CC1C#N N1(C(COC(C)C)=O)CCCC1c1nc(C(=O)NC(C)Cc2cnccn2)cs1 N1(C(C2CCCCN2CC(F)F)=O)CCC(F)(F)CC1c1ccco1 c1(C(=O)NCC2CCC(NC(c3onc(C)c3C)=O)C2)cc(N)ccc1O C(=O)(C(CC)C(=O)NCCNC(=O)C(c1ccc(C(F)F)cc1)C)OCC C(C(C(=O)NCCNS(=O)(=O)CC)NC(Cc1cc(OC)n[nH]1)=O)SCC C(=O)(CN=C(NCC(C)(C)C(F)(F)F)NC1CC1C(=O)N(C)C)N(C)C C1(CCNC(c2nnn(CC)c2C)=O)CCN(C(c2ccccc2F)=O)C(C)C1 N1(C(C2SCC(=O)C2)=O)CCC(C(=O)NCc2ccc[n+]([O-])c2)C(O)C1 Cc1ccn2cc(CCNC(=O)C(C(C)C)NS(N)(=O)=O)nc2n1 C(=O)(CCCn1cc(CCc2ccccn2)nn1)NCCSCCC(C)C C1(C(=O)N(CC(C)NC(=O)C(c2ccc(Cl)s2)=O)C)(OC)CCSCC1 N1(CC(CC)NC2CCCCC2)CC(=O)N(Cc2ccc(C(N)=O)cc2F)C1=O Cc1c(F)ccc(C(=O)NC2CC2NC(=O)CSc2cn[nH]c2)c1N C1(C(=O)NCCc2c(C)nc[nH]2)CCN(C(C2(CO)CCC2)=O)CC1C C12(C(=O)NCC3(F)CN(c4c(CC)c(Cl)nc(C)n4)C3)CCCCCC1OCC2 c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)C(C)C)cc2c(F)cc(Cl)cc2[nH]1 c1(CN2CCC(CNC(=O)CCC(F)(F)F)CC2)ccc2ccsc2c1 C(=O)(N=c1ccn(-c2ccc(F)cc2C#N)[nH]1)NCC(C1CCCO1)OC N1(C(Cc2cc(C)sc2)=O)CC2CC(NC(=O)Cc3ccnc(F)c3F)C(C2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(CC)N(C(c2ccn(C3CCC3)n2)=O)CC1 C1(NC(CCC(C)C)c2nnnn2Cc2cccs2)COC2(CCC2)C1 CS(=O)CCC(O)C(=O)NCC1(F)CC(CNC(=O)C=CBr)C1 C1(NC(C2CC23CCC3)=O)CCC2(CC1)CN(C(=O)CN1CC3CC3C1)CCO2 C(=O)(C(C)C(F)F)N(CCC(=O)N(CCC)C(C)CO)C c1(N(C(C2CCC(CC)C2)=O)C)ccc(OCC(O)CN(C)C)c(OC)c1 N1(C(C2(C#N)CC=CC2)=O)CC(C(=O)NC2CCCOC2C)C2(CCC2)C1 N(C1CCc2ccccc21)C(C1(C)N(Cc2c(C)nc(C)s2)CCC1)=O c1(C(C)NC(Cc2cncs2)CO)cc(C2CCCCC2)cc(Cl)c1O N1(C(C(CCN(C)C)O)=O)CCC(CC(=O)NCC2CCCC2CF)C1(C)C Cc1cc(Cl)cc(C(N2CCN(C(=O)CC34COC(C)(C3)C4)CC2C)=O)c1O C(c1c(Cl)cccc1Cl)=CC(=O)NCC(CNC(C=CCOC)=O)CO C12(NC(C3C(CC)C3)=O)CCC(NC(=O)Cc3cccc(OC(F)F)c3)(CC1)CC2 N1(C(C(C)NS(CC)(=O)=O)=O)CCC(CNC(=O)CSC(C)(C)C)C1(C)C c1(C(=O)NCC(C)N(C(C2CCC(C(N)=O)O2)=O)CC)ccc(Cl)cc1 CC12CC(C(=O)NCCC3CN(C(=O)Cn4cc(C5CC5)nn4)C3)(C1)C(C)(C)O2 C1(CNC(CCC(=O)OCC)=O)CC2CCC1N(C(=O)C(C)SC(F)(F)F)C2 c1(C(=O)NCC2(O)CCN(C(C3(C)CCCS3)=O)C2)ccc(Br)c(F)c1 c1(CCC(=O)NCc2cn(CCNC(=O)CO)nn2)nc2ccccc2s1 c1(OC)cc(C)cc(C(=O)NCC2COCCN2C(c2occc2C)=O)c1C N1(C(C2(OC)CCCC2)=O)CC(NC(=O)Cn2nnc(=O)[nH]2)C(O)C1 c1(CC)cc(CC(=O)NCC2CC(O)CN2C(=O)C(C(C)C)N(C)C)n(C)n1 C1(C(N2Cc3ccccc3C2)=O)C2CC(CC2F)N1C(c1cnnc(O)c1)=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC(C=CCN1C(=O)CCCCC1=O)C.CO N(C1c2cc(C)ccc2CC1C)C(=O)NCc1nnc(COC)s1 C(=O)(CC(C)CCC=C(C)C)N(CC(C)NC(C(C)=C1CCCC1)=O)C N1(C(CNS(C)(=O)=O)=O)CCC2(CCCCN(C(=O)CNC(N)=O)C2)C1 C=CC(C)C(=O)NCC1(C(=O)NC(C)C(=O)NCCCF)CCC1 c1(C(=O)NC2CCC(C)(NC(C3CC(CC)C3)=O)CC2)c[nH]c2cccc(C)c12 N1(C(c2cc(C)sc2Br)=O)CCC2(NC(C3CC3(F)F)=O)CCCC12 c1(Cc2nnnn2C2CC2)cc(OC)n[nH]1.C1CN1CCF.COC C1(C)(C(=O)NC(CN(C(=O)CC2(O)CCC2)C)Cc2ccccc2)CCCOC1 CC(C)C(C)C(=O)N1CCC1C(=O)NCCCC(O)CO c1(OC)cc(C(=O)NCC2CCN(C(=O)Cc3cncnc3)CC2C)ccc1C c1(OCC)ccnc(N(C2CNCC2C#N)Cc2ccc(OC(F)F)cc2)n1 CC1CCC(CC(N2CCCC2CN(C(=O)Cn2cccnc2=O)C2CC2)=O)CC1 c1(CNc2c(C)c(NC3CCC(C)CC3C)ncn2)n[nH]c2c1CCCC2 N1(C(CSCC(C)C)=O)CCC2C1CCCN2C(=O)C=CCF n1(CC(=O)NC2CCC(CNC(C3OCC(C)(C)C3)=O)C2)cnc([N+](=O)[O-])c1 c1(C(=O)NCCCCC(C)NC(C(F)=CC)=O)c(F)cc(Cl)cc1F N1(C(CC(CC)SC)=O)CC(=O)NC2CN(C(=O)CSc3nc[nH]n3)CCC12 N1(C(c2ccc(C)n2C)=O)CCC(NC(=O)Cc2cnoc2)C12CC2 CC(C)(C)CC(O)CC(=O)NC(CC1CC1)NC(=O)CCCc1ccc(Cl)cc1 C1(CN(C)C(C2(CO)CC2(F)F)=O)CCCN1C(=O)CN(C1CCC1)C1CC1 C(C(C)(C(C)C)NC(=O)CC(C)N(C)C)NC(c1cnc(CC(C)C)s1)=O S(=O)(=O)(c1ccccc1NC(c1cnc(-c2cnc(Cl)c(F)c2)cn1)=O)NCC c1(C(=O)NCC(C)CNC(C2C3CCC23)=O)nc(-c2ccco2)n2ccccc12 c1(C(N(C2CCN(C(CN(CCC)C)=O)CC2)CC)=O)cc2ccccn2c1 C12CC3(C1)CN(C3)C(=O)C(C)N2C(=O)COC.c1(OCC)ncccn1 N1(C(c2n(CC)ncc2)=O)CCC(NC(=O)CC(C)(C)CC(F)F)CC(C)(C)C1 c1(CN2C(CC(=O)NC3CC3)CCC2)ccc(C(F)(F)F)cc1I C1(C(N2CCC(NC(c3cccnc3S)=O)C(F)C2)=O)Cc2cccnc2C1 N1(C(CNC(=O)NC)=O)CCCC2(C1)CN(C(c1ccc(CF)cc1)=O)CCO2 c1(C(N2CCN(C(CCOCC#C)=O)CC23CC3)=O)c[nH]c2ccc(O)cc12 C(=O)(CC(C)COC)N(C(C(=O)NCCN(C(C)C)CC)C)C C(C(=O)N1CC(O)CC1C(=O)NCC1CN(C(=O)OC(C)(C)C)C1)(C(C)C)SC CC(O)CC(=O)NCC(O)CCNC(=O)CC1CCSC1 c1(CC(=O)OC)ccc(NC(C2CSCCN2C(=O)C=Cc2cnc[nH]2)=O)cc1 CC(C)C(O)C(C)C(=O)NCCc1n[nH]cc1C(N1CCOCC1CO)=O c1(N2CC(C)CC(C)(C)C2)ccc(S(=O)(=O)N2CC(CO)C3(CCC3)C2)cc1F c1(C(=O)NCC(C)CN(C(=O)C(C)(C)C)C)nccc2ccccc12 CCC(C)(CNS(=O)(=O)Cc1cccc(F)c1Cl)C(C)O CN1CCCCN(C(=O)C(c2ccco2)NC(C2CC23CCC3)=O)CC1 c1(NC)cnc(SC)nc1C(=O)NC(C)C(=O)Nc1ncn(C)n1 C(c1ccccc1)=C(OC)C(=O)N(C(C)CNC(=O)CCCN(C)C(C)C)C C1(C(=O)NCCNC(C2CC3(CSC3)C2)=O)CC(c2ccccc2[N+](=O)[O-])=NO1 c1(C(=O)NCC2CC(F)(CNC(C(CC)SC)=O)C2)cn2cc(C)nc2s1 CC(C)CC(F)C(=O)N1CC(NC(=O)CC2(C)CCCCC2)C1 N1(C(CCCSC)=O)CCN(C(C2C3COCC23)=O)CC1C C1(C(N2C(CCCC)CCC2)=O)CC(F)CN1C(c1ccc(Br)cn1)=O C1(CC=C)(NC(=O)CCC(F)F)CCN(C(c2cc(COC)no2)=O)C1 C(=O)(C1CCCc2ccnn21)NCCOC(CNC(CN(S(C)(=O)=O)C)=O)(C)C C#CCC(C(=O)N(CCC(=O)NC1(CO)CCSC1)CC1CC1)C1CC1 C(=O)(CCCCCc1cccs1)NCC(CNC(=O)CC(C)N(C)C)OC N1(C(C)CNC(C23CC(n4cc(Cn5nccn5)nn4)C2C3)=O)C(=O)CCC1=O N1(c2nc(C)cc(SC)n2)CCC2C(CCCN2C(C2CCN(C)CC2)=O)C1 C1(C(N(C2CC2)CC2N(C(CCc3n(C)ncn3)=O)CCC2)=O)CCCC12CC2 C(CCCCC(=O)NC1CCN(C(c2cc(C)ccc2Cl)=O)CC1CO)=CC CC(C(=O)NC1CCCN(C(C2(F)CCC(F)(F)CC2)=O)C1)C1=CCCC1 CCCC(O)(CCC)CC(=O)N1CCCC1Cc1ccc(F)cc1 c1(NC(CC2N(Cc3cc(C)nn3C)CCC2)=O)cc(F)cc(Br)c1 S(=O)(=O)(c1ccc(NCCCC2CCC2)c(F)c1)NCC(CCCCC)O c1(C(=O)NCC(N(C(C(COC)N(C)C)=O)C)C2CC2)ncc(Br)cc1F N1(C(C(C)OCC#C)=O)CCC(C)CC1CNC(=O)CCCOCC C1(C(=O)NCC(CCOC)NC(=O)C(C)(C)C(F)(F)F)CC2(C1)CC1(CCC1)C2 C1(CNC(C(C)Sc2ccc(Cl)cc2)=O)(CF)CC12CCOCC2 C1(CNC(=O)CC2(O)CCC2)CCN(C(c2nnc(O)cc2O)=O)CC1(F)F c1(-c2c(C(N3CC(C)OC(C)C3)=O)sc3c2CCC3)ccc2nc(O)[nH]c2c1 c1(CNC(C(C2CCC2)OC)=O)cccc(NC(=O)C=CC(F)F)c1 C(CC(=O)N1CCC(N2CCC2)C1)(C(F)F)NC(C=NOC)=O C(=O)(C(O)CCC(C)C)NC1(CC)CCN(C(C(CC)n2ccnc2)=O)CC1 C1(NC(=O)CCC2CC2)CC2CN(C(c3cccc(CO)n3)=O)CC2C1 C(=O)(CCCCC(C)(C)C)NC1(CNC(C(CC(C)C)=O)=O)CC1 C12(NC(N3CCN(CC(F)(F)C(F)F)CC3)=O)CC3CC(C1)C(O)C(C3)C2 c1(NC(C2N(Cc3cc(C)c(F)cc3)CC2)=O)cc([N+](=O)[O-])cnc1C N1(N(C(c2noc(-c3cccs3)n2)C)C)CCCC(O)(C)CC1 C1(C(=O)NOCC2CC2c2ccccc2)CCC(CC2CCCO2)C1.O=C1CO1 N1(C(c2c(CC)c[nH]c2)=O)CC(N(C(=O)CS(=O)(=O)NC(C)(C)C)C)C(C)(C)C1 C(CNC(C1(C)CCCS1)=O)(CC(C)C)NC(c1c(CC)non1)=O CC1C(C(=O)NC(C)(CCN2CCCC2)c2nn[nH]n2)CC1(F)F C(C(COC)CC(=O)NCC1CCN1Cc1ncccc1OC)OCC C1(C(=O)NC(C2CN(C(c3nonc3N)=O)CCO2)C)COC2COCC12 C#CCC(CC(=O)NC(C)(CC)CO)NC(c1ccnc(CO)c1)=O c1(C(=O)NC(C2CCCN(c3ncc(O)cn3)C2)C)cccc2ncccc12 c1(CS(N2CCC3(C(C(=O)NC4CCC4)C3)C2)(=O)=O)cc2ccccc2[nH]1 C1(C(N(C(C(=O)NCC(n2cccn2)C)C)C)=O)CN2CCC1C2 Cc1ccc(C(=O)NCCN2CCC(CN(C)C)CC2)c(OCC(C)C)c1 N1(C(C23C(NC(C4C5CC(=O)CC54)=O)C4CC2C3C4)=O)CCC(O)(C2CC2)CC1 c1(C(N2C(CNC(CC3(OC)CC3)=O)CC(O)C2)=O)ccc(Br)c(F)c1N C(=O)(C1CCCn2ccnc21)N1CCOCC(NC(C=NOC)=O)C1 N1(C(Cc2cc(COC)on2)=O)CCC(C)(CNC(c2ccn(C(F)F)n2)=O)C1 c1(C(N(C2CCCN(C(C3CCS(=O)CC3)=O)C2)C)=O)c[nH]c2nc(Cl)ccc12 c1(C(=O)OCC)ncc(F)cc1NC(=O)Nc1cccc(NS(=O)(=O)C(C)C)c1 c1(C(=O)NCC2(CO)CCN(C(c3c(CC)ncs3)=O)C2)c(F)cc(O)cc1F N1(C(c2cc(C)n(C)c2)=O)CC2CCN(C(c3cc[nH]c(=N)c3Cl)=O)C2C1 Cc1[nH]c(=N)sc1-n1cc(CN2CCN(C(=O)C(C3(O)CCCC3)F)CC2)nn1 C#CC1CCCCN1N1CCN(c2nc(C)c(C)s2)CC1 c1(C(N2C(C)CC(NC(=O)CCCCCC#N)C2)=O)c(Cl)cnc2ccccc12 N1(C(c2c(N)non2)=O)CC2(C1)CN(C(=O)CC1CC1(Br)Br)C2 N1(C(COCCC=C)=O)CCN(C(c2cocn2)=O)C(C)C1C CC1(C(=O)NCC2CNC2)CC12CCN(C(c1cc3ccc(Br)cc3o1)=O)CC2 CCCC(O)C(=O)NCC(C1CC1)NC(c1[nH]ccc1-c1ccccc1)=O C=CCC(C(=O)NC(CNC(c1sccc1C1CC1)=O)C1CC1)OC Cc1cc(C)c(C(=O)CN2CC3CC2C3C(=O)O)[nH]1 N1(C(CC2N(C(C3=NOC(C)C3)=O)CC2)=O)CCCC(F)(F)CC1 c1(C(C(=O)NCc2cccs2)N(C(c2ccccc2Cl)C)C)cc(Br)ccc1F C(=O)(CC1=Cc2ccccc2C1)OCCC(CCC)CCC C(=O)(C(C)CC(N)=O)NCC1C(C)CCN1C(=O)C(=O)Cc1cccc(F)c1 C1(CC(=O)N(CC(=O)NC(CC=C)CO)CCOC)CCCC(=O)C1 C1(CNC(C(C2(OC)CCCC2)(F)F)=O)CC(F)CN1C(C1(NC(N)=O)CC1)=O C(=O)(C(C)(C)C(=O)N1CC(N2CCN(C(C)=O)CC2)C1)OCC.C(=O)N C(c1ccc(F)c(Cl)c1)=CC(N1C(C)(CCNC)CC1)=O.C(C)(C)(C)OC(=O)N C(=O)(CC(CN(C)C)C(F)(F)F)N1CC1.CCCCC(C)C(=O)NCCOC C1(c2cn(CCCC(=O)NC(c3cccnc3)(C)C)nn2)(OCC)CCOC1 C1(C(N(C)CCOCCN(C)C(C2(C)CCC(=O)N2)=O)=O)CCC(C)(F)CC1 Cc1cc(C)n(CCCC(=O)NC(C)CCNC(c2cc(Br)c(C)o2)=O)n1 c1(C(N(CC(CNC(CCOCCC)=O)C)C)=O)cnc[nH]c1=N Cc1cc(CC(N2CC(OCC(=O)NCC3(O)CCN(C)C3)C2)=O)nn1C c1(C(=O)NCC(C)(O)CNC(c2cccc(F)n2)=O)cc(Cl)ccn1 N1(C(COCCC=C)=O)CCN(C)CC1CNC(=O)CNC(=O)CCC c1(C(N2CC(COC)(NC(=O)CC=C(C)C)C2)=O)cccn2c(C)nnc12 N1(C(CSc2c(C)n[nH]c2C)=O)CCC(C)CC1CNC(=O)C(F)CC1CCC1 C1(CNC(COCCOCC#C)=O)COCCN1C(=O)C(C)SC CCC(C)CCC(O)CC(=O)NC1CCN(CC2CCCN(CC(F)F)C2)C1C c1(C(=O)NC(C(C)NC(C2ON=C(C)C2)=O)(C)C)cc(OC(F)F)cc(F)c1 C(C)(CC(F)(F)F)NC(c1n(CC=C)nnn1)c1ccncc1 C1(C(=O)OC)OC(C(=O)OCCCc2nocc2C)CC1C C(=O)(CCC1=NNC(=O)CC1)N1CCC2(OCC(NC(CCOCC#C)=O)C2)C1 C(CCC(C)CC(=O)N1CCC=CC1C(=O)NC(c1cnccn1)C)=C(C)C c1(C(N2CC(NC(=O)CC3CCOC3)C(F)C2)=O)cc2c(cn1)OCCC2 c1(CN2CC(NC(C)=O)C(O)C2)cc(C)c(I)cc1C Cc1cc(Cl)ncc1NC(C1COC(CNC(c2cc[nH]c2)=O)C1)=O C1(C(=O)NC2(CC=C)CN(C(=O)CCC(=O)N(C)C(C)C)C2)CCCS1(=O)=O C1(CNC(Cc2c(C)ccnc2)=O)CN(C(=O)C(F)C(C)(C)O)CC12CC2 Cc1nn(C)cc1NC(=O)C(c1ccccc1)NC(=O)Cc1ccoc1 C(=O)(CS(=O)(=O)CC(=O)NCC1COC2(CCCC2)C1)OCC N1(C(C(CC=C)C)=O)CC(NC(=O)CC2(OC)CCC2)C2(CCCC2)C1 C1(C(C)(C)C)(CNC(CCC2C(C)(C)C2)=O)CCN(C(=O)CCn2cccn2)C1 Cc1ncnc(C)c1C(=O)NCC12CC(NC(c3snc(O)c3Cl)=O)(CO1)C2 C#CCC(C(=O)NCC(F)CO)NC(=O)Cc1cnnn1C C1(CNC(C2C(C=C)C2)=O)C(O)C(O)CN1C(c1sc(C)cc1Br)=O C(C(=O)Nn1cccn1)C1(NC(=O)C=Cc2ccoc2)C(C)CCC1 C(CCC(=O)NC(C)Cn1cc(CC(C)O)nn1)OCC=C c1(N2CC(C(C)NC(c3scc(OC)c3)=O)C2)nc(Cl)nc2c1cnn2C c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC(C)CNC(C1CC(C(F)F)C1)=O C(=O)(C(O)(CC)c1ccccc1)NCC(CC)NC(C1CC1C)=O c1(C(C(=O)NCC(CC)NC(C2CCC3CC3CC2)=O)C)ccc(F)cc1F c1(C(=O)O)ccc(S(=O)(=O)NCc2ccc(OC3CCCCC3)nc2)c(Cl)c1 c1(C(=O)NCC2CCCC2NC(C2(O)CC(F)(F)C2)=O)ncc[nH]c1=O C(=O)(C1(C)CCc2ccccc21)Nc1c(C)cc(NC(c2nonc2N)=O)cc1 Cc1cc(CC(=O)NC(C)CCC(=O)NCCCCC2CC2)ccc1O N1(C(=O)C(F)n2ccnc2)CC2(C1)CN(C(=O)COCC1CCC1)C2 Cc1ncccc1C=CC(=O)NC1CCC1CNC(C1CCN(C)C1C)=O C1(C(=O)NCC2(CNC(C3(O)CCSCC3)=O)CCC2)CCn2cnnc2C1 N1(C(CC(CC)NC(=O)CCOC2COC2)=O)CCCC(C)(O)C1 c1(CC)nc(C)c(C(=O)NCCNC(c2cc(Cl)sc2Cl)=O)o1 N1(C(=O)OCC)C=COCC1C(=O)OCCCCC1CC1C CC(C)(C)CCCC(=O)NC1CC(NC(C2CCOC(=O)N2)=O)C1 C1(CNC(C(C)O)=O)CCC(CNC(C2(Cc3cnn[nH]3)CCC2)=O)CC1 CCCC(C)(CCC)C(=O)NCCC1(O)CCN(C(C2CC2c2cccs2)=O)C1 C(=O)(C(C)(C)CCC(=O)OC)N1CCCC(CNC(CCSCCCC)=O)C1 N1(C(CCCC#N)=O)CCC(C2CCCN(C(C3Cc4cccnc4C3)=O)C2)C1 c1(CC(=O)NCC(CN(C)C(c2cc[nH]c(=N)c2)=O)O)ccc(Cl)c([N+](=O)[O-])c1 c1(CNC(C(=O)Nc2ccc(C(CC)C)cc2)=O)cccc(F)c1F CCCC(C(=O)N1CCOCC(NC(c2cnc(OC)c(C)c2)=O)C1)C(C)C CCCCCCCC(=O)NCC(CC1CC1)C(=O)Nc1cc(C)cc(C)c1 C1(F)(C(=O)NCC(COC(C)C)O)CCN(C(c2occc2C2CC2)=O)C1 CCC(CNC(c1ncn(C)c1C)=O)(CC)NC(=O)CC1C=NN(C)C1=O C1(O)(CCNC(C2CN(C)C2)=O)CCN(C(C2CCCC(C)CC2)=O)CC1 C1(C(N2CCC(NC(C=CSC)=O)(CF)C2)=O)CC(O)c2ccccc2O1 CCCCC(CC)C(=O)N1CCCN(C(c2cnc(OC)s2)=O)CC1 CC(CCNC(C1CCCCN1C(c1ccn(C)c1)=O)=O)C(F)F C(C(F)(C(=O)N1CCN(C(=O)CC)CC1)C(C)C)NC(C1(CCCC)CC1)=O C(=O)(C1=CCC2CCC1N2C(c1coc(C(N)=O)c1)=O)NCC1N(CC)CCC1 n1(CC(=O)NCC2C(CNC(CC(C)(F)F)=O)C2)cccc(O)c1=O c1(CC#N)cccc2c1CCN(c1ccnc(-c3ccncc3)n1)C2 c1(C(=O)NCCCC(C)NC(C2CCOC(=O)N2)=O)ccc2c(n1)CCC2 c1(C(N2C(CNC(CC3(C(=C)F)CCC3)=O)C=CC2)=O)ccc(OC)c(OC)c1 c1(NC(C2CCN(C(c3cc(C4CC4)on3)=O)CC2O)=O)cccc2occc12 c1(COC)csc(CNCc2ncoc2C2CC2)c1 N1(C(c2scnc2C)C(=O)NC(=O)NCCCOC)CCCC(C)(OC)C1 C1(C(=O)NCC(CC#C)(C)C)CCCCCN1C(=O)CCc1cnc(C)o1 Cc1sc(O)nc1C(=O)NC(C)CN(C)C(c1cncc(-n2cccn2)n1)=O c1(C(N2CCN(C(C3C(C=C)CC3)=O)C(C3CC3)C2)=O)nnc2n1CCCCC2 c1(CC)cc(OC)ccc1C(N1CCCC1C(C)NC(=O)C1=CCC1)=O CC1CN(C(=O)C(c2ccoc2)NC(C2CC2C(F)(F)F)=O)CCC1CO CC1(C)CCCCC1C(=O)NC1CC(C(=O)NOCC2CCC2)C1 c1(OCc2c(C(C)CC(=O)O)cccc2)ccccc1N=NN(C)C N1(C(CC(CC)(C)C)=O)CC2(CC(NC(=O)C(c3ccccc3)F)CO2)C1 N1(C(=O)CCCCCCCC2CC2)CCCC12CCN(C(=O)C(F)(F)C(F)F)C2 c1(C(=O)NCCC2C(C)CCCN2C(=O)CCCC2CC2)ccc(C#N)cc1F C1(C(=O)NCCS(=O)(=O)NC)CCCN(C(=O)CCCC2CC2)CC1 CC(=O)CCN=C(NCc1cccc(S(C)(=O)=O)c1)NCc1c[nH]nc1C(F)F c1(C(=O)OC(c2cccc(F)c2)C(=O)OC)cccc(C2(F)CC2(F)F)c1 N1(C(=O)C2CC2)CCCC(C2CCCCN2C(=O)Cn2cnc(Br)c2)C1 c1(OCC)c(C(=O)NC(C)C(C)NC(=O)COc2ccccc2)cccc1F N1(C(C2C(C#N)C2)=O)Cc2ccnn2CC(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1 N1(C(c2cc(C)cc(F)c2)=O)CCC(NC(c2cnsn2)=O)CC(C)(C)C1 C(=O)(C1CCCc2cccnc21)NC(CC)(CNC(=O)C1=COCCO1)CC C(=O)(CS(=O)(=O)CC(C)C)NCC1(F)CN(C(C=C(COC)C)=O)C1 C(CC1CCCO1)(C(F)(F)F)NC(N1CCC1COCC1CC1)=O C#Cc1ccc(C(=O)NC2CC(CNC(c3coc(C)c3)=O)C2(C)C)cn1 N1(C(C2(NC(C3CCCC(O)C3)=O)CCCC2)=O)CCC2OCCC2C1 c1(C(N2CCC(C(C#C)C)CC2)C(=O)NCC)cc(C)c(OC)c(C)c1 C1(NC(CN2CC(C)C2)=O)CN(C(c2cc3c(F)cccc3[nH]2)=O)C2(CCCC2)C1 C1(C)(C(=O)NCC2CCCC(NC(CN(C(C)=O)C)=O)C2)CC2CCC1O2 C1(CNC(=O)NCC2(C(C)(F)F)CCC2)C2C3CCC(C3)C12 CS(=O)(=O)C(CNC(=O)Cc1c[nH]ccc1=O)CNC(C1C2CC3C(C2=O)C13)=O c1(CCC(=O)NC(C(=O)NCC(C=C)O)c2cccs2)cc(C)[nH]n1 N1(C(C2(CC#C)CCCC2)=O)CCN(C(C2OCC2(C)C)=O)C(C2CC2)C1 N1(C(CC2N(C(C(SC)SC)=O)CCOC2)=O)CCC2=C(CCCC2)C1 C1(n2cc(CC)nn2)CC(c2nnnn2C)(NCC(C)(C)C2CC2)CCO1 C(C(C)C(=O)N1CCC(CCNC(c2csc(C(F)(F)C(C)C)c2)=O)C1)SC CON1CC(C(N2CCC(C)(CNC(=O)CSc3cn[nH]c3)C2)=O)CC1=O CCCCC(C)C(=O)NCC(C)(C)CN(C(c1cn(C)c(C)n1)=O)CC C1(CCC#C)CN(C(c2cc(NC(=O)OC(C)(C)C)c(C)o2)=O)CCO1 c1(OC)cc(C(C(=O)O)Nc2sc(C)nc2C)ccc1C(F)(F)F N1(C(C(=O)NCC(=O)N(C2CCCN(S(C)(=O)=O)C2)C)=O)CCCC2NCCC12 N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(C(=O)CCS(C)(=O)=O)C2)C1 N1(C(CC)=O)CC2(CC(C(=O)Nc3csc(C)c3)CO2)C1 C1(NC(c2cc(CNC(C3CCN(C4COC4)C3)=O)[nH]n2)=O)CCCC(CO)C1 c1(OC)c(Cl)cc(C(=O)N(CC(C)N(C)C(c2cnc(C)cn2)=O)C)cc1Cl CCC(CCCC(=O)N1CCS(=O)C(C)C1)NC(C1CCN1C(C)(C)C)=O N1(C(C(CC)n2ccnc2)=O)CCCN(C(c2cc(C(C)=O)cn2C)=O)C(C)C1 c1(C(N2CCC(CCNC(C(c3cccs3)SC)=O)CC2)=O)cc(F)ccc1N N1(C(C2CCC(C)CC2)C(=O)NC2CC2)CC=CCC2(CCOCC2)C1 N1(C(CNC(CNC(C)=O)=O)=O)CCC(CCNC(c2nn[nH]c2Cl)=O)C1 C=CCCCCCC(=O)N1CCCC(C)(C)C1CNC(=O)C(CC)C(C)(F)F N1(C(c2c(C)nccn2)=O)CCCCCC1CNC(=O)CCC(C)(C)C N1(C(c2ncccc2Br)C(=O)NCCc2c(OC)cccc2)CCC(O)C(F)C1 C(=O)(N1CCC(C(N2CC3CCC(C2)O3)=O)O1)C1C(C#N)C1 C1(C(=O)NCc2oc3ccc(OC)cc3c2)COc2ccccc2O1 c1(C(N2C(CNC(C3CC(OC)C3)=O)CC(OC)C2)=O)cncc(S(C)(=O)=O)c1 c12cnc(C)c(c1)C(=O)N2.N1(C(C)=O)CCC(C)C(NC(c2cccs2)=O)C1 Cc1cc(F)ncc1NC(C1CC2(CC2)CN1C(c1cnccc1N(C)C)=O)=O C1(C(N(CC(C)(C)NC(C2CC2c2ccccn2)=O)C)=O)(C(=O)OC)CCSC1 C(=O)(CCC(=O)NC(C1CCN(C(c2ccncc2NC)=O)C1)C)NCCC C1(OC)(CNC(=O)C(C(C)C)OCC(C)C)CCN(C(=O)CC2CNC(=O)C2)C1 N1(C(C2N(C(C(C)SCCCC)=O)CC(=O)C2)=O)CCC2(CCCO2)C1 CCC(CCC(=O)N1CCCC1C(O)CO)NC(=O)CS(=O)(=O)NC C1(CCOC)(NC(c2cn(CC)nc2)=O)CCN(C(=O)C(O)CSC)C1 c1(C(=O)Nc2ncc(SC)s2)cc2cc(C(=O)N=c3cc(C)[nH][nH]3)ccc2[nH]1 CC(C)C(C(C)C)C(C(=O)NCc1ccc(F)cc1)N(C1CC1C)C CC1CCC=C1C(=O)N1CCC2(CC2NC(c2cccc(F)c2F)=O)C1 c1(C(=O)NC2C(CNC(C3CC(OCC)C3)=O)CCC2)occ(C)c1C N1(C(C(CCC)N(C)C)=O)CCN(C)CC1CNC(=O)C(F)CC1CCCCC1 C1(CC)C(=O)N(C)CCN1C(=O)C(CCC1CC1)NC(=O)COCC(F)F C#Cc1cnc(C(=O)NCC2CC(F)CN2C(=O)CC2CNC(=O)O2)c(C)c1 c1(C(C)N(C(=O)CCOCCOC2CC2)CCCO)nnc(C(F)F)o1 CC1C(NC(=O)Cc2ccns2)CC2CCC1N2C(C1(NC(N)=O)CC1)=O NC1(CC(=O)NC2CN(C(N)=O)CCC2c2ccccc2)CC2(CCOCC2)C1 c1(C(=O)NC(c2ccccc2Br)C#N)nccc2c[nH]nc12 CC(C)C(C(=O)N1CCCC(C(C)N(C(C2(n3cccn3)CC2)=O)C2CC2)C1)C1CC1 Cc1oc(C(=O)NC(C)(CNC(=O)C(C)CO)CO)cc1Br CC1CN(C(C2CC23CC(O)C3)=O)CC1(C)CNC(c1ccc(F)cc1)=O N1(C(C(C(C)C)C#N)=O)CCCC(C)(C)C1C(N1CC(N(C)C)C(F)C1)=O N1(C(C(C2CCC2)OC)=O)CC(NC(c2nc(OC)c(C)s2)=O)C(C)C1 n1(CC)c(N2CCCC(C(=O)Nc3ccccn3)C2)nnc1-c1ccc(Cl)nc1 c1(-c2n(C)nc(-c3ccccc3N3CCOCC3)n2)cnn2ccc(O)nc12 C1(NC(c2ccc(C)o2)=O)CC2CC1CN(C(=O)C(C)(C)C1CCCCO1)C2 Cc1nc(NCCCc2nc3ccccc3[nH]2)cc(=NCC(C)CC(F)(F)F)[nH]1 N1(C(C2CC(NC(C3CN(C(=O)NC)C3)=O)C2(C)C)=O)CC(COC)C2(CC2)C1 Cc1cc(O)ccc1CNC(=O)C(C)N(C)C(c1cc[nH]c1)=O c1(C(=O)NCc2nccc(C(=O)NC(CCC)CCO)c2)cc(N)cc(F)c1 c1(C(N2CC(CNC(C=C(CC)C)=O)C(C)C2)=O)cc(N)c(OC)cc1OC C1(C(=O)NC(CNC(c2ccn(CCC)n2)=O)(C)C)NC(=O)CC1C(F)(F)F N1(C(C(C)=C2CC2)=O)CC(NC(C23COC(CF)(C2)C3)=O)CC1C CC(C)C(O)C(=O)NCCOC1CCN(C(C2CC(N(C)C)C2)=O)CC1 C1(C)(NC(CN(C2CCC2)C(c2cnc(CC)nc2)=O)=O)CC(C)(C)OC1=O Cc1nn(C)c(Cl)c1CC(=O)NC(CNC(C1CCC(O)C1)=O)C1CCC1 C1(NC(=O)COCCN(C)C)CC2(CCCN(C(C3CC3c3cccs3)=O)C2)C1 CC(C)CC(C(=O)NC(CC1CCC1)C(=O)N1CCC1(C)CCO)C(C)C CC1CCCN(C(=O)C2=NOC(C)C2)C1CNC(c1ccc(N)c(Cl)n1)=O C1(NC(CCC2COC(C)(C)O2)=O)COCCN(C(C2CC(CC3CC3)C2)=O)C1 Cc1cn2c(n1)C(C(=O)N1CC(NC(=O)C3=CCCSC3)C(O)C1)CCC2 c1(OCC)nc(Br)ccc1CCCNC(N1CCCCCC1CCO)=O N1(C(c2nnn(CC)c2C)=O)CC(F)(F)CC1CNC(=O)CS(=O)(=O)CC C1(C(=O)NCc2cnn(CC)c2C)CC2CC1CN(C(=O)CC(F)(F)F)C2 C(=O)(C(C)(CC)CCC(C)C)NC1CC2(CC(CNC(C(C=C)O)=O)C2)C1 c1(C(N2CCN(C(C(C(CC)C)OC)=O)CC(O)C2)=O)nc2nccc(C)n2n1 C1(C(=O)NCC2(C)N=C(C)SC2)CCN(C(C2(C)CCCCO2)=O)CC1C c1(OC)ccccc1C=CC(=O)NC(C)CCCCNC(C1CCCOCC1)=O c1(C(=O)NCC2(C)CCN(C(C3CC3C#N)=O)C2)ccc2c(c1)COC2 c1(CC(C(=O)NC2(C(=O)OC)CCCOC2)n2nnnc2C)cc(Cl)cc(Cl)c1 C1(NC(c2nnc(C(C)(C)C)s2)=O)CCC2CCN(C(C3CSCCS3)=O)C1C2 C(=O)(C(=O)N=S(C)(C)=O)NCC1(NC(C(NOC)=O)=O)CCCCC1C c1(C(=O)OC)cnc(=NCC2CC(NC(=O)CC3C=CS(=O)(=O)C3)C2)[nH]c1 C(=O)(CC(CC)C(C)C)NC(CCCCNC(C=CCOC)=O)(C)C C1(C(=O)NC(C2(CCCNC(C)=O)CCCCC2)C2CC2)CC(=O)CC12CCC2 C1(C)(C(=O)NC(CC)C(=O)OC)CCCN(Cc2cncc(F)c2)C1 Cc1nc(CC(F)(F)F)sc1C(=O)NC(C)COc1cccc(F)c1 c1(CCC(=O)NCCC(C)NC(c2cccc(C3(C)CC3)c2)=O)cncc(F)c1 C1(C(=O)NCCC2(CO)CN(C(CCOC(C)=O)=O)C2)CCCCC12CC2(F)F c1(NC(=O)NCc2scc(C)n2)c[nH]c2nccc-2c1 Cc1nn(C)c(C(=O)NC(CNC(=O)Cc2cnn(C)n2)CC(C)C)c1Cl C(=O)(C1CCCc2ncnn21)N(C)CCN(C)C(c1cnc(C(F)F)nc1)=O N(C(=NCC(C)C)NCc1ncccc1Cl)CC(NOCC)=O c1(C(=O)NC2C(CC)CN(C(=O)C(Cl)=CCl)CC2)cc2cc(OC)ccc2[nH]1 Cc1cccc2c(C(=O)NCCCCC(C)NC(=O)Cc3cnns3)coc12 c1(C(=O)NCC2(CN(C)C(C3CC3(C)Br)=O)CC2)nnc(O)cc1O C1(F)(CNC(=O)Cc2ccc(F)cc2)CCN(C(C2CC3(CCC3)C2)=O)CC1 c1(CNC(COc2cccc(C(=O)NC)c2)=O)cc(S(C)(=O)=O)c(OC)cc1C CC1CN2CCCC2CN1C(c1ccc2c(c1)CCC2)C(=O)NC1CCCCC1 C1(C(C)CNC(=O)Cc2cnoc2)CCN(C(c2cc(O)ncn2)=O)CC1 S(=O)(=O)(CC1=NOCC1)NC(c1nnc(-c2ccccc2)s1)C N1(C(C2C(C)CC2)=O)CC(C2(NC(c3cnc(C4CC4)nc3)=O)CC2)C1 n1(CCCC(=O)OC(C)(C)C)nc(-c2cc(Cl)ccn2)nc1C1CCC1F c1(C(c2n(CC(=C)C)nnn2)NCC(=O)OCC2CCOC2)cccc(C)n1 S(=O)(=O)(c1cccc(N2CC3(CCC3)OCC2C)n1)NCC(C(C(C)C)O)(C)C C(=O)(CS(N)(=O)=O)NC(C1CN(C(=O)CC2(C)CC2(Cl)Cl)CCO1)C c1(C(N(C(C)C)CCN(C)C(C2CC2F)=O)=O)cnc2c(F)cccc2c1 C1(CC(N2CC(NC(c3cnn(-c4ccccc4F)c3)=O)C2)=O)CCCNC1=O c1(CC)ccc(CC(N2CC3(CCC3NC(=O)C(C(C)C)SC)C2)=O)c(C)c1 c1(C(N(C2CCCC(NC(C3CCC=CCC3)=O)C2)C)=O)cc2n(n1)CCO2 c1(N2CC(CNC(c3c(N(C)C)nccc3)=O)OCCC2)ccn2nccc2n1 N1(CCc2cn(C3C(OC)COC3)nn2)C(=O)C2CCCCC2C1=O c1(OC(C(=O)OC)C)cccc(C(N2CCOC(CNC(=O)C(C)(C)C)C2)=O)c1 c1(C(=O)NCC(CN(C(c2[nH]cc(CC)c2)=O)C)C)cc(C)c2occc2c1 C(=O)(C1CN(Cc2ccnn2C(F)(F)F)Cc2ccccc21)OC c1(C(=O)NCC(C)NC(C(COC(C)C)NC(C)=O)=O)noc2c(F)cccc12 C1(NC(=O)CCc2cnn[nH]2)CC2CN(C(C3(F)CC=CC3)=O)CC2C1 C12(C(N3CCC(N4CCC(NC(C(F)=CC)=O)CC4)C3)=O)CCC(CC1)OC2 c1(N2CC(C(C)C)OCC2)nc2cccnc2c(=NC2CN(C)C2)[nH]1 C=CCC(C(=O)N(C1CCCN(C(c2ccc(CC)cc2)=O)C1)CC)OC N1(C(c2cncc(C(C)(C)C)c2)C(=O)NCC)CC(CO)C2(CC2)C1 CCC(CC(=O)N1CC(CC(F)C(N2CCCCC2C(C)(C)O)=O)C1)CC(C)C c1(C(N2CC(C)C(NC(=O)CCc3ccn(C)c3)C2)=O)csc2nnsc12 Cc1cc(C(N2CC3(CCN3C(=O)C(C)n3ccnc3)C2)=O)nnc1C N1(C(CCC(C)(F)F)=O)CCC2(CC1)C(NC(=O)C=Cc1ccsc1)CS2(=O)=O C1(C(=O)NCC(CC(C)C)NC(=O)CC2(O)CCCOC2)CCCCCCC1 N1(C(C2(COC)CCCO2)=O)CC(NC(=O)C(O)Cc2cnc[nH]2)C(C)(C)C1 C12(C(N(CCN(C(C)C)C(C3CC34CCOC4)=O)C)=O)CCCC(C)(C1)OC2 c1(C(=O)NC2CC(NC(CSCC=C)=O)C2)sc(CC)nc1C c1(C(=O)NC2(CC=C)CN(C(C3CCCOCC3)=O)C2)ccnc2c1CCO2 C12CCCN(C1)C2=O.c1(C(C)=O)nc(C(=O)NCCCNC(N)=O)cs1 C1(NC(C(COC)(C)OC)=O)CCC2(CCN(C(c3csc(Cl)n3)=O)C2)C1 c1(C(=O)NCC2C(C)(C)N(C(=O)CCc3ccoc3)CC2)ccc2ocnc2c1 Cc1c([N+](=O)[O-])c(C(=O)NC2CC3CN(C(=O)CCCN(C)C)CC3C2)nn1C N1(C(C=CC(C)(C)N(C)CCO)=O)CCN(C(=O)C(F)C2CC2)CC1 N1(CC(=O)NCCc2c(OC)ccc(Cl)c2)CCCCC2CCCCC12 C(=O)(C#CC1CCOCC1)NCc1ncc(C(N2CC(C(C)C)OCC2)=O)cn1 C(=O)(CC(C)(O)C(F)(F)F)NCC(C(C)C)(F)C(=O)NCC1=CCCN(C)C1 c1(C(N(CC(C)CNC(=O)CCC2CC2(F)F)C)=O)cc(N)c2ccccc2n1 C1(CC(N2CC(O)(CN(C(C3(COC)COC3)=O)C)C2)=O)CC(=O)NC1=O CCCC(C(=O)NCC1(C)CCCN1C(C1CC(N2CC(O)C2)C1)=O)OC C=CCCN=C(NC(=O)Cc1ccccc1)NC1CSC1(C)C c1(C(=O)NCC(CCNC(C(C)O)=O)(C)C)cc2c(s1)C(C)(C)CCC2 C1(NC(C(CCC)N(C)C)=O)CCOC12CCN(c1ncc(C)c(O)n1)CC2 c1(C(=O)NCCOCCCNC(CC2CC(=C)C2)=O)ccc(OC(F)(F)F)cc1 N1(C(COCC(=O)OC)=O)CCOC(Cc2cn(C(C)(C)C)nn2)C1 Cc1ccc2[nH]nc(CN(CC(=O)O)Cc3cccc(CS(N)(=O)=O)c3)c2c1 Cc1c(C(=O)NCC(F)CNC(=O)C(O)CN(C)C)cc(S(N)(=O)=O)cc1F CCCCCCCCC(=O)NC1CCN(C(c2coc(C3CC3)n2)=O)CC1C C(=O)(CC(C)(C)N(C)C)N(CCC(=O)NC(CCC=C)C)C(C)C O=C1CCc2cc(NC(=O)COC(c3ccc(Cl)c(I)c3)=O)ccc2N1 c1(C(N2CC(CNC(c3cc(CCOC)on3)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(CC(C)(C)C2CC2)=O)CCC(C2=NOCC2)C1.C1C(=O)NCCO1 N(C(=NCC(F)(F)F)NCC1(CC2CC2C)CC1)Cc1ccc(SC)cc1 c1(N2CCC(Cc3n(C)ncc3)C2)cc(C#N)ccc1Br C(=O)(C(O)CC(N)=O)NC(CSC)(C)C(=O)NCc1csc(C)n1 C1(NC(C=C(CC)C)=O)CC2CCC1CN(C(c1ncn(C)c1C)=O)C2 C(C(O)CC(=O)N1CC(C)(C#N)C1)NC(Cn1ccc(C)n1)=O c1(OC)cc(C)c(C(N2CCCN(C(=O)C=C(C)C(C)C)C(C)C2)=O)cc1Cl C1(C(=O)Nc2cccc(C3(N)CC(C)(C)C3)c2)NC(=O)OC1(C)C c1(OC)ccc(C(=O)NC2CC(F)CN(C(=O)C=CC3CCCC3)C2)nc1N C(c1scnc1C)=CC(=O)NCC(CNC(C=CCN(CC)CC)=O)CO C(=O)(C(C)(O)CC(C)C)N(C(C)C(=O)Nc1cnc2c(c1)CCC2)CCC C1(NC(=O)CN2CCCC2=O)CC2CC1N(C(=O)CC(O)C1CCCC1)C2 C1(OC)CC(C(N2CCCC2CC(=O)NCC(C)C(C)(F)F)=O)CC1O C1(C(=O)NCC(CNC(c2cc3nccnc3[nH]2)=O)OC)CCC2CC1C2(C)C c1(CC(=O)N(C2C3CN(C(C4COC4)=O)CC23)C)ccc(F)c(Cl)c1 CC1CN(C(=O)C=C2CCN(C)C2)CCN(C(C2CC(=O)C23CCC3)=O)C1 C(N=c1[nH]c2c(c(=NC3CSC3)[nH]1)CSC2)C1(N(C)C)CCSC1 Cc1nc(C(N2CCC(NC(=O)Cn3ncccc3=O)C(C)C2)=O)ccc1C#N C(=O)(CCCCCCN=[N+]=[N-])NC(C1(O)CCN(c2cc(C)nc(CO)n2)C1)C C1(F)(CNC(CCCC)=O)CCN(C(C2(Cl)CC2(C)C)=O)CC1 C(=O)(C(F)CC(C)(C)NC(=O)C(C)CC=CC(=O)OC)NCCOCC=C C#CC1CN(C(C2(n3nccn3)CC2)=O)CCN1C(=O)CC(O)C(C)C CC1(C)CC=C(C(=O)N2CC(CNC(=O)CNc3ccccc3Br)C2)CC1 C#CCC(CC(=O)N1CCC(C(N)=O)C1)NC(c1oc(C)nc1C)=O c1(C(=O)NCC2(NC(c3cc(Cl)c[nH]3)=O)CCOC2)ccccc1-n1cccn1 N1(C(CCCN(C(C)=O)C)=O)CC(N(C(=O)C=Cc2ccsc2)C)C(F)C1 c1(C(=O)OC)sc(NC(=O)C(=O)NCCn2ccc(C)n2)nc1C(C)C Cc1ccc(NC(c2cc(C(=O)NC3CC(NS(C)(=O)=O)C3)cs2)=O)c(C)c1 C(=O)(C(C)(O)CN1CCCC1)NC1(CC=C)CN(C(C2CCC(O)CC2)=O)C1 CCC(C)CC(C(=O)O)NC(c1ncccc1Br)=O C1(C(N(CC=CC(=O)N(CCC)C2CC2)C)=O)CC2CC1CC2O CC1(C)CCCC(CNC(=NCCc2cccs2)NCC2CCC=CO2)O1 C(=O)(CC(F)(F)C(C)C)NC1CCN(C(C=C(C)c2ccco2)=O)C12CC2 CCCC(C#N)C(=O)NCC1(CN(C(=O)CCc2nnc(C(F)F)o2)C)CC1 c1(C(N2CC(CC)N(C(c3csc(=NC)[nH]3)=O)CC2)=O)cc(C)c(=O)n(C)c1 c1(C(N(C2CCN(C(c3n(CC)ncc3)=O)CC2)C)=O)c[nH]c2cccc(F)c12 N1(C(CC(=C=C)C)=O)CCC2C(CCN2C(c2ccc(NC)c(F)c2)=O)C1 C(C)(C(=O)NC1CC(CCNC(=O)CCC2(C)CC2)C1)OCCCC CCC(CC)(CCNC(c1ccnc(OC)c1)=O)NC(C1CCCC(OC)C1)=O C(=O)(C(C)CO)N(C(C)CNC(=O)CCNc1ccncc1)CC C1(N(C)C(C)=O)(CC)CN(C(c2cccc(N3CCNC3=O)c2C)=O)CCC1O N1(C(c2cnc(CNC(Cc3n(C)ncc3)=O)nc2)=O)CC(C2CCCC2)C1 N1(C(CC(C(C)C)OCC)=O)CCN(C(=O)C(C)CC(C)(F)F)CC12CCC2 C12(C(N(C)CC3CCN(C(C4CN5CCN4CC5)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 Cc1nnc2n1CC(C(N)=O)N(N(C(=O)CSc1ccncc1)C)C2 C1(C(N2CC(SC)C(NC(C3CCOC3)=O)C2)=O)CCN(CP(C)(C)=O)CC1 N1(C(c2cccc(NCCC)c2)=O)CCC(C)C(CNC(C2(COC)CC2)=O)C1 C(=O)(C1=C(c2ccccc2)CCCC1)NCC(CO)N(C)CC1CC1 c1(CC)cccnc1C(=O)NC1CCCCC1CNC(=O)C(O)C1CCC1 C1(CNC(C(C)C2CCC2)=O)CN(C)CCN1C(=O)CC1CCC(C)(C)CC1 C1(CC(=O)NC2CCCCCC2CO)C2CCC(C2)N1C(c1ccn(CCF)n1)=O c1(C(N2CCOCC2)=O)cc(S(=O)(=O)Nc2cccnc2O)ccc1Cl C1(NC(C(CSC)O)=O)CCC12CN(C(=O)C(c1ccc(F)c(C)c1)=O)C2 N1(C(C(CC)NC(C)=O)=O)CC2(CC(NC(=O)CC3CC3)C2)C1 C=CCC(CC)C(=O)NC1CCN(C(c2snc(Cl)c2Cl)=O)C1CC N1(C(c2c(CC)nc[nH]2)=O)CCC(C2CCN(C(c3cn[nH]c3)=O)CC2)CC1 c1(C(N(CCCNC(C#CC(C)C)=O)CCO)=O)cc(=O)c2ccccc2o1 C#Cc1c[nH]nc1C(=O)NC(c1ccc(C(C)C)cc1)CNC(=O)C(CCC)OC Cc1cc(CNC(c2cccc(C)n2)c2nnnn2C2CC2)cc(Cl)n1 C1(CC)CCN(C(C2(CNC(=O)CNc3ccccn3)CCC2)=O)C1 N1(C(C(CC)F)=O)CCCC(CCCCNC(=O)C(=O)NCCOC)C1 c1(-c2scc(C)n2)nc(CN2CC=CC2)n(CCC(F)(F)F)n1 CN1CCCC(C(=O)NCC2(NC(=O)CCOC3CC3)CCCC2)C1 S(=O)(=O)(c1ccc(F)c(Cl)c1)C(=O)NCCCN(C)C(C1C2CC2C2CC12)=O S(=O)(=O)(c1c[nH]c(=NCCC2CC3C=CC2C3)cc1C)CCN1S(=O)(=O)CCC1 C1(N(C(c2c(C)[nH]c(-c3nn[nH]n3)c2)=O)C2CC2)CCC2(CCCCC2)CC1 c1(CN2CC(C)(CNC(C(C)C[SH](C)C)=O)C2)ccc(Br)nc1 C(=O)(N=c1[nH][nH]cc1I)C1N(Cc2cccc(OC)n2)CCC1 c1(C(=O)OCC)c(C)c(S(=O)(=O)NCCCc2cncc(F)c2)c(C)n1C Cc1nn(C)c(C)c1C(=O)NCC1(F)CN(C(c2cc(-c3ccns3)on2)=O)C1 N1(C(c2n(C=C)nnc2)=O)CCC(NC(=O)C(C(C)(C)C)NC(C)=O)C(CC)C1 C1(CC(=O)Nc2c(C)nsc2)C2CN(C(=O)CC3CCN(C)CC3)CC12 N1(C(C(C)SC)=O)CC2(COC(CNC(=O)CS(N)(=O)=O)C2)C1 c1(C(N2CCCC(NC(c3c(C)cns3)=O)C2C)=O)ccnc2c(F)cccc12 C1(CNC(C2C(NC(c3n(CC)nc(C)c3)=O)CC=CC2)=O)CN(C)CCN1C CC(O)C(F)(F)C(=O)NCC1CN(C(=O)C(O)C(C)(C)C)CCCO1 c1(C(C)=O)cc(C(=O)NC2CC(C)(NC(c3cn[nH]c3)=O)C2)c(C)o1 c1(N2CC(OC)CC(OC)C2)nc2c(c(=NCCC(C)N3CCCC3)[nH]1)CCC2 S(=O)(=O)(c1cccc([N+](=O)[O-])c1)N(C(C1C(c2c(C)ccc(Br)c2)C1)=O)C(C)C Cc1cnc2cc(-c3nc(Cc4ccccc4F)nn3CC3CC3C)ccn12 CC1CC(C(=O)NC2CN(C(=O)C(F)(F)c3cnn(C)c3)C2)CC(C)O1 c1(CNC(c2nc(C(=O)NC(c3nn[nH]n3)CC)sc2)=O)cc(C)nn1C Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC(C1CCOC1)NC(=O)C(F)=CCCF c1(N2CCN(c3ccc(C)cc3C)CC2)nccc(=NCC(F)c2ccccc2)[nH]1 c1(CC(=O)NCC2N(C(Cc3cc(CC)no3)=O)CC2)cccc(OC)c1Cl C=CCC(C)(C)C(=O)NCCOC1CCN(C(=O)CN2CCN(C3CC3)C2=O)C1 Cn1ncc(C(N2CC(NC(=O)CNC(c3ccsc3)=O)C2)=O)n1 C1(C(N2CCC(NC(CCc3cc(C)on3)=O)CC2C)=O)CCCC2C1C2(F)F c1(C(=O)NCC(C)N(C(CC2(CCC#C)OCCO2)=O)C)cccnc1C1CC1 C1(C(=O)NC2(CCC(=O)Nc3c(C)noc3C(C)C)CCC2)NC(=O)OC1(C)C C1(CC(=O)NCCNC(c2c(O)nc(C)c(Br)c2)=O)CCc2cnn(C)c2C1 c1(NC2(CNC(CCCC)=O)CCOCC2)ncnc2c(OC)cccc12 C1(CN(C(=O)C2CC2)CC)CCCCN1C(=O)CCCOC.C(=O)C(C)N1CCC1 Cc1nc(CNC(=O)CN(C)C(C2CCC=CCC2)=O)oc1C c12cccc(C)c1CNC(NC1CC1c1ccc(C)s1)=NC2.C1(OCC)CC1 FC1COc2ccccc2C1NCc1csc(I)n1 c1(CN(C(CN2CCC(C)(OC)C2)=O)C)ccc(C(F)(F)F)cc1C C1(CCNC(CCOC)=O)(C(=O)NCC2(N(C)C)CCCC2)CCCC1 C1(CCNC(C(C)C)=O)CC(F)(F)CN1C(=O)C=Cc1ccnn1C C(=O)(CCC(C)(F)F)NCC1C(C)(C)C1C(=O)NCC1CC(O)C12CCC2 C1(NC(c2n(CCC)nnn2)c2ccncc2)CC(=O)N(CCOCC)C1 C(=O)(C(C)(C)C(C)(C)O)N1C(CNC(CNC(CCC)=O)=O)CCC1 c1(N(CC(C)C)CCc2scc(C)c2)cnc2[nH]c(C(F)(F)F)nc2c1 c1(NC(N2C(C)COCC2)=O)ccc(Br)c2cccnc12 S(=O)(=O)(CCCOc1cccc(C(F)(F)F)c1)NCC(=O)OC C(=O)(C(C)(C)CC(=O)OC)N1CCC(C(N(C2CCNC2)CC)=O)(CC)C1.OC c1(C(N2CC(NC(C(c3ccccc3)C)=O)C(C)C2)=O)cc(Cl)nc(Cl)c1 c1(OC)ccc2nccc(C(=O)NC3(CO)CCN(C(c4cocn4)=O)C3)c2n1 C1(NC(CCP(C)(C)=O)=O)CCSC12CN(C(=O)CCc1ccc(N)cn1)C2 c1(C(=O)NC2CC(C)(NC(=O)CCCN3CCCC3)C2)cc(F)ccc1Cl Cc1cc(C(=O)NCC2(C)CN(C(=O)C(N)=O)C(C)(C)C2)c2c(O)nn(C)c2n1 c1(OC)ccc(O)cc1C(=O)NC1(CNC(C2CCN(CC(F)F)CC2)=O)CC1 c1(C(N(C2CCN(C(CC=CC=C)=O)CC2C)C)=O)ccn2cc(C)nc2c1 c1(C(N(C)CC2CCCN(C(c3ccccc3)=O)C2)=O)sc2ncccc2c1Cl Cc1cnccc1C(C)C(=O)NCC1(O)CCN(C(C2(CNC(N)=O)CC2)=O)C1 C1(C(=O)NCC2C(NC(c3c(CCC)n[nH]c3)=O)C2)CCOC2(CCC2)C1 CC(C)CC(O)CC(=O)NC1CCCCC1CC(=O)NC1CCCC1(C)C C=CC1CN(C(=O)C(C)OC(C)(C)C)CC1NC(c1cccc(C)c1Cl)=O N1(C(CC(C)SC)=O)CCN(C2CCN(C(c3ccc(C(N)=O)[nH]3)=O)CC2)CC1 C1(C(=O)O)(NC(c2ccc(F)c3ccoc23)=O)CCc2c(F)cccc21 C1(C(=O)NC(C2CCN(C(CC)=O)C2)C)CCCC(NC(=O)CC2CCCC2)C1 C1(NC(CC2(N(C(C(CC3CC3)NC(C)=O)=O)C)CC2)=O)C2CCC(C2)C1CO N1(C(c2c(C)onc2)=O)CCC(C2(NC(c3noc4ncccc34)=O)CC2)C1 C1(OC)CC(CNC(c2ncoc2CNC(C2CC(F)C(=O)N2)=O)=O)C1(C)C N(C1CCSc2c(F)cccc21)C(C(c1cccc(CC(C)C)c1)C)C c1(CC(=O)NCC2(OC)CCN(C(C(C)OCC#C)=O)C2)ccc2sccc2c1 C=Cn1nccc1C(=O)NCCCCC(C)NC(=O)C(F)CC1CCOC1 c1(OC)ccc(C(=O)NC(C)CCNC(=O)CC(=O)OC(C)(C)C)s1 CC1CCCC=C1C(=O)N1CCCC1(C)CNC(C1CCCN1C)=O CC1CC(NC(c2cncs2)=O)CCN1C(=O)C(C)N1CCCC1 C1(CC(C)C)COCC1(c1nnnn1CCCF)NCCc1ccccn1 C1(C(N(C)CCC2CCCN2C)=O)CC2CN(C(C3C=CCC3)=O)CC2C1 Cc1cc(C(=O)NC(c2cccnc2)C(=O)NC2CCCCC2(C)C)cnc1O Nc1ccnc(C(=O)NCC2CC(CNC(c3ncsc3Br)=O)CO2)c1 C1(Nc2nc3c(ccc(OC)c3)n2C)CCN(S(=O)(=O)N2CCCCC2C)CC1 C1(C(=O)NCCCOCCCNC(c2c(C)c[nH]c2)=O)CCN(C)S1(=O)=O C1(C(N2CCC(C)(CNC(C(C3CC3)OCC)=O)C2)=O)CNC(=O)CC1(C)C N(C1CCCc2nc(S(C)(=O)=O)ccc21)C(=O)NC1CCN(CC(C)O)CC1 c1(C(N2CC(C)C(C)(CO)C2)C(=O)NC2CC(F)(F)C2)ccc2c(c1)COC2(C)C c1(C(=O)NC2C(C)CN(C(=O)CS(C)(=O)=O)C2)cccc(N)c1Br c1(NC2(c3n(CC=C)nnn3)CC2(C)C)cccc2c1CCC2(C)C C(=O)(C1=NOC2(CCC2)C1)NC1C(CNC(C=CS(CC)(=O)=O)=O)CCCC1 Cc1cc(C)n2ncc(C(=O)NC3CCN(C(=O)CCOC(C)C)CC3F)c2n1 Cc1nsc(N)c1C(N1CCC(O)(C(C)NC(C2CCSCC2)=O)C1)=O N1(C(c2c(C)nc[nH]2)=O)CCC(CNC(c2cc(O)nc(O)c2)=O)C(F)(F)C1 C1(C)(CNC(CSC(C)C)=O)CCN(C(c2cc(-c3ccccc3)sn2)=O)C1 C1(c2nnnn2CCCF)(NCCc2c(C)ccnc2)CCCC(C2CC2)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCC(C(C)NC(C(C(C)C)CN(C)C)=O)CC1 C1(OCC(=O)NC)CCN(C(=NCCC2COCCO2)NCC2CCCC2)CC1 c1(C(c2nnnn2C2CC2)NC2(C)CC(=C)C2)cc2n(n1)CC(C)(C)CO2 C1(C(=O)NC2CC(CC(=O)N(C)CC3CC3(F)F)C2)(OC)CCCCC1 C1(NC(C)=O)CC2CCC1CN(C(=O)Cc1scnc1C)C2 CC1CN(C(c2ncn3ccccc23)=O)C(C)CN1C(=O)CN(CC(C)(C)C)C C1(CCC)C(C)CCCN1C(C12CC(c3ccc(Cl)cc3)(C1)C2)=O c1(CNC(c2c(NC(C)=O)cncc2)c2nnnn2C)ccc(F)cc1N(C)C C(=O)(C(C(C)(C)C)OC)N1C(C(=O)NCCC=CCCC)CC(O)C1 Cc1cc(C#N)cc(C)c1COCC(=O)NCC(C)(CO)CC(=O)O C(=O)(C1=CCC(NC(=O)CCc2cnco2)C1)NC(CC#C)CC C1(N=c2nc(C3CCCCC3)[nH]s2)(CNC(=O)C(F)n2cccn2)CCC1 Cc1ccc(C(=O)NCCC2CCC(NC(=O)C#CC3(C)CC3)C2)c(=O)n1C C#CCCCC(C)C(=O)N1CC2CC2(C(=O)NCCN2CC=CCC2)C1 c1(C(N2C(C)C(NC(=O)C=C3CCN(C)C3)CCC2)=O)cccc2c1CNC2=O C1(CNC(c2nc[nH]c2C2CC2)=O)CC(O)CN1C(=O)Cn1cc(C2CC2)cn1 C1(C(=O)NC(CC)COCC2CC2)CC(C)(C)CN1C(c1cnn2c1OCC2)=O C1(C(=O)NC(c2nc(C)on2)C)CCCCN(C(=O)Cn2ncn(C)c2=O)C1 c1(C(N(CC(CC)NC(=O)C(O)P(C)(C)=O)C)=O)ccc(O)c(C(=O)OC)c1 N1(C(CC(=O)OC)=O)CCC(C=CC(=O)NC2CCC3(CC2)N=N3)CC1 N1(C(c2csc(Br)n2)=O)CCOCC(CNC(C2(F)CCCC2)=O)C1 C1(CNC(c2c(C)con2)=O)CCN(C(=O)C(F)(F)Sc2cnn(C)c2)CC1C c1(OC)cc(C)c(C(N2CCC2CNC(=O)C2=CCOCC2)=O)c(C)c1 Cc1ccc(OCC(=O)NCC2(F)CCC(NC(=O)CSC3CC3)C2)cc1 C12(C(N3CCC(C(C)NC(=O)C(F)=C4CCCC4)C3)=O)CCC(CO)(CC1)OC2 CCC(CC)(CC)NC(=O)C(=O)NCCOCCOC.C(=O)(C(F)(F)F)N C1(C(N2CC(C(C)NC(c3ccc(C(F)F)o3)=O)C2)=O)CC(=O)CC12CCC2 c1(CN(C(=O)CCN(CCO)C(C2(CO)CCC2)=O)C)cncn1C C1(CC(=O)NCC2(NC(c3ncn(C)c3)=O)CCOC2)CCCS(=O)(=O)C1 Cc1cccc(Br)c1C(C(=O)NC1CC1(C)CO)NC(c1cc(C(N)=O)[nH]n1)=O CCC(C)(C#N)C(=O)N1CCC(CN(C(=O)C=Cc2nc(C)c(C)[nH]2)C)CC1 N1(C(c2nnc(C)s2)=O)CCCC(C)C1CCNC(c1cc(C2CCC2)no1)=O CC(C)(C)C(=O)CCC(=O)N(CCC(N1CCC(C)(C2CC2)C1)=O)CCO c1(C(=O)NC2CCC(NC(c3c(F)cc(Cl)cc3F)=O)C2)cccc2occc12 CCC(C)CCCC(=O)N(CCC(=O)NC(C)C(C)F)CCCO C1(NC(c2ncn(C)c(=O)c2)=O)CN(C(=O)CC2CC(F)C2)CC2(CC2)C1 c1(NC(C(CNC(C(C(C)C)C#N)=O)O)=O)cnc2[nH]cnc2c1 c1(C(C(=O)NCCN(C(C(F)=CCC)=O)CC(C)O)N(C)C(C)=O)ccccc1 C1(NC(N2CCn3c(Br)cnc3C2)=O)CCOC12CCS(=O)(=O)CC2 c1(CC)cc(N)c(C(=O)NC2CN(C(=O)C(O)C(F)(F)F)C(C)(C)C2)c(F)c1 Cc1cccn2ncc(C(=O)NCCCNC(C34CCC3CC4)=O)c12 c1(C(=O)NC2CC(O)(CNC(C3C(F)(F)C34CC4)=O)C2)cnc2ccccn12 N1(C(c2cncc(C(=O)OC)c2)=O)CC(C)(C)OC2COCC12 C=CC1CN(C(=O)CCCNC(C)=O)CC1NC(C1CC2(CCO1)CC2)=O c1(C(N2CC(N(C(C(CC)N(CC)CC)=O)C)C2)=O)ccc(OC)c2ccsc12 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C(C(=O)NCc2c(C)noc2C)CC(O)CC1 C1(OCCN(C(=O)COCC2CCC2)C)CCN(C(=O)CC2SC(=N)NC2=O)CC1 C1(C(=O)NCCC2(CNC(c3c(C)cn(C)c3)=O)CC2)CC2CCC1CC2 C1(OC)CCC(CC(=O)NCCCOCCNC(=O)CCc2ccsc2)C1 c1(COC)cccc(C(=O)NCC(C2CCC2)NC(C2(C(C)C)CC2)=O)c1 C(=O)(C1=C(C(C)F)N(C)C(=O)NC1c1cccc(S(N)(=O)=O)c1)Nc1cc(C)[nH]n1 c1(C(=O)NCCN(C(=O)C(C)(F)CC2CCCC2)C(C)C)coc2c1COC2 c1(C(CC(=O)NC2C(CNC(Cc3cnc(C)[nH]3)=O)C2)O)ccc(Cl)cc1 CC(C)CC(O)C(=O)NC1CCC(NC(=O)Cn2cnc(Br)c2)C1 N(C1CN(C(=O)CC2CCCC(=O)N2)CCc2ccccc21)C(C1(CC)CC1)=O c1(C(N2C(CN(C(COC(CC)C)=O)C)CCC2)=O)cc2ncccc2o1 c1(CC)c(Cl)nc(C2CCC2)[nH]c1=NCCN(C)C(C1CN(C)CCO1)=O c1(C(C)C)cnn(C)c1C(=O)N(C1CCN(C(c2ncccc2F)=O)C1)C C1(NC(c2c(C)csc2)=O)CCCCC1C(=O)N(C1CC1)Cc1ccccc1 N1(C(Cc2cc(C)[nH]n2)=O)CC2COCC2(C(N2CCOCC2C(C)(C)C)=O)C1 c1(OC)ccc2c(c1)N(C)CCN2C(c1ccn(C)c(=O)c1)C(=O)NCCC#N C12(CC(=O)NC3CC4C(C3)C4(F)F)CCC1CN(C(=O)C=CC(F)F)C2 c1(C(=O)NCC2CCN(C(CC(C)C(F)F)=O)CC2O)cc2c(s1)CC(C)(C)C2 Cc1ccnc(C(C)NC(=O)CCN(C(C2CN(C3CCC3)C2)=O)C(C)C)n1 CCC(C)C(O)C(C)C(=O)N1CC(C)(C)CC1CC(=O)NOC C1(CN(C(C=C)=O)CC)CCN(C(C2C(C(F)(F)F)C2[N+](=O)[O-])=O)CC1 C1(C(F)(F)F)(C(N(CC(C)NC(c2coc(C3CC3)n2)=O)C)=O)CCN(C)C1 c1(CC(=O)NC2(COC)CN(C(CCCOCCC)=O)C2)cccc(Cl)c1Cl N1(C(C(CC)OC(C)C)=O)CC2CC1(CNC(=O)CCCOc1ccccc1)C2 N1(C(C(C2CCCCC2)C)=O)CC2CCC1C2NC(=O)Cc1ccsn1 c1(SCC(=O)NC2C(CC)N(C(c3cccc(=O)o3)=O)CC2)cc(F)ccc1F N1(C(C(CC)F)=O)CC2CC(CNC(c3cccnc3N(C)C)=O)C2C1 N1(C(CCC2CCN(C(c3occc3Br)=O)CC2)=O)CCCC12CCC2 N1(C(C2(CC=C)CCCC2)=O)CC2(C(=O)Nc3ccccc3C(C)=O)CC1CO2 c1(OC)ncccc1C(=O)N(c1cc[nH]n1)CCSc1ccc(F)cc1 c1(OC)c(CNC2CC(C(=O)Nc3cnccc3C#N)C2)cccc1O CC(C)CCCCC(=O)N(C1CC(NC(=O)NC(C2CCCO2)(C)C)C1)C c1(C(=O)NCC(CNC(c2c(SC)csc2)=O)F)cnc(C)c(C)c1 c1(C(=O)NC(CN(CC)CC)C)cc(OCC(=O)OCC(F)F)ccn1 Cc1cc2ncn(CC(=O)NCCN(C)C(c3c(O)cccc3Cl)=O)c2cc1C CCCC(CCC)C(=O)N(C(C)CCNC(C1CC1(F)F)=O)C CN=c1[nH]c(=NCC2CC2Cl)[nH]c(=NC(C)Cc2nc3cc(Cl)ccc3n2C)[nH]1 C(=O)(C(F)(F)CC1CC1)N(CC)CC1CCCN1C(C1CCOC1(C)C)=O.C=O c1(C(N(CC(CN(c2ncc(C)c(O)n2)C)O)C)=O)cnc([N+](=O)[O-])cc1C c1(CN2CCOCC(NC(c3c(C)ncnc3)=O)C2)c(Cl)ccc(Cl)c1Cl c1(OC)ccc(N)c(C(N2CC(=C(F)CNC(=O)CC34CCCC3C4)C2)=O)c1 C1(CNC(c2ncc(C)nc2)=O)C(C)CCCN1C(c1n[nH]cc1C)=O c1(NC(c2c(CNC(c3c(C)c(F)cnc3)=O)cc[nH]2)=O)cccn2nccc12 n1(C(C)C(=O)NC2CCCC2NC(c2cc(O)cs2)=O)cnc2ccccc12 c1(C(=O)NC2CC3C2CCN3C(C2SC3C=CC2CC3)=O)noc2c1CCCC2 C1(CCCCC)(C(=O)NCC(CCNC(c2ccsc2)=O)OC)CCCO1 C(=O)(CC1=CCCCC1)Nc1cc(C)c(NC(=O)CC(O)CN(C)C)cc1 c1(CCC(=O)NCC(C2CCCC2)NC(C(CCC)C)=O)ccc(F)cc1F C(=O)(CC(C)(C)C#N)N1C(C(N2CCC2CC(C)(C)C)=O)(COC)C=CC1 C1(NC(Cc2cc(C)ncc2)=O)CCN(C(C2(n3cccn3)CC2)=O)C(C)C1 N1(C(=O)CC2CCCCN2C(C2CC(=C3CC3)C2)=O)C2C=CCC1CC2 S1(=O)(=O)c2ccc(Br)cc2NCC(OC)CN1.C1(CO)CCN2CCCC12 C(CC(C(=O)N(C1CCOCC1C)C)NC(=O)CCN(C)C)OC C(=O)(CC#N)NC(CNC(CSCCC)=O)C1CCC1 c1(OC)nsc(OC)c1C(=O)NC(C1CN(C(=O)CCOC2CC2)CCO1)C c1(C(N2CCC(CC(=O)Nc3cnoc3)C2)=O)c(F)cncc1Br C(=O)(C(=O)N=S(C)(C)=O)NCC1(COC)CN(C(=O)CCc2csc(C)n2)C1 c1(N2CCC(=O)NC(=O)C2)nc(NCC2CC3(CCC3)CO2)c2ncsc2n1 c1(C(=O)NCC2C(NC(C(CC)(C)O)=O)CC2)cc2cc(Cl)ccc2[nH]1 N1(C(c2ccc(Cl)o2)=O)CC(NC(C2(C(c3ccccc3)=O)CC2)=O)C2CC12 c1(CN(C(CC)C(C)C)CCOC)c(C)nn(Cc2ccccc2Br)c1C C1(CC(=O)NCCc2ccc(Br)cc2)COCCN1C(C1CCCC(O)C1)=O C1(NC(C2CCN(C(C=C(CC)CC)=O)C2C)=O)CN(C)C(=O)C12CC2 C1(NC(C=CSC)=O)CC2(CCN(C(=O)CC3CC4(CCCC4)CO3)CC2)C1 N1(C(c2c(C)cn(C(C)C)c2)=O)CC2CCCC2(CNC(c2c[nH]c(=N)s2)=O)C1 c1(C(N(CCNC(Cn2ccc(C)n2)=O)C)=O)ccc(F)c(F)c1C N1(C(C2(OCC)CCCCCC2)=O)CC2CN(C(=O)C(F)=C(C)C3CC3)CC2C1 c1(CC(N2CC(CNC(=O)C(O)C3CC3)OCC2)=O)ccc(F)cc1C(F)(F)F C(C(CC)CC(F)(F)F)NC(c1n(CCCCCC)nnn1)C1CCOCC1 Cc1cc(N)cnc1C(N1CCC(C(=O)NCC2(C)CCCC(=O)N2)C12CC2)=O N1(CC)CC(C(=O)NCC(C)C(=O)NC2(C)CCSC2)CC1=O c1(C(=O)NC(CC(C)NC(c2[nH]cc(C(=O)OC)c2)=O)C)c(F)cc(C)cc1F C1(C(=O)NCCN(C(C2CC2C2CCC2)=O)CC)CCCCC1(C)C c1(C(C)(C)C)cc(C(N2CCC(N3CCOC3=O)C2)C(=O)NCCCF)on1 n1(CC(N2CCN(C(c3nccc(C)c3)=O)CC2)=O)cnc2c1CCCC2 C1(C(=O)NCC2(CC)CCCN2C(=O)OC(C)(C)C)CCCCN1N=O c1(CC(=O)NC2CN(C(C(CC3CC3)SC)=O)C2)cn2ccccc2n1 S(=O)(=O)(c1c(C)o[nH]c1=N)NCc1c(C)cn(CC)n1 N1(C(=O)NC2(OC)CCCC(C)(C)C2)CC23CCCC2(C1)CN(C)C3 c1(CNC(C2CCCN(C(c3c(OC)nccc3)=O)C2)=O)nc(C)ccc1O OC1CCCCCC1C1CCN(c2nnc(-c3cncs3)n2CC2CC2)C1 Cc1cccc(C(=O)NCC23CC2CN(C(=O)CSCc2ccccn2)C3)n1 c1(OC)cc(C(=O)NCCCC(C)NC(=O)CNC(C)=O)cc(N)c1OC c1(C(=O)NC(C2CN(C(C3(c4ccccc4)CC3)=O)CCO2)C)cc(O)ncn1 c1(-n2cc(C3CCN(ONC(c4cc(C)ncn4)=O)C3)nn2)ccc(Cl)cc1Cl C#CC1CCCN(C(=NCCCCN2CCCC2)NCc2ccccc2)C1 C=CCCCCCC(=O)NC1CC2CCC1N2C(=O)CCc1nc(O)n[nH]1 c1(C(CN(C(C2CC(NC(COC(C)(C)C)=O)C2)=O)CCO)(C)O)ccccc1 C(=O)(C1=CC2CCCC12)NCCOC1CN(C(c2nccc(C)c2)=O)C1 c1(C(C)C)ccccc1C(=O)N(C1CN(C(C2CC2c2ccco2)=O)C1)C C(=O)(CCCCCN=[N+]=[N-])NCC1(O)CN(C(C2(N(C)C)CC(F)(F)C2)=O)C1 C(=O)(C(CCN(C)C)NC(=O)CC=C(Cl)Cl)NCCN(CCCF)C c1(NC(C(=O)NC(c2cn(CCC)nc2C)C2CC2)=O)cc(C)nc(NC)c1 C1(C(=O)NCc2snc(CC)n2)CN(C)CCN1C(=O)CCn1ccnn1 c1(N2CCC(S(=O)(=O)NCC)C2)nc(=NCc2ncoc2C)[nH]c2ncn(C)c12 N1(C(Cn2c(C(C)C)ncc2)=O)CCN(C(=O)CC2NC(=O)NC2=O)CC(C)C1 C1(C(=O)NCCCCN(C(Cc2ncc(C)o2)=O)C2CC2)CC1C1CCCCC1 Cc1nc(CCCNC(=O)CC2CCN(C(=O)Cc3sccc3C)C2)n[nH]1 Cc1cc(C(C)(C)C)ccc1C(=O)NCCCCC(C)NC(=O)Cc1ccno1 N1(C(CC=CCC)=O)CCCC1C(C)(C)NC(c1csc(C(=O)OC)c1)=O C(=O)(C(C)(C)C(=O)N(C)C)NC1CC(C(=O)NCC2C(=C)C2)C1 N1(C(C2CN(C)C2)=O)CCCC(C(=O)NCc2nccn2C)C1 c1(C(=O)NCC(C)NC(=O)C(C)C(C)O)cccc2c1CCOC2 C(c1ccc(F)c(Cl)c1)=CC(=O)NC(C1CCCC1)CNC(C(C)OCC#C)=O c1(C(C)NC(c2nnnn2C(C)(C)C)CCOC)ccccc1Br c1(CC(=O)OC(CCOC(CC)C)C(C)C)cccc(NC(C)=O)c1 C1(N(C(C(=O)NCCSC)C(C)C2CC2)C)CC2CC3CC(C2)CC1C3 c1(C(CSCC)C)cn(C2CN(C(=O)CC3CCSC3)C2)nn1 N1(C(C(CCc2cn[nH]c2)NC(C2CCCOC2)=O)=O)CCC(O)(CO)CC1 Cn1nc(C(F)(F)F)cc1CC(=O)NCC#CCNC(c1cc(C)on1)=O.C1CC1 c1(C(N2C3C(NC(C(C)OC4CCCC4)=O)C(C3)C2)=O)ccc2ncccc2n1 N1(C(c2scc(OC)c2)=O)CCC(C#N)(NC(C2CC=CCC2)=O)C1 c1(C(C)C)ocnc1C(=O)NCC1(O)CC(NC(=O)CCc2ccon2)C1 c1(C(CNC(=O)CN(C2CCC2)C)NC(CC(OC)OCC)=O)cccc(F)c1 N#Cc1ccc(F)c(NC(=O)CC2CCCC(NC(=O)CC=C(Cl)Cl)C2)c1 C1(NC(COCCCC#C)=O)CN(C(c2ccc(N)c(SC)c2)=O)CCC1CO N1(C(c2c(C(=O)OCC)ocn2)C(=O)NCc2cccs2)CCCSCC1C C1(NC(c2ncccc2F)=O)CN(C(C2CC3CCC(C2)C3)=O)CC12CCCC2 c1(NC(C2CC(c3cccc(F)c3)C2)=O)nnc2n1CCNC2 C1(CC)CCCCC1NC(=NC)NC1CCN(c2cccc(N(C)C)n2)C1 c1(C(=O)NC(C2CCN(C(c3ncc(OC)nc3)=O)C2)C)cccc(C#N)c1 C1(CNC(c2c(CC)ccc(C)c2)=O)COCC2(CCN(C(=O)C(C)C)C2)O1 C1(CC(F)(F)F)(OC(C)=O)CC(N)(C(=O)N(C)Cc2cccc(C(F)(F)F)c2)C1 Cc1nncn1NC(=O)C(C)C1CCN(C(=O)C(N)=O)C1 C1(C(=O)NC(CC=CC)C(=O)N2CCC(CC(C)C)CC2)CC2(CCC2O)C1 c1(CC(=O)NCC2N(C(COCCCC)=O)CCC2C)c(Cl)cccc1Cl CC1CC2CC(C(=O)OCc3cc(C(F)(F)F)ccc3Cl)(C2)O1 C#Cc1ccc(C(=O)NCC(F)CNC(c2cc(C)ccc2Br)=O)cc1C c1(CC)oc(C(=O)NCC2(CC(=O)NCC3C4CCCC34)CC2)cc1C c1(C(N2CC(C)(NC(C(C)OCc3ccccn3)=O)C2)=O)cc(F)c(O)c(F)c1 CC1(C)CC(CNC(C2CC(C)(O)C2)=O)N(C(c2coc(Cl)c2)=O)C1 c1(OCC(C(c2n(CC)nnn2)NCCCOCC(F)F)C)ccc(Cl)cc1Cl Nc1c(C(=O)NC2CCC(NC(c3ccnc4[nH]ncc34)=O)C2)cc(F)cc1F c1(CCC(N2CC(CN(C(CCNC(=O)OC)=O)C)C2)=O)ccc(CO)cc1F C(CC1=CCN(C(c2cc(Br)cc(F)c2F)=O)CC1)NC(C(C(C)O)C)=O C1(C(=O)NCC2C(NC(=O)CCCC(F)(F)F)CC2)CCc2nnc(O)cc2C1 C1(C(N2C(CC)C(O)CC2)=O)CC(C)CN(C(c2ccc(C#N)s2)=O)C1 Cc1nc2cc(CNC3CC3C(=O)Nc3nc(Br)cnc3Cl)ccc2s1 C1(C(C(=O)N(CC(C)NC(=O)CSCC(F)(F)F)C)O)CCC(C(C)(C)C)CC1 c1(C(=O)NC2C(CNC(c3c(CC)non3)=O)C2)c(N)cc(C)cc1F C1(C(=O)NCc2c(F)ccc(C)n2)N(C(=O)CC(C)C(C)C)CCCC1(C)C C1(C2CC2)(CNC(C2C(CC)OCC2)=O)CCN(C(=O)Cc2ccncc2Cl)C1 c1(NC(CNC(C(CCC)CCC)=O)C2CC2)ncnc2cc(C)[nH]c12 CN1C(=O)CCC1CC(=O)NCC(C)(C)NC(=O)CCN1CCCCC1=O C12(CN(C(=O)C(c3cn(C)nn3)NC(C3CC4(CSC4)C3)=O)C)CCC(C1)C(=O)N2 c1(N(CCC)CC)ccc(C(=O)NC2CC2NC(c2ncccc2O)=O)cc1 c1(C(=O)NCC(CC(=O)N(C)Cc2ccc(O)cc2)OC)cccc(F)c1C C1(NC(C(C)N2CCC2)=O)CN(C(c2ccnc(C(C)(C)C)c2)=O)C(C)(C)C1 c1(N2C(c3ccccc3)CCC(C)C2)ccc2c([N+](=O)[O-])cccc2n1 O=S(=O)(c1ccc(O)cc1)N1CC2(CN(Cc3ncc(-c4ccccc4)[nH]3)C2)C1 c1(C(C)CC(=O)NCC(O)COC(F)(F)F)cccc2ccccc12 c1(CCC)nnc(S)n1CC(=O)N(CC(C)NC(=O)C(C)Cn1ccc(C)n1)C C1(NC(NC(CC)CC)=NCCSC(F)(F)F)COc2c(C)cccc2C1 C12(CNC(C(C)(C3CCC3)NC(=O)COCCCF)=O)CCC(CC1O)C2 c1(OC)cc(N2CCC(C(C)NC(c3ccc(C(N)=O)cc3)=O)C2)ncn1 Cc1ccc(-n2cc(C(N3CC(NC(=O)OC(C)(C)C)C(C)C3)=O)nn2)cc1 CC(CCCCN=c1ccn2nccc2[nH]1)NC(=O)CSCC(N)=O C1(O)(CC(=O)NCC2CCN(CCCO)C2)CCCN(C(=O)CCC2CC2)C1 C1(CC(=O)NCCNC(c2cccc(CC3CCC3)c2)=O)CCC2CC2C1 C1(CC(C)C)(C(N2CCC(OCCNC(=O)CNC(N)=O)C2)=O)CCNC1=O c1(NC(N(C2CCCCCC2(C)C)C)=O)nccn2c(I)ccc12 C(=O)(C1=NOC(C)C1)N1CCCC(CCCCNC(c2c(C)nc(C)o2)=O)C1 CN1CCC(CC(=O)NCC2CC(NC(c3ccco3)=O)C2)C1=O Cc1ccnc(NC(=O)C(=O)NC(C(C)C)C(O)c2ccsc2)c1Br Cc1cc(Br)cc(F)c1C(N1CC2CN(C(c3cncc(O)c3)=O)C2C1)=O S(=O)(=O)(c1cc(C(F)(F)F)cs1)NC(CCOC(C)C)Cc1ccco1 N1(C(C(C)O)=O)CCC(O)(C(C)NC(=O)C(C(C)(C)C)SC(OC)CCl)CC1 c1(NC(C2SCCN(Cc3c(C#C)cccc3)C2)=O)c(C)cc(F)cc1[N+](=O)[O-] c1(C(N2CCN(C(CC(CC)CC)=O)CC2C)=O)ccc(S(=O)(=O)N(C)C)cn1 C1(NC(c2ccc(C(CC)C)cc2)=O)CC2CN(C(=O)C=CC3CC3)CC2C1 c1(C(N(C)CC2N(C(C(CSC)C)=O)CCCC2)=O)cc(C)cc(N)c1 C(=O)(CCCC(=O)N1CC(NC(=O)Cc2ccccc2)C2CC12)OCC N(C1CCc2cc(OC)ccc21)C(c1ccc(C=CC(=O)OC)cc1)=O N1(C(C(C)Oc2ccccc2)=O)C2CCCC1CN(C(c1ccsc1C#N)=O)C2 N1(C(c2n(C)cnc2)=O)CCN(C(C2C=CCCC2)=O)C(CO)C1 C#CCC(CC(F)F)NC(=O)CC1CCC(NC(c2ccc(CC)[nH]2)=O)C1 C1(CC)CCN(C(=O)C(C)N2CC(C)C2)C1C(=O)NC(CO)C(F)(F)F CC1(C)CN(C(c2n[nH]c(O)n2)=O)CCC1NC(=O)CC1CCC(C)CO1 c1(C(N(C2CCN(C(C(C)OCC)=O)C2)C)=O)ccc(S(=O)(=O)C2CC2)cc1 N1(C(c2n(C)ccc2)=O)CCN(C(=O)CCc2ccc(Cl)c(Cl)c2)C(CC#N)C1 CCC(CC)CC(F)C(=O)N1CC2(CCCC2NC(c2cc[nH]c(=N)n2)=O)C1 N1(C(=O)Nc2nc(F)ccc2Br)CCOCC1C1CCCO1 n1(CC)c(C)cc(C(=O)NC(C(C)NC(=O)CCS(N)(=O)=O)C(C)C)c1C C(=O)C1=CCCOCC1.N1CCOCC1C(N1CCC(N(C(C)=O)C)CC1)=O C(=O)(C1=COCCC1)N1C(C)CC(CNC(c2ccc(OC(C)(C)C)cn2)=O)C1 N1(C(COC)=O)CC2CCC2(CCNC(=O)CCP(C)(C)=O)C1 C(=O)C(C(C)CC)N(C)C.C(=O)(CC(C)(C)N(C)C)N(CC(CC)NC(C)=O)C C12(NC(C(CC=C)C)=O)CCCC1N(C(c1cc(C3(C)CC3)on1)=O)CCC2 C(=O)(CCC1=CCCCC1)N1CC(OC2CCN(C(c3c(SC)ccs3)=O)C2)C1 c1(C(=O)NC(C2CCCN2C(=O)C(c2ccccc2)F)C)cscc1Br N1(C(C(C)(C)OCC)=O)CCCN(C(=O)CCc2scnc2C)C(C)C1 C1(NC(C(C)c2ccsc2)=O)CCCC12CCN(C(=O)C=C(Cl)Cl)CC2 C1(CNC(C(C2CCOC2)OC)=O)CN(C(=O)CC(C)C(C)C)CC(C)(C)O1 C1(C(=O)NCCCNC(=O)C=CCN2CCOCC2)CCC(F)(F)C1 N1(C(Cc2cc(C)sc2)=O)CCC(CNC(c2ccc(N)cn2)=O)C(O)C1 C(=O)(C(C)CCCC(C)=O)NCCOC(CNC(C(C)OCCC=C)=O)(C)C N1(C(=O)NCc2cc(OCC3CC3)ccn2)CCc2nccnc2C1 CCC(C)CC(=O)NCC(C1CC1)N(C(=O)CCC(=O)N(C)C(C)C)C N1(C(C(F)=CCC)=O)CCOCC(NC(=O)CC2(C#N)CCOCC2)C1 C1(NC(COC)=O)CCCCC1CNC(C12CC(CO1)C2)=O.c12csc(n1)CC2 c1(C(N2C(C(=O)NC(c3ccc(F)cc3)C)CC3CC32)=O)cnc2ncccn12 C(C(=O)N1CCC(C(N2CC(N(C)C)C(C)C2)=O)O1)c1c(CC)cccn1 c1(N(CCC2CCN(C(c3c(C)cns3)=O)CC2)C)cc(=O)n2ccccc2n1 C1(C(=O)NCC(C(C)(C)C)NC(Cc2nn(C)c(Cl)c2)=O)CC2CCC(C1)O2 c1(C(=O)NCC2(F)CC(NC(CCC)=O)C2)ccc2c(c1)OCCCO2 C1(OC)CCC12CC(C(=O)NC1(CNC(=O)C=C(C)C(F)F)CCC1)C2 CC(C)(CC(=O)NCC1CC1NC(C1CNC(=O)N1)=O)C(F)(F)F Cc1cc(C(=O)OCc2ccn(C3CCCC3)n2)nn1C(C)(C)C C1(NC(CC2C(C(=O)OC)CC2)=O)CCS(=O)C1 c1(C(N2C(CC)C(C(=O)N(CC(O)CO)C)CC2)=O)ccc2occc2c1 c1(C(=O)NCCCN(C(CC2CC(=C)C2)=O)C2CC2)cccc(C2OCCO2)c1 N1(C(C=COCC)=O)CCC2(CCCN(C(=O)C(C)C(CC)CC)C2)CC1 c1(CC)nc2ccc(NC(=O)CN(c3ccc([N+](=O)[O-])cc3F)C(N)=O)cc2s1 Nc1c(C(=O)NCC2CC(NC(C3(F)CC4(CCC4)C3)=O)C2)cccc1[N+](=O)[O-] c1(C(=O)OC)cnc(Cl)nc1N1CCC(NC(C23CCCN(CC2)C3)=O)C(F)C1 N1(C(C=Cc2cc(C)no2)=O)CC(CC(=O)NCC(C)(C)C(C)C)CC1(C)C CC(C)C(O)C(F)(F)C(=O)N(CC(CO)(CO)NC(=O)C=Cc1cccnc1)C C(=O)(CCCN=[N+]=[N-])NCC1C(CNC(C2N(C)CCC2)=O)C1 c1(SC)cc(C(=O)NC2(CO)CCN(C(=O)CC3CC(F)C3)C2)oc1C C1(NC(C(C2CCC2)OCC)=O)CC2C(NC(c3cc[nH]n3)=O)C2C1 C1(CNC(C(COC)(C)O)=O)CC2CCC(C1)N2C(c1cc(C(C)=O)oc1C)=O c1(CNC(CC2N(C(c3nc(C)n(C)c3)=O)CCCC2)=O)cccc(F)c1O C1(C(N2CCCCC(NC(Cc3nc(C)sc3)=O)C2)=O)CCc2ncncc2C1 c1(NCCSCCOCC)nc[nH]c(=NCC2(OC)CCCOC2)c1C N1(C(c2c(C)nc(C3CC3)o2)=O)CCC(F)(CNC(c2cscc2F)=O)CC1 c1(C2N(C(C(=O)NC(CCC)C)=O)CCC2)ccc(C)nc1 N1(C(C2CCC(NC(c3c(C)cc(F)s3)=O)CC2)=O)CCC2(C1)CN(C)C2 c1(C(N2CCC(CC=C)(NC(=O)C(F)C(C)C)C2)=O)cccc2c1CCC2 N1(C(C(C)C2CCCO2)=O)CC(F)CC1CNC(=O)CC1CCC(=O)N1 c1(CNC(C(C)(C)c2ccns2)=O)cc(Br)c(Cl)c(Br)c1 CCC(CNC(c1nnsc1C)=O)(CC)C(=O)Nc1ccc2nonc2c1 c1(CN(C(CC(C)N(C)C)=O)Cc2ccsc2)ccc(Br)cc1 CC1COC(CNC(=O)CCOc2ccccc2)C1 c1(N(c2ccccc2)C)nccc(NC(N2CC3C(CN=[N+]=[N-])C3C2)=O)n1 c1(NCc2cn(C)nc2O)ccc2c(c1)CCC2(C)C c1(C(=O)NC(C)CNC(c2ncnc3sccc23)=O)cnc(O)c2ncccc12 C(=O)(CCCC(C)O)NCC1C(NC(c2c(C)nc(CC)o2)=O)CCC1 Cc1ccc(C(=O)NCC2(O)CCN(C(=O)CC3OCCC3(C)C)CC2)c(C)c1 N1(C(C(OC)OC)=O)C2CCC1C(F)C(NC(C1(CC(N)=O)CCCCC1)=O)C2 c1(OC)ccc2nc(C)c(C(=O)NC(C)CCF)cc2c1 C(N=c1[nH]nc(C(C)(C)C)o1)C1CC(NC(C(C)n2cncn2)=O)C1 C1(C(=O)NCCOC(C)=O)CCN(C(=O)CC2(C)CCOCC2)C1C(C)C c1(CNc2c(C)nc(-c3ccc(F)cc3Cl)s2)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC(CO)NC(C(C(C)C)C)=O)ccc2c(c1)CCCCN2 c1(C(=O)NCC2N(C(C(CCC)(C)CC)=O)CC2)c(OC)c(Cl)cc(O)c1Cl C1(SC)CCCCN1C(=O)CC1CC(C)=NO1.C1(=O)CCCN1.C(C)(=O)O Cc1cc(O)nc(C)c1C(=O)NC1CN(C(=O)CC(C)(C)CN(C)C)C(C)(C)C1 C1(NC(C(C)CN(C)C)=O)CN(C(=O)CSc2ccc(F)cc2)C2(CCCC2)C1 C1(CC(N2CC(NC(CCOCC#C)=O)(COC)C2)=O)CCC(C)CO1 c1(C(=O)NCC=CCNC(C(C)(C)COCC(F)F)=O)cc2n(n1)CCCC2O C1(CCNC(c2ccc(C3CC3)s2)=O)CC(F)(F)CN1C(C1C2CCCOC12)=O N1(C(c2c(C)nc(CC(F)(F)F)s2)=O)CCN(C(c2c(Cl)cnn2C)=O)C(C)C1 c1(NC(C2CC(O)CN2C(c2cc(Br)nc(Br)c2)=O)=O)cccc(F)c1OC(F)F O(NC(=O)CCNC(=O)NCCC(=O)C1OCCO1)CCCOC c1(N2CCCN(C(C3CCCS3)=O)CC2)ncc2c(n1)CCC2 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(C3CCCO3)C3CC3)C2)ncn1 c1(C(=O)NC2(C)CC(NC(C(C)O)=O)C2)cc2sc(F)cc2[nH]1 c1(C(N2C(C3(O)CN(C(C(C)C)=O)C3)CCC2)=O)ccc(N)c(N)n1 c1(C(N(CC(c2ccccc2)C)C2CC2c2ccsc2)=O)ncc(F)cn1 c1(CNC(Cc2ccc(C)s2)=O)ccccc1CNC(C1C=CCC1)=O C(=O)(C(C)C(F)(F)F)N(CC1CCN(C(c2cnc(CC)s2)=O)CC1)CC C=C(C)C(CC(=O)NC(COC)C(=O)Nc1cccc(CO)c1)OCC C1(C(=O)NCCC2C(C)C2)CN(C)CCN1C(=O)CC1(C)CC1 c1(C(=O)NCC2CCCN(C(C)=O)C2)cccc(N)c1O.c12c[nH]c(C)c1N2 c1(SCC(C)C)cn(CC(C)NC(=O)C(C)c2ccsn2)nn1 c1(C(=O)OC)nc(N2CC3CN(C(c4cc(Cl)ccn4)=O)CC3C2)c(F)c(Cl)n1 C1(NC(C(=O)NCC)=O)CN(C(=O)Cn2nnnc2C)CC12CCOCC2 N12CCc3cc(ccc31)CN(C1CC1)C2=O.C1(c2nn[nH]n2)(C(C)(F)F)CC(F)(F)C1 n1(CC)nc(C)cc1C(N1CCC(C)C1C(=O)N(C)CCn1cc(C)cn1)=O CCC(C)(C)C(C)CC(=O)N1CCC(F)(CNC(=O)CCC2CCCCO2)CC1 Cc1cc(CNC(c2cc(CNC(=O)C(C)n3ccnn3)no2)=O)nc(C)c1 c1(CC)ccc(C(=O)NCC2CN(C(=O)C3=CCCCC3)CC2C)c(O)c1 CCC(CC(F)F)C(=O)NCC1CN(C(=O)CSS(C)(=O)=O)CCC1C c1(C(N(CC(CC)NC(c2cc(OC)n[nH]2)=O)C)=O)ncccc1CSC CC1(C)C(CNC(=O)CC2CC3CC3C2)CCN1C(=O)CCCNC(N)=O c1(C(N)=O)ccc(C(=O)NCCNc2ccc(C(c3ccccc3)=O)cn2)cc1 C(CN=[N+]=[N-])(C(=O)N(C)Cc1c(C)noc1C)NC(c1ccc(OC)s1)=O CN1CCN(C(=O)Cc2cscn2)C(CNC(=O)COC2CCCOC2)C1 c1(-c2cn(CCC)nc2)ncn2c1CN(C(c1cc(Cl)c(C)c(Cl)c1)=O)CC2 C1(NC(C2CC(OCC)C2)=O)CN(C(c2cc(C)n(C)c2)=O)CC1N=[N+]=[N-] C(=O)(CC(CCC)CCC)N1C(CNC(C(C=C)C)=O)C2CCC1C2 CC(C)C(C(=O)OC(C)(C)C)C(=O)NCC(C)NC(c1cc2n(c1)CCSC2)=O C1(C(=O)NCC(CNC(=O)C=Cc2cnc[nH]2)OC)CCCCC1 C(C(C)(C)CC(=O)NC1(CNC(=O)CC(=O)NC)CC1)NC(C(CNC(C)=O)F)=O CC(C(F)C(=O)NC1CCN(c2cncc(Cl)n2)CCC1CO)C(F)(F)F c1(CC(=O)NC2CCN(C(=O)C(F)(F)c3cscn3)CC2O)ncc(F)cc1F c1(C(=O)NC(CC=C)CNC(=O)CCCn2ccnc2)cnn(CCC)c1Cl c1(C(=O)NC2CC3CN(C(CC(=C)C)=O)CC2C3)ccc2c(c1)CCCS2 C(CCCCC(=O)NCC1CC12CCOCC2)N(C(C1C(C(C)C)OCC1)=O)C N1(Cc2c(C)cc(F)cc2)CCC2CC(C(=O)NCC(O)CO)C2C1 c1(CC(C)Nc2ccnc(NCc3ccc(OC)cc3)n2)nc2ccccc2s1 c1(C(N2CC(NC(CC(CC)CN(C)C)=O)(CO)C2)=O)cc2ncc(C)cn2n1 c1(CC)n[nH]c2cccc(-c3cccnc3OC)c12.C12(C(=O)O)COCCN1C2 N1(CCc2cn(CC)nc2)CCC(NC(=O)Cn2cc(Cl)cn2)CC1C N1(C(c2cncc(OC)c2)=O)CC2CCCCC2(CNC(=O)Cc2nc[nH]n2)C1 Cc1cccc(-n2cc(C(C)(O)C(=O)O)nn2)c1Br.c1(N2C(=O)C2)ccccc1 C(=O)(C(C)(F)C(C)(C)F)NC(C(C)C)C(=O)NC1(C)CCCCCC1 N1(C(=O)Cn2cc(-c3ccccc3Br)nn2)CCN2CCOCC2C1 N1(C(CC(=O)NCC#C)=O)C2CCCC1CC(CNC(=O)C1=NOC(C)(C)C1)C2 c1(C(=O)NC2(CCNC(C(C)(C3CC3)OC)=O)CC2)ccc2c(c1)CC2 C1(c2ccc(CC)o2)CCCCCN1C(=O)C(c1cscc1Br)F CCC(C)C(O)C(C)C(=O)NCCc1cc(C(N2CC(C)CCC23CC3)=O)no1 C(=O)(C(C)C(C)c1ccc(F)cc1)N1CC(COC)(NC(=O)CC(C)OC)C1 CC1C=C(C(=O)NCC2CCC(NC(=O)CCn3cncn3)C2)C1 C1(C(C)C)CN(C(c2cnco2)=O)CCC1NC(c1ccn(CCN(C)C)n1)=O CC(CN(C)C)C(=O)NCCSCc1cn(C2CCCC2)nn1 CC(C)C(C)(CN=c1[nH]ncs1)NC(c1ncc(C(C)(C)O)cn1)=O C1(NC(CCCC#C)=O)CCC2CN(C(c3cc4ccoc4cc3F)=O)CC2C1 N1(C(CC2(C)CC2)=O)CCN(C(c2cc(Cl)cc3c2OCC3)=O)C2COCC12 N1(C(C(C)CC2CCCCC2)=O)CCN(C(=O)Cc2cncnc2)CC12CC2 c1(OC(C)C)nccc(NC(CCNC(C2CC(CN(C)C)C2)=O)C(C)C)n1 c1(NCC(=O)COC2CCCCC2)ncc(O)cn1.C12CN(CCO1)C2 c1(N2C(C)C(C(=O)OC(C)(C)C)CCC2)nc2ncc(Br)cc2o1 N1(C(CC(C)(C)N(C)C)=O)CC2(CCOCC2)C1c1cn(-c2cnnn2C)nn1 C1(CCNC(C2(CC)CCC2)=O)COCCN1C(c1ccnc(C(C)C)n1)=O C(CN=[N+]=[N-])(C(=O)N1CCCC(F)(F)C1)NC(CSC)=O c1(C(N2CC(NC(=O)Cc3c(F)cccc3Cl)C(F)C2)=O)cc2cccnc2s1 CC1CC(NC(C2CCCO2)=O)CCN1C(c1ccc(C(F)(F)F)c(O)c1)=O C(C)(C(=O)N1CCCCO1)N(C(COC(CC)C)=O)CC1CC1 N1(C(c2cc(CNC(=O)CC3CC(F)C3)[nH]n2)=O)CCC2(CNC(=O)C2)C1 C1(C(=O)NC2(CN(C(=O)CCOc3cccc(F)c3)C)CC2)CCCC(F)C1 CCCCC(C(=O)NCC(=O)NC)NC(C1CC1c1c[nH]nc1OC(F)F)=O N1(C(c2cc(CC)nn2C)=O)CCCN(CCNC(C2NC(=O)CC2C)=O)CC1 c1(C(=O)NC2CCN(C(CC(=O)Nc3nccs3)=O)CC2)n[nH]c2c1CCC2 C(=O)(C(CC(F)F)C1CCC1)NCC1C(C)(C)C(c2ccc(N)c(Cl)n2)C1 C1(C(=O)NC2C(NC(=O)CC3(CCC=C)CC3)CC2)(NC(C)=O)CCOCC1 c1(CN(C(C)CNC(c2cc(C#N)c[nH]2)=O)C)nnc(S(C)(=O)=O)s1 c1(CC(=O)NCC(CC=C)NC(=O)C=NOC)cccc2cnccc12 C(=O)(C(C)(C)c1nncn1C)NCCC(C)N(C(=O)CCCN(C)C(C)C)C Cc1nsc(C(N2CCC(C(=O)NC3CCC4CCC34)C2)=O)c1N N1(C(C2OCCN(C(C)C)C2)=O)CC(NC(c2ccnnc2S)=O)CC(F)C1 C(C)(CCC(=O)N1CCCC1CNC(c1cnc(C2CC2)o1)=O)OC Clc1cccc2c1OCC2Nc1nccc(=NCCc2ccoc2Br)[nH]1 C1(CNC(CCCC)=O)CCCCC1NC(c1cc(CCCO)on1)=O c1(C(N(CCn2cc(CCN3CCOC3=O)nn2)CC)=O)cnc2[nH]cncc1-2 c1(NC(C)=O)c[nH]c(C)c1C(N1CCOC(CNC(=O)C=C2CCC(C)C2)C1)=O C1(C2CCC2)(C(N(C(CNC(c2cc(O)cs2)=O)C2CC2)C)=O)CC1(F)F N1(C(C(C)OCCC=C)=O)CCN(C(=O)C2CCc3c[nH]nc32)CC(C)(C)C1 CC1(NC(C2(C#N)CC2C(F)(F)F)=O)CCN(C(=O)C(c2ccccc2)O)C1 N1(C(COCCC(C)C)=O)CCC2CN(C(c3ccc4c(c3)CCN4)=O)C2C1 C1(NC(C(COC)C)=O)CCN(C(C2CC2c2ccc(C)cc2)=O)CC1 N1(C(CC(C(C)C)C)=O)CC2(CCC(CNC(C34CC(CO)(C3)C4)=O)O2)C1 c1(NC(C2CCCCN2C(=O)NC2CN(C(=O)C3CC3)C2)=O)cccc(Cl)c1 C1(NC(CCC)=O)CCN(C(=O)Cc2cc(C)nn2C)CC(C)(C)C1 c1(C(=O)NCC2(NC(C3(O)CCOCC3)=O)CC3CCC2C3)ccn2nccc2n1 N1(C(CCCCOCC)=O)CCCCC12CN(C(=O)Cc1cc(C)on1)C2 Cn1c(CCCC(N2CCOC(CNC(C3(C(N)=O)CCC3)=O)C2)=O)nnc1S N1(C(c2cc(CC)on2)=O)CCCC(N(CC(=O)NC2CCCCCC2)C)CC1 N1(C(CC(C)NC(c2cc(C)c(C#N)cc2)=O)=O)CC(C)(C)C2COCC12 C1(N=[N+]=[N-])(C(N(CCC)CCO)=O)CCN(C(=O)C(F)CC2CCOC2)C1 c1(C(=O)NCC(CNC(c2c(C)cc[nH]c2=N)=O)F)ccnc2ccc(F)cc12 S(=O)(=O)(c1cn(C2CC2)nc1C1CC1)Nc1c(COC)ncs1 N1(C(C2C(C(C)C)C2)=O)CC(CNC(=O)Cn2cc(Br)cn2)C2(CC2)C1 c1(OC)ncc(Br)c(C)c1C(N1CC2(CC(N3CCN(C(=O)C(F)F)CC3)C2)C1)=O c1(CCC(=O)NCC2COCC2NC(=O)CC(F)F)ccncc1 c1(OC)cc(-c2nc(-c3cccnc3)nn2C2CC3CCC2C3)ccc1C(=O)O N1(C(CCN(CC)CC)=O)CCC(NC(C2CCN2S(C)(=O)=O)=O)CC1C C1(C)(CNC(c2cnc(OC)nc2)=O)CCC(NC(=O)CC23CCCC2C3)CC1 c1(OCC(CN(C)C)O)cc(F)cc(F)c1.N12CC=CC(C1)NCC2=O Cc1cc(=NC2C(C)CN(C(c3ccnc(CO)c3)=O)CC2C)[nH]c(C2CC2)n1 CC(C)CS(=O)(=O)CC(=O)NC1CC1NC(c1ccc(=O)n(C)c1)=O N1(C(C(=O)NCC)=O)CCC2(NC(=O)C(F)CC(C)(C)C)CCCCCC12 N1(C(c2nc(CCC)sc2)=O)CCCCC1C1(NC(=O)C(O)CSC)CC1 N1(C(C2(CSC)CC2)=O)CC(C(N2CC(O)(CN(C)C)C2)=O)C(F)(F)C1 C(=O)(C(F)(CNC(=O)CN1CSCC1=O)C(C)C)NCCN(C(C(C)C)C)C C1(NC(c2ccc(OC)s2)=O)CC(O)CN(C(=O)Cc2nocc2C)C1 c1(C(=O)NCCCC(C)(C)NC(C(C)C(F)F)=O)cccc(O)c1[N+](=O)[O-] C=CCC(C)(C)C(=O)NCc1ncc(C(=O)O)s1 Cc1cc(C)c(C(=O)NCCC2(NC(c3ccc(C#N)cc3F)=O)CC2)c(=O)o1 C1(CCNC(C(C)SC)=O)CC(F)(F)CN1C(c1cccc(C2CC2)n1)=O N1(CC(=O)NC(CC)CN(C)C)c2ccccc2CS1(=O)=O CC1=CCC=CC1C(N1CCCC(C(=O)Nc2scc(C)c2C#N)C1)=O Cc1nc(N(CC(O)CN(C)C(c2cc(C(N)=O)ccn2)=O)C)c2c[nH]nc2n1 C1(CNC(CC(=O)OCC)=O)CN(C(c2c(Br)noc2C2CC2)=O)CCO1 Cc1nc(C(N2CCCCC2CCNC(=O)CC2COC(=O)N2)=O)c(C)s1 C1(CC(=O)N(C2CCN(C(c3ccon3)=O)CC2)CC)CC2(CCC2)CCO1 c1(CC(N2CC(F)(C(N(C3CCNC3=O)CC)=O)C2)=O)cncnc1O c1(C(=O)NCCCN(C(CC2CC(CC)OCC2)=O)C)c(C)nn(C2CC2)c1Cl c1(OC)nn(C)cc1C(N1CCCC(C(C)NC(=O)C=CC2CCCCC2)C1)=O CC1CC2CCC(C1)N2C(C1C=CCCN1C(=O)COc1occ2c1CCC2)=O N1(C(c2cn(CCNC(Cc3ncn(C)c3)=O)nn2)=O)CCCC(CCO)CC1 c1(CC)nccnc1C(=O)NCCC(O)CNC(=O)C=C1CCCCC1 Cc1cc(C(N2CC(CC(C)NC(=O)COc3ccc(F)cc3)C2)=O)nc(C)c1 c1(C(=O)NC2CN(C(=O)CCNC(N)=O)CC2F)ccc2cncc(Br)c2c1 C1(C(=O)NC2C=CCN(C(CC3(OCC)CCOCC3)=O)C2)CCCC2(CC2)C1 CC(C)CC(C)CC(=O)NCCCCCNC(c1ccc2c(c1)CCC2)=O N1(C(c2c(OC)cccc2)=O)CC(NC(=O)C(C)C(C)(F)F)C2(CC2)C1 C1(C(N2C(C(C)NC(C(C)NC(COC)=O)=O)CCC2)=O)C(C)(C)C1(C)C C#Cc1cnc(C(N2CCC(C3CC3)C2CNC(C2(C(N)=O)CC2)=O)=O)c(C)c1 CC(CC(C)(C)C)C(=O)N(CCC(=O)NC1CCN(C2CCC2)C1)CCCO N1(C(C2(C)CC2(F)Cl)=O)CCN(C(N2CCN(CC(F)F)CC2)=O)C2(CCC2)C1 N1(C(CNC(=O)CN(C(c2cn[nH]c2)=O)C2CC2)=O)CCC(C2CCC2)C1 C1(C(=O)NCCC(C)(C)C)(CNC(C(C)OCCC=C)=O)CC=CC1 C(=O)(C1=NOC(C)(C)C1)NC1(CC(=O)Nc2c(OC)ccc(O)c2)CCC1 N1(c2nc(N3CC(=O)N(CCO)CC3)c3c(n2)scc3)CCCCC2(CCCC2)C1 c1(OC)ccc(C=CC(=O)Nc2cc(C)cc(Br)c2F)cc1C(F)(F)F c1(CN(C(C2CCCN2C(=O)C=Cc2cccs2)=O)C2CC2)ccccc1 Cc1csc(C(C)C(N2CCCC2CNC(=O)CC2CC(OC(C)(C)C)C2)=O)n1 Cc1ccc(C(N2CCCC(NC(C3(C4CC4)CCC3)=O)C2)=O)cc1C CC1CCN(C(C2CC(C)(C)C2)=O)CC1NC(=O)Cc1cccc(Cl)c1Cl c1(C(=O)NCC(CC)(C)NC(=O)C(F)F)cc(OC)ncc1Br N1(C(C(=O)N(C)C)=O)CCN(C2CCC(NC(=O)COC3CCCCC3)C2)CC1 CC(C)(C)CC(F)C(=O)NC1(C(N2CC(NC(=O)C3CC3)C2)=O)CCCCC1 N1(C(c2cc(OC)ns2)=O)C2CCC1CN(C(=O)C(C)(O)C1CCCCC1)C2 O=C1CCC(C(=O)NC23CC2CN(C(=O)C(F)=C2CCCC2)C3)n2cccc21 Cc1cc(C(=O)NC(C)(CNC(=O)COC(F)F)C(C)C)c(C)o1 C1(C(N(CC(C)C#N)C)=O)CCCC(NC(=O)C=CC2CCCN2C)CC1 N1(C(C2C(COC)C2)=O)CCN(C(=O)C=Cc2cncc(O)c2)C(CC(F)F)C1 Cc1sc(=O)n(CC(N2CCC(NC(C3CCN(C)C3=O)=O)C(O)C2)=O)c1C CC(C)C(CN(C)C)C(=O)NC(C)CC(=O)N1C(CO)CC1CO c1(NC(C2(CCNC(CC3CCCC(=O)N3)=O)CC2)=O)cncc2ccccc12 N1(c2onc(CCC)n2)CC(C(=O)OC(C)(C)C)C2CCCCC12 C(CCOCCO)(C(=O)NCCNC(=O)C(C)CC#N)NC(CCOC)=O C#CC1(O)CC(C(N2CCC(CO)(CNC(=O)C(C(C)C)SC(C)C)C2)=O)C1 CC1=C(C(=O)N(CCCCCNC(C2(C3CC3)CC2)=O)C)Cn2ncnc2N1C C(=O)(CCCCN=[N+]=[N-])NC1(C)CCN(C(=O)C#CC2CC2)C1 C12(C(N(CCN(C(=O)C(COC)OC)CC)CC)=O)CCCN(CC1)S2(=O)=O n1(CC(C)(C)C)nc(-c2ccc(N)cn2)nc1CCc1ccco1 c1(N(C(C)=O)Cc2nc(-c3ccccc3)no2)ccc(C(C)C(=O)OC)cc1F Cc1ccc(NC(C2CC3CCN(C2)C3)=O)c(-n2cc(C3(C)CC3)nn2)c1 CS(=O)(=O)c1ccc(Cl)cc1C(=O)NC1Cc2ccccc2C1C(=O)O C(=O)(C(CC(C)C)C(N)=O)N1CC(NC(C2CC3(CC(=C)C3)C2)=O)(CO)C1 C(=O)(C#CC1CCCCC1)NC(CN(C)C)C(N1CCC2(CCOC2=O)C1)=O C1(NC(=O)COC2CCC2)CN(C(=O)CCCc2cncs2)CC2(CCC2)C1 C(=O)(C1=CC2CCCCCC12)N1CC(CCNC(C2CC3(CCC3)C2)=O)C1 c1(C(=O)NC(C)CN(C(C2CC2c2nccn2C)=O)CC)ncccc1OC(F)F N1(C(C(C)OCC#C)=O)CC2(NC(=O)C(C3CCCN(CC)C3)(C)C)CC1C2 N1(CC)CC(C(=O)NC2CC(NC(=O)C=CCOC)C2)NC1=O c1(NCc2nc(C)sc2)nc2cc[nH]c2c(=NC2CC2c2c(Cl)cccc2Cl)[nH]1 CC(C)C(C(=O)NCC1CC(F)(CNC(=O)CCn2cc(Cl)cn2)C1)N(C)C C(=O)(C#CC1(C)CCCO1)N1CCCC(N(C)C(c2ccc(C(N)=O)nc2)=O)C1 C1(NC(C2C(C#C)C2)=O)CN(C(C2(CO)CC(F)(F)C2)=O)CC1C=C CCC(C(=O)OC)C(=O)NCc1csc(C(=O)NC2CC2c2cnn(C)c2)c1 N1(C(Cc2ccc(C)c(Cl)c2)=O)CC2CCC1C(NC(C1CCCOC1)=O)C2 Cc1cnn(CCC(=O)NC(CC2CC2)C(=O)N2CC=CC2)c1 CCCCCCCN(C(=O)CCN(C(=O)CCc1conc1C)C(C)C)C N1(C(C(c2n(C)cnn2)(C)C)=O)CCN(C(C2C=CCC2)=O)C2(CCC2)C1 CCC(C(C)(C)C(=O)OC)N(C(=O)CC(C(=O)O)c1ccc(Br)cc1)CC C1(C(=O)NCCCN(C)C(C23CC(C)(C2)C3)=O)CC12CCCCCC2 CSC=CC(=O)NC1CCCC1CNC(=O)Cn1cc(Cl)cn1 CCC(O)C(C)C(=O)N(C(C)CCNC(=O)C(c1ccc(Cl)cc1)C)C c1(NC(CC)=O)cccc(C(=O)NC2CCCC2NC(=O)C(C)c2ccsn2)c1 n1(CC(=O)N(CCN(C(C=C(CC)C)=O)C(C)C)C)ccc2c(C)cccc12 Cc1cc2ncnc(N3CCC(NC(C4CC(O)C4)=O)C(C)C3)c2[nH]1 C1(NC(CC2CCC(N)C2)=O)CCC2CCCC1O2 c1(C(N2CC(C)(C)CC2C)C(=O)NCCOC)ncc(Cl)cc1F N1(CC(N2CCC(C)C(CNC(C3(C)CCC3)=O)C2)=O)CCc2sccc2C1 c1(C(=O)NCC2CC(NC(CS(=O)(=O)NC)=O)C2)cc(=O)c2ccc(Cl)cc2o1 CCC1=NOC(CC(=O)NC2(CCC(N3CCC(CCOC)C3)=O)CCC2)C1 C1C(C)(C)OCC(=O)N1C.CCCCOCC(=O)NCC(C)C1CC1 Cc1ccc2ncc(C(c3nnnn3CCN(C)C)NC3CC4CCC4C3)n2c1 Cc1cc(=NCC2CN(C(c3ncc(F)cc3F)=O)CC23COC3)[nH]c(Cl)n1 C(CN=c1[nH]c(=NC(C)CC)[nH]c2c1CC(C)CC2)SCC c1(C(N2CC(CNC(c3c(C)nc(CCC)o3)=O)C2)=O)cc(OC)nc(Cl)c1 C1(NC(C(CCN(C)C)NC(C(C(C)C)C#N)=O)=O)CN2CCC1(C)CC2 C(CC(=O)N1CCN(C(c2cc(N)cc(O)n2)=O)CC1CO)(C(N)=O)NC(C)=O c1(C(=O)OC)ccc2c(c1)CC(C)N2C(=O)Cc1cnccc1OC Cc1cnc2c(cnn2CC(=O)NC2CN(C(C3(C4CC4)CCC3)=O)CC2C)c1 Cc1c(C(=O)NC2CC3(NC(=O)COC4CCCC4)COC2C3)cc(CO)n1C c1(OC)cnc(C)cc1C(=O)NC(C1CCCN1C(=O)Cc1sc(O)nc1O)C CCC(O)(CC(=O)Nc1cccc(NC(c2nsnc2O)=O)c1)c1ccccc1 c1(CC)c(C(=O)NCC2(C(F)F)CCN(C(c3cnsn3)=O)C2)cccc1F c1(OC)cc(F)c(F)cc1C(=O)NC1CC(NCc2ccc(COC)s2)C1 C1(C)(C(=O)NC(CC)CNC(c2cncn2-c2cnn(C)c2)=O)CCOC1C Cn1ccnc1CCC(=O)N(CC(C)(C)CC1CN(C(=O)CC(Cl)Cl)C1)C1CC1 c1(-c2c(C(F)(F)F)nsc2)nc(-c2cccs2)nn1C1CCCSC1 C1(C(N2CC(OC)(CNC(=O)CCCc3ccccc3)C2)=O)CCN(C)C1=O Cc1nc2cc(C(=O)Nc3ccc4c(c3)CCCC4)c(F)cc2[nH]1 c1(OCC)cc2cnccc2cc1C(=O)NCC1CCC2(CCCCC2)O1 C1(NC(Cc2ccc(OC)cc2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CCC1C c1(OCC(=O)N(CCNC(=O)CC2(CO)CC2)CC)nc(Cl)c(Cl)cc1Cl c1(C(=O)NC(CNC(c2cc(C)cc(O)n2)=O)CC(C)C)ccnc2[nH]nnc12 Cc1ccnc(C2CCN(C(=O)C(N3CCCC(C(=O)NC(C)CC)C3)=O)C2)c1 c1(C(N2CC(C)(C(=O)NC(C)CCO)C2)=O)ccc(F)cc1Br N1(C(c2ccc3nnc(C)n3c2)=O)CCCC2(C1)C(O)CC2O C(=O)(CCS(C)(=O)=O)NC(CCOCC)C(=O)NCC(O)C(C)SC N1(C(C(CC#C)C)=O)CCN(C(=O)C(F)(CC)C(=O)OC)CC2(CC2)C1 c1(C(=O)OC)cncc(CN2CCCC2CNC(c2c(Br)cnn2C)=O)c1 c1(OC)nccc(C(=O)NC2CCCC2NC(c2cnc(-c3ccco3)s2)=O)n1 C#CC(C)(C)C(=O)NCC(CCC)NC(=O)C(C1CCCCC1)O c1(OCC)c(C(C)NC2CCN(c3ccc(Cl)cc3)C2)c(C)nn1C c1(C(C(=O)NC2CCC(NC(C3CC=CC3)=O)CC2)O)ccc(Cl)c(F)c1 c1(-n2cc(CNC(n3ncc(C)c3)=O)nn2)ccc(CNc2cccc(F)n2)cc1 Cn1nc(C(N2CC3CC3C2CN)=O)cc1-c1cccnc1 C=C(Cl)C(C)(C)C(=O)N1CC(CC(C)NC(=O)CSCc2ccccc2F)C1 CN1CCOC(C(N2CCC(C)(CCNC(c3c[nH]c(=N)s3)=O)C2)=O)C1 c1(CNC(CCCC#C)c2nnnn2C2CCOC2)c(F)cccc1Br C1(CC(N2CCOCC2CC2CC2)=O)CC2(CC2)CN1C(C1CCC(F)CC1)=O c1(C(N(CC(=O)NCC(=O)NCC2CC2)CCC)=O)sc(C)cc1C Cc1ccc(NC(=O)CC2(NC(C3CCCC(C#N)C3)=O)CCCCC2)cc1F c1(C(=O)NCCCN(C)C(c2ccnc(CO)c2)=O)ccc([N+](=O)[O-])nc1 n1(CC(=O)NC(C(C)NC(c2ccn(C(C)(C)C)n2)=O)(C)C)cccnc1=O CCCC(CCCS(C)(=O)=O)C(=O)NC1CC(CO)N(C(c2ccccc2)=O)C1 N1(C(c2cc(C(=O)OC)no2)=O)CCC(O)(CNC(C2CCC(=O)NC2)=O)CC1 CN1CCCC(C(C)(C)C(=O)NC2(c3nn[nH]n3)CC(F)(F)C2)C1 N1(C(CC(CC)C)=O)C2CCC1CC(NC(c1cc(=O)cc(Cl)[nH]1)=O)C2 c1(C(N(CCNC(c2c(C)n(C(C)C)nn2)=O)C(C)C)=O)cccc(F)c1C C12(C(=O)OC)CCC(F)(F)CC1CN(C(c1csc(Cl)n1)C(=O)NCC1CC1)C2 C1(CC(N2CC(F)(CNC(c3csc(C(F)F)c3)=O)C2)=O)CN2CCN1CC2 Cc1ccc(C(N2CC=CC2CNC(=O)COC(C)C)=O)c(Br)c1 C1(C(N(CC(C)NC(CCc2cc(C)[nH]n2)=O)C)=O)CCC(=O)N1C N1(C(CC(C)Oc2ccccc2)=O)CC(F)CC1NC(C1(C)CCC(=O)C1)=O Fc1cccc(-c2ncc(-c3nccn3CCOc3ccc(Br)cn3)s2)c1 Cc1nc(CO)oc1C(=O)NOCCOC(C)C.C1(=O)CC2(CC2)CN1 C(CCCCC(=O)N(C(C)C(N1CCC(C(C)O)CC1)=O)C1CC1)OCC C(CC(C)CCNC(=O)C(O)c1ccsc1)NC(Cc1nc(C)[nH]n1)=O N1(C(C(=O)OC)C)CCC2(CC1)CC2C(N1CC2CCC1(C)C2)=O C=CC(CC)CC(=O)N1CC(CNC(c2cc(Cl)n[nH]2)=O)C(F)(F)C1 C1(CCNC(C2C(OCC)CC2)=O)CCCN(C(c2cc(CC)ccn2)=O)CC1 c1(C(N2CCC(C)(CCNC(C(CC)F)=O)C2)=O)c(C)cccc1N C(=O)(C(=O)N=c1ccn(CCN(C)C)[nH]1)N(CCN(C)Cc1ccsc1)C S(=O)(=O)(c1ccc(Cl)c(OC(F)F)c1)NS(c1cnn(C)c1Br)(=O)=O C#CC1(C(=O)Nc2cncc(Cl)c2)CCN(C(=O)C(CN(C)C)CC)C1 C1(C(=O)NCCC(C=C)C)C2CN(C(C3(O)CCSCC3)=O)CC12 CCC(CCC(=O)NCCN1C(=O)CNC1=O)NC(c1ccc(Cl)cc1)=O c1(C(=O)NC2(CC=C)CN(C(C(C)OCC=C)=O)C2)cc(C(N)=O)cn1C C1(CC(=O)N(CCCNC(C2CN(CC)C2)=O)C)CCCN1CC c1(NC(c2ccc(-c3c(C)cccc3)cn2)=O)ncc(F)c(Cl)n1 C#CCCCCC(=O)NCc1ccc(CCNC(=O)CC2CCC(C#N)C2)cc1 N1(C(CNC(C)(C)C)=O)CCCC(CC(=O)NC2CC(NS(C)(=O)=O)C2)CC1 C#CCC(C)(C(=O)NC(c1nccs1)C)NC(=O)CC1CC(CC)=NO1 c1(C(N2CC(CC)(CC)S(=O)(=O)CC2)=O)ccc(Br)c2[nH]c(=N)sc12 c1(CNS(=O)(=O)c2ccc(O)cc2)cc(C2=CCC(C(F)(F)F)CC2)[nH]n1 C=CC(F)(F)C(=O)NC(C1CCCN(C(c2cc(F)n(C)n2)=O)C1)C N1(C(c2cn(C(C)C)nn2)=O)CCC2CN(C(=O)C=CC3CCC3)CCC2C1 c1(C(=O)NCC(C)CN(C)C(C2CCCN(CC(F)F)C2)=O)ccc(F)cn1 N1(C(CC=CC)=O)CCC2(CC1)CC2(CO)CNC(=O)C(C(C)C)n1cncn1 c1(C(N2CCC(CC)C2C(=O)NCC2(CF)CCC2)=O)cc(O)cc(F)c1 C(=O)(C1CCCn2ncnc21)NCC1(OC)CN(C(c2cc(C)sn2)=O)C1 CC1(C)OCC2CC12C(=O)NCC1(O)CCCN(C(=O)CCc2nccs2)C1 C1(C2CN(C(C3(c4cc[nH]n4)CC3)=O)C2)(NC(C(c2cccnc2)C)=O)CC1 N1(C(CC(=O)OC)=O)CCN(C(c2cncc(CO)c2)=O)CC1C1CC1 c1(C(=O)NC2C(NC(C3C(SCC)CCC3)=O)CCC2)ccnc2c1ncn2C c1(C(N(CCNC(C2CNC(=O)O2)=O)C2CC2)=O)ccc(N(C)CCO)cn1 C1(CNC(c2cc(SC)oc2)=O)COC(C)(C)CN1C(=O)CC1CCCN1C N1(C(C)C)CC(C(N2CCN(C3CCN(C(=O)C=CBr)C3)CC2)=O)CC1=O C12(C(N3CCC(NC(CC4CCN(C)C4)=O)C(O)C3)=O)C3C4C1C1C2C3C41C#N N1(C(CC(C)C(C)(C)C)=O)CCC2(CC1)CC(NC(=O)CCC1OCCO1)C2 n1(CCC)cc(C(=O)NCC(C)(C2CC2)NC(=O)CC2CC(CF)C2)nn1 CCC(C)(C)C(O)C(=O)NCCC(N1CC2C(C1)C2(C)C)=O c1(C(=O)NCCCOCCNC(C(C2CCC(=O)N2)C)=O)cnn2c1NCCC2 CCCCC(C)(F)C(=O)N1CCCC(N(C)C(C2CCCCC2)=O)CC1 N1(C(c2nc(C)c(C)s2)=O)CCC(C(=O)OCc2c(Br)cnn2C)CCC1=O N1(c2nccc(NC(C)=O)n2)CCN(C(c2cccc(F)c2I)=O)CC1CO C(=O)(C1CCCc2ccccc21)NC1(CNC(c2cc(C#N)no2)=O)CC1 CCC(CC(=O)N(CC(O)CNC(C1(c2ccn(C)n2)CC1)=O)C)CC(F)(F)F N#CC1CCCC(C(=O)NCc2ccsc2C(N2CCC(O)(CO)C2)=O)C1 c1(OC)ccc(NC(=O)C(c2cc(OC)no2)N2CCCC2CC2CC2)cc1 CC1CN(C(=O)Cc2cncnc2)CCC1NC(C1C2(CC2)C12CC2)=O C1(C(=O)NCC(C)N(C(=O)CNC(C2CCC2)=O)C)CCCCS1(=O)=O C(=O)(CCCc1cnn[nH]1)NCC(CC)N(C(=O)Cc1occc1C)C C1(O)(CCNC(c2n(C=C)nnc2)=O)CCCN(C(C2(SC)CCCCC2)=O)C1 Cc1ccccc1C(=O)NCC(O)CNC(c1ocnc1C)=O C1(CN(C)C(C2CCC(=O)N2)=O)CN(C(=O)CC(C)(C)C)CCO1 N1(C(CCNC(C#CC(C)(C)C)=O)=O)CCC2CCC(C1)N2C CC1CCN(C(=O)C=Cc2ccnn2C)CCN1C(C1CCCNS1(=O)=O)=O N1(CC)CC(C(=O)NC(=O)C(C)(C)C#N)C2(COC2)C1 N1(C(=O)CC(F)F)CCOC2(CCN(C(C3CCN(C4COC4)C3)=O)CC2)C1 c1(OC)c(C)cc(C(N2CC(C3(NC(c4oc(C)cc4C)=O)CC3)C2)=O)cc1Cl Cc1cc(C(N2CCC(C)(C(=O)NC3CC3CN(C)C)C2)=O)cnn1 N1(C(C=CC)=O)CCC2C(NC(c3cc(C(C)(C)C)oc3C)=O)C2CC1 N1(C(CCNC(C)=O)=O)CCC2(CCCC2C(=O)Nc2cnc(Cl)nc2)C1 C1(NC(CC2(C=C)CC2)=O)CCCCC1CNC(c1c(Cl)n[nH]c1CC)=O c1(CC)ccc(C(=O)NC(CCN(C)C(C2(F)CCOC2C)=O)C(C)C)c(C)n1 CCC(O)C(F)(F)C(=O)NC(CNC(c1ccc(O)c(C(C)C)c1)=O)CO N1(C(C(C)NC=O)=O)CC2CN(C(c3ccc(C(O)C(F)(F)F)cc3)=O)CC12 C1(NC(c2cc(CC)oc2C)=O)CN(C(=O)C(C)Cc2cccnc2)CCC1F C1(C(=O)NCCC(C)NC(c2nnc(C)s2)=O)(CO)CCCCO1 C(CCN(C)C)(C(=O)N1CC(F)CC1CO)NC(C(N1CCNC1=O)C)=O C1(CCC)CN(C(C2CC(=C(F)F)C2)=O)CCN1C(C1CCN(C)C(=O)C1)=O N1(CC)CC(C(N2CC(OC)C(NC(c3ccoc3Br)=O)C2)=O)CC1=O C1(CCN(C(C2C(C)(COC)C2)=O)C)CCN(C(c2scnc2C2CC2)=O)CC1 c12ncccc1C(=O)NC1(CC1)CNC2=O.c1(NC)cc(OCCOC)n[nH]1 c1(C(=O)NC(C2CCN(C(=O)CC3(C#N)CC3)CC2)C)cc(O)cc(O)n1 C#CCC(C)(C)C(=O)N1CCN(C(=O)CCN2CCCCCC2)C(CF)C1 C#Cc1ccc(OC)c(C(=O)NCC2CCN(C(c3ccc(OC)s3)=O)CC2)c1 n1(C(=O)CC)nncc1N.C12CCC(C1)CN2.c1(C(C=O)c2cn[nH]c2)ccncc1 C(=O)(C1=COCCO1)NC(C1CN(C(=O)C(O)CCN(C)C)C1)C C12(CNC(CCCN(CCC)CCC)=O)CC1CN(C(=O)CCc1cnn(C)c1)C2 c1(CN(C2CC2(F)C(=O)O)CC(C2CC2)OC)cnn(C2CCCC2)c1C Cc1ncc(Br)c(C(=O)NCC(C(C)(C)C)NC(C2(Cl)CC2)=O)n1 c1(C(N2CC(C(=O)NC3COC(C(C)C)C3)(SC)C2)=O)cc(C)c(C)s1 Cc1ccc(C)c(C(N2CCC(O)(C(C)CNC(=O)CN(S(C)(=O)=O)C)C2)=O)c1 N1(C(CCSCCC)=O)CCCC1C1CCCN1C(=O)C=C(C)C1CC1 C1(C(=O)NCC(COC)(F)F)C(C)CCN1C(c1ccc(C#N)[nH]1)=O C1(O)(CC(N2CCC(CN(c3ccc(C#N)cn3)C)C2)=O)CCCN(C)C1 c1(CC(N2C(C3(NC(CNC(c4ccoc4)=O)=O)CC3)CCC2)=O)cccnc1O S(=O)(=O)(C=Cc1ccc(Cl)cc1)N1CC(CC(C)C)OCC1 C1(C(=O)NCC2N(C(c3n(C)[nH]c(=N)c3)=O)CCC2)CCCCN1N=O C1(O)(C(C)NC(C2CC(C(F)F)C2)=O)CCN(C(c2csc(Cl)c2)=O)C1 c1(C(=O)NCCCC(CCC)NC(=O)CC2CC=CCC2)n[nH]c2c1CCSC2 c1(OC)ccc(CCC(=O)NC(c2cn(CC(=O)N(C)C)nn2)C)cc1F c1(C(=O)NC(C)C(c2ccccc2)NC(=O)CC2(C)CC2)ccn(C)c(=O)c1O CCCCCS(=O)(=O)CC(=O)NC1CN(C(c2cnc(CC3CC3)s2)=O)CC1O c1(C(N(C2CC(C(N)=O)C2)C)=O)coc2c1CN(C(=O)C(C)(C)F)C2 C1(C(N2CCC(CN(C(C(OC)OC)=O)C3CC3)CC2)=O)CCCC12CCC2 N12CC3CN(CC3C1)C(=O)C(C)c1cccc(c1)O2.CCS(=O)(=O)NC1CC1 C1(NC(C2(COC)CCC2)=O)(NC(=O)C(=O)NC2CC2)CC(O)C1 C1(NC(CC(C(F)F)NC(CN(C)C(N)=O)=O)=O)CCn2nccc2C1 c1(CC(=O)N(CC(C)NC(=O)C(C)CSC)CC)cccc(F)c1OC C1(CNC(c2nc(C)sc2C)=O)CN(C(C2CC2C(F)F)=O)C2(CCOCC2)C1 Cc1ccc2cc(C(=O)NC3CCCCN(C(=O)CCCCCO)C3)ccc2c1 N12CCc3cc(ccc3C1)C2=O.c1(SC)cccc(C)c1NC(=O)CC1CC1 CCCC(O)(CCC)CC(=O)NC1CC(C)(N)C1.c1(C(=O)N)nn(C)c(C)c1Cl N1(C(c2c(OC)ccc(O)c2)=O)CCN(C(=O)C(C)=C2CCCC2)CC(C)(F)C1 c1(C(N2C(CNC(c3c(N(C)C)cccn3)=O)CCC2)=O)cc(O)c(F)cc1N C1(O)(C(=O)NCCCCCNC(c2c(NC(C)=O)c[nH]n2)=O)CCOCC1 N1(C(CNC(CNC(C)=O)=O)=O)CC2CN(C(c3cnsc3C)=O)CC2(C)C1 CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1cc(CO)[nH]n1)=O C(=O)(CCC(C)CN(C)C)NCC1(C)N(C(C(C(=O)OC)C)=O)CCC1 C(CC(=O)N1CC2=C(C1)CN(C(c1c(C)nsc1N)=O)C2)(C(F)(F)F)OC N1(CCNC(=O)CC2(NC(=O)C=CC3CCC3)CC2)CC=CC1 CN1CCc2cc(C(=O)NCC3CN(C(=O)Cn4cnnc4O)CCO3)ccc21 N1(C(C(CC)CC)=O)C2CCC1CC(NC(=O)C(O)Cn1cncn1)C2 CC(N=c1nc(N(CCCO)C)c2c([nH]1)CCS2)c1cnc2ccccn12 C(=O)(C1CCCc2nc[nH]c21)NC1CN(C(C(CC)(F)F)=O)CC1C C1(C(=O)NC2C(CNC(CCCC#C)=O)CC2)CC2(C1)CC(F)(F)C2 c1(CC)nc(CNC(=O)NN2CC3CC2C3)c(Br)s1 N1(C(Cn2c(C)csc2=O)=O)CC2(CCCC2NC(=O)Cc2cn[nH]c2)C1 C1(C(N(CCCN(C(COc2ccc(OC)cc2)=O)C)C)=O)CCC2C1C2(F)F C12(C(c3ncc(Cl)cn3)CNC(=O)CC(=O)NCC3CC3)CCC(CC1)C2 C1(NC(COC)=O)(CC(C)C)CCCCC1.C1(C)(C)C(=O)NC2CC(C2)O1 O=C(C1=CC2CCCCC12)NCC#CCNC(=O)C1Cc2ccccc21 Cc1ccnc(O)c1C(N1CC2CC(C1)N2C(c1ccsn1)=O)=O N1(C(CC(c2ccccc2F)C)=O)CCC2(CCCN2C(=O)Cc2cnc[nH]2)C1 c1(C(=O)NCC2CCN(C(C(C)(C)CCF)=O)C2)nc2ncccn2n1 Cc1cc(C(F)F)oc1C(=O)NC(C)CN(C)C(c1ncc(C(F)(F)F)n1C)=O C1(C(N(CC(C)(C)C(=O)NC2CC3CCCC3C2)C)=O)Cc2ccccc2C1 c1(N(C)CC2CCSC2)nnc(-c2ccccc2F)n1CC(=O)NCC(F)F c1(C(=O)NC2(CNC(C(C)=C(CC)C)=O)CC2)c[nH]c2cc(F)c(F)cc2c1=O Cc1nc(C)n(O)c1C(=O)NCCCC1CCCN1C(=O)Cc1cccc(F)c1 CON(C)S(=O)(=O)c1ccc(C(N2CCN(C(c3cc(F)c[nH]3)=O)CC2)=O)cc1 c1(-c2c(C(=O)NCCC(C)CO)cc(F)c(F)c2)ccc2cnccc2c1 N1(C(C(C)n2cccn2)=O)CCCC(NC(=O)CSCc2ccc(F)cc2)CC1 c1(NC(C2CCN(CCO)CC2)OC)nccc(=NCc2cc(F)ccc2Br)[nH]1 N1(C(C(c2ccc(C)s2)C)=O)CCCC(C)C1CNC(=O)CC1CC12CC2 N1(C(c2ccc(-c3ccccc3)s2)C(=O)NCC=C)CCSCC1c1nccs1 C(CCC(CCC)NC(=O)CC(=C)Br)NC(CCC(=C)Cl)=O C1(C(=O)NCC(C(=O)OC)C)CCN(C(C)=O)CC1C(C)C N1(C(COC)=O)CCOCC(NC(=O)NCC2(c3cc(C)cc(C)c3)CCC2)C1 C1(C(N(C(c2n3cc(c2)C3c2cnn(C)c2)=O)CCCCC(F)(F)F)=O)CCN2CCCCC2C1.C(C)=O.CC(C)CCC C1(CNC(c2csc(C(F)F)n2)=O)CCCN1c1nc(C2CC2)ns1 C1(C(C)C)CC(CC(=O)NC2CCN(C(=O)C3=COCC3)C2C)CCO1 N1(C(=O)C(O)c2ccco2)CC2CCC(C1)N2C(C1CN2CCN1CC2)=O C#CC12CC(CN1C(=O)CC(C(F)F)NC(C13CCC(CO)(CC1)C3)=O)C2 C(=O)(C1=CCN(C(c2ccc(C)c(C)c2)=O)CC1)NC(C1CCOC1)C#C Cc1cc(C(=O)NC2CC(C(=O)NC(CO)CCO)C2(C)C)n(C)n1 C(CS(=O)c1ccc(C)cc1)NC(=O)NC1C(SC)CCCC1 C(=O)(C1CCCc2ncnn21)NCC(CO)NC(c1c(SC)cccn1)=O C1(C(N2CC3CN(C(C=CC=CC)=O)C3C2)=O)CCc2ccccc2C1O c1(CC)ccccc1S(=O)(=O)N1CCCC(CCN)C1 N1(CC(=O)N(CC(=O)NC2CCC(OC)C2)C)CCC(C)CC1 C(=O)(C(C(C)C)N(C)C)N1C(CNC(CC2(CSC)CC2)=O)CCC1 C12(C(N3CC(N(C(C4(CC)CCCCC4)=O)C)C3)=O)CCC(F)(CC1)CC2 c1(CCCOC)nc(C2=NOC3(CCOC3)C2)n(-c2c(F)cccc2Cl)n1 CC1(C)CC2(CC(C(=O)NCC(N3CCN(C(C45COCC4C5)=O)CC3)=O)C2)C1 C12(C(=O)NCC(F)(F)F)CCOC1CCOC2.CCCNC(=O)C=CC=CC=CCO CC(C(=O)NCC(C)=CC(=O)NC(C(N)=O)c1cnc[nH]1)S(N)(=O)=O c1(CCC(=O)NC2C(C)N(C(c3sccc3F)=O)CC2)ccc(Cl)c(F)c1 C1(C(=O)NC(C(=O)NCCC)C)CC12CCN(C(=O)C(F)CCCC)CC2 C(CCC(C)(C)C(=O)NC(CC)C(C)O)NC(CCC=C=C)=O c1(OC)ccc(Cl)cc1CC(=O)NCCC1CN(C(=O)C(C)CSC)CCO1 Cc1c(O)ccc(C(N2CCC(CNC(=O)C3=NOCC3)C2(C)C)=O)c1C N1(C2(CCC(=O)CC=CCOC)COC2)c2ccccc2Sc2ccccc21 c1(OC)cc2c(c(S(=O)(=O)NC3c4ccc(C)cc4CCCC3C)c1)OCC2 c1(-c2cn(C(=O)Nc3coc(-c4ccc(Cl)cc4)n3)nn2)cnccc1C1CC1 c1(N(C(=O)NCC(C2CCC(C)(C)CC2)C)C)ccc(Br)cc1C#N CC(C)(C)CC(C(=O)NCCC1CC1)N(CCCN1CCOCC1=O)C c1(CC)c(C(=O)NCC2CCCC(NC(c3cc(C)on3)=O)C2)nnn1CC N1(CC)N=C(C(=O)N2CC(N(C(=O)C=C(C)C(C)(C)C)C)C(F)C2)CCC1=O CN1CCN(CC(C)(C)C(=O)NC2CCC3CC23C(=O)OC(C)(C)C)CC1 C1(NC(C(CSC)C)=O)CCC(O)CN(C(=O)CC(C)(F)F)C1 c1(C(N2CCN(C(COCC=C)=O)C(C3CCCC3)C2)=O)cc(Cl)c(F)cc1N Cc1cc(CCC(=O)NC2(C)CC(C(N3CC(O)(CO)C3)=O)C2)nn1C CC1(C)CC(C(=O)N2CC(F)CC2CNC(=O)CCCNC(=O)C2CC2)=NO1 Cn1cc(C(=O)NC2CN(C(c3cnc(OCF)cn3)=O)CC2F)c2ccccc12 C1(CNC(CC2CCN(C)C2=O)=O)Cc2ccccc2CN1C(=O)Cn1cncn1 CCC(CCCC(=O)N1CCSCC1C1CC1)NC(c1ccc(F)cn1)=O Cc1cccc(OCC(=O)NCC2(NC(=O)CC(C)C3CC3)CCOCC2)c1 N1(C(C(CCOC)C)=O)CC(NC(c2ccnc(C)c2N)=O)CC(C)C1 N1(C(C2N(C(C(C)N(C(C)=O)C)=O)CCCCCC2)=O)CCC2(C=CCO2)CC1 c1(C(N2C(C)CC(NC(C3(OC(C)C)CCC3)=O)C2)=O)cncc(Br)c1C N1(C(C(CCCC)C)=O)CCCC2(CCN(C(=O)C(c3c(C)noc3C)C)C2)C1 N1(C(C(C)NC(CC)=O)=O)CCCC(C2CCCN(C(c3cccs3)=O)C2)C1 c1(C(N2C(=O)CC2)=O)ccc(Cl)c(SCC(=O)NC2CCC2)c1N.C#CCNC C1(C(N2CC(n3c(C)nnn3)C2)=O)CC2CC1CC2NC(C1(NC(N)=O)CCC1)=O N#Cc1cc(F)ccc1C(=O)NCCC1CCC(NC(C2(C3CC3)CCC2)=O)C1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(=O)CNC=O)C4CCCCC34)cc12 C1(N(C(=O)CCn2cnnn2)CC)CCN(C(=O)CN2CCOCC2)C1 C(C(=O)Nc1cn(C)nc1C)(C(C)C)NC(CCc1onc(C)n1)=O C(=O)(CCC(C(=O)NC1(C)CN(C(c2cc(C)ccc2Cl)=O)C1)N(C)C)OC c1(C(=O)NCC(CNC(c2c(CC)cno2)=O)(C)OC)nc(=N)cc[nH]1 C1(NC(c2sccc2Br)=O)CCCCC1n1cc(C2CC=CCC2)nn1 C1(C2CCCN(C(=O)CCc3ccn(C)n3)C2)(NC(C(C(CC)O)C)=O)CC1 C1(CC(NOCCCC#C)=O)C2CN(C(C3CCC(C)(C)C3)=O)CC12 N1(C(C2OCCC(C)C2)=O)CC2CCCC(C1)N2C(=O)CCCc1ccccc1 CCCCC(O)CC(=O)NC1CCCCN(C(c2cc(C(C)C)on2)=O)C1 C(=O)(C(C)(C)C(=O)NCCC(C)N(C)C(C1CCS1(=O)=O)=O)OCC c1(C2(C(=O)NCC(CC)NC(C3(C)COC3)=O)CCCC2)c(F)cccc1F C1(C)(CC)CCN(S(=O)(=O)Cc2ncoc2CN)C1 O=C1OC(C(=O)N(C2CCCC2)CCN(C)C2CC2)Cc2ccc(F)cc21 c1(-c2cc(C)no2)cc(CNC(N2CCCCC2c2nnc(CO)o2)=O)c(C)o1 C(CCC(C(=O)NCCc1cccc(O)c1)NC(=O)Cn1nc(C)oc1=O)OC C(CC(C)C(=O)NCCCN(C)C(c1ccc(C(C)F)cc1)=O)=CCC c1(C(=O)NCC2OCCN(C(C=C(CCC)C)=O)C2)ccc(Cl)c(C(=O)OC)c1 N1(c2nnc(C)o2)CCC(C2CCCN(C(=O)CSc3nncn3C(C)C)C2)C1 N#Cc1cccnc1NC(C1CCN(Cc2cc(-c3cc[nH]n3)ccc2F)C1)=O CC1(C)C(C(=O)NCC2CC(NC(=O)Cn3cccn3)C(O)C2)CCS1(=O)=O C(=O)(C1=NOC2COCC12)NC1CC(NC(c2ccc(C(=O)OC)s2)=O)C1 c1(C(=O)NCC2N(C(CCC(CC)CC)=O)CCC2)cc2[nH]nnc2cc1OC N1(CC(=O)N(CC(=O)NCCC(C)(C)O)C)C(=O)CNC1=O c1(C(N(C)CC2(O)CN(C(c3cc(CC(C)C)on3)=O)C2)=O)ccc(O)c(F)c1 c1(CC)cc(NC(=O)CN(C(=O)C(C)C2(O)CCC2)C2CCC2)cc(F)c1 O=S(=O)(c1cccnc1N1CCOC(C2CC2)C1)NCc1c(F)ccc(Cl)c1Br C(=O)(C(C#N)C(C)(C)C)NCCC(=C)CNC(c1ccnc2ccsc12)=O CC(F)(F)C(C)(C)C(=O)NCC1(C2(O)CN(C(=O)C(c3ccccc3)O)C2)CC1 C(CCN=C(NCc1cn2cccc(F)c2n1)N1CCC(O)C1)NS(C)(=O)=O c1(C(=O)NCCN(C)C(C2(c3ccn(C)n3)CC2)=O)cc(CC(C)(C)C)c[nH]1 C(=O)(C1=C(C)OCC1)NCCCCC1CN(C(CNS(NC)(=O)=O)=O)C1 C(CC1=CCN(C(=O)CN(C2CCCC2)C)CC1)NC(C(C)OCC=C)=O c1(CC)sc(C(=O)NCCN(C(=O)CC2OCCCO2)CC)cc1Br c1(C(=O)NCC2N(C(C(CN(CC)CC)F)=O)CCC2)cc([N+](=O)[O-])ccc1O CC12CCCCC1CN2C(C1CN(C(C2CC2Cl)=O)CC12CC2)=O CCC(C)CC(=O)C(=O)NCCCN(C(=O)Cc1cnsc1)CC C(CCCN=[N+]=[N-])C(N(C(C)C(=O)NCCc1cn[nH]c1)C)=O c12ccc(cc1)CS2.N1(C(c2n(C)cnn2)=O)CC2CC1C2Cn1ccnc1 CCC(C(=O)N(C1CC1)C)OC.N1(CC=O)CCOCC1 c1(C(N(C(C)C(N2CC(C)(O)C2)=O)C)=O)cc(O)nc(O)n1 N1(C(C(Cn2cncn2)NC(c2cncs2)=O)=O)CC2CC2(CO)C1 C1(C)(CNC(C2CC(C)OCC2)=O)CCN(C(=O)CCSCC(N)=O)CC1 N1(C(CC2(CSC)CC2)=O)CCCCC(C(=O)NCC(O)CCO)C1 N1(C(C2COCCN(Cc3cc(C)[nH]c3C)C2)=O)CCC23OCCN2C(=O)CC13 C(=O)(CC(C)CNC(C=CC(CC)C)=O)N(C1CCN(C(C)C)C1)C c1(C(=O)NC(C(=O)N(CC(C(=O)NC)C)C)C2CCOC2)ccnnc1C C(=O)(C(C)(C)C1=CCSCC1)NC1C2CC(NC(CC(C)OC)=O)C(C2)C1 c1(CCC(=O)NC2CCN(C(c3coc(Br)n3)=O)C2)ccsc1Br C(=O)(C(CNC(=O)CNC=O)CC1CCCC1)N(CCN(CC)CC)C Cc1cccc2sc(NC(C3CN(C(c4cnn5cccc(C)c45)=O)C3)=O)nc12 C1(F)(CNC(CCCOCC)=O)COCCN(C(=O)CC(O)CC)C1 C(=O)(CC1=CCN(C)CC1)N(C1C2CN(C(c3cccc(C)n3)=O)CC21)C N1(C(C2N(C(C3CCC(=O)O3)=O)CCCC2)=O)CCC2(CCO2)C1 N1(C(N(Cc2n(C)ncc2)O)=O)CCCC(OCCO)C1 N1(C(c2onc(CC)n2)=O)CC2CC(NC(C3CCCS3)=O)C2C1 Cc1c[nH]c(CC(N)=O)c1C(=O)NCC1(C(N)=O)CN(C(=O)C(F)(F)CO)C1 CCC(C)C(O)CC(=O)NC1(C)CC(C(N2CC(CO)C(O)C2)=O)C1 N(C1c2cc(OC)c(C(=O)O)cc2CCCC1(C)C)C(C(CCC=C)(C)C)=O c1(CNC(=O)NCC(C2CCCOC2)OCC)ccc(C(=O)O)cn1 Cc1nn(C)c(C)c1OCC(=O)NC(C1CCN(C(=O)CCn2ccnn2)C1)C C(N=c1[nH]c(N2CC3CC2CN3CC(F)F)nc2c1SCC2)c1n(C)ncc1 C(=O)(CCC(C)(C)C(=O)N1CC(NC(=O)C(CO)C(C)(C)C)C(C)C1)OC CS(=O)(=O)C1(C(N2CCCC(F)(CNC(C3CC3Cl)=O)C2)=O)CCC1 c1(C(N2CC(NC(c3n(CC)ncc3)=O)C(F)(F)C2)=O)cc(C)c(OC)cc1C C(=O)(CC(C)(C)CNC(c1cncn(C)c1=O)=O)N(CC(CC=C)(F)F)C C(=O)(CCCCCCCC1CC1)N1CC2(C(NC(=O)CC3=CCOCC3)CC2)C1 CCCCC(O)C(C)C(=O)NCC1N(C(c2cncc(OC)c2)=O)CCC1(C)C C1(C(N2CCC(NC(C3CC(OC)(OC)C3)=O)(CF)C2)=O)CCn2ncnc2C1 c1(C(N2C(CCC(=O)NCC(COC)(C)CO)CCCC2)=O)cnc(O)cc1C C1(C(=O)OC)CC2(CC(NC(=O)N(CC(C)OC)C)CCO2)C1 N1(C(c2ccc(C(C)C)o2)=O)CC2CCC2(NC(C2Cc3nccn3C2)=O)C1 c1(C(N2C(C(=O)NC(c3ccccc3)CC)CC(O)C2)=O)ccc2nc(Br)sc2c1 c1(C(N2CCC(F)(C(=O)NC3(CC)COC3)C2)=O)c(O)cccc1F N1(C(C=CC)=O)CCCC2(NC(c3cc4cc(Br)sc4[nH]3)=O)CCCC12 c1(C(N(c2ccc(CC)cc2)C2CNCC2(F)F)=O)ncnc2[nH]c(C)nc12 C1(C(=O)NC)CCC2C(N1C(c1ccc(CNC(=O)OC(C)(C)C)cc1)=O)C2(F)F c1(C(=O)NC(CC)Cc2ccc(Br)cc2I)cc(Nc2ccnc(C)c2)nc(Cl)c1 Nc1nonc1C(=O)NC(C1CCOC1)CNC(=O)C=C1CCCC1 CCC(C(=O)NCCn1cc(CNC(C2CN(C3COC3)C2)=O)nn1)C(C)O c1(NC(N2C(C(CC)O)CCC2)=O)cc2cnccc2nc1C C(=O)(CC(C)(C)CNC(C1(F)CCCCCC1)=O)NC1CCCC(CC)C1 C(C(C)(C)CCNC(c1cscc1Br)=O)NC(C1(CC)COC1)=O C1(NC(c2cc(C3CC3)cc(F)c2)=O)CN(C(C2(CO)CCC2)=O)CCC1CO CN1C(C(=O)NC(C2CCCC2)CNC(=O)CC2(C3CC3)CC2)CCS1(=O)=O C(C1CCOCC1)=CC(=O)NCC(CNC(C1C(C(=O)OCC)C1)=O)C C(CCCC(=O)NCC1CC1NC(=O)Cc1cncn1C1CC1)SC C#CCC(CC#C)C(=O)N1CC(NC(c2cccc(OCC(F)F)n2)=O)C(F)C1 c1(CNC(C2(COC)CCN(C(=O)C=CCCC(C)C)C2)=O)nc(C)ccc1C N1(C(C2CCN(OC)CC2)=O)CCN(C(c2cnn(C3CC3)c2)=O)CCC1C N1(C(C=C2CCN(C)CC2)=O)CC(CNC(C2CCCCC2O)=O)OC(C)(C)C1 C(c1ccc(O)cc1)=CC(N1CCC(C(F)(F)F)(CNC(C(N)=O)=O)C1)=O c1(CC)cccc(C(=O)NCCCC(CO)NC(C2CCC(N(C)C)C2)=O)n1 c1(C(N2CC(C(=O)NC(C3(SC4CC4)CC3)=O)C2)=O)cccc(Cl)n1 Cc1c(C(=O)NC2CN(C(=O)C(F)C3CCC3)C3(CCC3)C2)c[nH]c2nccc1-2 C1(NC(CNC(=O)NC)=O)CCCC(NC(=O)C(C)CSC(F)(F)F)C1 N1(C(C(F)=CCC)=O)CCC2(CCCN2C(C2CCSC(C)C2)=O)C1 C(CC(C)(C)C(=O)N1CC(NC(C2CC=CCC2)=O)C(C(F)F)C1)SC c1(C(=O)NC(C(C)NC(CCSC)=O)(C)C)cc(Cl)c(Cl)cc1C C=CC1(C(=O)NCC(C)(C)C(C)C)CCN(C(=O)Cc2cc[nH]c2)C1 Cc1[nH]c2ccccc2c1C(=O)NC(C)Cn1ccccc1=O Cc1cc(NC(C2CCCCN2C(=O)CC(C)C)=O)c(N2CCCC2C)nn1 CN(C)NC(=O)CCC(=O)NCCCNC(c1cc(O)cs1)=O Cc1cc(F)c(C(N2CCC(N3C(=O)CNC3=O)C2)=O)cc1C(F)(F)F C(C1OCc2cc(Cl)ccc21)NC(c1cc(OCC)c(F)cc1)C N1(C(CCSCCCC)=O)CC(NC(C2(CC(C)C)CC2)=O)CC(O)C1 C=CCC(C(=O)N1CCC(CC=C)(C(=O)NCCN2CC(OC)C2)C1)N(C)C N1(C(C2CN(C)C2)=O)CC2CCC(N(C(=O)CC3(C)CC3)C)C2C1 C1(C(=O)NCCN(C(=O)CCCC(F)F)C(C)C)CCc2ncccc2C1 C1(C(N2CCCC(CNC(C(C=CC)O)=O)C2)=O)CNc2ccnn2C1 C1(CC(=O)NC(C)C(C)NC(=O)C(C)(C)C#N)CCC(F)(F)CC1 Cc1cc[nH]c1C(=O)N(C(C)CNC(=O)C(F)CC1CCCCC1)C Cn1cnn(CC(=O)NCC(C(C)(C)C)NC(C2C=CCC2)=O)c1=O c1(C(c2n(C(C)C)nnn2)NC(c2cccc(Cl)c2)CCO)csc([N+](=O)[O-])c1 CCC(CNC(=O)C=C(C)CN(C)C)(CC)NC(=O)OC(C)(C)C.C(=O)(CNC)N CCCCC(C)CCC(=O)NCCC(C)(C)C(=O)NCCCCC1CC1 c1(C(N2CC(NC(CNC(C)=O)=O)C(C)(C)C2)=O)c[nH]c2cc(F)ccc12 C1(NC(C2CC(OCC)C2)=O)(CF)CCN(C(c2cnn(C(C)C)c2C)=O)C1 c1(CC(=O)NC2(C)CCCN(C(C3CC(SC)C3)=O)C2)ccc2c(c1)CCC2 C(CN=c1cc(NC2CC2c2nc(C(F)(F)F)cs2)nc(C)[nH]1)NS(CC)(=O)=O N1(C(C(C)N(CC)CC)=O)CCC1(C)CC(=O)NOCC1(C)CC1 N1(Cc2c(C)ccc(C)c2)CCC(NC(=O)CCC2CCC(=O)N2)CC(C)(C)C1 CC(CC(F)(F)F)C(=O)NC1CCCCN(C(C2(C)CC2C(F)(F)F)=O)C1 C1(NC(C(C)(C2CC2)OC)=O)CC2(C1)CC1(CC(NC(=O)CSC(C)(C)C)C1)C2 C1(NC(=O)CCSCc2ccccn2)C2CN(C(C34CC(C3)C4)=O)CC12 c1(OC)ccccc1N1CCC(NC(=O)NC(C2(F)CCC2)C)C1 N1(C(=O)COCC2(O)CCCCC2)CCCCC1c1ccc(F)cc1 N1(C(C(CCC)=CCC)=O)CC(NC(C2(n3cccn3)CC2)=O)CC(O)C1 c1(C(=O)NC2(CNC(C3(OC)CC(C)C3)=O)CC2)cnn(C(C)C)c1N N1(C(CC(COC)C)=O)CCN(C(=O)Cc2ccsc2C)CCC1C N1(C(Cc2cc(C)sc2)=O)CCC(CNC(=O)CCc2c(C)noc2C)CC1C c1(C(=O)NCCN(C(C2C3C4CCC(C4)C23)=O)CC)cc2cnccc2[nH]1 CC1CC(C(=O)NCC2(CC3CCC3)CC2)CN(C(=O)CC2CCC(=O)N2C)C1 C12(CNC(=O)NCC)CCCC(C)(C1)OC2.C12C=CC(C1)C(=O)O2 C1(C(=O)NCC(C)Cc2ccco2)C2CN(C(C)C(=O)NC(=O)C3CC3)CC12 C1(C(N2CC(N(C(=O)C3=CCOC3)C)C(O)C2)=O)CC2CCC(C1)C2 C1(CNC(C(C)OCOC)=O)CCCCN(C(C2C3CCCCCC23)=O)C1 c1(NC(=O)CCCCCBr)cccc2cc(O)ccc12.n12cc(cn1)CNC(=O)C2C CC1(C(=O)NCCc2ccc(F)nc2)CCCN(CC2CCC(F)(F)CC2)C1 C(=O)(C(C)(F)C(C)(C)F)N1CCOCC(NC(C(c2ccccc2F)OC)=O)C1 CC1CCCc2cc(C(=O)NCC3CN(C(=O)C(F)C(C)(C)O)CCN3C)nn21 C(=O)(C(CCS(C)=O)N(C)C)N1CCC(CNC(C=Cc2ncc(C)[nH]2)=O)C1 c1(OCC(=O)NC(C)CCCNC(=O)CCNC(=O)CO)nn(C)cc1[N+](=O)[O-] C1(C(=O)NCCN(CC(C)O)CC)CN(C(c2oc(CO)cc2C)=O)CC(C)(C)C1 c1(CN2C(C)(C(N3CCC(Br)C3)=O)CC2)c(F)cc(Cl)cc1Br c1(C(=O)OC)ccc(NC(C2CC23CN(C(=O)Cc2ccsc2)C3)=O)cn1 CS(=O)(=O)c1ccc(CNC(=O)CC2CN(C(=O)Cc3cncnc3)C2)nc1 c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(c1nnc(O)nc1O)=O C1(CNC(C(CSC)C)=O)CCC(NC(=O)CSC)CC1 CCCCC(O)C(C)C(=O)N1CCC1C(=O)Nc1ccc(C2CC2)nc1 N1(C(C2CCN(C(c3cnn[nH]3)=O)C2)=O)CCCCCC1CCO N1(c2cc(COC)ncn2)CCCC(NC(c2ccc(C)cc2)=O)CC1 C(=O)(CCC(=O)NC(C)CN(C)C(C1CCCN1Cc1nnn(C)n1)=O)OCC CC12CN(C(c3c(O)cccc3Cl)=O)CC1CN(C(c1cc(C(F)F)no1)=O)C2 c1(C(N2CCCC(CCNC(C(CC#C)O)=O)C2)=O)ccnc2cc(C)ccc12 N1(C(c2nc(OC)nc(O)c2)=O)C2CCC1CN(C(=O)CC1OCCCO1)CC2 Cc1cc(NC(=O)C(C2CCOC2)NC(=O)C2=CCCC2C)c(C)c(C)c1 CC(C)(C(=O)OCC1(Cl)CCC1)Sc1ccccc1 C(=O)(CCCCC#N)NCC(C)CNC(C1CCCCCC1)=O N1(C(COCCOCC)=O)CCCC(CCNC(C2(C)CCCCC2)=O)C1 c1(C(N(CCN(C(=O)CN2CCC(C)(O)C2)C)C)=O)ccc2sc(O)nc2c1 N1(C(c2cncc(C)n2)=O)CCCC(C)C1CCNC(=O)C(F)(F)CC1CC1 c1(CC)nn(C)c(Cl)c1C(=O)NCC(O)CCNC(c1coc(OC)n1)=O CC(C)C(O)C(=O)N1CCCCC1CN(C(=O)CC=C(Cl)Cl)C N1(C(c2cccc(SC)c2)=O)CC2CCN(C(=O)C(C(C)O)N(C)C)C2C1 C1(C)(CC)CC(NC(=O)C2CC2)CN1C(C1(c2cccnc2Cl)CC1)=O C#CCCC(C(=O)NCC(=O)OC)NC(=O)C(CC)CC=C c1(C(=O)Nc2ccnc(OC(C)C)c2F)ccc2c(c1)C(=O)N(C)C2=O c1(CC(=O)NCC2CCN2C(c2cc(Br)cc(F)c2F)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC(C2CCOC2)NC(CC=CCC)=O)c(C)noc1CCC C12(C(N(C)CC3(CNC(c4ccc(N)cc4O)=O)CC3)=O)CCCCC1CCC2 C1(CC(=O)NCCOCCCN(C(C(C)n2ccnc2)=O)C)CCCC1(F)F c1(C(=O)NC2CC(C)N(C(=O)C=CCn3cncn3)C2)cc2ccc(F)cc2o1 C1(C(N(C)CC2CCCC3CC23)=O)CCC(C2CC2)N1C(c1ccccc1Cl)=O C1(C)(C(N(CCCNC(c2ccc(C)s2)=O)C)=O)CCc2ccccc2C1 O=C1OC2CNCC2N1C1CCN(C(c2cc(C(=O)O)co2)=O)CC1 c1(C(=O)NC2CC(CCNC(C3CCCN(C(C)=O)C3)=O)C2)ccc(F)cc1Cl N1(C(CN(C2CCC2)C)=O)CC(NC(=O)CC2CCOCC2)C2CC2C1 Cc1cc(NC(=O)Nc2c(F)cc(OC(F)F)cc2F)c(Br)nc1C C(=O)(C1=CCCCC1)NC(C(=O)NCCCOC(=O)NC)Cc1ccco1 CC(C(=O)N(CCCCN(C(=O)C(C)(C)c1ccsc1)C)C)C1=CCCC1 c1(OC)ccc(C(N2CCN(CCN3CCCCC3)CC2)C)cc1C(C)C N1(C(CCSC)=O)CC2(CNC(=O)Cc3ccon3)CC1CO2 C1(CC=C)CCCN(C(c2coc(CNC(c3c(C)n[nH]c3C)=O)n2)=O)C1 N1(C(C2(C)CCC(O)CC2)=O)CCC2(CCCCN(C(=O)Cc3cscn3)C2)C1 N1(C(CCC2CCCN(C(=O)Cn3cccn3)C2)=O)CC2CCCC(C2)C1 C1(NC(=O)CC2(CO)CC2)CCN(C(=O)CNCc2ccccc2)C(C2CC2)C1 CC1CN(C(c2ccsc2)=O)CCN1C(=O)CC1CC2C=CC1C2 c1(NCCCC=CCCC)ncnc(NC(C2CCC(C)(C)O2)COC)c1C C1(NC(C2(C#N)CCC2)=O)CCCCN(C(C2CC23CCOC3)=O)C1 C(=O)(CCCCCC#N)NC1(CO)CCN(C(c2c(CC)nc(C)o2)=O)C1 C(=O)(C(O)CC(C)(C)C)NCCC(C)NC(c1csnc1Br)=O C1(C(=O)OC)CC2(CCN(c3ccc(Br)cc3[N+](=O)[O-])CC2)CO1 c1(CN2CCC2N(C2CC3OC(=O)CC23)C(=O)OC(C)(C)C)n[nH]c2c1CCSC2 c1(CC)cccc(C(N2CCC(C)(CC(=O)NCCC3CC(=O)N(C)C3)C2)=O)n1 C(=O)(C1=CCCC1C)N1C(CN(C(CN(c2ccc(Cl)cn2)CC)=O)C)CCC1 C(=O)(CC(CC)C(C)(C)C)N(CCCCCC)CCNC(c1csc(=N)[nH]1)=O N1(C(c2n(C)nnc2)=O)CC(CNC(c2cnc(C3CC3)nc2)=O)N2CCC1C2 N1(C(c2ncc(OC)nc2)=O)CC(O)CCC1C(=O)NCCc1ccco1 Cc1c(C(=O)NCC(C)(C)CN(C)C(C2CCS(=O)(=O)N2)=O)ccn1C(C)C C1(C(=O)Nc2cccc(C(C)=O)c2)CC2(C1)CN(Cc1ccn(CCF)n1)C2 C(=O)(C(C)(C)CC1CC1)N1CCC(OCC(=O)NC(CCSCC)C)C1 CCC(CC)CC(F)C(=O)NC12CCC(C(=O)NCc3ncco3)(CC1)C2 CCC(CC(=O)N(CCC(=O)N1CC2CC1CS2=O)OC)C1CCC1 c1(C(=O)NC2C(CNC(c3c(CN(C)C)occ3)=O)C2)ccc(OC(F)F)cn1 CC1C(C)N(C(c2ccn(C)c2)C(=O)NCC2CCC(F)(F)CC2)CCS1=O CCC(C)CCCC(=O)NC1(C)CN(C(=O)CC2(CC)CCOCC2)C1 C1(NC(C(C)C2CCC2)=O)CCN(C(=O)Cc2ccc(Cl)cn2)CC1F c1(C(=O)NCCC(=C)CNC(=O)Cn2ncnn2)cc(S(=O)(=O)CC)cnc1O c1(C(N(CC(CC)NC(C2CCCCN2CC(F)F)=O)C)=O)c(C)n[nH]c1C N1(C(COC(CC)(C)C)=O)CCC(C2CC(NC(C3CC3C(C)C)=O)C2)CC1 c1(Cc2cc(OC)cc(C)c2)cc(F)c(F)c(F)c1.c12cncc(c1)NC2=O c1(C(N2CC(NC(c3n(CC)ccc3)=O)C3C2C3)=O)ccc2nc[nH]c2n1 c1(C(N2CC(OCCNC(=O)CCc3ncc[nH]3)C2)=O)cccc2c1CCOC2 c1(CCCC(=O)N(C(C)CNC2CC(=C3CCC3)C2)C)ccccc1Cl CC1(C)CC(CNC(=O)C=Cc2cccs2)CN1C(=O)CN1CCSCC1 N1(C(C(CC)N(C)C)=O)CCCCC2(CCN(C(=O)C=Cc3cccnc3)C2)C1 N1(C(C2=NOC(C)C2)=O)CC2CC(NC(c3cc(C(F)F)ccn3)=O)CC(C2)C1 C(=O)(CCCC(CC)CC)N1CCC(C(=O)NC(CC=C)(C)C)(CC=C)C1 N1(C(CC(C)O)=O)CC2CC(NC(=O)COCCc3ccccc3)CC1C2 N1(C(c2ccc(C)c(O)n2)=O)CCC2CN(C(=O)CCCCC3CC3)CC12 C(=O)(C1OCCn2ccnc21)NCC1C2CN(C(c3cc(C)nc(C)n3)=O)C1C2 c1(C(=O)NC(C(=O)N(C)Cc2cncnc2)c2ccoc2)ccc2nccn2c1 C1(N2CCCC(C)CC2)CC2(CCN(C(=O)C(c3ccc(Cl)cc3)C)CC2)C1 c1(CC(C)C)cnc(N(C)CCN(C)C(c2cccc(Cl)c2)=O)nc1 C(=O)(CCC(=O)c1ccc(Cl)s1)NC1CC(CNC(=O)C=Cc2ccsc2)C1 c1(C(C)=O)ccc(C(C)=O)cc1F.c12coc(c1)C(=O)NCC1(O)CN(C1)C2=O CC1(C)CC(CNC(C2CCC(=O)C2)=O)CN1C(=O)CC1CC(=O)NC(=O)C1 C#CC1(O)CC(C(N2CCCC2C2(NC(c3cnoc3CC(C)C)=O)CC2)=O)C1 Cc1c(CN2CC(c3cccc(C(F)(F)F)c3)C2)nnn1C1CCCCC1 Cc1sc(C(=O)NC2CCN(CCCNC(C3CCN(C)CC3)=O)C2)c(C)c1C c1(C(=O)NCC(C)(C)NC(CC2(C(=O)OC)CC2)=O)ccc(=N)[nH]c1Cl n1(CC)cc(Br)c(C(=O)NCCN(C(=O)CN2CCC(C)CC2)C2CC2)n1 C(=O)(C1c2ccccc2CN1Cc1c(C)scn1)Nc1cc2ccccc2n1C c1(OC)cc(C)c(C(=O)NC2CC2NC(c2nc(C)sc2Br)=O)cn1 C1(CC(N2C(CNC(c3c(C#N)scc3)=O)CC(F)C2)=O)CN2CCN1CC2 N1(C(CCc2nnc(C)o2)=O)CCN(C(=O)C(C)C(O)CC)CC(C)(F)C1 C1(C(=O)NCCCNC(C(c2cccc(Cl)c2)OC)=O)Cc2cc(F)ccc2O1 c1(NC(C2CC(CC)(CC)C2)=O)[nH]c2ccc(C(=O)NOCCOC)cc2c1C N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCc2ccccc2C1CNC(c1cnsn1)=O N1(C(c2cc(CCOC)on2)=O)CC(N(C(=O)C(CC)(CC)OC)C)C2(CC2)C1 N1(C(C2CN(C)C(=O)C2)=O)CCCC2(CCN(C(=O)C(C)(C)CC(F)F)C2)C1 Cc1ccc(SCC(=O)NCCC2CC(N(C)C)C2)cc1.C12(C)CCN(C1)C2=O N1(C(C2CCCCCC2)C(=O)NCC2CC=CCC2)CCc2sc(Cl)cc2C1 Cc1cc(Cl)c(C(=O)NC2CC3C2CCN3C(=O)C(C)C2CC2)c(Cl)c1 C1(n2cc(-c3n(C)ncn3)nn2)CON(C(=O)C(O)C2CN(CC(F)(F)F)C2)C1 c1(C(=O)NCCCN(C(C2CCCO2)=O)CC)cc(C)cc(OC)c1C CCCCCC(=O)NC(c1ccccc1F)CNC(c1nc(C(C)C)oc1C)=O N1(C(CC(CC)SC)=O)CCCN(C(c2cc(O)n(CC)n2)=O)C(C(C)C)C1 Cc1cc(C(N2CCN(C(c3sccc3Cl)=O)CC(C)C2)=O)c(F)cc1F N1(C(COCC(=O)OC)=O)CCC(C(F)CNC(C2(C)CNC(=O)C2)=O)CC1 Cc1nn(C)c(Cl)c1CC(=O)NC1CN(C(C2CC2F)=O)CCC1C(F)(F)F N1(C(C(=O)NC2CCOCC2)=O)CCCCC1C(N1CCSCC1)=O CCC(C(=O)NCCCC1CCCN1C(c1ccnc(OC)n1)=O)C(C)O c1(CC)cc(Br)cc(CC)c1NC(=O)CC(C)(O)CCC N1(C(C(C(=O)OCC)OC)=O)CC2(CC(C(=O)N(CC(O)C(F)(F)F)C)CO2)C1 C#CCCCCCC(=O)N1CCCC1C=CC(=O)NC1(c2cc[nH]n2)CC1 C(C(=O)NCc1ocnc1C(=O)NC1(C(F)F)CCCC1)(C(C)C)SC CC(=O)C(C)CC(C)C(=O)NC(CC(F)F)C(=O)NCCC(=O)NC1CC1 C(=O)(C1=CCCC1(C)C)N1CCN(C(CCCC(=C)C)=O)C(CCOC)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCCNC(=O)CC2NC(=O)NC2=O)c1Cl C1(CC(=O)NCC2=CCN(C(c3ccsc3Cl)=O)C2)CCC2CC2C1 n1(C(CC)CC)nccc1C(=O)NCC(C1CCOC1)NC(=O)CCSC CCC(CC(=O)NC1CC2CC(C1)CN(C(c1cc(F)n[nH]1)=O)C2)C(C)(C)C C(=O)(CC(C)C(F)F)NCC1(F)CCC(NC(C=C(COC)C)=O)C1 C=C(C)CCC(=O)NC1C2CCN(C(C3CC3c3ccccc3)=O)C12 C1(NC(CCNC(C(C=C)O)=O)=O)CCCC1C1CC1 N1(C(c2ccc(CCCCCC)s2)=O)CC(NCC2CCC(=O)N2C)C(SC)C1 C1(CN(C(C(C)OCCC=C)=O)CC)CCN(C(c2cccc(C)c2)=O)CC1 C1(C(N2CCC(O)(C(C)N)C2)=O)CCS(=O)(=O)C1(C)C.C(C(F)(F)F)C1(C(=O)NC)CC1 c1(C(F)F)cc(N(C2CCC2)C2CSC2)n2ncnc2n1 CN1C(=O)NCC1C(=O)NC1CCC(CNC(=O)CN2CCNC(=O)C2)C1 c1(CN2C(C(=O)Nc3c(C(=O)OC)n(C)nc3)COCC2)ccc(F)c(F)c1F c1(C(=O)NC(C)C(=O)Nc2ccsc2)n[nH]c2c1COC2 N1(C(C(C)NC(C)=O)=O)CC2(CCN2C(c2cnc(O)c(F)c2)=O)C1 Cc1c(C(=O)NOCC(N2CC3C(C2)C3(C)C)=O)cccc1C#N N1(c2nc(CC)nc(=N)[nH]2)CCC2(CCN(C(c3ccc(C(F)F)o3)=O)C2)C1 C(C)(c1cnccn1)=Cc1c(C(C)=O)cccn1.C12CCCN(C1)C(=O)CN(C)C2 c1(CN2CC3N(C(CCC)=O)C3C2)ccc2c(c1)C=CC(C)(C)O2 c1(C(=O)NC2C3CN(C(c4cc(OC)nc(C)c4)=O)C2C3)cc2ccccn2n1 c1(C(C)=O)ccccc1C(=O)NCCC1CCCN(C(c2ccc(Br)cc2)=O)C1 Cc1cncc(CC(=O)NCC(O)CNC(c2ccc(C(N)=O)[nH]2)=O)c1 N1(C(CCC(C)(C)C)=O)CCCC2CN(c3nc4ccc(N)cc4s3)CCC12 N1(c2n(CCCOC)c(C3CCCCN3C)nn2)CCN2C(=O)C(=O)NCC2C1 N1(C(C(CC=C)C)=O)CC2CCC1C(NC(=O)CNC(c1cscn1)=O)C2 c1(OC)cc(C(N2CCCC2(C)C(N2CCC(O)C(C)C2)=O)=O)cc(Br)c1Cl C(=O)(C1CCCn2nccc21)N(CCC(c1cccs1)NC(=O)C=CCO)C N1(C(CC2N(C(C)=O)CCC2)=O)CCN(C(c2csc(C(F)F)c2)=O)CC1C c1(OCCCCC)ccc(CC(=O)NCC(CC)NC(=O)C=C(Cl)Cl)cc1 C1(NC(C(C)NC(N)=O)=O)(CO)CCCN(C(c2ccc(CO)o2)=O)C1 N1(C(=O)Cc2c[nH]nc2O)CCC2CN(C(C3(c4cc[nH]n4)CC3)=O)CC2C1 CCC(C)C(O)CC(=O)N1CC(C(N2CC3CCCC2C3CO)=O)(SC)C1 N1(C(CC#CC)C)C(=O)CCN(CC(C(C)C)NS(C)(=O)=O)C1=O.c12ccc(o1)s2 C(=O)(C(F)(F)CNC(C)=O)Nc1cccc(CNC(C=COCC)=O)c1 C(C(C)C)(C(O)C(=O)NC1CCC(C(=O)NOCc2cc(O)ccc2C)C1)OC C(=O)(C1=CCC(C)CC1)NC1C(OC)CN(C(c2ccc(F)s2)=O)C1 c1(N2CCCC(NC(Cn3nnc(C)n3)=O)C2C)c(C#N)cccc1[N+](=O)[O-] CC(C)C(C)C(CNC(=O)Cc1csnn1)NC(c1cn(C2CCC2)nn1)=O Cc1c(Br)ccc(C(=O)NC(C)CCN(C)C(C2CC2F)=O)c1F N1(C(Cn2cnc(=N)[nH]2)=O)CCCCC(CNC(C2CC(S(N)(=O)=O)C2)=O)C1 c1(C(N(CC(C)N(C(C(CC#C)C2CC2)=O)C)C)=O)cc2n(n1)CCCC2=O N1(C(c2ccc(C(OC)OC)o2)=O)CCCCCC(NC(=O)CCS(C)=O)C1 C1(C(=O)NC2(CCNC(=O)C(O)c3ccsc3)CC2)CCC2CC12 CC1C(C)N(C(c2nncn2C)C(=O)NCC2CCCO2)CCS1(=O)=O C12C3CN(CC13)C(=O)CN(C)C(=O)NC(=O)C2.CCC(C)(O)C1CC1 C12(CNC(Cc3nc(C)sc3)=O)CCC1CCN2C(=O)C=Cc1cnc[nH]1 N1(c2c(C)cncn2)CCN(Cc2c(C)cccc2Br)CC1C#N c1(CC)onc(C(=O)NCC#CC(=O)N2CCC(COC)C2)c1C CC1(C)CCCC(CC(=O)N(CCCO)CC(F)F)O1 Cc1cccc(N2CCCC(C(=O)NCc3ccccc3O)C2)c1 C(CCCC(=O)NC(CCN(C)C(c1sc(F)cc1C)=O)C(C)C)OC N(C(=NCc1ccc(F)cc1)NCC(C)(F)F)Cc1n(C)cnn1 c1(OC)ccc(C(=O)C(=O)NCC(C)NC(c2cscc2F)=O)cc1 C1(O)(CNC(C(C)NC(CC)=O)=O)CCN(C(c2cnc(Cl)[nH]2)=O)CC1 c1(CCC(=O)N(C2CCN(C(Cc3cc(C)[nH]n3)=O)C2)C)cccc(N(C)C)c1 C=CCC(C)(C)C(=O)NC1CCC(CNC(c2c(C)nn(C)c2C)=O)CC1 Cc1oc([N+](=O)[O-])cc1C(=O)NC12CC1CN(C(C1CCC(=O)N1)=O)C2 c1(C(=O)O)ccc(C#N)nc1C.c1(OCc2cn(C(C)=O)nn2)cn(CC)c(C)n1 c1(CC(=O)N(C2CCN(C(=O)Cn3cncn3)CC2)C)ccc2ncsc2c1 C1(NC(COCCC(C)C)=O)CC(CNC(c2cc(F)ccc2Cl)=O)C12CCC2 c1(C(N2CCC(NC(CCOCCOC)=O)(CO)C2)=O)nncc2c1CCCC2 N1(C(c2c(C)ncnc2)=O)CCCCC2(C1)CN(C(c1cc(F)ccc1Cl)=O)C2 C1(C)(NC(CNC(C(CC)C)=O)=O)CCCN(C(c2ccoc2)=O)C1 N1(C(C(CCC)N(C)C)=O)CCC2C(CCN2C(c2cc[nH]n2)=O)C1 n1(CCOC)cc(C(=O)NCC(C(C)C)NC(C2(OC)CCOC2)=O)cn1 C1(CNC(C(C)(O)C2CC2)=O)CC2(CCN(C(C3CC(C#N)C3)=O)CC2)CO1 N1(C(C2(C)C(C)C2)=O)CCC(F)(F)C(CNC(=O)CCc2cn[nH]c2)C1 C1(=O)C(O)CSCCC(=O)N(C)CCCN1C.C(COCCOCCO)OC C=C(Cl)CC(C(=O)N1CCC(F)(CO)C1)NC(c1coc(CC)n1)=O c1(C(N2CCC3(C(C(=O)NCc4nnn(CC)n4)C3)C2)=O)cccn2cncc12 N1(C(C(C(C)(C)O)NC(COCC=C)=O)=O)CC(C)N(C)C(C)C1 C1(C(=O)NOCc2cn(C)cn2)(CC=C)CCCN1C(C1COC(=O)N1)=O CCCC(C(=O)N1CC(C(C)(C)O)(CNC(=O)C(=Cc2ccccn2)C)C1)OC CC1CCC(=CC(=O)NC(C)(C)CC=CC(=O)NC2COCC2F)CC1 c1(NC(c2cc(F)cnc2O)=O)ncc(Cl)cc1Cl.C12CCCCC1CNC2=O C1(NC(c2c(C)n(C(C)C)cc2)=O)CCC(C)N(C(c2c[nH]cc(Cl)c2=O)=O)C1 C(=O)(CC(C)(C)C(=O)NCC1CN(C(=O)COC2CCOC2)CC1O)OC CCCC(C)(O)C(=O)NC(C)CC1CCN(C(C2CCNC2=O)=O)CC1 C1(CNC(C2CCCC(NC(C=CC)=O)C2)=O)CN(C(=O)OC)CCN1C C12(CNC(C3C(C)OC(C)C3)=O)CC(CO1)N(C(c1cn(C3CC3)nn1)=O)C2 N1(C(C2N(C(C(C)OCC=C)=O)CC=C2)=O)CCOC(C(=C)C)C1 C1(C(N2CCC(CN(C(C34CCCC3C4)=O)CC)CC2)=O)CC(=O)NC(=O)N1 c1(NC(C2N(Cc3cccc(C)c3)CCNC2)=O)cc(Cl)cc(Cl)c1Br C1(CNC(CNC(CCCCC)=O)=O)CC(F)(F)CN1C(=O)CC1CC2(CC2)C1 CN1CCN(C(=O)C=CC2CC2)C(CNC(c2csc(-c3cnccn3)n2)=O)C1 C1(C(N2CCC(CN(C)CC)C2)=O)COC2(C1)CN(C(=O)C(C)(C)CSC)C2 C1(NC(CCCCC)=O)CC(C2CCN(C(c3c(C)cc(F)cc3C)=O)C2)C1 c1(C(=O)NCC(C2CCCC2)NC(c2c(C)n(C)nc2)=O)ccc(F)cc1Cl c1(NC(C(=O)NC2CCN(C)C2=O)=O)cc(Br)cc2[nH]ccc12 c1(C(=O)NC(C(=O)NCC(C)(C)SC)CC2CC2)c[nH]c(=O)cn1 N1(C(C2CCC(C)C2)=O)CC2CCCC(NC(c3ncc(Cl)n3C)=O)C2C1 C1(CC(N)=O)CCCC(NC(N2CCOCC2CCC(F)(F)F)=O)C1 c1(CNC(C2C(C)(C)C2)=O)nnc2n1CCN(C(=O)Cc1cc[nH]c(=N)c1)C2 N1(C(c2c(OC)cccn2)=O)CCCC(C)(NC(c2ncc(Cl)cc2F)=O)C1 N1(C(C(C)=CC=C)=O)CCOC(CC(N2CCC2CF)=O)C1 C1(C(N(CC(=O)O)Cc2cn(Cc3cnc(C)nc3)nn2)=O)CN2CCN1CC2 c1(C(=O)OC)nc(=NCCN(C(c2cc3sccc3cn2)=O)C(C)C)c(C)c(C)[nH]1 N1(C(C2(CF)CCC2)=O)CC2CCC(C1)N(C(=O)Cc1ccsn1)C2 c1(C2C(C(=O)NCCN(C(C)C)C(C3CCC4CC34)=O)C2)cccc([N+](=O)[O-])c1 c1(CC(N2CCCC(NC(c3n[nH]cc3F)=O)C2)=O)c(Cl)cccc1Cl c1(C(=O)NCC(CNC(C2CC(SC)C2)=O)O)ccc2c(c1)OCCO2 N1(C(CC)=O)CCN(C(C2CCCN2S(=O)(=O)CC)=O)CC1Cc1ccccc1 N(C1CCOc2c(C)cccc21)C(c1n(CC)nnn1)C1(C(C)C)CC1 Cc1cc(C(=O)NCC(C)(C)CNC(c2cc(O)n(C)n2)=O)cnn1 c1(OCC=C)ccccc1CN1CC2C(C(=O)NC3CCC(C(N)=O)CC3)C2C1 c1(OC)c(C(=O)NC2CC(O)CN(C(=O)Cc3ncoc3C)C2)ccc(Cl)c1Cl C=CCCCC(C(=O)OC)OC.c12cc(cc(N(C)C)c1)NC(=O)N2 C1(NC(C(CC=CC)CC)=O)CCN(C(=O)Cc2c[nH]nc2O)CC12CCC2 O=C1NCc2c(C(N3CC4CC(NC(C56CC5C6)=O)CC3C4)=O)cccc21 c1(NCC2CCN(CC)C2)[nH]c(=NCc2ccc(C)o2)nc2sccc12 CC1CCN(C(C2CCCCC2(C)C)=O)CCN1c1[nH]cnc2nc(Cl)cc1-2 c1(CN(C(=O)CC2CCC(C)(C)C2)C)cc(Cl)cc(Cl)c1 CC1CCC(NC(=O)Cc2cnoc2)CN1C(=O)CCOC1CC1 CC1CC(NC(=O)CC(C)(O)c2ccccc2)CN1C(C1(c2ccncc2)CC1)=O C=CC1(CNC(=O)CC=CCNC(C2(Cl)CC2C(C)=O)=O)CCOCC1 C1(=CCNC(c2cnc(C(C)(C)C)s2)=O)CCN(c2nc(C(F)(F)F)ns2)CC1 CC(C)CC(C(=O)NC1C=CC(CNC(C2CCCC2C)=O)C1)C(N)=O c1(CC)ncnc(NC2CC2NC(N2CCCC2c2ccc(Cl)cc2)=O)c1F c1(C(=O)NCCCC(C)NC(COCCC#C)=O)cc(-n2ccnc2)ccc1O CC(CN=c1[nH]c(=N)[nH]c(=NCc2cccc(Cl)c2Br)[nH]1)C(C)(F)F C(=O)(C(CC)CC(C)C)NC1(CC=C)CN(C(C2(OCC)CCSC2)=O)C1 n1(CCC(=O)NCCC(C)NC(c2n(CC)ncc2)=O)ccc2cc(Cl)ccc12 O=S(=O)(c1cccc(N2CCC3CCC(C2)S3)n1)N1CCCC2COCC12 c1(OC)cc(Cl)cc(CNC2CN(c3cc(C#N)ncn3)CC2O)c1O c1(OCCC(=O)N(CCCNC(C2C3CCCC23)=O)C2CC2)ccccc1Cl O=C(C1=Cc2ccccc2C1)N1CC2CC1CCN2C(C1CC2CC2CO1)=O c1(C(N2CC(C(=O)OC)C(C)(C)C2)C(=O)NCC(F)F)cc(Cl)c(F)c(Cl)c1 C1(CC)CN(C(=O)CC2CN(C(c3ccnc(OC)c3)=O)CCO2)CCN1C C1(CC(=O)NCCC2N(C(c3cncc(C)n3)=O)CCSC2)CCCCC12CC2 c1(C(N2CCC(CNC(=O)Cn3ccnn3)C2)=O)ccc(-c2cnn[nH]2)cc1 c1(N2CCCC(CNC(CSCCCSSC)=O)CC2)ccc([N+](=O)[O-])cn1 CC1(C2CCCN(C(C34CCCC3CCN4C(C3CCNC3=O)=O)=O)C2)CC1 S(=O)(=O)(c1ccc(N2CCC(C(F)F)C2)cc1Br)N1CC(CC(C)(C)C)OCC1 C1(NC(C2(OC)CCOC2)=O)CCN(C(c2cnc(CC3CC3)s2)=O)CC(C)(C)C1 N1(C(C2CC(OCC)C2)C(=O)NC(C)CC)CCOCC1 Cc1sc(Cl)nc1C(=O)NCC(C)(C1CCC1)NC(=O)CCCn1ccnn1 CC(C(=O)NCC1CCC(NC(c2coc(CO)c2)=O)CC1)C(=O)N1CCOCC1 c1(N2CCCC(C(C)O)C2)nc(=NCc2conc2Br)[nH]c2cccc(F)c12 CCC(C)(C)C(C)CC(=O)NC(C1CCCN1C(=O)CCS(C)(=O)=O)C c1(C(N2CCCCC(NC(C(CC)=CC)=O)C2)=O)cnc(O)c2cncn12 C1(C(=O)NCC2(CNC(CN(C)C(N)=O)=O)CCC2)COc2cc(O)ccc2C1 c1(C(N(CCC(C(C)C)NC(CSCCC)=O)C)=O)cc2c(F)c(F)ccc2[nH]1 C1(c2ccccc2)(NC(CC(C)C)=O)CCN(C(c2ccc(C(C)C)cn2)=O)C1 CC(CCO)C(=O)N(C)CCN(C)C(c1nnn(C)c1N)=O C1(N(C(CN(C(C)=O)C)=O)C)CN(C(=O)C(F)C2CCOC2)C1 N1(C(C=C(CCC)C)=O)CCC2(CC1)CC2NC(c1ccc(F)c(CC)c1)=O C(=O)(C1=CCCCC1C)N1CCCC(C(=O)NCCn2cccn2)(CC)C1 C12(NC(=O)C(F)F)CCN(C(=O)Cn3nc(C(F)F)cc3C3CC3)CC1C2 c1(C(N2CCC(COC)C2)C(=O)NCc2cccs2)cc(Br)cc2cccnc12 c1(CC)ncccc1C(=O)NC(C)(C)CNC(=O)C(c1ccc(Cl)nc1)(C)C C(CCC(C)C)=CC(=O)NCC1N(C(C2(C(=O)OCC)CC2)=O)CC1 c1(NC(C2CCC(NC(C3(CCCF)CC3)=O)CC2)=O)cc(Cl)ccc1O N1(C(C(n2ncc(C)c2)C)=O)CCCN(C(=O)CC(C)C)CCC1 c1(C(=O)NCC2(CNC(C3CCCC3O)=O)CC2)cnc2nc(O)nc(O)c2c1 C(=O)(C(C#N)CC1CC1)NCCCNC(=O)CCN(CCC(C)OC)C(C)C c1(C(C)OCC)nc(-c2cc(CO)n(C)n2)n(Cc2cccc(NC(C)C)c2)n1 C(=O)(C(F)C(F)(F)F)NCC(CNC(C1C(CN(C)C)C1)=O)(C)C c1(CNC(c2ccc(N3CCOCC3=O)cc2)=O)ccc(S(=O)(=O)CCO)cc1 C1(CCC(N2CC(CC=C)(NC(=O)C(=Cc3cccs3)C)C2)=O)CCCCN1C CC1(C)COCCC1CNC(=NCC1CCC(F)(F)C1)NC1CCC1 N1(C(Cc2cc(C(C)C)no2)=O)CCN(C(=O)CCc2cocn2)CC12CCC2 CC1(C)CN(C(C23CCCC2C3(F)F)=O)CCC1C(N1CCSCC1(C)C)=O c1(C(N(C(C(=O)NCC(CCC)O)C)CCC)=O)ccc2cc[nH]c2c1 C(=O)(C1CCCc2nnn(C)c21)NC1CC(C(C)NC(c2ccc(F)cn2)=O)C1 Cc1cc(C(=O)NCC(C2CC2)NC(C2CCCCS2)=O)[nH]c1C c1(C(N2CC3C(C(=O)NCc4n(C)cnn4)(C3)C2)=O)cc2cc(F)ccc2s1 C(=O)(C(C)(C)CN(C)C(c1cc(CC)no1)=O)NC1(CCCC)CC1 C1(NC(c2cn(CC)nc2)=O)CC(O)CN(C(=O)C(c2cncn2C)O)C1 C(=O)(CC(C)(C)C(F)F)NC1CC(NC(c2c(N(C)C)ccc(F)c2)=O)C1 C(=O)(C1=CC2CCCCC12)NCC1CCC(NC(CC(C=C)CC)=O)CC1 C12(CNC(c3cnc(C(C)OC)s3)=O)CCC(CN(C(C3CC3(F)F)=O)C1)C2 CC1C(NC(=O)C(CO)c2ccccc2)CCN1C(=O)CCC1CCCCO1 C(C(C)(O)CC(=O)N1CCOCC(CNC(C2CC3(CCC3)C2)=O)C1)OC C1(CCC(=O)N(C)CC2CCN(C(Cc3c(C)ccs3)=O)C2)CCCC(=O)N1 C1(C(=O)NCC2C(NC(CC=C)=O)C2)CCOC1c1nncn1CC Cc1ccc2cc(C(=O)NC(C3CCN(C(=O)C(C)(C)C(C)C)C3)C)oc2c1 C1(C(N(CCCN(C)C)CC)=O)CCC(NC(=O)C(C)CCOC)CC1 Cc1cc(C#N)sc1C(N1CCCN(C(=O)C=NOC)CC1)=O C(=O)(C#CC1CCOCC1)N1C(C)CCC(NC(c2c(O)nnc(C)c2C)=O)C1 c1(NC(CCNS(CC)(=O)=O)=O)ccc2cnnc(O)c2c1 N#Cc1cc(C(=O)NCC2(CO)CCCCCC2)ccc1Br N1(C(CCN(C(C(CCC)N(C)C)=O)CCO)=O)CCCOC(C)(C)C1 c1(OC(CC)CNC(c2coc(Br)c2)c2nnnn2CC(F)F)ccccc1Cl Cc1cc(NC(c2cc(Br)cn2C)c2nnnn2-c2ccccc2)cnc1Cl C1(C(=O)NCC(C)NC(C2CC=CCO2)=O)Cc2cc(F)cc(F)c2O1 CN1CC(C(=O)NCCC2(O)CN(C(c3cnc(S)nc3)=O)C2)NC1=O C#CCCCCC(c1nnnn1CC(F)F)NCc1occc1CC CCC(CCC(=O)NC1CC12CC(NC(=O)Cc1ccc(OC)c(Cl)c1)C2)OC c1(CN2C(c3cccs3)CCC(C)C2)n[nH]c2ccccc12 C1(CNC(CCC(C)OCC)=O)CCN(C(c2coc(Cl)c2)=O)C(C)C1 C1(C(=O)NC(C)CCNC(=O)CCCC2CCOCC2)CCC(C(C)(C)O)CC1 Cc1nc(C(=O)NC2CC(NC(C3CCCN3C3CC3)=O)C2)c(C(F)(F)F)[nH]1 N1(C(c2c(OC)cccn2)=O)CCC12CN(C(=O)CC1C=CCCC1)C2 c1(CC)nc(C(N2C3CCC2CN(C(=O)CSCC(N)=O)C3)=O)c2ccccn12 c1(OC)cc(CN=C(NCC2CC2)N(C)C)cc(OC)c1C C1(COC)(CNC(=O)CO)CCN(C(=O)CCc2cccnc2)C1 c1(NCC(C)CCCO)ccc(Br)c2cnn(C)c12 CCC(C)C(=O)C(=O)N1CCC(C(N2CC(CO)(CF)C2)=O)O1 N1(C(C(C(C)C)SC)=O)CCC2CCC(NC(c3cc(C)nc(Cl)c3)=O)C1C2 C1(CNC(C2N(C)C(=O)CC2)=O)CCN(C(=O)Cc2cn(C)nn2)C12CCC2 c1(C(N(C2CCC(NC(CC3C(C)CCO3)=O)CC2)C)=O)cc(F)cc(Cl)c1 CCCCCCC(=O)NCC12CC1CN(C(c1c(OC)ccnc1OC)=O)C2 N(C1CN(C(c2cccc(O)n2)=O)Cc2ccccc21)C(C(C)(O)C(F)(F)F)=O C1(NC(C(CC)CC)=O)COC2C(NC(c3nc(C)n(C)c3C)=O)COC12 C1(OC)CN(C(=O)C(C(C)C)NC(=O)CN2CSCC2=O)CC1(C)C C1(CS(C)(=O)=O)(NC(=O)NCC2CCC3(CC3)CO2)CCCCCC1 Cc1nnsc1C(=O)N(C(C)(C(=O)NC(CO)C1CC1)C1CC1)C C1(NC(C2(C)CCC(C)C2)=O)COC2(C1)CN(C(=O)Cc1c(Cl)cnn1C)C2 c1(NC(C(=O)N(CC(CC)OC)C)=O)cc(OC)c(S(N)(=O)=O)s1 C(=O)(CCCCC(=O)N1CCCC(CO)(NC(C2CN3CCN2CC3)=O)C1)OC C1(C(=O)NC2C(CC)CC2)CCC(CNC(c2ccc(C)o2)=O)C1 C12(C(N3CCC(N(C(=O)CSCCOC)CCC)C3)=O)CC(CO)(C1)OC2C N1(C(CN(C(CC(C)(C)C2CC2)=O)C2CC2)=O)CCOC2C(O)CC12 CC(C)CC(C)(CO)NC(C1CCCCN1C(C1OCC2CCCC12)=O)=O C1(C2CC(n3cc(CC(C(=O)O)NC(c4nc(CC)oc4)=O)nn3)C2)CCCCN1C c1(CC)nccnc1C(=O)NC(C1(C(=O)N(CCCCC(C)C)CC)CC1)C c1(C(=O)NC2CCN(C(=O)CSCc3ncc[nH]3)C2)cc(Cl)cc2ccncc12 C(CCCCCNC(=O)Cc1nncn1C)N(C)C(C1CCS(=O)(=O)C1)=O c1(C(N2C(C)(CNC(CC=C=C)=O)CCC2)=O)ccc2[nH]c(=O)cnc2c1 c1(N(C(=O)CC2CCN(C(=O)CN3CCCCC3)C2)C)ccc(Cl)c(F)c1 c1(C(N)=O)cnc(C(=O)NCC(=C2CN(C(=O)CC3CCS(=O)(=O)C3)C2)F)cn1 CC#CCC(C)NC(=O)C(C1CC1)N(C(=O)C(c1ccn(C)c1)C)C C1(NC(C(F)=CCC)=O)CCCN(C(c2cccc(C(C)=O)c2O)=O)C1C c1(OC)nccc(C(N2CSCC2C(=O)NC(c2cnccc2C)C)=O)n1 CC(C)(C)C(O)C(=O)NCC12CC1CN(C(=O)Cc1nc[nH]n1)C2 C(CCCC(C)C)(C(=O)NCCOC)N1CCN(CC(CC)O)CC1 Cc1nc(CCC(N2CC(CNC(=O)CCc3cc(Cl)no3)C(O)C2)=O)oc1C c1(C(=O)NC2C=CCN(C(CCCNC(N)=O)=O)C2)cc2cccc(Cl)c2[nH]1 c1(C(=O)NCC2(NC(c3nc(Br)c[nH]3)=O)CC2)c(Cl)ccc2ncccc12 c1(C(=O)NC2C(C(=O)NC3C(=O)NCC3)CCCC2)ccc2nccnc2c1 Cc1cc(CN2CCOC(C3CC3)C2)nc(N(C)C)n1 N1(C(c2c(C)cn(C)c2)=O)CCCC(C)(C)C1CNC(=O)CC(C)c1ccco1 c1(C(=O)NCC2C(C)CCN(C(=O)C(N)=O)C2)ccc2sccc2c1 C1(F)(C(=O)NC2CCC(NC(C3(C)CCC3)=O)C2)CS(=O)(=O)CC12CCC2 c1(N(C2CNCC2C#N)C(CCc2ccc(OC)nc2)=O)ncnc2c1CCCC2 N1(C(C(C)(C)C)=O)CC(NC(=O)CCCCc2cnc[nH]2)C2(CC2)C1 c1(C(=O)NC(CCNC(c2nc(C)oc2)=O)C)c[nH]c2nccc(Cl)c12 C1(NC(c2n(CCC(=O)OCC)nnn2)c2sccc2C)CCCCCC1 C1(C(N(CCC(O)C(=O)NC2CC(C)(C)C2)C)=O)CCCC2(CC2)C1 N1(C(CNC(CC)=O)=O)CCC(C)C(NC(=O)CC(C(F)F)C(F)(F)F)C1 N1(C(c2nc(C(C)NC(C3CCCCC3C)=O)oc2)=O)CC(C)CCCC1C C(c1ccccn1)=C(C)C(=O)NC(C)CNC(c1ccnc(N(C)C)c1)=O n1(CC)ncc(Cl)c1C(N1CCCC(C(C)(O)CNC(=O)Cn2nccn2)C1)=O c1(CC)ccccc1CCNC(N1CCCC(CNC(=O)C(C)NC(C)=O)C1)=O C1(NC(c2ccc(OC)cc2OC)=O)CN(C(=O)C(O)C(C)(C)C)C2(CCC2)C1 c1(CNC)cccc(N(C)C)c1.C12CCCN1C(=O)NCC(C)C2 N1(C(c2nc(CCC)oc2)=O)CCC(C(C)C)CC1CNC(=O)COC(F)(F)F c1(C(=O)NC(c2ccccn2)CC)nc(CNC(C2C(C)(C)C2(F)F)=O)oc1C N1(C(CCCOCCC)=O)CC(O)CC1(C)C(N1CCC(N2CCCC2)C1)=O C1(C(N2CC(CCCCNC(C(CC)OC)=O)C2)=O)CN(CP(C)(C)=O)C1 c1(C(N2C(C)CN(C(=O)Cn3cc(C(F)F)cn3)CC2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NCC2CC(CNC(CCCOC)=O)OC2)cc(Cl)cc(Cl)c1 c1(OC)cc(C(=O)NC(C2CCCN2C(C2OCC2(C)C)=O)C)ccc1C(N)=O N1(c2nnc(C(=O)NCCC)n2Cc2ccn(C(C)C)n2)CCC(S(C)(=O)=O)C1 CC1(C)CN(C(C2CC(F)(CO)C2)=O)C1C1CCN(C(C2C=CCC2)=O)CC1 N1(C(CC(=O)OC)=O)CCN2C(=O)C(NC(c3cncc(C)c3C)=O)CC2C1 n1(C(C(=O)NCC2(NC(CCCc3onc(C)n3)=O)CCC2)C)nc(C)cc1C c1(CC(N2CC(CCNC(=O)Cn3ncnn3)OCC2)=O)cc(F)c(F)cc1F C1(C(N2CC3CC2C3)C(=O)NCCSC)CCC(CCC(C)C)CC1 C1(NC(c2sccc2C2CC2)=O)(CNC(=O)CC2CCC2)CCCC1 CC1OCCN(C(c2ccncc2O)=O)C1C(=O)NCCC1(C)CC1(F)F CC(C)C(C(=O)N1CC2CCN(C(C3CC4CC3CC4(F)F)=O)C2C1)C(C)C CCC(CC)C(C(=O)NC(C)CC1CN(C(c2c[nH]nc2C(C)(C)C)=O)C1)OC c1(CNC(CCOC)=O)csc(C(=O)NC2CCN(CCF)C2)c1 C1(C(=O)NC2CC(CNC(C(CCSC)O)=O)C2)SC2C=CC1CC2 N1(C(c2c(OC)cccc2)=O)CC(CNC(=O)C(C)N(C)C(C)=O)C2(CC2)C1 c1(NCC(c2ccc(C(C)C)cc2)C)nncc2ccccc12 Cn1cc(C(=O)NC2CC2NC(C23CCCCC2NC(=O)C3)=O)c(=O)n(C)c1=O C1(C)(C(=O)NCC(CC)NC(=O)C(O)Cc2cnc[nH]2)CCCCNC1=O C1(CC(=O)NCc2c(C)nn(C)c2)CN(C(C2CCC3CC23)=O)C(C)(C)C1 c1(C(=O)NC2C=CCN(C(CC=C(C)C)=O)C2)c[nH]c2c(F)cccc2c1=O C1(C)(NC(C2CCC(NC(c3c(OC)n[nH]c3)=O)C2)=O)CCCCCC1 C(CN=C(NCC1CCCCCCC1)NCC1CCC(C)O1)OCC=C n1(CC)cncc1CC(=O)NCCCOCCOCCNC(C12COCC1C2)=O c1(OCC)cc(C(=O)N(C2(C(=O)NCC(c3n[nH]c(C)n3)C)CC2)C)[nH]n1 N1(C(=O)Cc2csnn2)CCC2CN(C(C3CCCC(F)(F)C3)=O)CC2C1 C(=O)(C1Cc2ccccc21)NC1CCC(C(=O)NC2CC(C)C2)C1 c1(C(N(C(CCC(C2CCCCC2)=O)=O)C2CC2)=O)cnc2ccc(Cl)cn2c1=O C1(CCCC)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CCCc1ccc(C)s1 Cc1cc(C(=O)N(C(C(=O)NC2CC3(CCC3)C2O)C2CC2)C)c(O)nn1 C=CCC(C)(CC)C(=O)N1CCC(C(=O)NCCc2cnco2)O1 Cc1cccc(C(N2CC(NC(=O)CCSC3CC3c3ccccc3)C(C)C2)=O)c1 c1(CC)c(C(N2CCOC(CC(=O)NCc3nnn(C)n3)C2)=O)nnn1C C1(NC(=O)NCCOc2c(C)occc2=O)CC(C)CC(C)(C)C1 C1(C(N2CC(CC(C(=O)NCCS(C)(=N)=O)F)C2)=O)CC2(CC2)CO1 Nc1cnc(C(=O)NCCCCC(=O)NCCC2(O)CCC2)cn1 CC1(NC(c2ccc(O)nc2)=O)CCN(C(C2CCN2C2CCCC2)=O)CC1 C1(CCNC(CC=CC=C)=O)CCN(C(c2scc(OC)c2OC)=O)C(C)C1 C(=O)(C(C)C(C)(C)C)NC1(CC=C)CCN(C(=O)CCc2ccccc2F)C1 N1(C(CCC(C)NC(=O)CNC(=O)CP(C)(C)=O)=O)CCc2ccccc21 N1(C(COC2CC(NC(c3c(CC)cncc3)=O)C2)=O)CCOC(C)(C)C1 Cc1cc(NC(=O)C(c2ccc(Cl)cc2Cl)O)ccc1NC(=O)C1=CCC1 C(=O)(N=c1[nH][nH]c2c(Cl)cccc12)C1N(C(CC(CC)O)=O)CC(F)C1 c1(C(N2CCC(C(C)NC(c3nn(C)cc3Cl)=O)C2)=O)ncncc1F N1(C(C(c2ccc(Br)cc2)CC)=O)CC2CCC2(C)C1 N1(C(CCCC#C)=O)CCC2CCC12CNC(=O)CNS(C)(=O)=O c1(C(=O)NC2C(CC)CN(C(=O)C=C(Cl)Cl)CC2)cc2cccnn2n1 C#CCCCC(=O)NC(C)CCNC(=O)CCNC(=O)C(CC)CC C1(C(N2CCC(F)(F)C2)=O)CN(C(=O)CCc2nncs2)C2(CCC2)C1 Cc1cc(C(=O)NC2CCCC23CCN(C(=O)C(C)(C)F)C3)c(N)c([N+](=O)[O-])c1 Cc1nc2c([nH]1)CC(C(N1CCC(C(F)F)(CNC(c3cnsn3)=O)C1)=O)CC2 c1(C(=O)NCC(CNC(c2cc(Cl)ns2)=O)O)cn2c(n1)CCCC2 CN(S(N)(=O)=O)CC(=O)NC1COCC1NC(=O)CCc1ccsc1 c1(C(CC(C)O)C2CC2)nc(Cc2ccc(C(N)=O)cc2)nn1-c1cnnn1C N1(C(C2C(C)C2)=O)CCN(C)CC1CNC(=O)C(c1ccccc1)C Cc1cc(=NCC2CCC(NC(c3cccnc3-n3cccn3)=O)C2)[nH]c(Cl)n1 Cc1cc(C(N2CCC(O)(C(C)NC(c3ccc(Cl)o3)=O)C2)=O)ccc1C(C)C c1(CC(=O)NCC(C2CC2)NC(C2(N(C)C)CC2)=O)c(Cl)cccc1Br C(CC(C(=O)N1CC2CC1CS2)NC(c1n[nH]c(=N)[nH]1)=O)OC N1(C(C23CCC(CN(C(C4CCC(C)(C)C4)=O)C2)C3)=O)CC2(COC(C)(C)C2)C1 C(=O)(C1=CNC2=NCCC2=C1)N1CCC(CNC(=O)C(F)C(F)(F)F)(CO)C1 c1(CC)ncc(C(=O)N(CC(CC)NC(=O)CNC(C)=O)CC)[nH]1 c1(C(N2C3(CCN(c4ncc(C)cn4)CC3)CC2)=O)n[nH]c2ccc(C#N)cc12 C(C(=O)NC1CCOC1)(C1=NOC2CC12)N1CCC(C)(CC(F)F)C1 C(=O)(C(C(C)CC)NC(N)=O)N(CCC)CCNC(C12CC(O)C1C2)=O N1(C(CCC(C)=O)=O)CCC(CNC(c2ccoc2)=O)C1(C)C c1(C(N2CCCC(NC(C3CC4C(C)(C)C4C3)=O)C2)=O)ccc(Cl)c(Cl)c1O CC1CN(C(=O)C(C2(O)CCCC2)F)CCC1Nc1nccc(C#N)n1 C1(C(=O)NCc2c(OC)n(C)nc2C)CCn2c(Br)cnc2C1 C1(CNC(Cn2ncc(CC)c2)=O)C2CC1N(C(=O)CC1(c3ccon3)CCC1)C2 c1(SC)ncc(C(=O)N(C(CNC(=O)CCCc2ccccc2)C2CC2)C)s1 C1(C(N(C2CC(NC(c3nc(OCC)oc3)=O)C2)C)=O)CCC(C)CC1 CC1(CCNC(C2CCN(C(=O)C(C3(O)CCCC3)F)C2)=O)CC1(F)F Cc1cc(CNCc2nc(C3CCNCC3)cs2)cc2c1CCC2 C1(N(C(CC2C(NC(CCSCC)=O)CC2O)=O)C)CCOCC1C C1(C(=O)NC2COCCN(C(C3(NC(N)=O)CC3)=O)C2)CCc2[nH]nc(O)c2C1 C1(CNC(CCC2CCC(NC(=O)CCCC3CCCO3)C2)=O)CC2C=CC1C2 C(CCC(=O)NCCc1ocnc1CNC(=O)C(n1cc(Br)cn1)C)=CC N1(C(CC(=O)OC)=O)CC2COCCC2(NC(c2cc(C(C)(C)C)n[nH]2)=O)C1 CCC(CN(C)C)CC(=O)NC(C1CCN(C(c2nc(OC)ccc2F)=O)C1)C N1(C(C(C2CCN(C(c3ncon3)=O)CC2)C)=O)CC2CCCCCCC12 N1(C(C2(C(N)=O)CC2)=O)CC2CCC2(CCNC(c2ccc(SC3CC3)cc2)=O)C1 CC1CCN(C(c2cnc(C(C)(C)C)nc2)=O)CCN1C(=O)Cn1nccn1 c1(C(N2C(CNC(CC3C(=O)NC(=N)S3)=O)CC2)=O)cccc2cc[nH]c12 C12(C(N3CC(C(C)NC(=O)CCOC4CCCOC4)C3)=O)CCCCC1C2(F)F C1(NC(=O)CC2COCCOC2)CN(C(c2cccc(C3CC3)n2)=O)C2CCCC12 c1(N(C)Cc2ccc(C)s2)nc(=NCP(C)(C)=O)[nH]c2c1CCCCCC2 C(C(=O)NC(C1CN(C(=O)C(=O)NCC2CC2)CC1C)C)(C(C)C)SC N1(C(C2(C)N(C)CC(NC(COC)=O)C2)=O)CCC(F)(Cc2nncs2)CC1 N1(C(c2cccnc2)C)CCN(C(c2scc(Cl)c2Cl)C(=O)NC2(C)CC2)CC1 C(=O)(C1=NOC2(CCN(C(c3cc(Br)c(F)cc3O)=O)C2)C1)NC(CC)CO c1(C(N2CC3C(C(=O)NC4CCC(COC)CC4)C3C2)=O)c(F)ccc(F)c1F N1(C(Cc2c(OC)cncc2)=O)CC=C(CNC(C2CCCC23CC3)=O)CC1 N1(C(C(COC)COC)=O)CC2CC1CN(C(c1ccn(C3CCCC3)n1)=O)C2 c1(C(N2CCC(N(C)C(c3ccccc3O)=O)C2)=O)[nH]nc2ncc(Br)cc12 c1(OC)ccc(Br)cc1CC(=O)NC1CN(C(=O)CSC(C)(C)C)C1 N1(C(C(C)(C)C)=O)CC2(CCOCC2)CC1CNC(=O)C(F)(F)C(C)(C)O c1(OCC)nc(C)cc(=NCC(C)(C2CC2)NCC2CCCC3CCCCC23)[nH]1 N1(C(C)=O)CCN(C(c2ccnc(NC3CCC3)c2)=O)C(CO)C1 c1(CNC(CN(CCC)C)=O)cc[nH]c1C(=O)NC.N12CCC(C1)C2=O c1(C(N(CCNC(C2(C)CC(=C)C2)=O)C)=O)c(C)ccc(F)c1Br C=CC(CC)CC(=O)N1CCC(CN)C1.C1(C(=O)N(C)C)(CO)CCCCC1 C1(CNC(c2cc(CCC)c(C)s2)=O)CC(NC(=O)CC(F)F)C12CCC2 c1(CNC(C(=O)NCC2CN(c3ccc(C)cc3)C(=O)C2)=O)cc(C)nc(C)c1 c1(C(C(=O)NCC2C(NC(C3(OCC)CCC3)=O)C2)=O)cnn(CC)c1 N1(C(C(CNC(C=CC(=O)OCC)=O)CC2CC2)=O)CCCC(F)(CO)C1 C1(O)(CNC(c2cn(CC=C)nc2)=O)CCCN(C(=O)COCCCC(C)C)C1 C12(C(=O)NCC3CN(C(CC4C(C)(C)COCC4)=O)C3)CCN(CC1)S(=O)(=O)C2 C1(C(N2CCC(O)(COC)C2)=O)(NC(C(C)SCCCC)=O)CCN(C)C1 C1(C(CNC(C(C)SCC)=O)(C)C)CCCCN1C(=O)Cc1cnc(COC)[nH]1 C1(C(=O)NC(CCCNC(C=CC(CC)C)=O)C)(C(=O)OC(C)(C)C)CCCCC1 Cc1nc2c(C(=O)NC3CCCCC3CNC(c3n[nH]cc3Br)=O)cccc2o1 c1(C(N2C(C(C)C)CN(C(C3(C)CNC(=O)C3)=O)CC2)=O)onc2ccccc12 CC(C)CC(C(=O)N(CC(C)(C)CNC(=O)CN1CCC(=O)NC1=O)C)C(N)=O C(=O)(C(C)(F)C(C)(C)F)NCc1ccc(C(=O)NC(C)C(=O)NCCF)cc1 N1(C2C(CCC=C)C2)CCCN(C(c2ccccc2)CC)CC1 CC#CCCC(=O)NCCCC1CN(C(C2(CN(C)C)CCCC2)=O)CCO1 c1(NC(C(=O)NCC(S(C)(=O)=O)c2ccccc2)=O)ccc2c(c1O)CCCC2 c1(C(CC)C(=O)NC(C)C(C)NC(c2cc[nH]c2C(C)C)=O)ccc(F)cc1 CC1(C)CCCC1C(=O)NC1C2CC(NC(c3ccns3)=O)CC12 C(CO)(CCCO)N(C)C(=O)OCCC(=O)NC(C#C)CC1CCCC1 N1(C(C(C)NC(N)=O)=O)C(C(=O)NC23CC(C)(C2)OC3(C)C)CC2CCCCC12 Cc1cc(C(N2CCNC(C(N3CCC(C(F)F)CC3)=O)C2)=O)nc(C)c1 C(=O)(CCC(=O)NN(C)C)NCc1c(C(=O)NCC(CC(=O)OC)C)scc1 CCC(O)C(C)C(=O)N1CCC(O)(CNC(c2ccncc2C(F)(F)F)=O)CC1 CCCCC(O)C(=O)NCCCCCNC(=O)C(CN(C)C)C(C)C Cc1cc(=O)c(C(=O)NC2(C)CCN(c3ncc(Cl)c(O)n3)CC2)cn1C1CC1 CC1=C(c2ccc(NCc3cc(OC(F)(F)F)cc(C#N)c3)s2)CCCC1 Cc1cccc(C(C)NC(=O)C(CCC2CC2)NC(c2conc2C)=O)n1 c1(NC(=O)NC2(c3ccccc3)CCC2)ccc(=NCc2ccc(Br)cc2)[nH]c1 C1(c2onc(-c3cnc(C)[nH]3)n2)C2CCCOC12 Cc1ccc(C(F)(F)C(=O)NC(C)CC2CCCOC2)nc1 CC(CCCC(=O)NCCNC(C1(C#N)CC1(C)C)=O)c1ccccc1 [N-]=[N+]=NCCCCCCC(=O)N1CC(F)(F)CC1(C)CNC(C1CC2CC2C1)=O c1(C(N2CCN(S(=O)(=O)c3cccs3)C3CC23)=O)c[nH]c2c(Br)cccc12 C(=O)(CCC(Cc1ccccc1)NC(=O)NCC1CCC(NC(C)=O)CC1)OC N1(C(C(CC)C(=O)OC)=O)CC2CC(C1)CN(C(C1C3CNC(=O)C13)=O)C2 C12(C(N3CCN(C(C(C(C=C)C)C)=O)C(CCCC)C3)=O)CCC(C)(CC1)OC2 N1(C(c2ccccc2F)=O)CCN(C(c2cscc2Cl)=O)C(C2CCC2)C1 C(=O)(C(C)P(C)(C)=O)NC1CC(NC(CCNC(COC)=O)=O)CC1O C1(NC(COCCCC#C)=O)CCN(C(=O)CSc2ccc(C)c(C)c2)CC1O C1(C)(C(=O)NC2CCC(F)(CNC(C(C#C)(C)C)=O)C2)CC(C(C)(C)C)=NO1 C1(CC)CCC(C)CN1C(c1ccc(C2CC2)cc1)C(=O)NC1CC1C1CC1 Cn1c(Cl)cnc1C(F)(F)C(=O)NCC1(NC(c2csnc2Cl)=O)CCCC1 C1(C)(C(=O)NC(C)CCN(C)C(c2cccc(=O)o2)=O)CC(C(C)(C)C)=NO1 C1(OC)CC(CNC(c2c(C)ccn2C)=O)N(C(c2cc(C(C)=O)cn2C)=O)C1 N1(C(COCCC#C)=O)CC(Nc2ccc(CN)cc2)CC(C)(C)C1 c1(CC(=O)NC(C(CC)C)CC(=O)NC(C)C)c(C)nc2cc(O)nn2c1C c1(CC)c(C(=O)NCC2(CNC(=O)CN(C)CC)CCCCC2)nnn1CC c1(-c2nn(C)c(-c3cc(C(F)F)n(C)n3)n2)cc(F)cc(F)c1.c1cn[nH]c1 C(=O)(C(=O)C(C)(C)C)NC1(CCCNC(c2cc(C)on2)=O)CC1 C(=O)(C1c2c[nH]nc2CN1C(C1CC1(C)C)=O)NC1CC(C(C)C)OC1 CCC(C)(C)C(O)CNC(=O)CCNC(=O)C(C1(O)CCCC1)F c1(C(CN(C)C(c2cc(C)ns2)=O)=O)cccc(N2CCCC2=O)c1 N1(C(C(CC=C)NC(C)=O)=O)CCN(C(=O)C=C2CCC(C)C2)CC1CCO C1(NC(C(C(C)(C)C)O)=O)COC2C(NC(=O)CCc3n[nH]c(=N)s3)COC12 N1(C(c2ccc(OCC(=O)OC)cc2)=O)C(CNC(=O)C(C)O)CC2COCC12 C(=O)(C1OC(=O)c2ccccc21)N(CC(C)(C)NC(c1ccc(OC)cn1)=O)C c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)CCCSC)C3)cc1Cl N1(C(C(CCCC)NC(N)=O)=O)CCC(NC(C2CCCSC2)=O)C(CO)CC1 Cc1cc2n[nH]cc2cc1C(=O)NC1CCC1NC(C1CC1F)=O C12(NC(C3C(CC)CCO3)=O)CCCCCC1N(C(c1ccc(OC)s1)=O)CC2 C1(C(N(CC(C)NC(c2cn(CCC)nc2)=O)C)=O)CCC2(CC2)C1 C1(CNC(C(C)(Cl)Cl)=O)CN(C(=O)CCNC(c2ccco2)=O)CC12CCC2 C(N=c1cc(Cl)nc(C2CCC2)[nH]1)C1(CNC(=O)CC2CCCS2(=O)=O)CCC1 C(=O)(C1=COCCO1)N1C(C2(NC(=O)Cc3ccc(Cl)s3)CC2)CCCC1 c1(C(=O)OC)cc2n(n1)CCN(N(C)C(C)c1ncc[nH]1)C2 C1(C(=O)NC(C)CNC(c2coc(-c3cccnc3)n2)=O)CN(C)C(=O)N1 c1(C(=O)NCC2CCCC(NC(C3(C)C=CCC3)=O)C2)nccn2nccc12 N1(C(CC2ON=C(C)C2)=O)CCC(C(C)(C)CNC(c2occc2F)=O)CC1 C(=O)(CCC(=O)NC1CCN(C(c2cc(O)nn2C)=O)C1)N(CC)CC Cc1cc(-c2cccs2)c(S(=O)(=O)N(C2CCC2)CC2CCCS2)cc1C C1(N(C)C)CCC(N(C(c2cncc(F)c2)C(=O)NC(C)(C)C)C)CC1 C1(NC(C2C(C)(C(C)C)C2)=O)CCC2(CCc3ccccc32)CC1 N1(C(C(C)(O)Cn2cccn2)=O)CC2(CCCN(C(=O)C(O)CC3CC3)C2)C1 Cc1c(C(=O)NCCOCCN(C)C(C2CCCC2O)=O)cccc1Br c1(CCNC(C(C2CCOC2)NC(C(C=CC)O)=O)=O)cccnc1F C1(C(N2CCN(CCF)CC2)=O)CC12CCN(c1nnc3ccccn13)CC2 C1(NC(C(C)OCCOC)=O)CC2C(NC(c3cc(SC)c(C)o3)=O)C2C1 N1(C(=O)C=CCF)CC2C3CCC(C2C1)N(C(c1cc(O)cs1)=O)C3 CN1CCc2[nH]nc(C(=O)NCC34CCC(CC3)N4C(=O)C=CBr)c2C1 N1(C(CC2CC(=C)C2)=O)CCC(C(=O)NC(C)COC(F)(F)F)(COC)C1 CC(C)CC(C(=O)NC1CCCC(NC(c2ccoc2)=O)C1)C(N)=O S(=O)(=O)(c1ccc(Br)cc1NCC(C)(C)CS(N)(=O)=O)NC(CN(C(C)C)C)C CCCC(O)CCNC(c1ncccc1OCCF)=O c1(C(N2CCCC(NC(C3(C)CCCCC3)=O)CC2)=O)ccc2c(c1)OCCC2 Cc1n[nH]c(C)c1SCC(=O)N(CCN(C(=O)CC(C)F)C)C(C)C N1(C(C2CCCN(Cc3c(C)ncs3)C2)=O)CCC2(CC1)CC(C)(O)C2 CC1(C(=O)NCC2CCN2C(c2cc(OCC(F)F)ccn2)=O)CCC(=O)N1 S(=O)(=O)(c1cc(C(=O)N(C)C)c(F)cc1C)N(C)Cc1c(OC)cccc1 C1(CNC(COCCCC)=O)CCCCN1C(c1cccc(C2CCCC2)c1)=O C1(NC(C)Cc2csc(=N)[nH]2)CCCCCC1CN1CCC2CCC12 c1(C(=O)NC2CC(N(C)C(c3cncc(N)c3)=O)C2)ccc(Br)c(F)c1F c1(C(N2CCC(C)C2c2cn(CC3(O)CCC3)nn2)=O)c(F)ccc(F)c1Cl c1(N(C)C)ccc(C(N2CC(n3cc(C(O)C(C)(C)C)nn3)C(O)C2)=O)cc1F N1(C(C2CC(N(C)C)C2)=O)CCC2CCN(C(c3cccc(CF)c3)=O)CC12 N1(C(CCC(C)(F)F)=O)CCCC(C2CCCN(C(=O)CCc3cncs3)C2)C1 c1(C(=O)NC23CN(C(c4cccc(OC)c4)=O)C(C2)C3)c[nH]c2nccc-2c1 C1(C(N2CC(C(C(=O)NCc3c(C)con3)O)C2)=O)CN(C)CCO1 Cc1cc2cc(C(=O)N(C3CCN(C(c4cn[nH]c4)=O)C3)C)ccc2cn1 c1(CCC)ccc(CC(=O)NC2CCC(NCc3ccc(OCC)cc3)C2)cc1 C(CCCCCCN1CCCC1)NC(C(C1(C)CC1)NC(c1cnc(C)s1)=O)=O N1(C2CN(C(C3(COC)COC3)=O)C2)CCN(C(=O)C(C)(C)c2ccsc2)CC1 C1(NC(C2CCN(CCC)C2)=O)CC2CC(NC(C3(SCC#N)CC3)=O)C2C1 N1(C(c2c(C)cc(F)c(Cl)c2)=O)CCC2(CC1)CCN(C(C13CC(C)C1C3)=O)C2 N#CC1(C(=O)OCC(C2CCCC3(CC3)O2)=O)CCCC(=O)C1 C1(OC)CCn2cc(C(=O)NCCn3c(C(C)C)nc4ccccc34)nc2C1 N1(C(C(CCC2CCC2)NC(C(C(C)(C)C)=O)=O)=O)CC2CC(CO)C(C2)C1 C=CC1(O)CN(C(=O)CCN(C(=O)C=CC2(C)COC2)C(C)C)C1 c1(C(C(=O)NCC2CC(O)(CNC(c3coc(Br)n3)=O)C2)O)ccc(F)cc1 CC1OCCCC1C(=O)N(CCNC(c1cc(N2CCCC2)ncn1)=O)C1CC1 c1(CN(C(=O)OCC2CCN(C(C)C)CC2)C)nn(C)c(Cl)c1Br c1(C(N2C(CN(C(C(C)=CC3CC3)=O)C)CC(F)C2)=O)ccc2n[nH]c(C)c2c1 CCC(C(=O)N(C1(CC(=O)NCC(c2ccccc2)F)CC1)C)SC C(=O)(C1=CC2(CCN(C(c3sccc3OC)=O)C2)C1)N(CCF)CC c1(NC(CCC)=O)ccc(C(=O)NC(c2cn(CC3CCOC3)nn2)CC)cc1 c1(C(=O)NCCC(C)N(C)C(c2cnc(C3CC3)s2)=O)cn(C)nc1Cl CCC(C(=O)NC(C1(O)CN(C(=O)C(O)C2CCC2)C1)C)C(C)O CCC(CC)CCC(=O)N(C(C)CCNC(c1cc(C(F)F)ccn1)=O)C c1(CC(=O)NCCCCN(C)C(C2(C)CC(F)C2)=O)cc(F)ccc1F C1(CNC(=NCCC)NC(C)COC)CCc2nncn2C1 CCC(C)CCCCC(=O)NCC1(C)CC(F)(F)CN1C(=O)COC(C)(C)C C(=O)(C(CC)C(C)(C)CC)C(CC1C(CC(N2CC3(CC(=C)C3)C2)=O)C1(C)C)=O c1(CC(=O)NCC2CC2NC(C2CCO2)=O)ccsc1Cl CCC(C)C(O)CC(=O)N1CC(F)CC1C(=O)NCC1(C#N)CC1 N1CCc2ncsc2C1.c1(C2(CC=O)CC2)ccccc1OC(F)(F)F N1(C(C2(COC)CC=CCC2)=O)CCC2(CC(NC(=O)Cn3nnc(=O)[nH]3)C2)C1 c1(NC(c2cc(CNC(C3(C#N)CCCOC3)=O)on2)=O)ccc2nc[nH]c2c1 c1(CC)nc(=NC(C)CC(C)NC(=O)C(C)=C2CC2)s[nH]1 C(=O)(C(O)CCNC(C1CCO1)=O)NC(Cc1cc(C)[nH]n1)C C1(C(=O)NCC2CCC(NC(c3sc(C)nc3C)=O)C2)(OC)CCSCC1 c1(CC(=O)N(C2CN(C(C34CCC3C4)=O)C2)C)ccc(F)cn1 C1(C(=O)NCC(CC)N(C)C(C2(O)CCCCC2)=O)CCN(C)C1=O N(C(=NCCCCl)NCc1c(F)cc(F)c(F)c1F)CC(C)(C)C(F)F N1(C(c2cc(CCNC(C3(C)CCC(=O)C3)=O)on2)=O)CCCC(O)(C(N)=O)C1 N1(C(c2c(CCCC)ocn2)=O)CCN(C(c2nc(C)ccc2C)=O)CC1CO N1(C(=O)Cc2n[nH]c3c2CCCC3)CCC2(CC1)CN(C(=O)C(F)n1cccn1)C2 N1(C(C(C2CCCC2)OC)=O)CCC2C(C1)CN2C(=O)CC(C)(C)O C1(C(N2CC(CNC(=O)COC3CCOCC3)C2)=O)CCCOCC1 C1(CNC(c2cnn(CCC)c2C)=O)CCN(C(C2(N(C)C)CCC2)=O)CC1C C1(C(N(CCC(C)C)C)=O)(CNC(C2CCCN2C(C)C)=O)CCCO1 C1(NC(c2n(CC)nc(C3CC3)c2)=O)CC2CN(C(=O)C#CC(C)C)CC12 N1(C(C(CC)N(C)C)=O)CCC(C(F)CNC(=O)Cc2ccsc2Cl)CC1 O=C(CCC(=O)c1ccc[nH]1)NCCC1CCN(C(=O)C(F)(F)CO)C1 C#CCC(C(=O)Nc1ccc(CCC)nc1)NC(c1csc(C)n1)=O C=C1CN2C(=O)CCC2(C(N2CCC(C)(NC(c3cn(CCO)nn3)=O)C2)=O)C1 N1(C(C(N2CCCCC2=O)C)=O)CC(NC(=O)CC2CCCCC2)C2CC2C1 N1(C(C(CC)C#N)=O)CC2(CCN2C(c2ccc(C(C)(C)C)cc2)=O)C1 C1(C(=O)NCC2C(C)C2C)(NC(c2cc(CCO)on2)=O)CCC(C)(C)C1 c1(CN(C(=O)NCC(COC)C(C)C)C)c(C)cccc1F N1(C(C(C(C)C)c2nn[nH]n2)=O)CCCCCCC1=O.C1(CC(=O)N)CCCCCC1 C1(N(C)C(C2CCN(C(c3ccc(Cl)cc3)=O)C2)=O)C2CCC1(C)C2(C)C CCCC(C(=O)OC)C(=O)NCC#CCNC(=O)CCc1ccn(C)n1 C(=O)(C1CCCc2nn(C)cc21)N1CC2N(C(C3C(C)C3)=O)CC(C2)C1 C12(C(N(C)CCNC(=O)CC3(O)CCCCC3)=O)CCC(C)(CC1)CO2 CCC(C)CC(C)C(=O)NCC(C)(C)CNC(c1ccc2ccnn2c1)=O N1(CCOC)CCCOC(C2CCN(C(C3CCC(=O)N3C)=O)CC2)C1 N1(C(C2(COC)CC=CC2)=O)CC(C)C(NC(=O)Cc2c(C)noc2Cl)C(C)C1 N1(CC(=O)NC(CC2CN(C(Cc3ccc(C)o3)=O)C2)C)CCCCC1C N1(C(c2cc(C)c(Cl)s2)C(=O)NC)CCCC(N2CCOCC2)CC1 c1(C(=O)NCCN(CC(C)O)C(=O)Cc2ccc(Cl)s2)ccc(C(C)(F)F)cn1 Cc1ncc(C(=O)N(CCCCN(C(=O)CC2(CSC)CC2)C)C)cc1N N1(C(C23C(NC(C45C(C)(C)C(CC4)C5)=O)C4CC2C3C4)=O)CC2CCCC(C2)C1 c1(OC)cc(NC(C2CC(F)(F)CN2C(c2ccccc2NC)=O)=O)nc(Cl)c1 N1(C(C=CCN(C)CC)=O)CCC2(CC1)CC(C)N(C(=O)C1=CS(=O)CCC1)C2 C(C)(CCC(=O)NCC1C(CNC(C2COC(=O)N2C)=O)C1(F)F)SC n1(CC)nc(C(C)C)cc1C(=O)NCCNC(C1C2CCC(=O)C12)=O C(=O)(C(C)(C)CS(C)(=O)=O)NCCCC(C)(C)NC(=O)Cc1ccc(F)cc1F N1(C(C2C(NC(=O)OC(C)(C)C)C3(C2)CCC3)=O)CCCN(C(=O)C(F)(F)F)CC1 C1(NC(CCC=CC)=O)CN(C(c2cc(C3CC3)n(C)n2)=O)C2(CCOCC2)C1 c1(C(=O)NC2CCC(C)N(C(C3CC3(Cl)Cl)=O)C2)cccc(N=[N+]=[N-])c1 C(=O)(CC1=NN(C)C(=O)C1)NCC(C)C(F)C(=O)NC1CC(C)N(C)CC1C C(C)(CCC#N)(c1nnnn1C1(C)CC1)NCCOCC(=O)OC C1(C(=O)Nc2c(C(=O)OC)n[nH]c2)CC(F)CN(Cc2occc2Br)C1 C12(COC1)C(=O)N(CCNC(CN(S(C)(=O)=O)C)=O)CCOC2.CC(C)O c1(C(N2CCCCC(Nc3cc(C)nc(C)n3)C2)=O)cc(C)c(C)cc1Cl Cc1ccc(C(=O)OCc2nccn2-c2cc(C(F)(F)F)ccc2F)cc1CO C12(CN)CCC(C(N3CC(c4ccc(F)cc4)C(N)C3)=O)(CC1)C2 Cc1ccc(CC(N2CCCC2(C)C(N2CCOC(C#N)C2)=O)=O)cc1[N+](=O)[O-] c1(N2CCCC(CSC)C2)ncc(S(=O)(=O)NC2CCSCC2)cc1Cl CCCC(C)C(CC)(c1nnnn1CCC)NCc1nnc(CC)s1 Cc1c(NCCCc2ccc(-c3cc[nH]n3)cc2)ncnc1NC1CCOC1C C1(C(=O)NCCOCCCN(C(COCC=C)=O)C)OC2CCC1CC2 N1(C(c2c(C)oc(CNC(=O)C(C)CC3CC3)n2)=O)CC[Si](C)(C)CC1 N1(C(C=CC2(C)COC2)=O)CCC2(CCN(C(C3C(C#N)C3(C)C)=O)C2)C1 c1(CC(=O)NC2C(C)N(C(C3CCSCC3)=O)CC2)ccc2oc(O)nc2c1 C(=O)(C(C)CC(C)(C)C)N(CCCNC(CCc1c(C)noc1)=O)C(C)C O=C1NC2CCN(C(C3CSC4(C)CCC(=O)N34)=O)CC2O1 CC1(C)CCCN(C(c2cc3ccccn3n2)=O)C1C(N1CC(F)(CF)C1)=O N#Cc1cc(C(=O)NC2CCN(C(c3ccnc(-c4ccccc4)n3)=O)C2)on1 C=CCCCCCC(c1nnnn1C1CCC(F)(F)CC1)NC1(CSC)CCOC1 N1(C(c2nc(Br)c[nH]2)=O)CCN(C2CCN(C(C3CCOC3)=O)C2)CC1 C(=O)(CCC(C)C)NC1(CC=C)CN(C(c2cncc(C)c2)=O)C1 c1(C2(F)CC(C(=O)NC3CC(NC(Cc4n(C)ncc4)=O)C3)C2)cccc(F)c1 N1(C(c2cnc(OC)s2)=O)CCC(C(N2CCCCC2C(N)=O)=O)(CO)C1 C1(NC(c2ccncc2O)=O)CC2CCC(C1)N2C(C1CC2CCC(C1)C2F)=O Cc1cc(CC(N2CCN(C(=O)CSC(F)F)CC2C(C)(C)C)=O)ccc1CO C(=O)(CCCC(C)(F)F)NCCC1CCCN(C(CCC(=C)Br)=O)C1 C1(CNC(C(CC=C)C)=O)CCC2(CN(C(=O)Cc3cccc(C(C)C)c3)C2)O1 Cc1ccnc(C)c1C(=O)NC1COCC1NC(=O)CCn1ncn(C)c1=O N1(C(CCC)=O)CCC2CN(C(=O)OC(C)(C)C)CCC12.C1C(=O)N1CC c1(C(=O)NCC(CC=C)NC(C2(Sc3ccccc3F)CC2)=O)cnc(C)cn1 c1(C(N2CCC(N(C(=O)C(C)C3CC3)CCC)CC2)=O)c(F)cc(F)c(O)c1F C(CCN(C)C(c1cc(CSC)on1)=O)(C(C)C)NC(CC1N(CC)CCC1)=O C(C)(c1ccc(F)cc1F)=CC(=O)NC1(C)CC(NC(C(C#C)(C)C)=O)C1 c1(Nc2c(C)c(NC(C)CS(=O)(=O)CC)ncn2)cnn2c1OCCC2 C(C(O)CC(=O)Nc1cccc(CSC)c1)NC(C1(OCC)CCCC1)=O c1(OC)cccc(C)c1C(N1CC(CCNC(c2c(C)cnn2C)=O)C(C)C1)=O CC(C)CC(C)(CNC(c1ccnc(C2CC2)c1)=O)NC(C1CC12CCC2)=O N1(C(COCc2nnc(C)s2)=O)CCOC2(CCN(C(=O)CCC3CC3)C2)C1 CC1OCCN(C(=O)COC(c2cnc3[nH]ccc3n2)=O)C1(C)C C1(OC)CCN(C(=O)C(CNC(c2ccc(C(C)=O)[nH]2)=O)C(C)(C)C)CC1(C)C C12(CC)CCC(C(N3CCCN(C(=O)C(C)OCCOC)CC3C)=O)(CC1)CO2 c1(C(N2CC3C(NC(CC(C)N(C)C)=O)C3C2)=O)cc(Cl)cc(Cl)c1O N1(C(C(C(C)C)N(C)C)=O)CCC(CNC(=O)CS(=O)(=O)CCO)C(F)(F)C1 NS(=O)(=O)c1cc(C(N2CCCC(Cn3cc(C4CC4)nn3)C2)=O)cc(Br)c1 Cc1ccccc1C(=O)NC(C(C)NC(=O)CCCCN1CCCC1)C(C)C Cc1ccn(CC(=O)NCC2C=CC(NC(=O)C(C#N)C(C)C)C2)c(=O)c1 N1(C(C(COC)O)=O)CCCC(n2cc(CSc3nccs3)nn2)C1 CCC(C)CCCCC(=O)NCC1CC1NC(=O)CSc1cccc(OC)c1 C1(C(=O)NCC(C)CN2CCCC2)CC(C)N1C(c1cncn1C1CC1)=O c1(C=O)n[nH]c2c1CCOC2.C12(C(=O)N(C)CN)CCC1CN(Cc1ncn(C)c1)C2 c1(N2C(C)C(NC(C3CC34CCSCC4)=O)CCC2)ccc([N+](=O)[O-])cc1 Cn1oc(C(N2CCC(C(F)F)(CNC(C3(c4ccno4)CC3)=O)C2)=O)cc1=O c1(C(=O)NCC(CC)(CC)Nc2nc(C)ncc2F)cnc(OC)c(Cl)c1 C1(C(=O)Nc2ccncc2OC2CCNC2)C2CCN(CC2)S1(=O)=O Cn1cc(S(=O)(=O)NC2CC(C(NC[Si](C)(C)C)=O)C2)cn1 CCC(C)(COC)C(=O)N(C)CC1(O)CCCN(C(=O)CCc2ccon2)C1 c1(C(=O)NC(CCNC(C(C(C)C)OC)=O)C(C)C)ccc2nc(C)[nH]c2c1 N1(C(C(Cc2ccc(OC)cc2)C)=O)CC2CCC(C1)C2CNC(=O)CC1CC1 CC(C)C(C(=O)NC1(CF)CN(C(C2CSCC(=O)N2)=O)C1)n1ccnc1 N1(C(C(C=C)C)=O)CCOC(CCNC(=O)Cc2c(C)cnn2C)C1 C12(C(=O)NCCOCCC(C)C)CCC(CN(C(=O)CN3CCN(C)CC3)C1)C2 C1(NC(C(c2nccc(C)c2)(C)C)=O)CC12CCN(C(C1(SC)CCC1)=O)CC2 c1(C(=O)NC2(C)CC(NC(c3ccc(C(C)=O)[nH]3)=O)C2)ccc2cnccc2n1 C1(CCNC(CC(=C)C)=O)CN(C(c2ccc(C)c(Br)c2)=O)CC(C)O1 CC(C)CC(F)(F)C(=O)NCCN(CC(C)O)C(c1cc2n(c1)CCSC2)=O C(=O)(C(C)(C)C(N)=O)NC(CCN(C(c1nc(C(C)C)sc1)=O)C)C C(CCN=c1[nH]c2ncc(Cl)cc2s1)N(C(C(CC=C)C)=O)CC1CCCC1 N1(C(CCC=C)=O)CCCC(CC)(NC(c2cnccc2N2CCOCC2)=O)C1 C1(NC(Cc2c(C)nc[nH]2)=O)CC2CC(C1)N(C(=O)CSc1cn[nH]c1)C2 C1(C(=O)NC(CC(C)NC(C2(C)C(C)(C)C2(C)C)=O)C)CCc2nncn2CC1 c1(C(N2C(C)CCC(NC(=O)C=C(Cl)Cl)C2)=O)ccc(S(N)(=O)=O)c(Cl)c1 C1(NC(C2CC(C)OC2=O)=O)(CNC(c2coc(Cl)c2)=O)CCC(F)(F)CC1 N1(C(C2N(C)CCC2)=O)CCCC2CN(c3c[n+]([O-])ccc3[N+](=O)[O-])CCC12 CC1=NOC2(C1)CC(C(=O)NCCC1CCCN1C(=O)C(=O)Cc1cccs1)C2 c1(C(N)=O)cc2cc(NC(C34CCCC3CC(=O)CC4)=O)ccc2[nH]1 C1(CNC(=O)C=CC=C(Cl)Cl)CC2CCC1N(C(=O)CCc1cccs1)C2 c1(OC)ccccc1C(C(=O)NCC1(NC(c2nnsc2C)=O)CCOC1)OC c1(C(N2CCC(O)(CN(C(C(=O)NCC=C)C)C)C2)=O)cn2c(C)cccc2n1 N1(C(c2c(SCC)cccc2)=O)CCCN(C(=O)C(F)C(C)(C)O)C(C)C1 C=CCCCCCCC(=O)NC1CN(C(c2ccc(C(C)(C)C)o2)=O)CC1OC C1(C(=O)NCC2CC(C(=O)NC3(CCCF)CC3)CO2)CC2(C1)CC2(F)F C(=O)(C(C(C)(C)C)n1ccnn1)N1CC2C(CNC(c3cc(OC)no3)=O)C2C1 C=CC1(C(=O)N=c2ccn(CC(C)C)[nH]2)CCN(C(=O)Cc2ccc(C)s2)CC1 c1(C(N2CCC(CC=C)(NC(=O)CC(C)(C)O)C2)=O)cc(=O)n(C)cn1 CC1CC2(CCN(C(C3CNC(=O)CN3C(=O)CCCn3ccnn3)=O)C2)CO1 c1(C(=O)NCC(CCOC)NC(c2csc(S)n2)=O)cc(COC)oc1C CC1C(NC(c2cnn(C)c2N(C)C)=O)CCCN1C(=O)CSc1ccccc1 c1(C(=O)NCCc2ccc(Cl)c(Cl)c2)nc(Br)n2c1CCCCC2 C1(NC(C(C)O)=O)CCCN(C(c2ncsc2C(F)(F)F)c2ccccc2)C1 c1(C(=O)NCCCN(C(C)C)C(c2nnc(O)s2)=O)cc(F)c(F)cc1Cl N1(C(C=CC(C)(C)SC)=O)CC2CC(C1)CN(C(=O)CC(C)(O)C(F)(F)F)C2 C(C(COC)C(=O)NCCCCCCN(C(=O)CC1SC(=N)NC1=O)C)OC c1(CC(N2CCC(C3CCCN3C(=O)Cc3ccsc3)C2)=O)ccc(O)c(F)c1 CC1CCCN(C(=O)C(=O)N(C)Cc2nc(-c3ccco3)no2)C1 CC1CCN(C(=O)CCCC(=O)C2CC2)CC1NC(=O)CC1CN2CCC1CC2 CON1CCC(C(=O)NC(C)CCN(C)C(c2ccc(C#N)cn2)=O)CC1 c1(OC)cccc(CC(=O)NCCNC(=O)C(n2nccc2C)C)c1Cl C1(C#N)(C(=O)NC(CC)CNC(=O)Cc2nncn2C(C)C)CCCOC1 C1(C(C)NC(C2CC(N(C)C)C2)=O)CCCN1C(C1(C(F)F)CCCC1)=O C1(OCC)CCC(C(=O)NCCCNC(=O)C(c2ccnn2C)C)CC1 CC(CNC(=O)CSC1CC1)CC(=O)N1CCCC1CC1CC1 C(=O)(C1=C(C)OCCS1)N1CCN(C(CCSCCCC)=O)CC1CCC C#CCC(C(=O)NCCC1CCCNC1=O)NC(c1ccn(C2CC2)n1)=O N1(C(c2c(C(C)C)onc2)=O)CCC(N(C(=O)CSc2cnn(C)c2)C)C(C)C1 N1(C(C2(CC)CCOC2)=O)CC2CC(O)C1C2NC(=O)CNC(=O)CNC(C)=O C1(CNC(CC2C(CNC(CCCOC(C)=O)=O)C2)=O)CCOC1(C)C CC1COc2ccc(C(=O)NCC(C)(C)CNC(=O)C(C)C(C)O)cc21 C1(NC(C2N(C(c3ncn(CC)c3)=O)CC=CC2)=O)CC=C(C(C)C)CC1 N1(C(CC(C)(C)O)=O)CCC2CC1CN(C(C1C(F)(F)C13CCC3)=O)C2 C=CC(C)(O)CC(=O)NCC1CCCC1NC(C1CC(C(F)(F)F)C1)=O CN1CC(F)CC1C(N1CCC1CNC(=O)CCc1cn[nH]c1)=O c1(C(=O)NCCC(C)N(C(CCc2scc(C)n2)=O)C)cnc2sccn12 CCC(CSC)N=c1[nH]c(N(CC(=O)NC2CC2)C)nc2ncn(CC)c12 O=C(CCc1ccc(C(F)(F)F)cn1)NNc1ccc(Br)c(F)c1F CCCCC(COC)NC(=O)C(CCOCC)NC(=O)CCC(=O)NCC C(=O)(C1=COc2ccccc2O1)NC1CC(NC(CCNC(=O)NC)=O)C1 c1(C(N(CCC(C(C)C)NC(CC2(C=C)CCC2)=O)C)=O)ccc(C)nc1C Cc1ccc(C#N)cc1C(=O)NCC1CC(NC(C2C3CC4C(C3)C24)=O)C1 N1(C(c2ccnc(C)c2C)=O)CCC2(CC1)CC2NC(=O)CC(C)CF C=CCC(C)(C)CC(=O)N1CCC(NC(c2cc(C(N)=O)cn2C)=O)C12CCC2 CC1(C#CC(=O)NC2CC3CCC2N3C(c2ccnc(N(C)C)c2)=O)CCCO1 C1(Cl)(C(N2CC(COC)(NC(C3CC=CC3)=O)C2)=O)CC12CCC2 c1(C(=O)NC2C(C(=O)NCC(CC)(C)OC)C2(C)C)cnc(Cl)n1C c1(C(N2CCN(C(c3cc(C)ns3)=O)C3C2C3)=O)ccnc2c1CC(=O)N2 c1(CNC(c2ccc(C#C)c(F)c2)=O)nc2c(s1)CN(C(=O)CCC(N)=O)CC2 CC1CC(C(C(=O)NCc2cccs2)N(C(C)(C)C)CC2CCCO2)CO1 C1(CC(N2CCC(OCCNC(=O)C=CC3CC3)C2)=O)(OC)CCCCC1 CC(=O)CC(C)(C)CC(=O)NC(CNC(c1ccc(Cl)cc1C)=O)C1CC1 C1(C(=O)NCCc2ccncc2)CCN(C(c2cccc(F)c2O)=O)CC1O c1(OC)ccc(C=CC(N2CC3C(C(=O)Nc4c(F)cccc4I)C3C2)=O)cc1 C1(CCNC(c2[nH]cc(C(N)=O)c2)=O)CCCCN1C(=O)Cc1cccc(Cl)n1 N1(C(C2ON=C(C)C2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)C)C2 N1(C(CC=CC=C)=O)CCC(NC(C2CCCN2C2CC2)=O)CC1C c1(OC)c(Br)cc(CC(=O)NCC2CCN(c3nccc(C)n3)CC2)cc1Br CC1CCC(C(=O)NCC2(CCO)CCC2)CN1C(=O)CC1(C2CC2)CC1 N1(C(=O)OC(C)(C)C)CCC(C(=O)NCC2OCC23CCC3)C12CCC2 C1(C(N(C(CN(C(c2cncc(OC)n2)=O)C)C)C)=O)CC2C(C1)C2(F)F CC#CC1CCN(C(=O)C(C)(CNC(=O)CCOC2COC2)CC)C1 Cc1nc2c(o1)CCN(C(=O)COC(C)(C)CNC(C1COCC1C(N)=O)=O)C2 C1(N(C(C2CC2c2ccco2)=O)CC)CCN(C(=O)CC2CCC(=O)N2C)CC1 C1(CNC(c2c(C)nc(CCC)o2)=O)CN(C(=O)CC2CCCSC2)CCN1C N1(C(C=C(C)c2ccsc2)=O)C2CCC(C2)C1NC(C)CNC(=O)OC(C)(C)C c1(C(N2C(C(=O)NCCOCC(C)C)C(C)CC2)=O)cc2cccnn2c1 c1(C(=O)NCCCN(C(=O)C(CO)C(C)(C)C)CC)cccc2ccoc12 C(=O)(C1=CC2CC=CCC12)N1CC(NC(c2cncn(C)c2=O)=O)(CO)C1 N1(C(=O)Nc2ccc(C(=O)OC)o2)CCC2CN(Cc3cc[nH]n3)CCC12 N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCN(C(=O)C(c2ccc(F)c(C)c2)=O)CC1 C1(NC(c2c(C)oc3cc(O)ccc32)=O)Cc2ccccc2C1C(=O)O c1(C(=O)NC2CCC(CCNC(c3cc(O)cs3)=O)C2)ccc(CCF)cc1 C1(C(=O)NC2C(N(C)C(C34CC(C(C)(C)C)(C3)C4)=O)CCCC2)C2CC3C(C2=O)C13 c1(OCCC(=O)N(CC(CC)NC(c2cnn(C)c2N)=O)C)ccccc1O N1(C(CCCN(C)CCO)=O)CC(O)CC1C(=O)NC1C2CCC1CC2 C(=O)(C(C)(C)CN(C(=O)CC(C)F)C)NCc1c(C)nco1 c1(C(=O)NCc2ccc3occc3c2)n[nH]c2ccc(-c3ccnc(F)c3)cc12 CC1(C)CCC(C(C(=O)COCC2CCC2)=O)(N)C1.c1(CNC2CC2)nc(C)no1 CN1CCCCC(C(=O)NC2(C)CCN(C(C3CC4CCC3C43CC3)=O)C2)C1=O N1(CCNS(C)(=O)=O)CCCC1CO.c12cc(cs1)NC2=O c1(C(N(CCCC(=O)NCc2cnc(C)n2C)C)=O)n[nH]c2c1CCC2 CC(N=c1[nH]c2c(c(=NC(CCO)C3CC3)[nH]1)CCCCC2)c1ncc[nH]1 N1(C(C(C)(C)OC)=O)CCC(C2CN(C(=O)C(CO)C(C)(C)C)C2)CC1 CCCCCCC(=O)NC(CCCOC)C(=O)NC1CCC(C#N)CC1 C(=O)(C(C)(C)C(C)(F)F)NC1CN(C(C2CCCC(C)O2)=O)C1 N1(C(C2(c3cccs3)C(C)C2)=O)CC(O)(CCNC(c2ccncc2)=O)C1 C1(CNC(c2cc(C(C)=O)oc2)=O)C(C)CCCN1C(=O)CC1C=CCCC1 N1(C(c2ccc(C=C)cc2)=O)CC2CC(C1)CN(C(c1csc(CC)n1)=O)C2 n1(-c2ccc(C(=O)NCC3CCC(C)NC3)cc2)cnc2ccccc12 N1(C(CCOCC#C)=O)CC(NC(=O)CCC2CCCC(=O)N2)C(F)C1 c1(C(N2C(CN=c3cc(C)nc[nH]3)C(C)CCC2)=O)ccn2c1CS(=O)(=O)CC2 N1(C(c2ccc(C(OC)OC)o2)=O)CCC(NC(=O)C(F)(F)CN(C)C)C1C c1(CC(N2CCC(CNC(CC3C(C)=NOC3=O)=O)C2)=O)ncc(F)cc1F c1(OCC)cc(NC(c2cccc(NC(c3[nH]c(C)cc3C)=O)c2)C)nc(C)n1 N1(C(C(CC2CCCC2)OC)=O)CCOCC1CNC(c1coc(Br)n1)=O c1(CC)cc(N)c(C(=O)NCCCC2(NC(=O)CCS(C)=O)CC2)c(F)c1 C1(Cl)(C(=O)NC(CNC(CSC)=O)C)CC1C(C)=O C1(C(C)(C)NC(=O)Cc2ccsc2)CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1 c1(C(=O)NCCC(CNC(CCCCC#C)=O)O)cc(C)c(OC)c(C)c1 CC(=O)CCCC(C)C(=O)NCC1(C)CCC(NC(C2SCCS2)=O)C1 C1(NC(C2C(C=C)C2)=O)CN(C(c2ccc(C(=O)OC)c(C)n2)=O)CC1N=[N+]=[N-] C(=O)(CCC(F)F)NC1CC(CNC(CC=CCC)=O)C1 Cc1ccc(N2CC(C(=O)NC(c3cccc(F)c3)C3(O)CCC3)CC2=O)cc1 CC1(CCNC2CCCC3CC23)CCN(C(c2cccc(Cl)c2)=O)C1 Cc1scnc1C(=O)NCCCNC(C1(Br)CC1)=O N1(C(N(CC)CC2CCC2)=O)CCC(C)CC1Nc1ccccc1 C=CCCCCCC(=O)N1CCC(C2CCCN2C(=O)CCC(=O)NC)CC1 C#Cc1cc(C(=O)NC2CN(C(C3CC4CC4C3)=O)CC2CO)cc(F)c1 N1(C(C=NOC)=O)CCC2CC12C(N1CCC(F)(F)C1)=O CN1C(=CC(=O)N(CCC(C)(C)C)CC(F)(F)F)C(C)(C)c2ccccc21 CC1CN(C(=O)CC2(NC(=O)C=C3CCCCC3)CC2)c2cccnc21 C(=O)(C(C)S(C)(=O)=O)NC(CC(C)C)C1CCOCC1.C1(=O)CO1 c1(C(N(C(CNC(C(C(C)C)NC(N)=O)=O)C2CC2)C)=O)cccc2c1COC2 N1(Cc2n(CC)ccn2)CCOC(C)(CNC(c2ccc(OC)cc2I)=O)C1 C1(CC(=O)N(c2cc(-c3cccs3)on2)CC)CCCN(C(=O)C(C)(C)OC)C1 C1(C(N2CCCCC(CC3CC3)C2)=O)CCN(C(=O)Cn2cnnn2)C12CC2 CC1(C)CCC(O)(C(=O)NC2CC(F)(CNC(=O)CCNC(=O)CO)C2)CC1 N1(C(CC(C)(C)OC)=O)C(CNC(=O)C(C)(C)C(C)(F)F)CC2COCC12 CC1CN(C(c2cnc[nH]2)=O)CCC1NC(c1cnnc(O)c1)=O CN1C(=O)CCC1C(=O)Nc1n[nH]cc1NC(=O)CCC1CCCCC1 C1(OC)CC(O)CN(c2nnc(-c3ccc(F)c(F)c3)n2C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(N(C(=O)CC2C=CCC2)C)CC1 c1(C(=O)NC2(CNC(C34CC(COC)(OC3)C4)=O)CC2)c[nH]cc(F)c1=O N1(C(CS(CC)=O)=O)CCC2CN(C(c3c(F)cccc3Br)=O)CC12 C#Cc1ccc(C(=O)N(C2CN(C(c3csc(CC)n3)=O)CCC2C)C)cc1C C12(C)CCN1C(=O)CCOC2.C(CC=CCNC(C)=O)OC CN1CCC(C(N2CC(NC(c3ccnc(C(F)F)c3)=O)C(C)(C)C2)=O)S1(=O)=O C(=O)(C(CCc1cnn(C)c1)N(c1cccnc1)C)NCCOCC C1(CCOC)(NC(c2cnc(C)o2)=O)CCN(C(c2cccc(CO)n2)=O)CC1 c1(C(=O)NC2CC3(C(NC(C(C)NC(C)=O)=O)C3)C2)cc(C(N)=O)cc(F)c1 C1(C(N2CCC(N(C(CCSC)=O)C)C2)=O)CCC(C(C)(C)O)CC1 N1(C(C2CCC(OC)CC2)=O)CC(C2CCCN(C(=O)C(F)n3cccn3)C2)C1 CC1CC(CNC(C2(F)CCCCCC2)=O)CN(C(C2(CN(C)C)CC2)=O)C1 c1(C(=O)NC(C2(CNC(c3n[nH]c(=N)[nH]3)=O)CC2)C)csc(C2CCCO2)n1 c1(C(N2CC(C=C)C(NC(=O)Cc3sccc3C)C2)=O)c(C)cc(C)oc1=O CC(CNC(c1ccnn1CCF)=O)(CO)NC(c1cn(CC(F)(F)F)nn1)=O CCCCC(O)CC(=O)N1CCCCC(NC(c2cc(OC)ccc2F)=O)CC1 CCCCC(O)C(=O)OCC1(COC)CC(C(=O)Nc2cc(O)nc(OC)n2)C1 c1(C(N2CCC(CC#N)CC2)=O)nnn2c1CN(C(C1CC(O)C1)=O)CC2 N#CC1(C(N2CC3CC3(CNC(=O)CCC3CCC3)C2)=O)CCCOC1 c1(C(=O)NCC2(CNC(C3N(C)CCC3)=O)CC23CCC3)cc2ccsc2n1C N1(C(CSSC)=O)CCC2(CCCN2C(=O)Cc2cnccn2)C1 c1(C(=O)NCC2CC(NC(C(C(C)O)C)=O)C2)sccc1S(N)(=O)=O C1(CC(=O)NC(CN(C(C(C)c2cc[nH]n2)=O)C2CC2)(C)C)CCC=CCC1 C(=O)(C1=CC2CCC(C1)C2)N1CCC(C(=O)NC2CCC(OCC)CC2)C1(C)C c1(OC)cccc(C(O)C(=O)NCC(C)NC(=O)Cc2cnc(C)[nH]2)c1 N1(C(c2cnc(C(C)=O)s2)=O)CC2CCC(CNC(=O)C(C)(C)C#N)(C2)C1 CCCCCC(O)CC(=O)N1CC(CNC(C2OC3CCC2C3)=O)OC(C)C1 N1(Cc2c(CC)cccc2)CC2(CN(C(c3ccc(C)nc3)=O)CC2C(=O)O)C1 N1(C(c2cccc(NC(CC)=O)c2)=O)CC2CN(C(=O)C(C#N)C3CC3)CCC12 c1(C(N2C(C(=O)NC(C)C)CCCC2)=O)cc2c(s1)CCC(C(C)(C)C)C2 N1(C(CC(C)(C)C2CC2)=O)CCC2CCCC12C(=O)NC1CCC(N=[N+]=[N-])CC1 CCC(C(=O)NC1(CO)CN(C(C2(O)CCC2)=O)C1)C1CCOCC1 CC(CC(=O)N1CC2CC2(NC(c2cnc(C3CC3)o2)=O)C1)P(C)(C)=O CP(C)(=O)COCC(N1CCCC1CNC(=O)Cn1nccn1)=O C1(CCNC(c2onc(C)n2)=O)CCN(C(=O)CNc2cccnc2)C(C)C1 CS(=O)c1ccc(-c2cn(CCCC(=O)Nc3cncc4c3CCC4)nn2)cc1 c1(CC)c(C(=O)NCC(O)CN(C(=O)C(F)=C2CCC2)C)ccn1C C=CCCCCCCCC(=O)N1CCC2(NC(c3cn(C)c(C)n3)=O)CC2C1 C1(c2nc(C)[nH]n2)CN(N2CC(F)(F)CC2c2ccccc2)C1 Cc1ccc(S(=O)(=O)NCc2ccc(F)cc2-c2ccc(F)cn2)cc1C C1(NC(=O)C(F)n2cccn2)C2CC(O)C1N(C(c1ccnc3cc[nH]c13)=O)C2 c1(C(N2CCOC3C(O)CC23)C(=O)NC)cccc2c1CCO2 C1(C(=O)NC2CCN(C(C3CC(CC)C3)=O)C2C2CC2)CCc2c[nH]nc2C1 N1(Cc2c(C)nn(-c3ccccc3Br)c2)CC2(N)CCCC2(F)C1 C1(C2CC2)(C(N2CC(N(C(C(C)OC(C)(C)C)=O)C)C2)=O)CC=CC1 N1(C(c2nc(OC)nc(O)c2)=O)CC2CC(CNC(=O)CC3CC(=O)C3)CC1C2 C(=O)(C(F)(F)CC)NCC(C)N(C(C1C(CC)C1)=O)C CC(C)CC(O)C(=O)NC1CN(C(=O)Cc2cc(C3CC3)no2)CCC1F C1(C(=O)NCc2cc(C)[nH]n2)CCC(C2CC2)N1C(=O)CCC(=O)C1CC1 c1(C(=O)NC2CCN(C(c3c(C)snc3)=O)C(C)C2)c(F)ccc(N)c1F Cc1c(NC(CC2CCN(C(c3ccns3)=O)CC2)=O)cccc1F c1(C(N2CC(N(C(CCC=C)=O)C)C3(C2)CC3)=O)ccc(O)c(C)c1C N1(C(c2n[nH]c(CC)c2Cl)=O)CC(NC(=O)Cc2cc(C)cs2)CC1(C)COC N1(C(c2ccc(CC)[nH]2)=O)CCC2CCN(C(c3coc(CC)n3)=O)C2C1 C1(N(CCC)C)CCN(C(=O)CCN(C(C2(CO)CCOC2)=O)CC)CC1 c1(OC)cccc2c1OCC(C(=O)NC(C)C(C)NC(=O)CNC(=O)N(C)C)C2 C12(C(=O)NCC(CNC(C=NOC)=O)(C)F)CC=CCN1CCC2 C1(C(C)NC2(c3n(CC)nnn3)CCC2)CC2(CCC2)C1 Cc1ncnc(C(N2CCC(C3OCC3(F)F)CC2)=O)c1NC1CC1 N=c1[nH][nH]cc1C(=O)NC1CC(CNC(c2[nH]nnc2C2CC2)=O)C1 CC(C)CCCCCC(=O)NC(C)CCCNC(=O)Cc1ccccc1CC#N c1(CN(CC(C(C)C)OCc2ccccc2)C2CC2)n[nH]c2cc(F)ccc12 C1(C(=O)NC(CNC(CN(C2CCCC2)C)=O)(C)C)CC2CC1CO2 c1(C(N(C2CCCN(C(C3(C(=O)NC)CC3)=O)C2)CCO)=O)ccnc(Br)c1N c1(OCC)cc(OC)cc(C(N2C3CN(Cc4cc(Cl)cc(I)c4)CC23)=O)c1 CCC(C)C(C(=O)NC1CCC(CO)CC1)N(C)C(c1cc(C)n(C)n1)=O C12(C(=O)NCCOCCN(C(C(C)CSC(F)(F)F)=O)C)CCC(CO)(CC1)C2 N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(=O)CN1CCN(C)C(=O)C1 C1(NC(C(=O)NCC)=O)CCOCC1C(=O)NCC1CCC1CO C(=O)(CC1=CCOCC1)N1CCCC(CNC(=O)Cc2ccsc2Cl)C1 C(=O)(C(CC)C(C)O)N1CC(CN(C(Cn2ncc(C(=O)OC)c2)=O)C)OCC1 c1(-n2ncc(C(N3CCC(c4cn(C5CCC5F)nn4)C3)=O)c2)ccccc1F CCCCCCCC(=O)NC(CC)CC(=O)Nc1cnc(C)c(CC)c1 C1(CC2C(NC(CC=C(C)C)=O)CC2)CCN(C(=O)C2CC2)CC1 N1(C(C2N(c3nc(OCC)c(Br)cn3)CC(F)C2)=O)CCc2cc(F)ccc2C1 C1(C(=O)NCCCCNC(C(C)C2CCCC2)=O)CC2(C1)CC(C)(C)C2 C=CC(F)(F)C(=O)N1CC(O)(CCNC(=O)COCc2ocnc2OCC)C1 O=C1CCCCC(C(=O)NC(CC2CC2)C(=O)NC2CCNC2=O)C1 c1(C(N2C(C)CC(NC(c3cnc(C)nc3)=O)C2)=O)cc(C)c(F)cc1Cl Cc1sc(=O)n(CC(=O)N(C)CC2CCCN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)c1C N1(C(Cc2cc(OC)ncc2)=O)CC2CN(C(c3nocc3Br)=O)CCC12 c1(C(N2CC(NC(c3nn(CC)c(=O)cc3)=O)C2)=O)ccc2c(c1)CCOC2 Cc1ccc(C(O)CN(C(C(F)(F)F)C(F)(F)F)CCCOCC(C)C)cc1Br CCCCC(C(=O)N(CC(C)(C)CNC(=O)C(C)CC1CCC1)C)N(C)C C1(CNC(C(C(C)C)F)=O)CC2(CCN(C(C3C4C5CCC(C5)C34)=O)C2)CO1 CC1Cc2cc(NC(=O)NCCCCCN(C)C)ccc2O1 Nc1ncccc1-c1cn(CCC2CCCN(C(=O)CNC=O)C2)nn1 C(=O)(CCCC(=O)N1CCOC(CN(C2CCCC2)C)C1)N(CCC)CCC Cc1cc2n(n1)c(=O)[nH]c1scc(n1)c(=O)[nH]2.c1(N)ccccc1Cl.C(C)C C(C(=O)N1CC(NC(C2(C3CC3)CC=CC2)=O)C1)(C(C)(C)C)OC S(=O)(=O)(c1ccc(NCC(C2CCOC2)F)c(C#N)c1)N(C)CC=C1CCSCC1 c1(C(=O)NCC(CC=C)NC(C23CCCC2C3Br)=O)cc(C#N)cn1C N1(C(CC(C)(C)O)=O)CCN(C(=O)C(C)(O)c2ccccc2)CC1c1cn[nH]c1 c1(C(N(CC(O)CNC(=O)CC2(CO)CC2)C)=O)cc(Br)c2nccnc2c1 C1(CC)CN(C(c2ccsc2C)C(=O)NCSc2ccccc2)CCO1 c1(-n2c(C(N(C(C)C(=O)OC(C)(C)C)C)=O)cnn2)cccc(Br)c1 N1(C(CC=C=C)=O)CCCC(NC(=O)CCc2cnn[nH]2)C1 c1(C(=O)NCC2(O)CN(CCc3cn(CC)nc3)C2)c(C)nn(C)c1C C(C(O)C(F)(F)F)NC(CC1N(C(c2ccccc2)=O)CC1)=O CCN=c1cc(C(=O)N(CCCCNC(C2CCCC2CF)=O)C)cc[nH]1 N1(C(CC(COC)C)=O)CC2CCN(C(c3ccc(F)cc3OC)=O)C2C1 C(=O)(C1Cc2c(Cl)cccc21)NCCN(CCOC)C(c1c(Br)nnn1C)=O N1(C(C(CNC(C)C)C2CC2)=O)CCC2(CCN(C(=O)C3=CCCCO3)C2)C1 c1(C(N2CCC(N(C(=O)CCc3nncn3C)C)C2)=O)ccc2oc(=O)oc2c1 c1(C(=O)NCC2N(C(C(C)C)=O)C3C(C2)C3)nc2c(Br)cccn2n1 N1(C(C(CCSC)NC(C2CCCCCCC2)=O)=O)CCOC(C2(C)N=N2)C1 CCC(C)(C)CCCC(=O)N1CCCC(C)(C(N2CC(=O)NC(=O)C2C)=O)C1 CC(C(C)(C)C(=O)NCCCCCCF)NC(=O)CN1CC(=O)NC1=O C1(OC)CC(CNC(c2ccc(C3CCOC3)s2)=O)N(C(c2cc[nH]c2C)=O)C1 c1(C(=O)NCC(C(=O)OC)NCCC#N)ccc(S(=O)(=O)NC)cc1 CC(C)C(C(=O)NCC1(O)CN(C(=O)C(c2ccc(Cl)cc2)C)C1)C(C)C c1(NC(C2CCN(C(C3(CC)COC3)=O)CC2O)=O)cc(C)c(Br)cc1[N+](=O)[O-] C1(CNC(c2csnn2)=O)CC2(CCN(C(c3cn4ccnc4s3)=O)C2)CO1 c1(C(=O)NC2CCCC(NC(C3(C=C)CCOCC3)=O)C2)cccc2nc[nH]c12 N1(C(C(COC)C)=O)CCC2CCN(C(c3cc(O)n(CC)n3)=O)C2C1 c1(CNC(C(CCOCCO)NC(C(C)CF)=O)=O)ccc(=O)n(C)c1 c1(C(=O)NC)ccc(C(=O)NC2(CF)CN(C(=O)Cc3cncs3)C2)cn1 Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(F)CNC(=O)C1=CCCCCC1 C1(N(C(=O)C(c2ccco2)NC(=O)CCc2ccsc2)C)CCCCC1O N1(C(C2CCSCC2)=O)CCC2C(CCN2C(c2cnc3[nH]ccc3n2)=O)C1 C(=O)(C(CC(F)F)NC)NN(C1C(OCC)CC1)C(=O)CC(C)=C(C)C N1(C(CC(C)SC)=O)CCCC2(CCN(C(=O)Cc3nc(C)sc3C)C2)C1 C(=O)(CCCCCNC(c1cccc(OC)n1)=O)NC(CCC)C(=O)N(C)C CCS(=O)(=O)CC(=O)N1CC(F)(C(=O)NCCC(=O)NC(C)(C)C)C1 c1(C(N(CCC(=O)NCCc2ccns2)CC=C)=O)cn(C)nc1OC C(=O)(C(=O)C(C)CC)N1CC(CCC)C(NC(C2(n3cnnn3)CC2)=O)C1 C(CC(C(=O)NCC(C)CNC(c1ccc[nH]1)=O)N(C)C)SC Cn1ncc2cc(CN3CC4CCC(C3)C4NS(=O)(=O)CC(F)(F)F)ccc12 O=C(C1=CC2CCC=CCCC12)N1CC2(CCN(C(C34CC(F)(C3)C4)=O)CC2)C1 C(=O)(C(C)CCC(C)(C)C)N(c1ncon1)CC(n1cc(C(C)(C)CO)nn1)C C1(CNC(CN(C2CCCCC2)C)=O)CC(NC(=O)CNC(C2CCC2)=O)C1(C)C c1(C(CC)O)nc(-c2cnoc2C)n(CCOc2ccccc2F)n1 C12(NC(c3cnc(CC)s3)=O)CCCC1N(C(=O)CCC=CC(C)C)CC2 C=CC(C)(CC)C(=O)NCC1CCN1C(=O)CC1(C#N)COC1 c1(OC)ccc(F)cc1C(=O)NC1(CNC(c2cc(C)cc(N)c2)=O)CCOC1 CN1CC2C(C(N3CCOCC3CC(=O)NC3CC(Cl)(Cl)C3)=O)C2C1 C1(C(N(C2CCN(C(C(CC)OCC)=O)CC2)C)=O)CCCC(C)CC1 C1(C)(CC)CC(NC(c2cn[nH]c2)=O)CN1C(=O)CSc1ccc(F)cc1 C#CC1CCN(C(=O)COC2CCN(C(c3ccc(C)cc3)=O)C2)C1 C1(C(N(CC(C)NC(C2CS(=O)(=O)C2)=O)CC)=O)CCC(C(=O)OC)CC1 C(CC(O)C(=O)NC1CC2(C1)CC2NC(=O)CC1(c2ccc(F)cc2)CC1)SC N1(C(CC2CCC(C)C2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC2C1 c1(C(N2CC(C3CN(C(c4ccccc4O)=O)C3)C2)=O)cc2n(n1)CCCC2O C(CNC(=O)C(c1ccco1)NC(=O)C(C)=C(C)C)(C(F)(F)F)OC C(=O)(C1=CCCOCC1)NC(CNC(C=Cc1nnc(C(C)C)o1)=O)(C)C S(=O)(=O)(c1ccc(Cl)cc1)N1CC(C(=O)NCCCN2CCOCC2)SCC1 C1(CCC)(NC(=O)CCS(N)(=O)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 CCC(C(=O)NCC1(NC(c2c(F)cccc2F)=O)CCCC1)C(C)O C1(N(C(C(C)SC)=O)C)CCCN(C(C2CC2c2cn[nH]c2)=O)CC1 c1(OC)n[nH]c(C(=O)NC(C)CN2CCN(C(=O)C(C)OC)CC2)c1Cl c1(C(N2C(CN(C)C(C3CCCCC3)=O)CCC2)=O)ccc(F)c(O)c1 c1(CC(C)(C)C)ccc(C(=O)NC2C3CN(C(c4cocn4)=O)CC23)cc1 C1(NC(c2scnc2C(F)(F)F)=O)CCN(C(C2CC3(C2)CC3F)=O)CC1 C(C(Cc1ccc(Cl)cc1)C(=O)NC1CCN(C(=O)COCC(=O)OC)C1)OC C1(NC(=O)COCCF)CCCCCN(C(C2CC3CCCC(C2)C3)=O)C1 C1(NC(=O)Cc2ccon2)CN(C(=O)CCC2CC2)CC2(CCOCC2)C1 CCCC(C)CCNC(=O)C(C1CCC1)NC(C1OC2CCC1C2)=O c1(C(=O)NC2CCN(C(C(CC=C)C(C)C)=O)CC2)cc(Cl)c2c(c1)OCCO2 CN=c1nc(N2CCC(CC3CCOC3)C2)[nH]c(=NCC(C)(C)NC(N)=O)[nH]1 C1(NC(CCn2c(C)ncc2)=O)CCCC12CN(C(=O)C(C(C)C)N(C)C)C2 N1(c2c(C)c(NC3C=CCCCC3)ncn2)CCC(C)C(F)(F)CC1 C1(N(C(C2CCN(C(C)=O)CC2)=O)C)CN(C(C2(C(=O)N(C)C)CC2)=O)CCC1O N1(C(c2ccn(CCNC(c3c(NC)cccc3)=O)c2)=O)CCNC(=O)CC1C C(=O)(C1=NOC2(CCC2)C1)N(C1CCN(C(=O)CC(C)CN(C)C)CC1)CCC C(=O)(C1OCCc2c(O)cccc21)N(CCCN(C)C(c1cccc(O)n1)=O)C c1(NC)cncc(C(=O)NCC2CC(NC(c3cncc(C)n3)=O)C2(C)C)c1 c1(C(C)C)ccc(O)c(C(=O)NC(C)C(C)NC(=O)C2=CCCSC2)c1 c1(NC(N2CC3N(C(c4nn(CC)c(C)c4)=O)C3CC2)=O)ccc2c(c1)OCO2 c1(N(CC(=C)Br)C)nc(N2CC(C(N)=O)C3(CC3)C2)c2c(n1)CCCCC2 C(=O)(CCC(=O)N(C1CN(C(=O)C(F)CC2CC2)C1)C)NCCNC(C)=O C1(C(=O)NC2(NC(C3CCCOC3)=O)CC(CO)C2)CC2(CC2)CO1 N1(C(c2ccncc2F)C(=O)NCCSC)CCC2CC(O)CCC2C1 C(CCCCCNC(=O)CN1CCCS1(=O)=O)N(C(=O)C1=CCCS1)C C1(C(N2CC(C)C(NC(=O)C(F)(F)CO)C2)=O)CC2(COC(=O)N2)C1 C=CC(C)C(C)C(=O)N(CCCNC(c1cc(OC)cc(OC)c1)=O)C(C)C c1(OC)csc(C(N2CC(NC(C3CC(SC)C3)=O)C(C)C2)=O)c1OC Cc1ncc2c(n1)CCC(C(N1CCCC1(C)CNC(=O)Cc1cncs1)=O)C2 C(=O)(C(O)CC(C)(C)C)NC1CN(C(COc2cccc(C(C)C)c2)=O)C1 C(=O)(C(C)(C)CN1CCCCC1)NCCOCCN(C)Cc1ncco1 c1(C(N(CC(CNC(C(C)C2CC2)=O)O)C)=O)ccc2c(c1)CN(C)C2 c1(C(=O)Nc2nc(C)c(C(=O)NCC3(F)CCC3)s2)cc(Br)ccc1Cl c1(C(=O)NCC(=O)NC(c2ccncc2)C(C)C)cncc(S(N)(=O)=O)c1 c1(C(N2CC(O)CC(NC(CP(C)(C)=O)=O)C2)=O)ccnc2cc(Cl)ccc12 C1(=O)C(CCOCCO)N1.c1(CC)nocc1CN(C(=O)Cn1cnnc1O)C N1(C(c2ccc(CC)cc2)=O)CC2(CC2)CC1CC(=O)NCc1cc(C)ns1 N1(C(CCSCC(C)C)=O)CCC(O)(CCNC(=O)C(C)(C)C(C)C)CC1 C(N=c1[nH]c2c(c(=NCC3CC(n4ccnc4)C3)[nH]1)CCC2)c1nnc(C)o1 c1(CC)ccc(CC(N2CCC(N(C)C(C3(C)CC3(F)Cl)=O)CC2)=O)cc1 C1(=O)C(COC)COC2CCN1C2.c1(C(CC)NC(=O)C=CC(C)C)nccs1 CC1CCN(C(c2ncccc2N)=O)C1CNC(=O)C(F)CC1CCCC1 CCC(C(C)O)NC(=O)C(C)(C1CC1)N(C)C(C1CC(=C2CC2)C1)=O C#CCCCCCC(=O)N1CCC2(NC(=O)CC(C)(O)C3CC3)CCCC12 Cn1ccc2sc(C(=O)NC3(C)CCCN(C(c4ccnn4C4CC4)=O)C3)cc12 c1(N(CC(N)=O)C)nc(=NC(CCO)C2CCC(F)(F)CC2)[nH]c2ccsc12 CCCC(C(C)CC)(c1nnnn1CC1CCC1)NCc1cccc(OC)c1 c1(C(=O)NC23CC(NC(=O)C4=CCCS4)(C2)C3)ccc2c(c1)Cc1ccccc1-2 C1(O)(CNC(C(C)CN(C(=O)COc2cccnc2)C)=O)CCOCC1 CCCC(CNC(c1cn(CCO)nn1)=O)C(=O)N(C)CCN1CCCC1=O CC1CC(NC(C2(C)CC2)=O)CN1C(=O)Nc1cccc(N2CCCS2(=O)=O)c1 N1(C(CCOCCCOC)=O)CCC(CNC(C2CCOC2C2CC2)=O)C(O)C1 C1(C(=O)NC(CCNC(CC(=O)NCC)=O)C)C2COC(C)(C)OCC12 c1(CC)ccc(Nc2ccccc2C(=O)NC2(CC)CCOC2C)cc1 Cc1ccn2cc(C(=O)NC3CC4CCC3N4C(C3C(C)(C)C3(C)C)=O)nc2c1 c1(OC)cc(=NC(=O)C(C2CCCC2)NC(=O)CC2(O)CCCCC2)[nH]n1C C1(CC2CC3C=CCC(C2)C3)CCc2ccccc2N1Cc1c(Cl)cccc1 C1(C(N2C(CNC(C(COC)(C)C)=O)COCC2)=O)CCC2(CC1)CC(O)C2 C1(C(N(CCC(=O)N(CC(C)CO)C)C(C)C)=O)CC(C)(C)CO1 CCC(C)(C)C(C(=O)N1CCC(NC(=O)C(C)(C)c2ccns2)CC1)OC c1(C(=O)NC2C(NC(=O)C=Cc3cn[nH]c3)CC2)cc2cc(F)ccc2o1 C1(CNC(c2cc(Cl)ccc2Cl)=O)C2CCC1CN(C(C1CCC1)=O)C2 N1(C(c2cc(C(=O)OC)on2)=O)CCOC(CNC(=O)Cc2cncn2C)C1 N1(C(C(C)(C)OCC)=O)CC2C(C(=O)N(C)C(c3ccncc3)C)C2C1 c1(OC)cccc2[nH]c(C(=O)NC3CN(Cc4cnc(Cl)c(Cl)c4)CC3F)cc12 C(C)(CCC(C)(C)C)NC(C(CC#C)NC(=O)CC=C(C)C)=O c1(C(=O)O)cccc2c1CN(C(c1cn(Cc3cccs3)nn1)C1CC1)C2 c1(C(=O)NCCC2CCCN(C(C(CC)(C)CC)=O)C2)cnc2n1CCCCC2 C(C)(CCC#N)(c1n(C(C)C)nnn1)NC(C)Cc1ccco1 C1(CC(=O)NC(C2CCCCC2)CNC(C2CCO2)=O)CC2CCC1CC2 C(=O)(CC(C)(C)CC(=O)N1CCCC(O)(CCNC(C2(CF)CC2)=O)C1)OCC Cc1[nH]nc(CO)c1C(N1CCC(C(=O)NC2CCCC(C)C2)CC1)=O C(=O)(C1CSc2ccccc21)N1CC(NC(CCC=CCC=C)=O)(COC)C1 c1(OCC#C)ccc(CNC(C2CNCCN2Cc2nccs2)=O)cc1 c1(C(C(=O)O)N(C(C(c2cnn(C)c2)OC)=O)C)ccc(C)s1 C1(N(C(c2c(CCC)nco2)=O)C)CCCN(C(=O)COCC(C)(C)C)CC1 c1(CC)cc(N(C=O)Cc2ccnn2C2CCC2)n(C)n1 O=C(CC(O)C(Cl)(Cl)Cl)NC1CC(OC2CCOCC2)C1 C(C(=O)N1CCCCCO1)(C1CCC1)NC(C1CCCN(C)C1)=O C1(CC)CN(C(C2CC(O)C2)=O)CC1NC(C1CC=CCC1)=O C1(CNC(CSCCC)=O)CN(C(=O)CCn2ccc(C)n2)C2(CCC2)C1 c1(CCC)onc(C)c1C(=O)NC1CCC(F)(CNC(C2(C)CCOC2)=O)C1 CCCCCC(C)(CC)C(=O)N=S1(=O)CCC2(CC1)CN(C(=O)CSC)CCO2 CC(C)C(C)CC(=O)N(C1CCCC1)CCn1cc(C2CC3(CCC3)C2)nn1 C(=O)(C(C)N=c1cc[nH]cc1)N1C(C(N2CCC(F)(F)CC2C)=O)(CC)CCC1 CC(C)CC(F)C(=O)N1CCCC(NC(=O)CCc2cccnc2F)C1C c1(C(=O)NC2CN(C(C(CCC)(C)C)=O)CC(O)C2)cccn2nncc12 c1(CN2CCC(NC(c3cc(Br)ccc3F)=O)C(F)C2)c[nH]c2c(Br)cccc12 C1(CCC(=O)N(C(C)CNC(C2CCN(C(N)=O)CC2)=O)CC)C(=O)ON=C1C c1(C(=O)NC(CC(N)=O)c2ccccc2)cc2c(s1)C1CCC2C1 N1(C(CC(C)(F)F)=O)CC2CCOC2(CNC(C2(Cl)CC2(F)F)=O)C1 c1(CNC(C2CC2C(=O)NC2(C)CC2)=O)cc(OC(F)F)ccc1F C1(C(=O)NCC(C)(C2CC2)NC(=O)CC2CCCC(C3CC3)O2)CCCCC1O C1(CC)(NC(C2C=CCCC2)=O)CCN(C(=O)C(O)COC)CC1 c1(C(=O)NCC(C)N(C(c2cc(OC)cc(F)c2)=O)C)cc2n(c(=O)c1)CCS2 C1(C)(CC)CCN(C(CCc2ccco2)C(=O)NCc2ccccc2OC)C1 C1(C(=O)NCC2N(C(CCNC(N)=O)=O)C3CCC2C3)CCCC2(CCC2)C1 N1(C(CCC(=O)NCC)=O)CCCN(C(c2cc(Br)co2)=O)CC1CO C1(C(CC)C)CCN(C(=O)CNC2(c3nnc(C)o3)CC2)C1 C=C(Br)CCC(=O)N(c1ccccn1)Cc1cc(C)n(C)n1 N1(C(C(C=CC)O)=O)CC(NC(C23CC(C#N)(C2)C3)=O)C(CO)C1 N1(C(=O)NC(C)CCn2cc(Cl)cn2)CC(C)OC(C)C1 CC1CC=CCC1C(=O)NCCC1CCCN(C(=O)C=C2CCOCC2)C1 C=C=CC(C)C(=O)N1CCCC(NC(=O)C(C)SCC)C1 N1(C(C(Cc2c(C)noc2C)C)=O)CC2CCCC2(NC(=O)C(C)C)C1 N1(C(C)=O)CCc2cc(NC3CCCCN(CCCOC(C)C)C3)ccc21 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(c2cc(Cl)nnc2Cl)=O)C(C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(C(C)(O)CNC(=O)Cn2cnnn2)C1 c1(C(N2CC(NC(C(c3ccno3)C)=O)C(C)C2)=O)cc2ccccc2cc1N N1(C(CCN(C)OC(CC(C)C)C)=O)CC2CC1(c1cn(CC3CC3)nn1)CO2 Cc1cc(OCCNC(N2CCC(C)C(N(C)C)C2)=O)ccc1Cl C(CN=C(NCC1CCCCC(F)(F)C1)N1CCN(c2ncccn2)CC1)SC CC1(C)CCN(C(=O)C(O)c2ccco2)CC1NC(c1cc2ncccn2n1)=O C1(CNC(C(C)OCCOCC)=O)CCN(C(=O)C=CC)CC1(F)F N1(C(C2C(C(=O)NCCc3ncc(C)cn3)C2)=O)CC(C)N(C)C(C)C1 C(=O)(C(O)CCNC(C1CC(O)C(F)C1)=O)NC1C(OC)C(O)C1 CC1ON=C(C(=O)NCC2CCN(C(c3cn(CC(F)F)cn3)=O)C23CC3)C1C CCC(C)C(=O)C(=O)NCCC(=O)N1CCC1CC(C)(C)C C1(NC(C2N(CC)CC2)=O)CCN(C(=O)C(COC(C)=O)OC)CC1O CCCCC(O)C(=O)N(CC(=O)NC(c1ncccc1C)C)CC1CC1 c1(C(=O)NCC(CC(C)C)NC(c2c(SC)ccs2)=O)ncnc2ccsc12 N1(C(CCCCSC)=O)C2COCC1CC(NC(=O)CC1CCCCN1C)C2 c1(N(C(=O)C(C)(F)F)C(C(C)C)=O)ccccc1N1CCOCC1.C1=CNC1=O C1(C)(CC(=O)NCCc2n(CC)cnn2)CCN(C(C2CCC2C)=O)C1 CCC(CC(=O)NCc1ncccc1C(=O)NC1CCCC(C)C1C)C1CCC1 C(C(CC(C)C)C(=O)NCCCN(C(=O)CCNC(=O)C=CCl)C)OC C1(O)(CNC(C=NOC)=O)CCCN(C(c2cc(OC)ccc2N)=O)CC1 C=CCCC(C(=O)N1CC(N(C)C)C(O)C1)NC(C1CC2(CC2)C1)=O C=CC1(C(=O)Nc2cnn(CCN(C)C)c2)CCN(C(=O)C2=C(Cl)CC2)C1 CC(C(=O)NCC12COC(CNC(=O)CCCN(C)C)(C1)C2)C(C)(F)F CC1CCC(NC(=O)C(C)CC(F)F)CN1C(=O)COc1ccsc1 c1(C(=O)NCC(CNC(=O)CC2C=CCC2)O)conc1-c1ccccc1 C(=O)(CC(F)(F)C(F)(F)Br)N(c1cocn1)CCOCC(C)C N1(c2nnc(SCC)n2CC)CC(COC)OC2(CCC2)C1 c1(C(=O)NC2CCC(NC(c3scc(OC)c3)=O)C2)c(CO)noc1C c1(CNC(C2CCN(C3CCN(Cc4scc(C)n4)C3)CC2)=O)c(F)cccc1F.O c1(NCC2(F)CN(C(c3ccccc3-n3ccnc3)=O)C2)ccc(Cl)c(Br)c1.C1(C)CCN1 c1(C(=O)NC(C)CCCNC(=O)CCC(N)=O)nc2cccnn2c1Br N1(C(C(CC)CO)=O)CCC(CNC(=O)CC2CCOCC2)C(F)(F)CC1 C(c1ccncn1)=CC(=O)NCC1CC(NC(C2(c3cccs3)CCCC2)=O)C1 c1(OC)ccc(F)cc1C1(C(=O)OC)CC1.C1(N(C2CCCC2)CCS)CCCC1 N1(C(C=C(C)C)=O)CCCC2CN(C(C3Cc4ccc(C)cc4S3)=O)CC12 c1(SC)cc(F)ccc1C(=O)NC1CN(C(c2cnccc2C)=O)CC1O C(=O)(C(C)CC(C)(C)C)N1CCC(NC(c2c(C)nc(C3CCC3)o2)=O)C1C c1(CC(=O)N(C2CC2NC(C=CCOC)=O)CC)cccc(C(C)(C)C)c1 c1(CC)c[nH]nc1C(N1CC=CC1C(=O)NCCNC(C1CCC1)=O)=O C1(CNC(c2cn(C3CCOC3)cn2)=O)CCCCCN1C(=O)Cc1cnns1 CC(C)(C(=O)O)C(C(F)(F)C(F)(F)F)NC(c1[nH]ccc1C1CC1)=O C1(CNC(CCOCC)=O)CC2CCC1N(C(c1ccc(=O)n(C)n1)=O)C2 N1(Cc2[nH]cc(C)c2)CC2CCN(C(c3cc(I)c(F)cc3F)=O)C2C1 c1(COC)ccc(NC(=O)CC2CCCN(C(C3(C)COC3)=O)C2)cc1N c1(CC)nnc(CNC(=O)C(C)C2CC(NC(=O)C(C)N3CC(C)C3)C2)o1 C1(NC(C(C)C(C)(F)F)=O)CC1C1CCN(C(=O)CC(C)(C)O)CC1 c1(C(=O)NCC2C=CC(CNC(=O)COc3cccnc3)C2)cc(Cl)nnc1O N1(C(C(CN(CC)CC)F)=O)CCCC2(CCCN2C(=O)C#CC2CC2)C1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2CN(C(C3CC=CCC3)=O)CC2C1 C1(C(=O)NCC(CC)OC)CCCN(C(c2c(C)cnn2C(C)C)=O)C1 N1(C(Cn2c(C)ccn2)=O)CCC2C(C(=O)NC3(C)CCC3)C2C1 c1(SC)ncc(C(=O)N(C(C)CNC(c2cnc(N(C)C)cn2)=O)C)c(O)n1 c1(C(=O)OC)[nH]c(=NCC2CC(NC(=O)CC3CNC(=O)C3)C2)sc1C c1(NCC2CCN(C(CC)CC)C2)cc(Cl)c(C)c(Br)c1 N1(C(CC(OCC)OCC)=O)CCCCC(NC(C2(C)CCCC2C)=O)C1 C1(NC(=O)NCCN(C(=O)OC)C)C2CC3COC1C3C2 C1(C(=O)NC2C3CC2N(C(=O)COCC2CCOC2)C3)CC1C1CCOCC1 CC1COC(C)(C)CN1C(=O)C(Cc1ccco1)NC(=O)Cn1[nH]cnc1=N C(C(Cc1ccccc1)C(F)(F)F)NC(CCN1CCN(C(C)=O)CC1)=O N1(C(C2(CC)CC2)=O)CCC2(CCC(NC(c3cnc(C4CC4)c(C)c3)=O)C2)C1 Cc1ccc2c(c1)CC(C(=O)O)N2CCN(C)C.c12cccc(Br)c1COC2C C12CCCN(C1)C2=O.C(=O)(CCN(C(CC)CC)COC(C)=O)N(CCC)C C1(CC(=O)NC)CN(C(=O)Cn2cccn2)CCN1C(c1cocn1)=O N1(C(=O)NCCS(=O)c2ccccc2)CCC2(CCCC(CC(=O)O)O2)CC1 C(=O)(C(O)CC(F)(F)F)NCC(CC(=O)Nc1ccc(F)c(CO)c1)C1CCC1 N1(C(C2NC(=O)C(F)C2)=O)CC2CCCC(C1)N2C(=O)CCOC1CCC1 Cc1c(C(N2CCC(CNC(C34CCCC3C4)=O)C2)=O)cnn1C(C)C(C)(C)O Cc1cc(O)cc(C)c1C(=O)NC1CN(C(c2cccn2C)=O)CCC1CO c1(C(CC)Oc2ccc(C3SCC(N(C)C)C3)nc2)ccc(OC)cc1C C1(C(=O)NCCCCC(C)NC(CNC(C)=O)=O)CCn2c(C)nnc2C1 N1(C(C(C)Cc2ccccc2)=O)CCC(NC(c2scnc2C2CC2)=O)CC1C C#CC1(C(=O)NCC2CCCN(C(=O)C(C)N(CC)CC)C2CC)CCCCC1 N1(C(c2c(C)nco2)=O)CC2(CNC(c3ccn(C4CC4)c3C)=O)CCC1CC2 C1(CC)CN(C(c2coc(CNC(c3cnc(OC)s3)=O)n2)=O)CC(=O)N1 N1(C(CCNc2scc(C)n2)=O)CC(CNC(=O)C(N)=O)OC2COCC12 c1(OC)c(C(N2CCC(NC(=O)Cc3ccoc3)C2C)=O)ccc(Cl)c1C C1(NC(C2C(C)(C)CC2)=O)CCC(F)(CNC(=O)CCc2ccccc2Cl)C1 CON1CCC(CC(=O)NCC2CC2CNC(=O)C=Cc2ccccc2C)CC1 N1(C(Cn2ccc(C)n2)=O)CC2CC(O)C1C2NC(C1CC(O)C1)=O CCCCCC(O)C(=O)N1CCCC1C(C)NC(c1cnoc1C)=O C1(C(=O)NCCC2(OC)CN(C(CC3CC(=C)C3)=O)C2)COC2(CO)CC1C2 CCC(C)(CNC(C1CCCC1)=O)NC(C1C=CCCC1)=O c1(NC(C(C)C)=O)ccc(C(CC2C(NC(=O)OC(C)(C)C)CC2)OC)cc1 C1(CNC(C2(CC#C)CC2)=O)CC(NC(=O)Cc2c(C)cnn2C)C1(C)C CC12CCC(C(N3CCCC(NC(=O)CC(F)(F)C(F)F)CC3)=O)(CC1)OC2 c1(CC(=O)NC(CC=C)CNC(C2CC23CCC3)=O)ccnc(C(F)(F)F)c1 CC(O)(C(=O)N1CCN(C(c2ccc(C3CC3)cc2F)=O)C(CF)C1)C(F)(F)F c1(NCCCN(C)C2CC2)ccccc1NC(c1ccccc1)=O C=C=CCC(=O)NCC(COC)NC(=O)CCCn1cccn1 O=C1CCCC(CC(N2CC=CC(NC(=O)CCCc3cc[nH]n3)C2)=O)C1 C1(C(=O)NC(c2ccc(C)cn2)C)CCC(O)CN1C(C1CCCN1C(C)C)=O C(=O)(CCCCC(F)F)N1CC(CNC(CC2CC(C)(C)C2)=O)C(C)(C)C1 C#CCC(C)(C(=O)Nc1ccc(CO)c(F)c1)NC(=O)C(CC)CC=C CC(C)CCCCCC(=O)NCCCCNC(=O)CC1C=CCCC1 C(=O)(C#CC1CCCO1)NC1(CNC(=O)C=Cc2ccccc2)CCOC1 CC(C(=O)N1CCC1CNC(c1cnn2c1OCC2)=O)C(C)(C)C C1(C)(C(=O)NCCCN(C)C2CC2)CCN(C(C2CC2C2CCCC2)=O)CC1 C(=O)(C(F)C(F)(F)F)N1CC(COC)(CNC(=O)C(C)CC2CCCC2)C1 CC1CCC(CO)CN1C(=O)COC1CC(NC(=O)C=Cc2ccco2)C1 C1(C(=O)OC)(NC(N2CCOC(CCOC(C)(C)C)C2)=O)CCC2CC12 N1(C(C(=O)NCCOC)=O)CCCC(O)(CNC(=O)C(CN(C)C)N(C)C)C1 CCC(CNC(=O)C(C)C#N)(CC)NC(c1cc(C2(C)CC2)n[nH]1)=O N1(C(CCCC)=O)CCC(C2CC2)(CNC(C2CCCC(CF)C2)=O)C1 c1(C(N2CC3C(NC(c4ccc(CC)o4)=O)(C3)C2)=O)ccc2ccncc2c1 C1(C(=O)NC2CC(NC(=O)COCC3CCC(O)C3)C2)CCCCNC1=O c1(CC(=O)NC2C(OC)COCC2)ccc(O)c(C)c1 C1(NC(c2cc(CCC)oc2C)=O)CCN(C(c2sc(OC)nc2C)=O)CC1F C=CCCCC(=O)NCC1CN(C(c2ccc(CC)cn2)=O)C2CC12 C1(CC(N2CC(C3CCC3)C2)=O)CC2(C1)CN(C(C1C=CCCC1)=O)C2 C#CCCCC(=O)N(CC(C)NC(=O)CNC(c1ccccc1OC)=O)C C(=O)(C1=NNC(C(F)(F)F)C1)N1C(CNC(=O)CSCCF)CCC1 c1(N)ccccc1OC.C1(CCNC(C)=O)CCCN1CCOCC(C)C C1(CNC(C2(CC#C)CC2)=O)C2CCCC1N(C(c1ccc3c(c1)CCC3)=O)C2 C12(NCC=C(C)C)CCC(CC1n1cc(CNc3c(C)ccnc3Br)nn1)C2 N1(C(c2c(C)nc(C)n2O)=O)CCC2CN(C(c3cnn(C(C)C)c3N)=O)CC12 n1(CC(=O)NCC2(C)CCCN2C(=O)Cc2cnccn2)cccc(O)c1=O Cc1oc(CNC(c2cc(C3CC3)on2)=O)nc1C(=O)NC1CS(=O)(=O)C1 C#CC1CN(C(C2CCN(C(=O)Cn3cnnc3)CC2O)=O)CCN1C c1(C(N(C2CCCC2)CC=C)=O)ncoc1CNC(=O)C(CO)OC N1(C(c2ccc(CNC(C(CC=CC)C)=O)s2)=O)CC2C=CCC(C2)C1 Cc1cc(C(=O)NC2CN(C(=O)Cn3cccn3)CCC2C)nc(O)n1 c1(C(c2cn(C)nn2)C2N(C(=O)Nn3nccn3)CCC2O)cccc(N=[N+]=[N-])c1 c1(C(N2CCN(C(C(C)C#N)=O)C(c3nccn3C)C2)=O)nc2ccccc2[nH]1 C(=O)(CC(C)CC(C)(C)C)N1C(C)C(C(=O)NC2CCC3(CCCC3)C2)CC1 c1(C(N(CCC)CCNC(=O)CCn2cccn2)=O)csc(C(C)(C)C)c1 C1(N(C(c2c(C)n(CCO)nc2)=O)C)CN(C(c2cc(Cl)ccn2)=O)CC1(C)C C1(C(=O)NCC2(CF)CC2)CC2CCC(C1)N2C(=O)CC1CCCOC1 c1(C(=O)NC2CC2NC(c2cc([N+](=O)[O-])c[nH]2)=O)ncc2ccccc2c1O C1(C(=O)NC2CC(C)(NC(=O)C(C3(O)CCCC3)F)C2)CN(S(N)(=O)=O)C1 Cc1ccc(C)c(-c2ncccc2NC(=O)NCC23CCN(CC2)C3)c1 Cn1nc2c(c1C(N1CCN3CC(F)CC3C1)=O)CN(C(=O)C(N)=O)CC2 C(=O)(C(C(C)NC(c1ccnc(C)c1N)=O)C(C)C)NCCCNC(=O)NC C1(C(N(CC(C)OC)C)=O)CCN(C(=O)Cc2ccc(O)cc2)CC1O C1(NC(c2ccn(-c3ccccc3)n2)=O)C2CCN(C(=O)Cc3cnco3)C12 c1(C(C)NC(=O)NC(C2CCC(=O)N(C)C2)CC)oc2ccc(OC)cc2c1C N1(C(C(C)OC(C)(C)C)=O)CC(C(C)(C)O)(CNC(C2CCCCS2)=O)C1 c1(NC(CC2OCCN(S(CCCC)(=O)=O)C2)=O)cc([N+](=O)[O-])c(F)cc1C C=CCC(C(=O)NCCCCC(CO)NC(c1ccc(OC)cc1F)=O)C(C)C c1(NC(C2COCCN2C(=O)NC2CCCCC2OC)=O)cccc2c1CCN2 CC(F)(F)C(C)(C)C(=O)NC1CN(CCCNC(=O)C2=CCCCC2)CCO1 c1(C(=O)NCCCC2N(C(C(CC)N(C)C)=O)CCC2)noc2c1CCCC2 c1(N2CC(NC(c3cccc(C(F)(F)F)n3)=O)C(O)C2)ncnc2cc(Br)sc12 N1(C(C2(SC)CC2)=O)CC(CN(C)C(C2(C)CCNC2=O)=O)C2(CC2)C1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC2CNC(=O)C=C(C)c1ccccc1C N1(C(c2c(C)nn[nH]2)=O)CCC2(CC2C(N2CC(O)C(O)C2)=O)C1 C(C(=O)N=c1cccn[nH]1)N1CCN(S(C(C)C)(=O)=O)C2(C1)CC2 N1(C(C(n2ncc(C)c2)C)=O)CC(F)CC1CC(=O)NCC1CC1Cl C(=O)(C(O)CC(C)C)c1cn(C2C(SC)CCC2)nn1.N12CC(C(F)C1)C2 c1(-c2cn(CC3CN(C(C4(C=C)CCOCC4)=O)C3)nn2)cc(Cl)cc(Cl)c1Cl c1(C(=O)NCCC2CCCN2C(c2sc(F)cc2Cl)=O)ccc2cccnc2n1 c1(C(=O)OC)ccc2c(c1)CCC2NC(=O)C(=O)NCCC1CC2CC1C2 C12(NC(Cc3nnc(C)o3)=O)CCC(CC1)N(C(=O)CCOCC1CCCO1)C2 c1(NC(=O)N(C2CC(C#N)C2)CC2C(C)C2(F)F)cccc(CC2CCOCC2)c1 c1(C(N2CCC(NC(CC3(N(C)C)COC3)=O)C2)=O)ccc(O)nc1Cl N1(C(c2cc(C)c(C(F)F)cn2)=O)CC2(CCCCN(C(C3CCCC3)=O)C2)C1 Cc1cccc(Cl)c1CCC(=O)NC1C=CCN(C(=O)CNC2CCCCC2)C1 c1(CNC(C2CCC(C)S2)=O)nc2c(s1)CN(C(=O)CC1(CO)CC1)CC2 N(C)(S(=O)(=O)N1CCNC(C2CCC(F)(F)CC2)C1)CCOC C1(C(N2C(CC(=O)NCCCS(C)(=O)=O)CCC2)=O)CC2C=CC1CC2 C1(OC)CC(CNC(C2CCC(F)CC2)=O)N(C(c2n[nH]c(C)c2Cl)=O)C1 c1(C(=O)NCCN(CCC)C(C2CCCS2(=O)=O)=O)cc[nH]c(=N)c1 N1(C(C2CC(C)(CC)C2)=O)CCC2(CCCN2C(=O)C(=O)N=S(C)(C)=O)CC1 c1(C(=O)NCC2C(CNC(CCOCCCOC)=O)C2(F)F)c(C)n[nH]c1C c1(CCC(=O)N(C)CCNC(c2ccc(N(C)C)s2)=O)ccc(O)nn1 Cc1c(C(=O)NC(C2CCN(C(C3CC3F)=O)CC2)C)cncc1Br C#Cc1ccc(CNC(=O)C(=O)NC2C3CC4C(C3)C24CO)cc1 c1(CC(C)NC(C2CC3CC3N2C(=O)CS(C)(=O)=O)=O)ccc(O)c(O)c1 N1(C(C2CC(=O)NC2)=O)CCC2C1CCCN2C(c1cnc2cccnc2c1)=O C1(OC)CC(NC(=O)CCC(C)SC)CN(C(c2ccc(CO)cn2)=O)C1 N=c1ccn(CC(N2CCCC(Cc3ccccc3)CC2)=O)c(O)n1 N1(C(C2(COC)CC2)=O)CCC2CN(C(c3ccc(Cl)nc3)=O)CCC12 C(=O)(C(F)C(C)CC(C)(C)C)NCC1(NC(C(CCSC)O)=O)CCCCC1 c1(C(C)=O)ccccc1OCC(O)CN(C(=O)CCCN(C)Cc1ccsc1)C CC1(C)CC2(CC(NC(=O)C(CC3CCOCC3)NC(c3ccsc3Cl)=O)C2)C1 N1(C(CC(=O)N(C)C)=O)CC2COCC2(C(=O)NC2CN(C(N)=O)CC2(C)C)C1 Nc1c(C(N2CCC(C(F)C(=O)NC3CC(O)C3)C2)=O)cccc1F C1(C(=O)NCC(C)N(c2nc(C3CC3)nc(=N)[nH]2)C)CS(=O)(=O)CC(=O)N1 c1(C(=O)NC(C2CCN(C(C3CCC(SCC)CC3)=O)C2)C)cc(O)ccc1F Cc1nc(O)c(C(=O)NC(C)CCNC(=O)C2=CCCC2C)nc1C c1(CC)c(C(=O)NC2CCN(C(=O)C(O)CCSC)CC2)csc1C N1(C(CCC#C)=O)C(C(=O)Nc2cccc(CCC)c2)CCC12CC2 Cc1nc(C(=O)NCC(C)(C(C)C)NC(=O)CC(C)C(F)F)ccc1C#N C1(CNC(CC2(COC)CC2)=O)(NC(=O)Cc2n[nH]c(=N)s2)CCOCC1 C1(C(N(CCN(C(CC2(N(C)C)CC2)=O)C(C)C)C)=O)CCN(C(N)=O)CC1 c12cccc(c1)CS2.c1(CC(C2(C)CC2)=O)ccccc1SC1(C(=O)OC)CC1 Cc1oc(C2CC2)nc1C(=O)N(C1CCN(C(c2coc(C#N)c2)=O)C1)C C(C)(CCC(=O)NC1(CCNC(C2CC(O)(C(F)(F)F)C2)=O)CCC1)SC c1(CNC(CC(C=C)C)=O)cc2n(n1)CCN(C(=O)CCCC#N)C2 Cn1cc(C(N)C(=O)NCC(=O)NC2COCCO2)nn1 CC(C)C(C(=O)N1CCCC1CNC(=O)Cc1cccs1)Sc1ccccc1 C1(OC)CN(Cc2cscc2Br)C2(CCC2)C1 c1(C(=O)NCC(C)N(C(C(C)C2CC2)=O)C)oc(Br)nc1C(F)(F)F c1(C(=O)NC2(CC(=O)NCCC(CCC)O)CC2)cc(C#N)ccc1N c1(OC)nccnc1-c1nc(-c2ccc(C(F)(F)F)nc2)n(CC2CCCO2)n1 C1(NC(c2nc(C)sc2C)=O)CCCN(C(C2C3COCC23)=O)CC1 c1(C(=O)NC2CCC(N(C(=O)CC3(C#N)CCC3)C)C2)ccc(F)c(F)c1 C(=O)(C1COc2cc(C)c(C)cc21)NC1CC(CCNC(CC=C)=O)C1 Cc1cc(C(N2CC(NC(C3C4C=CSC34)=O)C(F)(F)C2)=O)cnc1C c1(CCN=C(NC(C=C)C)NCc2ccsn2)c[nH]c2cc(F)c(F)cc12 N(C(=NCC1CCC(F)CC1)N(C)Cc1ccccc1)CCc1c(C)cccc1 C(=O)(CC(C)C(=O)NCC1CN(C(C2(OC)CCSC2)=O)CC12CC2)OCC C1(C(N(C2CN(C(c3ncccc3Cl)=O)CC2(C)C)C)=O)CCCCCS1(=O)=O C=CC(C)(C)CC(=O)NCc1csc(CNC(=O)CCCOCCC)n1 N1(C(c2cc(COC)[nH]n2)=O)CC2(CCCC(CNC(=O)C(C)(C)CSC)O2)C1 N1(C(c2sccc2OC(F)F)=O)CCC2(C1)CN(C(C1(F)CC=CCC1)=O)C2 N1(C(CCc2cc(OC)c(O)cc2F)=O)CC2CCCCCCC2C1 N(C1CCCn2ccnc21)C(C1N(C(Cc2c(C)scc2)=O)CCC(C)(C)C1)=O c1(CN(CC(CC(C)C)OC)C(CC)C(=O)OC)ccc2c(c1)CCC2 C1(C)(CC)C=C(C(=O)NCC2(O)CCN(C(=O)Cc3csc(C(C)C)n3)CC2)C1 C12(C(=O)NC(c3nc(C(N4CCC5CC45C)=O)co3)C)CC(C#N)(C1)C2 N1(C(CCC=C)CSc2ccccc2)CCc2c(ccnc2-c2nn[nH]n2)C1 c1(OC)ncc(NC(c2cc(F)cc(F)c2)C)cc1Br N1(C(N2CCCC2NC(=O)Cc2ccccc2)=O)CN(C(=O)C(N)=O)CC1CO C1(CC)CN(C(c2ccc(Cl)o2)=O)CCN1C(c1ccc(C#N)s1)=O c1(NC(C2C(CNc3c(C(=O)OC)nccn3)C2)=O)ccc(C)c(Cl)c1 c1(C(N2CC(C3OCCN(C(CCCCC#C)=O)C3)C2)=O)ccc2nnnn2c1 N1(C(C(n2cnc(C#N)n2)C)=O)CCC2(CC1)CC(NC(=O)C(C)CO)CCO2 c1(CCNCc2c(C(=O)OC)nns2)ccc(Br)cc1[N+](=O)[O-] C(=O)(C(C)(C)C(C)(C)C)NC(CC1CN(C(C2(C)ON=C(C)C2)=O)C1)C C#Cc1ccc(C23CC(CC)C(OC2)C3)cc1.N1(CC(=O)NCCC)CCCC1CC c1(C(=O)NCC2C(NC(CC=CCC)=O)C2)cc(Cl)c(Br)cn1 c1(C(C)C)ccc(C(=O)NC2(CNC(C3(C)CCOCC3)=O)COC2)c(Cl)n1 C(=O)(CCC1=NNC(=O)CC1)NCC1C(C)CCN(C(C2(F)CC=CC2)=O)C1 C(CC(=O)NC(C)(C)CC(C)(C)C)(C(F)(F)F)NC(C1C(=C)C1)=O CC(CC(C)(C)C)C(=O)N(CC(O)CNC(=O)C=C1CCC(C)(C)CC1)C c1(NC(N2CC(OC(C)(C)C)C2)=O)ccc(C(=O)OC2(C)CCCO2)cc1 c1(N(CC(CCC)C)C)nc(=NCc2cc(C)cc(Cl)n2)[nH]c2c(F)cccc12 CCC(C)CCC(=O)N1CC(C(=O)NCc2cnn(CCF)c2)CCC1C CN1CC=C(C(=O)NCC(C)(O)CNC(=O)C(C(C)(C)C)C2CCC2)C1.C(C)(C)(C)O C1(NC(c2cc(CC(C)C)on2)=O)COC2CN(C(=O)CS(N)(=O)=O)CC12 N1(C(c2cn(C3CCCC3)nn2)C(=O)NCCCF)CCCCC12CC2 c1(SC)nc2ncnc(NC(C)CC(C)NC(C3(F)CCOC3C)=O)c2s1 C(=O)(C1CCCc2nc[nH]c21)N1CC2C(CNC(C=CCCC=C(C)C)=O)C2C1 c1(C(=O)NCC2CC(CNC(=O)CCCCC3CC3)OC2)cnn2ncccc12 N1(C(C(C)=C(CC)C)=O)CC2CCCN(C(c3ncnc4c3CCC4)=O)C2C1 N1(C(c2c(C)noc2C)=O)CCCC(CCNC(C2CC3C(C2)C3(F)F)=O)CC1 C(=O)(CS(=O)(=O)CCOC)NC1C(CC)CN(C(=O)C(C)OCCOCCO)CC1 C1(CC(N2C(CN(C)C)C=CC2)=O)CC2(C1)CN(C(C1CCCCC1(C)C)=O)C2 c1(-c2c(C)cccc2F)nc(=NC(=O)NCC(=O)NCc2ccsc2)o[nH]1 N1(C(C2(CCCC)CC2)=O)CCC(C)(C)C(NC(=O)CCCCC(=O)NC)C1 Cc1cc2[nH]c(C(=O)NC3CC3CNC(=O)CC=Cc3cccc(F)c3)cc2o1 Cn1ccc(C(=O)NC2CCCC2(C)NC(c2cc(Cl)ccn2)=O)cc1=O C1(C(N2CCCC(c3onc(-n4c(C)ncc4)n3)C2)=O)COC2COCC2O1 c1(C(N(CCNC(C(C)OC)=O)C(C)C)=O)ccc2c(c1)CC(C)O2 c1(CC(=O)N(CC(CC)NC(=O)CCc2cc(OC)no2)C)csc(C)n1 c1(OC)ccc(Cl)c(C(c2nnnn2C2CC2)NC(C)CC2CCOCC2)c1Cl c1(C(=O)NCCCC(C)NC(c2cnn(C3CC3)c2)=O)cc(N(C)C)ccc1N C1(CNc2c(C)c(N3CCC=C(Br)C3)ncn2)CCCC2(CNC2)O1 N1(C(c2c(CC)nco2)=O)CCCC(NC(=O)CC(C)(C)OC)C1C C1(C(=O)NCC(CC=C)NC(=O)C=CC)CC2CC(=O)C1O2 C12(C(N(CC(COC)O)C)=O)CCCC1N(C(=O)CC1CC(C)C1)CC2 C1(CC=C)(NC(C2COC(=O)C2)=O)CCN(C(=O)CCF)CC1 N1(C(CCC(=O)NCC)=O)CCC2CCCC12CNC(c1nccnc1CC)=O C1(C(=O)NC(=O)CC2CCCCO2)CC(O)CN1NC(C1CC1)C1CC1 C(C(CC(=O)N(C1(C(N)=O)CC1)C)OC)NC(C1(CCC)CCC1)=O c1(NC(C2(c3c(C)cccc3)CC(ON)C2)=O)cc(C#N)ccn1 c1(OC)cc(C(=O)NC2(CF)CCN(C(=O)C(C)(C)C3(O)CCOC3)C2)n(C)n1 C1(NC(c2cccc(CSC)c2)=O)CCCCN(C(=O)C(O)C(C)(C)C)C1 C1(C(=O)NCC(CC=C)NC(c2cc(C)c(CO)cn2)=O)COCC2(CCC2)O1 c1(C(=O)NC(CC=CC)C(=O)N(C)Cc2cnccn2)nccc(C)c1N N1(C(c2c(CC)[nH]cc2)=O)CC2OCC(N(C(c3ccc(O)cc3)=O)C3CC3)C2C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)CC=C)ccc(Br)cc1 n1(CC)cc(C(=O)NCCC2(NC(=O)CCC3CCCN3C)CC2)c(C)n1 c1(OC)nc(CS(=O)(=O)NCC2CCC(C(F)(F)F)O2)ccc1C C(=O)(CCCC(=O)N(C)C(C)CC)N1CCCC(Nc2c(C)cccc2)C1 C(CC(C(=O)NC(c1ncc(C)cn1)C)NC(c1sc(O)nc1C)=O)OC c1(CN2CCC(CC(=O)NC(C(C)O)CO)C2)c(F)cc(Cl)cc1Br C(=O)(C1=C2CCCN=C2NN1)NC1C(NC(=O)C=CC(F)(F)F)CCOC1 c1(N2CC(NC(C3C(C(F)(F)F)C3[N+](=O)[O-])=O)C2)nc(C2CC2)nc2c1CCC2 C1(F)(CNC(=O)COc2ccccn2)CCCN(C(c2cc(O)ccc2Br)=O)C1 c1(C(N(C2CC(NC(c3ccc(O)cc3Cl)=O)C2)C)=O)coc2ccc(Cl)cc12 N1(C(CC=CCC)=O)CC(NC(c2coc(-c3cccnc3)n2)=O)C2(CC2)C1 c1(CC)ccc(F)c(C(N2CCCCC(NC(=O)C(C)(Cl)Cl)CC2)=O)c1F c1(NC(C2C=CC(NCc3ncn(C)c3)C2)=O)cc(F)c(Cl)cc1Cl C1(CNC(C2CCOCC2)=O)CC2(CCN(C(c3c(F)cccc3F)=O)C2)CO1 c1(C(N2CC(C3CN(C(C4CC(OC)C4)=O)C3)C2)=O)cc(F)cc2nn(C)cc12 O=S(=O)(c1cnc(NC2COCCC2O)c(Cl)c1)NCc1cc(F)ccc1F C1(NC(c2nc[nH]c2C(F)(F)F)=O)CCOCC1NC(C1CCOCC1)=O C(=O)(C1=CCCOCC1)N1CCCN(C(C2C(C#N)C2)=O)CC1 C1(CC(=O)NCC(C)C2CCC2)CCCCN1C(C1(C)CC(F)(F)C1)=O c1(C(=O)OCC)nnc(SCC)nc1NC1CCN(C(c2ccnc(C)n2)=O)C1 O=C1CC(C(=O)NCC23CCC2CN(C(=O)C=Cc2ccc(Br)s2)C3)=NN1 N1(CC(=O)OC(C)(C)C)CCN(C(=O)CCc2cocn2)CC1 c1(-c2onc(-c3ccc(N(C)C)nc3)n2)ccc2occc2n1 C(CC#CC(C)(C)C)NC(CCC(C)NC(=O)CC1CC(=O)NC1=O)=O C1(C(N2CC(C)(COC)C2)=O)N(C(=O)C(c2cnn(C)c2)C)CC12CCCC2 C1(NC(C(=Cc2ccco2)C)=O)C2CC(O)C1N(C(c1cnnc(O)c1)=O)C2 CC1CCCn2cc(C(N3CCC(NC(C4SCCS4)=O)C(C)(C)C3)=O)nc21 C1(C(N2CC(C)(OC)C2)=O)CC2CC1CN(C(=O)CC1CCC(C)(C)O1)C2 CC(C)(C)CCC(=O)N1CCC(CC(=O)NC2(c3ccon3)CC2)C1 N1(CC)CCC(NC(=O)C=CC(C)(C)SC)CC1.c12sccc1CNC2=O c1(C(=O)NC2(CNC(C(C)C3CCC3)=O)CCOC2)ccc([N+](=O)[O-])n1C C1(C)(CC)CCCC1NC(=O)NCc1cc(CO)nn1C n1(C(C)C)cc(C(=O)NC2CN(C(=O)C(C)N(C)C)CC23CC3)c(O)nc1=O C#CCC(C)(C(=O)Nc1cnc(C)c(C)c1)NC(=O)CC(C)C(F)F CC1(C)C2CCC1(C(=O)NCC1CC1CNC(=O)CCSc1ccccn1)CC2 C1(CNC(c2nc(OCC)oc2)=O)CC(C)N(C(c2cnn(CC)n2)=O)C1 c1(C(=O)NCC2CC2CNC(C23C=CC(CC2)C3)=O)cccc2nncn12 N#CC1(C(=O)NCC2CC2NC(c2cc(C(F)(F)F)ccn2)=O)CC=CC1 c1(C(=O)NCC2(CN(C(C(C=C)O)=O)C)CC2)cc2c(=O)[nH]ccn2n1 Cn1cc(C(N2CCC(CO)(NC(=O)CC3(C#N)CCC3)C2)=O)c2ccccc12 N1(C(CC2C(C)=NNC2=O)=O)CC2CCN(C(c3cc4sc(F)cc4[nH]3)=O)C2C1 [N-]=[N+]=NCC(F)CCNC(C1(CNC(=O)Cn2nccn2)CC1)=O C(=O)(CCCCC(F)(F)F)NCC12OCC(NC(c3nccc(C)c3)=O)C(C1)C2 C1(NC(C(C(C)C)C#N)=O)CN(C(C2CC3(C2)CC(O)C3)=O)C2(CCC2)C1 CC(C)CC(C(=O)NCCC(O)CO)ONC(C1CCC2(CCC2)C1)=O c1(C(=O)OC)nn(CC(=O)N(CC2CCC2)CC2CCOCC2)c(=O)o1 C1(CC(N2CCC(C(N3CCC3)=O)CC2)=O)Cn2c(nc3ccccc23)NC1=O c1(SC)cc(F)ccc1C(=O)NC(CO)C(C)NC(=O)Cn1ccc(C(F)F)n1 C1(C(N(C2CC(=C)C2)C)=O)CN(C(C2(C(=O)OC)CC2)=O)CC(C)(C)C1 C1(C(=O)NC2(CCNC(C3(CC)CCC3)=O)CC2)CC(OC)C(OC)C1 N1(C(CSc2ccc(OCC)cc2)=O)Cc2[nH]nc(-c3cccc(C)c3Cl)c2C1 N1(C(CC=CCC)=O)CCC(C)(CNC(C2C=CCS2)=O)C1 N1(C(C2(CC)CCCN2C(c2ccnc(OC)c2)=O)=O)CC(C)C(N=[N+]=[N-])C1 N1(C(C2(C(C)(C)C)CC=CC2)=O)CCCC(CNC(=O)C(O)C2CC2)C1 c1(CNC(N2CC(C(OC)OC)OCC2)=O)c([N+](=O)[O-])ccc(Cl)c1Cl CP(C)(=O)c1cnc(C(=O)NCc2cn(CCO)nn2)nc1 N1(C(CC(=O)NCC)=O)CCCC(N(C)C(c2ccc(C(N)=O)[nH]2)=O)C1 N(C(=NCCc1ccccc1)NC1CCOCC1)C1C(F)CCCC1 N1(C(=O)NCCCN2CCOCC2)CC2CC(F)C(C2)C1 C1(C(=O)NCC2N(C(C=CC=CCC)=O)CC(F)C2)CC2CCC(C1)C2O C(C(O)CC(=O)N(C(C)CC(C)C)C)NC(C1(C(=O)NC)CCC1)=O c12cc(c(Br)cn1)C(=O)N1CCC(CC1)C(=O)N2.N1(CC)CCCCC1C#N N1(C(C(F)OC)=O)CCC2(CCCN(C(=O)C(c3cccs3)SC)C2)CC1 Cc1cc(CN(C(C(=O)NCc2ccsc2)=O)C2CC2)c(C)s1 n1(CC)nc(C(=O)NCc2cnn(C)c2C(=O)NOCC(N)=O)c(C)n1 N1(c2nnc(C)s2)CCC2(CC1)CCN(C(=O)CCOc1ccc(Cl)cc1)CC2 S(=O)(=O)(c1ccc2c(c1)COC2)NCC(=O)NCCCNC(C1CCC1(F)F)=O S(=O)(=O)(c1ccc(F)cc1Br)N(C)Cc1cc[nH]c(=N)c1 c1(CC2N(C(CC=CC)=O)CC2)cccc(N=[N+]=[N-])c1.N12CCC(C1)C(C)C2=O C(=O)(C(COC)CC(C)C)NCC(CC=C)NC(c1nnc(C)s1)=O N#Cc1cccc(OC2(C(=O)NC3(c4ccccc4)CCC3)CCCC2)c1 C(C(F)(C(=O)N(c1ccsc1)C)C(C)C)NC(C(C1CC1)OC)=O C1(COCC)CCCN(C(=O)CC2CCN(C(C3(CCCF)CC3)=O)C2)C1 C1(NC(CCN(CC)CC)=O)CC2CCC(C1C)N2C(=O)C(CC(C)C)C(C)C N1(C(CCc2n(C)ccn2)=O)CC2CC2(CNC(=O)CCNC(C2CCC2)=O)C1 CCCC(O)(CCC)CC(=O)NCC(O)CNC(c1ccn(C2CC2(F)F)n1)=O C1(NC(=O)CC2COCCO2)CN(Cc2ccc(F)nc2F)CCC1(F)F c1(C(N2C(CNC(C(c3ccc(Cl)cc3)CC)=O)CCC2)=O)cccc(F)c1N C(N=c1c(Br)c[nH]cc1[N+](=O)[O-])C1(O)CN(C(CCC2CCC(C)O2)=O)C1 c1(C(N2C(CCNC(c3c(C)nsc3C)=O)CCCC2)=O)ccc(N)c(F)c1 N(C1CCCc2n[nH]cc21)C(c1c(F)ccc(Cl)c1F)CN1CCOCC1 CC1CC(NC(=O)Cn2cccn2)CCN1C(=O)CCc1cc(F)ccc1F c1(CC)ccc(C(=O)NCC(C)(F)CNC(C2(C)CCCC2O)=O)nc1 n1(CC(=O)NCC#CCNC(C(C)(F)c2ccccc2)=O)nc(O)ccc1=O Cc1cc(C(=O)NCC(C)(C)CNC(=O)CC(C)N2CCCC2=O)cc(C)c1O c1(C(N(C)CC2(CNC(c3ncc(CC)s3)=O)CC2)=O)cn2c(n1)CC(C)CC2 N1(C(C2OCCN(C)C2)=O)CCC(NC(c2cn[nH]c2)=O)C12CC2 C1(C(C)NC(c2cncn2C)=O)CN(C(c2cc(Cl)cs2)=O)CCO1 N1(CC(=O)NC(CN(C(=O)CC(=O)N(C)C)CC)C)C(=O)NC2(CCCC2)C1=O C(CS(=O)(=O)C(C)(C)C)c1nc(CC)nn1CCOc1ccccc1 C1(NC(c2cc(NC(C)=O)ncc2)=O)C2CCCC1CC(NC(C1(C)CC1)=O)C2 C1(n2cc(CCCOC)nn2)CN(C(=O)CNC(=O)CC2CCOCC2)CC1C C=C=CCCN=c1nc(N(C)C)c2c([nH]1)CCC2.c1(C=O)cc2n(n1)CCCO2 C1(F)(C(=O)NC(CNC(C(C(C)C)N2CCCCC2)=O)C2CC2)CCN(C)CC1 N1(c2c(C)non2)CCC(C2CCN(C(C3CCC4(C3)CC4(F)F)=O)CC2)CC1 c1(C(=O)NCC(C(C)C)NC(c2cc(OC)ns2)=O)ccc(CCF)cc1 c1(CC(=O)NC(C)CCCCNC(=O)C(C)S(C)(=O)=O)ccc2c(c1)CCCO2 C1(C(N2CC(C)(NC(c3cc(-c4cnccn4)[nH]n3)=O)C2)=O)CCCS1(=O)=O C(=O)(C(O)CC(C)(C)C)NC1CCN(C(Cc2c(O)ccc(C)c2)=O)C1 CCC(CC(=O)NC1(C)CC(NC(=O)CCN2CCCCC2)C1)OC CC1(C)CCCC(C(=O)NCC(C)(C2CC2)NC(=O)CCCCNC(N)=O)C1 c1(CNC(=O)CNC(=O)C(=O)NC2(c3nccs3)CC2)cccc[n+]1[O-] CC(C)CS(=O)(=O)CC(=O)N(CCNc1ccc(CN2CCOC(C)C2)s1)CC C(C)(C(C(=O)NCC(C)(C)CNC(=O)C(=Cc1ccccc1)OC)N(C)C)OC c1(NC(c2nn(C)cc2Cl)C)nc(N(C)Cc2nnc(O)o2)nc2sccc12 c1(N(C)C)nc(C(=O)NC2CC(CNC(=O)CCc3ccccc3)C2)[nH]c(=N)n1 CC1CN(C(=O)Cc2ccc3nn[nH]c3c2)CCCN1C(=O)C(=O)NCC1CC1 c1(C(=O)OC)cc(C(=O)N(C2CCC3(CC3)C2)C2CC2)c(C)o1 N1(C(CSCC)=O)CCC2(NC(c3nc(C)nn3C)=O)CCCC12 Cc1cc(C(=O)NC(CN(C)C)C(=O)NCC(O)C(N)=O)nc(C)c1 c1(C(N(CC(=O)NC(C(O)CO)C2CC2)C(C)C)=O)c[nH]c(C#N)c1 c1(NC)c(C(=O)NCC2CCN(C(c3scnc3COC)=O)C2)cccc1F c1(OC)ncnc(C(N2CC3CC(CNC(c4cc(CO)on4)=O)C3C2)=O)c1F C1(CNC(C2(CCCC)CCCC2)=O)COCCN(C(c2cc(C#N)no2)=O)C1 c1(C(=O)NC(C2OCCN(C(c3ccc(C)nn3)=O)C2)C)cnc(C)cc1C c1(C(=O)NCCC(C)NC(C2C(C)C2C)=O)nn(C)c2c(=O)[nH]cnc12 c1(C(=O)NCc2nccc(C(=O)NCCN(C)C)c2)c(F)ccc([N+](=O)[O-])c1Cl C(CC1CC1)(C(=O)NC1(CO)CCC1)NC(C(C1CCOCC1)C)=O C(=O)(C(C)(CNC(=O)C(C)CCC)CC)NC(C(CC)CC)C C(=O)(CC1OCCc2sccc21)NC1C(C)N(C(=O)C=CC(C)(C)C)CCC1 C=C1CCN(C(C2CCC(C)(C)CC2)=O)C(C(=O)NC(C2CCCCC2)C)C1 c1(CCNC(CC)=O)ocnc1CNC(=O)C(c1cnn(C)c1)NC(C)=O C1(CNC(CC2C=NN(C)C2=O)=O)CN(C(=O)CCCn2cccn2)CC1(C)C C1(CNC(n2cnccc2=O)=O)CCCC12CCN(C(=O)COCC1CC1)CC2 CC1CC(C)N(C(c2cc(Cl)cc(Cl)c2)=O)CCN1C(=O)Cn1ccnn1 C(=O)(C(C)CN)NCC(C)CN(C)C(c1ncccn1)=O.S(C)(=O)(=O)NC1CC1 c1(CCC)cc(C(=O)NC(C2CCCC2)CNC(=O)CC(C)COC)ccn1.SCC CC1CN(C(c2cc(O)ncn2)=O)CC(C)N1C(=O)C(C)(C)Cc1cnn[nH]1 C(C(CNC(C1CCCC(C)(C)O1)=O)S(C)(=O)=O)NC(C1(CC)CC1)=O C1(NC(CC2CC(C)C2)=O)CC2CCC1CN2C(=O)C=CCO c1(NC(C2CCN2C(=O)C(C)C(=O)OC)=O)ccc(N)cn1.c1(CSC)ccccc1 C(=O)(CC(C)C(F)F)N(CC(CNC(C(C)N)=O)C)C.CC(C)CNC(=O)CC(=O)N N1(C(c2nc(C)oc2C)=O)CC2CC(NC(=O)Cc3ccco3)CC2C1 c1(C(=O)NCCNC(C=CC(C)C)=O)ccc(NC2CC(CNC=O)C2)cc1 c1(C(N2CC(OC)C(NC(=O)C(c3cnccc3C)C)C2)=O)ccc(F)c(Cl)c1 C(CCCC(C)(C)C(=O)NNC(=O)c1c[nH]nc1Br)NC(C(C)=C(C)C)=O N1(C(c2n(CC=C)ccc2)=O)CCC2CCN(C(c3c(C)nn(C)c3C)=O)CC12 N1(C(CS(CC)=O)=O)CCC(C(=O)N(CC(O)COC)C)C1(C)C c1(CC(=O)NCCn2ncc(C(=O)NC3CC(C)OC3)c2)ncccc1F c1(C(=O)NCC(CC=C)NC(c2ccsc2C(F)F)=O)cc2n(c1)CCC2 Cc1c(C(=O)OC2CCOC(C)(C)C2)[nH]c2cc(Cl)ccc12 N1(C(CCc2ccc(C)o2)=O)CC(C)CN(C(=O)Cc2nc(C)sc2C)CC1C N1(C(=O)CSC2CC2)CCOC2CCN(C(=O)C(c3ccc(Cl)cc3)(F)F)CC12 C1(NC(Cc2ccc(OC)cc2)=O)CCN(C(C2CCCCN2N=O)=O)C12CC2 c1(COC)nc(=NC2CS(=O)(=O)CC2NC(c2c(Cl)ccc3c[nH]nc23)=O)s[nH]1 c1(C(=O)NC2CC3CC(C2)N(C(=O)C=CBr)C3)ccc2ncc(=O)[nH]c2c1 c1(C(N(CCC(C)NC(C2(O)CCC2)=O)C)=O)ccc2nc(O)cn2c1 C(=O)(C(C(C)C)n1cccc1)NC1(CCNC(C2(C)CC(=C)C2)=O)CC1 C1(CC(=O)NCCOC(CC)(C)C)CCCCC1NC(=O)C(N)=O CN1CC(C(=O)N(CC(N2CCOC(C3CCC3)C2)=O)C)CCC1=O C1(CC(=O)NC(C)CCN(C(=O)CC(C)F)C)(CC)CCOCC1 c1(C(N2CC3C(CNC(Cc4cc(C)on4)=O)(C3)C2)=O)ccc(Cl)c(F)c1 C1(NC(CNC(CCCCC)=O)=O)CCCCN(C(c2cccc(CO)c2)=O)C1 N1(CCC(=O)NCC2N(C(C(CCC)C#N)=O)CC=C2)C(=O)NC(C)(C)C1=O C1(CNC(=O)C(O)C2CC2)CCC2(CCN(C(=O)Cc3ccc(F)nc3)CC2)C1 c1(C(N2C3C(NC(c4c(C)cns4)=O)CC(C3)C2)=O)cnn2cccc(Cl)c12 C1(C(C)NC(C2CC(CN(C)C)C2)=O)CCN(C(=O)C(O)Cc2ccccc2)C1 N1(C(c2c(C)cc(F)s2)=O)CCC2(CC1)CC2C(=O)NCCCCN(C)C1CC1 C1(CNC(C(C)O)=O)CN(C(c2ncc(OCC3CC3)cc2F)=O)CC(C)(C)O1 N1(C(=O)C2CC2)CCCC2(CC2)C1.Cn1ncc2c1NC(=O)CC(=O)NC2 N1(C(c2ccc(C)nc2O)=O)CCC2(CC1)CN(C(=O)C(C)C#N)CC2C(=O)O Cc1cccc(NC(C2CN(C(c3cccc(CO)c3)=O)CCO2)=O)c1I C(CC(C(=O)NC(C)C(=O)NCCOC)NC(c1ccoc1C)=O)OC c1(C(N(CCN(C(Cc2cc(C)c(CO)cc2)=O)C)C)=O)cc(C#N)ccc1F C(C(=O)NCC(C)(C(C)C)NC(=O)Cn1ccnn1)(C(C)C)OCC N1(Cc2nnc(CC)o2)CC2CCCN(C(=O)C(C)OCCOCC)C2C1 c1(C(=O)NC2(CCOC)CCN(C(C(C(C)C)OC)=O)C2)cc2ccccc2[nH]1 C(=O)(C1SCCc2ccccc21)N1C(CNC(CCSCCC)=O)CC2(CC2)C1 C(=O)(N1C(=O)CN(CC(F)(F)F)c2ccccc21)CC1C(C(=O)OC)C1 CCCCC(F)(F)C(=O)N1CCC(N(C)C(c2ccc(CSC)o2)=O)C(C)C1 C(=O)(CCCC(C)(C)CC)NC1CCCN(C(C(c2ccccc2)OC)=O)C1 C12(C(=O)NCC3CCN(C(c4ccns4)=O)CC3)CCCC1OCC2 CC(C)C#CC(=O)NCC(C1CC1)NC(=O)CCCOc1ccccc1Br C#Cc1ccc(C(=O)NC2(CC=C)CCN(C(c3coc(C(F)F)c3)=O)C2)nc1 N1(C(CC(c2ccc(OC)cc2)C)=O)CCC(C)(C)C(NC(c2ccco2)=O)C1 c1(C(=O)NC(C2CCOC2)CNC(CC2CC(=C)C2)=O)cc(C(=O)OC)n(C)c1 N1(C(C2C(C(C)(C)C)CCCN2)=O)CCC2C(=O)OCC12C c1(OCC)cccc(NC(=O)C(C2(C)CC2)NC(=O)CC2CCCC(C)O2)c1 C1(C(N2CCCCC(NC(=O)C(O)CC(F)(F)F)C2)=O)CC2(CCOCC2)CO1 N(C1CCCc2occc21)C(C1(NC(c2ncc(C)c(C)c2)=O)CCN(C)C1)=O CN1CC(O)CC1C(=O)NCCCCCCN(C)C(C1CC2CCC2C1)=O C1(C)(OC)CCN(C(C2(C)CCCN2C(=O)CCc2ccccc2)=O)CC1 C1(NC(C(C)N(C(C2(CC=C)CCOC2)=O)CCC)=O)CC(=O)N(CC)C1 CC1=C(C(=O)N2CC3CC2C3NC(c2coc(C)n2)=O)CCCO1 c1(C(N2C3(CNC(CC4C(C)CCC4)=O)CC(C2)C3)=O)cc(N)cc(O)c1 c1(CNC(=O)NCC2(C)CCOCC2)ccc2c(c1)CC(=O)N2 C(C)(CN=c1ccc(S(=O)(=O)NC2CC(CC#N)C2)c[nH]1)c1c(C)cccc1 Cc1ccccc1C=CC(N1CCN(C(c2cccn2C)=O)C(C)C1)=O C#CCC(CC(=O)NCCCO)NC(=O)CCCCC=C c1(CC)cc(CC)cc(F)c1.C12CCOCCN1C(=O)C(=O)N1CCC2CC1 C1(C)(CC)CCN(C(C2(CNC(c3cnc(C)cn3)=O)CC=CC2)=O)CC1 c1(-c2cn(CC(=O)NC(C(=O)NC)Cc3ccccc3)nn2)cc(F)ncc1F c1(C(=O)NC2CN(C(C3(C(N)=O)CCC3)=O)C2)cc2nn[nH]c2cc1F C1(NC(C(C)(C)SC)=O)CCN(C(c2ccc(-c3ccc(F)cn3)o2)=O)CC1F c1(C(N2CCC(CSC)CC2)C(=O)NCCCCCC)ccc(C2CC2)cc1 C#CC1(C(=O)N2CC=CCO2)CCN(C(=O)CSC(F)F)CC1 CC(C)(CN=c1[nH]c(Cl)nc2[nH]cnc12)N1CCN(CCO)CC1 n1(CC(N)=O)cc(C(N2CC(CO)(NC(c3coc(Br)c3)=O)C2)=O)nn1 C1(C(=O)NC(C)CS(N)(=O)=O)(CC)CCN(C(=O)C(O)C(C)C)CC1 C(C1Cc2ccccc21)NCC(=O)Nc1ncc(C#C)cn1 c1(NC(C(CC2CC2)NC(C2CN(OC)C(=O)C2)=O)=O)cccc2c1CCC2 c1(C(N2C3CN(Cc4ccc(CO)cc4)CC23)=O)cc(F)c(Br)c(F)c1 C1(CC)CN(C(c2cn(C)cn2)=O)CCN1C(c1[nH]cnc1-c1cccnc1)=O n1(CC(=O)NC2C(CNC(CN(CCCCCC)C)=O)CCC2)ccccc1=O C1(C)(C(=O)NCCN(C2CCCC2)C(c2ccc(SC)o2)=O)CC2CC2C1 Cc1ccc(F)cc1C(=O)NC1CC(NC(C2CCC3CC23)=O)CC1O c1(C(=O)NCC2CCCN(C(CCCCC)=O)C2)cnn2c(Cl)cccc12 C1(C)(C(=O)NC(c2nc(C(=O)NC3CN4CCC3CC4)co2)C)CCCN(C)C1 c1(OC)ccc(O)c(C(=O)CNC(=O)CN(c2ccco2)C)c1 N1(C(C(C)=C(C)C)=O)CCC2(C1)CN(C(C1CC3(C1)CC3(F)F)=O)C2 C1(OC)CC2CC(C(N3CCN(CCN(C)C(C4(C)CCCC4)=O)CC3)=O)CC12 c1(C(N2C(C)C(NC(=O)CSC3CC3)CC2)=O)cnn2c1S(=O)(=O)NCC2 O=S(=O)(c1c[nH]ccc1=NCC1CCC12CCOCC2)NCCc1nncs1 N1(CC(=O)NC2C(CNC(CCS(C)=O)=O)COC2)C(=O)CC(C)(C)C1=O N1(C(c2ncc(CC)s2)=O)CC2CC1CN2Cc1c(C)nn(CC)c1C C1(NC(c2cc(CF)on2)=O)CC2(CCCCN2C(=O)CCC[N+](=O)[O-])C1 Cc1ccc(F)c(C(=O)NC(C2CCCN2C(=O)CCCc2sccc2C)C)c1 O=C(CCCC(F)(F)F)NCC(O)CNC(C1(CF)CCOCC1)=O c1(CNC=O)c(F)ccc(N)c1F.C1(COCCN(C)C2CC2)CC1(C)C(F)(F)F C(C)(C)(CC(=O)NCC1CC(O)CN1C(=O)C(F)CC1CCC1)N(C)C c1(NC(C2CCN(C(CC(C=C)CC)=O)C2)=O)ccc2ccccc2c1 C(=O)(CS(N)(=O)=O)N(C(C)C)CCNC(=O)CCN(C)Cc1ccccc1 c1(OC)cccc(C2CC2)c1F.c12ccc(s1)CNC(=O)NCC(=O)CCC2 C(C1C(C(=O)NCCCN(C(=O)CNS(=O)(=O)CCCC)C2CC2)C1(C)C)=C(C)C Cc1ncc(C(N2CCCC2(C(=O)NC2(C)CCSC2)C(C)C)=O)cn1 c1(C(C(=O)NC(C)CCNC(=O)COCC(C)(C)C)(F)F)nc2ccccc2s1 CC1(C)C(CNC(c2ccncc2)=O)CCN1C(C1COCCO1)=O Cc1ccc(C(=O)NCC2(NC(=O)CSC(C)C)CCCC2)c(=O)n1C CC1CCn2cc(C(N3CC(c4nnc5ccccn45)C3)=O)nc2C1 c1(CNC(C)=O)cccc(CN(C(=O)CN2CCNC2=O)C)c1 CC(CS(C)(=O)=O)C(=O)N1CC2CCN(C(=O)CSc3ccccn3)C2C1 N1(C(C)=O)CC2CCCC2(C(=O)NC2CC(=C3CCC3)C2)C1 c1(C(=O)NCC(=O)NC(C)CC(C)NC(c2cnnn2C)=O)ccc([N+](=O)[O-])cc1 CC1CN(C(=O)C(c2ccc(F)cc2)=O)CC1NC(=O)CC1CCC(=O)N1 C1(CNC(C(CC)(C)CC)=O)CN(C(=O)CCCC2OCCO2)C2CCN1C2 CCC(C(=O)NCC1CC1NC(c1sccc1CN(C)C)=O)c1ccccc1 CC1(C)CCN(C(C2CCCC2NCc2ccc(N3CCCCC3)cn2)=O)CC1 C1(F)(CNC(CC(C)OC)=O)CCC(CNC(=O)Cn2nccn2)C1 C1(NC(CCCC#CC)=O)COC2CN(C(C3C=CCCC3)=O)CC12 CCC(O)C(F)(F)C(=O)NCC1CN(C(c2ncccc2Cl)=O)CC1(F)F C1(CC=C)(C(=O)NC(c2csnn2)C)CN(C(=O)CCC2CC2(C)C)C1 C1(CN(C)C(c2cc(Cl)cnn2)=O)COCCN1C(c1sccc1-n1ccnn1)=O N1(C(C(C)CC2CCC2)=O)CCC(C(C)(O)CNC(C2(O)CCC2)=O)CC1 CC(C)CC(C)C(=O)NCC(C)(C)CNC(C1CSCN1C(=O)C(C)(C)C)=O C1(C)(CNC(C(n2cc(CO)nn2)C)=O)CCN(C(=O)C=C2CCOCC2)CC1 C1(CC(=O)NC(CCC)(C)CC)C2CCC(C2)N1C(=O)C=C=C(C)C CN=c1cc(C(=O)NCCCC(C)NC(=O)CCCc2ccsc2)cc[nH]1 c1(C(N2CCN(C(C(CC(=C)C)C)=O)C(C(F)F)C2)=O)cc(C)c2c(c1)CCC2 c1(CC(N2CCC(NC(C3CC4(CSC4)C3)=O)C2)=O)ccc2ccccc2c1 C1(CNC(c2nc(C)n(C)c2C)=O)CN(C(=O)C(C)O)C2(CCC2)C1 CC1CCC=C1C(=O)N(C1CCCC1)CCCNC(=O)COC1CC(F)(F)C1 CC(C)(CNC(=O)CC1C(NC(=O)Cc2cc[nH]n2)CC1O)CC(F)F C1(C(=O)NCCCCNC(c2occ(C)c2)=O)CSC(c2ccccc2)=N1 C1(CNC(=O)NC2(CC(N)=O)CCOC2)CCCOC1C1CC1 c1(C(N(CCOC)CCNC(=O)C(C)OC(C)(C)C)=O)cc(C(F)(F)F)n(C)n1 C1(CNC(C2(CCCC)CCC2)=O)CN(C(=O)Cc2cc(C)no2)CC12CC2 c1(C(C(=O)NCC(C)C)N(CC(=O)OCC)C)cc2ccccc2o1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC1OCCN(C(c2ccoc2)=O)C1 c1(C(c2nnnn2C2CCC2)NC(C(c2cccc(F)c2)C)=O)ncc(F)cc1F N1(C(C(CC=C)NC(CCCC=C)=O)=O)CCSC(C)CC1 C1(NC(c2[nH]cc(CC)c2)=O)CCN(C(c2cnncc2O)=O)C12CCC2 C1(CC)CN(C(=O)C#CC2CC2)CCC1NC(c1cc(-c2cnn(C)c2)[nH]n1)=O CCCCC(C(=O)NCCN1CCCC1=O)N1CCC(C)(CC)CC1 Cc1coc(C=CC(=O)N(CCNC(=O)CCC2CC2)CC2CC2)n1 N1(C(c2n(C)cc(F)c2)=O)CCC2(CC2C(=O)Nc2nccc(C(F)F)c2F)C1 CC1CN(C(c2ccc(N)c(O)c2)=O)CCC1CNC(=O)CCNC(N)=O C1(O)(CNC(C(C)n2cnnn2)=O)CCN(C(=O)CC(C)NC(N)=O)CC1 C1(NC(=O)CC2CC3CC3C2)CCC2CC1CN2C(C12CCCC1C2(F)F)=O c1(C(N(CC(C)NC(=O)Nc2ccc[nH]2)CC)=O)cccc(OC(C)C)c1 N1(C(CCCCCC)=O)CCCCC1C1CCCN1c1cc(O)ncn1 N1(C(c2ccc(F)s2)=O)CCOC2CN(C(=O)C(F)(F)C3CC3)CC12 C12(CC(=O)NC3C(OC)CN(C(=O)CN(C4CCSC4)C)C3)CCC(CC1)CC2 C1(COC)CN(C(c2coc(Br)c2)=O)CCN1C(=O)CCS(N)(=O)=O c1(OCCCC#N)ccc(CN2CCC3(CCC3)C2)cc1C(N)=O C(=O)(CCC(=O)NCC1CC(NC(=O)Cc2cc(Cl)n(C)n2)C(O)C1)NCCC c1(OC23CN(C2)C(=O)NC3)cn(C)cc1C(F)(F)F.C1(C(F)(F)F)(COC)CC1 N1(Cc2c(C)nn(C)c2)CCCC(NC(c2ccc(F)cc2Cl)=O)CC1 Cc1ccc(Cl)c(C(C(=O)NC2COC2)N(C)CC2CC2)c1 N1(S(CCC)(=O)=O)CCC(NC(c2cc(Br)cs2)=O)C(C)CC1 CC1CCN(C(C2CCSC2)=O)CC1NC(C1CC2CCC(C1)O2)=O C1(NC(c2cc(C(=O)OCC)n[nH]2)=O)CCCC(NC(C2CNC(=O)N2C)=O)C1 c1(C(=O)NC2CC(C(C(=O)N(C3CCCCC3)CC)F)C2)nnc(O)nc1O C12(C(N3CC(CNC(C4CCSCC4)=O)OCC3)=O)CCC(F)(CC1)C2 c1(OC(C)C)cccc(C(=O)N(C(CNC(=O)CCCC(C)C)C2CC2)C)c1Cl N1(C(CC(C)F)=O)CCC(C2(O)CN(C(=O)CC(C(F)F)C(C)(C)C)C2)CC1 CC1(OCC(=O)NCC(C2CCC2)NC(C2CC2C(F)(F)F)=O)CCOCC1 CC(N=c1cc[nH]cc1[N+](=O)[O-])C1CN(C(=O)CCCN(C)C)CCO1 C1(C(=O)NCCCCC(C)NC(CCC(=C)C)=O)CN2CCCC2CO1 C1(CNC(CC(CN(C)C)O)=O)CC(C(=O)NCC(F)(F)C(N)=O)=NO1 C1(CNC(CN(CCOC)C)=O)CC(F)(F)CN1C(c1cc(SC)ccc1C)=O CCC(CC)(CCNC(C1CC(C(C)C)=NO1)=O)NC(C1C2CCN1CC2)=O C1(NC(=O)CC2(NC(=O)CCn3ccnn3)CCC2)Cc2ccccc2C1 N1(C(CN(C)CC)=O)CCCC(C2CCN(C(c3cccc4sccc34)=O)C2)C1 Cc1c(C(=O)N(C(C)CNC(C2OCCC2(C)C)=O)C)csc1Br CCN=c1[nH]c(C(=O)NC2CN(C(=O)CC=C(Cl)Cl)C(C)(C)C2)cs1 c1(CC)noc(COCC(=O)N(CCC(C)NC(C2(Cl)CC2(C)C)=O)C)n1 c1(SCC)nc(C)c(C2CCCCC2NC(C2CC(=O)NC(=O)N2)=O)c(C)n1 c1(NC(CCNC(=O)NC)=O)ccc(F)cc1F.C12(C)CN(C1)C2=O c1(CC)nocc1C(N1CC(C(C)NC(c2cc(CO)[nH]n2)=O)C1)=O C1(C(=O)OC)(CN2CCC23CNC3)CCCOC1 N1(C(C(C(C)C)SCC)=O)CC(CNC(=O)Cc2nonc2C)C2(CC2)C1 c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(C)SC(C)C)C2)cnc1O CC1CCc2c(C(=O)NC3(C)CCC(NC(=O)Cc4ccoc4)CC3)csc2C1 c1(C(=O)NC2CN(C(=O)CNC(=O)C3CC3)CC2F)ccc(Br)c(Cl)c1F c1(C(C)NC(C(c2nccc(C)n2)C#N)=O)ccc2c(c1)c(C)c(C)n2C N1(Cc2ccc(C)nc2)CCC2(CC1)CC(CC(=O)Nc1nc(F)ccc1O)C2 C1(NC(c2c(CC(C)(C)C)cccc2)=O)CC2CC1N(C(c1cncs1)=O)C2 C=C(Cl)CC(C(=O)NCCOC1CC1)NC(c1cnn(C)n1)=O c1(C(=O)NC2CCN(C(C(C)OCC#C)=O)CC2C)nc(O)c(C#N)cc1C c1(C(N(CC(C)O)CCNC(C(CC)NC(N)=O)=O)=O)cnn2c1NCCC2 C1(NC(C2(C(N)=O)CCC2)=O)Cc2ccccc2C1NC(C1CCC(F)C1)=O c1(C(C(=O)NCC2CC2Cl)N(C)CC2CC2)ccc(C(C)(C)C#N)cc1 N1(C(c2nc(CC)[nH]n2)=O)CCCC12CCN(C(=O)C(F)C(C)C(F)(F)F)CC2 N1(c2cc(C(N)=O)nc(Cl)n2)CC2(CCC(NC(=O)C(F)C(F)(F)F)CC2)C1 N1(C(c2cc(C)c(O)nn2)=O)CCCCNC(=O)C(F)(F)C1 C1(C)(CNC(c2cc(COC)sc2)=O)CCCN1C(c1c[nH]nc1C)=O c1(CN(C(c2csnc2C)C(=O)NCC)C)cccnc1OC Cc1nn(CC(=O)NC2COCC2NC(C2CCC(C)(C)O2)=O)c(=O)n1C C1(OC)CC(C(N)=O)N(C(=O)C=CC2CCC2)C1.c12cn(C)nc1CNC2=O c1(OC)ccc(F)c(C(N2CCN(C(=O)Cn3cnnc3O)C(CO)C2)=O)c1N c1(C(=O)NC2C=CCN(C(C3CCN(C)C3=O)=O)C2)c[nH]c2nccc-2c1 C#CCCC(C(=O)NC(C)C=C)NC(C1(O)CCSCC1)=O CCCCC(CC)C(=O)NC1(CO)CCN(C(c2nc(Cl)c(Cl)s2)=O)C1 c12cc(on1)CNC2=O.c1(C(N2CC(N3CCCC3)C2)=O)ccco1 N1(C(C(CC)OC)=O)CCN(C(c2cccc(C#N)c2)=O)CC1C1CCCC1.C1CC1 c1(C(N2CC3C(NC(c4cnc(Cl)[nH]4)=O)(C3)C2)=O)cc2c(Cl)nccc2o1 N1(C(c2c(C)cc(C)cc2F)=O)CC2(CCCCN2C(=O)CC2CCCCC2)C1 c1(CNC2CCC(NC(c3ccc(OC)c(I)c3)=O)C2)ccc(Br)cc1[N+](=O)[O-] Cc1c(C(=O)NCCCCNC(C2(C)CCC(C)(C)CC2)=O)nn2ccccc12 Cc1ccc(F)c(-c2cn(CC(C)NC(=O)C(C)(C)CC3CC3)nn2)n1 C(=O)(C1=CS(=O)CCC1)NCC(C)(C1CCC1)NC(CCN1CCC(C)CC1)=O c1(NC(c2cnc(SC)nc2)c2n(CC=C)nnn2)ccnc(OC)c1 Cc1cnc(C(=O)NCC2CCCCC2NC(=O)C=Cc2sccc2C)c(F)c1 N1(C(c2ccnc(C)n2)=O)C2CCC1CC(N(C)C(c1cnoc1C)=O)C2 CC1CC2CN(C(=O)CC(C)(C)F)CC2N1C(c1cccc2ccncc12)=O C1(CNC(C2(SC)CC2)=O)CN(C(C2CC3(CCC3)C2)=O)C2CCCCC12 Cc1cc[nH]c1C(N1CCC(N(C)C(c2csc(CS(C)(=O)=O)n2)=O)C1)=O C=CC1COCCN1C(C1CC(F)CN1C(c1ncccc1N)=O)=O N1(C(C(C)OC)=O)CCC(NC(=O)CCn2nc(C)nc2C)C(OC)C1 C1(C(N2CCC(NC(C3CC3[N+](=O)[O-])=O)C(O)C2)=O)C2CCCCCCC12 CCCCCCCCN(C(=O)C(C)(C)NC(=O)COC(CC)CC)C Cc1c(CNC(c2nc(CC3CC3)nn2C)=O)noc1-c1ccc(Cl)cc1 c1(C(=O)NCCC=C)cc2ccc(-c3cc(C)cnc3OCC)cc2o1 C1(NC(c2cnc(C)s2)=O)CC12CCN(C(c1c(F)cncc1F)=O)C2 C(=O)(C(CNC(C1CC1Cl)=O)N(C)C)NCCCOC C(=O)(N=c1ccn(C(F)F)[nH]1)c1ccc(CNC(C2C(C)(C(C)C)C2)=O)s1 C1(CC(=O)NCC(C)(C2CC2)NC(c2cnc(C3CC3)o2)=O)CCCOC1 c1(CC)ncncc1C(=O)NC1CC2(C1)CC2C(=O)NCc1cc(C(N)=O)co1 N#Cc1cccc([N+](=O)[O-])c1N1CCC2C(NC(=O)CSS(C)(=O)=O)CC12 N1(C(CCC(C)NC(c2cc(=O)n(C)cn2)=O)=O)CC2CC1C(F)(F)C2 C(=O)(C(F)(F)C(C)O)NCc1ccc(CC(=O)NC)cc1.C12(CCCC1)SC2 c1(C(N2CCCC(F)(CNC(C(CO)N(C)C)=O)C2)=O)cc2ncccc2s1 c1(C(N(C)CCN(C)C(C2OCCCO2)=O)=O)n[nH]c2c1COc1ccccc1-2 C1(NC(C(CC)NC(C)=O)=O)CC(F)(F)CC1NC(=O)C=Cc1cccc(Cl)c1 C(C(=O)N1CCC(N(C(=O)CC2CCC2(C)C)C)CC1)(C(C)C)NC(=O)OC c1(C(=O)NC2(C)CC(NC(C=CC)=O)C2)ccc(C(C)(F)F)nc1 c1(C(N2CCC(C(C)NC(c3ccc(O)nc3)=O)C2)=O)ccc(O)nc1Cl C#CCC(C)(C)C(=O)N1CCCC1CNC(=O)C(c1cccc(C(F)(F)F)c1)O C(C(C)(O)CC(=O)NCCCN(C(C1C(C(=O)OC)C1(C)C)=O)C1CC1)OC c1(CC)cc(N)ccc1C(=O)NCC(C)(CC(C)C)NC(=O)CCc1cccs1 c1(-c2cn(C3CCC(C(N4C(C#N)CCC4)=O)CO3)nn2)nc(Br)ccc1F C1(O)(C(=O)NC2CN(C(CC3C(C)(C)CCO3)=O)C2)Cc2ccccc2C1 CC(C)C(C(=O)N1CCC(NC(c2ccc(OCCF)cc2)=O)C1)n1ccnc1 C1(C(=O)NCCC2CC(C)N(C(=O)CCOC3CC3)CC2)CCC2(CCC2)CC1 c1(C(=O)N)ccc2nccnc2n1.C(=O)(CC(=O)OC)N(CCC)CCC C(CCCCC(=O)NC1(CNC(C2(C)CCCC2C)=O)CCCC1)=CC c1(NC(C(C)C)CNC(c2cc(C(C)(C)C)no2)=O)cc(=O)n2ccccc2n1 c1(SC)ccc(CC(=O)NC2CC(C)(NC(c3ccc(C(C)=O)o3)=O)C2)cc1 C(=O)(CCC(C(C)C)NC(C1C2CC(=O)CC12)=O)N1CC(C#C)C(O)C1 C(=O)(C(F)C(C)CNC(=O)C(C)(C)c1ccno1)NCc1nc(C(C)C)on1 C(=O)(C1=CCC(NC(c2cc(C)nn2C)=O)C1)NCC1(CC)CCCO1 c1(C(N2CCC(O)(CCNC(C(CCC)(C)C)=O)C2)=O)cccc2occc12 c1(C(=O)OCC)cc(Br)ccc1N(C)Cc1sc(C)cc1C c1(NCCNC(c2c(C)cccc2)=O)cc(Cl)nc(-c2ccccc2)n1 C1(NC(CC)=O)(CNC(c2cc(C)[nH]n2)=O)CC2CCC1C2 C(C(C)C(C)(C)C)N(C(C(CSCC)NC(c1cnsn1)=O)=O)C C1(C(=O)NC(CNC(CC(=O)NCC)=O)(C)C2CCC2)CCC2CC1C2(C)C N(C(=NCCCF)NCC1(C2CC2)CC1)Cc1c(OC)nccc1 c1(OC)cccc(C(C)NC(=O)CO)c1.c1(C(=O)O)cc(CN)co1 CC(CC(=O)N1CCC(C)(NC(c2ccc3c(c2)CC3)=O)C1)CC(C)(C)C c1(C(C(=O)NCCN(C(c2c(CC)csc2)=O)CCOC)C)cccc(Cl)c1 CC(C)(CC(=O)NCC1CCCC(CNC(=O)CCCC2CCC2)C1)CC(F)F C(C)(CN=c1[nH]nco1)(C(C)C)NC(C=Cc1ccc(OC)cc1)=O N1(C(C2(CCC)CC2)=O)CCCC(CNC(=O)C(C(C)(C)C)C2CCCC2)CC1 c1(C(N2CC(C=C)OCC2)C(=O)NC2CCCC2)cccn2ccnc12 N1(C(c2n(CC#C)cnn2)=O)CCC(=C)CC1C(=O)NC(c1nncn1C)C O=C(C#CC1CCCCC1)NC(C(=O)NCC1CCC(=O)O1)C1CCCO1 C1(C(=O)NCCC2CC(NC(c3ncn(CC)c3)=O)C2)(CC)CC=CCC1 C1(OC)CC(C(N2CC(NC(c3cc(CO)n(C)n3)=O)C(CO)C2)=O)CC1OC N1(C(C(C)=CCSc2ccc(C)cc2O)=O)CC2CC(C1)N2C(=O)OC(C)(C)C C(=O)(C(C)(C)C(F)c1ccccc1)N1CCC(C(C)NC(C(CC)CC)=O)C1 C1(NC(C(C=C)O)=O)CN(C(=O)CCCOc2ccc(C(C)(C)C)cc2)CC1C C1(C(=O)NC2CC(CO)N(C(=O)COC3CCOC3)C2)C2CCCCC12 c1(NC(C2C(OC)CN(C(C3CN4CCC3CC4)=O)C2)=O)cc(C)cc(O)c1 c1(CC(C)N(C)C)ccccc1F.C12COCCN1C(=O)Cn1cc2nn1 c1(C(N2C(C)CC(CNC(=O)C#CC3CC3)C2)=O)ncc2ccccc2c1O N1(C(C(C)C(=O)N2CCOCC2)=O)C2CCC1CN(C(C1(CF)CC1)=O)C2 c1(C(=O)NCCC(=C)CNC(c2ccnn2CCC)=O)cc(OC)ccn1 Cn1nc(C(N2CCn3nccc32)C(=O)NC2CCCC2)c(Br)c1Cl c1(CC(CN(C(C(C)=C(C)C)=O)C)NC(C2CC(C)(C)C2)=O)ccccc1 c1(CN=[N+]=[N-])ccc2c(c1)CN(S(=O)(=O)C1CCOC(C(F)(F)F)C1)CC2 Cc1nc(NC(C2C3(CC3)C23CC3)=O)c2cnn(-c3ccccc3)c2n1 N1(C(=O)C2=CCCCCC2)CCC2CCN(C(c3cccc(Cl)c3)=O)C2C1 c1(C(N2CCCN(C(C3=NOC(C)C3)=O)CC2C)=O)cc([N+](=O)[O-])cnc1N c1(CCNC(CCN(C(=O)CC(=O)NC2CC2)CC#C)=O)ccccc1 Cc1cc(C(N(c2nnc(CN3CCC(C(N)=O)CC3)s2)C(C)C)=O)cc(C)c1 c1(C(N2CC(F)CC2C(=O)OC)C(=O)NCCCC)cc(C)c(OC)c(C)c1 c1(C(=O)NC2CCCN(C(C3(C)CC(C)OCC3)=O)CC2)ccc2c(c1)CCC2 N1(CC(=O)N(CCn2cc(Cn3ccnc3)nn2)CC)CCOCC1=O C1(NC(c2n(C)cc(F)c2)=O)CCCN(Cc2ccc(Cl)cc2Br)CC1 CCCCC(CNCc1cnc(-c2cccc(C#N)c2)s1)CC C1(C(C)NC(=O)C=CI)CCCCN1C(c1cccc(F)c1)=O C(=O)(CCCCC#N)N1CCC(C(=O)NOCC(F)F)(CC=C)C1 c1(C(=O)NC(CC)(C)CNC(=O)C(C)(C)CC(C)C)cc2cccc(Cl)c2o1 C(C)(CC(=O)NCCCCN(C)C(c1cn(C(F)(F)F)cn1)=O)SC C1(NC(C(C)Oc2cccc(C)c2)=O)CN(C(c2ncn(C)n2)=O)C(C)(C)C1 CC(C)C(F)C(=O)NC1CCC(CNC(c2ccccc2Br)=O)CC1 c1(OCC)cc(F)ccc1F.CC(O)C(=O)NCCOCCN(C(=O)CO)C c1(C(c2cnc(-c3noc(C4CCN(C)C(=O)C4)n3)cn2)OC)ccc(C)c(C)n1 C1(OCC)CC2(C1)CC2NC(=O)C=CCOC(C(=O)Nc1ccccc1)C C1(NC(C2C(=C)C2)=O)CN(C(=O)Cn2ncnn2)CC12CCOCC2 c1(C(=O)NC2CCCC(NC(c3onc(C)c3C)=O)C2)c2c(c[nH]c1=N)CCC2 C(=O)(C(C(C)(C)C)C1CCCCCC1)NC1CN(C(C2(C)CCCSC2)=O)C1 N1(C(C(CC)C#N)=O)CCCC(NC(=O)C=Cc2csnc2C)CC1 CN1CCCCC1CC(N1CCC(O)(CCNC(=O)C(C)(C)c2cnc[nH]2)C1)=O C(=O)(CC1COc2ccccc21)N1CC2C(CNC(C3CCC3)=O)C2C1 c1(C(=O)NC2C(F)CCN(C(CC#C)=O)C2)ccc2occc2c1O CC1COCC(CC(=O)N(CC(CO)(CO)NC(=O)COCc2nc[nH]n2)C)O1 N1(C(C)=O)CSCC1C(=O)N(C1CCCCC1)CCCN(C)C(C)C.C1(=O)CN1 C#CC1(NC(=O)NCCC2(C)CCCO2)CCN(C(=O)OC(C)(C)C)C1 C12(NC(CCCOCC)=O)CC1CN(C(C1COCCN1C)=O)C2 C(=O)(C(C(C)(C)C)NS(C)(=O)=O)N1CC(CCNC(c2c(C)cco2)=O)OCC1 N1(C(C2C(CC)C2)=O)CC2CC1CCC2NC(=O)CC1COCC(C)(C)O1 n1(CC(=O)NCC2(CCC=C)CN(C(CSCCCC)=O)C2)ccccc1=O N1(C(C(C)CC(C)(C)C)=O)C2CCCC1CN(C(=O)C(N1CCCCCC1)C)C2 N1(C(C(OC)OC)=O)CCN(C(=O)C(c2cncn2C)O)CC1c1ccncc1 CCCC(C(=O)N(CC(CC)OC)C)NC(=O)CC1C(CC)C1(F)F C(=O)(C1=CCCCC1)N1CCCC(C(C)NC(c2nc(Cl)c(Cl)s2)=O)C1 Cc1ccc(N)c(C(=O)N(CCCNC(=O)C(C)C)Cc2cccnc2)c1F C(=O)(CCC(=O)NC1CCCCC1CNC(C1CN(C(C)C)CCO1)=O)NC C1(NCc2c(CC)cccc2)CN(C(C2CCS(=O)(=O)C2)=O)CCC1F C(=O)(C(=O)N=S(C)(C)=O)NC1(C)CCN(C(C(CC(C)C)O)=O)C1 c1(C(N2CC3C(NC(c4ccnc(C5CC5)c4)=O)C3C2)=O)ccc(F)c(O)c1 C(=O)(C1=CCS(=O)(=O)C1)N(C(C)CNC(=O)C(c1ccccc1C(F)(F)F)O)C C1(C(N2CC(CNC(c3ccc(C(C)C)cn3)=O)C2)=O)CCC(C#N)CC1 C1(CNC(CSS(C)(=O)=O)=O)CC2(CCOCC2)CN1C(C1NC(=O)NC1=O)=O C1(C(N(C)Cc2scc(C)n2)=O)N(C(c2ncncc2C)=O)CCCC1(C)C CC1CC(CC(=O)NC(C)CC(C)(C)C)CN1C(C1CC1c1cccnc1)=O c1(C(N2CCC3(C2)CN(C(c2cc(O)no2)=O)C3)=O)cn2ncccc2n1 C(CC(=O)N1CC(CNC(=O)C(C2CC2)SC)C1)NC(=O)OC N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC2CCC1CN2C(C1CC1(C)Br)=O c1(-c2onc(C)n2)ccc(C(=O)NCC(CO)NC(=O)COC(F)F)cc1 c1(C(N(CCCNC(C=CC(CC)C)=O)CC2CCCC2)=O)ncn(C(C)C)n1 CCC(C(O)C(C)C)NC(C1C2CC3C(C2NC(=O)CCc2ccnn2C)C13)=O c1(C(C)(CO)NC(=O)CC2CC3CCC2O3)ccccc1Cl C1(NC(CN(C)S(N)(=O)=O)=O)CN(C(c2cc(N)cnc2Cl)=O)CCC1O C(=O)(C1=CCN(C(C2CC3C=CC2O3)=O)CC1)N(C1CSC1)C c1(NC2CC=C(C)CC2)ccc(S(=O)(=O)N2CCc3ccccc3CC2)cc1Br C1(CNC(=O)CNC(c2c(C)occ2)=O)CCCCCN1C(C1CC(O)C1)=O N1(C(=O)Cc2c(Cl)cccc2Cl)CC2CCCC(C1)N2C(=O)C(F)Br N1(C(Cc2cc(C)c(Cl)cc2)=O)CC(CNC(=O)C2=NNC(=O)C2)C2(CCC2)C1 C1(C(N(CC(C)NC(C2CC(=C)C2)=O)CC)=O)CC(c2ccccc2)=NO1 C1(C(COC(C2N(CC)C(=O)CC2)=O)=O)(OC)CCCC(C)(C)C1 N1(C(c2c(CC)n(C)nc2)=O)CC2(CCC2NC(=O)C(Br)=C(C)C)C1 C1(CNC(c2c(C)nc(CCC)s2)=O)CC(NC(=O)CCC(F)(F)F)C12CCC2 C(c1ccco1)=C(C)C(=O)NC1(CCC(=O)NC(CO)C2CCC2)CCCC1 N1(C(Cn2nc(C)oc2=O)=O)CC2CCC1CN2C(=O)CCNS(C)(=O)=O N1(C(C(=O)NCC2CCN(C(c3c(C(C)C)n[nH]c3)=O)C2)C)CCP(C)(=O)CC1 N1(C(C2(C)CCCNS2(=O)=O)=O)CC(NC(c2cocn2)=O)C2(CCOCC2)C1 N1(C(CN2C(C)CC2)=O)CCCOC(CCNC(=O)CN2C(=O)CNC2=O)C1 CC(C1CC1)=C(F)C(=O)N(C)CCN(C(C1CC1CC(C)(C)C)=O)C(C)C N1(C(C(=O)C2CC2)=O)CC2(CCCN2C(=O)CCN2C(=O)C=CC2=O)C1 c1(C(=O)NC(C2CCN(C(C3CN(c4nnnn4C)C3)=O)C2)C)ccncc1F c1(C(=O)NCC2CC(CNC(=O)CC3CSCCS3)OC2)ccc2cnccc2c1 c1(C(N2CC(C)OCC2)=O)ccc(-c2ccccc2C#N)c2c1OCO2 C(C(C)NC(=O)C=CCN(C)C)N(C(C1CC1CC(C)C)=O)CC n1(CC)nc(C)cc1C(N1CCOCC1CCNC(C1(CF)CC(F)(F)C1)=O)=O CC12OCC(COC(=O)C(F)(F)Oc3ccc(F)c(Cl)c3)(CO1)CO2 c1(C(=O)NCC(C(C)(C)C)NC(C(C)(C)OCC)=O)ccc(Br)c(N)n1 N1(C(c2c(C(C)(C)C)n[nH]c2)=O)CC2CCC2(CCNC(C2CC2[N+](=O)[O-])=O)C1 C1(NC(=O)Cc2ccsn2)CCC2(CCN(C(C3CC(F)(F)C3)=O)C2)C1 c1(C(=O)NCC2C3CN(C(c4cnn(C5CC5)c4)=O)CC23)cccc2[nH]ccc12 C1(F)(CNC(CN(C)CC)=O)CCC(NC(=O)CSc2cccc(C)c2)C1 Cc1cccc(CC(=O)NC(C)(CNC(c2c[nH]nc2C)=O)CO)c1Cl C(c1ccc(C)cc1)=CC(=O)NCCN(C(C=COCC)=O)CC C1(C(=O)NCc2cc(C(N(C)Cc3cccnn3)=O)on2)CN2CCN1CC2 N1(C(CC(CC)C2CC2)=O)CCC(NC(=O)CNC(c2cscn2)=O)C12CCC2 N1(C(C2(F)CCN(C(C3(C4CC4)CC3)=O)C2)=O)CC2CC3CC2C1C3 c1(NCC)ccc(C=CC(N2CC(NC(=O)COc3cccnc3Cl)C2)=O)cc1 c1(C(N(C2CN(C(=O)OC(C)(C)C)C2)C)=O)ccc2cc([N+](=O)[O-])ccc2n1 c1(C(N2C(CC#N)CN(C(c3sccc3Br)=O)CC2)=O)cc(F)cc([N+](=O)[O-])c1 C1(C(=O)NC2(CNC(C(CC)F)=O)CCCC2)CCCCC(=O)N1 c1(C(N2CCC(F)(CNC(C3CC(OC)C3)=O)C2)=O)n[nH]c2c1CC(C)CC2 CC(C)(CC(=O)NCC(C(F)(F)F)N1CCN(C(C2CSC2)=O)CC1)C1CC1 C1(CCNC(C2(F)C(C)C2)=O)CCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 c1(C(=O)NCC(CNC(C=CCCC)=O)F)cnc2ccc(Br)cn2c1=O c1(CNc2nc(C)nc(NC3CN(C)C4(CCC4)C3)c2)ccc2c(n1)NCCC2 c1(C(C(=O)N(CCOC)Cc2c(C)noc2C)(C)C)ccccc1C(F)(F)F Cc1ccc(C=CC(N2CC(NC(=O)C3=CCOCC3)C3CCCC23)=O)c(C)c1 C1(CC(=O)N(CCCNC(c2n(CCCC)ncc2)=O)C2CC2)COCC1(C)C N1(C(c2c(C)c[nH]n2)=O)CCC(C)(C)CC1C(=O)NC1CCOC2(CCC2)C1 C1(NC(Cc2ccc(C)nc2)=O)CCCC12CCN(C(=O)CSCC(N)=O)CC2 c1(CC)ccc(C(=O)NCCOCCCNC(C2CC3CCC2O3)=O)cc1 C1(C(N(C2CCN(C(c3cc(C)nn3CC)=O)C2)CCC)=O)CC12CCOCC2 C1(C(N2CC(N(C(C(C)CC3CC3)=O)C)C2)=O)CCN(c2cccc(Cl)c2)C1=O Cc1ccn2ncc(C(=O)NC(C)CCNC(C3(NC(N)=O)CCCC3)=O)c2c1 C12(CCCCC1)CC(=O)N2.N=c1[nH]cc(C(N2CCCC2CCN(C)C)=O)s1 C1(NC(C(N(C(Cc2scc(C)c2)=O)C)C2CC2)=O)CCCCCC1CO c1(C(=O)Oc2c(Br)ccc(C)c2)cc(F)cc2ccoc12 c1(C(N(CCN(C(=O)CC2CC23CC3)CC)CC)=O)ccc(C(=O)OC)nc1 n1(CC)c(C(N2CCC(CCOC)C2)=O)cnc1O.C12CC1C(=O)NC2 Cc1ncnc(C)c1C(=O)NC1CC(F)CN(C(=O)C(F)(F)c2cscn2)C1 N1(CC2C(C(C)C)C2)C(=O)CN(Cc2cc(Br)cnc2-n2cccn2)C1=O c1(OC)nccc(I)c1CN1C(C(=O)Nc2ccccc2SC)CC2CC12 C1(C(=O)NC2C3CC(NC(c4ccn(CC)c4C)=O)CC32)C2CCCCCC12 c1(C(=O)NC2(C(N3CCC(C#C)(O)C3)=O)CCN(C)C2)cc2cccnc2[nH]1 Cc1c(C(N2CC3CC2CN3C(=O)CCc2ccon2)=O)oc2ccc(Cl)cc12 Cn1ncc2cc(C(N3CC4CC4(CNC(=O)C(C)(C)C(F)F)C3)=O)ccc12 C1(C(=O)NCC2CCCC(NC(C3(CC)CCCCC3)=O)C2)COC(C)(C)CO1 C#Cc1ccc(C(=O)N(C2CCN(C(=O)C(C)=C3CC3)C2)C)c(F)c1 C1(CNC(c2cccc(OC)c2)=O)CC2CCCC2N1C(=O)CC(C)F C=C(C)CCC(=O)NCCCN1CCC(NC(=O)CC(C)(C)OC(C)=O)C1 N1(C(C2CCN(C(C)=O)C2)=O)CCN(C(=O)COCCN(C)C)C(CC2CC2)C1 C1(C(=O)NC(C)(C)CNC(c2cc3ccccc3o2)=O)CCc2ncccc2C1 C1(NC(C=C(CC)CC)=O)CCCC(CN(C(=O)CCc2ccc(Cl)cc2)C)C1 C(=O)(C(C)(C)C1=CCN(C(=O)C(=O)Nc2ccc(S(C)(=O)=O)c(C)c2)CC1)OC n1(CC(=O)N(CCCNC(C(N)=O)=O)C2CC2)cc(Br)c(O)nc1=O C(CNC(C1CC2C=CC1O2)=O)(CC(F)(F)F)NC(CC(C)(F)F)=O C=CCCCCCC(=O)N1CCN(C(=O)CC(O)COC)CC1N(C)C C1(N(C)C(C2CC2Nc2ccco2)=O)CCCN(C(=O)OC(C)(C)C)C1 N1(C(C(=O)NCC=C)C(C2COC2)NC(=O)OC(C)(C)C)CCOCC12CC2 C1(n2cc(C3N(CCn4cc(C(=O)O)nn4)CCC3)nn2)CCCCCC1 c1(C(=O)NCC2CCN(C(c3c(Cl)n[nH]c3C3CC3)=O)C2)cncc2nc[nH]c12 CCC(C)C(O)C(=O)NC1CC(C)(CNC(=O)C(F)(F)C=Cc2ccccc2)C1 CC1CCCCN(C(=O)C=CC(C)(C)NC(=O)CC2(O)CCC2)C1 N1(C(c2c(C)cccc2)=O)CC(C)N(C(=O)Cc2ccc(O)nc2)CC1C CCCC(CC(=O)N(C)Cc1nocc1C(C)C)NC(=O)C(C)(C)C(=O)NC Cc1cc(F)ccc1C(=O)NCCCCNC(C1COCC1c1ccccc1)=O CCCC(CC)CC(=O)N1CCCCC1C1CCCN(C(=O)CNC(=O)NC)C1 c1(NC(C2(CNC(C3C(C)C(=O)C3)=O)CCC2)=O)cccc(F)c1 N1(C(C(C(C)C)F)=O)CCN(C(c2cc(C3CCC3)on2)=O)CC1C1CCCC1 Cc1ccn(C)c1C(=O)N(CCNC(=O)C(C)CF)C c1(OC)ncccc1S(=O)(=O)NC(c1cc(C)ccc1F)(C)C C12(C(N(C(C(=O)NCC(Cl)Cl)C3CC3)C)=O)CCN(CC1)C2 N1(C(c2nc(-c3ccncc3)cs2)=O)CCc2c(F)ccc(O)c2C1 C(=O)(C(CCS(C)(=O)=O)OC(C)=O)NC1CCC(NC(CSCCCC)=O)CC1 N1(C(C(=O)NC(c2n[nH]c(-c3ccccc3)n2)C)=O)CCCC2(CCSC2)C1 C12(C(=O)NC(c3ccccc3)C(C)NC(=O)C(N)=O)CC(C1)C(C(F)(F)F)O2 N1(C(Cc2c(CC)con2)=O)CCCC2(NC(c3nccn3C)=O)CC2C1 C1(C(N2C(C(C)NC(CCSCCCC)=O)CCC2)=O)COCCN1C=O c1(OC(C)C)cc(-c2ccc(NC(c3c(F)ccc(Cl)c3F)=O)s2)cc(C#N)c1 CCC(CNC(c1cocc1C(N)=O)=O)(CC)C(=O)N(C1CCCC1)C N1(C(Cc2nc(C)on2)=O)CC(C(=O)O)CC(C)C1.c1ccccc1C C1(C(N2C(CNC(C(c3cnn(C)c3)OC)=O)COCC2)=O)C(C2CC2)C1(F)F CN1CCC(C(N(CCO)CCNC(=O)C(c2cccn2C)=O)=O)C(O)C1 c1(C(N2CCOCC(NC(C3(P(C)(C)=O)CC3)=O)C2)=O)cc2ncccc2[nH]1 c1(C(C(=O)NCCC(C)NC(=O)C(C)(C)CF)O)ccc(F)c(Cl)c1 c1(C(=O)NCC2(O)CN(C(C3C4CCCC34)=O)C2)cncc(O)c1 c1(C(=O)NC2CN(C(CCOCC#C)=O)C2)cncc(SC)c1 C(C1=NOC2OCCCC12)NC(=O)NCc1nnc(CC)o1 c1(C2(C)N(C(=O)NCc3nc(C(=O)OC)c(C)s3)CCC2)ccnc2ccccc12 Cc1cc(CCC(=O)NCCOCC(=O)Oc2ccccc2)cc(C)n1 C1(CC=C)(NC(C2(CCCC)CC2)=O)CCN(C(=O)CS(=O)CC)C1 Cc1nsc(C(N2CC=CC(NC(c3ccc(C(F)F)o3)=O)C2)=O)c1N c1(OC)cc(C(=O)NCC(CNC(c2cn(C)[nH]c2=N)=O)CO)nnc1C1CC1 c1(C(=O)NCC(CCOC)NC(C2(C(F)(F)F)CCCC2)=O)cnc(O)c(Cl)c1 c1(C(=O)NC2CCC(CNC(C(CC)(CC)CO)=O)C2)cc(=O)n2ccsc2n1 c1(C(N(CCNC(CC=C=C)=O)Cc2cccnc2)=O)cccc(CF)c1 c1(C(C)C)ccc(O)c(C(N2CC3C(NC(C4CCCCO4)=O)C3C2)=O)c1 c1(C(C)(C)C(=O)OC2CCC(OC(C3CC(F)(F)C3)=O)C2)ccc2ccoc2c1 Fc1cc(CSCC2CC23CCOCC3)cc(Br)c1 c1(C(N2C(CN(C(=O)CC3CC4(CC4)C3)C)CCC2)=O)ccc2cnnn2c1 C(CCC(C)(C)C)(c1nnnn1C(C)C)NCc1cnn(CC)c1C c1(OC)ccc2c(CC(=O)NC3CCN(C(=O)C=CBr)C3C)c[nH]c2c1 Cc1cc(=NC(C)C2CN(C(c3nccc4[nH]ccc34)=O)CCO2)[nH]c(C)n1 c1(CN(C2CCC(C)(CC(C)C)C2)C=O)ccc(Br)cc1Cl C(=O)(CC(C)(O)C1CC1)N(C1CCN(C(c2ncoc2C2CCCO2)=O)C1)CC C1(CC=C)(C(=O)NCCN2CCC(C)C2)CCN(C(=O)COCC(=C)C)C1 C(=O)(C#CC1(CC)COC1)NC(CC#CC)C(=O)NC1CCC(=O)NC1C n1(CC(=O)N(CC(C)NC(c2cc(=O)n(C)o2)=O)C)cnc2sccc2c1=O N1(C(C(C)C#N)=O)CCN(C(CNC(c2cscc2F)=O)C(F)(F)F)CC1 C(C(C)(C)C(=O)NC(c1nnc(C)o1)C)NC(C=C(C)C(C)C)=O CCC(C)C(C(=O)NC1CC1CNC(=O)C(C1CCCCC1)F)NS(C)(=O)=O C(=O)(C(O)CC(C)(C)C)NCC(C)(CO)NC(c1nn(CC)c(O)c1)=O CCCC(CNC(c1cc(COC)[nH]n1)=O)C(=O)N(CC(=O)OCC)C N1(C(c2ccn(C)c2)=O)CC(O)CC1CNC(c1cc(Br)nn1C)=O CN1CCN(C(c2cncc(O)c2)=O)C(C(=O)NC2CCN(C3CC3)C2)C1 c1(C(N2CCC(NC(COCCC)=O)C2)=O)ccc2ncc(=O)[nH]c2c1 C12COCC1C(=O)N2.C(CC(=O)OCCCCC)OC(COCCC=C)CCCC c1(NC(C23CC(NC(=O)Nc4cccc(C)c4)(C2)C3)=O)nc(Cl)c2c(n1)COC2 C1(CNC(CCC(=O)NCCC)=O)CC12CCN(C(=O)C(O)CCSC)C2 N1(C(C2C(C)(C)N(C(=O)CCCCN=[N+]=[N-])CC2)=O)CCCC(C2CC2)CC1 Cc1cc2[nH]c(CN3CCn4c(C5CCCN(C)C5)nnc4C3)cc(=O)n2n1 C1(CC)CC(CC(=O)NC2CN(C(C3(C)CCCC3)=O)CC2C)CCO1 N1(C(C(CC#C)C2CC2)=O)CC(C(=O)NC(c2ccccc2O)C)C(F)(F)C1 N1(C(C2CC(OCC)C2)=O)CC(C2(NC(c3ncccn3)=O)CC2)C1 c1(C(=O)NCC2N(C(CCSCCCC)=O)CC(C)CC2)[nH]nc2ncccc12 Cc1c(C(=O)N(CC(Cc2ccccc2)NC(c2cn[nH]c2)=O)C)c(Cl)nn1C Cc1cc2c(NC3CCN(C(=O)CN4C(=O)CSC4=S)CC3F)ncnc2[nH]1 C1(CN(c2nc(C(F)(F)F)ns2)C)CCCN(C(=O)COc2cccc(Cl)c2)C1 C1(NC(C=C(C)C)=O)COC2(CCCN(C(c3cc4cc(Cl)ccc4[nH]3)=O)C2)C1 O=C(N=c1nc(Cl)[nH]s1)C1=NOC2(NCC(F)F)c3ccccc3N2C1 Cc1ccc(N)c(C(=O)NCC2(CNC(C3(C)CC3F)=O)CC2)c1F C1(C(=O)NCC2N(C(Cc3nn(C)c(Cl)c3)=O)CC2)CCc2ccnn2C1 Cc1cn2cc(C(=O)NCCN(C(=O)CCC(C)N(C)C)C(C)C)nc2s1 C12(CNC(C3CCCCCC3)=O)CC1CN(C(=O)CCCc1ccccc1)C2 C(CC1CCc2ccc3c(c21)CCO3)NC(C1CCC2(CN(C(CC)=O)C2)O1)=O c1(CC)ccccc1C1(C(N2CC(OCC)C(NC(=O)C(CC)OC)C2)=O)CC1 c1(OC)ncc(Br)c(=NC(=O)C2CC3CC3N2Cc2occc2Br)[nH]1 C1(C(N(C2CC(OC)C2)C)=O)CC(C)(NC(c2cnn(C(C)C)c2)=O)C1 N1(C(CC2(COC)CCOCC2)=O)CCC(COC)(NC(C2(C)CC2F)=O)CC1 C1(CNC(Cc2n(C)ccc2)=O)C2CN(C(=O)CCNC(C3CCCO3)=O)CC12 C(CCCCC(=O)NCC12CCC(F)(CC1)C2)N(C(=O)C(O)C1CC1)C Cc1cn2c(C(=O)NCC3CCC(NC(=O)C(F)=C4CCC4)C3)c(C)nc2s1 c1(NC(C)=O)cncc(-c2cc(C)cs2)c1 C=C=CCCC(=O)N1CCC(N(C(=O)CSC(F)(F)F)C)C1 N1(C(c2c(CC)nccc2)=O)CC(NC(=O)C(C)(C)C2CCCO2)CCC(O)C1 Cc1nc(O)c(C(=O)NCC2CCCN(C(=O)C(C#N)C3CC3)C2)nc1C N1(C(CC(C)(C)OC)=O)CC2CC(NC(=O)CC3(n4cncn4)CC3)C(C2)C1 N1(C(c2n(C)ccc2)=O)C(CNC(=O)C=Cc2cncc(F)c2)CC2COCC12 N1(C(C2C(CN(C)C)CC2)=O)CCC2CCN(C(=O)COCC(C)(C)C)CC12 O=C(CC1CCc2ccccc21)N1CCCC(CNC(C23CCC2C3)=O)C1 c1(C(=O)NCC2CN(C(CC(C)C)=O)C(C)C2)cnc2c(c1)N(C)CCO2 c1(C(=O)NC2C(C(=O)NCC(CC)(C)COC)OCC2)cc(C)ccc1F C1(C(=O)NCCC2CCCCN2C(=O)C(Cl)=CCl)(OC)CCC12CCC2 Cc1cccc(OC(C)C(=O)N(C(C)CNC(c2cc(CC(C)C)[nH]n2)=O)C)c1 CC1(C(N2CCCC2CCNC(=O)CCC(F)(F)F)=O)CCCNC1=O C(C(CC(C)C)C(=O)NCC(C)(C)NC(C1CC(C2CC2)=NO1)=O)OC Cn1ncc2c(N(C3CCNC3)Cc3cc4ccccc4s3)ncnc12 C1(C#N)(CC(=O)N(CC(C)NC(=O)C(C)O)C)CC1 CCCCC(O)C(=O)OC1CCCC1OCC.c1(C(C=O)=O)ccc(Cl)cc1 C1(C(N(c2ccccc2)C)=O)CCC(NC(c2ccn(C(F)F)n2)=O)C1 C(C(C)(O)CC(=O)N1CCC(NC(=O)C=Cc2ccc(Br)cc2)C1)OC C(=O)(CS(=O)(=O)C1CC1)N1CC(CN(C(=O)C=CCN2CCCC2)C)C1 N12CCC1CCCC2.N1C(=NCc2ccccc2C(F)(F)F)N1.C=CC(C)(C)C.C CC1CCC(CC(=O)NC2C3CC2N(C(=O)CN(CC(C)(C)C)C)C3)CC1C C1(CC(=O)NCC(N(C)C(c2cnccn2)=O)C2CC2)CCCC2(CC2)C1 N1(C(c2c(NC(C3(C)CCCC3)=O)cncc2)=O)CCCC(F)(F)CC1 CCCCC(CC)CC(=O)NCC(c1ccccc1CC)NC(C1(O)CCCC1)=O C1(CNC(C(C)OCC)=O)CC2(CC2)CN1c1ccnc(C)n1 c1(CC(=O)NC(CC(=O)NCC(C)=O)Cc2cccs2)cc([N+](=O)[O-])ccc1C C1(C(N2C(C)(COC)CCC2)=O)CC2(C1)C(C(=O)O)C2(F)F C(=O)(C1=NOCC1)N(CC(C)(C)NC(=O)CSCCCN)C C1(NC(c2c(SCC)nccn2)=O)CCCN(C(=O)C(C)=C2CC2)C1C c1(C(=O)NC23CC(NC(C4CC4F)=O)(C2)C3)c2ccccc2cc2ccccc12 C(=O)(C(CCC1CCC1)OC(c1ccccc1)=O)OC.N12CCCC(C1)OC2=O c1(C(CC(=O)OC)NC(=O)NC(COC)(C)C)cc(Cl)ccc1Cl c1(CC(=O)NCCCN(C(c2nc(C(C)C)oc2)=O)C)ccc(Br)cc1 c1(C(=O)OC)c(C)noc1NC(C1CC(O)CN1C(c1cc[nH]n1)=O)=O C(=O)(CCCCN1CCOCC1)NCCNC(C(F)=CC)=O.C12CN(C1)C2=O C1(C(=O)NC2C(SC)CN(C(=O)C=C(C)c3ccsc3)C2)CCOCC12CCC2 c1(CNC(=O)NCC2CCCSC2)cccc2[nH]ccc12 c1(CC(=O)NC2CCCN(C(CC3CCC(=O)NC3)=O)C2)cc(F)ccc1Cl N1(C(c2c(C)nc(N(C)C)s2)=O)CC(C2(NC(=O)COC(C)(C)C)CC2)C1 c1(NC(C2C(NC(c3cc(C(C)(C)C)no3)=O)C2)=O)cnccc1[N+](=O)[O-] c1(CCOC(C)C)nc(COc2ccccc2Br)n(-c2cncc(Br)c2)n1 C(=O)(C(C)(C)C(F)(F)CC)N1CCC(C(C)NC(CC(CC)OC)=O)CC1 C1(C)(C(N2CC(=C(CNC(Cc3c(C)ncs3)=O)F)C2)=O)CC(O)CN1C C1(c2nnnn2-c2ccc(SC)cc2)(NC(CC)(C)C(C)C)COCCOC1 C=CC1(CC(=O)NC2(C)CCCN(C(c3cc(C#N)no3)=O)C2)CCOCC1 Cn1c(=O)c2cc(C(N3CCC(C)(c4ccc(CN)cc4)C3)=O)sc2n(C)c1=O CCCC(C(=O)NC1CCN1Cc1cn(-c2ccc(SC)cc2)nn1)C(=O)O N1(CCC(=O)NCC2CCCC2NC(C2CC2(F)F)=O)CCCS1(=O)=O C12(C(C)OC(C(CC)CCC(=O)OC(C)(C)C)=O)C3C4C1C1C2C3C41C C(C)(CCCNC(C1(COC)CCOC1)=O)NC(C1C(=C)C1)=O c1(C(=O)NC2CC(F)CN(C(C3(F)CC=CC3)=O)C2)ccn2nnnc2c1 C1(CNC(Cn2c(C)ccn2)=O)CC(C(C)C)CCN1C(=O)C(C)NC(N)=O c1(C(C(=O)NC2CCN(C(C3(C4CCC4)CC3)=O)CC2)O)ccc(F)c(Cl)c1 N1(C(C2C(C(N)=O)COC2)=O)CCOCCC1C(=O)NC12CCC(CC1)C2 C1(N(C)C(C2CCCNC2=O)=O)CCCN(C(C2(Nc3ccccn3)CC2)=O)C1 C1(C(=O)NC2(C(=O)O)CCCCC2)CCCN(C(C2CC2C2CC2)=O)CC1 C1(NC(=O)C(c2cccc(F)c2)O)CC2C1CCN2C(=O)CCCn1cccc1 C1(OC)(CNC(c2ccnnc2O)=O)CCN(C(=O)C2CC2)C1 Cc1cc(C(=O)NC2CCC(C(=O)NCC3CC4C=CC3O4)C2)ncn1 N1(C(c2c(C)n(C)cc2)=O)CC(NC(C2CC2C2CCCO2)=O)C2CCCC12 C1(C(N2CCC(C)C(CNC(=O)C(F)(F)C(F)F)C2)=O)CC2(COC(=O)N2)C1 c1(C(C(=O)NC(C)(C)C)N(CCS(CC)(=O)=O)C)ccc(C)cc1SC c1(CC)ccc(F)c(F)c1.c12nnc(-c3ccc[nH]3)n1CCC1(N)CCN2C1 c1(C(C)(C)CN2CCC(CCCC3CCCNC3)CC2)ccc(F)cn1 C(C(C(=O)N1CC(O)CCO1)NC(=O)CC(F)(F)CC)SC c1(C(=O)NCC(C)NC(=O)OC(C)(C)C)cnc(NCC2CCC2)nc1 C1(C(=O)NC2(CN(C)C(c3cnnc(O)c3)=O)CC2)CC2(CCCO2)C1 Cc1ccc(C)c(C(N2CCCC(NC(=O)C=Cc3ccccc3F)CC2)=O)n1 c1(C(N2CC3CCC(C2)N3C(C2C(F)(F)C23CC3)=O)=O)ccc2nn[nH]c2c1 N1(C(N2CCCC2CC(C)C)C(=O)NC)Cc2cc(OC)c(OC)cc2C1.O N1(CC(=O)NC(C2CCOC2)CNC(c2nn[nH]c2Cl)=O)C(=O)CCC1=O C1(C(N2CCCC2CCCO)=O)NC2CC1CC2O N1(C(c2ccc(N)c(OC(F)F)c2)=O)CC2OCCN(Cc3ccccc3)C2C1 C=C(C)C(C)(C)C(=O)N1CCCC(CC=C)(NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCC2(O)CCCN(C(=O)C(O)CF)C2)c1C C(c1cc(F)c(F)c(F)c1)=CC(=O)NCCCN(C(=O)CCCCN(C)C)CC c1(C(=O)NCCC(C)N(C(C(CC)F)=O)C)cc(C(F)F)ccc1F c1(C(N(C2CC(NC(=O)CCCCCn3cnnn3)C2)C)=O)ccc(F)cc1F C#CCCCC(C)C(=O)N1CC(CCC(=O)NOCCCN(C)C)(C)C1 c1(C(=O)NC2C(CC)CN(C(c3[nH]nnc3C)=O)CC2)cnc2c(Cl)cccn12 C1(C(=O)NCC(C2CCCC2)NC(C2(CCCC)CC2)=O)CC1(C)C C1(C(=O)NCc2ccc(F)c(N)c2)(CC)Cc2ccccc2C1 c1(C(=O)NCC2C(CNC(C=Cc3cn(C)nn3)=O)C2)cnc2ccc(F)cn12 c1(OC)ccn2c(C(=O)NCC3CCN3C(=O)Cc3ccc(N)cc3)cnc2c1 C=CC(C(=O)NC(C(=O)NCCc1cncn1C)c1ccco1)OC C1(CN(C(=O)OC(C)(C)C)CC2CC2)CC(C(=O)NC2CSCCO2)C12CCC2 C1(C(N(CCNC(c2cnoc2-c2cccs2)=O)CC)=O)CCC(=O)N(CC)C1 CC1(C(=O)NC2CCC(CSc3ccccc3)C2)CC2(CC2)C1 C1(C(=O)NCCCC(C)NC(=O)C(O)C(C)C)(OCCCC(C)C)CCOCC1 CC1CN(C(=O)NCC2(CN(C)C)CCC2)CCN1C1CC1 c1(C(N2CC(NC(CCC=C)=O)(CO)C2)=O)cc(OC)cc2ncccc12 N1(C(c2c(C)ccnc2)=O)CCC(O)C(NC(=O)C(C)Oc2cccc(Br)c2)C1 C1(N(C(CCOCCOC)=O)C)CCC(CNC(=O)C(C)(C)OC(C)=O)CC1 Cc1cc(F)c(C(=O)NC(c2ccccc2)Cc2ccc(Cl)cc2)c(F)c1 C(C)(C(=O)NCCC(C)CO)(N(C(C(C)OCC)=O)C)C1CC1 CCC(C)N=c1nc(N(C)CC2CN(C)C2)c2cccc(F)c2[nH]1 CC1OC(C)C(C)C1C(N1CC(=C(F)CNC(C2(C3CC3)CCC2)=O)C1)=O c1(OCC)ncccc1C(N1CC(NC(c2ncoc2C2CC2)=O)C(SC)C1)=O C(CN=c1[nH]c(=NCC(CC)(CC)SC)c2cc(Cl)ccc2[nH]1)(C(F)(F)F)OCC C(=O)(CCCN(C)N=O)NC1C(NC(COCCCC)=O)C1 C(CN=C(NC1COC2COCC12)N1CCCCC(S(C)(=O)=O)C1)OC CC1(C)CC(CNCC2CCCN2C2CC2)CN(Cc2ccc(F)cc2F)C1 N1(C(c2cc(C)ns2)=O)CCN(C(C2CCCN(C)C2)=O)C(c2cn[nH]c2)C1 N1(C(CC2CC(CNC(C(C)NC=O)=O)C2)=O)CC2COC(=O)C2C1 N(C1CCc2cc(CNC(=O)C3CC3)ccc21)C(C(C)Cc1ccccc1)=O N1(C(C(CCOC)NC(C2(C#C)CCCC2)=O)=O)CC(C)(C)CCC1C Cn1nnc2cc(C(=O)NC3CN(C(c4cccs4)=O)CC34CC4)ccc12 Cc1cnc(CN2CC(O)CC2C(N2CCC2c2ccccc2)=O)cc1Br C1(CNC(c2ccc(CC)[nH]2)=O)CCCCN1C(c1n[nH]cc1F)=O CN=c1[nH]cc(C(=O)NCCc2n[nH]cc2C(=O)NCC2(C)C=CCCC2)s1 n1(CC(=O)NCC2CN(C(C=CS(C)=O)=O)CC2O)cc([N+](=O)[O-])ccc1=O C1(CNC(C2CN(C(C)C)C2)=O)CCCC(NC(C2CC2c2cccnc2)=O)C1 CC(C)(C)CC(C)(C)C(=O)NCC12COC(CN=c3nc(O)c(Cl)c[nH]3)(C1)C2 c1(CC(C)CSCc2ccccc2)nnnn1C1CNC1 C(=O)(C1=C(C)N(C)c2ncnn2C1)NC1CN(C(C(C=C)O)=O)CC2(C1)CC2 c1(C(=O)NC2(CCNC(c3cc(CO)on3)=O)CC2)csc(-c2ccccn2)n1 N1(C(C(CC2CC2)OC)=O)CCC2C(NC(=O)CCc3cscn3)C12 N1(C(C2(CC=C)CCCC2)=O)CCC(NC(=O)CCC(C)C)C(F)C1 CCC(C)CC(C(=O)NCc1cccc(F)c1F)NC(=O)CCc1cscn1 C(=O)(C1=CCCN(C(c2ccc(O)nc2C)=O)C1)N(CCCC)CCOC Cc1c(C(N2CCC(CN(C)C(C3CCCSC3)=O)C2)=O)oc2c(F)cccc12 C(C1=NOC2CCCC12)n1c(N2CC(CC)N(C)CC2)nnc1-c1cnccn1 Cc1nccc(C(=O)N(CC(C)(C)C(=O)NC2COCC2N(C)C)C)n1 C1(C)(CNC(C(N2CC(C)(NC(=O)OC(C)(C)C)C2)=O)=O)COCCO1 N1(C(C2C(OC)C2)=O)CC(NC(c2csc(-c3ncccn3)n2)=O)CC12CCC2 C1(C(=O)NC(C2N(C(c3nc(CCC)sc3)=O)CCC2)C)CCOCC12CCC2 c1(C(N2CCC(C)(C(=O)NC)C2)C(=O)NCC(F)F)cnn2c1CCC2 c1(CC)c(C(=O)NCC(CNC(c2cc(C3CC3)sn2)=O)OC)cnn1C c1(-c2c(CN(C(CC#CC)c3nnnn3CC)CC=C)noc2)ccc(Br)cc1 C1(C)(NC(C(Cc2cnc[nH]2)NC(C)=O)=O)CCN(C(=O)C(=O)NC(C)C)C1 CC1CCC(CNC(=O)C=Cc2cnn(C)c2)N(C(=O)Cn2ncnn2)C1 CC12CC(CNc3cccc(-c4ccncc4)n3)(C1)C(NC(=O)C1CC1)O2 N1(C(CSCCC)=O)CCCC(C(=O)NCC2CCCCCC2)C1 c1(-c2c(C)ccs2)nc(C2CSC2)nn1CCC(F)(F)F N1(C(C=CSC)=O)CCC(C)(CCNC(C2CCCOCC2)=O)C1 N1(C(C(c2ccc(C)o2)C)=O)CC2CC(NC(=O)C=Cc3ccncc3)C2C1 c1(C(N2CC(C)(C)C(NC(=O)COC3CCCC3)C2)=O)cnc2[nH]ccnc1-2 N1(C(CC=CC)=O)CCCCC1C1CCCN(C(c2cccc(=O)o2)=O)C1 N1(C(C23CC(C2)C3)=O)CCN(CC2CN(C(=O)C=Cc3ccco3)C2)CC1 N(C(=NCCC(=O)Nc1ccccn1)N1CCC(COC2CCCC2)C1)C(C=C)C C1(F)(CNC(C2(CCC)CCC2)=O)CCN(C(=O)C(C)(C)CCSC)CC1 c1(C(=O)NC2C(C)(C)C(CNC(c3cn[nH]c3)=O)C2)sc(C#N)cc1Cl N1(C(C(CCC)NC(C)=O)=O)CC2CCCC(C1)N2C(c1nn[nH]c1Cl)=O C(=O)(C(C)(C)CS(N)(=O)=O)N(CCC(C)NC(=O)CC1Cc2ccccc2O1)C C1(C(N(CCOC)CCNC(C2CCN(C)C2CC)=O)=O)CCOC2(CCCC2)C1 C#Cc1ccc(C(=O)NCC(c2ccccc2)CNC(C2CC2CC)=O)c(C)c1 N1(C(C(CC)C)=O)CCC(O)(CCNC(=O)CCc2cn(C)nc2C)C1 C1(CNC(=O)Cc2csnn2)CCCCCN1C(=O)C=C1CN2CCC1CC2 CC(C(=O)N(C)Cc1ccc(Br)cc1)C(F)(F)F N1(C(c2c(C)c(Cl)ccc2)=O)CC23CCCC2(C1)CN(C(C1CCC(=O)C1)=O)C3 N1(CC(C)C)CC(C(=O)NCC(C(C)(C)C)NC(C2CC23CC(O)C3)=O)CC1=O c1(C(=O)NC2CN(C(C3C(SC)CCC3)=O)C2)c[nH]c(=NC2CCOCC2)cn1 N1(C(C2N(C)CCCCC2)=O)CCC(C(=O)NC(c2ncc[nH]2)(C)C)CC1(C)C C1(O)(CC(N2CCC(NC(C(C)Cn3ccnc3)=O)C2)=O)CCOCC1 C(=O)(C#CC1CCOC1)CC1C(Cn2cc(-c3cccc(N)n3)nn2)C1(F)F Cc1[nH]c(=NCC2CN(C(c3cc4occc4[nH]3)=O)CC2C)ccc1[N+](=O)[O-] c1(C(=O)NCC(C2CC2)NC(C(CC=CC)CC)=O)cc2c(C)n[nH]c2cn1 C12(NC(C3ON=C(C(C)(C)C)C3)=O)CCOCC1CN(C(c1cscn1)=O)C2 CSC1=C(C(=O)N2CCCC2(C)CNC(=O)C(C2CCOCC2)C)CCCC1 N1(C(C2(NC(C3C(C)OCCC3)=O)CCN(C)C2)=O)CC2CSCC2C1 c1(C(N2CCC(NC(=O)CSC(F)F)(CF)C2)=O)c(Cl)ccc2ccncc12 c1(C(C)C(=O)N(C2CN(C(=O)CCc3cnn(C)n3)C2)C)ccc(F)cc1 c1(CC(=O)NCC(C)(CO)NC(C=C(C)C(C)C)=O)cc(C)sc1C N#Cc1cc(C(N2CC3CC(C2)C3(F)F)=O)c(O)cc1N c1(N)cc(C)c(S(=O)(=O)N(OCC=C(C)C)CC2CC2)cn1.C1(C)CC(C)(C)CO1 C1(C(=O)NC2CC(CNC(Cc3n(C)ccn3)=O)OCC2)CCc2c[nH]nc2C1 N1(C(C=CCN(C(Cc2c(CC)con2)=O)C)=O)CCC2(CCCOC2)C1 CC1Cc2cc(CC(=O)NCC3CC(NC(=O)C(F)(F)CO)C3)ccc2O1 N1(C(C(CC)(C)CNC(=O)Cc2csc(C)n2)=O)CCc2ccncc2C1 Cc1ccc2c(C(=O)NC3CN(C(C4COC(=O)O4)=O)CC(C)(C)C3)c[nH]c2c1 c1(CNC(C(C2CC2)NC(CC2(COC)CC2)=O)=O)ccc(C)c(C)c1 N1(C(C(C)OC2CCCCC2)=O)CC(CNC(=O)C2=CCCC2)OC2(CCC2)C1 N1(C(c2cc(OCC)no2)=O)CCC(O)(C(C)NC(=O)C(CC)SC)CC1 c1(OC)ccc(Br)cc1CCNC(=O)C(=O)NC1CCN(c2ccc(F)cc2)C1 c1(C(N2CCC(CCNC(CC(C=C)CCC)=O)C2)=O)cncc2ncccc12 C(=O)(C(CC=CCl)c1ccccc1)NCC(CNC(=O)Cc1nonc1C)OC C(=O)(CCCC(C)NC(C1CCC2CC12)=O)NCC(C(C)C)(C)C N1(C(C2CCC(C)(C)N(C(=O)CCc3nccs3)C2)=O)CCCCC2(CCC2)C1 Cc1cncc(CCC(=O)NCC2CC(C)(NC(=O)C(C)CC3CCC3)C2)c1 C(=O)(C(C)(C)C(N)=O)N1CC(OC)C(C(N2CCC(C)(C(=O)OC)C2)=O)C1 c1(C(=O)NCCC(C)CCNC(C2COCC(C)(C)O2)=O)c(F)ccc(F)c1N c1(C(=O)NCC(CNC(c2cc(F)cc(F)c2)=O)OC)cncc2n[nH]cc12 N1(CCNC(C(c2ccccc2)NC(C=C(CCC)C)=O)=O)CC2CC2C1 C1(CC)C(NC(=O)C(O)C(C)C)CCN1C(=O)CSCCc1ccccc1 C1(CNC(C2CC(=C)C2)=O)CC(F)(CNC(=O)C(=O)NCC(F)(F)F)C1 c1(CNC(=NCCC=C)NC2CC(OC)C23CCC3)ccc(S(N)(=O)=O)cc1 C1(CC(=O)NCC(CC=C)NC(C2(C)CCCCO2)=O)CCC2(CCCC2)CC1 C(=O)(C(C)(C)CCN(C)C)NCC1(NC(C=Cc2ncc(C)[nH]2)=O)CCC1 C(C)(CCCCNC(=O)Cn1nnc(C2CC2)n1)NC(c1n(C(C)C)ccn1)=O c1(C(=O)NC(C2CCCN(C(=O)Cc3ccccc3)C2)C)c(F)cc(O)cc1F C1(NC(=O)Cn2cccn2)CCC2(CC1)CN(Cc1ccc(F)c(Cl)c1)C2 C1(CNC(CC(C)SC)=O)CC2(C1)CN(C(=O)CCc1nc[nH]n1)C2 CC1CCN(Cc2ccccc2SCc2nccs2)CC1c1ccc(O)cc1 Cc1nnccc1C(=O)NCC1(F)CC(NC(C2(c3ccc(Cl)nc3)CC2)=O)C1 Cc1ncnc(C)c1CC(=O)NCC#CCNC(c1ccc(N)c(Br)n1)=O c1(C(N2CCC(C(C)NC(c3c(SC)nccn3)=O)C2)=O)cc(C)c(CO)cn1 C12CN(CC1c1ccccc1)C(=O)N2.c1(COC)cncc(C(C)C)c1 C1(NC(C(CNC(C2CC(OC)C2)=O)C)=O)CC2CC1OC(=O)N2 N1(C(C(C)NS(CCCC)(=O)=O)=O)CCN(C(=O)CC2(C)CCC2)CC(C)(F)C1 N1(C(C2C(C)(C)COCC2)=O)CC(CNC(=O)C#CC2CCC2)OC2(CCC2)C1 N1(C(Cc2cnc(C)s2)=O)CCC(CO)C(NC(c2sc(CO)nc2C)=O)C1 C(C1(O)CCc2ccccc21)NC(CC(C)C)c1nnnn1CC1CCOCC1 c1(C(=O)NCc2cccc(-c3c(C)nn(C)c3)c2)cc2cc(F)ccc2[nH]1 c1(C(=O)NC(CC)CNC(c2conc2CC2CCCC2)=O)sc(NC)nc1C c1(C(=O)NC23CN(C(c4cc(OCC)n[nH]4)=O)C(CC2)C3)cc(Cl)cc(Cl)c1F C1(c2cn(Cc3c(CC)ccs3)nn2)COCCN1C(=O)Cc1nc(C)sc1Cl C1(NC(Cc2cccc(OC)n2)=O)C(CNC(=O)C=CI)CCC12CCC2 N1(c2nnc(CC)s2)CCN(C(c2cn(CC3CCOC3)nn2)=O)CC(O)C1 c1(OCCC)nc(C)ccc1C(N1CCN(C(=O)CCc2cncs2)CC1C)=O N(C(=NCCCF)N1CCC(C2CCC2)C1)Cc1scc(C)n1 c1(C(=O)NCCN(CCC)Cc2ccccn2)ccc(C(C)(C)NCC)cc1 CC1CCN(C(=O)CC(C)(C)O)CC1CC(=O)NCc1nnc(O)n1C c1(C(=O)NC2C(CNC(C3CCC(C)C3)=O)CCC2)cc2c(cn1)CCCC2 C1(C)(C(=O)NC(CC(C)C)CNC(=O)CCc2cnn(C)c2)CCS(=O)(=O)CC1 Cc1cc2ccc(C(=O)NC3(C)CC(NC(=O)C=Cc4sccc4C)C3)cc2o1 N12CCC(CC1C)OCCNC2=O.c1(-c2cccc(C)c2)cc2sccc2[nH]1 C=CCCC(C)(C)C(=O)NCC(C)(C1CC1)NC(C1CCCCN1C)=O C(c1c(Cl)nc2sccn12)=CC(c1ccc(C(F)(F)F)nn1)=O Cc1cccn2cc(CC(C)NCC3(C)CCNC3)nc12 O=C(O)CCCC(=O)NCC(c1ccc(Cl)c(Cl)c1)O C(=O)(C(CNC(C1CCCCNC1=O)=O)CCC)NCCC(=O)NCC#C N1(C=O)CCNCC1.CC1(C)CN(C2CCN(C(=O)C(F)n3cccn3)C2)C1 CC1CCCC1(C(=O)NCC1(n2ccnn2)CC1)NC(=O)Cc1ccsc1 n1(CCC)ncc(C(=O)NCCC2(O)CN(C(c3cccc[n+]3[O-])=O)C2)c1Cl Cc1nccnc1-n1cc(-c2cscn2)nn1.C12CCCN(C1)C(=O)C(C)C2 c1(C(N2CCC(C3N(C(C(CC)F)=O)CCC3)C2)=O)ccnc(C2CC2)n1 CCC(C)C(O)CC(=O)NC(C)(CNC(=O)CSC(C)(C)C)Cn1cccn1 N1(C(C2(C#N)C(C)C2)=O)CC(C2(NC(=O)CC=CC(C)(C)C)CC2)C1 C=C1CC2(C1)CC(C(=O)NC1CN(C(c3ccc(Cl)nc3OC)=O)CCC1C)C2 c1(-c2cn(CC(=O)NCc3c(C)nc(C)o3)nn2)c[nH]c2nccc-2c1 C1(O)(CNC(c2cnc(O)o2)=O)CCCN(C(=O)C2=CCCS2)CC1 c1(CC)nc2c(C(N3CCCC3(C)CNC(=O)CS(C)(=O)=O)=O)ccnc2[nH]1 C(C(=O)NC(C)CCNC(c1nc(=O)n(C)[nH]1)=O)(C(C)C)c1cnc(C)s1 CCC(O)C(F)(F)C(=O)NCCCN(CCO)C(c1cc(C(=O)OC)ccn1)=O c1(CCC(=O)NC2C(CNC(Cc3c(C)ncs3)=O)C2)c(C)n[nH]c1C N1(C(CCCOC)=O)CCCC(C2CN(C(=O)CC3CSC3)C2)C1 N#Cc1cccc(C(F)(F)CNC(c2nc(-c3cn[nH]c3)cs2)=O)n1 C1(N(C(CCN(C(c2cscn2)=O)CC)=O)C)CCCCCCC1 CC1(C(=O)NCc2cccc(O)c2)CC(O)CN1C(=O)CN1CCCCC1 CC1(C)OCC(c2cn(CCCC(=O)NCCN3CCC(CO)C3)nn2)O1 c1(C(=O)NC(C2CCN(C(CCCCSC)=O)CC2)C)cccc(C(C)C)c1O C1(NC(CCCC)=O)COC2(C1)CN(C(C1CC3(CCC3OC)C1)=O)C2 C1(C(=O)OC)CCOC1C(=O)NCC1(OC)CN(C(=O)C(CC)OC(C)=O)C1 C1(CNC(Cn2c(C(=O)OCC)cnc2)=O)C2CC1N(C(=O)C=C1CCCC1)C2 c1(OC)ccc(CN2CC3C(C2)N3C(C2CCC(=O)NC2)=O)cc1C(C)C C(=O)(CC(C)(C)CC(=O)NCC(C)(CC(C)C)NC(=O)C(C)C1CC1)OCC N1(C(c2c(C)[nH]cc2)=O)CCC(C)C(NC(=O)C=Cc2ccc(Br)o2)C1 c1(CCC)n[nH]c(=NCCC2CCC(NC(c3cc(C(C)C)[nH]n3)=O)C2)s1 c1(OCCNC(C)=O)ccccc1.C1(=O)C(C)OCCC2(CCC2)CCOC1=O C#Cc1cc(NC(C2(C)CCCN(C(=O)Cn3ccnn3)C2)=O)cc(F)c1 CC(C(=O)NCC(O)CNC(C1OCCCC1(C)C)=O)S(=O)(=O)C1CCOCC1 c1(C(N2C(COC)CN(C(=O)C(C)(F)C(=O)OC)CC2)=O)ncn2c1CCCC2 C(=O)(C1=CS(=O)CCC1)N(C(c1ccccc1)CNC(c1ncc[nH]c1=O)=O)C C(=O)(CC(C)(C)COC)NCCCN(C(C(C=C)c1ccccc1)=O)CCO c1(CC)ccc(C(N2CC(C)C2C(=O)NC(C)Cc2cn[nH]c2)=O)cn1 Cn1nnc2ccc(C(=O)NC3CCC3NC(C3CC(=O)OC3(C)C)=O)cc12 CC(C)CCC(O)C(=O)N(C)CCOCCCNC(c1ccc[n+]([O-])c1)=O c1(C(=O)NCCC(=C)CNC(C2CC2C)=O)cc2c(C)n[nH]c2cn1 C1(C(N(C(CC(=O)OC)C)C)=O)(CF)CCN(C(C2CCCN2C)=O)C1 Cc1ccc(F)c(C(C)NC2CCCC(N3CCOC3=O)C2)c1 C(=O)(C(C)CN(C(=O)CCCN(C)C(C1CCCN1C)=O)C)NC CCCCC(COC)NC(=O)CCN(C(c1ccn(C)c1)=O)C1CC1 c1(C(=O)NC23C(C)OC(CNC(=O)OC(C)(C)C)(C2)C3)cc(Br)c(F)cc1N c1(OC)cc(F)cc(C(=O)NCC2CCN(C(c3cc(F)n[nH]3)=O)CC2)c1N C1(NC(C(C)OCC(C)C)=O)CC1C1CCCN(C(=O)CN(C2CC2)C(C)C)C1 Cc1ccn(CC(=O)NC2CN(C(c3cccnc3)=O)C2)c(=O)c1 N1(C(CCN(C(=O)C(C(C)C)NC=O)CC)=O)CCOC2COCC12 CC1(CC(=O)NC2COCCOC2)CCN(C(=O)CCC2CCCC2)C1 CCCCCC=CC=CC(=O)NCCN(C(=O)CCC1CCOCC1)CC c1(C(=O)OC)cc(F)cc(S(=O)(=O)NCCCCCCCC2CC2)c1 CCCC(C(O)C(=O)N(C1CCOC1C)C1CC1)NC(c1cc(C)nnc1O)=O Cc1nocc1C(=O)NCC(F)CNC(C1C=CCCC1)=O N1(C(c2ccc(Cl)nc2)=O)CC2CCN(Cc3ccn(CCF)n3)C2C1 CC1(C)CN(C(=O)COc2ccsn2)CC1NC(c1cn(CCCF)nn1)=O c1(C(=O)NC(CNC(=O)C2=CCCS2)C2CCC2)nccc2cccnc12 C1(NC(c2c(C(C)C)ocn2)=O)COC2(C1)CN(C(=O)COCC1CCOC1)C2 N1(C(C2(CCC)CC2)=O)CC2(C)CN(C(=O)CCCC(C)O)CC2(C)C1 c1(C(N2CCCC(C(C)(O)CNC(=O)Cn3ccnn3)C2)=O)ccc(O)c(Cl)n1 c1(C(=O)Nc2cncc(F)c2)nc2n(c1Cl)CCN(C(c1ccno1)=O)C2 n1(CCOC)ccc(=NC(=O)C2CNC(=O)CN2C(c2n[nH]c(O)n2)=O)[nH]1 c1(C(N2CC(O)(CNC(c3cnccn3)=O)C2)=O)cc(Cl)c(F)cc1Cl C1(C(=O)NC2C(C)CN(C(c3ccc(F)c(Cl)n3)=O)C2)CCC2C(C1)C2(F)F CCC(CC(=O)NC(CNC(c1cn(C2CC2)nc1C)=O)C1CC1)C(F)F C(=O)(C(CC(F)F)C1CCC1)N1CC(NCc2ccc(N(C)C)cn2)C1 C1(CC)CN(C(c2cnc(F)c(C)c2)=O)CCN1C(=O)CCc1ccccc1F c1(NC(C(C(C)C)=O)=O)ccc(F)cc1CCNc1cc(O)ncn1 N1(C(CNS(CC)(=O)=O)=O)CCC(C2CCOCC2)(CNC(=O)C(C)(C)CF)C1 C(CSC)(C(=O)NC(C1CCCCC1)CNC(c1ccn(C2CCC2)n1)=O)OC C(=O)(C(CO)C(F)(F)F)NCCn1ccc(C(=O)NC(C(C)F)C)c1 c1(C(N2CCN(C(c3c(C)cco3)=O)C3C2C3)=O)c(F)ccc2cnn(C)c12 c1(C(N2CC(O)(C(C)NC(C(C)SC(F)(F)F)=O)C2)=O)c[nH]c2nccc(Cl)c12 C(c1ccccn1)=C(C)C(=O)NC1CC12CC(NC(=O)CC13COCC(C1)C3)C2 c1(OCC)ccc2c(c1)CC(C(=O)Nc1ccc(C=CC(F)(F)F)cc1)CO2 N1(C(=O)NCC=C)CCCC(N=c2[nH]nc(CCC)s2)C1 C(=O)(C1CCCc2nc[nH]c21)NCC(CN(C(=O)CC1C=CCC1)CC)(C)C N1(C(CCOCC)=O)CCCC(CNC(C2(C)CC(C)=NO2)=O)CC1 C=C1CCN(C(=O)CC(CC)CC)C(C(=O)NCc2ccn(CC)n2)C1 C(=O)(CCCCC(F)(F)F)NCCCN(C(=O)Cc1ccc(Cl)cn1)C C1(COC)(NC(=O)C(C)C)CCN(C(=O)Cc2csc(C3CCOCC3)n2)CC1 C1(C)(CN(C(C(C)C2CCCO2)=O)C)CCCC1NC(c1ccc(C(F)F)o1)=O C12(C(=O)NCCOCCN(C)C(c3cc(C4(C)CC4)n[nH]3)=O)CCC(CC1)OC2 S(=O)(=O)(c1ccc(C#N)cc1)NCC(=O)NC(C(C(C)C)Nc1ccccc1)C N1(C(C2C3CCC2CC3)=O)CCCC(C2CCCN(C(c3cnc(O)o3)=O)C2)C1 N1(C(CCCC)=O)CC2CC1C2NC(c1oc(SC)cc1C)=O Cc1cc(C(=O)NCC2CN(C(c3ccc(C4CC4)nc3O)=O)C2)cnc1Br c12cc(Br)nc(n1)NC(=O)N2.c1(OC)cccc(C(C)OC)n1 c1(C(=O)NC2(CNC(C(C)NC(N)=O)=O)CC2)cc2n(n1)CCO2 c1(OC)ccccc1C1CC(O)CN1Cc1cn(C)nc1C1CC1 C1(NC(=O)C(O)CC2CCCCC2)CC2CN(C(=O)Cc3ccccc3)CC2C1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2CN(C(C)C)C2)=O)CC(C)(C)C1 c1(C(=O)NCc2cn(CC)nn2)ccc(CS)cc1.C1(C=O)CCCC1C C(=O)(C(C)(C)C(C)(C)CO)NC1CC(OCC(=O)N(C)Cc2ncn(C)n2)C1 n1(CCN)c(C(N2CCCCCC2CCc2ccccc2)=O)cc2ccccc12 C1(NC(c2c(C)onc2)=O)COCCC1NC(C1CCC(=O)N1C)=O C1(C#N)(C(=O)NCCC2CN(C(C(C)OC)=O)C2)CCCO1 CCC(O)(CN(C(=O)C(C)N(C(=O)C=Cc1ccnn1C)C1CC1)C)CC N1(C(CCCCC#C)=O)CCCC2(C1)C(NC(=O)CC1CC=CCC1)CCN2C C=CC1(C(N2CC(CC(F)C(=O)NCC(CC)N(C)C)C2)=O)CCCCC1 c1(C(N2CCC(C)(NC(=O)C3=C(Cl)CCC3)C2)=O)nccc2ccsc12 C1(CNC(C(C(C)C)NC(N)=O)=O)CN(C(=O)CCc2nc[nH]n2)CCN1C N1(C(C=CC)=O)CC(O)CC1CNC(c1csc(C2CC2)n1)=O c1(-n2c(C3CC34CC4(F)F)nc(C3C(C)(C)C3)n2)ccc(Br)c(Cl)c1 N1(C(C(C)OCCC=C)=O)CCN(CC2CN(C(=O)C(C)OC)C2)CC1 C1(CC)CN(C)C(=O)CN1C(=O)COC1CC(NC(=O)Cc2nccn2C)C1 Cc1nc(N2CCC(NC(=O)C=Cc3cn(C)cn3)C(O)C2)c(F)c(C)n1 c1(C(=O)NC2CCN(C(C3C(F)(F)C34CCC4)=O)C2)ccc2c(c1)NCCC2 CC1OC(C)(C)OC1(C)C(=O)NCC(C)(C)NC(=O)Cc1ccc2c[nH]nc2c1 c1(CC)ccc(O)c(C(=O)NCC2CCC2NC(c2ccc(C(F)F)s2)=O)c1 C(=O)(CCS(N)(=O)=O)N1C(CC)C(C(=O)N(C(C)C)Cc2ccco2)CC1 c1(NC(C2CC(=O)NC2=O)=O)ccccc1C1CCOC1 N1(C(CNc2c(C)cccc2C)=O)CC2(CCCC2NC(=O)Cn2ccnn2)C1 N1(C(CC2CCN(C)C2=O)=O)CCOCC(F)(CNC(=O)CNS(N)(=O)=O)C1 C1(C#N)(C(=O)NCCC2CCN(C(COCC(C)(C)C)=O)CC2)CC12CCC2 N1(C(C(=O)NCCCC(C)NC(=O)C=Cc2cccnc2)C)C(C)CCC1C c1(C(=O)NCC(C)(c2ncc[nH]2)NC(=O)C=CC(=O)N(C)C)cncc(C2CC2)c1 c12cnn(c1C)CC(=O)O2.C1(NC(CC)=O)CCN(C(C)(C)C)C1 c1(NC(C2(COC)CCCOC2)=O)ccccc1S(=O)(=O)C(F)F C(C1=C(C)CCCC1(C)C)NC(c1n(CC)nnn1)c1cc(C(C)C)no1 C1(F)(C(=O)NCCCCC2CN(C(C3(CC(C)C)CCC3)=O)C2)CCOC1 c1(NC(CC(=O)OC)CC2OCCO2)ncnc2c1ncn2CC(O)CO C(C(C)(C)C(=O)N(CCC(=O)NC(C)CC(C)(C)CO)OC)OCC CCCCN(C(=O)CC1CCN1C(C1(CSC)CC1)=O)C C1(CNC(c2ccn(CCOC)n2)=O)(CO)CCN(C(=O)C2=CCCS2)C1 N1(C(C(C=C)(F)F)=O)CCC(C2(NC(=O)CCc3cncc(F)c3)CCC2)CC1 CC1(C(N2CC(O)(CCNC(=O)CCCCC(N)=O)C2)=O)CCCCCCC1 Cc1cc(Cl)cc(C(N2CC(C)(NC(=O)CCNC(C3CCCO3)=O)C2)=O)c1O CC(CCC(=O)NCC1CCN(C(c2ccccc2C(F)F)=O)C1)S(C)(=O)=O c1(C(C)C)ncncc1C(=O)NC1(C)CCN(C(=O)C(F)n2ccnc2)C1 c1(CC(O)C2CC2)nc(CC23CCC(CC2)C3)n(-c2ccccc2)n1 c1(C(=O)NCC(CNC(C2CCN(C)C(C)C2)=O)OC)ccc2c(c1)CC2 c1(-c2cn(C(C(=O)NC(c3ncc(C)s3)C)C)nn2)cnn(C)c1C c1(CC(=O)NCCNC(c2c(Cl)c(C)n(C)n2)=O)cc(Cl)c2c(c1)OCCCO2 N1(C(CCOCC)=O)CC(NC(=O)C(CC)Oc2ccc(F)cc2)C2(CC2)C1 Cc1ccc(O)c(C(N2CCC=CC2C(=O)NC(C)(C)CN2CCCC2)=O)c1 C1(C(N2CC(O)(C(C)C)C2)=O)CCC2(CC2)N1C(C12CC1CNC2=O)=O c1(NC(c2n(C(CC)C)ncc2)=O)ccc(-c2ccc(C)nc2)nc1 c1(CC)ccc(C(=O)NC(C(=O)NCC2(CCO)CCC2)C2CC2)o1 c1(NC(COC)(C)CO)cccc(CC(=O)OC(C)C)c1 c1(C(N(C(C)CNC(C2CCc3cncn3C2)=O)CC)=O)c(Cl)ccc(C)c1N c1(CC(=O)NCC2N(C(c3ccn(C(C)C)n3)=O)CCC2)ncn2c1CCCC2 C1(CNC(C2(C=C)CCC2)=O)CN(C(=O)C(C)Cc2ccco2)CC1C Cc1cc(Cl)ccc1OCC(=O)N(C(C)CCNC(c1ccc(N)c(Cl)c1)=O)C c1(NC(=O)CSCc2coc(Cl)n2)ccc(Oc2ccccc2)cc1 C(C(F)(C(=O)NCCCOC(=N)O)C(C)C)NC(COCCC)=O c1(C(N2CCC(C(C(=O)NC(C#CC#C)(C)C)C)C2)=O)cccc(C#C)c1 C(C1CN(C(c2ccc(CC)s2)=O)CC1C(N1CCC(C)(CCC)CC1)=O)=CC N1(C(CC2CN(C(C)=O)C2)=O)CCN(C(=O)CC2(O)CCOCC2)CC1C1CC1 CCS(=O)(=O)CCN(C1CC1)CC1CCCO1.c1(C2C(=O)O2)ccccc1 C(=O)(CC(C)P(C)(C)=O)NCC(C)CNC(C1(C)CCN(C)CC1)=O C1(NC(C(C2CC2(C)Br)N(CC)CC)=O)(CNS(C)(=O)=O)CCCCC1 c1(C(=O)NCC(CC=C)NC(=O)C(C)OCCC(C)C)cc(CC)cc(F)c1 c1(C(N2CCC(CC(=O)NCC(C(N)=O)(F)F)CC2)=O)cnc2cc[nH]c2c1 C1(CN(CC(S(C)(=O)=O)c2ccccc2)c2ccccc2F)CCc2nnnn2C1 N1(C(c2ncc(C)cn2)=O)CCCC(C)C1CNC(=O)C=Cc1ccc(C)nc1 C(=O)(CCCCn1ccnn1)N(CC(C)NC(=O)C(C)(C)c1ccccn1)C C1(NC(c2cccc(C(C)C)c2)=O)CC2CCC(C1)N2c1ncnc2[nH]ccc12 CC1CN(C(=O)Cc2cccc[n+]2[O-])CC1CNC(=O)CC(=O)Nc1nccs1 c1(C(C(=O)NCCn2cc(C(C)OC)nn2)N(CC(C)(C)C)C)c(F)cccc1Cl c1(C(=O)NC(CCC)CCCNC(c2ccoc2C)=O)ccc([N+](=O)[O-])cc1F CC(C#N)CCC(=O)NC(CNC(c1ccnc(-c2ncc[nH]2)c1)=O)C(C)C C1(CC)CN(C(=O)C(C)(C)c2ccn(C)n2)CCN1C(=O)CCN(C)C(C)=O C12(C(=O)NCc3cc(CC)on3)CCCC1CCN2C(c1cnn(CCO)c1)=O C1(CNC(C(C)C)=O)CN(C(=O)CCc2cccc(Cl)c2Cl)C2CCN1C2 C1(C(=O)NCc2c(C)nn(C)c2)CS(=O)(=O)CC12CC2 C(=O)(CC(C(C)CC)NC(C1(OC)CCSC1)=O)NCC(C=C)O C#CC(CC(C)(C)C)NC(C1CCN(C(c2cncc(C)n2)=O)CC1)=O c1(-c2onc(CNC(C)C(=O)NCC(F)(F)F)n2)cccc([N+](=O)[O-])c1 C1(C(=O)O)C2CC2CN1C(=O)C(F)(F)C1(O)CCC1 c1(CC)oc(C)cc1C(=O)N(C(C)(C)CC(=O)NC(c1nccc(O)n1)C)C N1(C(Cc2c(OC)nccc2)=O)CCC2CN(C(C3CC(SC)C3)=O)CC12 C1(C(N2CC(N(C)CCO)C2)=O)C2CCN(C(C3OCCC3(C)C)=O)CC12 C12(NC(c3c(CNC(C(CCC)OCC)=O)ocn3)=O)CCCN(CCC1)C2 c1(C(C)C)cccc(F)c1C(=O)NCC1CC(NC(c2cnc(C3CC3)s2)=O)C1 CC1CCCC(C(=O)NC2CCC(N(C)C(c3nccnc3N)=O)CC2)CC1 Cc1oc(Br)cc1C(N1CC=CC1CN(C(=O)COC1CCOCC1)C1CC1)=O N1(C(c2cccc(OC)n2)C(=O)NCC=C)CCC2C(C1)C2(F)F C(CCCCCC(=O)N1CC(O)C(O)C1CO)NC(c1c(C)cn(C)c1)=O c1(OC)ncc(CN2CCC(C)(C(N3CCC(CO)C3)=O)C2)cn1 N1(C(C2C(CC)C2)=O)CCCC1C1CCN(C(=O)CCc2cnn[nH]2)C1 c1(C(c2n(CC)nnn2)(C)NCC2CC=CC2)cnn2cc(Br)cnc12 N1(C(c2c(C)nc(CCC)o2)=O)CC(NC(c2sc(SC)cc2C)=O)CCC1C c1(CC(=O)NCC2C(NC(COCC#C)=O)CC2)cc(C2CC2)no1 C1(CC(=O)NC2COCC2CNC(C2CCS2(=O)=O)=O)(CC=C)CCCC1 N1(C(COCC#C)=O)CCCC(C2CN(C(c3ccc(O)cc3F)=O)C2)C1 c1(CNC2C3CN(C(C4=C(C)OCC4)=O)CC2CC3)n[nH]c2cc(Br)cc(F)c12 CN1N=C(CC(=O)NC2(CO)CCCN(C(C3CCC(C)(C)O3)=O)C2)CC1=O C1(CNC(C23C(C)OC(C)(C2)C3)=O)N(C(c2cc(Cl)sc2Cl)=O)CCCC1(C)C C(=O)(C(O)C1=CCCCC1)NC1C(C(=O)NC(C2CCCCC2)(C)C)CC1 CC1CN(C(c2cccc(F)c2O)=O)CC(C)N(C(C2CN(C(N)=O)C2)=O)C1 c1(C(=O)NC2CN(C(C(CC#C)O)=O)CC23CCC3)ccc(=O)n2c1COCC2 CCCCC(CC)CCCN(c1cc(NCc2cnn(CC)c2)ncn1)C Cc1ccccc1-c1cccc(C(=O)NCc2ncsc2C)c1 C(=O)(C(C)C(C)COC)NCCN(CCC)C(c1cncc(N)n1)=O C1(C(=O)NCc2cncc(C(=O)NC(C)CCC3CC3)c2)CCCCC1(C)C C1(CNC(C(COC)C)=O)CCC2(CCC2)CN1C(=O)C=C1CN2CCC1CC2 C=CCC(C(=O)N1CCC(CCNC(c2c(N)cc(Cl)nc2Cl)=O)C1)C(C)C C1(CNC(CC2(NC(c3c(C)snc3)=O)CC2)=O)CCC(=O)NC1C C1(NC(=O)OC(C)(C)C)CCC(NCc2cccc(C(C)(C)C)n2)CN1C1CC1 CC(C)CC(C(=O)N1CCC(=CC(F)(F)F)CC1)NC(N)=O N1(C(Cn2c(C)nc(C)n2)=O)CC2CC(NC(C3(S(N)(=O)=O)CC3)=O)CC2C1 N1(C(CCC=CC)=O)CCCC1(C)CNC(C1(C2CCCO2)CC1)=O C1(C(=O)NC2(C)CC(F)(F)C2)CCOCCN1C(C1OCCC1(C)C)=O C(C)(C(=O)NCC1CCCC1N(C)C)(N(C(C(C)=CC(C)(C)C)=O)C)C1CC1 C1(NC(c2c(C)noc2)=O)CCC2CN(C(=O)Cc3ccc4c(c3)COC4)CC12 N1(C(C2(CC#C)CCN(C(=O)CCC3CCCO3)C2)=O)Cc2ccc(C)cc2C1 N1(C(C)=O)CC2CN(C(C3CC(=O)N(C(C)C)C3)=O)CC2C1 Cc1oc(-c2nc(CCn3nccn3)nn2Cc2ccc(F)cc2)cc1CO N1(C(c2cncc(CC)c2)=O)CCN(C(=O)Cc2cc(C)cc(C)c2)C(C2CC2)C1 c1(C(=O)NC2C(CNC(CCP(C)(C)=O)=O)CC2)cc(F)c(F)cc1Br c1(C(=O)NCCC(C)NC(c2cccc(CC)n2)=O)cc2sc(C)nc2[nH]1 c1(C(=O)NC2C(C)CN(C(=O)CCc3nncn3C)CC2)cnn2ccncc12 c1(CN(C(c2ccc(CO)s2)C(=O)NC2CCOC2)C)ccc(C2CC2)c(F)c1 N1(C(C(c2cccs2)SC)=O)CCC(C)(C)C(NC(=O)Cc2cncn2C)C1 c1(C(=O)NC2C(CC34CC(NC(CCC(=O)OC)=O)(C3)C4)C2)[nH]cc2c1CCC2 N1(C(c2cc(CNC(=O)CCc3csnn3)sc2)=O)CCOC2(CC2)C1 C1(NC(C=C(C)Cl)=O)CC1C1CCN(C(c2cccc3sccc23)=O)CC1 N1(CC=C)CCCN(C(=O)C(CNC(c2ccncc2)=O)CC2CCCC2)CC1 C#Cc1cc(C(N2CC(NC(=O)CCN(C)CCC)CC2C)=O)cc(Br)c1 CC(C)(C)C(C(=O)NC1CCC(NC(C23CC4CC2C3C4)=O)C1)N1CCCCC1 c1(C(N(C2CCN(C(c3cc(C4CC4)on3)=O)C2)C)=O)cc2cccnc2o1 C1(C(N(C(CC)C)C)=O)CCCCC1(C)NC(c1c[n+]([O-])c(C)cn1)=O C1(CCNC(C(C=C)O)=O)CN(C(=O)CCc2c[nH]c(C)c2C(C)=O)CCO1 c1(NC(C(C)NCC(=O)NC(C)(C)C)=O)cc(-c2ccccc2)nn1C c1(OC)cccc([N+](=O)[O-])c1C(N1CC(O)(CNC(c2ccc(F)cn2)=O)C1)=O N1(C(C2C(C)C(=O)C2)=O)CCOCC1CNC(c1ccn(C(F)F)n1)=O CC1(C)CCN(C(=O)CNS(C)(=O)=O)CC1C(=O)NC1CCCC12CCC2 CC(C(N)C(C)C)NCCCCSCC.c1(O)ccc(Cl)cn1 C1(CC)CN(C(=O)C(=O)NC(C)C)CCC1NC(=O)C(=Cc1cccnc1)F N1(CCC(=O)NCCC(C)(C)NC(C23CSCC2C3)=O)CCCCC1=O N1(CCc2cccc(OCC)c2)CCC(=O)N(CCc2cc(Cl)ccc2C)C1=O N#CC1CCC(c2nnnn2CSc2ccccc2)(Nc2ccc(F)c(F)c2)C1 Cc1nsc(C(N2CCCC(CNC(c3cc(Br)nn3C)=O)C2)=O)c1N c1(C(N2CC(CC)SCC2)=O)ccc(F)c(-c2cn(-c3ccccn3)nn2)c1 Cc1c(C(N2CC3CC(O)C2C3NC(=O)C2=CCOC2)=O)oc2ccc(F)cc12 C1(CNC(COC)=O)CC2(CCN(C(c3c[nH]nc3OC)=O)CC2)CO1 N1(C(CC2(CC=C)CCCC2)=O)CCCC(CCNC(C2CNC(=O)O2)=O)CC1 c1(CC(=O)NCC(CNC(CC2(C(=C)F)CCC2)=O)F)ccc2c(c1)COC2 C1(NC(CSCC)=O)CC2(CCN(C(=O)CCc3ccc(C)cc3C)C2)C1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCC2(CCC2NC(C2CC(C)N(C)C2)=O)CC1 CN1CCC(C)(CNC(=O)CC2CCCN(C(C3CC(O)C3)=O)C2)C1 CCCC(C(=O)OC(C)(C)C)C(=O)NC1CCCC(C(=O)NCC(=O)OC)C1 C1(N(C(C2(C(=O)OC)CC2)=O)CC2CC2)CCN(C(C2(C)CCCCO2)=O)CC1 C(=O)(CCCCCCCBr)NC(C1CCN(Cc2cc(F)c(F)cc2Cl)CC1)C C(c1c(C)noc1C)=CC(N1CCN(C(CCCSC)=O)CC1)=O CC(C)C(O)C(C)C(=O)N1CCC(C(=O)N(CC(=O)NC(C)C)C)(OC)C1 CCCN(OC)C(=O)c1coc(CNC(c2cnncc2C)=O)n1 N1(C(c2c(C)scn2)=O)CC(C)(C)OC2(C1)CN(c1ccc([N+](=O)[O-])cc1Cl)C2 N1(CC(C)NC(c2nc(C(C)C)oc2)=O)CCN(C(=O)COC(C)(C)C)CC1 CCCCCC(C(=O)Nc1cccc(Cl)c1C)N1CCN(c2nc(C)ns2)CC1 c1(C(=O)NC(CNC(c2cc(CCCO)on2)=O)CO)ccc(Cl)nc1O C1(N(C(=O)C=CC(=O)N(C)C)C)CCCN(C(=O)C(C)OC2CCCC2)CC1 N12CCCN(CC1)CC(=O)N1CC(C)(C1)OCC2=O.C(C(C)(C)C)N(C)C c1(CC)nc(=N)[nH]cc1C(=O)NC1(C)CC(NC(=O)COC(C)C)C1 N1(C(CCNC(C)=O)=O)CCN(C(C2OCCOC2C)=O)C(CC(F)(F)F)C1 N1(C(c2[nH]cc(CC)c2)=O)CC2CCC(CNC(c3ccc(COC)o3)=O)(C2)C1 C1(OCCOC)(CO)CCN(C(c2ccc(C3CCC3)cc2)=O)CC1 c1(C(=O)NC(C(=O)NC(C)CC(F)(F)F)(C)C2CCC2)cc2cccnc2[nH]1 c1(NC(C2N(C(Cc3cnc(C)s3)=O)CC2)=O)cc(Br)ccc1[N+](=O)[O-] c1(C(N2CCC(C(C)(C)NC(CC=C=C)=O)CC2)=O)ccc(NCC=C)c(F)c1 N1(CCn2cc(CN(C(c3cnc(Cl)s3)=O)C3CC3)nn2)CCCS1(=O)=O c1(N2CC(C)C(NC(=O)CCc3cccnc3F)C2)nc2ncc(Cl)cc2o1 c1(C(N2CC(OC)CC2(C)CNC(=O)C=C(C)C)=O)cc2n(n1)CCOC2 N1(C(CCC(=C)Br)=O)CCCC(N(C(=O)CC2CCOC2)CC)CC1 c1(CCC(N2CC(C)C(NC(C3COC(=O)C3)=O)C2)=O)ccc2[nH]ccc2c1 C1(NC(CC=C=C)=O)CCC2(CC1)CN(C(=O)Cc1n[nH]c3ccccc13)C2 CCCC(CCC)CC(=O)N1CCCCC1CCCNC(C12CC(OC)C1C2)=O N1(C(Cc2ccc(N(C3C(C)C3)C)cc2)=O)CCCC(N)(c2nn[nH]n2)C1 CC1CCCN(Cc2ccccc2NC(=O)COCc2ccccc2)C1 C(C(=O)N(CCC(=O)NCC(C)(C)OCC1CC1)C)(OC)OC C1(C(=O)NCCCC(C)O)(CF)CCN(C(c2ccoc2Cl)=O)C1 c1(CCNC(C(C)n2cnnn2)=O)ocnc1CNC(=O)Cc1ccco1 c1(N(CC(C)C(C)(C)C)C)ncc(S(=O)(=O)NCc2c(CC)noc2C)cc1Cl C1(C(N2C(C)CSCC2)C(=O)NCc2ccccc2)CCCCC1(F)F Cc1sc(Br)nc1C(=O)N(C1CC(NC(C2(C3CCCO3)CC2)=O)C1)C C1(CNC(Cc2n(C)nnc2)=O)CN(C(C2(C)CCOC2)=O)CC12CCC2 N1(C2CCC(c3cn(C)nc3)C2)CCCc2c1cnn2CC1CC1 N1(C(c2ccc(C)s2)=O)CC2(NC(c3cc(C)n(C)c3)=O)CC1C2 O=C(CS(=O)(=O)c1ccc(Cl)cc1)NCCCOCCNC(c1ccncn1)=O C1(C(CC)CC)CCC(NC(=O)C(=O)NCCCOC)CC1 C(CCC(=O)N(CCCc1ccco1)C(C)=O)N(CCCC)CCC c1(C(N(C2CN(C(C(C)OCCOC)=O)C2)C)=O)nc(C2CC2)oc1C C(=O)(C(C(C)(C)C)N(C)C)N1C(C(CNC(c2ccc(C)o2)=O)(C)C)CCC1 CCC(C(C)C)C(=O)N1CCC2C(NC(C3CN(C4CCC4)C3)=O)C12 C#Cc1ccc(C(=O)NC23CCC2CCN3C(=O)C(=O)NCC)cc1C Cc1cnc(CCN(C(=O)C(C2CCCO2)C2CC2)C)s1.c1(CC(=O)NC)ccco1 C(C(C(=O)N(C)CC1CCOC1C)C(C)(C)C)NC(CC(C)C)=O c1(C(=O)NC(C)CC(=O)NCC2CN(C)CCO2)cc(O)ncn1 N1(C(CNS(C)(=O)=O)=O)CCCC(NC(c2cocc2C(N)=O)=O)C1 c1(NCC(=O)NC(C(C(=O)ON)NC(=O)OC(C)(C)C)=O)cc(Br)ccc1[N+](=O)[O-] C#CCCCCC(=O)NCC1CN(C(=O)C=CC(F)F)CCC1C N1(C(C2(C)N(C)CCC2)=O)CC(C2CN(C(=O)CN3CC4CC4C3)C2)C1 CC(C)CCC(=O)N1CCCC(NC(c2cc(C(F)F)cs2)=O)C1 C1(C(=O)NC2(CC#C)CCC2)(CSC)CCCO1.C12CCN1C2=O c1(OC)ccc(C(N2CC3(CCC3)C2C2CCOCC2)=O)nc1N c1(CC)nc(=N)[nH]cc1C(=O)N(C(C)CNC(C1CCCCC(=O)N1)=O)CC C1(NC(c2cn(CCOC)nc2)=O)CC(O)CN(C(C2(C(N)=O)CCC2)=O)C1 N1(C(C=CCCC)=O)CC(F)CC1CNC(=O)CC(C)NC(N)=O CC1(C)CCCC1(C)NC(C1CN(C(c2ccnc(O)c2)=O)CCO1)=O c1(NC(=O)CC2CCN(C(c3ncccc3I)=O)C2)cc(F)c(Cl)c(Br)c1 c1(Cn2cc(C3(O)CN(C(=O)CCCCC4CC4)C3)nn2)cc(Cl)ccc1Cl N1(C(CCc2c(C)noc2C)=O)CCCC(O)(CCNC(C2CC23CC3)=O)C1 c1(CS)ccncc1.C(=O)(CCOCNC(=O)CCC(=O)NCC1CC1)C1CC1 C1(NC(C(C(C)C)O)=O)CCCC2CN(C(=O)Cc3ccc(O)c(Cl)c3)CC12 c1(NC(CSC)C)ccc(S(=O)(=O)NCC2CCOC3(CCC3)C2)c(Cl)c1 c1(OC(C2C(c3ccc(C)cc3)C2)=O)cc(F)ccc1C C(c1cc2ccccc2o1)=CC(=O)NC1CC(NC(c2n(C)ccc2)=O)C1 C1(C)(CNC(C(C)(C)SC)=O)CCN(C(C2(C(C)(F)F)CC2)=O)C1 N1(C(c2c(OC)csc2)=O)CC(NC(C2CC23CCOCC3)=O)CC(F)(F)C1 c1(N2CCCC(CN(C(c3c(CC)noc3C)=O)C)C2)nc(OC)c(F)c(C)n1 N1(C(Cc2cn(CC)nn2)=O)CCC(C)(CC(=O)NCCCC(=O)NO)C1 c1(CC(=O)OCCOc2c(C)cc(Cl)cc2)ccccc1N=[N+]=[N-] C=CCC(C(=O)N1CCC(F)(F)C(CNC(=O)Cc2cnoc2)C1)C(C)(C)C C(=O)(CC(CCC)NC(C1COCCN1C)=O)Nc1ccc(CCC)cc1 CCCCCC(O)CC(=O)N1CCN(C(C2CC2C(F)F)=O)CC1C C#Cc1ccc(C(c2nnnn2C2CCOC2)NCC2(CO)CC2)cn1 c1(NCC(=O)N(C(c2noc(C)n2)CC)C)cc(OC)nn1C c1(OCC)ccc(C(=O)NCC(C)(CO)NC(=O)CCC=CC(C)C)cc1 C=CCC(C(=O)OC)NC(=O)CSCCNC(C1C2CC(=O)CC12)=O N1(C(c2ccc(COC)o2)=O)CCC(NC(C2CCN(C)C(=O)C2)=O)C(C)(C)C1 Cc1cc(C(=O)NC2CC2CNC(=O)C(C(C)C)N2CCCCC2)c(O)nc1C CC1CN(S(=O)(=O)Cc2ccccc2Br)CCN1c1ccncc1 C1(NC(c2nn(C)c(O)c2)=O)CCN(C(=O)C=Cc2cnccn2)CC1(C)C C(=O)(CC(C)C(C)(C)NC(c1ccn2cccc2c1)=O)NC(CC=C)CC=C c1(C(N2CCC3CN(C(C4C(C)C4C)=O)C3C2)=O)ccnc2ccccc12 N1(CCC)C(=S)NC(c2cc(Cl)ccc2Cl)C2=C1C1(CCCCCC1)NC2=O c1(C(N(CC(CNC(C(F)OC)=O)O)C)=O)ccc2nn(C(F)F)cc2c1 c1(C(=O)NC(C)C(CO)NC(c2ncncc2C#N)=O)ccccc1[N+](=O)[O-] N1(C(c2ccc(OC)c(I)c2)=O)CCCc2cc(OC)ccc21 C#CCC(CC(=O)OC)NC(=O)C(CC(C)C)NC(C1CC1C(F)(F)F)=O C1(CNC(c2ccc(C(F)F)cc2)=O)CN(C(=O)CN2C(=O)CNC2=O)CC1O N1(C(Cc2ccc(OC)cc2Cl)=O)CCC2CCN(C(=O)C(O)C3CC3)C2C1 Cc1cc(NC(C2CC(C)CN2C(c2ccc3cc[nH]c3c2)=O)=O)c(F)cc1F c1(C(=O)NCCn2cnnc2O)cc2cc(Br)ccc2cn1 N1(C(CCOCCOC(C)(C)C)=O)CCC(CCNC(=O)CCc2cnoc2)C1 c1(OC)ccc(CC(N2CC(NC(=O)CCn3ccccc3=O)C(C)C2)=O)cc1 c1(CNC(C(C)OCOC)=O)ncoc1CC(=O)NC1CCCC1C(C)(C)C c1(C(N2CC(NC(C3(CF)CCC3)=O)CC(O)C2)=O)cc2c(o1)CCCC2 N1(C(CCCCOCC)=O)CCC2(CCCN2C(=O)CC2NC(=O)NC2=O)CC1 c1(C(=O)NC(CNC(C2(OCC)CCC2)=O)CC)cnc(C)nc1 C1(O)(CNC(CCN(c2ccncc2)C)=O)CCSC1.C12(CCC1)C(=O)N2 c1(C(=O)NC2(C)CN(C(c3c(C)onc3O)=O)C2)cnc(O)c(F)c1 c1(C(c2noc(-c3csc(C4CC4)n3)n2)(C)C)ccc(C(F)(F)F)cc1 N1(c2ncc(C(=O)OCC)nc2)CCCC(C2CN(c3ncc(I)cn3)C2)C1 OCC(CC1CCOC1)CN=c1nc(N2C3CCCC2COC3)c2c([nH]1)CCC2 Cc1cn2nc(C(=O)O)cc2c(N(C(C2CCC2)=O)CC#N)n1 c1(C(C(=O)NCC(CNC(COCCC)=O)N(C)C)O)cccnc1 C1(C2(O)CCOCC2)(C(N2CC3CCN(C(=O)C4=C(Cl)CCCC4)C3C2)=O)CC1 C1(CNC(CCCN(C)C)=O)CN(C(c2c[nH]nc2C2CCCCC2)=O)CCO1 c1(OC)cc(C(=O)NC2CCN(C(c3cncc(F)c3)=O)C2)cc([N+](=O)[O-])c1O C1(CC(=O)NCC2CC2C(=O)NCc2ncoc2C2CC2)CCOC1=O n1(CCC(=O)NC2(CF)CCN(C(C(C#C)(C)C)=O)C2)ccc2ccccc12 C1(CNC(=O)CC2CCOC2)CC(NC(c2cnc(-c3cccs3)o2)=O)C(O)C1 N1(C(c2cc(C)oc2)=O)CCCC(N(C)C(c2ncc(Br)cc2N)=O)C1 C(=O)(C(CC#N)c1ccccc1)NCCN(CCC)C(c1cnoc1C(C)C)=O N1(C(C(CC)N(C(=O)C=Cc2cnn(C)c2)C)=O)CCC2CCN(C)CC12 O(NC(=O)C(Cn1cccn1)NC(=O)CC(C(=C)C)OCC)CC(=C)C CC1(C)CC2(CC(C(=O)NCC3(O)CCN(C(=O)CCn4ccnc4)C3)C2)C1 Cc1cc(Cl)n[nH]c1=NC(=O)C1CCCC1C(=O)NCc1cccc(Cl)c1 CC(F)(F)C(F)C(=O)NCCOC1(CC=CC(=O)NCC(=O)OC)CCC1 C1(c2n(CCC)nnn2)(NCc2cn(C3CC3)nn2)CCC(CC)C1 N1(C(c2cccc(C)c2Cl)C(=O)Nc2ccccc2Cl)CCC(O)C(C)(C)C1 N1(C(CC2CN(C(c3ccc(CC)nc3)=O)C(C)C2)=O)CCC(F)(C#N)C1 c1(C(N2CCC(CCC(=O)NCc3onc(CC)n3)C2)=O)c(C)ccnc1O C#Cc1cccc(C(N2CC3(C2)CN(C(c2ccnc(OC)c2)=O)C3)=O)c1F N12CC3CC1C3C(=O)NC(C)(C)C=CC2=O.C1(SC)CCCC1N(C)C N1(C(C(=O)NCCCCC2CCCC(C)C2)=O)CC(N)CC2(CC2)C1 C1(C(=O)NCc2c(C(=O)NCC(CC)C)n[nH]c2)CN(C)CC(C)O1 C1(c2n(C(CC)(C)C)nnn2)(NC(C)(C)COC)CN(C)CC1C c1(C(=O)NC2CCN(C(c3cc(C)nc(O)c3)=O)C(C)C2)ccc2oncc2c1 CC1CC2CN(C(C3C(C)(C)C3(F)F)=O)CC2N1C(c1ncncc1Cl)=O N1(C(C2CC(OC)C2)=O)CCN(C(c2oc(C)nc2C)=O)CC1CS(C)(=O)=O Cc1nn(CC(=O)NCC(C)(C)CN(C(=O)C(N2CCOC2=O)C)C)c(=O)o1 c1(C(N2C3CN(C(C(C)Br)=O)CC2C3)=O)ccc(I)c([N+](=O)[O-])c1 N(C1CCC(NC(=O)CC(C)(C)O)c2ccccc21)C(CC=C=C)=O c1(C(n2nnc(-c3ccccc3)n2)C(=O)NC)c(F)cccc1F C1(NC(C2(O)CCC(C)CC2)=O)COC2C(NC(C3C4CC5C(C4)C35)=O)COC12 N1(C(C(CC)=CCCC)=O)C(CC(=O)NCCC2CC2C)C2CCCC12 N1(C(C(C)=C2CCCC2)=O)CCCCC(CC(=O)NCC2CC[Si](C)(C)C2)C1 CS(=O)CCC(=O)NCc1cn(CCNC(C2(Cc3ccc(C#N)o3)CC2)=O)nn1 C1(C(=O)Nc2ccc(C(CC)C)cc2)CN(Cc2cncc(Br)c2)CCC1(F)F Cc1ccc(C(=O)NC2(C(N3CCN(C)C(C(=O)N(C)C)C3)=O)CCC2)cc1O C1(CC(=O)NC2CCC(NC(C)(C)C)C2)CCCC2(CC2)C1 CCCC(C)C(=O)N(C(C)(C(N1CCC(C)(CO)C1)=O)C1CC1)C N1(C(c2scc(C(C)=O)c2)=O)CCCC(N(C)C(c2cc(C)c(C)o2)=O)CC1 N1(C(CCC(=O)NCC)=O)CCOCC(NC(=O)Cc2cc(Br)ccc2C)C1 Cc1ccnnc1C(=O)N(CCCCNC(C1COC(C)C1)=O)C N1(C(CCCc2onc(C)n2)=O)CC2CCCC(NC(C34CC(O)C3C4)=O)C2C1 CC1(NC(=O)CC2(C3CC3)CC2)CC(NC(=O)C(O)C2CC2)C1 C1(NC(C2(NC(C)=O)CCC2)=O)CCN(C(c2ccc(CC#N)cc2)=O)CC1F C(C)(C(C)(C)C(=O)NCCOC(=O)C1CC1)NC(CCC(C)OCC)=O Cc1ccccc1C(N1CC(CNC(=O)Cc2ccnnc2O)C1)=O C1(OC)CC(C(c2c(C(N(C3CCOCC3)C)=O)cccc2)c2nn[nH]n2)C1(C)C c1(CC(N2C(C)CC(NC(CCOCCC)=O)C2)=O)c(Cl)cccc1Br C1(C(N2C(CN(C(C3(CNC(C)=O)CC3)=O)C)CCC2)=O)CCCN(C)C1 c1(C(=O)NC(CNC(c2c(C)c(N)cnc2)=O)C)cc2cc(F)cc(F)c2[nH]1 C1(CNC(c2cc(C)[nH]n2)=O)CC2CCC1N2C(c1cc(CO)on1)=O c1(NC(C2CN(Cc3ccccc3)CCO2)=O)ccnc(Sc2ccccc2)n1 N1(C(C2CN(C)C(=O)N2)=O)CCN(C(=O)CCc2cnoc2)CC1c1cn[nH]c1 Cc1cc(C(N2CC3CC3(NC(C3CC(Cl)(Cl)C3)=O)C2)=O)c2c(C)nn(C)c2n1 N1(C(C(CC)CC2CCCC2)=O)CCN(C(=O)Cc2ccnn2C)CC1C(C)C C1(NCC(CCC)NC(=O)OC(C)(C)C)CCCN(C(C)(C)C)C1 c1(OC)nccc(C(N2CCC(C)C(N(C(=O)C3=CCCC3)C)C2)=O)c1Br c1(C(=O)NC2CC(CCNC(=O)CN3CCOC3=O)C2)cnncc1O Cc1nc(N2C(C(N3CCC(O)C(F)C3)=O)CC3CC23)nc2ccc(Br)cc12 C12(CCOCC1)C(=O)NC1CCCC1CNC2=O.CCCOCC1CC1.CC C#CCC(CC(F)F)C(=O)N1CC(CNC(=O)C2=C(C)OCCS2)C1 c1(C(=O)NCC(CC)N(C(=O)CCCS(N)(=O)=O)C)cccc2oc(=N)[nH]c12 CN1CCc2c(C(=O)Nc3nc(C4CCNC4)cs3)cccc21 C1(C(N(C2CCN(C(=O)COC(F)(F)F)CC2)CCOC)=O)CCS(=O)(=O)N1 C12(CC)CN(C(C3CC(C)OC3=O)=O)C(CNC(=O)C(C)(C)CO)(C1)C2 C1(CC(=O)N(C(CO)C2CC2)C)CC2(C1)CN(C(=O)C(C)(C)C1CC1)C2 C(=O)(C1SCCc2sccc21)NC(C(C)C)(C)CNC(c1cnnn1C)=O C1(OC)CC2(C1)CC2NC(C1(CNC(c2cccc(NC(C)C)c2)=O)CC1)=O C12(NC(C(N3CCSCC3)C)=O)CC(NC(=O)CC3CCCO3)(C1)C2 c1(C(=O)NC23C(CN(C(CS(CC)=O)=O)C2)C3)ccc2ncncc2c1 C1(C(N2CCC(C)OCC2)=O)COC2(C1)CN(C(c1ccoc1Cl)=O)C2 C(C1(C)COC1)=CC(=O)NC1(CN(C(=O)Cn2ccc(Br)n2)C)CC1 c1(C(=O)NC(CN(C)C(C2CC3(CC3)CO2)=O)(C)C)ccccc1SCCO c1(C(=O)NCC2(C)N(C(c3nc(C)c(C)s3)=O)CCC2)cccc(F)c1Cl CCCC(C#N)C(=O)NCC1CCN(C(=O)Cn2cnc(Br)c2)C(C)C1 c1(C(=O)NC(C(C(C)C)NC(CCNC(=O)OC)=O)C)cc2c(s1)CCCCC2 c1(C(=O)NCCC(C)CCNC(C2CCC(C#N)CC2)=O)ccc2cncn2c1 C1(C(=O)NCC2(O)CCCN(C(CS(N)(=O)=O)=O)C2)CCCc2ccccc2C1 C1(CC=C)(NC(c2cnc(CCC)s2)=O)CN(C(C2CC2F)=O)C1 Cc1nc(C(N2CCC(O)(CCNC(c3ccns3)=O)C2)=O)c2n1CCCC2 CCC(CC)CCC(=O)N1CC2(C1)CN(C(C1CCCC(=O)O1)=O)C2 C1(C(N2CC(CCC=C)(C(=O)NCCC3(C)CCCC3)C2)=O)CC2CCC1C2 N1(C(C(CC(C)C)OC)=O)CCCN(C(c2cncc(N)c2)=O)C(C(C)C)C1 N1(C(CC2ON=C(CC)C2)=O)CCCC(NC(c2ccc(C(C)(C)C)s2)=O)C1C C(CC(C)C)(C(=O)N1CCC(NC(c2ccc(Cl)s2)=O)C1)NC(C)=O C1(CN(C(c2ccc(COC)o2)=O)C)CN(CC(C)C)CCO1 c1(C(=O)OC(c2c[nH]nc2-c2cnccn2)C(=O)OC)nc(Cl)c(Cl)s1 C(C)(CO)(CC(C)C)NC(c1cc(CNC(c2scc(OC)c2)=O)ncc1)=O Cc1ccc(C(N2CCN(C(c3ncncc3Cl)=O)C3CC23)=O)cc1OC(F)F CC(C)S(=O)(=O)C(C)C(=O)N(C1CN(C(c2ccon2)=O)C1)C c1(C(C)=O)cc(C(=O)NC(C2CCCCC2)CNC(=O)C(C)NC(N)=O)co1 C1(N(C)C(c2cc(=O)cc[nH]2)=O)CCCCN(C(=O)C(CN)c2ccccc2)C1 O=C1CC(NC(c2coc(CNC(=O)CC3CCCCO3)n2)=O)CC(=O)N1 CCC(CO)CCNC(=O)C(C1CCN(C(=O)Cc2ccnn2C)C1)C c1(NC(c2ccc(I)cc2Br)=O)ncnc2ncn(C3CC3)c12 c1(C(CC(=O)NC(CNC(CN(CCOC)C)=O)C(C)C)C)ccc(F)cc1F C#CCC(C)(CC)C(=O)NCC(CCNC(=O)C(n1cc(C)cn1)C)OC C1(CNC(c2c(Cl)cn(C)n2)=O)CN(C(=O)C2=COCCO2)CCC12CCOC2 c1(C(=O)NC2C(NC(CC3C(C)(C)CCC3)=O)CC2)cc(Cl)c2n[nH]cc2c1 N1(C(c2ccc(CCC)s2)=O)CCC2(NC(c3nc(Cl)sc3Cl)=O)CC2C1 C1(CN(C)C(c2ccn(C)c2)=O)CCCN(C(=O)COCC2CCCC2)C1 C1(C)(NC(c2nc(C)n(C)n2)=O)CCN(C(c2ccccc2SCCO)=O)CC1 N1(C(C(CC=C)C)=O)CC2CCCC2(Nc2ccc3nnnn3n2)C1 O=C(CCCCCn1cc(C2CCCCC2)nn1)NC(CNS(C)(=O)=O)C(=O)O C1(C)(CC)CCCN(C(=O)C(CCC2CC2)NC(c2ccc(CO)cc2)=O)CC1 N1(C(C2CC(N(C)CC)C2)=O)CC(C(N2CCC(CN=[N+]=[N-])C2)=O)C2(CC2)C1 C(CC1=CCCCC1)CNC(CCCC=C)c1nnnn1C CC1CC(C(N2CC(C)(C)CC2CNC(=O)C#CC(=O)N(C)C)=O)CC(C)O1 C(c1ccc(F)cc1)=C(C)C(=O)N1CCC1CNC(=O)C1=CCC1 S(=O)(=O)(c1cccc(Cl)c1)N1CC(NC(=O)Nc2cc(F)cnc2Br)C(O)CC1 c1(C(N2CCCN(C(C(CCC)(C)CC)=O)CC2)=O)cnc2c(c1)CCCC2 c1(C(N2CCCC(OC)CC2)C(=O)NCC(=C)C)cc2n(n1)CCCCO2 C12(CNC(=O)CCC3CCCC3)CC(C1)C(NC(=O)Cc1cnns1)CO2 C(=O)(CC(C)(C(F)F)N(C)C)N(C1CCN(C(CC(CC)C(F)F)=O)CC1)C C=C(Cl)C(C)(C)C(=O)N1CCCN(C(c2c(OC)ccnc2OC)=O)CC1 CC1CCCC1CC(N1CC(c2ocnc2CNC(=O)COCCO)C1)=O S(=O)(=O)(c1cccc(F)c1)NCC(=O)NCC(CCNC(C1C(OC)CC1)=O)O c1(C(C(=O)NCC2CCCN2C(c2cn(C)nn2)=O)OC)ccc(O)cc1 c1(OC)c(C(=O)NC2CCC(CO)C2)ncnc1C C#CCC(C(=O)NCCc1cc[nH]n1)NC(c1cnnn1C)=O c1(C(=O)NC2CCCCN(Cc3cn(CC(C)C)nc3)C2)cc(Cl)c(F)cc1F Cc1ccc(Cl)c(C(=O)NCC2(C(F)F)CCN(C(=O)COC(F)F)C2)c1 C=CC1(C2(C(=O)NCC3CN(C)CCN3C(=O)CCC(C)(C)C)CCC2)CCC1 C1(CNC(CC(C)n2ccnc2)=O)CCCN(C(c2cnn(C(C)(C)C)c2)=O)C1 C1(NC(C(CC)OCC)=O)CCC2(CC1)CCN(C(=O)CSCCC#N)C2 C1(NC(c2c(Br)n[nH]c2Br)c2n(CC(=C)C)nnn2)CCn2ncnc2C1 C=CC(C)(CC)C(=O)NC1C2CCN(C(c3ccnn3CC)=O)CC12 c1(CC(C(=O)NC2C(NC(C3(CC=C)CC3)=O)CC2)(C)C)nc2ccccc2[nH]1 c1(-c2scc(CC(N3CC(c4ccccc4)C(O)C3)=O)n2)ccc(O)cc1 n1(CC)nc(C(N2CC(C(C)NC(C3CCC(=O)N3C(C)C)=O)C2)=O)ccc1=O N1(C(CCn2cc(-c3cn(C(C)C)nc3)nn2)=O)C2CCC1CC(CO)C2 c1(C(N(CCC(C)NC(C2(CCC)CC2)=O)C)=O)cn(C2CC2)nc1C CCC(CC)CCCC(=O)NCc1ncc(C(=O)NCC(C2CCCO2)O)cn1 C#CCCCN=c1[nH]c(=NCC(C)(F)C(C)(C)F)[nH]c2cc(OC)ccc12 C(=O)(C(F)C(=O)NCC12CC(C(=O)Nc3cn(C)nc3C(C)C)(C1)C2)OCC c1(OC)cc(CO)ccc1OCC(N1CC(CNC(c2cn[nH]c2)=O)CC1C)=O c1(OC)cnc(Br)cc1CNC(=NCC1CCOC1)NCC(C)(C)F C(C(CC1CC1)C(=O)N1CCC(OCF)C1)NC(COc1ccn(C)n1)=O N(C1CCc2cc(C#N)ccc21)C(N(C)CC1CCC(F)(F)C1)=O C1(c2cccs2)CC(=O)N1.C(CC(=O)NCC(O)CNC(N)=O)NC(COC)=O CC1C(NC(C2(CF)CC2)=O)CCCN1C(c1cc(C(F)(F)F)cnc1O)=O c1(CC)cc(N)ccc1C(=O)NCCC(O)CNC(=O)CC1(CC)CCC1 N1(C(c2ccc(C(C)=O)o2)=O)CCC(CN(C(=O)C(O)CCN(C)C)C)CC1 C=CCCN=C(NCCC1C=CCC1)N1CCc2cc(Br)cc(F)c2C1 N1(C(CC2(C=C)CN(C(=O)C(O)C3CCC3)C2)=O)CCS(=N)(=O)CC1 c1(C(=O)OCC2CCC(C(=O)OCC)CC2)cc(F)c(F)cc1O C(=O)(C1=CS(=O)(=O)CCC1)NC1C(CC)CN(C(=O)C=Cc2cnc(C)s2)CC1 CC1(C)CC(C(C)(C)NC(=O)COc2ccccc2)N(C(C2CC(F)C2)=O)C1 C#CCC(CC(F)(F)F)C(=O)N1CCC(NC(=O)OC(C)(C)C)CC1 C12(C(=O)NC(CC=C)(C)C)CC(CN1C(=O)Cc1csc(C)n1)C2 C1(C(C)NC(CSCCOC)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 C(C(O)CC(=O)N1CC(C(N)=O)(CNC(c2nccnc2N)=O)C1)N(C)C C1(NC(C(C)OCC)=O)CC2CC(C1)N(C(=O)Cc1noc3ccccc13)C2 Cn1cc2c(n1)CCCC2C(=O)N1CC(O)(CCNC(=O)CC2(C)CC2)C1 c1(CN=C(NCc2n(CC)ncn2)NC2CC2C)cc(C)c2ncccc2c1C c1(C(=O)NC2C3CC(NC(CSCC)=O)CC32)ccc(C)c(S(=O)(=O)N(C)C)c1 N1(C(C2CC3(CC3)C2)=O)CCCC(C2CCN(c3nnc(C4CC4)s3)C2)C1 c1(C(C)C)cccc(C(N2CC(CF)(NC(=O)CN3CCCC3=O)C2)=O)n1 Cc1n[nH]c(C)c1CC(=O)NC1CCC(CCNC(c2cn(C)nc2Cl)=O)C1 c1(OC)cc(C=CC(N2CC(O)(CCNC(C3C=CCC3)=O)C2)=O)ccc1O C(=O)(C(C)C(C)O)N1C(CN(C(c2c(C)n[nH]n2)=O)C)CCC1 C1(C(=O)NC2C=CCN(C(c3nccc(Cl)c3Cl)=O)C2)CC2C=CC1C21CC1 N1(C(C2C(CCC)CCC2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)C)C2 C1(C(=O)NCC(C)NC(C(C2CC(F)(F)C2)OCC)=O)CCC(=C2CCC2)CC1 c1(C(N2C3CN(Cc4c(Cl)cccc4I)CC23)=O)cc(F)c([N+](=O)[O-])cc1F c1(C(C(=O)NC(CNC(C(C)Cc2ccccn2)=O)(C)C)=O)ccc(Cl)cc1 N1(C(C(c2c(C)cccc2Br)NC(C2CC2C2CC2)=O)=O)CC(C)(C)C12CCC2 O=C(CCCCNC1CCCC1)NCC1(C2CCCO2)CCOCC1 c1(CNC(=O)NCC23OCCCC2C3(F)F)cccc2c1OCCC2 C1(CNC(c2ccc3cc[nH]c3c2)=O)C(C2CC2)CCN1C(c1ccoc1Cl)=O N1(C(c2c(CCCC)ocn2)=O)CCC(CNC(c2cc(C)c(C)s2)=O)C(O)C1 c1(C(N2CCCC(C)C(C)C2)=O)noc2c1CN(C(=O)C=Cc1ccsc1)CC2 CCCC(C)(C)C(=O)NC(C)C(C(C)C)NC(c1cn(C)c(C)n1)=O C(CCCCC(=O)N1CC2C(N(C)C(c3cc(C)cc(C)c3)=O)C2C1)SC C12(NC(COC(CC)(C)C)=O)COC(C1)C(NC(C1(n3cc(Cl)cn3)CC1)=O)C2 C1(C)(C(=O)NCC(CCC)(C)O)CCCN(C(C)(C)C)S1(=O)=O N1(C(C(CC)OCC)=O)CC2CCCC2(NC(=O)CSc2ccccn2)C1 C1(NC(=O)CCCc2cccs2)(CF)CCN(C(C23CC2C3)=O)C1 CC#CCCC(=O)N1CCOC(CC(=O)NCC2CC2C2CC2)C1 N1(C(c2cnn(CC)c2C)C(=O)NCCOCCOC)C2CCC1CN(C)CC2 c1(CC)cccnc1C(=O)NC(C)(CNC(=O)C(C)NC(=O)CC(F)(F)F)CO c1(C(=O)NCC2(F)CC(NC(c3c(C)coc3C)=O)C2)ncn2c1CCCCC2 c1(C(=O)NCC(N(C(c2c(C)ccs2)=O)C)C2CC2)cccc(C2CCOC2)c1 C(=O)(C#CC1(C)CCCO1)N1CCC(C=C)(C(=O)N(CC(O)CCC)C)C1 c1(SC2(C(=O)NCC(C(C)C)NC(c3noc(CO)n3)=O)CC2)ccccc1F N1(C(C(C)SC(F)(F)F)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)CC1CCO c1(CC)n[nH]cc1C(=O)NCC1(CCNC(c2cc(C(F)F)cs2)=O)CC1 N(C=CC(=O)C(F)(F)F)C(C12C(CN(C(c3cc4ccoc4cn3)=O)C1)C2)=O C(CN=c1ccc(Br)c(S(=O)(=O)NC(C)C(C)(OCC=O)CC)[nH]1)C(C)C.CCS CCCCC(CCC)N=c1nc2c(ncn2C)c(NCC(C(C)C)N2CCCC2)[nH]1 C(C)(CO)(C(=O)NCC(C(C)(C)C)NC(=O)CCc1cc[nH]n1)OC C1(NC(=O)C=C2CCCCC2)CN(C(=O)CCCc2ccccc2)CCC1O C1(NC(c2cc(SC)c(C)o2)=O)CN(C(c2coc(C)n2)=O)CC12CCOCC2 c1(C(=O)NCC(C)NC(=O)CCCn2ccnn2)c(C(C)(C)C)sc2c1CCC2 C1(C(=O)NC2(C)CN(C(C(Cc3c(C)nc[nH]3)O)=O)C2)CCc2n[nH]c(C)c2C1 N1(C(=O)CC=C(Cl)Cl)CC2(C1)CN(C(C1CCOC3(CCC3)C1)=O)CC2CO N1(S(CC=C)(=O)=O)CC2OCCN(C(=O)Cc3ccc(OC)cc3Br)C2C1 CCC(C)C(C(=O)NC(C)C(C)F)N(C(=O)Cc1cc(C)on1)C c1(CC)cc(OC)ccc1C(=O)NCC(C)CNC(c1cnoc1CC(C)C)=O N1(C(c2cnc(OC)c(Cl)c2)=O)CCOCC(F)(CNC(c2cnco2)=O)C1 C1(C(=O)OCC)CN(c2ccnc(N3CCCC3)n2)CC1N(C)C C#CCC(C)C(=O)NC1COCC1NC(=O)COc1ccc(CC(=O)NC)cc1 c1(C(N2C(C)CN(C(=O)C3=CCCC3(C)C)CC2)=O)cc(=O)c2ccccc2[nH]1 C(C(CNC(C1(C#N)CCC1)=O)CO)NC(C1CC(C)C1)=O c1(C2C(C(=O)NCC(C)NC(CCCc3onc(C)n3)=O)C2)cccc(F)c1F C1(NC(c2cc(C(C)C)sc2)=O)CC12CCN(C(=O)C=Cc1cccnc1)CC2 c1(CNC(CN(C(CC(C=C)C)=O)C2CC2)=O)ccc(CC)cc1O C1(CNC(c2cc(C)sc2)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC1O CN1C(=O)CSC1=CC(=O)NC1CCCN(C(c2cccc(Cl)n2)=O)C1C C1(C(=O)NCC2C(CNC(c3c[nH]cc3C3CC3)=O)C2)CC1C1CCCC1 N1(C(c2cc(C)oc2)=O)CCOCC(NC(c2ccc(F)c(O)c2)=O)C1 N1(c2c(C)c(NCC3CCCC3C)ncn2)CCCC2(CC1)CCN(C)CC2 N=C1NC(=O)C(CC(N2CC3CC2C3NC(c2ccc(SC(F)(F)F)o2)=O)=O)S1 C1(C(N2CC(C)(NC(=O)C=Cc3ncc[nH]3)C2)=O)(COC)C=CCC1 c1(CN(C)C(C2C(CNC(=O)C(O)Cn3cncn3)C2(C)C)=O)cccc(O)n1 Cc1nn(-c2ccccc2Cl)c2ncc(C(N3CCC4CCC(C3)N4C)=O)cc12 Cc1ccc(C(O)C(=O)N(C)CC2COCCN2C(=O)C#CC2CC2)cc1 C12(NC(c3scc(C(N)=O)c3)=O)CCN(C(c3cnc(Cl)[nH]3)=O)CC1C2 C1(C(=O)NC(CC#C)CC)CCC(C)(C)N(C(=O)C(CC)C(=O)OCC)C1 CCCC(C(=O)NC1CCCCC1CNC(c1nnn(C)n1)=O)N(C)C CCCC(C)(C)CC(=O)N1CCN(C(c2cc(COC)[nH]n2)=O)C(CCOC)C1 C(=O)(CCCCN=[N+]=[N-])NCCC(C(=O)NCC1CCC(C)CC1)OC c1(NC(C2CSCCN2C(c2cnccc2Cl)=O)=O)ccc(Br)nc1F N1(C(C(C=C)O)=O)CC2(CCN(C(c3cnc(C)nc3C3CC3)=O)CC2)C1 N1(C(c2c(C)oc(C(C)C)n2)=O)CC(NC(C2CCCSC2)=O)C2CCCCC12 N1(C(CCN(C(c2c(C)cnnc2)=O)C2CC2)=O)CCOC(C)(C2CC2)C1 C1(NC(=O)Nc2ccnn2C(F)(F)F)CCOC2(CCS(=O)(=O)C2)C1 C1(C(=O)Nc2cnn(C3COC3)c2)(CC)CCN(C(C2CCC3(CC3)C2)=O)C1 c1(CCNC(=O)C(=O)NC2CCCC2n2ccnn2)cc(O)nc(C2CC2)n1 c1(-c2cn(CC3CN(C(C(CC)CC)=O)C3)nn2)cc(=O)n(C)c(=O)n1C C1(CNC(C(N2CC(C)C2)C)=O)CN(C)CCN1C(c1ccc(C2CC2)cc1)=O c1(C(=O)Nc2ccsc2)cc2n(n1)CCCN(C(C1(F)CCCC=C1F)=O)C2 C=C(C)CC(C)C(=O)Nc1cccc(NC(C2CC(F)C(=O)N2)=O)c1 Cc1cc(C(=O)NCC2(CNC(=O)C(C)(C)N(S(C)(=O)=O)C)CC2)ncc1Cl N1(C(c2c(OC)c(OC)cc(Cl)c2)=O)CCC2C1CCCN2Cc1ccccc1 N1(C(CCC=C)=O)CCCOC(CNC(c2occc2C(=O)OC)=O)C1 C1(C)(CC)C=C(C(=O)N2CCCC2CNC(C2CC3CCC3C2)=O)C1 C1(CC=C)(NC(=O)C(C2CCOC2)OCC)CCN(C(=O)CCC2CCOC2)C1 CC1CN(C(=O)COCCC2CCOC2=O)CC(C(=O)NCC(C)(C)C)O1 c1(C(N2CC(CNC(C3C(OC)C3)=O)OCC2)=O)ccn2cncc2c1 Cc1ccc(CC(=O)NCC2CN(C(C3CC3c3cncn3C)=O)C2)cc1[N+](=O)[O-] N1(CCC)CCCC(O)(C(N2CCCC2C(=O)OC)=O)CC1 N(C1CCCc2ccoc21)C(C(CCC#C)NC(=O)C(C(C)C)C(C)C)=O C12(CNC(C(CC)N(CC)CC)=O)CCC(CC1)N2C(c1cc(F)ccc1C)=O C1(NC(N(CC)CC2CCC(=O)N2)=O)CCC(C)(NC(=O)C(C)SC)CC1 Cc1cccc(N)c1C(=O)NC1CC(F)CN(C(C2CC2C(F)(F)F)=O)C1 C(CN=c1[nH]c(Cl)nc2c1COCC2)N(C(=O)C(F)CC1CC1)CC(F)(F)F c1(-n2c(COCCC)nc(-c3nc(C(F)(F)F)cs3)n2)ccc2[nH]ncc2c1 C(C)(C)(CCC(=O)NCCCCCCNC(=O)C(c1cnn(C)c1)O)OC C(=O)(C(F)(F)CC(C)C)N1CC(CNC(CC(=O)NCC)=O)C(C)(C)C1 C1(CN=c2[nH]nc(CO)s2)(NC(c2cc(CCC)oc2C)=O)CCCCC1C C1(=O)n2c(nnc2C(F)(F)F)N1.N1(C(CSCC(N)=O)=O)CCCCC1 C1(C(N(CC=C)Cc2ccccc2)=O)CN(C(=O)C(F)C(CC)CC)CC(C)(C)C1 C(=O)(C1=CS(=O)(=O)CCC1)NCC1(CNC(C=CSC)=O)CCOCC1 CC1CCC(C(=O)NCC2CC(F)CN2C(c2coc(Br)c2)=O)CC1 c1(C(=O)NC(C)CCNC(=O)CCOC2CCOCC2)csc(S(N)(=O)=O)c1 CCC(CC(=O)NC1(C(=O)NCc2nn(C)c(=O)o2)CCCCC1)CC(C)C c1(CC(=O)NCC(C)(C)NC(CSCC)=O)ccc2c(cnn2C)c1 c1(CNC(CC=C=C)c2nnnn2CCOCC2CC2)csc(=NC)[nH]1 C1(N(C(c2c(C)n(C3CC3)cc2)=O)C)CCN(C(C2(F)CCOC2)=O)CC12CC2 C1(NC(c2nccc(CC)c2)=O)CCCN(C(C2CC(C(C)=O)C2(C)C)=O)CC1 c1(SC)cccc(NC(=O)C(=O)NC(C2CN(NC(=O)OC(C)(C)C)C2)C)c1 c1(NC(C2N(C(C(CN)N)=O)C3C(C2)C3)=O)ncccc1C(F)F N1(C(c2cnc(S)[nH]2)=O)CC2CC(C1)CN(C(c1nccc3ccncc13)=O)C2 c1(C(=O)NC2C(C)(C)N(C(c3cc(Cl)ccc3F)=O)CC2)occ2c1CCOC2 C1(CCCC(=O)NCCC(=C)CNC(=O)CS(=O)(=O)N(C)C)CCC(C)C1(C)C c1(CC)cc(C)ccc1C(=O)NCC1C2CN(C(c3cc(O)ccc3Cl)=O)CC12 C1(CC)CCN(C(=O)Cc2cc[nH]n2)C1C(N1CCC(OCC(N)=O)C1)=O C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC(C)NC(C1(C(F)F)CCCCC1)=O C1(NC(c2ncc(C)c(Cl)c2)=O)CC2CCC(C1F)N2C(c1cccc[n+]1[O-])=O c1(C(N2CCCCC(NC(C)=O)C2)=O)cc(F)cc(F)c1C1CCCC1 O=C(C#CC1CCCC1)NCc1cccc(NC(c2ccsn2)=O)c1 CCC(O)C(C)(C)C(=O)N1CCN(C2CN(C(=O)CCCN=[N+]=[N-])C2)CC1 c1(C(=O)NCCN(C(C(C)OC(C)(C)C)=O)C)nc(Cl)ccc1OCC.C C1(NC(CS(CC)=O)=O)CC2CN(C(=O)C(O)C(C)(C)CC)CC2C1 N1(C(c2c(C)oc(C)c2C)=O)CCN(C(c2cncs2)=O)C2(CC2)C1 C1(CN(C(=O)Cc2cccs2)C)C2CN(C(=O)C(C3CC3)C3CC3)CC12 CC1CN(C(=O)CC(C2CC2)C2CC2)CCC1NC(c1cc(Cl)ccc1F)=O C1(C(N2CC(CNC(C(C)(C)SC)=O)C(C(F)F)C2)=O)CCCC2(CCC2)C1 C(=O)(C(C)CC(F)F)N(CCC)CCNC(C1(CS(N)(=O)=O)COC1)=O N1(C(CONC(C2C(C)CCO2)=O)=O)CCSCC1CO C(=O)(CCC(O)C(C)(C)C)NC1(C2CN(C(C3(C)CCN(C)C3=O)=O)C2)CC1 c1(CNC(=O)C(c2ccc3n[nH]cc3c2)=O)ccc2cc[nH]c2c1 C1(C(N(C)Cc2ccc(CC)o2)=O)CC12CC(NC(=O)Cc1ccsc1C)C2 C12(CNC(=O)C3=CCCOCC3)COCCN1CCN(C(c1cc(Cl)cs1)=O)C2 C1(CNC(=O)NC2CC(NCc3ccccc3)C2)CN(CC(F)(F)F)CCO1 c1(C(=O)NC(CCN(C(c2c(SC)cccc2)=O)C)C)cc[nH]c2nccc1-2 Cn1cc(C#N)cc1C(=O)NC(C(=O)NCCn1ncccc1=O)C(C)(C)C Cc1ccc(Br)c(NC(C2CC23CN(C(=O)Cn2cc(Br)cn2)C3)=O)n1 c1(OCC(C(=O)N(C)CCOCC)NC(C(CCC)C)=O)cc(C)cc(C)c1 c1(CNC(=O)NC2(n3cnnn3)CCOCC2)ccnc(-c2ccccn2)n1 O(NC(=O)C(C)(C)CC(F)F)C(CC(C)C)C(N1CCC2(CN(C)C2)C1)=O C(=O)(C1=CC2CC(C1)CC2O)NC12CC(CNC(C3C(CCC)C3)=O)(OCC1)C2 N1(C(CC=CCC)=O)CC(C2CCCN(C(c3c(Br)cc(Br)c(O)c3Br)=O)C2)C1 c1(C(=O)NC(C2CN(C(=O)C(C(C)O)N(C)C)C2)C)ccc2ccsc2c1 c1(C2(NC(C=CC=CCC)=O)CCC2)cn(Cc2ccno2)nn1 C1(CNC(c2cc(C3CC3)[nH]n2)=O)C2CN(C(c3sccc3F)=O)CC12 Cc1nc2c(F)cccc2cc1C(=O)NCCN(C(c1ccon1)=O)CC1CC1 c1(N(C)C(c2ccnn2C)=O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 c1(C(=O)NCC(CC=C)NC(c2csc(C(C)(C)C)c2)=O)c(C)coc1C CCCN=C(NCc1ccsc1S(C)(=O)=O)N1CCC(C(=O)OC)(CC)C1 c1(C(=O)NCC(CN(C(CCCOC)=O)C)C)cnc(C)nc1 C1(CNC(C2CC(O)C2)=O)CCC2(CCN(C(C3CCCCC3)=O)CC2)O1 c1(C(C(=O)NCCOCCNC(CC2CCN(C)C2)=O)(C)C)ccccc1Cl C1(NC(C(F)=CC)=O)CN(C(=O)CC2CCCC2(F)F)CCC12CCOCC2 CC(C)CC(CNC(=O)OC(C)(C)C)C(=O)NC(C)CNC(C1CC1OC)=O C1(CNC(C(C)(C)n2cnnn2)=O)CC2(CC2)CN1C(=O)COC1CCCOC1 N1(C(C(C)N2CCC2)=O)CCC(NC(c2occc2CN2CCOCC2)=O)C1C C(=O)(CCC(=O)c1cc(C)sc1C)N1CC(O)(CCNC(CCNC(C)=O)=O)C1 N1(C(c2c(CC)ccs2)=O)CCN(C(C2CCCS2(=O)=O)=O)C(C(C)C)C1 c1(C(N2C(CCNC(c3c(CC)n(C)nc3)=O)CCCC2)=O)ccc(O)c(Cl)n1 c1(CCN=C(NC(C=C)C)NC2CC23CC(C)(C)C3)cccc2cc[nH]c12 CC(C)CCCCC(=O)NC1CCCC(NC(=O)CS(=O)(=O)C2CC2)CC1 c1(C(=O)NC2CCN(C(COC)=O)C2(C)C)cc(CC)c2n[nH]cc2c1 Cc1cc(C(=O)NC2C3CCC2N(C(C2CC4(CC4)CO2)=O)C3)ncc1N C(=O)(C#CC(C)(C)CNC(C1CC12CCC2)=O)NCc1c(OC)cccn1 c1(CNC2CN(C(CC(C)O)=O)CC23CC3)n[nH]c2ccc(Br)cc12 Cc1nc(NCC2COC(C)(C)C2)ccc1S(=O)(=O)N1CCOCC1 C(=O)(C(=O)CC(C)C)N1CCC(CC=C)(C(N2CC(O)(C(N)=O)C2)=O)C1 C=CC(CC)CC(=O)N(C1CCCN(C(=O)C=Cc2ccncc2C)CC1)C N1(C(C(C)NC(=O)NC)=O)CCC2C(C1)CN2C(=O)Cc1c(C)nn(C)c1Cl Cc1c(C(N2CCCC(C)C2CNC(=O)Cc2cn[nH]c2)=O)sc2ccccc12 N1(C(CC2CCC(=O)NC2)=O)CCCCC(NC(=O)Cc2cc(F)ccc2Cl)C1 c1(OCCC(=O)NCC(C)CNC(C2CCC3(CC3)C2)=O)ccc(Cl)cc1Cl N1(CC)CC(NC(=O)C(C2CCN(C(=O)CCC3OCCO3)C2)C)C(C)C1 C1(NC(C2C(C(C)(C)C)C2)=O)CC2CCC1CC2NC(C1CCCCO1)=O C#CCCN=C(NCc1cc(F)ccc1Cl)NCC1CC1CF C1(C#N)(C(=O)NC(C)CN(C)C(C2CC(C)(C(C)(C)C)C2)=O)CC=CC1 N1(C(C=C(C)C(C)C)=O)CCC2CN(C(C3(C)C=CCC3)=O)CCC12 C(=O)(C1=CC2(CCN(C(c3nc[nH]n3)=O)C2)C1)NCCC(CCC)C1CC1 C1(NCC(=O)N(CCCNC(CC(C)n2cccn2)=O)C2CC2)CCS(=O)(=O)C1 CC1=C(C(=O)NC(CNC(C2CCS2(=O)=O)=O)C2CC2)CC1 C=CCC(C)(C)CC(=O)NC1COCCC1NC(C1CN(S(N)(=O)=O)C1)=O C1(C(=O)NC(CNC(c2ncc[nH]2)=O)C2CC2)(OC)CCOCC1 N1(C(C(C=C)(C)C)=O)CC2CC(C1)CN(C(C1CNC(=O)CC1C)=O)C2 CCCCC(O)C(C)C(=O)N1CC(O)CC1CNC(=O)C=CCOCCOC C1(NC(c2ncn3c2CCC3)=O)CC(O)CN(C(c2csc(C(F)F)n2)=O)C1 c1(CCC(=O)NC(CC)CNC(C2(CCOC)CC2)=O)ccc2ncsc2c1 c1(CC(=O)NCC2CCCN2c2ncnc3[nH]ccc23)c(F)ccc(F)c1O C=CCCC(C(=O)NCC=CCCC)NC(c1ccc(OC)nc1)=O n1(CC)nc(C(N2CC(F)CC2CNC(c2cnsc2C)=O)=O)c(Br)n1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC1CC(NC(C2(F)CCOC2)=O)C1 C(c1cncc(O)c1)=CC(N1CC(NC(C2(Cl)C(C)(C)C2)=O)C(O)C1)=O N(C(=NCCC(C)=O)NCc1c[nH]nc1-c1cccs1)C1CC(OC)C12CCC2 C1(C(=O)NC(C(C)C)CCNC(C2CCC(=O)N2C)=O)CCc2ncncc2C1 c1(C(=O)NC(CN(C(=O)Cc2ccnc(OC)c2)CC)C)ccc(C)c(C)c1Cl CC(CCCNC(c1cn(-c2cccnc2)nn1)=O)NC(c1ccsc1Br)=O Cc1ccc(CNC(=O)C(CC(C)C)ONC(=O)CCC2CCC2)c(C)c1 C12CCN(C3(CC3)C1)C(=O)O2.C(C(CO)OC(=O)OC(C)(C)C)OC CC1COCCC1C(=O)NCC1CC1CNC(c1cnn(-c2ccccc2)c1)=O C1(NC(CN(C(C2CC2CN(C)C)=O)CC)=O)CCC(CC(N)=O)CC1 Cc1cc(C#N)cnc1C(=O)NC1CS(=O)(=O)CC1NC(c1ccc(Cl)o1)=O Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(=O)C=Cc2cccc(Cl)c2)C1)=O C(=O)(C(C)(C)CNC(C)=O)NCC1CC(NC(C(C)(C2CC2)OCC)=O)C1.C(C)=O c1(NC(=O)NC2C(C(C)C)(CC)C2)ccnc(C#N)n1 C=CC1CN(C(c2cccc(Cl)c2O)=O)CC1NC(=O)C(C)(C)C(F)F CCC(C)C(C)C(=O)N(C1CCN(C(=O)C=CSC)CC1)CC1CC1 CC(CC(N)=O)C(=O)N(C)CC1CCCC1NC(c1ccc(=O)n(C)n1)=O CC1CCN(C(c2cscc2C#N)=O)CC1CNC(c1cncnc1)=O Cn1nc2c(c1C(=O)NC1CC(C)(NC(c3cnn(C(C)(C)C)c3)=O)C1)CCC2 CC1(C)CCC(CNC(C2(CNC(=O)Cn3cccn3)CCCCC2)=O)C1 C=CCC(F)(F)C(=O)NC1CC2CN(C(=O)CCCOCC=C)CC12 N1(C(C(C)NC(=O)NC)=O)CCC(CNC(c2n[nH]cc2[N+](=O)[O-])=O)(OC)CC1 c1(-c2cccc(C)c2F)cn(CC(F)(F)F)c(=O)nc1O c1(OC(CC)C)ccc(C)c(NC(=O)NCCN2CCOCC2)c1 N1(C(COCCC(C)C)=O)CC(NC(=O)C#CC2CC2)C2(CCC2)C1 C(=O)(C(C(C)(C)C)OC)NCC(=O)NCC(CNC(CC)=O)CO CN1N=C(CC(=O)NCC23CC2CN(C(C2(C(F)F)CCC2)=O)C3)CC1=O c1(C(N2C3CC(CNC(C4(SCC)CC4)=O)C2CC3)=O)cc2occc2n1C C1(C)(CNC(c2ccc(COC)cc2)=O)CN(C(=O)CCSC2CC2)CCO1 C12(NC(c3ncc4n3CCCC4)=O)CCCC1N(C(c1csnc1Cl)=O)CCC2 Cc1cnc(N2CC3C(C(=O)Nc4c(C(F)(F)F)cccc4Cl)C3C2)nc1C C(=O)(CCC(=O)N1CC(OC)CC1CNC(C1CCCO1)=O)NCC N1(C(c2c(OC)nn(C)c2)C(=O)O)CCN(C(=O)C(F)C2CCOC2)CC1 C(=O)(C1=CC2C=CC(C1)C2)NC1(CCCC(=O)Nc2c(C)noc2)CCC1 CC(C(=O)NCCC1CN(C(=O)CC2(C(F)(F)F)CCC2)CCO1)C(F)F C12(C(=O)NCC(C)N(C(C(C)=CC)=O)C)CCC(O1)c1ccccc12 n1(CC)ccc(CC(N2CC(C)C2C(=O)NCCOC2CCCCC2)=O)n1 C(=O)(CC1OCc2ccccc21)N(C(CCNC(c1cn(C(C)C)nn1)=O)C)C C1(C(C(=O)NC2CC(F)(CNC(c3c(C)snc3)=O)C2)O)CCCCCCC1 N1(C(CCc2ccc(C)o2)=O)CCCC(NC(c2ccsn2)=O)C1 C12(CNC(C(CO)OC)=O)CN(C(C3CC3C(=O)OC)=O)CC1CCO2 C1(CN=C(NC2C(C)(OCC)C2)NC2CCOCC2)CCC2(C1)OCCO2 C1(C(N2CC(C)C(NC(=O)Cc3cn[nH]c3)C2)=O)CC(C)(C)OC1(C)C O=C1COc2cc(NCC3CCCC3O)cnc2N1 C=CC(C)CC(=O)N1CC2CC1C2NC(=O)Cc1ccccc1C C1(C(C)NC(CCc2nnc(C)o2)=O)CN(C(=O)CSC(F)F)CCO1 N1(C(C2(N)C(C(C)(C)C)CC2)=O)CC(O)C(C#N)C1 c1(NC(N2CCC3(CC3Nc3ncc(C(F)(F)F)cc3Cl)C2)=O)coc2c1CSC2 C#CC1(C(=O)NC(c2ncc[nH]2)CO)CCN(C(c2ccsc2C#N)=O)CC1 C#Cc1cnc(C(N2CCC(C3CCCN3C(=O)C(F)C(C)C)CC2)=O)c(C)c1 C1(N(C)C(=O)C2CC2)CN(CC2CN3CCN2CC3)CC1(C)C.c1ccc(F)cc1 C1(C(F)(F)F)(C(=O)NC2CCC(C)(CC(C)C)C2)CCCCCC1 c1(NCC(N(C(c2ncn(CC)c2)=O)C)C2CC2)ncnc2c1SCCC2 c1(C(N2CC(F)(CNC(C3CCCOC3)=O)C2)=O)cnc2c(c1)CNC2=O c1(C(N2CCN(C(CCC3(C)CC3)=O)C(C(C)(C)C)C2)=O)cnc2ccnn2c1 C#CC1CN(C(=O)CCSC)CCN1C(C1CC(C2CC2)=NO1)=O c1(C(C)C)nccc(C(=O)NC2CCC(NC(=O)CCc3cccc(F)c3)CC2)n1 CCC(CC(=O)N1CCCC(c2n[nH]c(CNC(=O)CCF)n2)C1)C(C)C S(=O)(=O)(c1cccnc1)N1CC(CC(N2CCCC(N3CCCC3=O)C2)=O)C1 c1(C(N2CC(O)C(F)C2)=O)cc2n(n1)CCCN(C(C1CCCO1)=O)C2 C1(OC)CN(C(c2ns[nH]c2=O)=O)CC1NC(c1cccc(C(F)(F)CF)c1)=O c1(C(=O)NC2(CCNC(C(C)N(CC)CC)=O)CCC2)cccc2ccnn12 CC1CCN(C(=O)Cn2cccc(C)c2=O)CC1NC(C1CC(C2CC2)=NO1)=O C#CCC(CO)NC(=O)CCNC(=O)CCc1cnco1 C1(C(=O)NCCCSCC)CC(O)CCN1C(C12CCCC1C2(F)F)=O N1(C(C2C(CC)CCN2C(=O)C=Cc2ccccn2)=O)CC2CCC(C1)C(=O)O2 c1(COC(c2n[nH]c3c2COC3)=O)cc(O)nc2ccccc12 c1(CNC(C2C(NC(COCCCC)=O)CCCC2)=O)c(OC)ccnc1O C1(CNC(C=CCNC(CNC(C2C(C)C2)=O)=O)=O)CC(=O)N(C)C1 N1(CCN(C(CCCOC)=O)C)CCN(C(C)C(=O)N(C)C(C)C)CC1 C1(C)(C(N(CC(=O)NC2CC(CC(C)(C)C)C2)CCOC)=O)CSC1 c1(N2CCC(N(CCCC)C)C2)nc2c(c(=NCC3CC3C)[nH]1)CCCCCC2 CC(CC(=O)NC1(C(=O)NCc2cccnn2)CCN(C)C1)C(F)F C1(NC(C2CCC(C)O2)=O)C2CC3C(C2)C13C(=O)NC1CC(O)C(F)C1 c1(CCNC(=O)N)ccnc(SCc2ccccc2)n1.C(COC)(C1CC1)OC c1(C(N2CC(NC(C(CCCOC)C)=O)C(C)C2)=O)nccc(Br)c1O c1(C(=O)NCC(C2CCC2)NC(C(C2CC2)OCC)=O)ccn(C)n1 C12(C(=O)NC(CC)(C)CO)CC1CN(C(=O)CC=CC(C)(C)C)C2 Cc1cc(=O)n(C)cc1NC(C1CCC(C)(C)N(C(=O)CCCN(C)C)C1)=O N1(C(c2c(-c3ccc(C(=O)NCC)nc3)ncs2)=O)CC2COCC2C1 c1(NC(C2CC2F)=O)c(SC2CCN(C(=O)Cn3ccnn3)C2)cccc1F S(=O)(=O)(c1ccc(S(=O)(=O)NC(C)(CCO)C(=O)O)cc1)NC C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(C)NC(=O)C(F)C(C)(C)O)C1 N1(C(C2CC(=C)C2)=O)CCC(C)C(NC(=O)C=Cc2ccc(SC)s2)C1 CCC(C)CCC(=O)NCC(C)(CO)NC(=O)CCc1cc(Cl)no1 C=CCCC(C)C(C(=O)NCCCC)N(C)Cc1nc(C)cs1 N1(C(CO)=O)CCC(F)(F)C(C(=O)NCCNS(C)(=O)=O)C1.C=CCCCCS N1(C(c2nc(C(C)C)oc2)=O)CCCC(NC(=O)CCc2cccn2C)C1 c1(C(N2C(C(N(C(C=C)C3CC3)C)=O)C=CC2)=O)cc2ncccc2[nH]1 C1(C(=O)NCC(C(=O)NC(C)CN2CCCC2=O)OC)OCCC1(C)C c1(C(N(CC(CC)NC(=O)C(=O)C(C)(C)C)CC)=O)cccc(C#N)c1F C#CC1(C(=O)NC2CCC(=O)N(CC)C2)CCN(C(=O)CCCn2ccnn2)C1 c1(C(N2CCN(C(C(COC)OC)=O)CC2CCO)=O)cnc2cccc(C)n12 Cc1ccc([N+](=O)[O-])cc1C(N1CC2CC1CC2NC(c1ccco1)=O)=O Cn1nc(C(=O)NCC(O)CCNC(c2cc[nH]c2)=O)c(Cl)c1C(F)(F)F C(C(C)N=c1cc(C)[nH]c(=NCC2(OC)CCC2)[nH]1)c1ccc(OC)cc1 C1(CNC(c2cc(C)n(C(C)C)n2)=O)CCN(C(C2CCCCC2O)=O)C1(C)C C(=O)(C1CCc2nccn21)NC1(CCC(=O)NC(CC=CC)CO)CCC1 C(=O)(C(C)C(O)C(C)C)NC(CC#C)(C)C(=O)NC1CC2C=CC1C2 c1(C(=O)OC)cc(=NC(=O)C2CCN(Cc3cc(Br)c(F)cc3O)CC2O)[nH][nH]1 c1(C(=O)NC(CN(C(C2CC3CC3C2)=O)CC)C)cc(F)c(N)cc1OC c1(CNC(c2cc(Br)ccc2F)CCC(=O)O)cccc(O)c1Br Cc1nc(C2CC2)nc(C)c1C(=O)NC1CN(C(C2CN3CCN2CC3)=O)C1 C1(C)(NC(CCc2c(C)ncs2)=O)CCCN(C(=O)CNC(c2ccco2)=O)C1 N1(C(c2ccc(CNC(c3ccc(CC)o3)=O)o2)=O)CCCC(F)(F)CC1 C#CCCN=C(NCC(C1CC1)OCC(C)C)N1CCC(O)C(C)(C)C1 CC1CCN(CC(=O)N(C)C)CC1NC(=O)Cc1cnns1 C1(CN(C)C(C2CCNC(=O)C2)=O)COCCN1C(=O)C=Cc1cn(C)cn1 C(c1cccc(F)c1F)=CC(=O)NC1CCC(NC(c2c(C)scn2)=O)CC1 c1(C(=O)NCCOCCCN(C)C(c2cn(C)nn2)=O)ccc(Br)cc1 CC1=C(C(=O)NCC2=CCN(C(=O)Cc3ncc(C(F)(F)F)[nH]3)CC2)CCO1 C(=O)(C1=CCCOC1)NCC(C1CCCN(C(CCN(CC)CC)=O)C1)(C)O CC1(C)CCC(C(=O)NC2CC(=O)C(=O)C2)C1.c1(N)ccccc1.C1CC1 C(=O)(CCCN=[N+]=[N-])NCC(c1ccccc1)CNC(C1C(C(C)C)C1)=O N1(C(C(CC)(C)CNC(=O)CC(C)OC)=O)CCCOC(C)(C)C1 C1(NC(CCc2cc(C)on2)=O)CCCOC1C1CCN(C(=O)C(C)(C)F)CC1 CC(C)CCCCC(=O)N1CCCC(O)(CCNC(C2CC3(C2)CC(C)C3)=O)C1 c1(OC)cc(CC(N2CCOC(CNC(=O)C(C)(C)CO)C2)=O)ccc1O C(=O)(C(C)(C)CN(C(=O)CC(=O)N(C)C)C)NCc1n(C(C)C)ccn1 N1(C(NS(=NCC=C)(C)=O)=O)CC(OC(C)(C)C)C2CCCC12 Cc1nc(C(=O)NCC2CCCN2C(c2ncccc2O)=O)n(C)n1 C(=O)(C(C)(CO)NC(c1scnc1Cl)=O)N(C)CC1(C#N)CC1 N1(C(c2c(OCC=C)cccn2)=O)CCCC2CN(C(=O)C(C)(C)CC)CCC12 c1(NC(C)=O)ccc(F)c(C(N2CCCC(C)(NC(=O)Cc3cnsc3)C2)=O)c1 C(=O)(C(O)CC(F)(F)F)NC1(C(N2CC(C3(C)CC3)OCC2)=O)CCC(C)(C)C1 C=CCCC(C)(C)C(=O)NCC(C1CCCCN1C(c1[nH]c(C)nc1C)=O)(C)C N1(C(CC2C(CC)C2(F)F)=O)CC2CC1C2NC(c1n[nH]c(C)c1Br)=O CCC(CCC(F)(F)F)(C(=O)NNC(=O)CCF)c1ccccc1Cl CC(CCCNC(=O)C(C)OCc1ccccc1)NC(c1csc(C2CC2)n1)=O C1(C(=O)NC(C=C)(C)CC)CN(C(C2CC(OC3CC3)C2)=O)CC1F c1(CCNS(N(CC)CC)(=O)=O)c[nH]c2c(Cl)cc(F)cc12 S(=O)(=O)(c1cnn2ccc(=NCCC(F)F)[nH]c12)NC1CC(C=C)C1 c1(-c2cc(C)nn2C)ccc2c(c1)CN(C(=O)C(F)C(F)(F)F)CC2 N1(C(C2N(CC)CC2)=O)CCC(C)(CC(=O)NCC(C2CCC2)OC)C1 c1(C(N2CCC(NCc3c(OC)ccc(F)c3)CC2)=O)c[nH]c2ncc(F)cc12 Cc1ccc(C(N2CCN(C(=O)CSC(C)(C)C)C3CC23)=O)c2c1CCCN2 c1(C(=O)NC2CCN(C(C=C(CC)CC)=O)CC2CC)cc([N+](=O)[O-])ccc1N N1(C(C(C)(C)SC)=O)CCC2CCN(C(C3CCN(OC)CC3)=O)CC2C1 C1(N2CC3C(C(=O)NC)C3C2)CCN(C(C2CCC(=O)N2)=O)CCC1C C#Cc1ccccc1C(N1CCN(C(c2n[nH]c(=N)s2)=O)C(CC#N)C1)=O CC(C)(CNC(c1ccc(C(F)F)o1)=O)CCNC(=O)C=CC1CC1 C(=O)(C(F)(CNC(=O)CC1(CC)CCC1)C(C)C)NCCC(C=C)(C)C C(C(F)F)(C(C)(C)C)NC(CC1C(NC(c2c(CC)nccc2)=O)CCC1)=O C1(CNC(c2cc3ccccn3c2)=O)CCCC2CN(C(c3cncs3)=O)CC12 C1(F)(CNC(C(C2CCC2)OC)=O)CCN(C(=O)CN2CCC(O)CC2)CC1 N1(C(C(C)(C)SC)=O)CCN(CC2CN(C(c3nsnc3O)=O)C2)CC1 N1(C(Cc2ccc(C)o2)=O)CCC2(CC1)CCN(C(C1CN(C)C(=O)N1)=O)CC2 N1(C(CCCCCCC)=O)CCOC2(C1)CN(C(=O)C(C)C(=O)OC)C2 C(C(C(=O)NCCN1C(=O)CNC1=O)C(C)(C)C)NC(c1n(C=C)ncc1)=O c1(C(=O)OCC)cc(C)nnc1NC(C)CN(C(=O)CN1CC(=O)NC1=O)C c1(C(N2CC(C)(CNC(CCCC=C)=O)OCC2)=O)c(C)cc(O)nc1C O=C(CCC(CCl)[N+](=O)[O-])NCC12CC(C3CCCC3)(C1)C2 CC(Cc1cccc(F)c1)N=c1nc(N2CCC(C)(C)C2)c2c([nH]1)CCC(C)C2 CC(O)CC(C)N=c1[nH]c(=NCC2(c3ccc(F)cn3)CC2)[nH]c2c1COC2 Cc1ccc(CC(N2CCC(N(C)C(c3n[nH]cc3Cl)=O)C2)=O)cc1C CS(=O)(=NC(=O)c1ccc(CN2CCOCC2)o1)C1CC(c2nn[nH]n2)C1 Cc1cc(C(N2CC3CCC2CN3C(C2(C)CNC(=O)C2)=O)=O)c(C)nc1C N1(C(c2c(NC)cccc2)=O)C2CCC(C2)C1C(N1CC(n2cnnc2)C1)=O Cc1cc(C(N2CC(N(C)C(c3[nH]cc4c3CCC4)=O)C(F)C2)=O)ccc1Cl Cc1ccc(C(=O)NC(C2CCCN2C(C2CC3C=CC2C3)=O)C)c(C(C)C)n1 C=CCC(CC(=O)NC(C)CC(C)(C)O)NC(C1(C=C)CCCCC1)=O c1(C(CC(=O)NC(c2nccc(=N)[nH]2)C)N)cccc(F)c1 c1(N(CCOCC)C)nnc(C2COCCN2C)n1CC1CCCO1.C1CCOC1 CC(C)CC(C)C(=O)NC(C)(CNC(c1c[nH]cc(Br)c1=O)=O)C1CC1 C1(NC(C(NN(CC)C)=O)=O)CCCC12CCN(C(=O)OC(C)(C)C)C2 C=CC(CC)C(=O)N1CCC(C(=O)N(CC(C)CO)C)(C2CC2)C1 c1(C(N2C(CNC(=O)CC3C(C)C3(F)F)CC(OC)C2)=O)ccc2ccoc2c1 c1(C(CF)NC(N(c2cccc(OCF)c2)C(C)C)=O)ccc2c(c1)OCO2 N1(C(C2(C#C)CN(C(c3ccc(N)cc3)=O)C2)=O)CCOC(C)C1CO N1(C(C(COC)OC)=O)CCC2CN(C(C3CC4CCC3C4)=O)C(C)C12 C(=O)(C1=COCCO1)NC(c1ccccc1C(F)(F)F)C(=O)OC CC(C)C(CCNC(C1(C)CCOCC1)=O)NC(=O)C(C)NC(C)(C)C c1(C(C)NC(C(C)NC=O)=O)nocc1C(=O)NC1CC2CC2C1 c1(OCc2c(C(=O)OC(C)C#N)cccc2)cc(S(C)(=O)=O)co1 n1(C(C)C)nc(C2CC2)cc1NC(=O)CCCN(C)C c12ncccc1S(=O)(=O)NCCCCN2C.C1(Cc2cnn(C)c2)C=CCCC1 N1(C(CN(CCC)C)=O)CC2CCC1C(CNC(=O)Cc1ccccc1F)C2 C1(N(C(c2cnc(SC)s2)=O)C)CCCC(NC(=O)C(C)(C)NC(C)=O)C1 N1(C(C(C)SC)=O)CC2CCC(C(=O)Nc3cncc(C#N)c3)(C2)C1 C1(CNC(C=CC=CCC)=O)COC(CNC(=O)CCC2CC(OC)C2)C1 c1(C(N2CCC(N(C(C3C(CC)C3)=O)CC)C2)=O)ccc(F)cc1SC CC1=CC(C)=NS(=O)(=O)N1CC(=O)NCCCNC(c1cc2n(n1)CCCO2)=O C1(NC(c2c(C)coc2C)=O)CN(C(=O)C(C)c2cc[nH]n2)C2(CCCC2)C1 C1(SC)CN(C(c2cc(OC)n(C)n2)=O)CC1NC(=O)CN1CCCOC1=O N1(C(CC2N(C(C)C)CCC2)=O)CC(NC(c2ccc(Cl)cn2)=O)CCC1C C1(C(N)=O)C2CN(C3(OCCO)CCOCC3)CC12 C=CC(O)C(=O)NC1CCCC1CNC(=O)CC1(O)CCCC1 c1(C(N2CCC(O)CC2)C(=O)NC)cccc2cc(C)oc12.c1(CC=CCBr)cccc(C#N)c1 CCCC(C)CC(=O)N(CCCN(C)C)CCNC(=O)C(c1cccn1C)=O O=C(N=c1ccn(CCOCCCCO)[nH]1)c1ccc(CC(F)(F)F)c(Br)c1 C1(C(C)(C)C)CC2(CCCN(NC(c3ccc(C#N)cc3)C3CCCOC3)C2)C1 Cc1nn(CC(=O)NC2CN(C(C3CCC(C(N)=O)C3)=O)CC2(C)C)c(C)c1Cl C1(CNC(C(C)N(C)C)=O)CN(C(c2n[nH]cc2Cl)=O)C2COCC2O1 N1(C(C2(OC)CCCOC2)=O)Cc2[nH]nc(C(=O)N(C)CCF)c2C1 N1(C(c2c(C)c[nH]c2)=O)CCC2CCN(C(c3cc[nH]c4nccc3-4)=O)C2C1 C1(NC(C2CN(C(c3c(CC)nn(C)c3)=O)CC2C)=O)C(O)C2CCOC12 C(CCN=c1cc(C)nc(NC(C)CS(N)(=O)=O)[nH]1)n1ncc(C)c1 c1(CNC(C2CSCCN2C(c2cc(Cl)sc2Cl)=O)=O)ncccc1Cl N1(C(C=CCN(CC)CC)=O)Cc2[nH]nc(C(N3CCC(C)C3C)=O)c2C1 N1(C(CCC(C)OC)=O)CCN(C(c2cccnc2)=O)CC1CN(C)C C1(NC(C(C)(C)c2ccns2)=O)CN(C(C2CCC(C)CC2)=O)CCC1CO C1(NC(CCCN(CCCCCC)CCC)=O)C=CCN(C(C2CC23CC3)=O)C1 C1(C(C(=O)NC(CC=C)(C)C)(C)C)CCCN(C(c2c[nH][nH]c2=N)=O)C1 C1(C(=O)Nc2cnccc2C)(NC(CCSCC)=O)CC1(C)C C12(COC)CC(CNC(=O)CC(C)F)(CN1C(c1ccc(C)s1)=O)C2 c1(COC(c2ccc(C)cc2Br)=O)ccc([N+](=O)[O-])cc1Br C1(CC(N2CC(CC(=O)NC(c3ccccc3)C)C2)=O)NC(=O)NC1=O CC1CCN(C(c2cc3occc3[nH]2)=O)C(C(=O)NCC2CCC=CO2)C1 C(CC(C)C(=O)N1CCC(C(=O)N(CCC(N)=O)C)C1C)OC c1(C(N(C)CC2N(C(C(=O)NC(C)C)=O)CCCC2)=O)nc[nH]c2ncnc1-2 N1(C(c2c(C)nncc2)=O)CCC(NC(c2ccnc(F)c2F)=O)C12CCCC2 C(=O)(C(CCC(N)=O)N(C)C)NCC1N(C)CCN(C(CC(C)F)=O)C1 c1(C(N2CC(CCNC(C=CC=CC)=O)C(C)C2)=O)c([N+](=O)[O-])ccc(C)c1C N1(C(c2ccc(C=C)cc2)=O)CCC(NC(=O)C(N2CCCCC2)C)C(C)(C)C1 C1(OCC)(OC)CC(C)(C(N2CCCC(NC(C3(C)CCCO3)=O)C2)=O)C1 C(=O)(C(c1ccccc1)=CC(=O)O)NC1CN(C(c2c(C)n[nH]c2C)=O)CC1F C1(NC(c2c(CC)ocn2)=O)CCN(C(=O)C(C2CCOC2)OC)CC1C N1(C(c2cncc(OC)n2)=O)CCOCC(NC(=O)CC2COCCN2C)C1 C1(COCC)CCCCC1.C1(CC(=O)N)(NC(C2(CCN(C)C)CC2)=O)CCC1 N1(C(C2C(CC(C)C)C2)=O)CC=CC1C(=O)NCC1(O)CN(C)C1 C(=O)(CC1OCCc2ccsc21)NC1C2(CC(NC(CCC(=C)C)=O)C2)C1 c1(OC)c(CC(=O)NCC(C)N(C(=O)COC2CCCOC2)CC)cccc1F C(=O)(CCCC(=O)N1CC(NC(=O)CCn2ccnc2C(C)C)CC1C)NCC c1(CC)cscc1NC(=O)C(C)N(C(=O)COc1ccn(C)n1)C C1(CNC(c2cc(Cl)sc2Cl)=O)C2CCCC1N(C(=O)CC1CC=CC1)C2 c1(OC)ccnc(NC2C3CN(C(c4nnn(C)c4C(F)(F)F)=O)CC23)n1 c1(C(N2C3C(NC(c4c(C)scc4)=O)CC(C3)C2)=O)ccc2c(c1)C(=O)NC2 Cc1sc(Cl)c(C(=O)NC2(CNC(=O)CC3CC(C)C3)CCOC2)c1C Cc1cc(O)c(F)cc1NC(=O)CC1CN(C(c2csc(=N)[nH]2)=O)CCC1C c1(OC)cc(C(N2CCC(C(=O)NCCCOC(C)C)C2)=O)ccc1O c1(NC(C)(C)CNC(=O)C(c2ccccc2)O)nccc(CN2CCCC2)n1 C1(NC(c2c(C)onc2CO)=O)CCC(C)N(C(C2C3CCCCC23)=O)C1 CCC(C)(C)C(C)CC(=O)NCC1CCN1C(=O)CSc1ccc(OC)cc1 c1(C(=O)NCC(C)N(C(C(c2c(C)cccc2)C)=O)C)ccc(F)c2ccsc12 CC1CC(C(=O)N(C)CC2CCCC2(C)C)CN(C(=O)CCc2ncccn2)C1 C1(CNC(C(C=CCCC)O)=O)CC12CCN(C(=O)C=C(C1CC1)C1CC1)CC2 Cc1ccc(C=CC(N2CCCC(NC(=O)C3=CCCOC3)C2)=O)cc1C N1(C(C(C(C)C)c2cn(C)nn2)=O)CCS(=O)(=O)N2CCOCC12 CC1=C(C(=O)NCC2(C)CCN(C(=O)CCc3ccccc3)C2)C(=O)OC1(C)C CCC(C)(O)C(=O)NC1C2CN(C(c3cc(O)cs3)=O)CC12 c1(NCC(=O)N(C2CC2)CC2CN(C(c3c(CC)nns3)=O)C2)ccc(C)cc1 c1(CC)nc2ccc(F)cn2c1C(N1CCCCC1Cc1nn[nH]n1)=O C(CS(N)(=O)=O)N(C(C1CC(C(C)NC(=O)OC(C)(C)C)C1)=O)C c1(CN(CCNC(C(CC)OCC)=O)CC)ccc(C(F)(F)F)cc1 CC#CCC(CO)NC(=O)CN(C(=O)C(C)CC1CC1)C1CCC1 Cc1c(N)ccc(C(N2CC(F)(F)CC2(C)CNC(c2cncn2C)=O)=O)c1Cl c1(C(=O)NC2CN(C(C(CC(C)C)OC)=O)CC2O)cnn2ccc(C)cc12 C(N=C(NC1CC1)N1CC(C)CC(C)C1)C1Cc2c(ccc(OC)c2)O1 CC1(C)CC(OC(c2ccccc2CCC(N)=O)=O)C(=O)N1 C1(NC(CCCc2onc(CC)n2)=O)CCN(CC2CCC(C)O2)C(C)C1 c1(CC(=O)N(C(C)CNC(=O)CNC(=O)CC(C)(C)C)CC)ccc(O)nc1 c1(CC)ccc(O)c(CN2C(C(=O)Nc3cccc(C)c3OC)CC3CC23)c1 Cc1cc(N)ccc1C(=O)NC1COCC1N1CCN(C(=O)CCC2CC2)CC1 c1(OC)nc(C(=O)NCCC2COCCN2C(=O)C(C)CN(C)C)ncc1F c1(NC(c2ccccc2)CSC)nccc(=NCc2ccnc(NC3CC3)c2)[nH]1 C1(NC(C(CC)CCOC)=O)CC2CCC(C1)N2C(=O)C(c1ccccc1)=O c1(OC)cc2[nH]ncc2cc1NCCC(=O)N(C)CCN(C)C CC1CCN(C(=O)Cc2cc(O)no2)C1c1cn(CCO)nn1 c1(OC)cc(C(=O)NCc2nc(CNC(=O)CCC(C)C)cc(O)n2)ccc1C O=C1NC(=O)C(CNC(=O)C(CC2CCOCC2)NC(=O)CC2(O)CCOC2)N1 C1(C)(C(=O)NCC(C)(C)NC(CN(c2ccccc2)C)=O)CCCC(C)(C)C1 CCS(=O)(=O)C=CC(=O)N1CCC(CNC(=O)CC2CCOC2=O)C(C)C1 CCC(CC)CN=c1[nH]c(=NCC2(C)CC3CC3C2)c2cccc(F)c2[nH]1 CCC(CCC(=O)NCC1CC(C)=NO1)NC(=O)CCCOC(C)C C1(CC=C)(NC(=O)CN(C2CCSC2)C)CCCN(c2ncc(OC)c(C)n2)C1 c1(C(C(N2CC3(CC(NC(C(C=C=C)C)=O)C3)C2)=O)C)cccc2ccccc12 C1(NC(c2c(OC)cnnc2)=O)(CO)CCCN(C(=O)CC2=CCCC2)C1 C1(CC(=O)Nc2c(CC)cccc2)CN(C(c2cc(C(C)=O)c[nH]2)=O)CCC1C C(=O)(CC(C)CF)N(CCCNC(=O)C(F)(F)c1csc(C)c1)CC C1(C(=O)NC2C(OC)CN(C(=O)C(C)(C)CN(C)C)C2)CC2CCC1C21CC1 Cc1ccc2c(c1)CCC(C(N1CC(NC(c3ccn4c3CCCC4)=O)C1)=O)O2 c1(C(N2CC(NC(Cc3c(C)noc3C)=O)C2)=O)ccc(F)c(F)c1O Cc1ncc(C(=O)NCC2CC3CCC2N3C(=O)C2=CCCS2)c(C)n1 c1(OC(C)C)nccc(C(=O)NCC(CC2CCCC2)C(=O)OC(C)(C)C)c1F c1(CC(=O)N(CC(CC)NC(C2CCOC2(C)C)=O)C)cn2cc(C)sc2n1 C(=O)(C1=CCCCC1C)NC1CC2CC(NC(c3c[nH]cc(C)c3=O)=O)CC21 C1(C(=O)NCCS(CC)=O)CCCCN1C(=O)Cc1cncnc1 c1(C(=O)NC2CC(NC(C3CCOCC3)=O)C23CCC3)ccc2[nH]ccc2c1 C1(CC(=O)N(C)Cc2nccs2)CCCC(NC(=O)Cc2cccnc2)C1 c1(CC)ccc(C(=O)N(CCCCCCNC(C2(C#N)CCCO2)=O)C)cc1Cl C(=O)(CC(C)(C)C(F)F)N(C1CCCN(C(C2COC(=O)O2)=O)CC1)CC c1(C(CNC(C)C(=O)NCc2ccc(C(F)(F)F)cc2)O)ccc(F)c(Cl)c1 CCCCC(C)(CO)NC(=O)C(CN(C)C)NC(=O)CCN(C)CC C#CCC(C)(CC)C(=O)N1CCC(CNC(c2cccc(F)c2C)=O)C(F)(F)C1 c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(N)=O)oc2c(Cl)cccc2c1C C(C)(C)(CCC(=O)OC)N(C(N(CCC)C)CC)CC C1(OC)CC2CC(C(N3CCC(CCNC(=O)C(F)(F)CN(C)C)CC3)=O)CC12 Cc1ccc(C)c(C(=O)NCC2CC2NC(c2cnc(O)c(F)c2)=O)c1O C(CO)(C(C)(C)C)NC(c1nnnn1CSC1(C)CC1)(COC(C)C)C C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(C2CC2C)=O)C2(CCCC2)C1 Cc1cc(C(=O)NC2CN(C(=O)CSCC(C)C)CC2C)nnc1O N1(C(C(=O)N(CCOC)C)=O)CCCCNCC(F)(F)C1 C1(CC(N2CCCCC2C2CCN(C(C3CCSC3)=O)C2)=O)(COC)CCOCC1 N1(C(c2c(C)nc(Cl)s2)=O)CC2CCN(C(c3ccc(Cl)s3)=O)CC2C1 c1(C(=O)NC(CC)CNC(=O)CC2CCCO2)cc(C)oc1C(F)(F)F S(=O)(=O)(c1cccs1)NC(CCSC)C(=O)Nc1cc(CS(C)(=O)=O)nn1C C(CC(C(=O)N1CCCNCC1)NC(=O)CN)OC N1(C(CCOC)=O)CC2(C1)C(NC(=O)Cn1cccc(C)c1=O)CCS2(=O)=O N1(CC=C)CCN(CCn2cc(C(=O)OC)nn2)C(C)C1=O C1(NC(c2cnc(Cl)cn2)=O)COCCN(C(C2CCS(=O)(=O)CC2)=O)C1 CC1OC2(CO)CC1(C(=O)NCCN(C)C(C1CCCN(CC(F)(F)F)C1)=O)C2 N1(C(C(C)O)=O)CCOCC1CCNC(=O)CSc1ccccn1 c1(C(=O)NCCN(CCC)C(C2CC2C#N)=O)nnn(CC)c1CC c1(C(=O)NC(CC)(CC)C(N)=O)n[nH]c2c1CN(C(=O)C(C(C)C)SC)C2 Cc1c(Cl)cnn1CC(=O)N(CCCNC(=O)Cc1cnc[nH]1)C C1(C2CCN(C(c3cnn(CCO)c3)=O)CC2)(NC(CC(C=C)(C)C)=O)CCC1 C1(NC(=O)NC2CCCC(C(F)(F)F)C2)CCCN(c2ccccc2)C1 C(=O)(C(C)(O)C(F)(F)F)NC1CC(F)(CNC(CC(C)c2ccco2)=O)C1 C(=O)(CCCN=[N+]=[N-])NCCCC(=O)N(C)CC1(O)CCC1 N1(c2n(C)ncc2[N+](=O)[O-])CCC2(CCC2)C(CNC(=O)CC2CCCCC2)C1 c1(CC)cnsc1C(=O)NC1COCC1n1cc(-c2cnc(C(C)(C)C)o2)nn1 c1(C(=O)NCC23OCC(CNC(C4C(=O)NCC4)=O)(C2)C3)cnc2cccnn12 CN1CCN(C)CC(C(N2CCCC2CCNC(C2(C)CCC2)=O)=O)C1 C1(CNC(c2coc(Br)n2)=O)CN(C(=O)COCCc2ccccc2)CCO1 CCC(C(=O)NC1CC1NC(C1CC(O)C1)=O)Oc1ccccc1 c1(C(=O)NCC2(CN(C(C)C(=O)O)CC)CC2)c[nH]nc1-c1ccoc1 Cc1ncc(Cl)c(CN2CC(C(=O)O)C(c3ccccc3)C2)n1 CCS(=O)CC(=O)N(CC(O)CN(C)C(c1cc(Cl)ns1)=O)C N1(C(C(c2cc(C)sc2)(F)F)=O)C2CCC1CN(C(c1cc(O)cc(O)n1)=O)C2 N1(C(C(c2ccc(C)cc2)C)=O)CCC(NC(c2ccc(Br)cc2I)=O)C(F)C1 CCCCC(c1nnnn1CCCSc1cccs1)NCCCn1cc(C)cn1 C1(C(=O)Nc2ccc(F)cc2O)CCC2(CN(Cc3ccc4nc[nH]c4c3)C2)O1 C1(NC(CCCC#C)=O)CC2CCC(C1)N2CC1CCC(C)C1 CC1CCCCN1CCNC(=O)C(C)(C)NC(=O)CC(C)N(C)C C1(c2nn[nH]n2)(CC)CCCN(C(=O)CCCCC(O)c2ccccc2)C1 N1(C(CCCCC=C)=O)CC(CNC(c2cnc(C)[nH]2)=O)CC12CCOCC2 N1(CCC(=O)N(CC(C)(C)NC(C(C2CCOC2)OC)=O)C)CCOCC1=O C1(C(=O)NCCCCC#CC)CN(C(=O)C(CSC)OC)CCC1(C)C c1(C(=O)NC2C(NC(COCC=C)=O)CCC2)cc(F)cc2nc[nH]c12 C(=O)(C1CCc2cccnc21)NC1CCC(NC(C=Cc2c(C)cccn2)=O)C1 CC(C)(F)CN=c1[nH]c2c(c(=NCc3ccc(Br)cc3N)[nH]1)CC(C)CC2 CCC(CC(=O)N1CCN(CC(=O)NCCCC(O)CO)CC1)OC c1(OC)ccc2c(=NCCc3ccoc3)[nH]c(=NCc3[nH]c(C)nc3C)[nH]c2c1 CC1(C)CC(CNC(C2CNC(=O)N2)=O)CN1C(c1coc(C2CCC2)n1)=O C(=O)(C1Cc2ccccc21)NC(C1CC(NC(C2CCNC2=O)=O)C1)C n1(CC(=O)NC2CC(NC(=O)CCC3CCCC(O)C3)C2)ncc2ccccc12 C(=O)(CCC(=O)N1CC(O)(CNC(=O)C(c2ccc(C)cc2)(C)C)C1)OC C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(CC=C)CNC(c1onc(C)c1C)=O C1(CCNC(CN(S(CC)(=O)=O)C)=O)COCCN1C(=O)C(N1CCC(C)C1)=O c1(C(C)C)cc(C(=O)NCC(C)NC(c2ccncc2Cl)=O)cc(F)c1 C1(NC(C=C=C(C)C)=O)CC(F)CN(C(=O)C(F)(F)c2ccccc2)C1 CS(=O)(=O)c1ccc(C(O)CNc2ccc(-c3ccco3)cc2)cc1 C(=O)(C(O)C(C)CC)N(CC(CNC(CCCCC)=O)(C)C)CC C1(N(C)C)CN(C(C2CCC(NC(=O)Cc3ccsc3)CC2)=O)CCC1O C=CCCCC(C(=O)NCC(CC(C)C)N(C)C)NC(=O)C#CC(C)C Cc1cc(N(C2CNCC2C#N)C(=O)Cc2cncnc2)ncn1 c1(C(N2CCCC2C(=O)NC(C)(C)C)C(=O)NC)cc(Cl)cc(Br)c1F c1(CC)cc(COC)cc(S(=O)(=O)N2CCC(Cc3cnc[nH]3)CC2)c1 N1(CC(=O)N(CCCCNC(c2nc(CC)oc2)=O)C)C(C)CCC1C C1(NC(c2c(-c3cn(CC)nc3)n[nH]c2)=O)CCC(CNC(=O)C(C)(F)F)CC1 C(C(CC1CC1)C(=O)NC(C)Cc1nn[nH]n1)NC(CC(=O)OC)=O N1(C(N2C(c3onc(C)n3)CCC2)=O)CC(=O)Nc2cc(C(F)(F)F)ccc21 N1(C(c2c(C)noc2)=O)CCC(N(C(=O)Cc2cc(Cl)n(C)n2)C)C(C)C1 c1(C(=O)NC2CC(NC(C(C)c3ccon3)=O)C2)cc(O)nc2c1CCCN2 c1(CC)ccoc1C(=O)N(C)CCOCCC(=O)NC(c1cnsc1)C C1(NC(Cc2cc(C)on2)=O)COCCC1NC(=O)C(C)c1ccco1 C1(N(C(CCNC(C)=O)=O)C)CC2CCC(C1)N2C(C1C2CC3C(C2=O)C13)=O CCCS(=O)(=O)C(C)C(=O)NCC1CN(C(=O)Cc2nccn2C)C1 N1(C(c2c(CC)cno2)=O)CCC(NC(=O)CN2CCOCC2)C(C)C1 c1(OC)ccc2oc(C)c(C(=O)NC3CN(C(C4CCCCC4)=O)C4CC34)c2c1 C(C(=O)NCC1(O)CN(C(C2(C)CCN(C(C)=O)C2)=O)C1)(C(C)C)SCC c1(NCC2(O)CCN(C(CC(=C)C)=O)CC2)ncnc2sc(C)c(C)c12 c1(COC)c(C(=O)NC2CCCCC2NC(C2(C)CCC23CCC3)=O)cnn1C Cc1cc(C(F)(F)F)ccc1CC(N1CCC(NC(c2n[nH]c(C)c2C)=O)C1)=O c1(C(=O)OC)ccc(C(N2CCC(CC(C3CC3)OC)C2)=O)cn1 c1(C(=O)NC(C)CNC(=O)CCCCO)cncc(N=[N+]=[N-])c1 C1(CNC(c2c(C)sc(O)n2)=O)CN(C(=O)CC=C(Cl)Cl)CC(C(F)(F)F)O1 c1(-c2ccc(C(=O)NC)cc2)ccn2nc(C(=O)NC(CO)CO)cc2c1 n1(CCC(=O)NCC(C)(C)NS(=O)(=O)C2CC2)cc(CCOC)nn1 CCCCC(F)C(=O)N1CCSCC1C(=O)NCC1CCOC1 N1(C(c2n[nH]cc2-c2ccccc2)=O)CC(NC(C2(C(F)F)CCC2)=O)C(F)C1 C#CCCCCCCC(=O)N1CC(NC(c2nc(C)oc2C)=O)C(O)C1 C1(C(=O)NC)CCN(C(C2CN(C(=O)CN3CSCC3=O)CCO2)=O)C1C N1(C(C(C)c2cccs2)=O)CCN(C(C2(F)CCCC2)=O)CC2(C)CCCC12 C(C)(C(C)(C)C(=O)NC1CC(CCC(N)=O)C1)NC(C(C(C)O)N(C)C)=O C1(NC(CCC(C)=O)=O)CC(NC(=O)C=Cc2nnn(C)n2)C12CCC2 c1(-n2cc(CN3CCC(NC(c4nc(Br)cs4)=O)C3)nn2)ccc(F)cc1 C1(CC(=O)NC(C)C(C)NC(c2cnc[nH]c2=N)=O)CCS(=O)(=O)CC1 N1(C(c2cc(CNC(CCCCOC)=O)on2)=O)CC(C)SC(C)C1 c1(C(C)OCC)nc(C)c(C(N2CCC(C)(NC(c3snnc3CC)=O)C2)=O)s1 c1(N2CC(c3nc(C)[nH]n3)OCC2)nc(=NCCC2CC2)[nH]c2cccc(F)c12 N1(C(c2cncc(C)c2C)=O)CCC(NC(C2(F)CC=CC2)=O)C(CO)CC1 O=C(C#CC1CCCC1)NC1CCCCN(C(=O)CCc2nccs2)C1 c1(CC)cc(C(N2CC(CNC(c3ccn(COC)n3)=O)CC2C)=O)ncn1 Cc1cccc(C(N2CCCC2C2(C(=O)NC3CC4C=CC3CC4)CC2)=O)c1O N1(C(C2CCN(CC)CC2)=O)CCC(F)(F)C(C(=O)Nc2ccc(Br)c(C)n2)C1 C1(C(=O)NCc2cc(OC)nnc2OC)CCc2nc(C)nc(C(F)(F)F)c2C1 CCC(CC(=O)NCC1(CC(=O)NCC(C)(C)CO)CC1)SC Cc1nc(N(CCCCN(C(=O)CC(C)(O)C(F)(F)F)C)C)c2scc(C)c2n1 c1(CC(C)NC(C(=O)NCC2C(OCC)C2)=O)c(F)cccc1Cl O=C1CC(NC(C2CC(O)CCN2C(C2C3CCC(F)C23)=O)=O)CC(=O)N1 C1(C(=O)NCC(C(=O)NCC(CC)(C)Cl)C)C2CC3C(C2)C13 c1(COC2CCN(C(=O)NCC3(C)C(OC)CC3OC)C2)cc2ccccn2n1 C(CC(=O)NCC1(C)CC1(F)F)(C(F)(F)F)NC(C(C)(C)SC)=O Cc1nc(N)c(CC(=O)NCC(CNC(=O)CC2CC2(C)C)CO)c(O)n1 c1(CC)cnc(CNC(=O)CC=CCNC(=O)CSCCC#N)o1 N1(C(c2nccc(C)c2)=O)CCC(NC(=O)C(CCS(C)=O)N(C)C)C(C)(C)C1 C1(CNC(C2(CC)CC2)=O)CN(C(=O)C(F)C(F)(F)F)C2COCC2O1 N1(C(CCNC(C)=O)=O)CCN(C2CCN(C(C3(C)CCCN3C)=O)C2)CC1 C1(NC2(c3n(CCCC)nnn3)CC(OC)C2)CCCC(C(C)(C)C)C1 c1(CC(C(=O)N2CCC(OC)C2)NC(COCC)=O)ccccc1Br C1(C2(O)CN(C(=O)C(CC(C)C)n3ccnc3)C2)(CNC(C(C)NC(N)=O)=O)CC1 c1(C(=O)NC2CC3CC2N(C(c2ccsc2Cl)=O)C3)ccc2oc(O)nc2c1 C(=O)(C(C)(C)CC(C)C)N1CC(C)(C(N2C(CCC=C)CCC2)=O)C1 Cc1ccc2scc(CC(=O)N(C(C)CNC(=O)CC3CC=CCC3)C)c2c1 c1(CC(=O)N(CCC(C(C)C)NC(c2cnn(C)c2)=O)C)c(F)cccc1F C1(C(=O)NCC(CC2CN(C(C3CC(C)C3)=O)C2)(C)C)CC(Cc2ccccc2)=NO1 C1(CC(=O)N(CC(C)NC(=O)Cc2ccc(Cl)nc2)C)CCC(C)CC1 CCCC(O)CNC(C1(C(C)NC(=O)CNC(=O)OC)CC1)=O C(=O)(C(C)(C)CCCc1ccc(OC)cc1)OCC1(C(=O)OC)CCOCC1 C(=O)(CCCCCC(=O)NCC(C)NC(C1(C)CC1(F)F)=O)OC C(=O)(CCCCC(C)(C)C)N1CCC(CNC(C(CC)F)=O)C(F)(F)C1 C1(NC(C2C(C(=O)OC)C=C2)=O)CN(C(c2cc(C)cc(O)n2)=O)C2CCCC12 c1(N2CCCC(CC=C)(NC(=O)C(C)OCC)C2)ncnc2[nH]ccc12 c1(C(=O)NCC(CO)NC(c2[nH]c(=NCC)sc2)=O)nccc2occc12 N1(C(C(C)NC(N)=O)=O)CC2CCCC1C2CNC(c1c(Cl)n[nH]c1C1CC1)=O C1(NC2CCN(C(c3ccccc3)C)C2)CCC(Cc2ccccc2)C1 N1(SCCCOC)C(=O)CN(CCc2ccc(Br)s2)C1=O c1(CC(N2CCOCC(NC(CCC(N)=O)=O)C2)=O)c(F)cc(F)cc1F N(C1CN(C(c2ccc3c(c2)CC3)=O)Cc2ccccc21)C(CCOCC#C)=O C1(NC2CC2)CCCCN(C(c2c(OC(F)(F)F)cncc2Br)=O)CC1 Cc1cccc(C(N2CCOC(CN(C(=O)C(C)OCC3CC3)C)C2)=O)c1C C1(C(=O)NC2C(NC(=O)CCOC3COC3)C2)C2CC3C(C2=O)C13 Cn1cc(C(=O)NC2CC(NC(C3CSC3)=O)CC2O)ncc1=O N1(C(c2ccc(Cl)cc2O)=O)CCN(C(C2CCc3nnnn3C2)=O)CC(O)C1 N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ncncc2C)=O)C(CCOC)C1 C1(C(=O)NC2(c3ccccc3)CN(C(C(C)SC)=O)C2)CCS(=O)(=O)C(C)C1 N1(C(c2cc(C)n(C)c2)=O)CC(NC(C2(c3cccc(Cl)c3)CC2)=O)C(C#N)C1 c1(C(=O)NCC(C)(CO)NC(=O)Cc2ccccc2)ccc(F)cc1Br Cn1cnc(C(=O)NCC2(F)CCN(C(c3cc(C(N)=O)ccn3)=O)C2)cc1=O C(=O)(C(C(C)(C)C)n1ccnn1)N1C(CNC(c2cc(C)sn2)=O)CCC1 N1(C(CCCC(=O)OC)=O)CCC2C(CCCN2C(=O)CCC=C(C)C)C1 c1(OCC)ccc(OCCCOC2CCC(C(=O)NC(=O)CC(C)F)CC2)cc1 c1(C(C)NC(=O)NC2CCN(C3CCOCC3)C2)nccc2ccccc12 CC(C)CC(CNC(=O)C(C1(O)CCCC1)F)C(=O)NC(CN(C)C)C(C)C c1(-n2c(C(c3ccc(C)cc3)NCC(C)CO)nnn2)c(C)cccc1C c1(N(C)CC2CCN(C(c3c(C)scc3)=O)C2)ccc(NC)cn1 CC1CCCC=C1C(=O)N(C)CC1CCCN(C(=O)C(F)(F)c2cscn2)C1 C1(C(=O)NC2C(OC)CN(C(c3cccc(CC)c3)=O)C2)(OC)CCCC(C)C1 c1(C(=O)NCCC(=C)CNC(=O)Cc2ccc(Cl)c(F)c2)cc(O)nc(OC)n1 N1(C(c2c(C)snn2)=O)CCOC2(C1)CN(C(=O)CCC1CCCC1)C2 C1(NC(N(CCSC)C)=O)CCCC(F)C1 C1(NC(CN(S(CC)(=O)=O)C)=O)CN(C(C2CC2C(F)(F)F)=O)CC1C N1(C(Cn2ccc(C)n2)=O)CCCC(C)(NC(=O)CSCc2ccccc2C)C1 N1(C(C2C(CCC)C2)=O)CCC(NC(=O)C(=O)N(C)C)C(F)(F)CC1 c1(CC)cn2c(n1)CC(C(N1CCC(CNC(=O)C(F)CC)(OC)CC1)=O)CC2 C1(CC(=O)NCC2C=CCN2C(C2C=CCC2)=O)CCC(F)(F)CC1 N12CCC(C1)C2.c1(C(N(C)CCC2CC2)=O)ncoc1C(F)(F)F CC1(C)C(NC(c2n[nH]cc2F)=O)CC1CNC(=O)CCNS(C)(=O)=O c1(SC)cnn(C)c1C(=O)NC1CC(C)(NC(=O)C(C2CCCCC2)C)C1 c1(Cc2nc(C(C)(C)NC(C)=O)sc2)cccc(S(=O)(=O)C(N)=O)c1 C#CCC(C(=O)NCC(C)(C)C)NC(=O)C(F)OC(F)(F)F C(=O)(C1=NOC2(CCC2)C1)NC1CC(C)CN(C(c2cccn3nncc23)=O)C1 N1(C(=O)OC(C)(C)C)CC(OC(C2C3CCCCC23)=O)CC2CCCCC12 C(=O)(CCCCC(=O)OC)N1CCC(C)(CNC(COCC(=O)NC)=O)C1 CC(CS(C)(=O)=O)C(=O)N1CCCC(C(C)(O)CNC(c2cnc[nH]2)=O)C1 CC1CC2(CC2)CN1C(=O)CC1CCN1C(c1ccc(F)cn1)=O C(CN=c1cc(Cl)c(O)n[nH]1)(c1ccccc1F)NC(C(CCSC)O)=O N1(C(c2onc(C)n2)=O)CCC2(CC2C(=O)NC2(CF)CC2)C1 N(C1CCCn2cnnc21)C(C12N(C(c3cc(CO)on3)=O)CC(CO)(C1)C2)=O c1(C(=O)NCCC2CCN(C(=O)CCC(F)F)C2)ncc(Cl)cc1Cl c1(C(=O)NCC2N(C(C3ON=C(CC)C3)=O)CCC2)noc2cc(F)ccc12 c1(C(=O)NCC(C)N(C(CC(C=C)CCC)=O)C)cc2cccn2c(O)n1 C(=O)(C(O)CCNC(=O)C(C#N)CC)NCCCCCC Cc1ccc2nonc2c1C(=O)NC(C)CCNC(=O)CCCc1n[nH]c(=N)s1 CC(C(=O)N1CCC(C(=O)NC2CCC(=O)N(C(C)C)C2=O)O1)=C1CC1 c1(C(N(CCOC)CCNC(C2C3COCC23)=O)=O)cc(Cl)cnc1OC c1(C(=O)NCC(C)N(C(C(C)CO)=O)C)ccc(-c2ccc(F)cc2)n1C CC1CN2CCN1C(C(=O)NCC1CC(NC(c3sccc3C#N)=O)C(O)C1)C2 C1(C)(CC)NC(=O)N(CC(=O)NCCCNC(c2cccn3nncc23)=O)C1=O CC(C)(CCC#N)C(=O)N1CCCC2(NC(=O)C3=CS(=O)CCC3)CC2C1 C(=O)(C1CCCn2nccc21)NCCCN(C(C(C)Sc1ccccc1)=O)C C1(C(N2CCC(C3N(c4nnn(C)n4)CCC3)C2)=O)CCC(=C(F)F)CC1 c1(N2C(CC)CN(C(c3ncsc3C)=O)CC2)ncnc2c1oc1ccccc21 C#Cc1ccc(C(=O)N(CC(C)O)CCNC(C2(C)CCCS2(=O)=O)=O)cc1Cl C1(N(C(=O)CC2CCN(C(=O)CC3CCCNC3)CC2)C)CCCC(N)C1 c1(CNC(C2(C(C)(F)F)CC2)=O)ccoc1CN(C)C.C12CCN(C1)CC2=O c1(CC(=O)NC(Cn2cc(C3(COCC)CCCO3)nn2)C)ccc(OC)cc1 C1(F)(CNC(C2C(CC)C2)=O)CCCN(C(c2cnc3n2CCS3)=O)CC1 C1(C)(CC)CC(NC(=O)CCNC(C)=O)CN1C(c1ncc(Br)cc1C)=O CC1CC(N(C(=O)CCCN(C)C(c2csc(Cl)c2)=O)C)CC(C)C1 N1(C(c2ncc(OC)nc2)=O)CC(F)(F)CC1CNC(C12CCC(F)(CC1)C2)=O CC(C)(CNC(c1conc1CNC(C1CCCC(=O)CC1)=O)=O)CCCO Cc1cccc(O)c1C(=O)NC(CCCNC(=O)C(C)(F)F)c1ccccc1 Cc1c(F)c(F)c(CN2CC(Cn3cncn3)C2)c(F)c1F N1(C(c2c(C)nncc2)=O)CCC(C2CCN(C(C3(F)CC3C)=O)C2)CC1 c1(C(=O)NC(CNC(C(C)O)=O)CO)cnn(-c2ccccc2)c1F c1(C(N(C2CCN(C(c3nncn3CC)=O)C2)CCC)=O)ncc(Br)cn1 C1(C)(CC(N2C3CC(NC(c4n(C)ncc4)=O)C2CC3)=O)COC(C)(C)CO1 C(=O)(CCC(CC)CCCC)NCCC(=C)CNC(=O)CC(C)n1cccn1 N1(C(C2CN(C(CCC(C)OC)=O)CC(C)O2)=O)CC2NC(=O)OC2C1 c1(CC(=O)NCC(CNC(c2ccnn2C2CCCC2)=O)OCC)cccc(O)c1 N1(C(C(C)CF)=O)CCC(NC(=O)C(O)C2CCCC2)CC1 C(CC(CO)C(C)C)NC(c1cc(CNC(C#CC(C)C)=O)sc1)=O N1(C(C)=O)CCOCC1C(N1CC(C(C)NC(=O)CC2CCC2)C1)=O N(CP(C)(C)=O)(CC(=O)OCC)C(N1CCCC(c2ccn(C)n2)C1)=O C1(C(=O)NC(C(C)(C)C)CNC(c2cscc2C#N)=O)CC2CCC1CC2 C(=O)(NN1CCCC1C(=O)NCC1(C)CCC(=O)N1C)c1c(C)n(C)nn1 c1(C(N2CC(C(C)NC(c3cnc(CC4CC4)s3)=O)C2)=O)ccnnc1Cl C1(N(C(C=C(C)C)=O)C)CC2CCC(C1)N2C(=O)CCc1ccc(O)c(O)c1 C1(c2cn(CC3(O)CCN(C(c4sccc4Br)=O)C3)nn2)(N(C)C)CCCCC1 N1(C(c2cc(C(=O)OC)n(C)n2)C(=O)NC2CCCCC2)CCC2CCN(C)CC12 C(=O)(C1=CCCCO1)NC1CN(C(CCOc2ccc(C(N)=O)cc2)=O)C2C1C2 c1(CC)[nH]c(Cl)nc(=NCC(C(C)(C)C)NC(c2cnn(C)c2Cl)=O)c1C#N c1(CC)noc(CC)c1CC(=O)NC1CC(NC(C23CC(C)(C2)C3)=O)C1 C(=O)(C#CC(C)(C)C)N(C1CCCN(C(c2ccc(NS(C)(=O)=O)nc2)=O)C1)C C1(N)CCc2c[nH]nc2C1.C12(CCOC1)CCC(=O)N2C(=O)C1CC1.CO c1(C(N2CCN(CC(N3CCC(C#C)CC3)=O)CC2)=O)cccc2c1CCC2 C1(CNC(CN(c2ncccn2)C)=O)CN(C(c2cncn2C)=O)C(C)(C)C1 N1(C(c2c(C)nsc2)=O)CC(C(=O)NCC(O)C(C)C)C(F)(F)C1 C(=O)(C1CCCn2c(Br)cnc21)N1CCCN(C(C(C(C)C)(C)O)=O)CC1 c1(OC)ccc2c(c1)CCC2NC(c1nc(Cl)ccc1Cl)c1nnnn1C(C)C c1(C(=O)N(C2CCNCC23CC3)c2ccncc2)ccn2nccc2c1 C(=O)(C1=CC(O)C(NC(=O)C#CC2(C)COC2)C1)NC(c1cnn[nH]1)C N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)CC2CCC(C3CC3)O2)CC1CCO CCC(CC(=O)NCC1CN(C(=O)C(C)CC2CCC2)C2(CCC2)C1)CC(C)C CCCC(CNC(c1cc(OC)cnn1)=O)C(=O)N(CCO)CCOC CC1(C)C2CN(C(c3cc(O)nc(O)n3)=O)C(C(=O)Nc3cc(Br)cc(I)c3)C12 C1(NC(C=CC)=O)CCN(C(c2cc(CCO)on2)=O)C1C1CC1 C1(O)(CCNC(C(C)CC2CCCO2)=O)CCN(C(c2ccoc2Cl)=O)CC1 Cn1ncc(C(=O)NC(C(=O)NC2CCN(C(N)=O)C2)C2CCC2)n1 C#CC1CN(C(C2CCS(=O)(=O)CC2)=O)CCN1C(=O)C(COC)N(C)C c1(C(N2CCC(CCN(C(CCOCC)=O)C)CC2)=O)nc(O)nc(O)c1N c1(NC(=O)CC2CN(Cc3ccc(O)c(F)c3)CCO2)nccc(Cl)c1I c1(NC(C2CCCN2Cc2ccc(Oc3ccccc3)s2)=O)ccnc(Cl)c1F c1(CC(N2C(CNC(C3(CSCC)CC3)=O)CCC2)=O)cnn(C)c1C C1(C(=O)NCc2n(C)ccc2)CCC(NCC2CCC(O)CC2)CC1 c1(NC(c2n(CCCSCC)nnn2)C2CCCSC2)ccc(C(N)=O)cc1 C(=O)(C1Cc2ccc(Cl)cc21)NCC1C2CN(C(c3c(C)n(C)nc3)=O)C1C2 CC(C)(C(=O)N1CCC(CNC(=O)CCc2ccccc2Cl)C(O)C1)C(F)(F)F N1(C(c2ccn(CC(F)F)c(=O)c2)=O)CCc2nc[nH]c2C1c1ccc(Br)cc1 N1(C(C(C(C)C)(C)C)=O)C(CNC(c2ncoc2C(F)(F)F)=O)CC2COCC12 c1(C(=O)NC(C)(C)CCCNC(=O)CCCn2ccnc2)cccn2ccnc12 N1(C(c2c(C)n(C3CCOC3)nn2)=O)C2CCC1CN(C(=O)CC1(C)CC1)C2 C1(C)(C(=O)NCC(CC(C)C)OC)CC(O)CN1C(C12CSCC1C2)=O C1(C(=O)NCC(C)CCCO)CCCN1NC(=O)C1(C#N)CCCC1 C1(C(=O)NC(CCCCC)C)COCCN(C(=O)C2=CCCC2C)C1 N1(C(C(=O)NCCOC)CC2CCC3CC23)CCN(Cc2ccc(Cl)cc2)CC1 c1(SC)nn(C)cc1C(=O)NC1CCCC1NC(=O)CCC(=O)C1CC1 C1(NC(c2onc(CC)n2)=O)CN(C(=O)CCc2cncc(C)c2)CCC1C Cc1cc(C(=O)NC(C)(CO)C(=O)N2CC(F)(C#N)C2)oc1C N1(C(C(c2n(C)ccn2)(F)F)=O)CCOC(CCNC(=O)CCn2cnnn2)C1 C(=O)(CCCOC(C)(C)C)NCC1(CNC(C(C2CCCOC2)OC)=O)CCC1 c1(OC)cncc(C(=O)NC2CCC(CNC(C3CC4CCC3O4)=O)C2)c1 C1(C(=O)NCC2CCC(F)(CNC(C3C(=C)CC3)=O)CC2)CC2(CC(C)=NO2)C1 C1(CCNC(C2(C(F)F)CCCO2)=O)CCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 c1(CCCC(=O)NC2CN(C(=O)C3=CCCS3)CCC2F)c[nH]c2ccccc12 N1(C(C(CC)CCOC)=O)CCCC2(C1)CN(C(c1cccc(O)c1)=O)C2 N1(C(CC(CNC(C(N2CCOC2=O)C)=O)C)=O)CCOc2ccccc21 c1(C(=O)NC2(CC=C)CCCN(C(=O)C(O)C=CC)C2)cc(Cl)ccc1[N+](=O)[O-] C=CC1CN(C(c2cnn(C(C)(C)C)c2C)=O)CC1NC(c1cncs1)=O C1(CCNC(=O)C=NOC)(NC(C(C)NS(CCC)(=O)=O)=O)CCOCC1 N1(C(c2ccc(C)[nH]2)=O)CCC(C)C(NC(C2(CN(C)C)CCCC2)=O)C1 C1(C(=O)NCC2(C)CCCN2C(c2cnccn2)=O)CCn2nncc2C1 N1(C(=O)OC)CCN(C(=O)C2=NOC(C)C2)C(CO)C1.C12=CC=C(C=C1OC)C2 C(CN=C(N)NCC(F)F)C1CC(CC)C1.c1(SCC)cc(C)on1 C(=O)(C1=CC2(CCN(C(=O)C(F)(F)CC)C2)C1)NC(CCCC)CC CC(C)CCC(O)C(=O)N1CCCCC(CNC(=O)CCc2ccc(Cl)nc2)C1 C1(O)(CCNC(C2C(C(C)(F)F)C2)=O)CN(C(=O)C=Cc2ccco2)C1 N1(c2cccc(OC)c2)CCCC(C(N2CC(C(C)C)C(O)C2)=O)C1=O Cc1cc(C)c(NC(=O)C(=O)NCCC2CC3CCC2O3)cc1Br c1(C(=O)NCC2CC(NC(C(C3CC3)SC)=O)C2)c(C)nc2sc(C)cn12 C1(NC(c2nnn(CC)c2C)=O)CCN(C(c2cc(C)sn2)=O)CC1CO N1(C(CCC2C(C)(C)C2)=O)CCOC(CNC(c2ccoc2Br)=O)C1 C(=O)(C1CCCn2nccc21)N(CCNC(c1cc(OC)c(O)c(Br)c1)=O)C N1(C(=O)NC)CCN(c2nnc(COc3ccc(C)cc3)n2CCSC)CC1C N1(C(CCCCN(C(C)=O)C)=O)CC(CNC(=O)C#CC2(C)CC2)CCC1C N1(C(C(CC)NC(C)=O)=O)CCOCC(CNC(C2(C)CCOC(C)C2)=O)C1 N1(C(C(C)OC)=O)CCCC(C2CCN(C(c3nc(C)ncc3Cl)=O)CC2)C1 CC1CCN(C(=O)CCc2cnccn2)CCN1C(c1ccc(=O)oc1)=O c1(C(N(CC)CC2CCCN2C(C2COCCN2C)=O)=O)c(Cl)ccc(F)c1C c1(OCC=C)ccc(CNc2cccc(N3CCOCC3=O)c2)cc1Cl C1(NC(CN2CCN(C)CC2)=O)COC2C(NC(c3ccc(Cl)o3)=O)COC12 C1(C(=O)NCc2ccc(F)cc2)CC(C(C)C)=NO1.C12(COC)CN(C1)C2=O c1(CC)nc(Cl)c(CC)c(=NC2CCN(C(C3CCC(CC)O3)=O)C(C)C2)[nH]1 C12(CNC(CCCCC(C)C)=O)CCCC1N(C(C1C3(CC3)C13CC3)=O)CCC2 Cc1ccc2sc(C(=O)NCCOCC3CCCC3Oc3ccccc3)nc2c1 CCC(F)C(=O)NCC(O)CN(C)C(c1cnn(C(F)(F)F)c1)=O C1(N(C(C2N(C(C(CC)N(C)C)=O)CCCC2)=O)C)CCCC(C)(C)C1 c1(COC)sccc1C(N1CC(C(C)NC(C2CN(CC(F)(F)F)C2)=O)C1)=O C1(C(N2CC(O)(CNC(CNS(CC)(=O)=O)=O)C2)=O)CC2CCC1C2 O=S(=O)(c1ccc2c(Cl)ccc(Cl)c2c1)NCC(C(F)F)c1ccccc1 C=C1CC2(C1)CC(C(N1CCOCC(NC(=O)C(c3ccc(C)s3)C)C1)=O)C2 CC1(C)CCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1C(=O)Nc1cnc(Cl)nc1 C1(CNC(C(C2CN(C(c3c(CC)ocn3)=O)C2)O)=O)CC(C2CC2)=NO1 C1(CNC(C(C2CC2)OC)=O)CN(C(=O)CC=CC)C2(CCOCC2)C1.C1(C)CC1 c1(C(N2CC3(CN(C(C(C(COC)C)C)=O)C3)C2)=O)ccc2ccncc2n1 c1(C(N(C(CN(C(C(CC)=CC)=O)C)C)C)=O)ccnc(N2CCN(C)CC2)n1 c1(C(=O)NC(CC)(C)CO)nc(C)c(C)cc1N C1(CNC(CSCCCC)=O)CC12CCN(C(c1ccsc1CC)=O)CC2 Nc1c(C(=O)NC2CC(NC(=O)CCCc3ccncc3)C2)cccc1O c1(NC(c2c(CNC(c3c(CC)onc3C)=O)nccc2)=O)cccn(C)c1=O N1(C(CN(CCCCCC)C)=O)CCC2CCN(C(=O)Cc3nc(C)cs3)CC12 CC(CC(C)C(F)F)NC(=O)C(C1(C)CC1)NC(=O)CCC(=O)C1CC1 C(c1ncccc1C)=CC(=O)NC1C(CNC(c2c(COC)cco2)=O)CCC1 c1(CC(=O)NC2CN(C(CNC(CCC(C)C)=O)=O)CC2O)ccc(F)cc1Cl c1(C(N(CC(CNC(Cc2cc(C)on2)=O)(C)C)C)=O)cccc([N+](=O)[O-])c1Cl N1(C(C)=O)CCC(N(C(=O)Cc2csnc2C)Cc2cnncc2C)CC1 N1(C(CCC(C)OC)=O)CCCCC(C(=O)NC(CO)CCC2CC2)C1 N1(C(CCC)=O)CCC2(CCCCC2NC(=O)CN(C)CCO)C1 O=C(CCC(F)(F)F)NC1(CCCCNC(=O)COC2CCCO2)CC1 c1(C(=O)NC(C(=O)NC(CC)C2CC2)Cn2cncn2)cc(C)sc1N c1(CC(=O)NC2C(NC(C3C(CN(C)C)C3)=O)C2)cccc(OC(F)(F)F)c1 c1(C(=O)NCCC2CN(C(C(C)(C)C3CCCO3)=O)C2)ccc(N)cc1Cl c1(-c2ccn(CCCC3(F)CCN(C(=O)OC(C)(C)C)C3)n2)cc(F)ccc1F CCC(C#N)C(=O)N1CC(O)(CCNC(=O)C2CC2)C1 c1(OCCC)cccc(C(=O)NCC2(O)CCN(C(=O)Cn3ccc(C)n3)C2)c1 c1(C(=O)NC(CCc2ccc(OC)cc2)C(=O)O)sc2cccnc2c1Br C(=O)(CCC(=C)Br)N(CCNC(C1(CC#C)CCCO1)=O)CCOCCO C1(C)(C(=O)NCC23CC(NC(C(CC)CCOC)=O)(C2)C3)OC(C)(C)OC1C C#CCCCCCCC(=O)N1CCC(O)(CCNC(=O)C(O)CC2CC2)CC1 c1(OC)cc(C(N2CC(NC(=O)C(N3C(=O)CCC3=O)C)C(O)C2)=O)nc(C)c1 c1(C(=O)NC(CC)CN(C)C(C23CCCC2(C(N)=O)C3)=O)ccc(O)c(C)c1C c1(C(=O)NC2C(N(C(C(CCOC)C)=O)C)CCCC2)ccc2c(c1)CCCO2 c1(CC)cc(NC(c2nnnn2C2CCOC2)CC2CCC2)ccc1C c1(OC)cc(C(N2CC(NC(c3nc(=N)cc[nH]3)=O)CCC2C)=O)cc(C)n1 C1(CNC(C2C(C)(COC)C2)=O)CN(C2CC2)CC1(F)CO.c1(C=O)sccc1F c1(N(C)C(c2ccc(Br)cc2)=O)cc2cc(Br)ccc2s1 C1(NC(Cn2ccc(C)n2)=O)CCN(C(C2CSCCS2)=O)CC1O C(=O)(CC(C)(C)CC(F)(F)F)N1CC2C(NC(C3N(CC)CCC3)=O)C(C2)C1 C1(C(=O)NC(C#C)CC)CCN(C(=O)Cc2cccc(O)c2)C(C)(C)C1 N1(C(C(CNC(C2(CCOC)CC2)=O)O)=O)CC(C)(C)C1C(C)C C1(OC)CN(C(=O)C(N2CCOCC2c2noc(C(C)C)n2)=O)C1(C)C C1(NC(CC=CC)=O)CC2(C1)CC2NC(=O)CC(c1cccc(OC)c1)C c1(C(=O)NC2CC(CNC(C3CCNC3=O)=O)C(O)C2)ccn2c1CCCC2 N1(C(Cn2ccc(C)n2)=O)CCC2(CC1)CCN(C(C1CCCC1C)=O)C2 n1(CC(C(N2CCC(N(C(C(C(C)C)O)=O)C)C2)=O)C)ncc2c1CCCC2 c1(NC)cc(C(=O)NC2CCCC(NC(C3CC(C)(C)C3)=O)CC2)cc(Cl)n1 c1(C(C)(C)C)nc(SCC(=O)NC2CC(CCc3cn(CC4CC4)nn3)C2)cs1 N1(C(C2ON=C(C)C2)=O)CC2CCCC(N(C(=O)C=CC3CCOCC3)C)C2C1 C12(C(=O)NC(C3CCCCC3)C#C)CC(CO1)N(C(c1ccc(CO)s1)=O)C2 Cc1ccc(CC(=O)N(C)CCN(C(=O)C=Cc2nc(C)co2)C)cc1 N1(C(c2c(C)cccc2)=O)CC(NC(=O)C=CC(C)C)C(C2CC2)C1 C1(CC(=O)NCCCCCNC(=O)CN2CCCNC2=O)CC2CCC1CC2 N1(C(c2[nH]c(=NC)sc2)=O)CC2CCC(C1)N2C(=O)C(=CC1CCCC1)C C1(NC(C2C(=O)NCCCC2)=O)CN(C(=O)CSc2nncs2)Cc2ccnn2C1 N#CC1(CNC(=O)C(O)CCCNC(C2CC2C#N)=O)CCCCC1 Cc1cc(C)n(CC(N2CCCN(C(=O)CCC(N)=O)C(C)C2)=O)c(=O)n1 C=CC(C)(O)C(=O)NCc1ncoc1C1CN(C(=O)CSc2nc[nH]n2)C1 Cc1ccc(NC(C2CCCN(C(=O)Cn3cccnc3=O)C2C)=O)cc1C CS(=O)CCC(=O)N(C1CCCCC1)CCNC(=O)C=C(C1CC1)C1CC1 CCCCCCCNC(=O)COC1CC(NC(=O)C(O)CC2CCCC2)C1 c1(C(N2CCC(N(C)C(C3(CO)CC3(F)F)=O)C2)=O)ncnc2c1CCC2 CCC(C)C(CNC(=O)COC(C)C)NC(=O)CSCC(=O)NC C1(N(C(CN(CCC)C)=O)C)CN(C(=O)CNC(=O)NCC2CC2)C1 c1(C(=O)NCCCN(C)C(c2cc(Cl)cn2C)=O)ccncc1F c1(N2CC(O)(CCNC(C(c3c(C)n[nH]c3C)C)=O)C2)ncnc2c1CCC2 C1(NC(c2c(-c3ccccc3)nc(C)s2)=O)CN(C(C2CC2C)=O)CC(C)(C)C1 N1(C(CN(C)CC)=O)CCOC2(CCC(NC(c3cc(O)ccc3C)=O)CC2)C1 N1(C2C(NC(C3C(c4c(C)ccs4)C3)=O)CCC2)CCN(C(=O)C=CBr)CC1 C1(F)(CNC(c2cnc(O)o2)=O)CCN(C(C2CCN(CC(F)(F)F)C2)=O)C1 N1(C(CC(=O)NCC)=O)CCN(C(C23CC(CC(C)O2)C3)=O)CC1CCO C1(NC(C2C(C)CCO2)=O)CN(C(=O)CC2(C(F)(F)F)CCC2)CC1O CC(C(=O)NCC(C(=O)N1CCC(CC(C)(C)C)C1)N(C)C)C(C)(C)C c1(CNC(C(CC)N(C)C)=O)cccc(C2CCC2)c1 N1(c2cc(NCC3(Br)CC3(F)F)nc(C)n2)CCCNC(=O)C(F)(F)C1 c1(CNC(C2CSCCN2CC)=O)ccc2c(c1)OCCN2C c1(C(=O)NCC(CC=C)NC(=O)CCn2cc(Cl)cn2)cc(C)nn1C c1(C2C(C)C2)cc(C(=O)NCC(C)(C)CNC(=O)CC(C)n2cccn2)[nH]n1 c1(C(=O)NCCN(C(c2nc(C)n(C)c2)=O)C2CC2)cc2c(C)nn(C)c2s1 N1(C(C(C)OCC=C)=O)CC2CC(C(=O)NCC3CC3CC)(C2)C1 c1(C(=O)NC(CC(C)C)CNC(C2(F)CCCN(C)C2)=O)cncc2c[nH]nc12 N1(C(c2c(C)nc(CC)o2)=O)CC(N(C)C(C2CC2c2ccsc2)=O)C(C)(C)C1 C1(C2CCOCC2)(C(=O)NC(c2c(OC)cccc2)CNC(C2CCCC2)=O)CC1 n1(CC(N2CCC(N3CCN(C(C=C=C(C)C)=O)CC3)C2)=O)cc(F)ccc1=O C(C(C)(C)C#CC(=O)N(C)CC1CCCN(C)C1)NC(C(CC)C)=O c1(CC(=O)NC2C3CN(C(C(C)=C4CC4)=O)C(C3)CC2)cccc2c1OCCO2 C1(NC(C2(C)CCC2)=O)COC2(CCCN(C(C3CC(F)(F)C3)=O)C2)C1 C1(NC(Cc2n(C)ncc2)=O)CCCCC1NC(=O)Cc1cnc[nH]1 C=CCC(C(=O)NC(C)(C)CCNC(C1CC2CCC2C1)=O)NC(C)=O C1(CC(NOCC(C)(C)C)=O)CCCCN1C(=O)CN1CC=CC1 N1(C(C2C(CC)OCC2)=O)CCC(CCNC(=O)C(F)(F)c2cnn(C)c2)CC1 C1(C(=O)NC2(C(N3CCCC(O)C3)=O)C(C)CCC2)CC12CCOCC2 CC(Cc1cnco1)C(=O)NCCCC(C)NC(=O)C(=O)NCc1ccccc1 C1(CNC(C2CC=CC2)=O)CCN(C(c2cc(O)ccc2Br)=O)C12CCC2 C1(CNC(=O)Cc2cccnc2)COCCN(C(c2cn3c(n2)SCC3)=O)C1 c1(CCC)cnc(N(C2CCNCC2F)S(=O)(=O)C(C)C)nc1 O=C1CCC2(C(=O)NCCNC(c3ccc4occc4n3)=O)CCCCC2N1 C(c1ccc(Cl)cc1)=C(C)CN1CCC(O)(Cc2ccc(F)cc2)CC1 C1(OC)CS(=O)(=O)CC1N=c1[nH]c(=NCCC(C)(C)CC)[nH]c2c1CCCC2 C(=O)(C(C(C)(C)C)OC(C)(C)C)N1CC2C(NC(C(C)(C)SC)=O)(C2)C1 Nc1c(C(=O)NCC(O)CNC(c2cnn3cnnc3c2)=O)ccc(Br)c1F CC(C(=O)N)NC(=O)Cn1ccnc1.C(CCCc1ncc[nH]1)NC(N)=O C(=O)(CC(C)(C)CN(C)C)NCC(C)N(C(c1ccc[n+]([O-])c1)=O)C1CC1 N1(C(c2cnc(CC)s2)=O)CC2(CO)CC1(C(=O)NC(C)CN1CCCCC1)C2 C1(OC)CN(C(C2CC(O)C2)=O)CC1c1cn(Cc2cc(Cl)c(Cl)s2)nn1 c1(-c2cn(C(C(=O)N(CCOCC)C)C)nn2)cc(OC)ccc1Br Cn1nc(CNC(=O)C(C2CCCCC2)O)c2c1CCN(C(=O)C1=CCC1)C2 C(c1cncs1)=CC(=O)NC(CC1CCOCC1)C(=O)NCCC1CCCCC1 C1(C(N(CCCOC)CCO)=O)C2CCC(C2)N1C(=O)C1=NOCC1 Cn1c(=O)n(CC(N2CCOCC2C(=O)Nc2cc(O)nn2C)=O)c2c1CCC2 N1(SCCCC2CC(C(=O)NCc3ccc(COCC)o3)C2)CCN(C)C(=O)C1 N12CC3COCC3(C1)C2=O.Cc1c(C(=O)NCCCCCCF)cccc1F N1(C(C2OCCN(C)C2)=O)CC(CNC(C2(c3ccccc3)CC2)=O)C2(CCC2)C1 N1(C(C2CCC(C)O2)=O)CCC(NC(c2cnc(Cl)cn2)=O)C12CCC2 N1(CCN(C(CC(C)C2CC2)=O)C)CCN(C(c2cnc(C3CC3)nc2)=O)CC1 CCCC(CC)C(=O)N1CCC(C(N2CC=CC2CNC(N)=O)=O)C(C)C1 CC1(C(=O)NCC2COCCN2C(c2nnc(C(F)(F)F)s2)=O)CCOCC1 C1(CC(=O)NC(C(C)C)CNC(=O)CSCCN(C)C)CCC(=O)NC1 N1(C(CCOCC#C)=O)CC(CNC(=O)CN2CCNC(=O)C2)C(F)(F)C1 c1(CNC2CN(C(C(C)(C)CCl)=O)CC2F)ccc(Br)c(F)c1O c1(C(=O)NCCNC(C2CC=CCO2)=O)nc(-c2ccccc2)oc1C1CC1 C1(NC(=O)NC2CCC(NC(c3c(C)scc3)=O)CC2)CCn2c(C)nnc2C1 N1(C(C2C(CC)N(C)CC2)=O)CCC2CCN(C(C3CC(=O)N(OC)C3)=O)C2C1 C1(CNC(=O)C(F)=CCCF)CCCC12CCN(C(C1(O)CCCCC1)=O)CC2 c1(C(=O)NC(CC)(CNC(C2CC2(Cl)Cl)=O)CC)noc2c1COCC2 N1(C(c2ccn(CC)n2)=O)CC(NC(c2ccn(CC#N)n2)=O)C2(CC2)C1 CC1(NC(=O)C(O)CNC(=O)CCc2csnn2)CC2CCC1C2 C(N=c1nc2scnc2c(NCC23CC(C)(CCO2)C3)[nH]1)c1ccc(C)n1C N1(C(CCSCCC)=O)CC2CCOC2(CNC(c2cn(C)nc2O)=O)C1 C1(CC(=O)NCCCCN(C)C(c2cn(CC3CCOC3)nn2)=O)COC2(CCC2)C1 C1(NC(C(N2CC3CC3C2)C)=O)CN(C(c2cc(Cl)sc2Cl)=O)CCC1F C(=O)(C(F)C(C)CNC(C1(N(C)C)CCOCC1)=O)N(CC#CC)C c1(-n2cc(C3C(OC)CN(C(C4(CC=C)CC4)=O)C3)nn2)nnc2ccccn12 C1(NC(C(C)C2(O)CCC2)=O)CC(C(=O)NCc2ncc(CO)[nH]2)CC1O c1(C(N(CCC(C)NC(=O)CC2COCCO2)C)=O)cnn(C(C)C)c1F c1(C(=O)OC)cc(Br)sc1NC(c1ccnn1C1CCCC1)=O c1(NC(C2CC3(CC(OC)C3)C2)=O)ncnc2c1CCC2 c1(C(=O)NCC(CO)NC(=O)C(c2ccccc2)=O)ccccc1C(F)F CCCC(C)(O)CC(=O)N(C1COCC1NC(C1(O)CCC1)=O)C1CC1 C#CCCN=C(NCC(C)(F)F)NCC1(C2CC2)CC1 C(=O)(CCC1=NNC(=O)CC1)NC1CC(NC(c2c(C)ncnc2)=O)C(O)C1 C1(C(=O)NC(C2CCN(C(=O)Cn3cnnn3)C2)C)CN(C)C(=O)CCO1 c1(-c2c(OC)cnc(F)c2)ccn2cc(C(N3CCCC(N(C)C)C3)=O)nc2c1 CC(=NO)C1CC(C(=O)NCC2CC3(CC3)CN2C(=O)CC(=O)OC)C1(C)C Cc1cc(=NCC(C)CNC(c2[nH]c(C)c(C)c2C)=O)[nH]c(C(C)(C)C)n1 C1(NC(=O)CCn2cccn2)CCOCC1NC(c1nccc(C(F)(F)F)n1)=O CC1=CCSC1C(N1CCC(OCC(=O)NC2CC(F)(F)C2)C1)=O c1(CC)cccc(NC(=O)CONC(=O)Cc2ccon2)n1 CC(C)CC(C)CC(C)C(=O)NCC1CC(C)N(C(=O)C(C2CC(F)(F)C2)O)C1 c1(CC)ccc(C(=O)N(C2CN(C(C3CCN(CC(C)C)CC3)=O)C2)C)c(F)c1 CCC(CC)(CC)C(=O)N1CCCC(C)(NC(=O)C(n2ccnc2C)C)C1 CCC(C)C(CC(=O)NCCCCC1CC1C)NC(c1cocn1)=O C1(C(=O)NC(CCCC)(C)C)COC2(C1)CN(C(=O)CCCCCC#N)C2 C1(C)(NC(CCc2cc(C)[nH]n2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C1 c1(OC)cc(C(N2CC(C)(NC(=O)CO)C2)=O)cc(NC(C)=O)c1OC(F)F N1(C(CN(C)CCO)=O)CCOC2(CCN(C(C3CCC(F)(F)C3)=O)C2)C1 C1(O)(CN2CCC(NC(=O)Cc3coc(-c4ccccc4)n3)C2)CCSCC1 N1(c2n(-c3ccc(C)cc3)nnn2)CCC(CNC(C2CC3CC3C2)=O)C12CC2 c1(C(N2CCN(C(C3C(CC)CCO3)=O)C(CO)C2)=O)n[nH]c2c(C)cccc12 N1(CCC=CC)CC2CC2(C(=O)NC2CC2)C1 C1(OC)Cc2ccccc2C1NC(=O)Nc1cc(F)cc(F)c1 c1(COCC)ccccc1NC(c1nnnn1C)C1(OC)CCCC1 CC(C)C(CCC(=O)NCC1CC2(C1)CC(O)C2)NC(C1COCCN1C)=O c1(SC)ccc(CN2CC(C(=O)Nc3ccc(C(=O)O)cc3)CC2C)cc1 C1(NC(C(C(CC)C)N(C)C(c2ccn(CCF)n2)=O)=O)CCCCC12CCC2 c1(C(=O)NCCCc2cnoc2)cn(C2CC3(NCC4CCOC4)CC23)nn1 N1(C(Cc2c(C)n[nH]c2)=O)CCCCCC1CNC(C1COCCN1C=O)=O N1(C(C2CCN(C(=O)CC3CCOCC3)CC2F)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NCC(CC(=O)NCCCC)OC)ncc(F)cc1F c1(CC(=O)NC(C(CO)NC(C(CC)n2ccnc2)=O)C)ccc2c(c1)CCO2 C1(NC(=O)C=Cc2ccc[nH]2)CCC(NC(c2ccncc2C2CC2)=O)CC1 c1(OCC)ccc(NC(=O)C(=O)Nc2ccc(F)cc2F)cc1S(N)(=O)=O c1(C(N2CCC3CN(C(COC(C)=O)=O)CC3CC2)=O)cccc2nc(O)ccc12 C(=O)(CC1=NSC(=O)C1)NCC1N(C(CC23CC(C(=O)OC)(C2)C3)=O)CCCC1 C1(CNC(C(CCC)NC(=O)Cc2ccnn2C)=O)CCOCC1(C)C c1(SCC(N2CC(COC)(CNC(C3CC34CCCC4)=O)C2)=O)nc(C)cc(C)n1 c1(CC(C(=O)O)NC2CCCCCCCCC2)ccc([N+](=O)[O-])cc1Cl c1(C(=O)Nc2ccc(CNc3c(C(N)=O)cncc3)cc2)scc2c1OCCO2 Cc1cc(C(F)(F)F)ccc1C(=O)NCCOCCOCCNC(N)=O c1(C(C)NC(=O)NCC2CC(OCCO)C2)nc(Nc2ccccc2)cc(Cl)n1 c1(C(=O)NC(C2N(C(C3C(C=C)CC3)=O)CCC2)C)cc(C)c(Br)cn1 N1(C(C(CC)N(C(=O)CC(C)C)OC(C)=O)=O)C2CCC1CC(NS(=O)(=O)NC)C2 Cc1cc(C(=O)NCCC2(O)CCCN(C(=O)COC(F)F)C2)c2occc2c1 C12(C(N3CCCC(NC(C4C(C)(C)CO4)=O)CC3)=O)CCC(O1)c1ccccc12 C(CCCC(=O)NC1(C)CC(NC(c2cccc(N(C)C)c2)=O)C1)OCCC=C c1(OCC)ccc(Br)c(Cc2noc(C3C=CS(=O)(=O)C3)n2)c1F C(=O)(C(C(C)(C)C)NC(c1cnns1)=O)NC(C)CC1CCCC1 C(=O)(CC(CC)C(C)C)NC(CCC)CC(N1CCOC(C)(C)C1)=O N1(C(CCC#C)=O)CCC(C)(C)C1C(=O)NCCN1CCCCC1 C1(NC(C=CCN(C)CC)=O)CC2CCC1CN2C(c1cnoc1C(C)C)=O Cc1cc(C(N2CC3CC3(C(=O)Nc3cc(Br)nc(Br)c3)C2)=O)cc(C#N)c1 N1(C(CN(C(C)=O)C)=O)CC(NC(=O)C(C)(C)O)CCC1C C(=O)(CS(=O)(=O)C(C)C)NCC1C(NC(C(c2ccc(OC)cc2)(F)F)=O)CC1 N1(C(c2ccc(SC)o2)=O)CCC(O)C1C(=O)NC1(C)CCCC1C C=Cn1nncc1C(=O)N(C1CCN(C(c2ccc(C(C)=O)cn2)=O)CC1)C c1(NC(C2CC2C(=O)Nc2cc(O)ccn2)=O)cc(Br)ncc1[N+](=O)[O-] N1(C(c2c(C)scc2)=O)CC2CN(C(c3ccc(-c4ccc(Br)cc4)o3)=O)CC12 C(CC(O)CNC(=O)CCc1ccncc1)NC(=O)CCC1CNC(=O)N1 c1(-c2onc(C3(N(C)C)CCCOC3)n2)coc2c(F)cc(F)cc12 C(C(CC(C)C)C(=O)N1CC(=O)C1)NC(c1c(C)nc(Br)s1)=O C1(O)(CN(C(CC2(C=C)CC2)=O)C)CCCN(C(c2nc(Cl)sc2C(C)C)=O)C1 C(=O)(C1=CCCS1)N(C1C(C(N(CCCC)C)=O)CCC1)C.C1(=O)NCCN1 N1(C(CNC(C(CC)C)=O)=O)CC2(CCCN(C(c3n[nH]cc3F)=O)C2)C1 Cc1cc(C(=O)NCC2CCN(C(c3ncoc3C)=O)C2)ncc1F c1(OC)ccc(Cl)c(C(=O)NC2CCCN(C(=O)Cc3ccc(Br)cc3)CC2)c1 Cc1cc(Br)c(NC(C2CC3(C2)CN(C(=O)C(C)c2cccs2)C3)=O)cc1C C(=O)(C(C1=C(C)CCCC1(C)C)N1CCCC12CCN(C)C2)NC(CC)(C)C N1(C(C2(CNC(Cc3nc(C)oc3)=O)CC2)=O)CCn2cnnc2C1 c1(NCc2c(C)nc(Cl)s2)cccc2cccc(Cl)c12 N1(C(c2nc(C#C)sc2)=O)CC(NC(c2ccc(F)c(C)c2N)=O)CC(C)(C)C1 C1(NC(C(CCOC)C)=O)CN(C(=O)CCCc2nc(C(C)C)no2)CCC1C c1(CCC)cc(C(N2CCC2CNC(C2CCCN2CC(F)(F)F)=O)=O)c(C)o1 N1(C(CN2C(C)CC2)=O)CC=CC1Cn1cc(C2CCOC2)nn1 c1(NCCNCC(c2ccccc2)(C)OC)c(C(=O)O)nn(C)c1C n1(CC)nc(C(=O)NC(C)C(C)NC(=O)C=Cc2cn(C)nn2)c2c1CCOC2 C1(CNC(c2ccc(OC)s2)=O)CC2(CCOCC2)CN1C(=O)C(O)P(C)(C)=O c1(NC(Cc2nc(C)oc2)=O)ccc2c(ccn2CN(C)C)c1 c1(C(N2CCC(NC(c3c(C)cn(C)c3)=O)C(CO)C2)=O)cccn2nccc12 c1(C(=O)NC2C=CCN(C(C3C=CC=CC=C3)=O)C2)cc(C2CC2)nc(Cl)c1 C1(C(=O)NC(CCC)C2CCC2)N(C(c2csc(C)c2C)=O)CCCC1(C)C c1(CNC(C(=O)OC)Cc2ccc(O)cc2)cnc(C2CC2)nc1 C1(C(N2CCC(C)(CNC(c3cc(Cl)c[nH]3)=O)C2)=O)CCOC2(CCCC2)C1 C1(Cl)(C(N2CC(CC=C)(C(N3CCC3CC)=O)C2)=O)CCCCC1 c1(C(C)Nc2sc(Br)cc2N)cc(F)ccc1F c1(C(N(CC(CC)NC(c2ccnc(O)c2)=O)C)=O)cnc(C)c(C#N)c1 C(=O)(CCCS(C)(=O)=O)NCC1C(NC(CCn2ncc(C)c2)=O)CC1 N1(C(C=CC(C)C)=O)CC2(C(=O)NCc3ncco3)CC1CO2 c1(C(=O)NC2C(CO)CCN(C(CCC)=O)C2)[nH]nc2ncnc(O)c12 C1(NC(C(CC=C)C)=O)CC2CC1N(C(c1scc(Br)c1Cl)=O)C2 N1(C(C(=O)NCC(C)C)C2CC2c2cccs2)CCC2(CC(C(F)F)=NO2)C1 c1(CC)ncsc1C(=O)NC1CCCC1CNC(=O)CC1C(CC)C1(F)F CC(CCCNC(=O)C(C)Oc1ccccc1)NC(=O)C=CC=C(Cl)Cl c1(C(=O)NC(CC)CNC(=O)C(C(C)C)SCC)nn(CC(F)F)cc1[N+](=O)[O-] C1(NCc2cncc(C)n2)CCCN(C(C2CCC(O)CC2)=O)CC1 Cc1cc(=O)c(C(N2CC=CC2CNC(=O)C(n2cc(Cl)cn2)C)=O)cn1C C1(C(N2CCC(CNC(c3c(C)c(N)cnc3)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 C(CC(C(=O)Nc1ccc(OCC)nc1)NC(C1CNC(=O)O1)=O)OCC Cc1cc(N)c(C(=O)NCC(F)CNC(C2CCC3CC2CO3)=O)c(F)c1 C1(C(=O)NCC2N(CC)CCC2)CC12CC(NC(=O)C(C)=C1CCC1)C2 c1(N2CC(CC(=O)Nc3cccc(F)n3)OCC2)ncnn2cc(Br)cc12 CN1CC(O)CCC1C(N1CC(C(N2CCC(O)C(CO)C2)=O)C(F)(F)C1)=O c1(CC(=O)N(CCC(C)NC(=O)CSCC(F)(F)F)C)cc[nH]c(=N)c1 C1(C(=O)NCCOC2CCN(C(c3ccncc3F)=O)C2)CCC2(CC1)CC2 C(=O)(CCCCCCS(N)(=O)=O)N1CCC(C2(NC(C=COCC)=O)CC2)C1 C1(C(=O)OCC(=O)NC(c2c(C)cccc2)C)CCC2(COC2)OC1 C1(CC(C)NC(=O)C2CC2)CC2CCC(C1)N2C(=O)C=Cc1ccccc1 c1(CC)c(C(=O)NC2(C)CC(NC(=O)C(C)P(C)(C)=O)C2)[nH]c2ccccc12 C1(NC(CSc2c(C)n[nH]c2C)=O)CC(O)CN(C(C2(C3(O)CCC3)CC2)=O)C1 C1(C(=O)OC)CC2CCC(C1)N2C(=O)C(C(C)C)Nc1ccccc1N N1(C(c2c(CCCC)ocn2)=O)CCCC(CNC(=O)C(=O)NC2CC2)C1 C1(OC)CS(=O)(=O)CN(C(C2C=CCC(C(=O)OC(C)(C)C)C2)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)NCC(CNC(c1[nH]cc(OC)c(=O)c1)=O)O c1(OCC)cc(C(N2CCCC2CNC(=O)CC2CCC(F)(F)C2)=O)oc(=O)c1 C#Cc1ccc(OCC(=O)NCC2C3CN(C(=O)C(C)(O)COC)CC23)cc1 Nc1cccn(CC(=O)NCC2CC(CNC(c3cnc(S)[nH]3)=O)CO2)c1=O c1(C(=O)NC2CN(C(Cc3cc(C(C)C)no3)=O)CC2F)ccc(S(C)(=O)=O)s1 C1(CC(N2CC(NC(=O)CN3CCCNC3=O)(CF)C2)=O)CCC2(CCC2)O1 c1(CC)nc(-n2cccc2)sc1C(=O)NC1CC(C)(NC(c2sc(F)cc2C)=O)C1 CC(=CN=c1[nH]c(Cl)ncc1F)c1ccccc1 C(=O)(C1=CCC(NC(=O)Cc2ccoc2C)C1)NCC1(C(CC)=O)CC1 Cc1nc(C(N2CCC3(CCCN3C(C3CCCN3C)=O)C2)=O)c2n1CCCC2 c1(OC)ccc2[nH]c(NC(=O)C(=O)NCc3ccc(COCCO)cc3)cc2n1 C1(C(N2CC(C)CC(NC(CN(C(C)C)C)=O)C2)=O)CCC(=O)C(C)C1(C)C CCCC(C)(C)C(=O)NCCC1CN(C(=O)CC2CC3(CC3)C2)CC(C)O1 c1(C(=O)NC2(C)CN(C(=O)C=CC3CCCCCC3)C2)cc[nH]c2nccc1-2 NC(=O)CCC(=O)NCC(CNC(c1cccc(OCC(F)(F)F)n1)=O)CO N1(C(CC2CCC(C)O2)=O)CCOC2(C1)CN(C(c1cn3c(n1)SCC3)=O)C2 C#CC1(O)CCN(C(=NCCc2c[nH]nc2C)NCCN(C)C(=O)OC)C1 N1(C(c2c(C)cno2)=O)CC2CCCC(CNC(=O)C3=C(Cl)CCOC3)(C2)C1 CC1=C(C(=O)Nc2nccs2)C(c2ncc(S(N)(=O)=O)s2)NC(=O)N1CC1CC1 c1(C(=O)NC2CC(N(C(C(C)SCC)=O)C)C2)c(F)ccc(Cl)c1N C1(C(=O)NCC2CC(OC)CN2C(=O)C=C(C)C(F)F)CCc2c(cnn2C)C1 CCC(C)(C)C(=O)NCCCN(C(=O)CN1C(C)CCC1C)C c1(CN(C)C)c[nH]c(C(=O)NC(CNC(=O)CN(C)C2CC2)CO)c1 C1(CNC(c2ccc(OC)o2)=O)CC2CCC1N2C(c1cnnc(Cl)c1)=O C1(O)(C(CNC(C2C(=C)C2)=O)(C)C)CN(C(c2csc(CSC)n2)=O)C1 N1(CCCC)C(=O)NC(c2cnc(N(C)C)cn2)C(C(=O)OCC)=C1C(C)OC C(=O)(C(C)CC(C)(C)C)NC(C(CO)NC(CC(C)NC(=O)OC(C)(C)C)=O)C C#CCCCC(C)C(=O)NC1CC2CC1N(C(=O)Cc1ccc(C)nc1)C2 O=C(CC1=CCOCC1)NC1CCC(C(=O)NC2CN(CC(F)F)C2)C1 N1(C(CC=CCC)=O)CCC(C2CC2)C1CNC(=O)CCc1cnc(C)o1 CCCC(CCC)C(=O)N1CCOC(C(C)NC(c2ccc(N)c(F)c2F)=O)C1 O(NC(=O)C(C)(C)C1CCN(C(C2CC(O)C2(C)C)=O)C1)CCC=C N1(C(C2C(c3cn(CC)nc3)OCC2)C(=O)NCCCSC)CCC2C(O)CC12 C(C(C(=O)NC(C)(C)CNC(C1CC(F)(CF)C1)=O)C(C)(C)C)OCC=C C1(CN(C)C(C2C(F)(F)C23CC3)=O)CC(F)CN1C(c1ncc[nH]c1=O)=O CC(C)C(CCC(=O)N1CC(CO)C1(C)C)NC(=O)C(C)CC1CCC1 N1(C(C=CC=CCC)=O)CC(C=C)(CC(=O)NC(CC)C(=O)N(C)C)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCC(C)(C)NC(C(C)CN(C)C)=O C1(C(=O)NCC=CC)CC(C)(C)CCN1C(=O)C(N1CCOCC1)C C(N=c1cc(C)nc(Cl)[nH]1)c1cccc(NC(c2c(OC)cccc2)=O)c1 C(CCC(C(=O)NCC12CCC(CC1)O2)NC(c1ccncc1Cl)=O)OC Cc1ccc2sc(C(=O)NC3CC4CC3N(C(C3(C)CS(=O)(=O)C3)=O)C4)cc2c1 c1(C(C)C)noc(CCC(=O)NC(C2CCN(C(=O)C(F)C3CCOC3)C2)C)n1 C1(NC(CC(C)(C)O)=O)CCCC12CCN(C(=O)C=CC1CCCCC1)C2 c1(CC(=O)NCCSCC(=O)N(CC(CCC)C)C)ccc(F)nc1 C(=O)(C1=CCCOC1)NCCCCCCNC(C(c1ccn(C)n1)(C)C)=O C(C(=O)N1CC(C(C)NC(=O)CC(O)C2CCCC2)C1)(C(C)C)NC(COC)=O C(CCC(C(=O)NCc1cocn1)NC(=O)CCS(N)(=O)=O)OC c1(OC)ccc(CN2CC(CNC(=O)CCc3ccc(C)cc3)C2)cc1F C(=O)(C1=CCC(C)CC1)NCC1CCCCN(C(c2cncc(C)c2)=O)C1 c1(N2CCCC(C(=O)NC(C#C)C)C2)c(OC)c(Cl)nc2ccnn12 Cc1ccccc1-n1cc(-c2csc(C(=O)NCC3(C#N)CC3)n2)cn1 CCC(CCC(=O)N(CC(O)(CC)CC)C)NC(c1ccc(O)cn1)=O N1(C(C(c2nc(C)sc2)=O)=O)CCC(CO)C(NC(c2cocn2)=O)C1 CC#CCCC(=O)NCC(CNC(=O)COC1(C)CCC1)OC c1(CCC)ncoc1C(=O)N(CCCCCNC(=O)C(O)CN1CCCC1)C N(C(=NCc1ccc2nc(O)oc2c1)N1CCC(CSC)C1)C(CC)CC C(=O)(CC(CC)CCCC)NCC12C(CN(C(C(CCCCC)F)=O)C1)CCO2 C1(NC(=O)NC2C3CCN(C(CCCC)=O)C3C2)C2CCC(CC2)C1C(F)(F)F Cc1cc(C(=O)NNC(=O)c2cc[nH]n2)c(C)n1-c1ccco1 c1(C(=O)NC2CCC(NC(c3cncc(O)c3)=O)C2)c(F)c(F)cc(F)c1F N1(C(CCOCCN(C)C)=O)CCCC1(C)CNC(C1CCCC12CC2)=O Cc1cc2c(C(=O)NC3CCC(NC(=O)CC(C)C(F)F)CC3)ccc(C)c2[nH]1 c1(N2C(c3nc(C)[nH]n3)COCC2)ncc(I)cc1Br Cc1cccn2ncc(C(N3CCC4C(NC(=O)C=Cc5cccs5)C34)=O)c12 C1(C(=O)NC2(COC)CN(C(CC=C)=O)C2)CC2CCC(C1)N2C CC1(C(=O)NCCCN(C(c2cscc2C2CC2)=O)C2CC2)CCCC1O CC1(C)CCCN(C(=O)CCc2cn[nH]c2)C1C(=O)NC(C(C)(C)O)C1CC1 C1(OC)CCC2(CCN(C(N(C(CC#C)C(=O)C(=O)OC(C)(C)C)C)=O)C2)C1 Nc1cc(C(=O)NCC(CO)NC(=O)C(F)C(F)(F)F)cc(F)c1Br C1(C(=O)NCC(C(N2CC(C)(OCC)C2)=O)C)CC(=O)NC(=O)N1 C1(C(=O)OC)N(CCOc2cc(F)ccc2F)CC12CCC(F)(F)CC2 N(C1CCc2cccnc21)C(=O)C1CC1C(F)(F)F.c1(N)[nH]c2c(Br)cccc2c1-n1cccc1 c1(C(N2CCC(C(=O)Nc3c(C)cnc(F)c3)C2)=O)ccc(Br)c(O)c1Br C1(C(=O)NCCc2cc(C)cc(C)c2)CCN(Cc2sccc2Cl)CC(C)(C)C1 C1(OCC)CC2(C1)CC2C(N1CC(O)(C2CCCN2C(c2coc(C)n2)=O)C1)=O C1(NC(C(=Cc2ccco2)C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCC1CO N1(C(c2n(C(C)C)ccc2)=O)CCC2CN(C(=O)C=Cc3ccco3)C2C1 C1(N(C(CCSCCC)=O)C)CCC2CN(C(=O)Cn3cnc(C(N)=O)n3)CC12 N1(C(CCSC)=O)CC(NC(=O)CCc2cnn(C)n2)Cc2ccccc21 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(C2SCCCS2)=O)CCC1CO c1(OC)cc(C(=O)NC2CC(C(F)F)(CNC(=O)Cn3ccnn3)C2)sn1 C(=O)NNc1ccc(Cl)c(C)n1.c1(C(=O)OC)[nH]c2ccccc2c1CC(N)=O c1(C(=O)NC2CC(CNC(C(C)NC(CC)=O)=O)C2)ccc(S(C)=O)cc1 c1(CNc2scc(-c3ccc(OC)cc3O)c2)c(OC)cccc1C#N C(=O)(CC1=NNC(=O)C1)NC(CN(C(C(c1c(C)n[nH]c1C)C)=O)C)C n1(CC(N2CC3C(CNC(C#CC(=O)N(C)C)=O)(C3)C2)=O)ncc2ccccc12 N1(C(C(COC)COC)=O)CCC(C)(NC(=O)CC(C)C2CCCO2)CC1 Cc1ccc2[nH]c(C(=O)NC3CCC4CC3CN4C(C3CC3C)=O)cc2c1C CCCC(CNC(=O)Cc1cn(C(C)C)nn1)NC(=O)C=C(CC)CC c1(C(C(=O)NCC(=O)OCn2cccn2)N2CCCC2)ccc(C(C)C(F)(F)F)cc1 c1(C(=O)NCC(CNC(CC(CC)C)=O)C(F)(F)F)ncc2cc(Cl)ccn12 O=[N+]([O-])c1cccc(S(=O)(=O)Nc2cc(Cl)cc3nc(O)[nH]c23)c1 N12CCOCCC1NC2=O.Cn1cc(C(F)(F)F)nc1CN C1(CNC(CCOCC#C)=O)CCCCN1C(=O)CC1CCC(C)CO1 C(=O)(C1CCc2ccccc21)NCC1CC1C(=O)OC(C)(C)C c1(C(=O)NC(CC(C)NC(c2cnn[nH]2)=O)C)ccc(N)cc1 N1(C(C(CN(CC)CC)F)=O)CCCC(C)(CNC(c2cnncc2C)=O)C1 C1(NC(C(C(CC)O)C)=O)CCCC12CN(c1ncnc(C(C)(C)C)n1)C2 N(C(=NCCNS(C)(=O)=O)NCC1CC2CCC1O2)CC(C=C)(C)C C1(N(C(c2n(CC=C)ccc2)=O)C)CCCN(C(=O)C(C2COC(C)(C)O2)O)C1 N1(C(C2(CF)CCN(C(c3cc(C)cc(C)c3)=O)C2)=O)CC2CCCCC2C1C C1(NC(C(=O)NCCOCCCC)=O)CCN(C(c2ccccn2)=O)C(CC)C1 N#Cc1ccc(CN2CC(C(=O)Nc3nccs3)CC(C(F)(F)F)C2)c(Br)c1 c1(NC(C(c2n(C)cnc2)N)=O)ccc(C(F)(F)F)cn1 c1(C(=O)NC2CC(C)(NC(c3cc(OC)nn3C)=O)C2)cccc2c1OC(C)C2 c1(C(=O)NC2CCC(F)(CNC(=O)C=CCOC(F)(F)F)C2)c(F)ccc(F)c1F n1(C2(C(=O)NC3CC(NC(CCN(C)CC)=O)C3)CC2)cc(Cl)cn1 C1(NC(c2c(CC)nco2)=O)CC2CCC1CC2NC(=O)CCc1ncnn1C C1(COC)(NC(c2ccccc2C(F)(F)C(F)(F)F)=O)CCOC(C)(C)C1 O=C(C#CC1CCOCC1)NCC12CCC1CCN2C(C1CC(O)C1)=O c1(C(=O)NC23CC(CNC(C(C)CF)=O)(C2)OC3C)cccn2nccc12 c1(COC)ccc(C(=O)NC2CCC(NC(C3CCNC(=O)C3)=O)C2)cc1F c1(C(=O)NC)ccc(C(=O)N(CC(O)CN(C)C(c2nnc(C)s2)=O)C)cn1 c1(C(=O)NCC2OCC(CNC(C(CC)(C)C)=O)C2)c(N)sc2c1CCSC2 C1(NC(C(CC)n2ccnc2)=O)CCC(C)N(C(c2ccc(Br)cc2)=O)C1 C1(CN(C)C)CCCCN1C(C1C=CCN1C(=O)CCC1CCCC1)=O N1(c2c(C#N)c(F)ccc2)C2CCCC1CN(C(c1ccc(C3CC3)s1)=O)CC2 C1(CNC(CCCc2[nH]c(=N)sc2)=O)(CNC(C2CC23CCC3)=O)CCCCC1 N1(C(C=CCOCCOC)=O)CCC2CCN(C(=O)CCCn3ccnc3)C2C1 C1(C(=O)OC)CC(C)N1C(c1nn[nH]n1)=O.C1(N2C(=O)CCC2)CN(C2CCC2)C1 C1(NC(CC2(C)CCOC2)=O)CC(CO)N(C(C2COCC2C(N)=O)=O)C1 C(=O)(CC1(O)CCOc2ccccc21)NCC(C)NC(CCCC#C)=O C1(CCN(C(=O)CC2CCCCC2O)C)CCCCN1C(c1ccnc(O)c1)=O C=CCC(CC=C)C(=O)NC1CCN(CCCNC(=O)C(O)P(C)(C)=O)C1 C1(NC(c2csc(Cl)n2)=O)CC2(CCCN(C(=O)CC3CCCO3)C2)C1 C1(NC(c2c(C)nn[nH]2)=O)CC(C)N(C(=O)C=CC(=O)N(C)C)C1 Nc1ccc(C(N2CCCC(c3cc[nH]c(=N)n3)C2)=O)c(F)c1 C(=O)(C(O)CCCC)NCC1CN(C(CC=C)=O)CC1c1ccc(OC)cc1 c1(-c2nc(-c3c(C)ccc(SC)c3)n(C3CC3C)n2)cn2c(C)cc(C)nc2n1 C=CCC(C)C(=O)NCc1ccc(CNC(c2cc(C(F)(F)F)ncn2)=O)cc1 C1(C(=O)NC2CN(C(=O)C=C3CCC3)CC23CC3)CC(c2ccc(F)cc2)=NO1 C(C)(CCN=c1ncc(C(F)F)c[nH]1)NC(C1CCC(=C)CC1)=O S(=O)(=O)(c1c[nH]ccc1=NCC(C)(C)CC1CC1)C1C(C)CCC(C)(C)C1 C=C(C)C1CN(c2cc(NCc3nc(C#N)cs3)nc(C)n2)CCO1 C1(C(N2CC(C)C(NC(C3(C(F)F)CCCO3)=O)CC2)=O)CN2CCN1CC2C c1(C(=O)NC(C)CC2CN(C(C3(C)CC4(CCC4)C3)=O)C2)cnc2occc2c1 N1(C(CC(CCC)O)=O)CC2CC1CCC2NC(=O)CC1OCCCC1(C)C c1(CN2C(CC(=O)NCC3(CC(=O)O)CCC3)COCC2)ccc(Cl)cc1O CCCCC(C)C(=O)NCCCOCCC(=O)N(C)CC1CCCO1 C(=O)(C1SCCc2ccccc21)N1CC2(N(C(c3n(C)ccn3)=O)CC2)C1 C(=O)(C1=CC2(CN(C(C3C4CCCCCC34)=O)C2)OC1)NC1CCC(C)(C)CC1 c1(C(=O)NC(C)CCN(C)C(c2ccc(N)cc2)=O)cc2c(=O)[nH]ccn2n1 C(=O)(C(F)(C(=O)OCC)C(C)NC(N1CC(C)C2(CCC2)C1)=O)OCC C1(C(=O)NCC(CN(C)C(C23CCC2C3)=O)O)CCOCC1 c1(SC(C)C(=O)Nc2ccccc2)ccc([N+](=O)[O-])c(Br)c1 C=C=CC(C)C(=O)NC(c1nocc1C(=O)N(C)CCC1CN(C)C1)C C1(C(=O)NCC(CC)(C)Cl)CC(O)CN1C(c1nccnc1C)=O O=S(=O)(c1nc[nH]n1)NC1CCCC12CCC2 N1(C(c2n(C(C)C)ccc2)=O)CCC2(NC(=O)CCOC3CC(F)(F)C3)CC2C1 c1(CN)n[nH]c(=NC2CCCCC2NC(=O)C2=CS(=O)CCC2)s1 N1(C(C(c2ccccc2)NC(C)=O)=O)CCCN(C(c2cc(C)n(C)c2)=O)CC1 C(=O)(CCCC(C)C)N1C(CNC(C(CCSC)OC)=O)C=CC1 C(CCC(N)=O)(C(=O)N1CCC(C)(Cc2cnn(C)c2)C1)NC(=O)OC(C)(C)C Cc1cccc(O)c1C(=O)NCc1ccc(CCNC(C2CC2CF)=O)cc1 c1(C(=O)NCCN(C)C(C2CCSC2)=O)ccc(N2CCOCC2)cc1F C1(C(=O)NC2CC(O)(CNC(c3ccc(F)s3)=O)C2)CCc2nnc(O)cc2C1 C12(C(=O)NCC(C(=O)OCC)C)CC1CCN2C(=O)Cn1cnnc1 c1(C(=O)NCC(CNC(C(C)NC(N)=O)=O)O)cc(O)cs1 c1(C(N2CCC(CNC(=O)COc3ccc(F)nc3)C2)=O)c(Cl)cncc1Cl C(C(=O)NC1(C)CN(N2CCC(C(C)C)(CO)C2)C1)(C(C)C)SC.CC=O C1(CC(=O)NCC(CC)NC(=O)C(O)Cc2cccc(Cl)c2)CC2(CCC2)C1 c1(C(=O)Nc2cc(OC)c(C)cc2C)csc2c1CCN(Cc1ccccc1)C2 c1(C(N2C(C)CC(NC(c3cnc(S)nc3)=O)CC2)=O)nccc2c1NCCC2 C1(C(=O)O)(NC(C2CC2C2CCCO2)=O)CCS(=O)(=O)CC1 c1(CNC(C(CC)NC(=O)C=CC2CCC2)=O)cncc(C)c1 c1(C(=O)NC2CN(C(c3cc(C)c(C)[nH]3)=O)C(C)CC2)n[nH]c2c1NCCC2 c1(NC(CCC2N(C(c3c(C)cco3)=O)CCC2)=O)cc(C(N)=O)ccn1 N1(C(CC(CNC(C(C=C)(C)C)=O)C2CCC2)=O)CC2(CNC(=O)OC2)C1 c1(C(=O)NCC(C)N(C(C(CCC)OCC)=O)C)c(OCC2CC2)cccc1Cl C(C(=O)NC(C)(C)C=CC(=O)NOc1ccc(F)cc1)(C(C)C)OC C1(CNC(Cc2cc(C)[nH]n2)=O)C(C2CC2)CCN1C(c1cnccc1C#N)=O CC1CN(CC(O)COCC(F)(F)F)CCN1Cc1coc(C2CCOCC2)n1 CS(=O)(=O)c1ccccc1CN1CCCC(C(=O)NCc2c(Cl)cccc2Cl)C1 c1(C(=O)NCC2N(C(CC=CC)=O)CCC2)cc(F)c(F)cc1O Cc1cccc2c(C(=O)NC3(C)CN(C(=O)Cc4cc[nH]c(=N)c4)C3)n[nH]c12 N1(C(C=CC(C)C)=O)CCN(C)CC1CNC(c1[nH]c(=N)ccc1C)=O N1(C(C(CC)(C)O)=O)CCC(C)(Nc2ncc(C)cn2)CC1 Cc1cc(CC(=O)NCC2(C)CCN(C(C3CN(C(N)=O)C3)=O)C2)ccc1F Cc1cc(C)nc(N2CCCC(NC(=O)CCn3cccnc3=O)C2)n1 c1(C(N(CCN(C(C(C(=O)OC)(C)F)=O)C)C)=O)ccc(O)c(C)c1C Cc1csc(C(=O)NC2(c3ccc(-c4cncn4C)cc3)CCC2)c1C c1(OC)ccc(CC(C)CNC(=O)C(=O)N(C(C)C)Cc2ccoc2C)cc1F N1(C(C(CCC)CC2CCCC2)=O)CC2(CCN(C(C3(CF)CC3)=O)CC2)C1 CC(C)C(C(=O)NCC1C2CC1N(C(=O)CC(C)c1cccs1)C2)n1cnnn1 C1(CC(=O)N(CCCOCC)C)CC(C)(C)CN1C(=O)Cc1cccnc1 Nc1cc(Cl)cc(Cl)c1C(=O)NC1CCC1NC(=O)C=C1CCSCC1 C1(CCNC(C(C2CCCC2)OC)=O)CCN(C(=O)CCc2ccncn2)C1 c1(CC)nc(C)[nH]c1C(=O)NCC(C)N(C(=O)CCC1CC1(Cl)Cl)C n1(CCC(=O)OCC)nnnc1C(c1ccncc1)NC1(CF)COC1 C1(NC(c2c(C)snc2)=O)CC2C(NC(=O)CC3CCCN(C)C3)C2C1 Cc1nc(C=CC(N2CCOC(CNC(=O)CN(S(C)(=O)=O)C)C2)=O)cs1 N1(C2CC(=O)NC2)CCC2(CC(C(=O)N=c3cc[nH][nH]3)=NO2)C1 N12CCN(CC1)CC2=O.Cn1ccnc1SCC(=O)N(C1C2CCCC12)C1CC1 c1(C(=O)NCC23CC2CN(C(=O)Cc2nc(Cl)cs2)C3)c(Br)ccc2c1OCO2 c1(CC)oc(C)cc1C(=O)NC(CN(C(C1(C(F)(F)CC)CC1)=O)CC)CC c1(OCC=C)ccc(C(=O)NNC(=O)c2ccc(N(C)C)cc2)cc1[N+](=O)[O-] Cc1nc(CC(N2CCC(O)(CNC(=O)C(O)C(C)C)C2)=O)c(C)s1 C1(CC)CCCC1(C)C(N1CCC(CF)(NC(c2ccc(C(F)(F)F)[nH]2)=O)C1)=O CC1CC(C)N(C(=O)CNS(C)(=O)=O)CCN1C(c1ccc2nc(O)[nH]c2n1)=O CCCCCCC(F)C(=O)N1CCC(CN(C)C(C2(C(C)C)CC2)=O)C1 C#CCCCCCCC(=O)NCC(CC=C)NC(c1ccccc1)=O N1(C(C2CC(C)(C)O2)=O)CCC(O)(CCNC(=O)Cc2csc(Cl)c2)CC1 N1(C(=O)C=C2CCCCC2)CCOC2(C1)CN(C(=O)CNC(C1CCOC1)=O)C2 C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NC(C(C)NC(c1c(CC)cno1)=O)(C)C Cc1cc(=NC(=O)C(=O)NCC=CCNC(=O)Cc2ccc(C3CC3)cc2)[nH]o1 c1(C(N2CCC(C3CCC3)C2)C(=O)NCCOCC)cnc2ncccn12 C1(C(=O)NC2CCC(NC(c3ccc(F)o3)=O)CC2)CCc2nnc(O)n2C1 C12(C(=O)NCC(C)CN(C(=O)Cc3cncn3C3CC3)C)CC3CC1C2C3O c1(C(=O)NCC(CC)NC(C2CC(F)(CO)C2)=O)cncc(F)n1 S(=O)(=O)(c1cccc(F)c1)NCC(=O)NC1CCC(NC(C2(CO)CCC2)=O)C1 N1(C(c2c(C)cc[nH]2)=O)CC2OCC(NC(c3cccn4nccc34)=O)C2C1 C1(C)(CC)C=C(C(=O)NCC2CCC(NC(c3cc(SC)ccc3Cl)=O)CC2)C1 CC1=C(C)CC(C)(C(N2CC(CNC(=O)CP(C)(C)=O)C(C)(C)C2)=O)CC1 N1(C(CC2(CN(C(=O)CN3CCSCC3)C)CC2)=O)CC2(CCN2C)C1 C(C1CS(=O)(=O)c2ccccc21)CN1C(=O)CCN(C(=O)NCCCCl)CC1 CC(C)C(C(=O)N(CCC(C)NC(C1CC(C2CCC2)C1)=O)C)C(C)C c1(CC)cc(Cl)ccc1C(=O)NC1CCC(CNC(=O)CCC(N)=O)C1 c1(C(=O)NCC2C(C(N3C(CC(=O)OC)CCC3)=O)C2)ccc(C)c(C)n1 C1(CNC(C(=Cc2ccco2)C)=O)COCCN(C(=O)C(F)CC2CCCC2)C1 Cc1ccc(CNC(=O)C(C)NC(c2cnccn2)=O)c(F)c1 C=C1Cn2c(C(=O)NC34CCN(C(C5(C#N)CCOCC5)=O)CC3C4)nnc2S1 c1(N2CC=CC(NC(=O)CC3CC4(CC4)C3)C2)ccc2nnnn2n1 c1(C(N(C2CCCN(C(C3(CC)CCNC3=O)=O)C2)CC)=O)sc(C)cc1Cl N1(C(CSC)=O)CCCC2(NC(c3cnc(N(C)C)cn3)=O)CCCC12 Cc1cccc2cc(C(=O)NC3CCN(C(=O)CC4CCOC4)C(C)C3)[nH]c12 N1(C(C(CCC)C)=O)C2CCC1CN(C(c1cc(C(N)=O)cc(C)c1)=O)C2 C1(C(=O)NC2(CCCC)CC2)CCCCC1CNC(C1(C)CNC(=O)C1)=O C1(CC(N2CCC(F)(CO)C2)=O)CCCN(CC2CCCCO2)C1 C#CC1CC2(CC2)CN1C(c1ccnc(CNC(=O)C(C)(C)CC(F)F)c1)=O CC1CC(C(=O)OCC2CCCN2S(=O)(=O)CCCCC(=O)OC(C)(C)C)=NO1 N1(C(C(=O)OCC)=O)C2CC1CN(C(c1sc(C)nc1C(F)(F)F)=O)C2 N1(C(C(C(C)(C)O)F)=O)CCCC(C)(C)C1CNC(=O)CC1CCC1 c1(C(N(C)C)=O)ccnc2cc[nH]c12.C12CCCN1C2=O C1(OC)CC2(CCC(C(=O)NCC=CCNC(C3CC34CC(O)C4)=O)CC2)C1 C1(OC)C(N=c2[nH]c(=NCCc3c(C)noc3C)[nH]c3c2CCCC3)CC1(C)C C1(C(N2CCC(O)(Cn3cc(CC(C)(C)O)nn3)C2)=O)Cc2cc(Cl)ccc2O1 C1(CCCC)CN(C(=O)C(C)CSC)CCN1C(c1nn(C)cc1C)=O CC1=C(C(=O)N2CCC(NC(C3CC(F)(F)C3)=O)CC(C)(C)C2)C(C)(C)CCC1 C#Cc1cc(F)c(C(=O)NC2CC3(C2)CC3NC(c2coc(Cl)n2)=O)c(F)c1 N1(C(C(CSC)O)=O)CCCC2CN(C(=O)CNC(=O)Cn3cncn3)CC12 c1(C(N2CCC(CNC(c3cccc(C(C)C)n3)=O)C2)=O)ccc(N)c(F)c1 c1(CC)ccc(C)cc1C(N1CC(C(N)=O)(CNC(C2CCCC2C)=O)C1)=O C1(C(=O)NCC(CCOC)(C)C)C2CCCC2CN1C(=O)COCC(=O)OCC C1(CNC(C(c2ccc(C)cc2)C)=O)CCCCCN1C(c1nn(C)cc1Cl)=O Cc1ccc(C(=O)NCC2(CNC(=O)C(C)C(C)O)CCCC2)cc1Cl c1(CC)cc(C(=O)NC(C)CN(C(C23CC4CC2C3C4O)=O)CC)ccc1F Cc1cc(Br)cnc1C(=O)NCC(CC(F)(F)F)NC(C1CC1C1CC1)=O C1(NC(c2c(SC)cccc2)=O)CC1C1CCCN(C(=O)C=CBr)C1 C1(NC(c2cc(CC)nn2C)=O)CC2CN(C(=O)CC(=O)OC)CC12 C(=O)(N=c1ccn(C(F)F)[nH]1)C1(C)N(C(COCC(=O)NC)=O)CCC1 CN1CCN(C2CCN(C(C3C4CN(CCCC(F)(F)F)CC34)=O)CC2)CC1 O=C1N(CCc2cncnc2S)CC2CCCCN12 C(C(CC(F)(F)F)NC(c1ccnn1C1CC1)=O)NC(c1c(C(C)C)[nH]cc1)=O C1(C(N2CCCC(C(=O)NCCNC(C3CN(C)C3)=O)C2)=O)(CC)CCNC1=O c1(NCC(CCCCC)O)ncc(C)cc1S(=O)(=O)NC(c1ccccc1Cl)C Cc1cc(C(=O)NC(CCNC(c2csc(Cl)c2)=O)C(C)C)nn1C1CC1 c1(C(N2C(CO)CC(NC(CN(S(CC)(=O)=O)C)=O)C2)=O)cc2ccsc2n1C N1(C(C2C(OCC)CCC2)=O)C2CCC(C2)C1C(=O)Nc1cccnc1C(C)C CCC(CCCC(=O)N1C2CCC1(CO)CC2)NC(N1C(C(=O)OC)CCC1)=O c1(C(N2CCC(CNC(C(C)n3cnnn3)=O)C23CC3)=O)cn2ccncc2n1 C(C(C)CC(=O)N(C)CC1CCCN1C(C1(C(F)F)CC2(CC2)C1)=O)OC c1(CC)ccccc1OCCOCC(=O)NCCN(C(=O)C(C)CO)C(C)C N1(CC)N=C(C(=O)NCCC2CCCCN2C(=O)CCCCC(C)C)CCC1=O c1(NC(C(c2cc(Cl)cs2)N(CCN(CC)CC)CC)=O)cccc(Cl)c1C c1(C(N2CCCC(CC=C)(NC(CCC)=O)C2)=O)cc2c(cn1)OCCO2 C12(C(N3CCC(NC(C(c4ccccc4)C)=O)C3)=O)CC(C)(C1)OC2C c1(C(N2CC(C)C(CO)C2)C(=O)NC2CCC2)noc2cc(Br)ccc12 Cc1cccc(C2(C(=O)N(CC(C)N(C)C(c3cccnn3)=O)C)CCC2)c1 c1(-c2ccc(NC(C3C4CCC(F)(F)C34)=O)cc2)nnc2n1CCC2 CONC(=O)C(=O)NC(C)CNC(=O)Cc1ccc[nH]1 c1(OC)ccc(NC(=O)NNC(=O)c2cc(Br)c[nH]2)cc1.SC N1(C(c2c(OC)cc(C)s2)=O)CCCC12CCN(C(=O)C(C)NC(C)(C)C)C2 c1(C(=O)OCC)ccc2c(c1)CC(NC(=O)C(=O)NCCCCCCCO)C2 CC1CN(C(C2CC3C=CC2C3)=O)CCC1CNC(=O)CC1COC(=O)N1 c1(CNC2CN(C(Cc3c(C)ccc(Br)c3)=O)CC(F)C2)cc(F)cc(C#N)c1 Cn1c(=O)sc2cc(CNS(=O)(=O)c3ccc(Br)cc3Cl)ccc12 C1(CNC(C(N)=O)=O)CCCC(NC(=O)C=C2CCC(C(F)(F)F)CC2)C1 CC(CCc1ccccc1F)C(=O)NC1(CN(C)C(C2CC(=O)N(C)C2)=O)CC1 c1(C(=O)NC2(CC)CCCN(C(=O)CCC(C)(F)F)C2)ccc2nc[nH]c2n1 CC1CCCC1(C)NC(N1CCN(c2ccc(O)cc2)CC1)=O c1(C(N(CCCNC(=O)C=CC(N2CCC(F)C2)=O)CC)=O)cc(C)c(F)cn1 N1(C(C(N2CCOCC2)C)=O)CC(CNC(c2nn(C)cc2N)=O)CC12CCC2 N1(C(c2c(COC)noc2)=O)CC(NC(=O)CCC=CC(C)C)C2CCCC2C1 C=CC1(NC(C2(CC)CCN(C(C3COC(=O)N3C)=O)CC2)=O)CCCCC1 N1(C(C(CC)CC(C)C)=O)CCC(NC(=O)CC(F)(F)C(C)C)C2(CCC2)C1 C(=O)(C1=COCCC1)N1CCN(C2CN(C(C(OC)OC)=O)C2)CC1 C1(NC(c2c(O)nc(CC)c(C)c2)=O)CCC2(CC1)CN(C(=O)C(C)(C)F)C2 c1(C(N2CC(CC)C(NC(=O)C(F)F)CC2)=O)cc(S(=O)(=O)NC)cs1 C(=O)(C(O)C(C)C)N1CC(OCCNC(c2n(COC)ncc2)=O)C1 c1(C(N2C(CNC(C(C=C)(C)C)=O)C(C)(C)CC2)=O)ccc2c(c1)CCN(C)C2 c1(SC(C)C(=O)NCCCOCCC(=O)N(C(C)CO)C)ccccn1 C=CCC(C)(C)CC(=O)NC1CCCC1CNC(=O)COC(C)(C)C N1(NC(C23CC(n4cc(CN5CCC5CCO)nn4)C2C3)=O)CCC(O)CC1 N1(C(CCC=C=C)=O)CC(CNC(=O)CC2CCC(=O)NC2)C2(CCOCC2)C1 N1(C(c2ncc(C)nc2)=O)CCC2CN(C(c3ccc(F)c(F)c3Br)=O)CC2C1 N1(C(C2OCC(C)(C)C2)=O)CC(NC(=O)Nc2cncc(C#N)c2)C2(CCC2)C1 N1(C(c2cn(C)nc2I)C(=O)NC(C(=O)OC)CC(C)C)CCC(C)C(F)(F)C1 CC1CC(NC(C2(C)CC(C)(C)C2)=O)CCN1CCCN1C(=O)CNC1=O S(=O)(=O)(c1cc(NC(c2ccc(OC)cc2F)=O)c(Cl)c(F)c1)N(CC)CC N1(C(CCc2cnc(C)o2)=O)CC(O)CC1CNC(=O)CCN1CCCCC1 N1(C(CC2(C#N)CCC2)=O)CCCC2(CCCN2C(=O)CCc2nncs2)C1 C(=O)(N=c1cc(Br)n(C)[nH]1)C1CN(C(CS(Cc2scc(C)n2)(=O)=O)=O)C(C)CC1 Cc1ccc(O)nc1NC(=O)CSCCNC(C1CC(=O)C1(C)C)=O C(=O)(CC1=NN(C)C(=O)C1)N1CC(N(C(C2CCC(NC(CC)=O)C2)=O)C)C1 S(=O)(=O)(c1ccccc1)C(=O)NCC(N1CCC(C(C)NC(=O)C2=CCC2)C1)=O N1(C(C(CCCOC)C)=O)CCCN(C(=O)C(F)(F)CN2CCCC2)CC1C N1(C(C(CC=C)(C)C)=O)CCC(C2(NC(C3(SC)CCC3)=O)CC2)CC1 C(=O)(CCCCCC(C)C)NC(C(=O)NC1CCC(C)(OC)CC1)(C)CO Cc1nc2cccc(C(N3CCC4(CC3)CC4NC(=O)CO)=O)n2n1 CN1N=C(C(=O)N2CCC(n3cc(CC(=O)N4CC=CCO4)nn3)C(O)C2)CCC1=O c1(NC2C=CCN2)cccc(CC(=O)N(CCN(C)NC(CC)=O)C(C)C)c1.N c1(C(=O)NC2CN(C(C3C(C)(CC)C3)=O)C2)ccc(CCc2ccccc2)[nH]1 n1(CCCC)nc(C)c(C(N2CC(O)(CNC(=O)CC3CCOC3=O)C2)=O)c1Cl C(=O)(CCCC1CCC1)NCC(C1CCOC1)NC(C1(SC)CCC1)=O CCCCCCC(C)C(=O)N1CC2(C1)CN(C(=O)CCCn1nc(C)nc1C)C2 C1(CCNC(=O)Cc2cnccn2)COCCN1C(=O)Cc1cncs1 C1(C(=O)N(C)CC2(NC(=O)C(C)C(C)O)CC2)(COC)CCCCC1 n1(CC)nc(C2CC2)cc1C(=O)NCCC1CC(NC(=O)COC2CC=CC2)C1 C1(C(=O)NC2CN(C(C3CCC(C)CC3)=O)C2)CCCC2(CC2)C1 c1(CC(=O)N(C)CC2CCN(C(C3CC(F)(F)C3)=O)C2)csc2nccn12 C1(C(F)(F)F)(C(=O)NC(C)CCNC(C2(C(C)(C)O)CC2)=O)CC=CCO1 CON(CCO)C(=O)COC1CN(C(=O)C=C(C2CC2)C2CC2)C1 C(CCCC(CO)NC(C12CCC1C2)=O)NC(C1CCN(C)CC1)=O c1(C(N2CC(O)(CNC(C3CCn4cncc4C3)=O)C2)=O)ccc(F)c(F)c1F N1(C(CC)=O)CCN(C(=O)C(C(C)C)NC(N)=O)C2CCC12 c1(C(C)=O)ccc(SC(C)C(=O)NCc2ccc(Cl)cn2)cc1 C#Cc1cn(C)nc1C(=O)NCC(C1CCCCC1)NC(c1cn(CC)cn1)=O C1(OC)CCN(CC(=O)NC(=O)N(CC(N2CCCC(C)C2)=O)C)CC1O C(=O)(C1(C)CCCn2ccnc21)NC(c1ccc(Br)cc1F)(C)C C1(NC(C2CC3CCC3C2)=O)CCN(C(=O)C(F)(F)C2(O)CCCC2)CC1 c1(CNCC(CCC=C)O)cccn(C(c2ccccc2)C)c1=O CC(CC(=O)NCCCCO)C(C)(C)NC(c1cn2c(n1)CCC2)=O Cc1ccn(CC(=O)NCC2(O)CN(C(c3ccn(CC(F)F)n3)=O)C2)c(=O)c1 CCC(CC)C(C)C(=O)NCCCCNC(c1cnc2sccn12)=O c1(C(=O)NCc2c(CCNC(C(CC)N(C)C)=O)ocn2)nnc(O)cc1O C1(NC(C(c2cncnc2)C)=O)CCCC(C(=O)NC2(CCF)CC2)C1 c1(NCC(C2CCCCC2)OC)nnc(SC)n1CCC(C)(C)N1CCOCC1 N1(C(C=C(C)C2CC2)=O)CCC(C2CCCN(C(C3CCOC3)=O)CC2)CC1 c1(NC(C2C3CN(Cc4c(C)cc(C)[nH]4)CC32)=O)c(C)cc(F)cc1F CC1(C)CCC(NC(=O)CC(C2CCC(F)(F)CC2)N)c2ccccc21 C1(S(C)(=O)=O)(C(=O)NC(C2OCCN(C(C3C(CC)C3)=O)C2)C)CCC1 N12CCC(O)C(C1)C2=O.c1(C(=O)OC(C)(C)C)ccsc1CN1CCCCC1 c1(C(N2C(CNC(c3c(C)[nH]c(C#N)c3)=O)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(CNC2(C#C)CC(C(=O)OC)C2)ccc(C(F)(F)F)c(F)c1 c1(NC(C2(C)CCN(C(c3cc(F)cc(F)c3)=O)C2)=O)ncc(Cl)nc1Br C1(COC)(NC(c2ccn(CCF)n2)=O)CCCN(C(=O)C(F)C(C)C)C1 CCCCCC(O)CC(=O)NC(C)CCCNC(c1cc(F)cc(Cl)c1)=O c1(C(N2CC(NC(C3CCCSS3)=O)CC3(C2)CC3)=O)cc(F)c(F)c(O)c1F C1(CNC(=O)C=Cc2ccco2)CC2CCC(C1)N2C(=O)CCC(F)F c1(C(=O)NC(CN(C(C2(CC#C)CCOC2)=O)C)C)cc2nnn(C)c2s1 C1(C)(CC)CCN(S(=O)(=O)N(C)CC2CCCCC2)C1 C1(C2CC2)(NC(C(F)=C(C)C)=O)CCN(C(=O)C(c2ccc(Cl)cc2)=O)C1 c1(C(=O)Nc2nccc(OC)c2)ncn2c1CCCC2 Cc1nocc1NC(=O)CC1CCN(C(C)CC2(C)OCCO2)C1 c1(CCC(=O)NCCC2(O)CCN(C(C3CCSC3)=O)C2)nc2cccnc2[nH]1 c1(C(=O)NC2CN(C3CN(C(CSC(=N)N)=O)C3)C(=O)C2)csc2cncn12 Cn1nc2c(c1C(=O)Nc1ncc(Br)nc1I)CN(Cc1ccccc1I)CC2 C(=O)(C1=CCCOC1)NC(CN1CCN(C(COCCC#C)=O)CC1)(C)C C1(CC)CN(C(=O)CC2CCC(=O)N2)CCN1C(=O)CC1(COC)CCOCC1 CC1CN(C(=O)C(Cc2cnn(C)c2O)NC(=O)CC(=O)NC2CC2)CCN1C N1(C(C2CN(C(C)C)C2)=O)CCC2(COC(CNC(C3CC3F)=O)C2)C1 C1(NC(C(c2ccccc2)NC(=O)NC)=O)CCOCC1NC(C1(Cl)CC1)=O c1(C(=O)NC(CNC(C2CC(CC)OCC2)=O)(C)C)cn(C(C)C)c(=O)nc1O c1(C(=O)NC(CNC(C(CC)(C)C)=O)(C)CC)coc2c1CS(=O)(=O)C2 Cc1sc(C(N2CCCC2CCNC(=O)C(C)CC2CC2)=O)nc1O c1(CC(N2CCN(C(C(C(C)C)F)=O)C(C3CCC3)C2)=O)cccc2nonc12 N1(CCN2CCCC(NC(Cc3cc(C)ncn3)=O)C2C)C(=O)NC(C)(C)C1=O c1(C(=O)NC(C(=O)NC(c2n(CC)ncc2)C)CC2CC2)cccc2[nH]ccc12 C1(C(=O)OCCC2CC2(Br)Br)CC(=O)N(C2CCCCC2)C1 C1(C(=O)NCC2(CC(C)C)CC2)CCC(C)(C)N(C(C2CCCN2C=O)=O)C1 CCC(C)C(C(=O)NC1CC(CC(C)(C)C)C1)N(C(=O)Cn1ncccc1=O)C c1(C(=O)NC(C2CN(C(=O)C(F)C3CCC3)C2)C)ccc(OC(F)(F)F)nc1 N1(C(C2CC(C#N)C2)=O)CCCC12CCCN(C(c1cc(Cl)c(F)cc1Cl)=O)C2 CN1CC(=O)Nc2ccc(C(=O)NCC34CC(NC(C5COC5)=O)(C3)C4)cc21 CCC(C(=O)NCCCN(C(=O)Cc1cnn(C2CC2)c1)C(C)C)OC C1(C(C(=O)NCCc2cc(C)no2)C)CCCN(C(c2c[nH]cc2C)=O)C1 C1(CNC(C(N2CCNC2=O)C)=O)(CO)CCN(C(=O)Cc2cnn(C)c2O)C1 C(CCCC(=O)N1CCC(NC(c2cc(CS(C)(=O)=O)c(C)s2)=O)CC1)OCC CC1=C(C)CC(C(N2CCC(O)CC2C(=O)NC2CCCCCCC2)=O)CC1 C1(NC(c2cc(C(F)(F)F)ncc2Br)c2n(C)nnn2)CCCC12CCOCC2 n1(CC(N2C(c3c(C)cccc3)CCC2)=O)nc(C)c(C(=O)O)c1C c1(NC(c2nc(C(N3CC(O)C3)=O)cs2)=O)cc(O)ccc1Cl c1(SC)ccccc1C(=O)NC(c1ccccc1OCC1CC2(C1)N=N2)C1CC1 CCC(CC(=O)N(C)CC1(O)CCN(C(=O)CC2(C#N)CCCCC2)C1)C(C)C C1(S(C)(=O)=O)(C(=O)NC(C2CN(C(C3CC4CCC3C4)=O)C2)C)CCOCC1 C1(C(N(CCNC(c2cc(COC)on2)=O)CCOCCO)=O)C2COCC12 N1(C(c2c(C)cnn2C)=O)CCCN(C(C2CC(C)N(C)C2)=O)C(CO)C1 c1(C(N(C2CCN(C(=O)C(C)CO)CC2)CC)=O)noc2ccc(Cl)cc12 N1(C(C#CC(C)C)=O)CC=C(C(C)(C)C(=O)NCCCCCC2CC2)C1 c1(C(=O)NCC2CCN(C(CNC(CNC(C)=O)=O)=O)C2)cc(Cl)c(F)c(Cl)c1 c1(NC(CCC)CCOC)cc(Br)ccc1S(=O)(=O)NCc1cc(C)cc(C)n1 CN=c1[nH]cc(C(N2CCCC(N(C(=O)C(C)SC(C)C)CC3CC3)C2)=O)s1 C12(C(N(CC(C)NC(c3cc4cccnn4n3)=O)C)=O)CCC(CO)(CC1)CC2 c1(N2CC(C)C(NC(=O)CC3CCCC3(F)F)CC2)ncnc2sc3c(c12)CCC3 C(CC(C)(C)CNC(=O)CCCOc1ccccc1F)NC(C(CC)O)=O CCC(C)C(C(=O)N1CCC1Cn1cc(-c2ccc(OC)c(N)c2)nn1)N(C)C C1(CNC(N2CCCCC(C(=O)OC)C2)=O)CCCCCCCCCCCC1 C1(NC(C2(NC(CCCCC=C)=O)CCCC2)=O)CCCC(C2CC2)C1 CCCCCC(C)(c1nnnn1C1CCOC1)NCc1cc(Cl)cs1 Cc1nn2c(c1C(=O)NCC1(C)CC(NC(=O)CC3CC=CCC3)C1)CCCC2 n1(CC(=O)NCC2CC(F)CN2C(c2cnsn2)=O)cccnc1=O N1(C(c2cc(C)ns2)=O)CC(C(=O)NCc2nonc2C)C2(CCC2)C1 c1(C(=O)NC2C(NC(C3CN(C(=O)NCC)C3)=O)C2)nnc(O)nc1O CC1CN(C(=O)CCOCC(F)F)CC(C)C1NC(c1ccc(S(C)(=O)=O)o1)=O C(CC(C(=O)N(C(C)(C)CC(=O)NCc1cocn1)C)OC)OC c1(NC)ccccc1C(=O)NC(C(=O)N1CCC(F)(F)C1)C(C)C CC1=C(C)CC(C(=O)NC(C)CNC(c2cn(C)[nH]c2=N)=O)CC1 C12(C(=O)NCC(C)(CO)NC(c3ccc(O)nc3Cl)=O)CC3CC(CC(C3)O1)C2 C12(NC(CS(CC)(=O)=O)=O)CCN(C(c3cnc(O)o3)=O)CCC1C2 C(C)(C)(CCC(=O)NC1CC(CNC(C2CCO2)=O)C1)OC C1(NC(c2nc(C)sc2)=O)CCCN(C(C23COC(CF)(C2)C3)=O)CC1 C1(CC2C=CCOC2)CCN(CCc2csc(-c3ncccn3)n2)CC1 CN1CCC2(CCN(C(C3(CNC(C4CCCCN4C)=O)CC3)=O)C2)C1 c1(C(N2C(CNC(C(CCC)c3ccccc3)=O)CC2)=O)nc(O)[nH]c(=O)n1 N1(C(C=CC(CC)C)=O)CCCC(NC(c2cnc(C)c(Cl)c2)=O)C1C CC1(C)CC(CNC(=O)CC2(O)CCC2)CN(C(c2cnoc2C2CCC2)=O)C1 C1(NC(c2cn(C)nc2C(C)(C)C)=O)CN(C(C2(N=[N+]=[N-])CC2)=O)CC1C1CC1 Cc1ccc2c(=O)c(C(=O)NC(C)(C)CNC(=O)CC3CCCC3)c[nH]c2c1 c1(C(=O)NCC(CNC(Cc2c(C)cc(C)s2)=O)F)cnn2ccc(O)nc12 CCC(C)(C(=O)NCC1(O)CCN(C(=O)CN2CCS(=O)CC2)C1)C(N)=O C1(C(=O)NC(c2ccc(OC)cc2)CC)CC2COCC(C1)C2N c12ccc(C)cc1S2.c1(OCC)nccc(N2CC3CCC2C3)n1 c1(N(C2CN(C(C=CCCC=C(C)C)=O)C2)C(=O)CC23CC(C2)C3)ccccc1 C(=O)(C(F)(F)C(C)(C)O)NCC(CC)(C)NC(=O)C(O)Cc1ccccc1 c1(C(=O)NCCn2cc(C(=O)NC3(CC=C)CCC3)nn2)ccncc1N c1(N2CCC(O)(C(=O)Nc3c(C)nn(C)c3)C2)nc(S(C)(=O)=O)ncc1C N1(C(C(C2(C)CC2)NC(C(C(C)C)O)=O)=O)CCOC2(CCC2)C1 c1(C(C)C)ccc(C(OCOC(C)C)C)cc1.C1CCSCCN1 C(=O)(CC=C(Cl)Cl)N1CCC(CNC(C(CSC)=O)=O)C1 Cn1cc(C=CC(=O)NCCC(O)CNC(=O)Cc2cccc(Br)c2)nn1 Cc1sc(Cl)c(C(N2CCCC(C)(C(=O)NC3C4CC5C(C4=O)C35)C2)=O)c1C N1(C(C(CC(C)C)CNC(=O)CCCCN(C)C)=O)CCc2ccc(F)cc21 C1(C(NOC(C=C)C)=O)(NC(=O)CCC2CCOCC2)CCN(C)C1 c1(OC)ccc2c(c1)OCC1C2OCCN1C(=O)NCCc1cc(C)ccc1F C1(N(C(C2N(C(CCN(C(C)=O)C)=O)CC(C)C2)=O)C)CC(C)CC(C)C1 C(C)(CO)(C(=O)N1CC(C(O)C(N2CCOC(CN=[N+]=[N-])C2)=O)C1)OC c1(C(=O)NCC(n2cc(-c3c(C(=O)OC)n[nH]c3)nn2)C)ccc2sccc2c1 c1(C(N2CC=CC(NC(c3cnn(C)c3F)=O)C2)=O)cc2nccnc2cc1F N1(C(C(C)(C)C)=O)CC2CCC(NC(=O)CCc3cccc(C(=O)OC)c3)(C2)C1 N1(C(c2c(CC)nn[nH]2)=O)CCOC(C(C)NC(C2(CO)CCCC2)=O)C1 C1(CNC(=O)Cn2cc(Cl)cn2)CN(C(=O)Cc2ccsn2)C2CC12 CC1=CCC(C(=O)NCc2cn(C3CN(C(=O)CCCN(C)C)C3)nn2)CC1 CC(C)CC(CNC(=O)C(C)C(C)C)C(=O)NC(C(C)(C)CO)C1CC1 c1(C(N2CCCC(C)(NC(=O)CN3CCC(F)(F)C3)C2)=O)ccc(F)c(N)c1F C(=O)(CC(CC)CCCC)NC(CC=CC)C(=O)NCc1ccncc1Cl c1(C(=O)NC2C(C)CCN(C(C(CC)=CCCC)=O)C2)cnc2ccc(C)cn12 N1(C(C2OCCN(C(C=CC(C)C)=O)C2)=O)CCCC12CCOC2 C1(C(N(CCN(C(COCC(=C)C)=O)CC)CC)=O)CCc2nn[nH]c2C1 C(=O)(C1=CC2C=CC1C2)N(C(C(=O)N(C(CC(CC)C)C)C)C)C CCC(C(=O)NC1(C(=O)N(C(C)CC(C)C)C)CC1C)OC N1(C(CCCC(C)C)=O)CC2(CCC(CNC(=O)C(F)(F)c3nccs3)O2)C1 CCC(C)C(C(=O)N1CCC1CNC(=O)Cc1ccc(C)nc1O)NC(=O)OC CCN(C)NC(=O)C(C1CCCCC1)N1CCCC1 C1(CC(=O)NC(C2CN(C(c3cccs3)=O)CCO2)C)CC2CCC1CC2 Cc1ccc(C(N2CC(C)(C)CC2CNC(=O)C(C)n2ccnn2)=O)c(F)c1 c1(C(C(=O)NC2CCCN(C(c3c(C)nccc3)=O)C2)=O)ccc(Cl)cc1O N1(C(C(C)(C)n2ccnn2)=O)CCC2(C=C(C(=O)Nc3ccc(F)c(F)c3)C2)C1 c1(OC)ccc(C(N2CCC(NC(=O)C(C)CC(C)(F)F)CC2)=O)c2sccc12 c1(CCC(=O)NC(C(=O)OC)C2(C(F)(F)F)CC2)ccc(O)c(OC)c1 C1(NC(C2CC(NC(CN(C)C)=O)C2)=O)CC(N(C)C)C(O)C1 C#Cc1ccc(NC(=O)C(c2ccccc2)NC(C2(C#C)CCCCC2)=O)cn1 c1(N2CCC(NC(C3CCCN3C(C3CCC3)=O)=O)CC2)ncc(Cl)cc1Cl N1(C(C2(C(=O)OC)CCCC2)=O)CC2CC2(CN2CCNC(=O)C2)C1 C1(NC(CC(C)(C)F)=O)CCCN(C(=O)CCc2ccc(Cl)cc2Cl)CC1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(C)(C)C1C(=O)NOCC1CCCCC1 C1(NC(CN(C)CC)=O)CN(C(=O)CCC2CC2(C)C)C2(CCOCC2)C1 CCC(C(C)(C)O)NC(C1CCC(NC(C2CCC(=O)C2)=O)CC1)=O CC1(C)Cc2cc(C(=O)NC3CCN(C(C4CC(C)(O)C4)=O)C34CC4)sc2C1 C1(NC(CCOCC)=O)CCCC(C(=O)NCC2(C#N)CCC2)CC1 CC(C)CC(C(=O)NCC(C)CN(C)C)ONC(c1occc1C(C)C)=O c1(CC)nc(O)c(C(=O)NC2CCN(C(=O)CC3C=CCCC3)CC2)cc1C c1(OC)ccc(C#N)c(NC(C2CCCC(NCC3(F)CCC3)C2)=O)c1 Cc1ccc(C(=O)NC(C)CCNC(C2(CC(C)C)CCC2)=O)cc1Cl N1(C(C(C)=C(C)C)=O)CC2CCC(CNC(=O)Cc3cncs3)C2C1 C1(CC(=O)N(C2CCN(C(=O)CCc3ccoc3C)C2)CC#C)CC(=O)NC1=O O=NN1CCCC1C(=O)NCCC1CC(NC(C23CC(C#N)(C2)C3)=O)C1 Cc1noc(C)c1C(C)CC(=O)NC1CCN(C(=O)CCc2nc[nH]n2)C1 C1(C(=O)NC2CC(C)(NC(COc3cc(C)on3)=O)C2)CC(=O)N(O)C1 N1(CCC(=O)N(CC(C)NC(CCc2c(C)ccnc2)=O)C)CCSC(C)(C)C1 N1(C(C2C(C(=O)OC)C2)=O)C2CCC1(CNC(=O)CC1CCCC(F)(F)C1)CC2 N1(C(CC=C(C)C)=O)CC(O)CC1C(=O)Nc1cnoc1 c1(N2CC(C(=O)Nc3c(OC)nccc3C)SCC2)ncnn2ccc(Br)c12 C=CCCCCC(=O)NC(C)CNC(C1CC1c1ccccc1)=O c1(C(=O)NC2CC(NC(Cc3c(C)cccc3)=O)C(O)C2)c(Cl)ccc(F)c1N C(=O)(C1=CCCSC1)NCC1CC(N(C(=O)CCCNS(C)(=O)=O)C)C1 C(=O)(C1=CCCOCC1)NCC1N(C(C(C2CCOCC2)OC)=O)CC1 CCC(CC)CC(=O)N1CC2CC(NC(C3CCN(C(=O)NC(C)C)C3)=O)C2C1 CC1=CCN(CCNC(c2coc(C(=O)NC3C4CCCC34)n2)=O)CC1 N1(C(CN(C2CCCC2)C)=O)CC2CCC1C2NC(=O)COCCF.C1(C)(O)CCC1 Cc1ccc(Br)c(CC(=O)NCCOCCCNC(c2cc(C)on2)=O)c1 c1(C(N(C2CCN(C(C(CC#C)C)=O)C2)C)=O)ncc(C(=O)OC)cc1Cl C(=O)(CC(C)C(C)C)N1C(CCNC(c2nc(C)n(C)c2)=O)CCCC1 C1(NC(=O)C#CC2CCCO2)CCc2cnn(CCCC(F)(F)F)c2C1 c1(C(=O)NC2C(NC(c3cc(COC)no3)=O)C2)cnc([N+](=O)[O-])n1C CC1CC(c2ccccc2)CCN1CC1CCCC1.c12occc1C(=O)NC2 N1(C(c2cncc(N)n2)=O)CCCCC(CNC(c2cc(Cl)cs2)=O)C1 C=CCC(CNC(C1(SC)CCOCC1)=O)C(=O)N(CC)Cc1ccc(Br)cc1 C1(CN(C(C2(CC#C)CCOC2)=O)C)CN(C(c2ccoc2C)=O)CCO1 c1(C(=O)NC(C2CN(C(CNC(=O)OCC=C)=O)C2)C)ns[nH]c1=O.C(=O)OC Cc1cc(I)ccc1C(=O)NC1CC(NC(c2c(Cl)ccnc2Cl)=O)C1 c1(OC(C)C)ncccc1C(=O)NCC(C)NC(C1CCSC1)=O C1(CC=C)CC(OC2C#CCCCCC2)CC(CC(=O)OCC)O1 Cc1ccc(CC(=O)NC2CC23CCN(C(C2CCC(C)C2)=O)C3)cc1F N1(C(CCOC)=O)CCCN(C(=O)C(c2ccccc2F)C)C(C)C1 C1(C)(C(=O)OCC)CCCN1CC1CCC(C(F)(F)F)CC1 C(C(=O)NCC1(CC)CC(C)(C)C1)(C(C)C)NC(COCCC=C)=O C1(CNC(c2nc(C(C)OCC)sc2)=O)CC2(C1)CN(C(=O)Cc1csnn1)C2 N1(C(c2c(C)sc(O)n2)=O)CCCCCC1CNC(C12CCC(CO)(CC1)C2)=O Cc1cnc(NCC(C)NC(c2nn(C)c(Cl)c2Cl)=O)nc1S(C)(=O)=O C1(C(=O)OC)CC2(CCN(C(C3CC3CNCCOc3ccccc3Cl)=O)C2)C1 Cc1ccc(Cc2cn(NC(CCCSCCC3CCCC4CC34)=O)nn2)cc1 CC(F)CC(=O)NCCOCc1ccccn1.C12CCCN1CCCNC2=O C1(COC)(CNC(=O)Cn2cncc2C)CCCN1C(c1cc(C#N)no1)=O Cc1cccc2sc(C(=O)NC3CCC4CC3CN4C(=O)C(C)C)c(Cl)c12 c1(NC(C2N(C(C3C(C)=C3)=O)CC(F)C2)=O)sc(C)c(C)c1C(=O)OC C1(CCNC(c2n(CC)ncn2)=O)COCCN1C(=O)CCOCCCOC Cn1ccc(=NC(=O)C23CCCC2CN(C(c2c(Cl)cnn2C)=O)C3)[nH]1 n1(CC(N2C(C)CCC(NC(=O)CCC(F)F)C2)=O)cc2ccccc2n1 N1(C(c2nncc(NC)c2)=O)CC2CCC1C(CC)C2.C12CC(C1)C(=O)NC2 C=CCC(C(=O)N1CC2(CC(CC(=O)NCC3CCOC3=O)C2)C1)C(C)C N(C)(CP(C)(C)=O)C(C1(NC(c2cnc(C)o2)=O)CCSC1)=O Cc1ccccc1C(C)CC(=O)NC1CCC1CNC(c1c(C)cnn1C)=O C(=O)(C1CCCc2nn[nH]c21)NC(CCOC)CNC(=O)CCC1CCC1 c1(C(=O)NCC2(O)CN(C(C3(CC#C)CCCO3)=O)C2)nc(C)c(C)nc1O CC1CN(C(=O)CCc2nccn2C)CCCN1C(c1cnc2[nH]cncc1-2)=O N1(C(CSCC(=O)OC)=O)CC2CCC1C(NC(c1c(Cl)csc1Cl)=O)C2 C1(COC)(CNC(=O)C(N)=O)CCN(C(C2CCCN2C2CC2)=O)C1 C12(CNC(C(CC)(C)C)=O)CCCC1CCN2C(c1ccc(C(N)=O)o1)=O c1(CC)cc(C(=O)NC2CCC(NC(=O)CC3CC3CC)C2)ccc1F c1(C(=O)NCC(CC=C)NC(=O)C(CO)N(C)C)cnc(C(N)=O)cn1 C12(CNC(CC)=O)CCC(CNC(=O)C3=CCC3)(CC1)CO2 O(N1CCC(N=O)CC1)CC(=O)NC(CC(C)C)C(=O)O N1(Cc2cn(CC(C)C)nc2)CCC(O)C(C(=O)NCc2ccccc2F)C1 c1(OC)cccc(C(=O)N(C)CCN(C(=O)C=C2CCC(C)C2)C(C)C)c1 C1(C(=O)NCCCCC(=O)N2CC(C(CC)C)C2)CC12CCOCC2 Cc1nc(C=CC(N2CCCC2CNC(C2CC(C)(O)C2)=O)=O)[nH]c1C C(CC(C)(C)CC(=O)NCc1ccc(C(N2CC3CCC3(C)C2)=O)s1)OC C(C(CC1CCCC1)CO)NC(COCCNC(C=CC)=O)=O Cc1ccc2oc(C(=O)NCC(C3CC3)N(C(=O)C(C)C(C)(F)F)C)c(C)c2c1 CC1=C(C(=O)NC(CC(=O)NCC(C)(C)C2CCCO2)C(F)F)COCC1 N1(C(CC2C(C)CCN(C(=O)CCC(C)(C)C)C2)=O)CC2CC(C1)N(C)C2 CCCC(C#N)C(=O)N1CCN(C(CNC(c2cc(C)c(C)o2)=O)C(F)F)CC1 c1(C(=O)NCC(C)N(C)C(c2ccc(-c3ccncc3)s2)=O)nc(=N)cc[nH]1 c1(CC)ccc(OC)cc1C(=O)NCCC1COCCN1C(=O)C(C)C(C)(F)F N1(C(c2c(C)ocn2)=O)CC2CC2(NC(=O)C(C2CCCC2)C2CCCC2)C1 c1(C(=O)OC)cc(CC(=O)NC23CC2CN(Cc2cnccc2Cl)C3)ccc1C N1(C(c2nc(COC)oc2)=O)CCCC(CNC(C2(C3CC3)CC2)=O)CC1 N1(C(c2nc(CC)sc2)=O)CCC(C)C(N(C(=O)CCc2cncc(F)c2)C)C1 S(=O)(=O)(c1cccnc1N1CCC(C#N)C1)NCC1OCCN(C(C)(C)C)C1 c1(-c2ccc(C(C)(C)C#N)s2)ccncc1.CCC Cc1nc2cc(Br)cc(NC(c3ccc(Cn4cccn4)o3)=O)c2o1 c1(C2(C(N3CCC(N)CC3)=O)CC2)c(Cl)cccc1Cl N1(C(c2cc(COC)[nH]n2)=O)CC2CCC2(CNC(=O)CCC(C)N(C)C)C1 c1(C(=O)NC(C(C)NC(C2CCCCC23CC3)=O)(C)C)cc2cccc(F)c2s1 C1(=O)C(N)COC(=O)N2CC(C2)N1C.c1(Oc2ccccc2)ccccc1 N1(C2CCN(C(C(C)=C(C)C)=O)C2)CCN(C(=O)CC2OCCC2C)CC1 CC1OC2(CNCC(c3cccc(Cl)c3)O)CC1(CO)C2 c1(C(=O)NC(c2ccccc2F)CNC(c2ccc(C)s2)=O)cncc(N)c1 CC(C)(CC(=O)NC1CN(C(C2CCN(C(N)=O)CC2)=O)C2CC12)c1cccs1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CC2CCN(C(c3cn(C)nn3)=O)CC2C1 c1(NC(=O)CC2C3CCCC3N2C(C2CCCCC2)=O)cc(C(N)=O)cc(F)c1 C(=O)(CCCCC(C)C)NCCC(=C)CNC(c1c(Cl)sc(C)c1C)=O C(C(C)(C)NC(=O)C=CC(=O)OC)=CC(=O)NCC.C1(=O)C(C2CCOC2)N1 N1(C2CC(OCC#C)C2(CC)CC)CC2CN(C(C)C)CC2C1 CC(C)(C)C(C)(C)C(=O)N1CCOC(CC(=O)NCC(F)CO)C1 Cc1cc(C)c(S(=O)(=O)N2CCC(c3ccc(F)cc3Cl)C2)cc1[N+](=O)[O-] c1(C(=O)NCC(C2CCCCCC2)(C)O)cc2c[nH]nc2s1 c1(C(=O)NC(CNC(C2CC3C(C2)C3(F)F)=O)CO)cccc2nccn12 C12(C(=O)NC(CCN(C(c3ccc(C)cc3C)=O)C)C)C3C4C1C1C2C3C41C CC(C)CC(C)C(=O)NCC1(O)CC(C(=O)NCC(O)C2CC2)C1 C1(CC(=O)NC(CN(C(C)=O)C)C)CN(C(=O)CN2CCCNC2=O)CCC1C Cc1cnc(CN2CCC(C#N)(NC(=O)CC3COCCO3)C2)c(F)c1 c1(C(N2C(CC(=O)NC(c3n[nH]c(C4CC4)n3)C)CCC2)=O)ccc(C#N)cc1 N1(C(CNC(C(CC)C)=O)=O)CCN(C(c2coc(C3CC3)n2)=O)CC1C C1(CC(=O)NC(C)CCN(C)C)CN(C(=O)CC2CCCC(=O)N2)C(C)(C)C1 c1(C2CCOCC2)cccc(F)n1.C1(C(=O)NCCc2c[nH]nn2)C2CC3C(C2)C13 C(CNC(=O)CN1CC2CCC1C2)(CC(F)(F)F)NC(C=CC=C)=O.CCCCCC=C N1(C(C=C(COC)C)=O)CC(N(C(=O)CC(C)(N(C)C)SC)C)C2(CC2)C1 N1(C(C(C)=C2CCC2)=O)CC2CC(NC(=O)C(C)(C)c3cncnc3)C2C1 CCCS(=O)(=O)CC(=O)NCC12CN(C(=O)C(C)(C)n3cccn3)CC1CCO2 N1(C(c2c(C(C)C)c[nH]n2)=O)CCOC(CNC(C2CC3C=CC2O3)=O)C1 C12(CNC(C3(C#C)CC3)=O)CCC1CCN2C(=O)Cc1ccc(C#N)cc1 c1(CC)cc(N2CCC(C(C)NC(c3oc(C(F)(F)F)nc3C)=O)C2)ncn1 CC1CC(C(=O)NCC(O)CNC(c2ccnc(Cl)c2N)=O)CC(C)C1 c1(CC)oc(C)cc1C(=O)NCCCCC(C)NC(c1ccnn1C(C)CC)=O C1(C(N(CCOC)CC2CC2)=O)(CCNC(C2CC(OC)C2)=O)CCC1 N1(C(C(C)NC(=O)NCC)=O)CCCC(C(=O)NCC(c2ccccn2)O)CC1 c1(N2CCOCC(NC(c3c(C(C)C)cccc3)=O)C2)c(Br)cccc1[N+](=O)[O-] C#Cc1cccc(C(=O)NC2CCCC2NC(=O)CCCN=[N+]=[N-])c1 C1(CC)(CC)CC(C(N2CCC(C(F)C(=O)N3CC(CF)C3)C2)=O)C1 n1(CCC(=O)NCCCN(C(=O)C(O)C(C)CC)CCC)c(C)c(C)sc1=O C(=O)(CC(=O)NCn1cc(C)nn1)C1(C(=O)N(C)C)CC1.C12CCC(C1)C2.CO n1(CC(C)O)cc(C(=O)NC23CC2CN(C(c2nnc(S)n2C)=O)C3)ccc1=O CC1CCN(C(=O)CC2CCN(C(c3ccn(C)n3)=O)CC2)CC1N(C1CC1)C C1(O)(CS(=O)(=O)NCCCC)CCCC(C)C1 N1(C(c2ccc(CC)cn2)=O)CCOCC(CNC(=O)CC(C)n2ccnc2)C1 O=C1CCC(CC(N2CCCC(CCNC(=O)CCc3ncco3)C2)=O)CN1 c1(CC(=O)NCC2(F)CCN(C(C(C(=O)OC)F)=O)C2)ccc(C)c(OC)c1 N1(C(c2ccc(Cl)s2)C(=O)NCC2CC2)CCCCC1c1ccccn1 CN1CCC(C(F)(F)F)(CNC(C2CC2C(=O)NCCC2CCC3CC23)=O)C1 N1(C(C2CCCS2)=O)CCCC2(CCN(C(=O)Cc3csc4nccn34)CC2)C1 c1(NCC(C)CO)nc(N2CCCNC(=O)CC2)nc2ncn(C)c12 CC12CN(C(c3cccnc3S)=O)CC1(C)CN(c1ccnc(S(C)(=O)=O)n1)C2 N1(C(c2ccc(CC)o2)=O)CCCCC1CC(N1CCC(C)(F)C1)=O c1(OC)ccc(N)c(C(=O)NC(C)(C)C(C)NC(C2CCCNS2(=O)=O)=O)c1 C1(C(=O)NC2C(NC(CN3CC(C)C3)=O)COC2)CC(C2CCOCC2)=NO1 C(=O)(CC1=NNC(=O)C1)NC(CSC)OC.C12CC(C1)N2 CCCC#CC(C)(C)NC(=O)C(C)NC(=O)C(C)n1cccn1 C(=O)(CS(=O)(=O)CCOC)N1CCC(CC#C)(C(=O)N(CC(C)CCC)CC)C1 c1(CNC(C(CC)C)=O)ccc(C2(CNC(=O)CNS(=O)(=O)NC)CC2)cc1 C1(C(N2C(C)CN(C(c3coc(Cl)n3)=O)CCC2)=O)CC(c2ccncc2)=NO1 c1(SC)ccccc1C(=O)N(CCF)CCNC(C)=O C1(C(N(C2CC(C#N)C2)CC(=O)N(C)Cc2cnsc2)=O)CC12CCOCC2 C1(C(=O)NCC2OCCC(NC(C(CN(C)C)(C)C)=O)C2)C(F)(F)C12CCC2 c1(OCC)ccc(N)c(C(=O)NC2CC3CC(NC(=O)CS(C)(=O)=O)C2C3)c1 O(NC(=O)CN=c1ccnc(N2CCCC(NS(C)(=O)=O)C2)[nH]1)CC n1(CC)cc(NC(=O)NC2CCCC(C(=O)OC)C2)ccc1=O c1(-c2ccc(NC3C(OC)CN(C(C)=O)C3)nc2)ccc([N+](=O)[O-])cc1F CC1CC(C(=O)N2CC=CC2(C)C(N2CCOC(C)C2)=O)=NO1 c1(C(=O)NC(CNC(C(CCC)C)=O)COC)ccc2c(c1)N(C)C(=O)C2 c1(C(=O)NCCC2CCN(C(CCC#CC)=O)C(C)C2)ccc2[nH]c(=N)oc2c1 c1(OC)cncnc1C(N1CCC(C)(C(=O)OC)C1)=O.C(C=O)(C1CCC1)N c1(C(=O)NC(CN(C(=O)C(C)NC(C)=O)CC)C)cccc([N+](=O)[O-])c1N c1(C(=O)NCC(C)CNC(=O)C(C)(C)c2ccno2)ccc2nccn2c1 C1(C(=O)NCC2CCCN(C(C=CC3N(C)CCC3)=O)C2)CC2CCC1C21CC1 c1(C(=O)NCCCN(C2CCCC2)C(C2CCC(=O)N2)=O)ccccc1F c1(-c2cnc(OCC)nc2)cccc2[nH]nc(C(=O)NCCc3nn[nH]n3)c12 c1(CC(N2CC(N(C)C(c3cc(Br)no3)=O)C2)=O)ncc(F)cc1F N1(C(CSCCCC)=O)CCC(C(=O)NCC2CC2)C12CC2 Cn1cnc2ccc(C(N3CCCCC(CNC(=O)C(O)CC(N)=O)C3)=O)nc12 CCCC(C)C(=O)NCCC1CCCN(C(C2(CC)COC2)=O)C1 C(=O)(CN=S(C)(C)=O)NCc1c(CN(C)C(C2CC2C(C)(C)C)=O)cccc1 C12(C(N3C(C)CN(C)CC3)=O)CCC(CC1)N(C(c1cccc(F)c1)=O)C2 C1(C(N2CC=CC(C(=O)NC(c3ccn(C)n3)C)C2)=O)CCCCC1(C)C c1(C(=O)NCC2(NC(c3ccncc3Br)=O)CCC2)cc2cccnc2cn1 N1(C(C2CC2[N+](=O)[O-])=O)CC2CC(C1)N(C(c1ccc(-c3cccnc3)s1)=O)C2 c1(CNC(C2COC3CN(C(=O)OC(C)(C)C)CC32)=O)c2n(c(=O)n1C)CCCC2 Cc1cnc(C(=O)NCc2occc2C(=O)N(C)CC2CC2)cc1C CC(C)CC(c1nnnn1C1CCCCC1)NCCc1csc(Cl)c1 N1(C(Cc2cccc(C#C)c2)=O)CCC(F)(F)C(CNC(c2sccc2C)=O)C1 N1(C(c2c(CC)nccn2)=O)CCC2C(CCCN2C(=O)C(C)CSC)C1 C1(NC(CCCOC)=O)CC2CCC(C1)N2C(c1n[nH]cc1C(F)(F)F)=O c1(C(=O)NC2C(CNC(C(C)CF)=O)CC2)ccc(C(C)(C)C)nc1 CC(C)CC(=O)C(=O)N1CC2C(NC(=O)COc3ccsn3)C2C1 CCC(C)C(O)C(C)C(=O)NC(COC)CC(=O)N(C)CCN1CCCC1=O C(=O)(C(F)(F)C(F)(F)F)NC1CCC(N(C)C(C2CCC(C)(C)CC2)=O)C1 c1(C(=O)NC2CCCN(C(C(CCCC)N(C)C)=O)C2C)cc2cc(Cl)sc2[nH]1 C(=O)(CC(C)C(=O)N1CCCC(CO)C1C(N1CCOC(C(C)(C)C)C1)=O)OC CC(CC(=O)N1CCCC(C)(CNC(=O)CC2CC3CCC2O3)C1)P(C)(C)=O Cc1cc(F)ccc1C(N1CC(=O)CC1C(N1CCC(F)CC1)=O)=O C#Cc1ccc(C(=O)NC2CCCCC2CNC(=O)C2=CCSC2)nc1 C#Cc1ccc(F)c(C(C)NCC2CCN(c3ccc(F)cc3F)C2)c1 c1(C(=O)NCC2CCN(Cc3cccc(C)n3)C2)ccc(Br)nc1Br CC(C)(C)CCC(=O)NCC12CC(NC(c3coc(C(N)=O)c3)=O)(C1)C(C)O2 c1(CC(=O)NC2CC(C)N(C(=O)CP(C)(C)=O)CC2)cn(C)c2ccccc12 c1(C(C(=O)NC)NCCN(C(c2cnsn2)=O)CC2CCCO2)ccc(F)cc1 N1(C(C(N2CCSCC2)C)=O)CCC(CO)(CNC(=O)CN2CCOCC2=O)C1 Cc1cc(C)n(CC(N2CCCC(C(C)(C)O)C2)=O)n1.c1(SCN)ccccc1 C12(CNC(C(C)N(C(=O)C(C)NC(=O)OC)CCC)=O)COC(C1)C(O)C2 Cc1cc(=NCCCC(C)(C)NC(=O)C=Cc2ccco2)[nH]c(C(C)C)n1 CCC(CC)C(=O)N(CCCCNC(=O)CNS(C)(=O)=O)C CC(C)C(CNC(C1CC2COCC2C1)=O)C(=O)N1CCCC1CN(C)C c1(C(N2CC3C(NC(CN(CCC)C)=O)(C3)C2)=O)cc(Cl)cc2c1CCC2 n1(C(COC)C)nc(-c2ccc(N)cn2)nc1CCc1cc(C)no1 CC(N=c1nc(N2CC(=O)NC(C)(C)C2)c2ncccc2[nH]1)c1ccoc1 C1(C(=O)NC2CC(O)(CNC(=O)CC3CC=CC3)C2)CCC2(CCCCC2)CC1 C1(NC2(CC(=O)OC)CCCOC2)CC2(CCCCCC2)C1 c1(OC)ccc(CNC2CC2C(=O)NCC2CCC(O)CC2)c(OC)n1 CCC(C(=O)NCCOCCNC(=O)Cc1c(C)nn(C)c1Cl)C(C)(C)CC C(=O)(C(C)(C)N=[N+]=[N-])NCc1c(C(=O)NCCc2nc(C)[nH]n2)occ1 C1(C(N2CC(COC)C2)=O)CCC(CNC(c2ccn(C(F)F)n2)=O)C1 C(=O)(CC1=CCCC1)N(C1CCCN(C(C(C)OCC(C)C)=O)C1)C N1(C(C2C3(CC(OCC)C3)C2)=O)CC(NC(C2CC3CC3C2)=O)CC2(CC2)C1 C1(CNC(CC(C)C(F)F)=O)CCCC2(CN(C(=O)Cc3c[nH]nc3O)C2)O1 CCCCC(O)C(C)C(=O)NCC(C)=CC(=O)NCc1cnc(C)s1 Cc1ccc(F)c(O)c1C(N1CC2(C1)SCCC2NC(C1CC2CCC1O2)=O)=O c1(NC(=O)N(CCc2cccc(F)c2)CCO)ccc(NC2CCOCC2)cc1 CC(=O)CCCC(=O)NC(C)(CO)C(=O)N(c1csnc1C)C CCCC(F)C(=O)N1CCC2CC12C(=O)NCc1cc(C#N)c[nH]1 c1(CC(=O)NCc2nocc2C(=O)NC2(CO)CC=CC2)cncnc1O CC(C)C(O)C(F)(F)C(=O)NCC1CCCC1NC(=O)C(C)Cc1cnc[nH]1 C1(CNC(COC(CC)CC)=O)CCCN(C(=O)CCCC2(N(C)C)CCC2)C1 c1(C2(C)CC2NC(C2CC(O)(C(F)(F)F)C2)=O)cccc(Cl)c1 C(=O)(CCP(C)(C)=O)N(CC1(O)CCN(C(c2nc(CCCC)sc2)=O)C1)CC C(CCCCCCCO)=CC(N1CC(CNC(=O)C=CCO)OC(C(F)(F)F)C1)=O C(N=c1cc[nH]c(-c2nccs2)n1)C1CN(C(=O)NC2C(C)(C)CCC2)C1 c1(C(C)OC)nc(C)c(S(=O)(=O)N2CCCCC2C(=O)OC)s1 Cc1ccc(CNC(=O)CCC2CCCN2Cc2ccccn2)o1 C(N=c1ccn2nccc2[nH]1)C1CCCN(Cc2c(OC)cccc2F)C1 c1(C(N2C(CNC(C(C)CC3CC3)=O)CC(F)C2)=O)ccc(S(N)(=O)=O)cn1 c1(C(N2CC(C)(C)C(C(=O)NCC3(O)CC(O)C3)C2)=O)c[nH]c2cnccc12 N1(C(C(CC)OC)=O)CCCCC(C(=O)NC2CC2(C)C)C1 C1(NC(C(CCCC)O)=O)COC2(CCN(C(c3cnc(C)cc3C)=O)CC2)C1 Cc1ccc(C(C)NC(=O)C(CN(C)C)NC(=O)C(O)C2CCCC2)nc1 Cc1nc(C(N2CCN(C(C3(Cl)CC3(F)F)=O)CC(C)(F)C2)=O)c2ccnc-2[nH]1 c1(CC(=O)NC2CC2)cccc(Nc2ccns2)c1 C(=O)(C1CCc2c[nH]nc21)N1CCC2(C(NC(c3n(C)c(S)nc3)=O)C2)C1 C(=O)(C(C)CCO)N(C1CCCC1)CCNC(CN1C(C)CC1)=O C1(CNC(=O)Cc2cscn2)CCN(C(C2CCOC(=O)N2)=O)C12CCC2 c1(C(=O)NCC(CNC(CSCCC)=O)F)cnn(CCF)c1 C1(C2(NC(CC(=C)Br)=O)CC2)CCCCN1C(c1ccccc1SC)=O c1(C(N(CC(C)O)CCNC(C2N(C(C)=O)CSC2)=O)=O)ccc(C)n1C c1(OC)cc(C)c(CCC(=O)OC(CC(F)(F)F)c2ccc(F)cc2)c(C)c1 N(C1CCCc2ccoc21)C(C1CC(C)N1C(=O)CCc1cn[nH]c1)=O C1(COC)CCN(C(c2cc(CNC(=O)C(=O)N(C)C)oc2C)=O)CC1 c1(OC)cc(OC)c(C(N2CCCC2C2CCN(C(=O)C3=CCC3)C2)=O)cn1 Cc1cc(C(=O)NC2CCN(C(=O)C(C)(C)CCC#N)C23CC3)cc(C)c1Cl N1(CC)CCOCC1CC(=O)NCC1(NC(C2CCCC(C(=O)OC)C2)=O)CC1 N1(c2ncc(C)cn2)CCOCC(C(=O)NCC2CCCCCC2)C1 c1(C(CNC(C2(C3CCCO3)CC2)=O)NC(C2C(C)CCO2)=O)ccccc1F N1(C(C(C)C(C)O)=O)CCCC(C)(NC(=O)C=Cc2cccc(Cl)c2)C1 C12=CNC(=NCCNC(=O)C(=O)NC1)C=C2.c1(OC)ccc(C)c(C(C)(C)C)c1 C1(CNC(c2cc(CC)[nH]n2)=O)CCCC(NC(C2(Br)CC2(F)F)=O)C1 C1(CONC(=O)Nc2cc(-c3cccs3)on2)CS(=O)(=O)CC1C(F)(F)F c1(OC)ccc(C)cc1C(N1CC(O)(CNC(c2cc(C)ccc2O)=O)C1)=O CCC(CC(=O)NCC1CC(C(=O)NC(C)Cn2ccnn2)C1)OC C12(CNC(=O)C=Cc3cocn3)CCC1CN(C(=O)COc1ccc(F)nc1)C2 S(=O)(=O)(CC(=O)N1CCC(O)(C(C)NC(=O)COCc2cccc(C)c2)C1)NC Cc1nc(N2CC(O)(CCNC(c3ccco3)=O)C2)cc(-c2ccco2)n1 Cc1cn2cc(C(N3CCC(C)(NC(c4cc5n(n4)CCCC5)=O)C3)=O)nc2s1 C1(C)(CC)CC(NC(=O)C2=CCCC2)CN1C(=O)CN1CCSCC1 C1(CNC(C2C(=C)C2)=O)CC2CCC(C1)N2C(=O)C=Cc1ccccc1 CCCCCCCCNC(=O)C(=O)NCC(c1ccc(OC)c(OC)c1)C C(=O)(C(F)C(C)C(F)(F)F)NCC(CNC(c1cc(C)c(C)s1)=O)O CCCCCC(O)C(C)C(=O)N1CC(F)(CNC(c2cc3ccccc3o2)=O)C1 c1(C(N2CCC3CN(C(CCC(C)C#N)=O)CC32)=O)ccc2cccc(F)c2n1 C(=O)(C(O)C(F)(F)F)N1CCC(CNC(c2ccc(CC(C)C)s2)=O)C1 C1(C(=O)NCCN(CCC)C(C2(N(C)C)CC2)=O)CCCC(CF)C1 c1(C(n2cc(C3CCN3C(=O)COCCC(C)C)nn2)C)nc2ccccc2o1 c1(C(N(C)NC(C(=O)NCC)=O)=O)cnn2cccc2c1.c12cccc(c1)CC2 C=CC1(C(=O)NCCCC2CCCCC2)CCN(C(=O)C=C2CCCCC2)CC1 CC1(C)CN(C(=O)C=CC2CCOCC2)CC(CNC(=O)C(C)(C)CF)O1 c1(NC(=O)Nc2csc(=NCc3c(Cl)cc(Cl)cc3Cl)[nH]2)ccnn2cccc12 C(=O)(C(CC(C)C)C(N)=O)NC1CCC(C(N2CC(F)=C(C)CC2)=O)C1 C1(O)(CNC(C2C(C(N)=O)C2)=O)CCN(C(=O)CNS(=O)(=O)C2CC2)C1 N#Cc1cnccc1COC(=O)C=Cc1cccc(-c2ccc(Cl)cc2)c1 O=C1C2CCCCC2C(=O)N1CCNC(c1cc2c(cn1)COCC2)=O C(S(=O)(=O)c1cc(Cl)ccc1F)C1CCN(C(=O)NCCCCOC(C)C)CC1 c1(OC)ccccc1-c1nc(C2COCCO2)n(Cc2cccs2)n1 C1(CNC(C(CO)N(C)C)=O)CCC(CNC(C2(C)CC=CCC2)=O)CC1 C#CC1(C(N2CCC(CCO)C2)=O)CCN(C(=O)CC(C2CC2)C2CC2)C1 N1(c2nccc(OCC)n2)CCC2(CCN(C(c3ccc(Br)c(F)c3F)=O)C2)C1 C1(C)(NC(c2ncc(OC)cn2)=O)CCC(NC(=O)Cc2ccccn2)CC1 c1(-c2c(C3(C(=O)OC)CC3)cccc2)cc(OC(C)C)c(F)c(F)c1 c1(CC)cc(C(N2CC(OCCNC(C3CC(C#N)C3)=O)C2)=O)c(C)o1 c1(C(N(CCCN(C(=O)C(C)(C)c2ccccn2)C)C)=O)cnn(C)c1N c1(C(=O)NC2CN(C(=O)Cc3ccc(F)cc3Cl)C2)cccc(C#CC2CC2)c1 c1(C(=O)NCC(C)CN(C(=O)CCC2(C#N)CCC2)C)sccc1Cl N1(C(c2cn(C)nn2)=O)CCC(C2CCCN(C(c3ccc(F)nc3)=O)C2)C1 Cc1ccc(C#N)cc1C(N1CCC(C(C)NC(=O)C(O)C(C)C)CC1)=O c1(OC)cc(CCC(=O)NCCCCCC2(NC(c3ccc(C)s3)=O)CC2)on1 N1(C(C(=O)NC)C)CCCC(NC(=O)CC(C)OC)CC1 N1(C(CCC=CCC=C)=O)CCC(CNC(c2scc(C)c2C)=O)(OC)CC1 CC1(C)CCOC(CN=C(NCc2nnc(COC)s2)NC2CCC2)C1 C1(NC(COCCCCC)=O)CC2CC(NC(=O)CC(C)CC(C)C)CC2C1 N1(C(CC2CC(C)(C)OCC2)=O)CCC2(CC1)CN(C(c1ncc(F)cn1)=O)C2 C1(C2(O)CCOCC2)(C(=O)NC(C2CN(C(c3cnoc3)=O)CCO2)C)CC1 c1(C(=O)NCC(CCNC(C(C)OCC)=O)O)ccnc2ccncc12 C(=O)(CCCC(=O)N(C1CCCN(C(c2coc3c2COC3)=O)C1)CC)NCC S(=O)(=O)(c1ccc(C(=O)N(CCC(C)NC(=O)C(O)CCSC)C)cc1)NC c1(C(=O)NCCC2(OC)CN(C(c3ccc(F)c(C)c3)=O)C2)sc(C)c(C)c1C c1(C(=O)NC(COC)CNC(=O)CC2COC(=O)C2)ccc(F)c(F)c1 N1(C(C2N(CC(C)C)CCC2)=O)CCC(O)(CNC(=O)CCc2cnoc2)CC1 c1(C(N2CC(NC(C(CCC)O)=O)CC(C)(C)C2)=O)cnn2c1OCCCC2 N1(C(CSCC(=O)OC)=O)CC2CC1CN2C(C1(c2cnn(C)c2)CCCO1)=O C1(C(=O)N(CC(C)C(C)C)C)(CC)CCCN(C(c2ccc(C(C)C)o2)=O)C1 c1(C(=O)NC2C(CNC(c3n(C)ccc3)=O)CCC2)c(C(F)(F)F)cccc1O c1(CC)nn(C)cc1C(=O)NC1CN(C(c2sccc2C(C)(C)C)=O)CC1C N1(C2CCC(NC(COC)=O)C2)CCN(C(=O)CN2CCC(O)CC2)CC1 N1(c2c(C)c(NC(c3nc[nH]n3)C)ncn2)CCC2(CCCN2C)C1 N1(C(Cc2ccc(CC)cc2)=O)CCC(C2(NC(=O)CP(C)(C)=O)CC2)C1 CC1(C(=O)NCC2C3CN(C(=O)Cc4cnco4)CC23)CNC(=O)C1 Cc1ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CC4CCC4C3)=O)CC2O)c1C N1(C(=O)Cc2ccc(Cl)cn2)CC2CCC(C1)N2C(C1CC1F)=O C1(N2CCC(COC)CC2)CCC2(CC1)CN(C(c1c(F)cccc1Br)=O)C2 C12(CNC(=O)Cc3ccon3)CC(C1)C(NC(=O)COC1CC=CC1)CO2 C1(C(N2CC(C3CN(C(c4csc(O)n4)=O)CCO3)C2)=O)CCN(CCO)CC1 N1(C(C(CCC)OC)=O)CCC(C2CCCN(C(c3cscn3)C)C2)CC1 Cc1cccc2nc(C(=O)NC(C)(C)CCN(C(=O)C3=COCCC3)C)cn12 C1(C)(COC)CCCN(C(C2CCN(C(=O)CC3(C)CCOC3)C2)=O)C1 C(=O)(C(O)CCCNC(C1CC(C)N(C)C1)=O)N(CC(=C)C)C C1(NC(=O)NC(Cc2ccc(C)cc2)(C)C)Cc2cccnc2C1 CC1(C)C(CNC(C2CCCO2)=O)CCN1c1ncc(O)cn1 N1(C(CCNC(COC)=O)=O)CC(N(C)C(C2CC23CCCC3)=O)C(C)(C)C1 N1(C(CC2CC(=O)NCCC2)=O)CC2CN(C(=O)CSC(F)(F)F)CC2C1 N=c1[nH]c2ccc(C(N3CCC(NC(=O)C4=CCCC4)CC3)=O)cc2[nH]1 N1(C(C#CC(C)(C)C)=O)CC23CCCCC2(C1)CN(C(C1CC(C#N)C1)=O)C3 N1(S(CC)(=O)=O)CCC2CCC(C1)N2C(c1cncc(CN(C)C)c1)=O CC1CCCC(C(=O)NC2CC(C)(NC(=O)CCCNC(N)=O)C2)C1 N1(C(c2ccc(C=O)s2)=O)CCC2(CCC(C(=O)NC3CCCCC3)O2)CC1 C1(C(=O)NCC2(NC(C(C)C3CC3)=O)CC2)CN(C)CC1c1ccccc1 c1(C(=O)NCCN(CCC)NC(c2nsc(CC3CC3)n2)=O)c(C2CC2)noc1C Cc1nc(NC(=O)C=CC(F)(F)F)sc1NC(=O)NCC1CN(C)CC1O c1(CCNC(N2CC(C(N3CCC(O)CC3)=O)C2)=O)cccc(Br)n1 N1(C(C(CC)=O)=O)Cc2ccc(-c3cc4ccc(F)cc4[nH]3)cc2C1 c1(C(N2CC(O)(C(C)NC(CC=CCC)=O)C2)=O)cccc(C)c1Br C1(NC(c2c(C(=O)OC)csc2)=O)CCS(=O)(=O)C1.c12cn(nn1)CC(=O)S2 c1(OCC(C)C)ccc(SCC(N2CC(NC(=O)CNC=O)C3CC23)=O)cc1 N1(C(C(CC)CNC(C)=O)=O)C2CCC1C(NC(=O)C(C)C(=O)N1CCOCC1)C2 c1(N(C(=O)C#CCNC(C2COCCO2)=O)CC)ccc(O)cc1 C12(C(=O)NCCC(C)NC(c3csc(-c4cnc[nH]4)n3)=O)CCC(CC1)CO2 CN1N=CC(CC(=O)NCC(C(C)(C)C)NC(c2ccn(C(C)(C)C)n2)=O)C1=O C(=O)(C(C(C)NC(C1CCCC1O)=O)C(C)C)NCc1nccc(C)n1 c1(C(=O)NC(C)Cn2cc(CN3CC4CC4C3)nn2)c(Cl)nc2ccccn12 C1(C(=O)OC)CC2(CCC(CNC(c3ccc(-n4ccccc4=O)cc3)=O)O2)C1 CC1CN(C(=O)CC2CC3(CC3)CO2)CC1NC(c1cnc(O)s1)=O c1(C(=O)NCCOCCCN(C(c2cc(OCC)n[nH]2)=O)C)ccccc1C c1(CC)nnc(O)c(C(N2CCC(CNC(=O)C(O)CCC(C)C)C2)=O)c1CC CCCCCC(C)(C)C(=O)N(CC(C)CNC(C1CCCN(CCC)C1)=O)C c1(NC(C(=O)N(S(C)(=O)=O)CC2CCCC2)=O)cc(F)ccc1N1CCCC1=O CC(C)C(F)(CNC(=O)CCN1CCOC1=O)C(=O)NCc1ccccc1C#N N1(C(c2c(C)ccs2)=O)CCC2(CC1)CN(C(=O)C(C)(C)N1CCCC1)C2 C12CCCC1C(=O)NCCCCCN(CC)C2.c1(CC)nncs1 C12(C(=O)NC(CN(C(c3coc(C4CC4)n3)=O)CC)C)CCCN1CC(OC)C2 C1(CNC(CC(C)NC(CCCOCCOCC)=O)=O)CNC(=O)CO1 Cc1cccc(C(=O)NC2(CCCCNC3CC4CC4C3)CC2)c1 N1(C(C2(NC(C34CCC(C3)C4(C)C)=O)C(C)CCC2)=O)CC=CCC(C)(C)C1 c1(COC(COC(C(C(C)CC(C)OC(C)=O)OC)=O)=O)cccn2c(C)cnc12 c1(C(N2CCC(OC(C(=O)NCC(C#C)CCC)C3CC3)C2)=O)nnccc1C C1(OC(=O)N(C)CC)CCCCC1.C(=O)(CCNC(=O)CCOC)NC.CC(C)N c1(C(N2CCC(CNC(C(C)N(C(C)=O)C)=O)C2)=O)cc2c(nn1)CCCO2 c1(C(N2CC(NC(C(C=CCCC)O)=O)C(C(F)F)C2)=O)c(F)ccc(F)c1Cl N1(C(CC2CCN(C(C3CCN(C)CC3)=O)C2(C)C)=O)CCC12CCOCC2 C(=O)(CCCCN1CCCC1)NCCN(C(=O)C(C1CC1)Sc1ccccc1)C N12CCC(O)(C1)C2=O.N1(Cc2nc(C)sc2)CC2C(C(=O)ON)C2C1 c1(CN2C3CN(C(c4ccc(COC)cc4)=O)C(C3)C2)c(O)cc(F)cc1F c1(C(N2CCC(C)(NC(=O)C3=C(C#N)CCC3)C2)=O)cnn2c(Br)cccc12 CCS(=O)CC(=O)NCC1(F)CC(NC(c2cccn2-c2ccc(F)cc2)=O)C1 c1(OC)ccc(Cl)cc1CC(=O)NCC(CO)NC(c1cc(C2CC2)ncn1)=O C1(NC(C=COCC)=O)CCCCCCC1NC(=O)CC1CCC(C)CO1 CCCC(CCCN(C(=O)CNC(c1ccsc1)=O)C)NC(=O)COCCOC C(=O)(C(C(C)(C)C)c1cc[nH]n1)NCC(C)N(C(=O)CO)C C#Cc1ccc(Br)c(C(=O)NCC2CC3(CC3)CN2C(C2CC2C=C)=O)c1 N1(C(c2nn(CC)c(O)c2)=O)CC2OCC(NC(c3ncc(Cl)cc3Cl)=O)C2C1 c1(C(N2C(CNC(=O)CC3CC34CC4)CC(OC)C2)=O)ccc(F)cc1Br c1(N(C)Cc2ccncc2)nc(=NC2CN(CC(F)F)C2)[nH]c2ccsc12 c1(C(=O)NCCC2(O)CN(C(C3OCCN(C)C3)=O)C2)ncnc(O)c1F O(N(CC)C(=O)C1CCC(NC(=O)Cc2ccccc2NC(C)=O)CC1)CC Cc1noc(C)c1CC(=O)NCC1C2CN(C(C3CC(=O)N3)=O)CC12 c1(CC)cncc(CC(=O)NCC2CN(C(=O)C=Cc3ccc(C(F)F)o3)C2)c1 C1(NC(CN)=O)CC(NC(C=CC=CC)=O)CN1.n1(C(COC2CC2)=O)cnnn1 C(=O)(C#CC1CCCOC1)NCC(C(C)C(C)C)NC(c1cccc(CC)n1)=O N1(C(Cn2nnc(=N)[nH]2)=O)CCOC2(CCN(C(c3ccc[n+]([O-])c3)=O)C2)C1 N1(C(COC)=O)CC(NC(=O)C=Cc2ccc(C)cc2OC)CC12CCCCC2 CC(C)CC(CNC(=O)C(C1CCOCC1)F)C(=O)N(CCC(N)=O)C c1(N(C)Cc2cccc(F)c2)nc2ccsc2c(=NCCN(S(C)(=O)=O)C)[nH]1 C1(C(N(CC(C)CNC(=O)CC(C)NC(N)=O)C)=O)COCCN1C=O Nc1c(C(=O)NC2COCC2CNC(C2OCCC2C(F)F)=O)cc(Cl)cc1Cl C(c1cscn1)=CC(=O)NCC1(CN(C(C(C)=CC2CC2)=O)C)CC1 N1(C(C2(CNC(c3n(CC)ncc3C)=O)CC2)=O)CCC(O)CC1C C1(C(=O)NC(C(=O)NC(CC)C(=O)N(C)C)CO)CC2CCC1O2 C1(CNC(C(CCC)(C)C)=O)CC2CCCCC2N1C(=O)Cc1ncc(C)o1 N1(c2n(CCC=C)c(CCCS(N)(=O)=O)nn2)Cc2c[nH]nc2C(C)(C)C1 C(C(=O)N1CC(CS(C)(=O)=O)C1)(C(C)(C)C)NC(=O)OC(C)(C)C c1(C(N2C(CC(c3cccc(C)c3)=O)CCCC2)=O)cc2nc(C)sc2[nH]1 c1(CNc2c(C)scn2)c(OC(F)F)cccc1Cl c1(CNC(c2cnco2)=O)ccc(CNC(c2cncn2C2CC2)=O)c(F)c1 C12(NC(=O)Cc3ccccc3)CCOCC1CN(C(=O)CCC1OCCO1)C2 CC1CCCC1(C)C(=O)NCC1CC(NC(c2ccc(C3(C)CC3)cc2)=O)C1 C=CCC(C(=O)NC(CNC(=O)CCCc1c(F)cccc1F)C1CC1)C(C)C c1(C(=O)NC)ccc(O)c(NC(C2CCCCC(=O)C2)=O)c1 C(=O)(C#CC(C)(C)C)NCC1CC(NC(c2cc(C(=O)OCC)sc2)=O)C1 CC(=O)C(C)(C)CC(=O)N1CC2COCC2(C(N2CCOC(CC(C)C)C2)=O)C1 C1(CNC(=O)C2=CCSC2)CC2CC1CN2C(c1ccc(F)c(CO)c1)=O Cc1ccc(CC(=O)NCC(O)CNC(C2(C)COCCO2)=O)c(Cl)c1 Cc1cc(CNC(c2occc2CNC(C2CCCOC2)=O)=O)nnc1C C1(NC(=O)CC2CC3(CC3)C2)C2CC3C(C2)C13C(=O)NCC1(F)CC(CO)C1 c1(C(CC)CC)cc(C(=O)NC2CC2CNC(=O)CCCn2cccn2)on1 C1(NC(c2c(SC)ccs2)=O)C2CC1N(C(c1cc(=O)cc(Cl)[nH]1)=O)C2C C1(C2N(C(=O)C(F)C3CCCC3)CCC2)CCN(C(C23CC(C2)C3)=O)CC1 CC1CCC(CNC(=O)C(C2CCN(C(=O)C(N)=O)CC2)C)CC1.C1CC1 N1(C(C2N(C=O)CCC2)=O)CC2(CCN(C(=O)C(=Cc3c[nH]cn3)F)C2)C1 C(CN=c1[nH]c(=NC2CCOCC2F)c2[nH]ccc2[nH]1)N(CC(C)C)C Cc1nc(C=CC(N2CC(NC(C3(C#N)CC3(C)C)=O)C(C)C2)=O)[nH]c1C N1(C(C(CC=C)OC)=O)CC2CC(C(=O)NC3CCCC3(C)N(C)C)(C2)C1 N1(C(c2cc(CC(=O)OC)on2)=O)CCC2CN(C(=O)CCC(C)C)CCC12 C=C(Cl)CCC(=O)N1CCCCC1CC(=O)NCc1ccn(C(C)C)n1 C1(CNC(C=Cc2nnn(C)n2)=O)CCN(C(C2CCC(N(C)C)C2)=O)C1(C)C N1(C(c2c(CC)non2)=O)CC2CC(C1)N(C(=O)C(C)Cc1ccc(O)cc1)C2 c1(CC)ccc(C(=O)NCC(CC)N(C(=O)C(c2ccnn2C)C)C)s1 N1(C(C#C)=O)CCC2(CCCC2C(=O)Nc2ccc(F)cc2C)C1 c1(N(c2scnc2C(=O)Nc2c(C)nn(C)c2)C(C)=O)ccc(Br)cc1I C(=O)(C1=NOC2COCC12)NC1C(NC(=O)C2=CSCCO2)COC1 c1(CC)nc(C)oc1C(=O)NCCOCCC(=O)N(C)Cc1occc1C CC(CC(C)(C)C)C(=O)NC1CN(C(c2csc(O)n2)=O)CC1c1nccn1C C(C1CCc2nccn21)NC(CC(CNC(CSCC)=O)O)=O C1(NC(CC2(OC)CC2)=O)CCCC(NC(c2cccc[n+]2[O-])=O)CC1 c1(C(N2C(CN(C)C(c3cc(N)ccc3Cl)=O)CCC2)=O)nccc(Cl)c1F c1(SC)cccnc1C(=O)NCC1CCCCN1C(C1CCCC(C)C1)=O c1(C(=O)NC2C3(CCC(NC(C(N)=O)=O)CC3)C2)c[nH]c2nc(F)ccc12 C#Cc1ccc(C(=O)N(C)CC2CC(F)CN2C(C2CN(CC)CCO2)=O)cc1 C1(C(N2C3(CNC(C4N(C)CCOC4)=O)CC(C2)C3)=O)C2Cc3ccccc3C12 Cn1ncc2ncc(C(N3CC4CCCC(NC(=O)C(N)=O)C4C3)=O)cc12 C1(CNC(CCCCC=CC)=O)CCC2CN(C(=O)Cc3ccn(C)c3)CC12 c1(C(=O)NC2CN(C(c3cc[nH]n3)=O)C2)ccc2nnc(O)n2c1 N1(C(C(C)CF)=O)CCC(CO)(CNC(=O)C(C)CSCc2ccccc2)CC1 c1(CC)ncc(C(N2CC(CN(C)C(C3CCC(CN(C)C)O3)=O)C2)=O)c(C)n1 CN1C(=O)CCCC1C(=O)Nc1ccns1 CC1CC2(CC(C(N3CC4CC(NC(=O)Cc5cocn5)C3C4)=O)C2)C1 N1(C(C(COC)C(F)(F)F)=O)CCc2sccc2C1CNC(=O)CCC(N)=O CCCCCCC(C(=O)NC1CC(NC(C2CNC(=O)C2)=O)C(O)C1)NC(C)=O C#CCCCCCC(=O)NC1(C)CCN(C(=O)CSc2cc(C)ccc2C)C1 c1(CC)cc(Cl)ccc1C(N1CCC(NC(C2CCN2CC)=O)C1(C)C)=O n1(C(C)C)ccc(C(=O)NCC(C2CCOC2)NC(=O)CCCF)n1 CN1C(=O)CCC1C(N1CC(NC(c2ncc(Br)cn2)=O)C(CC2CC2)C1)=O c1(C(=O)OCc2ccc(-c3cn(C)nc3)s2)cncc(N(C)C)c1 Cn1cnc2cccc(C(=O)NC3CCC3NC(c3cnc(S)n3C)=O)c12 C1(CC)(NC(=O)Cc2n[nH]c(=N)s2)CCCN(C(c2cccnc2)=O)C1 CC(O)(CNC(=O)CCc1cnccn1)CNC(=O)CCC1OCCO1 N1(C(C(C(C)C)O)=O)CCN(C)C(CNC(c2ccc(C(F)(F)CF)cc2)=O)C1 CCC(C)CCC(=O)N(C1CC2CC1N(C(=O)Cc1cc(Cl)n(C)n1)C2)C C#Cc1ccc(C(=O)OCCC2CCN(C(=O)OC(C)(C)C)C2)nc1C C1(NC(C(CCC)NC(N)=O)=O)CC2CC(NC(=O)CCCSC)C2C1 C1(C(N2CC(=C(F)CNC(=O)CCc3nnc(C)o3)C2)=O)(OC)CCCSC1 C12(CC(=O)NCCc3c(C)n[nH]c3)CCC1CN(C(=O)C(F)C(C)(C)O)C2 c1(C(=O)NC(CCCC)CNC(c2ccncc2F)=O)cccc2c1COC2 c1(C(=O)NCCN(C2CCCC2)C(C2CC2(Cl)Cl)=O)cnoc1-c1ccccc1 C1(NC(CCSCCC)=O)CN(C(c2c[nH]cc2CC)=O)CCC12CCC2 C1(OCCNC(CCC=CCC=C)=O)CCN(C(=O)CC(C2CC2)C2CC2)CC1 C(=O)(CC(C)CC(F)(F)F)NC1CC(CCNC(c2c(C)ncnc2C)=O)C1 C1(C(=O)O)CC2(COCCN2C(=O)C2=CC3(CCOC3)C2)C1 Cc1nn(-c2ccc(F)cc2)c(NCc2nocc2CN(C)C)c1Br C(C(C)(C(C)C)NC(=O)CP(C)(C)=O)NC(CC1CC(NC(C)=O)C1)=O N1(C(C(N)=O)=O)CC=CC1C(=O)NCC1CCC1C(F)(F)F c1(C(N2CCC(C)N(C(=O)C(C)CCN(C)C)CC2)=O)c2c(nn1C)CCCC2 C1(C)(C(N(C)CCNC(=O)CCCc2ncco2)=O)CCCCC1(F)F C1(C(=O)NC2CCCN(C(c3cccc(=O)o3)=O)C2)Cc2ccccc2C1 N1(CCc2cn(CCC3CC3)nn2)CCN(C(=O)CCCn2cccc2)CC1.CS N1(C(COC2(C)CCCC2)=O)Cc2nccn2CC(NC(C2CC=CCO2)=O)C1 c1(C(=O)NCCCOCCNC(CC=CC=C)=O)cnn(CC)c1C c1(C(C)C)nc(NCCSc2nccn2C)cc(N2CCC(CO)C2)n1 c1(C(=O)NCCOC)ccc(Cl)c(S(=O)(=O)NCC2CC3CC2C3)c1 C1(NC2(c3nnnn3CCC3CC3)CCN(C)C2)CC2CCC(C1)C2(F)F N1(C(c2c(OC)cccc2)=O)CCCN(C(C2CC(=O)N(OC)C2)=O)CCC1 c1(N(C(C(C)Cc2ccco2)=O)CCC(N)=O)ccccc1C=O N1(C2(CC(=O)Nc3ccnnc3)CCC2)CCCNCC1 c1(C(C)CNC(=O)C(=O)NCC(C2CCCCC2)F)ccc(F)cc1 Cc1cc(C)n2nc(C)c(C(=O)NC3(CC(C)(C)C)COC3)c2n1 c1ccnc2ncnn12.c1(NC(C2N(C(=O)OC(C)(C)C)CCS2)=O)ccc(F)cc1 c1(C2C(C(=O)NCC(CC)NC(c3n[nH]c(C)c3O)=O)C2)ccncc1Cl c1(C(=O)OC)cncc(S(=O)(=O)NCCc2ccc(Br)cc2F)c1 CCC(C)C(C)C(=O)NC(C)(C)CNC(=O)NC1(C)CC(C(F)(F)F)C1 C1(=O)CCN(OC)C(=O)C(CO)N1C.CCC(CC)n1cccn1 C=C(C)C(C)(C)C(=O)NC1CCCCCC1C(=O)N(C)CCc1ncon1 N1(C(Cc2ccn(C)n2)=O)CCCC(C)(C)C1C(=O)NCCCn1cccn1 c1(C(N2CCC3CN(C(C(CC#C)C)=O)CC32)=O)cc(S(N)(=O)=O)sc1C C1(NC(C(C)OCC=C)=O)CN(C(c2ccc(-c3cc[nH]n3)cc2)=O)CC1F C1(NC(C2OC3CCC2C3)=O)CCC(NC(C2C(Cl)(Cl)C23CC3)=O)CC1 c1(OC)ccc(C(C)C(=O)NCCNC(=O)C(c2cnn(C)c2C(F)(F)F)C)cc1 N1(C(CCC(c2ccc(C)cc2)=O)=O)CCN(C(C2CC2C)=O)CC1CO Cc1nnc2n1CCN(C(=O)C(=O)NC(C1CCCCC1)Cc1ccccc1)C2 n1(CC)nc(C(=O)NCC2C3CC3CN2C(C2CC2F)=O)ccc1=O C1(NC(c2c(C)sc(O)n2)=O)CCN(C(=O)C(C)CC(C)C)CC(C)(C)C1 N1(C(C(c2n(C)ncc2)O)=O)CCCN(C(C2(C(=O)N(C)C)CC2)=O)CCC1 C=CC1(CNC(=O)C(CC2CCC2)NC(=O)CC(C)n2cccn2)CCC1 Cc1cc(NC(=O)CC23CCC2CN(C(=O)C(C)(C)CCF)C3)cnc1C C1(CC)(CC)CN(C(=O)CC(C2CCC2)NC(=O)CC(C)C2CC2)CCO1 c1(C(N2C(C(=O)NCCOc3cccnc3)CC(OC)C2)=O)ccc(O)cc1Cl C(=O)(C(C)(C)CCNC(c1cc(Cl)n[nH]1)=O)N(C1C(C)COCC1)C CN=c1nc(C(N2CCCC2N2CCC(C)(C)C2)=O)cc(C)[nH]1.CC1=NOC(C)C1 C=Cc1cncc(C(N2CCC(F)(C(N3CC4CC(C)(C)C4C3)=O)CC2)=O)c1 N1(C(CSCCC)=O)CCC(C2(O)CC(NC(=O)Cc3nccn3C)C2)CC1 C1(NC(CCc2onc(CSC)n2)=O)CN(C(c2[nH]c(C)nc2C)=O)CC1C c1(OC)ccnc(C(N2CCC(NC(C3CN(C(C)=O)C3)=O)CC2C)=O)c1OC C12(C(N3CCCN(C(CC4OCC(C)OC4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 Cc1ncc(Cl)cc1NC(C1OCCC1NC(=O)CC1CCC(C)(C)C1)=O O(NC(=O)CCC1CCCN1C(C1CCCCO1)=O)CCOCCOC C#CC1CCC(NC(c2ccc(CNC(c3ccc(C(N)=O)[nH]3)=O)nc2)=O)C1 c1(OC)cc(C=CC(=O)NCC2(O)CCCC2C)sn1 C1(C(=O)NC(CCCC)COC)CC(F)CCN1C(c1cc(C2CC2)no1)=O c1(OC)cc2nn[nH]c2cc1C(=O)NCC1CC2CC2N1C(C1CC(=C2CC2)C1)=O Cc1nc2c(CCC(=O)NCC3CCN3C(c3c(C)nsc3C)=O)cccc2o1 Cc1c[nH]c(C(=O)NC(C(N2CC(C(C)C)C(SC)C2)=O)c2ccoc2)c1C c1(OC)c(C)cc(C(N2CCN(C(c3ccc(C)cc3)=O)CC2CO)=O)cc1C N1(C(c2n(CCC)ccc2)=O)CC2(CCC2NC(c2ccc(OC)cc2)=O)C1 CC1(F)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN(C(C2(C)CC2(F)Cl)=O)C1 c1(C(N2CC(NC(C3CN4CCN3CC4)=O)CC(C)C2)=O)ccc2ncnn2c1 N=c1cc[nH]c(C(=O)NCC23CC(NC(C4CCCCC4O)=O)(C2)C3)n1 C1(O)(C(N2CC3=C(CN(C(C45CC(OC)C4C5)=O)C3)C2)=O)Cc2ccccc2C1 N1(CC2CN(S(c3c(C)onc3)(=O)=O)C2)Cc2ccccc2-c2ccccc2C1 n1(CC(N2CCN(Cc3c(O)cccc3O)C3CC23)=O)ccc2c(F)cccc12 c1(-n2c(-c3ccc(-c4n(C(C)C(=O)N(C)C)ccn4)s3)nnn2)cc(=O)cc[nH]1 Cc1ccnc(C(=O)NCC2(CO)CCN(C(=O)CC3CCCCO3)C2)c1O C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(c2cc(Cl)c(O)c(Cl)c2)=O)CC(C)(C)C1 CC1C(NC(c2snnc2C2CC2)=O)CCCN1C(c1cc(C2CC2)on1)=O C(CN=C(NCCc1ccsc1Br)N(C)CCSC(C)(C)C)SC c1(C(=O)NC(c2cccc(F)c2)C(N)=O)scc2c1CCCC2 CCCN=c1[nH]c(=NC2CCCCN(c3ccccc3)C2)c2sccc2[nH]1 C1(C(=O)NC2C(NC(c3n[nH]c(CC)c3C)=O)CC2)CC2OC1C1CC21 N1(C(C(=O)N(C)C)=O)CC2CCCC(N(C)C(c3cnc4sccn34)=O)C2C1 C1(C)(CNC(C(C)CO)=O)COCCN(C(c2cccnc2C(F)(F)F)=O)C1 Cc1nc(CNC(=O)C(CNC(=O)CC23CCCC2C3)N(C)C)sc1C CC(C(=O)NCCN(C1CCCCCC1)C(=O)CC1CCOCC1)S(N)(=O)=O c1(C(=O)NCC(C2CC2)NC(C(C)(C)OCC)=O)cc2c(F)ccc(F)c2s1 n1(CCN(CC)Cc2ccc(-c3ccccc3CO)nc2)ccc2ccccc12 CC1CC(C)(C(=O)NC(CCN(C)C(C2(CF)CC2)=O)c2cccs2)C1 N1(C(c2c(C)nns2)=O)CCCC2(CCN2C(C2CCCSC2)=O)C1 C(=O)(C(F)C(F)(F)F)NCCCOCCNC(Cc1c(CC)cccc1)=O CCCCCC(C)(C)C(=O)NCc1ncccc1C(=O)N(CCC(N)=O)C N1(CCC)CCCC1C(=O)NC(C)CCNC(c1cnoc1C1CC1)=O C(C(C)CC(=O)NCCCC(C)NC(=O)CSCCCc1ccccc1)OC C1(C(=O)NCC2N(C(C=CCC)=O)CC(F)(F)C2)CCOC2(CCCC2)C1 CC(C)CS(=O)(=O)CCC(=O)NCCCN(C(=O)CCc1cscn1)CCO N1(C(COC(C)=O)=O)CC2C(NC(c3ccc(CF)cc3)=O)C2C1 c1(OCC(=O)N(CC(CC)NC(=O)C(C)(C)C2CC2)C)ccccc1C N1(C(CC(C)(C)CBr)c2nnnn2C2COC2)CC2CCC(O)CC2C1 c1(CC)cc(C)ccc1NC(=O)CC1CCCCC1NC(c1c[nH]ccc1=O)=O c1(CNC(C2CC2Cl)=O)n[nH]c2c1CN(C(=O)Cc1ccsc1)C2 O=S(=O)(c1ccc(NC(c2ccccc2)CO)c(Cl)c1)N1CCC=C(F)C1 CC(C(=O)NCc1cscn1)NC(=O)C(C)C1CCCC1 C1(C(=O)NCCC2OCCN(C(c3c[nH]c(=NC)o3)=O)C2)CC(C)(C)OC1(C)C C12(C(N3C(COC)CC3)=O)CCCCC1C2Br C1(NC(C2(OC)CC2)=O)CCCC2CN(C(c3cnsc3C)=O)CC12 CCCCC(C)C(=O)N1CC(CNC(=O)CCC2(NC(=O)OC(C)(C)C)CC2)C1 N1(C(C(N(C)O)=O)=O)CCC(O)(CNC(=O)C(F)OC(F)(F)F)CC1 C1(C(C)NC(c2cccs2)=O)CCCN(C(C)C(=O)Nc2ccccc2F)C1 c1(CC)cc(C(=O)NCC2(O)CC(NC(=O)CC3CC=CC3)C2)c(C)nn1 c1(C(N(C2CC(NC(=O)CCn3cc(Cl)cn3)C2)C)=O)csc2nccn12 CC(C)(C#N)CC(=O)NCC1(C)CCCN(C(c2cncc(C3CC3)c2)=O)C1 c1(CC)ccc(F)cc1C(=O)NCC12CC(NC(=O)C(F)CC)(C1)C(C)O2 N1(C(C2C(=C)C2C(=O)OC)=O)CCCC(F)(C(=O)NCCn2cnc(C)c2C)C1 c1(CN(C(CCCOC)=O)C)cnn2c1CN(C(=O)C(C)S(N)(=O)=O)CC2 c1(CN(C2CC(N)C23CCC3)C(c2ccc3c(c2)OCO3)=O)nc2ccccc2s1 C1(NC(C2C(NC(=O)C(c3ccccc3)F)COCC2)=O)CC2OC(=O)CC12 Cc1cn2c(C=CC(=O)NCCc3cnc(C#N)cn3)c(C)nc2s1 C=C(C)CC(C(=O)N1CCN(C)C(CNC(=O)C(O)CCSC)C1)OC CCC(CC(=O)NC1(CCNC(=O)Cc2ccc(F)cc2)CC1)C(C)(C)C C1(CC(N2CC(CSC)C2)=O)CC(F)CN1C(C1CC12CC2)=O c1(C(=O)NCC2(F)CC(NC(c3cc(CCC)on3)=O)C2)n[nH]c2c1CSCC2 C(=O)(C1=CCC(C)(C)CC1)N1CCCC(Nc2nc(O)n(C)c(=O)c2)CC1 c1(C(N2CCC(OCC(=O)OC)C2)=O)cc(C#N)[nH]c1C C#Cc1cc(NC(=O)C#CCNC(C2CCC(=O)N2)=O)ccc1C C(=O)(C(CN=[N+]=[N-])NC(C1CC2C=CC1CC2)=O)NC1CCN(C)C1 N1(Cc2ccn(C(C)C)n2)CCC(CO)CC12CC2 c1(CN2CCCC(C(=O)Nc3c(OC)nnc(Cl)c3)C2)cc(C)c(Cl)c(C)c1 c1(CNC(=NCC)NCC2CC=CCO2)cc(C)ccc1O N1(C(=O)NC2(c3cn(CCCCCO)nn3)CC(F)(F)C2)CCCCCC1 c1(C(=O)NCC(CC)(C)NC(=O)C(F)=C(C)C2CC2)ccc(C)c(F)c1 N1(C(CN(CCC#C)C)=O)CCCC2(CNC(C3CC(C)=NO3)=O)CCCC12 Nc1cccc(C(=O)CCC(=O)NCCCCNC(C23CCCC2C3)=O)c1 c1(C(C(N2C(CC)C(NC(c3cnnn3C)=O)CC2)=O)=O)ccc(Cl)cc1O C=CCC(CNC(=O)C#CCNC(C)=O)NC(=O)CC1CSCCS1 N1(C(c2c(C)noc2)=O)CCCC(CNC(c2coc(-c3cccnc3)n2)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)NCC1(O)CCN(C(C=C2CCC(C)C2)=O)C1 C1(C(=O)NCC2OCC(CNC(CCC#C)=O)C2)CC2(C1)CC(C)(C)C2 N1(C(C(CC)(C)O)=O)CC(CNC(c2ccoc2C2CC2)=O)CC(C)(C)C1 C1(NC(C2CC(C(C)O)C2)=O)(CF)CCN(C(=O)C(C)CC2CC2)C1 c1(OC)ccc(C(N2CCC(CNC(=O)CC(F)F)C2)=O)c(Br)c1F N1(C(CCCC2(C)N=N2)=O)CC2CC(C1)CN(C(c1ocnc1C1CC1)=O)C2 c1(C2C3C(CC3)N2)nnnn1CCCOC(C)C.C(C(C)(C)OCC1CC1)OC C1(C(N2CCC(O)(CC)C2)=O)CCCCC1(C)NC(=O)CC1CCC(C)(C)O1 CN1CCC(C)(C(=O)NCC23CC2CN(C(=O)CC2CSCCO2)C3)CC1 c1(OC)cc(N2CC(n3nccc3C)C2)nc(-n2cc(C3(CO)CC3)nn2)n1 C=CC(CC)C(=O)NC(CO)C(C)NC(c1cnn(CC)c1CC)=O N1(C(COCCSC)=O)C(C)CC2CN(C(=O)CCn3cccc3)CC12 c1(N(C)CC2CC2)ccn2ncc(S(=O)(=O)NC3(C)CCOC3C3CC3)c2n1 c1(C(N2CCCC(N(C(=O)CCC3CCCC3)CC)C2)=O)c(F)ccc(C#N)c1F c1(C(=O)NC2CC(CNC(c3n(C)c(O)nc3)=O)C(O)C2)cccn2nnnc12 C1(F)(CNC(C(c2ccc(F)cc2)OC)=O)CCN(C(=O)CC2CCC(=O)N2)C1 C1(C)(C(C)C)CCN(C(C23CC(C)(CN2C(=O)C(C)C#N)C3)=O)CC1 c1(C(=O)O)ccn(CC(=O)NC2CN(C(C3CC(N4CCCC4)C3)=O)C2)n1 c1(N2CCCN(C(c3ncc(C)[n+]([O-])c3)=O)CC2)ccc(C)n(C)c1=O Cc1cc(F)c(C(N2CCC3(C2)CN(C(c2cnc(O)s2)=O)C3)=O)cc1F O=C(CCCCCCNC(c1ocnc1C1CC1)=O)NCCC(F)F C1(NC(c2ccnn2CCF)=O)CCCCC1CNC(C1CCCO1)=O CC1(C)C(NC(=O)Cc2ccc(F)cc2F)CCN1C(C1COC(=O)O1)=O C1(CNC(CC=C=C)=O)CCN(C(=O)CNC(C2CCCCC2)=O)CC1C Cc1nc(F)ccc1-c1cn(CC2CCN(C(C3C=CCC3)=O)C2)nn1 C1(C(=O)NCC2(NC(c3ncn(CC)n3)=O)CCC2)CCn2c(cnc2C)C1 N1(C(C(C(=O)OC)C)=O)CCCN(C(c2ccc(F)c(Cl)c2)=O)C(C)C1 c1(OC)cc(C(=O)NCC2COCCN2C(c2ccsc2)=O)cc(C2CC2)c1 C1(NC(CC(CC)C)=O)CC2CC(NC(c3cc(CO)[nH]n3)=O)C1C2 CN1CCC2(OC(F)(F)F)CCCCC2(C(=O)Nc2ccc(C#N)cc2[N+](=O)[O-])C1 C1(CCNC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1 C1(NC(C=Cc2ccc(C)o2)=O)C(C)CN(C(C23CC(CO2)C3)=O)CC1C C1(C2CCCN(C(=O)C=CCO)C2)(NC(CC2C(C)=NN(C)C2=O)=O)CC1 Cc1nn(C)c2cc(-n3cc(C4CCC(C)C(C)C4)nn3)ccc12 C(c1nnn(C)n1)=CC(=O)NC1(C2CCN(C(C(N3CCOCC3)C)=O)C2)CC1 N1(C(C2CCOCC2)=O)CCN(C(C23CC(O)C2C3)=O)CC1C1CCC1 N1(C(CSC)=O)CCOC2CN(C(=O)C(C(C)C)n3cc(C)cn3)CC12 C=CCC(C(=O)N1CCC(C(C)(C)C)C1)NC(c1ccc(OCC)nc1)=O c1(C(N2CCC(C(=O)NCC3CCC(F)C3)C2)=O)ccc(F)c(Cl)c1 c1(OC(C)(C)C)ccc(C(N2CC(NC(=O)C=C3CCCCC3)C3CC23)=O)cc1 C12(NC(C(C)OCC)=O)CC(C)(C1)OC21CCN(C(C2CCC(F)(F)C2)=O)CC1 c1(OC)ccc2c(c1)CCCC2C(=O)NC12CC(NC(=O)CO)(C1)C2 c1(C(N2CCN(C(C(C=C=C)C)=O)C(CC)C2)=O)nncc2ccccc12 c1(NC(C2CCCC(NC(C3(Br)CCC3)=O)C2)=O)cccc(F)c1Br c1(CNC(c2nc(CNC(C=C(C)C(C)C)=O)oc2C)=O)cncc(C#N)c1 N#Cc1ccc(F)c(S(=O)(=O)Nc2csc3nccnc23)c1 CCS(=O)(=O)c1ccccc1CCNC(=O)NC1CN2CCC1C2 C(=O)(C(C)(C)CC(F)F)NC1CCN(C(c2c(CC)cccc2C)=O)C1 N1(C(C(C2CN(C(C3(OC)CCOCC3)=O)C2)O)=O)CCCC(N=[N+]=[N-])CC1 c1(C(C)NC2CC2)ccc2c(c1)CCO2.N1(C2CN(C=O)C2)CCOCC1 C(=O)(C(F)(F)F)NCC(=O)NC1CCN(C(=O)C(O)c2ccco2)C1 Cc1ncnc(C(=O)NCC2(F)CN(C(=O)C(c3ccccc3)F)C2)c1C Cc1cccc2[nH]cc(CC(=O)NC3CCCN(C(c4coc(C#N)c4)=O)C3)c12 C=CCCCC(=O)N(CC(CC)NC(C12CC(C#N)(C1)C2)=O)CC Cc1cc(C(=O)NC(C)CCN(C(=O)CNC(=O)CCC(C)C)C)c(O)nc1C c1(OC)ccc(NC(C2CCCCN2C(c2ccc(O)cc2O)=O)=O)c(F)c1 c1(OC)ccc(Cl)cc1CC(=O)NCCOC(C)(C)CNC(=O)CCCN(C)C C(=O)(C(CC)CCC)N1CCC(C)(NC(COCCCCOCC#C)=O)C1 C1(C(=O)NCc2ccc(C)o2)CC2C=CC1N(C(=O)CC1CCC(=O)C1C)C2 c1(C(C)C)cccc(C(=O)NCCN(C(c2ccc(F)s2)=O)CC(C)(C)C)n1 N1(C(c2c(OC)csc2)=O)CC2(CCN2C(c2ncccc2Cl)=O)C1 C(=O)(CCCN=[N+]=[N-])NCCN1CCNC(=O)C1.CC12CC(C1)C(=O)N2 N1(C(C2C(C)(C)C2)=O)CCN(C(=O)Cc2cnc[nH]2)CC1c1ccc(F)cc1 N1(C(Cc2nc(C(C)C)sc2)=O)CCCC(C2CC2NC(c2cnsc2)=O)C1 C1(CC(=O)NC(CNC(=O)CC23CCC(CC2)OC3)C2CC2)CC2(CCC2)CO1 c1(CC)cc(C)nc(NC2CCCCC2CNC(=O)C(F)=CC2CC2)n1 N1(C(C2(C)CCCO2)=O)CCCC(NC(C2(F)CC=CC2)=O)CC1 c1(C(=O)NC(CCNC(C=C(C)C(C)C)=O)(C)C)ccc2cnoc2c1 c1(CC(=O)NCC2OCCN(C(c3c(C)cncc3)=O)C2)ccc2[nH]ccc2c1 C(=O)(C(C)(C)C(C)(F)F)N1CCN(C)CC1CNC(C1(CCF)CC1)=O Cc1cccc(C(=O)NCC(C)(C)CNC(=O)CN=S(C)(C)=O)c1C#N C1(CC#C)(C(=O)NCCC(O)CN)CC=CCC1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(=O)C=Cc2cn(C)cn2)CC12CCCC2 C1(C(C(=O)NCC(C)F)C)CCN(C(c2ccc[n+]([O-])c2)=O)CC1 c1(OC)ccccc1OC1CCN(C(C2(N)CCSCC2)=O)C1 N1(C(C=CCCC)=O)CCC(CNC(=O)Nc2cnn(C3CCC3)c2)C12CCC2 Cc1ccc(CNC(=NC(C)CC2CCOC2)NCC(F)F)c(=O)n1C C1(C(C)C)CCC(C)CC1(O)CNC(=O)Cc1c(F)ccc(Br)c1F C(=O)(C1=CC2CCCCCC12)N(C)CC1COCCN1C(C1CCC(=O)N1)=O C(=O)(CC(C)C(F)(F)F)NC1C(CNC(c2c(-c3ccc(C)o3)onc2)=O)CC1 c1(CC)cnc(C(C(=O)NCC2CCOC2)N(C2CCCC2)C2CC2)o1 C(C(C(C)(C)C)NC(=O)C=Cc1ccsc1)NC(CCCc1onc(C)n1)=O C1(NC(c2ccc(C(=O)OC)o2)=O)CCC(NC(=O)C(C)c2ccon2)CC1 N1(CC(=O)NCC)CCC(NC(=O)NC(=O)COCC2CCCO2)C(C)C1 CN1CC(C)(C(=O)NC2CCN(C(=O)CCc3cncc(F)c3)CC2F)CC1=O c1(C(=O)OC)cc(C)cnc1NC1CN(C(=O)C(C)(C)C(C)C)CC1C C1(NC(C(CC)SCc2ccccc2)=O)CN(C(=O)Cc2scnc2C)CC1C c1(C(N(CC(CNC(CCc2cc(C)on2)=O)O)C)=O)cccn2ccnc12 N1(C(c2cc(CC)no2)=O)CCC2(CCCCC2NC(=O)CCCN(C)N=O)C1 N1(C(CNC(CCCC)=O)=O)CCN(C(C2(n3cncn3)CC2)=O)C(CCO)C1 c1(C(c2c(CNC(C(n3c(C)cc(C)n3)C)C)cccc2)=O)cccc(F)c1F c1(C(N(CCNC(c2cnccc2Cl)=O)CC)=O)cn2ncnc2nc1C C1(CN(C(c2ncn(C(C)C)n2)=O)C)COCCN1C(=O)Cc1cscn1 C(=O)(C1=CC2CCC=CCCC12)N1CC(CCNC(c2ocnc2C)=O)(OC)C1 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)C(NC(=O)C(C)(C)N2CCCC2)C1 C1(NC(C2CCCC(CF)C2)=O)CCCC2CN(C(=O)C=C3CCCC3)CC12 c1(C(N2CCCC(CNC(C3ON=C(C)C3)=O)CC2)=O)cc(C)cc(C)c1C CC1CN(C(c2cc(C(N)=O)no2)=O)CC1NC(=O)CC1CCCN(C)C1 C12(C(=O)OC)CC(CO1)N(CC1CCCN1Cc1ccccc1)C2 C=CCC(CC(F)F)C(=O)N(C)CC1(O)CCCN(C(=O)CCC(C)CC)C1 N1(C(C2(C#N)CC3CC3C2)=O)CC(NC(c2cnc(Cl)s2)=O)CC(F)(F)C1 N(C(=NCC1CCCN1C)NCc1sccc1C)C(C#C)CC1CCCO1 N1(C(C(CC)(C)F)=O)CC(NC(=O)CCn2cccn2)CC(F)C1 C1(C(=O)NCCNC(=O)CC2CCCNC(=O)C2)CCC(C2CCC2)CC1 c1(C(N2CCOC(CN=[N+]=[N-])C2)C(=O)NCCCC)ccc(COCC)cc1Br Cn1c(C(F)F)nc2cc(C(=O)NCC(O)CNC(C3CNC(=O)C3)=O)ccc12 CC1Cc2cccc(O)c2N(CC2(C#N)CCCCC2)C1 CC1CC=C(C(=O)NC2CC3CC2N(C(c2ccccc2CC#N)=O)C3)CC1 C1(CNC(CCS(C)=O)=O)CCN(C(=O)CCSCc2ccc(F)cc2)C12CC2 C1(CC(=O)NC(C2CSC2)C)CCN(C(C2CC3C(C2)C3(F)F)=O)C1(C)C n1(CC)ncc(Cl)c1C(=O)NC(CNC(=O)C=C1CCOCC1)CO C1(C(N2CC[Si](C)(C)C2)=O)CN(C(=O)C2=CCCOC2)C2(CCC2)C1 Cc1noc(Cl)c1CC(=O)NC1CCCC(CNC(=O)CCn2cnnn2)C1 CCCC(CCNC(C1OCCC1CNC(c1occc1C(C)C)=O)=O)CCC N1(C(C(=O)NC(CCCCC)C(C)(C)C)=O)CCSC2(CCCCC2)C1 CC1CCOC(C(N2CCC(NC(c3ccc(CN=[N+]=[N-])cc3)=O)C2)=O)C1 C1(Nc2cc(N3CCC(C=C)C3)nc(C)n2)CCc2nn[nH]c2C1 c1(C(C(=O)NC2CCC2)N(CCCC)CC)nscc1Br CC(C)(C(=O)N(CC(S(C)(=O)=O)c1ccccc1)C(C)(C)C)C(=O)N1CCCC1 Cc1c(Cl)ccc2[nH]c(C(N3CCCN(C(C4CCOC4)=O)C(C)C3)=O)cc12 O=C1OCCCN1CC(N1CCOC(C2CN(C(=O)Cc3ccco3)C2)C1)=O N1(C(CC=CC=C)=O)C2CCC1CC(CNC(c1cc(O)nc(Cl)c1)=O)C2 c1(C(=O)NC2(CO)CN(C(Cc3c(C(C)C)con3)=O)C2)cccc(O)n1 c1(N2C3CS(=O)C(C3)C2)nc2ccccc2c(=NCc2cccc3nc[nH]c23)[nH]1 C(=O)(C1CCC(=O)c2cccn21)NCCN(C(C1CCC(C)(C)CC1)=O)C1CC1 CC(CC(=O)NCCCCC(=O)N1CCCC1)C(F)F c1(CC(=O)NC2CN(C(CSC)=O)CC2n2ccnn2)cncc(C#N)c1 CCC(F)(F)C(=O)NCC1(O)CC(NC(c2ccnc(NC(C)C)c2)=O)C1 Cc1cc(N(C(C)CNC(=O)C(C)C(C)S(C)(=O)=O)C)n2ncnc2n1 CCCCC(C(=O)N1CCC(F)(CNC(c2c(C)cccc2O)=O)CC1)C(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)NC2=O)N.Cc1c(C(=O)C2CC2)nn(C)c1 c1(CNCC2(F)CCCN(c3ccnc(OC)n3)C2)cnc2ccccn12 C1(CCC(=O)NCc2nc(C)sc2)COCCN1C(=O)C(C)C N1(C(C(CCC)C)=O)C2CCC1C(NC(c1sc(Cl)c(Cl)c1C)=O)C2 C=CC(C)(CCOC)C(=O)NC1CCCN(C(=O)Cc2cnc(C3CC3)[nH]2)C1C CCCCC(C)C(=O)NCC1(CN(C(=O)CC2CCCC2O)C)CC1 c1(C(=O)NC2(COC)CN(C(C3CCOC3C)=O)C2)ccc(Cl)cc1 Cc1ccc(C(=O)NC2COCCN(C(c3cn(C)nc3C)=O)C2)c(I)c1 O=C(CC=C(Cl)Cl)NC(C(=O)NCC1CC1C1CCC1)c1ccoc1 Nc1cccnc1C(=O)NCC(c1ccccc1)CNC(=O)CNC=O c1(NC2CCN(C(=O)OCC)CC2OC)ccc2ncc(Br)cc2c1 CC1CCN(C(C2COC(C)C2)=O)CC1NC(=O)CNC(c1ccc(N)cc1)=O CCC(C(=O)NCCCCN(C)C(c1cn(C)[nH]c1=N)=O)C(C)(F)F N12CC3(C1)CN(C3)C(=O)OCCN(C)C2=O.c1(OC(C)(C)C)cn[nH]c1 N1(c2ccnc(C(CC)C)n2)CCn2ncc(CNC(=O)CCC(C)OC)c2C1 Cc1cnn(CC(C)NC(=O)C(n2cc(C(c3ccccc3)O)nn2)C)c1 c1(C(N2CCOCC(NC(C(C)O)=O)C2)=O)c2c(nn1C)CCSC2 N1(C(c2cc(CC)n(C)n2)=O)CCC2(NC(=O)CC(CN(C)C)CC)CC2C1 C(=O)(C(Cc1cnc[nH]1)NC(=O)CC(C)F)NC(c1cnn[nH]1)C c1(C(=O)NC2CC(CNC(CN3CC(C)C3)=O)C2)cnc2c(ccn2C)c1 c1(Nc2cn(C)c(C(=O)NCc3ccc(O)c(O)c3)c2)ccc(C#N)nc1 C1(O)(C2CN(C(C(Cc3ccccn3)NC(=O)OC(C)(C)C)=O)C2)CCCN(C)C1 c1(C(=O)NCC2(C)CC(NC(c3c(OC)ccs3)=O)C2)cccc(C2CC2)n1 C1(C(N(CCC#N)CC)=O)(C(=O)OC)CC1(C)C N1(C(C2CCCN(C(CC3CCCN(C)C3)=O)C2)=O)CCC(F)(CO)CC1 N1(C(C(CCC)NC(C)=O)=O)CCN(C(=O)CC2=CCCC2)C(CC(F)F)C1 C1(C(N2CC(CNC(CSCC(N)=O)=O)OCC2)=O)C2Cc3ccc(Cl)cc3C12 C1(C(=O)NCC(COC)OC)CCCCCCN1C(=O)C1=CCCCO1 C1(NC(c2ccc(C)nn2)=O)C2CC1CN(C(=O)C(F)CC1CCCC1)C2 c1(C(N2CCC(C)(NC(CCN(S(C)(=O)=O)C)=O)C2)=O)nc(Cl)ccc1N Cc1[nH]c(C(N2C3CCC2COC3)=O)c(C)c1C(N1CCC(C)C1)=O N1(C(c2c(COC)n(C)nc2)=O)C2CCC1CC(NC(C1CCNC1=O)=O)C2 C1(CNC(c2cccc(C(C)C)c2)=O)(NC(c2cscn2)=O)CCCCC1C c1(C(=O)NCC(C)N(C(C(CC)O)=O)CC)cccc(-n2ccnc2O)c1 Cc1[nH]nc2c1CCC(C(N1CC(C)(NC(c3ccccc3Br)=O)C1)=O)C2 c1(C(=O)NC2(C(=O)NCCCN=[N+]=[N-])C(C)(C)C2)ccc(O)cc1F C1(CNC(c2c(C)ocn2)=O)CC12CCN(C(C1CCCC(=O)C1)=O)CC2 Cc1nsc(C(=O)N(C2CCN(C(=O)Cn3nnc(=N)[nH]3)C2)C)c1Br N1(C(C(C)N2CCC2)=O)CCN(C(c2cnn(CC(F)(F)F)c2)=O)CC(C)(F)C1 c1(-c2c(C)csc2)cnc2c(C(=O)Nc3cnc(Br)c(C)c3)c[nH]c2c1 Cc1nc(C(=O)NC(C)C(=O)N(C2CC(C)C2)C)ccc1C#N c1(OC)cccc(S(=O)(=O)N2CCC23CN(c2cc(C#N)ncn2)C3)c1 c1(CN(C)C(C2(CNC(=O)COC3CCCOC3)CCCO2)=O)ccncn1 N1(C(c2c(C)scc2)=O)CC(NC(=O)CC2CCSC2)C(O)C1 N1(C(C)=O)CCCCC1C(=O)NC1CCC(CNC(c2cc(CCO)on2)=O)C1 c1(OC)cncc(C(=O)N(CC(=O)NCCC2CC(C)(C)C2)CC(C)C)c1 Cc1ccc2occ(C(=O)NC3CCCN(C(=O)C#CC4CCCO4)CC3)c2c1 C1(NC(Cc2c(C)non2)=O)CC(O)CN(C(=O)Cc2ccc(F)cc2)C1 c1(C(N2CCC(NC(c3nnn(C)c3C(F)F)=O)C2)=O)cccc2c1CCOC2 CCCC(CCCNC(=O)C(C)Cc1ccco1)NC(=O)CS(=O)(=O)NC c1(C(=O)NC(CNC(c2ccc(OC)c(C)c2)=O)C(C)C)cnn2cnccc12 N1(C(C2CCCN(Cc3cccn4nccc34)C2)=O)CCCC2(CCOC2)C1 N1(C(c2cc(C(C)=O)on2)=O)CC(F)CC1CNC(=O)CC(C)(C)N(C)C C1(CCC)CN(C(=O)C(C2CCC2)OCC)CCN1C(=O)C1=CCCSC1 Cc1cc(=NCc2nnn(-c3ccc(F)cc3)n2)nc(-c2cccnc2)[nH]1 C(=O)(CCC(=O)NN(C)C)NCC(CC)NC(=O)Cc1[nH]cnc1C C(CC(C(C)(C)C)NC(=O)CCOCCN(C)C)N(C(CCCC#C)=O)C CC1CCC(CNC(c2ccc(N)c(Cl)c2)=O)CN1C(c1ccns1)=O C1(NC(c2n[nH]c3c2CCCC3)=O)CCCCN(C(c2ccoc2)=O)CC1 C1(C(N2CCN(C)CC2)=O)C2CCC(C2)C1NC(=O)CC1CC=CC1 N1(C(C(C)(C2CC2)OC)=O)CCN(C(c2csnn2)=O)C2(CCC2)C1 C#CC#CC(C)(C)NCC1CCN(C(=O)OC(C)(C)C)C1CC Cc1cc(=NC(=O)C(F)C2CCN(C(=O)CCCN3CCCC3)C2)[nH]n1C CC1=NN(C)C(=O)C1CC(=O)N(C)CCN(C)C(c1ccnnc1S)=O C#CC1(C(N2CCOCC(O)C2)=O)CCN(C(=O)OC(C)(C)C)C1 CC1C(NC(C2CC3(CC3)CO2)=O)CCN1C(=O)CC1(C)CC1 c1(OC)cc(OC)cc(C2CCN(C(C3CCCC3C(F)(F)F)=O)C2)c1 C(=O)(CC(C)(C)CNC(C1CC=CCO1)=O)N(CCC(C)C)C c1(SC)cccc(C(=O)NC(CO)C(C)NC(=O)CC2(C3CC3)CC2)c1Cl C(=O)(C1=CCCCCC1)NC1(C)CCCN(C(c2coc3c2CCCC3)=O)C1 C1(C(C(=O)OC)N(c2ccc(NCC)cc2)C)CCC2(CC(C(=O)OC)C2)O1 c1(NCC(=O)NC2CN(C(c3cn(CCC)nn3)=O)C(C)C2)cccc(C#N)c1 C1(NC(C(C)N(C(c2c(F)ccc(C)c2)=O)C)=O)CCc2nn[nH]c2C1 C1(NC(CC2(COC)CCCC2)=O)CC2CCC1N(c1ncc(C)c(O)n1)C2 c1(OC)cc[n+]([O-])c(C(N2CC(N(C)C(c3cc(C)cc(C)c3)=O)C2)=O)c1 C1(C(=O)NCC2CCCCN(c3ncnc(C(F)(F)F)n3)C2)CCCCC12CCC2 c1(C(=O)NCC2C3CN(C(=O)CCC4CCCC4)CC23)cn2c(n1)COCC2 c1(C(N(C2CCN(C(C3CCC(N(C)C)CC3)=O)C2)CC)=O)cncc(Cl)c1C S(=O)(=O)(C1CCCCC1)CNC1CC(c2ccc(Br)cc2)(C)C1 C=CCC(C(=O)N1CCC(=C(F)CNC(=O)C(O)CC(=O)OCC)CC1)C(C)C c1(NC(C2C(C(N3CCN(CC(=O)NC)CC3)=O)C2)=O)c(C)cc(Br)cc1Cl C1(CNC(=O)CC2NC(=O)NC2=O)CC2(CCN(C(=O)CC(O)C3CC3)C2)CO1 O=C1CC(C(N2CC(NC(=O)CO)C(CC3CC3)C2)=O)CC(=O)N1 CCCC(C(=O)NCC1CN(C(C2CC(N3CC(O)C3)C2)=O)C1)C(C)C C1(NC(=O)CCNC(C2COC(=O)N2)=O)CN(C(c2cnns2)=O)CC12CC2 Cc1nc(-c2ccsc2)sc1C(=O)NC1CCCN(C(=O)CC2CC3(CC3)C2)C1 N1(C(C(c2ccccc2)OC)=O)CC(NC(c2ccc(Cl)c(O)c2)=O)C2(CC2)C1 c1(C(=O)NCCC(C)NC(c2cc(N(C)C)ccn2)=O)cc(F)n(C)n1 CCC(C(=O)NCC1CN(C(=O)CCOC(C)C)CCN1C)C(C)(F)F C1(NC(C(c2ccc(F)cc2)(C)C)=O)CCCN(C(c2ccncc2)=O)CC1 c1(C(C)=O)ccc(C(=O)N(C(C)C(=O)NC(c2nc(C)cs2)C)C)o1 c1(CC)ccc(C(=O)N(C)CC2CN(C(=O)Cn3cccc3)CCO2)cc1F C1(NC(CC(=C)C)=O)CC2(C1)CC2NC(C1CCC(CC#N)CC1)=O C1(CCCC)CN(C(C(=O)NCCNC(C)=O)C(C)C2CCC2)CCO1 C1(NC(CCCC(C)=O)=O)CCC2(CCCN2C(=O)C2Cc3ccccc32)CC1 c1(CNC(C2CCCCO2)C)cc(Br)cc(Cl)c1O C1(C(=O)NC2(C(=O)OC)CCCC2)CC2CC2N1C(=O)Cc1cccc(Cl)n1 C1(C(=O)NCc2occ(C(N(CC(C)(C)C)CCC#C)=O)n2)CN(C)CCO1 c1(OC)ccc(NC(=O)C(C)(C2CC2)NC(=O)NC(C)(C)C)c(C)c1 N1(C(C2(C)CC(C)C2)=O)CC2(CCCC2NC(=O)Cc2cn3ccccc3n2)C1 C(c1ccc[nH]1)=CC(=O)NC12CC(CNC(c3cnoc3C3CC3)=O)(C1)C2 C=C(C)CCC(C)NC(=O)CC1(N(C(=O)C(C)COCC)C)CC1 N1(C(c2n(C)ncc2)=O)CCN(C(C2CCCCN2C(=O)CCS(C)=O)=O)CC1 N(C(=NCCN1CCn2nccc2C1)NC(C)CC(F)F)C(CC)CC C1(CNC(CCC=C)=O)(OC)CCN(C(c2cnn(CC3CCCC3)c2)=O)CC1 CC(C(=O)NCC1CC2(CC(NC(C3(CF)CC4(CCC4)C3)=O)C2)C1)C(F)(F)F N1(C(C(=O)NCC)c2ccns2)CCCCC1CNC(c1ccccc1)=O c1(C(=O)NC(CNC(C(CCCC)=O)=O)CCCC)cc(S(=O)(=O)NC)c[nH]1 C1(NC(C(=Cc2ccccn2)C)=O)CCC2(CC1)CC2NC(=O)COCC1CC1 C(=O)(C1CCc2ccccc21)N1CCN(C(C(=O)NC2OCCN(C)C2)=O)CC1 N1(C(C2CC(OC)C2)=O)CCN(C(C2CCC(c3ccccc3)O2)=O)CC1CF C12(NC(CC3CC(SC)C3)=O)CC1CN(C(=O)Cc1sc(O)nc1O)C2 c1(CC(=O)N(C2CCN(C(C(C)C)=O)C2)C)ccc(Br)cc1[N+](=O)[O-] c1(CC)nc(C(=O)NC2CC2CNC(c2cc(F)cnc2O)=O)c2ccccn12 C1(N(C2C(C(=O)O)CCC2)Cc2ccccc2)CCc2nc(C(F)(F)F)cn2C1 N1(C(=O)CCC2CCC(O)CC2)CC2CCC(C1)N2C(=O)C(O)c1ccsc1 c1(C(=O)NCC2CCN(C(C3CC3F)=O)CC2(F)F)ccc2ccnc(O)c2n1 c1(C(N2C(C(C)NC(C3CCSC3)=O)CCC2)=O)cc2ncccc2cc1Cl C1(NC(C(CCCC)C)=O)CN(C(=O)COCC(C)C)CC2CCCC12 c1(N2CC=CC(NC(c3n(CC)nnc3)=O)C2)ncnc2sc(C(F)(F)F)nc12 c1(NCC(=C)Br)ccc(S(=O)(=O)NCC2(S(N)(=O)=O)CCC2)cc1F CC1=C(C(=O)N2C3CCCC2CC(CNC(=O)C(O)C(C)C)C3)CCC(C)(C)C1 c1(C(N2CC(C(C)NC(=O)CCC(=O)N(C)C)C2)=O)cc2cnccc2[nH]1 Cc1cnc(F)c(C(N2CCC(C(C)NC(=O)C(C)(C)C3(O)CCOC3)C2)=O)c1 c1(OCC)ccnc(N2CC(CN(C(=O)CCn3ccnc3)C)C2)n1 C1(N(C)C(C2CC2C2CC2)=O)CN(C(C2CCCCC2)=O)CC1O CC1=C(C(=O)N2CCOCC2CNC(=O)CSc2nccn2C)CCC1 C(=O)(C1=CCC2CCC1N2C(c1nccn1C)=O)N(c1ccc(F)cc1)C C1(NC(CN(C2CCC2)C)=O)COCCC1C(=O)N(C)OCC#N c1(OCC)cc(-c2ccc(N(CCCn3ccnc3C)C)c(F)c2)ccc1C N1(C(CC(C)(C)C2CC2)=O)CC2C3CCC(C2C1)N(C(C1CC=CCC1)=O)C3 N1(C(C2CC(SC)C2)=O)CC2CCCC(CNC(c3cc(C#N)c[nH]3)=O)(C2)C1 N1(C(c2ccnc(C)c2C)=O)CCC(C)(C)C(CNC(=O)COC2CCOC2)C1 CC1=CC(C)C(C(N2CC(CO)CC2C)C(=O)NCCOCC2CC2)CC1 c1(C(N2CCC(CCOC)(NC(c3csnn3)=O)C2)=O)cccc2nonc12 c1(C(=O)NCC(C)NC(=O)CC(=O)NC2CC2)ccnc2c1nnn2C C1(CN(C(C(C)NC(=O)NC)=O)C)CCCCN1C(=O)CC1(O)CCC1 N1(C(c2c(CC)cno2)=O)CCOCC(NC(=O)C=Cc2scnc2C)C1 C1N=C2C=CN=C(N2)C(=O)N2CCOCC12.C(=O)(CNC(=O)N)OC.C1CC1 c1(C(N2CCCC(NC(c3n(CC)nc(C)c3)=O)C2)=O)cc2ccccc2o1 C1(CNC(COC)=O)CCN(C(c2cccc(C)c2O)=O)CC1C C(=O)(CC(C)CC(C)C)N(CCNC(c1cncc(C(N)=O)c1)=O)CC C1(C(C)NC(C=C(C)C(C)(C)C)=O)CCCCN1C(=O)C(=CC1CCCC1)F C1(CN2CCCC(NS(CC)(=O)=O)C2)NCCC12CCCC2 c1(C(=O)NCC23C(CN(C(C(F)=C(C)C)=O)C2)C3)cc(Br)cc(N)c1C N1(C(CCOCC#C)=O)CCCC2CN(C(c3ccc(NC(C)=O)s3)=O)CCC12 C(=O)(CCCC(=O)OC)N1CC(NC(C2CCC(OCCC)C2)=O)C(SC)C1 N1(CC(C)(C)NC(Cc2c(C)ncs2)=O)CCN(C(C2(C(N)=O)CC2)=O)CC1 N1(C(C2(C)CC3CCC2O3)=O)CC2(C1)C(NC(c1ccns1)=O)CCS2(=O)=O n1(CC(=O)N(CCCNC(C2CC2(C)CC)=O)CCC)ccc(=O)cc1C C12(CCCO1)C(=O)NC2.N1(C(C2CN(C(=O)NC)C2)=O)CCC(CO)C1 C(C(=O)N(C1CN(C(=O)CC2CC=CCC2)C1)C)(C(C)C)c1cnc(C)s1 C1(CN2C3(COC)CC(c4ccc(C(C)C)cc4)(C2)C3)CCS(=O)(=O)C(C)C1 O=[N+]([O-])c1cc(C(=O)O)c(Nc2ccc(Cn3cccn3)cc2F)s1 C(C(=O)Nc1ccc(Cl)cc1F)(C1=CCCSC1)N(CCC)CC1CCOC1 N1(C(CSc2n(C)nnn2)=O)CC(C2CN(C(c3cccc(N)n3)=O)C2)C1 C(=O)(CCS(=O)(=O)N(C)C)N1C(C)CC(NC(C(=Cc2ccncc2)C)=O)C1 c1(C(=O)NC(CCNC(C(C)Cn2cccn2)=O)C)cc(Br)cnc1O O=C1Nc2c(C(N3CC4CN(C(C5CC5Cl)=O)CC(C3)O4)=O)cccc2C1=O c1(OCC)ccnc(N2CCN(C(=O)CCN3CCOCC3)CC2)n1 C(=O)(C(O)CC(F)(F)F)NCC1C(C(=O)NCC(CC=C)(F)F)CCCC1 C#Cc1ccc(C(=O)NCC(C)N(C)C(c2ccc(F)c(CC)c2)=O)cc1Cl c1(NCC(CC)OC)ccc(S(=O)(=O)NC2CCOC3(CCCCC3)C2)cc1Br N1(C(C2(C#N)CCC2)=O)CCC(CNC(=O)CC(F)(F)C(F)F)C(F)(F)CC1 c1(CN2C(C(=O)Nc3ccc(C(C)=O)cc3)CSCC2)ccc(C)nc1F c1(OC)nc(CN2CCN(C3CCC3)CC2)ccc1-c1nn[nH]n1 Cc1cnc(NC(c2ccnc(-c3ccccn3)n2)=O)c(Br)n1 C1(N(C(CC2CC(=C)C2)=O)C)CCC2CN(C(c3cnc(NC)cn3)=O)CC12 C1(C)(CC)C=C(C(=O)N2CC(F)(F)CC2C(=O)NC2CCC(C)CC2)C1 Cc1ccc(C(N2CC3CC2C3NC(=O)CC(C)C)=O)nn1 Cc1noc(C)c1CC(N1CCC(C(C)(C)NC(C2COCCO2)=O)C1)=O c1(C(N2C(C)(CNC(CC3C(C)CCC3)=O)CCC2)=O)cc(S(C)(=O)=O)co1 Cc1ncn(C)c1C(=O)NC(C)CCNC(=O)CCCCC1CCCCC1 C(=O)(C(C)CC(F)(F)F)N1CCC(CNC(C(CCC)(C)O)=O)CC1 C1(C(=O)OC)Cc2n[nH]cc2N(C(=O)C(c2ccc(Cl)cc2)O)C1 C1(CC(N2CC3C(NC(C4C5CC6C(C5)C46)=O)C3C2)=O)CCC2(CCC2)O1 c1(C(=O)OCC)ccc(NC(C2CC2NCc2ncco2)=O)cc1 CCCC(C)(CC)C(=O)N1CCC(O)(CNC(=O)COC)C1 C(CC(C)(C)C)(C(=O)N(C(C)C(=O)NCCC1CC1)C1CCSC1)OC Cc1cc(C(N2CCCC2C(C)(C)C(N2CCNCC2C(C)C)=O)=O)nc(C)c1 C(=O)(C1c2ccccc2C2CC1C2)N1C(CC)CN(C(=O)CC(C)SC)CC1 N1(CC(=O)Nc2ccccc2OC2CCCC2)CCc2nc(O)ccc2C1 CN(C)S(=O)(=O)N(C)CC(=O)NC1CN(C(=O)CCc2ccoc2)CC1O C=CCCC(C(=O)OC)NC(=O)CC(C1CC1)NC(c1cnc(O)n1CC)=O C1(COCC(CN(c2ccccc2F)C)O)CCCC(C(C)(C)C)C1 N1(C(=O)OCC)CCC(C(=O)NC(Cc2cncn2C)C(=O)O)CC1 C(C)(CC(=O)N1CCC1(C)CC(=O)NCC1COCCO1)=C(C)C c1(C(=O)NCCCCCNC(c2cc(CC)sn2)=O)cc(C)nn1C(C)(C)C c1(CC(=O)OCCCCN(C(C)C)C)c[nH]c2cccc(-c3cnc(F)c(Br)c3)c12 C(CS(=O)(=O)NC1(CCCC(C)C)CC1)(C1CCOC1)OC.OC O=C(C1CCCn2cnnc21)NC1C2CC1N(C(C1CCCC3(CC3)C1)=O)C2 C12(NC(C(CC)O)=O)CC(CNC(c3cnc(S)[nH]3)=O)(C1)OC21CCC1 N1(C(c2[nH]nc(C(=O)OCC)n2)C(=O)NC2(COCC)CC2)CCCS1(=O)=O c1(C(=O)NC2C(CNC(C3(C(=O)NC)CC3)=O)C2)ccc2cc(OC)ccc2c1 C1(C2CC2)(C(=O)NC(C)C(=O)N(C)C)CN(C(=O)CC(C)CN(C)C)C1 C1(C)(C(=O)NC(CCC)CC)CCCN(Cc2cccc(SC)c2)C1 CC1CCN(S(=O)(=O)CC(=O)N(CCCNC(C2CC3(C2)CC3F)=O)C)CC1 c1(C(=O)O)cccc2c1N(CC(C1NCC13CCOCC3)=O)CC2 c1(NC(C)=O)ccc(F)c(C(N2CC=CC2CNC(=O)C(O)C(C)(C)C)=O)c1 c1(C(=O)NC(CC#C)C(=O)N2CCCC2C2CCCC2)cccc2occc12 c1(C(N(C(C)C(=O)N2CC(C3CCC3)C2)CCC)=O)cnc(C2CC2)o1 c1(NC(c2cccc(C(=O)NC3CC(F)C3)c2)=O)cc(Cl)ccn1 N(C)(C1CN(C(=O)CCCCSC)CCc2ccccc21)C(C1(CC)CCC1)=O c1(NC(=O)NC2C(CC=C)C(O)C2)cccc(P(C)(C)=O)c1 c1(CC)cc(C(=O)NC2(CC=CC(=O)NCC(C#N)CC)CCC2)c(C)o1 c1(C(=O)NC(C2CCN(C(=O)C(C)(C)c3ccsc3)C2)C)cnc2[nH]nnc2c1 c1(C(N2CC(CCC)C(NC(=O)Cc3cccnc3)C2)=O)cc(C)ccc1CC C1(N(C(=O)CSCC2CCCO2)C)CCN(C(c2cscc2Cl)=O)CC1 C(C1CCC(=O)c2ccccc21)N1CC(=O)OCC12CCC2 c1(C(N(CCC)CCNC(c2ccnn2C2CCC2)=O)=O)cccc2c1OCC2 C(C(CO)(CO)NC(c1occc1C)=O)N(C(CSCCOC)=O)C c1(CN(C(c2ccccc2)C(C)C)C2CC2)ccc(Br)c(C(F)(F)F)c1 N1(C(CC2CCC(=O)NC2)=O)CC2(C1)CN(C(=O)C=C1CCC1)CC2CO N1(C(C2(C)CN(S(c3c(C)n[nH]c3C)(=O)=O)C2)=O)CCCC2(C1)OCC1CC21 C1(C(N(C(CC)CC)CC(F)(F)F)=O)(OC)CCN(C(c2cocn2)=O)C1 CC(CC(C)NC(c1ccnn1-c1ccccc1)=O)NC(C1CCOC1)=O C1(C(=O)NC2CCCC(CNC(Cn3c(C)ncc3)=O)C2)CC2CC(=O)C1O2 C1(Cl)(C(N(CC(CNC(C=C(C)C2CCCCC2)=O)O)C)=O)CC12CCOCC2 C1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CC(O)C2O)CCn2c(C)cnc2C1 N1(C(C(CCC)F)=O)CC2CC(C1)CN(C(=O)CNC(=O)C(C)CC)C2 c1(COC)c(C(=O)NC2C=CCN(C(C3(CF)CCC3)=O)C2)cnn1C c1(C2(C(=O)NCC(CNC(C3(OC)CC3)=O)(C)O)CC2)ccc2c(c1)OCCO2 C1(C)(NC(CC2(OC)CCCC2)=O)CCN(C(c2cc[nH]n2)=O)CC1 Cc1cc(N(C)CCN(C)C(c2ccc(F)cc2Cl)=O)nc(-c2cccs2)n1 C(=O)(C(CCS(C)(=O)=O)c1cn(C2CCCNCC2)nn1)NCC(C(C)(C)C)OC c1(CNC(c2nc(CC)oc2C)=O)nnc2n1CCN(C(=O)C=CCOC)C2 c1(C(=O)NC2(C)CCN(C(C3COC(=O)N3)=O)C2)ccc2c(c1)CCC2=O CC1CC(C(=O)NC2CC(C)(CNC(=O)CCNC(c3ccoc3)=O)C2)CN1C c1(CNC2CC(=O)NC2c2ccccc2)cccc2ncccc12 C#Cc1ccc(C(=O)NC2CCN(C(c3cnn(C4CC4)c3Cl)=O)C(C)C2)cc1 N1(C(CSCC#C)=O)CC2CC(C1)CN(C(=O)CCCCCC(C)C)C2 N1(C(c2cnc(CCCC)s2)=O)CC2(C1)CN(C(c1ccnnc1)=O)CC2CO n1(CC(=O)NC2CC(NC(CN3C(C)CCC3C)=O)C2)cc(P(C)(C)=O)cn1 CC(C)C(C(=O)N1CCOC(CC(=O)N(CC(O)CO)C)C1)C(C)C c1(C(N(CCNC(C(CN(CC)CC)F)=O)C2CC2)=O)c(C)coc1CC(N)=O Cc1cc(C(=O)NCCCCNC(C2(C)CNC(=O)C2)=O)cc2ccoc12 C(=O)(CCCC(C(=O)NCC1CCOCC1)N(C)CCOC)OC C1(C(C)NC(=O)C2=CCC2)CCCN(C(C2CC(=O)N(c3nccs3)C2)=O)C1 C#CCCC(C(=O)NCC1CC(C)(O)C1)NC(C1CCS1(=O)=O)=O CCC(CC)CCC(=O)NCC1(C)CCCN1C(c1cncnc1)=O C1(CCC(=O)NC2(CNC(CC3(N(C)C)COC3)=O)CCC2)CCCC(=O)N1 Cc1cnc2c(C(N3CC(NC(=O)Cc4ccco4)CC(O)C3)=O)cnn2c1 c1(OC)ccnc(CN2CCOC(C(=O)NCc3cncn3C)C2)c1 C(=O)(C(CCOC)C1CCC1)N(CCn1cc(C2(COC)CCCC2)nn1)C C12(CNC(CN(C)C3CC3)=O)CC(C1)C(NC(=O)CCc1nnc(C(F)F)o1)CO2 N1(C(c2c(N)c(Cl)ccc2)=O)CC2(CCC(CNC(=O)CCc3cnn[nH]3)O2)C1 CCC(C)CC(C)C(=O)NCC1CN(C(=O)C=CCCC(C)C)CCC1C C=C(C)C1OCCCC1C(=O)NC(C)CN(C(=O)CCNC(=O)C(C)(C)C)C N1(C(c2c(C)ccnn2)=O)C2CC1CN(C(=O)C(N1CCOCC1)C)C2 Cc1c[nH]cc(C(=O)NC(C2CCN(C(=O)CCCOC(C)(C)C)C2)C)c1=O N1(C(CCCc2cc(C)no2)=O)CCC2OCCN(C(c3csnc3C)=O)C2C1 Cc1cccc(C)c1CN(CCNC(C1CN(C)C1)=O)C1CC1 N1(c2snc(C)n2)CC(C)(C)CC1CNC(=O)C1=NOC(C)C1 N1(C(c2ccn(C)n2)=O)CCC(C2CCN(C(c3snc(Cl)c3Cl)=O)CC2)C1 C1(C(=O)O)CC(c2ccccc2)CCN1C(C12COCC(C1)C2)=O c1(C(N2CC(NC(c3c(C)cccc3)=O)C(CC3CC3)C2)=O)ncnc(O)c1F N1(C(C2CCC(C(C)(C)C)O2)=O)CC2(CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)C1 c1(C(=O)NC2(C)CC(NC(C3C(C)(C)C3(C)C)=O)C2)cc(Cl)ccc1C(F)(F)F c1(C(N2CCC(N(C(=O)C(F)OC)CC)C2)=O)ccnc(C)c1C C(CC1=CCN(C(c2nncs2)=O)CC1)NC(c1ccc(Cl)cc1C(F)F)=O N1(C(c2cc(CC)on2)=O)CCOC2(C1)CN(C(C1(S(C)(=O)=O)CCCC1)=O)C2 C(CCCC(CO)NC(c1ccc(F)s1)=O)NC(COCCCCCC)=O CC(C(=O)N(C)CCOCCNC(=O)C(C)O)NC(c1cccs1)=O C(C(O)C(F)(F)c1ccccc1)N(C)C(c1ncn(C(C)(C)C)n1)=O C1(C(=O)NCC(C)(C2CCC2)NC(C(C=C=C)C)=O)CCOC2(CCOCC2)C1 N1(C(c2cnc(Cl)s2)=O)CCN(C(c2cc(O)ccc2F)=O)C(CC(F)(F)F)C1 Cc1cc2ncc(C(N3CCC(C(=O)Nc4ccc(CCO)cc4)C3)=O)cn2n1 C1(C(F)(F)F)(C(=O)NCC(=C2CN(C(CCCOC(C)C)=O)C2)F)CCOCC1 C(CC(C(=O)N1CC(C)(CN(C)C)C1)NC(C1CCCC1)=O)=CC C(=O)(C1=CCCN(Cc2cnc(Br)c(F)c2)C1)NC(CC=C)CO N1(C(CNC2CCN(C)CC2)=O)CCN(C(c2ccccc2)=O)CC1CCO Cc1nc(C(C)C)nc(O)c1C(N1CCC(CF)(NC(=O)C(C)O)C1)=O C1(CNC(C(C=CCCC)O)=O)CC(NC(c2ccc(CC)cc2)=O)CCO1 C1(CC(=O)NC(c2ccccc2OC)CC)CN(C(=O)C(C)n2cccn2)C(C)(C)C1 C1(C(N(CCO)CC)=O)CC(C)(C)CCN1C(=O)C(c1cncnc1)C C(=O)(C(O)CCNC(=O)CCOC)NCC(=O)OC(CC)C CC1=C(C)C(NCCc2cccc(OC(C)C#N)c2)CCC1 C1(CNC(c2cc3ccsc3s2)=O)CC2CN(C(=O)C=Cc3ccncc3)CC12 c1(CC)conc1C(=O)NCC1CCCC1NC(c1ccc(-c2ccco2)o1)=O N1(C(Cc2nc(C)sc2)=O)C2CCCC1CN(C(C1CCCC(F)(F)CC1)=O)C2 C1(C(N(C2CCCN(C(c3ncn(C)c3C)=O)C2)CC)=O)CCCCC(=O)N1 Cn1cc(C(=O)NC2CN(C(=O)C(=Cc3cccnc3)F)CC23CC3)ncc1=O c1(C(C(=O)NCC2(OC)CN(C(=O)CCC3CC3)C2)O)cccc(F)c1 S(=O)(=O)(c1cc(C(=O)NCC23CCC2CCN3C(=O)C(F)F)c(C)o1)NC c1(CNC(C2(COC)COC2)=O)cncc(C(=O)NCC(O)(CO)CO)c1 C(=O)(C1=COCCO1)NC1C(CNC(c2cnc(C(C)(C)C)nc2)=O)CCCC1 N1(CCNC(=O)COC2CCCOC2)CCC(C(=O)Nc2nccs2)CC1 C1(C)(CC(=O)NC2CCC(NC(C(CC)CC)=O)C2)CCS(=O)(=O)N1 N1(C(C2N(CC)CC2)=O)CCC(O)(CNC(=O)CC2CCCC(OCC)C2)CC1 c1(C(N(CC(CNC(Cc2ccc(CC)cc2)=O)O)C)=O)ccc2nn[nH]c2c1 c1(OC)cccc(OC)c1C(=O)NCC1CCC(NC(=O)C=C(Cl)Cl)CC1 O=C(CC1COc2ccccc21)NC1CN(C(c2ncc3ccccn23)=O)C1 c1(C(=O)NS(=O)(=O)Cc2ccccc2Cl)ccc(F)c(N)c1.CC12CN(C1)C2 C1(NC(CC2(CNC(c3cc(C)n(C)n3)=O)CC2)=O)CCn2cnnc2C1 C1(C(=O)NCC2CC3(CC(NC(CC(C)(F)F)=O)C3)C2)CCC2C(C1)C2(F)F N1(C(CC(CC)CC)=O)CCC2(NC(c3ccc(SC)o3)=O)CCCC12 N1(C(C(CC)SC)=O)CC(CC(=O)NC2C(C)(C)C2(C)C)C2(CC2)C1 C1(C(=O)NC2COCCC2O)CC2(CC2)CN1C(c1ccncc1O)=O C1(NC(=O)Cc2ccc(O)cc2)CC(C(=O)NC2CC3CCC2O3)C12CCC2 N1(C(c2c(OC)nc(-c3nc[nH]n3)s2)=O)CC2CCC1C2N C(=O)(CCC(C)(F)F)N1CC(C(C(=O)N(C)Cc2cncnc2)O)C1 C=CCC(C)(C)C(=O)NCCCC1CN(C(=O)CNC(=O)CN(C)C)CCO1 c1(C(N2CCN(c3ccc(C)c(C)c3)CC2)=O)cnc2c(Br)c(C)ccc2c1 C(N=c1[nH]c(=NCCCC2CC2)c2ccccc2[nH]1)c1c(C)c(F)c(F)cc1 C1(F)(c2cn(CCCC)nn2)CCN(C(=O)Cc2ccc(C)c(I)c2)CC1 C1(S(N)(=O)=O)(C(N(C2CCCCC2)CCNC(CN(CC)CC)=O)=O)CCC1 c1(CC)nn(C)c(Cl)c1CNC(N1CCOCC(CO)C1)=O N1(C(C2CN(C(c3cc(Br)cc4[nH]ncc34)=O)C2)=O)CCc2cccnc2C1 CCC(C)C(O)C(C)C(=O)NCC(C)(C)CCNC(c1cccc(O)c1F)=O Cc1nc(Cl)nc(N2CCC(N3CCN(C(C4CCCN4C)=O)CC3)CC2)c1Cl CC1CNCCN(C)C1=O.c1(C(=O)NCCO)coc(C(C)(C)C)n1 c12ccccc1CC(=O)N2.C1(C(N(CC(COC)(C)C)C)=O)CNC(=O)N1C c1(C(=O)NC2C(CNC(CCC3CCC(C(N)=O)O3)=O)C2)ccc2n[nH]cc2c1F c1(N(CC(C)NC(c2cc(CC)c(C)s2)=O)C)nc(C)nc(=N)[nH]1 c1(OC)csc(C(N2CCN(C(C3(CCF)CCC3)=O)CC2)=O)c1OC C1(CNC(C(C=C)OC)=O)CN(C(C2CCC(C)NC2=O)=O)CC(C)(C)O1 n1(CC)nc(C(=O)NC2(CNC(=O)C(O)CC3CCCC3)CCCCC2)cc1O C1(OC)CC2(C1)CC(C(=O)NC1COC(C3CC3)C1)C2.C12(CC1)CC(=O)N2 N1(C(c2cccc(SCC)c2)=O)CC(N(C)C(C23CC(OC)C2C3)=O)C2(CC2)C1 c1(C(=O)NCCCC2N(C(C(COC)C)=O)CCC2)cccc2c1nc(O)n2C N1(C(C=Cc2c(C)ccs2)=O)CCN(C(=O)C(n2nccc2C)C)CC1CCO N1(C(Cc2c(C)cccc2)=O)CCN(C(=O)C(CO)c2ccccc2)C(C#N)C1 Cc1cncc(C)c1C(=O)NC1CCCC1NC(=O)CC(F)(F)F C1(CN(C(C(=O)NCC#C)C)C)CCN(C(c2coc(C3CC3)n2)=O)C1 C=CC1(C(=O)NC2CN(C(=O)C(C)CC3CCCC3)CC2C)CCOCC1 CCCC(c1ccco1)NC(=O)CCN(C(=O)C(=O)NCC1CC1)C C=C1CC(C(=O)NCC2CN(C(N)=O)C2)(CNC(C2CC2(C)C)=O)C1 c1(C(N)=O)csc(C(=O)NCC2CC2NC(c2cn(-c3ccccc3)cn2)=O)c1 C1(NC(C(C)(C)CC2CC2)=O)CCOC12CCN(C(C1CC13CCC3)=O)CC2 C(=O)(CCN=c1[nH]ccs1)N1CCC(CCNC(c2cnc(CC)[nH]2)=O)C1 c1(-c2cccc(CNC(C3(O)CC3)C)c2)c(O)cccc1O N1(C(CCCC#C)=O)CC(CNC(c2nc(Br)c(C)s2)=O)C(F)(F)C1 C1(C)(C(=O)OC)CCCN(C(c2ccc(-c3ccc(C)c(OC)c3)nc2)=O)C1 CC1CN(C(c2cscc2C(F)(F)F)=O)CC1NC(=O)C(C)(C)c1cnn(C)c1 CC(CCC(F)(F)F)NC(=O)CCNC(C1CCCCC(=O)C1)=O Cc1c(C(=O)NCCCN(C(=O)C(C)N2CC(C)C2)CCO)[nH]c2c(C)cccc12 N1(C(C(C)S(N)(=O)=O)=O)CC(C)CN(C(C2CCCC(C)(C)C2)=O)CC1C N1(C(C)C)CCCC(CC(=O)NC2CCCC(NC(=O)Cc3ncc(Cl)s3)C2)C1 O=C(CC(F)(F)C(F)(F)F)NCC1C2CCC(C2)N1C(C1C2CC3C(C2=O)C13)=O C(CCOCCO)(C(=O)NCC)NC(CC1CCN(C(C(CSC)OC)=O)C1)=O c1(C(=O)NCC2(NC(C3C(C)=C3)=O)CC2)ccc(F)c(C)c1Cl Cc1n[nH]c(C)c1SCC(N1CC(CNC(=O)CSCC(C)C)C(C)C1)=O C(=O)(C(CN(C)C)C(C)C)NC1(C)CN(C=O)C1.C1(CC#C)(CC)CCOC1.C c1(C(N(C2CCCN(C(=O)CC(C)(C)C#N)C2)CC)=O)c(OC)cccc1Cl C(=O)(CC(C)C(F)F)N1C(CNC(C=CCN(CC)CC)=O)(COC)CCC1 CCCC(C)(CC)C(=O)N1CCCC(CC(=O)NCCCS(C)(=O)=O)CC1 C(=O)(CC(C)C(=O)OC)N1CCC(N(C(C2CC3(CC3)CN2C)=O)CC)C1 C1(N(C(=O)C(O)C2CCCC2)C)CN(C(c2ccccc2Cl)=O)CC1O C1(CNC(CCC(=O)NC)=O)N(C(=O)CN2CCCCS2(=O)=O)CCC1(C)C c1(OC)ccccc1C(C)C(=O)NCCCCCCNC(C1(C)CC(F)C1)=O n1(CC(=O)NCc2c(OC)ccc(OC)n2)c(C)cc(C)nc1=O.C1C(SC)CCO1 Cc1ccc(Cl)c(C(=O)N(C)CC2(NC(=O)C(c3ccc(Cl)cc3)CO)CC2)c1 N12CCCCC1Cc1cn(nn1)CC2=O.c1(C(=O)O)cc(C2CCCC2)no1 C1(CC)C(NC(=O)CCc2ncccn2)CCCN1C(c1ccc(Cl)cn1)=O CCC(O)(CC)CCNc1ncnc(NC2COCC2OCC)c1C CC(C)(C(=O)NC1CC(O)(CNC(c2cscn2)=O)C1)Oc1ccccc1 c1(C(N2CCN(C(C(CCC)CCC)=O)CC2C)=O)ccc2c(C#N)c[nH]c2c1 C1(C)(CNC(Cn2c(C)cnc2)=O)CCN(C(=O)CC2CCC(F)(F)C2)C1 CC1CCC(O)(C(=O)NCC2CCN2C(C2CCC(C)(C)C2)=O)CC1 C(N=c1cc(C)[nH]c(=NCC2COCC(C)O2)[nH]1)c1n(CC)c(O)nn1 c1(C(=O)NCC2(O)CN(C(C(C)N(C(C)=O)C)=O)C2)[nH]nc2ncc(Br)cc12 N1(C(CCCSC)=O)CCC(C(F)(F)F)C(NC(c2cc(C(N)=O)no2)=O)C1 C1(C(N(CC(C)NC(=O)C(F)(F)C2CC2)C)=O)CC(c2cc(F)ccc2F)=NO1 N1(C(C(CC)C)=O)CCN(C(c2cc(C)sc2C)=O)CC(C)(F)C1 c1(C(C)NC(C(C)OCCOC)=O)nc(C(=O)NCc2cncn2C2CC2)co1 c1(C2(CNC(=O)NCCC3C(C)OCC3)CC2)cccc(C(F)(F)F)c1 C(CC(=O)N=c1[nH][nH]c(-c2cccc([N+](=O)[O-])c2)c1C)(c1ccccc1SC)OC N1(CCCNC(CC(C)NC(N)=O)=O)Cc2ccccc2C1 C(=O)(C1=CCN(C(=O)C2=NOC(C)C2C)CC1)NC(C1CCOC1)C#C N1(C(CNC(CNC(C)=O)=O)=O)CCC(CO)(NC(c2n[nH]c(C)c2C)=O)C1 c1(N(C)Cc2ccoc2)cc(NC2CCCSC2)ncn1 c1(C(C2CCOCC2)CNC(c2cc(C)no2)=O)cnc(C(F)(F)F)nc1 N1(C(C)=O)CCCCC(CNC(=O)Cn2c(-c3ccccc3)c(C)sc2=O)C1 C1(C(N(CC=C)CC2CC2C)=O)CCN(C(=O)CCCSC(C)(C)C)CC1 c1(C(N(C(C)CN(C(=O)CCNC(=O)C=CCl)C)C)=O)cnn(C(F)(F)F)c1 C1(O)(CCNC(C2CN(C3CCC3)C2)=O)CCCN(C(c2cnnc(O)c2)=O)C1 CC(C)(CO)CCN=c1[nH]c(=NCc2cccc(N)n2)[nH]c2c1CCCC2 C1(NC(C(C)=C2CCC2)=O)CCC2(CC1)CCN(C(=O)C(C)NC(=O)C1CC1)C2 C1(C(N(CC(C)C)CC(=O)N(C)CCOCCN(C)C)=O)CC(N=[N+]=[N-])C1 C(=O)(C(CCSC)OC)NC(CC=C)CNC(c1nncn1C1CC1)=O O(NC(=O)C1=CC2(CCN(C(=O)C(C)SC(C)C)C2)C1)CC(C(C)C)O C(=O)(CC(CC)CC(F)(F)F)N1CC2C(CNC(C(CC)(C)CC)=O)(C2)C1 C1(CC=C)(NC(C2CC(C)(C)CO2)=O)CCN(C(=O)C(F)C2CCC2)CC1 Cc1cc(C(=O)NC2CCN(C(=O)COCC(C)(C)C)C2C)nc(C)c1 N1(C(C(C)=C2CCCC2)=O)CC2CCC1CN(C(=O)CN1CCCNS1(=O)=O)C2 c1(CNC(=O)NC2(C3CC3)CCCCC2)cc2cc(Br)ccc2[nH]1 c1(OC(COC)C)cncc(NC(C2CCCC2c2ccccc2)=O)c1 N1(C(C2C3CN(C(c4cccc5[nH]ccc45)=O)CC32)=O)CCC2(CC1)CC(F)C2 C1(C(=O)NC(C2N(C(CNC(=O)NC)=O)CCC2)C)CCn2ncnc2C1 CC(C)C(F)(CNC(=O)CN1CCN(C)CC1)C(=O)N1CCC1C1CCCC1 C1(O)(CNC(c2sc(C)c(O)n2)=O)CC2CCC(C1)N2C(=O)CC1CCC(=O)N1 CCCCC(CCC)NC(=O)C(O)C1CN(C(c2cc(C)co2)=O)C1 c1(C(=O)NC2CC(C)(NC(CC(CC)OC)=O)C2)cc(Cl)c2c(c1)OCCO2 c1(NC(C)C)ccc(F)cc1C(=O)NC1CC1CNC(=O)CCS(C)(=O)=O c1(CCOC)cccc(NC(C(C)CC2CCOCC2)c2nnnn2CC2CC2)c1 N1(C(C2(CC)CCCC2)=O)CC(C)(C)OCC1CNC(c1coc(SC)c1)=O C1(C)(C(=O)NCCN(C(=O)COCC2CCCCO2)CC)CCN(C)C1 C12(CNC(C(C3CCC3)OC)=O)CCCC1N(c1ncc(F)cn1)CCC2 C1(CNC(C(C)(C)c2cc[nH]n2)=O)CC2CC2N1C(C1CCC(F)CC1)=O c1(COC)nc(N)cc(N(CCCCCCO)C)n1.c1(C)ccn(C(F)F)n1 C(=O)(C(CC(C)C)C(C)C)NC1(CC)CCCN(C(c2cn(C)nn2)=O)C1 c1(OC)ccnc(C(=O)NCCC2CC(NC(C3(C)CC3(Cl)Cl)=O)C2)c1N C#CCCCCCCCC(=O)N1CC=C(CNC(=O)CP(C)(C)=O)CC1 N1(CCNC(C(C)NC(CC)=O)=O)CCN(C(C2CN(C(=O)CC)C2)=O)CC1 N1(C(CC2(C)CC2F)=O)CCC2(CCN(C(C3CCn4c(O)nnc4C3)=O)C2)C1 C1C(C(C)(C)C)N1.C1(C(=O)OCC)CCC1C(=O)OC(C)(C)C N1(CC(C)C)CCN(C(c2n[nH]c3c2CCCC3)=O)C(C)C1=O c1(C(N(C2CN(C(Cc3cn(CC)nc3)=O)CC2F)C)=O)cc(C)c(C)nn1 c1(C(N(C2CCOC2)CC)=O)ccn(CCNC(=O)CCC2CCCC2)c1 C(C)(C(=O)C(=O)C1CC1)NC(C)=O.C12CC(O)(C1)CNC(=O)CNCCC(=O)NC2 c1(C(=O)OC)cccc(S(=O)(=O)N2CCC(c3nnn(C)n3)CC2)c1Br CC12CN(C(C3CC4CCC3O4)=O)CC1(C)CN(CCC1=CCCCC1)C2 Cc1nc2cc(C(=O)NC3CCC3NC(c3c[nH]nc3C(C)C)=O)c(F)cc2[nH]1 Cn1cc2c(C(=O)NC3CNCC34CC4)cccc2n1 CC1(C)CC(C)(CNC(=O)CN(C2CCC2)C(C23CC(F)(C2)C3)=O)C1 N1(C(c2cc(C)[nH]c2C)=O)CCCC(CCNC(c2ocnc2C)=O)CC1 C(C(C(=O)NC(C)C(=O)N(C(C)C)C(C)C)NC(=O)C(F)=C(C)C)OC c1(N2CC3CN(C(c4sc(Br)cc4Br)=O)CC32)ncc2sccc2n1 c1(C(N2CC(COC)N(C(C3CC3C3CCC3)=O)CC2)=O)c[nH]c(C)c(Cl)c1=O N1(C(c2cnn(C)c2F)=O)CCC(NC(=O)Cc2ccc(F)cc2F)CC(O)C1 N1(C(C2CCN(CC)C2)=O)CC2(CC2)CC1CC(=O)NCC1CC2(CC2)CO1 N1(C(C(c2ccccn2)C)=O)CCC(F)(C(=O)NC2CCC2)C1 C(C(C(=O)NCCCNC(=O)C(C)C)n1cc(CC(C)(C)C(=O)O)nn1)OCC C(CC(O)C(=O)N1C(C(=O)NCCC2CCN(C)CC2)CCC1C)N(C)C c1(CNC)c(-c2sc(-c3nccn3CCc3n[nH]c(=N)s3)cc2C)cccc1F N1(C(c2c(CC)c[nH]c2)=O)CC(C)OC2(CCN(C(C3(C)CC3Br)=O)C2)C1 c1(CN2C(C(=O)Nc3cc(OC)ncn3)CC2)ccc(F)c(F)c1Br N1(C(C(CCCCC)O)=O)CC2(C=C(C(=O)N3CC(N(C)C)CC3(C)C)CO2)C1 CN1C(=O)CCC(NC(C2COCCN(C(c3cc4n(n3)CCO4)=O)C2)=O)C1=O C1(NC(CCCC)=O)CN(C(=O)C2=C(C)OCC2)CCC1c1ccccc1 Cc1nc(C(=O)NCc2ccsc2C(=O)NCC2CCSC2)cc(O)n1 c1(NC2CC(OC)C2)cc(C)c(S(=O)(=O)N2CCCN3CCCCC3C2)cn1 N1(C(C2CCS(=O)(=O)N2)=O)CCC(F)(F)C(CNC(C2(C3CC3)CCC2)=O)C1 C1(NC(=O)Cc2cnns2)COCCN(C(=O)CCc2cc(Cl)cs2)C1 N1(C(=O)CCc2ccc[nH]2)CCC2CCC(C1)N2C(=O)CCOC1CCOCC1 C(=O)(C(CC(F)F)NC(C1CC(F)(CF)C1)=O)NCC(CC)C(C)C N1(C(C(C)C#N)=O)CC(F)(F)CC1CNC(=O)COc1cn[nH]c1 C1(NC(CCC(C)OC)=O)COC2C(NC(=O)Cc3cc(C)cc(F)c3)COC12 Cc1ccc(C(=O)NC2CC(NC(C3CCCC3(F)F)=O)C2)c(C)c1 C=CCC(F)(F)C(=O)NCC(C1CCC1)NC(=O)CN(CC)CC c1(CNC(N2CCCC(c3ncc[nH]3)C2)=O)cc2c(s1)CCC2 C12(NC(CCCOCC)=O)CCN(C(c3conc3CC)=O)CC1C2 n1(CC(=O)NCC(CCNC(CCCOC)=O)O)c(O)nc2ccccc12 C=C(C)C(C)(C)C(=O)NCC1(NC(c2cnns2)=O)CCOC1 N1(C(Cc2cnc(C)[nH]2)=O)CC2(CC2)CC1CNC(C1(c2cccnc2)CC1)=O C1(NC(C(C)C(F)F)=O)CC(C2CCN(C(c3c[nH]nc3C(C)(C)C)=O)CC2)C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CCN(C(=O)C(C)Cn2ccc(C)n2)C(C)C1 c1(C(N2C(CNC(C(C)SC)=O)CCC2)=O)cc(F)ncc1Br CC1CC(C)CN(CCN2CC(c3nn[nH]n3)CCC2=O)C1 c1(NC(c2c(OCC)cc[nH]2)=O)ccc(-n2ccc(C(=O)OCC)n2)cc1 C1(NC(CN(CCC)C)=O)CCOCC1NC(=O)CCc1ccc(F)cc1 CCC(CC(F)(F)F)C(=O)NCC1(CN(C)C(c2cccc3nc[nH]c23)=O)CC1 C(CCCC(=O)NCC12COC(CNC(=O)CC(C)N(C)C)(C1)C2)N(C(C)=O)C N1(C(c2c(C)ccnc2F)=O)CC2(CCC(C(=O)NCc3ccnc(Cl)c3)O2)C1 N1(C(C(C(CC)C)N(C)C)=O)CCN(C(c2ncccc2O)=O)CCC1C CCC(CC(=O)NC1CCCC1NC(=O)C(C(C)C)OCC)OC N1(C(C(CSC)O)=O)CCCC2(CCN(C(=O)CC(C)=NOCC#N)C2)C1 C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cc(C)oc2C)=O)CC1 c1(C(=O)NCC2(F)CN(C(C(F)=CCC)=O)C2)ccc2sc(C)nc2c1 C1(CC=C)(C(=O)NC2CCC3CC23)CCN(C(c2ccsc2OC)=O)C1 n1(CC(=O)NCC(CNC(C2N(C(C)=O)CCOC2)=O)CO)cc(F)ccc1=O S(=O)(=O)(c1ccc(NCCn2cnc([N+](=O)[O-])c2)c(Cl)c1)NCC C1(C)(CNC(C(C)OCC2CC2)=O)CN(C(=O)C(C)C(C)(C)C)CCO1 C12(C(=O)NC(C(C)NC(C3CC=CCO3)=O)C)CC3CC(F)(C1)CC(F)(C3)C2 C(CCCCC(=O)N1CC(OC(=N)O)C1)NC(c1ccc(C)n1C)=O Cn1nc(C(=O)NCCC2(CNC(C3CC34CCC4)=O)CC2)c(Cl)c1Cl N1(C(CCC#C)=O)Cc2cccn2CC(C(=O)Nc2ccc(I)cc2F)C1 C=CCCCC(=O)NCCCOCCN(C(=O)CCCOC(=O)NCCOC)C N1(C(C2N(C(C34CC(C#N)(C3)C4)=O)CC3(CC3)C2)=O)CCC2(CC(F)C2)C1 N1(C(CSCC)=O)CCOCC1C(=O)NCc1cc(C)no1 C(=O)(CC1OCc2ncccc21)N1CCC(NC(c2c(C)ccnn2)=O)C1 N1(C(C(CC(=O)OC)(C)C)=O)CC2(C1)CN(C(C1C=CCCC1)=O)CCO2 C1(C(=O)NCCCNC(Cc2nc(=N)[nH][nH]2)=O)SC2=CCC1C2 c1(C(=O)NCC(=C2CN(C(c3cc(OCC)n[nH]3)=O)C2)F)cncc(C(F)F)c1 N1(C(C2C(NC(CCc3ccc(C)o3)=O)CCO2)=O)CC(C(N)=O)C2(CC2)C1 c1(NC(C(n2cc(CN3CCC(OC(F)F)CC3)nn2)C)=O)ccc(C#N)cn1 CCC(C(=O)N1CC(NC(c2ccc(OC)cc2Cl)=O)C(OC)C1)C(F)(F)F C(CCCCCNC(c1coc(-c2cccc(Cl)c2)n1)=O)NC(C(CSC)C)=O C1(CNC(C2N(CC)CC2)=O)CN(C(C2(CO)CC(F)(F)C2)=O)CC1OCC c1(C(=O)NCC2N(C(c3cnc(COC)s3)=O)CC2)ccc(NC(C)=O)c(F)c1 c1(-c2onc(CNC(CO)C3CCC3)n2)cccc(Br)c1 N1(C(c2[nH]c(=N)sc2)=O)CC2(C1)CN(C(=O)CCOCC1CCCO1)C2 C1(CN(C(CCc2onc(CC)n2)=O)Cc2ccccc2)C(=O)OCC1(C)C Cn1nnc2cc(C(=O)NC3CCN(C(C4C(F)(F)C45CC5)=O)CC3)cnc12 CCC(C#N)(CC)C(=O)N1C2CCC(C(=O)NCC(C)N(C)C)C1CC2 N1(C(C(CC)SC)=O)CC(NC(c2cc(Cl)c(Br)s2)=O)C(C)C1 c1(C(N(C2CCN(C(C3CCCC3O)=O)C2)CC)=O)sc2cncn2c1C c1(CNC(CCCOCCC)=O)nc2c(s1)CCN(C(c1cncnc1)=O)C2 C1(C(=O)NC2(C(O)CO)CCC2)CC1C1(C)COC1.C12(C(=O)OC)CN(C1)C2=O c1(N(C2CC2)CC2N(C(=O)OC(C)(C)C)CCC2)cc2sccc2s1 c1(N2CCC(OC)C(F)C2)nc2c(c(=NCC(C)(C)N3CCCCC3)[nH]1)COC2 c1(C(=O)NC(CN(C(=O)CC2COCCO2)C)(C)C)n[nH]c(C2CC2)n1 N1(C(C=CCOCCOC)=O)CCCCC1CC(=O)NCCCCC1CCCC1 N1(S(C)(=O)=O)CCS(=O)(=O)CC1C(=O)N(C)C.N12CCC13CCCC3CS2(=O)=O CC(CNC(=O)C=CCN(C(=O)C(C)n1cncn1)C)CO c1(C(=O)NC(C)(CNC(=O)C(O)C2CC2)CO)cc(F)ccc1F C1(C(N(CCC)CCC)=O)CCN(C(C2C=CCCC2)=O)C(C)(C)C1 CCCCCC(F)C(=O)NC1CC(CNC(=O)C(n2ccc(C)n2)C)CC1O N1(C(C(CSC)C)=O)CCCC(CCNC(=O)C(F)CC2CCOC2)CC1 c1(N2CCCN(C(C)C)CC2)ccc2cnc(C#N)cc2c1 C=CCC(C)(C(=O)NCC1CC(C)N(C(c2nn(C)c(Cl)c2Cl)=O)C1)N(C)C N1(C(CCOCC)=O)CC2(C1)SCCC2NC(=O)C=Cc1cccnc1 c1(CNC(c2cc(C)ns2)=O)ccc(CN(C(=O)CC2C(C)(C)C2(C)C)C)cc1 c1(CC)ccc(C(C)C(=O)NC2C=CC(CNC(c3ccccc3)=O)C2)cc1 c1(OCC)ccnc2sc(C(=O)NC(C3CN(C(=O)C(C)OC)CCO3)C)cc12 c1(SC)nc2ncnc(N3CCCC(C(C)NC(c4ccc(F)s4)=O)C3)c2s1 Cc1cc(N)cnc1C(=O)NCC1CCN(C(C2CCOC2C)=O)CC1O c1(CNC(C2N(C(C=C=C(C)C)=O)CCC2O)=O)ccc(C)cc1F CC1CCC2(CC2)N(C(c2ncn(C)n2)C(=O)NC2CCOC2)C1 N1(C(CCCCSC)=O)CCCC(NC(=O)Cc2ccc(F)cn2)C(F)C1 CCC1=NOC(C(=O)NC2CCC2NC(=O)CN2CC(=O)NC2=O)C1 CC1CC(CNC(c2ccc(C3CC3)s2)=O)CN1C(c1cc(O)nn1C)=O CC1(C)CC(CC(=O)NC2(CO)CCN(C(c3cccc(Cl)c3F)=O)CC2)CCO1 Cc1ncc(S(N)(=O)=O)cc1C(N1CC(N(C)C(c2ccc(CO)o2)=O)C1)=O c1(C(=O)NCCCCNC(CCCOC(C)C)=O)ccc2c(c1)COC2 c1(C(N2C(C)(C(N3CCCC(O)C3)=O)CC2)=O)c(Cl)cccc1Br c1(C(=O)NC2(CNC(C(c3cn(C)nc3C(F)(F)F)C)=O)CC2)cc[n+]([O-])cc1 CC(C)CC(C)CC(=O)NCC(C)(C1CCC1)NC(=O)CCc1cnn[nH]1 C1(NC(CCNC(N)=O)=O)CCCN(C(c2cc(Cl)ccc2N)=O)CC1 C#CCC(C)C(=O)N1CC(CNC(=O)Cc2ccccc2OC(F)F)C(O)C1 c1(C(N2CCC(CCCNC(C(COC)(C)OC)=O)CC2)=O)cn2ccsc2n1 N1(C(CCNS(CC)(=O)=O)=O)CC(C)(CNC(=O)Cc2nc[nH]n2)CC1(C)C c1(C(=O)NCCCC(N2CCC(CC)(CC)CC2)=O)cncc2[nH]ccc12 C12CCC3(CN(C3)C(=O)CC(=O)N1)O2.c1(C(=O)OC)cnc(OC)c(Br)c1 N1(C(c2cn(CCC)nc2C)=O)CCC2(C(N3CCCC(C)CC3)=O)CCCC12 C1(NC(c2c(OC)scc2)=O)CN(C(c2ccncc2)=O)C(C)(CO)C1 c1(C(=O)NC2CC3CN(C(CCOCCN(C)C)=O)CC32)ccnc2[nH]nnc12 N1(C(C(C)CC(F)F)=O)CCOC2(CCN(C(C3(Cl)CC3(C)C)=O)CC2)C1 CN1CCCC(CC(N2CCC(NC(C3CC(C(F)(F)F)C3)=O)CC2)=O)C1 C(C(C)(O)CC(=O)N1CCN(CCCNC(=O)CC2CCC=CCC2)CC1)OC C1(NC(C2(CC)CCCCCC2)c2nnnn2C2CCC2)CC(C)(C)OC1=O N1(CC(=O)NC(c2cn(C)nn2)C2CC2)CCOC2(CCN(C(=O)C3CC3)CC2)C1 C(=O)(C1=NOC2(CCN(S(=O)(=O)CCBr)C2)C1)Nc1c(C)ccc(O)c1 c1(C(N(CC(C)(C)CNC(=O)CC2=CCCC2)C)=O)cncc(P(C)(C)=O)c1 c1(OC)cc(C)c(Cl)cc1C(=O)NCC(C)(CC(C)C)NC(=O)C(C1CC1)OC N1(C(CNC(C(CC)C)=O)=O)CC2CCCC(C(=O)Nc3oncc3C)(C2)C1 N1(C(C)=O)CC(NC(=O)COc2ccsc2Cl)C(O)C1 N1CC2(CCN(C(=O)CCC3CC3(C)C)C2)C1.C(c1ccncc1)=C(C)C C#CC1(C23C(S)CC(CC2)C3)CCOCC1.c1(-n2ccnn2)ccccc1Cl N1(C(C(CC)N(C)C)=O)CCC(CCN(C(=O)C(=O)Cc2ccccc2)C)CC1 c1(C(N2C(C)CC(CNC(C(C(CC)C)OC)=O)C2)=O)cc(F)cc2nn[nH]c12 CC1OCCC1CN(C)C(C1CC(CCNC(=O)Cc2ccn(C)n2)C1)=O c1(C(=O)NCC(CC(C)C)NC(c2n(CC)nnc2C)=O)cnc(C)nc1C C(=O)(C(CC(C)C)C(C)C)N1C(c2onc(CN3C4CC(=C)C(C4)C3)n2)COCC1 CC(CC(=O)NCC1CCOC1C(=O)NC1CCCC(C)(C)C1)CC(C)(C)C c1(OC)cc(C)c(C(=O)NCC2CCCCC2NC(C2(O)CCOCC2)=O)cn1 N1(C(C(C)CO)=O)CC2CC3CC2C1C3C(=O)Nc1cc(=O)n(C)cn1 Cc1cc(C(=O)NCC2CCC(NC(c3ocnc3C)=O)CC2)cc([N+](=O)[O-])c1 c1(C(N(C2C3CN(C(CC(C=C)C)=O)CC32)C)=O)cccc(=S)n1O C1(C(N2CCC(N(C(c3ccn(CC)n3)=O)CCO)C2)=O)CC2(C1)CC(F)C2 C1(C(N(CCCCCC)CCNC(=O)CSC)=O)CCc2n[nH]cc2C1C Cc1cc(C(N2CC3=C(C2)CN(C(C2(CO)CCCO2)=O)C3)=O)cc(N)c1O N1(CC)CCCCC1C(=O)NCC1CCC1NC(=O)C(=Cc1c[nH]cn1)F N1(C(C(C)C2CC2)=O)CCN(c2ccc(C(=O)NCc3cccc(F)c3)cn2)CC1 N1(C(C2(OC(C)C)CCC2)=O)CC(NC(=O)C(F)=C2CCCC2)C2(CCC2)C1 C1(C(=O)NC(CC=C)CC=C)COCCN(C(=O)C(C)(C)C2(O)CCC2)C1 NS(=O)(=O)c1cc(C(=O)NC(C)(CNC(C2(F)CCCC2)=O)C2CC2)cs1 c1(CCC(N2CC(C)(NC(c3cncs3)=O)C2)=O)cccc(C#N)c1 N1(C(c2cncc(-n3ccnc3)n2)=O)CCC(F)C(NC(C2(CF)CCC2)=O)C1 c1(C(=O)NC2CC(NCc3ccc(C)nc3Cl)C2)cc(F)cc([N+](=O)[O-])c1Br Cc1ccccc1OCCCC(=O)NCC1(CNC(=O)CCC=CBr)CC1 C1(C)(C(=O)NC(CNC(C2(C(C)=O)CC2)=O)C2CC2)CCCC1 Cc1snc2sc(C(N3CC4COCC4(C(N4CCC(O)CC4C)=O)C3)=O)cc12 C1(NC(CCCCCOCC)=O)CCN(C(=O)C(C)S(C)(=O)=O)C12CCC2 C(CC(C)(C)C(=O)NCC1(C)CCN(C)C1)NC(C(C)n1ccnc1)=O N1(C(C2(C)CC2)=O)C2CCC1CC(C(=O)N)C2.c1(SCCOC)ccc(F)cc1 c1(CNC(C2(CC#C)CCCO2)=O)nc2c(s1)CN(C(c1csnn1)=O)CC2 CCC(=O)CCC(=O)NCC1CCCCC1C(=O)NCCSCCCO c1(C(=O)NCC(CCCC)NC(=O)C(C2CCCCC2)SC)c(C)cccc1Cl c1(CC(=O)OC(CNCC)C2CCC2)ccc(OC)c(F)c1.N12CCC(C1)C2=O C(=O)(C(F)C(C)(F)F)N1CCN(CC(=O)NC(CC=CC)CO)CC1 C(CC(N)=O)(C(=O)NC(C)CCC1CC1)NC(C1C(C(C)C)CCO1)=O C1(NC(CC2CCN(C)CC2)=O)CCCCCC1C(N1CCC1CO)=O C1(NC(C(F)OC)=O)CCN(C(=O)CNC(=O)CC2CCCC2)C12CCC2 N1(C(c2cn(CCC)nc2)=O)CCC(CNC(C2CCC2C(F)(F)F)=O)C12CC2 c1(-c2cccc(NCc3cnc(CCOC)s3)c2)cc(C)ccc1C C1(NC(C2CCSC2)=O)CCN(C(=O)Cc2cc3ccccc3o2)CCC1CO C(=O)(N=c1ccn(CC2CC(CSC)C2)[nH]1)C1C(C)(CNC(CC2CC(=C)C2)=O)C1 C=CCC(C)(C)C(=O)N(CC(C)(C)CNC(=O)CC(=O)NCC(F)(F)F)C CC1CN(C(c2cccnc2)=O)CC1(C)CNC(=O)CSCc1ccccc1Cl C1(N=[N+]=[N-])(C(=O)OCC)CCN(C(c2cnccc2Br)=O)C1 C#CC1(C(=O)NC(C)CC2CCOC2)CCN(C(c2ccc(C)cc2)=O)CC1 C1(NC(CCC#C)=O)C2CC3CN(C(C4CCC5(CCCC5)CC4)=O)C1C3C2 c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ncc(Br)cc1C N1(C(CCCOCC=C)=O)CCC(C2CCN(C(c3cnc(C)n3C)=O)C2)C1 c1(C(=O)NC2CC2C(F)(F)F)ncc(C)s1.C(=O)(C(N1CCCC1)C1CC1)NC N1(C(N2CC(O)(C(C)N)C2)=O)CCC12CCC(O)CC2.n1(CCCC)nnnc1C C1(CC(N2CCC(F)(CNC(=O)CCOCC(F)F)C2)=O)CN2CCN1CC2 C1(NC(CC(=O)NCC#C)=O)CCC(CN(C(=O)CC2CCC(=O)NC2)C)CC1 c1(NCCC(=O)NCCC2CC(NC(COC)=O)C2)ccc(F)cc1F N1(CC2CN(C(C(C)OCC(C)C)=O)C2)CCN(C(=O)Cc2cn[nH]c2)CC1 c1(CC(=O)NCC2(F)CN(C(C3OC4CCC3C4)=O)C2)cccc2c1OCCO2 c1(NC(=O)CCC(C)OCC2CC2)n[nH]c(=NCc2ccc(CO)c(F)c2)o1 C1(NC(CC2CCN(C)CC2)=O)CN(C(=O)CP(C)(C)=O)C2(CCCCCC2)C1 Cc1cc(-c2csc(C(F)(F)F)c2)c[nH]c1=NCc1ccc(Cl)c2[nH]ccc12 c1(C(N(C)CC2(O)CCNC2)=O)nnc(-c2cccc(Cl)c2)c2ccccc12 Cc1cc(CC(N2CC(CN(C(=O)C(c3cccc(F)c3)(C)C)C)C2)=O)n(C)n1 C1(CNC(CCN2CCN(CC)CC2)=O)CC2(CC2)CN1C(=O)CC1CC=CC1 C1(C(=O)NCC2(Cn3cc(-c4cccnn4)nn3)CC2)CC(F)(F)C12CCC2 c1(C(=O)NC2CN(C(C(CSC)C)=O)CC2O)ccc(S(=O)(=O)N2CCCC2)o1 C(=O)(C(C#N)=CC=NO)NC1C=CC(C(=O)NC(C(=O)OCCC)(C)C)C1 C(=O)(C(O)C(C)(O)CC)NCC(COCC)NC(COCCC)=O c1(C(N2CCC(COC)(NC(=O)CCF)CC2)=O)ccc2c(n1)OCC(=O)N2 C1(CNC(C(CC)C)=O)CC12CCN(C(c1sc(Cl)cc1Cl)=O)CC2 C(=O)N=c1nc2n([nH]1)CC(C(F)(F)F)CC2.C(CCC(C)C(=O)OC)N(CCO)CC C1(C(=O)NCCC(C)NC(CSC)=O)CC12CCOc1ccc(Cl)cc12 N1(C(c2c(CC)nc(C)[nH]2)=O)CC(C)CN(C(=O)COC2CCCC2)C(C)C1 N1(C(CCC(C)SC)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CCC1C C1(N(C(=O)CCn2ccnn2)CCO)CCCN(C(=O)C=Cc2ccco2)CC1 c1(CNC(C2C(CC)C2)=O)cccc(NC(=O)C(F)(F)c2ccccc2)c1 Cc1cc(C(=O)NC2CN(C(c3cc4ncsc4[nH]3)=O)CC2F)ccc1Br C(CC(C(=O)NCC(C)(C)CSC)NC(c1cncnc1)=O)OCC C(=O)(C1=NOC2(CCC2)C1)N1CC(N(C)C(c2ccn(C)c2)=O)C(C)(C)C1 CCCCC(CC(=O)NC1(C(N2C(C(=O)NC)CCC2)=O)CCCCC1)NC(C)=O C1(NC(=O)CCF)CCN(C(=O)CC2(N3CCCCC3)CCCCC2)CC1F N1(C(CCOCCOC)=O)CCCC(NC(=O)C(c2ccc(OC)cc2)O)C1C CC(C)C1=NOC(C)(C(=O)NCCCCNC(=O)CCc2ccn(C)c2)C1 c1(-c2cn(C3CN(C(C(C)NS(C)(=O)=O)=O)C3)nn2)cc(F)ccc1F C1(NC(=O)Cn2cncn2)CN(C(C23CCCC(CO2)C3)=O)CC12CC2 c1(C(N2C(CNC(c3cnn(CC)n3)=O)CC2)=O)cc(OC)ccn1 C#CCC(C(=O)NCCC(C)NC(C1CC(N(C)C)C1)=O)C1CC1 C1(NC(CC2CN(C(=O)Nc3c(-c4n(C)ncc4)[nH]nn3)C2)=O)NC(=O)NC1=O S(=O)(=O)(CC(=O)NCC(C(C)(C)C)NC(=O)CC1CCCCN1C)NC C(C(F)C(=O)NCCn1cnnc1)C1CN(C(C2(CC)CC(=O)C2)=O)C1 N1(C(C(CCC)C)=O)CCC2(CNC(c3oc(CC(C)C)nc3C)=O)CCCC12 C12(C(N3CC(C)NC(=O)C3)=O)COCC1CN(C(C1C3CNCC13)=O)C2 n1(C(C)C(=O)NCC2CCN(C(C34CC(O)C3C4)=O)C2)c(=O)oc2ccccc12 Cc1ccc(C(=O)NC2CCN(C(=O)Cc3cnoc3)C(C)C2)c(O)n1 c1(C(C)C)nnc2n1CCN(Cc1cccc(C3(O)CCCC(C)(C)C3)c1)C2C CC(C(C)C(=O)NCC1CCC(C)CC1)NC(=O)C=Cc1cncn1C c1(OC)ccccc1COCCNC(=O)N(C)CC1CCCSC1 C(c1ccc(CC)cc1)=CCN(C1(CNC(CC(=O)OCC)=O)CC1)C c1(C(N2CC3CCC(O)C3C2)C(=O)NCCCSC)cc(F)c(F)cc1F CC(CO)C(C)NC(=O)CCN(C(=O)CSCC(F)F)C c1(-c2cn(CCCNC(=O)CC(c3cccnc3)C3CC3)nn2)ncccc1CO C1(NC(c2ccc(C)cc2)=O)CCN(C(c2nc(O)[nH]c(=O)n2)=O)CC1C N1(C(C(N(CC)OC)=O)=O)CCCC2CN(C(=O)Cc3nc[nH]n3)CCC12 c1(NC(c2nc(-c3c(OC4CC4)ccc(C)c3)sc2)=O)cccc(F)c1[N+](=O)[O-] C1(C(N(CCNC(=O)C(C)CN2CCCCC2)CC)=O)CCCC(=O)C1 Cc1ccn(CC(C)C(=O)NCC2CC2NC(c2cnc(C(N)=O)s2)=O)n1 N1(C(C(CCC)NC(C)=O)=O)CCC(C)(C)C1CNC(=O)CNC(=O)CC C=C1CCN(C(c2cccc(C#N)c2)=O)C(C(=O)NCc2ccccc2OC)C1 c1(C(=O)NCCC2CC(NC(c3c(C)cn(C)c3)=O)C2)cc2c(s1)COCC2 c1(C(N2CCCC(NC(C=C(CC)C)=O)CC2)=O)ccc2snnc2c1 CCC(C)(CCC(C)C)C(=O)NC1CC(NCc2cnn(C)c2Cl)C1 CCCCC(C(=O)NCCCN1CCCC1C)NC(c1ccc(=N)[nH]n1)=O C(=O)(CCCC(F)(F)F)N1CC2(C(NC(C(CC)Sc3nc(=N)[nH][nH]3)=O)CC2)C1 c1(CNC(=O)Nc2c(C)n(CCC(C)C)nc2)cccc2c1OCCO2 CC1(C2CC2)CCN(C(=O)C(Cn2cncn2)NC(c2ccoc2)=O)C1 Cc1cc(Cl)cc(C)c1C(N1CCOC(CNC(=O)Cn2c(C)csc2=O)C1)=O c1(CC)nncn1NC(=O)C1CCN1C(=O)CC(C)(C)O O=C(CCCN1CCOCC1)NCC(C1CCC1)NC(=O)CCCC1CCCC1 C1(C(C)C)CCC(C(=O)NCC2(C#N)CCC2)N1C(=O)C=CCN1CCC1 c1(CC)c(C(=O)NCC(C)NC(=O)C(C)c2ccsn2)cnn1C(C)(C)C C1(NC(c2ncccc2F)=O)CS(=O)(=O)CC1N=c1nc(C2CCCCC2)[nH]s1 N1(C(C(CC)N2CCCC2=O)=O)CC2CCC2(CNC(=O)C(=O)C(C)(C)C)C1 c1(C(N2C(CCNC(C3(C)CN(C)C3)=O)CCC2)=O)cncc(C#N)c1 C1(C)(CNC(C2(SC)CC2)=O)CCC(NC(=O)CCc2cccs2)C1 N1(CC(N2CC(N(C(=O)CC3CCC(O)C3)C)C2)=O)CC2CCC1C2 N1(Cc2onc(C(C)C)n2)CCN(C(C)(C)CNC(=O)C(=O)N(C)C)CC1 Cc1nc(Cl)[nH]c(=NCCCC(c2ccccc2)NC(=O)CCC2CC2)c1F c1(N(C(C)CC2CC2)C)nc2c(c(=NCC(C)(C)OCC(C)(C)C)[nH]1)COCC2 C1(NC(c2n[nH]c(CC)c2Cl)=O)CCCCN(C(c2cc(N)ccc2F)=O)C1 S(=O)(=O)(c1ccc2[nH]c(=NCc3csnc3C)sc2c1)N1CC(CC)N(C)CC1 c1(C(N(CCC(=O)NCC2CC(OC)C2)CCCO)=O)c[nH]nc1C(F)F c1(NC(C2CC(O)CCN2C(C2CC(O)C2)=O)=O)cc(Br)ccc1OCC1CC1 C(=O)(C1CCCc2nncn21)N1CCCC(NC(c2cc(C)c(C)[nH]2)=O)C1 C1(N(C(CC(CCC)C)=O)C)CCC2CN(C(=O)CN(C)C(N)=O)CC12 N1(C(C(c2ccc(F)cc2)C)=O)CCC(CF)(NC(c2cc(Cl)ns2)=O)C1 N1(C(COC(CC)C)=O)CC2(C1)CN(C(c1sc3cncn3c1C)=O)CCO2 C(C(=O)N(OC)C1CCCC1)n1cc(-c2c(CC)n[nH]c2)nn1 N1(C(c2cnc(CC)[nH]2)=O)CC2CCCC(CNC(=O)CC3CC3)C2C1 c1(OC)ccc2c(c1)CCC(NC(c1cc(Cl)ccn1)=O)C2=O C(=O)(C(O)CCCNC(C12CCC(CC1F)C2)=O)N(CC)CC1CCC1 C1(=O)CCC(C)(C)N1.c1(C(NOCC(=O)OCC)=O)cnc(C)c(C)c1 N1(C(C2=NOC(C)C2)=O)CC2CCC1CN2C(=O)COCC1CCOCC1 C#CCC(CC(=O)N1CCC(O)(CC)C1)NC(c1sccc1C#N)=O C(=O)(C(C)C(C)(C)C)N1CC(OC)C(NC(=O)CCn2cnccc2=O)C1 N1(C(C(=O)Nc2ccc(C)cc2Cl)C)CCS(=O)(=O)C(CCNC(=O)COC)C1 c1(NC(C(C)OC(c2cccc(C3CCC3)c2)=O)=O)cc(C(F)(F)F)ccc1F C1(C)(C(=O)Nc2cnc(C)nc2)CCCN(C(C2CCCCO2)=O)C1 c1(C(=O)NCC2CCN2C(c2cnn3ncccc23)=O)cc2c(nn1)OCCS2 c1(CC(=O)N(CCOC)CCNC(=O)CC2CS(=O)(=O)C2)cnc(Cl)cc1C Cc1cc(C(N2CCC(NC(=O)CCc3ccn(C)n3)CC2C)=O)cc(C)c1Cl C1(C)(NC(C(CCC)O)=O)CCCN(CC(=O)Nc2ccccc2C)C1 CCC(CC)C(C)C(=O)N1CC(N=[N+]=[N-])CC1C(N1CC2(CCC(=O)N2)C1)=O CC(C)(C#N)C(=O)NCc1ccccc1CNC(=O)CNc1nncs1 c1(NC(C(C)N(CCC)C(c2ccc(C(C)=O)[nH]2)=O)=O)cccc(CSC)c1 C1(CNC(C=C(C)C(F)F)=O)CC12CCN(C(=O)CN(C1CC1(F)F)C)CC2 c1(C(N(C(C)CNC(C2CCC(C)CC2)=O)CC)=O)nc(C(C)C)ncc1Cl N1(C(CC(C=C)CC)=O)CCCCC12CC(NC(=O)COC1CCC1)C2 C1(C(N(C)Cc2c(C)nsc2)=O)CC(NC(c2cncs2)=O)CCO1 C(CC(=O)NCC1CCCSC1)(C(C)(C)C)NC(c1c(C)nc(C)o1)=O Cc1ccc(C=CC(=O)NC2CCC(CCNC(c3ccc(C)nc3)=O)C2)nc1 N1(C(CN(C(C)C)CC)=O)CCCC(CNC(C2CCN(C(=O)NC)C2)=O)C1 C1(O)(CC)CN(C(C2CC(C)(C)C2)=O)C1 c1(-c2cn(CCCC(=O)NC(C)CC3CC=CCC3)nn2)nccnc1C(=O)O C1(C(N(C2CCN(C(=O)CC3CCCOC3)C2)CCO)=O)COC2CC1C2 CCCC(C(=O)N1CC(C(C(=O)NCC2CC2C2CCC2)OC)C1)C(C)C C(=O)(CCC(C)NC(=O)C=Cc1ccnn1C)N(CCCCC)C C1(NC(C=Cc2n(C)cnc2)=O)CCCC12CN(C(C1NC(=O)OC1C)=O)C2 c1(OC)cc(C(=O)NCCC(C)NC(=O)C=C(C)c2cnn(C)c2)cc(Cl)c1 C#Cc1ccc(C(=O)NCCC(C)NC(=O)C(c2ccc(F)cc2)(F)F)c(F)c1 c1(C(=O)NC(C2CCOC2)C#C)cc(COC)on1.C12(CC1)C(=O)NCC2 C1(C(=O)NC2CN(C(C3(C4CCOCC4)CC3)=O)C3CC23)CN2CCCN1CC2 C1(C(=O)NC(C)(C)CCNC(c2ccccc2CC#N)=O)CCc2ccnn2C1 C1(C(C)C)CN(C(c2ccc(O)nn2)=O)CCN1C(=O)Cc1nc[nH]n1 O=S(=O)(c1ccccc1-c1ccccc1)N1Cc2ccc(CN=c3cc(F)nc[nH]3)cc2C1 CS(=O)(=O)CCc1cn(C(c2nnnn2NCC2CCCO2)c2cccs2)nn1 c1(-c2cn(CC3CCC(NC(C4CC(=C)C4)=O)C3)nn2)ccccc1OC Cc1nscc1C(=O)NC(Cc1cn[nH]c1)C(=O)NCC1(CF)CC1 Cc1cc(O)c(F)cc1NC(C1(CNC(=O)C(C)CO)CCOCC1)=O c1(C(=O)NC(C(C)NC(C(C)Cc2cnc[nH]2)=O)(C)C)cc(Cl)c(F)cc1O c1(CC)cc(Br)ccc1NC(C1CN(S(=O)(=O)CC(C)C)CCN1)=O C(C(C)C(C)C(=O)NC1(CCC(=O)N(CCO)CCO)CCC1)OC C12(C(=O)NCCN(C(=O)COCc3nccn3C)C(C)C)CSCC1C2(F)F c1(C(C(=O)NCCCCN(CCCNC(C2SCCS2)=O)C)F)ccccc1 c1(C(N2CCC(c3cn(Cc4cnn[nH]4)nn3)CC2)=O)ncccc1Br C1(C(=O)NC(C2CCN(C(C3(C#N)CCOCC3)=O)CC2)C)CCC(=O)N(C)C1 N1(C(=O)Nc2c(SCC)nccc2)CC2(NC(=O)C(F)(F)F)CCC1CC2 c1(OC)ncnc(NC2CS(=O)(=O)CC2NC(c2ncccc2F)=O)c1C N1(C(C(=O)N(CC(C)OC(C)(C)C)C)=O)CC2CCCC12 Cc1nc(Cl)sc1C(N1CCC(CC(=O)NC(c2cncnc2)C)CC1)=O c1(C(=O)NCC(=O)NCC(=O)NC(C)C)ccoc1 N1(C(c2sc(C(=O)OC)c(C)c2)=O)CC(CNC(c2nccn2C)=O)CC(C)C1 N1(C(C(C(C)C)OC)=O)CC(C(=O)NC2CSC2)C(C)(C)C1 C1(CNC(CCc2cccc(OC)c2)=O)CCN(C(=O)CC(C)O)C12CCC2 N1(C(C#CC2(CC)CC2)=O)CCC(C2CC2)C1CNC(=O)C=C(Cl)Cl c1(CC)ncc(C(N2CCC(N(C)C(c3ccn(C4CCC4)n3)=O)CC2)=O)cn1 N1(C(C(CNC(C)=O)(C)C)=O)C2CCC1CC(N(C(=O)CN1CCCC1=O)C)C2 C(=O)(C(C)CC(C)(C)C)N1C(C(=O)NCC(CC(=O)NC)C)(COC)C=CC1 C12(C(N(CCCC=C)CC)=O)COCC1CN(C(c1ccc(C(C)C)cc1)=O)C2 C1(C(N2CCC(C)CC2)=O)C(CC)CCCN1C(=O)C(=O)NOC CC1CCC(CO)CN1C(=O)NCc1csc(C(=O)O)n1 N1(C(c2c(C)ccc(C)c2)=O)CCCC12CN(Cc1cc(F)cc(I)c1)C2 C(C1CN(C(=O)C(C)=C2CCCC2)CC1C(N1CCCC(F)CC1)=O)=CC C1(CNC(CC2(OC)CCC2)=O)C2CN(C(c3ccn(CCO)c3C)=O)CC12 CCS(=O)(=O)c1ccccc1N1CCN(C(C2CCCNS2(=O)=O)=O)CC1 N1(C(C(C)n2ccnn2)=O)CCC2(CC1)CC2CNC(c1cocc1C(N)=O)=O CCCC(CC)CCC(=O)N1CC(CCCCNC(=O)CC(C)C2CCCC2)C1 C1(CC(=O)NCC2(Nc3nc(C)nc(O)c3)CC2)COc2ccccc2O1 Cc1cc(C(=O)NCC2COC(C)(C)CN2C(=O)CN(C)C)c(C)cc1Br C12(CNC(C3C(C)(C)C3)=O)CC(CCO1)N(C(C1CC3C=CC1O3)=O)C2 C1(O)(CC(=O)NC2CN(C(C3(C4CCCCO4)CC3)=O)CC2F)CCOCC1 C12(C(N3CC(C)(NC(c4n(C(CC)C)ncc4)=O)C3)=O)CCC(CC1=O)C2 C1(NC2CCN(C(C3N(CC)CCOC3)=O)C2)CC(C(=O)OC)=NO1 C1(N(C)C(C2CCCC2(C)C)=O)CCCCN(C(=O)NCc2ccoc2)C1 c1(C(=O)NC2C=CCC(C(=O)NC(CCCC=C)C)C2)c(C#N)ncn1C C(=O)(C(C(C)(C)C)N1CCCC1=O)N(C)Cc1cn(C2CCOCC2)nn1 c1(C2(NCC3(C)N(C)CC(OC)C3)CCOC2)c(F)cc(Br)cc1F C1(C(N2CC3CC2CN3C2CCC2)C(=O)NCC)CC12CCC(F)(F)CC2 C1(O)(CNC(CSCC(N)=O)=O)CCCN(C(c2cncnc2C2CC2)=O)C1 C1(C(=O)NC2CC(C)(NC(c3[nH]cc(C)c3)=O)C2)OC2CCC1CC2 c1(CN(C(C(=O)NC(C2CCOC2)C)=O)C)cnc(C(F)(F)F)s1 c1(OC)ncc(C(=O)N(C2CCCN(C(C3CCCS3(=O)=O)=O)C2)C)c(C)n1 c1(NC2CCN(C(Cc3c(C)ocn3)=O)C(C)C2)ncnc2cc(C3CC3)nn12 c1(NC(CCC2(NC(C3CC(OC)C3)=O)CCCC2)=O)ccccc1N=[N+]=[N-] Cn1nc(C(=O)NCC2CC3(CC3)CN2C(=O)CC2(C)CC2(Cl)Cl)c2c1CCC2 C(=O)(C(C)(C)CNC(C1CCC(NC(C2CCCN2C)=O)C1)=O)NC C12CCCC(C1)NC2=O.c1(CN(C(=O)CC2C=CCC2)C)nn[nH]c1C1CC1 c1(COC)ccc(C(=O)NCC2(F)CN(C(c3ncoc3C3CC3)=O)C2)s1 C1(NC(C2(CC)CCNC2=O)=O)CCC2CC1CN2C(=O)Cn1cncn1 C1(C(=O)NCCOCCN(C(=O)CCC2OCCO2)C)CCCC(C(F)(F)F)O1 c1(C(=O)NCC2CCN(Cc3cc(Br)cs3)C2)cnn2cccc(F)c12 C12(NC(c3c(C)n[nH]c3)=O)CCCN(C(c3c(Cl)csc3Cl)=O)CC1C2 c1(SC)cc(C(N2CCCC2CCC(=O)NCC(C)(C)C2CCCO2)=O)co1 N1(C(c2c(C)nc(CCC)s2)=O)CCC(C)C(NC(=O)CC2(O)CCOC2)C1C C(=O)(C1=CS(=O)CCC1)NCCCCNC(CC(C(C)C)C)=O C1(N(C(=O)CC(C2CC2)C2CC2)C)CN(C(=O)CC2CC(F)(F)C2)CC1F N=c1[nH]c(CC(=O)NCC2CCC(NC(=O)C(=O)Nc3ncc[nH]3)C2)cs1 C(C(C)(C)C(=O)N1CC(CCNC(C2C3CCC2CC3)=O)C(C)C1)SC CC(CCCCNC(=O)CC1CC1(Cl)Cl)NC(C1CC(F)(CO)C1)=O c1(C(=O)NC2C(NC(CCc3nnc(C(C)C)o3)=O)CCCC2)n[nH]cc1[N+](=O)[O-] c1(C(=O)NC2CC(C)(CNC(c3nscc3Br)=O)C2)n[nH]c2c1COC2 CCCC(C)(CCC)C(=O)NCC1=CCN(C(c2ccccn2)=O)CC1 CC1(C)CCC(C(=O)NC2CC(CNC(c3cnn(CC(F)(F)F)c3)=O)C2)C1 CCCC(C(=O)NCCCNC(=O)Cc1cccc(OCC2CC2)c1)N(C)C c1(-c2cccc(CN3CCC(NC(CCSC)=O)CC3)c2)nc2ccccc2s1 C1(NC(C(C)CN(C)C)=O)CCN(CCNC(C2C3CCC2CC3)=O)CC1 c1(CCC(=O)NCCC2CCC(CNC(C(C)(C)C)=O)C2)ccnc(Cl)c1 C1(OC)CC(NC(=O)CCc2ccccc2)CN(C(C2CC23CCC3)=O)C1 Cc1cccn2nc(C(=O)NC3CCN(C(c4cncnc4)=O)C(C)C3)cc12 N1(C(c2cccc(C=CC(F)(F)F)c2)=O)CCC2CCC(F)(F)CC2C1 N1(C(=O)Nc2c(OCC#C)cccc2)CCc2[nH]c3ccc(F)cc3c2C1 c1(C(=O)Nc2cncc(C)n2)cnc2ccc(-c3ccc(F)c(C#N)c3F)cn12 c1(-c2nc(C(C)C3CC3)nn2C2CCOC2(C)C)ccc(S(=O)(=O)C(F)(F)F)cc1 N1(C(C2(c3c(C)c[nH]n3)CC2)=O)CCC(CNC(=O)C(F)CC2CC2)C1(C)C C1(OC)CN2CCCC2(C(=O)NCC(C)(C)CNC(=O)Cc2cnoc2)C1 N1(C(C2(CNC(c3cc(C)oc3C)=O)CCCC2)=O)CCC(C)(C2CC2)C1 N1(C(CCSCCCC)=O)C(CNC(=O)CCc2csnn2)CC2CC12 CC(CCC(C)(C)C)C(=O)NC1CCCC(CC(=O)Nc2cc(O)ccc2F)C1 CC(C)C(O)CC(=O)N1CC(C)(C)CC1CC(=O)NCc1nn(C)c(=O)n1C c1(N2C(C)CN(C(=O)CC(=O)N(CC(F)(F)F)C)CC2)nc2ccc(F)cc2o1 CCCC(C(O)C(=O)NC(C)(CC=C)CC=C)NC(=O)C(=O)CC(C)C C1(CCNC(C#C)=O)C(C)CCCN1C(=O)C=C(C)Cl c1(C(N2C(CC)CC(C)C2)C(=O)NCCCF)cc(OC)ccc1Cl c1(CC(N2C(CNC(CSCC)=O)C(C)(C)CCC2)=O)cnc2n1CCCC2C C1(CNC(C(C2CC2)NC(C2C3(CC3)C23CC3)=O)=O)CCCC2(CC2)C1 c1(NC(C(C)Sc2c(C)n[nH]c2)=O)cc(C(=O)O)cc(C(=O)OC(C)C)c1 C1(C)(OC)CC(NC(=O)C(CNC(c2cc(C)nc(O)c2)=O)OC)C1(C)C C(=O)(C1=CCN(C(=O)Cc2cc[nH]n2)C1)NC1CC(CCC(=O)OC)C1 C1(CC(N2C(CC)CC(O)C2)=O)CCN(C(=O)C2=COCC2)C1(C)C C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCNC(c1cncc(C=C)c1)=O)C C=C(CNC(c1ccccc1)=O)CCNC(=O)CCNC(=O)CC12COC(C1)C2 c1(NC(C2(OC)CCSC2)=O)cc(NC(c2ccc[n+]([O-])c2)=O)ccc1C C1(CC(=O)NC(C)CN(C)C(C2CCN(C3CCCCC3)C2)=O)C(C)(C)C1(C)C CC1CC(C)CCN(C(C2CC2CNC(C2CC3(CCO2)CC3)=O)=O)C1 c1(C(=O)Nc2c(C(=O)OC)c(C)cs2)ccc(-c2ccc(F)cc2)nc1C c1(CC)c[nH]cc1C(=O)NCC1OCCC1C(=O)NCc1ccsc1C C1(CNC(COCCCCC)=O)N(C(=O)CC(C)OC)CCCC1(C)C CC(C(=O)N1CC2CC(NC(C3CCCCCC3)=O)C1C2)C(C)(F)F CCCCC(F)C(=O)NC(Cc1cc[nH]n1)C(=O)N1CC(C(C)C)(OC)C1 C1(O)(CNC(c2c(CC)c[nH]n2)=O)CCCN(C(c2cc(OC)ccn2)=O)CC1 c1(OC(C(=O)NCC(CNC(C(C)CC2CCC2)=O)(C)C)C)ccccc1F n1(C2CN(C(C(CC)CC)=O)C2)ccc(=NC(=O)CCNc2nccs2)[nH]1 Cc1cccc(CCN(C2CCOC(c3ccncc3)C2)C)c1 C1(CNC(C(CSC)OC)=O)CC(C)(C)CN1C(=O)Cc1cncc(C)c1 C=CCCC(C)N=c1nc2c(cnn2C(C)C)c(NC(C2(COC)CC2)C)[nH]1 N1(C(C2CC(C)SCC2)=O)CC2CC(C1)C2NC(c1c[nH]nc1C1CCOC1)=O S(=O)(=O)(c1ccccc1Cl)NC1C(NC(c2c(OC)cccn2)=O)C2CCC1C2 c1(C(=O)NCC2CCC(NC(c3c(SC)snn3)=O)C2)nn(C)cc1[N+](=O)[O-] C(=O)(C1CCCc2c[nH]nc21)N(C1CCN(C(=O)CSCCOC)CC1)CCC CC1=C(C(=O)N2CC3CC3C2CNC(C2C3CCCOC23)=O)CCC1 C=CC1(O)CCN(C(=O)CC2CCCC(NC(=O)CCCCOCC)C2)C1 CC1CCC(NC(C23CC(C2)C3)=O)CN1C(C1CCC(C(N)=O)C1)=O c1(C(N2CC(CCCCNC(c3cnc(CC)s3)=O)C2)=O)nc(O)nc(O)c1N c1(NC)ccccc1CNC(C1(CC)CCCN1C(=O)C(O)C1CC1)=O O=C1CC(C(=O)NC(C2CC2)C2CC2)N(C(C2CC=CC2)=O)C1 C1(c2cn(CCCCC=C)nn2)CCCN(C(c2ccnnc2O)=O)C1 N1(C(C(C)OCC=C)=O)C2CC1CN(Cc1ccc(CC)cc1)C2 C1(N(c2ccccn2)CC(C)O)CCN(C(=O)NCCc2cccs2)CC1 c1(C(N2CC(C)(CNC(CSCC)=O)OCC2)=O)cc2nccnc2cc1F C#CCCCCCC(=O)NC1CCC(C)(CNC(=O)CCc2cc(OC)no2)C1 C1(C(=O)NCC(C)NC(C(CCC)C)=O)CC2(C1)CC(C)(C)C2 N1(c2ncc(C)cn2)CCC2(NC(=O)CCC3CCCCCC3)CCCC12 C=C=CCCC(=O)NC(CNC(=O)CCC(C)c1ccccc1)CO c1(C(=O)N)cc(Cl)c(C)cc1[N+](=O)[O-].N1(C(CO)=O)CC(CO)(OC(CC)=O)C1 CC(C)(C)[Si](C)(C)OCc1cccc(CCC(=O)NC2CCCCC2)c1 C(=O)(C1=C(C#N)CCC1)N1CCCC(C(C)C(=O)N(C2CCCC2)C)C1 C1(NC(c2ccc(F)s2)=O)CN(C(c2cc3c(o2)CCCC3)=O)CC2CCCC12 Cc1cc(F)ccc1C(N1CC(C)(C)CC1CNC(=O)CCc1ccnn1C)=O C(C)(c1cccs1)=CC(=O)NCCN(C(=O)C(CN(C)C)N(C)C)CC.C(C)(C)C C1(CC(=O)N(C)CC2CCCC2NC(C2CCSC2)=O)CCc2ccccc2C1 N1(C(CCCC#CC)=O)CCC2(C1)CN(C(C13CC(C1)C3)=O)CC(C)O2 Cc1n[nH]c(C)c1CC(N1CCCC(C(C)C(=O)N(C)CCO)C1)=O Cc1cc(=NC(CN(C)C)CCO)nc(N2CCOCC2)[nH]1 Cc1cnnc(O)c1C(=O)NCCC1CC(F)(F)CN1C(c1ccnnc1O)=O CCC(CC(=O)N1CCC=C(C(=O)NCc2ncoc2C(C)C)C1)C(F)F N1(C(C2C(C)C2)=O)CCN(Cc2ccc(Br)o2)CC1.c12ccccc1NC2 c1(CC)n[nH]c(=NCC(C2CCCCC2)NC(c2ccc(C(C)(C)C)o2)=O)s1 c1(OCCC(=O)NCCNC(CC2C(C)CCC2)=O)ccc(F)cc1 Cc1nc(N2Cc3ccc(-c4cccc5ccnn45)cc3C2)c2ccsc2n1 c1(OC)ccc2onc(CC(=O)NC3C4CC3N(C(=O)C(C)(C)F)C4C)c2c1 Brc1ccc(-n2nnnc2C(c2csc(C3CC3)n2)NCc2cnccn2)cc1 c1(C(F)(F)F)cncc(CCC)c1.C(C1CCCC1)=C.C1(=CCN2CCC2)CCCC1 CC(C)C1=CCC(C(N2CC(C)N(C(C3CC34CCCC4)=O)CC2C)=O)CC1 Cc1cc(C(N2CC(C)CCC2C(=O)NCCC(C)F)=O)ccc1C#N N1(C(c2c(CC)nc(C)[nH]2)=O)CCCC(C)(NC(c2nn(C)cc2Cl)=O)C1 C=CCC(C(=O)N1CCN(C)CC1CNC(c1cc(OCC)n[nH]1)=O)C(C)C C=CCCCCCC(=O)NC1CN(C(=O)Cc2cncnc2O)CC1C c1(C(=O)NCC23CC(CNC(C(CC)O)=O)(OC2)C3)cccc(F)c1F N1(C(C2C(C)C2)=O)CC(F)(F)CC1CNC(c1cccn1Cc1ccccn1)=O C1(NC(c2c(CCNC(C3(COC(C)C)CC3)=O)n[nH]c2)=O)CN(C)CC1C1CC1 c1(CN2C(C(=O)Nc3cc(C)c(F)cc3)C(O)CC2)cc2c(Br)cccc2[nH]1 CC(C)(CC(=O)NCC1CCCC(NC(c2cc(=O)cc[nH]2)=O)C1)CC(F)F c1(C(N2C(C)(CC(=O)N(C(CO)C3CC3)C)CC2)=O)cc(C#N)ccc1N C1(C(=O)NC2(CSC)CC2)CC(O)CCN1C(c1cnnc(C)c1)=O CC1CCN(C(=O)CCS(C)(=O)=O)CCN1C(=O)C(C)CC1CCC1 C1(N(C(CN(CCOC)C)=O)C)CCCN(C(c2ccnn2C2CC2(F)F)=O)C1 C1(C(N(CC=CC(=O)NCc2nc(C)[nH]n2)C)=O)CC=CCC1C CC(C)C(N=c1[nH]c(Cl)ncc1F)C(C)NC(c1cnnn1-c1ccccc1)=O c1(C(=O)OC)cc(C(=O)NC(COC)C(=O)NCc2cn(C)cn2)no1 c1(CC)ccc(Nc2cccc(OCC(=O)OC)c2)cc1S(N)(=O)=O C1(C)(C(N2C(CNC(C(CC)(F)F)=O)CCCC2)=O)CCCNC1=O C1(C(=O)NCCC2N(C(c3c(CC)nns3)=O)CCC2)CCC(O)CC1 Cc1cc(C(=O)NCC(C)NC(C2CCN2Cc2ccccc2)=O)ncc1CO c12ccc(cc1)CNC1(CCC1)CNC2=O.C(=O)(C(F)C1CCC1)NCCl.C1CC1 C12(NC)CCC(CNC(c3ccc(F)cc3CCC(=O)NC3CC3)=O)(CC1)OC2 N1(C(C2CC(C)(O)C2)=O)CCOC2(CCN(C(C3(c4cc[nH]n4)CC3)=O)C2)C1 c1(NC(c2c(C)nn[nH]2)=O)nc(Cl)ccc1C(=O)Nc1ccccc1C(C)(C)C N1(CCNC(C2CC3CCC2(C(F)(F)F)C3)=O)CCCC(C2CCCCC2)C1 c1(C(=O)NC(C)CN(C(=O)C(O)C2CCC2)C)cccc(-c2cc[nH]n2)c1 c1(NC(C)=O)cnccc1C(N1CCCC1(C)CNC(=O)Cc1cc(C)cs1)=O c1(CC(=O)NCC2CC2NC(=O)C(c2cccc(Br)c2)O)ccc(O)nc1 Cc1ncnc(C)c1CC(=O)NC(C)C(CO)NC(C1CCC(C)(C)CO1)=O CC1(C)CN(C(C2CC2)C2CC2)C(=O)C1.C(C(F)(F)F)OCCNC(CS)=O C1(NC(C(C)=CC)=O)CC2(C1)CC(CNC(=O)C(c1cccn1C)=O)C2 C1(C(=O)NCCCCN(C(C=Cc2c(C)ccs2)=O)C)CCn2nccc2C1 C(=O)(C(C)CC(C)C)NCC(C)(CNC(=O)C(c1c(C)n[nH]c1C)C)OC c1(NC(C(C)O)C(=O)OC(C)(C)C)ccnc2c1CCO2 C1(NC(C(C)OCC)=O)CC2CC1N(C(=O)C(c1ccc(C3CC3)cc1)(C)C)C2 C1(NC(C2C(CNC(C)=O)C2)=O)(CNC(=O)C=Cc2ccoc2)CCCCCC1 N1(C(CC2(COC)CC2)=O)CC2COCCC2(NC(c2csc([N+](=O)[O-])c2)=O)C1 C1(OC)CC(CCNC(=O)CCCSC)N(C(=O)CCOc2ccccc2F)C1 c1(C(=O)NCC2N(C(CCCC=C)=O)CC(O)C2)ccc2cc(C)ccc2c1 N1(C(C2CC(C#N)C2)=O)CCC(N2CCN(C(C3CCC4CC4C3)=O)CC2)CC1 C1(C(=O)Nc2cccc(C(C)C)c2)CNC(=O)CN1C(=O)CCc1ccsc1 Cc1c(NCC(C)CO)nc[nH]c1=NCCC1CC=CCC1 c1(OCC)ccnc(CNCC2CCN(Cc3ccccc3)CC2)n1 N1(C(CC2CC(OC)C2)=O)CCC(NC(=O)Cc2coc(C(F)F)n2)C(CO)C1 N1(C(C(CNC(C(C2CC2)SC)=O)C(C)C)=O)CCc2c(F)cccc21 N1(C(c2c(CC)nns2)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)C(C)C1 Cc1[nH]nc(C(=O)NC2CCCC2CNC(c2sccc2Br)=O)c1C c1(C(N2CCC(CNC(C3CC4CC4C3)=O)C2)=O)c(Cl)cncc1Br c1(C(=O)NCC2(F)CC(NC(C=CC(C)(C)SC)=O)C2)cc(Cl)ncc1NC N1(C(C(C)(C)C#N)=O)CCC(C2CN(C(=O)CC3OCCOC3(C)C)C2)CC1 Cc1nc(C(C)C)nc(O)c1C(N1CCN(C(C2C3CCCC23)=O)CC1)=O c1(C(=O)NCCCC(C)NC(c2cc(OC)c(C)cc2)=O)cc(Cl)cc(Cl)c1O C1(OCCOC)CCCCC1NC1CCCC(c2ccc(F)cc2)C1 C=CCCC(C(=O)NC1CCOC(C)C1)NC(=O)CCC(C)(C)C c1(C(=O)NC(CN(C(C2CC(CCC)C2)=O)C)C)ccn(-c2ccccc2)n1 C1(NC(C(CCNC(C2C(C)CC2)=O)(C)C)=O)CCC(C2CC2)CC1 c1(OC)cc(F)c(CNC(=O)C(N2CC3CC(C2)CN(C(=O)C2CC2)C3)=O)cc1F CC1OC(C)C(C(N2CCC(O)(C(C)NC(=O)C3=CCCS3)C2)=O)C1C c1(C(C)C(=O)NC2(C)CCN(C(=O)Cc3ccoc3)C2)ccc(C#N)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC1CC(NC(C(COC)C)=O)C1 C(CC(C(=O)NCC12CC1CN(C(=O)COCCF)C2)N(C)C)SC C=CCC1C(=O)N1CC.C(C)(C(=O)NOCC1CC1)NC(C)=O C1(NC(c2cccc(CN(C)C)c2)=O)CCN(C(=O)COC2CCCC2)C12CC2 C1(=O)CC(C(F)F)CC(CC)N1.C(CC1CC1)(C1CC1)NC(=O)NC Cc1ncncc1C(=O)NC(c1ncoc1C)C(=O)NCC1CCCO1 C(=O)(CS(=O)(=O)CC)N1C(C(N2CCC2C(C)O)=O)(COC)C=CC1 N1(c2nnc(C(=O)OCC)c(CC)n2)CC2CC(NC3CC4CCC3CC4)C2C1 C1(F)(CNC(COCCOC)=O)CC(CNC(C2CCC2c2nc[nH]n2)=O)C1 Cc1ccnc2c(C(=O)NCCN(C(=O)CCCCCC(C)(C)C)C)cccc12 Cc1cc(F)cc(C(=O)NC2CCC2NC(c2c[nH]nc2F)=O)c1N Cc1cc(C(=O)N(CCCNC(C2CC2Cl)=O)C(C)C)c(C)n1NC(N)=O CC(C(=O)NCCOCCNC(=O)CCN1CCC(F)C1)C(C)(C)O c1(C(N2CC(COC)N(C(=O)CCSC)CC2)=O)ccc2ncn(C)c(=O)c2c1 c1(C(N(CCN(C)C(c2cc(Br)cnc2N)=O)C)=O)cc([N+](=O)[O-])nn1C c1(NC(C2C(CC)CN(C(=O)CC(C)NC=O)C2)=O)cc(CO)cc(F)c1 c1(SC2C(C(N(C)C)=O)CCC2)cc(Cc2ccn(C)n2)ccc1O C1(C)(CC)CCC(=O)NC1.N1CCC(CCC(=O)N2CC(n3cnnc3)C2)C1 C(C(CCC)C(=O)NCC)NC(C(C)OC1(C#C)COC1)=O C1(C(=O)NC(C)C(=O)NCC2CC2)CCCC1Cn1cc(CCCN(C)C)nn1 c1(C(N2CC(NC(CC3(COC)CC3)=O)C3C2C3)=O)cc(Cl)cc2c1OCC2 C1(C(=O)NCC(=C2CN(C(CCCNC(=O)OC)=O)C2)F)CCCCC1F C(=O)(C1CCCc2nn(C)cc21)N(C)CCNC(=O)Cc1cnn(C)c1 N1(C(c2ccc(C(C)C)cc2)C(=O)NCCSC)CCC(C)C(CO)C1 CCCCC(=O)C(=O)NCC(C(C)(C)C)NC(c1scnc1COC)=O CC1(c2ccccn2)CCN(C(N2CCOC(c3cc[nH]n3)C2)=O)C1 CCCC(C(=O)N1CCC(C)(CNC(c2ccc(C(F)F)nc2)=O)C1)NC(N)=O C=C(C)CCC(=O)NCC1(C)CCN(C(=O)C(N2CCNC2=O)C)C1 C(CN=c1c(C2CCCCC2C(=O)O)c[nH]c2ccccc12)NS(N(C)C)(=O)=O N1(C(c2[nH]cc(C)c2)=O)CCN(C(C2CC(C#N)C2)=O)C2CCCC2(C)C1 c1(NCC(C)CN(C)C)[nH]c(=NC2C3CC(Cl)CCC23)nc2sccc12 c1(C(C)=O)c(CCC(=O)N2CC(NC(C3CCC(C)C3)=O)C2)c[nH]c1C N1(C(=O)CCc2cccnc2)CCCC(C2CCN(CC(F)(F)C(F)F)C2)C1 N1(C(C(CC)NC(N)=O)=O)CCC2(CC(C(=O)NC34CC(C3)C4)C2)C1 c1(SCC(=O)NC2CC(NC(=O)C=CC3CCOC3)C2)ccc(C(F)(F)F)cn1 C(=O)(CCCC(F)(F)F)NCC(C1(O)CN(C(CC(C)n2ccnc2)=O)C1)(C)C c1(C(=O)NCCC2CC(NC(c3cc(OC)n[nH]3)=O)C2)nn(C)cc1Cl CC1=NN(C)C(=O)C1CC(N1CC=CC1CNC(C1(CC2CC2)CC1)=O)=O C=CC(C(=O)N1CSCC1C(=O)NCC=C=C)OC C(CCCCCNC(C1CCCC(=O)O1)=O)N(C(CC1N(C(C)C)CCC1)=O)C c1(OC)cc(C(N2CCC(CNC(c3ccccc3F)=O)C(C)C2)=O)ccc1F CC1CN(C(=O)Cc2cccc(O)c2)CCN1C(c1ccc(O)c(=O)cc1)=O C1(NC(C(CN(C)C)NC(CNC(CCC)=O)=O)=O)CCC(CO)CC1 N1(CC(=C)C)CC=C(CCNC(c2cc3oc(-c4ccccc4)cc3[nH]2)=O)CC1 N1(C(c2c(CC)ocn2)=O)CCC(CNC(c2cc(C(N)=O)no2)=O)C12CC2 c1(C(=O)OC)ncc(OC)cc1NC(=O)CCC1NC(=O)NC1=O C1(NC(C(C)(C)SCCC)=O)CCCCC1CNC(c1ccc(C)nc1)=O Cc1ccc(Cl)cc1C(=O)NCC1C(C)CCN1C(=O)CNC(=O)CC(F)(F)F Cc1cccc2nc(N3CCC4(CNC(=O)CN5CCOCC5)CCCC34)oc12 Cc1cnc(C)c(C(N2CC(CNC(=O)C=Cc3cnccc3C)C(O)C2)=O)c1 C1(NC(CCC#CC)=O)CC2(C1)CN(C(c1c(C(F)(F)F)coc1C)=O)C2 C1(NC(c2c(OC)ccs2)=O)CCN(C(C2CC2F)=O)CCC1c1ccccc1 C#CC1(NC(=O)CC(C)(C)CNC(C2(CO)CCOC2)=O)CC2CCCC12 C12(CNC(C3C(C(N)=O)C3)=O)CCC(CN(C(=O)CN3CC4CCC3C4)C1)C2 C12(CN3CCCN(C(C)=O)CC3)COCC1CN(CCCOc1ccccc1)C2 C1(C2(NC(N3CC(C(N4C(CN=[N+]=[N-])CCC4)=O)C3)=O)CC2)CCC(C)(O)CC1 CC1(C)CC(=O)c2[nH]c(=NC(CNC=O)CCOC(F)(F)F)oc2C1 c1(OCC(C(=O)N(CC(C)NC(c2cocn2)=O)CC)OC)ccc(Cl)cc1C C1(CCNC(c2c(COC)occ2)=O)NC(=O)NC1=O.C12(CCOC1)C(=O)N2 N1(C(CCN(C(C)=O)C)=O)CCN(C(=O)CCS(N)(=O)=O)C(C2CCC2)C1 C1(NC(CCCCC(=O)NCC)=O)CCS(=O)(=O)C12CN(C(=O)C1=CCSC1)C2 c1(C(N(CCCNC(c2coc(O)n2)=O)CC)=O)ccc(Br)nc1N C=CCCCCNC(=O)CC1(C)CN(C(=O)COC(C)(C)CC)C1 c1(C(N2CC=CC(NC(C(CO)NC(N)=O)=O)C2)=O)cc2occc2s1 c1(CCCNc2cn(C3CN(C(C(=O)OC)=O)C3)nc2)cccc(C)c1 c1(OC)nc(C)c(C(c2nnnn2C(C)C)NCCn2cnnn2)c(C)c1Cl Nc1sc2ccccc2c1C(=O)N(C1CS(=O)(=O)C12CCC2)CCO N1(C(CCC=C)=O)CCC2(CC1)CC2C(N1CCOCC(C(=O)O)C1)=O C#CCC(CC(F)F)C(=O)NC1(C(F)F)CC(C(=O)NC2CC2OC)C1 Cc1cc(F)cc(C)c1C(=O)NCC1CN(C)CCN1C(=O)C(O)CF Cc1ncc(C(N2CCSCC2CCNC(=O)CSCc2cccs2)=O)n1C C1(NC(Cc2ccc(SC)cc2)=O)CN(C(=O)C(C#N)C(C)(C)C)C2CCCC12 CC1CN(C(c2ccoc2C(F)(F)F)=O)CCN1C(c1cc(F)cnc1O)=O N1(C(COCC(=C)C)=O)CC(NC(c2nc(C)n(-c3nc[nH]n3)n2)=O)C(SC)C1 C(=O)(C(CC)C(C)(C)CC)NCc1occ(C(=O)NC(CCCC=C)C)n1 C1(NC(C(C)OCc2ccc(C)cc2)=O)CCN(C(C2CCCCO2)=O)C1(C)C C1(NC(CNC(c2cc(C)oc2C)=O)=O)CN(C(C2CC2F)=O)CC2(CCC2)C1 C(N=c1[nH]c(=NC2CCC3CCC23)[nH]c2c1CCC2)n1c(C)nc2cc(Cl)ccc21 N(C1CS(=O)(=O)c2ccccc21)C(CC1C(C(=O)OCC)C1)=O n1(CC)nc(C(=O)NC2CN(C(C3CCCCC3C(N)=O)=O)CC2C)c(C)n1 N1(C(c2cc(CCC)on2)=O)CC2CCC1CN2C(=O)C1=NOC(C)(C)C1 C(C)(CCCC(=O)N1CCC1CN=[N+]=[N-])NC(CCCC=C)=O C(=O)(C1=CC2C=CC1C2)NCC1(C)C(C)CN(C(CCc2ccnc(C)n2)=O)C1 c1(C(C(N)=O)NC(C2(F)CN(C(C3CC3F)=O)C2)=O)ccccc1Br C1(CC(=O)NC)CN(C(=O)CCCN(C)C(C)=O)CCN1C(=O)CC(C)C1CC1 Cc1ccc2c(c1)CN(C(C1(NC(=O)CC(=O)NC3CC3)CC1(C)C)=O)C2 C1(CC(=O)NCCCCN(C)C(c2c[nH]c(Br)c2)=O)CCOC(C)(C)C1 C=CC1(O)CCN(C(=O)COC2(C)CN(C(=O)C=C(C)C)C2)C1 C1(NC(C(C)n2cnnn2)=O)CN(C(c2ccc3occc3c2)=O)CC2(CC2)C1 C(N=c1ccnc(N2CC(OC)C3(CC3)C2)[nH]1)c1c(C)nc(CCC)o1 N1(C(CC(C=C)C)=O)CCOCC(C)(CNC(c2c(Cl)c(C)nn2C)=O)C1 c1(NC(C2CCN(c3cncc(OC)n3)CC2)C)cc(C(C)O)ccc1[N+](=O)[O-] N1(CC(=O)NC(C2CCN(C(=O)CSc3ccccn3)C2)C)CCOCC1 c1(C(C(=O)NC(C2CCN(C(C3C=CCS3)=O)C2)C)=O)cccn1C c1(OC)cc(C(=O)NC2CC3CN(C(=O)C(C)O)CC3C2)c2c(c1)CCO2 O=C(C1CCOc2ccccc21)NCC12CCCN(C(=O)Cc3cscn3)C1C2 C1(C(N2CCCC(c3cccc(C)c3)C2)=O)CCC2(CC1)NC(=O)N(C)C2=O N1(C(CC2C(C)C(=O)CC2)=O)CCC2(CC1)CC2CNC(c1ncn(C)n1)=O c1(C(CO)N(C(C2(CC3CCCC3(C)C)CN(CC)C2)=O)CC)ccccc1Cl Nc1c(C(=O)NCC(CNC(c2cncc(C3CC3)c2)=O)CO)cccc1F c1(OC)ccc(Cl)c(C(N2CCC(O)(C(N3CCCC(F)(F)C3)=O)C2)=O)c1Cl c1(OCC(=O)NCCCC(C)NC(CSCCC)=O)ccc(Cl)c(C)c1 CC1NC(=O)C(N(C)C)=C1NCC(O)C(C)(F)F C1(NC(c2cccnc2O)=O)CCCN(C(C2(Cl)CC2(F)F)=O)C1 Cc1ccc(F)cc1-c1noc(C2C3CN(C4(c5nnn(C)c5N)CC4)CC23)n1 N1(C(c2c(C)csc2)=O)CCC(C)C(CC(=O)NC(Cc2ccco2)CO)C1 CC1CCN(C(c2cccc(Cl)c2)=O)CC1NC(=O)CC1CC2CCC1C2 N#Cc1cc(COc2ccccc2C#N)nc(-c2ccc(F)cc2)c1 C1(C(=O)NCc2c(C)ocn2)CC(=O)CN1C(C1CC(=O)C1(C)C)=O CC1(C(F)(F)F)c2ccccc2CCN1C(CCc1ccsc1)C(=O)NC1CC1 c1(C(=O)NCC2CC(C)N(C(c3ccncc3)=O)C2)ccc(N=S(C)(C)=O)s1 c1(C(=O)OC)nc(NCCN(C2CCCCC2)C(=O)C=CCO)c(F)c(Cl)n1 C1(NC(C(C2CCCCC2)OCC)=O)CC12CCN(C(C1(CN(C)C)CC1)=O)C2 C(=O)(CCCCCCN(C)C(C)=O)NCCCCC(=O)NC(C1(OC)CCC1)C CC(C(=O)NCCCC1CN(C(c2cc(C(F)F)ncn2)=O)CCO1)S(C)(=O)=O C(c1ccc(F)cc1)=C(C)C(=O)NCC(C)NC(c1ccc(N)cc1F)=O C12(CNC(C(CC)(C)C)=O)CCC1CCN2C(c1cc(C2CCOCC2)on1)=O N1(C(C2C(CC)CCC2)=O)CC2CC1(CNC(C1(C(F)F)CCCO1)=O)C2 N1(C(CC(C)CN(C)C)=O)CC2(C)CC1(C(=O)NC1C=CCCCC1)C2 N1(C(C#CC(C)C)=O)C2CCC1CC(N(C(=O)CCC1CC1(Cl)Cl)C)C2 N1(C(COC2CCN(C(C(C=C)CC)=O)C2)=O)CC(O)C(C2CC2)C1 Cc1cn2c(n1)C(C(=O)NC1(C)CCN(C(C3(CF)CC3)=O)CC1)CCC2 C(CSC)(C(=O)NCC1CC(NC(=O)CCCn2cc(C)cn2)C1)OC c1(CCC(=O)NCCCNC(C(C)OCCOCC)=O)cc(F)ccc1Br CCC(C)C(O)C(=O)N1CC2(NC(=O)C(N3CCC(C)CC3)=O)CC1C2 c1(CC(=O)NC2(C)CCN(C(C(C(C)C)C#N)=O)C2)nc2c([nH]1)CCCC2 c1(OC)ccnc(C(=O)NC2(C)CC(NC(C3CC3(Cl)Cl)=O)C2)c1OC c1(CC(=O)OCC(c2cncs2)=O)ccco1 N1(C(C2CC2(F)F)=O)CCC2(C(=O)NN(c3ccc(F)cc3)C3CC3)CC2C1 CC1(NC(=O)CCc2cc[nH]n2)CCN(C(C2CC2C(F)(F)F)=O)C1 c1(OC)ccc(O)c(CNC2CC(C)CN(C(=O)Cc3ccc(F)cc3I)C2)c1 OC12CC1C2.c1(CN2CCCC2)cnc(-c2ccccc2)o1 C=CCCC(C(=O)N1CCCC(C)C1)NC(c1cc(C)cc(F)c1)=O C=CC1(C(N2CC(NC(c3ccoc3C3CC3)=O)C2)=O)CCCCC1 C1(C(=O)NCCN(C(CCCC(N)=O)=O)CCOC)Cc2n[nH]cc2C(=O)N1 C1(C(=O)NC(CCC)C2CCCC2)CCC(C)(C)N(C(=O)C2=CCC(C)CC2)C1 N1(C(C=CC=CC)=O)CCc2sc(CNC(C3(F)CC3(Cl)Cl)=O)nc2C1 c1(C(=O)NC2CCCCCC2NC(C2CCCSC2)=O)ccc2nonc2c1 N1(C(CCC#N)=O)CCC(NC(c2c(C3CC3)cccc2F)=O)CC1C1CC1 N1(C(C)C(N2CCCC2C2(NC(C3SCCCS3)=O)CC2)=O)CCCCCC1 c1(CC(=O)NC(CNC(CC(C)=C(C)C)=O)(C)C2CCC2)ccc(F)c(C)c1 C1(NC(C2C(CC)CCO2)=O)CN(C(c2coc(Cl)n2)=O)CCC1C C(N=c1cc(C)nc(C)[nH]1)C1N(C(C(c2cccc(C)c2)(F)F)=O)CCCC1 Cc1ccc(C(=O)NCC=CCNC(C2CC2C(C)O)=O)c(F)c1F C1(O)(C(=O)NCC2CCC(NC(c3ccc(C)[nH]3)=O)C2)CCCC(C)CC1 C1(CNC(c2cc(=O)cc[nH]2)=O)CN(C(=O)CCc2nc(O)n[nH]2)C2CC12 C1(C(N2CCC(NC(CNS(CCOC(C)C)(=O)=O)=O)C2)=O)CC2CCC1O2 N1(C(C(CCNC(C2CCCCN2C)=O)O)=O)CC2CN(Cc3ccccc3)CC12 c1(C(=O)NCC(C(C)C)NC(C(C2CCCC2)OC)=O)sc(C)cc1C N1(C(C(C)C2CCC2)=O)CCC2(CC1)CN(C(=O)Cn1nccn1)C1COCC21 C1(F)(C(=O)NC(C)CCCCNC(C2CCC2C)=O)CCCCCC1 N1(C(c2cc(C(C)=O)oc2)=O)CCC(C(C)(C)NC(C2CCN(C)C2C)=O)CC1 c1(CN2C(NC(=O)NCc3ccco3)CCC2)cc(F)cc(Br)c1 c1(CCC(=O)O)ccc2nc(C(N3CC(C(F)(F)F)C(C(F)(F)F)C3)=O)oc2c1 c1(C(N2CC3C(NC(CCCC(=C)C)=O)C3C2)=O)cc2c(=O)[nH]ccn2n1 Cc1csc(C(=O)N(CCC(C)NC(=O)C(C)C2CC2)C)c1C N1(C(c2cccc(SCCCC)c2)=O)CCC2CN(C(c3cscc3F)=O)C2C1 N1(C(=O)OC)C2CCC1CC(C(=O)NCCCC(CSC)Cc1ccccc1)C2 Cc1c(C(=O)NC(CNC(C2(Cl)CCCCC2)=O)CO)cccc1F c1(C(=O)NCC(=C)CCNC(=O)COC(F)(F)F)ccc(=O)n(C)n1 c1(N(CCC)C)ccc(C(=O)NC2CCN(C(=O)C(C)CC34CC(C3)C4)C2)cc1 C1(C(N2C(CCN(C)C)CCC2)=O)COCC(=O)N1CCC(F)(F)F C1(C2CCN(C(c3cc4c[nH]cnc-4n3)=O)C2)(NC(c2cnco2)=O)CC1 c1(C(N2CCN(C(=O)CC3C=CCC3)CC2C2CCC2)=O)nccn2ccnc12 N1(C(CC(CC=C)(C)C)=O)CCC2CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)CCC12 c1(COC)cc(=NCC23CCC(CN)(CC2)CO3)[nH]c(Cl)n1 C1(C(C(=O)OC)N)CCCN(C(=O)Cc2nc(-c3ccc(F)cc3)cs2)C1 C12(C(N(C3CN(C(c4cc(C(C)C)on4)=O)C3)C)=O)CCOC1CCOC2 C(=O)(CC(C)NC(=O)CCC1CCC(NC(=O)CC(C)N(C)C)C1)OC C(=O)(C#CC1(C)CCCO1)N(CC(O)CN(C(=O)Cc1nncn1C)C)C O=C1CC(CC(=O)NC2C3CN(C(c4ccc([N+](=O)[O-])s4)=O)CC23)CC(=O)N1 c1(C(=O)NCC2C(CNC(C(C)=CC3CC3)=O)C2)cnc(S(C)(=O)=O)s1 c1(NC2CC3CC3C2)cc(C(=O)OC)[nH]n1 N1(C(C(CC)CC)=O)CC2CCC2(NC(=O)C=CS(C)=O)C1 CCCCC(O)CCC(=O)N1CCCOC(CNC(c2csnc2Cl)=O)C1 C1(CC)CCC(C(=O)NC2(C)CN(C(C3(CF)CCOCC3)=O)C2)CC1 C(=O)(C(C)(C)CCCO)NC1CN(C(c2c(=O)ccn(C)c2)=O)CC1(C)C N1(C(C2C(C)(C)OCC2)=O)CCC2(CCC2)C(CNC(=O)C2=C(Cl)CC2)C1 CC1CCC(NC(c2cc(=O)n(C)cc2Br)=O)CN1C(=O)Cc1cnc[nH]1 Cc1oncc1C(N(C1CCN(CC(=O)NC2CC2)C1)C(C1CNC(=O)N1)=O)=O CCCC(C)C(C)(c1nnnn1CC)NCc1ccc(CCO)cc1 C1(NC(c2nc(C(C)=O)sc2)=O)CCCN(C(C2(C)CCCC2)=O)CC1F C1(CC(N2CCCC2CO)=O)CCN(C(c2cncnc2C2CC2)=O)CC1 N1(C(C(=O)NCC(C2CCCO2)OCC2CCCO2)=O)CCC2(CC1)CS(=O)(=O)C2 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCCC(C)(NC(C2CN(C(C)C)CCO2)=O)C1 N1(C(C(=O)NC(C2(C)OCCO2)C)=O)CC(O)(C(=O)OCC(C)(C)C)C1 c1(C(C(=O)N(C)CC2N(C(CC)=O)CC(F)C2)(C)C)c(C)[nH]c2ccccc12 CCC(C(=O)N(CCC(=O)NCC(C)(C)C1CC1)CCO)OC Cc1ccccc1CC(=O)NC1CN(C(C2(CO)CC2)=O)CC1CC1CC1 c1(OC)ccc(C(N2CCNC(C(=O)NCCC(C)C)C2)=O)cc1OC C1(C(N2CC(Nc3nccc(OC(C)=O)n3)C2)=O)CN2CCN1CC2C c12c(OC)cnnc1OC2.C1(C(=O)OC)COCC1NC(=O)OC(C)(C)C c1(NC(C2N(S(c3c(C)n[nH]c3C)(=O)=O)CC2)=O)cccc(C#N)c1[N+](=O)[O-] c1(NCC2C(C)C2(F)F)[nH]c(=NCC2CNC(=O)C2)nc2c1ncn2C c1(N(C(=O)CC2CC(=O)N2)C(c2c(SC)scc2)=O)c(F)cc(Br)cc1[N+](=O)[O-] c1(C(N(CCOCCCN(C(C2C(C)(CC)C2)=O)C)C)=O)cccc([N+](=O)[O-])c1 c1(CC(=O)NC2(C)CCN(C(C3(C)CC=CCC3)=O)C2)c(F)cccc1F N1(C(CSC)=O)CC2=C(C1)CN(C(=O)Cn1nc(C)c(Br)c1C)C2 C1(C(=O)NCCc2c(C)nsc2)(NC(=O)C(O)Cc2cnc[nH]2)CCOCC1 c1(C(=O)NC2CC(CNC(C3(OC)CCSC3)=O)C2)cnc2c(c1)COCC2 c1(C(C)=O)cnc(Cl)[nH]c1=NC1CCN(C(c2nnn(C)c2C(F)F)=O)CC1C C1(NC(CCCCC#C)=O)CC2(CCC(CNC(c3cnccc3Cl)=O)CC2)C1 N1(C(C2C(C)(C)C2)=O)CCCC(C2CN(C(=O)C(c3ccc(Cl)cn3)(F)F)C2)C1 c1(CN2CC2)c(Br)cncc1Br.C(=O)(C1=CCCS1)N(C)C N1(C(C(C)NC(=O)C2CC2)=O)CCCC2(C1)CC2(F)F Cc1ccc(CC(=O)NC2CCN(C(c3cc(C(F)(F)F)cn3C)=O)CC2)cn1 c1(C(=O)OC)cnc(NC(c2cnc(-c3cnccn3)s2)=O)s1 c1(C(=O)OC)cc(C(N2CC(=O)N(C)CC2C(=O)OC2CC2)=O)c(Cl)cc1Cl N1(C(C(CCC)NC(C)=O)=O)CCCC(C2CN(C(=O)C3=NOC(C)C3)C2)C1 CN1CCC2C(CCN2C(C2(C)CN(C(C3CCC4(CC4)C3)=O)C2)=O)C1 C12(NC(CC=CC)=O)CCOCC1CN(C(c1cccc(C#N)c1)=O)C2 CCCCC(CNC(c1cnccc1N(C)C)=O)NC(=O)CC(=O)NC1CC1 C1(C)(CC)CC(NC(c2ccc(C(C)(C)C)s2)=O)CN1C(=O)CC=C(C)C Cc1sc(Cl)nc1C(N1CCCC(n2cc(CN3CCCCC3)nn2)C1)=O C(=O)(CCCC(=O)N1CCCC(NC(=O)C(C)(C)n2ccnn2)CC1)OC C1(CN(C)C(C2CCC(=O)N2)=O)CCCCN1C(c1ccc(=O)oc1)=O C(CC1=CCCCC1)N(C(CC1CC2CC(=O)C1C2)C(=O)NC1COC1)C C1(CC=C)CCCCN1C(=O)CNC(=O)CC#N c1(C(=O)NC(CNC(C(F)=CC)=O)(C)C)nn(CC)cc1Cl N1(C(Cc2cc(C)sc2)=O)CCC2(CC1)CC(NC(=O)CCn1cnnn1)CO2 c1(NCC(CC)Oc2ccccc2)cc(C)c(S(=O)(=O)N2CCCC(O)CC2)cn1 c1(NC(C2(c3c(-c4cccs4)csc3C)CC2)=O)ccc2nc(C)oc2c1.CO c1(C(=O)NCC(C)NC(c2cc(C(F)(F)F)c[nH]2)=O)cccc2cccc(O)c12 C1(CCOC)(NC(c2cnc(OC)s2)=O)CCN(C(=O)CC(C)n2cccc2)C1 C1(NC(CCC2C(C)(C)C2)=O)CC2(C1)CC(NC(c1ccc(Br)c(N)c1)=O)C2 C1(CNC(C(CC)(C)OC)=O)CCC2CN(C(C3C=CCS3)=O)CC12 CC1CN(C(=O)Cn2nnc(=N)[nH]2)CC1CNC(c1cn(C2CCCC2)nn1)=O C1(C(N2CCC(SC)CC2)=O)CN(C(=O)C=CC(F)F)C2(CCC2)C1 c1(C(N2CCC(NC(C3(C)CC(=C)C3)=O)C2C(C)C)=O)ccnc(F)c1OC c1(C(=O)NCC2CCC(C)N(C(=O)COC(C)(C)C)C2)cccc2[nH]ncc12 N1(C(C(C)CCN(C)C)=O)CCOCC1(C)c1cn(-c2cccc(Cl)c2)nn1 C1(C(N(CCCCO)C)=O)C2CCCC2CN1C(C1CCC(=O)N1C)=O O(N(CC)C(=O)C1CC=CC(NC(c2ccnc(OC)c2)=O)C1)CC C1(CCCNC(C(COC)OC)=O)CCCCN1C(=O)C=C(C)c1ccco1 C1(CCNC(CCC(=O)NCCC)=O)CCCN(c2nccc(CC#N)n2)CC1 N(C)(C(=NCCF)NCC1C2CCC(CNC1=O)O2)C(C(F)(F)OC(C)C)(C)C Cc1cccc2c1C(=O)NC(C)(C)N2C(=O)Cc1coc2ccccc12 S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(CSC)cc1F)N(C(CC)CC)CC O=C1CC2(CCC2)C(C(N2CCN(C(C3(CO)CCOC3)=O)CC2)=O)CN1 c1(C(=O)NCC2C(NC(c3cn(CCOC)nn3)=O)CCC2)cc2ncccn2n1 C(N1CCC(P(C)(C)=O)C1)N1C(C)c2ccccc21 Cc1ccnc(C)c1C(=O)NCCN(C(=O)C(O)C1CC1)Cc1ccccc1 C1(F)(C(=O)NCc2cc(OC)no2)CCN(C(=O)C(F)C(C)C)CC1 c1(C(N2C(C)CCN(C(C3CC(OC)C3)=O)CC2)=O)cc(O)nc2cnccc12 c1(C(=O)NC2CS(=O)(=O)CC2NC(c2ncccc2O)=O)cnc2n1CCOC2 Cc1c(C(N2CCN(C(C3CNC(=O)C3)=O)CC2)=O)sc2[nH]cnc(=O)c12 C1(CCNC(C(C)C)=O)CN(C(=O)C(C)(O)c2ccccn2)CCO1 N1(C(CCNC(=O)OCC)=O)CC2C(CC(=O)N(CC(F)F)C3CC3)C2C1 c1(CNC(=O)OCC2CCOC2)ccc(CO)c(Cl)c1 N1(C(C2C(C(=O)OC)C2)=O)CC(NC(c2cccc[n+]2[O-])=O)CC2(CCC2)C1 C(=O)(CCC(C)CN(C)C)NC(CCCC)CNC(=O)CCNc1ccccn1 C1(C2CN(C(CC3(C)CC3)=O)C2)CCCCN1C(=O)C=CC1CCOC1 n1(C2(C)CC2)nnnc1C(c1cc(Cl)cs1)NCC1(n2ccnn2)CC1 c1(CC)cc(C(N2CCC(NC(c3ncccc3F)=O)C(O)C2)=O)cc(Cl)c1 N1(C(c2ccc(C)cc2C)=O)CC2CCCC1CN(C(=O)COC(C)C)C2 C1(CNC(C(c2ccc(F)cc2)C)=O)CC2CN(C(C3CCCS3)=O)CC12 C1(C(=O)NCC2(F)CN(C(C(CC=C)NC(C)=O)=O)C2)CCC2(CCOCC2)O1 c1(C(=O)NCC2CCC(NC(c3ccc(CC#N)cc3)=O)C2)cc2n(n1)CCC2 N1(C(Cc2c(C)n[nH]c2)=O)CC2CC1C2NC(C1(CC(F)F)CCC1)=O c1(C(N2CCCC(OC)C2)C(=O)NC)cccc(C(=O)Nc2ccccc2Cl)c1 C1(NS(Cc2c(Cl)ccc(OC)c2)(=O)=O)CNCC1C1CCOCC1 N1(C(C(CSC)C)=O)CCC(CF)(NC(=O)Cc2ccccc2F)C1 c1(C(=O)NC2(CC=C)CN(C(c3nsnc3O)=O)C2)coc2c1COC2 CC(C)(C)CC(O)C(=O)NCCCCCCC(=O)NCCCC1(O)CC1 C1(OC)CC2C1CCN2C(c1ccncc1Cl)C(=O)NCC1CCOC1 C1(C(=O)NCC2N(C(C(c3cn(CC)nc3)=O)=O)CC2)CCCC2(C1)CC2(F)F c1(C(=O)NCC2(O)CCN(C(C(CCC#C)O)=O)C2)c[nH]c2ccc(C#N)cc12 c1(C(=O)NC2C(NC(=O)OCCOC)CCCC2)nc(Br)ccc1N c1(C(N2CC(CC(=O)Nc3cc(C#N)c(Cl)cc3)C2)=O)ccc(O)c([N+](=O)[O-])c1 N#CC1(C(=O)NCCCCCNC(c2ccc(C3CCOC3)s2)=O)CC2CC2C1 n1(CCC#C)c(N(C(C)(C)C)CC2CCCOC2)nnc1CC(O)C(C)C O=C(C(F)(F)CCn1cc(-c2ncccn2)nn1)NCC1CCS1(=O)=O C1(NC(=O)C=CCO)CN(C(=O)COc2ccccc2Cl)CC1CC(O)CO C1(NC(CC2(CNC(=O)Cn3nccn3)CC2)=O)(CC2CC2)CC2CCCC12 CCC(CCCC(=O)NC(C)(CO)C1CCC1)NC(c1coc(C(C)C)n1)=O c1(C(N2C(CNC(c3cc(OC)no3)=O)C(C)CC2)=O)cnc2[nH]c(C)nc2c1 c1(C(=O)OC)cc2c(s1)CCC2NC(=S)Nc1cccc(F)c1C#N c1(CNC(C(CC=CC)NC(=O)OC(C)(C)C)=O)ccc(CS(C)(=O)=O)c(Cl)c1 n1(CCOCC)nnnc1C(c1ncoc1C(F)F)NC1CC(C)C1 c1(OCC)cc(-c2nccn2CCCn2cccc2)cc(C2CC2(F)F)c1O C(=O)(C(C)CCCC(C)C)N1CC(CC(=O)NC(CC)C(=O)NC)OCC1 CC(C)CC(CNC(=O)CN1CCSCC1)NC(c1ncccn1)=O C1(OC(N2CC3(C(=O)OC)CC2(C(=O)O)C3)=O)CC(O)CN(C(C)(C)C)C1 N1(C(C=C(C)c2ccccc2)=O)CC2CC(C1)CN(S(=O)(=O)CC(C)C)C2 C(=O)(C1SCCc2sccc21)NC(CNC(c1cc(C)n(C)c1)=O)CO N1(C(CCC2CCCCN(C(c3cccc[n+]3[O-])=O)C2)=O)CC2CCC(C1)C2O C1(C(C)(C)NC(CNC(CC)=O)=O)CCN(C(=O)C(F)=C2CCCC2)C1 C(CC(O)C(=O)NCC1CCN(C(C2CCCC2c2nncn2C)=O)CC1)SC N1(C(C2CCC(CNC(C(C3CCC3)OCC)=O)CC2)=O)CC2CCOC2C1 Cc1nc(C=CC(N2CC(F)(CNC(C3CCC3C(F)F)=O)C2)=O)cs1 C12(NC(C=CC(C)C)=O)CCN(C(C3(c4ncc[nH]4)CC3)=O)CC1C2 N1(C(c2c(CC)cno2)=O)CC(NC(=O)CCCOc2cccc(C)c2)CC1C n1(C(CNC(Cn2cc(C(CC)N(C)C)nn2)=O)C)ncn(C)c1=O C(C(C)(C)CC(=O)N(C1CCCN(C(=O)C(C)CC(N)=O)C1)C)OC N1(C(C2(CC#C)CC2)=O)CCC2(CC(NC(=O)CCOC)c3ccccc3O2)C1 C1(C(=O)OCC)CCC(CC(=O)NCCn2cc(CC(C)(C)CO)nn2)CC1 Cn1nccc1C=CC(=O)NC(C1CCOC1)CNC(=O)C(C)(C)n1cc(Cl)cn1 CCC(C)(C)CCCC(=O)N1CC(C(=O)NC(CO)CC(C)(C)C)C(C)C1 C1(C2CCC2)(C(N2C(C3(O)CN(C(C4(COC)CCCC4)=O)C3)CCC2)=O)CC1 N1(C(CCC#C)=O)CCC2(NC(=O)CCn3ccc(O)nc3=O)CCCC12 CC(C)CC(O)C(C)C(=O)NC1CCCC(CC(N2CC(N(C)C)C2)=O)C1 C1(C(N(CC(CN(C(=O)CN2CC(=O)NC2=O)C)O)C)=O)CC2CCC(C1)S2 C1(C(=O)NC2(CC(=O)NCCCn3cccn3)CC2)CCS(=O)CC1 c1(CC)ncc(C(=O)NC2CCN(C(c3cc(CC)ccc3N)=O)C2)c(C)n1 C1(CC)CN(C(=O)COC(F)(F)F)CCN1C(C1CCN(C)C(=O)C1)=O N=c1[nH]c(CC(=O)NCC2(CNC(=O)CC3CC3)CC2(F)F)cs1 C1(NC(C(C)C)=O)CCN(C(C2(CF)CC2)=O)CCC1(F)F c1(C(C)C)nc(C(=O)NCCOCCCNC(=O)CCc2cnc(O)[nH]2)cs1 c1(C(=O)NC2(CN(C(CN3C(=O)CN(C)C3=O)=O)C)CC2)nccc2cc[nH]c12 C1(CC=C)(NC(C2CC2=C)=O)CCN(C(=O)C(=Cc2ccco2)C)C1 c1(C2(C(N3C(CNC(c4ccc(Br)o4)=O)CCC3)=O)CC2)ccnc2ccccc12 C1(CC(N2C(CNC(CN(CC(=O)NC(C)C)C)=O)CCC2)=O)SC(=N)NC1=O Cc1c(C(N2CC(CO)(NC(=O)Cc3cccs3)C2)=O)ccc(F)c1F C1(NC(C2CCC(=C)CC2)=O)CCCC12CCN(C(c1[nH]c(C3CC3)nc1C)=O)C2 C1(CCNC(C(SC)SC)=O)CN(C(=O)Cn2ccccc2=O)CC1C CCCCC(CNC(=O)CCS(C)=O)NC(c1cnc(N(C)C)o1)=O c1(C(=O)OC)cnc(N=S(C)(C)=O)c(N(c2ccc(F)cc2)C)c1 c1(Cn2nnnc2C(COCC)(C)N2CCCC2)noc2c1CCC2.C1CCO1 Cc1ccc(NC(=O)CSC2COC(C(F)(F)F)C2)cc1 N1(Cc2cc(C)on2)CCCC1C1CCCCN1C(c1cc(C2CC2)no1)=O N1(C(C(C)CF)=O)CCCC(C)C1CNC(c1cnn(C2CC2)c1)=O C1(NC(C=CC=CC)=O)C2CC1N(C(C1CC1c1ccccc1Cl)=O)C2 Cc1cc(C(=O)NCC(C2CC2)NC(C2CCC3(CCC3)C2)=O)cc(C)c1C N1(C(C(C)C2CCC2)=O)CC(NC(C2(c3cccnc3Cl)CC2)=O)C(C)C1 CC(C(=O)NC1CN(Cc2cn3cc(Br)ccc3n2)C1)C(F)(F)C(F)F N1(C(CCCCCOCC)=O)CCC2CN(C(=O)CC3CC(C)(C)C(=O)N3)CC12 N1(C(c2c(C)n(C)cc2)=O)CCC(N(C(=O)CSC(C)(C)C)C)C(C)C1 C1(CC=C)CCCN(C(=O)C(O)Cn2cncn2)C1 Cc1nc(C(N2CCCC(N(C(=O)CCCc3ccc(Cl)cc3)C)C2)=O)nn1C c1(-c2nc(-c3cccc(SC)c3)on2)cnn2c(C)c(C)ccc12 c1(C(=O)NC(CN(C)C)C(=O)NCC23CC(CCO2)C3)ccccc1C(N)=O C12(CNC(CSCCOC)=O)CCC(CNC(=O)C(C)c3ccco3)(CC1)CO2 N1(CCC)CCN(C(=O)C(C)CNC(=O)CC(CC)SC)CC1 C1(C(=O)NCCCNC(=O)CSCC2CCCO2)CNC(=O)CC12CCC2 N1(c2cc(COC)ncn2)CCC2(CC1)CC(NC(C1(OC)CCC(C)C1)=O)C2 C1(CN(C(C(COC)OC)=O)C)CN(C(c2cc(C)c(C)o2)=O)CCO1 c1(C(N2CC(C)C(NC(c3cc4ncccc4s3)=O)C2)=O)coc(S(N)(=O)=O)c1 Cc1cccc(F)c1C(=O)N(CCC(C(C)C)NC(=O)CC1SC(=N)NC1=O)C C1(CNC(C2(C(C)(F)F)CCC2)=O)CC2(CC2)CN1c1nc(CC2CC2)ns1 CC1(C)CCC(O)(CNC(C2(CNC(=O)CCC3(C)N=N3)CCCCC2)=O)C1 C(=O)(CC(F)(F)C(F)(F)F)NCCCCCNC(C1(OC)CCC12CCC2)=O CC(C)(C)C(C#N)C(=O)N1CCN(C(c2ccc(C3CC3)cc2Cl)=O)C2CCC12 Cc1cnc(N2CCC(C)CC2)c(S(=O)(=O)NC2CCCCN(C)C2)c1 Cc1ccc(Cl)c(O)c1C(N1CCCC(NC(C2CNC(=O)C2)=O)CC1)=O c1(NC(C2NCC(C(=O)OC)C2)=O)ccc2nccn2c1C c1(C(N2C(CNC(C=CSC)=O)CCC(C)C2)=O)onc2c1CCCC2 N1(C(CC2C(C)=NOC2=O)=O)CCC(CNC(=O)Cc2nc(C)sc2C)C(C)C1 N#Cc1cc(C(N2CC3CN(C(C4CC45CCOCC5)=O)CC23)=O)ccc1F C1(CC(=O)NC(C2CCN(C(C3CC(O)C3)=O)C2)(C)C)CC2CCC(C1)N2C c1(OC)c(NC(=O)NCCCN(CC)Cc2cncc(OC(C)C)c2)cccc1Cl C(=O)(CN=c1cc[nH]cc1)N1CCC(NC(N)=O)C(F)C1.N12CCC(CC1)C2=O c1(C(N2CCN(C(C(C)OC)=O)C(C3CC3)C2)=O)cccc2ccccc12 C=CC1(O)CCN(C(C2CC=CCN2C(C2CC(C3CC3)C2)=O)=O)C1 C1(CNC(Cc2cc(C)sc2)=O)CN(C(=O)CCCC(C)(F)F)CCC12CCC2 CC(C)C(C(=O)Nc1ccc2ncnn2c1)C(C)NC(=O)CNC=O N1(C(CCN(CCC)C)=O)C2CCC(C(=O)NCc3n[nH]c(C)n3)C1CC2 c1(N2CC(NC(c3c(OC)cncc3)=O)C(C)CC2)ncn(C)c(=O)c1Br c1(CC)cccc(C(N2C(C(N3CC(COC)CC3O)=O)C2C)=O)c1 c12ccccc1CCOC2=O.C1(C(=O)SC)CCCS1(=O)=O C1(C(N2CC(CN(C(c3c(C)nsc3N)=O)C)C2)=O)CCc2c[nH]nc2C1 N1(C(CC2(C(=O)OC)CC2)=O)CCC(O)(CNC(=O)CC2CCCC2C)CC1 c1(C(N2CCN(C(C(C)O)=O)CC(O)C2)=O)ccnc2c1ccn2C N1(C(c2c(Cl)nc3sccn23)C(=O)NC(CC)C)CCN(C)C2(CCC2)C1 C(=O)(C1=CCCN(C)C1)N1CCC(C(=O)NCc2ccc(C#C)cc2)(CC=C)C1 C1(CC(=O)NCC2(COC)CCCO2)CC(C)N(C(c2cc[nH]c2)=O)C1 CC1(C)CC1(NC(c1cccnn1)=O)CN.c1(C(C(=O)O)N)ccccc1 C1(N(C(CSCC=C)=O)C)CC2CCC(C1)N2C(c1cnc(N(C)C)o1)=O Cn1c(C(=O)NCc2cn(CCSc3ccccc3)nn2)ccc1C#N N1(C(c2c(CCC)n[nH]c2)=O)CC(O)CC1(C)C(=O)NCc1cccnc1 Cc1ccnc2c(S(=O)(=O)NCC(c3ccc(=N)[nH]c3)=O)cccc12 C1(C(=O)NC(CCC)C(=O)NCC2(C)CCC(=O)N2)CN(C)CC(C)O1 C=Cc1cc(C(=O)NCCC2CCCN2C(c2c(F)cccc2F)=O)cc(F)c1 c1(C(c2ccc(Cl)cc2)NC(N(C)CCN(C)C)=O)ccccc1F C1(C#N)(C(N2CC(C(C(=O)N(CCCC(=O)NC)C3CC3)OC)C2)=O)CC(F)(F)C1 c1(C(=O)NCC2C(CNC(c3cnc(S)[nH]3)=O)C2)cc2ccsc2c(O)n1 c1(C(=O)NC2(CNC(c3ccc(Cl)cc3Cl)=O)CC2)coc(=O)c2ccccc12 CCC(C)C(C(=O)N(CCCNC(=O)CC#N)C(C)C)N(C)C C1(CCC(C)(C)NC(=O)CSC(F)F)CCN(C(=O)C(F)C2CCC2)CC1 N1(C(C2N(C)C(=O)CCC2)=O)CC(F)(F)CC1(C)CNC(=O)CC1CC1(C)C CCC(C)C(C(=O)NCCN(C)C(c1ncc(C)cc1OC)=O)NC(=O)OC N1(CC(=O)NC(CN(C(CN(CCOC)C)=O)C)C)CC2CCC1C2 CC1C(C(F)(F)F)CCN1C(=O)CSCC(=O)OC(C)(C)C S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC(NC(CCc2scc(C)c2)=O)C(C#N)C1 c1(OCC)ccc(N)c(C(N2CCCC2CNC(c2ccn(C3CC3)n2)=O)=O)c1 c1(C(N2CC(NC(c3c(OC)cccc3Br)=O)C(C)C2)=O)nc2ncccn2n1 C1(NC(c2c(CC)ccs2)=O)CCC12CN(C(c1csc(C(F)F)c1)=O)C2 C(=O)(C1=CS(=O)(=O)CCC1)N1C(CNC(c2cnc(SC)n2C)=O)CCC1 S(=O)(=O)(c1ccc(N2CC(C)SC(C)C2)c(F)c1)NCC(C)CN1CCOCC1 C1(CNC(=O)CC2(NC(c3cn(CCO)nn3)=O)CCC2)CC1C1CCCC1 [N-]=[N+]=NC1CCC(NC(=O)CC(C(F)(F)F)N2CCOCC2)CC1 CC1CCC(NC(=O)CCN2CCCC2=O)CN1C(=O)CNC(N)=O C12(O)CCN(CC1)C2=O.C1(C2(O)CCC2)(C(C)NC(=O)C(O)C2CC2)CC1 c1(CN2C(COC)CCCC2)c(C)nn(C2CCS(=O)(=O)C2)c1Cl C1(NC(c2nc(C)[nH]n2)=O)CC(=O)N(C2CN(C(=O)Cc3ccc(Cl)cc3)C2)C1 N1(C(CCC=CC(C)C)=O)CCC(NC(=O)COc2ccsc2)CC1C C(=O)(C1=CCC2CCC1N2C(c1ccc(N)cn1)=O)NCCCC(C)C C=CC(C)N=c1[nH]c(=N)[nH]c(=NCCC(=O)Nc2cccc(F)c2)[nH]1 c1(C(=O)NCC(C2CCC2)NC(C(C)O)=O)ccc(S(C)(=O)=O)cc1Br Cc1cnn(CC(=O)NC2CCC2NC(=O)Cn2ccc(C)n2)c1 C(=O)(C1NCCc2nc(C)ncc21)Nc1c(C(=O)NCC)cccn1 C1(N(C(C(C2CN(C(C3CC3CC(C)C)=O)C2)OC)=O)C)CCOC(C)(C)C1 C(C(CC1CC1)C(=O)N1CCOC(C(C)(C)C)C1)OC.C=C1CC2(C1)C(=O)NC2 c1(CCOC)cc(C)cc(F)c1.N12CCC(CN(C(CC)CC)C)(C1)NC2=O c1(-c2cn(C3CN(C(CNC=O)=O)C3)nn2)ccc(CCO)c(F)c1 O=C(C(F)CC1CCOCC1)NC1(CNC(C2CC2(Cl)Cl)=O)CC1 C1(NC(C2(CNC(=O)Cc3cocn3)CC=CC2)=O)CC2(CCC(O)C2)C1 C=CCC(CNC(c1scnc1C)=O)NC(=O)CC1CCCCO1 C(CC)(C(=O)NCC1CC1NC(c1c[nH]nc1F)=O)=CC c1(NC(c2n(CCOC)nnn2)CC2CCC2)ccc2cc(N(C)C)ccc2c1 C(=O)(C(C(C)(C)O)NC(C1CCCS1)=O)NCCC(CCC)O C1(CCNC(CC=C=C)=O)CCCN(C(=O)CCc2ccc(CC)cc2)C1 c1(SC)nccc(C(N2CCC(C)(CNC(=O)CCSC(F)(F)F)C2)=O)n1 N1(C(CCCC#N)=O)CCCCCC1C(=O)NCCn1cnnc1 C1(C(N2CC=C(CNC(CC3(C)CC3(F)Cl)=O)CC2)=O)CCCCC(=O)C1 CC1N(C(C2CC23CC(NC(=O)COCCN(C)C)C3)=O)CCC1(C)C C1(CNC(C(C=CC)O)=O)CCCCCN1C(c1sc(C(C)C)nc1C)=O c1(-c2onc(-c3nc(N4CCC4)ccc3)n2)ccc2n[nH]cc2n1.c1cscn1 c1(NC(=O)OCCCC)cc(C)c(NC(=O)NN(C)C)cc1C Cc1ccc(C2CN(C(C3CCN(C(=O)CC4CCCN4)CC3)=O)C2)cc1 Cc1cc(F)c(C(=O)N(CCC(=O)N2CC(O)CO2)C(C)C)cc1[N+](=O)[O-] N#Cc1ccsc1C(N1CC(NC(=O)CN2CCC(F)CC2)C(CO)C1)=O C1(c2nnnn2C)(Nc2cccc(CC(=O)OCC)c2)CCC2CCCC2C1 C1(NC(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(=O)CC2(N(C)C)CCCC2)CC1 c1(C(N2CCN(C(CC3(C=C)CC3)=O)CC2C)=O)cc2oc(Br)cc2s1 CN1CCOC2CN(C(C3(C)C=CCN3C(c3coc(C(N)=O)c3)=O)=O)CC12 c1(C(N(CC(CNC(COCCC=C)=O)C)C)=O)cccc(-c2nc(C)cs2)c1 c1(C(=O)NC(CC)CNC(=O)Cn2cccn2)ccnc2c(C)c(C)ccc12 c1(NC)ccc(C(=O)NC(C)CNC(=O)C(C)(C)CF)cc1F C1(C(=O)NCC(C)N(C(=O)CNC(=O)NCc2cccnc2)C)C2COCC12 C1(CC(=O)N(C)CC2CCCN2C(=O)CCn2cncn2)COC2(CCC2)CO1 C=CCC(CC)C(=O)NCC1(C(=O)NCc2cc(CC3CC3)n[nH]2)CCC1 C1(CNC(C(C)=C(C)C)=O)CCC(NC(c2cn(Cc3ccccc3)cn2)=O)C1 c1(OCC(N2CCN(C(C3(C)CC3)=O)CC2CCO)=O)ccc2c(c1)CCCC2 c1(C(=O)NC(C2CCOC2)CC)ccc2c(c1)NC(=O)CCS2 c1(C(=O)NC(CCOC)CNC(C2CN3CCC2CC3)=O)ccc(O)c(F)c1F C1(NC(COCCCC)=O)CCCOC12CCN(C(=O)C(C)(C#N)CC)CC2 c1(CCC(=O)N(C(C)CCNC(=O)CCC[N+](=O)[O-])C)c[nH]c2ccccc12 c1(C(=O)NCC(C(C)C)NC(c2c(C)cns2)=O)ccc(S(C)=O)cc1 CC1CCCC1NC(=O)CCC1CC(CNC(=O)Cc2ccn(C)c2)C1 c1(NC(CC2CCN(C(c3n(C)c(C(F)(F)F)cc3)=O)C2)=O)cc(Br)cnc1O CCC(CC)C(=O)NCC(=O)N(C)Cc1cc(Cl)ccn1.C1C(=O)N(C)CCO1 c1(C(=O)N(Cc2ccccc2)Cc2nn[nH]c2Cl)cccc(Cl)c1 n1(C2C(C)C2)cnc2cc(NC(=O)Cc3cccc(C(F)(F)F)c3)[nH]c2c1=O c1(-c2cn(CCN(CCC(=O)OC)C(N)=O)nn2)ccc(-c2cncnc2)cc1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(C2CC2NC(c2cscc2C)=O)CC1 N1(C(c2cnc(OC)nc2C)=O)CC2(COC(CNC(=O)C(C(C)C)SC)C2)C1 c1(NCc2c(OC)cnc(F)c2)ccc(C2=CCSCC2)cc1C c1(C(N(C(C)CNC(C2(n3ccnn3)CC2)=O)C)=O)cc2c(F)c(F)ccc2[nH]1 C(CC(CC)C(=O)N1CCC(F)(CNC(c2cccc(OC(F)F)c2)=O)C1)=CC c1(C(=O)NCC(CC)NC(c2nn(C)cc2Cl)=O)cccc(C#N)c1C CC1CN(C(=O)CCc2ccc(C3CCC3)cc2)CC1CNC(=O)CCF N1(CC(N2C(C3(NC(=O)C=CCF)CC3)CCC2)=O)C(=O)CNC1=O c1(NC(C(=O)NCCOC)CC2CC2)cc(NC(=O)CC2CC(F)C2)on1 C1(N2C(C)CCCC2)CCC2(CC1)CN(C(C1(c3ccc(O)cc3)CCC1)=O)C2 c1(C(=O)OC)cccc(C(N2CCCC(C3CC(N)CCO3)C2)=O)n1 C1(NC(C(C(C)C)SCC)=O)CC2CCC1CC2NC(=O)Cc1csc(C)n1 N1(C(c2cnc(C(C)C)nc2)=O)CC2(CNC(C34COCC3C4)=O)CC1CCO2 N1(CC(N2C(CN(C(Cc3ccn(CC)n3)=O)CC)CCC2)=O)CCN(C)CC1 C1(CCNC(c2c(C)coc2C(C)C)=O)CC(F)(F)CN1C(=O)Cn1cncn1 c1(OC)cncnc1C(=O)NCC(C1CCOC1)NC(c1nncs1)=O C1(CC(=O)N(C(CCCC)C)C)CN(C(C2(CC)CC2)=O)CCO1 c1(C(=O)NC(C2CCN(C(=O)C(C)n3cnnn3)C2)C)cccc2c1CC(=O)N2 C1(NC(c2ccc(CC)o2)=O)(CF)CCN(C(c2c[nH]c(=O)cn2)=O)C1 C(=O)(CCS(C)(=O)=O)NC(C(=O)NC(C=C)C1CCC1)Cc1cc[nH]n1 c1(C(=O)NC(CNC(C(CC)CC2CCCC2)=O)C(C)C)cc(N)cc(F)c1 c1(C(=O)NC2(C)CCN(C(C3(CC=C)CC3)=O)C2)ccc(Br)nc1O c1(CC(=O)NC2C(NC(=O)C=Cc3cc[nH]n3)C2)ccc2ccccc2c1 c1(C(N(CC(C)NC(c2cc(C)cc(F)c2N)=O)C)=O)cc2c(s1)CC(C)(C)C2 CC1(C)OCC2CC12C(=O)NCC(C1CCCC1)NC(c1nocc1Cl)=O c1(C(=O)NCCC(=C)CNC(C2(CO)CC2)=O)cc(C(C)C)ncc1Br CCCC(C(=O)NCC(C)NC(=O)C(C)(COC)OC)OC c1(C(=O)NC2CC(CC(C)C)OCC2)cc(S(C)(=O)=O)ccc1F CC1(C(=O)NC2CCCC2NC(=O)C(=O)NCC(F)(F)F)CCn2ccnc21 CC1(C(=O)NC2CCCC2NC(C2(C3CCCO3)CC2)=O)CC1(F)F c1(N(C2N(C(C(CCC)C)=O)CCCC2)C)cc(C(F)(F)F)nc2ncnn12 c1(C(N2CCN(C(C#CC3(CC)CC3)=O)C(C)CC2)=O)ccc2oc(=O)oc2c1 N1(C(c2c(C)nccc2)=O)CCCN(C(=O)C(F)CC2CCCCC2)CC1C C(=O)(C(=O)N=c1ccn(Cc2cccc(Cl)c2Cl)c(O)n1)OC.c1(C=O)nccs1 CC1C(NC(c2cc3c(F)cccc3[nH]2)=O)CC2CCC1N2C(=O)C1=CCCS1 c1(CC(=O)N(C2CC(C(=O)NC34CSCC3C4)C2)C)cccc2cn[nH]c12 Cc1oc2ncnc(O)c2c1C(N1CCC(NC(=O)CC2(C)CC2F)CC1)=O C=CCC(CC)C(=O)NC(C)(C)CCCNC(c1cnn(-c2ccccc2)c1)=O C1(Sc2n(C)ncc2)COCCC1C1CC1.C1C(=O)NN1C(=O)OC(C)(C)C CCC(C(=O)NCCC1CC(NC(=O)CCC2CCCN2C)C1)C(C)(C)CC N1(C(c2cc(OC)ncn2)=O)CCCC2(CCC2NC(=O)C(F)C(F)(F)F)C1 Cc1[nH]nc(C(N2CCC3(NC(C4C=CCC4)=O)CCCC23)=O)c1[N+](=O)[O-] C12(CNC(COCC)=O)CC(NC(=O)C(C)NS(C)(=O)=O)(CO1)C2 CC(=O)CCCCCCC(=O)N1CCC(C)(NC(=O)C2=CS(=O)(=O)CCC2)CC1 C(=O)(CCC(=O)NCC1CCCCC1NC(=O)CSCC(=O)OC)NC C1(C)(C(=O)NC(CNC(C(N2CCOCC2)C)=O)C)CCCS1(=O)=O c1(C(N2CCC(OC)C2)C(=O)NC2CCCCC2)ccc(C)c(C)c1F CCC(CN(C)C)C(=O)N1CC(CCC=C)(C(=O)Nc2cscc2C)C1 C(=O)(CCC(C)(C)F)NC(C1(O)CCN(C(C2CCC(C)O2)=O)C1)C N1(C(c2cscn2)COC)C(=O)NC(c2cccc(F)c2)C1=O c1(NC)ccc(C(=O)NC(CC2CCC2)C(=O)NCc2nnnn2C)cc1 Cc1oc(-c2cccs2)nc1C(=O)NCC1(F)CC(NC(=O)C=C2CCC2)C1 c1(CNC(CC(C)C)=O)cnn(C)c1C(N1CCOCC1CC1(C)CC1)=O c1(C(N(C2CCCC2)CCNC(C=Cc2ncc(C)[nH]2)=O)=O)ccc(O)c(F)c1F C1(C)(CCC(=O)NCCCCC2C(C)C2)CCCN1C(C1CCCCCC1)=O N1(C(c2cc(C(CC)CC)no2)=O)CC2(CCN(C(C3(F)CCOC3)=O)C2)C1 c1(CNC(Cn2cc(CN(C(C(=O)OC)C)C)nn2)=O)cc2cc(C)ccc2s1 N1(C(c2c(CC)cco2)=O)CCCCC1CC(=O)NCCc1ncccc1F C1(C(C)=O)Cc2c[nH]nc2CN1C(c1ccc(OC)cc1OCC(F)(F)F)=O C1(C(=O)NCCCC2(CNC(C(C)OC3COC3)=O)CCCC2)CCCC12CC2 c1(C(=O)NCC(CO)NC(c2cc[nH]c2)=O)cc(Br)n[nH]1 c1(C(=O)NCC(C)(CO)NC(c2cccs2)=O)cccc(-n2ccnc2O)c1 O=C(C(O)CC(F)(F)F)NCC12CCC(CC1)N2C(=O)CC1CCCO1 C1(C(N(C(CNC(c2c[nH]c(=NC)o2)=O)C)C)=O)CC2C=CCC(C1)C2 COn1cnc(C)c1C(=O)NC1CCCCC1CC(N1CC(O)(CN(C)C)C1)=O Cc1cc(F)ccc1NC(=O)C(N1CCOCC1c1nc[nH]n1)c1ccon1 c1(CC)cc(=NC(C)c2cc(Br)ccc2F)[nH]c(N2CCOCC2)n1 CC(Cc1ccncc1)C(=O)NC1CC(CCNC(c2[nH]ncc2Cl)=O)C1 C(CN=C(NCCC1(C)CC1(F)F)NC(C)C1CC1)c1cccc(OC)n1 c1(CC(=O)NCC2N(C(c3c(C)csc3)=O)CCC2)ccccc1I C1(CNC(C2C(C)CC=CC2)=O)CN(C(=O)CCCC#N)C2CCN1C2 c1(OC)ccc(Cl)c(C(=O)NC2CC(CNC(c3ccnn3C)=O)C2(C)C)c1 N1(C(CCSCCCC)=O)CC=CC(NC(=O)CC2CNC(=O)O2)C1 C1(NC(C2(C(=O)NC)CC2)=O)CCCC2CN(C(c3conc3CC)=O)CCC12 N1(C(c2c[nH]c(=NC)o2)=O)CCC(CNC(=O)C(C)CS(C)(=O)=O)C(F)(F)C1 CC(C(=O)NC1CN(C(C2CC(F)(CO)C2)=O)CC(C)(C)C1)C(C)S(C)(=O)=O Cc1cccc(C)c1C(N1CCC(CCC(=O)NC2CC(O)C2)C1)=O N1(C(=O)Nc2cccc(O)n2)CCCN(C(c2cnc(C(F)(F)F)cn2)=O)CC1 c1(OC)ccc(C(=O)OC(N2CCN(CCOC3CC3)CC2)=O)c(N)c1 c12cccc(F)c1-c1ccc(nc1)N2C1CCCC1.n1(CC(=O)OC)nc(C)cc1C C1(C(=O)NC(C(C)C)C)CC(NC(=O)OC(C)(C)C)CN1C c1(C(=O)NC2CC(O)(CNC(C(C)C#N)=O)C2)ccc(OCCF)cn1 c1(-c2scc(C(N3CCN(c4nccs4)CC3)=O)c2)cccc(C(F)(F)F)c1 c1(CS(=O)(=O)NC(c2cccc(C(=O)OC)n2)=O)c(C)cccc1C CCC(CC)(CC)C(=O)NCC1CC(C)CCN1C(=O)CS(C)(=O)=O c1(OC)cccc(C)c1C(N1CCC(c2ccccc2)(NC(=O)COCCF)C1)=O N1(C(C(C)OC)=O)CC(C)(C)OCC1CNC(=O)CCSc1cccc(Cl)c1 c1(OC)ncc(CN2CCC(CC(=O)Nc3ncccc3CO)C2)cc1Br Cc1cnn2cc(C(=O)NCCCN(CCC(C)(C)C)C)cnc12 C1(C(N2CC(OC)C(F)C2)=O)CC2(CC2)CN1Cc1ccc(OC(F)F)nc1 C(C)(C)(CCCF)NC(C(CN(C)C)NC(C1CC(=O)C1)=O)=O c1(C(C(=O)NCC(CN(C(c2c(CC)scc2)=O)C)O)OC)ccccc1OC c1(C(=O)NC(CN(C(=O)C2=CCCSC2)CC)C)cc(C(C)C)n(C)c1C c1(C(=O)NC(c2nc(Oc3cc(CCC)no3)sc2)=O)ccc(C)cc1C C1(CNC(C=CCCC)=O)CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1 CC1CC2CN(C(c3cnc(C(N)=O)s3)=O)CC2N1C(=O)COCc1nc[nH]n1 N1(C(c2c(OC)ccs2)=O)CC2CCC(CNC(=O)CC3CCCC3O)C2C1 Cc1nc(-c2ccco2)sc1C(C)OC(=O)CCc1ccsc1 C1(NC(c2c(C)coc2)=O)CC2(C1)CC(NC(c1ccn(C)n1)=O)C2 O=C(CS(=O)(=O)C1CC1)NCC1CCC(CNC(=O)COCC2CCOC2)C1 c1(C(=O)NCCC(=O)NC2CCN(C(=O)C3CC3)C2)ccc2c(c1)C(=O)OCC2 C=CCCCCCC(=O)N1CCC(F)(CNC(C2(C(C)(C)C)CCCC2)=O)CC1 C=CCCCCC(=O)NC(C)(CNC(c1ccc(C(C)C)cn1)=O)CO C1(C(=O)NC2C(CNC(c3cccc(N)c3O)=O)C2)Cc2cc(F)cc(F)c2O1 Cc1nn(-c2ccc(F)cc2)c(C)c1C(=O)N(CCCN(C)C)C C#CC1CCCCN1C(c1cccnc1CNC(=O)C(C1CC1)OC)=O c1(-c2cn(C3CCN(C(c4n(CC)ccc4)=O)C3)nn2)cc(C)cc(C)c1 CC(=O)C(C)CC(C)C(=O)NC1CC2C1CCN2C(=O)CCCN(C)C C=CC1CC1C(=O)NCC1(CC(=O)OCC)CC1 c1(C(N2C(CNC(CC=C(C)C)=O)COCC2)=O)cnc2n1C(C)CCC2 N1(C(C(F)=CC)=O)CCN(C(=O)Cc2sc(C)cc2C)C2CCCCC12 C1(C(=O)OC)CCC(=O)N1C(=O)C(CN1CCCCCC1)Oc1cccc(F)c1 CN1CCC(C(=O)NC2CCC(F)(CNC(=O)CC(=O)NCC3CC3)C2)CC1=O C1(C(=O)NC(C)CC(=O)O)C2CN(C(=O)CN3CC4CC4C3)CC12 c1(CC)ccoc1C(=O)NCC(C)CN(C)C(C1CC(OC(F)(F)F)C1)=O c1(CNC(C2CCC(C)C2)=O)ccc(CC(C)NC(c2cccs2)=O)cc1 c1(C(C)C)cccc(F)c1C(N1CCN(C(=O)Cc2nn(C)cc2Cl)CC1C)=O C(=O)(CCCN=[N+]=[N-])NCCCN(C(c1cccc(CC)n1)=O)CC n1(C(C)C)ncnc1C(=O)NC(C1CCCC1)CNC(=O)CCC1CCC(=O)N1 c1(-c2c(OC)scc2)ccc2nnc(C(N3CCC(O)C3)=O)n2c1 C(=O)(C1=CCC(C)(C)CC1)NC1C(CNC(c2c(C)cc(Cl)cc2)=O)CC1 N1(C(C2(O)CCN(C(c3ccc(OC)c(Cl)c3)=O)C2)=O)CCCCC(C)(F)C1 C1(OC)CCCCC1C(=O)N(C)CCN(C(=O)C(F)(F)c1cccnc1)C c1(C(=O)NC(CNC(C2C(C=C(C)C)C2(C)C)=O)(C)C)ccc(S(C)(=O)=O)s1 C1(C(C(=O)OC)NCCN2CCCC(C(=O)OC)C2)CCN(C(=O)OC)CC1 O=C1COc2ccc(S(=O)(=O)Oc3cnn(N4CCOCC4)c3)cc2N1 Cc1ccc2c(c1)CCN2C(C1CCC(F)CN1C)=O N1(C(C2C(CC)CCCC2)=O)CC(CNC(=O)C(C)(C)C(C)C)C2(CCC2)C1 Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CC(C)(C)c2cccs2)nc1C c1(C(=O)NCC2(NC(CC(CC)OC)=O)CCC2)cccn2cncc12 C1(C(=O)NC2(CCC)CC2)C=CCN1C(=O)C=CCN1CCOCC1 C(=O)(C1=C(C)CC1)NC1(C(=O)NC(c2cnn(C)c2)CC)CC1C C1(CNC(c2cc(C)c(Cl)s2)c2nnnn2C(C)(C)C)CCCC(C)(C)C1 c1(C(=O)NCC(C(C)C)NC(C(NOC)=O)=O)cc(C)cc(F)c1 c1(C(=O)NC(CNC(C2OCCN(C)C2)=O)C2CC2)cc(F)cc(F)c1 c1(C(N(C2CCCN(C(=O)CN3CCCCCC3)C2)C)=O)ncccc1Cl N1(C(C2(CC=C)CCN(C(c3cnn(C(C)C)c3)=O)C2)=O)CCC(=O)N(C)CC1 C(=O)(C(C)SC(F)(F)F)OCC(F)(F)F.C(CCCCCCCO)N(CC)CC C12(CNC(C3C(CCC)C3)=O)CCC(CNC(=O)CCCS(C)(=O)=O)(CC1)CO2 C1(CC)CC(C(=O)NCCCc2ccsc2)CCN1C(=O)CC1CC(C)(C)CO1 C#CC1CCCC(NC(=O)CCCOc2cc(Cl)cc(Cl)c2)C1 C(=O)(C(O)C(C)CC)NCC(CC)NC(C1(c2cccnc2)CCC1)=O N1(C(CC(CC(=O)OC)C)=O)CCC2(CC1)CCN(C(=O)C(C)S(C)(=O)=O)C2 c1(C(N(CCCNC(C(C(CC)O)C)=O)C2CC2)=O)ncccc1N=[N+]=[N-] C(=O)(C1=C(Cl)CCOC1)N(C)CC1COCCN1C(C1CNC(=O)N1C)=O C1(CNOC)CC12CCC2.c1(SCC)cc(C2CC2)no1.C1(C=O)(CNC=O)CC1 C(CC(C)(C)O)NC(C(C)(C)C)=O.CC1C=CC(=O)N1C1CC1 Cc1cc(C)c(C(=O)NCC(CC(C)C)NC(=O)Cc2ncc(C)[nH]2)cn1 N1(C(C2N(C)CCN(C)C2)=O)CCC2CC2(C(N2CCCCCC2)=O)CC1 N1(Cc2ncn(C)c2)CCC2(CC1)CN(C(C1(C)C=CCC1)=O)C2 N1(C(C(=O)Nc2c(C)cccc2C)=O)CCN(Cc2cn(C)nc2Cl)C(C)C1C N1(C(CC)=O)CCC2CCC12CN1c2c(I)c(n(C)n2)C1.C1=CCCCC1.NC c1(C2(C(=O)NC3(C(F)F)CCCNC3)CC(O)C2)ccc(Cl)cc1 N1(C(C(C)NC(c2cc(I)ccc2N(C)C)=O)=O)Cc2ccccc2C1 CC(c1ccccc1Cl)=CC(=O)NC(C1CCCC1)CNC(=O)C#CC(C)C c1(CC)ccc(Cl)c(C(=O)NC2CC2CNC(C2CCOC2=O)=O)c1 CCCCC(CNC(C1(SC)CC1)=O)NC(C1CCS(=O)(=O)C1)=O C=CCC(CC)C(=O)NC1(CO)CCN(C(=O)C(C)(C)c2cscc2Cl)CC1 N1(C(c2c(CC)[nH]nc2Cl)=O)CC2CCC(NC(=O)CNC(N)=O)(C2)C1 C1(C(=O)NCC2ON=C(CC)C2)CN(C(C2CCOC2)=O)C2(CCC2)C1 c1(C(N2C(CN(C(=O)C(c3cncn3C)O)C)CCC2)=O)cccc(F)c1 N1(CC)CCc2cc(-c3ccnc(NC(=O)NC(C)CF)c3)ccc21 C(CC(CS(C)(=O)=O)N(C=O)Cc1ccccc1)OC.c12cccnc1OCC2=O C1(CNC(CCCC(=C)C)=O)CCC(C)(C)CN1C(=O)CSc1ccccc1 c1(C(=O)NC(C(C)C)C(C)NC(c2c[nH]cc2C2CC2)=O)cc2sccc2n1C CC1CC(C(=O)NCC2CCC(NC(=O)COc3cccc(F)c3)CC2)C1(C)C Cc1noc(C)c1CC(C)NC(=O)Cn1nnnc1C.C1(=O)CN1CC(=O)O c1(C(=O)OC)cnc2c(c1)c(C)nn2C(C1(C)CCC1)C.C1(CN)C(C)(C)C1(C)C c1(-n2cc(CN3CC(O)CC(C4(C=C)CC4)C3)nn2)ccnc(P(C)(C)=O)c1 Cc1nc(C)c(-c2nnc(SC(c3ccccc3)C(=O)N(C)C)n2C)s1 N1(C(C(C)(C)SC)=O)CCC2(CC1)CCN(c1ncc(O)cn1)C2 c1(C(=O)NCC2CN(C(C(CC)C)=O)CC2O)c(C)nn2cc[nH]c(=O)c12 c1(OC)c(CC(N2CCC(O)C(NC(C3CC3C)=O)C2)=O)cccc1F N1(C(c2ccc(N)cc2O)=O)CCC(C2CC2)(NC(=O)CSCc2ncc[nH]2)C1 N1(C(c2c(C#N)cccc2)=O)Cc2[nH]nc(C(=O)Nc3c(C#N)cccc3Cl)c2C1 C#CCCCC(C)C(=O)NCC1(NC(=O)CCN2CCCCCC2)CC1 c12cc(c(C)o1)C(=O)C2.C1(C)CCCCC1n1cc(C2CN(C(=O)C(CC)CO)C2)nn1.C=CC C1(CN(C)C(c2snc(Cl)c2Cl)=O)CCCN(C(=O)C2=CCCO2)C1 N1(C(Cc2cc(C)[nH]n2)=O)CC2CCCC2(C(=O)NC(c2cccc(F)c2)C)C1 Nc1cnc(N2CCC(NCc3cccc(C(F)(F)F)c3)C2)cn1 C1(NC(C2CC(F)C2)=O)CCCCN(C(=O)Cc2cccnc2O)CC1 c1(OC)ccc(SCCC(=O)NCC2CCCN(C(=O)CN(C)C)C2)cc1 C1(C(=O)NC(C(=O)NC(CC(=O)OCC)C2CC2)C)C2CCCCC12 N1(C(C(C)(CO)OC)=O)CCOC(C)(CNC(=O)CSC)C1 C1(C(=O)NC2CCSC2)CCCCCN1C(c1n[nH]c2c1CCC2)=O C1(C(N2C(CNC(c3ccnc(C)c3N)=O)CC2)=O)Cc2ccc(F)cc2O1 Cc1c(Cl)nc[nH]c1=NCC(O)CNC(c1cc2cccnc2s1)=O C1(C(N2CCC(=CCNC(C3CCCN(C)C3)=O)CC2)=O)CN=C2N=CNN2C1 N1(C(c2cc(C)no2)=O)CCC(CCNC(c2ccc(O)c(N)n2)=O)CC1C Cc1nn(C)c2c(N(C)Cc3ccncc3)nc(N3CCC(C4CC4)C3)nc12 CC1(C(N2CC3CC3(CNC(c3cccnc3Cl)=O)C2)=O)CCCOC1 c1(C(=O)NCC2N(C(CC(C=C)(C)C)=O)CC(F)(F)C2)cnc2c(c1)CCCC2 N1(C(c2c(C)n[nH]c2)=O)CCOC(C(C)NC(=O)C(F)CC2CCCCC2)C1 C12(C(N(CC(=O)NC(C)(C)C)C)=O)CC(CO)(CN1C(C1CC3(CC3)C1)=O)C2 c1(C(N2CCC(NC(C3(OC)CC3)=O)CC2C2CC2)=O)ccc2c(n1)CCC2=O c1(N2CC(C(C)C)NCC2)cc(NC2CCC(C)(C)OC2)nc(C(C)C)n1 CN(C1CCc2ccc(Cl)cc21)C(=O)C(=O)NCCc1ccc2c(c1O)OCO2 C12CCN(CC1F)C(=O)N2.c1(C(c2ccnn2C)C)coc(OCC(F)(F)F)n1 c1(OCC(=O)NC(C)CCCNC(C2(Cc3ccco3)CC2)=O)ccc(Cl)cc1 N1(C(c2cn(CCNC(CSCC#C)=O)nn2)=O)Cc2ccc(O)cc2C1 c1(SC)ncc(CNC(c2nnnn2CC2CC2)c2cscn2)s1 c1(SC(F)F)cc(C(F)(F)F)nc(C2CCOCC2)n1.C1CCCC2CCCC2N1 c1(C(=O)NC2CC(NC(CN3C(C)CC3)=O)C2)cnc(O)cc1C(F)(F)F C1(NC(c2nn(C)c(F)c2)=O)CC2CN(C(c3cnn4cc[nH]c34)=O)CC12 c1(C(=O)NCCCC(=O)NCc2nc(C)sc2C)ccc(C)c(C#N)c1 c1(C(N(C2CN(C(C3CCC(C)(C)C3)=O)C2)C)=O)nc2ccccc2[nH]1 C1(CNC(C2CN(C(C)C)C2)=O)CCCCN(C(=O)CC(C)O)C1 N1(C(CN(C(C(C)SC(C)C)=O)CC2CC2)=O)CCC2(CCC2)C1 c1(C(=O)NCc2c(CNC(CC(=C=C)C)=O)nccc2)nnn2c1C(=O)NCC2 c1(C(=O)NC(C(C)(C)C)CNC(C2CCCC23CCC3)=O)cccc(C#N)c1F c1(OC)ccc(C=CC(=O)NC2(CF)CCN(C(C3(C#N)CC3)=O)C2)cc1F c1(OC)cccc2c(CCNC(c3c(F)cc(I)cc3F)=O)c[nH]c12 N1(C(C(CC)N(C(N)=O)C)=O)CC2CC1CN2C(=O)C(c1cncn1C)O CC1CCN(C(c2cn3c(n2)SCC3)=O)CC1CNC(=O)C1=COCCO1 CC1CCC(C)(C(=O)N(CC(C)N(C(=O)Cn2ncnn2)C)C)CC1 C(=O)(CC1=CCN(C(C2CC(F)(F)C2)=O)CC1)NC(C#C)C(C)C CC(CCS(C)=O)N(C(=O)C(=O)C1CC1)C CCC(C(=O)NCC(C(C)C)NC(c1cc(O)cs1)=O)Sc1ccccc1 c1(C(=O)NCC(CC)NC(=O)Cn2nnc(C)n2)coc(-c2ccccn2)n1 C1(C(=O)NC(C2CN(C(C3CN(C4CCOCC4)C3)=O)C2)C)COC(=O)C1 C1(NC(c2cc(CO)[nH]n2)=O)CN(C(=O)Cn2ncc(Br)n2)C2CC12 c1(CC)ccccc1-n1nnnc1C(C1(C(F)(F)F)CC(O)C1)Nc1ccsc1 S(=O)(=O)(c1cc(C(=O)NC2COCCN(C(=O)CCN)C2)ccc1OC)NCC C1(CNC(CCC#N)=O)CCCCC1NC(c1nncn1-c1ccccc1)=O C=C1CCN(C(c2cc(OC)cc(C#N)c2)=O)C(C(=O)NC)C1 c1(C(=O)NCCCCNC(C2C(C)(C(=O)OCC)C2)=O)cnc(C2CCC2)s1 O=C(C1=NOC2(CCN(Cc3cnco3)C2)C1)Nc1ccc(F)c(C(F)F)c1 c1(C(=O)NCC(CC)C#N)cc(C)ccc1NC1CCCCC1 C1(NC(=O)C(O)CCNC(C2CCC(=O)NC2)=O)CCCCC12CC2 C(CN=c1[nH]c2cccc(C)c2s1)C(NNC(c1cc(OC)c(OC)c(OC)c1)=O)=O C(=O)(CCCC(C)C)NCC1(CO)CCN(C(c2c(C)nc(C3CC3)o2)=O)C1 c1(CN2CC(C(N(c3oncc3C#N)C)=O)SCC2)c(O)cccc1Cl C1(CC(=O)OC)(CC)COCCN1C(=O)CC(N)CN(C)C Cc1nc2cc(C(=O)NCCC3CCCNCC3)c(F)cc2[nH]1 c1(CN2C(C(N(C)Cc3ccccc3)=O)C=CC2)cc(F)c(O)cc1F CCCCC(O)C(=O)NCC1(NC(=O)CCC2OCCO2)CC(OC)C1 N1(C(C(=O)NCC)=O)CCCC(NC(c2oc(CC(C)C)nc2C)=O)C(F)C1 Cc1c(C(N2CCC(CN(C)C(C3CCC(N(C)C)CC3)=O)C2)=O)cncc1N c1(C(N2CCC(C(=O)OC(C)(C)C)C2)=O)cc(Cl)nc2n[nH]cc12 CC1CCC(C(=O)NC2(C)CCCN(C(c3cc(O)cs3)=O)C2)CC1C CC1CCN(C(=NCCC2(C)CC2(F)F)NCCF)C1 c1(CC)ccc(CCC(=O)NCCCOCCN(C)C(C2CC2C(N)=O)=O)cc1 C1(NC(C(C=C=C)C)=O)CCCN(C(=O)OC(C)(C)C)CC1 N1(C(C(C=C)CC)=O)CCN(C(C2CCCN2CCC)=O)C(CCC)C1 c1(CN(C)C)cc(NC(=O)C(N2CCN(c3ccncc3Cl)CC2)=O)nn1C c1(OC)cccnc1C(=O)NC1CN(C(c2cc(C3(C)COC3)no2)=O)C1 C1(CNC(c2ccc(F)cc2O)=O)CC2CCCC2N1C(=O)CCC1CC1(F)F O(NC(=O)C(O)C(CCC)NC(C1(C#N)CCOC1)=O)CCCC=C c1(CC)cccc(C)c1C(=O)NCC1(F)CCCN(C(C2ON=C(C)C2C)=O)C1 c1(C(=O)NCCN(C(=O)CC2CCCOC2)C2CC2)cnc2ccccc2n1 c1(C(=O)NC2CN(C(C3C(OCC)C3)=O)CC2C)cc2ccoc2cc1F O=S(=O)(c1cccc(=NC2CCCc3sccc32)[nH]1)N1CCOCC1C1CC1 c1(OCC)ncc(C(=O)NC(C)CCCNC(=O)CC(C)SC)cn1 N(C(=NCCCF)NCC(C)OC)Cc1c(OC)nccc1 C1(CNC(C(CC=C)C)=O)CCC12CCN(C(=O)C(C)(C)F)CC2 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(Cn2cc(CCOC(C)=O)nn2)C1 N1(C(c2nc(C)oc2)=O)CC2CCCC2(NC(c2cccc3[nH]ccc23)=O)C1 c1(C(=O)NC2C(C(=O)Nc3c(C)csc3)OCC2)csc(C#N)c1 c1(C(N2CCCCCC2c2ccc(Cl)cc2)=O)cc(Br)c(F)cc1Cl c1(C(=O)NCC23C(CN(C(C(C(C)(C)C)O)=O)C2)CC3)cccc2ncsc12 N1(CC)CC(CNC(c2ccc(CNC(C3CCO3)=O)s2)=O)CC1=O c1(N2CCCC(N(C)C)C2)nc(=NCc2cccnc2)[nH]c2c1CCC2 c1(C(=O)OC)cc2c(s1)CCOC21CCN(N2CCCC(N3CCC3)C2C)CC1 C(CNC(=O)C(COC)N(C)C)(CC(C)C)NC(C1(CC#C)CCOC1)=O C(=O)(CCCCc1cnc[nH]1)N(C1CN(C(=O)C=C(Cl)Cl)C1)C c1(C(=O)NCC(C)NC(=O)Cc2cnc[nH]2)cccc2nc(O)n(C)c12 c1(CC)[nH]nc(C(=O)NC2CC(CCNC(=O)COCc3nc[nH]n3)C2)c1Cl C(C(F)(F)C(=O)N1CCC(F)(CNC(=O)CN2CCCC(N(C)C)C2)C1)N(C)C C(C(C)(C(C)C)NC(=O)C(=O)N(c1ccc(Br)cc1)CCOC)NC(C(CC)C)=O C(c1cnn(C)c1)=C(C(=O)NC1C(CNC(c2c(CC)noc2)=O)CCC1)C C(=O)(C(CNC(c1ccc(O)nc1)=O)C(C)(C)C)NC(c1ccccc1O)C c1(C(=O)NCC2N(C(C(CC)COC)=O)CCCC2)cc2c(nn1)CCC2 c1(CC)noc(C)c1CNC(=O)CCCN(C(C1C2CC3C(C2)C13)=O)C1CC1 C1(C)(CNC(C2(N(C(=O)CP(C)(C)=O)C)CC2)=O)CCC(=O)N1C C(=O)(CC(=O)NCCCNC(=O)C(C)COC)OCC N1(C(C(N2CCC(C)CC2)=O)=O)C2CCC1CC(NC(=O)C(C)(C)CC(C)(C)C)C2 N1(C(c2c(-n3cnnc3)ccc(C)c2)=O)CCc2nc(C)sc2C1 c1(C2N(C(CSCC(C)C)=O)C(C)(C)CC2)cccc(-c2nn[nH]n2)c1F C=C(C)CCCC(=O)N1CCN(C2CCN(C(=O)C(C)C3CCCO3)C2)CC1 N1(C(C2N(C(C3C(C)C3)=O)CCC2)=O)CCC2(CC1)CC(=O)N2 C(=O)(C(CCC1CC1)NC(C1CC1)=O)N(c1csc(Cl)n1)C(C)(C)CC1CCC1 O=C(CCCCCc1ccc(F)cc1)NC1CC(NC(=O)Cc2ccccn2)C1 c1(N(C)C)ccc(Cl)cc1-c1nc(-c2ccn(C)n2)nn1CC1CCCOC1 C1(CC(=O)NC(CC)CNC(C2(Br)CC2)=O)CCC1(F)F C1(NC(C2CCCCS2(=O)=O)=O)CC2CN(C(=O)CC3CCC4CC4C3)CC12 CCCCCC(C)(C)C(=O)N=CC=CCC1=CCN(C(=O)Cn2cccc2)CC1 C1(NC(C(NOC)=O)=O)CC2CCC1C(NC(C1CC3COCC3C1)=O)C2 C=CCCC(CC(C)C)C(=O)N1CCC(NC(C2(O)CC2)=O)C1C N1(C(C2N(C(CN(C3CC3)CC)=O)CC(=O)C2)=O)CCC(O)CC(C)(C)C1 Cc1ccc(NC(=O)COC(c2nccn2C)C)cc1Br C1(CNC(C2C(C)=C2)=O)CN(C(c2occ3c2CCC3)=O)CCC1(C)C c1(C(=O)NCCCNC(C(C(CC)CC)OC)=O)c(O)nnc2c1CCC2 C1(C(C)(C)C)(C(=O)NCC2(C(C)(C)O)CN(C(C3CC3C#N)=O)C2)CCCC1 c1(SC)nn(C)cc1C(=O)NC(C1CCN(C(C2OCCO2)=O)CC1)(C)C N1(C(C)=O)CCc2ccc(NC(=O)C(C)Oc3ccc(CO)cc3)cc21 C1(OC(C(c2cc(C)no2)(C)C)=O)CCC(F)(F)C1 C1(C(=O)NC(C)CC(C)NC(=O)Cn2cc(N)cn2)(CC)CCNC1=O C(=O)(C(C)(C)C(=O)N1CC(NC(=O)C=CCN2CCC2)C(CO)C1)OCC N1(C(C)=O)CCN(C(=O)NCc2ccc(N3CCCC(O)C3)cc2)C(C)C1 c1(NC(C2CC(NC(c3cc(Cl)sc3Cl)=O)C2)=O)c(Cl)ccc2cccnc12 C1(C(=O)NC2CCC(CNC(c3cc(C)oc3C)=O)C2)CC2CC2CC1C Cc1ccc(C)c(SCC(=O)NCCCCN(C)C(c2ccc(CSC)o2)=O)c1 c1(C(C)=O)cn(C)nc1C(=O)NC(C)CC(C)NC(C1CCCS1)=O O(NC(=O)C(C)C(C)NC(c1coc(CC)n1)=O)CC C(C)(C)(C(C)CC(=O)NC1CN(C)CC1(F)F)NC(CCSCC)=O c1(C(=O)NC(CN(C(=O)CCNC(C)=O)CC)C)csc2c(OC)cccc12 Cn1cnc(C(=O)NCC2CC(O)(CNC(c3ccc(CSC)s3)=O)C2)cc1=O C=CCC(C(=O)NC1CN(C(=O)C(F)OC)CC1SC)OC N1(C(C(n2ncc(C)c2)C)=O)CC2CCOC2(CNC(C2(N(C)C)CC2)=O)C1 N1(C(C2N(CC)CCC2)=O)CCN(C(c2cc(C(C)=O)cs2)=O)CC1C(C)(C)C Cc1noc2nc(C(C)C)cc(C(N3CCc4ccnc(O)c4C3)=O)c12 C(=O)(C1CCc2ccccc21)NCC(C)(C)NC(=O)C(F)=CC1CC1 n1(CCC)cc(C(=O)NC23CC(CNC(=O)C(c4cccnc4)C)(C2)C3)cn1 C(CCCCN=c1cc(C)c(S(=O)(=O)N2CCC(CN(C)C)CC2)c[nH]1)OC c1(CC(=O)NC2CC(NC(CCC3C(C)=NOC3=O)=O)C2)c(C)nc(C)nc1O C1(CN(C(CC2(COC)CCCC2)=O)C)CCN(C(=O)C(C)NC=O)CC1 CC(C)C(C)(C)C(=O)NC12CCC(CNC(C34CC5CC3C4C5O)=O)(C1)OC2 c1(C(N(CC(O)CN(C)C(C2(C(F)(F)F)CCCC2)=O)C)=O)cc(C#N)ccn1 C(=O)(CS(=O)(=O)NC(C)(C)C)NCC(C)(C1CCC1)NC(C(C=CCCC)O)=O c1(OC(C)C)c[nH]nc1C(=O)NCCOC1CC(C(=O)NCCc2cscn2)C1 C1(Cn2cc(C(CCC)NC(C3(CCN(C)C)CC3)=O)nn2)CCCS1(=O)=O C(C(O)C(C)(C)C)NC(C(=O)N(C=O)C(C)C)C.CO C1(C(=O)NC2(CNC(C(C)O)=O)CC2)CCCC(F)C1 c1(C(=O)NC2C3CN(C(c4cc(C)ncc4)=O)C2CC3)cccc2cc[nH]c12 N1(C2CCN(C(c3c(SC)ccs3)=O)C2)CCC(NC(=O)C2=CCC2)CC1 CN1N=CC(CC(=O)N(C2CCCC2)Cc2ccccc2)C1=O C1(OC)CC(C(=O)NC2CCC(SC)C2)N(C(=O)CCC2CCC2)C1 C#CCCCCC(=O)N1CC(=O)NCC1C(N1CCC(O)(C#C)C1)=O C1(C)(CNC(C(C)OC2CCCC2)=O)CCN(C(=O)CSC2CCCCO2)CC1 C1(NC(C2CCN3CCOCC23)=O)CN(C(c2cncs2)=O)C2CCCCC12 c1(C(N(C)CC2CN(C(C3(C=C)CCCCC3)=O)C2)=O)c(Cl)oc2ccccc12 N1(C(C2(C#C)CN(C(=O)C(C)=C3CCCC3)C2)=O)CC(C)C(C)C1C C12(CNC(C3(C)CCC(=O)N3)=O)CN(NC(C=CC(=O)N(C)C)=O)CC1CCO2 Cc1ccc(C=CC(=O)NC(C)(C)CNC(c2cc(O)nc(C(F)F)n2)=O)cn1 c1(N(C)CC2CCC(CC)O2)nnc(-c2ccccc2C)n1CC1CCOC1 C(=O)(CC(F)(F)F)NCC(=O)N(CCNC(C1C(C)CC1)=O)CC1CC1 N1(C(C(C)(C)c2cnsc2)=O)CC2CC(O)C1C2NC(C1CCCS1)=O C(=O)(CSC)NCCN(C(=O)CN(C)CC)CCC.CCO N1(C(CC(=O)OCC)=O)CCN(C(c2cnnc(O)c2)=O)C(CC(F)F)C1 Cc1ccc(C(=O)NCCC2CN(C(=O)COC3CCOC3)CC(C)O2)c(Cl)c1 c1(-n2cc(CSCC(=O)Nc3c(C)ccnc3C)nn2)sccc1S(N)(=O)=O N1(C(C(C)SCC)=O)CCN(C(=O)C(O)C2CCCC2)C(CC(F)F)C1 CCCC(O)(CCC)CC(=O)N1CC(O)(C2(CNC(=O)CCNC(N)=O)CC2)C1 Cc1ccc2scc(C(=O)NC3CCN(C(=O)CCCC(C)(C)C)CC3F)c2c1 C1(F)(CNC(C2(CC)CC2(F)F)=O)CCCN(C(c2ncccc2O)=O)C1 c1(CC(=O)NCC(CN(C(C(C)O)=O)C)O)ccc(Sc2ccccc2Cl)cc1 C(=O)(C1CCSc2ccccc21)Nc1c(C#N)cc(Br)cn1 c1(C(N(C(C)CCNC(C2(C3CCCCO3)CCC2)=O)C)=O)ccc(Cl)cc1F Cc1cc(C(=O)NCc2ncccc2C(N2CCCC(C)CC2)=O)ccc1O C(C)(C)(CC(=O)N1CC(O)(CN(C(=O)C(c2ccccc2F)(C)C)C)C1)OC c1(NC(C2CCCCN(c3cc(Cl)c(O)nn3)C2)=O)cccc(C2CC2)c1F CCCC(C)(O)C(=O)N(C1CCC(CNC(c2ccc(C)n2C)=O)CC1)C C1(CCC)CN(C(C2CC3(CCCC3)C2)=O)CCN1C(N1CCCC1C)=O c1(C(=O)NCC(CCOC)NC(c2ccc(C)o2)=O)ccc2c(c1)OCCC2 c1(OCC(C)(C)NC(C2CCC(CN)C2)=O)ccc(F)cc1 c1(CN2C(C(=O)Nc3cccc(NC(C)=O)c3)CCC2)cc(Br)ccc1O N1(C(CC2C(OCC)CC2)=O)CCC(OC2CN(N3CCNC3=O)C2)CC1 C(N=c1[nH]c2cccnc2s1)C1CCN(C(c2c(C)n(C(C)C)nn2)=O)C1 c1(CN=c2cc(NCC(CC=C)(C)CO)nc[nH]2)cnc2ccccc2n1 c1(CC)n[nH]c(=NCC2CN(C(c3ccc(OC(F)F)cc3)=O)C2)s1 Cc1cc(Cl)ncc1NC(C1(CCNC(=O)CC2OCCC2(C)C)CCCC1)=O C1(C)(NC(C2(CF)CCN(C(CC(COC)NC(C)=O)=O)C2)=O)CCCCC1C N1(C(C2C(C)(C)CC2)=O)CCOCC(NC(=O)CCNC(C2CCCCC2)=O)C1 CCC(C)C(C)C(=O)NCC1CN(C(=O)C(=O)C(C)(C)C)CCC1C c1(CC)ccc(C)c(C(N2CCC(C)(CCNC(C3CC(OC)C3)=O)C2)=O)c1 N1(c2c(-c3cn(Cc4ccccc4C)nc3)ncs2)CCCCC1SCC n1(C(COC)C)cc(C(=O)NCC(n2cc(-c3csc(C)c3)nn2)C)cn1 c1(C(=O)NCc2cc(N(S(C)(=O)=O)C)nn2C)ccc2ccoc2c1 N1(C(=O)Cc2ccsc2)CC(C2CN(C(=O)CC3CCSC3)C2)C1 c1(CNCC2N(C(C3CCC(F)(F)C3)=O)CCOC2)cnc2n1CCOC2 c1(C(=O)NCC2CC(Nc3nc(C)nc(=N)[nH]3)C2)cnc2[nH]c(O)nc2c1 N1(C(C(CSC)C)=O)CC(C(N2CCCOCC2)=O)C2(CCC2)C1 C1(NC(C)=O)C2CC3C(C2)C13C(=O)N(C(C)CN(C)C(=O)N(C)C)C CC1CCCC(C(=O)NC2(CC=CC(N(C)CP(C)(C)=O)=O)CCC2)CC1 N1(C(CCOC)=O)C(CNC(=O)C(C)(C)OC(C)C)CC2CC12 c1(C(=O)NCCC2CCCN(C(CC(COC)C)=O)C2)cn2cccnc2n1 n1(CC(=O)NCC2CCC(NC(CCCOCCC)=O)C2)cnc2ccccc12 c1(C(=O)NC2CCC(NC(C3N(C)CCCC3)=O)CC2)ccc(O)c(CO)c1 N1(C(CNc2c(C)nccc2)=O)CC2(CCN(C(c3cccs3)=O)CC2)C1 C1(NC(=O)C=CC(F)(F)F)CCC(O)CN(C(=O)C(F)CC2CCCC2)C1 N1(C(C2C(=C)CC2)=O)CCN(C(c2cccc3cncn23)=O)C2(CC2)C1 N1(C(CC(C)CF)=O)CC(NC(c2cncc(C(F)(F)F)n2)=O)CC(F)C1 c1(NC(C)CNC(c2cncc(Cl)n2)=O)ncnc2ccc([N+](=O)[O-])cc12 N1(C(c2cnccc2Cl)=O)CCC(N=c2[nH]c3cc(F)cc(F)c3o2)C1 N1(C(CNC(C)=O)=O)CC2CCC1CN2C(c1ccc(Br)c(F)c1N)=O CCC(CCOC)C(=O)NCC1(CNC(=O)CSC)CC1 C1(CC(=O)NCC2(F)CC(CNC(c3cc(C(F)F)no3)=O)C2)CCC2CC12 c1(CC)cc2c(N3CCN(C(C4CC4C4CC4C)=O)CC3C)ncnc2s1 c1(-c2onc(C)n2)ccc(C(=O)NC(C)C(C)NC(C2(O)CC2)=O)cc1 C1(CNC(CC=CC)=O)CN(C(c2nnn3c2COCC3)=O)CCC12CCOC2 C(=O)(CS(=O)CCC(F)(F)F)NC(CNC(C=CC)=O)(C)CC CC(O)(CC(=O)N1CCCC(F)(CNC(c2ncc(Cl)cc2F)=O)C1)C(F)(F)F C1(CNC(c2cc(CC)oc2C)=O)CC2(CC2)CN1C(=O)CC(O)CN(C)C C(CCCCN(C(=O)CCc1cn[nH]c1)C)NC(CSC)=O c1(CNC(C2CC(N(C)CC)C2)=O)nc(C(=O)NCC2CC=CC2)c(C)o1 c1(C2N(C(C3(C)CCC4CC4C3)=O)CCC2)ccc2c(c1)OCCO2 C(C)(CC(=O)NC1CCC(NC(=O)C(F)C2CCCC2)C1)(C(F)F)N(C)C N1(C(COCCOCC#C)=O)CCC(C(=O)NCC2C=CCCC2)C(C)(C)C1 C12(NC(c3c(C)nc(-c4ccsc4)s3)=O)CCN(C(=O)CC3(C)CCC3)CC1C2 N1(C(=O)NC(c2ccc(SC(F)(F)F)cc2)C)CCN(C)C(C)C1C N1(C(c2ccnc(C)n2)=O)CC2CCC2(C(N2CCC(OCC(N)=O)C2)=O)C1 Cc1c(C(N2CC3CCN(C(=O)CN4CC(=O)NC4=O)C3C2)=O)sc2nccn12 Cc1oc(CO)cc1C(=O)NCC(C)(F)CNC(C1(C)CCCC1C)=O N1(C(Cc2ncc(CC)[nH]2)=O)CCC2C(CCN2C(=O)C(C)NS(C)(=O)=O)C1 C(CCCCCC(=O)N1CC(CNC(C2(C)CC=CCC2)=O)C(C)C1)SC c1(C(C)C)ccc(C(=O)NCC(C)CN(C(C2CCOC2)=O)C2CC2)o1 C1(NC(C(C)C(C)O)=O)CCN(C(=O)Cc2cccs2)CCC1CO C1(CN(C2CCN(C(C)=O)C2NC(c2cc([N+](=O)[O-])n[nH]2)=O)C)Cc2cscc2C1 c1(C(=O)NC(C)C(CO)NC(C2(F)CCOCC2)=O)ccc(N(C)C)nc1 N1(C(c2cnccc2F)=O)CC2CC(NC(=O)C3(c4ccccc4)CC3)CC2C1 C1(C(=O)OCC)CCc2sc(NC(=O)Nc3ccc(I)c(Cl)c3)nc2C1 c1(CCC(=O)NC(C(C)NC(=O)OC(C)(C)C)C)nc(-c2ccoc2)no1 CC(C)S(=O)(=O)CC(=O)NCC1C=CC(NC(=O)COc2ccccc2O)C1 Cc1cc(C(N2CCCN(C3CC3)CC2)C(=O)NC(C)C)c2c(c1)CCC2 C=C(C)C(CC(=O)N(C1CCC(NC(=O)C(C(C)(C)C)SC)CC1)C)OCC c1(C(=O)NCC2C(CNC(C(C)(O)C3CC3)=O)C2)cnc2c[nH]nc2c1 N1(C(C2C(COC)C2)=O)CCCC(C(=O)NCCc2ccc(C)s2)C1 N1(C(C(=O)NCC)=O)CC2CC2(NC(=O)CCC2CC(C)(C)CO2)C1 C#Cc1ccc(C(=O)N(CC(C)NC(c2cccc(C3CC3)c2F)=O)C)nc1 C1(NC(c2cscc2F)=O)CCN(C(C2CCC(F)CC2)=O)C1C1CC1 c1(C(C)=O)cnc(Cl)[nH]c1=NC1CCCC(NC(c2cnc(C)o2)=O)C1 C1(C(N2CC(C)N(C(C34CCC(C)(CC3)OC4)=O)CC2)=O)CNC(=O)CC1(C)C Cc1cccc(C(N2CCCC2CCC(=O)N(C(C)CC(C)C)C)=O)c1 C1(NC(C(c2ccco2)NC(CCC=CCC=C)=O)=O)CNC(=O)C12CC2 C1(COC)CCC(NC(=O)C(C2(O)CCC2)NC(=O)CCN(C)CCO)CC1 C(=O)(CCCCCSC)N1CC(C(C)(C)O)(CNC(CCC2CCC(C)O2)=O)C1 N1(C(C(c2ccccc2Cl)C)=O)CC(NC(=O)CCCC2CCC2)C(O)C1 C1(CC(=O)NCC(CNC(C(c2cccnc2)OC)=O)C)CCCC(F)(F)C1 CCCCC(C(=O)N1CCC(CCC(=O)NCCCn2ccnc2C)C1)N(C)C c1(C(N(C2CCN(c3nc(Cl)ncc3Cl)C2)C)=O)ccnc2[nH]ncc12 N12CCC(CC1)C2=O.C1(N(C)C)CCC(N(C(=O)CCC2OCCO2)C)C1 CCC(C(C)(F)F)NC(=O)CC(C1CCC1)NC(=O)OC(C)(C)C c1(C(=O)NCC(C(C)C)(C)NC(c2ccnnc2)=O)cccc2c1OC(F)(F)O2 C#CCC(C)(CC)C(=O)NCCC1CC(NC(C2(C#N)CCSCC2)=O)C1 c1(CC)ccc(C(=O)N(C)CCn2cccn2)c(C(F)(F)F)c1 Cc1sc2nc(SCC(=O)NCCN3CCP(C)(=O)CC3)nc(O)c2c1C N1(C(C(COC)C)=O)CC2CCCC(CNC(=O)CN3CCC(O)CC3)(C2)C1 c1(CC(C)NC(c2ccc(OC)cc2)=O)ccc(-c2nn[nH]n2)c(O)n1 C(c1cn(C)cn1)=CC(=O)NCCC1(NC(C(C)N(CC(F)(F)F)C)=O)CC1 C(=O)(C(C)(O)C(F)(F)F)NC(C(C)(C)C)CNC(c1nnc(O)nc1O)=O Cc1nc(NCCC2CCC(NC(c3ccc(O)nc3)=O)C2)c2cnn(C)c2n1 c1(CC)oc(C(N2CCCC(CNC(C3CCCC(CF)C3)=O)C2)=O)cc1C c1(C(=O)OC)nccc(N2Cc3ccc(cc3)C2)n1.C(=O)(CCc1ccoc1)OC C1(C(N(CCCCC=C)C)=O)CC2C=CC1N(C(c1cnc(=N)[nH]c1)=O)C2 N1(C2CC(NC(CCCOCC=C)=O)C2)CCN(C(C2CCC(CC)O2)=O)CC1 c1(C(N(CC(C)NC(C2CCN(C(=O)NC)C2)=O)CC)=O)sccc1C#N C#CCCCCC(=O)Nc1cccc(CC(=O)NCCCN2CCC(O)C2)c1 c1(C(C(=O)OCCC=C(C)C)C)cccc(Br)c1 N(C(=NCCC1OCCC1(C)C)NCC1CCOC1)Cc1c(Br)cn(CC)n1 C1(NC(CC2(OC)CCCC2)=O)CCC(CN(C(=O)CC2(C)CCCO2)C)CC1 Cc1ncc(F)cc1NC(C1CCCN1C(=O)Nc1ccc(C#N)cc1)=O N1(C(CC2CCC(C)C2)=O)CCOCC(CNC(C23CC(CN2C2CC2)C3)=O)C1 C1(OC)(CNC(=O)C(C2CN(C(=O)C(CO)N)C2)SC)CCCCC1 C1(C(=O)NCCCC(C)NC(=O)CCC(F)(F)F)CCCC(C)(C)C1 c1(C(N(CCN(C(=O)CCNC(=O)CO)C(C)C)C)=O)c[nH]c(Br)c1 C1(NC(C=CCC)=O)COC2(C1)CN(C(=O)C(c1ccccc1)OCC)C2 C(=O)(C(CCC)S(N)(=O)=O)N1CCC(CC=C)(NC(C2CC(C)CCO2)=O)CC1 N1(C(C2C3CNC(=O)C23)=O)CCCC(CNC(C2(c3ccno3)CC2)=O)C1 N1(C(CCc2scc(C)n2)=O)CCC(NC(C2(C)CC2C(F)(F)F)=O)CC1C C1(O)(C(=O)NC2CCCC(NC(c3ccsc3Cl)=O)CC2)CC2(CCOCC2)C1 N1(C(C(C(C)NC(C(CC)=CCCC)=O)(C)C)=O)CC2CCN(C)C2C1 C1(C(=O)NCCC(C)(C)NC(=O)Cc2cc(C3CC3)no2)CCC(C#N)C1 Cc1ccc(OCC(=O)NCC(C)CN(C)C(c2ccc(O)c(N)c2)=O)c(C)c1 C1(NC(=O)Nc2cccc(C(N)CO)c2)CCn2nnnc2C1 C1(NC(C2N(C=O)CCC2)=O)CN(C(c2cncc(F)c2)=O)CC2(CCC2)C1 N1(C(C2(NC(c3cc(C)on3)=O)CCCC2C)=O)CC2CC(C)C2C1 C1(O)(C(C(N2C(CN(C(Cc3c(C)ccs3)=O)C)CCC2)=O)(F)F)CCCCC1 C1(C(=O)NC2CCN(Cc3cn(-c4ccccc4)nn3)C2)CCCC(O)C1 C1(c2n(C)cnc2)CN(C(=O)C2=CCC2)CC1NC(c1cc(Br)c[nH]1)=O Cc1ccc(Cl)c(O)c1C(=O)NCCNC(C1(C)C=CCCC1)=O Cc1cccc(S(=O)(=O)N2C(C(N3CCC4(CCCCC4)C3)=O)CC3CC23)c1 C(=O)(C(F)CC)N1CC(OCCC(N2CC(SCC)C2)=O)C1 c1(C(=O)NCCC2(NC(CCC#C)=O)CCCC2)c(OC)cccc1Cl CC(C)(O)CC(=O)NCC1(F)CC(NC(c2ccnnc2NC2CC2)=O)C1 c1(C(N(CCNC(CC(C)C(C)(C)C)=O)CC2CC2)=O)cc2c(cn1)COCC2 N1(c2ccnc(N3CCC(CNC(=O)NC)C3)n2)CCC2(CCCCC2)C1 Cc1conc1CC(=O)NC1(CNC(c2ncc[nH]2)=O)CC1 N1(C(C2(C#C)CC2)=O)CCCC(C2(NC(=O)C(C)OCCN(C)C)CC2)C1 C(=O)(CC(C(F)F)c1ccccc1)NC(CC(C)NC(c1cnc[nH]1)=O)C c1(CNC(C(C)(C)COC)c2n(C(CC)C)nnn2)ccc2ccccc2c1C C(C(C)C)(C(O)C(=O)NCCN(C(C1(c2ccccc2)CC(C)C1)=O)CO)OC c1(CCNC(C2CN(CCN3CCCC3)CCC2O)=O)ccc2c(c1)OCO2 CC(=Cn1ccnn1)C(=O)NC1CCC(NC(c2c([N+](=O)[O-])cnn2C)=O)C1 C(=O)(C(C)(O)C(C)(C)C)NCC(C)NC(c1nccn2ccnc12)=O C1(NC(C(Cc2c(C)nc[nH]2)O)=O)CC2(C1)CC(NC(c1onc(C)c1C)=O)C2 CN1CC(NC(=O)CC2CCCN(C(c3ccn(C4CC4)n3)=O)C2)CC12CCC2 c1(-c2[nH]ccc2)ccn2ccnc2c1.n1(CC)nnnc1N1CC2CC1C2 N1(C(c2cc(OC)no2)=O)CCN(C(=O)CC2(CO)CC2)C(C)CC1C CC(C)C(CC(=O)NCC(CNC(=O)OC(=O)C#CC(C)(C)C)C)N(C)C CC(C)C(O)CC(=O)NC1CN(C(c2scnc2C(C)(C)C)=O)CC1CC1CC1 C1(F)(CNC(C=CCOC)=O)CC(NC(=O)C=Cc2cocn2)C1 N1(C(C2CCCC(C(=O)OC)C2)=O)C(C)CC2CN(C(c3coc(C)n3)=O)CC12 C(CC(C)C(=O)N1CCC(CC(=O)NC(CCOC)C(C)C)C1)=CCC c1(CNC(C(F)(F)F)C2CC2)ccc2cccc(Cl)c2n1 CC(C)C(CNC(=O)C(C1CC1)C1CC1)C(=O)NC1(C(F)(F)F)CCCC1 c1(NC(C2(NC(CC=C)=O)CC(CO)C2)=O)cnc(Cl)c(C)c1 c1(C(N2CCCC(NC(c3cc[nH]n3)=O)(CO)C2)=O)cc(Br)ccc1[N+](=O)[O-] N1(C(CCC(C)(C)F)=O)CCC2(CC1)CCN(C(=O)CN1CC3C=CC1C3)CC2 c1(CCNC(N(CC(CCC=C)O)C)=O)ccc(Br)c(OC)c1 Nc1cccc(C(=O)NCCCNC(C2(Cc3cnn[nH]3)CCCC2)=O)c1F C(=O)(C1CCc2c[nH]nc21)N1CCC(C(=O)NC2(C#C)CC2)C(O)C1 C1(CC(=O)NC2COCCN(C(c3csc4cncn34)=O)C2)CC2(CCC2)CO1 C=CCC(C)(C)CC(=O)NC(CC(=C)Cl)C(=O)NCCC1CCCC12CC2 c1(CC)nc(N2CCCC(NC(c3c(C(F)(F)F)cnn3C)=O)CC2)[nH]c(=N)n1 c1(CNC(=O)CC2CC2)nnc2n1CCN(C(c1ccc3cccnc3n1)=O)C2 Cc1ccc(C(=O)NC(C)C(C)NC(c2cnn(C)c2C(F)F)=O)c(N)c1Cl N1(C(C2CCN(c3nc(C)cc(C(=O)OC)n3)CC2)=O)CCC2(CCC(O)C2)C1 N1(C(C(COCC)NC(=O)C#CC2CCC2)=O)CCc2nc[nH]c2C1 c1(NCC2CCC(C)O2)ccc(=N)[nH]c1Br Cc1ccoc1CC(=O)NC(C)CC1CN(C(c2cn[nH]c2)=O)C1 O=C(C#CC1CCOCC1)NCC1CCN(C(C2CN(S(N)(=O)=O)C2)=O)C1 N1(C(c2ccc(CCC)s2)=O)CCN(C(=O)CC2CC(F)(F)C2)C(COC)C1 C1(CNC(c2cc(CNC(CC#N)=O)sc2)=O)CC(O)C12CCC2 N1(C(=O)Cc2ccc(Cl)cc2)CCCC2C1CCN2C(=O)Cc1ccncc1 N1(C(C(CC)C)=O)CC(C2CCCN(C(c3[nH]c(=N)ccc3C)=O)C2)C1 c1(C(=O)NC(C2CCCN2C(C2CC2c2ccccn2)=O)C)nn(C)cc1Cl CC(C(=O)N1CCN(C)C(CNC(c2cnn(C)c2C2CC2)=O)C1)C(C)(F)F c1(C(=O)NCC2C(CC)C2)c(C(=O)Nc2cnc(OC)cn2)cccc1C c1(CC)cccc(CC)c1CC(=O)NCC(C)CN(C)C(C12CC(F)(C1)C2)=O c1(C(c2nnnn2CCCC2CC2)NC(C(=O)NCC(C)C)C)ccnc(F)c1 c1(C(N2C(CNC(CCC#C)=O)CC(OC)C2)=O)cccc2ccc(C)nc12 C1(CNC(COC(C)C)=O)CC(F)CN1C(=O)C(C)O c1(C(N2C(CNC(C3CCO3)=O)CCC2)=O)ccc(Cl)c(C(F)(F)F)c1 C1(C2CCNCC2)(C(=O)NCC(C(C)C)=O)CCOCC1 C#CC(C)(C)C(=O)NCC1CCCCN1C(c1c(C)noc1C)=O c1(C(=O)NCC2N(C(C(C)n3cccc3)=O)CCOC2)noc2ccc(Cl)cc12 c1(CC(=O)N(C2CCC23CCNCC3)C(C)C(F)(F)F)cccc2ccccc12 C(CC(O)C(=O)NCC1CN(C)CCO1)NC(CCC=C)=O N12CC(C)(C)CC1CC2=O.N1(C(Cn2c(C)nnn2)=O)CCCC1(C)C(N)=O c1(C(N2CC(CC(C)(F)F)C2)=O)cc(=O)c2cc(Cl)ccc2o1 C1(C(=O)NCC=CCNC(c2c(C)nn(C(C)C)c2)=O)CN2CCN1C(C)C2 c1(C(CNC(=O)C(C)c2ncco2)NC(CC2CC(OC)C2)=O)cccc(Cl)c1 C(c1ccnn1C)=CC(=O)N(C)CC1(CNC(=O)C=CCN2CCCC2)CC1 CCC(CN=c1[nH]c(=NCC2(CC#N)CC2)[nH]c2cc(C(F)(F)F)ccc12)OC c1(CCC2CC2)cc(NCC2C(C(=O)NC(C3CCC3COC)=O)C2)n(C)n1 C=CC(C)(O)CC(=O)N1CCC(N(C(=O)C(C(C)C)NS(C)(=O)=O)C)CC1 c1(CCC(N2C3(CN(C(c4ccc(=O)oc4)=O)C3)CC2)=O)nc2ncccn2n1 C1(C)(C(=O)NC(CCCNC(C2C(C)=CCS2)=O)(C)C)CCCCNC1=O N1(C(CC(CCC)CC)=O)CCC2(CCCN2C(=O)C(C(C)C)SC)C1 CC(C)(CC(=O)N1CC(NC(c2sc(F)cc2Cl)=O)C(O)C1)CC(F)F c1(NC(c2cncc(NC(C#C)=O)c2)=O)c(F)cc(Cl)cc1Br c1(CC)cnccc1C(N1CC2C(C(N3CCCC(C(C)C)C3)=O)C2C1)=O CC(CNC(=O)CC(=O)N(C)C)CC(=O)Nc1ccc(F)nc1 N1(C(C(C)(C)NC(=O)NCC)=O)CCCC(CNC(c2cccc(CO)n2)=O)C1 c1(CC(=O)NCC(CNC(c2csc(-c3ccc(C)o3)n2)=O)OC)n[nH]c(C)n1 c1(NC(C)CCCNC(C23CCC(CC2)CC3)=O)ccc(NC=O)c([N+](=O)[O-])c1 c1(OC)nn(C)cc1-c1nc(-c2nc[nH]n2)nn1Cc1ccc(C)cc1 N1(C(C(C)=C(C)C)=O)CC(C2(NC(=O)CCOCc3ccccc3Cl)CC2)C1 C(CC1=CCOCC1)NC(c1c(C(C)NC(C(COC)(C)C)=O)noc1)=O C1(C(=O)Nc2cccc(NC(CCCCC(N)=O)=O)c2)Cc2c[nH]cc2S1(=O)=O N1(C(C2C(CC)C2)=O)CCCC(C2CCN(C(c3ncn(C(C)C)n3)=O)CC2)C1 C1(NC(CN(CCC)C)=O)CC2(CCN(C(=O)C(C)CC(F)(F)F)CC2)C1 C1(CC)C=CCN(C(=O)C(C(C)O)N(C)C)C1.C12(CC1)C(=O)N2 Cc1ncc(C(N2CCCC(C(=O)Nc3nc(Br)ccc3Br)C2)=O)c(C)n1 C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(C2C3COCC23)=O)CC1S(C)(=O)=O c1(C(C)=O)cnccc1C(N1CCC(CO)(NC(=O)C=Cc2ccco2)C1)=O N1(C(C2C(C)C2)=O)CC2OCCN(C(=O)C(O)Cc3cnc[nH]3)C2C1 C(=O)(C(CC)CC(F)F)NCC1C(NC(CC=C)=O)CCC1 c1(COC(C(=O)NC2CCC(CNC(CSC)=O)C2)C)cccc(C)c1 N1(C(COC(CC)C)=O)CCC(C2(NC(=O)C3=CCCOC3)CC2)CC1 C(C(=O)N1CCCC1(C)C(N1CCC(CN=[N+]=[N-])C1)=O)(C(C)(C)C)OC Cc1cc(N2CCCN(S(C)(=O)=O)CC2)nc(=NCCNC(=O)C2CC2)[nH]1 c1(C(=O)NC2C3CCC2CN(C(=O)CC(F)(F)F)C3)cncc2cnccc12 C(=O)(C(F)CC(CC)CC)NC1C(C(N2CCC(=C)C2)=O)CC1 C1(NC(C=CCC)=O)CC2CC1N(C(c1cccc(OCC(C)C)c1)=O)C2 C(=O)(C#CC1CCCO1)N1CC2C(CNc3nc(OC)nc(OC)n3)C2C1 N1(C(C(CC)SC)=O)CCCC(NC(=O)Cn2nc(C)cc2N)C1 C1(C(=O)NCCC2(NC(C(CCSC)O)=O)CCCC2)CC(=O)N(C)C(=O)N1 Cc1ccc(NC(C2(CO)CCN(C(=O)CCc3ccsc3)C2)=O)c(Br)c1 C1(CN(C)C(C2CCC(C(N)=O)CC2)=O)COCCN1C(C1CC(F)(F)C1)=O C(=O)(C1=NOC(C)(C)C1)NC1C2(CCN(C(C=CCNC(=O)OC(C)(C)C)=O)C2)C1 C1(NC(=O)CCCc2nccs2)(CO)CCN(C(=O)CC2CCC=CCC2)C1 C1(C)(NC(CN2CCC(C)CC2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 C(=O)(C(CC)CCCCC)NC1C2(CC(NC(C3(CC#C)CC3)=O)C2)C1 C(=O)(C(C)(F)C(C)(C)F)N(C)Cc1n[nH]c(CO)n1.C12C=CC(C1)NC2=O C1(C(=O)NC2C(NC(CCC(C)(C)F)=O)COC2)CSC(c2ccccc2)=N1 Cc1cn2cc(C(=O)OC3CCC(C)CC(C)(C)C3)nc2c(C)n1 C#Cc1cnn(C)c1C(=O)NCc1ccsc1C(N1CCC(CC)CC1)=O CC1CCCC(C)N1CCC(N1CC2(NC(=O)C(=O)N(C)C)CC1(COC)C2)=O c1(CN2CC(NC(Cc3ccc(OC)cc3)=O)C(C)C2)cc(Cl)c(O)cc1F N=c1[nH]nc(CCC(=O)NC2CC(F)(CNC(C3COCCO3)=O)C2)s1 C1(NC(C2CC23CC(O)C3)=O)CCCCN(C(c2ncoc2-c2ccon2)=O)C1 Cc1cc(=NCC2CC=CCC2)[nH]c(N2CCC(N3CCC(O)C3)CC2)n1 Cc1ncnc(C)c1CC(=O)N(C1CCN(C(C2CC(C)(C)O2)=O)C1)C c1(N(C)C)nc(C(N2CCC(CNC(C3CCCC(=O)O3)=O)C2)=O)cc(O)n1 C(=O)(N1OC2CC1C(O)C2O)C1C2(CC(NC(=O)CCc3nc[nH]n3)C2)C1 C(=O)(C(O)Cc1cnc[nH]1)N(CC(O)Cc1cnn[nH]1)C.c1(=O)c(=O)[nH]1 c1(C(N2CCC(NC(c3nc(C(C)OC)sc3)=O)C2)=O)cc(CO)c(C)o1 CC1CN(C(c2ccc(CF)cc2)=O)C(C)CN1C(=O)C(O)CC1CCCC1 C(C(C)CC(=O)ONC(c1cc(Cc2cccc(OCF)c2)on1)=O)OC Cc1cc(Cl)cc(Br)c1NC(C1CCSC(C(F)(F)F)C1)=O O=C(CC1OB(O)c2ccccc21)Nc1ccc(Cl)c(I)c1F C(=O)(C(F)(F)C(O)C(C)C)NC1CCCN(C(c2c(CC)n(C)nc2)=O)CC1 c1(C(=O)NCCCNC(C(C)C(C)C2CCCCC2)=O)cccc2nc(O)oc12 c1(CNC(c2cnc(CNC(=O)CCN3CCCC3)[nH]2)=O)cccc2oncc12 C1(C(=O)NCC(C2CC2)NC(c2cc(C(=O)OC)on2)=O)CN(C)C(=O)N1 Cn1cc2ccc(C(=O)NC3CN(C(C4(Cl)CC4(F)F)=O)CC3C3CC3)cc2n1 Cc1ccc(C)c(C(=O)NCCC2CCCCN2C(C2CC3(C2)CC(C)C3)=O)c1 C1(C(N(C)CC2CCCN(C(c3c(OC)noc3C)=O)C2)=O)CCCCN1N=O N1(C(C(C)(C)c2cccnc2)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)C2 c1(NC(C2CC(C(=O)NC(C(N)=O)CO)C2)=O)nc2ccccc2o1 CC1(C)C(CNC(=O)COc2ccon2)CCN1C(=O)CCC(N)=O N1(C(c2ncc(Br)cn2)=O)CC2CCC(C1)N(C(=O)Cn1cccn1)C2 C(=O)(C1CCCc2nc[nH]c21)NCCC(CNC(Cc1c(C)cccn1)=O)O N1(C(CS(=O)(=O)NC)=O)CC(C)N(C(=O)CCc2cscn2)CC1C c1(C(=O)NC2(C3CN(C(CCOCC#C)=O)C3)CC2)cncc2nnn(C)c12 C(C1CCC(=O)O1)=CCN1CCC(C(C)C(=O)N(C)C)C1 CC1COC2(C1)CN(C(=O)CC1CC(NC(C3(CO)CCOC3)=O)C1)C2 c1(C(=O)NCC2(O)CCN(C(C3CN(C)C(=O)C3)=O)C2)cc2sc(Cl)cc2[nH]1 C(=O)(C(C)CCCC(C)=O)N1CCC(CC#C)(C(=O)NC2CCCNC2=O)C1 CCC(C(=O)NCC(O)CNC(C1CCCN1c1ccncn1)=O)C(C)C Cc1nc2cncc(C(N3CCC(CNC(=O)C(C)CO)C34CCC4)=O)c2[nH]1 N1(C(CC(C)(F)F)=O)Cc2ccnn2CC(NC(=O)COCc2ccccn2)C1 C(CN=c1[nH]nc(C2CC2)o1)NC(C1N(C(N)=O)CCCC1)=O C(=O)(C(C)(O)CCN(C)C)NCC(C(=O)NCC(CC)N(C)C)N(C)C c1(N2CC(CNC(C)=O)OCC2)nc2cc[nH]c2c(=NCCc2ccccn2)[nH]1 c1(C(=O)NCC(C(C)C)NC(C(=Cc2cnc[nH]2)C)=O)cc(C(F)F)nn1C c1(C(=O)NC2CC(C)(NC(CCC(C)C)=O)C2)cc2sccc2[nH]1 CCCCC(CCC)NC(c1ccnc(CNC(C2CC(C)(C)CN2C)=O)c1)=O CC(CNC(C1CN(C2CCC2)C1)=O)(C1CC1)NC(N)=O C(=O)(C(CCC(N)=O)N(C)C)N1CCCCC(NC(CCCOC)=O)C1 c1(C(=O)NCC2(C(C)(C)O)CN(C(CN(C)C)=O)C2)cc2cn[nH]c2cn1 C#CCC(C)(CC)C(=O)NCCC(C)(C)NC(c1nc(C)n(-c2nc[nH]n2)n1)=O Cc1cccc(C(=O)NC2C=CC(CNC(=O)Cc3csc(C)n3)C2)c1 N1(C(c2cc(CC)nn2C)=O)CCN(C(=O)C(c2cccc(Cl)c2)O)CC(O)C1 c1(C(=O)OC(C)(C)C)ccncc1C(=O)NCC1(NCCC2CCOC2)CCC1 c1(C(=O)NC2C(NC(=O)CCc3ccncn3)C2)c(O)cc(F)cc1F C1(NC(c2cn(C)nn2)=O)CCN(C(=O)CCC(F)F)C1c1ccccc1 c1(OC)ccc(C)cc1C(N1CCCC(NC(c2ncc(F)cc2F)=O)CC1)=O C=CC1COCC1NC(=O)CC1CC2(CC2)C1.c1(=O)c(=O)n1C c1(-n2cc(CNC(CNC(CNS(CC)(=O)=O)=O)=O)nn2)ccc(CO)cc1 N1(C(C(C)(C)O)=O)CCC2(CC(NC(c3ccnc(C(F)F)c3)=O)CO2)C1 c1(C(=O)NCC(c2c(F)cccc2Cl)O)cc2n(n1)CCCCC2=O N1(C(C(CCC)NC(c2cc(OCC)no2)=O)=O)CCCC(C)(CC)CC1 CS(=O)(=O)c1coc(COC(C2CCN(CC(F)(F)F)CC2)=O)c1 Cn1ncnc1CCNC(=O)C(C1CCN(C(C2(C3CC3)CC2)=O)C1)F c1(C(N(CC(CC)NC(=O)CC(C)(C)C(F)F)C)=O)cccn2cc(C)nc12 Cc1cc2c(Br)ccc(C(=O)NCCCC(C)NC(=O)CC3(O)CCC3)c2o1 N1(C(c2c(CNC(CCC(=O)NC)=O)nnn2C)=O)CCOCC12CC2 N1(C(C2C(CCC)CCC2)=O)CCC2(CC1)CC(NC(=O)CC(C)C(F)F)CO2 CC1(CNC(C2(CO)CCOCC2)=O)CCN(C(=O)C(F)(Cl)c2ccccc2)C1 C(=O)(C1CCCc2nn(C)cc21)N(CCNC(C=Cc1c(C)cccc1)=O)C N1(C(COc2cccc(C)c2)=O)CC2(CC(NC(=O)CCC[N+](=O)[O-])CO2)C1 C1(NC(C2CCCCNC2=O)=O)CN(C(=O)C2=CCCSC2)Cc2ccnn2C1 CC1CCC(NC(=O)CCCn2cccn2)CN1C(c1ncc[nH]1)=O c1(OC)ccc2c(C(=O)NCC3(NC(=O)CC4CCOC4=O)CC3)cnn2c1 C(C(O)CC(=O)NCC1(NC(C2(c3cccnc3)CC2)=O)CC1)N(C)C C(C1=CCCOC1)N(C(CCN(C(CNC(C1C(C)C1)=O)=O)C1CC1)=O)C C1(C(N2CCOCC2)=O)(CNC(=O)CSCC(F)F)CC2(CC2)C1 CC1CCN(C(c2cnc3n2CCC3)=O)CC1CC(=O)NCc1cn[nH]c1 Cc1cc(NCC2CCCOC2)ncc1S(=O)(=O)NCCc1ccc(Br)o1 C1(NC(C(c2cn(C)nn2)NC(=O)CCOCC2CC2)=O)CCC2(CC1)CC2 N1(C(c2cc(C)nn2C(C)(C)C)=O)CC2CC(NC(c3sccc3C)=O)C2C1 Fc1ccc2c(c1)C1C(C2)C1(F)F.c1(C2NCCCC2)nc2ccccc2o1 c1(N(C(C)=O)Cc2ccn(CC)n2)ccccc1OCc1ccncc1 c1(C(=O)NC(CC=C)CNC(C)=O)ccc(OC)c(S(C)(=O)=O)c1 CC1CCN(c2nnc(C(O)C(C)C)n2CC2CCCCO2)CC1F c1(C(=O)NC2CN(C(c3ccc(N(C)C)cc3)=O)C2)cc2cc(Cl)ccc2[nH]1 c1(C(=O)NCC(=O)NCC(F)(F)F)c(O)cccc1[N+](=O)[O-].C12CNCCN1C2=O c1(CN(C(CC)C)C)ccc(S(=O)(=O)NCCC(CC)CO)cc1C#N c1(CC(N2CCCC(CCNC(C3CCOC3)=O)C2)=O)coc2cc(Cl)ccc12 C(=O)(CCC(C)(F)F)NC1(C)CC(NC(C2N(C(C(C)C)=O)CCCC2)=O)C1 c1(CC(=O)N(CC(C)NC(C2CCCC(C)(C)O2)=O)C)ccc(F)cc1[N+](=O)[O-] C1(C(N2CCC(C(CC)CC)C2)=O)CC2CN(C(=O)C(C)(C)OC)CC2C1 N1(C(C(C=C)(C)CCOC)=O)CCC2(CCC2NC(c2ccc(O)nn2)=O)CC1 C(=O)(CCCC(F)(F)CO)N1CCCC(C)(NC(c2cc(C)n(C(C)C)n2)=O)C1 c1(CC(C(=O)NC2C(CNC(C=C(COC)C)=O)C2)NC=O)ccc(C)cc1 CC1=C(C(=O)NC2CC3(C(N4CCC(CC(N)=O)C4)=O)COC2C3)CCCO1 c1(C2CCOC2)ncc(C(N(CCCNC(C2CC(O)C2)=O)C)=O)s1 N1(C(C2CCN(CC)C2)=O)CC2CCCC2(NC(=O)C2=CCCCO2)C1 c1(C(=O)NCC2(C)CCN(C(C3CCC(C)C3)=O)C2)cc2c(s1)CN(C)CC2 CCC(C)(C)C(=O)N(CC(C)(C)NC(=O)CCc1ccc(C(C)C)cc1)C N1(C(CC2CC(OC)C2)=O)CC(NC(=O)C(C)CC#N)CC(O)C1 C(C)(C(C)CC)N(c1ccccc1)C(CSCC)=O C1(C(C)NC(=O)CC2CNC(=O)O2)CCN(C(c2cn(C)cn2)=O)CC1 N1(C(C(C2CCC2)NC(=O)CCc2ccsc2)=O)CCCN(C=O)CC1 c1(CNC(c2ccccn2)CCC)coc2ccc(OC)cc2c1=O S(=O)(=O)(c1ccc(NC2CCCC(F)C2)nc1)N(CCOCC)C CCC(C)(CO)C(=O)NC1CCC(CC(N2CCOCC2CCO)=O)CC1 N1(C(C(C(C)NC(=O)Cn2ccnn2)C)=O)CC2(CCCCC2)C1 CC1CCCC1C(=O)NCc1c[nH]nc1C1CCN(C(=O)CSc2nc[nH]n2)C1 CC1CN(C(c2ccc(Br)o2)=O)CCC1NC(=O)C=CC(N)=O C(=O)(CCCCCS(N)(=O)=O)NC(C1CCN(C(CCNC(=O)NC)=O)C1)C C1(C(N2C(C#C)CC2)=O)CN(C)CCN1C(c1cscc1OC)=O N1(Cc2c(OC)cco2)CC2CN(C(c3cc(C)cnc3Cl)=O)CC2C1 C(=O)(NNC(=O)CC12CC(c3ccccc3)(C1)C2)C1CC1.C12(CN=[N+]=[N-])CC(N)(C1)C2 C(CC1=CCCCC1)N(C)C(C1(NC(C2CC2c2ccccc2)=O)CCSC1)=O N1(C(C#CC(C)C)=O)CCCC12CCN(C(c1ccn3ncccc13)=O)C2 C1(NC(C=CC)=O)CC(F)(CNC(C23CCCC2C3)=O)C1 Cn1c(Cl)c(CN2CCN(c3nc(C(N)=O)cs3)CC2)c2ccccc12 C1(C(=O)NC2CCC(Cn3cc(C(CC)N(C)C)nn3)C2)CC(C)(C)CN1C Cc1cc(C(=O)NCC2CCN(C(=O)C(C)SC(F)(F)F)C23CC3)cc(C)n1 C1(OC)CN(C(=O)Cc2cscn2)C(C)(CNC(=O)CNS(N)(=O)=O)C1 N1(C(C2(CC)CCC2)=O)CC2C3CCC(C(NC(c4cc(C)no4)=O)C3)C2C1 C1(NC(C(COC)O)=O)CCN(C(=O)CCCC2OCCO2)CC1 CCCC(C)(C)CC(=O)N1CCC2(CC2)CC1C(=O)N(C1CCN(C)C1=O)C Clc1ccc(-c2csc(CSc3cccc(Cl)c3)n2)cc1 N1(C(C(CCC)O)=O)CC2CC(C1)CN(C(C1CCCN1C1CCCC1)=O)C2 c1(C(=O)NC2(CC=C)CCN(C(C3CCCCS3)=O)C2)ccc(N=[N+]=[N-])cc1 CC1(C#N)CCCN(C(=NCc2ccc3c(c2)OCO3)NCC2CCOC2)C1 C1(C(=O)NCCCC(C)NC(C=C(CCC)C)=O)CCC(C(=O)N(C)C)CC1 C1(C(=O)NC2C(C)CCN(C(c3n(CC)cnn3)=O)C2)CCc2nc(C)cn2C1 C(C(C(C)C(C)C)NC(=O)CN1CCC(F)(F)C1)NC(c1c(C)cccn1)=O Cc1ccc(O)c(C(N2CCCC(CO)(NC(c3cn(C)c(=O)n3C)=O)C2)=O)n1 N1(C(C(CC)OC)=O)CC2CC(CNC(C3(C(F)(F)F)CCCC3)=O)C2C1 N1(C(CC(CC)(F)F)=O)CC2(C1)CN(C(c1cc3c(=O)[nH]ccn3c1)=O)CCO2 N1(C(C2CN(CC)C(=O)C2)=O)CC2CCCN(C(C3CCN(C)C3=O)=O)C2C1 c1(C(=O)NC2C(C(N(CC)Cc3cc[nH]n3)=O)C2)ccc(F)c(F)c1Cl C1(NC(CCCOc2cccc(C)c2)=O)CN(c2ccnc(Cl)n2)CC(C)(C)C1 c1(NC)cnccc1C(=O)NCC(C)N(C(=O)C(C)c1ccon1)C C(=O)(C(C)(CC)CC)NCC(CC(=O)N(C(CC#C)C)C)O CC1C(C(=O)N2CC(NC(c3ccc(F)cc3F)=O)CC2(C)C)=NOC1C C1(CNC(CP(C)(C)=O)=O)CCC2(CO1)CC(NC(C1CC(O)C1)=O)C2 c1(C(N(CCCOC)CCNC(=O)CSC2CCCO2)=O)ccccc1C C(C(O)C(=O)Nc1ncccn1)NC(=O)C1CC1.C12CCCC1N2 C1(C)(C(=O)NC2(CNC(C3C(C)CCCC3)=O)CC2)CCC2(CC1)OCCO2 N1(C(c2cc(C)c(Cl)cc2)=O)CC2CN(C(=O)C=C3CCN(C)CC3)CC2(C)C1 c1(C(=O)OC)ccc(S(=O)(=O)NC2(C)CCCC2c2cccc(F)c2)nc1 N1(C(c2cc(Cl)nc(Cl)c2)C(=O)NC(C(=O)OC)C)CCCN2CCCC2C1 N1(C(C2CC(OC)C2)=O)CCC(=O)NC2CN(C(=O)C(C)CO)CCC12 C(=O)(CC(CC)CC(C)C)N(C(C(=O)OC)CC(F)(F)F)C.c1(C)nn[nH]n1 C(c1ccc(N)c(N)c1)=CC(N1CCC(CC=C)(NC(C2CC2(C)CC)=O)C1)=O n1(CC)cc(C(=O)NCC2COCC2NC(=O)Cc2cc(C)nn2C)c(C2CC2)n1 C12(C(=O)NCc3cc(C)[nH]n3)CCCC1CCN2C(c1cc2ncccc2[nH]1)=O C(=O)(C(C)CC(C)CC)NC1(CC=C)CN(C(=O)Cc2ccccc2C(C)C)C1 CCC(CC)(CO)C(=O)NC1CCN(C(c2cccc(C3CCC3)c2)=O)CC1F N1(C(c2c(C)ccnn2)=O)CCC(C(N2CC3CC=CC2C3)=O)C(C)(C)C1 c1(CC(C(=O)NC(C#C)CC2CCCC2)NC(=O)C(O)C(C)C)ccccc1Br c1(C(COC)NC(=O)C(c2sc(Br)nc2Cl)N2CC(O)CC2C)cccc(F)c1 N(C1CN(C(=O)CCS(C)=O)CCc2ccccc21)C(c1cnc(C)nc1)=O N1(C(C2(CSC)CC2)=O)CCCC1C(C)(C)NC(=O)COc1cc(C)on1 N1(C(c2c(CC)nco2)=O)CC2CC(C1)N2C(C1COCC(C)O1)=O Cc1cc(=O)ccn1CC(=O)NC1CC2CC(NC(=O)Cn3ccnn3)C1C2 CCC(CSc1ccccc1)CCO.c12nnc(n1C)c(=O)[nH]2 N1(C(c2cc(CCC)on2)=O)CCCC(O)(CCNC(C2(C)CC3CC3C2)=O)C1 c1(C(=O)NC2CCCC(NC(Cc3cc(OC)no3)=O)C2)sc(F)cc1Cl C(=O)(CCN=[N+]=[N-])NC(C(=O)NCCCC#C)CC1CCCC1 Cc1ccc2nc(C(=O)NC3CCCC34CCN(C(=O)CC3CC3)C4)cn2c1 CC(CCC(C)(C)C)C(=O)N(C)CC1(NC(=O)C2=CSCS2)CC1 Cc1cnn2c(SCC(=O)Nc3ccc(O)cc3)cc(Cl)nc12 c1(C(=O)NC2CN(C(c3c(C)cc(C)nc3)=O)C(C)C2)ccc2c(c1)COC2=O CCC1=C(C(=O)N2CCC(NC(c3cnc(S)[nH]3)=O)C2(C)C)CCCO1 N1(C(CCC2(NC(=O)C=C3CCC3)CCCC2)=O)CC2CCCC1C2 n1(CC)cncc1CNC(=O)CSCCNC(=O)C=CC1CCOC1 C1(NC(c2cnc(NC(C)=O)o2)=O)CN(C(=O)C(C)(C)c2ncco2)CC1F N1(C(CCC)=O)CC2(CCC(NC(=O)C=Cc3ccc(OC)cc3)C2)C1 c1(C(N2CC(N(C)C(C3CCC(=C4CCC4)CC3)=O)C2)=O)ccc(N)c(CO)c1 N1(C(C2CCCN(C)C2)=O)CC2(CCCC2NC(=O)CCCN2CCOCC2)C1 N1(C(C(C)OCC2CC2)=O)CC(C)CN(C(=O)CC2CCC(=O)C2)C(C)C1 C(=O)(C(CC(F)F)N(C(=O)CC(C)SC)C)NCC(CO)OC N1(CC(=O)NC(C)Cc2cnc[nH]2)CCN(C(c2cccs2)=O)CC1 CC(CCNC(=O)C(c1ccccc1Br)(F)F)CCNC(=O)C=CCF C1(C(=O)NCC2CCN(C(CCc3cn(C)nc3)=O)C2)CCOC(=O)CC1 C1(NC(C=C(C)c2ccsc2)=O)CCN(C(C2CCCC(C)(C)O2)=O)C12CCC2 c1(C(N2CC(O)(CNC(=O)COCc3nc[nH]n3)C2)=O)cc(C(F)F)ccc1F C(=O)(C1CCCn2ncnc21)NC1CN(C(c2c(C)nc(CC)s2)=O)CC1(C)C C(CC#CC(C)(C)C)N1CCCC(C)C1 CCC1=NOC(CCNC(C2(CC)CCN(C(C3CC(C)(C)CO3)=O)C2)=O)C1 C1(C(=O)NC(C)CNC(=O)CC2C=CCC2)Cc2cc(C(F)(F)F)ccc2O1 C1(CC#C)(C(=O)N(CCCNC(=O)CC2CC2(Cl)Cl)C2CC2)CCOC1 c1(OC(C)C)cc(CC(=O)N(C)Cc2cn(C3(C(F)(F)F)CC3)nn2)cc(Cl)c1 C12(CNC(C3N(CC)CCC3)=O)CCC(C1)N(C(C1(C(F)(F)F)CC1)=O)C2 C(Cc1cnc[nH]1)(C(=O)NCCC(C)O)NC(C=C(COC)C)=O CC1CC(NC(=O)CC2CCCC2C)CN1C(=O)Cc1ccc(SC2CC2)cc1 c1(-c2cc(OC)c(C)nc2)ccc2ccnc(NC(=O)CSC(C)=O)c2c1 c1(OC)ccc(O)cc1C(=O)NC1CCCC(CNC(C2CC(O)C2)=O)C1 N1(C(C(CC)NC(N)=O)=O)CC(CNC(C2CN(CC(C)C)C2)=O)C(O)C1 N1(C(C(C(C)C)N(CC)CC)=O)CCC(CNC(=O)CCSC)C(F)(F)CC1 CC(C)C(C)(CO)NC(C1OCCC1NC(C1CCOC1)=O)=O c1(COC(=O)CCNC(C2CC3(CC3)CN2CC)=O)cc(C)c2c(c1)CCCC2 c1(C(N2C(C(=O)NCC(C)NC(=O)OC)C=CCC2)=O)ccc(C)nc1C c1(C(N2CC(N(C(CCCCSC)=O)C)C(F)C2)=O)cc(C)nc(O)n1 c1(COC)ccc(C(=O)N(CC(=O)NCC2CCC2)C2CC2)cc1 C12CC(F)(C1)CNC2=O.C(=O)(C(C)(O)C1CCC1)N.C(C(=O)N)SCCN(CC)CC N1(C(c2c(C)c[nH]n2)=O)CCc2nc(CNC(C3CC3C3CC3)=O)sc2C1 C(=O)(C1=CCCN(C(=O)CC2(CSC)CC2)C1)N(C(C=C)C1CC1)C c1(NC(c2ccc(CNC(C(c3cccnc3)OC)=O)s2)=O)cc(C)ccc1C c1(C(=O)NC(C2CCN(C(c3cccc(OCCF)c3)=O)C2)C)cnnc(O)c1 N1(C(CC2N(C(Cn3c(C)ccc3C)=O)CC(O)C2)=O)CCCC2CCCCC12 N1(C(C2C(CC)OCC2)=O)CCC2(CC1)CC(NC(c1ccoc1Br)=O)CCO2 c1(CN2CC(C)(C(=O)NCc3ccc(Br)nc3F)C2)c[nH]c2cccc(C#N)c12 C(=O)(C(COC)CC(C)C)N1CC(C(=O)NCC(F)C2CCC2)(COC)C1 CC1CN(C(c2ccco2)=O)CCC1CNC(=O)CCc1ccc(C(F)F)cc1 c1(C(C)NC(c2cn(C)nn2)=O)ccccc1-c1ccc(C(N2CCCC2)=O)nc1 C1(N(C(CN2CCN(C(c3c(CC)noc3C)=O)CC2)=O)C)CC2CCC1CC2 CC1CCC(=CC(=O)NC2(CC(=O)NCCCC(N)=O)CCC2)CC1 C1(CC(=O)NC(CCN(C(CN(CCOC)C)=O)C)C)CC(C)=NO1 c1(C(N2CC(CC)N(Cc3ccc(O)cc3)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C(C)(C)F)=O)CCC(F)(F)C(CNC(C2(CC3CCCC3)CCCC2)=O)C1 C1(C)(CC)C=C(C(=O)NC2(C(=O)NCC(O)CC3CCC3)CCCCC2)C1 C1(C(=O)NC(C2CCN(C(C3(SCC)CC3)=O)C2)C)CC=C(C)CC1 c1(C(=O)NCCC2(OC)CN(C(C3(CN(C)C(C)C)CC3)=O)C2)c(C)cnnn1 N#CC1CC(C(=O)NCCN(C(c2ocnc2C2CCC2)=O)C2CC2)C1 N1(C(C(N2CCC(C)C2)=O)=O)CCN(C(=O)C=Cc2ccc(C(N)=O)o2)CC1CF c1(C(C)C)ncc(C(=O)NCC2CCCC2NC(=O)Cc2ccoc2)cn1 c1(NC(=O)CC2CCCN2C(c2ccc(Br)nc2F)=O)ccc(Cl)c2cc[nH]c12 c1(SCC(N2CCCC(NC(C(C(=O)OC)C)=O)C2)=O)ccc(C)c(C)c1 C1(S(N)(=O)=O)(C(c2n(CCSC)nnn2)Nc2ccc(F)c(SC)c2)CCCC1 N1(C(C#C)=O)CCC(O)(CNC(=O)CCc2cc(OC)no2)C1 N1(C(CNC(CCC)=O)=O)CCCC1CCNC(=O)C(C)(C)c1cncs1 N1(C(C2CN(CC)C(=O)CC2)=O)CCC2(NC(=O)Cc3cc(C)on3)CCCC12 C1(N(C(Cn2ncc(C)c2)=O)C)CC2CC1N(C(C1CCC(=O)C1)=O)C2 CC(C)C(O)C(=O)NCC1(CCCNC(=O)Cc2csc(=N)[nH]2)CCCC1 c1(OCC(C)N(C)Cc2ccccc2)ccnnc1S C1(NC(CC2ON=C(C)C2)=O)CCC(F)(CNC(=O)Cn2ccc(C)c2)C1 c1(C(=O)Nc2c(CC)ccc(F)c2)cc([N+](=O)[O-])ccc1OC C=CC(C)(C)CC(=O)NCC(C(F)(F)F)N1CCN(C(=O)CC2CSC2)CC1 N1(C(c2n(CCOC)ncc2)=O)CC(NC(C2(COC)COC2)=O)CC1C C(=O)(CS(=O)(=O)C(C)(C)C)NC1CC(NC(C2C(C)(C)C3CCC2C3)=O)C1 C12(C(=O)NC(CCOC)CNC(=O)CCc3ccn(C)c3)CC(C)(C1)OC2(C)C c1(N(C)Cc2ncc[nH]2)nccc(=NC2CCCCCC2F)[nH]1 C1(COC)(NC(C2CC2(C)C(C)C)=O)CN(C(C2(C(=O)N(C)C)CC2)=O)C1 C(C1=CCN(C(C2CCC=CO2)=O)CC1)NC(CC1(OC)CCC1)=O c1(CC)ccc(C)cc1C(=O)NCCC(C)NC(C1(C)CCNC1=O)=O c1(C(N2CC(N(C(=O)CC3CCC4CC34)C)C2)=O)cc2c(s1)CCC2 c1(NCC2CN(C(CC(C)N(C)C)=O)C2)ncnc2cnccc12 NC(=O)CC(O)C(=O)N1CCCC(F)(C(N2CCCC(O)CC2)=O)C1 C1(OC)(NC(N2CCCC2c2cccc(F)c2)=O)CS(=O)(=O)C1 N1(C(C(CCC)CC)=O)CCC(C2CC(NC(c3sc(C)cc3C)=O)C2)CC1 C12(C(=O)NC3CC(NC(C(CCC)c4ccccc4)=O)C3)CCN(CC1)CC2 CC(CS(C)=O)C(=O)NC12CC(CNC(=O)Cc3csc(Br)n3)(C1)C2 c1(CC)ccc(CCC(C)NC(C)(CCI)c2nnnn2C2CC2)cc1 N(C1CCCn2ncnc21)C(C(CN=[N+]=[N-])NC(=O)CSC1CC1)=O C1(C(N(C)Cc2c(C)n(C)nc2)=O)CC2CCN(CC(N)=O)CC12 N1(C(CN(CCOC)C)=O)CC(CNC(=O)CN2CCOCC2)CC1C C1(CC)C(C(=O)N(C2CCC2(C)C)C)CCN1C(=O)CNC(=O)OC c1(C(=O)NC(CC)CN(C(C2CCCC(N(C)C)C2)=O)CC)nc(C)ccc1C n1(CCC)ccc(C(=O)NC2(CCC(=O)NC(c3cnn(C)c3)CO)CCC2)n1 CCC(CC(=O)NCC(C(C)C)NC(C1(F)CCCCC1)=O)SC C(=O)(C1=CCOCC1)NCC(CNC(c1cc(C2CC2)no1)=O)OC C(C)(C)(C(=O)N(CCNC(c1cn(CC2CCCOC2)nn1)=O)C1CC1)N(C)C Cc1ccc(Br)cc1C(=O)NCCCCCCN(C(=O)C(C)C1CCCO1)C N1(C(C2CCCNC2=O)C(=O)NC)CCC(C)=C(Br)C1 c1(C(=O)NCCCN(C)C(c2coc(Br)c2)=O)cc(OC(F)F)cc(F)c1 C(=O)(C1=CCCSC1)NC1C(CCC)CN(C(c2c(C(C)C)cnn2C)=O)C1 c1(NC(=O)NCCOc2ccccc2Cl)ccc(NC2CNC(=O)C2)c(Cl)c1 c1(CN2CCC(C(=O)Nc3c(C(=O)OC)cnn3C)CC2)cc(F)c(Br)cc1F C(=O)(N=c1cc2n([nH]1)CCCC2)C1C(C)N(C(=O)CC=C(Cl)Cl)CC1 C1(CNC(C(C(CC)C)=O)=O)CCC2CN(C(=O)C=Cc3cnn(C)c3)CC12 C1(O)(CNC(=O)COCCF)COCCN(C(c2csc(-c3ncc[nH]3)n2)=O)C1 N1(C(C2(CC#C)CCCO2)=O)C2CCC1CN(C(c1cccc(CCO)c1)=O)C2 C12CC(F)CN1C(=O)C[SH2](=O)CC(=O)NC2.c1(CSC(C)(C)C)ccnc(O)c1 c1(CS(=O)(=O)NC(C#C)C2CCC2)ccc2ccccc2c1 C1(NC(C2(CNC(CCSCC(C)(C)C)=O)CC2)=O)CCCCC1 CN1C(=O)CCC1C(=O)N(C1CCCCC1)CCNC(=O)CC1(CO)CC1 c1(-c2n(-c3ccc(OC)cc3)nc(CO)n2)cc(F)ccc1O N1(C(=O)NC(C(=O)NC)Cc2cccc(Br)c2)CC(C(=O)OC)CC(C)C1 c1(N2CC(C(C)NC(=O)CCc3cnn(C)n3)C2)ccnc(-c2nccs2)n1 n1(CCC)nc(C(=O)N(C2CCNCC2)C(C)C)ccc1=O C1(NC(CC2(COC)CC2)=O)CN(C(=O)C(C)(C)CC2CC2)CC1C(F)(F)F C1(C)(CNC(c2cnn(CC)c2C2CC2)=O)CCN(C(=O)C2=CCOC2)CC1 Cc1cnc(NCC2CCCC2NC(=O)CSc2nc[nH]n2)nc1 Cc1cc(NC(c2nncs2)=O)ccc1NC(=O)CCn1cncn1 c1(C(=O)NCC#CCNC(C(C)OCCCC)=O)ccccc1NC(=O)CCC C1(NC(=O)C=Cc2cocn2)CC12CCN(C(=O)Cc1ccsc1)C2 N1(C(CSCC(=O)OC)=O)CCCC(CCC(=O)N)C1.N1(C(C)(C)C)CCN(C)CC1 CCC(C)(C)CC(=O)NCCCC(C)NC(=O)C(C)C1CC1 CCCCCCCN(C(=O)CCNC(C1CN(CC)CCO1)=O)C1CC1 c1(N(C)C)ncc2c(n1)CCC(NC(=O)C(=O)NCc1c(F)cc(F)cc1F)C2 C1(C(=O)NCCC2CC(C)C2)CCCC1CNC(c1coc(C(F)F)c1)=O c1(CC)oc(C(=O)NCC2CCN(C(c3cn(C)cc3C)=O)C2CC)cc1C N1(C(=O)Nc2cc(Cl)ccn2)CC(NCc2ccc([N+](=O)[O-])cn2)CC(F)(F)C1 C1(N(C(C2N(S(CC)(=O)=O)CCC2)=O)C)CC2CC1N(C(=O)CSC(C)C)C2 c1(CC)ccc(NC(C23CC2CCN3C(c2nnc(S)n2C)=O)=O)c(C)c1 c1(OC(F)F)cc(C)ccc1C(N1CCCC(N(C)C(C2(OC)CC2)=O)CC1)=O CC1CN(C(c2cnco2)=O)CCC1Nc1ncncc1Br C12(C(N3CCN(C(CCc4cc(C(C)=O)c(C)o4)=O)CC3)=O)CCN(CC1)CC2 C=C(C)CCCC(=O)N1CC(CNC(=O)CCC(=C)C)C(F)(F)C1 c1(C(N2CCC(N(C)C(c3ccc4[nH]ccc4c3)=O)C2)=O)ccc(C#N)cc1F CCCC(CC(C)C)C(=O)NCC=CC(N1CCOCC1C1CC1)=O C1(NC(CCSCC)=O)CC(CC(=O)NCc2ccc(SC)o2)C1(C)C N1(C(C(CC)=CC)=O)CCC(C)N(C(=O)C(c2ccncc2C)C)CC1 c1(C(N2CCC(NC(C(c3cnn(C)c3)OC)=O)C2)=O)n[nH]c(C2CC2)c1Br Cc1n[nH]c(C)c1S(=O)(=O)N1CCC2(CC1)CN(C(C1CC1F)=O)C2 c1(CC(=O)NC2CCC(CNC(CCC3CC(OC)C3)=O)C2)ccc(C)nc1Cl Cc1ccc(C(N2CCN(C)C(CNC(C3(CC(C)C)COC3)=O)C2)=O)c(O)n1 CCC(C)C(C)CNC(c1conc1C(C)NC(c1cnn(C)c1OC)=O)=O c1(C2N(C(=O)Nc3cccc(C(C)(C)C)c3)CCC2)ccc(F)cc1Br C1(NC(=O)C=Cc2c(F)cccc2F)CCC2(CCCN2)CC1 C(=O)(CC(C)C(C)(C)C)N(C(CC(=O)NCCCC#C)(C)C)C c1(CC)cc(C(=O)NC2CC2C(OC(F)(F)F)=O)cc(C)n1.CC Cc1coc(C(N2CC(NC(C3CC(C)CO3)=O)CC2C)=O)c1C C(C1c2ccsc2CCN1C(=O)C(C1CCOCC1)O)NC(=O)CCOC1CC1 Cc1c[nH]c2ncc(C(=O)NCCC3CCCCN3C(C3CC(C)(F)C3)=O)cc12 C(c1ccc2ccccc2n1)=CC(=O)NC12C(CN(C(c3c(OC)ccs3)=O)C1)C2 c1(CC)ccc(Br)cc1C(=O)NCC1(F)CCCN(C(c2nc[nH]n2)=O)C1 N1(C(COCCOCC)=O)CC(=O)NCC1C(=O)N(C)Cc1ccon1 C(=O)(C1=CC2(CCOCC2)C1)Nc1nc(CN2CCCC2)cs1.c12ncoc1c2=O N(C1c2ccccc2CC1NC(C12CCC(CC1)OC2)=O)C(CC1CC(=O)C1)=O c1(NCCC2(C(=O)OC)CCCC2)ccccc1C(=O)NC(C)CS(=O)(=O)O Cc1cc(=O)n(C)cc1C(=O)NC1(C)CCCC1C.c12cn(nn1)CCNC2=O Cc1ccc2[nH]c(C(N3CCC(C)C3CNC(C3C=CCCC3)=O)=O)cc2c1C c1(C(=O)NC2CC(NC(CC(C)n3cccc3)=O)C2)csc2c1CCCC2 Nc1ccc(C(N2CC(CO)(NC(C34CC=CC(C3)OC4)=O)C2)=O)cc1Cl N12CCCC3(CC(CO3)OC1=O)C2.C(=O)(C(=O)NCC(F)(F)F)C(C)(C)C C1(NC(Cc2ccc(CC)cc2)=O)CC2CC(C1)N(C(C1(C)CCN(C)C1)=O)C2 C1(C#N)(C(N2CCCN(C(C(=O)NC(C)C)=O)C(CO)C2)=O)CC2CCC1CC2 c1(C(=O)NC2CC(CCN(C(CNC(CC)=O)=O)CC)C2)[nH]nc2ncccc12 c1(-c2c(C#N)nccc2)nc2c(s1)CC(C(=O)NCCn1cc(CO)nn1)CC2 CC(C)(F)CC(=O)NC1CCN(C(=O)C2CC2)C1n1cccn1 Cc1cccnc1S(=O)(=O)CN1CC(O)C(F)C1 Cc1nc(C)n(CCC(=O)NC2CCN(C(=O)CSCCC(C)C)C2C2CC2)n1 c1(-c2scc(SCCNC(C(n3cc(C4(O)CCC4)nn3)C)=O)n2)ccc(F)cc1 c1(C(N(C)CCC2CCN(C(C3CC3Cl)=O)CC2)=O)ccnc2ccccc12 CCC(C)(CNC(=O)C(n1cc(Cl)cn1)C)NC(c1ccn(C)c1)=O c1(C(N2CC(NC(c3cc(C(C)=O)sc3)=O)C2)=O)cc(C)nc(O)c1[N+](=O)[O-] N#Cc1ccc(C(N2CC3CCN(C(C4CC(C(F)F)C4)=O)C3C2)=O)cc1F C1(C(=O)NCCN(C(=O)C(F)(F)CO)CCC)CC2CCCN2C(=O)N1 N1(C(C2CCCC2)=O)CCCC(O)(Cn2cc(CCC3CC3)nn2)CC1 Cc1ncnc(C)c1CC(N1CCC(NC(C2CC2(C)C(C)C)=O)CC1)=O N1(C(Cc2cn(CC)nn2)=O)CCOC(CCNC(=O)C(C)(C)CC2CC2)C1 C1(C(=O)NCCOCCNC(C(C)NC(CC)(C)C)=O)CCC(F)(F)CO1 N1(C(c2cc(C)sn2)=O)CCC2(CCC2NC(C2CNC(=O)CC2(C)C)=O)CC1 N1(C(C(CCSC)O)=O)CCN(C(=O)CC(C)N(C)C)CC2(CC2)C1 N1(C(c2ccc(OC)cn2)=O)CCN(C(=O)C=Cc2cncnc2O)C(CO)C1 CC1CC(NC(=O)CCC(C)(F)F)CN(C(c2cccc(C(F)F)c2F)=O)C1 N#Cc1cccc(CC(N2CCC(CN(C(C3CC4CCC(C3)O4)=O)C3CC3)C2)=O)c1 C1(c2cccs2)(CS(=O)(=O)N2CC(CCC(F)(F)F)C2)CCCCC1 Cn1ccc(-c2cc(C(N3CC(n4cc(C5(O)CCOC5)nn4)C3)=O)no2)n1 C1(NC(COC(C)=O)=O)CCCC(NC(=O)C(=O)Nc2cncc(C)c2)C1 c1(CC(=O)NCCN(C(=O)CC2CC=CC2)CC)ccc(O)cc1Cl c1(NC2(COC)CC=CCC2)nc(C(F)(F)F)nc2ccccc12 C(CCN=C1NCC2CCCCC2N1)c1c(F)cccc1 Cc1nc(Cl)ccc1CC(=O)NC1(C)CCN(C(c2[nH]nnc2C2CC2)=O)C1 N1(C(c2c(F)ncc(C)c2)=O)CC2CC1CCC2NC(=O)CSCCC(C)C C1(C(=O)NC(C#C)C(C)(C)C)CCC2(CC2)N1C(=O)CS(=O)CC Cc1cc(C(N2CCC(CCNC(c3csc(Cl)n3)=O)CC2C)=O)c(N)c(F)c1 c1(N2CCC(N(C)CC3CC3)CC2)nc(=NCC(CO)C2CC2)[nH]c2ccsc12 Cc1cnc2n1C(C(=O)NCC1CC(NC(=O)CNS(=O)(=O)C3CC3)C1)CCC2 C1(C(=O)NCC(CN(C)C(C2(C(C)(F)F)CC2)=O)O)CCOC1(C)C c1(CC(=O)N(CC(C)NC(C2(C(F)(F)F)CC2)=O)CC)cc(C)on1 c1(N2C(CCNC(c3ccc(CC4CCCC4)cc3)=O)CCC2)nccnc1F c1(C(N2C(C)CCCC2)=O)cc(F)c([N+](=O)[O-])cc1F c1(OC(C(N2C(CNC(c3cc(C)ncn3)=O)CCC2)=O)C)cccc(C)c1C N1(C(c2cc(-c3ccccc3F)on2)C)CCN(N2CCCC2=O)CC1C N1(C(C(CO)OC)=O)CC(C)(C(=O)NCCC2CC3C=CC2C3)CC1(C)C C12(C(N3CCN(C)CC3CCO)=O)COCC1CN(C(=O)CN=[N+]=[N-])C2 N1(N(C)Cc2cnn(C)c2)CC(C)(C)CC1C=O.C1(CC)CCOC1C=O C1(F)(CNC(C(C)NC=O)=O)CCCN(C(C2CCC2c2nc[nH]n2)=O)C1 CCC(O)C(C)(C)C(=O)NCC(CC(=O)NC1(CCOC)CC1)C1CCC1 Cc1cc(N2CCC(CC(=O)N(CCC#N)C)C2)nc(CO)n1 c1(C(N(C)CC2N(c3cc(OC)nc(C)n3)CCC2)=O)cc2cccnc2[nH]1 C1(CC(=O)NC2CN(C(C3CCC(CC)CC3)=O)CC2O)CCC(C)(C)CO1 N1(C(Cc2c(C)occ2)=O)CCC2(CCCCC2NC(c2cc(O)nc(Cl)c2)=O)C1 C=Cc1ccc(C(=O)NC2CCCN(C(=O)C=CSCc3ccco3)CC2)cc1 CCC(C)C(C(=O)Nn1nnc2c1CCCC2)NC(=O)C=CC(C)(C)C N1(C(CC(=O)Nc2c(OC)cccc2)c2ccccn2)CCCC2(C=CCO2)C1 CC(C(=O)N1CCC(CNC(c2ccc(C3CCC(=O)N3)cc2)=O)C1)C(F)F C(=O)(C(C)(C)CCOC)NCC12C(CN(C(C(C=C)(F)F)=O)C1)C2 c1(NC2(c3n(CCCOC)nnn3)CCCSCC2)ccc(F)c(S(N)(=O)=O)c1 Cc1csc(=O)n1CCC(=O)NCC1C=CCN1C(=O)CC1CCOC1 c1(OC)cc(CC(=O)NCC(CC(C)O)c2ccccc2)cc(OC)c1OC N1(C(Cc2cc(OC)c(Br)cc2)=O)CC2(CCC(N3CCC(F)(CO)C3)CC2)C1 O=C(CCCCCCCCCO)NC1CC2C1CCN2C(c1ccnc(S)c1)=O C1(CNC(CCc2onc(CCC)n2)=O)CN(C(c2ccc(F)o2)=O)CCO1 C(=O)(CCS(=O)(=O)CC(C)C)NCC(CCNC(C1CC=C(C)CC1)=O)O CCC(C)C(C(=O)NCC1CC2C=CC1CC2)N(C(=O)CSC)C CC1(NC(=O)CC2OCCCO2)CCC(NC(=O)C=Cc2cn[nH]c2)C1 C1(CN(c2ncc(C(=O)OCC)s2)C)C(C)CCN1C(=O)C=CC(=O)NC1CC1 CCC(CN(C)C)CC(=O)N1CCCC(NC(=O)C=Cc2cccs2)C1C C1(C)(C(=O)NC(CC=C)CC)CCCN(C(c2cc(CCC)nn2C)=O)C1 c1(C(=O)NC2C3CN(C(CCSC)=O)C(C3)C2)cc(Cl)cc2cccnc12 CCN=C(NCCC(C)F)N1CCC(F)(C#N)C1 S(=O)(=O)(c1c(Cl)cccc1Cl)N(C1CCNCC2CCCCC12)c1n(C)nnn1 N1(C(COCC(=C)C)=O)CCCN(C(=O)CSc2ccc(F)c(F)c2)CC1C C1(NC(c2c(C)nc(C)o2)=O)COC2(C1)CN(Cc1ccc(Cl)cc1F)C2 C1(COC(CC(C)C)=O)CC2OC1C1CC21.C(=O)(C)NCCNC(=O)NOC.C N1(C(CCC=CC)=O)CCC(O)(C(C)NC(=O)Cc2ccc(C)nc2)C1 C1(C)(CNC(CS(CC)=O)=O)CC(F)(F)CN1C(C1CC2(CC(=O)N2)C1)=O c1(-c2c(C)n[nH]c2)ccc(C(=O)N(c2ncncc2Cl)Cc2ccccc2)cc1F N1(C(C2N(C(CC)=O)CSC2)=O)CCC(NC(=O)CC(CC)CC)C12CCC2 N1(Cc2ccc(-c3ccc(C(=O)NC(C)(C)C)cc3)cn2)CCn2cncc2C1 Cc1ccc(Cl)c(OCC(=O)NCCN(C(C2C3CC4C(C3)C24)=O)C(C)C)c1 c1(N2CC(NC(C(=O)OCC)=O)C(F)(F)C2)ccn2ncc(I)c2n1 C=CCC(C(=O)NC(CO)C(=O)NCc1ncc(CC)s1)C(C)C N1(CC)CCC2=C(C1=O)C(c1ccc[nH]1)NC(=O)N2c1cccc2c1CCO2 C=Cn1nncc1C(N1CC(O)(CNC(=O)CC2CC2C)C1)=O Cn1ccc(C=CC(N2CCC(CCC(=O)NCC[Si](C)(C)C)C2)=O)c1 N1(C(COCCOCC)=O)CCCN(C(c2ccccc2-n2cncn2)=O)CC1 C(=O)(CN=c1[nH]c2ccccc2s1)N1CCCCC(NC(C(C)C)=O)C1 N#CC1(C(=O)NCCc2nc(O)n[nH]2)CC2CCC1C2 N1(C(C(C)(Cl)Cl)=O)CCC(OCCNC(=O)COc2ccsc2)CC1 Cc1cc(C(=O)NC2CC2NC(=O)CSCc2ccncc2)nn1C(F)F C1(NC(c2c(CC)n(C)nc2)c2nnnn2CCCF)CNC(=O)C12CC2 Cc1nnccc1C(=O)N(C(CNC(=O)CC1CC(C)(C)C1)C1CC1)C c1(C(N2CC(=C(CNC(COCCC=C)=O)F)C2)=O)cc(F)ccc1Br c1(C(N2CC(CCc3cn(CC(CC)CC)nn3)C2)=O)cc(C)ccc1F CC(C)C(C)CC(=O)NC(C1CC(NC(C2CCC(C(N)=O)C2)=O)C1)C N1(C(CC2CC(CC)C2)=O)CCCOC(CCNC(=O)CCn2cncn2)C1 c1(C(=O)NC2C(NC(=O)CCc3ccoc3)CC2)ccc(Br)o1 C1(CN(C)C(c2sccc2F)=O)CCCCN1C(c1ccc(Cl)nc1)=O C1(CNC(c2cc(CCC)nn2C)=O)C(C)CCCN1C(c1csnc1OC)=O Cc1nc(-c2ccccc2)ncc1C(N1CCCN(C(C2C(C)C2C)=O)CC1)=O c1(CC(=O)NC2CC(NC(c3c(CC)c[nH]n3)=O)C2)coc2c(F)c(F)ccc12 c1(C(=O)NC2CC(NC(C3CC(CCC)C3)=O)C(O)C2)ccc(C)nc1N C(=O)(C1=CCCC1(C)C)NCC1N(C(Cc2cccc(NC(CC)=O)c2)=O)CC1 C(CC(F)F)(C(=O)NC(C)CCN1CCCC1)NC(CCCC)=O N1(C(C(C)(C)OC(C)C)=O)CCCCC(COC(=O)NCc2ccc(Cl)cc2)C1 C1(C(=O)OC)N(C(C2(NC(=O)C=Cc3ccccc3)CC(F)(F)C2)=O)CC1(C)C C(=O)(C1=C(C#N)CCC1)N1CCN(C(Cn2c(=O)sc(C)c2C)=O)CC1C(C)C CC(=O)CCCCCCC(=O)N1CCC2(CCOC2)C(C)C1 C1(C(=O)NC(c2nccn2C)CC)CCCCC1CNC(=O)CCC=CC(C)C N1(C(=O)C(O)CC2CC2)CC(F)CC1CNC(=O)C(F)(F)Cc1ccc(F)cc1 C1(NC(C2C(OCC)C2C)=O)CN(C(=O)CN2CCC(C)CC2)CC1C N1(C(C2CN(C(C(CC)NC(N)=O)=O)CC2C)=O)CC2CC1CN2C C1(NC(c2cnc[nH]2)=O)CC2(C1)CN(C(C1CC=CCC1)=O)C2 C1(C(=O)NC2CC(CNC(C34CCCC3C4)=O)C2)CCCN2CCCC12 N1(c2n(CC)c(C(O)Cc3ccccc3)nn2)CCCCC(S(C)(=O)=O)C1 C1(CNC(CN(C)C(=O)C2CC2)=O)(NC(C2CCSCC2)=O)CCOC1 c1(NCc2c(C)nn(-c3ccccc3)c2Cl)cc2ccncc2c(O)n1 C1(COC)(NC(=O)CCCc2nc(C3CC3)no2)CC1(F)F c1(C(=O)NCC(CC)NC(C2(N(CC)CC)CCCC2)=O)ccc(SC)s1 C1(C(=O)NCCCCN(C)C)CCOCC1NC(c1nccnc1N)=O C1(CNC(CCCc2ccc(OC)cc2)=O)CN(C)CCN1C(=O)C1=CCCC1 N1(C(C(C)CF)=O)CC=C(CCNC(c2cc(-c3ccccc3Cl)no2)=O)CC1 CC(C(=O)OCc1ccccc1)=NOCc1nc(C(F)(F)F)no1 C1(C(=O)NCc2cccc(-n3cc(C(CSCC)C)nn3)c2)CCC2(CCC2)C1 C(CNC(c1cccc(OC(F)F)n1)=O)(C(C)(C)C)NC(C(CN(C)C)O)=O n1(CC(N2CCCC(NC(c3cccnc3Br)=O)CC2)=O)cnc2ccccc12 c1(OC)cc(C(=O)NC2(CNC(C3CC(O)C3)=O)CC(OC)C2)sn1 C1(NC(C2(OC)CCC2)=O)CCN(C(=O)CC2CCC3CC23)CC1O C(=O)(C#CC1CCC2(CC1)OCCO2)NC1CCN(CC(=O)OC(CCCCC)C)C1 Cc1c(C(=O)NC(C)CC2CN(C(c3cn(C)nc3C3CCC3)=O)C2)nnn1C C1(C(=O)NCCC(C)(C)NC(c2c(C)cc(C)o2)=O)CC2(C1)NC(=O)NC2=O N(C1CCc2cc(CNC(=O)C3CC3)ccc21)C(c1ccc(C(C)(C)C)cn1)=O Nc1ccc(F)c(C(=O)NCCCOCCNC(c2ccc([N+](=O)[O-])o2)=O)c1F C(CC(C)(C)CC(=O)N(C)CCOCCC(=O)NCc1ccc(C)s1)OC CCC(CC(C)C)C(C(=O)NCCOCC1CC1)N1CC2COCCC2(CSC)C1 C1(C(C)C)COCCN1C(=O)CCN(CCCO)C(=O)COC(F)(F)F CCCCCC(O)C(=O)N1CCC(NC(c2nn(-c3ccccc3)nc2Br)=O)C1 C1(NC(C=Cc2ccc(CC)o2)=O)CC2CN(C(=O)C=CS(C)(=O)=O)CC2C1 n1(CC(=C)C)nc(-c2ccccc2)nc1C1CCCCN1C(=O)N(C)C c1(OC)cc([N+](=O)[O-])ccc1C(N1CCN(C(=O)COCCSC)CC(O)C1)=O Cc1nc(C(=O)NCC2CC(NC(=O)CCc3ccc(Cl)s3)CC2O)n(C)n1 c1(C(N2CCC(CC)C2C(=O)NCc2nnn(C)n2)=O)cc(O)cc(F)c1 N1(C(C(C)C2CCCO2)=O)CCN(C(c2ccno2)=O)CC1CCO c1(C(=O)NCCOCC(N2CCC(CC)C2)=O)ccc(C)cc1C c1(C(=O)NCC2CCN(C(CCC=C=C)=O)C2)cc2cccc(C)c2[nH]1 Cn1cnc2c(C(=O)Nc3ccc(NC(c4n[nH]cc4Cl)=O)nc3)cccc12 c1(C(=O)NCC(CN(C)C(C2CCCN2CCCO)=O)(C)C)ccc(CO)cc1 C1(CNC(CC(CC)C)=O)CC(C)CN(C(c2cccc(-n3ccnn3)c2)=O)C1 c1(C(N2C(CNC(C3C(=C)CC3)=O)CCCC2)=O)cc(C)c(N)cc1F C(=O)(C1CCCn2nccc21)NCCC1(OC)CN(C(=O)CC(C)(O)C2CC2)C1 CC(C(=O)NCC(C1CC1)N(C)C(C12CC(C)(CCO1)C2)=O)C(C)(C)C C12CC(O)CN1C(=O)CCC1CCC(C1)NC2=O.C1(CC)(OC)CCC1 c1(OC)cnc(Cl)cc1C(=O)N(CCCNC(C1CC12CC2)=O)C(C)C C1(C(N(C(C)CNC(=O)C(C)(C)C2CCCC2)C)=O)CC(O)CN1C c1(CCC(=O)NC(CCOC)CNC(c2ocnc2C2CC2)=O)ccccc1Cl N1(C(c2c(C)nc(C)c(C)n2)=O)CCCC2(CCN(C(=O)CC(F)(F)Cl)C2)C1 C1(NC(Cc2n(C)ncc2Cl)=O)CC(O)CN(C(c2cnc(O)cc2O)=O)C1 c1(C(=O)NC(COC)CC(=O)NC2C=CC(CO)C2)cc2cccnc2[nH]1 c1(C(=O)NCC2C(CNC(c3c(C)cc(F)cc3)=O)C2)cc(N)cc(O)c1C c1(C(=O)NC(C2CCCN2C(C2CC2C2CC2)=O)C)cccc(C2CC2)c1 c1(NC(C)=O)c(C(=O)NC2CC3CN(C(c4ccnnc4Cl)=O)CC23)cccc1C C1(C(=O)NC(CNC(C(CSC)O)=O)(C)CO)CN2CCN1CC2C C1(CNC(c2ccn(C(C)C)n2)=O)CN(C)CCN1C(=O)C(N1CCNC1=O)C N1(C(C2(C)C(C)CN(C(C(CSC)OC)=O)C2)=O)CCN(C)C2(CCC2)C1 N1(C(C2CCn3ncnc3C2)=O)CCN(C2CCC2)c2ccccc21 c1(C(=O)NCC2CCN(C(c3ccc(C(=O)NC)nc3)=O)CC2)cc(O)cc(=O)o1 c1(C(C(=O)N(CCNC(c2cnn(C(F)F)c2)=O)C(C)C)OC)ccccc1F C1(C(CNC(C(C)n2cnnn2)=O)O)(C(=O)NC2(Cl)CCC2)CCCC1 N1(c2nnc(-c3c(OC(C)C)c(Cl)ccc3)n2C)CCC2(C1)CN(C)C2 c1(OC)cccnc1C(=O)NCC12CC1CN(C(C1C3COCC13)=O)C2 N1(C(CCCOC)=O)CCCCC(NC(=O)C=CC2(C)COC2)C1 c1(CC)ccc(N)c(C(=O)NC2CCCCN(C(=O)CC3CCC4CC34)C2)c1 N1(C(c2ccn(CC)n2)=O)CC(NC(c2ncccc2OC)=O)CC2(CC2)C1 c1(C(=O)NCC(CN(C(C2CC(CC)C2)=O)C)O)cccc2[nH]ccc12 c1(C(=O)NC2CCCCCN(C(C(C(C)O)(C)C)=O)C2)cn(C)c2ncccc12 C(C1CCOc2ccccc21)NC(C(=O)N(C)Cc1ccc(OC)c(OC)c1)=O N1(C(C(=O)NC2C(=C)COC2)=O)CCOC(c2ccccc2C(F)(F)F)C1 c1(CC)ccc(C(=O)NCC(C2CCN(C(C3(O)CCOC3)=O)CC2)F)cn1 c1(CC)cc(C(=O)NC2CN(C(=O)CC3CCOC3=O)CC2F)cc(Cl)c1 C(N=c1[nH]nc2ccc(Cl)cn12)N.c12cccc(c1)N2C(=O)OCC.C(C)(C)(C)O c1(NC(c2c(C)nns2)C)nccc(=NCC2C(F)(F)C23CCCC3)[nH]1 C#CCC(CC#C)C(=O)N(CCCNC(C1(O)CN(C)C1)=O)C(C)C C1(CC(=O)NCCCOCCN(C(=O)CCF)C)(C(F)(F)F)CCC1 C(C(C)(C)CNC(=O)COCC1CCCOC1)N(C(C1C(OCC)CC1)=O)C N1(C(C(C)NC(CC)=O)=O)CC2CCN(C(c3ccc(NC)cn3)=O)CC2C1 C1(C2CC2)(C(=O)NCC2(F)CC(NC(CN(C)CCO)=O)C2)CCOCC1 CC(C)C(C(C)NC(=O)CC(C)(C)C)NC(c1ccnc(C(F)(F)F)c1)=O C1(CNC(c2cc(OC)cc(F)c2)C)C2CC1N(C(=O)OC(C)(C)C)C2C c1(C(=O)NCC2CN(C(C3CC34CC4(F)F)=O)C2)cccc2c3c([nH]c12)CCC3 N1(C(C(C=C)(C)O)=O)CCN(C(c2cc(C3CC3)n(CC)n2)=O)C(CC)C1 c1(NC(C2CC(O)CN2C(=O)C2CC2)=O)cnc2cccc([N+](=O)[O-])c2c1 c1(C(N2CCC(O)(C(C)NC(c3nc(CCC)sc3)=O)C2)=O)cnc(O)c(F)c1 C1(C(N(C(C(=O)OC)C)C)=O)(NC(=O)CCc2nccs2)CCC(C)(C)C1 c1(OC)cccc(C=CC(N2CC(NC(c3scnc3C)=O)C(C)C2)=O)c1 C1(NC(CC(CNC(CCCCCSC)=O)O)=O)CCC(=O)NC1(C)C C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NC(CCOC)COC C(=O)(CCCC(F)(F)CO)N1CCCC(N(C(C(C)C2=CCCC2)=O)CCO)C1 C1(CNC(c2ccc(COC)cc2)=O)(NC(=O)CNC(C)=O)CC2CCC1C2 C1(=CC(=O)NCC(CCNC(C2CC=C(C)CC2)=O)O)CCOc2ccccc21 N1(C(C(C)OCCC=C)=O)CCCC(NC(C2CCCC(=O)N2)=O)CCC1 CC(C)C1=NOC(C(N2CC(F)(F)CC2CNC(=O)C=Cc2ccc(Cl)s2)=O)C1 O=C(O)CC(CN(C(c1cnn(CCN2CCCC2=O)c1)=O)CCO)C1CCCC1 c1(C(=O)NC2(C)CCN(CCCCCC)CC2)cccc2occc12 C1(NC(C2C(=C)C2)=O)CN(C(c2cnn(Cc3ccccc3)c2N)=O)CCC1O CC1(C)CC(F)(F)CCC1C(N1CCN(C(c2ccccc2)=O)C2(CC2)C1)=O c1(OC)cc(C)c(CC(N2CC3(CCCN3C(c3ccoc3C)=O)C2)=O)c(C)c1 c1(C(=O)NC(CC=C)CNC(C2C=CCCC2)=O)ccc(CO)cc1F c1(COC)cc(C(=O)NC(Cc2ccc(C(F)(F)F)cn2)CC(=O)O)sc1C N(C1CCc2c(C)cccc21)C(=O)Nc1n(C)nc(C)c1Cl C1(OC(C)(C)C)CCCC(CCNC(=O)NCc2cc(=N)[nH]o2)C1 CC(O)C(C(N)=O)NC(c1ccc(CNC(c2ccc(N)cn2)=O)cn1)=O N1(C(C2(SC)CC2)=O)CCC2CN(C(=O)C3=NOC(C(C)(C)C)C3)C2C1 CC1CC(c2cn(CC(F)(F)F)nn2)CCN1C(c1cc(Cl)sc1Br)=O CC1CN(C(c2ccccc2C(=O)NC2CCC2(C)C)=O)CCC1.C(CO)NC C1(CSC)CCN(C(c2ncnn2C(C)(C)C)C(=O)NCC(C)C)CC1 c1(C(=O)NCC2N(C)CCN(C(c3ccsn3)=O)C2)nc2cncnc2nc1O C1(OC)CN(C(=O)CCC2CCCOC2)CC1NC(c1cc(C)cs1)=O N1(CC(C)NC(C2C(C)C2(F)F)=O)CCN(C(C2CC3C=CC2C3)=O)CC1 C(=O)(CC1COc2ccccc21)N(CC(C)(C)NC(c1ccc([N+](=O)[O-])[nH]1)=O)C Cc1ccc(C)c(OCCC(N2CC3(NC(=O)CC4CC(CF)C4)CC2C3)=O)c1 C1(C)(C(=O)NC2CC3C(NC(CC(CC)C4CC4)=O)C3C2)CC2C=CC1C2 N1(C(C2CCC(C)(CC)O2)=O)C2CCC1CC(NC(=O)CN1CCCCCC1)C2 C12(CCC(=O)OCc3ccn(C)c3)CCC(CC1)C2 c1(NC(=O)NCCC(=O)NCc2ccccc2Br)cccc2c1NCC2 c1(C(N2CCC(NC(CCC=C(C)C)=O)C2C)=O)nc(Br)n2ccccc12 C1(NC(C(CC)CC2CCCC2)=O)CN(C(C2(O)CCOCC2)=O)CC(F)(F)C1 C1(NC(C(C(C)C)N2CCCCC2)=O)CCc2nnc(-c3ccccc3)n2C1 N1(C(CSCC=C)=O)CC2CC1CCC2NC(c1ccc(C(C)(C)C)c(Cl)c1)=O N1(C(C2(C#C)CC2)=O)CCC(N(C(=O)Cc2ccn(CC)n2)C)C1 Cn1cc(C(N2CC=CC2CNC(=O)CCN2CCOCC2)=O)cn1 C1(c2n(CCCSC)nnn2)(NC2CCC3(CC2)CC3)CCCC(C2CC2)C1 c1(CN(C(=O)NNC(=O)c2coc(N(C)C)n2)CCC)cccc(Cl)c1 N1(C(c2nc(SC)sc2)=O)CCCCC(NC(c2cncc(N(C)C)c2)=O)C1 CN1CCC(C(N2CCN(CC(C)NC(=O)C(C)(C)CO)CC2)=O)CC1=O C(c1cc(F)c(O)c(F)c1)=CC(=O)NC(CNC(c1cnnc(O)c1)=O)C1CC1 c1(CC2CC(N(C)C)OC2)ccc(C(=O)NOCCOCCOCC2CCC2)[nH]1 N1(C(CCc2ccc(C)o2)=O)CCC(NC(C2CCN2S(C)(=O)=O)=O)C(O)C1 N1(C(C(=O)N(CC(CC)(C)OC)C)=O)Cc2ccc(O)cc2C1 N1(C(c2scc(C)c2C)=O)CC2(CCN(C(=O)Cc3ccsn3)CC2)C1C(C)C C12(C(=O)NC3CCN(C(COCCC)=O)C3C(C)C)CC=CCN1CCC2 c1(C(=O)NCC(C)CNC(=O)CCc2ccc(O)c(F)c2)ccc2nn[nH]c2c1 c1(C(N(C)Cc2ncon2)=O)cn2c(n1)CCN(C1CCC(C)(C)C1)CC2 N(C(=NCCc1cccc(C)n1)NCC1CCCCO1)C(C#C)C(C)C N1(c2ccnc(C)n2)CC2CCC(NC(c3coc(C(C)C)n3)=O)CC2C1 c1(CC(=O)NCCOCCNC(=O)Cc2ccns2)ccc([N+](=O)[O-])cc1Cl C(=O)(CC(C(F)F)NC(C1(CC2CC2)CCC1)=O)N(C(c1ccccc1)C)C1CC1 C(=O)(C(C)(O)C(C)(C)C)N(C)CC1CCCN1C(C1CC2(CCC2)C1)=O c1(OC)ccc(CN2CCC2C(=O)Nc2nc(Br)ccc2C)cc1C(F)(F)F C1(COC)(CNC(=O)CCC2CC2(Cl)Cl)CCCN1C(=O)Cc1c(C)noc1Cl C1(NC(CCc2ccc(C#C)cc2)=O)CC2CCCC(C1)N2C(=O)CC Cc1ccncc1C=CC(=O)NCCCN(C(c1cc(=N)[nH]c(=N)[nH]1)=O)C(C)C C#Cc1ccc(C(=O)NC2(CF)CCN(C(=O)C(C)NS(C)(=O)=O)C2)c(F)c1 CC1CN(C(=O)C(C)N(C)C)CC1CC(=O)NC(C(N)=O)C1CC1 C1(C(=O)N(C2CCN(CCOC)C2)C2CC2)CN(C(=O)CN2CCCC2)CC12CC2 Cc1occ(C(F)(F)F)c1C(N1CC(CCNC(c2cn[nH]c2)=O)C(C)C1)=O c1(C(N(CC(C)NC(C=CCC)=O)C)=O)ncnc(C)c1C N1(C(C(CC2CCC2)NC(Cc2c(C)n[nH]c2)=O)=O)CCOC(CN=[N+]=[N-])C1 c1(C(=O)NC(CNC(C2(COCC)CC2)=O)(C)C)nn(C)c(=O)cc1C C1(C(N2CCC(N(C(=O)C(C3CCC3)OC)CC)C2)=O)CCC(C(=O)OC)CC1 C1(C)(CNC(C2C(NC(C(C)OCOC)=O)CC2)=O)CC=CCC1 Cc1c(NCc2conc2C(F)(F)F)ncc2ccccc12 N1(C(C2(Cc3ccccc3)CC=CCO2)=O)CCCCC1CC(O)C(F)(F)F c1(C(=O)NC2(C)CN(C(C3(CO)CC(C)(C)C3)=O)C2)cc2ccsc2s1 S(=O)(=O)(c1cccnc1NCC1CC1NC1CC1)N1CCC(=C)CC1 c1(CC)ccc(Br)cc1C(=O)NCC12CC1CN(C(=O)C(C1CC1)OC)C2 c1(C(=O)NC2(CF)CCN(C(c3c(C)n[nH]c3C)=O)C2)ncc2[nH]ncc2n1 c1(N(CCC)C(C23CC(CO)(C2)C3)=O)ccc(Cl)c(OC)c1.c12cnc(nc1)[nH]2 C1(NC(c2cnc(OC)c(C)n2)=O)CCC12CCN(C(=O)CC(Cl)Cl)CC2 Cc1sccc1C(=O)NCC(F)CNC(=O)C(F)(F)C1CCOCC1 C1(CC)CN(C(=O)CC2CCN(C)C2=O)CCN1C(=O)Cc1ccc(OC)nc1 C1(CNC(COc2cc(C)on2)=O)CC12CCN(C(=O)Cc1ccc(Cl)s1)CC2 c1(OC)cc(C(N2CCC3C(NC(=O)CCN4CCCC4=O)C23)=O)ccc1C#N O=C1CN(CCCCCc2cccs2)C(=O)N1CCCC1CCCCC1 C12(CNC(C(c3cccnc3)C)=O)CC(CN1C(=O)CNC(c1cccnc1)=O)C2 C(C(C)(C)C(=O)NC1CC2(C1)CC2NC(=O)CCNS(=O)(=O)C(F)(F)F)OC c1(CCC(=O)NCCCNC(C2CC=CCC2)=O)cnc2n1CCOC2 C1(NC(c2nc(COC)sc2)=O)CN(C(c2cc(C3CCC3)[nH]n2)=O)C(C)(C)C1 N1(C(C(C)OCC2CC2)=O)CCC2(CCCCN(C(=O)C(=O)NC3CC3)C2)C1 N1(C(CC)=O)CCCCC1CNC(C1(CS(N)(=O)=O)COC1)=O c1(CC2CCC2)cc(O)ncc1-c1nc(C2(C)CC2)nn1Cc1ccc(Cl)cc1 C1(C#N)(C(=O)NC2(C)CCN(C(C3CCCS3)=O)C2)CC2CCC1CC2 C(CC(C(=O)NC(C)(C)CN(C(=O)CCc1ccco1)C)OC)OC C=CC1(C(=O)NC2CC(NC(=O)CSC)C2)CCCCC1 C1(NC(=O)Nc2c(OCC)ccs2)CCCCCC1c1ccccc1 CC1CN(C(c2cnc(C3CCCO3)s2)=O)CCN1C(c1cc[nH]n1)=O c1(C(N2CCC(O)(C(=O)Nc3ccncn3)C2)=O)ccc(F)cc1 C1(CC(C)NCCCc2ccn(C3CCCC3)n2)CCN(C(C(C)(C)C)=O)CC1 c1(C(N2C(C(C)(C)CNC(C34CC(C3)C4)=O)CCC2)=O)cnc2n1CCOC2 C=CCCC(C)(C)CNC(C(CC)CC)c1nnnn1C1(C)CC1 N1(C(c2nc(NC(c3cc(I)ccc3F)=O)sc2)=O)Cc2ccccc2C1 N1(C(C2N(C(CSCCC(C)C)=O)CCC3(CC3)C2)=O)CCc2ccncc2C1 c1(N(C)CCN2CCCCCC2)cc(N2CCC(c3cc[nH]c(=N)n3)CC2)ncn1 CC(C)CC(C)(CNC(=O)CCOC1CC1)NC(=O)CSCc1cscn1 Cc1nc(CNC(C2CC3CC3C2)CO)no1 C(=O)(CC1=NN(C)C(=O)C1)N(C)CC1(O)CCCN(C(C(C)SC(C)C)=O)C1 CC1CN(C(c2ccnc3ccnn23)=O)CCCN1C(C1CC=CCC1)=O N1(Cc2cnc(CC)s2)CC(NC(c2cc(Cl)c(Cl)c(Cl)c2)=O)CC(F)(F)C1 C1(NC(C(C(C)C)O)=O)CS(=O)(=O)CC1NC(c1c[nH]ccc1=N)=O C(=O)(C(CC(C)C)C(C)C)NCC#CCNC(c1c(C)nc(N)cn1)=O N1(CC(=O)NC(C2CCCN2C(c2cc(Cl)ns2)=O)C)CCC(C)(O)C1 C(C)(CC(=O)N1CC(F)(CNC(C2(C)CC2(F)F)=O)C1)(C(F)F)N(C)C Brc1ccc(CN2CCOCC2)c(N2CCOC(c3cccs3)C2)c1 N1(C(C(CCC)c2ccccc2)=O)CCCC(NC(=O)C(F)(F)CN(C)C)C1C C1(C(N2CCC(O)(CCNC(C(CC)C#N)=O)CC2)=O)CCC2(CCOCC2)O1 c1(C(=O)NCCc2c(OC)c(Cl)ccc2)ccc2nc(F)ccc2c1O c1(C(N2C(C(=O)NCC(C)(O)CCO)CC(C)C2)=O)ccc2n[nH]cc2c1 c1(CNC2C3CN(C(C4CCC(OC)CC4)=O)CC32)cc(C)c(Br)cc1F N1(N2CCc3ccc(Cl)cc32)CC2CCN(C=O)CCC2C1.C1(C(=O)O)(C)CC1 CCC(CC(=O)NC(C)C(C)(C)CO)N(C(=O)C=CC1(C)COC1)C Cc1c(C(N2CC(O)CC2(C)C(=O)NC2CC(C)C2)=O)[nH]ccc1=O CCCC(O)CC(=O)NC1CN(C(=O)Cc2ccc(C3CC3)cc2)CC1CO c1(C(=O)NCCNC(C(CC2CCCC2)OC)=O)cc2c(Br)cccc2[nH]1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC(C(C)NC(CCC(C)C)=O)C Cn1ncc2cc(C(=O)NCC3CCC3NC(c3cc(O)nc(O)n3)=O)sc12 c1(OC)cc(OC)cc(C(=O)N(C)CC2CCCN2C(=O)CN(S(C)(=O)=O)C)c1 C(N=c1[nH]c(=NC(C)c2ccc(Br)c(F)c2)[nH]c2c1SCC2)c1cc(C)on1 C(C1CC1)(C1CC1)=CC(=O)NCCOCCC(=O)NC1CN(c2ncco2)C1 c1(C(N2C(C)CCC(NC(Cc3cc(C)sc3)=O)C2)=O)ccc(N)cc1[N+](=O)[O-] C1(NC(c2c(C)scn2)=O)CN(C(=O)CC=CC(C)(C)C)CCC1CO N1(C(C2CC2CNC(C2(NC(C)=O)CC2)=O)=O)CCCN(C=O)CC1 N1(C(=O)Nc2c(COC)occ2)CC=C(c2cccc(C)c2C)CC1 C1(NC(CCc2c(C)cccc2)=O)CN(CC(C2CCCOC2)=O)C(C)CO1 N1(C(C(CC)C#N)=O)CCOC(C)(CNC(c2ccnn2CC)=O)C1 Cc1c(C(=O)NC(C)C(C)NC(c2cncc(F)c2)=O)cccc1C#N C(=O)(CC(C)C(F)F)N1CC(OC)C(C(=O)NCc2cccc(C)c2O)C1 C(CCC(=O)NCCc1ocnc1CNC(C1(C)CC1(F)F)=O)OCCC C(CCCC(=O)N(C)CC1CCCN(C(=O)CCSc2ccccn2)C1)OC N1(C(C2=NOC(C)C2)=O)CCN(C(=O)Cn2ncccc2=O)CC(O)C1 c1(C(N2CCCC(CNC(C3CCC(O)C3)=O)C2)=O)nnn2c1CSCC2 C(C(CNC(=O)C(CSC)NC(=O)CNc1ccccn1)C(C)C)OC c1(OC)ccc(C(=O)C(=O)NCC2CCC(C)CN2C(c2cccs2)=O)cc1Cl c1(C(=O)NC2CC3(CN(C(CC(COC)COC)=O)C3)C2)ccn2nncc2c1 c1(NC(c2nnnn2CC2CCOC2)(c2ccccc2)COC)cncnc1C C1(CNC(C2CC=CCO2)=O)CCN(C(c2cnnc(O)c2)=O)CC1O N1(C(c2nc(CC)oc2)=O)CCC(O)(C(C)CNC(=O)CCCC2CCCC2)C1 c1(OC)c(O)cc(C(N2CCCC2C(=O)Nc2cnc(C)c(Br)c2C)=O)cc1Br C12(C(N3CCC(O)(C(CNC(C(CCSC)O)=O)C)C3)=O)CCC(O)(CC1)CC2 C(=O)(C(O)CC(C)C)NC(C(C)(C)NC(C1(CCOCC)CCCC1)=O)C C1(C(=O)NC(COC)CNC(=O)C(F)C2CCOC2)CCC([N+](=O)[O-])CC1 N1(C(CC2(C=C)CC2)=O)CCC(O)(CNC(c2cnc(C(C)(C)C)[nH]2)=O)C1 C(=O)(C#CC(C)(C)C)NC1CC(N(C(CC(c2c(C)cccc2)C)=O)C)C1 C1(C(=O)NCCn2ncc(C)c2)CN(C(=O)CC23CCCC2C3)C(C)(C)C1 c1(OC)cc(OC)c(Cl)c(C(N2CC3(NC(=O)C(C)N4CC(C)C4)CC2C3)=O)c1 CC1(C#N)CCN(C(C2(C)CCN2C(C2C3COCC23)=O)=O)CC1 CC1C2CCC(C2)C1C(N1CC2(C)CC1(C(=O)NC1CCCCCC1CO)C2)=O c1(C(N(C)CC2CCC(F)(F)CC2)=O)cc(S(=O)(=O)N2CCCC2)cn1C C=CC(C)C(=O)NCC(C)CNC(=O)C(c1cncn1C)O C(=O)(C(CO)C(F)(F)F)N(C1CC(C(=O)NC(C2CCCO2)CC)C1)C C1(C2(NC(=O)CN3CCCC3)CC2)CCCCN1C(=O)CCN1CCCCC1 Nc1c(NC(=O)NCC(=O)NCC2CCOC2)cc(F)cc1F C(CC(C)C)(C(=O)NC(Cn1cncn1)C(=O)N1CCC(c2nn[nH]n2)C1)OC CC1CCCC(C)CN1C(=O)CC(C)(C)CNC(C1(C#N)CC1(C)C)=O C(c1cc(OC)cc(OC)c1)=CC(=O)NC(C(C)NC(C(CC)CC)=O)C C1(C)(C(=O)NC(C(=O)OCCC)C)CC(O)CN1C(=O)CCc1cc(C)on1 c1(CC(=O)N(CCN(C(c2c(NC)cnnc2)=O)C)C(C)C)csc2nccn12 C1(C)(OCC(=O)N(C(C)CN(C(=O)Cc2ccsn2)C)C)CCCC1 C1(C(=O)NCC2(C(=O)NOC(c3nnc(O)o3)C)CC(=C)C2)CSCC(=O)N1 C1(NC(c2c(OC)nsc2)=O)(CO)CCCN(C(c2n[nH]cc2C)=O)C1 N1(C(C2=CC(C)(C)C2)=O)CCC(NC(C2CCC(C3CC3)CC2)=O)CC(C)(C)C1 C(=O)(CCC(C)(C)CC)NCCOC(CNC(c1nc(CC)oc1C)=O)(C)C N1(C(CSC)=O)C2CCCC1CN(C(c1cn3ccccc3n1)=O)C2 c1(N2CC(C(C)NC(C(c3cccnc3)OC)=O)C2)nn2cc(C)nc2s1 N1(C(c2c(C)ocn2)=O)CC(N(C)C(C2CC2[N+](=O)[O-])=O)C(C)(C)C1 C1(C(=O)NCCN(CCOC)C(c2cc(Cl)ncc2O)=O)CC2COCC(C1)C2 N1(C(c2c(C)cc[nH]2)=O)CC2(CCN(C(C3CC3c3ccccn3)=O)CC2)C1 N1(C(C2CCSC2)=O)CC2CCC1C(CNC(C13CCCN1CCC3)=O)C2 N1(C(CC(COC)C)=O)CCN(C)C(C(N2CC(CO)C2(C)C)=O)C1 C1(NC(C2(OC)CCOCC2)=O)CC1C1CCCN(C(=O)CCC2CCOC2)C1 Cc1cc(Cl)ccc1OCC(=O)Nc1ccc(NCC(C)(C)NC(=O)CO)nc1 C1(NC(c2cnnc(Cl)c2)=O)CCCCC1NC(c1occc1Br)=O C1(C(=O)NCC(C)C)COCCN1C(c1cnc(Br)s1)=O C1(C(=O)NC(C2CCOCC2)CC)CCCCC1NC(c1nnsc1C)=O N1(C(C=C(C)c2cnn(C)c2)=O)CCC2(CCC2)C(CNC(=O)C(F)=C(C)C)C1 c1(C(C(=O)N(CC=CC(=O)N(C)CC2CCO2)C)F)ccccc1 C1(CCNC(C(F)=C(C)C)=O)CCCN(c2nnc(C#N)s2)C1.C12CN(C1)C2=O C1(C(=O)NC(C)(C)CCNC(C2CC2(C)C)=O)CCS(=O)(=O)C12CCC2 N1(C(c2c(COC)cno2)=O)CC=CC1(C)C(=O)NCCNC(=O)C1CC1 c1(C(C(=O)N(CC(=C)C)C2CCC2)(C)C)c[nH]c2ccc(Br)cc12 c1(C(=O)NC2C(CNC(C3N(CC)CC3)=O)CCC2)ccc(N)c(F)n1 N1(C(CCCCN(C)C)=O)CCCC(C2(NC(=O)C3Cc4ccccc43)CC2)C1 C1(C)(NC(c2ccn(C)c2)=O)CCC(NC(=O)Cc2c(Cl)cccc2Cl)CC1 c1(C(=O)NCC(N(C)C(C2(Cl)CC2)=O)C2CC2)cc(Br)cc([N+](=O)[O-])c1 Cc1ncnc(O)c1CCC(=O)NCC(C)(CO)NC(C12COCC1C2)=O C1(F)(C(=O)NCC2(C(C)(C)O)CN(C(c3cnc(C)n3C)=O)C2)C2CCCCC12 O(C1CCSc2ccccc21)C(C1CCCCN1C1CCCC1)=O C1(=O)C(C(C)O)N1.c1(CC)cc(C(=O)N(CC(=O)NC)C)[nH]n1 N1(C(=O)CC2(c3ccccc3)COC2)CC(C(N2CCCC2)=O)C2(CC2)C1 C1(CNC(CSCCOC)=O)CN(C(=O)Cc2ccnnc2O)CC(C)(C)O1 C1(C(=O)NCc2ccncc2)(CC)CCCN(C(=O)CC2CCC(=O)N2)C1 c1(C(=O)NC2CC(C)(NC(C(CC=C)N(C)C)=O)C2)ccc(N)cc1Br C1(SCC)CCC(C(N2CCCC2(c2ccccc2)C(=O)N(C)C)=O)CC1 N1(C(CN2C(=O)CSC2)=O)CCN(C(c2cccc3cc[nH]c23)=O)C2CCC12 c1(CC)[nH]nc(C(N2CCCC2CN(C(C2C=CC=CC=C2)=O)C2CC2)=O)c1Cl N1(C(C2C(CC)C2)=O)CCC(CNC(=O)C2=CC(C)(C)C2)C(CC)C1 c1(SC2(CS(=O)(=O)Nc3cnc(OC)s3)CC2)ccc(Br)cc1 C1(C(=O)NC2(c3cn(C)nc3)CC2)CC(O)CN1C(=O)C(C)(F)c1ccon1 O=C(O)CC(CC(=O)Nc1cccc(CF)c1)c1ccccc1 Cn1nncc1Nc1cnc(CC(F)(F)F)s1 C1(CC)C(NC(=O)C=C(C)C2CC2)CCN1C(=O)CCCOc1ccc(C)cc1 Cc1ccc(C)c(CNC(=NCCF)NCc2ccncc2Cl)n1 N1(CC=CC(=O)NCC(n2ccnn2)C)CCCC1 N(C(=NCCc1cccs1)NCC(C)(C)C1CC1)C(C)CC1CCOC1 c1(C(=O)NC2CC(C)C2)cnc2nc(NS(=O)(=O)C3CCCCC3)ccc2c1 C1(CN(C(C2C(C)(C(=O)OCC)C2)=O)C)CCN(C(=O)Cn2ccc(C)c2)CC1 c1(CC)nocc1C(=O)NCC1(O)CN(C(=O)CN2CC3CC3C2)C1 c1(NC(C)=O)cccc(C(c2nnnn2CCCF)Nc2ncc(C)o2)c1 C=C1COCCN(C(c2cnc(C(C)(F)F)s2)C(=O)NC2(C)CC2)C1 CC(C)(CS(C)(=O)=O)C(=O)NCCNC(=O)CC1(OCc2ccccc2)CC1 c1(CCC(=O)NCCC(C)NC(=O)C(C)(C)CO)ccc(Cl)cc1Br C#Cc1ccc(C)c(NC(C2CC3CC3N2C(=O)C(C)(C)CC2CC2)=O)c1 c1(C(N2CCN(C(C(C)OCCC=C)=O)C(C)C2)=O)ccc2c(C)noc2n1 N1(C(C2C(C)C2)=O)CC2CCC(C1)N2C(c1ccc(C(F)(F)F)cc1I)=O CC1(C)C2CN(CC(c3nnnn3C3CCC3)NCc3c[nH]cc(Cl)c3=O)CC12 CC1C(=O)N(CC(=O)NCC2CCC(C)C2)C(=O)C1C C(=O)(C(C)S(=O)(=O)C(C)C)N(CC(C)NC(c1c(NCC)ccc(Cl)c1)=O)C N1(C(CSC)=O)CCC(O)(C2CCN(C(C3CC4C(C3)C4(F)F)=O)CC2)C1 N1(C(C(CC)N(CC)CC)=O)CCC(C2(NC(=O)C(C)(C)NC(C)=O)CC2)C1 C1(NC(COC(C)C)=O)CC2CC(NC(C3(F)CCCCC3)=O)CC12 CC1CC(C(=O)NCC2CCC(CNC(=O)C(=O)NCC3CC3)CC2)CCS1 c1(CC)noc(CC)c1CC(N1CC(O)(C(C)NC(c2ncn(C)n2)=O)C1)=O N1(CC)C(=O)CCC1CC(=O)NC(C1CN(C(c2cc(COC)ccn2)=O)C1)C N1(C(CCC=C)=O)CCOCC(CNC(c2nn(C)nc2Br)=O)C1 C(CCO)(C(F)F)N(C(C(C1(O)CCC1)NC(CCC)=O)=O)C C1(NC(N2C(CC)CCCC2)=O)Cc2c[nH]nc2CC1C Cc1cc(C(=O)NC2C=CC(C(=O)NCCC3CC=CC3)C2)[nH]c1C c1(OC)ccc2c(NC3CC3C(N3CCC(C#N)C3)=O)ncnc2c1 Cc1c(OC(F)(F)F)cccc1NC(=O)COC1CCCNC1 N1(C(CC2(C=C)CC2)=O)CCC(C2CCN(C(=O)C(C)CCCC(C)C)CC2)C1 c1(OC)ccc(NC2(CC3CC3)CCCCC2)cc1OC N1(C(C(CSC)OC)=O)CCN(C(c2cccc(Br)c2)=O)CC(O)C1 N(C(=NCC(C)C)N1CCC2(CC(C(F)F)=NO2)C1)Cc1ccc(CCC)cc1 c1(C(C)C)ccc(NC(C2CC(NC(=O)Cc3cccc(F)c3)C(O)C2)=O)cc1 c1(SCC)ccccc1C(=O)N(CC(C)CNC(C1CC1c1nccn1C)=O)C c1(C2C(C(=O)NC3CCN(C(=O)CC4CC4C(F)(F)F)C3)C2)cccc(OC)c1 N=c1nnn(CC(=O)NC(c2ccccc2)CNC(c2nn[nH]c2Cl)=O)[nH]1 c1(OC)nn(C)cc1C(N1CCCC1(C(=O)NC1(CF)CC1)C(C)C)=O O=C(C#CC1CCCC1)NC1COCCN(C(=O)CN2CCCC2CO)C1 CCCC(C)CC(=O)N1CC2(CNC(C3CN(C)C3)=O)CCC1C2 C(=O)(CCC(O)C(C)(C)C)N(CCCNC(C1CCC(=O)C1)=O)CC(=O)N.CO c1(CC)cccc(NC(C2(NC(=O)CC3CCCC3C)CC2)=O)c1 c1(C(N2CC(CC)N(C(=O)C3=CCSC3)CC2)=O)cnc2n1CCOC2 CCC(C)C(C)(O)CNC(=O)CCC(C)(C)NC(c1cnc(C)nc1)=O CN1CCC(n2cc(NC(c3csc(-c4cccs4)n3)=O)cn2)CC1 c1(OCC)cccnc1C(=O)NC(C)CNC(=O)C=Cc1csnc1C O=C1NCCCC1n1cc(COC2CCCCC2CO)nn1.C12CCN(C1)C2=O C#Cc1ccc(CC(N2CCC(NC(=O)C=C3CCOCC3)C(O)C2)=O)cc1 c1(NCC2(CNC(c3nnn4ccccc34)=O)CC2)c(Br)cccc1[N+](=O)[O-] C(C(=O)N1CC(O)CCO1)N(C(C)CC(N(C)C[Si](C)(C)C)=O)C C#Cc1cccc(C(=O)NC2(C)CCN(C(C3CCC4(CCC4)OC3)=O)C2)c1Cl c1(OC)c(C(N2CC(OC)C(NC(=O)Cn3ncn(C)c3=O)C2)=O)cccc1N C(=O)(CC(CC1CC1)NC(=O)CCCOC(C)(C)C)OCC(C(C)C)N(C)C O(N=C1CCCCCC1)CC(=O)NC1CN(C(CCc2ccc(C)o2)=O)C2C1C2 c1(OCC(=O)NCC(CC)NC(C2CCCC2(C)C)=O)ccc(F)cc1 N12CC(CC(C)C1)C2=O.c1(NC(C)=O)ccc(C(=O)NCCN(C)C)cc1 C(C1=NOC2CCCC12)NC(CC12CN(C(C3(CN(C)C)CC3)=O)C(C1)CO2)=O c1(C(=O)Nc2c(Oc3cc(CN)c(Br)cc3)cccc2)cccc([N+](=O)[O-])c1O c1(OC)noc(C)c1C(=O)NC(C)CCCCNC(c1cc(SC)c(C)o1)=O C(CC(C)C(=O)N1CCC(C)C1C(=O)NCCC(=O)NCC)=CCC c1(N(C)C)cc(C(=O)N(C2CC(NC(=O)CC(=O)N3CCCC3)C2)C)cc(Cl)n1 C1(OCC)COCCC1CC(N1CCCC1CNC(=O)CC1CCCC1)=O C(C(C)CC(=O)N(C1CCC(F)(F)C1)CC1CC1)NC(C1(CCOC)CCC1)=O C1(C(=O)NC2CN(C(c3cc(CCC)n(C)n3)=O)CC2C)CN2CCN1CC2 C1(NC(C(C)SCCCC)=O)CC(C)CN(C(c2cncc3c2CC3)=O)C1 CC1=NOC(CC(N2CC(O)(C(C)NC(c3ccoc3C)=O)C2)=O)C1 C(=O)(NNC(=O)C(=O)NC1CC1)OC(C1CC(C)CC(C)C1)=O C1(NC(c2c(C)ccnc2C)=O)CN(C(c2ccccc2F)=O)C2(CCCC2)C1 c1(CCC)sc(C(=O)NC(C)(CNC(=O)C(C)c2ccsc2)CO)cc1CC C12(CNC(CC3CC(CC)OCC3)=O)CC(NC(c3cncnc3)=O)(C1)C(C)O2 c1(OCC)ccc(C(=O)NCC2CCCN2C(C2CCC=CCC2)=O)cn1 C(=O)(CCCC(=O)NCC1C(NC(CSCCC)=O)CCCC1)N(CC)CC O=C(C#CC1CCCCO1)NC1CCC2(CC1)CC(NC(=O)C1=NNC(=O)C1)C2 C1(C(C)NC(C2(CCC)CC2)=O)CN(C(c2cncnc2C2CC2)=O)CCO1 c1(N(C)C)ccc(F)c(CNC2(CO)CCCC2)c1.N12CCC(F)(C1)C(=O)N2 O=C(N=c1nc(O)[nH]c(O)n1)c1[nH]nc2cc(-c3cc(CO)cnc3F)ccc12 C12(NC(c3c(Cl)ccc(OC)c3F)=O)CCCC1N(c1nnco1)CCC2 c1(C(=O)NCC23C(CN(C(C4(NC(C)C)CC4)=O)C2)C3)nccn2ccnc12 N1(C(COC(C)(C)C)=O)CCC2CN(C(c3ncc(Cl)cc3Br)=O)CCC12 N1(C(c2c(C)onc2Br)=O)CCN(C(C2CC2F)=O)C(CO)C1 C(=O)(C(C)(C)CN1CCOCC1)N(CC(C)N(C(CCN(CC)CC)=O)C)C C#Cc1ccc(C(N2CC3(CC3)CC2C(=O)Nc2cnccc2CC)=O)c(C)c1 C1(NC(C2CCC(C)O2)=O)CC=CCC1C(N1CC(C)(C(F)(F)F)C1)=O C(=O)(C(O)C(C)(C)CC)NC(CC)(C)CNC(=O)Cn1nnc2c1CCCC2 Cc1nn(C)cc1C1CCC(CO)N1C(=O)C(c1cccc(Cl)c1)(C)O N1(C(CCN(CCC)C)=O)CCSCC1CCNC(c1cc(C)n(C)n1)=O C1(CC(=O)NCCCN(C(=O)C2=CCOC2)Cc2ccccc2)CCCC(O)C1 N1(C(C2CCCC(OC)C2)=O)CCCN(C(=O)Cc2ccc(C)cc2F)CC1 c1(C(=O)NCC(CNC(CC2C(COC)C2)=O)(C)O)cc(Cl)n[nH]c1=N Cc1cc(C(=O)NC2CN(C(c3ccc(Br)c(O)c3)=O)CC2F)cc(C(F)F)c1 CC(C)(C)C(O)C(=O)NCC(C)(C1CCC1)NC(=O)C(c1cc(Cl)cc(Cl)c1)=O C1(CNCCCN(S(C)(=O)=O)C)(CO)COCC2CCCCN12 c1(-c2cc(C)cc(C)c2O)cccc2c(NCc3cc(Cl)ccc3Br)cccc12 C1(C(N2CCCCC2C(F)F)=O)CCC2CCC1N2C(=O)CC1CC(F)(F)C1 C#CCC(C)(C(=O)NCc1cccc(C#N)n1)NC(=O)C(CC)CC C12(NC(CC(CC=C)NC(=O)Cc3cc(C)cs3)=O)CC3CC(CC1C3)C2 c1(OC)ccc(CN2CC(=O)N(Cc3cnn(-c4ccccc4)n3)C2=O)cc1F C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC2C(CNC(CS(CC)(=O)=O)=O)(C2)C1 C1(C(=O)NC2C3CC2CN(C(=O)C=Cc2nccs2)C3)CC2C=CC1C21CC1 C(CN=c1[nH]c(C2CC2)nc(=N)[nH]1)N(C(C1C(OCC)C1)=O)C C(=O)(C1=CCC(C)(C)CC1)N1CCN(C2CCN(C(C(CC#C)C)=O)C2)CC1 C1(CC)C(NC(C2(SC)CC2)=O)CCN1C(c1csc(-c2cccs2)n1)=O C(C1CCOCC1)=CC(=O)NCC(C(C)C)NC(=O)Cc1ccn(C)n1 c1(C(=O)NC(CNC(C(=O)NCCOC)=O)CCOC)cccc(F)c1Cl C1(C2(NC(C3C(=C)C3)=O)CCC2)CCCCN1C(c1nnc(S)n1C)=O C(C(C)CCCC(C)C)NC(CC1(C)N(C(c2c(CC)nns2)=O)CC1)=O C(=O)(C1=CCC2(COC2)OC1)NC1C(NC(c2cc(OC)c(C)cc2)=O)C1 c1(C(N2CC3(C(C(=O)NC(c4cnccn4)C)C3)C2)=O)ncc(Cl)cc1Cl C1(C(N2CC(CC)C2)=O)CC(O)CN1C(=O)CCCCNC(=O)C1CC1 c1(C(C)NC(C(CC(F)C(N)=O)C(N)=O)=O)nc2ccccc2n1C c1(C(=O)NCC2CCN2C(=O)CCOC2CC2)c(C(F)(F)F)nc2n1CCCC2 N1(C(=O)OC(C)(C)C)CCOCC1.C12CC(C1)C(=O)C1(CC1)C(=O)N2.C1(=O)CON1 c1(OC)cccc(O)c1C(N1CCCC(CO)(NC(=O)CC2CCCCC2)C1)=O c1(NC(c2cncc(CNC(C(CC=CCC)C)=O)c2)=O)cn(CC)nc1C#N C12(C(=O)OC)COCCC1(F)CN(C(=O)NCc1ccnc(S(N)(=O)=O)c1)C2 c1(C(N2CC(O)(C(C)NC(c3c(C)ccs3)=O)C2)=O)cc(C(F)(F)F)cnc1C CC(CS(C)(=O)=O)C(=O)NC1CCC1NC(c1cc(O)nc(N(C)C)n1)=O C1(OC)CC(CNC(=O)CC(C)n2ccnc2)N(C(C2CC(C)OC2C)=O)C1 c1(-c2onc(C3C(OC)(OC)CC3)n2)cc2ccccc2[nH]1 c1(C(=O)NC(CC)CNC(=O)C=CC(=O)N(C)C)cccc(C(C)(F)F)n1 C1(C2CCN(C(C3(CF)COC3)=O)C2)(NC(C(CC(C)C)OC)=O)CC1 n1(CC)nnnc1C(c1ccncc1)NC(c1ccc(C)o1)C C1(C(=O)OC)CCCN(CC#CCCNS(C)(=O)=O)C1 C1(NC(CC(CC)O)=O)CCN(C(C2(N3CCCCC3=O)CC2)=O)CC1C C1(OC)CN(C(=O)C(F)=CC2CC2)C(C)(CNC(=O)C=CC2CC2)C1 C(N=c1[nH]c2ccccc2cc1[N+](=O)[O-])C1CN(C(c2c(C)cccc2C)=O)C1 C(=O)(C1=NN2CCCN=C2N1)NCC(CCOC)NC(c1cc(Cl)ns1)=O C1(NC(C2CN(C(C)C)C(=O)C2)=O)CC(F)CN(C(=O)Cn2cc(CO)nn2)C1 C1(CC(N2CC(CNC(c3c[nH]c(=NC)o3)=O)C2)=O)COC2(CCC2)CO1 N1(C(C(N2CCSCC2)C)=O)CCCCC2(CCN(C(c3ccc(Br)o3)=O)C2)C1 c1(NC(c2ccc(OC(C)C)cc2)=O)cc(C2=CCC(O)CC2)ccn1 c1(COC)nn(C)cc1S(=O)(=O)NC1CCCCC1c1ccnn1C c1(OC)ncc(Cl)cc1C(=O)NCC1CCN(C(c2ccn(C)c2)=O)C1(C)C C1(OC)CC(CNC(=O)COCc2ncc(C)o2)N(C(=O)CC(C)F)C1 N1(CC)Cc2ccccc2CC1C(N(CC(C)N(C)C)C(C1C=CCC1)=O)=O c1(NC(C)=O)ccc(C(=O)N(C(C)CCNC(=O)C2=CCCS2)C)nc1 C(=O)(CC(F)(F)F)NCCCC(C)NC(C1CCC(c2ccccc2)O1)=O O=C(C1=CCSC1)N1CCOC(CNC(C2(Cc3ccccc3)COC2)=O)C1 c1(C(N2CCN(C(C3=NNC(=O)C3)=O)CC2CO)=O)cccc2[nH]cc(Cl)c12 c1(SC)ncc(C(=O)N(CCCCN(C(=O)CC(C)F)C)C)c(O)n1 N1(C(C)C(=O)NCC(=O)Nc2ccccc2)CC23CCCCC2(C1)CN(C)C3=O c1(C(=O)NC(CNC(c2onc(CC)c2C)=O)C)ccc2c(c1)C(=O)OC2 c1(C(=O)Nc2[nH]cc(C(=O)O)c2)ccc(S(=O)(=O)NC=O)cc1 C(CCC(=O)NC(C)CCN(C(=O)Cc1csc(C(C)C)n1)C)=CC CC(C)C(C(=O)NCCC(C)NC(c1cnccn1)=O)c1cnn(C)c1 N1(C(C(C)C2CCCO2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 C#Cc1ccc(C(=O)NC2CC2NC(=O)C(C)CN2CCOCC2)cc1Cl C1(c2ccc(Br)cc2)(SCCCn2cc(CNC(C(C)O)=O)nn2)CC2(CC2)C1 c1(NC(C2CCN(Cc3ccc(OC)cc3Br)C2)=O)ccc2c(c1)c(Br)nn2C C(=O)(C(O)CC(C)(C)C)NC1CC(NC(C(C)(C)OCC)=O)C1 c1(NCC2N(C(CCCC(C)C)=O)CC2)ccc([N+](=O)[O-])cc1S(C)(=O)=O N1(C(c2cnc(Cl)cn2)=O)CC2CCN(C(=O)COCC(F)(F)F)C2C1 c1(CC)c(C(=O)N(CCCCN(C)C(C2CCCN(C)C2)=O)C)ccn1C CC1CCCC1(C)NC(=O)NCC(=O)N(C(F)C(=O)O)C1CCCC1 C(N=c1[nH]cc(Cl)c(C)c1C#N)C1CN(C(C(C(CC)C)C)=O)CC1C(F)(F)F CN(Cc1ccc(Cl)c(F)c1)N1CC2(CC(C(=O)OC(C)(C)C)CO2)C1 c1(C(=O)NC2C(NC(C3(CN(C)C)CC3)=O)CCC2)ccc(Cl)c(O)c1N c1(CC)c(C(=O)NCC(C(C)(C)C)NC(=O)CCOC2COC2)cccc1C C(CN=c1ncc(C(F)F)c[nH]1)N(C(C1CC(C)=NO1)=O)CC C(=O)(CS(=O)(=O)CC(F)(F)F)NC(CN(C(c1c(CC)ccc(OC)c1)=O)C)C CC#CCC(C(=O)N(CC)CC1CCOC1)NC(=O)C(C)C(C)(C)C C12(NC(c3c(CC)nn(C)c3)=O)CC(CNC(=O)Cn3ccnn3)(C1)OC2C N1(C(c2c(SC)ccs2)=O)CCCC(NC(=O)Cc2c(C)noc2C)C(F)C1 c1(C(N2CC(O)(C(C)NC(c3cn(C)nn3)=O)C2)=O)ccc(F)cc1 CC1CN(C(=O)Nc2cccc3c2CCO3)CC2(CCOC2)O1 C(C)(CC1CCC1)(C(=O)NCCNC(=O)Cn1ccc(C)n1)OCC N1(C(c2c(CCC)n(C)nn2)=O)CCN(C(c2cccnc2O)=O)C(C2CC2)C1 n1(CC(=O)NC2CC(NC(CC(C)(C3CCC3)N(C)C)=O)C2)nnc2c1CCCC2 C12(C(=O)NC(CCN(C)C)C(=O)NC(c3nn[nH]n3)CO)CCCC1OCC2 Cc1[nH]c(CN2C3CCC(C3)C2c2ccccc2)c(C)c1C(N1CC(O)C1)=O N1(C(c2cccc(OCc3ccc(F)cc3)n2)=O)CCCC2(CCNC2)CC1 C1(OC)CC(C(=O)N(CCCNC(=O)C(C)n2cccn2)C)CC1OC N(C(=NCCCCl)NCc1cscc1C(F)(F)F)C(C1CCCO1)C C=CCC(C)C(=O)NC(CN(C(=O)CN1CCCNC1=O)CC)CC n1(CC)nc(C(=O)NC(CC2CC2)CC(=O)NCc2ccc(C)s2)cc1C N1(C(C2CC(OC)C2)=O)CC(NC(C2COC(=O)O2)=O)CC2(CCC2)C1 Cc1ncccc1C=CC(=O)NC(C)C(C)NC(=O)C(c1cccc(O)c1)(C)C c1(C(N(C)CC2CN(C(=O)CCc3nccs3)C2)=O)nn(C)c2c1C(O)CCC2 N1(C(c2ccn(C)n2)=O)CC2CC(NC(c3cc(C4CC4)on3)=O)CC2C1 c1(C(N2CCC3(CN(C(C4(SC)CC4)=O)C3)C2)=O)cc(C)ccc1S(N)(=O)=O c1(C(N2C(C(=O)Nc3c(C)noc3C)CCCC2)=O)cc(Cl)cnc1Br C(C(COC)CC(=O)NCC1CN(C(C2(C(C)(F)F)CC2)=O)CCCO1)OC C(=O)(C(C)C(O)C(C)C)NC(CC)C(=O)NCC(C)(C1CC1)OC(C)=O c1(N(C2CCCC2)C)ccccc1C1CCN(C(=O)C(N)Cc2ccc[nH]2)CC1 c1(CC)ccc(F)c(C(=O)NCC(C)N(C)C(c2cnsc2C)=O)c1F C(=O)(C(COC)CC(C)C)N1CC(F)(C(=O)OCC2OCCN(CC)C2)C1 C(CCC(=O)N(C(C)C)C)NC.C(C=O)=CCC1(CC(C)C)CC1 CCC(CNC1CCC(C)(C(C)C)C1)(CC)c1ccccn1 CC(CC(C)(C)C)C(=O)NCC(c1ccccc1)NC(=O)CC(C)(C)C C(=O)(CC(CC)CC)NCC1C(C(=O)NC(CC)CC)CCC1 C1(CNC(COCC(C)C)=O)(CNC(=O)Cc2ccco2)CC1(F)F C(C1=CCN(C(=O)Cc2cccc(Cl)c2)CC1)NC(C(n1cc(C)nc1)(C)C)=O C(=O)(C(CNC(=O)CC(F)(F)F)CC(C)C)N(CCC(N)=O)CC CC1CCN2CCN12.C1(CC(=O)NCc2cc(C=O)sc2)C=NN(C)C1=O N1(C(C=CC=CC)=O)CCCC(N(CC=C(C)C)CC2CCCCC2)C1 Cc1nc(S)sc1CC(N1CCC(C)C1CNC(=O)CC12CC(C1)C2)=O c1(OC)cc(C)[nH]c(=NCC2CCCCC2NC(c2cc(C)oc2C)=O)n1 c1(CC(=O)NC2C(C)CCN(C(C3COC(C)C3)=O)C2)cc2ccccc2o1 C(=O)(C1CCCc2c[nH]nc21)N1CC(SC)C(NC(=O)C=CC(=O)N(C)C)C1 C(CN=c1[nH]c(=NCc2ccno2)[nH]c2c1CS(=O)(=O)CC2)c1n(C)ncn1 C1(CNC(=O)COC2COC2)CCCN(C(c2scnc2Cl)=O)C1 C1(NC(C(C)N(C(c2c(C)[nH]cc2)=O)C)=O)CCN(C)CC1C C1(C#N)(C(=O)NCC2CC(NC(C(COC)O)=O)C2)CCCCC1 C1(C(N2CC(CCC)N(C(c3[nH]nnc3C)=O)CC2)=O)CCC2CC1C2(C)C C1(NC(CC2N(C(c3nn(C)c(Cl)c3)=O)CCC2)=O)CC(C2CCCC2)C1 Cc1cccc(C(=O)N(C(C)CCNC(=O)CSC2CCCCO2)C)c1Cl Cc1sc(C(=O)NCC2(C)CCCN2C(=O)CC(C)F)c(C)c1C c1(C(=O)NC2CCN(C(c3ncc(OCC)nc3)=O)C2)cnc2cc(C)ccn12 C1(C(N2CCC(O)CC2)=O)(COC)C=CCN1C(=O)C(C)OCC(C)C N1(C(C(C(C)C)NC(=O)CCN(c2ccccc2)C)=O)CCCC(C)(CCO)C1 C1(C(=O)NC(C(=O)NC2CN(CC)CC2C)Cc2cc[nH]n2)CC(=O)CC(=O)N1 c1(OCC)cc(C(N2CC(C(F)F)C2)=O)c(CNC(C2(C(F)F)CCC2)=O)n1C C(CC(C(=O)NCCC1CCCN1C(C1CC1F)=O)OC)OC C1(NC(CC2(OC)CCC2)=O)CC2CC(C1)N(C(c1cc(O)ccc1F)=O)C2 c1(C(=O)NCCCNC(C2CC3(C2)CC(F)C3)=O)cc(F)c(F)c(O)c1F C1(NC(Cc2c(C)n(C)nc2)=O)CC2(CCC(CNC(c3ccoc3)=O)OC2)C1 Cc1cccc(=O)n1CCCCN(C(=O)C(C)C1CCOC1)C1CCNC1 C1(CNC(c2cnc(C)n2C)=O)CN(C)CCN1C(=O)CCc1cccs1 N1(C(C(CC2CC2)NC(CC2(CC)CCC2)=O)=O)C2COCC1C2 CN1CCc2ccc(C(N3CCC3CNC(=O)Cn3ccc(Br)n3)=O)cc21 CCCC(C(=O)NCC1(CCNC(c2ccccc2OC)=O)CC1)N(C)C C1(NC(C(C(C)C)SCC)=O)CC2(C1)CN(C(c1ccnn1C(F)F)=O)C2 C=C=CC(C)C(=O)NC1(CNC(=O)CC(F)(F)F)CN(C(c2ccccc2)=O)C1 c1(OC)cc(CN2CCOC(CN)C2)cc(-c2ccc3c(c2)OCCO3)c1OC c1(C(=O)NC(CCCCNC(CC(C=C)C)=O)C)c[nH]c2c(Br)cccc12 c1(C2(C)CCN(C(=O)NCC3(C)CC(F)(F)CO3)CC2)n[nH]c2ccccc12 c1(C(=O)NCCOC2CCN(C(CCC(C)OCC)=O)C2)cc(F)cc(F)c1N C1(NC(C=Cc2cc(C)no2)=O)C(C)CN(C(=O)Cn2ncccc2=O)CC1C n1(C(C)C)ncc2c(NCCNC(C34CCCC3C4(F)F)=O)nc(Cl)nc12 c1(N2CCCC(C(C)NC(C3CCCSC3)=O)C2)ccc(F)cc1[N+](=O)[O-] C(=O)(C1=CCCCO1)N1CCCC(C2N(C(CC=C=C)=O)CCC2)C1 c1(C(=O)NC2CC(C(C(=O)NC)F)C2)cnc(C)nc1 c1(C(N(C(=O)C(O)CCSCC)CC(C)O)=O)cc2ncccc2[nH]1 C(=O)(C1=CC2(CCOC2)C1)NC1CCC(NC(CN2C(C)CCCC2)=O)CC1 C1(C)(C(N2CC(C(=O)NC(c3ccns3)C)(CC)C2)=O)C=CCCC1 CCC(CC)(CO)C(=O)N1CC(CCNC(c2ccnc3c2CCO3)=O)C1 N1(Cc2cc(C(C)=O)[nH]n2)CCC(C(C2CC3CCC2C3)C(=O)O)CC1 C1(NC(CN(C(C)=O)C)=O)CCCC(C(=O)NCCCOCCO)CC1 c1(C(=O)NC2CN(C(C(C)C#N)=O)C(C)C2)cn2cnnc2cn1 C1(CNC(=O)C=CC2CCC2)CCCC(NC(=O)C=C2CC2)C1 C12(NC(CCc3ccc(C)s3)=O)CC1CN(C(c1cc(CO)oc1C)=O)C2 Cc1noc(C(=O)NC23CC(NC(=O)C(C4(O)CCCC4)F)(C2)C3)c1C c1(NC2CCC(NC(c3c(C)ccc(C)c3)=O)CC2)ccc([N+](=O)[O-])c(C)n1 C1(CNC(C2C(C(=O)OCC)C2)=O)CCC(C(N)=O)O1.C1CC(=O)NCCO1 c1(SCC(N2C(CNC(c3cc(CC)on3)=O)CCC2)=O)nc2ccccc2o1 C1(C(N(CCNC(CCNC(COC)=O)=O)C)=O)COCCC1c1ccccc1 C(C(C)(C)CNC(c1nocc1C(C)(C)C)=O)N(C(C(C1CCC1)OC)=O)C C1(C(N2CC(C3(C)CC3)C2)=O)N(C(=O)C(CO)C(F)(F)F)CCCC1(C)C C1(NC(c2c(OC)csc2)=O)CC(CNC(c2csc(=N)[nH]2)=O)C1(C)C c1(C(N2CC3CC(CC(=O)NCC(C(CC)CC)O)(C2)C3)=O)cccn2ccnc12 CCCCC(C(=O)NC1CN(C(=O)C=CCOCCOC)CC(F)(F)C1)C(C)C N1(c2n(C)c3c(n2)c(Cl)ncn3)CCc2c(Cl)c(Br)cc(F)c2C1 N1(C(c2c(CC)occ2)=O)CC(O)CC1(C)C(=O)Nc1cc(C)cc(C)c1 C(=O)(C1=NOC2COCC12)NC1CCCC(CC(=O)NC(C)(C)CCCF)C1 C1(NC(C=NOC)=O)CCCC(CN(C)C(c2cnc(-c3ccsc3)s2)=O)C1 CCCCC(C(=O)NC(CNC(=O)CC(=O)N(C)C)CC)C(C)C C1(C)(NC(C2N(C(Cc3cc(C)sc3)=O)CC(O)C2)=O)C(C)(C)C1(C)C c1(C(N2CCC(N3CCCC3)C2)C(=O)NC)cccc(C(N)=O)c1.CSC C1(NC(C2CC(=C)C2)=O)CCCC2CN(C(C34CC(CO)(C3)C4)=O)CC12 Cn1cc(C=CC(=O)NC2(C(=O)NCCC(N)=O)CSC2)cn1 N1(C(CCc2onc(C)n2)=O)CC(NC(=O)CC2CCCC(C)O2)C2CCCC12 C1(OC)CC2CCC2C1.C12(O)CN(C1)C(=O)NC1CC21.CC(C)(C)OC(=O)NC Cc1ncc2n1CCC(C(=O)NC1CC(F)CN(C(C3CN(C)C(=O)N3)=O)C1)C2 CCCC(CC)CCC(=O)NC(c1nocc1C(=O)NCCCN1CCC1)C N(C(=NCC=C1CCOCC1)N1CCCC(n2ccnn2)C1)CC(=C)C C=Cn1nccc1C(N1CCCC1C(C)NC(=O)C(C)N1CCCC1)=O c1(CNC(C2=CCSC2(C)C)c2n(C)nnn2)sccc1S(C)(=O)=O N1(C(=O)CCC2CCCO2)CCC(C(N2CCC2Cc2ccccn2)=O)(CO)C1 c1(CCN=C(NCC(CC(=O)OC)C)NC2CCCCC2)cc2ccccc2o1 C(=O)(CC(C)CCC)NCCN(C(C(CCC)NC(N)=O)=O)C1CCCCC1 N1(C(CCCC(C)O)=O)CCC2CCN(C(c3c[nH]nc3C3CC3)=O)CC12 O=C(C1=COCC1)NC1CCOC(C(N2CC(c3ccon3)C2)=O)C1 NC(=O)CC(O)C(=O)NC1CN(C(=O)Cc2cccc(OCCN(C)C)c2)C1 CC1CN(C(N2CCOCC2=O)=O)CC1n1cc(CC(C)(C)NC(N)=O)nn1 c1(C(=O)NC2CCCN(C(CS(C)(=O)=O)=O)C2)c[nH]c2c(Br)cccc12 c1(C(=O)NC2C3CN(C(CC(CCC)(C)O)=O)C2C3)cc2cccc(OC)c2o1 c1(C(N(C)CC2CCCCN2C(c2ccc[nH]2)=O)=O)ccccc1S(C)(=O)=O c1(CC(=O)NCC(C2CCCCC2)NC(C=COCC)=O)ccc(C)nc1Cl C=CC1(CC(=O)NCCCN(C(C2C3CCCCC23)=O)C(C)C)CCCCC1 Nc1cc(F)cc(C(=O)NCc2ncoc2C2CN(C(c3cnoc3)=O)C2)c1F C1(NC(C(C)(C)NC(Cc2c(C)n(C)cn2)=O)=O)CCCCCC1(C)C c1(NCCCC)ccccc1C(=O)NC1CC(NC(=O)Cc2ccc(O)nc2)C1 C1(C(=O)NCc2nnc(C)o2)(NC(CSCC)=O)CCC(C)(C)C1 C1(n2cnnn2)(CC(=O)NC2C(NC(CC(=O)N(C)C)=O)C2)CCOCC1 C1(CCNC(CC2N(C)CCC2)=O)COCCN1C(c1ccccc1C(F)F)=O c1(C(=O)NCC(C(C)C)NC(CCC(=O)N(CC)CC)=O)cc(Cl)c(F)cc1Cl N1(C(c2cc(C)nn2C)=O)CCC(NC(C2(C)CCCCCC2)=O)CC1C c1(C(=O)NCC2(F)CCN(C(C3N(C)CCC3)=O)C2)cn(C)c2c(Cl)cccc12 C(=O)(CCCC1(NC(=O)C(C)c2ccco2)CCC1)NC(CCOC)C CC1CCCCC1n1cc(CC(O)Cc2ccccc2)nn1 C(CC(C)C(=O)N(C1CCCN(C(=O)C(=O)NCC2CC2)C1)C)OC N1(CC)CCOC(C(=O)NC2(C(=O)NC3C(C)CCC3C)CC(F)(F)C2)C1 C(C(C)C(=O)NC1CCN(C(C2(NC(=O)OC(C)(C)C)CCC2)=O)C1)OCC C(=O)(C(C(O)C(F)(F)F)C(C)(C)C)Nc1cncc(CCN(CC)CC)c1 C1(C(=O)NCC2(F)CN(C(CCSc3n(C)ccn3)=O)C2)CCCC2CCCN12 C1(N(C)C)CCC2CN(C(c3cccc(OC(F)(F)CF)c3)=O)CC12 c1(CC=C)cccc(C(N2CCCC(CN(C)C(C3CC3F)=O)C2)=O)c1 c1(C(=O)NC(COC)C(=O)NCC(C)(C)N2CCCC2)cc2ccccn2n1 CCCC(C(=O)N(C(C)CN(C(=O)COc1cccc(Cl)c1CC)C)C)C(C)C c1(CC)c(C(=O)NC2CCCC(NC(=O)CCn3nc(C)nc3C)C2)nnn1C c1(C(=O)NCCCOCCC(=O)NCCc2ccc(F)nc2)c[nH]c(=S)cn1 CCC(CCCC(=O)NC1CC2(CCCC2)C1)NC(C1(C)CC(F)C1)=O C1(C(N2CC(C3(NC(CCC(=C)Br)=O)CC3)C2)=O)CCc2nncn2C1 O=C(C1=COCC1)NC(Cn1cncn1)C(=O)NCCCc1cccs1 c1(NC)ccc(C(N2CC=CC2(C)C(=O)NC(C)Cc2ccncc2)=O)nc1 c1(C(=O)NC(CC)CNC(C2CCC(N(C)C)CC2)=O)ccc2oc(C)nc2c1 N1(C(C2C(C)CC(=O)NC2)=O)CCC(C2CN(C(C3CC(O)C3)=O)C2)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)CS(C)(=O)=O)ccc2c(O)n[nH]c2c1 N1(c2cc(NC3CC(OC(C)(C)C)C3)nc(C(C)C)n2)CCCCC(F)(F)C1 C1(NC(C(C)=C2CCC2)=O)CC=C(C(=O)N2CCCC(CO)CC2)C1 C1(C(=O)NCC(c2ccc(F)cc2)NC(c2c(C)n[nH]c2)=O)CC2CC1CO2 N1(C(C2(OC)CC2)=O)CC2CC1CC2NC(=O)CCc1cccc(C(F)F)c1 Cc1cc(O)cc(C)c1C(N1CCC12CN(C(c1ccccc1CO)=O)C2)=O N1(C(C=C2CCC(C)C2)=O)CC2(C)CN(C(C3CCC(C)C3)=O)CC2(C)C1 CC(C)CC(CC(=O)NCC1OCCC1(C)C)NC(c1c[nH]c2cnccc12)=O C(=O)(C1CCc2cccc(F)c21)NCC(C)(O)CNC(c1cncc(N)n1)=O c1(C(=O)NCC2=CCN(C(C(C(C)C)C)=O)CC2)c(F)ccc2ccncc12 C(N=c1[nH]cc2ccnc-2[nH]1)C1C(C)CCN(C(c2cccc(OC)n2)=O)C1 c1(N2CCC(C)(C(F)(F)F)CC2)nc(N2CC3CCOC3C2)nc2ccccc12 c1(C(=O)NC(C)CNC(=O)Cn2ccc(O)nc2=O)c(F)cccc1[N+](=O)[O-] C1(NC(c2scc(C)c2)=O)CCC2CC1CN2C(=O)Cn1nc(C)n(C)c1=O C(=O)(C1CCCc2cncn21)N(CCCN(C(C1N(C(C)=O)CCOC1)=O)C)C c1(C(N2CCC(CN(C(C(=O)NCC=C)C)CC)C2)=O)nccn2nc(C)cc12 N1(C(C2CCCN(CC)C2)=O)CCC(C(=O)NCCCSC)(OC)CC1 N1(C(=O)OCC(=O)NC2CCN(CC(=O)OC)C(C)C2)CCc2sc(Br)cc2C1 c1(C(=O)NCC(C)CC2CCCC2)cc(=NC(=O)N2CCCC2)[nH]o1 O=C(C1=CCCN(C(=O)Cc2ccc(F)cc2F)C1)Nc1cc(Cl)cc(Cl)c1Br c1(C(N(C2CCCCC2NC(C2CCC(F)(F)CC2)=O)C)=O)cc2scnc2[nH]1 C1(C(=O)N(CC(C)CO)C)(CC)CCCN1C(=O)Cn1cnc(C#N)n1 Cn1cnc2[nH]c(=NCC3(C)CCOC3)nc(N3CCCOCC3)c12 N1(C(CC2(OC)CCC2)=O)CCC2(CC1)CN(C(=O)C(C)(C)c1csc(C)n1)C2 CC1(F)CCC(C(N2CCCC(C)(NC(c3ccnc(C(F)F)n3)=O)C2)=O)CC1 c1(C(c2nnnn2CCCF)NCC2(CC)COC2)ccnc(Cl)c1 C#CCC(C)(CC)C(=O)N(C)CC1CCCN1C(=O)C=CCF C12(C(N(CCC)CCN(C)C)=O)CCC1CN(C(=O)Cc1ccc(F)cc1)C2 C1(C(=O)OC)N(C(=O)C(CC2CC2)OC)CCOC1(C)C N1(C(C(C)=CC)=O)C(C(=O)NC2CONC2=O)CC2CCCCC12 c1(CC(=O)NC2(CC=C)CN(C(c3cc(C4CC4)no3)=O)C2)cn2ccsc2n1 N1(C(CCN(C)CC)=O)CC2CC2(C(=O)NC(c2ccco2)C)C1 c1(C(N(CCCCCC)CCNC(=O)CC(=O)NC2CC2)=O)cc(CN)ncn1 C1(NC(CCc2onc(COCC)n2)=O)CCN(C(=O)C=C(C)C)CC1CC C1(C(=O)NCCNC(CN(C)C(=O)C2CC2)=O)CC=CCC1C(F)(F)F C(=O)(CC(CC)C(C)C)N1CCC(C(=O)Nc2cnc(CCC)nc2)C1C N1(C(c2c(C)n[nH]c2C)=O)CCC(C(=O)N(C23CC(F)(C2)C3)C2CCC2)C(C)(C)C1 CC(C)C(C#N)C(=O)N1CCCC1C(C)(C)NC(=O)C=Cc1cc(CC)cs1 C(=O)(C1=CC2CCCCCCC12)NCCC1(NC(COCCCC)=O)CC1 c1(C(=O)NC2CC(OCC(=O)NCC(CCC)C)C2)cncnc1C.O c1(COC)ncc(CNC(=O)CNC(C2(C#N)CC2)=O)[nH]1 Cc1c(NCC(=O)Nc2ccc(Cl)cc2)nc[nH]c1=NCc1cocn1 C(=O)(CCCCCn1cnnn1)NC1CN(C(c2cc(CCC)c(C)s2)=O)C1 c1(CC)cc(F)ccc1C(=O)NCC1CCCC(NC(C2(O)CCSC2)=O)C1 Cc1csc(=NCC(=O)N2CCCC(C)(NC(C3(C4CCC4)CC3)=O)C2)[nH]1 C1(CC(=O)N(C(CNC(C2(C#N)CC2)=O)C2CC2)C)CC2(CCC2)C1 c1(SC2(C(N(CC(CN(C(=O)CC#N)C)O)C)=O)CCC2)nnc(O)n1C C1(Cc2nc(C3(C4(N)CCC4)CC3)on2)CCN(C(C(C)(C)C)=O)CC1 N1(C(COC(CC)C)=O)CCC(CO)(CNC(C23C=CC(CC2)C3)=O)CC1 CCC(C)(CNC(=O)CC1CC(NC(=O)CC2C=NN(C)C2=O)C1)CC CN1CCC(C(N2CC(CNC(c3csc([N+](=O)[O-])c3)=O)C3CC23)=O)CC1=O c1(C(=O)NC2C3CN(C(C4C(COC)C4)=O)C2C3)c[nH]c2cc(Cl)ccc12 N1(C(c2ccc(OC)nn2)=O)CC(N(C(=O)CC2CC=CC2)C)C2(CC2)C1 C1(C(=O)NCc2cc(C)sc2)CC=CCN1C(C1CCCCN1C)=O C(CCS(=O)(=O)c1ccc(C)cc1)NC(C(C)(C)NC(C)=O)=O C(=O)(C1OCCn2ccnc21)NC(C)CNC(c1cc2c[nH]nc2s1)=O Cc1[nH]c(=N)sc1C(=O)NCC1(F)CC(CNC(=O)CCN2CCCCC2=O)C1 N1(C(c2c(C)n[nH]c2)=O)CC(F)CC1C(=O)NCC1CC1[N+](=O)[O-] CC1CN(C)CCC1N(C)C(C1CCC(NC(c2ccnc(O)c2)=O)CC1)=O C(CN=c1ccc2c([nH]1)CCCC2)C1CCN(CC(C)(C)O)CC1 N1(C(C2(CC=C)CN(C(=O)CCSCC)C2)=O)CC2(CC2)CC1C c1(C(=O)NCC2N(C(C3C(C)=C3)=O)CCC2)ccc(C)c(S(=O)(=O)N(C)C)c1 N1(C(c2c(OC)cc([N+](=O)[O-])cc2)C(=O)NCCC#N)CCc2cccnc2C1 C12(NC(c3ccc(C#C)o3)=O)CCCCC1CN(C(=O)CC(C)CCCCC)C2 C1(N(C(N(C(C)C)CCc2ncon2)=O)C)CC2CC2C1 c1(NC(c2c(C)csc2)c2nnnn2C)ccc(O)c(CO)c1 C1(NC(C(C)OCC#C)=O)CC2CC1CN(C(=O)C(C)SC(C)C)C2 c1(C(=O)OC)n[nH]c(=NC2C(C)CN(C(=O)C(C)(C)F)CC2C)s1 N1(C(C(CCC)C#N)=O)CCC2CCN(C(c3ccc([N+](=O)[O-])s3)=O)C2C1 CC(=O)CCCCC(=O)N1CC(OCC(=O)NCc2c(C)cccc2F)C1 c12ccccc1S2.C(=O)(C(C)(C)C)N(CC(C)NC(=O)COC1CCCOC1)C Cc1cccc2c1CC(C(=O)NCC(O)CNC(c1ccc(CO)o1)=O)O2 N1(C(C2C(=C)C2)=O)CCC2(C1)CN(C(=O)Cn1cc3ccccc3n1)CCO2 C#Cc1cccc(CNC(=O)C(C)(CO)NC(c2ccn(C)c2C)=O)c1 N1(C(C=C(C)C(C)C)=O)CC(CCNC(=O)C=Cc2ccc(F)cc2)OC(C)C1 C1(NC(CCCC)=O)CN(C(c2cc(C)n(CC3CCCC3)n2)=O)CCC1CO C#CCC(CC(=O)NCC(C)(O)CO)NC(=O)CS(C)(=O)=O C(=O)(C(C(C)(C)C)NC(C1C2COCC12)=O)NCc1ccc(OC)nc1 CCC(C)C(C(=O)N(C)Cc1ncco1)NC(C1COCOC1)=O CC1(C)COCC1C(=O)NC(c1ccccc1F)C(=O)NC(C)(CO)C1CC1 C1(NC(C(CCN(C)C)NC(=O)CC2CCC(=O)CC2)=O)CN(C)C(C)(C)C1 C(CC(O)C(=O)NCC=C1CCN(C(C2C=CCS2)=O)CC1)SC N1(CCNC(CCCC(C)C)c2ccccc2)CCC2(CCCC(=O)N2)C1 C1(COC)CCCN1C(=O)CC(C)NC(c1cccs1)=O N1(C(C)=O)CCC(C)(C(=O)N(C)CC2CCCCN2C(=O)CCC2CCOC2)C1 c1(CC)cc(C)nc(NC2CCC(NC(=O)CC3CCCCC3C)CC2)n1 c1(C(=O)NC(Cn2cc(-c3ccc(SC)cc3)nn2)C)cc2nc[nH]c2cc1Br c1(NC(=O)C=CS(C)=O)ccc(C(F)(F)F)cc1[N+](=O)[O-].CC1(C2CCC2)CN1 Cc1cn2cc(C(N3CCCC3C(C)(C)NC(C3CCCN(C)C3)=O)=O)nc2s1 C1(NC(=O)C=CC2CCCC2)(CO)CCN(C(=O)CC2CCN(CC(F)(F)F)C2)C1 CCS(=O)(=O)CC(=O)N1C(C(=O)NC(CCO)C(C)C)CC2CC12 c1(C(=O)NCC2(NC(C(C3CCOC3)OC)=O)CC2)cc(C)cc2ccncc12 C(=O)(CCC(=O)NCC1(OC)CN(C(C2(COC)CC2)=O)C1)N(CC)CC c1(CC(=O)NC)ccccc1NC(C1(NC(=O)CC2CCCC(=O)N2)CC1)=O CCCS(=O)(=O)CC(=O)N1CC(NC(=O)C(C)Oc2ccc(Cl)cc2)CC1(C)C c1(C(N(C)CC2(CNC(C3CCCCN3C)=O)CC2)=O)cnccc1N(C)C CC(C)CCC(O)C(=O)NC(C1CC1C(=O)Nc1cccc(F)c1)C N1(C(C(c2ccc(C)o2)C)=O)CCC2C(C1)CN2C(c1cn(C(C)C)nc1C)=O C(=O)(C(CO)C(C)(C)C)N1CCN(C(C2(CC)CC2=O)=O)C(C)C1 N1(C(C(Cn2cccn2)NC(C(c2n(C)ncc2)O)=O)=O)CCCC2(CC2)C1 c1(C(=O)NC2CC(CNC(CCC(=C)C)=O)C2)cnc2cccnn12 c1(C(=O)NCC2CCN(C(C(CC)(C)F)=O)C2)ccc2c(c1)OCO2 c1(N(C)Cc2cnc(CC)s2)nc(N2CCCC3(CCCO3)C2)c2c(n1)CSC2 C1(C(=O)NC2CC(C(F)F)(NC(C3CCCO3)=O)C2)CCC2CC1CO2 C1(C(=O)NC2C(C)N(C(=O)C3=NOC(C)C3)CC2)CC12CCCCC2 C(=O)(C(C)C(C)(C)C)N1CC(c2c(CNC(c3c(C)cn(C)c3)=O)nco2)C1 C1(CN(C(=O)C=C(C)CNC(=O)C(c2cnn(C)c2)C)CC)CCC(=O)N1 O=C(C1=C(Cl)CCOC1)NC1CCC(C(F)F)CC1 C(=O)(CCCCC(F)(F)F)N(C1C2CN(C(c3cnc(N(C)C)nc3)=O)CC21)C N1(C(c2n(CCCC)ncc2)=O)CCC(C)C(NC(c2ncc(C(F)F)s2)=O)C1 C1(C(N2CCC(C)(N(C)C)C2)=O)CCc2ccnn2C1 C1(NC(COCCCCC)=O)CC2CC(C1)N(C(C1CCCC3(CC3)C1)=O)C2 CN=c1nc(N(CC(C)OC(C)(C)C)C)[nH]c(=NCC(c2ccsc2)OC)[nH]1 c1(-n2c(C3CCC(=O)N3C3CC3)nc(CCOC)n2)ccc(S(C)(=O)=O)cc1 S(=O)(=O)(CCC(=O)N1CCCC(N(C)C(c2sc(CO)nc2C)=O)C1)NC N#CC1CN(C(c2cc(O)nc(Cl)c2)=O)CCN1C(=O)CCc1ccoc1 C1(CNC(N(C)Cc2cccc(-n3cccn3)c2)=O)CCC(C)c2ccccc2C1 S(=O)(=O)(c1cccc(C(F)(F)F)c1)NC(C1CCC(OC)CC1)C(=O)O N1(C(C(C(C)C)C2CCC2)=O)CCC2(CCC(NC(=O)CC3CCCC3)C2)C1 N1(C(CCC#CC)=O)CCCN(C(=O)C(C#N)Cc2ccc(C#N)cc2)CC1C CC(C)CC(C)CC(=O)N1CCCC(C)C1CNC(=O)CC1(C)CCCCC1 C1(NC(c2cccn2C2CC2)=O)CC2CC1N(C(C1CCC1)=O)C2 N1(C(CCCOCC)=O)CCN(C(c2cnc(OC)nc2)=O)C(CC)C1 Cc1cn2ccc(C(N3CC4CC(NC(=O)C(C)(O)C5CC5)CC3C4)=O)cc2n1 C1(COC)(NC(=O)CCc2nncs2)CCN(C(c2nccnc2C(N)=O)=O)C1 Cc1cc(C)n(CCCC(=O)NC2CCN(C(=O)Cn3ccnn3)C2)n1 N1(CC(C)NC(c2cccc(Cl)c2)=O)CCN(C(=O)C(O)c2cnc[nH]2)CC1 c1(NC2(c3n(CCSC)nnn3)CCC2)cc2n(n1)CC(O)CO2 CCCC(C)CCCC(=O)NC1CCC(NC(c2c(C)nsc2N)=O)C1 c1(N)nc2ccsc2c(=NC2CCCSCC2)[nH]1.Cc1cn2c(n1)CN(CO)CC2 Cc1ccc(C(=O)NCCN(C(=O)C(CC(N)=O)c2ccccc2)C2CC2)c(O)n1 c12ccc(c(NC(=O)C(=O)NCCCOCC(F)F)c1)o2.S(C)(=O)(=O)N(C)C C12(CNC(C3(CCC)CC3)=O)CC(C1)C(NC(C1(C)CC(F)C1)=O)CO2 c1(C(N2CC(C)C(NC(=O)COc3cn[nH]c3)CC2)=O)cnc2ccoc2c1 CC1OCCOC1C(=O)N(C(C)CC(=O)NCC1CC1c1ccoc1)C C1(NC(c2n(CCOCC)nnn2)C(C)C)CCOC1(C)C C(=O)(C(C)CC(C)(C)C)N1CCC(C)C1CNC(c1ccnc(C(F)(F)F)c1)=O N1(C(C(C)CNC(c2ncc[nH]2)=O)=O)CCCC(CC2CC2)C1 Cc1cccn2nc(C(=O)NCC3CC3Cl)cc12 C1(CC(=O)NCCCN(C(C2(n3cncn3)CC2)=O)C2CC2)(CC)CCCC1 CCC(C(=O)N(CC(=O)NCc1ccccc1)C)NC(c1ccco1)=O CC1CN(C(c2cnc(C3CC3)[nH]2)C(=O)NCc2ccc(F)cc2)CC(C)(C)C1 C1(C(=O)NC2(CO)CC(F)(F)C2)(CO)CCN(C(=O)COC2CCCOC2)CC1 C(C(C)C)(C(O)C(=O)NCCC(C)NC(C1(C)CCN(C)C1=O)=O)OC C12(CCN(C(c3ncccc3C)=O)C1)C(=O)NCC2.C1(O)(CC#C)CCOC1 C1(C(=O)NC2C(NC(C34CC(C(=O)OC)(C3)C4)=O)CCCC2)COCCN1C=O CC(C)CC(C(=O)N(C)Cc1cnccn1)ONC(c1n[nH]cc1[N+](=O)[O-])=O c1(C(=O)NC2(C3N(C(CCN(c4ccncc4)C)=O)CCC3)CC2)ccc(F)cn1 c1(C(=O)NCC(CC=C)NC(C2CCS2(=O)=O)=O)cc(C(F)(F)F)cn1C N1(C(C(C)n2ccnc2)=O)CCSCC1C(=O)NCC(O)(CO)CO CN1CC2CN(C(=O)C(C3CC3)N(C)C(C3CC=CCC3)=O)CC2(C)C1 c1(NC2CC(F)(CNC(=O)CC3CCC(O)C3)C2)nc2c(cc1C#N)CCOC2 C1(C(N2CCCCC(NC(=O)COC3CCOC3)C2)=O)CCCC12CCOCC2 C1(C(=O)NCC(CNC(c2c(CCC)n[nH]c2)=O)F)CCCCN1S(N)(=O)=O C1(C(N2CC(OCC)C(CNC(C3CCCC3CC)=O)C2)=O)CC(C(C)C)=NO1 CC1(CNC(c2csc(-c3ccsc3)n2)=O)CCCN1C(C1CC1F)=O CC(C)(O)CC(=O)N1CCC(C)(NC(c2cc(-c3ccccc3)ccn2)=O)C1 N1(C(C)C)CCN2C(=O)C(NC(=O)CS(=O)(=O)N3CCCC3)CC2C1 c1(C(=O)Nc2n(C(=O)OC)ncc2C)ccc(F)c(F)c1 C1(C(=O)NCC(CC=C)NC(=O)Cc2cccc(F)c2Cl)CCc2nc[nH]c2C1 C1(C)(OC)CC2CC1CC2CNC1(c2nnnn2C2CC2)CC2(COC(C)C2)C1 C1(OC)CC(CNC(=O)CS(=O)(=O)NC)N(C(=O)C=CCO)C1 N1(C(C)C(=O)NC2(c3cn[nH]c3)CN(C(=O)CC(Cl)Cl)C2)CCC(O)CC1 N1(C(C(C)(C)c2ccccc2)=O)CC2CN(C(c3c(F)ccnc3Cl)=O)CC12 Cc1ccnc(C)c1CNC(=O)C1=CCC(NC(C2CCNC(=O)C2)=O)C1 c1(C(=O)NCC(=O)N(C)CC2(O)CN(C(C3C(C)CCS3)=O)C2)cc(Cl)ccn1 C1(C)(C(=O)NCc2ccc(C)cc2)CC(O)CN1C(=O)C=Cc1ccncn1 c1(OC)ccc2c(C(N3CC(CNC(=O)CNC=O)C(C)C3)=O)coc2c1 C1(C(N2CCC(C)(NC(C(=Cc3cccs3)C)=O)CC2)=O)CC2CCC1CC2(F)F C(=O)(C(C)(C)C(F)F)NC1CCN(C(c2cc(CC(C)C)[nH]n2)=O)C1C1CC1 C(C(C)(C)CNC(=O)Cc1csc(S)n1)N(C(=O)C(C)(C)c1cncs1)C C1(NC(CC(c2c(C)nn(C)c2C)CC)=O)CC1C1CCCN(C(=O)CCC)C1 N1(C(C(CC)O)=O)CCC(C)(CNC(=O)C(C)(C)OC(C)=O)CC1 C1(OC)(CO)CN(C(=O)C(F)CC2CN(C(C3(c4ccno4)CC3)=O)C2)C1 Cc1c(NC(=O)C(=O)NC2CN(C(N)=O)C3CC23)cccc1F O=C(C1Cc2c(Cl)cccc21)NC1(CNC(C2Cc3nccn3C2)=O)CCC1 N1(C(C(CC#C)(C)C)=O)CC=C(CC(=O)NCC2(n3ccnn3)CC2)CC1 C=C(Cl)C(C)(C)C(=O)N1CC(NC(C2(C(F)F)CCN(C)CC2)=O)C(O)C1 CC(CC1CC1)N=c1ccnc(NC2CC3(CCC3)C2c2cc(F)ccc2F)[nH]1 C1(C(=O)NC(C)CNC(c2ccccc2Cl)=O)CCCCC(=O)C1 C1(NC(C(CN(C)C)O)=O)CC(F)CN(C(c2c[nH]c(=N)o2)=O)C1 N1(C(CC=C)=O)CC2(COC(CNC(c3c(C4CC4)cccc3F)=O)C2)C1 C(=O)(C(C)(O)C(F)(F)F)N1CCCCC(C(=O)NC2CC(OC)C2)C1 C1(C(N(CCSC)C)=O)CN(C(=O)C(N2CCOCC2)C)CCC1O C1(C(N2CC(CNC(=O)CC3CSCCS3)C2)=O)OCC2CCCCC12 N1(Cc2cnc(OCC)nc2)CCC(NC(C2CCCCN2C(C)C)=O)C(C)C1 CCCCC(C)C(=O)NCC=C1CCN(C(c2cnc(C(N)=O)cn2)=O)CC1 C1(C(=O)NC2CCC(CNC(C(C)C)=O)C2)CC2CCCCCCC12 N1(C(C(C)SCCCC)=O)CCCC1(C)CNC(=O)CO.C1(N)CCCC1 CC1(C)Nc2ccccc2C1NC(C1CCC(C)(CN)CC1)=O N1(CC(=O)NC2C(OCC)(OC)CC2)CCCC(C)(CCSC)C1 C1(C#N)(C(=O)NCC2N(C(CCCSC)=O)CCC2)CC12CCC2 C1(OCC(=O)N(C2CCN(CC(C)C)C2)C(C)C)CCC(C)CC1 c1(CNC(=O)CCC2CCOC2)cc(C(N2CCCC2C(F)F)=O)cs1 C(=O)(CCCCCC(C)C)NCC12C(CN(C(CCC(C)OCC)=O)C1)CCO2 Cc1cc(F)ncc1-c1cn(C2CCN(C(=O)CC(C)N(C)C)C2)nn1 c1(CN2C(C(=O)Nc3cccc(CCC)n3)CSCC2)c(Cl)cncc1Cl N1(C(C(CC#C)(C)CC)=O)CCCCC2(CCN(C(C34CCC(CC3)C4)=O)C2)C1 c1(N2CC(CC(C)NC(c3c(C)[nH]nc3C(F)(F)F)=O)C2)ncc2ccnc-2[nH]1 C1(C)(C(N(C)CC2(C#N)CCC2)=O)CC(O)CN1C(C1CC(F)C1)=O c1(C(=O)NC2CCCN(C(C(CC)OC3CCCC3)=O)C2)ccn2ccccc12 c1(C(N2CC(O)(C(C)NC(c3csc(CO)n3)=O)C2)=O)cc2ccccc2nn1 N1(C(c2nn(CC)c(O)c2)=O)CCC(O)C(NC(c2oc(C)nc2C)=O)C1 n1(C(CC)C)ncc2c(C(=O)NOC(c3ccccc3C)C)cc(C)nc12 C1(C(=O)NC(c2n(C(C)C)ncn2)C)CCCN(C(C2CCC(=O)N2C)=O)C1 c1(C(N(CC(F)(F)F)CC)=O)ccncc1C1=CCC(C(F)(F)F)CC1 C(=O)(CCC(C(=O)OCC)NC(c1cn(-c2cc(Cl)c(F)cc2Cl)nn1)=O)OC Cc1cccc(CCC(N2CCC(NC(=O)CCC=CBr)C2C)=O)c1 n1(Cc2ccc(C(=O)NC3CNCC34CCC4)cc2)cnc2cccnc12 C1(C(=O)NC(C=CC(=O)NC(COC)C)(C)C)CCC(C)O1 c1(C(=O)NCC2N(C(C3(CC=C)CCC3)=O)CCCC2)nc(C)n(C)c1C c1(OC)ccc(C(N2CCN(C(C3CC3F)=O)C(CC3CC3)C2)=O)c(F)c1 C#CCC(C)(C(=O)NC1CC2CC(C(N)=O)CC12)NC(=O)COCC1CCCO1 N1(C(c2cn(C)c(C(N)=O)c2)=O)CC(C)(C)CC1CNC(C1CC(F)(CO)C1)=O c1(C(=O)NCC2CC(NC(c3n(CC=C)ccc3)=O)C2)c(C)nc2ccccn12 C1(C)(C(=O)NCC(CCOC)NC(=O)CCCC#N)CCCCCC1 c1(C(=O)NC2CCC(C(=O)Nc3cn(CC)nn3)C2)ccc(Cl)nc1Cl c1(OC)ccc2c(c1)CC(C(=O)NCCCNC(C1(C)COCCO1)=O)O2 Cc1oc(-c2cnn(C)c2)nc1C(=O)OC(C)C(C)F c12c(OC)ccc(C)c1NC2.C1(CCOC)CC(=O)N(C)C1c1cccc(Cl)c1 N1(C(C(CC)OC2CCCC2)=O)CCC(F)(NC(c2cnc(S)nc2)=O)C1 C1(NC(C2(C)CCCS2)=O)C=CCN(C(c2cnn(C(C)(C)C)c2N)=O)C1 c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccn2)cc(C)c2c(c1)CCC2 N1(C(CCN(C2CC2)Cc2ccoc2Cl)=O)CC2CCC2(OCC)C1 N1(C(c2cn(CCC)nc2)=O)C2CCC1CN(C(c1cn(C(F)F)c(C)n1)=O)C2 c1(C(=O)NC(C)C(C)NC(c2cc(O)ncn2)=O)cccc2c1nnn2C C1(CC)(NC(C2CN(c3nncs3)C2)=O)CCN(C(=O)C(C)OC)CC1 N1(C(CC2ON=C(C)C2)=O)CC(C(N2CCC(C3CC3)C2)=O)CC12CCC2 C1(CC)CCCCC1C(=O)NC(C)(C)CNC(=O)CC(C)(C)c1cccs1 C1(CNC(C)=O)CC(O)CN1C(=O)CC1(CC2CC2)CCC1.N12CSCC1C2=O C12(C(=O)NCC3CCCN3C(C3(N4CCCC4)CCC3)=O)CCC(CC1)OC2 c1(C(=O)NC2CN(C(CCCC#C)=O)CC2O)cc2cc(Br)cc(F)c2o1 C1(CNC(CN2CCC(OC)C2)=O)(CO)CCN(C(c2c(C)nsc2N)=O)C1 N1(C(CC(=C)Br)=O)CCOC(CN(C)C(C2CC(=O)N(CC(C)C)C2)=O)C1 N1(C(c2c(C)onc2)=O)CCC2(CC1)CC2C(=O)NC1(C(=O)O)CC2CC(O)C1C2 C1(CNC(C(C)SCCCC)=O)CN(C(c2cc(Br)co2)=O)C2(CCC2)C1 C1(CC(N2CC(CN(C)C(c3cc(C(F)F)nn3C)=O)C2)=O)CN2CCC1CC2 CC1(C)COC(C(=O)NCC2CCN2C(=O)COC2CCCCCC2)CO1 n1(CCC)nnnc1C(c1cn(CC(=O)OC)cn1)NC(C1CCCCC1)CO C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(=O)C(C)OCC2CC2)CC1C1CC1 C(=O)(C(O)CCC(C)C)N1C(CN(C(c2noc(CC)c2C)=O)CC)CCCC1 c1(NC(N(C)CC2OCCN(C)C2)=O)cccc2c1CCCC2 c1(C(N2CCN(C(C3CC(O)C3)=O)CC2CC(F)(F)F)=O)ccnc2[nH]ncc12 C1(C(=O)OCC#CCNCC)CN(C(c2cccc(C)c2)=O)CC1O N1(C(C2(CNC(c3cc(C)c(C)nn3)=O)CC(C)(C)C2)=O)CCCC(C)(O)CC1 c1(C2(CNc3nccc(N(C)CC4CCC4)n3)CCC2)ccc(F)cc1F c1(OCC(=O)NCCC(C)NC(CC(C)C)=O)ccc(F)cc1O c1(C(N(CCN(C(COCCCC#C)=O)C)C)=O)c(F)cc(OC)cc1F C1(C(C)=O)CC(C(=O)NCC(C)CNC(=O)CC2(CSC)CC2)C1(C)C Cc1cn(C)cc1C(=O)N(C(C(=O)NCc1ncc[nH]1)C1CC1)C C(CC(C)C(=O)NC(C)CNC(=O)Cc1ccccc1OC(C)C)OC c1(C(N(CC(C)O)CCNC(C(CC)C)=O)=O)cccc(C(F)F)c1Cl N1(C(C=CC=CC)=O)CCCC(C)(NC(c2ccc(Cl)nc2Cl)=O)C1 C1(C(N2CC(N(C(c3c(C)c(Br)sc3)=O)C)C2)=O)SC2C=CC1CC2 C1(CC(N2CCC(CNC(c3nnn(C)n3)=O)C2)=O)CCCC(=O)N1 c1(C(N2CCC(O)C(O)CC2)C(=O)NCCCSC)ccc2ccc(Br)cc2n1 c1(CC(=O)N(C2CCCCC2)CCNC(C(C2CCC2)OCC)=O)sccc1Cl C1(C2CC2)(NC(C(C2CCCN(C(c3ccc(C)n3C)=O)C2)C)=O)CCCC1 c1(C(=O)NCC2CCN(C(C3CC(=O)NCC3)=O)C2)cccc2nccn12 c1(C(C(=O)N(C2CCN(C(C3C=CC=CC=C3)=O)C2)CCC)C)ccc(F)cc1 C1(NC(CC2(C=C)CN(C(=O)COC)C2)=O)CCc2n[nH]cc2C1 c1(NCC(C)(C2CC2)NC(c2cc(C3CC3)on2)=O)ccc([N+](=O)[O-])cc1C#N C1(C)(CNC(C(C)NC(CC)=O)=O)CN(C(=O)CCNC(C)=O)CCO1 C1(CC(N2C(CN(C(C3ON=C(C(C)C)C3)=O)C)CCC2)=O)CCCNC(=O)C1 c1(C(N(CCCCNC(c2coc(CC3CC3)n2)=O)C)=O)ccn2ccsc12 N1(C(c2n(C)ncc2C2CC2)=O)CCN(C(c2ccnc(Cl)c2Cl)=O)CC(O)C1 C1(C(C)N(C(c2ccon2)=O)C2CC2)CCCN(C(=O)CCC2OCCO2)C1 N#Cc1csc(C(=O)NC2CCOCC2C(=O)NCCc2cccnc2O)c1 N1(C(C2CC(OC)C2)=O)CC(C)CN(C(=O)C=CC=C(Cl)Cl)C(C)C1 Cc1cc(C(N2CCC(CO)(NC(=O)C=CC(=O)N(C)C)CC2)=O)cc(C)c1O C(N=c1[nH]c2c(c(=NCCC3CC(=O)N(C)C3)[nH]1)CSC2)C1N(CC)CCCC1 C(=O)(C(O)CCCCC)NCC1(F)CC(CNC(C2C(=C)C2)=O)C1 S(=O)(=O)(c1cccc(=NCCCn2ccnc2)[nH]1)NCC(C)(C)F c1(C2C(C(=O)NCC3(N(C)C)CC3)(COC)C2)ccccc1 S(=O)(=O)(c1[nH]c(=NC(CO)C2CC2)ccc1Br)NCCc1scc(CSC)n1 C1(CNC(c2c(C)ccs2)=O)CN(C(C2CN(C(C)C)CCO2)=O)CC12CCC2 C(=O)(C(C)(C)C1CCN(C(=O)C(C)SC)C1)NCCN(C(=O)C(C)(C)C)CC c1(C(=O)NC(CN(C(c2c(C)nc(C(C)C)o2)=O)C)C)nc(Cl)ccc1Cl C1(S(C)(=O)=O)(C(=O)NC2CC(C)(NC(C=C3C(C)(C)CCCC3)=O)C2)CCCC1 c1(NCCOCC(CC)C)ccc(S(=O)(=O)NC(C)CCC2CC2)cc1C#N C1(NC(C2C(OCC)CC2)=O)CCC(C)(NC(=O)CCC2NC(=O)NC2=O)CC1 N1(C(=O)NC2(C(=O)O)CCCC(C)C2)CCC2(C1)CC2(F)F C(=O)(C1Cc2c(Cl)cccc21)NCC(C)N(C(C(CC(=O)OCC)(C)C)=O)C C1(CC)CCCCC1N(C(C1CCCSC1)C(=O)NCc1cccc(Cl)c1)C CC1C(C(=O)NC2(CCF)CCC2)CCN1C(=O)Cc1ccsn1 N1(C(Cn2c(C)ncc2)=O)CCC(C2CC2)C1CNC(C1CCCCCC1)=O N1(C(C2CCCCCC2)=O)CC2(CO)CC1(C(=O)NCc1cn(CCO)nn1)C2 C(CCCCC(=O)N1CCC(C(=O)NCc2ccc(C)nc2O)C1)OCC C1(OC)CCC(CC(N2CCCC2C2(O)CN(C(C3CC3CF)=O)C2)=O)CC1 C(=O)(CC(C)(C)CC(=O)NCCC(O)CNC(=O)CCC1CC(C)C1)OC CC(C)(CC(=O)N1CC2(CCCC(CNC(c3ccoc3)=O)O2)C1)CC(F)(F)F N1(C(CC(C)F)=O)CC2(CO)CC1(C(=O)NCC(C)OCCO)C2 Cn1c(C(=O)NCCC2CCCN(C(C3CCC(=O)O3)=O)CC2)ccc1[N+](=O)[O-] C1(CC(=O)NC2(COC)CC2)CN(C(=O)Cc2ccon2)CC12CC2 C(=O)(C(CCC(C)C)N(C)C)N(CC(CC)C#N)C1CNC(=O)C1 C(=O)(C(F)(CNC(C1CNC(=O)N1)=O)C(C)C)N1CCC(C(CC)C)CC1 CC(C)C(CNC(=O)CN(C1CC(C#N)C1)C(C1CCC1)=O)C(C)C C1(C(=O)NC(CN(C(=O)C2=CCC2)CC)C)OCC2CCCCC12 c1(NC(C)=O)cnc(C)c(C(N2CCC(NC(=O)CC3(C)CC3(F)Cl)CC2)=O)c1 N1(C(C2C(OC)CC2)=O)CCN(CCN(C)C(C2CCCN2C2CC2)=O)CC1 N1(C(C(COC)OC)=O)CCC(COC)(NC(C2Cc3nccn3C2)=O)CC1 c1(OC)cc(Cl)ccc1-n1nc(CC2(C)CC2)nc1CNC1CCOCC1 c1(CN(C(=O)NOC(F)F)CCO)cccs1 CC1(C)C(CNC(c2ccnc(F)c2)=O)CCN1C(c1ncc(Cl)cc1Cl)=O c1(C(=O)NCC(C(C)(C)C)NC(CCC=C=C)=O)nn2cccnc2c1Cl c1(C(=O)NC(C2CN(C(=O)CC3OCCO3)CCO2)C)cc2c(Cl)cccc2s1 C(C)(CO)(C(=O)NCCC1CCC(NC(=O)Cc2cccc(C(N)=O)c2)C1)OC N1(C(C2C(C)CCO2)=O)CC2CN(C(c3occc3Br)=O)CC2C1 C1(NC(c2cn(CC)nn2)=O)CC(O)CN(C(=O)CCC=CC(C)C)C1 N1(C(CN2CCC(OC)C2)=O)CCC(C(c2nccn2C)O)CC1 C1(C(=O)NCC2(CN(C(c3c(C)csc3)=O)C)CC2)CC2COCC2C1 CCCCC(CNC(=O)CCCCCN(C)C(C1(C2(O)CCC2)CC1)=O)CCC O=C(NNc1cc(F)c(Br)cc1Cl)c1ccccc1-n1cc(C2COC2)nn1 c1(C(=O)NC2C(NC(COc3cccc(C)c3)=O)C2)cnc(Cl)c(N)c1 C1(CC(=O)N(C)Cc2cnc[nH]2)COCCN1C(c1cncc(C(F)(F)F)c1)=O N1(C(CCC2CCN(C(N)=O)C2)=O)CCOC(C#N)C1.CC(C(=O)NCC)SC N1(C(C2(CC)CCC2)=O)CCC(CC)(NC(c2sc(C)nc2C(F)(F)F)=O)CC1 N1(C(CNS(CC)(=O)=O)=O)CC2CC(NC(=O)CCCCC(=O)NC)CC2C1 c1(C(=O)NCCC(=O)N(c2ccnc(C)n2)CC)cncc(OC)n1 C(C(C)CC(=O)Nn1cnc2ccccc12)NC(CCCCCNC(C)=O)=O c1(OC)ccc(CC(N2CCC(N(C(=O)CSC)CC3CC3)CC2)=O)cn1 c1(COC)nc(C)c(C(N2CCCC2C(C)NC(C2(O)CC2(C)C)=O)=O)s1 O=C1NC(=O)C2CN(C(C3(F)CN(C(c4cc(F)cc(F)c4)=O)C3)=O)CC12 c1(C(C)=O)ccc(CNC(=O)CCc2ccc(Cl)cc2Cl)cc1F C(=O)(C(C)(C)C(=O)NC)N1CCC(c2c(CNC(C(C3CC3)OC)=O)c[nH]n2)C1 c1(C(=O)NC(CNC(C(CC)C#N)=O)(C)C2CC2)cc(Br)c(C)cn1 c1(C(=O)NCCCCC(C)NC(C2(CC)CCOC2)=O)ccc2c(n1)CCC2=O N1(C(c2c(CC)c[nH]c2)=O)CCC2CCCC12C(=O)NC1(C)CC(O)C1 C1(NC(C(CC)(O)c2ccccc2)=O)CCN(C(=O)Cc2ccsc2C)C(C)C1 c1(C(N(C)CC2N(C(C3C(C#C)C3)=O)CCOC2)=O)cc(O)nc(C2CC2)n1 c1(OC)ccc(Cl)cc1NC(c1cc(-n2nnnc2C)cc(F)c1)=O CC1CN2CCN1C(C(=O)NCC1CC(NC(=O)CC(C)(C)O)C1)C2 C1(F)(C(N2CC(C(C)NC(C(CC)C)=O)C2)=O)CC=CCC1 O=C(C(O)C(F)(F)F)NC12CC(C(N3CC(O)C(O)C3CO)=O)(C1)C2 C(=O)(C1(O)CCCc2ccccc21)NCC(Cc1c(C)c(Br)ccc1)CO C1(N(C(=O)CCNC(=O)Cc2cnnn2C)C)CC2C=CC1CC2 c1(OC)nc(C(N2CCCCC2C)C(=O)NCc2ccco2)sc1C c1(N2CCC(CC)C2)nc(N2CCn3nc(C(C)(C)C)cc3C2)nc2c1CSC2 C(c1ccc(Cl)nc1)=CC(=O)NCCCC(C)NC(C1C=CC=CC=C1)=O C(=O)(C(O)CCC(C)C)N1CC(C#C)(C(=O)NCc2cc(CC)no2)C1 c1(C(=O)NCC(CCC)C(=O)NCC(F)Br)ccc2n[nH]cc2c1 Cc1cccc(C(N2CCOC(C)(CNC(C3CC3CF)=O)C2)=O)c1C#N C(=O)(C(F)C(C)(C)O)NCC1C(CC(=O)N(CCC(N)=O)CC)C1 C1(C(=O)NCc2ncc(OC)nc2)CCCN(C(=O)C(CO)OC)CC1 c1(N2C3(CC(COC)C3)CC2)ncnc2ccc(F)cc12 c1(CN2C(COC)CN(C(C3CCCCN3C)=O)CC2)cc(Br)cc(C)c1O c1(NC(C)=O)nc(CC(=O)N(C(C)CNC(c2ccon2)=O)C)cs1 Cc1ccc2c(N3CCN(C(=O)C(C)(O)CC(C)C)CC(O)C3)ncnc2c1 C1(NC(c2cc(C)c(C)[nH]2)=O)CC=C(C(=O)NCC(C)C2CCC2)C1 CS(=O)C=CC(=O)NCCC1CCN(C(C2CCCN2C(=O)C(F)(F)F)=O)CC1 N1(C(C(=O)N(C)C)=O)CCC2CCC(NC(c3cc(Cl)nnc3O)=O)C1C2 N1(C(C(C)NS(CC)(=O)=O)=O)CCOC(C(C)NC(c2cnn(C)c2N)=O)C1 O=C1CS(=O)(=O)CC(C(=O)NCC(O)CNC(=O)CC(O)C2CCCC2)N1 N1(C(CSCC#C)=O)CC2CCCCN2CC1CNC(=O)CC(=O)NCC C(=O)(C(CNC(=O)C(O)CN(C)C)C(C)(C)C)N1CCCC(C#C)C1 N1(C(c2c(C)csc2Cl)=O)CC2OCCN(C(c3c[nH]c(=O)cn3)=O)C2C1 c1(CNC(C=CCN(C)C(C2CCSC2)=O)=O)ccc(Cl)cc1 N1(C(CCCOC)=O)CCC(C#N)(NC(c2cccc(OC(C)C(=O)OC)c2)=O)C1 CC(CC(=O)N1CCCC1C1(NC(=O)C=CC(C)(C)C)CC1)CC(F)(F)F c1(C(=O)Nc2nnc(C(=O)NCCCC)s2)ccc2c(Br)cccc2n1 C1(C(=O)NC2(CF)CN(C(C(C)CN(C)C)=O)C2)CCCCN(C)C1=O N1(C(Cc2c(C)scc2)=O)CCOC(CCNC(=O)CC2CC(F)C2)C1 N1(C(c2c(CC)n[nH]c2)=O)CCC(NC(c2scc(C)c2Cl)=O)C(C)C1 N1(C(C(CC)C)=O)CCCCC(NC(=O)CN2CCCCS2(=O)=O)CC1 Cc1ccc(C(=O)N(CC(C)NC(=O)C2=CCOC2)C)c(F)c1F c1(-c2ccc(OC)nc2)cc(C(=O)Nc2ccc3c[nH]nc3c2)cc2cc[nH]c12 C(C(=O)OCc1nc(C2CCCCO2)cs1)(C(C)C)N(C(C)=O)Cc1ccccc1 c1(C(=O)NCC(C)(C(C)C)NC(c2ccc(OC)cc2)=O)cnn2c1N(C)CC2 N1(C(COCCCC#C)=O)CC(CC(=O)NCCn2cnnc2)CC1C C(C(F)(C(=O)Nc1cc(C)ccc1OC)C(C)C)NC(c1cccc(OC)n1)=O C12(CNC(=O)CC3CCOC3=O)CC(CN1C(=O)CCC1CCCO1)C2 O=C1NC(=O)C2(CCCN(C(=O)C(F)(F)c3cccnc3)C2)N1 C=C1COc2c(C(N3CC(F)(F)CC3C(N)=O)=O)cnn2C1 C1(OCCNC(=O)CC2CC3(CC3)C2)CCN(C(=O)Cn2nccn2)CC1 c1(C(=O)NC23CC(C(=O)NC4CCC(N(C)C)C4)(C2)C3)cnc[nH]c1=N n1(C(C)(C)C)nnnc1C(C1CC1c1cccs1)NCC1CCCO1 CC1CC=C(C(=O)N2CC3CN(Cc4cc(C#N)ccc4F)CC3C2)CC1 Cc1nc(F)ccc1CN1CCCCC1C(=O)NCCC(C)C N1(C(=O)NC)CCCC1(C)C(=O)N(CCCNC(c1ccncc1C)=O)C C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1ccoc1C)NCc1c(C)cccc1 c1(C(N2CC(CC)C2)=O)ccnc(-c2ncc[nH]2)c1.C12(CC1)C(=O)NCCN2C c1(OC)ccc2cc1NC(=O)COc1ccccc1NC(=O)N2.C(C)(C)O O=C1CC(=O)NC(C(=O)NC2(CC(N3CCOCC3CO)=O)CCCCC2)C1 c1(C(N2CC(CC)C(NC(=O)C=CCO)C2)=O)ccc(S(=O)(=O)NC)o1 C1(O)(CNC(CS(N)(=O)=O)=O)CCN(C(=O)CCC(=O)c2ccc(F)cc2)CC1 C1(C(C)NC(COC(CC)CC)=O)CCN(C(=O)C(=O)NCC(F)F)C1 N1(C(CC=CC)=O)CCC(N(C)C(C2CC(CC(C)(C)C)C2)=O)CC1 c1(C(N2CC(CNC(C3(C)N(C)CC(OC)C3)=O)C2)=O)c(O)ccc(Cl)c1F C(=O)(CCCCCC(C)O)NC(CC=C)CNC(c1cncc2ccsc12)=O C1(C(C)NC(c2ccccc2)C(=O)N(C)C)CCN(Cc2n[nH]cc2F)C1 C#Cc1ccc(OCC(=O)NCC2(C)CN(C(c3cnn[nH]3)=O)CCO2)cc1 CCCC(C(=O)N1CC=CC1CNC(=O)CC1CCN(C(C)=O)CC1)C(C)C C(C1=CCN(C(=O)C2=CCCCO2)CC1)NC(C1CCC1c1nc[nH]n1)=O C=CC1(CC(=O)NCC2CCC(NC(c3cnccc3OC)=O)C2)CCOCC1 C1(N(C(=O)CC#N)C)CCCC(CNC(c2csc(CO)c2)=O)C1 N1(C(C(C)=CC)=O)CC2(C1)CN(C(c1cccc(I)c1)=O)CCO2 C1(C(=O)Nc2cn(C)nc2)C2CCC(C2)C1NC(=O)Cc1csnn1 C1(NC(C(C)=C(C)C)=O)CC(CC(=O)NCc2ccsc2)C1(C)C C1(C(=O)NC(C)CC2CN(C(C3(C(F)F)CCCO3)=O)C2)CC2(C1)CC(F)(F)C2 N1(C(C(CC)COC)=O)CC2(C1)CN(C(c1cc(C3CC3)ns1)=O)CCO2 C1(C(=O)NC2CC(NC(=O)C(C)SCC3CCCCO3)C2)(OCC)CCCC1 C(C(F)(F)CCC(=O)NC(C12CCCCC1C2)C1CCCO1)n1cc(C(C)O)nn1 CC1(C)C(CNC(=O)CCOC2CCOC2)CCN1C(=O)CC(F)(F)F C(C1=CCCSC1)(c1n(CC(=C)C)nnn1)NC(c1ccccc1)C c1(OC(C)C(=O)N(CCCNC(C2(C)CSC2)=O)CCO)cccc(F)c1 c1(CC(=O)NC(CC=C)CNC(=O)CC2(C(=O)OC)CC2)ccc(O)c(Cl)c1 CC1CN(c2cc(Cl)ncn2)CCC1C(=O)NCc1cc2c([nH]1)CCC2 CN=C(NCC=Cc1ccccc1)N1CN(C)C(=O)C1C CC1(N(ONC(C2CC23CCCC3)=O)C(C2CCCCCCC2)=O)CCCC1(F)F c1(OC)ccn2cc(C(=O)NCC#CCNC(c3ccn(CC#N)n3)=O)nc2c1 C1(C(N2CC(C)(CC)C2)=O)CC(C)(C)CN1C(C1CC(=O)C1)=O C1(C(N2CC(NC(c3cc(CCC)on3)=O)C(C)C2)=O)CC2(CCC2OC)C1 c1(C(C)NC(c2nc(C)sc2C)C)ccccc1[N+](=O)[O-] N1(C(c2ccn(C(C)(C)C)n2)=O)CC2(CCCC2NC(=O)Cc2cnsc2)C1 c1(CCCC(=O)N(C2CN(C(c3cnc(C)[nH]3)=O)C2)C)ccc(F)cc1Br C1(OC)(CNC(c2c(Cl)cncc2Cl)=O)CCN(C(C2CC(=O)C2(C)C)=O)CC1 c1(C(=O)NCCC2N(C(C(CC)O)=O)CCCC2)cnc(Cl)c(F)c1N O(NC(=O)C(CNC(c1cnn(C2CC2)c1)=O)C(C)C)CC(C)C CC(C)C(C)CC(=O)NCC12CC(NC(=O)CN3CC4CCC3C4)(C1)C(C)O2 c1(C(N2CC3CCN(C(c4c[nH]c(=N)o4)=O)CC32)=O)cc2cc[nH]c(=O)c2s1 S(=O)(=O)(c1ccccc1F)NCCCC(N1CC(C#N)(CC(=O)OCC)C1)=O C1(C(=O)NCC2CCN(C(CC3CC(SC)C3)=O)C2(C)C)CCOCC12CCC2 c1(C(C)NC(CC2CC(NC(C3C(=C)C3C(=O)OC)=O)C2)=O)nn(C)cc1O c1(CC)nccnc1NC(C1CCCC1Cn1cc(-c2cccnc2)nn1)=O C1(NC(c2cc(CCC)on2)=O)CCN(C(c2ccc(C3CC3)o2)=O)CC1(C)C N1(c2n3c(nn2)C(F)(F)C3OCC)CCC2SC(=O)C=C2C1.C1CC1.OC c1(SCC(=O)NCCCOCCNC(C(=O)OCC)=O)n[nH]c(C)n1 N1(C(CCc2nnc(C)n2C)=O)CC2(CNC(c3cnc(Cl)[nH]3)=O)CCC1CC2 C=CCN=c1nc(N2CC3CN(C)CC3(C)C2)c2[nH]ccc2[nH]1 C(=O)(C1=CC2CC=CCC12)N1CC(O)(CNC(c2[nH]c(CC)c(Cl)n2)=O)C1 N1(C(CSCC#C)=O)CCC2(C=C(C(=O)N(C)CCOC(F)F)C2)C1 C1(NC(c2cc(Cl)nnc2Cl)=O)CC2CN(C(=O)COc3cccc(F)c3)CC12 C(=O)(C1CCCc2sccc21)N1CC(O)(CN(C)C(C2COCC(C)(C)O2)=O)C1 c1(C(=O)NCC2OCCN(C(c3c(C)ccnc3Cl)=O)C2)cccc2cnnn12 C1(CNc2cccc(COC)c2)OC2CCC1CC2.c12ccc(nn1)c(=O)o2 N1(CC=C)CCN(C(=O)CN2CCN(C(=O)C(C)CCO)CC2)CC1 N1(C(C2CC(N(C)C)C2)=O)CC(F)CC1CNC(=O)C=CC1(C)COC1 C(CCCC(C)(C)C)NC(C(C(C)O)NC(=O)CCCCOC(C)(C)C)=O C1(C(N2C3CN(C(C(N4CCC(C)C4)=O)=O)C(CC3)C2)=O)CCc2c(cnn2C)C1 n1(CC)ccc2cc(Sc3nc(-c4nc(C)ccc4OC)n(CCF)n3)ccc12 C(C#CCCCC)(OC(C1C(c2n(CC)cnn2)C1)=O)OC CC1CN(C(=O)Cc2cnco2)CCC1NC(=O)CCCC(=O)N(C)C CC1(NC(c2cnc(S)[nH]2)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)C1 C1(CC(=O)N(C2CC(C#N)C2)CC(=O)N(C(CCO)C(F)F)C)C(C)(C)C1(C)C c1(C(=O)NCCC(C)N(C)C(C2CCC(=O)N2)=O)csc(-c2cnc[nH]2)n1 CC(CC(=O)NC(C(=O)NCc1ncco1)c1cccs1)n1cccc1 CC(C)S(=O)(=O)c1cccc(C(=O)NCCCCNC(=O)CC(C)(C)C)c1 CC(N=c1[nH]c2c(c(=NC3CCCS(=O)(=O)C3)[nH]1)CCCCCC2)c1cnc[nH]1 c1(C(=O)NC2CC(NC(c3ncc(OC)cc3F)=O)C2)cc2cc(F)ccc2[nH]1 C(CC(C(=O)Nc1cnn(CCOC)c1)NC(C1CC12CCCC2)=O)OC C1(CCCNC(c2c(C)nco2)=O)CN(C(c2cnccc2N(C)C)=O)CCO1 N1(C(=O)Cc2cnns2)Cc2ccc(CNC(C3CC4CCC3C4)=O)cc2C1 c1cnc(Cl)c(C)c1.c1(NC(C#C)=O)cccc(C(=O)N(N2CC(N)C2)C)c1 N1(C(C(CC#C)C)=O)CCC(CCOC)(NC(=O)CC(C)c2cnn(C)c2)CC1 c1(OC)cccc(C(C(=O)NCC(F)CNC(c2nc(C)sc2C)=O)OC)c1 c1(C(N(CCCN(C(=O)CCc2cccnc2F)C)C)=O)ccccc1O C1(CN(C(=O)Cc2cncnc2O)C)CCCN(C(=O)COc2ccsn2)C1 O=C(C1Cc2ccc(Cl)cc21)NC1CN(C(c2ccc(Cl)o2)=O)CC(F)(F)C1 c1(C(=O)NC2CC(NC(C(CO)N(C)C)=O)C2)ccnc(Oc2cccnc2)c1 N1(C(C(C(=O)OC)C)=O)CCC12CCN(Cc1cc(Br)cc(C)c1O)CC2 CC(CC(C)NC(=O)CCC1CC1)NC(c1n[nH]c(-c2ccccn2)n1)=O N1(C(CC(CCC)O)=O)CCC(C(=O)N2CC(C(N)=O)C(C)C2)=C(F)C1 C1(N(C)CCN2CCC(O)C2)CCN(c2nnnn2-c2ccccc2)CC1 C(c1ccccc1F)=CC(=O)C(N1CCCC(CNC(C2CC2(Cl)Cl)=O)CC1)=O N1(C(CCC(C)C)=O)C2CCC1C(F)C(NC(=O)CC1(CS(C)(=O)=O)CC1)C2 C(=O)(CC(C)C(C)(C)NC(CO)C1CCC1)NC(C12CCC(CC1)CO2)C CN1C(=O)CN(CC(N2CCC(NC(c3ncnc4sccc34)=O)C2)=O)C1=O C(=O)(CCCn1cncn1)N(C(C)C(=O)NC1CCC1N(C)C)CC C1(C(=O)NC(C2CCN(C(c3csc(-c4cnc[nH]4)n3)=O)C2)C)CC(F)(F)C1 C1(C(N(CCNC(C2(N(C)C)CCCC2)=O)C2CC2)=O)CC12CCC(F)(F)CC2 C(=O)(C#CC1CCOCC1)NCC1N(C(c2cc(S(=O)(=O)N(C)C)oc2)=O)CC1 c1(C(N2C3CN(C(c4cc(C)[nH]c4C)=O)C(C3)C2)=O)c(C)ccc2ccccc12 C1(C(C)C)CCCN(C(=O)CN(C(c2ccnnc2)=O)CC2CC2)CC1 CC1(C)CC(C(=O)NC(C(=O)N2CC(c3cc(O)no3)C2)C2CC2)=NO1 C1(=O)C2=NOC(C2)CN1.c1(C(=O)NCCc2c(C)nc[nH]2)c(C)oc(C)c1C c1(C(C)C)cc(C(=O)NCCC(O)CNC(=O)CN(C2CCSC2)C)ccc1O c1(C(=O)NCCCCC(CO)NC(C2(C)CC2)=O)cc(Cl)c(F)c([N+](=O)[O-])c1N C1(=O)C(O)CCNC(=O)NC2CN1C2.C12(CNC(CCC)=O)CC(C(=O)OC)(C1)C2 N1(C(C2CCCC(NC(c3nc4ccccc4[nH]3)=O)C2)=O)CC(=O)NC2(CC2)C1 CCCS(=O)(=O)C(C)C(=O)NCC(C1CCCN1C(c1ccncc1O)=O)(C)C C1(CC(=O)Nc2ncc(C#C)cn2)CCN(C(=O)OC(C)(C)C)CCC1(F)F Cc1ccc(-c2cc(NC(=O)C(C)OC(c3cnn(C)c3C)=O)n[nH]2)cc1 N1(C(C(C)=CC2CC2)=O)CC(CNC(c2c(F)cccc2Cl)=O)CC1(C)C C(=O)(C1=C(Cl)CCC1)NC(C1CCN(C(=O)CCc2nncn2C)C1)C N1(C(C2N(C)CCCC2)=O)CC2(CC2)CC1CNC(=O)COCC1CCCC1 c1(CC)cc(N)c(C(=O)NCC(CNC(=O)CCCCCN(C)C)OC)c(F)c1 c1(OC)ccc2cc(C(=O)NC(c3cnc(C)nc3)(C)C)[nH]c2n1 c1(C(N(CC(C)NC(=O)CC23CCCC2C3)CC)=O)ccnc(C(N)=O)c1 c1(C(=O)NC2C3(CC(NC(C(COC)(C)OC)=O)C3)C2)cnc2c(C)cccn12 c1(Cc2onc(C(C)(C)NC(c3ccccc3)=O)n2)ccc(N)c(Cl)c1 C=CCC(C(=O)NC(CNC(=O)CCNS(C)(=O)=O)CC(C)C)NC(C)=O C1(CCC)CN(C(c2ccncc2Br)=O)CCN1C(C12CC(O)C1C2)=O c1(C(=O)C(N2CCCCC(CN3CCNC3=O)C2)=O)cc([N+](=O)[O-])c[nH]1.C1CN1 Cc1cc(C)n(CC(N2CC(NC(C3CN(CC(C)C)C3)=O)C(O)C2)=O)n1 Cc1cc(C)c(C(=O)NC2CC(NC(c3cc(C4CC4C)on3)=O)C2)cn1 CCCC(C(O)C(=O)NC1C2CCC(C2)C1CO)NC(C1(C#N)CC(=O)C1)=O C1(C(=O)NC(c2cccnc2)CC)CC12CCN(C(=O)CC1CC=CC1)CC2 C#CC1CC2CCC1N(C(=O)C(CNC(=O)C1=C(Cl)CCCC1)CC=C)C2 CCC(CNC(C12COCC1C2)=O)(CC)NC(=O)CCc1cncnc1 C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CCC(CNC(C3CCC(C)CC3)=O)O2)C1 CCC(CCC(=O)NCC(O)CC(F)(F)F)NC(c1cccnc1NC)=O N1(C(CCN(C)Cc2nc(C#N)cs2)=O)CCN(C(N)=O)CC1 C1(C(N(C2CCN(C(=O)Cn3nnc(C)n3)C2)CC#C)=O)CC2(C1)CC(C)(C)C2 C(N=c1ccc(Br)c(S(=O)(=O)N2CCC(C(N)=O)C2C)[nH]1)c1c(CC)c[nH]n1 C(CCC(C(=O)NOCCC(F)F)NC(C1OCCOC1C)=O)OC CC1CCC(NC(c2ccc(C3CC3)cc2)=O)CN1C(=O)Cc1cccnc1 N1(C(c2cc(C)nnc2O)=O)CC2ON=C(CNC(=O)C3=CCCCC3)C2C1 c1(NC(=O)NCCC(Cc2ccccc2)NC(=O)OC(C)(C)C)ccc(O)nc1 c1(OC)ccc2cnc(N3CC4(CCC(C(=O)NCCCO)O4)C3)nc2c1 c1(C(N2CCC(C)(NC(CN(C3CCCC3)C)=O)C2)=O)cncc(O)c1Cl C1(C2CCN(C(=O)CC3CCC4(CCC4)O3)C2)(NC(CCCCOCC)=O)CC1 Cc1cccc2cc(C(=O)NC3CC4(C3)CC(CNC(=O)COC(C)C)C4)sc12 c1(C(=O)Nc2cccc(NC(N3C(CSC)CCC3)=O)c2)ccc2nccn2c1 c1(C(=O)NC2(CCNC(CC3(C)CC3)=O)CC2)cc(C(F)F)ccc1Cl C1(C)(NC(C2OCCN(C)C2)=O)CCC(NC(=O)CCCC#N)CC1 c1(CC)ccc(C=CC(=O)NC2CC2CNC(=O)Cn2ncc(Cl)c2C)cc1 CC(C)CC(CNC(c1ccnn1CCN(C)C)=O)NC(c1ccc(F)s1)=O C1(CNC(CSCC#C)=O)CC(C)N(C(c2oc(-c3ccccc3)nc2C)=O)C1 c1(C(C)C)ccc(C(=O)NCC2CCC(NC(C3(C)CSC3)=O)CC2)cc1 N1(C(c2ccc(COC)s2)C(=O)NC2CC(OC)C2)CCC(CC2CC2)C(C)C1 Cc1sncc1N(C(=O)C(C)NC(=O)NC1CN(C(N)=O)C1)C CCCCC(F)C(=O)N(CCCNC(=O)C(C)(C)C(F)F)C1CC1 C1(CC(=O)NC)CN(C(C2CC2c2ccno2)=O)CCN1C(=O)C1CC1 C1(C2CC2)(CNC(CCC=CC)=O)CCN(C(C2OCCOC23CCC3)=O)C1 C#Cc1cccc(NC(=O)N(C2(C)CCS(=O)(=O)CC2)CC(=O)OC(C)(C)C)c1C N1(C(C(CC2CCC2)OC)=O)CCN(CC(C)NC(C2(C)CC(C)(C)C2)=O)CC1 N#CC1CCC(C(=O)NCCCCCCNC(=O)C(F)C2CCC2)CC1 c1(CC)cc(C)cc(CC)c1NC(C1CC1NC(=O)C=CC(=O)OCC)=O c1(OC(C)C)ccc(CNC(c2cnc(Cl)s2)c2nnnn2C(C)(C)C)cc1F CC1(C)C(O)CCCN1C(C1CCN(C(=O)CC2C=CCC2)CCO1)=O c1(NCCOC)cncc(C(=O)NCCN(C)C(C2CC(C)(F)C2)=O)c1 N1(C(c2ccc(C(=O)NC)nc2)=O)CCOC(C)(CNC)C1.C(C)(C)C N1(C(CCC=CC)=O)CCCCC1C(=O)NCC(O)CF C(CSC)(C(=O)N1CC(O)(C(C)NC(C2(CCO)CC2)=O)C1)OC C1(CC(N2CC(C#C)(F)C2)=O)CC2(C1)CN(C(c1cnsn1)=O)C2 C1(C(=O)NCC(C)CN(C(=O)C(c2cccc(F)c2)O)C)CN(C)CCO1 C(=O)(CCC(C(=O)Nc1cccc(CNC(c2ccccc2F)=O)c1)OC)OC N1(C(CC(CC=C)NC(=O)C(O)C2CCCC2)=O)CCC(C)C(C)(C)C1 C(=O)(C(C)CC1CC1)NCCCOCCC(=O)N(CC)Cc1cccs1 C(=O)(CC(CC(C)C)n1ccnc1-c1cc2cccc(F)c2o1)OCC N1(C(C(CC)=CC)=O)CC=C(CNC(=O)C(C)NC(=O)OC(C)(C)C)CC1 C(CC(=O)Nn1ccnn1)N(C(=O)C(CC)C=O)C1CC1.CC N1(Cc2cc(C)sc2)CCCCC1CF.n12cc(nn1)-c1ccc(s1)NCCC2 c1(C(C)=O)ccc(Br)c(C(=O)NC2CN(Cc3cc(Br)c(Br)s3)CC2(F)F)c1 c1(CC)ccc(C)cc1C(=O)NCC(n1cc(CN(C)C(C)C)nn1)C Cn1c(=O)ccn(CC(=O)NCC2CN(C(=O)CC3(O)CC3)CC2(C)C)c1=O CC1(C)CC(C(=O)NCCOCCNC(c2cn3cnnc3cn2)=O)CNC1=O c1(C(N2CC(NC(C(c3c(OC)cccc3)=O)=O)C(C)C2)=O)cc(Cl)ccc1N Cc1ccc(C(N2CC(NC(=O)CC3CCC(=O)N3)CC23CCC3)=O)cc1C#N CC(CCCC(=O)OC(C)(C)C)NCCS(C)(F)N C1(NC(=O)C=Cc2cnc[nH]2)CC2CN(C(C3COC(=O)C3)=O)CC2C1 CC1CC1C(=O)NC.N1CCOC(c2nncn2C)C1.c1ccccc1 C=CC1(c2ccccc2)COCCN1C(=O)CS(=O)(=O)CC1COCCO1 C(C(C)(O)CC(=O)NCP(C)(C)=O)OCC.C1CCCCC1C#N C1(NC(c2coc(CO)c2)=O)COC2CN(C(C3CCC34CCOCC4)=O)CC12 c1(C(=O)NCCCCN(C(C2(C)N(C)CC(OC)C2)=O)C)ccc2cncn2c1 c1(NC2(CNC(c3c(OC)ccs3)=O)CCOCC2)cc(O)nc(=O)n1C C(=O)(C1Cc2ccc(F)cc21)N1CCC(CCNC(C(CC(C)(C)C)F)=O)C1 Cc1cc(OCC(=O)NC2CCC(NC(=O)C(C)SC3CCCC3)C2)ccc1Cl c1(-c2cc(CNC(C(C(C)C)O)=O)sc2)cc(O)c(F)c(F)c1 CC(=O)CCCCC(=O)NCc1nc(C)c(C(N2CCC3(CCO3)C2)=O)o1 Cn1nnnc1C(c1nc(C2OCCO2)cs1)NC1(CCC(C)(C)C)CC1 c1(C2N(C(C(C)(C)NC(C)=O)=O)CCC2)ccc(Cl)c(F)c1.C12CN(CCO1)C2 C1(NC(c2cnc(N(C)C)o2)=O)CN(S(=O)(=O)Cc2ccccc2Cl)CC1O c1(C(=O)NCC2(C)CC(NC(c3nc(C)oc3)=O)C2)nnc(O)nc1O N1(C(CCC=CC)=O)CC(NC(=O)CCn2nc(C)c(C)c2C)CC12CCC2 CCCC(CNC(c1ncccc1N)=O)C(=O)Nc1ccccc1F N1(C(CS(=O)(=O)NC)=O)CCC(NC(=O)CC2CCC(C)(C)C2)C(F)(F)CC1 C12(C(=O)NC3CCN(C(CC4CCC(C)C4)=O)C3)CC3CC1(CO)CC3C2 C1(C(=O)NC(C2N(C(CCCOCC)=O)CCC2)(C)C)CS(=O)(=O)CC12CC2 c1(OC)cccc2c(C(=O)NC(C3CC3(F)F)C)coc12 c1(CC(=O)NCCC(C)NC(c2nccnc2C(N)=O)=O)ccc2c(c1)COC2 c1(OC)cccc2[nH]c(C(=O)NCCC(C)NC(c3ccc(F)o3)=O)cc12 N1(C(C(C2(O)CCC2)NC(C(CCOC)C)=O)=O)CCCOCC1C c1(C(N2C(C(N3CCC(C(=O)NC)C3C)=O)CCC2)=O)cc(=O)n(C)cn1 CC1Cc2cc(NC(=O)C(CO)c3ccccc3)ccc2O1 C1(CNC(=O)NCCc2c(C)ccnc2)CCC2(CCC2)CO1 n1(CC(=O)N(C2CCS(=O)(=O)C2C)C(=S)SC(C)C)ccc(S(C)(=O)=O)cc1=O.CO Cc1nc(C(N2CCC(O)(C(C)CNC(=O)COC3CCCC3)C2)=O)c(C)s1 C=CC1OCCC1C(=O)NC1(CF)CCN(C(=O)CC2(CS(C)(=O)=O)CC2)C1 C1(C(C)C)C(=O)NCCN1C(C1CCN(Cc2ccc(Cl)cc2)C1)=O C1(C(=O)NCC2(C(=O)NC3CCCC(C)CC3)CC(=C)C2)C2CCCCCC12 C(=O)(C(O)CC(N)=O)N1CC2C(NC(CSCCN(CC)CC)=O)(C2)C1 c1(C(N(C)CC2(NC(C3ON=C(C)C3C)=O)CC2)=O)sc2cccnc2c1Cl CC(=O)CCN=C(NCc1[nH]c(C)nc1C)N1CCC(C)(F)C1 C(=O)(C1SCCc2sccc21)NCc1ccc(CN(C(CC(C)C)=O)C)cc1 c1(C(=O)NCC(CN(C)C(c2ccnc(CO)n2)=O)O)cccc2oc(O)nc12 C=C(C)CCC(=O)NC(CNC(c1ccncc1OC(C)C)=O)C(C)C c1(C(=O)NCC2CCCCN2C(c2cc(F)ccc2F)=O)ccc2cncn2c1 N1(C(=O)CCCC2CCC2)CCCC(F)(CNC(C2(C3CCCO3)CC2)=O)C1 C1(CCNC(c2cc(CN(C)C)on2)=O)COCCN1C(=O)CCc1cccs1 C(C(C)C#N)N(C(=O)C=C(C)CCC)CC.C1C(=O)N1CCOC c1(C(N(CC(CN(C(=O)CC2C(C)(C)C2(C)C)C)O)C)=O)ccc2c[nH]nc2n1 c1(C(=O)NC2CC(C)(NC(CC34CC(C)(OC3)C4)=O)C2)ccc2oc(=N)[nH]c2c1 C(=O)(C#CC1(C)CCCO1)NCC1(O)CC(CNC(c2c(F)ccc(C)n2)=O)C1 c1(C(=O)NC2C(NC(C3(C)CNC(=O)C3)=O)CC2)nc2cccnc2s1 N1(C(C2CC(C)C2)=O)CCC2(CC1)CCN(C(=O)CCC(N)=O)C2 C=C(C)CN=C(NCC(=O)NCC(F)F)N1CCC(OC2CCCC2)CC1 C1(C(=O)NC2CCN(C(CCSC)=O)CC2)CCc2n[nH]cc2C1C C(CCN(C)C)(C(=O)NOC1CCOC1)NC(c1nc(OCC)oc1)=O c1(C(=O)NCCC(C)NC(c2ccn(CCOC)n2)=O)coc2c1COC2 C1(CNC(C(C)=C2CCCC2)=O)CN(C(c2cccc(N)n2)=O)CCN1C N1(C(C(C(C)C)O)=O)CC2(CO)CC1(C(=O)NCC(O)CCC1CC1)C2 c1(C(=O)NC(CNC(C(C)=C(C)C)=O)C)cnnn1C N1(C(=O)C2CC2)CCC2CN(C(c3ccsc3)C3CN(C4COC4)C3)CC12 N1(C(C2C(OC)CCC2)=O)CCC(O)(CNC(=O)Cn2cc(F)ccc2=O)CC1 c1(C(=O)NCCCCNC(C(CC=CCC)C)=O)cc(C(F)(F)F)ccc1F C=C=CC(C)C(=O)NCC(C)CNC(C1(c2cccc(F)c2)CCCC1)=O N1(C(C2C(C(=O)NC(c3ccccc3)C)C2)=O)CCCC1c1ccccc1 N1(C(c2c(NC)cncc2)=O)CC(NC(=O)C(C)CC(N)=O)CC(F)(F)C1 CC(CNC(=O)OC(C)(C)C)CC(=O)NCC(C)N(C(=O)C(F)=C1CCC1)C c12cc(ccn1)OCC(=O)N2.C(CCCN(CC(N)=O)C)N(C)C(C1CCOC1)=O c1(OC)cccc2c(N3CCOC(c4ccc(F)c(F)c4)C3)nccc12 c1(C(N(C(CC)C(=O)NC(c2n[nH]c(CO)n2)C)C)=O)c(SC)cnn1C N1(C(CCCCC)=O)CCCC2CN(C(c3ccc4c(c3)OCO4)=O)CCCC12 N1(C(CC2CCC(C)CO2)=O)CC2CCN(C(=O)CCC3CCOCC3)C(C2)C1 c1(Sc2cccc(C(=O)NC)c2)nc(=N)[nH]c(=NCC2CC(N(C)C(C)=O)C2)[nH]1 C1(C(=O)NCC(CC2CN(C(COC(CC)C)=O)C2)(C)C)CC2(CCOCC2)C1 c1(NCC2(N(C(=O)CCc3cn(C)cn3)C)CC2)cc(O)nc(=O)n1C CN1CCOc2c(C(=O)N(C3CCN(C(c4cnc(O)s4)=O)CC3)C)cccc21 C1(NC(C2CC(OC(C)C)C2)=O)CN(C(=O)CC2CCCOCC2)CC1C1CC1 C1(NC(CCCn2cc(-c3n[nH]c(C)c3C)nn2)=O)CCNC2(CC2)C1 C1(CNC(CCC(C)OC)=O)CC(C)CCN1C(c1ccco1)=O C(=O)(C1CCCc2nc[nH]c21)NC1CCN(C(c2c(N)nc(Cl)cc2)=O)C12CC2 N1(C(CNC(C(CC)C)=O)=O)CC2CC(C1)C2NC(C1CCCCO1)=O N1(C(C2CCCSC2)C(=O)NC(C)C)CCCCC2(CCC2)C1 N1(C(C(C(C)C)F)=O)CCCC(O)(CNC(C2CN(C3CCC3)C2)=O)CC1 c1(OCC(N2CCC(C)(NC(C(CC=CC)C)=O)C2)=O)c(C)cc(Cl)cc1C Cn1nc(C(=O)NCCC2CCCN2C(=O)C(F)C2CCC2)c2c1CCCC2 C#CC1(C(N2CCC(N(C(=O)Cc3ccc(C)nc3)CC3CC3)CC2)=O)CCCC1 C1(F)(C(N2CCC(OCC#C)C2)=O)CCN(C(c2n[nH]c(O)n2)=O)CC1 c1(OC)cccc(F)c1C(C)NC(=O)C(=O)N(CC(c1ccc(C)cc1)O)C c1(C(=O)NCC(=C2CN(C(c3[nH]cc(C)c3)=O)C2)F)ccccc1C1CC1 Cc1coc(C(=O)N(C(c2ccccc2)CNC(=O)Cc2ccsc2)C)c1 C1(C(=O)NC(CNC(COc2c(C)cc(Cl)cc2)=O)C)CC2CCCCN2C1 C1(N(C)C(c2ccco2)=O)CN(C(c2cc(Cl)ccn2)=O)CC12CC2 c1(CCNC(CCSCCCC)=O)n[nH]cc1C(=O)NCCSCCOC S(=O)(=O)(c1ccc(C#N)c(N2CCC=CC(O)C2)c1)N(CCC(F)(F)F)C n1(C(C)C)nc(C(=O)NCCCC(C)NC(C2(C)CCCO2)=O)c(Br)n1 c1(C(=O)NC(C(C)NC(c2cc(C(F)F)n(C)n2)=O)C)sc2cccnc2c1Cl C1(CNC(=O)Cn2cccc2)CCCC1NC(c1nsnc1O)=O C1(CCNC(C2C(OC)C2)=O)CSCCN1C(=O)C(=O)Cc1ccc(Cl)cc1 C#Cc1ccc(C(=O)NCCCN(C)C(c2ccn(CC(C)C)n2)=O)cn1 N1(C(C2C(C)CCCC2)=O)CCCC(C2CCN(C(C3CSCN3C)=O)CC2)C1 CC1(c2nn[nH]n2)CCCN(CCS(C)=O)C1 CCC(C)(C(=O)N1CCC(N(C(=O)Cc2cc(-c3ccccc3)on2)C)C1)OC N1(C(C2CC3(C(OC)CC3)C2)=O)CC2CCC(C1)N2C(C1CC(OC(C)=O)C1)=O N1(C(C=CC)=O)CCC(C)N(C(c2ccc(CN(C)C)c(F)c2)=O)CC1 C1(NC(c2ccccc2Cl)=O)CN(C(C2CC2c2cccc(F)c2)=O)CC1O C#CC1(C(=O)NC2CC2C(C)C)CCN(NC(C2CC23CC3)=O)CC1 c1(C(N2CCN(CCNC(C(CC=C)C)=O)CC2)=O)ccc2c(c1)COC2=O C(CN=[N+]=[N-])(C(C)C)NC(C(CCC)NC(=O)CCCC1CC1)=O C(c1cncc(C)c1)=CC(N1CCC(N(C(C2CC2(F)Cl)=O)CC)C1)=O C=CCC(CC=C)C(=O)NC(C)CCC(=O)N1CC(CC23CC(C2)C3)C1 c1(C(=O)NC2C(C)CN(C(=O)CNS(N)(=O)=O)CC2)[nH]nc2c1CCC2(C)C N12CC3C(C3C1)C(=O)N(C)CCC2.c1(CC(C2CC2)N)ccc(F)cc1.COC C(=O)(C(=O)CCC(C)C)N1C(C(=O)NC(CC=C)(C)CC=C)CSCC1 c1(SC)ccc(O)c(C(=O)NCC2CC2CNC(=O)C(N2CCNC2=O)C)c1 c1(CCC(=O)NCCOCCNC(CC(C)(C)F)=O)nc2cc(Cl)ccc2s1 c1(C(CC)C)ccc(C(C(C)C)Nc2ncc(C3CC3)s2)cc1 C1(NC(c2c(OC)nc(Cl)cc2)=O)CN(C(C23CCCC2C3)=O)CC(F)(F)C1 C(=O)(C(O)CNC(c1coc(C)n1)=O)NC(c1ncc(C)[nH]1)CC Cc1ccc(Br)c(C(=O)NCC2CCCC2NC(=O)CC(C)C)c1 CC1CC(CNC(c2cc(C3CCC3)on2)=O)CN1C(=O)CN1CCSCC1 CS(=O)(=O)CC(=O)N1CCC(C2N(C(c3ccsc3)=O)CC2(C)C)CC1 C(N=c1[nH]c2ccc(O)cc2s1)C1CCCN(C(C2(CC=C)CCCCC2)=O)C1 C1(C(N(CCCO)C)=O)CC(C)N1C(=O)CCC1CCCC1 N1(C(CCS(=O)(=O)NC)=O)CCC2CCC(NC(c3cnncc3C)=O)C1C2 CCC(O)C(C)C(=O)NCC1(NC(C2CN(CC)CCO2)=O)CC(F)(F)C1 C1(C)(CC)CC(NC(=O)CN(C(=O)CN2CC(C)(OC)C2)C(C)C)C1 C(=O)(C1(C)OCCc2ccccc21)NC1C(NC(C2(CC)CC2)=O)CC1 C(C(=O)NOCC1CCCO1)(C1CCOC1)NC(c1cc(OC)n[nH]1)=O c1(C(=O)NC(C)CCCNC(C2(C)C(C)(C)C2(C)C)=O)ncc(Cl)c(N)c1Cl c1(C(C)CC(=O)NC2(CNC(c3cnn(C)c3)=O)CCCC2)ccc(F)c(F)c1 n1(CC(=O)N(CCC)CCNC(c2csnc2C)=O)nc(C)n(C)c1=O C1(C(N2C(CNC(c3c(CC)[nH]cc3)=O)CC(F)C2)=O)Cc2ccccc2C1 C(=O)(CCCC(=O)OC)N1CC(CNC(C2(COCC)CCCC2)=O)C(C)C1 Cn1nc2c(c1CNS(=O)(=O)c1cscc1Br)CCCC2 C1(CC=C)(NC(C2CCCC2CC)=O)CCCN(C(C2COC(C)(C)C2)=O)C1 C(=O)(CC(C(C)(C)C)NC(c1ccc(O)c(C)c1)=O)NCC(=O)OCC#C C1(NC(c2ccc(Br)nc2O)=O)CCCN2CCCC12 n1(CC)cc(Cl)c(C(=O)NCC(C2CCCCC2)NC(C2CCC(C)(C)C2)=O)n1 Cc1ccc(-c2cncc(C(=O)N(CC(O)CNC(C3CC3F)=O)C)c2)cc1 C12(CNC(C3(C(C)(C)C)CCCC3)=O)CC1CN(C(=O)CC1CCCC13CC3)C2 c1(C(N2CC(NC(C3CC(OCC)C3)=O)C(O)C2)=O)cn2c(n1)CC(C)CC2 S(=O)(=O)(c1ccccc1F)NC(NC(C#C)CC1CCCO1)=NCCOC(C)C C1(CCCCCNC(C(C)OC2COC2)=O)CCN(C(c2nonc2N)=O)CC1 C12CN(CCO1)C(=O)C2.N1(CC(N2CC(N(C)C)C2)=O)CCCC1CO Cc1c(C(=O)NCC2(NC(=O)C=C(Cl)Cl)CCOC2)cnn1-c1ccccc1F Cc1cc(C(N2CC(CNC(C3SCCC3C)=O)C2)=O)n(C(C)(C)C)n1 N1(CC(=O)NCCOC(CNC(COCCC#C)=O)(C)C)CC(=O)NC1=O C1(NC(c2c(OC)cc(C)s2)=O)CC(NC(C2CN(CC(C)C)C2)=O)C12CCC2 CON(CCC(=O)NCCC1CCCC1)C(=O)C(C)ON.N1CCCCCC1 C(N=c1[nH]c2c(c(=NCCc3c[nH]nc3CC)[nH]1)CCCCC2)C1(C=C)CCC1 c1(OC)ccc(Cl)c(CN(C)C(c2ccc(NC(c3ccccn3)=O)o2)=O)c1F C1(CC)CC(C(=O)NC23CCCC(NC(=O)C=CCO)(C2)C3)CC(=O)N1 O=C1CCC2CCN(C(=O)Cc3cccc(C4CC4)c3)C1C2 CCC(CC)CC(F)C(=O)NC1CC2(C1)CC2C(=O)NCC1CC(C)CO1 C1(CNC23CC(NC(c4c(=N)[nH]c(C5CC5)nc4)=O)(C2)C3)CCCCC12CCC2 c1(C(N(C2CN(C(C(C(C)C)SCC)=O)C2)C)=O)ccc2ccccc2c1C c1(C(=O)NCCC(=C)CNC(C2CCC(C)(COC)C2)=O)onc2c1CCCC2 c1(OCC)nc(C)ccc1C(N1CC(NC(=O)CCNS(C)(=O)=O)CC(C)C1)=O c1(NC)c(C(=O)NCCCN(C(=O)Cc2cc(O)nc(O)n2)C)cccc1N Cc1cc(C(=O)NCc2ccc(CN(C(=O)C=CS(C)=O)C)cc2)c(C)nc1C c1(C(=O)NCC(=O)NCCC2CN(C(c3c(CC)noc3)=O)C2)cccc(C)c1 c1(-n2c(C(CC)C)nc(-c3ccncc3)n2)ccc(OCc2ccccc2)c(C)c1 c1(C(=O)NCCOCCCN(C(=O)CCn2cnc(=N)[nH]2)C)ns[nH]c1=O c1(C(N(CC(C)NC(C(C(C)C)SCC)=O)C)=O)nn(C)c(Br)c1C c1(C2(C(=O)NCC(CO)NC(C3(C)CCC(=O)N3)=O)CC2)cccc(F)c1F C(=O)(CC(C)(C)SCC)N(CCCCN(C(C1(CCC=C)CC1)=O)C)C CC(C)CC(CCO)NC(C1C2CCC(C2)N1C(c1c[nH]cc1C1CC1)=O)=O Cc1c(NC(C2CCN(C(C3CN(C)C3)=O)C2)=O)cccc1F N(C(=NCC(O)c1cccc(F)c1)N1CC2C(C)C2C1)C(C)C c1(Cn2c(N3C(C(C)C)CN(C)CC3)nnn2)ccc2c(c1)CCCN2 Cc1[nH]nc(C(=O)NC2CN(C(C3CCC=CCCC3)=O)CCC2F)c1[N+](=O)[O-] CCCCCCC(C(=O)N1CC(NC(=O)CCCCC(=O)OC)CC(O)C1)OC C(=O)(C1CCCn2ccnc21)NC1(C)CCN(C(CC2CCN(C)CC2)=O)CC1 C12(C(=O)NCCC3CCN(C)C3)CC(CO)(CN1C(=O)C#CC1CC1)C2 C#Cc1cccc(C(N2CCCC(C)(CNC(c3ncn(CC)n3)=O)C2)=O)c1Cl C1(NC(C(CC)c2ccccc2)=O)CCc2onc(C(=O)N(C3CC3)CC)c2C1 Cc1nc(N2CC3C(NC(=O)C(C)Cc4ccccc4)C3C2)c2cnn(C)c2n1 Cc1cncc(C(=O)NCc2ccc(C(=O)NC3C(C)CCC3C)nc2)c1 C1(NC(C(C2CCCC2)OC)=O)CN(C(=O)C(C)O)C2CCCC12 C1(C(=O)NCC(C(C)(C)O)F)C2CC(O)C(C2)N1C(c1cc[nH]n1)=O c1(C(=O)NCC(CN(C)C(c2cn[nH]c2)=O)(C)C)cccc2c1CCCCC2 Cc1cc(CC(N2CCCC(NC(=O)CN3CCC(C)(O)C3)C2)=O)cc(F)c1 N1(C(c2cc(CCC)[nH]n2)=O)CC(CNC(C2CC(CF)C2)=O)C(C)C1 CCC(CC(=O)N1CC(CNC(c2sc(=N)[nH]c2C)=O)CC1(C)C)C(C)C N1(C(C2CC(C)(O)C2)=O)CC2(CC(NC(=O)C=Cc3cncnc3O)CO2)C1 N1(C(C(C(C)C)OCC)=O)CCC2(CC2NC(c2cc(C#N)c[nH]2)=O)C1 CC1(C(=O)NCC2CCCN(C(=O)CCOC3CCCC3)C2)CCOCC1 Cc1cc(C(N2CCC(OC3CN(C(=O)C(C)(C)C(N)=O)C3)CC2)=O)n2nccc2n1 N1(C(c2ccc(C)s2)=O)CCC2(CCCN(C(=O)CCCCN(C)C)C2)CC1 C=CCC(F)(F)C(=O)NCC1CC(CNC(C2CCC(CC)C2)=O)C1 c1(C(=O)NC23CC(NC(c4cc5cccnc5o4)=O)(C2)C3)cnc2[nH]cncc1-2 C1(NC(c2cscn2)=O)C=CCN(C(=O)CCC(F)F)C1 C(N=c1[nH]cnc2ccccc12)C1CN(C(c2c(OC)cccc2)=O)C(C)C1 C1(NC(CSCCNC(CCCSC)=O)=O)CC2CCC1(C(=O)NC)C2 N1(C(c2c(CC)nc[nH]2)=O)CCCC12CCN(C(c1nnn3c1CCC3)=O)C2 CCCCC(=O)NCC1(C(=O)NC2COCC2CC)CC=CC1 c1(C(=O)NC2CCCC(NC(c3cc(C)no3)=O)C2)cc(O)cc(Cl)c1Cl CC(O)CC(C(=O)O)NC(c1ccc(Cl)[nH]1)=O C(C)(CN=c1nc2[nH][nH]cc-2c(O)n1)N(C(CCNC(COC)=O)=O)CC1CC1 CC1CCOCCN1C(C1(C)C=CC=C1C(F)(F)F)=O Cn1nc(C(F)(F)F)c2cc(C(=O)NC3CCOCC3NC(=O)CC#N)sc12 N1(Cc2nc(C)sc2)CCCCC1CNC(c1c(Cl)cnn1C)=O c1(C(=O)NCC(C)N(C(C(C)OC)=O)C)cccc(C2(O)COC2)c1 c1(CC(N2C(CNC(CC(C)C3CC3)=O)C=CC2)=O)nc2ccccc2s1 C(=O)(C1CCCc2scnc21)NCC1N(C(c2cccc(NC)c2)=O)C2C(C1)C2 c1(SC)ncc(C(=O)NC(C)CC(C)NC(=O)Cc2c(C)cccc2C)c(O)n1 C1(NC(c2c(C)n(CC(C)(C)O)nc2)=O)CCN(C(c2n[nH]cc2Br)=O)C1(C)C N1(C(C=Cc2c(C)n(C)nc2)=O)CCCN(C(c2ns[nH]c2=O)=O)CC1C N1(C(C2C(C)C2)=O)CCCC(NC(=O)CC2C3CC2N(C(=O)CC2CC2)C3)C1 CN(C)C(=NCC1(C(N)=O)CC1)NCC1(c2ccc(Br)cc2)CCC1 c1(O)ccc(C2CCCCC2)cc1C.C(C1CONC(=O)N1)OC c1(C(N2C(C)(CNC(C3CCCSS3)=O)CCC2)=O)cc(O)c2ccoc2c1 C1(C)(CC)CC(NC(C2(C(=O)OC)CC2)=O)CN1C(=O)Cc1cnc(C)o1 C(=O)(CC(F)(F)C(=O)OC)NCCCCCN(C(C1CC(=C)C1)=O)C n1(SCC)nc(C)c(CC(=O)NCC2CC(C)(C)CN2C(=O)C(C)C2CC2)c1C C1(C(=O)NCCN(C(C(CC)F)=O)C)CCc2cnn(CC)c2C1 CCC(CC(=O)NC1CCC(C)(CNC(=O)C(=O)C(C)C)CC1)C(C)(C)C c1(C(=O)NCC=CCNC(c2cc(=O)cc(Cl)[nH]2)=O)ccn2ccnc2n1 N1(C(C2CCC(=C)CC2)=O)CCC(CCC)(NC(c2c(C)cccc2C)=O)CC1 C1(C(=O)OC(c2ccccc2)CC)CCN(c2cnccn2)CC1 c1(C(=O)NC(CCNC(C2C(C)(CC)C2)=O)(C)C)ccc(C=CC(=O)OC)cc1 CCC(CC)(CN=c1[nH]c2c(cc1C#N)c(C)nn2C)NC(C1CC(C)CO1)=O C(CCC(C)C(=O)N1CC(CC(=O)NC2CCN(C(C)C)CC2)C2(CC2)C1)OC Cc1nc2ccc(C(=O)NC3(C)CN(C(=O)Cn4ncnn4)C3)cc2n(C)c1=O CCCCCCCCC(=O)N1CC2CCC2(CNC(c2ccccc2OC)=O)C1 C1(OC)CN(C(C2CC(SC)C2)=O)CC1NC(c1cc(SC)c(C)o1)=O Cc1nnsc1C(=O)NC1(C)CC(NC(=O)C=CCCC(C)C)C1 C1(NC(C(F)(F)F)c2ccccc2N2CCCC2)CC2CCC(C1)C2CO C1(NC(c2ccn(C)n2)=O)CC2(C1)CC2C(=O)N(CCC1CC1)CC1CC1 C(=O)(CC(CC)C(=O)NCC)NC(C(=O)NCCNC(=O)OC)CCOC C1(CNC(c2c(CC)cco2)=O)CN(C(=O)C(C)C(F)F)C2(CCOCC2)C1 Cc1cc(C(C)(C)C)ccc1CNC(=NCC1CCCO1)NCC(C)(C)CO N1(C(C2CC(CC)C2)=O)CCOCC1CN(C)C(c1sccc1C(=O)OC)=O C1(NC(c2c(C)cn(C(C)C)c2)=O)CC2CC1CN(C(=O)C(c1ccn(C)n1)C)C2 C1(C)(C(N(CCC(C)NC(c2cc(-c3ccccn3)[nH]n2)=O)C)=O)C=CCC1 Cc1cccc(C(N2CC(NC(c3nc[nH]c3C)=O)C(C)C2)=O)c1Br c1(C(=O)NC(C)(C(N2CC(F)C(F)C2)=O)C2CCC2)ccc2cc[nH]c2c1 C(c1ccc(F)cc1F)=CCN1C(C(=O)NCCc2ncco2)CCCC1 O=C(C1CS(=O)(=O)c2ccccc21)NC1C=CCN(C(C2(C3CC3)CCC2)=O)C1 N1(C(=O)NCC(c2cccc(Cl)c2)OC)CCC(S(=O)(=O)C(F)F)C1 Cc1c(Cl)c(C(N2CCC(NC(c3cc(Cl)c(Cl)n3C)=O)CC2)=O)nn1C Oc1ccc2c(n1)CCCC2N=c1ccc2nnc(C(F)(F)F)n2[nH]1 c1(OCC)cccc2c1OCC(C(=O)NC1CC1NC(=O)C(CC)C(C)C)=C2 CCC(CC)CCC(=O)NCC1CCCN1C(=O)C(c1cccc(F)c1)F c1(C(N2CC(C)CC(NC(CNC(=O)NC)=O)C2)=O)cc(C)c(O)c([N+](=O)[O-])c1 c1(C(=O)NC23CC2CN(Cc2ccc4sccc4c2)C3)ccc(F)c([N+](=O)[O-])c1 CN1CCOCC1CC(=O)NC1CC(CNC(=O)C(c2ccccc2)N(C)C)C1 CCC(CCC(=O)NCC1(O)CCCC1(C)C)NC(C1CCC(CC)CC1)=O C1(NC(c2cccc(CC=C)c2)=O)CN(C(C2CNC(=O)N2)=O)C(CC)(CC)C1 Cc1nc(C2CC2)oc1C(=O)NC(C1CN(C(c2c(Br)nnn2C)=O)C1)C Cc1ccc(C(N2CC(NC(=O)Cc3cn(C)cn3)C(O)C2)=O)c(C)n1 c1(OC)ccc(C(N2CCC(NC(=O)CSS(C)(=O)=O)C2C(C)(C)C)=O)c(F)n1 N1(CC(NOCC(C)O)=O)CCN(C(C2CCC(=O)CC2)=O)CC1 CC1CN(C(C2COCCN2C2CCCC2)=O)CCN1C(C1CC(=O)C1(C)C)=O N1(C(C2(CC(C)C)CC2)=O)CCC(C(O)CNC(=O)CC2CSCCO2)CC1 c1(C(N2CCC(C)C2)C(=O)NC(C(=O)OC)C)cn(C)nc1Br C1(NC(C(CCC)OC)=O)CCC2(CC1)CN(C(=O)C=C1CCC1)CCO2 c1(CN(C(C2N(C(C=CCN(C)CC)=O)CC2)=O)C)ccccc1C c1(CN2CC(NC(c3n(C)ncn3)=O)CC(F)(F)C2)ccc2cc(Br)ccc2c1 C1(NC(C(C)NC(N)=O)=O)CCN(C(=O)Cc2cccs2)CC1F S(=O)(=O)(c1ccccc1[N+](=O)[O-])NCC(=O)NCc1noc(-c2ccccc2F)n1 C1(CC)CN(C(=O)CCC2CCCN2C)CCN1C(=O)Cc1sccc1Cl C1(NC(C2(C)COC(=O)N2)=O)CN(C(C2CC(=C3CC3)C2)=O)C2(CCCCC2)C1 C1(NC(c2ccc(OC(C)C)nc2)=O)CCN(C(c2cnn(C)c2F)=O)CC1O C1(NC(C(C)CC#N)=O)CC(C(=O)NC(N)=O)=CC1O.C1CC(=O)N1 c1(C(=O)NC2CCC(NC(=O)C3=CCCS3)CC2)cnn2cc[nH]c(=O)c12 N1(C(C2CCS(=O)(=O)N2)=O)CC2(CCN2C(=O)CCc2cccc(F)c2)C1 N#Cc1ccc(OCc2coc(-c3ccccc3)n2)cc1C(F)(F)F CC(C)CC(CNC(=O)Cc1cc(C(F)(F)F)n[nH]1)NC(=O)CSc1nc[nH]n1 c1(SC)ncc(C(N2CC(F)CC2CNC(C2(CO)CC2)=O)=O)n1C C(CCCC(=O)NC(C)C(C)NC(c1cnn(CC(F)F)n1)=O)OCCC=C c1(C(=O)NC2CN(C(c3cnc(N)c(Cl)c3)=O)C3C2C3)ccc2c(c1)COC2 N1(C(c2cn(CCC=C)nn2)=O)CC2CN(C(c3ccsc3Cl)=O)CC2(C)C1 c1(OC)ccnc(C(=O)NCCCCN(C)C(c2cc(C3CC3)ncn2)=O)c1F C#CCC(C)(C)NC(=O)CC1C(NC(=O)Cc2ncoc2C)CC1O c1(NC(=O)N(C2CC2)CC2CCC2)cc(I)cc(Br)c1Cl CC1Cc2ccccc2N(C(c2cc(F)c(N)c(F)c2)=O)C1C C1(CCNC(=O)Cc2cc[nH]n2)CCN(C(=O)Cc2ccc(F)cc2)CC1 c1(CNc2cccc(C(=O)NC(C(C)C)CO)c2)sc2ccccc2c1Cl N(C1CCCc2occc21)C(C(CCSC)NC(C1CCN(C)CC1)=O)=O N1(C(CC2(N(C)C)CC2)=O)CC(NC(=O)CC2(C(=O)OCC)COC2)CC(O)C1 N1(C(c2cc(C)oc2)=O)CCCC(N(C)C(c2cc(C3(C)CC3)n[nH]2)=O)C1 c1(CNC(Cc2nc(NC(c3c(C)ncs3)=O)sc2)=O)ccc(Br)cc1Cl C(CC(C)C(=O)NCCN(CCOC)C(C1(c2ccc(F)cc2)CCC1)=O)=CC N1(C(C(CC=CC)NC(C2CCC(C)(C)OC2)=O)=O)CC2COCC2(C)C1 O=S(=O)(c1ccc(Br)cc1NC1(C2CCCO2)CCC1)NCC1(n2cccn2)CC1 C1(CC)CN(C(C2COCCC2(F)F)=O)CCN1C(c1cnccc1Cl)=O C12(NC(c3c(C)n[nH]c3C)=O)CCC(NC(c3c(O)cccc3O)=O)(CC1)C2 Cc1nc(C)c(-c2nc(CCN(C)C)nn2CCC(C)C)nc1C N1(C(CC2CN(C(C3(F)C(C)(C)C3(C)C)=O)CC23CC3)=O)CC2(CCNC2=O)C1 Cc1oc(C)c(C(=O)NCC2CC(C)CN(C(c3cc(F)n(C)n3)=O)C2)c1C c1(OC)nc(N(C2CCNCC2O)C(c2nccc(Cl)c2I)=O)ncc1F c1(OC)ccc(-n2nnnc2C(c2nc(C)n(C)n2)NC(C)CCCF)c(F)c1 C1(NC(=O)CCCCCC2CC2)CC2CN(C(=O)C3=CCS(=O)(=O)C3)CC2C1 c1(CNC(C2(CCCC)CC2)=O)ncc(N(C)C(c2ncn(C3CC3)n2)=O)cn1 CC1C(=O)NCCCN1.C1CCCN1C.c1(CC)ccsc1.C(=O)C N1(CCCCC2(C)OCCO2)CC(C2=NOCC2)C1 c1(C(N(C)CC2N(C(C(CC=C)C)=O)CCOC2)=O)ccc(F)c(F)c1F C1(O)(C(C)NC(c2c(CCC)[nH]cc2)=O)CCN(C(=O)C(C)SC(F)(F)F)C1 N1(C(COCCOCC#C)=O)CCC2CC12C(=O)NC(CSC)CO c1(C(CC(=O)N(C)CC2(NC(C3C(OC)C3)=O)CC2)C)cccc(F)c1 N1(C(C(=O)NCC)=O)CCCC1(CNC(=O)C1=CCOC1)COC C1(CNc2c(C(=O)OCC)scc2)CCC(NC(c2ncccc2C)=O)CC1 c1(OC)cc(Cl)c(C(N2CCC(c3cn(CCO)nn3)(N(C)C)C2)=O)cc1Cl c1(C(=O)NC2CN(C(c3c(C)nn(C)c3)=O)C2)ccc2cccc(C)c2n1 c1(C(N(CCCCN(C(c2nc(CC)sc2)=O)C)C)=O)cc2n(n1)CCCC2=O C1(OCC)(OC)CC(C(c2nnnn2CC(F)F)NCc2csnc2C)C1 CCCC(CNC(C1CCCCC1OCC(F)(F)F)=O)C(=O)O C1(N(C)C(C2CC(C)(C)CN2C)=O)CCC2CN(C(=O)Cc3cnoc3)CC12 C#CC1(NC(=O)CCC2(C)CCCN2C(C2CS(=O)(=O)C2)=O)CC2CCCC12 C1(O)(C(C)NC(=O)CCc2ccc[nH]2)CCN(C(c2c(N)cccc2Cl)=O)CC1 N1(C(C(C)Sc2ccncc2)=O)CC2(C1)CN(c1cc(O)ncn1)C2 c1(C(=O)NC2(CF)CCN(C(CC(CC)C)=O)C2)ccc(F)c2ccsc12 OC1CC2CC1CC2CN(c1cccc(C(F)(F)F)c1)C1CC2CNC1C2 C1(CCOC)(NC(=O)COCCCC(C)C)CCN(C(=O)C(O)CN(C)C)C1 c1(C(N2CC(NC(C3CC(C)(CC)C3)=O)C2)=O)cncc(-n2cnnn2)c1 c1(SCCC(=O)N(c2c(C)nn(C)c2C)C2CCOCC2)ccc2c(c1)CCCO2 c1(C(N(C)C(c2cncc(OC(F)(F)F)c2)=O)=O)cc(C#N)cs1 C1(NC(=O)CCCc2cc[nH]n2)CCCC(n2cc(Cl)cn2)C1 N(C(=NCCc1cccs1)NCC1CN(S(C)(=O)=O)C1)C(c1cnccn1)C CCCC(C(=O)NCCC1CCOCC1)NC(c1ccc(F)cn1)=O c1(OC)ccccc1OCC(=O)NC1CCCC1CNC(=O)C1=COCC1 N1(C(CN(CCOC)C)=O)CCCC1C1CCCN1C(c1csc(CO)n1)=O N1(C(c2cccc(C(C)=O)c2)=O)CCN(C(=O)C(n2nccc2C)C)CC12CC2 c1(C(=O)NC(C)CNC(=O)CC2CCNC2=O)cn(C)nc1-c1ccco1 C(C1CN(C(c2sccc2Cl)=O)Cc2ccccc21)NC(c1[nH]n(C)c(=O)n1)=O c1(C(=O)NCCCN(C)C(c2ccc(C3CC3)c(Cl)c2)=O)cc2cccnc2[nH]1 c1(NC(C2C3CN(C(=O)C=Cc4cnccn4)CC23)=O)ccc(F)c(F)c1F N1(C(c2ncc(-c3c(OCC)c(O)ccc3)cn2)=O)CC(O)C(O)C(O)C1CO C1(NC(c2c(C)ncn2O)=O)CC12CCN(C(=O)COCc1cccc(Cl)c1)C2 C(=O)(C(O)CC(C)(C)C)N1C(C(C)C)CCC1C(=O)NCCC1COCC1O C1(C(=O)NCC(C(C)C)NC(C2CCCCS2)=O)CCCC(C)CC1 c1(OC)nc(N(c2cnn(C)c2)CC2CC2)ncc1F NS(=O)(=O)c1ccsc1C(N1CCCCC(NC(=O)CC2CCOC2)C1)=O C1(NC(Cc2ccc(OC)nc2)=O)CC2CC1CN(C(=O)C=C(C)Cl)C2 c1(C(N2CC(C(C)NC(=O)C=Cc3cccc(O)c3)C2)=O)cc2n(n1)CCCC2O CCC(C(N)=O)NC(C1CCN1C(c1cnn[nH]1)=O)=O C1(C(=O)NC2CC(OC)CN(C(C=CCC)=O)C2)CCn2c(C)nnc2C1 CC(C)C#CC(=O)N1CC2C(NC(c3nocc3C(C)(C)C)=O)C2C1 c1(C(C)C)ccc(C(=O)N(C)CCOCCNC(=O)CCc2ccoc2)nc1 c1(-c2scc(C(N3CCCC3c3nc(O)n[nH]3)=O)n2)ccc(O)cc1F C12(C(=O)NCC3N(C(C4CCOC(=O)N4)=O)CC3)C3CC(CC13)C2(F)F c1(C(=O)NC2CC(C)N(C(c3cccs3)=O)C2)ccc2nnn(C)c2n1 c1(C(N(CC(CC)NC(=O)CCC2CC2(C)C)C)=O)cc(Cl)c(F)cc1F C(=O)(C1=CCC2CCC1N2C(=O)CCOCC(C)C)NCC(CC=C)(C)CO C1(CC)(CC)CC(NC(=O)CCC2CC2(F)F)CN1C(c1ccon1)=O C1(C(=O)OC)CCN(C(C2C(CNC(c3cc(CO)on3)=O)C2(C)C)=O)C1C FC1(F)CCC(N=c2[nH]c(=NCc3cc(Br)ccn3)c3sccc3[nH]2)C1 c1(C(N2CCCN(C(C3C(COC)C3)=O)C(C)C2)=O)cc2nc(C)cc(C)n2n1 c1(C(N(C2CN(C(C(C)O)=O)CC23CC3)C)=O)ccc2c(c1)NC(=O)CS2 Cc1ccc(O)cc1C(=O)NCCC1CCN(C(=O)CCC2CC(C)C2)C1 CCCC(C)CCCC(=O)NCC12CC1CN(C(c1cc(Cl)cn1CC)=O)C2 C(=O)(C(F)(F)C(F)F)N(C1C2CN(C(=O)CSC3CCCCO3)CC12)C c1(C(=O)NCC(CNC(=O)CC2CC2)F)ocnc1-c1ccccc1 CCCCCCC(C)C(=O)NCCC(C)N(C(=O)C=Cc1cncc(OC)c1)C C12(C(=O)C3CC3)CC1CCN2C(=O)CC1CC(OCC)C1.C(=O)(C(C1CC1)N)NCC C1(CC#C)(C(N2CC(F)(CC)C2)=O)CCN(C(c2cnn(CC)c2)=O)C1 c1(C(=O)NCCC(C)N(CCC)C)c[nH]nc1CNC(=O)C(O)C1CCCC1 CON(CCCO)C(=O)C12CCC1CN(C(c1cc(C)c[nH]1)=O)C2 N1(C(c2cc(C)nnc2C)=O)CC2(C=C(C(=O)N3CCC(C)(O)C3)CO2)C1 N1(C(CCCC#C)=O)CC(NC(c2sccc2F)=O)C2CCCCC12 n1(CC=C)ccnc1C(=O)NCC1C=CCN1C(c1cnc(C2CCCO2)s1)=O N1(C(c2n(C)c(=O)ccc2)=O)CCC=C(C(=O)Nc2cc(C(C)(C)C)no2)C1 C(=O)(C(C)CCCC(C)C)N1C(C(=O)NC(CC(C)C)C)CC2(CC2)C1 n1(CC(N2CCCCC2CCC2CCCC2)=O)nc2ccccn2c1=O Cc1ccc(C#N)cc1NC(C1CCCC(NC(C2(O)CCC2)=O)CC1)=O N1(C(C2CC(OC)C2)=O)CC2(CNC(=O)C(C(C)(C)C)SC)CC(F)(C1)C2 CC1(C)CCCC(C(N2CC3CC2C3NC(=O)Cc2ccns2)=O)CC1 C1(CC)CCCN(C(=O)CC(C)C(F)F)C1C(N1CC(C)(C(C)O)C1)=O N1(C(c2cc(C)sc2)=O)CC(C)CN(C(c2n[nH]c(O)n2)=O)CC1C c1(OC)ccc(CC(=O)NCC(O)CNC(c2sccc2C2CC2)=O)cc1 C1(CNC(C(C)NC(CC)=O)=O)CN(c2nc(CC)cc(CC)n2)CCCO1 C(N=c1[nH]c2c(c(=NC3CCC3C3CCCC3)[nH]1)CCC2)C1CS(=O)(=O)NC1 c1(OC)ncc(F)c(=NC(=O)c2cc(C)c(-c3ccc(N(C)C)nc3)cn2)[nH]1 CCC(C)(CCNC(C1CCOC(C)C1)=O)NC(c1cn(CCO)nn1)=O N1(c2n(CC(c3c(OC)ccc(OC)c3)O)nnn2)CC=CCC2(CCCC2)C1 CCCCC(F)C(=O)N1CC(C(C)NC(=O)CC2CNC(=O)O2)C1 c1(C(=O)OC)oc(SC2(C(=O)NCc3ccco3)CC2CO)nc1C C1(NC(=O)CC2(NC(C3CCCCO3)=O)CC2)CCCC(F)C1 C(CC(C(=O)NCC1(F)CC(NC(c2cncn2C)=O)C1)NC(N)=O)SC C(N=c1cc(C(C)=O)nc[nH]1)C1N(C(C2(C=C)CCOCC2)=O)CCC1 C1(O)(CNC(C2C(OCC)C2)=O)CCN(C(c2nc(C)ccc2Br)=O)CC1 N1(C(C(C)NC(c2ccoc2)=O)=O)CC(NC(C2CC2(Cl)Cl)=O)C(C)C1 Cc1coc(C=CC(=O)NCC(CNC(C2(c3cc[nH]n3)CCC2)=O)CO)n1 N1(C(c2c(CC)cncc2)=O)CC2(C=C(C(=O)N3CCC(CC)C3)CO2)C1 C1(NC(c2nccc(C)c2)=O)C2CC1CN(C(C1CCS(=O)(=O)N1)=O)C2 CC1(C)CN(C(=O)CN2CCC(O)CC2)CC1NC(c1cc2ccsc2[nH]1)=O N1(C(=O)NC)CCC(C)(C(=O)OC(=O)NCCOC(C)(C)C)CC1 C=CC1(CC(=O)NC(c2ncco2)(C)C)CN(C(=O)C(F)CC2CC2)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(C)(C)NC(C(CC)n1cccn1)=O Cc1cc(N2CCC(F)(CF)C2)nc(=NCC2CCC(C(F)(F)F)O2)[nH]1 c1(CC(=O)NC2CCN(C(C(c3cnn(C)c3)OC)=O)C2)ccc(C#N)nc1 CCC(C)(CCC(C)C)C(=O)NCC1CCCCCN1C(=O)C1=C(C)CCCC1 C1(CNC(C(C)CC2CCCC2)=O)C(C)CCCN1C(=O)CCCOC(C)(C)C c1(N2CCC(CC=C)(NC(c3cc(CC(C)C)[nH]n3)=O)C2)ncc2ccsc2n1 C(=O)(C(CC(C)C)ONC(c1oc(C)nc1C)=O)NC1C(CCOC)C1 c1(OC)ccc(C(=O)NC2CCCC2NC(=O)C(c2ccc(Cl)cc2)C)cc1N C12C3CC(O)C1N(C3)C2=O.c1(NC(C(C)C)=O)ccc(CC2(O)CCC2)cc1 c1(C(C)=O)cc(C(N2CCC(O)(C(C)NC(C3CCOC3C)=O)C2)=O)ccc1C c1(NC(=O)OC)ccc(C(N2CC(NC(C3CC(O)C(F)C3)=O)C(C)C2)=O)cc1 C1(C2(O)CN(C(c3cnc(N(C)C)o3)=O)C2)(CNC(C(C(C)C)SC)=O)CC1 C(=O)(CC(C(F)F)n1cccn1)NC(CNC(c1n(C(C)C)ccn1)=O)C C1(C(=O)NC2CN(C(c3c(OC)cnnc3)=O)CC2SC)COCCC1(F)F N1(C(CCN(C)C)=O)CC2(CCC(NC(c3nc4ccccc4[nH]3)=O)C2)C1 c1(C(=O)NC(CC)C(=O)NO)cc(C(=O)NC)cc(Br)c1 CC1CN2CCN1C(C(=O)NC(CNC(=O)Cc1ccccc1CO)C1CC1)C2 C(=O)(C(F)CCC(C)(C)C)N1CC2C(C(N(C3CCC4CC34)C)=O)C2C1 C1(CNC(=O)Cc2cscn2)CCN(C(c2cc3cccnn3c2)=O)CC1(F)F c1(C(C)=O)cc(C(=O)NC2CC(CCNC(=O)Cc3csc(C)c3)C2)oc1C c1(C(=O)NCC(COC)NC(=O)Cc2ccnc(F)c2F)ccc2cccnn12 CCC(C(=O)NC(C(N1CC2(C1)CN(C(C)=O)C2)=O)c1ccco1)C(F)(F)F N1(C2C(NC(C(C)NC(N)=O)=O)C2)CCCCC1 C1(OC)CC(NC(C2(N(C)C)CC2)=O)CN(C(=O)C=Cc2ccc(C)s2)C1 C1(C(=O)OC(C)(C)C)CCCN(C(=O)CCCNC(=O)C2CC2)CC1 CCCC(CCC)C(=O)N1C(C(=O)NCCc2nc(C)no2)CC1C C12(C(=O)NC(C)C(C)(C)NC(c3cc(Cl)cc(F)c3F)=O)CC(C)(C1)OC2(C)C N1(C(C=NOC)=O)CC2CCCC2(CNC(C2C3CCCC23)=O)C1 c1(C(=O)NCCC(C)(C)NC(=O)OC(C)(C)C)c(F)ccc(Cl)c1F C1(NC(CCc2ncc(C)[nH]2)=O)CCN(C(=O)COc2ccccc2O)CC1C CC1CN(C(C2CCN(C(=O)NC(C)C)CC2)C(=O)NC2(C)CC2)CC(C)O1 c1(C(=O)NC(CNC(C2(COC)CCC2)=O)C)ccc(N)c(F)c1 C1(OC)C(NC(=O)CN(C(=O)C=CC2CCCC2)C(C)C)CC12CCC2 S(=O)(=O)(c1ccc(=NCCN2CCOCC2)[nH]c1)NC(C1(C)OCCCO1)C C1(C(=O)NCC(=O)NC2CC2)(NC(C2(C)C(C)C2)=O)CC(O)C1 C(=O)(C(O)CC(C)(C)C)NCC1(C(N(C2CCN(CC)C2)C)=O)CC1 N1(CC(F)Cc2ccccc2)CCCC(C(F)(F)CO)C1 C1(C)(CNC(C=CC(=O)N(C)C)=O)CCN(C(=O)C(c2cccnc2)N(C)C)C1 C1(N(C(CC(=C)I)=O)C)CC2CC1N(C(c1ccncc1)=O)C2 C1(C)(CNC(C(=O)NCC)=O)CCC(NC(c2cc(-c3ccns3)on2)=O)C1 C1(C(=O)NCc2onc(C)n2)CC1C1CN(C(=O)Cn2cccc2)C1 C1(CNC(c2c(C#C)c[nH]n2)=O)C2CCCC1N(C(=O)Cc1c(Cl)cnn1C)C2 c1(CC)cccc(NC(C2CC(O)CN2C(c2ccc(OC)nc2)=O)=O)c1F c1(N2CC(CC(=O)Nc3cc(C#C)c(C)cc3)C2)ncnc2sc(CC)cc12 Cn1ncc([N+](=O)[O-])c1COC(C1CCCN(S(=O)(=O)C(F)(F)F)C1)=O CCCC(C)C(=O)NCCC(O)CNC(=O)CCCN(C)C C1(C)(CNC(=NCC2CC(OC)C2)NC2CCCCC2C)CCS(=O)(=O)CC1 c1(CNC(c2cncc(O)c2)=O)ccc(CNC(C2CC3(CC3)C2)=O)cc1 CCCCC(C)CCC(=O)N1CC(C(C)NC(c2cn(C)nc2C2CCC2)=O)C1 C1(NC(C(C)C)=O)COC2(C1)CN(C(=O)CCC1(C)CCC(=O)N1)C2 O=C(C1=CCOCC1)NC1(C(=O)NCC(O)CC2CCCC2)CCCCC1 N1(C(CCSC)=O)CC(OC)C(NC(c2ccc(CN3CCOCC3)cc2)=O)C1 C1(C(=O)NC2CC(NC(c3cn(C)nc3Br)=O)C2)CC2(C1)CC2(F)F N1(C(C(C)OC)=O)CCOC2(CCC(NC(=O)Cn3ncc(Br)n3)CC2)C1 c1(CC)cscc1C(=O)NCC=CCC(=O)N1CCC1CO C1(CNC(c2cc3ccoc3cn2)=O)CC2COCC2N1C(C1(O)CCC1)=O N1(C(c2c(C)ncs2)=O)CC(NC(c2cnn(C3CCC3)c2)=O)CC1C C(=O)(CCC(F)(F)F)N1CC(=O)N1.C=CCOCCOC N1(C(C2CCCC(C)C2)=O)CCC(CNC(=O)CNC=O)C1(C)C C1(NC(C=Cc2ccc(C)o2)=O)CC2CC1CN(C(c1cc(C(C)C)no1)=O)C2 c1(C(N2CC(C)(C(=O)NCC3CNC(=O)CO3)C2)=O)cccnc1C#N N1(CCNC(c2cc(Cl)cnn2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC1 c1(C(=O)OCC)c[nH]cc1C(=O)N(C)CCNC(C1(c2ccc(C)s2)CC1)=O C(CCCNC(=O)CC#N)(c1ccccc1)NC(COC1(C)CCC1)=O N1(C(C=C(COC)C)=O)CCCC(CC)C1C(N1CCCNC(=O)C1)=O C(=O)(C1CCCc2c[nH]nc21)N1CC(NC(c2c(C)cc(=O)n(C)c2)=O)(CO)C1 C(=O)(CCc1cccs1)NC1(CCNC(COCCN(C)C)=O)CC1 C1(NC(=O)CCCN2CCCC2)CCC(F)(CNC(C2(F)CCCC2)=O)C1.C1CC1 Cc1ccccc1C=CC(=O)NCC12CC(CO1)N(C(=O)C(C)OCC1CC1)C2 C1(C(N2C(C)(CC)CC2)=O)CCC(=O)N(Cc2ccccc2)C1 C(CC(O)CC(=O)NCC1COCCN(C(c2cncc(Cl)c2C)=O)C1)SC c1(C(=O)NC2(CNC(C=CC3C(C)C3(Cl)Cl)=O)CC2)cccc([N+](=O)[O-])c1 c1(NC(CNC(C2(C)CCC(=O)N2)=O)C2CCC2)ncnn2c(Br)ccc12 C1(C(N(C)CC2CCN(C(c3occc3F)=O)C2)=O)CC(C2CC2)=NO1 c1(C(N2CCCC(OCC(C)C)C2)C(=O)NC2(C)CC2)ccc2ccccc2c1 c1(CNC(c2ccc(OCOC)cc2)=O)cc2cc(C)ccc2[nH]1 N1(C(C(Cc2ccco2)NC(COCCCN(C)C)=O)=O)CCC(C(=O)NC)C1 n1(CC#C)cccc1C(=O)NCCN(C(=O)C(F)C1CCC1)C(C)C CCC(CNC(c1cc(C)c(CC)o1)=O)(CC)C(=O)NCC1CCN1C(C)(C)C C1(SC)CN(C(C2CCC(=O)NC2)=O)CC1NC(=O)Cn1cc(CC2CC2)nn1 Cc1cc(Cl)ccc1OCC(=O)NC1CCCC1CNC(c1cnoc1C)=O c1(NC2CCCCN(C(c3c(C(C)C)ncnc3)=O)C2)ncc([N+](=O)[O-])cc1F C(=O)(C(C)CC(C)C(C)=O)NC1C(C(=O)NC2C(CC)C2)CC=CC1 C1(c2cn(CC(CC)C)nn2)CN(C(=O)CNC(=O)Nc2ccsc2Cl)CCO1 S(=O)(=O)(c1cc(NCC(c2cccs2)=O)ccc1C)NC C(C(C)C(F)C(=O)NC(C)CN1CCCC1)NC(c1cncc(OC)c1)=O c1(NCCNC(C2(SC)CC2)=O)cc(Cl)nc(C2CC2)n1 Cc1cc(CCN2CC(c3cncn3C)C2)ccc1Br N1(C(c2cnc(C(C)C)nc2)=O)CCN(C(=O)C(C)N(C)C)CC1C1CCCC1 C1(CNC(c2cccc(OC)n2)=O)CC2(C1)CN(C(C1CCOC1C)=O)C2 c1(CC(=O)NCC(C(C)(C)C)NC(C(CCC)C#N)=O)cncc2ccccc12 C(c1ccc(F)cc1)=C(C(=O)NC(C(C(C)C)NC(c1ccn(CC)n1)=O)C)C c1(C(N2C(CNC(C(C(C)C)F)=O)CCCC2)=O)cc2oc(Cl)cc2[nH]1 N1(CC)CCOC(CO)C1c1ccccc1.C1(C(C)C)CCNC(=O)N1 O=C(C1=CCCCCC1)NCCN(C1CCCC1)C(c1cnc(Cl)s1)=O CC1CN(C(=O)CC2CC2(C)C)CC1NC(=O)CC1CSCCS1 CC(C)CC(O)C(C)C(=O)NCC(C)C(=O)NCC(C)C(C)C CC(C)CC(C)(O)CNC(CCn1cccn1)C(=O)O n1(CC)nc(C(=O)NC2CN(C(c3cnnn3CC)=O)C2)c(=O)c2ccccc12 C(=O)(CS(=O)(=O)CC)N1CC(CC=C)(C(=O)NC(COC)C(C)C)C1 N1(C(c2c(COC)n(C)nc2)=O)CCCN(C(=O)CCCc2ccsc2)CC1 c1(N(C)CC2CCC(SC)C2)ccc(S(=O)(=O)NCCF)c(Cl)c1 N1(C(C(C)(C)C2CCCO2)=O)CC2OCCN(C(=O)Cc3ccoc3)C2C1 c1(CCC(N2C(CN(C)C(c3nncn3C(C)C)=O)CCC2)=O)ccccc1C#N Cc1ncc(NC(C2CCCN(C(C34CCCC3C4(C)C)=O)C2)=O)c(C)n1 CC(C)C(CCc1ccccc1)C(=O)NCCN(C)C(c1ccc(N)c(O)c1)=O N1(C(C2CN(C)C2)=O)CCN(C(=O)C(C)(C)F)CC1Cc1cncs1 CC(CNC(=O)CC1C=CCC1)(CO)NC(=O)CC(C1CCC1)C1CCC1 CC1(C)OC2(CCCN(C(=O)NC3Cc4ccc(NC(N)=O)cc4C3)C2)NC1=O N1(C(CSCC)=O)CCCC(N(C(=O)Cc2cc(C(F)(F)F)n[nH]2)CCF)C1 C=CC1(C(=O)N(C)CCc2cnc[nH]2)CCN(C(=O)COCCSCC)C1 c1(CC(=O)NC(CN(C(C(C2CC2)OCC)=O)CC)C)cc(C(F)(F)F)n(C)n1 CC1CN(C(c2csc(-c3ncccn3)n2)C(=O)NC)CC(C)(F)O1 c1(C(N2CCC(NC(C3(CC#C)CCCO3)=O)C2)=O)csc2cc(C)ccc12 C1(F)(C(N2CC3C(NC(C(C)C4CC4)=O)C(C3)C2)=O)CS(=O)(=O)CC12COC2 C12(CNC(C(CC)CC)=O)CCCC1N(C(=O)COCCCF)CCC2 c1(CN(C)C)ccc(C(=O)NC2CCC(C)(CNC(=O)CC(C)(C)C)C2)cc1 c1(OC)c[nH]c(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCCC2)cc1=O C1(OC)CCCC12CCCN(C(=O)N=c1cnn(-c3cccc(Br)c3)[nH]1)C2 C1(CC)CC(C(N2CC(=C(F)CNC(=O)CC3COC(C)(C)C3)C2)=O)CCC1=O O(C=C(C#N)C(=O)N1CCCC1CCNC(c1cc(C(C)C)on1)=O)CC CCCCCCN(CCNC(C1CCOC1CC)=O)C(C12CC(F)(C1)C2)=O N1(C(c2nc(C)sc2)=O)CCC(O)C1C(N1CCC(C(N)=O)C1)=O N1(C(c2n(CC)nnc2)=O)CC2CCC(C1)N2C(c1cc(C)c(F)cc1Cl)=O C1(NC(c2cc3ccccc3s2)=O)CN(C(C2(F)CCOC2)=O)CC2(CCC2)C1 C1(CN(C(C(C)=C(C)C)=O)C)CCCN1C(c1cc(Cl)no1)=O c1(-c2nnc(C)o2)cccc(COC(C2CC(=O)N(c3ccccc3F)C2)=O)c1 C12(NC(C=CSC)=O)CCN(C(c3cnc(C4CC4)nc3)=O)CC1C2 C1(N(C(=O)C=Cc2ncc(C)[nH]2)CC)CCCN(C(C2CC3CC3C2)=O)C1 CN1CCC(C(=O)NCc2csc(CNC(=O)Cc3cccnc3)c2)CC1 C12(C(=O)NC)C(NC(C3CC3C(C)C)=O)C3CC1C2C3.Cc1cc(CO)oc1C Cc1ccc(O)c(CC(N2CCCC2(C)CNC(=O)COc2cc(C)on2)=O)c1 n1(CC(=O)NCC(CCOC)NC(=O)CC(C)C)nc(-c2cccs2)oc1=O N#Cc1cccc(Br)c1C(=O)NC1CCC(NC(c2cc(F)c(F)cc2Br)=O)C1 C(=O)(CCCCCSC)NCC(C(=O)OC)Oc1ccc(COC)cc1 CC(C(C)(C)C)=CC(N1CC(F)(CNC(=O)CCCNC(c2ccco2)=O)C1)=O Cc1c(-c2ccccc2F)o[nH]c1=NC(=O)NCC1CCNC(=O)C1 c1(NC(c2ccc[n+]([O-])c2)=O)c(F)cc(I)cc1[N+](=O)[O-] CCC(CC(C)C)C(=O)NCCC(C(C)C)NC(C1CNC(=O)CC1(C)C)=O n1(C(C)C)cccc1C(=O)NC1CCC1NC(=O)C(C)OC1CCCCC1 C(C)(C)(C(C)NC(c1ccnn1CC1CCC1)=O)NC(CN(CCC)C)=O c1(NC(c2ncc(C)s2)=O)nc(C)c(NC(c2cccs2)=O)s1 CC1CCc2nc(N3CCC(=C(F)F)CC3)[nH]c(=NC3CCOCC3)c2C1 c1(C(C(=O)NCCC#C)NC(=O)C(C)NC(N)=O)cnn(C)c1 C1(NC(C2C(=C)C2)=O)C2CC3C(C2)C13C(N1CC(C)(C(F)(F)F)C1)=O Cn1cc(-n2cncc2C(=O)NCC(F)CNC(c2csc(C(N)=O)n2)=O)cn1 c1(OC)ncc(F)cc1CNC1CC(C)CN(C(c2cc(F)ccc2I)=O)C1 C1(NC(=O)C=Cc2cscn2)COC2(CCN(C(c3ccccc3CO)=O)C2)C1 C=C(C)CCC(c1nnnn1CCOCC)NCC1CCN(CC(C)(C)C)CC1 c1(C(=O)N(CCC2(C(=O)NCCC3CC=CC3)CCC2)C2CC2)cc(O)cc(=O)o1 c1(C(=O)NC(CNC(C(C)=C(CC)C)=O)(C)C)cncc2c[nH]nc12 C#CCCC(O)C(=O)N1CCN(C(C2SCCS2)=O)C(C)C1 CC1(C(N2CC3CCC3(CNC(C34CCC(F)(CC3)C4)=O)C2)=O)CCC12CCC2 c1(CNC(=O)CCC2CCCOC2)cnn(CCNC(=O)CCc2cnco2)c1 N1(C(c2c(C(C)NC(C3CC3c3ccco3)=O)nn[nH]2)=O)CCCCC(C)C1 C1(CNC(c2cnc(C)s2)=O)CC12CCN(C(=O)CCn1cc(Cl)cn1)CC2 c1(C(=O)NCC2(OC)CN(C(C3C(CCC)C3)=O)C2)ccc(-n2cnnn2)cn1 c1(OCC(=O)NC2CCCCC2NC(=O)CCC2CCC2)cc(F)cc(Cl)c1 C12(CC)CN(C(c3sccc3Cl)=O)C(CNC(c3cc(Cl)cs3)=O)(C1)C2 c1(NC(=O)C(=O)NC2COC3(CCCC3)C2)ccc2sccc2c1 C(=O)(CC1=CCCCC1)NC(C(C)NC(c1ncc(CC)cn1)=O)C(C)C C(=O)(CCCC(=O)N(C1CCCCN(C(c2cc(C)oc2C)=O)C1)C)OCC Cc1nc(C(=O)NC2(C)CCN(C(=O)CN3CCCC3)C2)ccc1C#N N1(C(=O)CCOC2CC2)CCC2CN(C(c3cnn4ncccc34)=O)CC2C1 C(=O)(CC(C)(C)CC(C)=O)NC(CNC(CCCCCOC)=O)CC(F)(F)F N1(C(C(C#C)(C)C)=O)CCN(C)C(C(=O)NCc2ccccc2C)C1 CC1(C(=O)NCC2(C)CCCN2C(=O)CCC[N+](=O)[O-])CCc2ccccc21 CCCC(C)(CC)NC(c1cn(C)nc1Cl)c1nnnn1CC(F)F C1(C(=O)ON2CCC(Cc3nccs3)C2)CCN(C(N2CCCC2)=O)C1 c1(C(N2CC3CN(c4ncccn4)CC3C2)=O)ccc(F)c(F)c1Cl N1(C(C(CNC(C)=O)(C)C)=O)CCC2(CCCC2CNC(C2CC23CC3)=O)CC1 C(C(C(=O)NCC(N1CCCCC1)C)C(C)(C)C)NC(C(c1ccc(C)o1)C)=O N1(S(CCC)(=O)=O)CCCC(C(=O)N(CCNC(c2conc2C)=O)C(C)C)C1 CC(C)C(C)(CNC(=O)C(O)Cc1cn(C)cn1)NC(=O)CCCn1ccnn1 C1(C(=O)NCCN(CCC)CC)CCC(NC(=O)CCCC2CC2C)C1 N1(C(c2nncn2C)C(=O)NC(C(=O)OC)C)Cc2nccn2CC(CO)C1 c1(C(=O)NC(C(C)NC(c2cc(CC)nc(O)c2)=O)C)cnc2ccnn2c1C N1(C(c2c(C)ccnc2)=O)CCC2CN(C(=O)C(=O)NCC3CC3)C2C1 N1(C(c2ccc(CCC)cc2)C(=O)NC2CCCC2)CCOC2(CCCSC2)C1 CC1CN2CCN1CC2C(=O)NCC1CCN(C(=O)CCS(C)=O)C1(C)C N1(C(c2c[nH]nc2C2CCCC2)=O)CCN(c2ncnc3[nH]ccc23)CC(O)C1 c1(C(C)(O)C(=O)NC2CN(C(=O)C(O)C3CC3)C2)ccc(Cl)cc1 C(=O)(C(C)CC(C)C(C)=O)N1CCC(C(N(CCCC)CC)=O)(CO)C1 Cc1cc(C)n(C(C)CC(=O)N(CC(C)CNC(C2(O)CC2)=O)C)n1 c1(C(=O)NC2(C)CC(NC(C(C(C)C)c3cnc(C)s3)=O)C2)cc(N)cc(F)c1 C1(NC(C(C)OC)=O)C2CC3CN(C(=O)CCc4cnc(C5CC5)o4)C1C3C2 C(c1ccc(SC)s1)=CC(=O)NCC(CC)NC(C12CC(CCO1)C2)=O CC(C)C(C)CC(=O)NC1CCN(C)CC1.C12(CC3(CC3)C1)c1cn(nn1)C2C C1(C(=O)Nc2c(C#N)ccs2)Cc2c([nH]c3ccccc23)CN1C(=O)C=CCBr C1(C(=O)NC(C(C)(C)C)CNC(C2(CC#N)COC2)=O)Cc2nnsc2S1 C#CCC(CC(F)F)C(=O)NC(CNC(=O)Cn1nnnc1CC)C1CCC1 N1(C(C(C)OCCCC)=O)CC(C)(C)OCC1CNC(=O)CC(F)(F)C(F)F N1(C(c2cccnn2)=O)CCC2(CC1)CC(NCc1ncccc1F)C2 c1(C(=O)NC2CCN(C(c3c(CC)cccn3)=O)CC2)c(C)nn(CC)c1C Cc1cccc(-c2nc(C(N3CC(C#N)C3)=O)cs2)c1C N1(C(CCC2CCC(C)O2)=O)CCN(C(=O)CCC(=O)OC(C)(C)C)CC1CF N1(C(c2nc(C)nc(O)c2)=O)CC2C3CCC(C2C1)N(C(c1oncc1C)=O)C3 C(=O)(C(C)CSC)N(CC(CC)NC(c1cnn(C2CC2)c1)=O)CC.CO.O c1(C(=O)NC(C(C)C)(C)CNC(=O)CC2CCCO2)cnc2ccccn2c1=O c1(NC(C2C(C)(CNC(CCc3cn(C)nn3)=O)C2)=O)ccc2c(c1)OCC2 C1(NC(C(C2CCCC2)OCC)=O)CCCC2CN(C(C3COC(C)C3)=O)CC12 CC(C(=O)NC1CCN(C(=O)COC(F)(F)F)CC1O)C(F)(F)F C1(NC(C(CC)C(C)(F)F)=O)CN(C(C2CC(O)C2)=O)CC2CCCC12 CCC(CC)(CO)C(=O)NC1CCN(C(c2cc(OC)c(OC)cc2O)=O)CC1 c1(-c2c(C(=O)NCc3cc(C)on3)ncs2)ccccc1C C1(CC)CSC(=Nc2ccccc2)N1C(=O)C(c1ccc(OC)cc1)O CCC(C(=O)NCc1ccon1)N(C)C(C1CC(C)(F)C1)=O c1(CCC)nc(C(=O)N(CC(=O)NCCCCCC2CC2)C(C)C)co1 C12CCN(C1)C2=O.c1(NCCNC(C(=O)NC)=O)ccn(C)n1 N1(C(c2ccc(SCC(=O)O)o2)=O)C2CCCC1CC(NC(CC1CC(=O)NCC1)=O)C2 CCC(C)(C)CCCC(=O)NCC1CCC(F)(NC(=O)CC2CCCO2)C1 C1(O)(CCNC(c2cnn(C(C)C)n2)=O)CCN(C(=O)CC2(O)CCCOC2)C1 C1(NC(CCc2cc(OC)no2)=O)CCCN(C(c2ccncc2)=O)C1C C1(NC(=O)CC2CCCOC2)CCC2CN(C(c3ccnn3C3CC3)=O)CC2C1 N1(C(C=NOC)=O)CCCC2(CNC(c3cc(F)c(F)c(F)c3)=O)CCCC12 Cc1[nH]nc2c(C(=O)NC3(CNC(=O)CC(C)F)CCCC3)cccc12 c1(C(=O)NCC2CN(C(C3C(C)(C)COC3)=O)C2)ccc(O)c(F)c1 C1(CC(=O)NC(C2(NC(C3CC(O)(C#N)C3)=O)CC2)C)CCC(=O)NC1 Cc1ccc(COC(=O)CCc2csc3ccccc23)c(=O)n1C N1(C(Cc2cn(CC)nc2)=O)CC2CC(OCC)CC1C2.C1C(C)CC(=O)O1 Cc1cnc(C(N2C3CC2CN(C(=O)CC(C)C(C)C)C3)=O)cc1Cl Cc1cc(C(=O)NC2CC(C)N(C(C3(C(=O)NC(C)C)CC3)=O)C2)cc(Cl)n1 c1(C(=O)Nc2c(C)nc(Br)cc2)cn2c(n1)CN(C(=O)C=Cc1cnc[nH]1)CC2 C(=O)(CCCCC(C)C)NCC12C(CN(C(CCCCCOCC)=O)C1)C2 c1(OC)cccc(I)c1C(=O)Nc1ncc(CCNC(=O)CCC(C)C)s1 CCC(CCC(=O)NCC1(C2CCCCO2)CC1)NC(C1CC(n2cncn2)C1)=O C1(OC)CC(NC(c2ccc(C)cc2)=O)CN(C(=O)C(C(C)C)SC)C1 N1(C(C2(COC)CCOCC2)=O)CC2(C1)CN(C(C1(COC)CCOC1)=O)C2 c1(C(=O)NCC2N(C(C(CCC)C(C)C)=O)CCOC2)ccc(C=NOC)cc1 C1(C)(CC)CC(NC(=O)C(F)F)CN1C(=O)CCCCCc1ccccc1 CCCC(C)CC(=O)NCC1(O)CCN(C(=O)C(c2ccccc2)C2CC2)C1 c1(C(C)(C)CNC(=O)C(=O)Nc2ccccc2)ccc([N+](=O)[O-])cc1 C(=O)(CC(C)(C)C(=O)NC1CCCCC1NC(C1CCCCS1)=O)OCC C1(CCC(=O)Nc2cn(CCCN3CCOCC3)nn2)CCc2ccccc2C1 c1(C(N2C(C)CC(CNC(=O)Cn3cncn3)C2)=O)cc(N)cc(F)c1 CCCCCC(F)C(=O)N1CCC(NC(c2c[nH]nc2CC)=O)C1 c1(NC(N(CCO)Cc2cnn(CCOC)c2C)=O)cc2sc(C)nc2cc1Cl c1(CN(C)C(C2NC(=O)CC2c2ccccc2)=O)ccc(NC(C2CC2)=O)cc1F c1(CC(N2CCC(CCOC)(NC(C(CC#C)C)=O)C2)=O)cccc(C)c1C Cn1nc(O)cc1C(N1CCC(Cn2cc(Cn3ccnc3)nn2)CC1)=O c1(C(N2CCC(C(=O)NC3N(S(C)(=O)=O)CCC3)CC2)=O)ccc2nc[nH]c2c1 C1(NC(C(c2cccs2)SC)=O)CC(F)(F)CC1NC(c1cnccc1Cl)=O C12(CNCCS(=O)(=O)NCCOC)CCCCC1NC(=O)CC2 C1(C)(CNC(C2C(CC)C2)=O)CCCN1C(c1cc(Cl)c(Br)[nH]1)=O c1(NC(N2CCC(SC(C3CC(c4ccccc4)C3)C)C2)=O)nn(C)cc1Br n1(CC)ccc(CC(N2CCCC2)=O)n1.C1(CSC)C(=O)N2CCC2(C)C(=O)N1 C1(C(=O)NC2CC(CCC(=O)NCc3ccc(C)o3)C2)(CC)CCNC1=O N1(C(c2c(NC)cnnc2)=O)CCC(C(=O)N(C2CN(C)C2)C)CC1C c1(OC)ccc(CCC2OCC(NC(=O)NCC3(CSC)CC3)C2)c(Cl)c1 Cn1nc(C(N2CCCC2(C)CNC(C2C3CCCC23)=O)=O)c2c1CCCC2 CN(C)S(=O)(=O)N(C)CC(=O)NC(C)(C)CNC(c1cc(Cl)ccc1O)=O c1(C(=O)NC2(COC)CN(C(C3CCCCC3O)=O)C2)cnccc1C(N)=O c1(C(=O)NCC2CN(C(c3c(CC)n(C)nc3)=O)CC2C)sccc1S(C)(=O)=O C1(CNC(=O)CCC2CCC2)CC2CC2N1C(C1CC(=O)N(CC(F)(F)F)C1)=O C=C(Cl)C(C)(C)C(=O)NCC1CC2(CC2)CN1C(C1CC(C#N)C1)=O c1(NC2C(C)CN(Cc3ccc(Br)cc3Cl)C2)nc(Cl)nc2[nH]c(O)nc12 N1(C(C(SC)SC)=O)CC2CCCC(NC(C3CCS(=O)(=O)C3)=O)C2C1 C=CC(CCC)CC(=O)NCCOCCCN(C(=O)CC1CC=CC1)C c1(C(=O)NCC2N(C(C(CCCC)O)=O)CCC(C)C2)cc([N+](=O)[O-])cn1C C#CCCN=C(NCC12CCC(CC1)CC2)NC1CCN(c2cccc(C)c2)C1 C12(C(N3CC(CC)SCC3)=O)CC(C)(CN1C(=O)CCCC(C)C)C2 N1(C(c2c(SC)cccc2)=O)CCCN(S(=O)(=O)CC2CC2)CC1C Cc1conc1C(=O)NC1(CN(C(=O)C(n2ccc(Br)n2)C)C)CC1 N1(C(C2(c3ccc(OC)c(C)c3)CCC2)=O)CCC(C2CC(F)(F)C2)C1 C(=O)(C(C)(O)CC(F)F)N1CCCC(CN(C(C(CCSC)NC=O)=O)C)C1 N1(CCC)CC(C(N2CC(NC(c3nocc3C3CC3)=O)C(F)C2)=O)CC1=O N1(C(Cc2c(C)ccs2)=O)CCC(CNC(=O)C(C#N)=CC(C)C)C(O)C1 N1(C(C(CC(=C)C)C)=O)CCN(C(c2nocc2C(C)(C)C)=O)CC(O)C1 C1(CNC(CCN(S(C)(=O)=O)C)=O)CC(C)(C)CN1C(=O)C1=COCCO1 c1(NCc2ccc(C)nc2)cc(C2=CCN(c3ccccc3[N+](=O)[O-])CC2)cs1 c1(C(=O)NCCC2CCC(NC(c3scc(C)c3)=O)C2)cc(C)cc2c[nH]nc12 N1(C(CSC)=O)CCCC(N(C(=O)C(CO)OC)CC)C1 c1(N(C)Cc2cc(C)no2)ncc(N)c2ccccc12 CC1(C)CCN(C(=O)C(N2CCOCC2)C2CC2)CC1NCC=Cc1cccs1 c1(CNC(C(=O)N(CCNCC)CC)=O)c(C)cccc1C.c1(OC)cccnc1 C1(C(N(CCC(=O)OCC)C)=O)C2CCN(C(=O)C(c3cncn3C)O)CC12 N1(C(Cn2c(C)nnn2)=O)CCC(CNC(c2ncccc2OC(F)F)=O)C(C)C1 c1(CN2CC3(CN(C(C(C)(C)C)=O)C3)C2)cc(Br)cc(Cl)c1O C(C(F)C(=O)NCCC1CCCN1C(C1CCCC1)=O)N(CC)CC c1(C(=O)NCC2(F)CN(C(c3c(CC)n(C)nc3)=O)C2)c(C)oc(C)c1C C1(F)(CNC(C2(C)CC2(F)F)=O)CCCN(C(=O)C(F)=C2CCC2)CC1 N1(C(C2(C)CCOC2)=O)CCCCC(NC(=O)CC2CC=CC2)C1 C1(C(=O)NCCn2nnnc2C2(CC)CCN(CC)CC2)C2Cc3ccccc3C12 N1(C(C(CC)(C)O)=O)CCN(c2ncc(COC)cn2)C(CC)C1 C1(NC(c2cc(C)no2)=O)CN(C(c2cc(Cl)ccc2C)=O)CC2(CCC2)C1 C1(O)(CN(C(Cc2c(CC)con2)=O)C)CCN(C(c2ccc(CO)nc2)=O)C1 C(=O)(C1=CCC(NC(=O)C(C(C)C)OCC)C1)NC(C(=O)NCCC)C C(C(C)(C)C(=O)N1CCCC(OCc2cn(CCOC(C)=O)nn2)C1)N(C)C CC(C)(CCF)C(=O)NCC(O)CC(=O)NCCCC1CCOC1=O c1(NC(C2CCN(C(CN(CC)CC)=O)CC2(C)C)=O)ccc2c(c1)OCCC2 c1(OCC)sccc1C(=O)NC(c1ccccc1)CNC(c1ccc(CO)s1)=O c1(C(=O)NCCCc2cn(C(C3(S(N)(=O)=O)CC3)C)nn2)ncccc1F c1(OC)ccc(CN(c2ncnc3occc23)C2(C#N)CCNC2)cc1C#N c1(N(CC(C)C#N)C)ccc(S(=O)(=O)N2CCCC2c2cccc(Cl)c2)c(Cl)c1 c1(CN2CC(C(C)NC(c3cn(-c4ccccc4)nn3)=O)C2)cnccc1Cl c1(C(=O)NC(CNC(C(CC)CC)=O)CO)c[nH]c2nc(Br)ccc12 C(CC(O)CC(=O)N1CCC(C(C)NCC(=O)Nc2ccccc2OC)C1)SC C=C(Cl)CC(C(=O)NCCC(CC)CO)NC(C1CC2(C1)CC21CC1)=O C1(CC(=O)NCC2(CO)CN(C(C3(C(F)F)CCCO3)=O)C2)CCS(=O)(=O)CC1 CC(CCCc1ccccc1)C(=O)NCCN(CCCN(C)C)C(C1CC1C)=O CCC(C(=O)NC(C1CN(C(=O)C(C)n2cncn2)C1)C)OC1CCCCC1 c1(CN(C)CC2(Cl)CC2(F)F)ccc(C(F)(F)F)cn1.n12cc(nn1)C2 c1(C(C)C)ccc(Cl)c(C(=O)NC2CC(F)CN(C(=O)Cc3ccoc3)C2)c1 c1(COC)nc(NC(C)COCC(F)(F)F)cc(=NCC(CO)SC)[nH]1 C1(OC)(CNC(=O)CC2(C(F)(F)F)CC2)CN(C(=O)CC2CCCN2C(C)C)C1 C1(NC(C2CN(C(N)=O)C2)=O)CCOCC1NC(=O)Cc1cc[nH]c1 c1(C(=O)NCC(CN(C)C(C2C(F)(F)C23CC3)=O)O)cc(F)cc2nc[nH]c12 C1(C(=O)NC(CC2CC2)CC2CC2)C2Cc3c(Cl)cccc3C12 c1(CC2(C(=O)NCC3OCCN(C(C(N)=O)=O)C3)CC2)cccc(F)c1F c1(C(=O)NCC(C2CC2)NC(c2c(CC(C)C)onc2)=O)cccc(F)c1 C1(C(=O)NC2C=CCN(C(c3ccc(C(C)C)cn3)=O)C2)CNC(=O)C(C)(C)C1 N1(C(CCC=C)=O)CCC2CN(C(=O)CCc3nccn3C)CC12 c1(C(N2CCN(C(CC(CCC)C)=O)CC2COC)=O)c(F)ccc(Cl)c1F C(=O)(C(COC)CC(C)C)N(C(C)CCC(=O)OC(C)(C)C)C.CS c1(OC)cc(C(=O)NC2CCCC(O)C2)cc(N)c1O.N1(C2(C(=O)N)CC2)CCCC1 C1(C(N2CC(CC(CNC(C3C(C(C)C)C3)=O)(C)C)C2)=O)(N(C)C)CCCSC1 c1(C(N2CCCCC(NC(C3(n4cnnn4)CC3)=O)C2)=O)cccc(Br)c1O CN1CCc2cc(C(=O)NC3CC(NC(c4ccc(F)cc4F)=O)C3)sc2C1 N1(C(c2cccc(NC(C)=O)n2)=O)CC(F)(F)CC1C(N1CC(=O)NC(C)C1)=O N#Cc1ccccc1NC(C1(c2ccc(-c3nn[nH]n3)cc2)CCC1)=O CCC(F)(F)C(=O)N1CC(CNC(c2ccncc2C(F)F)=O)(OC)C1 C1(C(C(=O)NCCOCC)N(c2ccc(Br)cn2)C)CCCC(C)(C)C1 N1(C(CC(C(=O)OC)C)=O)CC2(CCN(C(c3cccn4nnnc34)=O)C2)C1 C1(C(=O)NCC(C)CNC(=O)C(c2ccccc2F)(F)F)Cc2nnsc2S1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1CCC2(CN(C(CCC3(C)CC3)=O)C2)O1 CC(C)(C)C(CNC(c1c[nH]c(Br)c1)=O)NC(C1(C)CC2CC2C1)=O C1(C(=O)NCC2CC(OCC)C2)CN(C(c2coc(C(N)=O)c2)=O)CC(C)(C)C1 C1(CNC(C(C(C)C)O)=O)CCC2CN(C(=O)C(C3(O)CCCC3)F)CCC2C1 C(=O)(C(C(C)CC)CCC)NC1(C)CN(C(C(=O)NCCOCCCC)=O)C1 C(N=c1cc(C)nc(-c2ccccn2)[nH]1)C1CCN(C(C(CC)C)=O)C1 C1(CC(=O)NCCCOCCNC(CN(C(=O)OCC)C)=O)C=NN(C)C1=O C1(C(N2C(CN(C(=O)Cc3ccc(N)cc3)CC)CCC2)=O)CCCC(C)(C)C1 Cc1cc(-c2nc(C3CC(O)C(F)C3)n(Cc3ccccc3F)n2)c(C)o1 Cc1ccc(CC(=O)NCC2CCN(C(c3nn(C)cc3N)=O)CC2O)c(F)c1 N1(C(C(CC)O)=O)C(C(=O)Nc2cnc(Br)cn2)CCC1C C12(CNC(CC(=O)N(C)C)=O)CC(NC(c3cc(F)c[nH]3)=O)(C1)C(C)(C)O2 C(=O)(CC(C)CC(C)C)N1C(CC(=O)NCC2(OC)CC2)CCCC1 N1(C(c2c(-c3ccc(OC)nc3C(F)(F)F)ncs2)=O)CCc2n[nH]cc2C1 CC(C)(C)C(C#N)C(=O)NC1(C(F)F)CC(NC(=O)C=Cc2cccc(Cl)c2)C1 N1(C(c2nc(OCC)sn2)=O)CCCCC1C(C)NC(c1cc(Cl)c(Cl)[nH]1)=O C1(C2(O)CCN(C(C34CCCCC3CCC4)=O)CC2)(NC(C2CC2F)=O)CC1 c1(OC)cccc(Cl)c1C(=O)NC1CC1C(=O)Nc1ccc(C)nc1F C1(N(C(=O)CCSc2ccccn2)C)CCCCN(C(C2CCC2C#N)=O)C1 c1(C(=O)NCC2C(CNC(c3cnc(CC)s3)=O)C2)c(OC)ccn2ccnc12 c1(C(N2CCN(C(C(CCC)NC(N)=O)=O)C(CC)C2)=O)c(F)cc(N)cc1F c1(-c2ccc(-c3n(CC(C(C)C)(C)O)ccn3)s2)cc(F)cc(Cl)c1 C1(NC(C=C(C)C(F)F)=O)CN(C(=O)C=CBr)C2(CCCOC2)C1 C1(CNC(C=C(C)C(F)F)=O)CCCCCN1C(=O)CC1COC(C)(C)C1 c1(OC(C)C(=O)NC2CCCC2NC(=O)C(C)CF)cccc(Cl)c1 C1(O)(CC(=O)NC(C)CN(C)C)CCN(CCCc2ncccn2)CC1 C(=O)(C(S(C)(=O)=O)C1CC1)NCC(C)(C1CC1)NC(C(C)C1(O)CCC1)=O CCC(CCC(=O)N1CCCC(F)C1)NC(C1CC2(CC2)CO1)=O C1(C)(C(N2CC(N(C)C(C3CC(F)C3)=O)C2)=O)C=CCC1 N1(C(c2c(OC)ccs2)=O)CCN(C(C2C(OCC)C2)=O)C2CCCC12 N1(C(CC)=O)CC(Nc2nc(OC)cc(OC)n2)C2(CCOCC2)C1 C1(NC(C2CCS(=O)CC2)=O)CCCN(C(C2CC(OC(F)(F)F)C2)=O)CC1 N1(C(C(C)NS(CCC)(=O)=O)=O)CCC(NC(c2cc(=O)cc[nH]2)=O)C12CC2 CC(C)C(C)(O)C(=O)N(C)CC1CCCN(C(=O)C2=CCCOC2)C1 c1(C(=O)NCC23CC(NC(CCCC(C)O)=O)(C2)C3)cnc2ccccn12 CC1(C)COCC1CNC(=O)CC1(NC(C2CC=CC(O)C2)=O)CCC1 c1(OC)cc(CC(C)NC(=O)C(=O)NC2CCN(CC(C)C)C2)ccc1O c1(C(C(=O)N(CC(CNC(c2c(CC)c[nH]c2)=O)O)C)(C)OC)ccccc1F C1(C(=O)NC(C(C)NC(C(C)C)=O)C)CC2CS(=O)(=O)CC2C1 C1(CNC(CCC(CC)OC)=O)CC12CCN(C(C1CC(N(C)C)C1)=O)CC2 c1(OC)cnc(C(=O)NCC2CCCN(C(C3CC4CCC3C4)=O)C2)nc1 c1(C(=O)NCC2C(CNC(C3CCC(C)(F)CC3)=O)C2)noc2ccc(Cl)cc12 C(CC(C(=O)N1CC2CC2(CO)C1)NC(=O)Cc1ccc(F)nc1)OC c1(CNC(C2CCN(Cc3cc(CO)[nH]n3)CC2O)=O)nc2c([nH]1)CCCC2 c1(NCC2CCC(C)S2)ncccc1S(=O)(=O)NCc1nc(C(N)=O)cs1 CC1(C)C2CCC1(C)C2C(=O)NC1CCN(C(=O)CNC(=O)C2CC2)C1 c1(CC)c(C(=O)NC2CC(C)(CNC(=O)CCC(=O)N(C)CC)C2)cccc1F c1(C(=O)NCC(C(C)C)NC(=O)CCc2cccc(F)c2F)cc(O)cc(O)n1 c1(C(=O)NC(C)CCNC(=O)Cn2cnccc2=O)c(Br)ccc(F)c1N Cc1oc2nc(Cl)ccc2c1C(=O)N(CC(O)CNC(C1OCCO1)=O)C C(=O)(CCC(C)(C)C)NC1CCCC(C)C1.c12ccc(cc1)COC2=O c1(C(N2CCC(CNC(CC3(C)CC3)=O)C2)=O)ccc(Cl)c2occc12 c1(C(=O)NCC(=O)NCC(C)NC(c2ccno2)=O)cccc(O)c1 CON(CCC(=O)NC1CCn2ccnc2C1)C(=O)C1CC2(CCO1)CC2 O=C(N=c1cc(CCO)[nH][nH]1)c1cc(F)ccc1Oc1ccc(Br)cn1.CC(F)F c1(C(N2CCC(NC(c3c(CC)nn[nH]3)=O)C2C2CC2)=O)c(C)cc(Cl)cc1N C1(CC(C)NC(c2cc(C)sc2)=O)CCN(C(=O)CC(C)O)CC1 N1(C(C2C(NC(C3(C)CC(F)C3)=O)CCO2)=O)CCNC(=O)CC1 Cc1ccc(C(=O)C(=O)NC(C)C(C)NC(=O)C(C)n2ccnn2)cc1 C1(C(N2CCN(C(C(=O)OC)=O)CC2)=O)COCCN(Cc2cccn2C)C1 c1(CC(=O)N(CCCN(C(C=C2CCN(C)C2)=O)C)C)cnccc1Cl C1(C)(CC)C=C(C(=O)NCC(=O)NCC(=O)NC(Cc2ccco2)CO)C1 CCCC(CC)CCC(=O)N1CCCCC1CNC(C1CCC(=O)NC1)=O Cc1cc(F)c(C(C)C)cc1NC(c1c[nH]c(-c2ccco2)n1)=O c1(CC)oc(C(=O)NCC(=C2CN(C(=O)C(CC)c3ccccc3)C2)F)cc1C C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CCCC(NC(=O)Cn2nccc2C)C1 c1(C(=O)OC)ccc(C(=O)NC(C)Cn2cc(CSC)nn2)cc1C(F)(F)F c1(C(=O)NCC(CNC(CCCCSC)=O)C)nc2c(Br)cccn2n1 c1(C(N2CCC(=CC(=O)N(CCO)CCO)CC2)=O)cc2c(F)c(F)ccc2[nH]1 C(=O)(C1=CCSC1)NC1CCC(CCC(=O)N(CC)CC2(O)CCC2)C1 C12(C(=O)NC(C)C3CC3)COCC1CN(C(=O)Cc1ccccc1Br)C2 c1(OC)cncc(C=CC(=O)NC2CN(C(c3ccoc3Br)=O)C3CC23)c1 c12ccccc1n(CC(C)C#N)c(=O)n2C1(O)CCCOC1.CC(C)N(C)C c1(N(CCN(C(c2cn(CCOC)nn2)=O)C)C)ccnc(-c2nccs2)n1 c1(C(=O)NCC(CC(C)C)NC(=O)CCn2cccn2)ncc(C(N)=O)cc1Cl N1(C(CC(C(C)C)NC(c2ccc(CF)cc2)=O)=O)CCN(C)C(C)(C)C1 c1(CN2CCCC(C(=O)NC(CC)CN3CCCC3)C2)cc(C#N)ccn1 N1(C(CC(CC)C2CCC2)=O)CC2CCC1C2NC(c1ccc(OC)cc1N)=O C1(CC(=O)NCC(CNC(C(CCOC)C)=O)(C)OC)CCC(C)(C)CO1 C(CC(C)P(C)(C)=O)NC(c1cncc(-c2cnn(CC)c2C)n1)=O N1(C(C2(CC=C)CCN(C(c3cc(CC)no3)=O)C2)=O)CCC2(CC(OC)C2)C1 n1(C(CC)CC)nc(-c2cscn2)nc1-c1cc[n+]([O-])cc1 CC1(C(=O)NCC2CN(C(=O)CCc3cncc(N(C)C)c3)C2)CC2CCC1O2 CN1C(=O)CCCC1C(N1CCOCC1CNC(C12CC(CO1)C2)=O)=O C=CCC(C)C(=O)N1CC(CC=C)(NC(=O)CCCn2ccccc2=O)C1 c1(-c2n(CC)c(N3CCCC(C(C)(F)F)C3)nn2)cn(C)c(=O)n(C)c1=O C(=O)(C1CCCc2n[nH]cc21)N1CC(F)CC(NC(c2c(C)ccc(C)n2)=O)C1 n1(CCC)nnnc1C(C1CCCCC1)NCC1(CCC)CCC1 C1(C(N2CCC(C(N(C3CCN(C)C3)CC#C)=O)C2)=O)CCN(C)C(=O)C1 c1(C(=O)NC2CC(NC(c3sccc3Br)=O)C2)cn2cccc(F)c2n1 c1(N2CCN(N3CC(C)CC(C)C3)CC2)cccc(C#N)c1[N+](=O)[O-].CCO c1(OC)ccc(S(N)(=O)=O)cc1C(N1CCC(C)C1CNC(=O)CC1(O)CC1)=O C(CO)(C(=O)N1CC2COCC2O1)NC(C(COC)C)=O CC1CN(C(C2(O)CCOCC2)=O)CCC1C(=O)N(C)OC1CCCC1 N1(C(C2CCCN(C)C2)=O)CC2CC(NC(C34CC(C)(C3)C4)=O)CC1C2 N1(C(C(C=C)(F)F)=O)CC2(CCC2)CC1C(N1CC(CS(C)=O)C1)=O C(N=c1[nH]c(N2CCc3ccnc(O)c3C2)nc2c1CSC2)C1C(C(C)C)C1 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC1(C)N(C(c2cncc(C)n2)=O)CCC1 c1(OC)ncccc1C(=O)NCCC(Cc1ccccc1)NC(=O)C1=CCCS1 N1(C(c2c(OC)ccs2)=O)CC2(CCCCN2C(c2cc(C)c(C)nn2)=O)C1 C1(CNC(c2ccc(C)c(Cl)c2)=O)CN(C(C2CNC(=O)C2)=O)CC(C)(C)C1 C(=O)(C(C)C(=O)NC(C(=O)NC(c1cncc(F)c1)C)C1(O)CCC1)OC Cc1cnn(C(C)C(=O)NC2CCC(NC(=O)Cc3cnn(C(F)F)c3)C2)c1 c1(OC)ccc(O)c(CN2CC3CN(C(c4cc(OC)nc(Cl)c4)=O)CC23)c1 C(C(CO)N=c1nc[nH]n2c(Br)ccc12)NC(=O)C=C1CCC1 C(=O)(C(F)CC(CC)CC)N1CC2C(C(NOCC(=C)C)=O)(CCC2)C1 c1(C2(C(=O)NCC(CNC(c3cc(C4CC4)on3)=O)OC)CCC2)ccc(C)cc1 c1(CN(c2ccnc(-c3ccccc3)n2)C)nc(Cl)ccc1Br c1(C(=O)NCC(CNC(C2CCS(=O)(=O)CC2)=O)OC)nn(C)c(N)c1C Cc1c2c(-c3cnc(F)c(C(=O)NCC(N4CCCC4)=O)c3)cccc2nn1C c1(SCCNC(C(=Cc2ccc(Br)cc2)C#N)=O)cc(O)nc(-c2ccncc2)n1 CCS(=O)(=O)CC(=O)N1CCC(CNC(=O)Cc2cncnc2)C(C)C1 CN1CCCC1C=CC(=O)NCC(C)(C)NC(C1C=CCCC1)=O N1(C(c2c(NC(C)=O)snc2C)=O)CCN(C(c2occc2C)=O)C2(CCC2)C1 C1(C(N2CCCC2C2CCN(c3nncs3)C2)=O)CC12CCC2 C1(C(F)(F)F)(C(N(CCCN(C)C(c2cnccc2Cl)=O)C)=O)CC2C=CC1C2 c1(C(=O)OC)cc(CN)cc(S(=O)(=O)NC2(CC(F)F)CC2)c1 c1(OC)ccc(C(=O)NC(C2(O)CN(C(=O)C=CC(C)C)C2)(C)C)cc1.C1=NC1 Cc1occc1C(=O)NCC1CCN1C(=O)C(C)c1cc[nH]n1 C1(NC(C(CC)NC(C)=O)=O)CC2CCC1(C(=O)NCCCCCCCO)C2 c1(C(N2C(CNC(c3cccnc3O)=O)COCC2)=O)ccc2c(c1)CCCO2 N1(C(C2(C)N(C)CC(OC)C2)=O)CCCc2ncccc21 C1(C)(C(N2CC(NC(c3cc(C)ncn3)=O)C3(C2)CC3)=O)CCCCNC1=O C1(NC(CC=C)=O)CN(C(c2cc(N(C)C)nc(Cl)c2)=O)CCC1O C1(NC(c2c(C)occ2)=O)CCN(C(c2ccc(-n3nnnc3C)cc2)=O)C1C C1(CNC(c2cc(C)[nH]n2)=O)CCCCN1C(=O)CCC1(C)CCC(=O)N1 c1(C(N2CC(CCNC(C=CSC)=O)C2)=O)c(C)cnn1CC(F)F C1(C(=O)NC2C(C=C)CN(C(c3ccc(O)nn3)=O)C2)CC2(C1)CC(C)(C)C2 CCC(C)(CO)C(=O)N1CCCC(CCNC(=O)Cc2cnc[nH]2)CC1 C1(CC)CCN(C(c2cnc(C)n2C)=O)C(C(=O)NC(C)CN=[N+]=[N-])C1 Cc1ccc(Oc2ccc(Cl)cc2C(F)(F)F)c(Cl)c1O.C1(=O)C(C)N1 C(CC(=O)NC1CCC(NC(=O)C2=CS(=O)CCC2)C1)(C(F)(F)F)OC C(=O)(C(C)=Cn1ccnn1)NCC12CN(C(C(C=C=C)C)=O)C(C1)CO2 c1(C(=O)NC(C)(C)CCC=CCNC(c2cc[n+]([O-])cc2)=O)ncccc1F C(=O)(C(C)C(C)NC(c1sc(F)cc1C)=O)NC(C1CCCCC1)CC C(CN=C(NCc1ccc(F)cc1)N1CC2C(CF)C2C1)N1CCS(=O)(=O)CC1 CCC(CCOC)C(=O)NC(C)(CO)C(=O)N1CC(C)(C(F)(F)F)C1 C(CC)(CS(=O)(=O)c1ccccc1)N(c1cc(N(C)CP(C)(C)=O)ncn1)CC C1(C(=O)NCCC(C)NC(=O)C(C)(O)C2CCC2)COC(=O)N1C c1(CN(C2CCN(C(c3ccc(C#C)cc3)=O)C2)C)cccc(F)c1C#N N1(C(C2CC(C)OC2)=O)CCC(C(O)CNC(=O)CCCN(C)C)CC1 N1(C(c2cc(C)oc2)=O)CC(CNC(C2C3CCC2(c2cccs2)C3)=O)C(C)C1 c1(NC(c2cc(F)ncc2NCc2ccc(Br)o2)=O)ccc2c(c1)OC(F)(F)O2 c1(CC)cc(OC)cc(C(N2CCC2CNC(c2cc([N+](=O)[O-])c[nH]2)=O)=O)c1 CC1CN(C(=O)Cn2cnnn2)CCC1NC(c1cc(Cl)n(C)n1)=O CC1(C)CC(CNC(c2cnn(C)c2F)=O)CN1C(=O)CCF.CC N1(C(Cc2c(C)cccc2C)=O)CCN(C(=O)C2=CCSC2)C(C)C1C c1(C(C)C)cc(C(=O)NC2(C)CC(NC(=O)CC3(n4cccn4)CC3)C2)n(C)n1 c1(C(=O)NC2C(CNC(c3ccccc3)=O)CCCC2)[nH]nc2ncnc(O)c12 c1(CC(=O)NCCCCNC(C2N(CCC)C(=O)CC2)=O)cnn2c1CCCC2 C1(C(=O)NC(C(=O)NCCOC(CC)(C)C)(C)C)CC12CCOC2 c1(CCC)cc(C(=O)NCC2COCCN2C(=O)Cc2ccccc2C)ccn1 c1(OC)cnc(N(C2(C(=O)OC)CNC2)C(C2CCCN(C)C2)=O)nc1 Cc1cc(C(=O)NCC2C(C)CCN2C(=O)COc2ccccc2Cl)c(C)cn1 c1(C(N2CC3C(NC(c4c(C)noc4)=O)C(C3)C2)=O)c(C)oc2ccccc12 C(=O)(NN=c1[nH][nH]c(=Nc2ccccc2Cl)s1)c1ccc(C(N)=O)nc1 C#CC1(O)CCN(C(C)C(=O)NC2CC(C)N(C(C3C4CCCC34)=O)C2)CC1 CCCC(C(=O)OC)C(=O)N1CC=CC1C(=O)NOCCCCC1CC1 c1(OC)ccc2cc(N(C(=O)NCC3CCSC(C)C3)CC#N)[nH]c2c1 c1(OCCN(C)C)c(C(N2CCCC(C3CC(N)CCO3)C2)=O)cccc1N c1(C(=O)NCC2CC(NC(C3(OC)CC(C(F)F)C3)=O)C2)ncc(C)cn1 c1(C(N2C(CCNC(C3OCC(C)(C)C3)=O)COCC2)=O)cnc2ccccn12 C1(CCN2CC(O)CC(OC)C2)Sc2ccccc2NC1=O N1(C(c2n(CC)ccc2)=O)CCCC(CCNC(c2cnc(N(C)C)s2)=O)CC1 c1(C(CNC(C=C(COC)C)=O)N(C)C)ccc(OC(C)C)cc1.C1C=CC1 C(C(C)CC(=O)N(C)CCC1CCOCC1)NC(c1ccn(CCC)n1)=O c1(NCCCOC=C)ccc(S(=O)(=O)NC(c2cn(C)nn2)C)cc1C#N C1(NC(c2c(N(C)C)cccc2)=O)CN(C(=O)CC2(C#N)CCC2)CCC1O Cc1nc(C(C)(C)C)sc1C(=O)NCC(O)CN(C(=O)CCCN(C)C)C C(N=c1nc(O)c2ccccc2[nH]1)C12OCC(NC(C(C)N3CCC3)=O)(C1)C2 CS(=O)CCC(=O)N1CC2CC2(CNC(C2SCCS2)=O)C1 C1(C(=O)NCCn2c(C)nnc2)(NC(=O)C=CC2CCCN2C)CCC(C)(C)C1 c1(C(=O)NC2C3(CCN(C(C4N(C)C(=O)CCC4)=O)C3)C2)ccc([N+](=O)[O-])cc1 FC1CCCCCC1N=c1[nH]c(-c2ccc3c(c2)COC3)nc2cc[nH]c12 N1(C(C)=O)CCC2(CO)CN(C(=O)CC3CCC(C)(C)CC3)CC2C1 C1(CCC(=O)NCC2C(NC(c3n(C)ncc3)=O)CCC2)CCCC(O)C1 C=CCC(C(=O)NCc1c(CC)noc1C)N(C(C(CC)NC(C)=O)=O)C N1(C(c2c(C)nn(C3CC3)c2)=O)CCCC(NC(=O)CC2CCOCC2)C(F)C1 CC1COc2ccc(C(=O)NC3CCC3NC(=O)COC3CCC3)cc21 C1(C(C)NC(C2CCC(C(N)=O)C2)=O)CCN(C(=O)CN2CC(C)(C)C2)C1 Cc1ccc2c(c1)CCC2C(=O)N1CCC2(CC1)CC2NC(=O)CC(F)(F)F C1(CNC(CCCOCC)=O)CCCC(CNC(=O)COCc2ccccc2)C1 c1(OCC)nc(Cl)ccc1C(=O)NC1CC(CNC(=O)CCC(F)F)C1(C)C C1(=CCNC(Cn2ccc(C)n2)=O)CCN(C(C2(C#N)CC2C)=O)CC1 N1(C(C(=O)NC)C)CCC2CC(C(N3CC(C(=O)O)OC(C)(C)C3)=O)C2C1 CC(C)CC(C(=O)N(C)Cc1cocn1)ONC(C1CCCCC1)=O CC1(C)CC(CC(=O)Nc2cccc(CNC(c3ccsc3)=O)c2)CCO1 C1(CNC(C=C(C)Cl)=O)C2CC1N(C(c1cccnn1)=O)C2 c1(C(COC)CNSC(F)F)ccc(Cl)cc1 c1(NC(C2CN(C(c3cc(C)nn3C)=O)CC(F)C2)=O)cc(C#N)c(F)cc1Br C12CN(C(=O)C(c3ccc(OC)cc3)(C)C)CC1NC2.C1(CC)(CC)CC1 CC1(F)CC2(CN(C(c3cc(F)c(-c4cn(CCC=CCO)nn4)c(F)c3)=O)C2)C1 C(CC(=O)N1C2CCC1CN(C(C1COC(=O)C1)=O)C2)(C(F)(F)F)OC C1(CNC(COCP(C)(C)=O)=O)CC12CCN(C(C1CCNC1=O)=O)CC2 c1(OC)c(C(=O)NCC2CCN2C(c2cc(C(C)(C)C)n(C)n2)=O)cccc1Cl CC1=C(C(=O)NCc2cc(C(=O)NCC(c3cnc[nH]3)C)on2)SCCO1 c1(-c2ccccc2)nc(=NC(=O)C2=COCCO2)s[nH]1 c1(N2CCC(C)C2)c(Cl)nc[nH]c1=NCCc1ccc(CN=[N+]=[N-])cc1 c1(C(=O)NCC2CC2NC(=O)C(O)CCc2ccccc2)cc(O)nc(O)c1 C1(C)(C(=O)NC(C2CCCC2)CNC(Cc2cc(C)sc2)=O)CCC(=O)C1 c1(CS(Cc2cc(C)no2)=O)sc2ccccc2c1C C#CCCCCCC(=O)NC(CC#C)C(=O)N(C)CCC1CCCN1C c1(C(N(C(C)C)CCNC(C2CCC2(F)F)=O)=O)cnc(C2CC2)nc1O c1(C(N2C3CCC(NC(c4c(C)nsc4)=O)C(C3)C2)=O)cccc(P(C)(C)=O)c1 c1(C(=O)NCC2(CN(C(=O)CC3(C)CC3)C)CC2)cc[nH]c2nccc1-2 CC(CC(=O)c1ccc(F)cc1)C(=O)NC(c1cc(Br)sn1)=O CN1CCC(C)(C(N2CC(NC(=O)C(F)=CC3CC3)C3(CC3)C2)=O)CC1 c1(C(N2CCC(CNC(c3cnn(C4CC4)c3)=O)C2)=O)cccc(F)c1C(F)F N#CC12C3C4C1C1C2C3C41C(=O)NC(CNC(=O)CCSCC(N)=O)C1CCC1 N12CCC(C)(CC1)C2.c1(C(=O)NCc2ccn(CC)n2)cnc(OC)cc1C C=CCCC(C)(C)C(=O)N1CC(CCCCNC(=O)C#CC(=O)N(C)C)C1 N1(C(=O)CCNS(=O)(=O)c2cccc(Br)c2)CCc2c(O)ccc(F)c2C1 C1(C(=O)NCC(C)NC(c2cnc(C3CC3)[nH]2)=O)CCCC2C1C2(F)F CCC(CC(=O)N1CCC1C(N1CCCOCC1)=O)c1ccccc1.CCO C(=O)(C1=C(Cl)CCOC1)N(C(C)CNC(C1(COCC)CCCCO1)=O)CC CC1=C(C(=O)NC2(CO)CN(C(=O)C(C)(O)C(C)C)C2)CCC(C)(C)C1 Cc1c(C(=O)NC2COCCN(C(=O)C(C)n3ccnc3)C2)sc2nnc(S)n12 C(c1cnn(C)c1C)=CC(=O)N(CCOCCNC(C(n1ccc(C)n1)C)=O)C N1(C(COC(CC)C)=O)CC2(CNC(=O)COC(F)(F)F)CC1CO2 C(=O)(C1=C(Cl)CCCC1)NC1CC(NC(c2cccc(CC)c2C)=O)C1 C(=O)(C(C)(C)CCF)NCC(C)CC(N1CC2CC2C2CC12)=O S(=O)(=O)(c1cccc(N2C3CCC2CC3)n1)N(C)Cc1nc(CC)sc1 C1(C)(CN(CC(C)(C)NC(=O)C(F)(F)F)C)Cc2ccccc2C1 N1(C(c2c(CC)n(C)nc2)=O)CCC2(CC2NC(=O)CCc2cncnc2O)C1 C(=O)(C(C)CCC(C)(C)C)N1CCC(CN(C(=O)CC2=CCCC2)CC)CC1 C1(NC(c2cc(C)ncn2)=O)COCCN(C(=O)CCc2ccc(F)cc2Cl)C1 c1(SCCCNC(C2(Cl)CC2(F)F)=O)nc2ccccc2s1 n1(CCN(C)C)cc(C(=O)NC2(CCNC(C3CC(C(F)F)C3)=O)CC2)nn1 N1(C(=O)C2=COCCO2)CC2C3CCC(C2C1)N(C(c1ncc[nH]c1=O)=O)C3 CC1(NC(=O)CC2(O)CCC2)CCCN(C(C2CCCC2N2CCOCC2)=O)C1 CCCCC(O)C(=O)NC1(CC)CCCN(C(c2scc(C)c2Br)=O)C1 CCCCC(CC)NC(C1C=CCCN1C(c1ccccc1OC)=O)=O C(=O)(C(CN(C)C)OCCCOC)N(C(CC)CC)C(=O)CSCCC#N C1(CNC(C=CCC)=O)COCCN(C(=O)C(C)C(=O)OC(C)(C)C)C1 C(=O)(CCCC(C)(C)C)N1C(C(=O)NCCSCCOC)C=CCC1 C1(C)(C(N2CC(CCCCNC(C(C)NS(C)(=O)=O)=O)C2)=O)CC(=O)C1 c1(NC(C2(NC(C(C)=C(CC)C)=O)CCCC2C)=O)cc(F)ccc1OC C#Cc1cncc(C(=O)N(C2(C(=O)NOCC=CCl)CC2)C)c1 S(=O)(=O)(c1cccc(F)c1C)N1CC2CCN(Cc3nc(OC)c(Br)cc3)C2C1 c1(C(N2C(c3c(C)noc3C)CCC2)=O)cc(Br)cc(=N)[nH]1 N#Cc1ccc(C(=O)NCC2CC(NC(C3CC4CCC4C3)=O)C(O)C2)cc1 C(=O)(CC1NC(=O)c2ccccc21)N1C(C)CCN(C(COC)=O)CC1 C12CCC(CC1)CC(=O)NCCN(C)C2=O.c1(C(C)C)cc(C2CC2)[nH]n1 c1(C(=O)NCC2CCC(NC(Cc3c(C)cnn3C)=O)C2)ccn(C)c(=O)c1 C1(CC(=O)NCC(C(=O)NC)O)N(C(=O)C=CC(F)(F)F)CCC1(C)C C1(C(N(C)C)=O)(NC(=O)C(F)=CCCF)CCC1 c1(CNC(C(c2cccc(Br)n2)C)=O)ccccc1OC(F)(F)F N1(C(c2c(C)cc(C)nc2)=O)CCC2(CC1)CC2C(N(CC(C)C)CCO)=O c1(C(=O)NC(CC(C)NC(CCN(CC)CC)=O)C)cc(C)cc2c1CCC2 C1(NC(C(c2cn(C)nc2)=O)=O)CN(C(=O)C(N2CCCC2)C2CC2)CC1F c1(CC(=O)NC2CC(NC(C(CC)(C)C)=O)C2)c[nH]c2cccc(Cl)c12 Cn1ccc(C(N2CC3CC3(CNC(=O)CCOC3CCCOC3)C2)=O)cc1=O c1(C(=O)OC)cccc([N+](=O)[O-])c1NC1CC(NC(C2CCCC2(F)F)=O)C1 N1(C(Cc2sc(C)c(C(C)C)n2)=O)CCC(C)(NC(=O)CC(C)(C)C)CC1 CC(C)(O)CC(=O)NC1CCOC(CNC(c2cn(C(F)F)cn2)=O)C1 C#CCC(CC(F)F)C(=O)N1C2CCCC1CN(C(=O)CC1CCCN(C)C1)C2 c1(C(=O)NCCN(C(=O)Cc2cccc(C(F)F)c2)CC)ccc2ccoc2c1 C1(CC)CN(C(=O)C(C2CCCCC2)NC(c2cnc(OC)s2)=O)C(C)CO1 CC(=O)CCCC(C)C(=O)NC1CC(C(F)C(N2C3CSCC2C3)=O)C1 CC(CS(C)(=O)=O)N=c1[nH]c(ON2C(=O)CCc3ccccc32)nc2c1CCCC2 C1(CNC(C2(OC)CCOCC2)=O)CC2CCCC2N1C(=O)C(C)C1CC1 N1(C(C(C)=C(C)C)=O)CCC2C1CCCN2C(=O)COCCCC(C)C C1(NC(CC2(C(=O)NC3CC3)CCC2)=O)CCC2CCN(C(C3(C(N)=O)CC3)=O)C12 N1(C(Cc2cnc(C)o2)=O)CC(NC(=O)C(C)Sc2nncn2C)CCC1C C1(C(N(C2CCN(C(C=CCOC)=O)CC2)C)=O)CC(COC)C12CCC2 N1(C(C)C)CCN(C(C2CN(C(=O)OC(C)(C)C)CC(C)O2)=O)CC1C Cn1c(C(=O)NCCCNC(C2CC2C(N)=O)=O)ccc1-c1ccccc1 N1(C(Cc2cn(CC)nn2)=O)CCC(C)C1CNC(c1ccc(C)n1C)=O C1(NC(C(C=CC)O)=O)CN(C(=O)Cc2cc(F)ccc2Cl)CCC1F C1(C(N2CCC(C(=O)NCCCCCO)CC2)=O)CCC(=O)N2CCOCC12 c1(C(CC(N2CCN(CCCO)CC2)C)(C)C)ccccc1Br CC1CCN(C(=O)C(CCN(C)C)NC(c2cc(=N)[nH][nH]2)=O)CC(C)O1 CC1(C)CCCCN(C(C23CC(NC(=O)C=CC(F)F)(C2)C3)=O)C1 C(=O)(C(CC(C)C)OC)N1CCCC(CC(=O)NCC(CC2CC2)OC)C1 C1(CC#C)(C(=O)NCc2cccc(C)n2)CCN(C(C2CC23CC3)=O)C1 C(N=c1cc(C)nc(C#N)[nH]1)C1C2CN(C(CC)=O)CC21 Cc1cc(CCC(N2CCOCC2CCNC(=O)CCC(C)N(C)C)=O)nn1C c1(C(=O)NC(CCC)CNC(c2cnc(CC)s2)=O)cccn(C)c1=O CCC(C)C(O)C(=O)N1CC(OCC(=O)NCC2CCC(C)(C)CC2)C1 C=C1CC2(C1)CN(C(C1CCCC(NC(c3ncccc3F)=O)CC1)=O)C2 N1(CC(=O)Nc2ccccn2)CCCc2ccccc21.C12CCCC1CNC2=O c1(C(=O)NC2C3CN(C(C(C4CCC(C)CC4)CC)=O)C2C3)nc2ccccc2s1 N1(C(C(CSCC)(C)C)=O)CCN(C(c2ccc(COC)[nH]2)=O)C(CCO)C1 CC(C)C(C)C(CNC(c1cc(C(F)(F)F)ccc1O)=O)NC(=O)CC(F)F C1(NC(C=CC=CC)=O)CS(=O)(=O)C12CCN(C(=O)C(C)CCC)CC2 c1(CNC(=O)NCCOCCNC(COCCCC)=O)sc(C)c(C)c1Br C(=O)(CCC(C)(C)C#N)N(CC(N1CCC(OC(C)=O)C1)=O)CC1CC1 C(CCN=C(NCC(C)(C)C(C)(F)F)NC1CCCN(c2ncccn2)C1)OC N1(C(C2(OC)CC(CF)C2)=O)CCC(CCNC(C23CC(O)C2C3)=O)CC1 CC1CC(C(N2CCC(C(C)C(=O)NC3CCC(CO)C3)CC2)=O)CN1C N1(c2c(C)c(NCCc3cnc[nH]3)ncn2)CCC(C2CCCOC2)CC1 c1(C(N(CCNC(C(C)(C)OC)=O)C)=O)cc(C)ncc1Br C1(C(=O)NCCNC(C(c2scc(C)n2)(F)F)=O)CC2CCC2C1 N1(C(c2nccc(Cl)c2F)=O)CCC2CCN(C(=O)C(F)(F)CO)CC2C1 CCC(CC)(CO)C(=O)NC(C)C(C)NC(c1cc(C2CC2)n(C)n1)=O C12(C(N3CC(F)(F)C3)=O)C3C4C1C1C2C3C41C(N1CC(CCO)C(O)C1)=O N12CCCC1(c1cccc(Br)c1)C2.N1(CC(O)c2ccsc2)CCCC1 C1(C)(CN(C(=O)C=Cc2cocn2)C)CCCC1NC(=O)CN1CCSCC1 c1(C(=O)NCC2CC(NC(CCOCCCOC)=O)C2(C)C)ncc(F)cc1F c1(CC)nc(C)c(C(=O)NCCOC2CN(C(=O)CC3(O)CCC3)C2)o1 N1(C(CCCC(C)(F)F)=O)CCC2(CCN(C(C3(CF)CC(F)(F)C3)=O)C2)C1 C1(CNC(c2ccc(CC)s2)=O)CCC(C)N(C(C2CCC(O)C2)=O)C1 c1(CC(=O)N(CCNC(C2CC2(C)Br)=O)CC)nc(C)c(C)s1 C(CC(C(=O)NCc1cn(CC(N2CCC(O)(C(F)F)C2)=O)nn1)OC)OC C(c1ccccc1)=C(CC)C(=O)NCC1CCC1NC(=O)CCc1cc[nH]n1 c1(C(=O)NC2(c3ccccc3)CN(C(C(CC)OC)=O)C2)ncc(F)c(OC)n1 Cc1ccccc1C(C)CC(=O)NCC(C)NC(=O)Cn1nnnc1C1CC1 c1(C(CC)NC2CCOC2)nc(C)cc(=NCCc2cc(F)ccc2OC)[nH]1 c1(C(=O)NCC(CC=C)NC(=O)C(C)(C)c2cccs2)c[nH]c2nccc-2c1C N1(C(C(COC)(C)O)=O)CCC(CO)(NC(=O)C=CCF)CC1 c1(C(=O)NCC2(O)CCN(C(c3cncc(OC)c3)=O)C2)cc2c(s1)CCSC2 C(=O)(CCCC(F)(F)CO)N1CC(NC(=O)COc2cccc(F)c2)C(CO)C1 N1(C(C(C)OC2CCCCC2)=O)CCC(C2(NC(C3CC=CCC3)=O)CC2)CC1 C1(NC(CC2C(C)C2)=O)CN(C(=O)CN2CCC(N(C)C)CC2)CC1(C)C Cn1nc(Br)cc1CC(=O)NCC(C)(C)CNC(C1CC2(CC2)CO1)=O CN1CCC(C(=O)NC(C)(C)CNC(=O)CCc2ccc(N(C)C)nc2)S1(=O)=O C1(CNC(C=C(CC)CC)=O)CCCCC1NC(=O)COC1CC(F)(F)C1 c1(CNC(C2C(NC(C(CCC)C)=O)C2)=O)cnc2[nH]ccc2c1 Cn1ncc2c1CC(NCC(=O)Nc1ccc(F)c(F)c1F)CC2 C1(N(CC(C)C)C(=O)CC2CCC(=O)N2)CCN(C(C2CC2(F)F)=O)CC1 C(CCN(C(=O)CCN(C)CCO)C)(C(C)C)N.C1(OC)CN(CC(=O)NCC)C1 c1(C(=O)NC2CC(CC(=O)NCc3c(CC)n[nH]c3)C2(C)C)cc2occc2[nH]1 C1(N(C(Cc2cc(C(C)=O)sc2)=O)CCO)CCCN(C(C2CC(C)=NO2)=O)C1 c1(C(N2CCC(C)N(C(=O)CC3C=CCC3)CC2)=O)cc2ccccc2c(O)n1 C1(CCNC(=O)CCOC2CCOC2)CCN(C(=O)CSn2cnnn2)C1 C(C)(C)(CCC(=O)NC(C1CCCN(C(c2nn(C)nc2C)=O)C1)C)OC c1(C(=O)NC(c2c(C)c(F)ccc2)C)ccc2nc(C3=CCCC3)cn2c1 c1(CC)cc(C(=O)NCC(O)CN(C)C(c2cn(C)nc2C)=O)cc(N)c1 C1(C(=O)NCC#CCNC(Cc2n(C)ccc2)=O)CN2CCN1CC2 C1(CCN(C(C2(CSCC)CC2)=O)C)CCCCN1C(c1[nH]c(O)nc1C)=O c1(C(N2CC3C(NC(CC(COC)C)=O)(CC3)C2)=O)cccc2c1CCC2 Cc1ccc(CC(C)C(=O)NCC2CCN2C(=O)Cc2ccco2)cc1 N1(CCN=C(NCC(=O)NC(C)C)NC2CC(N=[N+]=[N-])C2)CCn2nccc2C1 C1(N(C(C(C)=CCC)=O)C)CCC(C(=O)NCC(=O)NC(C)(C)C)C1 c1(NC(NC2CCCn3ncnc32)=O)cc2ccc(OC(F)F)cc2o1 N1(C(CCc2scc(C)n2)=O)CCC(F)(CNC(c2cc(Cl)cn2C)=O)C1 C=C(C)CCCC(=O)NC1(c2cn(-c3cncc(SC)c3)nn2)CC(F)(F)C1 N1(C(C(COC)NC(C)=O)=O)CCCOC(CNC(=O)CCC(C)CN(C)C)C1 C(=O)(CCCn1ccnc1)NCC(C)(C)NC(=O)CC1CCCO1 c1(C(N(CCCN(C)C(c2c[nH]nc2C(F)F)=O)C)=O)cc(C2(O)COC2)on1 c1(C(=O)NC2C(C)(C)CCN(C(COC(C)(C)C)=O)C2)coc2c(Cl)cccc12 Cc1ccc(F)c(CNC(=O)C=CC(C)NC(c2occ3c2CCC3)=O)c1 C1(CC)CN(C(C2(CCOC)CC2)=O)CCC1NC(=O)Cc1cnsc1 N1(C(CSc2c(C)cccc2)=O)CC(NC(C2(OC(=O)N(C)C)CC2)=O)CC(O)C1 N1(C(c2cc(SC)oc2)=O)CCC(C)C1C(=O)NCC#CC1CC1 CC12CCOC(C(N3CCC(NC(c4ncnc(O)c4Cl)=O)CC3)=O)(C1)C2 c1(C(N2C(C3CCN(C(CCC(N)=O)=O)CC3)CCC2)=O)cc2n(n1)CC(F)C2 N1(C(c2n(C(C)C)cnc2)=O)CC(N(C(=O)CN2CCOCC2)C2CC2)C(C)C1 CCC(C)(CC)C(=O)N1CC(CNC(c2cncs2)=O)OC(C(F)(F)F)C1 C1(C(CNC(C(C)OCC)=O)(C)C)CCN(C(=O)C(C)CC2CC2)CC1 N1(C(C(=CC2CCCC2)C)=O)CC(O)CC1(C)C(=O)NOCCC(C)O C(=O)(C1CCc2ccccc21)N(CCC(=O)NC(COC)CO)C(C)C CC(C)C(C(C)NC(c1ccnn1CC(F)(F)F)=O)NC(=O)CSCC(N)=O C1(NC(CN(CCNC(=O)CC(=O)NCC=C)C)=O)CC2CCC1C2 C1(C(=O)NC(CNC(C2CCC(C)(CC)O2)=O)CO)CN2CCN1CC2 N1(C(C(C)NC(C2CC(N=[N+]=[N-])C2)=O)=O)CC(C)C12CCOCC2 c1(CC(=O)NC23C(CN(C(c4cccc(OC)c4)=O)C2)C3)cc(Br)ccc1C C12(NC(C(CC=C)NC(C3C(C)(C)C3(F)F)=O)=O)CCCN(CC1)C2 CCCC(C)(O)C(=O)N1CC(NC(c2cn(C)nc2I)=O)C1 Cc1c(C(=O)NC2CCN(C(=O)CC3OCCO3)CC2O)sc2[nH]cnc(=O)c12 C(=O)(C1=NOC(CNC(=O)CCCC2CC2)C1)N(CCn1cccn1)CC C1(C(=O)NC2(C)CCN(C(c3cc(Cl)cs3)=O)C2)CC(S(C)(=O)=O)C1 N1(C(C(C=CC)O)=O)CCC2(CC2)CC1C(=O)NCc1ncc(C)cc1C C(=O)(C#CC1CCOCC1)N1CCC(C(N2CC(C)=C(C)C2)=O)C(C)C1 C1(Cc2ccc(C)o2)CCN(C(=O)C(=O)NCc2c[nH]cc2C(F)(F)F)CC1 N1(CC(=O)NCCC(CNC(=O)C(C)C2CCOC2)OC)CCC(C)(C)C1 N1(C(C2CC(OCC)C2)=O)CCC(C(C)NC(=O)CC2(C)CC2)C1 c1(-c2c(C(=O)NCCOc3c(SC)cccc3)ncnc2)cccc(Cl)c1F C(CC(C)(C)C(=O)NCC1(C)CCC(NC(C2(C(C)(F)F)CCC2)=O)C1)OC c1(C(=O)NCC2C(C(N(CCOC)C)=O)CCO2)ccc(O)nc1C c1(C(N(C(CC)CNC(=O)C(c2ccn(C)n2)C)C)=O)ccc(C)c(Cl)c1 C1(NC(CCC#C)=O)(COC)CCN(C(=O)CCc2nc(SC(C)C)no2)C1 C1(NC(c2ccc(C)[nH]2)=O)CN(C(=O)CCC(=O)NC2CCCC2)CC12CCC2 n1(CCC(=O)NCC2(O)CC(NC(C3CCSC3)=O)C2)nc(O)c2c1CCCC2 C(C(C)C(F)C=O)O.C1(CN2CCC(C(=O)OC)CC2)CCCS(=O)(=O)C1 C(=O)(C(C)(C)C(C)NC(=O)CCCN(C)C(C)C)NCCn1c(C)nc(C)n1 c1(C(CC(=O)NCCOCCNC(C2(C)C(C)C2)=O)C)ccc(Cl)nc1 C1(c2c(C)ncs2)CCCN(CC(O)COCC2CCOC2)C1 N1(C(C(C)C(C)O)=O)CCC(NC(c2cnc(Br)s2)=O)C(F)(F)CC1 c1(CN2CCC(NC(=O)Cc3cccc(Cl)c3F)C(F)C2)cc(F)cc(Br)c1F C1(C(=O)NCCN(C(C(C(C)C)c2ccc(Cl)cc2)=O)C)CCCCCN1C C=CCCC(F)(F)C(=O)NCC(O)C(=O)NC1COC(C)(C)C1 Cc1cccc2cc(C(=O)NCCCNC(c3c(Br)noc3C3CC3)=O)nn12 C#CCC(C)(C)C(=O)N1CCC(NC(=O)CCCCCn2cnnn2)C(F)C1 c1(C(=O)OC(C2CCCOC2)C(=O)OCC)ccc(C(F)(F)F)nc1 N1(C(C(C)CO)=O)CCC2(NC(C3CCCC(C)CC3)=O)CCCCCC12 c1(CC(=O)N(C2CCC(NC(C3(C)CC=CCO3)=O)CC2)C)c(O)ncnc1O c1(C(=O)NCC(N(C)C(C2(C(C)(F)F)CC2)=O)C2CC2)c(N)cccc1[N+](=O)[O-] c1(N2CCC(CC)(CO)C2)nc2c(c(=NCc3nnc(C)s3)[nH]1)CCCC2 C(C(=O)NC1CCN(C(c2c[nH]nc2C(F)(F)F)=O)C1C1CC1)(C(C)(C)C)SC C(CC(C(=O)NCCC1CC(C)=NO1)NC(=O)C(C)N1CC(C)C1)=CC C(CCCCCC(=O)N(CC(O)CNC(C1CCC1C(F)F)=O)C)SC C(=O)(C(C)(F)C(=O)NCC(C)CNC(c1cn(C)nc1C)=O)OC CCC(O)C(=O)NC1(CNC(C2CC2(C)C)=O)CCCC1 C1(CC(=O)NCCC2(NC(C3N(C(=O)OC)CC3)=O)CC2)CC(C)(C)CO1 C1(C(N2C(C=C)CCC2)=O)CCN(C(=O)c2cc(C(C)C)no2)O1 CC1CN(C(c2ncc(Cl)cc2F)=O)CCCN1C(C1CCC(C(F)(F)F)O1)=O c1(C(=O)NCC2(O)CCN(C(Cn3c(=N)[nH]nc3)=O)C2)[nH]cc2c1CCS2(=O)=O c1(COC)nccc(=NC2CS(=O)(=O)CC2NC(c2ccc(O)nc2)=O)[nH]1 CCC(C(=O)NC)NC(=O)CC1CC1CNC(C1(C)CC=CC1)=O.C1CC1 C#CC1(F)CN(C(=O)CC2CCCCN2C(C2CCC(=O)N2CCC)=O)C1 CC1CCCN(C(=O)CCn2ccnn2)C1CNC(=O)CCC(=O)N(C)C C(C(CNC(=O)COCc1ccco1)CO)NC(C1C(C)C1)=O Cc1nc(F)ccc1CNC(=O)NC1(N(C)C)CCCC1 c1(NC(c2nc(C(=O)Nc3ccc(OC(C)C)nc3)sc2)=O)cnnc(O)c1Cl C(CC(C)(C)NC(=O)CC1CCCOC1)N(C(=O)CC1CCSC1)C C1(C(F)(F)F)(COC(C(CC)F)=O)CCOCC1 C1(C(C)NC(C=CSC)=O)CN(C(=O)Cc2csc(C(F)(F)F)n2)CCO1 C1(C2CCCC2)(NC(C2CC(C)CN(C(=O)C=CCF)C2)=O)CCC1 C1(NC(c2cc(Cl)c[nH]2)=O)CC2(C1)CC(NC(C1CC(n3ccnn3)C1)=O)C2 c1(C(=O)NCC2(NC(C=CCC)=O)CC(C(F)(F)F)(OC)C2)sc(C)c(C)c1C c1(OC)cccc(CC(=O)NC(C)CC(C)NC(C2CCC(C)C2)=O)c1 C(N=c1[nH]c(=NCC(CO)OC)c2c(F)cccc2[nH]1)c1ncc(CC)s1 c1(CN(CC)Cc2ncc(C(C)(C)O)s2)ccccc1 C1(NC(CS(N)(=O)=O)=O)CN(C(C2CCCC3(CC3)C2)=O)CC12CCOCC2 N1(C(C(CCCC)O)=O)CCC2C1CCCN2C(=O)Cn1ncc2cccnc12 CC(C)(C#N)CCC(=O)NC1CC2(C1)CN(C(C1CCCCCC1)=O)C2 c1(C(=O)NCC#CCNC(c2cc(CC)oc2C)=O)ccc(C#N)cc1O Cc1ccc2[nH]nc(C(N3CC4(CNC(=O)C=CCO)CCC3C4)=O)c2c1 N1(C(C(CC)=CC)=O)CCOCC1CCNC(=O)C(O)C(C)C CC1CN(C(=O)CCC2CC2)CC(C)C1NC(c1cc(Br)ccc1F)=O CCS(=O)CC(=O)NC1(CNCc2ccc(C(F)(F)F)cn2)COC1 C(=O)(CC(C)C(F)F)NCC1(F)CC(C(=O)NC(C)CN2CCOCC2)C1 c1(C(N2C(CCNC(c3sc(F)cc3Cl)=O)CCC2)=O)ccn2ccnc2c1 c1(C(=O)NCC2(NC(=O)C=Cc3nccs3)CCOC2)nccc2[nH]ccc12 C1(C(N2C(CCCNC(=O)CSC(F)F)CCC2)=O)CN2CCN1CC2 S(=O)(=O)(c1cc(C)cnc1N1CCCCC(C)(F)C1)NCC(C1CCC1)OC C1(C(=O)OCC)(CC)CCN(CC(=O)OC)CC1.C(c1ccccc1)=CC(=O)NCCC CC1(C)CCCC(C(=O)NC2CC(NC(C3CCOC(=O)CC3)=O)C2)CC1 c1(NC(c2c(C(=O)Nc3cn(OC)nn3)[nH]cn2)=O)cc(F)c(Br)c(C)c1N c1(C(=O)NC(CC#C)Cc2ccccc2)ccnc(N2CCCS2(=O)=O)c1 CC(CN(C)C)CCC(=O)N(C)CC1CN(C(=O)Cc2c[nH]ccc2=O)CCO1 c1(C(N2C(C(=O)NCC(C#C)OC)CCCC2)=O)cccc(C#C)c1C C(=O)(C1=CC2CC(C1)CC2O)N(CC(c1ccc(Cl)c(Cl)c1)=O)CC1CC1 C(N=c1[nH]cnc2[nH]ccc12)C1N(C(CN(C)CC)=O)CCC1 c1(SC)nc(N2CCC(O)C(C(N3CCn4nccc4C3)=O)C2)ncc1F C1(NC(CCCCN(C)C)=O)CC12CCN(C(=O)CC(C)(F)F)C2 c1(OC)cccc2cnc(N3CCCC(C(=O)N(C)C(C)C)CC3)nc12 c1(C2(O)CC(C(N3CC(NC(C(C)OC(C)(C)C)=O)C3)=O)C2)cccc(Cl)c1 c1(CN2CC(CCO)OCCC2)cc2nc(OC)cc(Br)c2o1 N1(C(CC2C3CN(C(CCc4cnc(C)o4)=O)CC32)=O)CC2(CCN2C)C1 S(=O)(=O)(c1ccc(Nc2c(O)noc2C)cc1)N1CCN(CCCC)CC1 c1(C(N2CC(CNC(CCSCCCC)=O)(OC)C2)=O)cc2n(n1)CC(F)C2 CCC(C)(C)C(C)CC(=O)N1CCCC(C)(C)C1CNC(=O)COCCOC N1(C(c2cccc(-c3cc[nH]n3)c2)=O)CCC2CC1CN(C(C1(O)CCC1)=O)C2 C(C)(CCCNC(=O)C(O)COCc1ccccc1)NC(COC(C)C)=O N1(C(CCn2c(C)ncc2)=O)CC2CC1CN2C(C12CCC1CC2)=O Cc1ccn(CC(N2CCC(C(=O)NC(c3ncc(C)o3)C)C2C)=O)n1 C1(CCC)CN(C(=O)Cc2ccc(Cl)cc2C)CCN1C(=O)Cc1ncc(C)o1 C1(CNC(C(C)CC(F)F)=O)CN(C(=O)CCC(C)(C)F)C2(CCC2)C1 N#Cc1ccc(Cl)c(C(=O)NC(Cc2cn(-c3ccccn3)nn2)C(=O)O)c1 Cc1ccc(C(=O)NC(C)CN(C)C(C2CC(C3OCCO3)C2)=O)c(N)c1 N1(C(CC(C=C)CC)=O)CCC2(CC1)CC2CNC(c1conc1C1CCC1)=O O(NC(=O)CC(C)C(C)(C)NC(C1CCCCO1)=O)CCCOCC C1(NC(CCCc2scc(C)n2)=O)C2CC1CN(C(C1(C3CC3)CCCO1)=O)C2 C1(CNC(c2c(C(C)C)n(C)nc2)=O)CC2(CCC2)CN1C(C1COCCO1)=O c1(CC)cccc(CC)c1CC(=O)NCC1CC(O)CN1C(=O)CC1(C)CCC1 c1(N2CCC(C(C)NC(C3C(OCC)C3C)=O)C2)ccc(C#N)nn1 C(C#CC#CCO)NC(C(C1CN(C(C2CCCCN2C)=O)C1)OC)=O C1(CC)CCC(C(=O)NCC(F)CNC(c2ncsc2COC(C)(C)C)=O)C1 C1(F)(CNC(c2ccc(C)o2)=O)COCCN(C(c2ccc(CO)c(F)c2)=O)C1 C1(NC(COC(CC)CC)=O)CC2CC(NC(=O)CCc3cccs3)CC12 C1(C(=O)NCC(C)N(C(=O)C(=O)C2CCCC2)C)CCC2(CCOCC2)O1 C1(C(N2CC(O)(C3CCCN3C(C3CC(=C4CC4)C3)=O)C2)=O)CC12CCOCC2 c1(NC(C23C(CN(C(CCN(C)C)=O)C2)C3)=O)ccc2[nH]c(=O)ccc2c1 c1(C(=O)NC(CC(C)NC(C(CC#C)O)=O)C)cc(F)cc(Br)c1 C1(C(=O)N(C)CC2(O)CN(C(c3cc(Cl)ncc3O)=O)C2)(OC)CCCC(C)C1 CCC(C)C(C)C(=O)N(C)CCN(C)C(c1cnnc(Cl)c1)=O c1(OC)ccc(C(CNC(=O)C(C)(C)F)NC(C23CC(F)C2C3)=O)cc1 C1(C(=O)NCC2C=CC(NC(c3cnc(CC4CC4)s3)=O)C2)(COC)CC=CC1 C1(CC)CC(C(=O)NC2CC(N(C(=O)CC=CC(C)(C)C)C)C2)C1 CC(CCCC(=O)NCc1cn(C2CC2)nn1)NC(=O)C(C1CC1)N(C)C c1(OC)ncc(Cl)c(C(=O)NC(C)C(C)NC(=O)C(O)C2CCC2)c1Cl C1(NC(C(CC)C(C)(F)F)=O)CCC12CCN(C(=O)CCCCOC)CC2 C1(CC(=O)NC(CCC=C)C)CCCN(C(C2CCCN2CCC)=O)C1 C1(NC(NCC(C2CC2)NC(=O)OC)=NC(C)C)CCC2(CC1)CS(=O)(=O)C2 C(=O)(CCCCCN=[N+]=[N-])NCCC(C(=O)N(CC(=C)C)CC(=C)C)O N1(C(C2CCCN(C)C2)=O)CCC(NC(=O)CN2CC(=O)NC2=O)C(F)(F)CC1 N1(C(Cn2c(C)cnc2)=O)CC(O)CC1(C)C(=O)NCCC(F)(F)CO c1(C(N2CCC(N(C(=O)C(CO)N(C)C)CCC)C2)=O)ccc(=O)n(CCF)n1 c1(CNC(=O)C(c2cc(Br)cs2)=O)ccc(C2CCCCC2)cc1 O=S(=O)(c1ccc(N2CCC(CCO)C2)c(Br)c1)NCC1CCC1(F)F c1(C(=O)NCC(n2cc(CCN(C)C)nn2)C)ccc(-c2cnco2)cc1 c1(C(N2CC(O)(C(C)NC(c3c(CC)nc[nH]3)=O)C2)=O)ccc(N)c(N)n1 C1(CN(CC(F)F)C)COCCN1C(c1cc(NC(=O)OC(C)(C)C)ccn1)=O C(=O)(CCS(N)(=O)=O)N1CCC(OCCNC(C2CC(N(C)C)C2)=O)C1 C1(NC(C(C)=CC)=O)CC2(CCN(C(c3cc(C(C)(F)F)ccn3)=O)C2)C1 C(C)(C)(CCC(=O)NCc1csc(C(=O)NC2CN(C(C)=O)CC2C)c1)OC c1(OC)ccc(C)nc1C(N1CC2CC1CC2NC(=O)CCOCC(F)(F)F)=O c1(C(N2CCN(C3CCC3)CC2)C(=O)NC(C(=O)OC)C)ccc(Cl)c(C)c1 C1(C(=O)NC2CC3(C(NC(c4c(CC)n(CC)nc4)=O)C3)C2)CN2CCN1CC2 N#CC1CC2(CNC(=O)Cn3cc(C4CC=CCC4)nn3)CC1C2 C1(C(N2CC(CC(C(=O)N(C(CC)C)CCO)F)C2)=O)CC2COCC2C1 C(=O)(C1CSc2ccccc21)N1CC(C2CN(C(c3cccc(C#N)c3)=O)C2)C1 C1(N(C(=O)C=CC=CCC)CC#C)CCN(C(=O)C=Cc2c[nH]nc2C)CC1 N1(C(Cc2c(C)occ2)=O)CC2CN(C(C3CC(C)(C)C3)=O)CC2C(F)(F)C1 N1(C(C(CCC)CC)=O)CCC2(CCCN2C(c2cnc(C(F)F)cc2C)=O)C1 N1(C(c2cc(C)[nH]c2)=O)CCSCC1CCNC(c1ncccc1C(C)(C)C)=O C(=O)(C1Cc2ccccc21)NCCC1CC(C(=O)Nc2cc(Cl)ccc2F)C1 C(c1nc2ccccc2o1)=CC(=O)N(CCNC(c1c(C)cnnc1O)=O)CC C1(CNC(CC(C(CC)C)O)=O)(NC(=O)Cn2ncnn2)Cc2ccccc2C1 C(=O)(C1CCc2nccn21)N1CC(NC(c2c(CC)nco2)=O)CC12CCC2 C1(NC(c2c(OC(C)C)cncc2)=O)CC2CN(C(c3cccnn3)=O)CC2C1 C1(NC(c2[nH]cc(C)c2)=O)CC2CC(C1)N(C(c1cnc(C3CCOC3)s1)=O)C2 C1(NC(c2cn(C)c(=O)n2C)=O)CC12CCN(C(=O)C#CC1CCOC1)CC2 c1(C(=O)NC2COCCN(C(C(C)(F)F)=O)C2)occ2c1CCCC2 N1(C(C(CC)(C)OC)=O)CC(NC(=O)Cn2ccc3ccccc23)CC(C)(C)C1 c1(C(N(C(C(=O)Nc2c(OC)cccc2)(C)C2CC2)C)=O)cc(C)n(C)c1C N1(C(C2CC2c2ccccc2Cl)=O)CCN(CC2CC(c3ccccc3)C2)CC1 CCC(CC(=O)NCC1(C)CCCN1C(=O)C(COC)C(F)(F)F)C(F)F C1(OC)CC2CCC(C1)N2N1C(C=O)C2CC2C1.n1(CC=O)cnnc1 n12ccnc1C2.c1(NC(=O)NC2CCN(CC)C2)ccccn1 CCCCC(C)C(=O)NCCCN1CCC(CNC(=O)CN2CCCC2)CC1 c1(C(=O)NCCCCNC(CCOCC(C)C)=O)cc2c(s1)CCS(=O)(=O)C2 N1(C(C2(C)CC=CCO2)=O)CC2CCCC2(CNC(=O)Cn2cnnc2)C1 CCC(CC(=O)NCCCCCSC)NC(=O)CC1CC=CCN1C N1(C(C2N(C(c3n(CC)ccc3)=O)CC(F)C2)=O)CCS(=O)C(C)C1 C1(CC)CCN(C(C2CC(NC(C3CC=CCC3)=O)C2)=O)CCO1 CN1CCOC(C(=O)NCC2(F)CCCN(C(c3cc(N)c(F)cn3)=O)C2)C1=O c1(C(=O)OC)ccccc1N1CC(NC[Si](C)(C)C)CC1=O CC(CC(=O)NC1(C2CCCN2C(=O)C(C)(F)F)CC1)C1CCCC1 Cc1nc(CC(=O)N(CCCNC(c2ocnc2C2CC2)=O)C(C)C)c(C)s1 C=C(C)CC(C(=O)NC(C)Cc1cn[nH]c1)NC(=O)C(C(C)C)C1CC1 n1(CC(=O)NC(CCCNC(C(CCSC)O)=O)(C)C)cccc(C)c1=O C(C(C)(C(=O)NCCOC1CN(C(C2CCN(C)C2=O)=O)C1)OC)OC Cc1nc2c(o1)CCN(C(C1CCCCCN1C(C1CCC(=O)NC1)=O)=O)C2 N1(C(C2C(C)(C)C2)=O)CCC(O)(CCNC(=O)C2=CCCCC2)CC1 C12(NC(c3c(C#C)cn(C)n3)=O)CC(C)(C1)OC21CCN(C(C2CC2F)=O)CC1 C(=O)(C1=CCC(C)(C)CC1)N(CC(C)NC(c1cc(OC)ccc1O)=O)CC c1(OC)ccc(N)c(C(=O)NCCC(C)NC(=O)CCOC2CCCOC2)c1 CCC(N=c1[nH]c(N2CCN(C(c3cncs3)=O)CC2)nc2cc[nH]c12)C1CC1 c1(C(=O)NC2C(NC(=O)CCOCC(F)F)CCC2)cn2c(n1)CCCC2 Cc1ccc(C(=O)NC(C)(C)CCCNC(=O)Cc2cncs2)c2cccnc12 C1(NC(C2(CNC(c3cn(CC)nn3)=O)CC2)=O)CCCC(C(N)=O)C1 c1(C(C)C)cccc(C(=O)NCCCCC2(NC(=O)CSC(F)(F)F)CC2)c1 C1(C)(C(=O)NC2CC(C)N(C(c3cnn(C)c3F)=O)C2)Cc2ccccc2N1 c1(C(N2CC(NC(CC=C)=O)C(C)CC2)=O)ccc2nc(O)n(C)c2c1 C1(C)(C(N(CC(=O)N(C(C)C)C)C)=O)COC(=O)N1 c1(C(N)=O)oc2ccccc2c1CNC(C1CC2CCC(C1)C2(F)F)=O c1(CC)cccc(C)c1C(=O)NCC1(F)CN(C(c2nc(C(C)C)oc2C)=O)C1 C1(NC(c2c(CCC)n(C)nn2)=O)CCCCN(C(=O)Cc2ccnnc2O)C1 C1(CNC(c2cc(C)n(C(C)C3CC3)n2)=O)CN(C)CCN1C(=O)C=CCO c1(COC(C2N(C(C(=C=C)C)=O)C(C)(C)OC2)=O)cc(Br)cc2c1OCC2 C(=O)(C1=CCC(C)CC1)NCC(C)CNC(c1ccc(-c2ncn(C)n2)cc1)=O C1(CNC(=O)C=Cc2cocn2)(CO)CCN(C(C2CC23CCC3)=O)C1 c1(OC)c(N)c(C(=O)N(CC(C)NC(C2CC2CF)=O)C)cc(Cl)c1Br N1(C(COCCCCC)=O)CC2CC2(CNC(c2cc(C(C)(C)C)c[nH]2)=O)C1 C1(CN(C(=O)COCCF)C)CCCN(C(c2ncc(Br)cn2)=O)C1 Nc1ccc([N+](=O)[O-])cc1C(N1CCOCC1CNC(C1COCCO1)=O)=O c1(C(c2n(CCOC)nnn2)NCCCC(F)(F)F)noc2c1CCC2 CC1CCC(O)CN1C(=O)C(c1ccc(Cl)cc1O)(C)C O=S(=O)(c1cnc(NC2CCC3CC23)c(Cl)c1)NCCCOc1ccc(F)cc1 c1(C(=O)NCCCCNC(c2ccn(C)c(=O)c2)=O)c(F)cc(F)c(F)c1F N1(C(=O)Cc2nc(F)c(F)cc2F)CCCC2C1CCCN2C(=O)CC1(CSC)CC1 N1(Cc2ncc(OCC)nc2)CCC(NC(=O)Cc2ccc(Cl)c(F)c2)C(C)C1 c1(CNC(C2N(C)CCCCC2)=O)ccc2c(c1)N(C)CC2 C1(NC(=O)Cc2cc[nH]c2)CC2(C1)CC(NC(c1sccc1Br)=O)C2 C1(CN(C(C=C(C)C)=O)C)CCCCN1C(=O)CC(C)c1ccncc1 N1(C(c2nccc(C)c2)=O)Cc2ccc(C(=O)Nc3cc(Cl)cnc3C)cc2C1 C(=O)(CCCN(C)C(C)=O)O.C(=O)(CCCn1cc(C)cn1)NCC CC1CC=C(C(=O)N(C(C)(C)CC(N2CC(=O)NCC2C(N)=O)=O)C)CC1 N1(C(C(CSC)(C)C)=O)CCOC2(CCN(C(=O)Cc3sc(C)cc3C)C2)C1 C1(C)(C(=O)NC(C)C(C)NC(C2(F)CCOCC2)=O)CC(c2ccccc2)=NO1 CC(CCCC(=O)NC1CCCC1C#N)NC(=O)C=C1CCC1 c1(C(=O)NC(CNC(C2CC2c2ccoc2)=O)CO)cc2ncccc2[nH]1 c1(C2(C)COC2)cc(Cl)ncc1F.c1(Cc2n(C3(C)CC3)nnn2)cnc(F)nc1 Cn1cc(Cl)c(C(=O)NC2CC3C(NC(C4CCS(=O)CC4)=O)C3C2)n1 c1(C(=O)NCC2C(NC(CCC(CC)CC)=O)C2)cc2cccc(OC)c2o1 c1(CN2C(CC)CN(C(c3cccc(C(N)=O)c3)=O)CC2)ccc(F)cc1C#N N1(C(COCCN(C)C)=O)CC(NC(=O)C(=C2CCCCC2)F)CC(F)C1 c1(C(N(C)CCOCCNC(=O)Cc2cnccn2)=O)cncc(Cl)c1Cl N1(C(c2cccc(C)c2)=O)CC(NC(C23CCC(CC2)CC3)=O)C2CCCC2C1 C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(c1snc(Cl)c1Cl)=O C1(C(=O)NCCC2CCCN(C(=O)CCc3nncs3)C2)CC2CCC(C1)C2 c1(CC(=O)NC2CC(CCNC(=O)CC3CC3)C2)cn2cc(Cl)cc(Cl)c2n1 N1(C(C2N(C(C)C)CCCC2)=O)C2CCC1CN(C(=O)C(O)C1CCC1)C2 N1(C(C=CC=CC(=O)OC)=O)CCn2c(CNC(=O)C(F)n3cccn3)nnc2C1 C(CCCCCC(=O)NC1CCN(C(c2cc(C)c(C)nn2)=O)CC1CO)SC N1(CC(=O)NC2CCC(NC(C(C)(C)C)=O)C2)CCCS1(=O)=O N1(C(c2n(C)nc3c2CCC3)=O)CCC2C1CCCN2c1ncncc1F c1(-c2cn(C(C)C(N3CCOC4CC34)=O)nn2)cccc2[nH]ccc12 C1(C(N(CCOCC=C)C)=O)CN(C)CCN1C(=O)CC(C)(O)C=C C12(CNC(C(CCOC)C)=O)CC(NC(=O)CC(C)C(C)C)(C1)C(C)O2 N1(C(CCCOCC=C)=O)CC2(CCCC2NC(=O)C=C2CN3CCC2CC3)C1 c1(OC)cccc2[nH]cc(CC(N3CC(NC(C4CSC4)=O)CC3C)=O)c12 C(c1cccc(O)c1)=CC(N1CCC(NC(c2c(CC)nc(C)o2)=O)C1)=O c1(C(=O)NCC#CC(=O)NCC(F)C2CCC2)cncc2[nH]ccc12 C1(NC(=O)NCC2C(c3ccc(Br)cc3)(C)C2)CCCC2OCCC12 C1(OC)CN(C(=O)Cc2ccc(C)o2)CC1NC(C1CCCN1C(=O)C1CC1)=O O=C1CC(C(=O)NCc2ccc(C(=O)N(C3CC3)CC3CCOC3)nc2)=NN1 c1(OCCC(C)C)cccc(C(=O)NC2CC(C(=O)NC(=O)C(C)(C)C)C2)c1F c1(C(=O)NCC(=O)NCc2ccco2)cccc(-n2cncn2)n1 c1(C(=O)NCCN(C(C2CCSC(C)C2)=O)CC)coc(C#N)c1 c1(OC)cccc2[nH]cc(C(=O)NC3CCC(NC(c4ccccc4I)=O)C3)c12 N1(C(c2n(CC=C)ccn2)=O)CCCC(C2CCCN(C(=O)C(F)OC)C2)C1 c1(C(=O)NCC(CC=C)NC(=O)CC(C)n2cccn2)cc2c(C)cccc2o1 C(=O)(C(O)CC(C)(C)C)Nc1n(CC)nc(-c2ccccc2)c1 c1(CCC(=O)NCC2C(NC(CC3(OC)CC3)=O)C2)nc(C)c(C)[nH]1 c1(C(=O)NC2(C)CC(NC(C3(CCC)CCNC3=O)=O)C2)ccc(C#N)cc1C C(=O)(C(C)(C)C(F)(F)F)N1CC(CCCC(=O)NC2C3(CC(OCC)C3)C2)C1 C1(NC(CSCCC)=O)CN(C(c2cc(OC)cc(Cl)c2F)=O)CC12CCC2 c1(CNC(C(C(CC)O)C)=O)c(C)nn2c1CN(C(c1cn(CC)cn1)=O)CC2 C1(C(=O)NC2CC(C)(NC(CC3CCC(C)CC3)=O)C2)C2C3CCC(C3)C12 C(=O)(C1=CC2CCC(C1)C2)NCC(C(=O)N(CC(C)C)CC(C)C)CC1CC1 C(=O)(CC1CS(=O)(=O)c2ccccc21)N(C1CCN(C(C)=O)CC1)CCO C1(NC(c2c(C(F)F)c[nH]c2C2CC2)=O)CN(C(=O)C2=COCC2)C2(CCOC2)C1 C1(NC(=O)OC(C)(C)C)CC12CCC(C(=O)NCc1n[nH]cc1C1CC1)CC2 N=c1cc(C(=O)NC2CCC(NC(=O)Cn3cccn3)C2)c(Br)c[nH]1 C1(NC(CN(CCOC)C)=O)CC12CCN(C(c1csc(C(C)C)n1)=O)CC2 c1(C(=O)NCC(=O)N(CCNC(C(CC)N2CCCC2=O)=O)C)ccccc1C N(C1CCCc2c1cnn2C)C(C1CCC(F)(CC(C)C)C1)=O c1(OC)cc(C(=O)NC(CNC(=O)C(C)SC)CC(F)(F)F)ccc1Cl C1(C(=O)NC2CC(F)(F)C2)CN(C(c2cccc(F)c2O)=O)CCC1O c1(CCC)ncoc1C(=O)NC(C)(C)CCNC(=O)C(F)OC(F)(F)F C1(C2CN(C(CC(C)N(C3CC3)C)=O)C2)CCCCN1C(=O)CN1CCCCC1 C1(NC(c2cnc(C3CC3)nc2)=O)CN(C(C2CC2F)=O)CC2(CCC2)C1 C(=O)(C(C)CN(C)N1CCOC2(CCCN(c3nc(C)ns3)C2)C1)OC C1(O)(CNC(c2c(C)noc2C)=O)CCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 C1(CNC(C(C)NS(C)(=O)=O)=O)CC2(CCOCC2)CN1C(=O)C(F)(F)CO N1(C(C(CCC)C)=O)CCN(C(c2ccc(Cl)cc2NC(C)C)=O)CC1C Cc1cccc(O)c1C(=O)NC1CC1CNC(c1cc(C)n(C2CC2)n1)=O N1(C(c2scc(COC)c2)=O)CC(CNC(=O)Cc2nccn2C)C(O)C1 c1(CC)cc(C(=O)Cn2nccn2)ccc1C(=O)NC1CCC(C)(CN)C1.OC c1(C(C)(C)C)ccnc(C(=O)NCC2CCCC2C(=O)NC2CCC(CO)O2)c1 C1(C(N(CC(=C)C)C)=O)CC12CCN(C(c1ccnc(OC)n1)=O)CC2 N1(C(C2CN(C(C(CCC)C#N)=O)C(C)(C)C2)=O)CCC2OCCC2C1 c1(C(=O)NCC2C(CNC(c3nc(C)nc(O)c3)=O)C2)nc2nccc(C)n2n1 CC1(C)CCC(C(=O)NCC2(O)CCN(C(=O)CCc3cnoc3)C2)CO1 c1(OC)cc(OC)c(C(=O)N(CC(=O)O)C2CC2)cc1OC C12(C(=O)NCc3c(C(=O)NC(C(=O)OC)CO)n(C)nn3)CCCC1C2(F)F C1(O)(CCNC(=O)CCC2CC2)CCN(C(=O)Cc2c(Cl)cccc2Cl)CC1 C(=O)(C(COC)CC(C)C)NC1C(CN(C(CCCCC#C)=O)C)CCC1 C1(N(C(C2C(=C)CC2)=O)C)CCC2CN(C(c3cc(S(=O)(=O)NC)co3)=O)CC12 N1(C(C2(CCN(C)C)CC2)=O)CC2CCC1C1CN(c3nnco3)CC21 CCC1=C(C(=O)NCCCCNC(=O)CCOc2ccccc2)CCCO1 C=CC1(CC(N2CCCC(OCCNC(=O)CNC(=O)OC)C2)=O)CCCCC1 c1(C(=O)NCCC(C)NC(=O)Cc2nc[nH]n2)csc(-c2ncc[nH]2)n1 N1(C(C2(OC)CCN(C(C3CC4CCC3O4)=O)CC2)=O)CCCC2CC1C2(C)C C(C1=NOC2CN(C(C3(c4c[nH]nc4OC)CC3)=O)CC12)NC(CCC(=C)Cl)=O c1(N(C)Cc2cnc3c(c2)CCC3)nc2c(c(=NCc3cnn[nH]3)[nH]1)SCC2 N1(c2nccc(C(=O)OC)n2)CC(C(N2CC3CNCC3C2)=O)CC(F)C1 Brc1ccc2c(c1)OCCN2Cc1cnc2n1CCC2 C1(CN(C(=O)C(F)OC(F)(F)F)CC)CCCN1C(=O)CCN(C)C(C)=O C1(C(=O)NCC2CN(Cc3ccccc3)CCO2)CCOCC12CCCCC2 C1(C(N(CCOCCC(=O)NC(C(=O)OC)C)C)=O)COC(C)C1 C1(CC(=O)N(c2cccc(CC)c2)C)CC2C=CC1C2.C12CC(C1)NC2=O O=C(CCC(=O)c1ccc(Br)cc1)N(C1CCOCC1)CCCO C(C(C)(C)C#CC(=O)NC1(CO)CC2CCCC12)NC(c1nc(C)oc1)=O C(CCC(C)(C)C(=O)N(C)Cc1nccn1C)NC(CC(CC)CC)=O C1(C(=O)NC(CCC)C(=O)N(C)C)CCCCCN1C(=O)CS(=O)CC C1(CCC)CCN(C(=O)C(C2(O)CCCCC2)NC(=O)CN(C)CC)CC1 N1(C(c2ccc(-c3scc(C)c3)cc2)=O)CCCCC2(CCN(C(=O)CO)C2)C1 c1(C(=O)NCC(CC)NC(C2(O)CCCCCC2)=O)cc(C)cc(Br)c1 Cc1ncn(C)c(=O)c1C(=O)NCCC1(O)CN(C(C2CC3CCC2O3)=O)C1 c1(C(=O)NC2CN(C(C(C3CCC3)OC)=O)CC2O)ccc(F)c2ccccc12 c1(CC)cc(C(N2CC3C(CNC(=O)C(C)(CC)CO)C3C2)=O)ccc1O C1(NC(=O)NCCOC)CCC(C)(C)N(C(=O)OC(C)(C)C)C1.C1C(C)C(=O)O1 c1(C(=O)NC(C2CCCN(C(C3CC(C#N)C3)=O)C2)C)cnc2c(c1)CCC2 N1(C(C(CCNC(C2(CC=C)CC=CC2)=O)OC)=O)CCc2ccccc2C1 N#Cc1ccc(N)c(C(N2CCCN(C(=O)CCS(N)(=O)=O)CC2)=O)c1 C=CC1(C(N2CCC(CC(C)C)CC2)=O)CCN(C(c2ccnc(C)c2)=O)CC1 C(=O)(C1CCc2snnc21)NC(CCCNC(CCNS(C)(=O)=O)=O)(C)C C(=O)(CCCCC(=O)N1CCCC1CCNC(C1(C)CC1(Cl)Cl)=O)OC C12CCN(CC1)C(=O)n1nnnc1C(c1cc(C)on1)NN2CC1CC1.CC.CC N1(C(c2c(NC(C)=O)cccn2)=O)CCCC12CCN(C(C1CC(F)C1)=O)C2.C(=O)C=O CC(CNC(c1cc(C(F)F)[nH]n1)=O)C(F)C(=O)NC1(C)CCCC1O C1(C(N(C(C)C(=O)NC23CSCC2C3)C(C2CC2)C)=O)(CO)CCCO1 c1(C(N2CCN(C(c3cc(CCC)oc3C)=O)CC2)=O)ccc(S(C)(=O)=O)cc1 C1(NC(c2ccn(CCOC)n2)=O)CC2CC1N(C(c1cnn(CCF)c1)=O)C2 N1(C(=O)OC(C)(C)C)CCC1CCCNC(CCCC1CCCO1)=O C=CCC(C)(C)C(=O)N1CCC(C(=O)NCc2cc(O)ccc2O)C1 c1(C(N2CC(NC(c3[nH]nc(OC)c3Cl)=O)(CO)C2)=O)nnc2ccccc2n1 CC(C)(O)C(C)(CO)NC(C1C2CCN(C(=O)CCc3cnco3)CC12)=O c1(C(N2CC(C(C)NC(c3ccoc3Br)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl c1(C(=O)NC23CCN(C(C=Cc4nc(C)sc4)=O)CC2C3)cc(N)c(Cl)c(O)c1 C1(F)(COC)COC1.C(CC(=O)NCO)N1C(=O)CC2(CC2)OCC1 N1(C(C(CC=CC)CC)=O)CC(O)(C2(CNC(c3cccc(SC)c3)=O)CC2)C1 c1(COC(C(C)C(C)c2ccccc2Cl)=O)cn2ccccc2n1 c1(C(C)C)ncc(C(=O)N(C(C)CNC(=O)C(C)C2CC2)C)s1 n1(CC(=O)NCC2CC(NC(C3CN(CC(C)C)C3)=O)C2)ncc(O)nc1=O N1(C(C=C(C)C2CCCCC2)=O)CC(NC(=O)CCc2nccs2)CC(C)(C)C1 Nc1c(C(=O)NCCCNC(c2ccnc(OCCO)c2)=O)sc2ncccc12 C1(C(=O)NCC(C)O)CCC2(CN(C(c3ccn(C)c3)=O)C2)O1 CCC(C)C(C)N=c1[nH]c(C(N2CCOC(Cn3cc(C(C)O)nn3)C2)=O)cs1 C1(CNC(C=CC(CC)=CC)=O)CN(C(=O)CNC(C2CCCC2)=O)CC1C C1(C2CCN(C(=O)C(C)(C)C(C)(C)O)CC2)(NC(C(C=CCCC)O)=O)CC1 N1(C(CCC=C)=O)CCN(C(c2nccc(C(F)(F)F)n2)=O)C(C2CC2)C1 c1(C(=O)NC2C3CN(C(CCSCCCC)=O)C(C3)C2)cc(F)c(F)c(F)c1 c1(C(N2C3C(CNC(CC4(OC)CCC4)=O)C(C3)C2)=O)cnc2[nH]cnc2c1 CC1COC(C(F)(F)F)CN1C(=O)NC1CCC2(CC2)C1 c1(C(=O)NCCC(C)(C)NC(C(C)NC(CC)=O)=O)ccnn2ccnc12 CC(C)C(C(=O)N1CCC(NC(=O)C(O)C2CCCC2)CC1)n1cccc1 S(=O)(=O)(c1cccnc1NCCOCC1CCCC1)NC1C2CC(OC)C(C2)C1 N1(C(c2nc(CC)oc2)=O)CCC(CC(N2CCOCC2)=O)CC1 C=CC(C)(O)CC(=O)NCCN(C(c1ccc2c(c1)CC2)=O)CC1CC1 c1(OC)cc(C(=O)N(CC(C)(C)CNC(=O)Cc2ccc(F)cn2)C)ccn1 CC1(C)COCC(C(N2CC(CNC(c3nn[nH]c3Cl)=O)C(F)(F)C2)=O)O1 c1(CCC)nc2cc(C(N3CCC34CN(C(C3CC3(C)C)=O)C4)=O)cc(C)c2[nH]1 C1(C2CC2)(NC(=O)CCc2ccsc2)CCN(C(C2CCNC2=O)=O)C1 c1(OC)cccc(OCc2cc(C)on2)c1N(C)C(=O)NCCCC(C)C C1(CC(=O)OC)CCCC(NC(C2CC(C(F)F)(NC(=O)OC(C)(C)C)C2)=O)C1 Cc1cn(C)cc1C(=O)NC(C)CN1CCN(C(C2(CN(C)C)CC2)=O)CC1 C(C(=O)NC1CCC1NC(=O)CCOC(C)C)(C(C)C)n1ncc(C)c1 N1(C(c2cc(CN(C)C)ncc2)=O)CCCCCC1CNC(C1(C)CC1(C)C)=O O=C(CN1CCCC(O)(c2cnn[nH]2)C1)C1Cc2ccccc21 Cc1ccc([N+](=O)[O-])cc1C(N1CC(NC(c2ccc(Br)c(F)c2)=O)C(F)C1)=O CS(=O)(=O)c1ccc(NC(=O)Cc2csc(-c3ccsc3)n2)nc1 CC1(C)OCc2cc(C(N3CCOCC3CNC(=O)Cc3ccon3)=O)ccc21 C(C(F)(F)CCC(=O)NCCCNC)n1cc(C2(C(=O)OC)CC2)nn1 c1(CNC(CC(C)N(C)C)=O)cccc(NC(=O)CSc2ccccc2Cl)c1 N1(C(C2CCN(C(CC(C)C3CC3)=O)CC2)=O)CCC12CCC(O)CC2 C(CC(CC)C(=O)N1CCCCC1CCN(C(=O)COCCOCCO)C)=CC Cc1ccc(CNC(=O)C(Cc2ccoc2)NC(=O)CCc2cn[nH]c2)o1 CC(C)(C)C(O)C(=O)NCC1CN(CC(N2CCCCC2CO)=O)CCCO1 C1(C(N2C(C)(CC(N3CCC(CC(F)F)C3)=O)CC2)=O)CC2CC(=O)C1O2 CC1N(C(C2C3CCC(C3)N2C(C2CCC2C#N)=O)=O)CCC1(C)C CC1CN(C(C2(c3cccc(F)c3)CC2)=O)CC1CNC(c1ncn(C)n1)=O c1(C(=O)OC2CN(S(=O)(=O)C(F)(F)F)C2)cccc(I)c1Cl C(=O)(C1=NOC2COCC12)C(N1C(C(N2CCC(N)C(O)C2)=O)CCC1)=O N1(C(C(CCCOC)C)=O)CC2(CCCCN2C(c2snnc2C)=O)C1 C(C)(CCC(=O)NCC(c1ccccc1)NC(c1cc(C)nn1CCO)=O)OC C1(N(C(CCCN(C)C)=O)C)CN(C(C2C(Cl)(Cl)C23CC3)=O)CC12CC2 c1(CSC)cc(C(=O)N(C)CC2CCCN2c2nccc(CO)n2)sc1C NS(=O)(=O)c1ccc(C(=O)NC2CCN(C(C3CCOC3)=O)CC2F)cc1 C1(NC(C2SCCS2)=O)CCC12CN(C(=O)Cc1ccccc1F)C2 CC(C)C(O)CC(=O)NCC1(NC(C2(CCCCO)CC2)=O)CC1.C(=O)O c1(C(N(CCOCCNC(C=C(CCC)CCC)=O)C)=O)ccc2c(n1)CCC2 N1(C(c2n[nH]c3c2CC(C)CC3)=O)CC2CCN(C(=O)CC(C)(C)C)CC(C2)C1 N1(C(C=Cc2c(C)n(C)nc2)=O)CCCN(C(=O)C2=COCCC2)CC1C c1(C(N2CC(C)(NC(c3ccc(-n4cccc4)nc3)=O)C2)=O)cc(=O)cc(Cl)[nH]1 C1(NC(c2c(OCC)scc2)=O)CCN(C(c2ccc(OCC)cn2)=O)CC1F CCC1C(=O)Nc2ccc(C(=O)N(CC(C)N(C)C(c3cn(C)nn3)=O)C)cc21 C(C)(N=c1nc(N2CC3CC3C2)c2c([nH]1)CCS2)c1c(C)noc1C CC1(C)CC(CC(=O)NCCC(F)(F)F)CN1C(=O)C=CC(F)F C1(NC(C2(OCC)CC2)=O)CC1C1CCN(C(C2CCCN2CC)=O)CC1 C(CC(C(=O)N1CCC(COC)CC1)NC(=O)CC1CCC(=O)CC1)OCC O=C1CCN(CC(=O)NCCC2CN(C(c3cc(Cl)ccc3Cl)=O)C2)C(=O)N1 C(CCCCC(=O)NC(C)C(CO)NC(c1ccc(C(C)C)c(Cl)c1)=O)SC N1(C(C(CC)SC)=O)CC2CC(N(C(=O)CC3CCN(S(C)(=O)=O)CC3)CC)C1C2 C1(O)(CN(C(=O)C(F)n2ccnc2)C)CN(C(=O)CCc2cncs2)C1 N1(C(C(C)C)=O)CCC2CCC(NC(=O)C(C(C)C)n3cnnc3)C1C2 c1(CC(=O)NCCNC(c2c(N(C)C)cc(Br)cn2)=O)cc(Br)cc2c1OCC2 c1(C(N2C3CN(Cc4c(OC)c(Cl)ccc4)C(C3)C2)=O)ccc(F)c(F)c1O C(c1ccccc1F)=CCC(=O)NCC1(O)CCN(C(=O)CC2COC(=O)N2)C1 N1(C(=O)COC(F)F)CCC(O)(CCNC(c2cn(C3CCCC3)cn2)=O)C1 C1(NC(=O)CCn2ccnn2)CN(C(=O)Cn2ncnn2)CC12CCC2 c1(OC(c2cc(C=O)on2)C)ccn(C)n1.N12CCC(C1)OCC2=O.C1(O)CCC1 c1(C(=O)NC2(CNC(c3cn(CCC=C)nn3)=O)CCCC2)ccc(C)cc1C c1(OC)nc(C(=O)NCC2CN(C)CCN2C(c2cc(Cl)no2)=O)cc(O)n1 c1(C(=O)NCCC2(O)CN(C(C3(CC)CC3(F)F)=O)C2)cc2[nH]nc(C)c2cn1 C1(F)(CNC(=O)CSCn2cncn2)CCN(C(=O)CSC2CCOC2=O)C1 C1(NC(Cn2c(C)ccn2)=O)CCCCC12CCN(C(=O)C(C)(C)N(C)C)C2 N1(C(C2CC(C)=C(C)CC2)=O)CCC(NC(=O)C2=CCC2)C(C)(C)C1 O=C(C(O)C1=CCCCC1)N1CC(C(N2CCCC23CCCCC3)=O)C(F)(F)C1 c1(CNC(=O)C(=O)NCC(CO)C2CCCC2)ccc(Br)cc1 N1(C(c2c(C)noc2C(C)C)=O)CCCC2CN(C(c3occc3F)=O)CCC12 c1(C(=O)NCC2(O)CC(NC(C3CC(=C)C3)=O)C2)sc2ccc(C)cc2c1C c1(C(=O)N(C2(C(N3CCC(F)(F)CC3)=O)CCC2)C2CC2)nnc(O)nc1O C1(C(=O)NC2CC(NC(C3CC(C(=O)OC)C3)=O)C2)Cc2nn[nH]c2C(C)C1 C1(COC(Cc2cccc(OC)c2)=O)CC(C)(C)CC(C)(C)C1 Nc1cc(Cl)cc(Cl)c1C(N1CC2CCC1CN2C(C1CCCC12CC2)=O)=O N1(C(c2ccc(Br)cn2)=O)CC2CCC2(C(=O)NC2CCC(F)(F)CC2)C1 CC(C)(C(c1nnnn1CC(F)F)NCCC(N)=O)c1ccncc1 c1(OCc2n(CC)ncn2)cnccc1SC.C(CC(C)(C)OC)=CC(=O)N c1(OC)ccc2oc3c(c2c1)CCCC3NCc1cnc(C)cn1 C1(C)(CNC(C2CCCN(c3c(C)cccn3)C2)=O)COC(C)(C)CO1 C1(CC(N2CCC(c3cn(CCCC)nn3)C2)=O)CCN(C)CC1 N#Cc1ccc(N2CCN(c3ccnnc3)CC2)cc1C(F)(F)F c1(C(=O)NC2CN(C(C(C)CF)=O)CC(C)(C)C2)c2c(nn1C)CCSC2 C1(NC(CCN(S(C)(=O)=O)C)=O)CN(C(=O)CC2CSCCO2)CC1CO C1(OC)CN(C(c2cnncc2C)=O)CC1C(N1CC(O)C1(C)C)=O c1(NC(C(n2cc(C(C)(C)C(=O)OC(C)(C)C)nn2)C)=O)cnn(C)c1S(N)(=O)=O CS(=O)C=CC(=O)NCCOCCn1cc(NC(=O)CC2CCCNC2=O)nn1 n1(CC)nnc2c(N3CCC(NC(=O)CSc4ccccc4)C(C)C3)ncnc12 C=CC1(NC(=O)CC2CCCN(C(=O)CC3CCOC3C)C2)CCCC1 c1(C(N(CCCNC(C2CC(C#N)(OC)C2)=O)C)=O)c[nH]c(=O)c2ccnn12 C1(NC(c2c(OC)scc2)=O)CC2(CCCN(C(c3ccc(O)nc3Cl)=O)C2)C1 CC1(CC(=O)NC2CC(CNC(c3c[nH]cc3CC3CC3)=O)C2)CCCO1 C1(NC(=O)CCCO)CC2CC(C1)N(C(=O)CNCCCOc1ccccn1)C2 N1(C(c2cc(SC)oc2C)=O)CCCN(C(c2cn(C)nc2Cl)=O)CCC1 c1(OC)ccc(C(=O)NC2CC(C)N(C(C3CCCC(=O)N3)=O)C2)nc1Cl N1(C(C(C)CN(C)C)=O)CCN(C(c2cc(C3CCC3)on2)=O)CC(C)(C)C1 c1(N(CCC)CCNC(c2ccnc(C)c2)=O)cc(C)ccc1[N+](=O)[O-] C1(C)(C(=O)NCC2(O)CN(C(c3c(COC)nn(C)c3)=O)C2)CCCCNC1=O C1(NC(c2c(CC)cno2)=O)CCCCC1NC(=O)Cn1cccc1 CC1(C)CC(CNC(C2CC(C(C)(C)C)C2)=O)N(C(C2CCOC2(C)C)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)CCCNC(N)=O)N1CCN(CC)CC1C c1(C(N2C(C)(CC)CC(NC(c3n[nH]cc3C)=O)C2)=O)cc(S(N)(=O)=O)cs1 N1(C(CCC(=C)C)=O)CCC(NC(=O)C(C)OCCc2ccccc2)CC(O)C1 O=C1OCC2CN(CCc3ccc(Cc4ccccc4)cc3)CCC12 CC1(C)CCCOC1C(=O)NCCCC(=O)NCC1C2CCCCC12 C(=O)(CCC(=O)N(C)C)NC(C)C(CO)NC(C1CC(=O)N(O)C1)=O C1(NC(C=C(C)c2cccs2)=O)CN(C(=O)CC2CN(C)C2)Cc2ccnn2C1 C(=O)(CCCS(C)(=O)=O)NC(C)C(CO)NC(c1cc(-c2ccccc2)co1)=O c1(NC(C(N2CCC(C)(CC#N)C2)=O)=O)cc(Br)c(F)cc1Cl CC1CCCCCCN1C(c1coc2c1CN(C(c1cn(C3CC3)nn1)=O)C2)=O C(=O)(C(C)(C)C(C)O)N1CCC(C)(C(=O)NC(C)Cc2cnccn2)C1 N(C(=NCC(F)(F)Cl)NCc1ccccc1)CC(C)(C)F c1(C(N2CCC(NC(COCCCC#C)=O)C(CC)C2)=O)ncnc2ccsc12 C1(COC)CN(C(=O)CC=C(C)C)CCN1C(=O)C(c1ccc(Cl)cc1)C N(C1CN(c2cccc(F)c2C#N)CCc2ccccc21)C(COC(CC)C)=O C(=O)(C#CC1CCCCC1)NCC(CC)NC(Cc1c(CC)con1)=O C1(NC(Cc2cc(OC)no2)=O)(CNC(=O)CC(C)OC)CCCCC1C CCC(C)C(=O)NCC(=O)NCCCNC(c1cc[nH]c1C)=O CC1CCC(NC(=O)C(C)(C)c2cnc[nH]2)CN1C(c1cnco1)=O N1(C(c2c(CNC(C3(CC)CCCO3)=O)nnn2C)=O)CC23CCC2(COC3)C1 C1(F)(CNC(C(Br)=C(C)C)=O)CCC(NC(=O)Cn2cc(C(C)O)nn2)C1 C1(C)(CNC(c2n(C)ncc2)=O)COCCN(C(=O)Cc2csc(Cl)n2)C1 c1(N2CCCC(C(C)C)C2)nc(N2CC3CC3C2)c2c(n1)CCC(C)C2 N12CCC(C)(C1)C2=O.c1(C(=O)NC(CC)CSC)ccsc1C(C)C c1(CCCNC(C(=O)NCc2ncc(CC)o2)=O)ccc(N2CCOC2=O)cc1 c1(C(=O)NC2CCN(C(C3CC4C=CC3C4)=O)CC2)ccn2ncnc2c1 C(C1CCOC1)=CC(=O)NCC1(O)CC(CNC(C2CNC(=O)N2)=O)C1 Cc1ncc2n1CCC(C(=O)NCC1CN(C(=O)COCCO)CCC1(C)C)C2 O=C1CN(Cc2cccc(F)c2)C(=O)N1C1CCN(C(=O)Nc2ccccc2)C1 Cc1nc(COCCC(=O)NCC2CC(NC(c3cnoc3C)=O)C2)cs1 CC1CC(NC(c2c(C3CCC3)cnn2C)=O)CN1C(=O)C(C1CCC(=O)N1)C N1(C(c2c(CC)cns2)=O)CCC(F)(CNC(C2(C(C)C)CCCO2)=O)CC1 c1(C(N2CC(CC)N(C(C3C(F)(F)C34CC4)=O)CC2)=O)cn2ccc(C)cc2n1 C1(O)(COC)CCN(C(=O)C(C2CCCO2)NC(=O)C=C(C)C)C1 Nc1cc(C(N2CC3CC(NC(c4coc(O)n4)=O)C3C2)=O)cc(O)c1Cl c1(C(N(C2CN(C(C3CCCC3O)=O)C2)C)=O)cc(C2CCC2)no1 Cc1ccc2c(=NCCNC(N)=O)[nH]c(N3C4CNC(=O)CC3COC4)nc2c1 N1(C(C(CC)F)=O)Cc2ccc(CNC(c3cncn3C3CC3)=O)cc2C1 C1(CNC(CC2(C)CC2)=O)CN2CCCCC2CN1C(C1CN2CCC1CC2)=O N1(C(C(C)N2CCCC2)=O)CCC(NC(C2(C)CCSCC2)=O)C(C)C1 n1(CC(=O)NC(C2CCCN(C(c3cc(C(C)(F)F)on3)=O)C2)C)ncccc1=O C=CCC(CNC(=O)C=C(C)CCC)C(=O)NCC(C)(C)CCCO C1(COC(=O)CC2(NC(C(=O)NC3CC3)=O)CCC2)C=CCOC1 C1(C(N(CC(CN(C)Cc2cc(C#N)ccc2F)O)C)=O)CCC2(C1)CC2(F)F N1(C(C2CC(C)(NC(C3N(CC)CCC3)=O)C2)=O)CC=CC(O)C1 c1(CN(C)C(C2(C(F)F)CC2)=O)cccc(CNC(=O)CC2CC(O)C2(C)C)c1 n1(CC)cnc2[nH]c(=NCCN3CCCOCC3)nc(N3CCCC(C)C3)c12 c1(C(N2C(C(C)(C)NC(C(CCCC)O)=O)CCC2)=O)cc2sccc2cn1 c1(C(=O)NCC(C)N(C)C(c2c[nH]nc2C(F)(F)F)=O)cccc(C2CCC2)c1 N1(C(C=CCCC)=O)CCN(C(=O)C(CC(C)C)NC(=O)OC(C)C)CCC1C C=CCC(C(=O)NCc1cncc(OC)n1)NC(=O)Cn1[nH]cnc1=N Cc1c(C(=O)NC2CC(O)CN(C(=O)C#CC(C)(C)C)C2)sc2cncn12 C1(C(=O)NCCCN(C(c2c(C)coc2)=O)C(C)C)CCCN(CC(C)C)C1 N1(C(C2CCN(C)C(=O)C2)=O)CCC2(CCCN2C(=O)C(Cl)=CCl)CC1 C1(C(=O)NC(CCC)(C)CC)CCC2(CC2)N1C(c1c[nH]nc1C)=O Cc1cc(F)cc(C(N2CC3CC(NC(c4ccon4)=O)CC3C2)=O)c1O N1(C(C2N(CC)CC2)=O)CCC2CCC(NC(c3cccc4[nH]ncc34)=O)C1C2 c1(NC(C2CCOCC2)CC)ccc(S(=O)(=O)NC(C)C(C)(C)OC)cc1Br C1(CC(=O)NC(C)Cc2nnc(C(CCl)OC(=N)O)s2)COCC(C)O1 Cc1ccc(CN2CCN(C(C3CCCCN3CC(F)F)=O)CC2)c(C)c1 C(=O)(C1=CCCOCC1)N1CCC2C(C(N3C(C)CC(O)CC3)=O)C2C1 c1(C(=O)NC2(CC=C)CCN(C(=O)C=CC)C2)cc(OC)cc2c1OCC2 CCC(C)(C)C(O)C(=O)N(CC(C)C(N1CCN(CC2CC2)CC1)=O)C N1(C(C)=O)CCC2(C(=O)N(S(=O)(=O)Cc3cccc(Cl)c3)C(C)(C)C)CC2C1 C(=O)(C(F)CCC(C)(C)C)NC1C(F)CCN(C(C2C(C)=CC2)=O)C1 C1(OC)CC(CCNC(=O)COCCOC)N(C(=O)C=C2CCCC2)C1 CCC(C)CC(C(=O)N(C1CCCC1C)C)NC(=O)CC(C)C1CC1 Cc1cn2cccc(C(=O)NC3(C)CN(c4nc5ccc(N)cc5s4)C3)c2n1 c1(OC)ccc(C(=O)NCc2n[nH]cc2C(=O)NCc2ncon2)cc1 c1(NC(=O)Nc2c(C)cc(N3CCN(C)CC3)cc2)noc2cc(Cl)ccc12 CCC(CO)C(=O)N1CC(=C(F)CNC(C2CCCS2)=O)C1 C=C(C)C(C)(C)C(=O)NC(CNC(c1cnc(C2CC2)s1)=O)CC(C)C c1(C(N2CCCC(NC(C(C(C)C)SCC)=O)CC2)=O)cc2c(ccn2C)[nH]1 N12CCN(CC1)C(=O)CC(=O)NC(C)(C)C2=O.C=C1CC(C)(c2nn[nH]n2)C1 C(=O)(C#CC1CCOCC1)N1CC(O)(C(C)NC(C2(C)CCCC2(F)F)=O)C1 c1(C(=O)NCCN(C(c2cc3n(c2)CCSC3)=O)CC)c(N)cccc1[N+](=O)[O-] c1(C(=O)NCC2C(NC(C3N(C)CCOC3)=O)CC2)ncc(Cl)cc1O CCC(CC(=O)NC1(CCCC(=O)N(CCC(=O)NC)C)CCC1)SC Cc1nc(C(N2CC=CC2CNC(=O)CC2CCCC(O)C2)=O)sc1C Cc1cccc(Br)c1C(C(=O)NC1CC2CC1CC2=O)NC(=O)COC(C)C C1(NC(CSCCC)=O)CCOC12CCN(C(=O)Cc1cnc(C3CC3)[nH]1)CC2 c1(C(N2C3CC(NC(CN(C)CC)=O)C(CC3)C2)=O)cc(F)c(C#N)c(F)c1 c1(OCC)cc(NC(=O)C(C)(C)C)c2cc1OC2.C1(C)(CNC)CNCCC1O C1(C)(C(N(C2CCN(C(c3ccc(N)cn3)=O)CC2)C)=O)CCC(=O)N1 S(=O)(=O)(c1cc(C(=O)OC)ccn1)NC(C1CCOCC1)C(=O)OC C(CC(=O)N1C(C)C(=O)C1CC)(CC(C)C)NC(C(COCC)C)=O.OC C1(C2CC2)(C(=O)NC(CCCC)CC)CN(C(=O)C(CC2CC2)OC)C1 n1(CCOC)ccc2c(C(=O)NC(C)CN(C(=O)CCCC3CC3)C)cccc12 n1(CC)nc(C)c(=NCCN2CCN(C(C)CNC)CC2)[nH]1 N1(C(c2c(C)[nH]nc2Cl)=O)CC2(C1)CN(C(C1CC=CCC1)=O)CCO2 c1(N(C)CCc2ccccc2)nc(N2CCC(COC(F)F)C2)c2sccc2n1 CC(O)CCCCCC(=O)N(CC(O)CN(C)C(c1ccc2c(n1)CCC2)=O)C c1(C(=O)NC2CN(C(=O)C=CBr)CC23CC3)cccc2[nH]cc(Cl)c12 c1(C(=O)NCC2N(C(c3c(C)nc(C)o3)=O)CCCC2)cncc(C)c1Cl C=CCC(CC(=O)NC1CCOC(C)(CC)C1)NC(c1cnn(CCF)c1)=O C1(C(=O)NCCN(C)C)CC12CCN(C(=O)C(c1ccccc1)O)CC2 C1(C(N(CC(CC)NC(=O)COCC(=O)OC)C)=O)COC(=O)N1 c1(C(N2CCC(OCCNC(C(C)OCCCC)=O)C2)=O)ncnc(O)c1F N1(C(CC2(COC)CCCC2)=O)CC2CCC1C1CN(C(=O)C(F)OC)CC21 N1(CC(=O)NCCC(CNC(=O)C(C)C(F)F)OC)CCCCC1C c1(N2CCCC(CN(C(C3(OC)CCCCC3)=O)C)C2)ncnc2c1COC2 C(C(=O)NC1CCC(F)(F)CC1)(C(C)CC(C)(C)C)N(CCC=C)CC S(=O)(=O)(c1ccc(S(=O)(=O)COCCO)cn1)N1CCCC(C)(SC)C1 C1(NC(C(CC)(C)O)=O)CC2CC(NC(C3CN4CCN3CC4)=O)CC2C1 c1(C(=O)NCC(CNC(C2C(C(C)C)C2)=O)(C)C)ccccc1CCC(F)(F)F C1(NC(C2CC23CC3)=O)CCN(C(=O)C=Cc2ccc(Cl)cc2)CC12CCC2 C(=O)(CCCCC(F)F)N1CCC(CNC(C(C2CCCCC2)OC)=O)C1(C)C N1(C(c2nnc(C)s2)=O)CCC(NC(=O)C(C)Oc2ccccc2C)C1(C)C c1(C(N2C(C)(C(=O)NCCC(CCC)O)CCC2)=O)cc(C)cc(O)n1 C(CCc1cnn(C)c1)(C(=O)NCc1nnn(C)n1)N(CCC(=O)OC)C1CC1 CS(=O)(=O)c1nccc(N(Cc2c(Cl)ccnc2Br)CC2CCCNC2)n1 Cc1cn2cc(C(N3CCCOC(CNC(C45CCCC4C5)=O)C3)=O)nc2s1 c1(N(C)C)ccccc1C(N1CC(OCC(=O)NC2CC(NC(N)=O)C2)C1)=O Cc1cnc2ccc(C(=O)NC3CC(NC(=O)CCC(C)S(C)(=O)=O)C3)cn12 C1(C(CC)O)CCCCN1C(=O)Cc1ccc(NC(c2cnsc2)=O)cn1 N1(C(CC2CCC(=O)C2)=O)CC2CCCC(NC(C34CCC(CC3)OC4)=O)C2C1 N1(C(C(C)NC(=O)C(C)NC(=O)C2CC2)=O)CCC(F)(CNC(C)=O)C1 c1(SC)cccc(Br)c1CC(=O)NCC(C)(CC(C)C)NC(=O)C(C)O CC1(C)NC(=O)OC12CCN(C(c1cnc(CN)cn1)=O)CC2 CCCCC(O)C(=O)NC1CN(C(c2cc(N)ccc2SC)=O)CC1F c1(C(CNC(=O)C(C)(C2CCC2)N(C)C)NC(CC2CC(C)C2)=O)cccc(Cl)c1 Cc1ccc([N+](=O)[O-])c(C(=O)NCC(CNC(=O)Cc2cncn2C)CO)c1C CCCCC(C)CCC(=O)N1CCC(CC(=O)N(C2CC(O)C2OC)CC)C1 CC1(C)CC(C)(C(N2CCCCC(CO)C2)=O)CN1C(=O)C1=NOCC1 Cc1nccc(C(N2C(C(=O)Nc3ccc(C(C)C)nc3)CC2C)=O)n1 C12(C(N3CCN(CCN(C)C(C4CC(C)(O)C4)=O)CC3)=O)CCCN1CC(O)C2 C(C)(CC(C)(C)CO)NC(C1N(C(C(C)C2(O)CCC2)=O)CCSC1)=O N1(C(c2cccc(C)n2)=O)CCC2CCCN(C(c3ccccn3)=O)C2C1 C(=O)(CC1CN(C)c2ccccc21)NCC(CC=C)NC(C1CN(C(=O)NC)C1)=O N1(C(=O)Nc2ccc(CCC(=O)OC(C)(C)C)cc2)CCC2(C1)CC(F)(F)C2 c1(CC)cc(C(N2CCN(C(=O)CC(O)CN(C)C)CC2C)=O)ccc1OC c1(C(C2CN(c3cc(C)ncn3)C2)CN2CC(F)(F)C(F)(F)C2)cc(C)c(F)c(F)c1 CCS(=O)c1ccccc1C(=O)NC(CCN(C)C(c1cc(Cl)cs1)=O)C(C)C N1(CC(=O)NCC(=O)N(CC2N(CC)CC2)CC2CCCOC2)CCCCC1C Cc1nc(Br)c(C(N2CCC(CF)(NC(=O)C(C)C3CC3)C2)=O)s1 N1(C(c2c(OC)oc(C)n2)=O)CCC(O)(CN(C)C(c2cnc(C#N)s2)=O)CC1 CC1CN(C(=O)COC2CC2)CC(CCNC(c2ccnc(O)c2Br)=O)O1 Cc1cnc(F)cc1C(=O)NC(C)CCCCN C(CCCCC(=O)NCc1cnc(C)o1)N(C(C(CC)COC)=O)C c1(C(=O)NCC(CCC)NC(=O)C(C)(C)N2CCCC2)sc(F)cc1C c1(C(=O)NC2(CNC(CCCC)=O)CC2)ccc(NC2CC2)cc1C S(=O)(=O)(c1ccc(NCC2CCC3(CCCC3)C2)c2cnccc12)N(C)CCF C=CC1CC(N=c2[nH]c3ccc(Br)cc3s2)CN1CC(C)C C1(NC(c2cc(OC)ncn2)=O)CCN(C(=O)CSCC(=O)NC)C1(C)C C=CC1CN(C(C2CCC(NC(c3coc(CO)c3)=O)CC2)=O)CC1O c1(OC)cc(COCC(=O)NCC2(O)CCN(C(=O)Cc3cncs3)C2)ccn1 c1(CC)ccc2cc(C(=O)NCC3CC3CNC(c3csc(C#N)c3)=O)[nH]c2c1 CCC(C)C(O)C(C)C(=O)N1CCCC1C1(C(=O)NCc2cc(C)ncn2)CC1 Cc1cccn(CC(N2CCC(NC(c3ccc(C(C)C)o3)=O)C(O)C2)=O)c1=O c1(C(c2nnnn2CCSC)NC2CC(=C)C2)ccc(Br)cc1OC(F)F CC#CC1CCN(C(=O)CCCN(C)C(c2ccsc2C)=O)C1 c1(Nc2ccc(C(N3CCN(C(C)=O)CC3)=O)cn2)cc(Cl)c(C)cn1 c1(C(=O)NC(CC)(C)CNC(=O)CN2CCCC2)cccc(C(=O)OC)c1C CC(C)CCCCC(=O)N1CC(CC(=O)NC2C3CCCOC23)C(C)C1 c1(C(N2CCC(C(=O)Nc3nc(Br)ccc3Cl)C2)=O)cc(F)cc(F)c1Br C(CNC(c1cccnc1C)=O)(C(C)C(C)C)NC(CCn1ncc(C)c1)=O N1(C(C2CC(=O)NC(=O)C2)=O)C2CCC1CC(CNC(c1cc(F)c[nH]1)=O)C2 c1(C(=O)NC(c2ccccc2)C(C)NC(=O)CNC=O)sccc1C#N CC1C(NC(c2cncc(N=[N+]=[N-])c2)=O)CC2CCC1N2C(c1nccn1C)=O C(=O)(CC(CNC(=O)CC(C)C1CCCO1)C1CCC1)N1CC(C)(CC)C1 C1(C(N2CC(C)C(CC(N3CCOCC(CO)C3)=O)C2)=O)CC2CC(=O)C1O2 N1(C(C2C(=C)C2)=O)CC(NC(=O)C(C)CC=CC)C(O)C1 c1(C(C)C)ncc(Cl)c(C(=O)NC2CCN(C(c3ccoc3)=O)CC2O)n1 C1(C(=O)NC(CNC(c2n(CCC)nc(C)c2)=O)C(C)(C)C)CC2(C1)CC(C)C2 c1(C(C(=O)NC(C(=O)OC)C)N(Cc2nonc2C)CC2CC2)ncc(CO)s1 C=CCN=c1[nH]cc(C(=O)NC2CN(C(=O)CSCC(N)=O)CC2C)s1 C1(CC(=O)NCCCCNC(C(C)OC(C)(C)C)=O)CCC(=O)N1C c1(OCC)nc(NC2(CNC(C3(C)CCCCO3)=O)CCCC2)ncc1C CCC(CNC(=O)C=CCOCCOC)(CC)C(=O)NC1CCNC(=O)C1 C1(C(=O)NC2(C)CN(C(CCCNC(=O)OCC)=O)C2)CCC(=O)CC1C C1(C(N2CCCC(CCNC(CC(=O)OC)=O)C2)=O)CCCN2CCCC12 C(=O)(CCCC(C)(F)F)N1C(C(C)C)CN(C(C2CC=CCC2)=O)CC1 C1(NC(CC(CC)(O)c2ccccc2)=O)CCN(C(=O)C2=COCC2)CC1(C)C C1(C)(C(N(CC(C)(C)CNC(c2csc3cncn23)=O)C)=O)CCCNS1(=O)=O C1(CNC(COCCCOC)=O)CN(C(c2cncc(C(C)C)c2)=O)C2CC12 c1(C(N2CC(CNC(c3scc(C)c3)=O)C(C)CC2)=O)cccc2ncc(C)n12 N1(C(C2N(C(C3OCCC(=O)C3)=O)CCCCCC2)=O)CCOCC(C2CC2)C1 C=CCCC(F)(F)C(=O)NCC(O)C(=O)NC(CC1CCCC1)CO c1(C(N2CCC(COC)(NC(C3C=CCC3)=O)C2)=O)ccc(Cl)c(Br)c1 C=CC1(NC(=O)C(CNC(c2cnoc2C(C)C)=O)N(C)C)CCC1 C1(NC(=O)NCCCC(C)N2CCCC2)CS(=O)(=O)CC1C C1(N(C(=O)C(=O)NCC2CC2)CC)CCCN(C(=O)Cn2ncn(C)c2=O)C1 C12(C(=O)NCC3N(C(C(N4CCSCC4)C)=O)CC3)CCCC1(C(N)=O)C2 N1(C(CCCN(C(C)=O)C)=O)CCC(CO)(CNC(=O)CCS(C)=O)CC1 c1(OCC)ccc(C(=O)NCCNC(c2cncc(C(N)=O)c2)=O)cc1Cl Cn1c(C(=O)NCCNC(=O)C(C2CCCCC2)F)cc(Cl)c1Cl N1(CCC(CC)C)CC2CC(C1)C1CCCCN1C2 C1(C(=O)NCC2N(C(C(N3CCNC3=O)C)=O)CC2)C(CC2CC2)C1(C)C C1(Cc2ccc(C)cc2)CCCCC1N=c1[nH]c(=NCC(C)F)[nH]c2c1CSC2 n1(CCC)nc(C)c(C(=O)NCCC(C)NC(c2nnn(C)c2CC)=O)c1C c1(C(N2C(CCC(=O)NCCCc3ccncc3)CCC2)=O)ccc(F)nc1F c1(C(=O)NC(c2cn(C)nc2)C(=O)N2CCC2c2ccnn2C)sccc1C#N c1(C(=O)NC2CCC(N(C(CCC(=O)N(C)C)=O)C)CC2)c(F)cc(N)cc1F c1(C(N2CC(C(C(=O)NCC3CCCSC3)O)C2)=O)ncccn1 C1(CCNC(c2ccsc2)=O)CCCN(C(=O)COC2CCCC2)CC1 C(CCN=C(NCC(O)Cn1ccnn1)NC1CC(=O)N(CC)C1)OCC C(=O)(C1CN2CCN1CC2)N1CC2C(C(=O)NCCCC3C(C)(C)C3)(C2)C1 N1(C(C(c2cnn(C)c2)C)=O)CC2CC(O)C1C2NC(c1snc(O)c1Cl)=O C(=O)(C(C)CC(N)=O)N(CCC(=O)NC1C(C=C)OCC1)C1CC1 N1(C(c2cnc(C)nc2)=O)CC2(C1)CN(C(C1CC1(C)Br)=O)C2 O=C(C1=COCCC1)NC1CC(F)CN(C(c2cc(O)nc(O)n2)=O)C1 N1(C(C=CC)=O)CC(NC(=O)C(C(C)C)OCC(C)C)C2(CC2)C1 c1(CC)nc(C)c(C(=O)NC(C2CCCC(C)C2)CC)o1 N(C(=NCCF)N1CCOC(C2CCCO2)C1)CC(CSC)(C)C Cc1c(Cl)cnn1CC(=O)NC1CC1CNC(=O)CCCc1cncs1 N1(C(C(C)(C)C#N)=O)CC2CC(C1)N(C(c1cn(CC(F)F)cn1)=O)C2 C1(CNC(C2CCC(N(C)C)CC2)=O)COCCN(C(C2(C)CCNC2=O)=O)C1 c1(C(N(CCC(=O)NCCC(=O)OC(C)C)C(C)C)=O)cn(C)nn1 C1(OC)CC(NC(c2c[nH]nc2C2CCOC2)=O)CN(C(c2occc2C)=O)C1 C(=O)(C1=CC2CCCCCC12)NC1CN(C(CC(CCC)CCC)=O)CC1O C(=O)(C(CN)C(C)C)NC(C1CCCC(C)C1)c1n(CCCC)nnn1 c1(C(N(CC(=O)NCC=C(C)C)C2CC2)=O)cc2ccccc2[nH]1 N1(C(CN(CCC#C)C)=O)CCN(C2CCC(NC(=O)C=CC)C2)CC1 N1(C(C(C(=O)OC)OC)=O)CCc2ccccc2C1CNC(c1csc(C)n1)=O c1(NC(=O)CC2(CNC(=O)Cn3cnnn3)CC2)cncc(F)c1 c1(C(N2CC(NC(C(CSC)(C)C)=O)C(C)(C)C2)=O)cc(N)c(C)c([N+](=O)[O-])c1 C=CCCCCC(=O)N1CCCC1(C(=O)NC)CCc1ccccc1 N1(CCC(=O)NC2(CNC(=O)C(F)=C3CCC3)CCCC2)CCCCC1=O CCS(=O)(=O)c1cccc(CCN2CCNCC2c2cccc(Cl)c2)c1 C(=O)(C(O)CC(N)=O)NC1C(C(=O)NC2C(OC)C(O)C2)CCC1 N1(CC(=O)NCCOCC(C)(C)C)CCCC2(CC=CCO2)C1 c1(C(N2CCC(C)C2CNC(c2cnn(C)c2F)=O)=O)ccc(Br)c(N)c1 N1(C(CC(C=C)C)=O)CCN(C(=O)CN2CCCCCC2)CC(C)(C)C1 C(CN(C)N1CC(O)(c2ccc(C(C)C)cc2)C1)c1c(C)n(C)nc1 c1(C(=O)NCC2C(NC(CC(C(F)(F)F)OC)=O)C2)cccc2nn(C)cc12 c1(C2(C(=O)NC(C)CNC(=O)CCc3cccn3C)CCC2)cc(F)ccc1Cl c1(C(=O)NC(CNC(CC=CCCCCC)=O)CCOC)cc(O)ncc1F CCCCC(C)C(=O)NC12CC(NC(C3CCCCN3C(C)=O)=O)(C1)C2 c1(C(=O)NCC2N(C(C3CCC(=O)NC3)=O)CCC2)c(F)cc(F)cc1Cl C=CCC(CNC(c1nonc1N)=O)C(=O)N(C)Cc1ccns1 CN1C(=O)CCc2cc(C(N3CCCC(NC4CCCCC4)C3)=O)ccc21 CCC(CCCC(=O)N1CCC(CCOC)CC1)NC(C1(OC(C)=O)CC1)=O c1(CC(C)NCC2(OC(C)C)CS(=O)(=O)C2)ccc(Cl)cc1Cl N1(C(c2n(C)ncc2)=O)CCC(C2CC2)(CNC(C2CC(=O)N(C3CC3)C2)=O)C1 C1(NC(Cn2ncc(CC)c2)=O)CCN(C(=O)CCc2ccsc2)CC1CC O=C1Cc2ccc(-c3ccc4nnc(NC(=O)CC(F)(F)F)n4c3)cc2N1 CCCCCCCCCC(=O)N1CCN(C(=O)C(O)CF)CC1CCC CC1CC2CCCC2N1C(=O)C(CN)C1CCOC1 c1(NC)ccc(C(=O)NC(C(=O)N2CCCC2CC(C)O)C(C)OC)nc1 c1(C(N2C(C(=O)NCc3cc(C(C)C)no3)CC(F)C2)=O)cnn2ccccc12 c1(CO)cscc1CNC1CCC1c1nc[nH]n1.N#CCCC1C(C(=O)OC)C1 N1(C(CCSC)=O)CC2CN(C(C3(Cl)CC3(F)F)=O)CC2C1 c1(CC(C(=O)NC(C)CCCNC(C2CC(F)(F)C2)=O)O)ccc(Cl)cc1 c1(C(=O)NC(=O)C(C)Cn2cccn2)cn(CCCCNC(CCOC)=O)nn1 C(=O)(CC(C(F)(F)F)NC(=O)C=Cc1cn(C)cn1)NCCC(C)(C)N(C)C Cc1nc2c(F)cccc2cc1C(=O)NC1CCC1NC(C1(CN(C)C)CC1)=O N1(C(C2(CC#C)CCCC2)=O)CCCCC(CNC(=O)CC2CC=CCC2)C1 Cc1ccn2ncc(C(N3CC4=C(C3)CN(C(=O)C(C)C3CCOC3)C4)=O)c2n1 c1(CC)cc(C(=O)NCCN(C(=O)CCC2CCC(O)CC2)C)nn1C C(=O)(C1=NOC(CC2(O)COC2)C1)N1C2(CNC(C(C(C)C)F)=O)CC(C1)C2 c1(OCCC(C)(F)F)ccc(NC(NCP(C)(C)=O)=O)cc1 CC(C)(C)C(CC(=O)NCC1OC(=O)CC1(C)C)NC(=O)CSCC(N)=O N1(C(c2c(=O)ccn(C)c2)=O)CC(CNC(C2CC3CCC2C3)=O)CC12CCC2 CCC(C)C(CC(=O)NCC(C)(C)n1cccn1)NC(c1ccnc(CO)c1)=O c1(COC)cc(C(N2CCCCC2CCNC(c2ccnnc2O)=O)=O)n(C)c1 c1(CC(=O)NC(CN(C(CC(CC)OC)=O)C)CC)cc(F)ccc1F C(N=c1[nH]c(=NCCC(O)C2CC2)[nH]c2c1SCC2)C1(OC)CC1 c1(C(=O)NCC2C3CN(C(C(CCC)C)=O)CC32)cc(O)cc(Br)c1 CN1N=C(C(=O)N2CCC(F)(CNC(c3cccc4c3OCC4)=O)C2)CCC1=O C=CC(CC)CC(=O)NCC1CN(C(c2cnc3n2CCS3)=O)CC12CC2 O=C(N=c1cc[nH]cc1O)C1CCCC2C1C2(F)F.c12cccc(c1)NC2=O C1(NC(CC(CC)C2CCC2)=O)C2CC1CN(C(=O)CC1(C)CCS(=O)(=O)N1)C2 N1(C(C)NC(=O)CC2COCCO2)CCN(C(=O)CCOCC2CCCO2)CC1 c1(CC)ncc(C(=O)NCC(c2ccccc2)CNC(=O)C(O)CSC)o1 Cc1c(C(N2CC(CNC(c3ccc(C(N)=O)cn3)=O)C(C)C2)=O)nnn1C c1(C(C(=O)NCC(C)N(C(c2ccc(OC)o2)=O)C)OC)ccc(Cl)c(F)c1 CC(C(C)C(=O)N(C)Cc1nccs1)NC(=O)CCC1CCCOC1 CCCCCC(C)CC(=O)NCC1(O)CC(NC(=O)CCCCC(=O)OC)C1 C12(NC(Cc3nc(C)[nH]n3)=O)CCN(C(c3ccc(F)cc3Cl)=O)CC1C2 Cc1cc(O)ccc1N(C(=O)CNC(=O)CC=CC(C)(C)C)C CC1CCc2[nH]nc(C(=O)NC3CC3)c2C1.C12(CCN(C(=O)CO)C1)COC2 N1(C(c2nc(CC)sc2)=O)CCOC(CCNC(=O)C(F)CC2CCCCC2)C1 C1(CC)CCCCC1OCC(=O)NCC(C)NC(=O)Cc1coc(C)n1 N1(C(CC(C=C)C)=O)CCC2CCC(NC(c3cc(CC)cc(Cl)c3)=O)C1C2 N1(C(c2cccc(C)c2)=O)CC2CN(c3cc(C)nc(C(C)C)n3)CC2C1 C(F)(F)(C(F)(F)F)CC(=O)NCC1(F)CN(C(c2ccncc2C(F)(F)F)=O)C1 C1(C(=O)NCC2CCCO2)CCCC(NC(=O)CCc2cccc(Br)c2)C1 N1(C(C2CC(CC)C2)=O)CCCC(C)C1CNC(c1cc(C)ccc1C)=O c1(C(=O)NC(CNC(CC2(C=C)CC2)=O)(C)C2CCC2)cnn(C(C)C)n1 N1(C(C2(CCOC)CCC2)=O)CC(NC(=O)C=Cc2ccc[nH]2)C(C)(C)C1 c1(C(N2CCC(C(=O)Nc3c(OC)c(F)ccc3)C2)=O)cc(C)cc2[nH]ccc12 C1(NC(Cc2cccc(C)c2Cl)=O)COC2(C1)CN(C(C1CC3C=CC1O3)=O)C2 c1(OC)cc(OC)c2sc(NC(c3ccnn3C3CCCCC3)=O)nc2c1 C12(NC(C(C)C3(O)CCC3)=O)CCCN(C(=O)CCc3ccccn3)C1C2 c1(CC)ccc(C(=O)NCCC2CC(NC(c3cnccc3CC)=O)C2)cc1 c1(C(C2CC2N(C)C)N)ccc(Br)cn1.C12(O)CN(C1)C2=O.CC1C(=O)N1C c1(C(N2CCC(CC)OCC2)C(=O)Nc2ccccc2)ccc2ccccc2c1 C1(NC(C2C(CC)CC2)=O)CCC(CCC(C)C)C1 c1(C(=O)NC2CCCN(C(CC(COC)C)=O)CC2)[nH]c2cc(F)ccc2c1C N1(C(C2(N(C(C(CC)CN(C)C)=O)C)CC2)=O)CCn2nccc2C1 CC1CCN(C(c2c(F)cncc2Cl)=O)CC1CNC(=O)CSc1cccs1 C1(C(=O)NCC(C)=CC(=O)NC2(CF)CCC2)CNC(=O)CC12CCC2 C1(CNC(CCNC(C)=O)=O)CC2CC2N1C(c1ccsc1C)=O CN1CCC(NC(=O)CNC(C2CCCNC2)=O)S1(=O)=O C1(C)(NC(C2CCN(CC(C)C)C2)=O)CCN(C(=O)CO)CC1 N1(C(C(CO)N(C)C)=O)CC2CC1C2NC(=O)C(c1cccc(Cl)c1)(F)F c1(C(N2C(C(=O)NCCc3cccnc3)CC3CC32)=O)cccc2c1CCCO2 N1(C(c2cc(OC)ncn2)C(=O)NCCCSC)CCC(C2CC2(F)F)C1 c1(OCC)ccc(CCC(=O)NC2CC(CNC(C3(C)CC(F)(F)C3)=O)C2)cc1 C1(CNC(C2CCC2)=O)CC2(CCN(C(C3OC4CCC3CC4)=O)CC2)CO1 C(=O)(C1=C(C)OCC1)NCCCC(C)(C)NC(C(C)OCCC=C)=O c1(CC)nc(C)c(C(=O)NCCCOCCN(C(=O)CN2CC3CC3C2)C)o1 N1(c2c(C)cncn2)CC(C2CCN(C(c3cccc4ccn(C)c34)=O)CC2)C1 N1(C(=O)NC2C3CCN(C(C)=O)C32)CCc2nccc(Br)c2C1 c1(C(=O)NC(C)(C)CNC(C2(O)CCCCCC2)=O)ccc(P(C)(C)=O)s1 C(=O)(CCCCC(=O)OC)c1c(SCc2onc(CC)n2)c(F)ccc1 c1(NC(C(C(=O)OCC)(CC)CC)=O)cc(S(N)(=O)=O)c(Cl)cc1Cl C1(NC(c2ccc(F)o2)=O)CCN(C(c2cnc(S)n2C2CC2)=O)CC1F c1(C(CNC(CN(CCC)C)=O)NC(c2ccc(CC)s2)=O)ccc(F)cc1 C1(C(=O)NCc2ccoc2)(NC(C(CN(C)C)N(C)C)=O)CCCCC1 c1(C(=O)NC(C)CNC(C2CCC(=O)C2)=O)cc(F)cc2ccncc12 C(=O)(CC(O)C(C)C)N1CC(SC)C(C(F)(F)F)C1.C1(C#N)(CN2CC2=O)CCC1 N1(C(c2ccc(SC)s2)=O)CCC2(CC1)OCCCC2NC(=O)C(C)C(C)O N1(C(C(CSC)OC)=O)CC2CCC1CC2NC(=O)C(C)n1cccn1 CC(C)CCC(F)C(=O)NC(c1nocc1C(=O)NCCCS(N)(=O)=O)C N1(C(C=CCCC=C(C)C)=O)CC2CCN(C(C3CN(C)CCO3)=O)CC2C1 C1(NC(c2ccc(CCC)[nH]2)=O)CN(C(=O)C(C)(O)CCC)CCC12CCC2 N1(C(c2c(C)nccc2Cl)=O)CCCN(C(=O)Cc2csc(S)n2)C(C(C)C)C1 Cc1ccc(S(=O)(=O)Nc2cccc(NCCC(=O)Nc3ccsn3)c2)c(F)c1 CC1(CNC(c2cccnc2)=O)COCCN(C(C2(C#N)CCCOC2)=O)C1 c1(C(N2CCC(O)(C(=O)Nc3cncc(Cl)n3)C2)=O)ccc(Cl)c(Cl)n1 C1(CNC(=O)CC2CCC(=O)O2)CC2CCC1N(C(C1(C(F)(F)F)CC1)=O)C2 CN1CCCC1CC(=O)NCCOC1CCN(C(=O)CCc2cnoc2)C1 N1(C(C(C(=O)OC)C)=O)CCCC(F)(C(=O)NCCC2(COC)CCC2)C1 C1(C(=O)NCC(COC)(C)C)CCN(C(c2ccsc2C#N)=O)CC1C C(=O)(C(CC(C)SC)N1CCCC(C(C)(C)C)CC1)NC(c1ccccc1)C C(=O)(C(C#N)(CC)CC)N(C(C(=O)NCC(=O)N(C)CCO)C)C c1(C(=O)NCCCNC(C=Cc2cn(C)nc2)=O)cc2c(s1)C(C)(C)CCC2 C(=O)(C(CNC(=O)Cc1ccc2c(c1)CC2)(CC)CC)N(CC(CC=C)(F)F)C C1(C(=O)NC2CC(CNC(c3ccc(C4CC4)s3)=O)C2)CCCC2(CCC2)O1 C1(F)(CNC(c2cnc(SC)[nH]2)=O)CCC(NC(C2CCCCS2)=O)C1 C(=O)(C1(C)CC(C(C)C)C(C)C1)N1CCC(N(C(C=C(C)Cl)=O)CC(C)C)CC1 C(C)(N=c1nc2sccc2c(N2CCC(CC(N)=O)CC2)[nH]1)c1c(C)noc1C N1(C(CC2(OC)CCC2)=O)CCCC(NC(c2cc(C(C)=O)[nH]n2)=O)CC1 CC1CSCCN(C(=O)C=CCC(C)(C)NC(=O)CC2CC3(CC3)CO2)C1 N1(C(C2(CCOC)CC2)=O)CCCC(O)(CCNC(c2cccc(N)c2F)=O)C1 c1(C(=O)NCC2C(CNC(CC(OC)OC)=O)C2)ccc(OC(F)(F)F)c(F)c1 C(=O)(CCC(N)=O)NC(c1cccc(Cl)c1)CNC(c1c(OC)n[nH]c1)=O CC1(C#CC(=O)NCCC2(C)CCN(C(c3cccc(F)c3O)=O)C2)CCCO1 C(=O)(C(C)C(=O)N(C)CC1CCN(C(=O)CCN(CC(C)C(C)C)C)CC1)OC C1(C(=O)NC(C#C)CO)CCn2cncc2C1 c1(CC(=O)NCC2CN(C(CC=C=C)=O)C(C)C2)ccccc1[N+](=O)[O-] C=C(Cl)CCC(=O)N1CC2CC1C2NC(=O)Cc1csc(C2CC2)n1 c1(C(=O)NCC2C=CCN2C(=O)C2CCc3c[nH]nc32)csc2ncnc(O)c12 c1(CNC(C2CCCC(CN)O2)=O)nc2ccccn2c(=O)c1Br C1(N(C(C(C=C)(C)C)=O)C)CCN(C(=O)CCCC(=O)N(C)C)CC1C Cc1cc(N)cc(C(N2CCC(NC(N)=O)CC2)=O)c1F c1(C(=O)NCCOC)[nH]c(C)c(C(N2CC(C)SC(C)C2)=O)c1C N1(C(CCCn2cc(C3N(C)CCC3)nn2)=O)CCC12CCN(C)C2 C(C1=CCN(C(c2c(C(F)(F)F)coc2C)=O)CC1)NC(C(C(C)C)SC)=O N1(C(C)=O)CCCC1CNC(C12CC(C)(C1)C2)=O C(=O)(C1=COCCC1)N1C(C(C(=O)NCc2cc(C)nn2C)(C)C)CCC1 C(c1cccc([N+](=O)[O-])c1)=CCNC1CC1C(=O)NCCc1cccc(O)c1 c1(C(N2CC(CCCNC(COCC)=O)OCC2)=O)cnc2[nH]c(C)nc2c1 C(CC(CNC(c1ccc(C)o1)=O)NC(=O)COCCCN=[N+]=[N-])OC C1(NC(c2ccc(C(N)=O)cn2)=O)CCCCN(C(c2ccnn2C2CC2)=O)C1 N1(C(c2c(C)scc2)=O)CCC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C(C)C1 C1(N(c2n(CCC=C)c(C(C)(C)O)nn2)C)CCCC(C(N)=O)(C(=O)OC)C1 C1(NC(CS(=O)(=O)NC)=O)CC2CC(NC(c3ccc(C(F)(F)F)[nH]3)=O)CC2C1 CN=S(C)(=O)c1ccc(C(=O)NCC(C)N(C)C(c2ocnc2C)=O)cc1 C1(CNC(CCN(C)C)=O)CCCCN(C(=O)C(C)(C)CC2CC2)C1 c1(OC)ccc(F)nc1NC(C1CC1C(=O)Nc1cccc(C#N)c1)=O C1(NC(C2CCN(CC)C2)=O)(CC)CCCN(C(c2ccn(CCO)c2C)=O)C1 N1(C(C(CO)N(C)C)=O)CC2C(CNC(c3cncnc3C3CC3)=O)C2C1 C1(C)(CC(=O)NCCc2nc(C)[nH]n2)CCCN1C(=O)CC1CCCCC1 Cc1nc(C(C2CCOC2)NCc2c(C(=O)O)cnn2C)c(C)o1.C12CCC1C2C C1(NC(C(C)SC)=O)CCSC12CN(C(=O)C(C)Cc1ccc(F)cc1)C2 C=CCCC(C(=O)OC)NC(=O)C(CC)NC(c1nscc1C)=O c1(C(=O)NCCC2OCCN(C(C3C(C)(C)CCC3)=O)C2)cc(Cl)cc(Cl)c1F FC1(F)CCN(C(=NCCc2ccccn2)NCC2CCCSC2)C1 N1(CCn2c(C)cc(C)n2)Cc2ccc(O)cc2CC1C(N1CCOC(C)C1)=O c1(OC)c(Cl)cc(NC(=O)C(=O)Nc2cn(C)nc2C(F)(F)F)cc1Cl c1(C(=O)NC)cc(NC(=O)NC(C)Cc2cccc(O)c2)ccc1F c1(NC)ccc(C(=O)NC2CC(CC(N3CCC3C3CCC3)=O)C2(C)C)cc1 N1(C(CCC(C)C)=O)CC2(CCCC2)C1C(N1CCN(C(C)C)C(=O)C1)=O c1(N2CC(=C(CNC(C3CSC3)=O)F)C2)cc2c(cn1)C(=O)CCC2 C1(CNC(c2c(C)ccnn2)=O)CN(C(c2coc(C(F)(F)F)c2)=O)CCC1C C1(OC)CCCC(NC(c2ccccc2-c2cccc(Cl)c2)=O)C1 C1(C(N(C2CCN(C(=O)CCc3cnn[nH]3)C2)CC)=O)CCCN(CC(F)F)C1 c1(C(=O)NC(CNC(c2cc(CC)c(F)cc2)=O)C)coc2c(C)cccc12 c1(C(=O)Nc2c(O)cc(OC)c(Cl)c2)c(Cl)nc(SC)nc1Cl.N12CCC(C1)C2 C1(CC(=O)N)CCCC(=O)C1.C1(CC(=O)NCC(C)NC)CCC(O)C1 N1(C(=O)CC2CCCOC2)CCN(C(C2CCC=CCC2)=O)C(C(F)F)C1 Cc1csc(CN(C)C(C2CCOC2CNC(=O)CCc2cc(C)on2)=O)c1 N1(C(C2C(C=C)C2)=O)CC2CCN(C(c3ccc(Br)c(OC)c3)=O)CC12 CCC(O)C(F)(F)C(=O)N1CC(CNC(c2cc(Br)nn2C)=O)C(O)C1 N1(C(c2cc(Cl)nn2C)C(=O)NC(C(=O)OC)C)CCN(C)C2CC12 N1(C(C2CCN(C(c3c(C)cn(C)n3)=O)C(C)C2)=O)CCC12CCOCC2 N1(C(CC=CC=C)=O)CC(C)(C)CC1C(N1CC(C(=O)OC)(OC)C1)=O N1(C(C2C(OCC)CC2)=O)CCC2CC12C(=O)NOCC1CCOC1C CCC(CNC(C1CC1(F)Cl)=O)(CC)NC(c1cncn1C)=O C1(NC(CCc2cc(OC)no2)=O)CC12CCN(C(C1CC1F)=O)CC2 c1(NC(C(=O)NC(C)CCCOc2cccnc2)=O)cnc2ccnn2c1 C1(C)(C(N(CCOC)CCNS(C)(=O)=O)=O)CCC2CC2C1 CC(C)(CC(=O)NC1CCC1NC(c1c[nH]nc1C(C)(F)F)=O)CC(F)F C=C(C)CC(C)C(=O)N1CCCC(CNC(=O)CCCOc2ccccc2F)C1 c1(CN2CC(C(=O)Nc3ncncc3Cl)C(O)CC2)c(O)ccc2ccccc12 c1(C(c2nnnn2C2CCC2)NCCS(N)(=O)=O)ccnc(Cl)c1Br c1(C(N(CC(C)NC(c2c[nH]nc2C(F)F)=O)C)=O)cc(CO)ccc1Cl N12CCCC(F)(C1)C2=O.c1(OC)cccc(NCC(=O)N(CCC(F)(F)F)C)c1 c1(OCC)c(OC)cc(C(=O)NCCNC(C23CC(C)(C2)OC3C)=O)cc1Cl C(C(C)(C)C(=O)NC1CCOCC1NC(=O)CC1CNC(=O)O1)SC N1(C(c2c(COC)n(C)nc2)=O)CC2CCN(C(=O)Cc3cc(C)no3)C2C1 CCN=C(NCC(C1CCCCC1)N(C)C)N1CCC(CCOC)C1 N1(C(c2c(C)nsc2)=O)CCC(O)(CNC(=O)CC2CCC(=O)N2)C1 c1(C(CC)NC(CC)(COC)c2nnnn2C(C)C)ccc(C#N)cc1 C1(CNC(c2c(C)scc2)=O)CC2CCC1N(C(=O)CNC(=O)NC1CC1)C2 c1(CC(N2CCC(O)(C(CNC(CCC#C)=O)C)C2)=O)cccc2sccc12 c1(C(=O)NCC(CN(C(CC(=O)OCC)=O)C)C)cc2n(n1)CCN(C)C2 C1(C(=O)NCC(C)NC(c2ccnn2C2CC2)=O)CCCCC1C(C)(C)C C(=O)(C(C)(CNC(=O)C(C)SC(C)C)CC)NC(CCC)CO C(c1ccncc1)=CC(=O)NC(CC(=O)NCC1(F)CN(C)C1)C1CC1 c1(CNCC2N(C(c3cocn3)=O)CCOC2)ccc2c(c1)Cc1ccccc1-2 c1(OCC)ccccc1Cl.C1(C)CC(=O)NCCC2CCN(C2)CCCN1 Cc1cn(CC(=O)NC2CCN(C(c3cc[nH]c3)=O)C2)c2ccccc12 c1(C(=O)NCCCCN(C)C(C2CC=CCC2)=O)cncnc1-c1ccccc1 C1(NC(C2C(COC)C2)=O)CCN(C(=O)CCCc2c(F)cccc2F)C1(C)C C(=O)(C1=CCC(C)CC1)NCCOCCCNC(c1c(C)cccc1)=O c1(C(=O)NCC(CC(=O)NC2CC2CF)OC)c[nH]nc1-c1ccoc1 c1(OC)cc(C(=O)NCC2(NC(C3CCC(=O)N3)=O)CCCC2)ccc1F Cc1c(OCC(=O)N(C)CC2CCCN2C(C2(C#N)CCOC2)=O)cccc1Cl N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC2CC2(C)C)C(C)(C)C1 CCCC(Cl)C(=O)N1CCC(O)(C(=O)NC(c2cccc(Cl)c2)C(C)C)C1 C1(S(C)(=O)=O)(C(N2CCC(NC(C(CC=C)OC)=O)CC2)=O)CCC1 Nc1nc(C(=O)NC2(CF)CN(C(=O)CC3CCC4(CCC4)O3)C2)ccc1O N1(C(C2CCC(C)(C)OC2)=O)CC2(CC(C(=O)NC(CO)C(C)(C)C)CO2)C1 c1(OC)cc(O)ncc1C(N1CCC(NC(=O)C=Cc2ccoc2)C1(C)C)=O Cc1ccnc(C(=O)NC2CCC2CNC(c2c(C)c[nH]c2CC(N)=O)=O)n1 c1(C(N2CC(C)C(NC(C3(c4cccnc4)CCC3)=O)C2)=O)cnc2n1CCC2 C1(CC(=O)NCC(CC)(CC)NC(C(CC)F)=O)CCCCC1(F)F Cc1cc(F)c(NC(=O)C(=O)NCC2C3CCC2(c2ccco2)C3)c(I)c1 CCC1=NOC(C(N2CC(NC(=O)C(C)OCC(F)(F)F)C(CC3CC3)C2)=O)C1 C1(C#N)(CC(=O)NCCC(C)N(CCC)C)CCOCC1 Cc1c(NC(C2CC2c2cccnc2)=O)n[nH]c1C1CC1 C1(C(=O)Nc2c(C)c(F)ccc2)COC2(CCN(C(=O)C(C)n3cccn3)CC2)C1 C(=O)(CC1=NN(C)C(=O)C1)OC(C1CCCN(CC(=O)N(CC=C)CC=C)C1C)=O CC#CCCC(=O)NC1CCC(NC(c2cc(Cl)sc2NC(C)=O)=O)CC1 C#CCCCCCCC(=O)NCC(O)CN(C)C(c1ccc(P(C)(C)=O)s1)=O C1(NC(c2[nH]nc(OC)c2Cl)=O)CCN(C(c2ncsc2C)=O)C(C)C1 C1(COC)(CNC(=O)CC2CCC2)CCN(C(C2CCC(=O)N(C)C2)=O)CC1 Cc1ccc(F)cc1NC(C1CC2(CC2)CN1C(c1ccnc(C(F)F)c1)=O)=O N1(C(=O)CC2CCCCCCC2)CCC2CCN(C(=O)CCc3ncco3)C2C1 C(=O)(CS(=O)(=O)CC(C)C)N1CCC(OCCNC(c2n[nH]c(C)c2C)=O)C1 Cc1csc2c(C(N3CC(C)(NC(=O)CC4CCCC45CC5)C3)=O)ncnc12 C1(NC(=O)CC2CC2)CCN(C(c2cnc(C3CC3)nc2O)=O)CCC1CO Cc1cc(C)c(C(N2CCC(NC(c3nncn3C)=O)C(F)C2)=O)c(=O)o1 C(=O)(C(O)C(F)(F)F)NCCN(CCOC)C(c1cc(C(F)(F)F)n[nH]1)=O N1(C(=O)CSc2cccnc2Cl)CC(NC(=O)C(O)Cc2cnc[nH]2)C2(CC2)C1 c1(OC)ccccc1C(N1CCC(C)(NC(C2CC2(Cl)Cl)=O)C1)=O N1(C(C(C)NC(=O)C2CC2)=O)CCC2(CC1)CCN(C(c1ccn(C)n1)=O)C2 N1(C(C(C(CC)C)NC(c2cc(O)cc(=O)o2)=O)=O)CCC2(CC(OC)C2)C1 Cc1nc(N)cnc1C(=O)NCC1CCCCN1C(c1cc(C(C)C)n(C)n1)=O CCC(CC(=O)NCCN1CCN(C(C2CCCCNC2=O)=O)CC1)C(C)C N1(C(CC2CN(C(CCC(C)OCC)=O)CC23CC3)=O)CCN2CCCCC1C2 CC1(C)CC(CNC(c2ccsn2)=O)CN1C(c1coc(O)n1)=O Cc1ccc(C(N2CCCC2C2CCN(C(c3csc(Cl)c3)=O)C2)=O)nc1 C1(CC(N2CCC(CCNC(C3(C4CCC4)CC3)=O)C2)=O)CCC2(CC1)CC2 c1(C(N2CCC(C(C)NC(c3n[nH]cc3Cl)=O)C2)=O)ncsc1S(N)(=O)=O n1(CCCN(C)C)nc(-c2ccccn2)nc1CCn1ccnc1 c1(CC(C(=O)NC(C(N)=O)C2CC2)NC(c2c(C)scn2)=O)cnn(C)c1O C1(c2cc(CNC(c3ccc(Br)c(Br)n3)(C)C)on2)CCC(F)(F)CC1 CN1N=CC(CC(=O)NCC(C)(C)C(=O)NCC2CC(C)(O)C2)C1=O C(=O)(CCCCCc1csc(C(=O)Nc2cc(C)nc(Cl)c2)n1)OCC C1(NC(CCC=C(C)C)=O)CS(=O)(=O)CC1NC(c1cccc(Cl)c1)=O c1(C(=O)NCCCNC(C2N(CCC)CCC2)=O)ccc(OC2CC2)cc1 c1(C(=O)NC2C(NC(CNS(N)(=O)=O)=O)CCC2)ncn2ccccc12 Cc1cc(Cl)ccc1C(=O)NC1CN(C(c2cc(Cl)on2)=O)CCC1C c1(C(=O)NC2CCN(C(C3C(CN(C)C)C3)=O)C2)cccc2c1OCC2 C(CNC(C1CCCC(O)C1)=O)(C(C)(C)C)NC(c1[nH]cc(C(C)=O)c1)=O C(=O)(CN=c1cc[nH]cc1)N1C(CC(=O)NC(CCC)CO)C(C)(C)CC1 C(=O)(C1CCCc2nncn21)N(C)CC1CN(C(=O)CCn2cnnn2)CCO1 c1(SCC(=O)NC(C2CN(C(=O)CCCN=[N+]=[N-])C2)(C)C)ccc(F)cc1Cl CON1CCC(C(N2CCC(O)(C(C)NC(=O)C(=CC3CCCC3)C)C2)=O)CC1 Cc1cc(C=CC(=O)NC(C)CN(C)C(C2CCC3(CC2)CC3)=O)c[nH]c1=N c1(OC)cc(=O)n(C)cc1C(=O)NCC1(C)CCCN1C(=O)C=C1CCN(C)C1 N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CC2CN(C(=O)CC(C)(C)O)CC2(C)C1 C(C)(C)(CC(=O)NCc1nc(CNC(=O)CC2CC(OC)C2)cs1)OC c1(NC(CC)CNC(=O)C=Cc2cnc[nH]2)nc(Cl)nc2c1ncn2CC C1(NC(CC2C(OC)CC2)=O)CC2CCC(C1)N2C(=O)CSc1cccc(C)c1 CC(O)CCCCCC(=O)NCCCCCNC(C1CCC(C2CC2)O1)=O c1(C(=O)NC2C3CN(C(CCc4ccn(C)c4)=O)C2C3)ccc(F)c(CO)c1 C1(C(=O)Nc2[nH]c(=N)sc2)CCCOC1C1CCN(C(=O)COC2CCC2)CC1 C=Cn1nccc1C(=O)NC1CCN(C(=O)CCCOCC)C1C(C)C Cc1cccnc1C(N1CCOC(CCC#N)C1)=O c1(OC)cc(C)c(C(N2CC(NC(c3ccc4n[nH]cc4n3)=O)C2)=O)cc1Br C=C=CCCC(=O)NC1COCC1C(N1CC(C)(F)C1)=O c1(OC)cc(Cl)ccc1CN(C(=O)COC(F)F)CC1CCCOC1 C1(CC)CCC2CN(CCC(c3ccccc3)O)CC12 Cc1ccc(C(=O)NCCOC2CCN(C(C3CC(=O)CO3)=O)C2)n1C c1(C(=O)NCCN(C(CC=C)=O)CCCN(C)C)cc(Cl)cc([N+](=O)[O-])c1O c1(N(C(C)CNC(=O)C=C2CCN(C)CC2)C)nc(C#N)ncc1Cl C1(CNC(CC(N)c2nccs2)=O)CC2CCN1CC2 Cc1cc(C#N)cnc1C(N1CCC(C2CCCN2C(C2CC(F)C2)=O)CC1)=O N1(C(c2cncc(Nc3ncc(F)c(C)n3)c2)=O)CCCC(C)C1CC.CO CC(COCCN(C)C)N=c1[nH]c(=N)[nH]c(=NCc2cc(O)nc(C3CC3)n2)[nH]1 Cc1nc(N(C)C)sc1C(=O)NCC1CCC1NC(c1ccccc1Cl)=O c1(C(=O)NCC2CCC(F)(CNC(C3(C)CCC(=O)C3)=O)C2)cnn2c1CCC2 c1(CC(c2cccs2)NC(C(=O)NCCC(C2CCCO2)OC)=O)ccccc1 c1(C(c2nnnn2C)NCC2C(C)C2C)cccc(C2CC2)c1F c1(C(N(C2CC(C(=O)NCC(C(C)C)OC)C2)CC)=O)ccc2c[nH]nc2n1 N1(C(C2N(CC)CCC2)=O)CCCC(NC(=O)C(O)CN(C)C)CC1 CN1C(=O)CCC1C(=O)NCC1(F)CC(CNC(=O)Cc2ccccc2Cl)C1 C(CC(C)CCCC(C)C)OC(c1c(SCC)cc(Cl)cc1)=O C(C(CC(C)C)C(=O)NCC12CC(C)(CCO1)C2)NC(C(C)=C1CCCC1)=O C1(CC(=O)N(CCC(C)NC(=O)Cc2cccc(Cl)c2)C)CCCCCO1 C12(NC(C=CCN(C)CC)=O)CCCC1(F)CN(C(c1cc(C(C)C)[nH]n1)=O)C2 Cc1occc1CC(=O)NC1CCN(C(C2(C)CSC2)=O)C1 C(=O)(C(C(C)CC1CC(F)(F)C1)N1CCC(OCC(N)=O)C1)NCC=C c1(C2N(C(C3C(P(C)(C)=O)CCC3)=O)CCC2)ccc2cnccc2c1 c1(C(N2CCCC(NC(C(CC)C(C)(F)F)=O)CC2)=O)nc2sc(C)cn2c1C CC1(NC(C2CC2c2ccncc2F)=O)CCC(NC(c2nn[nH]c2Cl)=O)CC1 Cc1c(F)cc(C(=O)Nc2nc(-c3cc(Cl)ccc3F)cs2)c(F)c1F C1(C(=O)NCc2c(C)nc[nH]2)CSCCN1C(=O)CO N1(C(C(C)NS(CC)(=O)=O)=O)CCC(O)(CN(C)C(c2cc(CO)on2)=O)C1 C1(CNC(=O)C(C2CC(F)(F)C2)O)CC(F)CN1C(=O)CC1COC(=O)N1 c1(C(=O)NCCOCCN(C)C(C2C3CCC23)=O)c[nH]c2cc(F)c(F)cc12 N1(C(C2(CCOC)CCCC2)=O)CCC2(NC(=O)CCCCC#N)CC2C1 c1(C(=O)OCc2ccc(N(CCCC)C)cc2)cc(C)c(CC)nc1O C(=O)(C1CCCn2ccnc21)N1C(CNC(c2coc(C(N)=O)c2)=O)CCCC1 c1(C(=O)NCCCCC(C)NC(C2CC(C)(C)CO2)=O)ncnc2c1CCC2 N1(C(C=CCCC)=O)CCOC(CCNC(=O)C(C)(C)c2cnn(C)c2)C1 c1(C(N(C2(C3CC3)CC2)C)=O)cccc(CNC(=O)C=CC2CCC2)n1 C1(C(=O)NCC(CN(C)C(c2c[nH]c(C#N)c2)=O)(C)C)C2CC2C2CC12 Cc1ccc(F)cc1C(N1CCC(O)C(NC(=O)CC2CN3CCC2CC3)C1)=O c1(SC)cc(C(N2CC(O)(CNC(=O)CC3CC(F)C3)C2)=O)ccc1[N+](=O)[O-] C(CCC(C)C)(C(=O)N1CCNC(=O)CC1C)NC(c1cc(C)no1)=O C(CCC(O)C(=O)NCC(C)CN=[N+]=[N-])NC(Cn1c(C)nnn1)=O C(CC1=CCCCC1)N(C(=O)C(C1CC=CCC1)NC(C1CCNC(=O)C1)=O)C C(=O)(CCS(C)(=O)=O)N1CCC(N(CC(C)C)C(c2cccs2)=O)CC1 Cc1cnc2n1CCC(C(=O)NC1CN(C(=O)CN(C)C(N)=O)CC1C)C2 c1(CNC(C2CC2C(N2CCCC2c2ncc[nH]2)=O)=O)cccc(C2CC2)c1 C1(C)(CNC(c2c(CC(C)C)onc2)=O)CCN(C(c2ccc[nH]2)=O)C1 N1(C(c2cnc(CC)[nH]2)=O)CCN(C)CC1CNC(C1CCCCC12CC2)=O C1(NC(C(C)NS(CCC)(=O)=O)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC1C N1(C(C2(CCF)CCC2)=O)CCC(C(CO)NC(C2(CO)CCCO2)=O)CC1 C1(C(N(CCN(C(=O)C(C)CC2CC2)C(C)C)C)=O)CC(O)(c2ccccc2)C1 c1(C(N(CCCNC(C2CCN(C)C2=O)=O)C)=O)cc(Br)c(F)cc1F C#CC1CCN1C(C1C(CNC(c2conc2CC)=O)C1(C)C)=O c1(NC)cnc(C(=O)NCC(C(=O)NCCCSC)N(C)C)cn1 N1(C(C2C(CCC)C2)=O)CC(NC(c2ccc(-c3cc[nH]n3)cc2)=O)CCC1C Cc1noc(C)c1CCC(=O)N1CC(N(S(=O)(=O)CCCl)C)C1 c1(CCCC)noc(CCC(=O)N(C2CCN(C(=O)CCSCC)C2)CCO)n1 N1(C(CC(CC)CC)=O)CC(C)CN(C(=O)CSc2ccc(C)c(C)c2)CC1C C1(C)(CNC(c2cc(OC)ns2)c2nnnn2CC2CC2)CNC(=O)O1 c1(C(=O)NCC2(OC)CN(C(c3ncccc3Br)=O)C2)ccc2c(c1)N(C)CC2 C1(CCCCNC(C=C(CC)C)=O)CCN(C(c2cnn(C3CC3)c2C)=O)CC1 C1(C(=O)NCC(C)N(C(=O)CC2CC2(Cl)Cl)C)CC12CCc1ccccc12 c1(C(N2CC(NC(C=C(CCC)C)=O)C(OC)C2)=O)cccc2c1CCCCN2 c1(C(N2CCC(C(N(CC(=O)N(C)C)CC)=O)C2)=O)cnc(O)c(C)c1 c1(C(=O)NC2CCN(C(c3c(CC)c[nH]c3)=O)CC2CC)cc(C)c(F)cc1Cl c1(C(N(CC(C)NC(c2c(CC)occ2)=O)C)=O)ccc2cccc(O)c2c1 N1(C(c2ccn(CC)n2)=O)CC2CC1C2NC(c1nc(-c2cccs2)oc1C)=O C(=O)(C(C)(C)CNC(c1ccns1)=O)NC(c1ccsc1)C C(=O)(C(C)(C)C)NCC(C)N(C)C(C12COCC1C2)=O c1(C(=O)NC)cc(=O)c(N2C(C)(CC)CC(NC(c3cnc(C)s3)=O)C2)cn1C C1(C(=O)NC(C)Cc2nn[nH]n2)CCCCCCN1C(=O)CC(F)(F)C(F)F c1(C(N2CCC2Cc2ccccc2)=O)cnn(CC2CC(C(=O)NC3CC3)C2)c1 N1(C(COCCC=C)=O)CCCC(C(=O)NCc2cnc(C(C)C)[nH]2)C1CC C1(C(=O)NCCCC(=C)Cl)CC2CC1CN(C(c1ncc(F)cn1)=O)C2 c1(C(=O)O)cccc(Cn2cc(CN3CCC(CCCl)CC3)nn2)c1 C1(NC(C(CCOC)OC)=O)CC12CCN(C(=O)C1=CC3C=CC1C3)CC2 c1(C(=O)NCC(C)NC(=O)CN2C(C)CCC2C)cc(CC2CC2)nc(O)c1 N1(C(C(CC)F)=O)CCCCC1C1(NC(=O)C(C)OCCC(C)C)CCC1 C12(NC(CCC=CC)=O)CC1CN(C(=O)COc1ccccc1O)C2 CCCC(C)CCCC(=O)N1CCC(O)(CCNC(=O)C2=CCOCC2)C1 C(CC1=CCN(C(=O)CC2CC3CC3C2)CC1)NC(C1(CC(C)C)CCC1)=O N1(CC2(C#N)CCC2)C(=O)CN(CCc2ccc(Br)c(Cl)c2)C1=O CC1=C(C(=O)NCCN(C(=O)C2=CC3CCCCC23)C(C)C)C=C2CCCN=C2N1 C1(C(=O)Nc2cn(CC(C)C)nc2)CC2(CCN(C(=O)C(F)C(C)(F)F)C2)C1 C1(N(CCc2ccc(OC)cc2)C(c2cnc(C)cn2)=O)CCNCC12CC2 N1(C(CCOC)=O)CC(C(=O)NCC2CC(C(=O)OC)C2)C2(CC2)C1 C=C(Cl)CC1C(=O)N1.c1(C(=O)NC2(CC)CCC2)cc2n(n1)CCO2 CC1CCN(C(c2ccoc2)=O)CCN1C(=O)CCN1C(=O)NC(C)(C)C1=O N1(C(COC(C)C)=O)CCC2(C1)CN(C(c1ccnc(P(C)(C)=O)c1)=O)CCO2 C1(CNC(C(CC)OCC)=O)CCN(C(c2cc3c(s2)CCC3)=O)C12CCC2 c1(C(=O)OC)cc(Br)c(NC(=O)Nc2ccc(F)cc2NC(C)=O)nc1C C(=O)(CC(=O)NC1CC1)N(C(C)CCNC(=O)C(=O)NCCC(N)=O)C N1(C(C=C(C)C)=O)CCC2(CC1)CC(C)N(C(c1ncoc1C)=O)C2 N1(C(C2N(CC(C)C)CCC2)=O)CCC(NC(c2cc(O)nn2C)=O)C(C)C1 Cc1nc2nccc(N3CCC(CCNC(c4cc(C)c(Cl)cc4C)=O)C3)n2n1 C(CC(O)CC(=O)N(C)CCNC(c1cc(-c2ccncc2)[nH]n1)=O)SC C1(NC(C2(OC)CCOCC2)=O)CC2CN(C(=O)Cc3ccon3)CC12 S(=O)(=O)(c1ccc(OC)c(-c2cccc3c2OCC3)c1)NC(CC)C(=O)OC N1(C(C2(CCOC)CC2)=O)CCC2(CCC(NC(=O)Cc3cncs3)CC2)C1 Cc1ccc2cc(C(=O)N(C3CCC(NC(=O)CCOC4CC4)C3)C)ccc2c1 N1(C(C2C(C(C)(C)C)C(=O)C2)=O)CC=CC(NC(=O)C(C)(C)Cc2cnn[nH]2)C1 C(=O)(C(=O)N=S(C)(C)=O)N1C(CN(C(Cc2c(C)cco2)=O)C)COCC1 c1(N2CCC(SCC)C2)ccncc1S(=O)(=O)NC(c1ccc(F)c(F)c1)C C1(CC(=O)NCC(CC)NC(c2c(C)nn(C)c2F)=O)CCCC(C)(C)C1 c1(C(=O)NCC(CC(=O)N(C(C)CS(C)=O)C)(C)C)cncc2[nH]ccc12 Cc1ccc(Br)nc1C(N1CCN(c2cccs2)CC1)C(=O)NCCC#N c1(C2C(SCC(=O)N(C3CCN(C(c4cncnc4)=O)CC3)C)C2)cccc(Cl)c1 C1(NC(=O)C(C2CCOCC2)O)CC2CCC1CC2NC(C1(C(F)(F)F)CC1)=O C(=O)(C(CC(C)(C)C)NC(=O)C(C1(O)CCCC1)F)N(CC(CC)O)C C1(C(=O)NC2C(n3ncc(C)c3)C2)C2CCC(C2)C1NC(=O)C=CCN(C)C N(C1CC2CCCc3cccc1c32)C(c1ccc([N+](=O)[O-])c(F)c1)=O CCCCC(CC(=O)NCCCC(C)(C)CO)NC(=O)CCOCCCOC C1(NC(C2ON=C(C)C2)=O)CC(C)CN(C(c2cnn(CC(C)C)c2)=O)C1 c1(C(=O)NCC(C)(C)CNC(C23CC2CNC3=O)=O)nccc2[nH]ccc12 C1(CC(N2CC(CCO)(NC(C(C)NC(=O)NC)=O)C2)=O)CCCCN1C C1(C2CC2)(NC(CN(C)C(C2CCC(CO)CC2)=O)=O)CCOC1 N1(C(Cc2cc(C)no2)=O)CCC2(CC(C(=O)Nc3ccns3)=NO2)C1 C1(C(N2CC(C(C)NC(C3CCOC3(C)C)=O)C2)=O)CCC(=O)N(C)C1 c1(C(N2CCC(CNC(c3c(C)nn[nH]3)=O)C2(C)C)=O)ccc(S(C)(=O)=O)o1 c1(OC)ccnc(CN2CC(c3cccc(C)c3)(O)C2)n1 N1(C(C=C(CCC)C)=O)CCCCC1CN(C(=O)CCc1ccon1)C CC(=O)CCN=C(NCc1ccn(C)n1)N1CCC(C(F)(F)F)(OC)C1 C1(CNC(C(CC)CO)=O)CN(C)CCN1C(=O)Cc1cccnc1OC N1(C(=O)Cc2cncs2)CCC2(CNC(=O)C(F)(F)c3nccs3)CCCC12 c1(N2C(C(=O)Nc3c(OC)ccc(F)n3)CC(F)C2)nc2ccccc2[nH]1 C(=O)(C(=O)C(C)CC)N1CCC(CC=C)(C(=O)NCc2ccnc(F)c2)C1 C1(C(=O)NCC2CNC(=O)CO2)CCCCCC1NC(C1CC2(CC2)C1)=O c1(CC(N2CCC(C)(NC(c3c(C)cccc3)=O)CC2)=O)cccc2nsnc12 C1(NC(C=C(C)Cl)=O)CC2CN(C(=O)C=Cc3ccncn3)CC12 Cc1cncc(C=CC(=O)NC2CN(C(=O)CC(C)c3ccncc3)CC2C)c1 C1(NC2(c3onc(C)n3)CCCC2)CC(NC(=O)OC(C)(C)C)C(O)C1 c1(OC)cccc2cc(C(=O)NC3CCCCNC3=O)c(=O)oc12 Cc1cc(=O)n(C)cc1C(=O)NCC1CCN1C(=O)CN1CCCCCC1=O C(CC(C)(C)C(=O)N1CC(O)(CCNC(=O)CC2(C)CC2(F)Cl)C1)SC c1(OC)c(Cl)cc(C(=O)NCCNC(=O)C(CCO)N(C)C)c2ncccc12 c1(C(=O)NC(CC#C)C(=O)NCCCN2CCOCC2)ccnc(C)c1N N1(C(=O)C=Cc2cccc(Cl)c2)CC(C2CCCN(c3ncc(Br)cn3)C2)C1 C1(NC(c2cn(C)nc2C(F)F)=O)CCN(C(C2CCC=CO2)=O)CCC1CO C12(C(=O)NC3CCN(c4nccc(C(C)C)n4)CC3C)CC(C)(C1)OC2(C)C N#CC(CC1CC1)C(=O)OCCC1CCCC12CC2 N1(C(C(CNC(c2ccc(Br)s2)C2CC2)C)=O)CC2CC2(C(C2CC2)=O)C1.CO CCC(C)(C)C(C)CC(=O)N1CC2(C1)CN(C(c1cncc(C(=O)OC)c1)=O)C2 C#CC1CCCC(NC(=NCc2ccccc2OCCOC)NC2CC2)C1 C1(C(NOC(C=C)C)=O)CN(C(C23CC(C#N)(C2)C3)=O)CC1(F)F CC(C)(CC1CCCO1)C(=O)N1CC(OCCNC(c2cnc(NC)cn2)=O)C1 c1(NC)cncc(C(N2CC(C(N3CCC(CCO)CC3)=O)(SC)C2)=O)c1 c1(C(=O)NC2CCC(CNC(c3cc(C#N)no3)=O)C2)cnc2ccccc2n1 N1(C(C(COC)NC(CCCOCC=C)=O)=O)CCC(COC)C(C)C1 c1(C(=O)NCC2C(NC(CCc3ccn(C)c3)=O)C2)c(C2CC2)cccc1F c1(COCCNC(c2c(COC)cco2)=O)cc(OC)c(O)c(OC)c1 Cn1nnc(CNC(C2CC2Cl)=O)c1C(=O)NC1CNC(=O)C1 c1(C(C(=O)NCC2C3CN(C(C4N(CC)CC4)=O)CC32)=O)ccc(F)cc1F c1(C(=O)NCC(CNC(Cc2c(C)nc[nH]2)=O)C)ccc(CO)cn1 Cc1c(F)ccn2c(NC(=O)CCSc3ccc(Cl)cc3)cnc12 CC(CC(=O)N(C)CCOCCNC(=O)C(O)c1ccco1)CC(F)(F)F C(=O)(C(F)(F)C(C)O)N(CC(CNC(c1c(C)[nH]nc1C(F)(F)F)=O)O)C c1(C(N2CC3CCN(C(=O)C=CC4CC4)C3C2)=O)ccn2c(O)nnc2c1 N1(C(c2c(CNC(c3nn(CC)nc3C)=O)cc[nH]2)=O)CCC2(CCCO2)CC1 C1(NC(C(C)CC2CC2)=O)CCCC(NC(=O)CSCc2ccccn2)C1 CC(C)CCN=C(NCc1ccc(C(C)O)cc1)NCC1CN(C(C)C)CCO1 N1(CC(CNC(=O)NC2(C(F)(F)F)CC(O)C2)CO)C(=O)c2ccccc2C1=O C(=O)(C1=CCC(C)CC1)NCC1OCCCN(C(C2(COC)CC2)=O)C1 CC1CCC(C)N(C(C23CC(CC4CC4)(CN2C(C2CC24CCCC4)=O)C3)=O)C1 C1(c2cc(C)no2)(NC(C2(C3(C(=O)O)CCCCC3)CC2)=O)CCOCC1 N1(C(C(C)(C)OC(C)=O)=O)CCC(CNC(=O)CN2CC(=O)N(C)C2=O)C(C)C1 CC1CCC2(CC1)CCN2C(=O)CCC1CCN(C(C2(CF)CC2)=O)C1 c1(CN2C(C(=O)Nc3ncc(F)cc3Br)CC2)ccc(Br)cc1[N+](=O)[O-] c1(OC)ccc(C(=O)NCC(C)NC(C2(O)CCC(C)CC2)=O)c2[nH]ncc12 N1(C(C2CCN(C(CCOC)=O)C2)=O)CCC2(CC1)COC(=O)N2 Cc1cc(C#N)cc(C(=O)NC2CC3CC(C2)N(C(c2ccc(=O)oc2)=O)C3)n1 CC1C(NC(=O)CCc2ccncc2)CC2CCC1N2C(c1ccnc(Cl)c1)=O N1(C(c2c(C(C)C)noc2)=O)CC2CCCC2(CNC(=O)CSCC(F)(F)F)C1 c1(NC(C)=O)ccccc1CC(=O)NC1CCCCC1CNC(=O)CC N1(C(=O)C(Cl)=CCl)CC2(C1)CN(C(C1(C(F)F)CCCC1)=O)CCO2 CC1(O)CCCN(C(=O)C2=CCN(C(=O)CCc3ccco3)CC2)CC1 c1(C(N(CC(C)(C)NC(c2ccc(CN(C)C)o2)=O)C)=O)cnc2n1CCOC2 c1(C(=O)NC(c2cn(C(c3cccnc3)C)nn2)(C)C)cc2scc(Cl)c2[nH]1 N1(C(C2(Oc3ccccc3)CC2)=O)CCC(O)C(c2ccccc2)C1 N1(CC(=O)NC(CC)CNC(=O)CC2CCCC2C)Cc2ccccc2C1 C1(CNC(c2ccsn2)=O)CCCCCN1C(c1ccc(O)cc1)=O n1(CC(C)C)cc(S(=O)(=O)NC(c2nc3c(s2)CCC3)C)cn1 Cc1ccccc1C(C)CC(=O)OCCN1C=C1NC(=O)C(c1cccnc1)O c1(NC(C(N2CCC(CSC)C2)c2cccs2)=O)ccccc1C c1(CCC)nc(C(=O)N(C)CCN(C)C(C2CCCN2C(=O)NC2CC2)=O)co1 CCCCC(O)C(=O)N1CCCC(N(C)C(c2ccc(O)cc2F)=O)CC1 C1(CC(=O)NCC(c2ccccc2)CNC(CCSCC)=O)CCCC1(F)F CCC(C)C(O)CC(=O)NC(CCCOC)C(=O)NC1CCC(=O)NC1(C)C N1(C(CC2CN(C)C2)=O)CCC(CO)C(NC(c2ncccc2OC(C)C)=O)C1 c1(C(N2CCC(NCc3nn(CC)nc3C)C2)=O)nc[nH]c2nccc1-2 Cc1cc(C)c2nc(N3CCC(NC(c4ccnn4CCF)=O)C(F)C3)sc2c1 CC(C)CC(C)(C)C(=O)NCC1CCN(C(=O)CN2C(C)CCC2C)C1 Cc1cccc(NC(C2CC3CCC2N3C(=O)Cc2cccs2)=O)c1C c1(CC(N2CCC(C)(OC)C2)=O)ccc2c(c1)CCCC2=O Cc1cc(C(N2CCOC(CC(=O)NC3CC3c3ccn(C)n3)C2)=O)ccn1 C1(C(=O)N(C2CC(NC(C3CCOCC3)=O)C2)C)(CC)CCOC1 N1(C(C=CCN(C(C(CCCC)=O)=O)C)=O)CCCC2NC(=O)CC12 C(c1ccccc1[N+](=O)[O-])=CC(=O)NCC1(F)CC(NC(=O)C=CCF)C1 N1(C(c2ncc(N)nc2)=O)CCOCC(CNC(=O)COCC2CC2)C1 c1(C(C(=O)NC(CN(C(C2CC3(CC3)C2)=O)CC)C)C)ccc(C)s1 C(C(CC(C)C)NC(C12CCCC1C2)=O)NC(c1cc(C)on1)=O c1(CCC(N2C3C(NC(C4C(C)(C)CCC4)=O)C(C3)C2)=O)ccc(F)c(F)c1 CC(C)C(O)C(F)(F)C(=O)N1CC(C2(NC(=O)COCCN(C)C)CC2)C1 O(NC(=O)C(CCSC)NC(c1cc(C)c(C)o1)=O)CCCC#C C1(CC)CCC(C(N2CCC(CNC(=O)CCCC3CCCCC3)C2)=O)O1 c1(OC)cccc(C(=O)NC2CN(Cc3c[nH]nc3C)CC2O)c1Br Cc1cnc(C(=O)NCC2C3CC2N(C(c2ccc(C(F)F)cn2)=O)C3)c(F)c1 Cc1cccc(CC(=O)NCC(CC(C)C)NC(C2COC(=O)O2)=O)c1 N1(c2cc(OCC)nc(C)n2)CCC(C2CCCN(C(=O)C3=C(Cl)CC3)C2)CC1 c1(C(=O)NC2CN(Cc3cccc(Cl)c3)CC2F)ccc2cccc(Br)c2n1 CC(C)C(CNC(C1CCN1C)=O)N=c1nc(Cl)[nH]c(C)c1C#N CC1(C(=O)NCc2cn(CCNC3CCN(C4CC4)C3=O)nn2)CC2CCC1O2 CC1CN(C)C(C)CN1C(C1CN(C(=O)C#CC(=O)O)CCO1)=O C1(C(N(OC)CC2CCCC2)=O)COC2(C1)CN(C(=O)CC1COC(=O)C1)C2 c1(OCC(=O)NC(C)(C)CNC(=O)CC2COCCO2)ccc(C#N)cc1Cl n1(CC=C)nnnc1C(c1cnoc1-c1ccccc1)NCCC1CC=CCC1 C12(NC(CCC#C)=O)CC3CCC(C1C2)N3C(c1nn(C(C)(C)C)cc1OC)=O c1(C(C(N2CC(N(C(CC3(OC)CCC3)=O)C)C2)=O)O)ccc(Br)cc1F C(=O)(C(C)C(O)C(C)C)NC(CCNC(CC1(C=C)CCC1)=O)(C)C N1(C(=O)OC(C)(C)C)CC2CCCC2(NC(C2COCC2(C)C)=O)C1 c1(-n2ncc(NC(CC(=O)NCC(COC)(C)OC)=O)c2)ccc(C)cc1 C1(NC(=O)NC(C(O)C(F)(F)F)C2CC2)CCC2(CCOCC2)C1 N1(C(c2nncc(OC)c2)=O)CC(C)CN(C(C2SCCS2)=O)C(C)C1 N1(C(c2cc(I)ccc2Cl)=O)CC(N=c2ncc3cc(F)cc(Br)c3[nH]2)C1 Cc1c(C(N2CC(N(C(=O)C3CCc4c[nH]nc43)C)C2)=O)[nH]c2c(C)cccc12 C(CC(=O)NCCCCC1CN(C(=O)COC2COC2)C1)NC(C1C(C)C1)=O CC(C)CCCCCC(=O)NCCC(N1CCCC1CCC(C)C)=O c1(C(N(C2CN(C(=O)C(C3CCC(O)CC3)(C)C)C2)C)=O)cc(O)cc(F)c1F Cc1c(C(=O)NC(CNC(=O)CCCF)CC(C)C)nn(C)c1Br C1(C(N(CCCCN(C)C)C)=O)(NC(C2COCOC2)=O)CCSC1 N1(C(CCCC(C)C)=O)CCC2CN(C(=O)CSCCN(C)C)CC2C1 C1(CNC(CC2(OCC)CCC2)=O)CC2CCC1N(C(=O)CC#N)C2 CC1CCC(c2cccs2)N(N(CCN2CCOCC2)CCO)C1 c1(C(N(CCCN(C(CSCCC)=O)C)C)=O)cc2c(=O)n(C)c(=O)n(C)c2s1 N1Cc2ncccc2N2CCCC2C1.CC(O)(CC(=O)c1ccc(SC)cc1)CC(=O)O CON(CCC(=O)NCC1(CF)CCC1)C(=O)C1CC2C(C1)C2(F)F Cc1ccc2[nH]nc(CN3CCC(NC(c4ncnn4C)=O)C3)c2c1 N1(C(C(CC=CCC)C)=O)CCCC2C(NC(c3cc(C)sc3N)=O)C(C)(C)C12 C=CCC(C(=O)NC(C)(C)CCCNC(=O)C(C)OCOC)c1ccccc1 C(=O)(C(O)CC(C)(C)C)N1CC(CC(C)NC(=O)CCNC(=O)C(C)(C)C)C1 N1(Cc2c(OC)c(Br)ccc2)CCC=C(C(=O)N=c2ccn(CCN(C)C)[nH]2)C1 c1(C(N2CC=CC(NC(c3c(CC)nn(C)c3Cl)=O)C2)=O)coc2c1CCCC2 C12(C(N(CC(CC)NC(c3cc(C(N)=O)no3)=O)C)=O)CCC(C)(C1)OC2 n1(C(C)C)cc(C(c2nnnn2C(C)(C)C)NCCC2CCCC2)cn1 c1(C(=O)NCC(C)NC(C2C(OCC)C2)=O)c[nH]c2cc(C)ccc12 N1(CC(=O)NC2CCC(C)N(C(=O)CC(F)(F)F)C2)CCc2sccc2C1 N1(C(C(C)(C)F)=O)CCC2CCCC12CNC(c1ncc(Br)cn1)=O N1(C(c2coc(Cl)c2)=O)CCN(C(=O)Cc2sc(O)nc2O)C(CCO)C1 C1(C(=O)NC(C2CCN(C(c3cccc(C(N)=O)c3)=O)C2)C)CC2CCC1C2 C1(=Cc2ccn(C)n2)N=C(c2cc3c(s2)CCC3)NCC1=O C(=O)(C(C)(O)CC(F)(F)F)N(CCCNC(C(C1CC1)OC)=O)C1CC1 C1(CNC(C(C(CC)C)O)=O)CCC2(CN(C(=O)CCc3ccc(F)nc3F)C2)O1 Nc1cc(C(=O)NCC2CCN2C(C23COCC2C3)=O)ccc1-n1cncn1 Cc1cncc([N+](=O)[O-])c1N1CCCC1CNC(c1ccc([N+](=O)[O-])[nH]1)=O N1(C(CC(C)C)=O)CC2CC1C2NC(=O)C(C)Oc1ccccc1F C(=O)(CC(C)CC(F)(F)F)NCC(C(C)C)NC(=O)Cc1cnnn1C n1(CC(=O)NC2CCN(C(COCCCCC)=O)C2C(C)C)cc(F)ccc1=O CC(F)(F)CCC(=O)N1CCN(C(c2cc(CO)on2)=O)C(c2cn[nH]c2)C1 c1(C(N2CCC(N(C(C(CC)NC(N)=O)=O)C)C2)=O)nnc(C)cc1O C(CO)(C(=O)NCc1ncco1)NC(C(c1ccn(C)c1)C)=O n1(CC(=O)NCC(CC)(CC)NC(=O)C(C)NS(C)(=O)=O)ccc(=O)cc1C c1(NC(C)=O)cc(C(=O)NCC(C)CNC(c2ccc(C)c(O)n2)=O)ccc1C c1(C(C(=O)NCCNC(c2nnc(CC)s2)=O)C2CCCO2)ccccc1OC N1(C(c2ccc(CN(C)C)o2)=O)CCCC(CN(C)C(C2CC2F)=O)C1 N1(C(C2CC(C)(CC)C2)=O)CCc2c(c(CNC(C3CC3(Cl)Cl)=O)nn2C)C1 C1(C(=O)OC)CC(C2CC2)=NO1.c12cc(sc1C)CNC(=O)NC2 c1(C(=O)NC2CCCCN(C(c3cncc(C)c3C)=O)C2)cc2ccncc2[nH]1 C(c1cccc(Br)c1)=CC(=O)NC(CNC(C=COCC)=O)CO CC1(C)CN(c2ncnc3ccsc23)CCC1NC(=O)COC(F)(F)F Cc1sc(C(=O)NC2CC(NC(C3CN4CCCC3CC4)=O)C2)cc1S(N)(=O)=O N1(C(CNC(CCNC(CN(C(C)C)C)=O)=O)=O)C(C)CCC1C c1(C(=O)NC23CC(NC(CSC)=O)(C2)C3)ccc(Br)cc1O c1(Nc2scc(CC(=O)NCC(c3ccccc3)(C)O)n2)c(Br)cnn1C C(=O)(C#CC1CCCC1)NCCC1CC(C(=O)NC2(C)CCC(O)CC2)C1 C1(CCNC(C2C(C)(C(F)F)C2)=O)CN(C(=O)CNC(=O)C2CC2)CCO1 c1(CC(=O)NC2(CCNC(CNC=O)=O)CCC2)cnc(C2CC2)[nH]1 c1(C(=O)OC)cn(CC2CCN2C(=O)C(=O)Nc2ncc[nH]2)c2ccccc12 C1(NC(=O)NC(c2ccco2)COC)CCCCN1CC1CC1c1ccco1 C1(OC)CN(C(c2cnc(C(C)C)o2)=O)CC1NC(C1(c2cc[nH]n2)CC1)=O N1(C(c2c(C)[nH]cc2)=O)CCC(C2CCCN(C(c3cnnc(O)c3)=O)C2)C1 Cc1ccc(C(=O)NCC2CC(C(=O)NCC3(F)CC(N(C)C)C3)C2)cc1C C1(C(=O)NC2(CO)CCC(C)CC2)CCN(C(=O)C(F)(F)C2CC2)CC1(C)C c1(-c2c(OC(C)C)cccc2)cn2c(n1)CN(Cc1cc(Br)cc(Br)c1F)CC2 C1(C2CC2)(CNC(=O)CCF)CCN(C(=O)Cc2nc(-c3ccccc3)no2)C1 CC1CN(C(=O)CC(C)(C)C)CCN1C(=O)C(O)Cc1ccc(F)cc1 C1(CNC(C2CC(c3ccc(O)cc3)C2)=O)CCCN(c2ccncc2)C1 C(C(CC)CC)c1onc(CCC(=O)OCCCC)n1.c1ccccc1 N1(C(C(CC(CC)CC)F)=O)CCC2CN(C(=O)C(C)C(O)C(C)C)CCC2C1 CCC(C#N)(CC)C(=O)N1CCCC(CN(C(=O)CCc2ncccc2C)C)C1 c1(C(=O)Nc2nc(-c3cc[nH]n3)cs2)ccc(S(=O)(=O)Cc2ccc(Br)cc2)cc1 Cc1ccc(=O)n(CC(=O)NC2CCCC2CNC(=O)CS(C)(=O)=O)n1 C1(CNC(c2c(C)onc2C2CC2)=O)N(C(c2cncs2)=O)CCC1(C)C c1(OCC)cccc(C(=O)NC2CC(NC(=O)CC3(CO)CCCCC3)C2)c1N S(=O)(=O)(c1ccc(NCC2(N(C)C)CC2)cc1Cl)N1CC(CC=C)C(N(C)C)C1 N1(C(CC(CC)(F)F)=O)CC2(CCC2)CC1C(=O)NC1CN(C)CC1C C(CCO)(C(F)(F)F)NC(C1CC(N(C(=O)CN2CCN(C)CC2)C)C1)=O c1(OC)ccc(Cl)cc1C=CC(=O)NCC=CCNC(C1CCOC(=O)CC1)=O C(c1c(Cl)cccc1Cl)=CS(CCNC(CCCCNC(=O)OC(C)(C)C)=O)=O N1(C(COCc2c(C)cccc2)=O)CC(C)N(C(=O)CCC2OCCO2)CC1C c1(C(N2CCC(NC(CC(c3ccc(CC)cc3)C)=O)C2)=O)cc(=O)cc(Cl)[nH]1 C(CCc1cn[nH]c1)(C(=O)NCC(O)CF)NC(=O)OC(C)(C)C C1(NC(CCc2ccn(C)n2)=O)CCC2CC1CN2C(=O)C1=CCOCC1 c1(C(=O)NCCC23CCC2CN(C(=O)C(Cl)=CCl)C3)cc2ccccn2n1 CC(C)(C)CC(O)C(=O)N1CC(F)(F)CC1CNC(=O)C(F)(F)c1ccccn1 N1(C(c2cccc(OC)c2)=O)CCC2(NC(=O)CCC3CC3(C)C)CCCC12 Cc1nc(C(=O)NC(C23CCC(CC2)C3)CNC(=O)Cc2c[nH]nc2C)c(C)s1 C(=O)(C(C)(C)C(N)=O)NC(CCOC)CNC(=O)CSc1ccccc1 CC1(C)CC(CC(N2CC(CC3CC3)C2)=O)N(C(C2Cc3nccn3C2)=O)C1 CC1(C(=O)NCC2CCN2C(=O)Cc2csc(Cl)n2)CCc2ccccc2C1 C1(C(N2C(CNC(CCCCCSC)=O)CCC2)=O)Cc2ccncc2C1 c1(C(=O)NCC2CN(C(CCC(=C)C)=O)CC2O)ncn2c1COCC2 c1(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)c[nH]c2cccnc12 C1(C(N2C(CNC(CCCC(N)=O)=O)CCCCC2)=O)CCc2nncn2CC1 c1(CNC(=O)OC(C)(C)C)ccncc1NS(=O)(=O)CCCN1CCCC1 N1(C(c2cc(OC)cc(Cl)c2)=O)CC2CN(C(C3CCCC34CC4)=O)CC2C1 C12(CNC(C3CCC(=O)NC3)=O)CCC(CC1)N2C(c1cc2n(c1)CCC2)=O C(CCC1CC1)(C(=O)N1CCCCCC1)NC(c1ncncc1Cl)=O C(=O)(CS(=O)(=O)CCO)NC(C1CCCCC1)CNC(c1n(CC)nnc1C)=O N1(C(c2nc(COC)oc2)=O)CCCC(NC(C2CCCC2C(F)F)=O)C1 N1(C(C2(CNC(C(CCC)F)=O)CC=CC2)=O)CC2C3C=CC(O3)C2C1 c1(C(=O)NC(CCC)CNC(=O)CN2CCC(C)C2)cc(O)ccc1C C1(CC=C)(NC(c2[nH]nc(C(F)(F)F)c2CC)=O)CCN(C(C2(C)CC2)=O)C1 c1(C(=O)NC2CCCC(CNC(C(C)(C)SC)=O)C2)ccc(O)c(CO)c1 C1(C)(C(=O)NCCCCN(C)C(C2CC3CCC2O3)=O)CCC(=O)C1 c1(CC(N2CCC(C(C(=O)NCC(C)OCCO)C)C2)=O)cccc(F)c1 c1(SCC(N2CC(O)(CNC(C3(C(C)C)CCCO3)=O)C2)=O)cc(F)ccc1F n1(CC)nc(C)c(CC(N2CCOCC2CCNC(c2csnn2)=O)=O)c1C N1(C(Cc2c(C)noc2C)=O)CCCC2(NC(=O)Cc3cccs3)CC2C1 C1(C#N)(C(=O)NC2CC3(CN(C(C4N(CC)CCC4)=O)C3)C2)CC2CCC1CC2 N1(C(C2(C#N)CC2)=O)CC(C(=O)NCCC2CCCC23CC3)C2(CCC2)C1 Cc1cc(=NCC(C)CNC(=O)C(=O)Nc2ccccc2)[nH]c(N(C)C)n1 N1(C(c2nc(C)sc2)=O)CC(C2CCN(C(c3cn(C)cc3C)=O)CC2)C1 C1(C(=O)NCC(C)CNC2(C(O)CO)CC2)CCC(=O)C1 c1(C(=O)NC(CNC(c2nc(CCC)sc2)=O)C)cc(C)c2[nH]nnc2c1 Cc1[nH]nc(C(=O)NC2(C(N3CC(n4cnnc4)C3)=O)CC2(C)C)c1Cl C1(CCN(C(C(CC)=CC)=O)C)CCN(C(=O)C(C)N(CC)CC)CC1 CCS(=O)(=O)CC(=O)N1CC=CC1CNC(=O)CC1CCN(C(C)=O)CC1 C=C=CCNC(=O)CN(C(=O)C1CC1)CC n1(CC)cc(C(=O)NC2CCC(NC(=O)COCCS)C2)c(C2CC2)n1.C1CC1 c1(SCC)cnc(O)c(C(=O)NCCC(C)(C)NC(c2nc(O)c(C)s2)=O)c1 c1(CC(C)NC(=O)NCC2CC3(CC3)CO2)csc2ccccc12 CC(C)CCOC1(CCC(=O)N2CC(NC(N)=O)C2)CCC1.C1C(=O)N1 C(=O)(C1=NOC2(CCC2)C1)NCCOCCNC(CN(C)CC)=O N1(CCNC(C(C(C)OC)O)=O)CCCN(C(c2nocc2C(C)C)=O)CC1 Cc1ncc(C(=O)NC2CCCCN(C(c3ccnc(O)c3)=O)C2)c(C(C)C)n1 N1(C(C(=O)NCC(F)F)=O)CC(C(=O)NOCC2CCCC2)CC12CCC2 c1(N(n2cc(CNOc3ccccn3)nn2)C)ccc([N+](=O)[O-])cc1F N1(C(C(=O)NCCOCCCC)=O)CCC(C)C1CNC(c1ccc(C)nn1)=O c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)CN(C)C)C)ccnc2ccsc12 C(=O)(C(F)(F)C(C)O)N(CC(C)CNC(c1ncccc1CO)=O)C N1(C(c2c(C)ncc(N)c2)=O)C2CCC1CC(N(C)C(C1CCCC(C)C1)=O)C2 c1(C(=O)NCCC2CCCN2C(=O)CSCc2ncc[nH]2)cc2n(n1)CCCO2 Cn1ncc2cc(C(=O)NCC3C4CN(C(C5CC(=O)CCO5)=O)CC34)cnc12 Cc1c(C(N2CC(NC(C3(C)CNC(=O)C3)=O)C(F)C2)=O)ccc(F)c1F c1(CCC(=O)NC2C(NC(c3c(C)ccnn3)=O)CCCC2)ccccc1C#N C12(NC(CCOCC#C)=O)CCC(CNC(=O)C(C)CC(=O)OCC)(CC1)CC2 Cc1cc(C(N2CCC(C)(CNC(=O)CC(O)C3CCCC3)C2)=O)nn1C1CC1 C1(C(CNC(CN(S(CC)(=O)=O)C)=O)C)CCN(C(C2C(C)C2C)=O)CC1 CC1CC(N=c2[nH]c(N3CCC(C)(C)CC3)nc3c(F)cc(F)cc23)CS1 c1(CNC(C2(N(C)C)CCC2)=O)cc(C(=O)NCC2COC(=O)N2)n(C)n1 c1(OC)ccc(CN2CCCC(NC(=O)NC(C)(C)C)CC2)c(Br)c1OC CCCCC(O)C(=O)NCC(C)(C)CNC(c1ncsc1C(C)C)=O Cc1nc(O)nc(O)c1CCC(=O)NC(CNC(=O)C(C(C)(C)C)N(C)C)CO N1(C(Cc2c(C)ocn2)=O)CCCC12CCN(C(C1C(C)(C)C1(F)F)=O)C2 C1(C2CC2)(CNC(c2cccs2)=O)CCN(C(c2cc(CC3CC3)[nH]n2)=O)C1 N1(C(CC(CC)(F)F)=O)CCC2OCCN(C(c3cnc4[nH]nnc4c3)=O)C2C1 C1(NC(C)(C)C)C2CCCOC2C1(C)C.C12CC3(COC(C3)CNC(=O)O1)C2 N1(C(c2c(C)cc(CC)o2)=O)CC2CCCC2(C(=O)NC2(C)CC(O)(CO)C2)C1 C(=O)(C(F)C(C)CNC(c1cnc(O)cc1C)=O)NCc1cn(CC)nc1 C(=O)(C(CC)CC(F)(F)F)N(C1CCN(C(c2c[nH]c(C)c2)=O)CC1)CC#C CN1C(=O)OCC1NC(=O)NCCCCCCn1cc(-c2cnccc2Cl)nn1 C1(CNC(c2c(OC)cnnc2)=O)(CO)CCCN(C(C2CC2(C)C(C)C)=O)C1 c1(CC(=O)NC2(C)CN(C(c3ncccc3F)=O)C2)c(F)cccc1C#N N1(C(c2n(C(C)C)ccn2)=O)CC(C(=O)NC2CCC3(CCC3)C2)CC(C)(C)C1 C1(OC)CCC(C)(C(=O)NC2CCCN(C(C3CCCN3C)=O)C2C)CC1 c1(CCC(N2CCC(F)(CNC(C3CC4(CCC4)C3)=O)C2)=O)ccc(F)cc1F c1(OC)cccc(CCCN(C)C)c1F.S1(=O)(=O)CCN1 N=c1[nH]c(C(=O)NCCOCCOCCNC(C2CCCO2)=O)ns1 C1(C(=O)O)CC2CCCCC2N(C(=O)CCn2ccnc2)C1 c1(C(=O)NC)cc(C(=O)NCCSCCOCCC(=O)N(CCCO)C)on1 CCC(C)CCCC(=O)N(C(C(N1CC2(C1)CN(C)C2)=O)C1CC1)C CCCS(=O)(=O)CC(=O)NC12CC1CN(C(c1ccc(C(=O)OC)s1)=O)C2 C12(C(N3CCC(C(C)NC(c4cc(=O)cc[nH]4)=O)C3)=O)CCCCC1OCC2 C(=O)(C#CC1CCCOC1)N1CCCCC(NC(c2ccc([N+](=O)[O-])o2)=O)C1 c1(-c2n(CC=C)c(N3CCNC(=O)C3)nn2)ncc(C)cc1F c1(C(N(CC(O)CN(C)C(c2cc(C(F)F)no2)=O)C)=O)n[nH]c2c1CCOC2 N1(C(C2CC(C)C2)=O)CCN(C(=O)CCC(=O)c2ccccc2)CC(C)(C)C1 c1(C(N2C(C)CC(NC(=O)C=Cc3ncc[nH]3)C2)=O)cc(F)cc(Br)c1O C1(CC)CCCCC1C(=O)NC1(CO)CN(C(c2cc(C3(O)COC3)on2)=O)C1 C1(CNC(Cc2cnc(C)s2)=O)(CO)CCN(C(c2sccc2C)=O)C1 c1(C(=O)NCC2C3CN(c4ncc(C)cn4)CC32)ncc(Cl)cc1F c1(C(N(CCNC(=O)CCc2ccon2)CC)=O)c[nH]c2ccc(F)cc2c1=O C1(CNC(COC2CCN(C)CC2)=O)CCCCCN1C(=O)CCc1cccs1 N1(C(c2c(C)onc2)=O)CCCC2(C1)CN(C(C1CCCN1C=O)=O)CCO2 C(CCCCCNC(=O)Cc1cc[nH]c1)N(C(=O)CC1CC1(C)C)C O=C1CCC2(CC1)C(=O)NCCN2C(=O)NCCCc1ccc(Cl)cc1F c1(NC(=O)OC)ccc(C(N2CCC(NC(=O)CCSC)C2C2CC2)=O)cc1 c1(OC)cc(Nc2nc(CCCO)nn2-c2ccnc(Cl)c2)nc(C(F)(F)F)n1 c1(CC)ccc(F)c(C(=O)NC2(COC)CCN(C(=O)CCN3CCCC3)C2)c1 CCCCS(=O)(=O)NC(C)C(=O)N(CC(C)NC(=O)COCCOCC)C c1(N2CC(CN(C(c3c(C)cn(C)n3)=O)C)OCC2)cc(C(N)=O)nc(Cl)n1 C1(CNC(=O)CC2CCSCC2)CCCCN1C(=O)CC1CCCCC1 c1(NC)snc(C)c1C(=O)NCC1CCCCN1C(=O)CSC(F)F N1(C(c2c(C(C)C)occ2)=O)CC2C(NC(C3C4CN(C)CC34)=O)C2C1 C(C(=O)NC1(CNC(C2CC(CC)=NO2)=O)CC1)(C(C)C)SCC c1(C(=O)NCC2(C)CN(C(C3CN(C(CC)C)C(=O)C3)=O)C2)cc(Cl)ccc1Br c1(CNC(C(C)N(C(COCC(=O)OC)=O)C2CC2)=O)cccc(F)c1F CC(C)CS(=O)(=O)CC(=O)NC1CS(=O)(=O)CC1NC(C1CCCC1)=O CC(C)(C)C(CNC(=O)NCCc1ccc2[nH]ccc2c1)C(F)F N=c1ccc(C(=O)NC2(CNC(=O)Cc3cc(C(F)F)on3)CCC2)c[nH]1 C(N=c1nc(N2CCC(OCCF)C2)c2c([nH]1)CCCCC2)C1(P(C)(C)=O)CC1 CCCC(C)(O)C(=O)N1CC(CCNC(=O)COc2cccc(C)c2)(OC)C1 c1(C(=O)NC2C(C(N3CCc4c(nc(C)o4)C3)=O)C2)c(F)c(F)c(F)c(F)c1F C(=O)(CCCC(=O)OC)N(CCCOCCN(C(C1CC(=C)C1)=O)C)C C1(NC(C2C(=C)C2)=O)CCC2CC1CN2C(=O)CCc1ccc(N(C)C)cc1 c1(C(=O)NC2CC(N(C(C(C=C)O)=O)C)C2)cc(OC)cc2c1CCC2 C1(C#N)(C(=O)NCCC(C)NC(=O)CC2CCCN2C)CC1C(F)(F)F c1(CN2CC(CNC(Cc3c(C)noc3Cl)=O)C2)nc2c(s1)CCCC2 c1(C(=O)NC2CCCC2CNC(C2(c3ccno3)CCC2)=O)cc[n+]([O-])cc1 c1(C(=O)NCC=CC(=O)NC(c2ccccc2O)C)ncc[nH]c1=O N1(C(c2ccc(OC)cc2)C(=O)NC2CC(F)(F)C2)CCCC(C)(O)CC1 N1(C(Cc2onc(C)n2)=O)CCCC(N(C(=O)CC2CC2(C)C)C)CC1 C1(F)(CNC(C=C(CCC)C)=O)CCC(NC(c2cc[nH]c2CC)=O)C1 N1(C(CC=C(C)C)=O)CCN(C(C2CC(F)C(=O)N2)=O)C(CCO)C1 N1(C(C(CC=CC)NC(=O)CN(C)C(=O)C2CC2)=O)CCOC(C)(CC)C1 c1(C(=O)NCC(C)NC(c2c(COC)cccn2)=O)cncc(Cl)c1C c1(OC)ccc(C(=O)NC(C2CCN(C(c3cccnn3)=O)C2)C)nc1Cl C1(NC(c2ccc(Cl)o2)=O)CCC2CCN(C(C3C4CNC(=O)C34)=O)C1C2 N1(C(C2C3(CC(NC(COCC=C)=O)C3)C2)=O)CCC2(CC1)CC2CO C1(NC(c2scc(C)c2Cl)=O)CCC2CN(c3cnc4ccccc4n3)CC2C1 C(C(C)(C(=O)NC1CCC(C(=O)N(C)CC2CCCC2(C)C)C1)OC)OC N1(C(c2c(C)noc2N)=O)CC(CNC(=O)C(C)OC2CCCC2)CC(C)(C)C1 Cc1nc2ccnn2c(C)c1CCC(=O)NC(CNC(=O)CNS(C)(=O)=O)CO C(=O)(C(F)(F)C(C)(C)O)N1CCC(C)C(NC(=O)C(O)Cc2cnn(C)c2)C1 c1(OC)c(C(=O)NC(C)C(C)NC(=O)CCOC2CCCC2)cnn1C C#CC1CCN(C(=O)Cn2cc(CNC(C3CC3Cl)=O)nn2)CC1 c1(CNC(C2CCN(C(C(N3CCC(C)CC3)=O)=O)C2)=O)cnn2ccncc12 Cc1oc(CNC(C2(O)CC2)=O)nc1C(=O)NC1CCOC1C C1(NC(C(C=C)(C)C)=O)CC(C(=O)N(C)CCOC(F)F)=CC1O N1(CCC(C)C)CCCC1C(=O)NC1CC1CNC(c1ncnn1C(C)(C)C)=O O(N(C)C(=O)CN=c1nc2c(cnn2C)c(N2CC3CCOC3C2)[nH]1)CC N1(C(C(C2CN(C(C3CCc4cnnn4C3)=O)C2)OC)=O)CCC(C)C(C)(C)C1 N1(c2nccc(CC(=O)OC)n2)CC(C)CN(C(=O)CC(C)(O)COC)CC1C CC1CCC(CC(=O)N(CC(=O)NCc2ccnn2CC(F)F)C)O1 N1(C(c2c(CC)nn(C)c2)=O)CC2CCC2(CC(N2CC3C(CO)C3C2)=O)C1 c1(NC(C2(C)CCN(C(Cn3ncn(C)c3=O)=O)C2)=O)ccc(O)c(F)c1 N1(C(C2C(C)(C)C(=O)C2)=O)CC(NC(=O)CCCCCF)CC2(CC2)C1 C=C1CC2(C1)CC(C(=O)NCCCOCCNC(=O)C(C1CCOCC1)C)C2 C1(C2CN(C(=O)C(c3ccc(Cl)cc3)O)C2)(NC(=O)CC2CCC2(F)F)CC1 C1(C(=O)NC(CC)CNC(=O)Cc2cnco2)CC=C(C)CC1 C1(NC(CCc2c(C(=O)OC)nco2)=O)CCN(C)C(=O)C1 CCCCC(O)C(=O)NCC1CCCC1C(=O)Nc1ccc(Cl)c(CO)c1 c1(C(N2CCC(C)(CNC(C3(CF)COC3)=O)C2)=O)cccc(Br)c1F C(=O)(C1CCCn2ccnc21)N1C2CC(NC(=O)CSc3ccccc3)C2CC1 c1(CC(=O)NC2CC(C)(NC(CCOC)=O)C2)cnc(Cl)cc1C C1(CCCNC(c2cc(Br)n[nH]2)=O)CCCCN1C(c1cn[nH]c1)=O Cc1c(CNC(C2CC(C)(F)C2)=O)sc2cncn12 N1(C(C)C)C(=O)NC(c2cn(C)c3cccc(Cl)c23)C2=C1CN(C(C)(C)C)C2=O C1(C(F)(F)F)(C(=O)NCC2N(C(c3cnc[nH]3)=O)CC=C2)CC=CCO1 O=[N+]([O-])c1cnn(C2CCCC2)c1NCCCc1ccc(C(F)(F)F)c(F)c1F c1(CNC(C2CN(C(=O)CCN3CCCC3)CCO2)=O)cc(Cl)nc(Cl)c1 c1(COC)ncc(C(=O)NCC23CCC2CCN3)cc1Cl C1(C)(CNC(C(CCC=C)C)c2nnnn2CCCSCC)CCS(=O)(=O)CC1 c1(N2CC(COCCOC)OCC2)[nH]c(=NCC(CO)C2CC2)nc2sccc12 C1(NC(N2CCCC(O)(Cc3n(C)ccn3)C2)=O)CCC2CCC1OC2 c1(N(c2cccc(C(F)(F)F)c2)Cc2c(C)cn(C)n2)ccc(O)c(COC)c1 C=C1CC2(C1)CC(C(=O)OCc1ccc(CNC(=O)OC(C)(C)C)[nH]1)C2 C(CCCC(C)(C)C(=O)NNC(=O)C(C)C(C)NC1CC1)NC(CSCC)=O C(C#Cc1cn(C(c2nccc(F)c2Cl)(C)C)nn1)NC(C(CC(C)C)=O)=O N1(C(CCC#CC)=O)CCC=C(CNC(c2cnc(C)nc2)=O)C1 N1(C(CC(CC)(C)C)=O)CC2CC1CCN2C(=O)C(C)Cc1cnn(C)c1 N1(C(C(N2CCOCC2)C)=O)C2CCC1CC(CNC(=O)CC1CC(F)(F)C1)C2 C1(CNC(c2nc(CCCCC)sc2)=O)CN(C(=O)CCC(C)SC)CCO1 C1CS(=O)(=O)CC(=O)O1.c1(C(=O)OC)ccc(C)c(OCc2cnn(C)c2)c1 N1(C(c2n(C=C)ncc2)=O)CC(C)(C)OC2(C1)CN(C(=O)CCC(=O)NC)C2 Cc1nc2cc(C(=O)NC(c3cn(Cc4csc(C)n4)nn3)C)c(F)cc2[nH]1 Cc1cc(N)n(CC(=O)NC2(CNC(C3CC4C=CC3C4)=O)CC2)n1 Cc1scc(C(=O)NCC(C(C)C)NC(=O)C(N2CCOC2=O)C)c1C1CC1 C(=O)(C1=CC2(CCOC2)C1)NC1CC(OC)CN(C(C2CCCO2)=O)C1 C1(C(=O)NCCCCNC(CCC(C)(C)OC)=O)CC2CCCCN2C1 c1(OC)cnc(CNC(c2ccccc2-c2cccnc2O)CC(=O)O)nc1 N1(C(c2cccc(C(=O)NC)n2)=O)CCCC(NC(C2(Cl)CC2(F)F)=O)CC1 c1(OC)c(N(C2CCN(C(c3ccc(Cl)nc3Cl)=O)CC2)C)ncnc1C Cc1nn(C)cc1S(=O)(=O)N1CCN(c2cc(NCc3ccsc3)ncn2)CC1 c1(C(=O)NCC(CO)NC(c2c(C(C)C)onc2)=O)ccc2c(c1)OCC(=O)N2 N1(C(C2ON=C(C)C2)=O)CCC2(C1)c1ncn(C)c1CCN2C(=O)CC1CC1C C#Cc1cc(C(=O)NCC2CN(C(=O)Cn3ccccc3=O)CCO2)ccc1C C1(C)(C(N(C2CC(NC(=O)CS(=O)(=O)C3CC3)C2)C)=O)CCCNS1(=O)=O CCC(CC(F)(F)C)C(=O)NC1CCSC12CN(C(C1CCSC(C)C1)=O)C2 C1(c2cn(C3(C(=O)OC)CN(C(C4(CO)CCO4)=O)C3)nn2)CC2(CC(=O)C2)C1 C#CCC(CC(F)F)C(=O)N1CCC2(CCC2NC(=O)CC2CCOC2)CC1 Cc1ccc(C(C)N(C(c2[nH]nnc2C)C(=O)NC(C)C)C)cc1 C1(CC)(NC(c2nocc2Cl)=O)CCCN(C(=O)COC2CCCCCC2)C1 S(=O)(=O)(c1cnc2c(C#N)cnn2c1)N1CC(C(N2C(C#C)CC3(CC3)C2)=O)C1 c1(C(=O)NCC(C)CNC(=O)CC(C)n2cccn2)ccc(Cn2cccn2)o1 CC1C(NC(c2cnn(C3CC3)c2)=O)CCN1C(C1CCCSC1)=O C1(C)(CNC(C2C(C(N(c3ccccc3)CC=C)=O)CCC2)=O)CCC(C)CC1 N1(C(C(C)N2CCCC2)=O)CC=CC1(C)C(N1CCC(c2cnco2)C1)=O C1(C(=O)NC23CC(CNC(CC4C(C)OCC4)=O)(C2)C3)CN2CCC1CC2 Cc1cc(NC(C2CC(F)CN2Cc2nc(C)c(C)nc2C)=O)cc(C)c1C C1(C(C)C)(NC(=O)C(C2(O)CN(C(=O)COC3CCC3)C2)F)CCCC1 C1(C(=O)NC(C)CCNC(c2cc(N)c(F)cc2F)=O)Cc2ccc(F)cc2O1 CC(CCNC(c1cc(CNC(C2CC3(CCCO3)C2)=O)no1)=O)C(F)(F)F C1(C)(C(=O)Nc2scc(-c3cc(C(=O)OC)c(C)o3)n2)CCC(C)=C(C)C1 N1(C(=O)NC(c2cccc(OC)c2)CC)CC2CC1CN2C(=O)C=C(C)C(C)C CC1(NC(c2cnc[nH]2)=O)CCCN(C(c2c[nH]c(C#N)c2)=O)C1 c1(C(=O)NC2CCC(N(C(=O)CC3CC(C)(C)CO3)C)C2)cc2ncccc2o1 C(=O)(C1=NOC2COCC12)N1CC2(CN(C(C3(C(=O)OCC)CC3)=O)C2)C1 C1(N(C)C(c2nn(C)cc2Cl)=O)CCCC2CN(C(C34CC(F)(C3)C4)=O)CC12 c1(CCNC(C(C)(C)C(C)C)=O)ccc([N+](=O)[O-])cc1Br CCC(C)C(O)C(=O)N(CC(C)CNC(c1ccnc(CO)c1)=O)C c1(C(=O)NCc2nc(C)c(C(N3CCC(OCCO)C3)=O)o2)ccc(=O)n(C)c1 C1(NC(Cc2cc(C)nn2C)=O)CC(F)CN(C(c2cncn2C(F)(F)F)=O)C1 C1(C(C)NC(c2ccoc2)=O)CCN(C(c2csc(-c3cccnc3)n2)=O)CC1 C=CC(C)CC(=O)N(C(C)C(=O)NC1CC(N(C)C)C1)C C1(NC(c2cnc(OCC)nc2)=O)CN(C(C23CC(CC(C)O2)C3)=O)CC1(C)C c1(C(CO)NC(CONC(c2cc(CCC)[nH]n2)=O)=O)c(C)cccc1Br C1(NC(CC2CC(C)(C)C2)=O)C2CC1N(C(c1ccccc1F)=O)C2 CCC(C)C(O)CC(=O)NC1CC(C(=O)NCC2(C)CCN(C)C2)=CC1O C=CCC(C(=O)NC1CCN(C(=O)CC2CCOCC2)C1CC1CC1)C(C)C c1(CC(=O)NC2CC(NC(CN(C)C3CC3)=O)C2)cc(C(F)(F)F)ccc1Cl c1(C(=O)NC2CCC(C)N(C(c3ccc(Cl)s3)=O)C2)ncc2c(F)cccn12 c1(-c2cc(C(c3ccc(F)cc3)OC)sc2)nnc(CCc2ccccn2)n1N c1(OC)ccc(-c2nc(C3CCCN(C(C)=O)C3)n(CCS(C)(=O)=O)n2)nc1 c1(C(C(C)NC(=O)CN2CCC(c3nncn3C)C2)OC)ccc(F)cc1 c1(CC(=O)NC(C2(O)CN(C(=O)Cc3ccnc(F)c3)C2)C)ccc(F)cn1 C1(C(=O)NC2(CO)CN(C(CC3(CO)CC(C)(C)C3)=O)C2)CC12CCCCC2 c1(NC)nn(C)cc1C(=O)NCCN(C)C(c1cc(C(=O)OC)no1)=O CC1CCCCC1(CNC(=O)COc1ccsc1)NC(C1CC(n2cnnc2)C1)=O Cc1nc(Cl)[nH]c(=NC2CCC3CN(C(c4ncc(F)cn4)=O)CC23)c1[N+](=O)[O-] c1(C(C(=O)NC)N(C)Cc2nnc(C(C)(C)C)o2)ccc(C)cc1 N1(C(c2cnc(CCC)s2)=O)CCN(C(c2coc(C(N)=O)c2)=O)C(C)C1C C(C(=O)NCCOC1CN(C(=O)C(C)COC)C1)(C(C)C)NC(CC)=O N(S(=O)(=O)N1CCC(C)CC1)CC(N1CC(C)OC(C)C1)C C(=O)(C(F)C(F)(F)F)NCC1C(NC(c2cnc(=N)[nH]c2)=O)CC1 c1(C(C(=O)NCCN(C(CNC(C(CC)C)=O)=O)C2CC2)C)ccc(F)cc1 C(C(=O)NOCCCCF)(c1ccoc1)NC(=O)CCCC1CCCC1 c1(CC(=O)OC)ccc([N+](=O)[O-])cc1Br.C1(=O)C(=O)CCO1 c1(C(CNC(=O)C(C)O)NC(C2(C#C)CCCC2)=O)ccc(OC)cc1OC N1(C(c2cc(C)cc(Cl)n2)=O)CC(F)C(N=c2ncnc3[nH][nH]c(I)c2-3)C1 c1(C(C)C)ccc(C(=O)NC2CCC(CNC(=O)C(O)C3CCCC3)CC2)nc1 N1(C(Cc2scc(C)c2)=O)CCC(C(O)CNC(C2CC(C(F)F)C2)=O)CC1 C1(C(N2C(Cn3cc(C(C)(C)NC(N)=O)nn3)CCCC2)=O)CC(S(C)(=O)=O)C1 C(C(=O)Nc1cncc(C(=O)NC2CCCN(O)C2=O)c1)(C(C)(C)C)OC C=CCCC(C)(C)C(=O)N1CC(CN(C)C(c2csc(C(C)=O)n2)=O)C2(CC2)C1 C1(C(=O)NC2(C)CC(NC(=O)C3=CCCOCC3)C2)CCN2CCCC2C1 c1(CC)ccc(NC(c2cc(OC)ccn2)=O)cc1.C12(F)CN(C1)C2=O C(=O)(CCS(=O)(=O)N(C)C)N(C)CC1CCCN(C(C2(N(C)C)CC2)=O)C1 c1(CC(=O)NCC(C(=O)NCC(C#C)CC)OC)ncccc1C C(=O)(CCCCCN(C)C)NC(CNC(c1c(-c2ccc(C)o2)onc1)=O)(C)C c1(C(N2CCN(C(CN(C(CSC)=O)C)=O)CC2)=O)ccc(O)c(F)c1 N1(C(c2cc(CC)c(=O)n(C)c2)=O)CCOC2(CCN(C(c3cscn3)=O)C2)C1 c1(CC(=O)NCC2(CNC(CSC)=O)CCCCC2)ccnc(F)c1F c1(CNC(c2cc(-c3ccccc3)cs2)=O)cccc2c1CNC2 N1(C(c2ccc(NC)cn2)=O)CCC(C2CCN(C(c3snc(Cl)c3Cl)=O)C2)C1 c1(C(=O)NC(C(=O)N(CC(=O)OC)CC)CC(C)C)cccn2nccc12 C1(C(N(CC(C(C)C)OC)C)=O)(OC)CCN(C(=O)C(C)Cn2ccnc2)C1 C(=O)(C1CCCCc2ccccc21)NC1(C(C)NC(=O)C2=CCCCC2C)CC1 C1(C2CCN(C(=O)C(F)C3=CCCCC3)C2)(NC(C=C(C)C(C)(C)C)=O)CC1 C1(COC)(CN)CN(C2CCC(Oc3ccncc3)C2)CCO1 N1(C(C(C(C)C)CO)=O)CCC2(CC1)CCN(C(=O)CCc1ccc(F)nc1)C2 Cc1sncc1C(N1CCC(N(C)C(c2cc(C3CC3)no2)=O)C1)=O C1(NC(c2cccc3c2CCCN3)=O)CC1C1CCN(C(=O)CC2CCC2)CC1 N1(C(c2cc(CC(C)C)nn2C)=O)CCCC(O)(CNC(C2(C)CCOC2)=O)C1 c1(NCC2CCCN(C(c3c(N(C)C)cccc3)=O)C2)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC(CNC(C=C(C)Cl)=O)C3C2C3)=O)cc2ncccc2[nH]1 C1(NC(C(F)=CC)=O)CCCN(C(c2ccc(C)c(N)c2)=O)C1C c1(C(=O)NCc2cccc(C(=O)NC(C#C)CC3CCC3)n2)c(C)cnnc1O N1(C2N(CC3(CC)CC3)CCS2)CCCC(C(=O)NCCNC(=O)C(C)=O)C1=O C1(C)COCC2(CCN(C(=O)O)CC2)O1.CC(C)CC(C)(C)C.C1C(=O)N1C1CC1 c1(C(N(C(C)C)CCNC(c2cc(Cl)ccc2Cl)=O)=O)cnn2cccnc12 C1(NC(C(COC(C)(C)C)NC(C2(O)CCCN(C)C2)=O)=O)COC2(CCOCC2)C1 C1(C(=O)NCC2C(C(=O)NCc3c(C)nsc3)CCC2)(CO)CCCCO1 CC(CCCCNC(C1CCCN1C)=O)NC(c1c[nH]nc1N(C)C)=O c1(OC)ccccc1NC(=O)C(N1CCCC1CC(N)=O)C1CC1(C)Br C(C(=O)O)(C1=CCC2CC2C1)NCC(c1nccs1)C Cc1ccc(C#N)cc1NC(C1C2CCC(C2)C1NC(c1ccc(O)nc1)=O)=O c1(C(=O)NCC(C)(C)NC(c2cncc(-c3ccoc3)c2)=O)cc(F)cnc1O C12(CNC(c3ccc(C)nc3N)=O)CCC(CC1)N(C(C1CSCCS1)=O)C2 c1(C(=O)NC(C2(CNC(C(C)NC(CC)=O)=O)CC2)C)cc(C)ns1 Cc1cccc2c1CC(C(=O)OC(c1cnccn1)Cc1ccccc1)N2 Cc1[nH]nc2c1CCC(C(N1CCN(C(c3ccc4c(c3)OCC4)=O)CC1)=O)C2 C1(O)(CNC(=O)COCC2CCOCC2)CCCN(C(C2CC3CC2CO3)=O)CC1 c1(C(N2CCC(N(C(=O)CN(C)CC)CC#C)CC2)=O)cccc2nc(C)nn12 N1(C(c2c(C)ccc(SC)c2)=O)CCC2(COC(CNC(=O)CSC(F)F)C2)C1 C1(CNC(=O)Cn2cccnc2=O)CC2(CC2)CN1C(c1cnn2c1OCC2)=O c1(NC(C2C3(CC(NC(C(=O)NCC)=O)C3)C2)=O)ccc(O)c(F)c1 C1(CNC(C2CC3(C2)CC3F)=O)CCCC2(CN(C(c3nncs3)=O)C2)O1 N1(C(C)NC(c2nscc2C)=O)CCC(NC(C2(C(=O)NC(C)(C)C)CC2)=O)CC1 c1(C(=O)NCC2C(C)(C)CCC2)cc(F)cc([N+](=O)[O-])c1 N1(C(c2n(CC(C)C)ncc2)=O)CCN(C(=O)C(C)O)C(CC(F)(F)F)C1 C(=O)(CC(F)(F)C(F)(F)F)NC(CC=C)CNC(c1cccc(C)c1N)=O C(C(CC1CC1)C(=O)NCc1cccc(C2CC2)c1)NC(C(C)C)=O CC1CN(C(=O)C(F)(F)c2csc(Cl)n2)CC1NC(=O)C(F)CC1CCCCC1 N1(C(c2c(C)cnnc2)=O)CC(F)(F)CC1(C)CNC(=O)C(c1ccnn1C)O Cc1cc(C(F)(F)C(=O)N(CC(C)N(C(=O)C(C)N(C)C)C)C)cnc1Cl N1(CCC)C(=O)NC(c2cccc(F)c2)C(C(=O)NCCOC)=C1C c1(OC)cc(C)ccc1NC(=O)NCCOCCSC N1(C(C(F)=CC)=O)CCC(C(C)(O)CNC(c2ccnc(C(F)F)c2)=O)CC1 CCCC(C(=O)N(CCCCN(C(=O)C(=O)C=Cc1cccs1)C)C)NC(N)=O c1(C(=O)OC)sc(=NCC2(O)CCCN(C(C3CC3CCN(C)C)=O)C2)[nH]c1Cl C(CN=c1[nH]c(=NCCC2CC2)[nH]c2cc[nH]c12)=CCOC c1(C(=O)NCCNC(C23OC(C)C(CC2)C3)=O)cc2nnn(C)c2s1 C12(C(=O)NC(C)(C)CCF)CCC(NC(=O)CC(Cl)Cl)(CC1)C2 N1(C(CC(C)C2CC2)=O)CC2(CCC(NC(C3CCC(C)(C)O3)=O)CC2)C1 O=C(CN=c1cc[nH]cc1)N1CC2CN(C(=O)C(Cl)=CCl)CC2C1 c1(OC)cccc2c1OC(c1nc(CS(=O)(=O)NC)no1)C2 c1(C(N(C2(C(=O)NC3(CC=C)CC3)CC2)C)=O)cc(CC)[nH]n1 c1(C(N(C(CCNC(c2c(C)noc2)=O)C)C)=O)cccn(SC(F)(F)F)c1=O Cc1nc(C(=O)N(C(C)CN(C)C(c2cc(C(F)F)on2)=O)C)c(C)o1 C#CC1(N)CCCCCC1.C(N=c1ccnc(CO)[nH]1)C1(C(C(CC=C)(C)C)=O)CC1 CC1CCN(C(c2cn(C)[nH]c2=N)=O)CC1C Cc1ccnc(C(N2CCOC(CN(C(=O)C(C)C(F)F)C)C2)=O)c1F C1(NC(=O)CCCF)CCC2(CC1)CCN(C(C13CC1COC31CCC1)=O)CC2 c1(C(N(C2CN(C(C(C(C)C)SC)=O)C2)C)=O)cc2ccc(Cl)cc2c(=O)o1 C1(CNC(C=CC=CCC)=O)(COC)CCN(C(c2cnccn2)=O)C1 c1(CNC(CC2CCN(C(C3(C)CCOCC3)=O)CC2)=O)cc(Cl)ccc1O n1(CC(N2C(NS(CC(=O)OCC)(=O)=O)C=CC2)=O)nc(Cl)ccc1=O N1(c2cc(N3C4CC(N(C)C)C4CC3)ncn2)CCCC(N=[N+]=[N-])C1 CCCCCC(O)C(=O)N(CC(C)CNC(=O)CCCCO)C N1(C(c2cc(NS(C)(=O)=O)sc2)C(=O)NCCCC2CC2)CCS(=N)(=O)CC1 C1(O)(C(C)NC(CNC(CC(C)C)=O)=O)CCN(C(C2CC2(Cl)Cl)=O)C1 N1(CC2CCCC(C)(N)C2)CCCc2cc(NC(=O)C(F)(F)F)ccc21 N1(C(C=Cc2n(CC)ccn2)=O)CCC(C)CC1CNC(c1c[nH]nc1F)=O c1(NC(C(=O)N(C(C)C)C2CC2)=O)cc(F)ccc1N1CCOCC1 CCCC(C)CC(=O)NC1CC1CNC(c1cccc(NC(N)=O)c1)=O c1(C2C(C(N(C3CCC(NC(=O)COC4CC=CC4)C3)C)=O)C2)ccccc1F CCCCC(CC)CCC(=O)NC(C)CNC(=O)CCn1ccnn1 O=C(CCCCCNC(c1cccs1)=O)NCCc1ccc(O)nc1 c1(C(=O)NCC(CNC(c2cc(CC)ncc2)=O)F)cc2ccc(Cl)cc2s1 c1(CCNC(CN(c2ccccc2)C(C=C)C)=O)snnc1C C1(CNC(=O)Nc2c(C(=O)OC)ncc(Br)c2)CCCCC(F)(F)C1 CC1(C)CC(NC(=O)CC2(NC(c3ccccc3)=O)CCC2)CC(C)(C)N1 c1(CNC(c2ccc(F)c(I)c2)=O)ccc(C(F)F)c(Br)c1 C1(NC(CC(C)c2ccco2)=O)CN(C(=O)CC2CC=CC2)CC12CC2 CCC(C)(C(=O)N1CCC(NC(c2c[nH]nc2OC(C)C)=O)C(CO)C1)C(N)=O CC1(C)NC(=O)CC1C(N1CCC(C(=O)NCC2=CCCCC2)C12CC2)=O Cc1c(NCCCNC(=O)N(C)C)ncnc1N1CCN(C)C(c2ccccc2)C1 C(N=c1[nH]c(=NCC2CCOCC2)c2[nH]ccc2[nH]1)c1cn[nH]c1 N1(C(CCCc2c(C)ccs2)=O)CCC(C2CC(NC(=O)CCC(C)C)C2)C1 c1(C(=O)NC2CC3CN(C(=O)CC(F)F)CC3C2)cc2ccccc2c(O)n1 C1(NC(C2CCN(C(CC)=O)C2)=O)CCC2(CC1)CC2NCCCNC(C)=O O=C(C1=NOC2(CCN(Cc3cc(Cl)cnc3Br)C2)C1)Nc1cc(Br)ccc1Cl C1(NC(CCC)=O)(CC)CCCN(C(=O)CC2CCC(F)(F)CO2)C1 C1(C(=O)NCC2C(C)(C)CCN2C(=O)C=CC2CCC2)CCC2(CC1)CC2(F)F c1(C(N(C)CC2N(C(CCc3ccc(C)o3)=O)CCC2)=O)nnc2n1CCCC2 CCCC(CCCNC(=O)CC(=O)NCC)N=c1[nH]nc(C(F)F)o1 C1(CC(=O)NCc2cc(C(C)C)no2)CC(NC(=O)C(F)C2CCCC2)C1(C)C C1(NC(C2(CC)CCC2)=O)CC2CC1CN(C(C1(CF)CC1)=O)C2.C(C)=O N1(C(C2CC(CN)CN(C(C)=O)C2)=O)CCC2(CCCNC2=O)CC1.CO N1(C(C2(F)CC(C(=O)OC)C2)=O)CC(CNC(c2cn(C3CC3)cn2)=O)C(C)C1 S(=O)(=O)(c1cc(C(=O)O)[nH]n1)NC(CNC(CC)C)=O CCC(CC)(CCNC(c1cc(C2CC2)cs1)=O)NC(c1oc(C)cc1C)=O Cc1ccc(F)cc1CC(=O)NC1CC2CCC1N2C(=O)Cc1ccon1 c1(C(=O)OC)cc(Br)cc(I)c1NC(=O)CC1COC(=O)N1 C1(NC(C2CC2(F)F)=O)CC1C1CCCN(C(=O)C=CC2CCOCC2)C1 c1(C(N(C(CNC(C(C2CC2)SC)=O)C)CC)=O)ccc(Cl)c(C)c1 C(c1nc(C)c(C)[nH]1)=CC(=O)NCCC1(O)CCN(C(C2C(C=C)CC2)=O)C1 C(=O)(C1=CC(O)C(NC(=O)CCCC2CCCC2)C1)NCC1CCC(=O)NC1 C1(c2nnnn2CC2CCCOC2)(NCC2(CC#N)CC2)CCSC1 C1(NC(c2c(OC)c[nH]n2)=O)CCCN(C(=O)Cc2ccsc2C)CC1 c1(OC)cc(OC)c(C(=O)NCCCN(C(=O)C(C)C2CCOC2)C)c(F)c1 C1(C(=O)NCC(C)(O)C2CCCC2)CCCCN(C(=O)CCCCC2CC2)C1 c1(C(C(=O)N(C(C)CNC(C2CC(C)(F)C2)=O)C)OC)ccc(Cl)cc1 c1(CC(=O)NCCCN(C(C(CC2CC2)OC)=O)C)ccc2nn[nH]c2c1 c1(OC)nccc(C(=O)NC2CCCC2CNC(C2(OC)CCC2)=O)n1 C1(C(=O)NC(C2(OC)CCC2)C)C2CCN(C(c3cc(O)cc(F)c3)=O)CC12 C1(OCCCNC(C(CC)n2ccnc2)=O)CCN(C(C2(C)C=CCC2)=O)CC1 c1(C(=O)NCC(C)NC(C(F)=CCC)=O)cccc2c1CCC2 C1(N(C)C)CN(C(C2(F)CCCC2)=O)CC1CNC(=O)CC1CCC(=O)CC1 C(CC(=O)N1CCOCC1CC1CC1)(C(F)(F)F)NC(=O)C(F)OC(F)(F)F C1(C2C(CN(C(CCC3CC(C(=O)OCC)C3)=O)CC(C)O)C2)CSCCO1 C1(NC(CC2CC(=C)C2)=O)CCC(NC(c2ccco2)=O)C1 c1(C(N(CCC)CCNC(=O)C(CC)CC)=O)cc(CNC(N)=O)ccc1Cl O=S(=O)(c1ccc(NC2CCCCC2)cc1Br)N(c1ccccn1)CC(Cl)(Cl)Cl c1(CCN=C(NC(CC)CC)NCC(C)C)c[nH]c2cc(Cl)cc(Cl)c12 c1(C(N2CCC(NCc3ncn(C)c3)C(C(=O)O)C2)=O)cc(I)c(F)cc1F CCCC(C#N)C(=O)NCC1(CCNC(c2nccc(C(=O)NC)c2)=O)CC1 N1(C(CCOCCC)=O)C2CCC1CN(C(C1CC=CCO1)=O)CC2 c1(C(=O)NCC(CN(C(=O)Cc2ccon2)C)O)ccc(OC(F)(F)F)cc1F N1(C(c2c(C)con2)=O)CCCN(C(c2cccc(C(=O)N(C)C)c2)=O)CC1C N1(C(C(c2cccc(C)c2)O)=O)CC2(CC(NC(C3(C)CC3C)=O)C2)C1 C1(O)(C(=O)NCC2CCN(C(=O)CCc3nccs3)C2)CN2CCC1CC2 Cc1ccc(O)c(CN2CCC(F)(C(=O)NCc3cccc(F)c3)C2)c1 CC1=C(C(=O)NCc2nc(C(=O)NCC3(CO)CCCCC3)c(C)o2)COCC1 C1(C(=O)OCC2N(C(C(C)O)=O)CCCC2)CC2(CCC2O)C1 c1(CNC(C(C=C)O)=O)ccc(CC(C)NC(c2csc(CC)n2)=O)cc1 C1(NC(C(CC)SC)=O)CC(F)CN(C(=O)CC23CCCN2CCC3)C1 c1(N2CCC(CCNC(=O)C(c3ccc(Cl)c(Cl)c3)O)CC2)nc(Cl)ncc1Cl Cc1nc(C(=O)NCCNC)c(C)o1.c1(C=O)cnc(C2CC2)[nH]1 N1(C(C(N)=O)=O)CC2(CNC(=O)CC3COC(=O)C3)CC1CCO2 c1(NC(C(N2CC(CC)OC(C)C2)=O)=O)ccc(S(C)(=O)=O)nc1 C1(C(N(CC(CC)NC(=O)C(S(C)(=O)=O)C2CC2)CC)=O)CCC(O)CN1C C1(NC(C2C(C)CCO2)=O)CC(F)CN(C(C2CC(C)CCO2)=O)C1 C1(CC(=O)NC2CC(CNC(C(CC)(C)C)=O)CC2O)CN2CCN1CC2 C1(NC(CC(C)OC)=O)CN(C(c2ncncc2Cl)=O)C2(CCOCC2)C1 N#Cc1ccc(Cc2noc(C3CC(OC(F)F)C3)n2)cc1 C1(C(=O)NC(C2CCCC2)C)CCCN1C(=O)Cc1cnn(C)c1 c1(C(=O)NCC(CN(C(=O)CCc2cncs2)C)O)ncn2ccccc12 CC(C)(C(=O)N1CCC(N(C(=O)Cc2cc[nH]c2)CCO)C1)C1CCOCC1 C(CCS(C)(=O)=O)(C(=O)NC(C)(C)CN(C)C(C1CC1C(C)(F)F)=O)OC N1(C(c2c(C)nc(C(N3CCCC(C(C)C)CC3)=O)o2)=O)CCCC(CC)C1C C1(NC(C(C)O)=O)CS(=O)(=O)C12CCN(C(C1Cc3cncn3C(=O)N1)=O)CC2 c1(C(C(=O)NCC2(F)CC(CNC(CC(C)SC)=O)C2)=O)ccc(F)cc1 N1(C(C2CN(C(C)=O)C2)=O)CC2(C(=O)NCCOCCO)CC2(C(F)(F)F)C1 C1(NCc2c(C)nn(-c3ccccc3)c2Cl)CCCNCCC1(F)F CC1(C)CC(CC(=O)NC2(C)CC3(CC3)C2)N(C(=O)C2=COCCC2)C1 c1(C(N2CC(N(C)C(c3cc4sccc4n3C)=O)C2)=O)ccc([N+](=O)[O-])cc1F C(=O)(C(F)(CNC(c1nonc1CC)=O)C(C)C)NCC(CCC)(C)O C1(NC(=O)NC2CC(CN)C2)CCC2C3C=CC(C3)C12 C(CC(C)C)(C(=O)NC1CN(C(C2(F)C(C)(C)C2(C)C)=O)CCC1CO)NC(C)=O C1(NC(Cc2nc(CC)sc2)=O)CCCCN(C(c2cnc(CC3CC3)s2)=O)C1 c1(C(=O)NCC(c2c(OC)cccc2)C)ccc(Br)c(C)c1C C1(C(C)NC(CCSCCCC)=O)CCCN(C(=O)CCc2csc(=N)[nH]2)C1 C(=O)(CS(N)(=O)=O)N(C(C)CNC(=O)C(c1cscn1)N(C)C)C c1(CC)nc[nH]c1C(N1CC(O)(CN(C(=O)Cn2cc(C)cn2)C)C1)=O C1(NC(Cc2scc(CC)n2)=O)CC2CCC1N(C(C1CC(=O)NC(=O)C1)=O)C2 c1(C(=O)NC2CCCC(NC(Cn3nc(C)oc3=O)=O)C2)cc([N+](=O)[O-])oc1C CCC(C)C(O)C(C)C(=O)NC(CC(=O)NC(C)(CSC)CO)C(F)F CC(C)C(C(=O)NCc1ccc(C#N)o1)C(C)NC(C1CS(=O)C1)=O Cc1ccc(C)c(C(=O)NC2(C)CCN(C(=O)Cn3nc(Cl)ccc3=O)C2)n1 n1(CCCC)nc(C)c(C(=O)N(C)CC2(NC(C3COC(=O)N3)=O)CC2)c1Cl CC1(C(=O)NCC2CCN2C(C2CC(O)(C(F)(F)F)C2)=O)CC2(CCC2)C1 Cc1cc(NC(=O)C(CC2CCOCC2)NC(=O)CC2CSCCO2)cnc1Cl c1(NC(c2cccc(C)n2)C)ncccc1S(=O)(=O)N1CC2CCC2(C)C1 Cc1ccc(N2CCN(C(=O)C(=O)NC3CCCCCC3)CC2)cc1N N1(C(C(C)(N(C)C(C23CC(F)(C2)C3)=O)C2CC2)=O)CCC(C2CC2)C1 c1(C(=O)NCC(CN(C(=O)CC2(C)CCCO2)C)O)cc([N+](=O)[O-])c[nH]1 Cc1cc(C)n(CC(=O)NC2CN(C(=O)CC(C)C)C3CC23)c(=O)n1 CCCCCCCC(=O)NCC(O)CCNC(c1c(F)ccc(F)c1N)=O C(=O)(C#CC1(CC)COC1)N1CC(C(C(=O)NC(CCC=C)CO)O)C1 C1(C(N(C)CC2C(NC(c3c(C)onc3)=O)CCC2)=O)OCC2CCCC12 C1(C(N(CC)CC2CCN(C(=O)C(C)(C)SC)CC2)=O)CCCS(=O)(=O)N1 N1(S(CC2(COC)CCOCC2)(=O)=O)CCC12CCOC(C)(C)C2 C1(N(C(CC2N(C(c3c(COC)cco3)=O)CCC2)=O)C2CC2)COCC1(C)C CCCC(O)CC(=O)NCCCC(C)NC(c1ccc(C#N)o1)=O c1(-n2cc(C3N(C(C(c4cccnc4)OC)=O)CCC3)nn2)ccc(Br)nc1 C1(C(N(C2CCN(C(=O)CCC#N)C2)CC)=O)CC2(CCCCO2)C1 Cc1cnc(N)c(C(=O)NCC2CCN(C(c3cnc(C4CC4)s3)=O)CC2C)c1 C(=O)(C1CCCc2nnn(C)c21)NC(C)CNC(C1(c2ccccc2)CC1)=O C(=O)(CC(C(F)F)NC(=O)C(F)C(C)(F)F)NC(C(=O)N(CC)CC)C N1(C(C(CC)C#N)=O)CCC2(CC1)CC(CNC(C1(OCC)CCCC1)=O)C2 S(=O)(=O)(c1c[nH]ccc1=NCC1CCN(CC)C1)NCCCCCC=C CC1CC(C(=O)NC2(C)CCCN(C(=O)CC(C)(C)C3CC3)C2)CCS1(=O)=O N1(C(C2(CC)CCCC2O)=O)CCCN(C(=O)C(=O)Nc2ccc(C)cc2)CC1 c1(C(=O)NCCCCCN(C(CCOC(C)C)=O)C(C)C)cc(F)ccc1O C(=O)(CC(O)C(C)CC)NCC(=C)CCNC(c1ccccc1CO)=O c1(-c2[nH]c(C)cc2C(=O)N=c2cc(C)n(C)[nH]2)ncnc2cccc(F)c12 c1(C(=O)N(CC(C)CNC(=O)CC2(c3ccccc3)CC2)C2CC2)cc(Cl)c(Cl)[nH]1 c1(C(N2CCN(C(c3cc(C=C)cc(F)c3)=O)CC2)=O)cc2ccc(O)nc2s1 c1(NC2CC(C)N(Cc3ccccc3)CC2)cccc2cccc(Br)c12 C1(CNC(c2ccncc2)C)CCN(C(=O)CSC2CCCS(=O)(=O)C2)CC1C C(=O)(CCN1C(=O)CSc2ccccc21)Nc1nnc(CCC(=O)OC)s1 N1(C(C(=O)NCCOC(F)F)=O)CCCC2(C1)C(O)CC2O C1(NC(C(C)OCC#C)=O)CN(C(c2cccc(CN(C)C)c2)=O)CCC1F N1(C(CN(C)C(=O)C2CC2)=O)CCC(C(C)(C)CNC(C2CNC(=O)C2)=O)CC1 S(=O)(=O)(c1ccc(Br)c([N+](=O)[O-])c1)NC(c1ncn(C)n1)(C)C C1(CC)CCCN(C(c2cnccn2)=O)C1C(=O)NCCOc1ccccc1 C=CCC(CC)C(=O)N1CC(NC(C2CC23CC3)=O)CC1(CC)CC O=C(C1=CC2CC(C1)CC2O)NCC1(NC(c2csc(O)n2)=O)CCC1 c1(C(=O)NC(CN(C(CNC(CCCCC)=O)=O)C)C)nc(OC)ccc1OC CCC(CC(=O)N1CCC(CN(C)C(c2ccnc(C(F)F)c2)=O)C1)SC C1(NC(C=CCCC(C)C)=O)C=CCCC1C(=O)NCc1nncn1C(C)C Cc1[nH]c(C(=O)N(CC(C)NC(=O)CC(C)n2cccn2)C)c(C)c1C CCC(C)CC(=O)NC1CCC1CNC(C1CC(CC(C)(C)C)C1)=O C1(CNC(Cn2nnc(C)n2)=O)CC(C(F)(F)F)CN1C(C1CCNC1=O)=O C12(NC(c3c(C)con3)=O)COCCC1CN(C(=O)CNc1ncccn1)C2 N1(C(C=CC)=O)CC(NC(c2coc(C(C)C)n2)=O)CC12CCOC2 C1(C(N2C(C)CN(C(=O)CCN3CCCCC3C)CC2)=O)CC2C=CCC(C1)C2 C(c1cc(F)cc(F)c1)=CC(N1C2CN(C(c3c(C)ccc(I)c3)=O)C(C2)C1)=O C1(C(N2CC(C)C(NC(C3(S(N)(=O)=O)CC3)=O)C2)=O)CNC(=O)CC1(C)C C(=O)(C(C)CC(C)C)N1C(C2CCN(C(c3c(Cl)cc(C)s3)=O)C2)CCC1 C1(CNC(CCSC)=O)CCN(CCNc2csc(-c3nc[nH]n3)n2)CC1 C1(O)(CNC(CN(C(CCC=CCC=C)=O)C)=O)CCCCCC1 N1(C(C2C(=C)CC2)=O)CC2CC1CN(C(=O)CCC(C)O)C2 c1(OCC)ccc(CNC(c2ncc(Cl)n2C)C2CCCCC2)cc1 C(=O)(C1CCCc2nn[nH]c21)NC1C=CCN(C(c2cc(CC)no2)=O)C1 c1(C(=O)NC(C)CNC(c2cnc3ccsc3c2)=O)ccc2c(c1)C(=O)NC2=O C(C(C)(O)CC(=O)NCC1(CNC(=O)Cc2ccco2)CC1)OC N1(C(C2CCC(C)(CC)O2)=O)CCCC(NC(c2cc(Br)co2)=O)CC1 c1(SC)ccc(Cl)c(C(N2CC=CC(NC(C3CC3C(C)C)=O)C2)=O)c1 CCC(CC)C(C)C(=O)NCC1CCN(C(c2ccc(C(C)(F)F)nc2)=O)C1 C=CCC(C(=O)NC(CNC(=O)CCN1CCNC(=O)C1)CO)c1ccccc1 c1(OC)ncc(Br)cc1C(=O)NCC12CC1CN(C(=O)C(C)(F)F)C2 Cc1ccc2cccc(C(=O)NC3CC(NC(c4sncc4C)=O)C3)c2n1 C(CCCC(C)(C)C)(C(=O)NCC1CCOC1)N(C1(C(=O)OC)CCCCC1)C CC(N=c1[nH]c(=NCC(C)C2CC2)c2cccc(F)c2[nH]1)c1ccc(Cl)c(F)c1 N1(C(c2occ(C)c2)=O)CC2(CCC2NC(c2cc(-c3ccc(Cl)s3)on2)=O)C1 C(=O)(C1CCc2cccc(OC)c21)NCC(CCNC(C1C(C=C)C1)=O)=C c1(C(N2C(CN(C(C3C(C)(C(C)C)C3)=O)C)COCC2)=O)ccc(N)c(O)c1 c1(NC(C2(F)CN(Cc3c(O)ccc(C#N)c3)C2)=O)ccc(Br)c2c1CNCC2 C1(C(N(CCN(C(C)C)C(c2ccon2)=O)C)=O)CCCN1S(=N)(=O)N(C)C c1(C(=O)NCc2ccc(CNC(C(C)SCCCC)=O)cc2)ncc(F)cc1C C1(NC(C=CC(C)C)=O)C2CC3CN(C(=O)C(C)Oc4ccccc4Cl)C1C3C2 c1(C(=O)NC(C)(C)CNC(c2ccc(Cl)o2)=O)nnn2c1CCCC2 N1(C(C(C)=CC)=O)CCCC(O)(CCNC(C2(OC)CC(CF)C2)=O)C1 c1(C(=O)NCCC(=C)CNC(=O)Cc2cccc(OCC)c2)cncn(C)c1=O CCCC(C)(C)C(=O)NCCCC(C)NC(c1ccnc(OC)c1Br)=O c1(OC)nc(=NC2CC(F)(CNC(=O)CCc3cn[nH]c3)C2)[nH]c2[nH]cnc12 c1(C(N2CC(NC(c3cc(Cl)nc(Cl)c3)=O)C(F)C2)=O)cccc2cc[nH]c12 C1(NC(c2c(CC)onc2)=O)CC(C)CN(C(c2csc(C)c2OC)=O)C1 c1(CN(CCCNC(C2CCC2)=O)C(c2[nH]cc(CC)c2)=O)ccc(Cl)nc1C Cc1nc2cc(-c3noc(CC4CSc5ccccc5O4)n3)cc(O)c2o1 c1(NC(C(C(C)C)NC(c2cocn2)=O)=O)ccc2c(c1)CCO2 C12(C(N3CC(NC(c4cc(C(N)=O)cc(C)c4)=O)C3)=O)CCOC1CCOC2 N1(C(CCCCCCSC)=O)CCCC1C1CCCCN1C(=O)CCC(F)F C12(C(=O)NCCc3ncc[nH]3)CCN(C(c3cc4ncccc4[nH]3)=O)CCC1C2 C1(C(=O)NCCC2CC(C)(C)C2)CCC(O)CN1C(=O)C(O)C(C)(C)C c1(C(N(C2(C#N)CCNC2)C(c2cnn(CC)c2C)=O)=O)cc(F)ccc1C(N)=O Cc1c(C(=O)NCC(C)(C)CNC(=O)C(c2ccc(F)cc2)F)cnn1C1CC1 N1(C(CCC=CC)=O)CC2CC(C1)N(C(c1cnc(CC(C)(C)C)s1)=O)C2 c1(C(=O)NCC2(COC)CN(C(C3CC(N4CCOCC4)C3)=O)C2)[nH]c(O)nc1C Cc1nccc(C(=O)NC2CC2CNC(=O)Cc2cn(C)nc2C)n1 c1(CC(N2CCC(CNC(C(CCC)OCC)=O)C2)=O)cccc(F)c1O c1(NC(CNC(c2nc(C)nc(O)c2)=O)C)ncc([N+](=O)[O-])cc1C#N c1(NC(=O)NCCCN(C(C)=O)C)ccc(N=[N+]=[N-])cc1 CC(F)(C(=O)NCC1(NC(c2cnc(Cl)c(N)c2)=O)CC1)C(F)(F)F N1(C(=O)C=Cc2cnco2)CCC2(CCCN(C(c3[nH]cc4c3CCC4)=O)C2)C1 N1(C(CCSC)=O)CCCC2CN(C(C3(C)COCCO3)=O)CCC12 N1(C(c2nn(CC)c(C)c2)=O)CC2CCC2(CNC(c2nccnc2C)=O)C1 C(=O)(C(C)C(=O)c1ccc(Cl)cc1)NC(c1c(C)ocn1)=O C1(C)(CNC(C#CC2(C)CC2)=O)CN(C(c2ncccc2Cl)=O)C(C)(C)C1 Cc1nc2cc(C(=O)NCCC(C)NC(=O)CC3OCCO3)ccc2n1C CC1(C)CCC(C(N2C3CC2CN(C(C2CCCCS2)=O)C3)=O)CO1 N1(C(C(C=CC)O)=O)CC(NC(c2cnn(CCC(C)C)c2C)=O)CC(F)C1 c1(C(=O)NCC(C)N(c2nnc(C3CCCC3)s2)C)csc(CO)n1 Nc1c(C(=O)NC2CCN(C(C34COC(CF)(C3)C4)=O)C2)nnn1CCN N1(C(=O)C(O)Cc2ccc(Cl)cc2)CC2CCCC2(NC(C23CC(F)(C2)C3)=O)C1 C(=O)(C1CCc2c[nH]nc21)N1C(C)CC(CNc2cc(Cl)ncn2)C1 CCCCC(CC(=O)NCCC(C)N1CCC1)NC(c1cncc2[nH]ccc12)=O C1(O)(C(C(=O)NC(CSC)(C)C)F)CN(C(=O)CNC2CCCC2)C1 C1(C(N2CCC(C)(NC(c3cnc(Cl)s3)=O)C2)=O)CC2CCCCCC12 c1(SCC#C)cccc(C(=O)NC(C)CCCCNC(=O)CC2(C)CC2)c1 CC(C(=O)NCCN1CCC(NC(=O)CCS(C)=O)CC1)C(C)(C)O C(=O)(C1Cc2ccccc21)NCCN(C(=O)CC1(C2CC2)CC1)CCC Cc1cc(C)n(CC(=O)NCC(CO)NC(=O)CCC2CCCO2)c(=O)n1 c1(SC)nc(C(N2CCC(O)(CCNC(c3ccco3)=O)C2)=O)c2ccccn12 c1(C(=O)O)sc2cccc(F)c2c1CN1CC(COCC)(OC)C1 CC(C)(C)C(CNC(C1(C)CNC(=O)C1)=O)NC(c1cc(-c2ccco2)[nH]n1)=O c1(OC)cnc(C(=O)O)cc1C(=O)NC(c1cnc(F)c(Cl)c1)c1ccccc1 CC1(C)CC(NC(C2CCS(=O)(=O)C2)=O)CCN(C(=O)COCCCF)C1 N1(C(C(CC)CC)=O)CC(NC(=O)Cc2sc(S)nc2C)CC12CCCOC2 c1(CC(=O)NCCC(C)(C)CO)c(C(F)(F)F)cccc1C(F)(F)F c1(OCCC(=O)NCC2(F)CC(NC(C3CCC(C)O3)=O)C2)ccc(F)cc1Cl CC1(C(=O)NCCNC(=O)COc2ccc([N+](=O)[O-])cc2)CCS(=O)(=O)CC1 c1(C(N(CC(CN(C(C(CC)COC)=O)C)O)C)=O)ccc2c(c1F)CCC2 C(C#Cc1cn(-c2ccc(F)nc2)nn1)NC(=O)NC1CCS(=O)(=O)C1 N1(C(C2(C(N)=O)CC2)=O)CCCC(C)C1CNC(c1[nH]c(=NC)sc1)=O C1(C(=O)NC(CNC(C2CCCO2)CSC(C)(C)C)=O)CCCC(C#N)C1 c1(SC)cc(F)ccc1C(=O)NC(C)CCCCNC(C1CN(C)C(=O)N1)=O CC12CSCC1CN(c1cccc(CC3CCCCCC3)n1)C2 C1(C(=O)NC(CNC(c2c(C)onc2CO)=O)C2CC2)CCCCN1N=O Nc1ccc(C(=O)CCC(=O)NCCC(O)CNC(=O)CCc2cn[nH]c2)cc1 C(C)(CCC(=O)N(C1CCCN(C(=O)CC2CSC2)C1)Cc1nncn1C)OC C12(C(=O)NCc3c(C)nn[nH]3)CCCC1CCN2C(=O)C(C)SC(C)C c1(C2(C(N3CC(CC=C)(NC(c4csnn4)=O)C3)=O)CCC2)ccccc1F N1(c2cn(CCOCCN(C(=O)CC3CSCCO3)CCO)nn2)CC(=O)CCC1=O Cn1cc(Cl)cc1-c1nnc(N2CCOC(COC)C2)n1CC1CC1 CCCCC(C(=O)NC1(CNC(=O)C(F)=CC2CC2)CCC1)C(C)C Cn1ccc(S(=O)(=O)N2CC3CCN(C(=O)Cc4ccccc4Br)C3C2)n1 Cc1ncc(C(=O)N(C)CC2CCCN2C(C23CCCC2C3(F)F)=O)cc1C#N C(=O)(CCCC(=O)OC)NC(CN(C(C(C(C)C)NC(CCCC=C)=O)=O)C)C C1(NC(c2nc(CCC)oc2)=O)CN(C(=O)C(CC)OC)CC12CC2 c1(C2C(=O)N(C)CC(=O)C2)ccc(OCC)c(OCC(C)C)c1.C1(COCC)CC1 S(=O)(=O)(c1cc(C(F)(F)F)cc(O)c1)N(C12CC3CC(O)(C1)CC(O)(C3)C2)C Cc1cc(Cl)c(C(=O)NC2CCC(N(C)C(c3nccnc3Cl)=O)CC2)s1 CC1(NC(=O)CCC2CCCCO2)CC(C(=O)NCC2C3CCCC23)C1 CCC(C)(CNC(=O)C(C)n1cncn1)C(=O)N(C)Cc1nncs1 c1(C(C)NC(c2nnnn2C)C2CC(OCOC)C2)cccc(F)c1C c1(C(=O)NCC2C3CC2N(C(=O)Cc2cc[nH]c2)C3)nc2ccccc2[nH]c1=O N1(C(CN(C)C)=O)CC(NC(c2cc(Cl)nc(Cl)c2)=O)CC2(CC2)C1 N1(C(c2nc(CC)sc2N)=O)CCC(C)(C)C(CNC(c2sccc2CC)=O)C1 c1(C(N(C)CC2(CNC(C3(CC)COC3)=O)CC2)=O)cc([N+](=O)[O-])cc(C)n1 CCCC(O)C(=O)NCc1ccc(-c2cnn(CCOC)c2)cc1 C1(NC(c2nc(C(C)=O)sc2)=O)CCN(C(C2(C)CC3(CC3)C2)=O)CC1C C1(C)(CNC(c2c(C)coc2C(C)C)=O)CC(F)(F)CN1C(=O)CC1CCCC1 c1(SCC)ccc(CNC(=O)C(=O)NCCc2cc(Cl)c(Cl)s2)cc1 Cn1cc(C(=O)NC(COC(F)F)CO)c(Cc2ccccc2)n1 CN1CCCCC1C(N1CC(C)(NC(=O)CCc2cccc(F)c2)C1)=O C1(CC(=O)NCCCC(=C)Cl)C2CCCC2N1C(=O)C=CCN1CCC1 c1(C(=O)NCC(CC)N(C(=O)CC2(C)CCC2)C)cccc(OC)c1 N1(C(c2ccc(CC)s2)=O)CC(C)N(C(=O)C(C)CC(N)=O)CC1C Cc1[nH]ccc1C(=O)N(C1CCN(C(=O)CN2CC3CC3C2)C1)CCO N1(C(C=COCC)=O)CC2CCCC2(NC(c2c[nH]c(=N)cc2C)=O)C1 Cc1ccc(-c2ccccc2)c(NC(=O)Cc2cc(C)nn2C)c1 C1(C(=O)NC2C(CNC(C(C=C)C)=O)CC2)CC(C(C)C)=NO1 N1(C(c2cc(C)nnc2)=O)CCC(C2CC2)(NC(C2CC(F)(F)C2)=O)C1 c1(CN2CCC(CNC(c3cccc(CCC)c3)=O)C2)c[nH]c2cc(C)ccc12 C1(NC(c2scc(C)c2Br)=O)CCN(C(=O)CN2CC=CC2)C12CC2 N1(C(CCOCCC)=O)CCCC2(CCC(NC(=O)C(C)(C)c3ccns3)C2)C1 C1(CNC(c2cc(OC)ns2)=O)CCC(C)CN1C(=O)CCSC1CCCC1 c1(C(N2CC3(N(C(C(C)CO)=O)CC3)C2)=O)ccc(S(=O)(=O)NC(C)(C)C)cc1 c1(C(N(C2C3CC(NC(=O)C(O)CN4CCCC4)CC23)C)=O)cccc(O)n1 c1(C(=O)NCCC(C)(C)NC(C(c2ccno2)C)=O)cncc2c1CCNC2=O c1(C(C)NCC(c2ccc(Cl)cc2)C)nnc2n1CCC2 c1(C(N2CCC(CNC(C3CC=CC3)=O)C2)=O)cccc2c1OCCO2 CC1(C)CC(O)(C(=O)NCC2(O)CC(NC(=O)CCCSc3ccccc3)C2)C1 c1(OC)ncc(NC(=O)COC2CN(C(c3cnc(Cl)n3C)=O)C2)cn1 N1(Cc2ncc(OC)nc2)CCC2(CC2C(=O)Nc2sc(C)nc2C(F)(F)F)C1 c1(-n2c(C(=O)NCC3(O)CN(C(C(CSC)C)=O)C3)cnn2)cccnc1Cl c1(NCC(O)CNC2CCC(c3ccccc3)C2)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC2CC(CSC)(N)C2)cc(C)n(C)n1.C1(CC(=O)C2CC2)(C)CC1 C1(F)(C(N(C2(CCO)CC2)C)=O)CCCN(C(=O)C(F)=CC2CC2)C1 CC(C)(CC(=O)NC1(CNC(=O)Cc2cc(F)cc(F)c2)CCOCC1)C(F)F c1(C(=O)NCC2N(C(C#C)=O)CCC2)nc(CC)ncc1Cl CCC(C)CC(=O)C(=O)NC(C(=O)NC1(c2cc[nH]n2)CC1)C1CCC1 N1(C(c2c(C)n(C)cc2)=O)CCC2(CC2)CC1C(=O)NC1(C(N)=O)CC1 c1(NC(CSC(COC)C)=O)c(C(=O)OC)cc([N+](=O)[O-])cc1[N+](=O)[O-] C(=O)(C(C)S(N)(=O)=O)N1C(CN(C(CS(CC)=O)=O)C2CC2)CCC1 N1(C(c2cc(CC)on2)=O)CCc2ccccc2C(NC(=O)C(C)C2CCC2)C1 N1(C(CC2CCN(OC)CC2)=O)CC2CC(C)N(C(C3C(C)C3C)=O)C2C1 CC(O)C(=O)NNC(=O)NC1C(C)(C)C1(C)C.n12cc(nn1)C(=O)NC1CC2C1 C(=O)(CC1CCOc2ccccc21)NC(CC=C)CNC(=O)C1=CCCCC1 N1(C(c2cc(Cl)cc(Cl)n2)=O)CCC2CN(c3ccn4nccc4n3)CC2CC1 C1(N(C)C)CCC(NC(=O)COCCOCCNC(=O)C(C)(F)F)CC1 c1(OC)cc(C)ccc1NC(=O)C(c1ccoc1)NC(C1CC2C=CC1O2)=O N1(C(C(CCC)C#N)=O)CCCC2CN(C(C34CSCC3C4)=O)CC12 C12(NC(c3cn(C)nc3)=O)CCN(C(c3cc(O)ncn3)=O)CC1C2 c1(C(=O)NC(CNC(c2cc(OC)c(F)cc2)=O)C)ccc2c(c1O)CCC2 C1(SC)OCC2CCCCC12.C12(NC(=O)CSCCSC)CCCC1C(=O)NC2 N1(CC=C)CCCC(NC(c2cnc(C3CCNCC3)[nH]2)=O)C1 N1(C(CCCCC(C)C)=O)CCCCC12CC(NC(C1CCCCC1(C)C)=O)C2 N1(C(C=C(CC)C)=O)CC(NC(c2cnoc2-c2ccccc2)=O)C(O)C1 C#CCC(CC(F)F)C(=O)NC1CCCCC1NC(=O)C(N1CCOCC1)C CC1OCCN(C(=O)CCCN2CCCC2)C1C(N1CCCC(C)CC1)=O Cc1ccc2c(c1)C(NC1CCCCC1c1ccnn1C)CCC2 C1(NC(=O)CCCc2cccc(Cl)n2)CN(C(c2cnc[nH]2)=O)CCC12CCC2 C1(C)(OC)CCN(C(C2CC(C)(NC(=O)CCn3cnccc3=O)C2)=O)CC1 c1(OC)cc(C(N2CC(C(=O)NCC3CCCOC3)C(F)C2)=O)ncn1 C1(CNC(c2cc(CC)ncc2)=O)CCCC2CN(C(=O)C(C)(C)C#N)CC12 c1(C(=O)NC(C2CN(C(=O)COC(F)F)CCO2)C)[nH]nc2c1COC2(C)C Cc1cc(C(=O)NC2CN(C(c3ccccn3)=O)CCC2F)cc(Cl)c1 S(=O)(=O)(c1ccc(NC(CO)C2(C)CC2)c(C#N)c1)NCC(C1CCCCC1)C c1(CNC(=O)C(N2CCCC(NC(C3CC4(C3)CC4F)=O)C2)=O)ccc(F)nc1 S(=O)(=O)(c1c[nH]c(=NCCCNc2nccs2)cc1C)N(C)Cc1cnc(C)o1 N1(C(CC(C)(C)O)=O)CCOC2CN(C(c3ccc(-c4ccco4)nc3)=O)CC12 C1(F)(OC(=O)NCC(C2CCCC2)NC(CNC(COC)=O)=O)C2CCCCC12 C1(CNC(C2ON=C(C)C2)=O)CN(C(c2cc(Cl)n(C)n2)=O)CCC1(F)F C1(NC(c2cnc(O)o2)=O)CC2(C1)CC(CNC(C1CC3CCC1O3)=O)C2 C1(CCOC)(NC(c2cc(C)sc2C)=O)CCN(C(=O)Cc2csc(C)n2)C1 c1(NC(C)=O)cccc(F)c1C(N1CC2CCC2(CNC(=O)C=C(C)C)C1)=O C1(N(C(c2cc(CNC(c3cc(OCC)n[nH]3)=O)no2)=O)C)CC(C)CC(C)C1 C(=O)(CC(C)CC(C)C)N(C1CC(C#N)C1)CC(=O)NC(CCCC)(C)C C(=O)(CC1COc2ccccc21)NC1CC(NC(C(C)C#N)=O)C1 N1(C(C2CCN(C)CC2)=O)CCOC(C)(CNC(C2(S(N)(=O)=O)CCC2)=O)C1 C1(C(=O)NC(CC)CN(C)C(C2CCCCN2C)=O)CCC([N+](=O)[O-])CC1 c1(C(N2CC(NC(c3c(CC)scc3)=O)(CO)C2)=O)cnc([N+](=O)[O-])n1C c1(OC(C)C(=O)NC2CCC(n3cccc3)CC2)ccc(Cl)cc1Cl N1(Cc2nc(C)[nH]n2)CC2CCN(C(C34CC5CC(C(=O)N3)C4C5)=O)CCC2C1 C#CC1(C(N2CCCN(C(C3CC=CC3)=O)CC2)=O)CCCCC1 N1(C(CC=CCC)=O)CCC2(CC1)CC2C(N1CCC(C)C1(C)C)=O NS(=O)(=O)C1(C(=O)NC2CCC2NC(C2(Oc3ccccc3)CC2)=O)CCC1 CSC1=C(C(=O)N2CCC3(NC(=O)CN4CCCCCC4)CC3C2)CCCC1 C1(NC(c2c(CCC)occ2)=O)CN(C(c2c(F)cccc2Cl)=O)CCC1CO c1(CC(=O)NCC2(CCNC(CC3CC(=C)C3)=O)CC2)coc2cc(C)ccc12 C1(C(N(C)CC2(NC(c3csc(=N)[nH]3)=O)CC2)=O)CCC(C(C)(C)C)CC1 c1(C(=O)NCCOC2CCN(C(C(C)N(C(C)=O)C)=O)C2)nn(C)c2c1CCC2 C1(CN(C)CC)CCN(C(c2ccc(Br)s2)C(=O)Nc2cnn(C)c2)C1 N12CC3CCC3(C1)NCc1c[nH]nc1C2=O.C(C(=O)O)(OCC)OCC.C1CC1 C(CN=C(NCc1cn(C2CCCCC2)nn1)NCC(C)(C)C=C)SCC#C c1(COC)n[nH]c(=NCC2(F)CCN(C(=O)CC3CS(=O)(=O)C3)CC2)s1 c1(CNC(C2CCCCC2)C(=O)NCC(C)OC)ccccc1OC(F)F c1(C(=O)NC2(C)CC(NC(=O)CCCn3cccn3)C2)ncn2ccccc12 Cc1nn2c(c1I)CN(C(=O)NCCCN1CCC(C(N)=O)CC1)CC2 c1(C(=O)NCC(CNC(Cc2cc(C)nn2C)=O)O)cc2cccnc2cc1F N1(C(CN(C(CC2(N(C)C)CCC2)=O)C)=O)CC2CCC1C(O)C2 C1(C(=O)NCC(N)=O)CCC2(CCN(C(C3CCn4c(Cl)cnc4C3)=O)CC2)O1 N1(C(c2cc(CCOC)on2)=O)CCC(NC(c2ccnc(COC)n2)=O)CC1 C(C)(C(CO)NC(c1cc(-c2ccco2)no1)=O)NC(C1C(OCC)C1)=O CCC(C)CC(C(=O)NC1CC(O)C1OC)NC(c1nnc(S)n1C)=O Cc1c(C(=O)NC(C)C(C)NC(c2ccn(CCF)n2)=O)c(C(F)F)nn1C c1(C(=O)NC2(C)CC(C(=O)NCC(c3cccnc3)C)C2)ccc(F)cn1 c1(CC)n[nH]c(CC)c1CC(=O)NC1CC1NC(=O)Cc1cc(C)[nH]n1 n1(CC(=O)NCC(CNC(c2ccc(O)cn2)=O)OC)nc(C)ccc1=O N1(C2CCC(NC(CC3(C#N)CC3)=O)C2)CCN(C(=O)C=Cc2ccoc2)CC1 C1(c2nnnn2C2CCOCC2)(Nc2c(COC)n(C)nc2)CCCCCC1C c1(Nc2cccc(NC(N3C(C#C)CCCC3)=O)c2)c(Br)cc(Cl)c2occc12 C1(NC(C(C)C)=O)(CO)CCN(C(c2cccc(Oc3cccc(F)c3)c2)=O)C1 C1(C)(C(N(CC(C)C(=O)NCCN2CCCCC2)C)=O)CCN(C)CC1 N1(CC)CCCCC1C(=O)NC(C)CCCNC(=O)Nc1cnn(CCOC)c1 C1(NC(C(C2CCCC2)OC)=O)COC2CN(C(c3c[nH]c(=N)nc3C)=O)CC12 N1(C(c2cnc(C)s2)=O)CC(C(=O)NC(C(O)CO)C2CC2)C(C2CC2)C1 N1(C(CC(CC)O)=O)CC2C(C1C(=O)Nc1c(Cl)cc(Cl)cc1Br)C2(C)C CCCCC(C(=O)OC)N1CCC(C(=O)NC2CCCCC2)(OCC)CC1 c1(C(=O)NCCOCCCNC(C2(COC)CCOC2)=O)ccc2n[nH]cc2n1 C(=O)(CS(=O)(=O)CC)N1CCC(C(CNC(C(C)(C)OCCC)=O)C)CC1 Cc1cc(C(N2CC3CC(C2)N3C(c2cnc(C)s2)=O)=O)cc(Cl)c1 c1(C(N2CC(C)(CNC(c3c(C)nc(C)s3)=O)OCC2)=O)cc(C#N)ccc1O c1(CCC(=O)NC2CCN(C(c3ccc(OC)nn3)=O)C2)ccc(Br)c(C)c1 c1(CNC(=NC)NCC(n2cc(C(F)(F)F)cn2)C)ccc(F)cc1 n1(CC)ncc2cc(C(=O)NCC(F)CNC(=O)C(C)C(C)(C)C)c(C)nc12 C1(C(N2CC(C)C(NC(=O)CCc3ccc(Cl)nc3)C2)=O)CC12CCOCC2 c1(OC)cc(C#N)c(NC(C2CC2NC(c2ccc(Cl)c(F)c2)=O)=O)cc1OC CC(C)C(C(=O)NCCNC(=O)N(C)C)NC(C1CCCC1)=O.C(N)(=O)N C12CCC(CC1)CN2.C12CC(C1)OC(=O)C2.CCC(=O)OCCC c1(C(N(C2CC(NC(C(C)Cc3cccnc3)=O)C2)C)=O)nccnc1C(N)=O C(=O)(C(O)CCS(C)=O)N1CCN(C(c2c(OC)n[nH]c2)=O)CC1 C1(C)(CNC(C(F)OC)=O)CC(F)(F)CN1C(=O)CCN1CCCC1 C#CCC(C)C(=O)N(CCCCN(C)C(c1cn(C)nc1C(C)C)=O)C CCC(CC)(C(=O)NC12CC1CN(C(C1COCCN1CC(F)(F)F)=O)C2)OC CC1CN(C(c2coc(C(N)=O)c2)=O)CC(CCNC(c2cnc(S)n2C)=O)O1 N1(C(CN(CCOC)C)=O)CC2CC2(CNC(C23CCC(CC2)C3)=O)C1 N1(C(C2CC(C)(C)OCC2)=O)CCc2ccccc2C1CNC(=O)C1=CCCO1 N1(C(C(C)Sc2ccc(OC)cc2)=O)CCC2(C1)CN(C(=O)CCOC(C)=O)C2 C1(C)(C(=O)NC(C2CCOC2C)C)CCCN1C(=O)CCc1cocn1 C1(C)(NC2CC2)CC(F)(F)CN1C(C1(C(=O)NCC2(C(=O)OCC)CC2)CC1)=O Cc1ccc2c(=NCC(C)S(C)=O)[nH]c(N(C)Cc3cnc[nH]3)nc2c1 C1(NC(CC(C2CC2)NC(c2c(C)cc(CC)o2)=O)=O)CC2CC3C(C2)C13 Cc1cnc(Cl)cc1NC(C1CCN1Cc1ccc(-n2cccn2)cc1)=O C1(OC)CN(C(=O)N(C)Cc2ccccc2Br)CCC1NC(=O)C(O)CC(C)C N1(C(C(=O)Nc2cccc(CC)c2)=O)CCC(O)(Cc2ccc(C)c(F)c2)CC1 C1(C(=O)NCC(NOC)=O)CN(C(c2csc(C)c2)=O)CC(C)O1 C1(C)(C(N(C(CC)C(=O)NCC(=O)N(C)C2CC2)C)=O)CC(C)=NO1 C1(C)(NC(C(C)Cc2cnc[nH]2)=O)CCCN(C(C23CCCC2C3(F)F)=O)C1 C1(C(N2CCC(CNC(=O)CC3CSCCS3)CC2)=O)CCCCCS1(=O)=O c1(C(N(CCCN(C(=O)C(F)(F)C(F)F)C)C)=O)ccc2nc(CO)[nH]c2c1 c1(SCC(=O)NCCC(CNC(CN2C(C)CC2)=O)O)ccc(Cl)cc1 c1(C(C(=O)NCCCNC(C(C2CCOC2)OCC)=O)=O)ccc(Cl)s1 c1(C(=O)NCC2C(C)CCCN2C(c2cc(Cl)cn2C)=O)cc(F)c(N)cc1F C1(OC)CC(C(F)(F)F)CN(C(=O)CCC(C)C)C1.C12CCC(CC1)NC2=O C1(CNC(=O)C2=NOCC2)CCN(C(=O)CN2C(=O)CNC2=O)CCC1(F)F c1(C(=O)OC)ccccc1CNCC1(Cc2ccc(Cl)cc2)CC1(F)F Cc1cc(C(=O)NCC2(F)CC(NC(c3ncccc3Cl)=O)C2)cc(F)c1 CN1CCC(C)(C(N2CC3CC(CNC(=O)CCc4ccsc4)C3C2)=O)CC1 C(=O)(CCS(=O)(=O)N(C)C)NC(C(C(C)C)NC(C1C(C)=C1)=O)c1ccccc1 CCCCC(CC)C(=O)N1CCC(CO)C(NC(=O)CC(CCC)OC)C1 N1(C(c2ccc(S(C)=O)cc2)=O)CC(C2CCCN(C(=O)C3=CCOCC3)C2)C1 c1(C(=O)N(CC(C)C(c2cc(NC(=O)C(=O)N(C)C)no2)C)C)ccc(F)cc1 c1(CCC(N2C(CN(C(C(C3CC3)OC)=O)C)CCCC2)=O)cnc2n1CCC2 c1(C(N2C(CNC(=O)CC3CSCCS3)CC2)=O)cnccc1Br C(CCCCCCO)NC(N(C(Cc1c(C)cccc1)C)C)=O N1(C(CCN(CC)CC)=O)C2CCC1C(F)C(NC(=O)C(CC1CC1)OC)C2 C(=O)(C1COc2ccccc21)N(CCCNC(Cc1cccc(C)c1F)=O)C C1(NC(C(CC(N)=O)NC(C2CCC(O)C2)=O)=O)CC2CC1CC21CC1 CC1CC(CNC(c2cnc(Cl)s2)=O)CN(C(=O)CC2CC(=O)NC2=O)C1 c1(NC(C)=O)cccc(F)c1C(=O)N(C1CCN(C(=O)C(C)(C)O)CC1)CCO c1(N2CCC(C)(C(=O)NC)C2)nc(=NCC2CCCC2C)[nH]c2c1CCCCC2 C1(C(N2CCCC(C(N)=O)C2)=O)(CC)CCN(C(C2CCC3(CC3)C2)=O)C1 c1(C(CCC)=O)ccc(S(=O)(=O)NCC(O)CC=CCOC)cc1 c1(NC(C)=O)cccc(C(=O)NCCC2CC2NCC2C3COCC23)c1 C1(C(N2CCC(CNC(c3c(CCC)occ3)=O)C2)=O)Cc2cc(C)ccc2S1 N1(C(c2cc(F)ccc2CC)=O)CCC2CN(C(c3cc(O)no3)=O)CC2C1.N1CC1 c1(NC(C)C)cccc(-c2nnc(N3CCC4CC34)n2C2CC2C)c1 c1(C(N2C(C)CC(NC(c3ccsn3)=O)C2)=O)ccc(C(F)F)cc1Cl C(CCSC)(C(=O)N1CCCC1CNC(N)=O)NC(c1c(CCC)nco1)=O C1(NC(c2ccc(CC)c(F)c2)=O)CC1C1CCN(C(=O)C(C)(O)C2CC2)CC1 CC1CCN(C(=O)CNS(N)(=O)=O)C1c1cn(C(c2ccncc2)C)nn1 C#CCC(C)(C)C(=O)N1CCN(CC(=O)NC(C2(O)CCCCC2)C)CC1 CC(C)C(O)C(C)C(=O)NC1(C(=O)N(C)CCNC(N)=O)CCCC1C N1(C(C(C(C)C)NC(COC)=O)=O)CCC2(CC1)CC(C)N(C(C)=O)C2 CC1CCCn2c(C(N3CC(CNC(c4cccc(F)c4)=O)C(C)C3)=O)cnc21 c1(OC)cc(C(C(=O)NCC2CCCO2)N(CC(C)(C)C)C)cc(C(F)(F)F)c1 C123CC(C1)(C2)CNC3=O.C(C)(C(=O)N)OCCOCC.C1(CC)CCC1 C1(O)(C(=O)NCCCCC(=O)NCC(CC)(C)CC)CC2CCC1C2 c1(CS(C)(=O)=O)nc(C(=O)NCCN(C(C2CC2C(N)=O)=O)C2CC2)cs1 C(=O)(C1CCCc2ncccc21)NC(C)CN(C(=O)Cn1nnc(=O)[nH]1)C N1(C(c2c(C(=O)OC)c(C)on2)=O)CCC2(CC1)CC2CNC(c1cnc[nH]1)=O c1(CN(C(CC(N)=O)c2ccccc2)CC)cccc(F)c1 Cc1ccc(C)c(CNC(C2(F)CCN(C(=O)C=CC(=O)NC3CC3)C2)=O)n1 C1(CNC(COC(CC)C)=O)CN(C(=O)C(F)CC2CCC2)CCC1CO C1(C2CN(C(=O)C=CC(=O)NC3CC3)C2)(NC(C(CC=C)C)=O)CC1 C1(OC)CC2CC(C1)N(c1cc(F)cc(Cl)c1)C2 C1(C(N(C(CC#C)C)C)=O)CC2CCC1N2C(=O)CN(C1CCC1)C CCC(C)(C)C(O)C(=O)N1CC2CN(C(c3cc(Br)c(Cl)s3)=O)CC2C1 C=Cc1cnn(C)c1C(=O)NC(CNC(c1cnn(CCC)c1C)=O)CCOC c1(C(C(=O)NCCC2CC(NC(CN(C)C3CC3)=O)C2)(C)C)cccc(F)c1 C(=O)(C(C)C(O)CCCCC)N1C2(CCN(C(C(C=CC)O)=O)C2)CCC1 C1(C(N2CCC(CNC(CCC=CC(C)C)=O)C2)=O)CCS(=O)(=O)C1(C)C C1(CNC(C(C)OCCOC)=O)CC2CCCC2N1C(=O)CC(C)(F)F CC1CCN(C(=O)Cc2ccc(O)nc2)C(C(=O)N(CCC(C)(C)C)C)C1 N1(C(=O)NCc2scc(C)c2)CCC(C2(C)CC2)C1 Cc1cnc2cccc(C(=O)NC(CO)C(C)(C)F)c2c1 CCCCCC(O)CC(=O)NC(C)(CNC(=O)CCCS(N)(=O)=O)CO C1(O)(C(N2C(C3CCN(C(C(CCCC)O)=O)C3)CCC2)=O)CN2CCC1CC2 C#CCCCCCC(=O)NCc1cccc(CNC(=O)CC2CCCCC2O)c1 c1(C(=O)NCC=C(C(=O)NCCCC=CC)C)cccnc1 C(=O)(C(CCC(C)(C)C)N(C)CC12CCC(CC1)CC2)NCCCSC N1(C(c2cc(C)c(C)nc2)=O)CCN(C(=O)CC2CCCCC2O)CCC1C CC(O)CCCCCC(=O)N1CC(NC(c2ccc(OCC(F)(F)F)cc2)=O)C1 C1(NC(C2=NNC(=O)C2)=O)COC2(CCN(C(c3cncc4nc[nH]c34)=O)C2)C1 N(C1c2ccccc2CC1NC(=O)C=C(C)Cl)C(C(CC=C)(F)F)=O C1(NC(C(C)(C)NC(=O)NCC)=O)CN(C(=O)CCF)Cc2nccn2C1 c1(OC)nn(C)cc1C(=O)NC(C)CC(C)NC(C1CC(=O)N(C(C)(C)C)C1)=O C1(CC(C2CCCC2)N)CCCCN1C(=O)Nc1cccc(C2CCOC2)c1 c1(C(=O)NC2C(OC)CN(c3ncncc3C#N)CC2)nc2ncccn2n1 c1(CCSC)nc(-c2cn(C(C)(C)C)cn2)n(-c2ccnc(Cl)c2)n1 CC1(C)OCC(CNC(=O)CC2CCC(C3CC3)O2)C(O)CO1 N1(C(Cn2nc(C)oc2=O)=O)CCC(CNc2ncccn2)C(C)C1 C1(NC(CSCCN(C)C)=O)CCC12CN(C(c1ccn(C)c1)=O)C2 C1(CC(=O)NCC(CCCC)O)N(C(=O)C(F)CC2CCOC2)CCC1(C)C c1(C(=O)NCCOCC(=O)N(C(CCC)C)C)cccc(CC#N)c1 S(=O)(=O)(c1ccc(N2CCC3(CCCC(C(=O)O)O3)CC2)c([N+](=O)[O-])c1)N(C)C C1(C(N2CCC(C(C(=O)N(C(C)C)CC3CCC3)C)CC2)=O)CC2(C1)CC(C)C2 N1(C(COC2CCN(C(C=CC(=O)N(C)C)=O)C2)=O)CCCC(C)(O)C1 O=C1COc2ccc(C(N3CCC4(CC4NC(C45COCC4C5)=O)C3)=O)cc2N1 O=C1CC(C(N2CC3CC(NC(C4CC5(CC5)CO4)=O)C3C2)=O)Cn2ccnc21 CCCCC(CNC(=O)CN(C)C(c1ccsc1C)=O)CCC C1(C(=O)NCC(C)N2CCC2)CC(=O)NC(c2ccccc2)C1 c1(C(N(C(CNC(C2C(C=C)C2)=O)C)C)=O)csc(C2CCCCC2)n1 C(CC(=O)N1CC(C)CC1CC)(C(F)F)NC(CCC=CCC=C)=O Cc1cc(N)cnc1C(N1CCC1CC(=O)Nc1ccc(O)cc1O)=O c1(C(=O)NCC(CC=C)NC(C2(C)CCCS2(=O)=O)=O)nccc2ccncc12 C12(NC(C(COC)(C)C)=O)CN(C(c3ccnnc3)=O)CC1CS(=O)(=O)C2 c1(C(=O)NC(CNC(c2c(CC)occ2)=O)C)cc2c(=O)cc[nH]c2s1 C(=O)(C1CCCc2nn[nH]c21)NC1(CC)CCN(C(C2(CC#C)CCC2)=O)CC1 N1(CC(=O)NCC=CCC(=O)N(CCOC)C2CC2)CC(=O)NC1=O Cc1cc(C(N2CC(NC(C3CCCC3)=O)CC2CO)=O)cc(N)c1O C12(C(N3C(C)C(NC(c4cccc(CO)c4)=O)CC3)=O)C3C4C1C1C2C3C41C C(=O)(C(C)(C)N(S(C)(=O)=O)CCO)N(C)CCN(CC(F)(F)F)C(C12CCC1C2)=O N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)Cn2ccc(C)cc2=O)C(CF)C1 c1(C2N(C(C3CC4CC4N3)=O)CCC2)cccc(F)c1F C1(=CC(=O)NC2C(CNC(C(C)n3cccn3)=O)C2)CCCCC1 C#Cc1c[nH]nc1C(=O)NCc1cncc(C(=O)N(CC(N2CCCC2)C)C)c1 Cc1cc(-n2cccc(C(N3CCCOC(CN)C3)=O)c2=O)cc(C)c1 C1(CC2(CS(C)(=O)=O)CC2)Cc2cc(Br)ccc2N(C(C(C=C(C)C)F)=O)C1 C(=O)(CCC(C)(C)C#N)N1CC(C(=O)OC)(CNC(c2c(CC)cns2)=O)C1 C1(N(C(C(C)OCC2CC2)=O)C)CCCCN(C(=O)C=Cc2ccccc2)C1 Cc1ccc(-c2cn(CC3CCN(C(c4nn(C)cc4N)=O)C3)nn2)cc1Cl N1(C(C2(C)C(C)CCCC2)=O)Cc2occ(C(=O)N3CC=CCO3)c2C1 CN1CCC(C(N2CC3(CC3)CC2C(=O)NC2CC3(C2)CN(C)C3)=O)CC1=O c1(CC(=O)NC(CC)CN(C)C(C2CC2C)=O)coc2cc(CC)ccc12 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2(CC2)CC1C(N1CCCC(O)(CO)C1)=O CC(C)C(CO)C(=O)NC(C)CC(C)NC(=O)C(C)CCNC(=O)OC(C)(C)C C(=O)(CCCC(F)(F)F)N(C1CCCN(C(=O)CC2CCCOCC2)C1)CC c1(NC(=O)NC2CCOC(c3ccncc3)C2)cccc(Cl)c1N1CCCCC1 C#CCC(C)(CC)C(=O)NCC1CCC1NC(c1nc(C)sc1C)=O C1(CNC(c2cnc(OC)c(C)c2)=O)CN(C(=O)CSC)C2CCCC2O1 CC1(C)CC(NC(=O)C(C)(O)C2CCCCC2)CN1C(=O)CCNS(C)(=O)=O c1(OC)cc(OC)c(CN2CCOCC2C(=O)NCC2CCC(F)(F)C2)cc1Br N1(C(CCNC(C)=O)=O)CC(NC(C2CCC(C)(C)CC2)=O)CC12CCCOC2 C1(C(=O)NCCN(C(=O)Cc2cncnc2O)C)OCC2CCCC12 N1(C(CC(CC)C2CC2)=O)CCCC(N(C)C(C2(F)CCCCC2)=O)CC1 c1(C(N(C)CC2N(C(CC(C)C(F)F)=O)CCCC2)=O)cc2ccnn2cn1 N1(C(C(C)(C2CCC2)NC(C2C(C(C)C)CCO2)=O)=O)CCS(=O)CC1C N1(C(Cc2n(C)ccc2)=O)CC2ON=C(CNC(=O)Cc3ccc(Cl)cc3)C2C1 c1(C(N2CC(NC(CC(CC)SC)=O)C(C)C2)=O)c(N)sc(C)c1C c1(OC)cc(C(N2CCC(CNC(c3ccoc3)=O)(OC)C2)=O)ccc1[N+](=O)[O-] C(=O)(C1=CCCCO1)NC(C1CCN(C(c2cnc(C)[nH]2)=O)C1)C N1(C(C2C(C)=C2)=O)CCC2(CC1)CN(C(C1CC1F)=O)CC2CO N1(C(C=CCOC)=O)CC(NC(c2cccc(-n3cncn3)n2)=O)C2(CCC2)C1 c1(CC(=O)NCC2C=CCN2C(c2cc(O)ccc2Cl)=O)nnc2n1CCCC2 Cc1ccc(C(=O)NCC2(C)CN(C(=O)C(c3cncn3C)O)CC2C)c(N)n1 CC1=CC(NC(=O)C(CC2CCOCC2)NC(=O)C(C)C#N)CCC1 c1(C(N2C(C(C)(C)NC(c3cnc(O)o3)=O)CCC2)=O)cc(O)c2ccsc2c1 C1(c2ccccc2)(CNC(=O)NCC2COCOC2)CCOCC1 S(=O)(=O)(c1ccc(Cl)cc1)NCCOC1CCS(=O)(=O)CC1 N1(C(=O)CCc2ccon2)CCN(C2CC(NC(C3(O)COC3)=O)C2)CC1 c1(-n2ncc(C(=O)NCC(CC=C)NC(=O)C(C3CC3)OC)n2)ccc(F)cc1 Cn1ccc(C(=O)NCC2(C(=O)NCc3cc(C(N)=O)no3)CCC2)n1 c1(NC(C2COCCN(c3c(C)cncn3)C2)=O)cccc([N+](=O)[O-])c1Cl C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC1CCCCN(C(CCC=C)=O)C1 N1(C(c2oc(CC)c(C)c2)=O)CCCC(C(=O)NC2CN(C(N)=O)C2)CC1 C1(C)(CNC(Cc2c(C)n[nH]c2)=O)CN(C(=O)Cn2cccc2)CCO1 N1(C(COCCCC)=O)CCC2CCN(C(=O)C=CCOC)C2C1 CCC(CNC(=O)C(C)C(C)c1ccc(F)cc1)(CC)NC(=O)CCC1CC1 c12cc(nn1C)CN2.c1(C2(C(C)NC(=O)C(C)SC3CC3)CC2)ccccn1 c1(C(=O)NCC(CC=C)NC(C2(CCOC)CC2)=O)ccc2cc(Cl)ccc2n1 N1(C(c2ccc(N)c(F)c2)=O)CCCC(O)(CNC(c2ccoc2)=O)CC1 CC1(CO)CN(C(c2cccc3ccncc23)=O)c2ccccc2O1 N1(C(c2nccc(C3(C)CC3)n2)=O)CCCC2(CCOC2)C1 c1(C(N2C3CN(C(c4cccc(C)c4C)=O)CC32)=O)ccc(C#N)cc1O O=C1CC2CC1CC2C(N1CCCC(F)(C(=O)NC2(CO)CC(F)C2)C1)=O C1(C(=O)NC(C(=O)NC)C(C)C)CN(C(=O)CCNC(=O)OC)CC(C)(C)C1 C=C(Cl)CC(C(=O)NOC1CCCC1)NC(=O)CC(C)CN(C)C CN1CCN(c2ccc(-c3nc(-c4cscc4C4CC5CC5C4)no3)cc2)CC1 CC#CCCCC(=O)N1CCC(NC(c2ccncc2SCC)=O)C(CO)C1 N1(C(C)C)CC(CNC(N2CCC(O)(Cc3ccccc3F)C2)=O)CC1=O c1(C(=O)NCC(CN(C(C2(C(=O)NC)CCC2)=O)C)C)ccc2cc[nH]c2n1 C1(NC(=O)CCN2CCC2)CC2(CCN(C(=O)CNCC(F)(F)F)CC2)CO1 Cc1[nH]c(C)c(C(=O)NCC2(O)CC(C(=O)NCC3(O)CCC3)C2)c1C c1(C(=O)Nc2cccc(NC(c3cccc(C#C)c3)=O)c2)ccc(F)c(C)c1Cl C1(C(=O)NCC2(OC)CCN(C(C3CCCOC3)=O)C2)CCn2c(C)cnc2C1 N1(C(c2ccc(OC)s2)=O)CCN(C(=O)COCc2nc(C)no2)C2CC12 C(=O)(C(F)C(=O)NCC1CCN(C(=O)C(SC)SC)CC1)OCC C(=O)(C1=C(C(C)(C)C)N(c2ccc(F)cc2C)C(=S)NC1c1cn(C)cn1)OC C1(C(=O)NC2CC(F)(CNC(CCC#C)=O)C2)(CC)CCCC1O c1(OCC(=O)NC2C(NC(c3cc(C)no3)=O)C2)c(F)cccc1F N1(C(c2c(OC)c(C)sc2)=O)CC(NC(c2ccnnc2O)=O)CC(C)C1 C1(NC(C(C2CC2)OCC)=O)CCCN(C(=O)COCC(C)C)C1C CC(C)C(O)C(=O)N1CC(CCn2cc(CN3CCC(F)CC3)nn2)C1 N1(C(C2CN(CC)C(=O)CC2)=O)CCN(C(=O)C2=CCCC2)C2CS(=O)(=O)CC12 C1(C(=O)NCC(C)CC(=O)N(C)Cc2ccccn2)Cc2nccn2C1 C1(O)(CNC(CC(C=C)C)=O)CCCN(C(=O)Cc2ccccc2Br)CC1 N1(CCCNC(CN2CCC(OC)C2)=O)CCN(C(C2CC2C2CCC2)=O)CC1 CC1(C(N2CC(NC(=O)CCn3c(O)nnc3O)C2)=O)CC=CCC1 N1(C(c2nn(C)c(O)c2)=O)CCCC2C(NC(c3nncs3)=O)C(C)(C)C12 c1(C2CN(C(C(F)(F)C3(OCC)CCC3)=O)C2)cccc(C#N)n1 N1(C(COC(CC)(C)C)=O)CCN(C(=O)CN(C)C(=O)OC(C)(C)C)C(CO)C1 N(C1CC(C)n2ccnc21)C(COCc1c(C)cccc1)=O c1(NC(C2CCC(NC(c3cc(C)[nH]c3)=O)C2)=O)cccnc1F CC1CC(C)N(C(c2cn[nH]c2)=O)CCN1C(=O)C=C1CCSCC1 C=CC(C)C(=O)NC1CCN(CCCNC(=O)C(n2ccnc2C)C)C1 N#Cc1ccc(N2CCCC2C(N2CCC(C(=O)NCCCO)C2)=O)cc1 C1(CNC(c2nnc(C)s2)=O)CC(F)CN1C(c1cc(C)n(C(F)F)n1)=O C1(C(C)C)(CNC(=O)C=Cc2cnn(C)c2)CCN(C(C2(C)CC(F)(F)C2)=O)C1 N1(C(CNC(CC)=O)=O)CC(C2CN(C(=O)C=Cc3cccc(CO)c3)C2)C1 C(=O)(C1=C2CCCN=C2NN1)N1CC(NC(C2CCCCC2)=O)CC12CCC2 C1(CNC(C2(P(C)(C)=O)CC2)=O)CC2CCC1N(C(=O)CN1CCCC1=O)C2 c1(C(N2CC(CN(C(=O)CCCn3ccccc3=O)C)C2)=O)cccc(C#N)c1 CC1(F)CN(C(=O)C(c2ccc(Cl)c(Cl)c2)O)CCN(C(C2CC(O)C2)=O)C1 c1(NC(=O)NC2CCCN(Cc3ccccc3)C2)ccc(C(F)(F)F)cn1 C1(C(=O)NCC(C)OC(F)F)CCN(C(=O)C2(C)CCCC2O)O1 N1(C(=O)CSc2ccc([N+](=O)[O-])cc2)CCC2(CC1)COCCO2 N1(C(CN2C(C)CCCC2)=O)CCN(C(=O)C(O)CC(F)F)C(CO)C1 Cc1ccc(C(=O)NC2CC3CC(NC(=O)CCc4cnc(O)[nH]4)C3C2)c(O)n1 C#CCC(C(=O)NC(C)CCN(C)C(c1cnn(CC(C)C)c1CC)=O)C1CC1 C(=O)(C1=CCN(C(=O)CCOCC(F)F)C1)NCc1c(C)nccn1 CC1CN(C(c2ccccc2Cl)=O)CCCN1C(C1CN(C)CC1C(F)(F)F)=O O=[N+]([O-])c1cccc2ccnc(OCC3CCCCN3)c12 O=C1NC(CNC(=O)C(=O)NC(C2CCCCC2)C2CCCO2)CO1 CCC(CC(C)C)C(=O)N1CCC(F)(C(=O)Nc2cnc(Cl)nc2)C1 Cc1ccc(C(=O)NC(C)CNC(c2ccc(-c3cnc[nH]3)cc2)=O)c(Cl)c1 c1(C(=O)NC2CC(CNC(C(C)CS(C)=O)=O)C2)ccc2nnn(O)c2c1 N1(C(c2c(OC)cccn2)=O)CCN(C(c2ccc3c(c2)CCO3)=O)C2CCC12 N1(C(C(C)(C)c2nccs2)=O)CCC(C2CCN(C(C3CCCOC3)=O)CC2)C1 N=c1[nH]ccc(C(=O)NC2CCCC2NC(C2CC3CCC2C3)=O)c1[N+](=O)[O-] C1(NC(C(CC)C)=O)COC2(CCN(C(c3ccc4c(c3)OCCN4C)=O)C2)C1 CC12CN(C(c3cscn3)=O)CC1CN(C(C1CCCCC13OCCO3)=O)C2 C(=O)(CCCCCN=[N+]=[N-])N1CC(C)C(CNC(C2CN(C)CCN2C)=O)CC1 C1(C(=O)OC)CCCN(C(C)CCSc2cccc(OC)c2)C1 c1(C(=O)NC2(C)CC(NC(=O)CN3CC4CCC3C4)C2)cccc(O)c1Cl C1(CNC(CCN(C)CCO)=O)CC2(C1)CN(C(=O)C(F)C1CCOC1)C2 c1(C(N2C(CCNC(C(C)OCCOC)=O)COCC2)=O)ccc(Cl)c(O)c1 N1(C(C(C)CO)=O)C2CCCC1CN(C(C1(c3ccccc3)CC1(C)C)=O)C2 C1(NC(CCC(=C)C)=O)CCSC12CN(C(C1CC(=O)N(CCC)C1)=O)C2 c1(C(=O)NCCSCC(=O)NCCC2CCCC3CC23)cc(O)cc(F)c1 c1(CC)nnc2cc(N3CC(NC(C4CC4(C)Br)=O)CC4(CCC4)C3)ncn12 N1(C(C2CCC(C(C)C)CC2)=O)CC2CCC(C1)N2C(=O)Cc1cncn1C c1(C(=O)NC(CCCCNC(CC)=O)CO)cc2c(ccc3ccccc23)[nH]1 CC1CC(CC(=O)Nc2cc(F)ccn2)C(C)O1 CCCC(C)(CCC)C(=O)NC1CCCC(NC(c2c(C)nc(O)nc2S)=O)C1 C(=O)(C1(C)OC(=O)c2ccccc21)NCC1(c2cn(CC(CC)O)nn2)CCC1 C(CC(C(=O)N(C)CC)NC(=O)CCc1csnn1)=CC C1(=CC(=O)NCC2(O)CN(C(C=C(CCNC)Cl)=O)C2)CCC(C(C)(C)C)CC1 CC1OC2(C(=O)NCC=CCNC(c3cnccc3Cl)=O)CCC1C2 C=CCC(CC=C)C(=O)NC1CN(C(=O)CCc2cc(C)no2)C1 N(C1CN(C(c2cnn(CCO)c2)=O)Cc2ccccc21)C(C(CCCC)F)=O n1(CC(=O)N(C)CC2CC(OC)C2)cncc1C c1(C(=O)NC2(CC=C)CN(C(=O)C(F)(F)c3ccccc3)C2)cc(C)ccc1F C1(NC(=O)Cc2csc(Br)c2)CC2(C1)CN(C(c1ccoc1)=O)C2 c1(C(=O)NC2CC(C)N(C(=O)CCC3CC(F)(F)C3)C2)ncc(C#N)cc1Cl N1(C(CC(CC(=O)OC)C)=O)CCC2C1CCCN2C(c1cc(Cl)ccn1)=O c1(C(N2C3CN(C(C(CC)C)=O)CC32)=O)ccc(Cl)cc1Cl Cc1ccnc(C(N2CCC(N(C)C(c3cnc(-c4ncccn4)s3)=O)C2)=O)c1 c1(OC)cc(C)ccc1C(c1cccs1)Oc1cc(C)nc(-c2cnccn2)n1 N1(C(CNC(=O)Cc2ccc(F)cc2)=O)CCC2CCN(C(=O)CC(F)F)C2C1 c1(C(CC(=O)NCC(C)(C)NC(CCSCCC)=O)NC(N)=O)ccc(O)cc1 CC(O)C(C(=O)NCCC1OCCC1(C)C)NC(C1CC(OC2CC2)C1)=O C(=O)(C1=CS(=O)(=O)c2ccccc21)NCCC(C)NC(c1coc(Cl)n1)=O C1(CC(C)C)CNC(=O)CN1C(=O)CC1(F)CN(C(C2CCCCC(=O)N2)=O)C1 N1(CC(CC)O)C2CCCC1CC(NC(C1CCC(C(=O)OC)CC1)=O)C2 N1(C(C(CC)CNC(C)=O)=O)CCCC(C)(NC(=O)C(=O)OC(C)(C)C)C1 N1(C(C(C)(C)C(N)=O)=O)CC2C3CCC(C2C1)N(C(c1ccnnc1)=O)C3 N1(C(C(C(=O)OCC)F)=O)CCN(C(=O)CCC(C)(C)C)C2COCC12 c1(C(N(C)CC2CCCN2c2ccnc3ncnn23)=O)cc2cc(Cl)ccc2o1 C(=O)(CC(C(F)F)C(C)(C)C)NC1CN(C(C2(c3c(C)c[nH]n3)CC2)=O)CC1O C1(C(=O)OC)N(C(c2cc(C(F)(F)F)ccc2F)=O)CC12CCC2 CC1CC(NC(C2CCCCC2)c2cscc2Cl)CCO1 c1(C(=O)Nc2cncc(Cl)n2)cn2c(n1)CCN(Cc1cnoc1)CC2 CC(C)(C)CCC(=O)NC1(C(F)F)CC(NC(C2CCC3(CCC3)O2)=O)C1 c1(OC)cc(Cl)ccc1CNC1CC(C(=O)Nc2c(F)cccc2Br)C1 N1(C(c2cccc(C(=O)OC)c2)=O)CCC2(NC(c3cc(C(C)=O)on3)=O)CC2C1 c1(C(=O)NCC(C)(C2CC2)NC(C23CCCC2C3(F)F)=O)ccc(Cl)c(O)c1N c1(C(=O)NC2CN(C(C3CCCCO3)=O)CC2F)c[nH]c2c(Cl)cccc12 CCCC(C(C)CC)NCC(C)(C)CC C(=O)(C(C)(C)C1=CCSCC1)NC1CC(CNC(C(C(C)C)SCC)=O)C1 C1(NC(CCSCCC)=O)CCN(C(c2cc(C(N)=O)co2)=O)C1CC C1(CC(N2CCC(N(C)C(c3cnn(C(F)(F)F)c3)=O)CC2)=O)CCCOCC1 CC1=NOC(C(N2CC(CO)(NC(C3CC(C(F)F)(OC)C3)=O)C2)=O)C1 c1(C(N2C(CC(=O)NC(CNC(=O)OC)C)CCC2)=O)cncc(CO)c1 c1(C(N2CCC(N(C(=O)C(C)n3ccnc3)CC#C)C2)=O)cc(N)nc(Cl)c1 S(=O)(=O)(c1cccc(N2CCC(C)(N3CCCC3)C2)n1)N1CCC(C(C)O)CC1 Cn1cnnc1C1CCCC1C(=O)NCC=CCNC(c1cnsc1)=O.C1(C)(C)CC1 c1(C(=O)NCCC2(O)CN(C(C(C)(C)SC)=O)C2)ccc2cnoc2c1 CC1(C)CCC(C(N2CC(C)(CCC(=O)NCC(F)C(C)(C)O)C2)=O)C1 c1(C(=O)NCCCC(C)NC(=O)CN(C)CCO)c(F)ccc(F)c1F CC1=C(C(=O)NCC2CC3(CC3)CN2C(=O)C=CCF)CCS1(=O)=O c1(COC)cc2cc(c1)S(=O)(=O)N2.C(C)(CCc1ccncc1)(C(=O)OC)OC c1(OC)ccc(CC(=O)NCC2CN(C(=O)Cc3ccc(C)s3)C3CC23)cn1 C=CC1(C(=O)NC2(C)CCC2)CCN(C(c2c[nH][nH]c2=N)=O)C1 C(=O)(C(=O)C(C)(C)C)NCC1CC(C)N(C(=O)Cc2ccnc(Cl)c2F)C1 c1(C(=O)NC2CCC(CNC(CC3CC(=C)C3)=O)C2)c[nH]c(=O)c2ccncc12 N1(C(c2cc(OC)ns2)=O)CCN(C(c2ncc(C(F)F)cc2F)=O)C(CF)C1 C1(C(N2CC(NC(CC)=O)C2)=O)CC12CCC(F)(F)CC2 C1(OC)(CNC(=O)CCC2(C)CC2)CCN(C(c2cnn(C)c2Cl)=O)C1 C1(NC(C2CC(CNC(C(C(CC)C)NC(N)=O)=O)OC2)=O)CCCCCCC1O N1(C(C2CN(S(N)(=O)=O)C2)=O)CC2CC1CCC2NC(C1(C(F)(F)F)CC1)=O CC1CCC(NCCOc2cccc(Cl)c2)CS1(=O)=O c1(C(=O)NCC(COC)NC(=O)C(C)CN(C)C)cc(C)c[nH]1 c1(N2CCC(C(=O)NC)CC2)cc(NC(C)CCc2cn[nH]c2)nc(C(C)C)n1 C1(CC)CCCN(CCCNC(=O)NCc2nc(C)nn2C)C1 N1(C(C(C2(O)CCC2)NC(C(C(C)C)C#N)=O)=O)CCC2CN(C)CC2C1 c1(SCCCC(=O)OC(C(=O)OC2CCCOC2)c2ccoc2)ccc(F)cc1 c1(C(=O)NC2CN(C(=O)CC(F)F)C2)cncc2c(F)cccc12 C1(NC(c2c(C)n(C3CC3)nc2)=O)CN(C(C2CC(C)(O)C2)=O)CC(F)(F)C1 n1(CCSC)nnnc1C(c1csc(-c2ccsc2)n1)NC(C)CSC C(=O)(C1Cc2c(Cl)cccc21)NC1CCN(C(c2c(CN(C)C)cco2)=O)C1 CC1(C)CN(C(=O)CCCC(F)F)C(CNC(=O)Cc2ccc(Br)cn2)CO1 C1(NC(CN(CC#C)C(=O)OC(C)(C)C)=O)COCC1NC(=O)Cc1ccccn1 C1(C(=O)NCC(CNC(C2CCCCC2)=O)OC)CN(S(N)(=O)=O)C1 C12(CNC(C(CSC)(C)C)=O)CCC(CC1)N2C(c1c(C)nn(C)c1Br)=O c1(-n2c(SC)ncc2)ccc(C(=O)NCCCN(C(=O)Cc2ncco2)C)cc1 C(=O)(C(C)(C)COC(C12CCCC1(C(N)=O)C2)=O)OC N1(C(CCCC)=O)CCC2CC2(NC(c2sc(C3CC3)nc2C)=O)CC1 C1(COC(C2C(C)(C)CC(F)(F)CC2)=O)CC(c2ccncc2)=NO1 C(=O)(CCC(C)NC(=O)C=CC(C)(C)C)NCC(CC1CC1)OC N1(C(C(n2cc(COCC)nn2)C)=O)CCC2CCCC12 c1(C(C)C)cccc(NC(=O)C(C2CCCC2)NC(=O)C#CC2CC2)c1 N1(CCC2CCCNC(=O)C2)CCCc2cc(NS(C)(=O)=O)ccc21 C1(NC(=O)C(N2CCC(C(F)F)C2)=O)CCC(CO)CC1 N1(C(C=CC(C)NC(c2cc(C)nn2C)=O)=O)CCN(C)CC(C)C1 C1(C)(OC)CCN(C(=O)C(C2CCN(C(=O)CN(C3CC3)C(C)C)CC2)C)CC1 C(=O)(C(C)CC(N)=O)N1CC(CC=C)(C(=O)NC(c2ncccn2)CC)C1 C(=O)(C(CNC(c1cc(C)c(C)s1)=O)(CC)CC)NCC(=O)NCC=C C1(C(=O)OCC)C2COC(C(=O)NC3CCC(NC(C4CCCO4)=O)CC3)CC12 C1(C2CCN(c3cc(Oc4ccccc4)ncn3)C2)(NC(CCC(=C)Cl)=O)CC1 C1(CN(C(c2cc(SC)c(C)o2)=O)C)CCC=CCCC1.C12(CC1)C(=O)N2 c1(OC)ccc(C(=O)NC2CCCCC2CNC(=O)C=CC(C)C)cc1N Nc1ccc(C(=O)NCC2CC3CCC2N3C(=O)C(F)=C2CCCC2)nc1N C1(C(N)=O)COCC1C(N1CCC(c2nn[nH]n2)C1)=O.C12(CCC1)CC(=O)N2 Cc1cnc(C(N2CCCC(NC(=O)C(=C3CCCCC3)F)C2C)=O)c(F)c1 C1(n2cc(NC(c3cc(C#N)cs3)=O)nn2)CCCN(C(C2(C)CC2(Cl)Cl)=O)C1 Cc1cc(C(=O)NCC2CN(C(C3C=CCC3)=O)C3COCC3O2)cc(=O)n1C Cc1c(C(=O)N(C)CC2CCCN2C(c2nncn2C2CC2)=O)cccc1C#N N1(C(c2cnc(OC)nc2C)=O)CC2(CCN(C(=O)CC(F)(F)Cl)C2)C1 c1(-c2cn(C3CC(CC(=O)NC4C(C)SCC4)C3)nn2)cnn(C)c1C#N c1(C2(NC(N3C(C(CC)(C)C)CCC3)=O)CCCO2)ncccc1Br C=CCC(C(=O)NCC1CC(CNC(C2(SC)CCC2)=O)CO1)OC C1(C(=O)NCCOC(C)(C)CNC(c2nc(C3CC3)cs2)=O)OC2CCC1C2 c1(OC)ccc(C=CC(=O)N(C(C)CNC(=O)Cc2ccncc2F)C)cc1 c1(OC)cc(NC(C2CCCCC2NC(c2cncc(Br)c2C)=O)=O)c(F)cn1 N1(C(CC(=C)C)=O)CCC2(CO)CN(C(c3cc(CC(C)C)c[nH]3)=O)CC2C1 N1(CCNC(Cn2ncc(C)c2)=O)CCN(C(=O)C(C)(C)c2ccncc2)CC1 CC(C)C(C)(O)C(=O)N1CC(CNC(=O)Cc2ccc(O)nc2)CC(C)C1 CC(CCO)N(C(=O)CC1(NC(=O)CSC2CC2)CCC1)C C1(C(=O)Nc2cccc(NC(c3cc(C)sn3)=O)c2)(CC)CCC(O)CC1 C(=O)(C(C)(C)CCNC(=O)C=Cc1ccncn1)NCC(C(=O)OC)O NC(=O)CCCCC(=O)NCC1(F)CC(NC(C2CCC3(CCC3)C2)=O)C1 CC1(CNC(C2CC3(CC3)C2)=O)CN(C(c2ccnc(Cl)c2O)=O)CCO1 CC(C)CC(C)C(=O)NCC1CN(C(c2ncncc2F)=O)CCN1C CC#CCCC(=O)NCC1CCCC(NC(C2CCCN2CCCCC)=O)C1 c1(NC(CC(CC)N(C)C(C2CCCCC2)=O)=O)ccccc1C#N Cc1ccc(O)c(NC(=O)CC2(C)CCN2C(c2ccc(=N)[nH]c2Cl)=O)c1 C1(CNC(CCC)=O)CC2CN(C(=O)Cc3ncc(C)s3)CC12 CCC#CC(C)(C)NC(C1CC(C)N1C(c1ccccc1OC)=O)=O C1(NC(=O)CCc2ccccc2F)COC2(CCN(C(c3coc(Cl)c3)=O)C2)C1 c1(C(=O)NCC2N(C(c3c(CC)occ3)=O)CCC2)cc2c(cc1N)OCCO2 Cc1cnccc1C(=O)NCC1CC(F)CN1C(=O)C=Cc1ncco1 c1(OCC(=O)N(C2CC2)CC2CCCN2C(=O)C(O)C2CCC2)cnc(Cl)cn1 C(C)(C(=O)N(CC(C)N(C(=O)CSC(C)C)C)C)(C1CC1)OC N1(C(c2n(CCOC)ncc2)=O)CCC2(CCCN2C(C2CCN(C)C2)=O)C1 c1(NC(C(=O)N(CCC(COCCC(=O)OC)O)C)=O)cccc(F)c1F C1(CCC)(C(N2CC(O)(CNC(=O)CCn3nc(C)cc3C)C2)=O)CCNC1=O c1(OC)ccc(F)c(C(=O)NCC2CCCC2NC(=O)CSCC(N)=O)c1Cl C1(C(C)C(N2CCC(CO)C2)=O)CCN(C(c2cn(C(C)C)cn2)=O)CC1 CC(CC1CC1)C(=O)NC1(C(=O)NCCNS(C)(=O)=O)CCCO1 C(=O)(N=S1(=O)CCNC(C)CC1)c1c(OC)cc(C)cc1F N1(C(C)C(N2CC3CC3C2)=O)CCC2CN(c3ccn4nccc4n3)CCC12 C1(C(=O)NCCCN(CCCNC(c2cscc2C(F)F)=O)C)CS(=O)(=O)C1 c1(C(C)C)n[nH]cc1C(=O)NCC1(CNC(c2cn(CCO)nn2)=O)CC1 C#CCC(CC(=O)N(CCCCO)C)NC(c1cc(C)c(N)cn1)=O Cc1cnnc(O)c1C(N1CC2(C1)CN(C(C1(C)CCN(C)C1=O)=O)C2)=O CN1N=C(C(=O)N2CC(N(C(=O)Cn3ncc4cccnc34)C)C2)CCC1=O c1(C(=O)NCC(C)(C2CC2)NC(=O)C=Cc2cccs2)cc(O)ccc1F N1(C(C(C)C2CC2)=O)CCCCC1CN(C(=O)CCc1cccnc1Cl)C1CC1 c1(C(=O)NCC2CCC(NC(C3(CC4CC4)CC3)=O)C2)ccc(O)nc1 N1(CC)CC(C)N(C(C2CCN2C(=O)Cn2nc(C)cc2C)=O)CC1C c1(C(C)C)ncc(Cl)c(C(N2CC(C)CCC2CNC(=O)CCP(C)(C)=O)=O)n1 c1(OC)nc2ccc(C(N3CC(NC(c4cc(CO)ccc4Cl)=O)C3)=O)cc2[nH]1 c1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCCC2C)[nH]cc2c1CCCC2 c1(-c2nc(NC(c3cc[nH]n3)=O)sc2)cccc(Br)n1 c1(C(=O)NCCC2(C)CNC(=O)C2)ccc2cccc(F)c2n1 N1(C(c2n(CC)ncc2)=O)Cc2ccccc2C1C(=O)N1CC(C)(O)C1 C(=O)(CC(C(F)(F)F)n1ccnc1)NCC1(C)CCN(C(C=CSC)=O)C1 Cc1cccnc1CC(=O)NCCC1CCN(C(C2CCC(O)C2)=O)CC1 c1(N2C(CNC(CC3C(C)=NOC3=O)=O)CCC2)nc(C)cc(C)c1C#N N1(C(C2(CC)CCN(C(c3cccnn3)=O)C2)=O)CC2CCC(C1)O2 n1(CC)nnc(C)c1CNC(=O)C(C)=CCNC(C1(O)CCCC1)=O C(C(=O)NCC(O)C(C)C)(C(C)C)NC(C1(CC=C)CC=CC1)=O N1(C(c2cn(CCC=C)nn2)=O)CCC(F)C(NC(c2ccc(Cl)cc2F)=O)C1 N1(C(Cc2scc(C)c2)=O)CCN(C(c2nnc(O)cc2O)=O)CC1CC(F)F c1(C(N(CCN(C)C(c2cc(Cl)c(Cl)[nH]2)=O)C)=O)cn(C)c(=O)n1C Cc1sc2ccccc2c1C(=O)NC1CC2(C1)CN(C(=O)C=CC(C)(C)C)C2 c1(C(=O)NC2C(NC(C(C)N(C(C)=O)C)=O)CCC2)ccc(CC(C)C)cc1F C1(CC(N2CC(NC(c3cccs3)=O)C2)=O)CCCS(=O)(=O)C1 N1(C(CSc2cn(C)nc2)=O)CCC(CC(=O)NCC2CC2Cl)CC1 N1(C(c2c(C)nncc2)=O)CC2(CC2)CC1CNC(C1(F)CCOC1)=O CC(C)CCCCC(=O)NC1CC2(C1)CC2C(=O)NCC1CCCN1C c1(C(=O)NC2CC3N(C(C4(OC)CCC4)=O)C(CC3)C2)cnn2c1C(C)CCC2 C(=O)(CC(C)(C(F)(F)F)N(C)C)NC1(CO)CCN(C(COCCCC)=O)C1 C1(C(=O)NCc2cncc(C)n2)C2CCC(C2)N1C(=O)C(c1ccccc1Cl)O C1(NC(C2CC3C=CC2O3)=O)CCN(C(c2ccc(Br)s2)=O)C12CC2 C1(NC(C2C(C)CCC2)=O)CCCC(C(=O)NC2CC3CCC2C3)C1 C1(C(CNC(CCOC)=O)NC(C2CCSCC2)=O)CCCCC1 c1(C(N(C2CCN(C(C3(CC)CCC3)=O)C2)C)=O)cc(Cl)ccc1N CCCCCC(O)CC(=O)NCCn1cc(C(N2CCC(n3cccn3)C2)=O)cn1 c1(CC(=O)NC2CCC3(CN(NS(CC=C)(=O)=O)C3)O2)sc2ccccc2c1Cl CCCC(C)CC(=O)NCC1CCN(C(=O)Cc2cc(F)ccc2O)C1 C1(C(=O)NC(C)CNC(=O)Cc2csc(-c3ccccc3)n2)CCN(C)CC1 c1(C(=O)NC2(CNC(CCCOCC)=O)CCOC2)cc(Cl)c(Cl)[nH]1 N1(C(C2CCC(CC)O2)=O)CCC(NC(c2ccc(CO)s2)=O)C(CO)CC1 C1(CNC(C2(NC(C)=O)CCCC2)=O)CN(C(C2CC2C(C)C)=O)C2(CCC2)C1 c1(CC(=O)NC2CN(C(C=C(CCC)C)=O)CC(C)C2)c[nH]c2cc(OC)ccc12 Cc1cc(C(=O)N(C2CC(C#N)C2)CC(=O)NCC(c2ncc[nH]2)C)ccc1O O=C1NCc2ccc(NC(C3(C(F)F)CCCO3)c3nnnn3C3CC3)cc21 CC1CC(CCNC(C2(C(N)=O)CC2)=O)CCN1C(c1ccc(Cl)o1)=O c1(C(N2CC(CNC(C(CC)C(C)O)=O)(OC)C2)=O)coc2cc(OC)ccc12 c1(OC(C(=O)NCC(C)NC(C(C(C)C)NC(N)=O)=O)C)ccccc1C#N Cc1cccc(C(=O)NCC2CC(NC(c3cccn3Cc3cccs3)=O)C2)n1 c1(CC(=O)NC2C=CCN(C(C3CSCCS3)=O)C2)cccc(C(F)F)c1 CC1CN(C(C2CCS(=O)CC2)=O)CC1CNC(C1CN(S(C)(=O)=O)C1)=O C=CC12CCN(CC1)C(=O)NC2.c1(CC(=O)OC(C)(C)C)cc(O)c(O)c(O)c1 C(=O)(C1=C(Cl)CCOC1)NC1C(C(=O)NCCC=CC=C)C2CCC1C2 CCCC(CC(C)C)C(=O)NC(C)(C)CCCNC(=O)COCC(F)(F)F N1(C(c2ccc(SC)s2)=O)CC2CC2(CNC(C2CC(F)(CO)C2)=O)C1 c1(CC)cnn(CNC(C2(C(C)NC(C3CC(OC)C3)=O)CC2)=O)c1 C1(C(=O)NC(CC)C(N)=O)CCC2(CCN(C(=O)CCc3cccnc3)CC2)C1 c1(CC(C(=O)NC2CC2c2cocn2)NC(N)=O)ccc(O)cc1 O=C(NNc1ccc(-c2nn[nH]n2)cc1F)C1CCN(c2ncccn2)CC1 N1(C(c2cc(Br)c(F)cn2)C(=O)NC)CCc2cc(OC)cc(OC)c2C1 c1(SCC2C(C(=O)OCC)(C(=O)OCC)C2)cncnc1O.C(C)(C)C c1(C(C)NC(=O)CC2CCCN(C)C2)ccc(CNC(c2cnn(C)c2)=O)cc1 CCCCCC(=O)NC1CC(NC(=O)COCP(C)(C)=O)C(O)C1 CCCCC(C)CCC(=O)NC(C)CCCC(=O)NC1CC1(CO)CO C1(CCC)(C(=O)NCC2CCC2NC(c2sccc2C)=O)CCNC1=O Cc1cc(C(=O)NC2CCN(C(c3cnc(O)n3C)=O)C2)nn1C1CCOCC1 C(=O)(C(C)N=c1cncc[nH]1)N1C2(CCN(C(C3CC=C(C)CC3)=O)C2)CCC1 c1(NC(N2CCC(c3scc(C#N)n3)CC2)=O)ncc([N+](=O)[O-])cc1C#N S(=O)(=O)(c1cncc(Br)c1)N1CC(NC(c2cc(Br)c(Cl)cc2F)=O)C2(C1)CC2 c1(CCC)[nH]nc(C(=O)N(CC(C)NC(c2ccc(Cl)c(N)c2)=O)C)c1[N+](=O)[O-] O=C(CC1OCc2cc(Cl)ccc21)NCC12CC(CN1C(C1CC13CCC3)=O)C2 N1(C(c2ccc(COC)o2)=O)CC(NC(c2cc(C#N)oc2C)=O)CC12CCC2 c1(C(=O)NCCCN(C(=O)C(F)CC2CCC2)C2CC2)ccccc1S N1(CC)CCOC(C(=O)N(CCC(=O)NCC(N2CCCC2)C)C(C)C)C1 N1(C(c2cnc(OC)c(Cl)c2)=O)CC2(CCCN(C(=O)C(C)C3CC3)C2)C1 C12(CCOCC1)C(=O)N2.C1(CN)CCCC(NC(=O)C(C)c2cc[nH]n2)C1 CC(C)(CC(=O)NCc1ccc(CCNC(c2coc(CO)c2)=O)cc1)C(F)F CC(C)C(O)C(=O)NCC(C)(F)CNC(c1ccn(C)c1C1CCC1)=O c1(N2C(C)CC(NC(C3CCC(=O)N3C)=O)CC2)nc2cccnc2s1 N1(Cc2onc(-c3c(Cl)cccc3)n2)CCC2CCNC2C1 C(CC(=O)N1CCC2C(C1)CN2C(c1cnc(C2CCC2)s1)=O)(C(F)(F)F)OC c1(C(C)NC(C(COCC)NC(=O)Cc2nccn2C)=O)cccc(C)c1 c1(C(N2CCOCC(C3CC3)C2)C(=O)NCC(=C)C)noc2ccc(Br)cc12 CC1(C)C(CNC(=O)CC2CCC(O)C2)CCN1C(=O)Cc1ccc(O)c(Cl)c1 C1(C(N(CCCCNC(c2ncoc2C2CC2)=O)C)=O)CC12CC(C)(C)C2 C(=O)(C1=C(Cl)CCOC1)NCC1N(C(c2ccc(C#C)cc2)=O)CCC1CC N1(C(c2c(COC)cccn2)=O)CC2=C(C1)CN(C(C1(C)CC(C#N)C1)=O)C2 N1(C(CN(C(CSCC=C)=O)CC)=O)CCC(C(=O)NC)C1C c1(OCCNC(C2(Br)CC2)=O)ccc(-c2ccc(OCC3CC3)nc2)cc1F C(C)(CO)(C(C)(C)O)NC(CC1CCN(C(C(CC)CC2CC2)=O)C1)=O c1(C(N(C(CNC(C)C(N)=O)=O)C)C)nc(-c2ncccn2)no1 C1(C(=O)NCc2cc(OC)no2)CCN(C(=O)C(CC2CCC2)OC)C12CCC2 C(=O)(C(C(C)C)OC)NC1(CCC(=O)N(C(C=C)C)C)CCCC1 Cc1nc(O)ccc1C(=O)NC(C)CNC(=O)C(CO)c1ccccc1 c1(OC)ccc(C(N)=O)cc1C(=O)N(C1CN(C(C2CCN(OC)CC2)=O)C1)C C1(C(=O)NC2CN(C(CCOC)=O)CC2C(F)F)CC(c2cnn(C)c2)=NO1 C(=O)(C#CC1CCOCC1)N(CC(O)CNC(c1scc(F)c1Br)=O)C N1(C(c2c(CC)noc2)=O)CC2CC(NC(c3cnn(C(C)C)c3C)=O)C2C1 C1(C(N(CCOC)Cc2ccc(OC(C)C)cc2)=O)CC(C)SC(C)C1 Cc1ncc(C(N2CCC(CNC(c3cc(C(F)F)cs3)=O)C(C)C2)=O)c(C)n1 C(=O)(C(C(=O)N1CC(CC(C)NC(=O)C(CCSC)SC)C1)C(C)C)OCC C(C(CC(C)C)C(=O)NCC(C)CC(=O)N1CC(c2ccccc2)C1)OC Nc1ccc(Cl)c(C(N2CC=CC2CNC(=O)Cn2cnc([N+](=O)[O-])c2)=O)c1 n1(CC)cc(C(=O)NC2(C)CC(NC(c3cc(C(N)=O)cs3)=O)C2)c(C)n1 CCC(C)CCCC(=O)N(CCCNC(C1CC2CCCC(C1)C2)=O)C1CC1 N1(C(c2scc(C)c2)=O)CC(F)(F)CC1CNC(C1COCC(=O)N1C(C)C)=O S(=O)(=O)(c1cnc(NCC(O)CN(C)C)c(Cl)c1)N(CC(COCC(C)C)O)C CCS(=O)(=O)c1cccnc1NC(=O)C(=O)NCCCCOC(C)(C)C C1(NC(c2cc(C)c(O)cc2)=O)COC2C(NC(C3COC(C)(C)C3)=O)COC12 N1(C(c2c(CC)ncnc2)=O)CCN(C)CC1C(N1CC2CC1(CO)C2)=O Cc1cc(C(N2CC(c3cn(CCCF)nn3)C(C)C2)=O)c(C)o1 C1(C(N(CCCCNC(c2cc(Cl)c(Cl)s2)=O)C)=O)CCN2CCOCC12 c1(OC)ncc(Cl)cc1CC(=O)NC(c1ccc(Br)nc1)C(F)(F)F N1(Cc2cc(N(C(C)C(=O)NC)C(C)=O)sc2)CCC(C)(NC2CCCCC2)C1 C1(C(N(CC(C)N(C(CC(C)C)=O)C)C)=O)CCC(F)CC1 N1(C(CSCC=C)=O)CCC(CCC(=O)NCCN2CC=CCC2)CC1 C(=O)(CC(C)(C)OC)NC1CCC(CCC(=O)NC(C(=O)OC)CO)C1 c1(C(=O)NC(CNC(c2n(CCC)ncc2)=O)(C)C)cn2nc(C)cc2[nH]c1=O C1(CC=C)(NC(=O)C=CS(C)=O)CCCN(C(=O)CCc2cncc(O)c2)C1 C1(C(=O)OC)CCCCC1O.C(C(=O)N(CC(O)CO)C)(C1CC1)N c1(C(=O)NCC(C)N(C(=O)CCc2ncc[nH]2)C)cc(Br)c(F)c(F)c1F c1(NC(CCC2N(C(c3cc(C)on3)=O)CCC2)=O)cccc(Cl)c1F Cc1cncc([N+](=O)[O-])c1N1CCCCC(NC(=O)CC2CCC(=O)NC2)C1 N1(C(CC)CC)CC(C(=O)NCCC(C)NC(=O)CC(=O)OC)CC1=O CCCCCC(CC)C(=O)NCC(C(=O)NCCOC1CC1)C(C)C CC(C)(CC(=O)N1CC2CCC1CN2C(C1(S(C)(=O)=O)CC1)=O)CC(F)(F)F N1(C(c2nc(CCC)oc2)=O)CCC(NC(c2cc(C)c(C)[nH]2)=O)C(F)C1 N1(C(CN(C(=O)CCc2nccs2)C)=O)CCN(C(=O)CC(F)(F)F)CC1 N1(C(c2ccc(C)cc2O)=O)C2CCC1CC(NC(c1cccc(C)c1O)=O)C2 C#Cc1cccc(C(=O)N(C2CCC(NC(=O)CC3=CCOCC3)C2)C)c1C CCC(CC(=O)N(C)CCc1cnc[nH]1)NC(c1ccc(NC)cc1)=O N1(C(C2C(C(C)(C)C)CC2)=O)CC(=O)NCC1C(N1CCC2(CCC2)C1)=O Cc1nn(C)c(NC(C2(Cl)CC2C(=O)OC(C)(C)C)=O)c1-c1ccccc1 N1(C(c2cncc(Cl)c2)=O)CCCN(CCCCNC(=O)C(F)(F)C2CC2)CC1 CCC(C(=O)NCC1CN(C(C2CC23CC3)=O)C1)c1cccnc1 N1(C(c2c(C#N)ccs2)=O)CC2(CCCC2)C1C(=O)NC.C(C(=O)NC1CC1)N c1(OCCCC(=O)NC2(C)CN(C(C3CCCCN3C)=O)C2)cc(Cl)ccc1Cl S(=O)(=O)(c1c[nH]c(C(N2CC(=O)NC(C)C2)=O)c1)NCC(C)O C12(NC(C(c3ccc(OC)cc3)CC)=O)CC(C1)N(C(c1ccnnc1S)=O)C2 CCCC(C(O)C(=O)N1CCC(F)(C#N)C1)NC(=O)CC(C)CC N1(C(CC(C)SC)=O)CCCC(C(N2CCC(c3ncn(C)n3)CC2)=O)CC1 C12(CC(F)(F)C1)C(=O)N(C)CCOC2=O.CCC(C)C(=O)NC(C)(C)C c1(C(=O)NC2CC(CNC(C(C)SC(C)C)=O)CC2O)ncsc1S(N)(=O)=O OC1CCC2(CCCN(Cc3ccc(F)cc3Br)C2)C1 Cc1c(Cl)ccc(Cl)c1NC(=O)CN1CCN(C(=O)C=CC2CC2)CC1=O c1(NCC(CC)(C)CC)cc(Br)ccc1S(=O)(=O)N1CCn2nc(C)cc2C1 N1(C(c2c(C)coc2)=O)CC(NC(=O)CCCn2ccnc2)C2CC12 C(c1ccnn1C)=CC(=O)N(C)CC1CCN(C(COCC(=O)NC)=O)C1 c1(C(N2CC(NC(CCCCCSC)=O)C(C)C2)=O)cc(F)cc2cnccc12 C#Cc1cc(C(=O)NC(CC(C)CC)C(=O)NCC2(OC)CCC2)ccc1C C1(C(=O)NCC(C)(C2CC2)NC(c2coc(Br)n2)=O)CC12CCOC2 C(=O)(C1=C(C)CCC1)N1CC(C(=O)NCC(C(CC)C)C)OCC1 CC(C)CCCCC(=O)N1CC2CCC(C1)N2C(C1(n2nccn2)CC1)=O Cc1cnc(N2CC3(CCC(C(=O)NCC(F)CO)O3)C2)c([N+](=O)[O-])c1 N1(C(C2ON=C(C)C2)=O)CCC2C(CCN2C(c2cc(C(C)C)oc2C)=O)C1 C1(NC(c2n(CCC)ccc2)=O)CCCCCN(C(C2CCCNS2(=O)=O)=O)C1 c1(NC(C)=O)cc(SC(C2CCCCC2)C(=O)Nc2ccccc2)ccc1F C(=O)(C(CC)CC)NC1C(C(N(CCC#C)CCO)=O)CC1 Cc1cnc2n1CCC(C(=O)N(C1CN(C(C3CC34CCSCC4)=O)C1)C)C2 C1(NC(CCC(=O)NC)=O)CC1C1CCCN(C(c2c[nH]nc2OC)=O)C1 C12(C(=O)NC(C)CN(C)CC3CC3)CC(CC3CC3c3ccsc3)(C1)C2 N1(C(CC2N(C)CCC2)=O)CCC2(CC(NC(=O)CCCc3cccnc3)C2)C1 C1(CC)(COCC)CCN(Cc2ccccc2)C1 C12(CN(C)C(C3CN(c4ncc(C(C)(C)O)cn4)C3)=O)CC=CC(C1)OC2 Cc1cnc(CC(=O)NCC2CCC(NC(C3(C(F)F)CCCC3)=O)C2)[nH]1 N1(C(C2(OC)CCSC2)=O)CC2CCC(C1)C2NC(c1ccnc2ccnn12)=O CC(C)C1=NOC(C(=O)N(C)CCNC(=O)C(C(C)(C)C)OC(C)(C)C)C1 N1(C(c2n(C)ncc2)=O)CC(NC(=O)Cc2cc(-c3ccco3)on2)C(F)C1 C#CC1(C(N2CCC(C(C)C(=O)NCCCCC=C)C2)=O)CCCC1 C1(CNC(c2n(C(CC)C)nnn2)c2ccn(CCF)n2)CCC(C)(C)CC1 c1(OCC)cccc(C(=O)NCC#CCNC(=O)C(C)(C)C(C)O)c1N Cc1cc(F)cc([N+](=O)[O-])c1NC(c1nc(NC(C2CCCS2)=O)cn1C)=O CN(CCCC(=O)NCCC1CC(NC(=O)C#CC2CCC2)C1)N=O c1(CNC(CCCSC)=O)cccc(CN(C(=O)C2=CCC2)C)c1 C(N=c1nc(O)c(Br)c[nH]1)C1(C)CCN(C(c2c(C)n(C)nc2)=O)C1 c1(ONC(n2cc(CN3CCCC3c3nc[nH]n3)nn2)=O)cccc(F)c1 CC(C)(CCNC(=O)Cc1csnn1)C(=O)Nc1ccc(O)c(F)c1 c1(CNC(=O)CC(Cl)Cl)cccc(C(N2CC(c3nc(=O)o[nH]3)C2)=O)n1 c1(C(N2C(CCNC(c3n[nH]c(CC)c3C)=O)CCCC2)=O)ccc(N)c(F)n1 Cc1nn(CC(=O)N(C(C)CCNC(C2(C)CNC(=O)C2)=O)C)c(C)c1Cl Cc1cc(NC(N2CC3CCCC(C2)C3(C#N)C)=O)c(Br)cc1I CC1CN(C(C2CCCC(O)C2)=O)CC1NC(c1cc(-c2ccccc2)co1)=O CC(=O)CCCC(=O)N1CCC(O)(CCNC(C2CN3CCN2CC3)=O)C1 N1(C(CCSC)=O)CC2(C(=O)NC(C)C(F)F)CC1CO2 c1(CC(CNC(=O)CC2CCCNCC2)OC)cccc(Cl)c1 Cc1n[nH]c(C)c1CN(C(C)C)Cc1ccccc1-c1ccccc1 N1(C(c2cc(COC)cn2C)=O)CCC2CCN(C(c3cccnc3N)=O)CC12 C1(C(=O)NCC2C(CNC(CC3(COC)CC3)=O)C2)CC2CC2C1 CS(=O)(=O)c1ccc(CNC(C2CCN(C(=O)CC(O)C3CCCC3)CC2O)=O)cc1 C1(CC(=O)OCCOC2CCNC2=O)CCC(C2CC2)O1 C12(C(N(CC(C)NC(c3ccccc3CC#N)=O)C)=O)CC(C1)C(C)(C)O2 c1(OC)cc(C)ccc1C(=O)N(C1CCN(C(=O)CCCC(C)=O)CC1)C c1(C(N2CCCC(CN(C(CSCC=C)=O)C)C2)=O)ncc(Cl)cc1Cl c1(C(=O)NCC(=O)NC(C)CNC(c2coc(Cl)n2)=O)ccccc1CC#N C1(CNC(CCC)=O)CCN(C(=O)C(C(C)(C)C)N2CCNC2=O)CC1O c1(C(=O)NC(C)C(C)NC(c2ccc(C(F)F)c(F)c2)=O)ccc(O)c(Cl)n1 C1(C(N(C)CCOCCNC(C2CCCC(=O)N2)=O)=O)Cc2ccccc2O1 Cc1nn[nH]c1C(=O)N(CCO)Cc1cc[nH]n1 c1(C(=O)NC(C(C)C)C)cc(CNC(=O)C=Cc2cncs2)on1 N1(C(c2nc(OC)oc2)=O)CCCC12CCN(C(=O)CSc1nncn1C1CC1)C2 N1(C(C(=O)NCC)=O)CC(NC(C2CS(=O)(=O)CCO2)=O)CC2(CC2)C1 N1(C(C(CC)C(C)O)=O)CC2CC(NC(=O)C(F)CC3CC3)CC2C1 Cc1cnc(C(N2C(C(N3CCCC3C(O)CO)=O)CC2C)=O)c(C)c1 c12ccc([nH]1)CNC2=O.C(C#CCNC(C=CCOC)=O)N(C)C C1(N(C(c2c(CCC)n(C)nn2)=O)C)CCCCN(C(=O)C(C)(C#N)CC)C1 C1(CNC(=O)Cn2cccn2)C(C2CC2)CCN1C(c1ncc(C(F)F)s1)=O N12CCC(C3CC3)C1C2=O.C(=O)(CCC(=O)NCC(c1ncc[nH]1)C)NCCC c1(NC(CN(CCCCO)C(c2ccncc2)C)=O)ccc(C#N)cc1F N1(C(C(C2(C)CC2)NC(C(C(C)C)C(C)C)=O)=O)CCC2(CCOCC2)C1 c1(C(N2CC(F)(C(=O)NC(C3CCOC3)C)C2)=O)cc(C#N)ccc1Br N1(C(Cc2c(C)n[nH]c2C)=O)CCCCC(N(C)C(c2ccncc2Br)=O)C1 N1(C(C2CC(C)N(C)C2)=O)CCC2(C=C(C(=O)N3CC(NC(N)=O)C3)C2)C1 N1(C(C2(C)CC(C)C2)=O)CC2CCN(C(=O)C=Cc3ccc(Cl)cc3)C(C2)C1 CN1CC(N(C(=O)CC2CN(CCC3(C4CC4)CC3)CCO2)C)CCC1=O c1(C(N(CCCNC(C(COC2(C)CCC2)=O)=O)C2CC2)=O)cc(F)cnc1O CC(C)C(C#N)C(=O)N(CCCC(=O)NC1(CCO)CCCC1)C S(=O)(=O)(c1cccc(F)c1)NCC(N1CCN(C(c2ncn(C)n2)=O)C2C1C2)=O C(=O)(C#CC1CCCC1)N1C(C(CNC(CN(C(C)=O)C)=O)(C)C)CCC1 C(=O)(C1CCc2oc(C)nc21)N(C(C)CNC(c1cc(C)no1)=O)CC CC(C)C(CO)CCNC(=O)CC1CC(C)N(C(=O)COC2CCCC2)C1 c1(CC)cc(C(=O)NC(C)(C)CNC(c2ccc([N+](=O)[O-])[nH]2)=O)cc(O)n1 C12(C(N3CC4C(CNC(C5CCC(=O)NC5)=O)C4C3)=O)CCC(CC1=O)C2 C1(C)(C(=O)NCC(C)(C)NC(C(CC)n2ccnc2)=O)CCC(=O)N(C)C1 N1(C(C(COC(C)C)NC(C)=O)=O)CC=CC(NC(C2(C)CS(=O)(=O)C2)=O)C1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1CC(F)(CNC(C2CC(C)C2)=O)C1 N1(C(C2CN(C(C)C)C(=O)C2)=O)CCCN(C(C2CC(CF)C2)=O)C(C)C1 c1(C(=O)N(CCOCCNC(c2cc(CCC)on2)=O)CC)cc2nc[nH]c2cn1 CCCCC(C)(C)NC(=O)C(COC(C)C)NC(c1nc(O)sc1C)=O c1(C(N2C(C(=O)NCC3(OC)COC3)COCC2)=O)cc(C)c2ccccc2n1 C1(C(=O)NCC(C)CN(C(=O)Cn2ncn(C)c2=O)C)CCC2(CCC2)CC1 C(=O)(C(C)CC(N)=O)N1CCC(CN(C(C(=O)NC)C)C)C1 C1(C(N2CC(C(CC)C)C2)=O)CSCCN1C(c1ccc(Cl)o1)=O CC1(C)COC(CC(=O)NCC(=O)NCC(=O)NCC(F)F)C1 N1(C(c2c(OC)nccc2)=O)CC(C)C(NC(c2cccc(Cl)c2)=O)C(C)C1 C(=O)(C(C)(C)C(O)C(C)C)NC1(CC=C)CCN(C(=O)C(C)CS(C)=O)CC1 c1(C(C)=O)cc(F)ccc1OCC(N1CCCC1)=O.C(C)(CN=[N+]=[N-])O CC(C)C(CCNC(c1nccnc1N)=O)NC(=O)CC1CCC(C)C1 N#Cc1cccc(C(=O)NCC2(NC(c3cccnn3)=O)CC2)c1 Cc1coc2c(C(N3CCCC(CCNC(=O)C(C)CC(F)F)C3)=O)cccc12 C1(CC(=O)N(CC(CC)NC(=O)CC2OCCCO2)CC)OCCC1C N1(C(C(C)(C)C)=O)CCN(C(C2CCC(=O)O2)=O)C(CC(F)F)C1 CCC(CC(=O)N1CCCC1(C(=O)NC1CC(C)(O)C1)CC)CC(C)C c1(C(=O)NCCCN(C(C2ON=C(C)C2)=O)C2CC2)cccnc1-n1ccnc1 c1(C(N2C(CCNC(C3CC3C3CC3)=O)COCC2)=O)cccn(C2CC2)c1=O N1(C(c2ccc(CC)cc2)=O)CCN(C(=O)C2=NNC(=O)C2)CC1CC(F)(F)F C(=O)(C(C)N1CC(C)C1)NCC(=O)NCC(=O)N(C(CC)C)C C12(C(=O)NC3C(N(C)C(c4conc4C4CC4)=O)CCCC3)C(=O)C3CC1C2C3 C1(O)(C(=O)NC(C(C)NC(=O)Cn2cnnc2O)C)CC(F)(F)C1 C1(NC(C=C(CCC)C)=O)CC2(C1)CC2NC(c1ccc(C2CC2)nc1)=O C12(C(N3C(C(C)(C)NC(C4CCS(=O)(=O)N4)=O)CCC3)=O)COC(CCO1)C2 N1(C(c2cc(CC)c(C)s2)=O)CCC(O)(CNC(=O)C(F)CC2CC2)CC1 c1(C(=O)NCC(C)(C)NC(=O)Cc2ccncc2)csc(-c2ncccn2)n1 CC1CN(Cc2noc(-c3cccc(=O)o3)n2)CC(C)O1 C(=O)(C(CC1CC1)NC(c1ccn(CCF)n1)=O)N(CCOC)CC N1(C(c2c(C)nns2)=O)CCC2C(CCN2C(C2CC3(C2)CC3F)=O)C1 N1(C(c2c(C)noc2)=O)CCN(C(C)CNC(=O)C=CCF)CC1 c1(CNC(C(COC)C)C)cc(-c2cn(CC3CC3)nn2)nn1C C1(CCC)CN(C(c2cncc(N)c2C)=O)CCN1C(C1CC1C1CCCC1)=O c1(CNC(C2(CF)CCCC2)c2nnnn2C2CC2)ccc(C(F)(F)F)nc1C c1(CC)ccc(CC(=O)NCC2CCC(NC(=O)CC(F)(F)F)C2)cc1 c1(C(=O)NC(CCCNC(C(c2ccc(F)cc2)CC)=O)C)cc([N+](=O)[O-])n[nH]1 c1(N(C(N=c2nc(CCC)[nH]o2)=O)c2ccc(C)cc2)ncnc2cnccc12 CC(C)CC(C)CNC(=O)NC(C(F)(F)F)C1CCC1 c1(NC(C2C(C(=O)Nc3c(C(=O)NC)cccc3)C2)=O)cnc(O)nc1O Cc1ccc(C(=O)N(C2CCC(NC(c3ccc(O)nc3Cl)=O)C2)C)c(F)c1 CN1CCC(C)(C(N2CCC(C(N3CCC(CC(C)(C)C)C3)=O)C2)=O)C1 CC1CCC(CC(=O)NCC(O)CN(C(=O)C(F)=CCCF)C)OC1 N1(C(C(C2CCOCC2)C)=O)CCCC(CN(C)C(C2CC23CC3(F)F)=O)C1 C1(CC(=O)NC)CN(C(=O)CCc2cc[nH]n2)CCN1C(=O)C=C(C)C O=C(NN=Cc1ccc(Br)c(Cl)c1)c1cccc(F)n1 N1(C(c2ccc(OC(C)C)cn2)=O)CCC(C(=O)O)C(F)(F)C1 CC1(C#N)CCN(C(C2C3CCC(C3)C2NC(=O)C(F)C2CCCC2)=O)C1 N1(C(CN2CC(C)(C)C2)=O)C2CCCC1CN(C(C1CCc3nnnn3C1)=O)C2 C=CC(CC)C(=O)NC1CCN(C(C2C3CC(=O)CC23)=O)C1C Cc1nn(CCO)cc1C(=O)NCCC1CCN(C(=O)CCc2nccn2C)C1 C1(CNC(c2n(C(C)C)nnn2)c2ccc(C3CC3)o2)CC2(C1)CC(F)(F)C2 n1(CC)nc(C)c(C(=O)NC(C)C(CO)NC(=O)CC2CCCOC2)c1C(F)F C1(NC(C(CC)C)=O)CCN(C(=O)COc2ccc(F)c(Br)c2)C12CC2 C1(CN(C(C2CC(C3CC3)C2)=O)CC)CCN(C(=O)CCc2nccs2)CC1 c1(CNC(C2(C3N(C(=O)C=C4CCCC4)CCC3)CC2)=O)ccc2nc[nH]c2c1 c1(OC)ccc(-c2noc(COC(=O)C3CC3)n2)cc1NC1CCCCC1C c1(C(N2CCN(C3CC(C)(C)OC3=O)CC2)=O)cnc2c(c1)CCCO2 C1(CNC(C=CC(N)=O)=O)CC(O)CN1C(c1cc(-c2cccs2)on1)=O Cc1ncc(Br)cc1NC(C1CCC(NS(=O)(=O)Cc2ccccc2)CC1)=O c1(C(=O)NCC2C(NC(C(c3cscn3)N(C)C)=O)CC2)ccc2nonc2c1 C(=O)(C(C1=C(C)CCCC1(C)C)N1CCCC1C1CCCCO1)NCC C1(CNC(C2CCC(COC)C2)=O)CC2(C1)CN(C(=O)C=C(C)Cl)C2 N1(CC(=O)N(CCC)CCC)CC(NC(c2c(C)cccc2F)=O)CCC1C c1ccc(N2CCC2C2CCC2)cc1.c12csc(n1)CN2 N1(C(CCc2n(C)ncc2)=O)CC(NC(C2(CO)CCOC2)=O)CC2(CC2)C1 CC(C)(C(=O)NCC(=C1CN(C(=O)COc2ccon2)C1)F)N1CCCCC1 N1(C(CC2CCC(=O)N2)=O)CC(C(N2CC(CO)(CO)C2)=O)C(C2CC2)C1 C1(S(N)(=O)=O)(C(=O)NCC2CN(C(c3ncn(CC)n3)=O)C2)CC1 N1(C(C2CCN(C(c3cc(CC)[nH]n3)=O)C2)=O)CCC(C)(CCO)CC1 c1(C(N2CC3CCC(O)CC3C2)C(=O)NC(CC)(C)C)ccc2ccccc2c1 N1(C(C(c2ccccc2)OCC)=O)CCCCC(NC(C2CC=CCC2)=O)C1 c1(CC(=O)NC2C(CNC(C3(C)ON=C(C)C3)=O)C2)cccc2nsnc12 c1(C(N2CC(OCCNC(=O)CCCCC3CC3)C2)=O)cc[nH]c2nccc1-2 C1(CC(=O)C(C2CN(C(C)=O)C2)=O)C=CC(OC)C1.C(C)(C(=O)NCCN)=CC C1(C2CCCN(C(c3cscn3)=O)C2)(NC(C2CCC(=O)NC2)=O)CC1 N1(C(c2cc(CC)oc2C)=O)CC2CCN(C(C3CC34CCOC4)=O)CCC2C1 c1(C(=O)NC2(CC=C)CCN(C(=O)CCC3CCCCO3)C2)cc(O)nc(C)n1 CCC(CC)C(C(=O)NCC(CC1CC1)C(=O)NCC1CC(F)C1)OC CCCCC(O)CC(=O)NC1CCCC1CNC(c1ccc(CO)c(F)c1)=O C1(CNCCC2CCCN(C(CC3(C(=O)OCC)CC3)=O)C2)CCCC(C)(C)O1 C(=O)(C(F)(F)C(C)(C)O)NCc1ncc(C(N(CC(COCC)O)C)=O)cn1 C(CC(=O)NCc1c(F)cccc1F)(C(F)(F)F)NC(=O)C=CC1CCCC1 CCCC(O)(CCC)CC(=O)NC(C)(C)C(C)NC(c1ccn(CC(F)F)n1)=O N1(C(C(C2CCC(=O)N2)C)=O)CCCN(C(=O)C(N)=O)CCC1 C=C=CCCC(=O)NCC(C)(C)CN(C(=O)Cc1nocc1C(C)C)C c1(C(=O)NCC(CC)NC(=O)CC2CCN(C)CC2)ccc(C)nc1C(C)C N1(C(COCCCC(C)C)=O)CC2COCCC2(NC(=O)C(C)NC(N)=O)C1 C(CC(=O)N(C)OCC(=C)C)NC(C1CC2COCC2C1)=O.C(CCO)CC#C c1(C(=O)NCCN(C(C(c2ccc(C)o2)C)=O)C)scc(C)c1Cl Cc1ccc(C)c(C(N2CC(NC(c3cc4c(ccn4C)s3)=O)C2)=O)c1C C1(C(N2CC(NC(c3coc(C(N)=O)c3)=O)C(O)C2)=O)CCOCC12CCCCC2 N1(C(C(CC(=O)OCC)(C)C)=O)CCC2C1CCCN2C(=O)C(F)CC C(=O)(C(C)CNC(=O)C(Cn1cccn1)NC(=O)CCC1CC(C)C1)OC C1(CNC(=O)NCC(C(C)C)F)CCCCC12CC2(F)F C#Cc1c[nH]nc1C(=O)NC(C1CC=CCC1)C(N1CC(C#N)C1)=O c1(SC(CC(C)=O)C)ccc(OC(C2(C(=O)O)CCOC2)=O)cc1F c1(C(=O)NC2C(C(C)C)CN(C(=O)Cc3cnns3)CC2)cccc2cncn12 N1(NCCCC(C(=O)OCCCSCC)O)C(=O)NC(C)(C)C1=O Cc1cc(Cl)ccc1-n1cc(CC(O)C(=O)N(C)CC2CCC(=O)N2)nn1 C#CC1CCCN1C(C1CCCCN1C(c1conc1CC)=O)=O Cc1cccc(Br)c1-n1cc(CSC2CN(C(C3CCOC(CO)C3)=O)C2)nn1 C(=O)(CN=c1cc[nH]cc1)NC1(C)CCCN(C(=O)CCOCC2CCC2)C1 N1(C(C(C)N(C(=O)C(C)(C)C2CC2)CC)=O)CCN(C)C(COC)C1 Cc1ccc(F)nc1N1CCN(C(=O)C(=O)Nc2ccc(C(C)(F)F)cn2)CC1 C(=O)(C(C)CCC(C)(C)C)NC(C)CCNC(c1nnn(C)c1N)=O Cc1nc2ccc(C(N3CC(NC(C4CC4C)=O)CC(F)C3)=O)cc2[nH]1 c1(C(=O)NC(C)(C)CNC(=O)C=Cc2cnc[nH]2)c[nH]c2ccncc12 C(=O)(C(CNC(=O)CNc1cncn1C)CCC)NC(C#C)C(C)OC C1(CNC(CC(C)c2cnn(C)c2)=O)CN(c2ccnc(Cl)n2)CC(C)(C)O1 Cc1ccc(C(=O)C(=O)NC(C)CC(C)NC(=O)C(F)n2cccn2)cc1 c1(C(=O)NC(C)CCNC(c2ccc(Cl)nc2O)=O)ccc2oc(O)nc2n1 N1(C(Cc2c(C)nn(C)c2)=O)CCC2(CC1)CC2NC(c1nc(=O)n(C)[nH]1)=O c1(C(N(CC(C)NC(C2CC2C2CC2)=O)C)=O)cc2ccc(F)cc2o1 C1(O)(CNC(C(C)(Cl)Cl)=O)CCCN(C(=O)C(O)c2ccco2)C1 C1(CC(=O)NCCCOCCNC(c2c(CC)nc[nH]2)=O)CC2C=CC1CC2 C(c1ccc(Cl)cc1)=CCN1CC(O)(CC(=O)N(CCCCCCN(C)C)C)C1 c1(C(=O)NC(C2CCCN(C(=O)C(C)n3ccnn3)C2)C)cn(C)c(=O)nc1O N1(C(C(C=C)O)=O)CCCC(CCC)(NC(=O)Cc2ccc(CCCC)cc2)C1 C(CC1=CCN(C(C2CC3(CCC3)CO2)=O)CC1)NC(CC(C)C(F)F)=O c1(OC)cc(C(=O)NCC2(OC)CCN(C(=O)C(F)(F)C(C)O)C2)cnc1O c12ccc(F)c(F)c1C(=O)N1CCC1C(=O)N2.N1(CC)CCN(CCCO)CC1 c1(C(=O)OC)cc(C)c(S(=O)(=O)NC2(CS(=O)(=O)N(C)C)CCOCC2)cn1 CC(C)C(C(=O)N(C)CCOCCNC(=O)Cc1nc(=N)[nH][nH]1)C1CCC1 C1(C(N2CC3(CC(NC(C4OCCC(=O)C4)=O)C3)C2)=O)CCc2nccn2C1 N1(C(=O)COCCC2OCCO2)CC2CCN(C(c3cccc(F)c3)=O)C2C1 C1(COC)(NC(c2cccc(C)n2)=O)CCCN(C(C2COC3(CCC3)C2)=O)C1 Cc1ccc(C(=O)NCC2CC3(CC3)CN2C(=O)C(C)S)cc1C CCC(O)C(C)(C)C(=O)N1CCN(CC2(NC(=O)C(C)c3ccco3)CC2)CC1 c1(CNC(C(N2CCC(C=C)C2)CC2CCOC2)=O)ccc2c(c1)OCO2 N1(C(=O)C=Cc2cnccn2)CC2(C(N3CC(O)(C4CC4)C3)=O)CC1CCO2 C(c1ccccc1C#N)=CC(N1C2CC(CNC(C3CCC(C)O3)=O)(OC2)C1)=O c1(OC)cc(OC)c(CC(C)N(CC(c2ncc[nH]2)O)Cc2sccc2C)c(C)c1 c1(NCCC(=O)NCC2CC(NC(C(CC)N(CC)CC)=O)C2)cccc(C)c1 c1(C(N2CCC(N(C(=O)C(c3cccnc3)C)CC)C2)=O)nccnc1N c1(C(=O)NC(CN(C(=O)CCC2CCOCC2)CC)C)coc2c1COC2 c1(C(N2C(CC)CN(C(=O)C(C)CC#N)CC2)=O)ccc2cnc(C)n2c1 S(=O)(=O)(c1cnc(NCCC(C)(C)C#N)cc1C)NC(CNC)C1=CCCCC1 c1(CC(=O)NCCC(CCNC(CC(C)C(F)F)=O)C)ccc2c(c1)CCCO2 N1(C(C(c2ccccc2Cl)OC)=O)CC2CC(C1)N(C(c1cc(C)n(C)n1)=O)C2 C1(CNC(C2N(C)C(=O)CC2)=O)CC2(C1)CN(C(c1cc(Cl)sc1Cl)=O)C2 C1(C(=O)NC(C)(CNC(c2ccc(CO)s2)=O)CO)COc2ccc(F)cc2C1 C1(C(=O)NCC#CCNC(=O)Cc2ccc(Cl)s2)CC2CCCCN2C1 N1(C(CC(=C)C)=O)Cc2ccnn2CC(NC(c2nc(C(C)(F)F)cs2)=O)C1 C1(NC(C=CC2N(C(c3cccc(CC)n3)=O)CCC2)=O)CCCCCC1CO S(=O)(=O)(c1cnc2ccsc2c1)N1Cc2c(nn(C)c2C(N)=O)CC1 C1(NC(C(C)OCC#C)=O)C=CCN(C(C2(c3ccc(F)cn3)CCC2)=O)C1 c1(C(N2CC(N(CC(C)(C)C(=O)Nc3ccccc3)C)C2)=O)cnn(C)c1C#N c1(N2CCCC(CCC)CC2)nc(=N)[nH]c(=NC2CCC(C)(C)C2)[nH]1 CCCC(C#N)C(=O)N1CC(CNC(c2csc(C)c2OC)=O)(OC)C1 C1(CCNC(C2(C(=O)NC)CC2)=O)CCN(C(c2cncc(CO)c2)=O)C(C)C1 N1(C(C2(CC#C)CCOC2)=O)CCCCC1CCNC(c1cncnc1)=O CCC(C)CC(C)(c1nnnn1C1CCCCC1)NC(c1ccc(Br)nc1)(C)C C(=O)(C(F)C(C)(C)O)N1CC(C(=O)NCC(c2ccnn2C)C)OCC1 N1(C(CSCCOC)=O)CCCC(CCNC(=O)CC2CCC(OC)CC2)CC1 N1(C(CC=CCC)=O)CCN(C(C2CC(F)(CCO)C2)=O)CC1CO Cc1ccc2cc(C(N3CCNCC3c3ccncc3)=O)nn2c1 Cc1cnc(C(=O)NCC(CNC(c2cc(=O)cc[nH]2)=O)CO)c(F)c1 CCCCC(C(=O)N1CCN(C(c2ccc(C(=O)OC)nc2)=O)C(C)C1)N(C)C N1(C(C(C(CC)C)NC(C)=O)=O)CCCC2(NC(=O)C(N)=O)CC2C1 C(=O)(C(C)(C)CC(C)(C)C)NCC(=O)N(CCC(C)C)C1CCC1 c1(C(N2CCC3(C(NC(COC)=O)C3)CC2)=O)oc2c(C)ccc(C)c2c1C c1(CC(=O)NC2CCCCC2NC(C2CC(C3CC3)C2)=O)cccc(Br)c1 Cc1c(CC(=O)NCC2(F)CC(CNC(=O)CC3(C)CC3(F)F)C2)ncn1C Cc1cc2c(cc1C)OC(C(=O)NCC1CCCN1C(C1(O)CCOCC1)=O)C2 CC1(C)C(NC(c2ccoc2CN2CCCC2)=O)C2CCCOC12 CC(C)CCC(C)NC(=O)C(C1(C)CC1)NC(=O)CCCc1ncco1 C1(C(N2CCCC(O)(CNC(=O)Cc3ccno3)C2)=O)CCC(=C(F)F)CC1 c1(C(=O)NCC(C)(CO)NC(C2N(CCC)CCC2)=O)c(C)cnnc1O N1(C(c2n(C)nc(C)c2Cl)=O)CCCC(C2CCN(C(c3ncoc3C)=O)C2)C1 c12ccccc1C(=O)N2.N1(CCC)CCCCC1C(=O)O C12(C(=O)NCCCC(C)O)CC(CN(C(C3(C)COC3)=O)C1)C2 c1(N2CCC(C(=O)O)C(O)C2)ncnc2c1nnn2CC.C1CC(C)CN1CC S(=O)(=O)(c1ccc(NCCCCCF)c(F)c1)N(C)CC1COC(C)(C)O1 c1(OC)c(C(=O)N(CCCN(C)C(C2CC(F)C2)=O)C)cccc1Br N1(CCNC(c2cn(CCNC(c3cc(CC)on3)=O)nn2)=O)CCCCCC1 CC(C(=O)N(C(C)CN(C(=O)Cn1nnnc1C1CC1)C)C)S(C)(=O)=O c1(C(=O)NCCNC(CSC(C(N2CC(OCC)C2)=O)C)=O)ccc(F)cc1 c1(C(N2CCC(NC(C(CC)N(C)C)=O)CC2)=O)ccc(Cl)c2c1OCCO2 c1(CCC)cc(C(=O)NC2CCCC2C(=O)NCC2CN(CC)CCO2)n(C)n1 C1(NC(C(c2ccccn2)OCC)=O)CCN(CC)C1=O C(=O)(C1SCCc2sccc21)N1CCN(C(=O)CC2CC3(CC3)C2)CC(C)(F)C1 N1(C(Cc2nc(C)sc2Cl)=O)CCc2sc(CNC(=O)C=CCO)nc2C1 C1(NC(c2cncnc2)=O)CN(C(=O)Cn2cccn2)CCC1CO C(=O)(C(CCS(C)=O)N(C)C)NCC1(O)CC(CNC(CSCCOC)=O)C1 c1(NC(=O)C(F)n2cccn2)nc2ccccc2o1.C12(CC13CCC3)C(=O)NC2 N1(C(C=CCCC)=O)CC2(CCC2)CC1CNC(c1c(C)nn(CC)c1C)=O Cc1c(C(=O)NC(CNC(=O)COc2c(F)cccc2F)C(C)C)c(Cl)nn1C CC(C)(C)CC(O)C(=O)N1CCC(CO)C(CNC(=O)CN2CC3CC3C2)C1 c1(C(N2CCOCC(C)(CNC(=O)CC3=CCCC3)C2)=O)cc(S(C)(=O)=O)co1 n1(CC)cc(Cl)c(C(=O)NCCNC(C2CN(C)C2)=O)n1 C1(CNC(c2n(C)cc(Cl)c2)=O)CN(C(=O)C2=C(Cl)CC2)CCC1(F)F C(CN=c1[nH]c(=NC2CC(C)CC(C)(C)C2)[nH]c2c1CCCCCC2)C1C(C)C1 C(=O)(C(C)S(=O)(=O)C(C)C)NC(CCCNC(C(C)(C)OC(C)=O)=O)(C)C CC(C)(C)C(C(=O)N1CC(N(C(C2CSC2)=O)C2CC2)C(C(=O)O)C1)c1cc[nH]n1 N1(C(C(c2ccc(C)cc2)=O)=O)CCC(NC(=O)CO)C12CC2 C(=O)(CC(C1CC1)NC(C1(C(C)C)CCC1)=O)NC1(CC=C)CCC1 C1(NC(CN2CCC(OC)C2)=O)CCN(C(=O)Cn2nccc2C)CC1F c1(NCC2N(C(C(CC)CC(C)C)=O)CCCC2)ncc([N+](=O)[O-])cc1Br N1(C(C2CC(=C)C2)=O)CCC2CCN(C(=O)CS(=O)(=O)NCC)C2C1 N1(C(c2c(C)nc(O)cc2)=O)CC(C)CN(C(=O)C(C2CCCCC2)=O)CC1C C(=O)(CC(CC)N(C(=O)CCN1CCOC1=O)C)N(CC(CCC)O)C c1(OC)ccc(C)c(NC(=O)CC2CN(C(=O)OC(C)(C)C)CC(C)O2)c1 N1(C(c2ccn(C)c2)=O)CC2CCOC2(CNC(c2ccncn2)=O)C1 N1(C(c2c(-c3cn(C)nc3)ocn2)=O)CCCC1C1CCCN1C(=O)COCCF C1(F)(C(=O)NCC2(O)CC(C(=O)NCC3(OCC)CCC3)C2)CCCCCC1 CCCC(C(=O)OC)C(=O)NCC(CC)NC(=O)C(c1cccc(Cl)c1F)(C)C Cc1cnc(C(=O)NCCOCCn2cc(-c3cccs3)nn2)cn1 S(=O)(=O)(c1ccccc1C(=O)NC1(CNC(=O)C(C)NC(C)(C)C)CC1)NC N1(C(c2cc(C)no2)C(=O)NC)CCCc2c(OCC(=O)OC(C)C)cccc21 C1(CCNC(c2cccc(F)c2F)=O)CN(C(=O)Cc2ccoc2)CCCO1 C(=O)(CCS(N)(=O)=O)NC1(CNC(Cc2cc(C)[nH]n2)=O)CCCCC1 C=CCC(CC=C)C(=O)N1CCCN(C(c2cc(C(N)=O)co2)=O)C(C)C1 C(CC(C)C)(C(=O)N1CCOCC(NC(=O)CCCc2cc[nH]n2)C1)OC C(=O)(C1=CCCN(C(=O)CC(CC)C(F)F)C1)N1C(C)(CCC)CC1 C(=O)(CC(O)CC(C)(C)C)NC12C(CN(C(c3cccc(C)c3Br)=O)C1)C2 C1(CNC(CCN(C(C)C)C(c2cccc(=O)o2)=O)=O)CC(O)C12CCC2 C1(CC(=O)NCCP(C)(C)=O)C2CCCC2N1C(=O)CC1C=CCC1 Fc1ccc(C2CNCCN2Cc2ccn(Cc3ccccc3)n2)cc1 c1(C(=O)NCC2CCN(C(=O)CC3CN(C4CC4)C3)C23CC3)cnc2ccnn2c1 CC1(C(=O)NCC(C)(CO)NC(=O)COc2ccc(C(N)=O)cc2)CC=CCC1 N1(C(Cc2cc(C)[nH]n2)=O)CCC2CCCC12CNC(c1nc[nH]c2ncnc1-2)=O N1(C(c2c(C)oc(C(C)C)n2)=O)CCN(C(c2ccc(N)cn2)=O)C(CCO)C1 N1(C(C)=O)CCN(CC2C(C(=O)NC(c3ccccc3I)=O)C2)CC1 C(C(C)C(C)C(=O)N1CCCC1CNC(=O)C(F)(F)CCn1ccnn1)OC CCC(CC)C(C(=O)NC1CC(C)CN(C(c2ccccc2O)=O)C1)OC C(CCC(C)(C)NC(C1CCCCN1S(C)(=O)=O)=O)NC(Cc1nc(C)sc1)=O C#CC1(NC(C2(C(C)NC(C3CCN(OC)CC3)=O)CC2)=O)CCCOC1 Cc1cc(CCC(=O)NC23COC(CNC(C4CCC(C)C4)=O)(C2)C3)c(C)s1 C1(c2n(C(c3ccccc3Br)C)nnn2)(NC2CCC(O)C2)CCCSCC1 C1(C(=O)NC(CCC)(C)CC)CN(C(C2CC2C(F)F)=O)C2(CCC2)C1 c1(COCc2cccc(OCC)c2)cc(OC(F)F)ccn1.C1C(O)CC1N N1(C(C(CNC(C2CC3(CSC3)C2)=O)O)=O)CCC2(CCC2)CC1 c1(CS(=O)(=O)N(C)CC2(C(F)(F)F)CC2)cccc(Cl)c1 C1(NC(Cc2scc(C(C)(C)C)n2)=O)CCCCC1NC(=O)Cc1cscn1 c1(C2(NC(c3ccccc3OC)CCC)CC2)ccccc1I Cc1ccnc(C)c1NCc1nccnc1CC(N1CCCC(COC(C)C)C1)=O Cc1occ(C(F)(F)F)c1COC(C1CCCN1C)=O N1(CCCC)CCC(C(=O)N(CCN(c2sccc2Cl)C)C(C)C)CC1 C1(Cc2cccc(NC(C=NOC)=O)c2)C2CC3CN(C(C4CC4F)=O)C1C3C2 C(=O)(C1CCc2cccnc21)N(CCCNC(c1n[nH]c(C)c1Br)=O)C1CC1 CCC(C)(CNC(=O)CCc1ncccn1)NC(=O)COC1CCC1 n1(CC)cnc(=NC(=O)OC)[nH]1.N12CCOC(C1)CNC2=O C(=O)(CCCC(C)=O)N1CC(CCC=C)(C(=O)NC(C)CC(N)=O)C1 c1(CC)c(-c2nc(CN(C)Cc3ccc(C)cc3)nn2CC(N)=O)c(C)nn1C C(=O)(C1=CCCC(C)(C)C1)NC(C(C)C)(C)CNC(=O)C#CC1(C)COC1 c1(CC2N(C(C3CC(n4cc(C(C)C)nn4)C3)=O)CCCC2)ccc(C#N)cc1 C1(C)(C(=O)NCC(CC)(CC)NC(=O)Cc2ccccc2F)CC(C2CC2)=NO1 c1(N(CC(C)CNC(C2CCn3cncc3C2)=O)C)nn(C)cc1[N+](=O)[O-] CC(C)(C)C(=O)NCC(O)C(=O)N(CC1CC1)C.C1(C(=O)OC)CCC1 O=C(C1=CS(=O)CCC1)NCC1CCCC1NC(c1ccnnc1Cl)=O C1(O)(C(N2CCCN(C(CC(C)C3CC3)=O)CC2)=O)CCCC(C)(C)C1 c1(COC)nc(C)c(C(N2CCC(COC)(NC(C3CCCOC3C)=O)C2)=O)s1 c1(C(N2CC(CC)N(C(=O)CSc3nc[nH]n3)CC2)=O)ccc(Cl)c(OC)c1Cl CC1CCC(Cl)=C(C(=O)NC2(CNC(c3nc(Cl)c(=O)[nH]c3N)=O)CC2)C1 CC1CCN(C(c2ncccc2C(F)(F)F)=O)CC1NC(=O)CCSCC(N)=O N1(C(C(C2(O)CCC2)NC(c2c(C)cc(O)nc2)=O)=O)CCCC2(CCCO2)C1 c1(CN(C2CCCN(C(c3c(CC)cccc3)=O)C2)C)ccncc1[N+](=O)[O-] C1(NC(CCCNC(c2scc(OC)c2)=O)=O)CC(C)CC(C)(C)C1 C1(OC)CC(C(=O)NC2CCC(F)(F)C2)N(C(=O)CCC2CC2)C1 C=CCCCCCCC(=O)N1CC(NC(=O)Cc2c(C)nc3n2CCCC3)C1 C1(C(N(C)CC2C(C)C2)=O)(N(C(=O)CC2CC(=O)C2)C2CC2)CCC1 CC(CC(F)F)C(=O)N1CCC(O)CC1C(=O)Nc1ccccc1 c1(OCC(N2CCC(N(C)C(C3CC34CCC4)=O)C2)=O)ccc(F)c(F)c1 Cc1ncc(N)cc1C(N1CC=CC1CNC(=O)CCc1ccon1)=O N1(C(c2cc(C(C)C)no2)=O)CCN(C(=O)C2CC2)C(C(C)C)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)N(CCCCO)C2CCCC2)C2(CC2)C1 C1(OC)(OC)CC(CNC(=O)C(N2CC(C)(CCCC(=O)O)C2)=O)C1 N1(C(C2CCN(C(C(CC)N(C)C)=O)C2)=O)CCC2(COC(C)C2)C1 C(C(CO)(CO)NC(c1cncc(CSC)c1)=O)N(C(C=COCC)=O)C CN1N=C(C(=O)N2CCOC(C(=O)NCCc3cccc(Cl)c3)C2)CCC1=O CCC(C)C(CC(=O)N1CCCC1CNC(=O)C(O)CCC(C)C)NC(C)=O c1(C(C)C)n[nH]c(=NCC2CC(CNC(C34CC3COC4(C)C)=O)CO2)o1 C(=O)(C1Cc2ccc(F)cc21)N1CCC(N=[N+]=[N-])(C(=O)NCC(C(C)(C)C)OC)C1 N1(C(c2c(C)ccnn2)=O)CCC(NC(C2CC23CCCCC3)=O)C12CC2 c1(NC(COCC)=O)cccc(C(C2(C)CCNCC2)C)c1 C(CC(C)(C)C)(C(=O)NC(C1CCN(C(C2(C(F)F)CCC2)=O)C1)(C)C)OC c1(N(C)Cc2n(CC)cnn2)nc(=NCC2CCCCS2)[nH]c2ccccc12 c1(OC)ccc(OCC(=O)NC2(CF)CCN(C(c3cc(F)n(C)n3)=O)C2)cc1 C1(CC)CN(C(=O)CCCCN(C)C)CCN1C(C1CCCCCC1)=O C12(C(=O)NC(C(=O)OCC)C3CC3)CCC(C)(C1)OC2.C1(=O)CC2(CC2)CO1 CCC(O)C(C)(C)C(=O)NC1CCC1CNC(=O)CCc1cnco1 N12CC(C)(C1)C2=O.C1(CNC(CC)=O)CN(CC(F)F)C1 c1(OC)ccc2c(c1)CC(C(=O)NC1CC3(C1)CN(C(=O)CC1(OC)CC1)C3)O2 c1(C(=O)OC)sc2ccccc2c1C(=O)NCC1CC(NC(=O)C(O)C2CCC2)C1 c1(CC(N2C(CNC(C(C)(C)C)=O)CCC2)=O)c(F)c(F)cc(F)c1F O(N1C(=O)c2ccccc2C1=O)CC(=O)NCC1C=CCN1C(C1CC12CC2)=O C1(C#CC(=O)N2CCCC2CC(=O)NCC2(F)CCOC2)(CC)COC1 c1(Cn2cc(CN(C(c3n(CCC)ccc3)=O)CCO)nn2)cc(Br)c(Cl)s1 C(=O)(CCCCC(C)C)N(C(c1ccccc1)CC1CC(C)(C)NC1=O)CC c1(C(=O)NCC2(C(C)NC(c3c(C)cno3)=O)CC2)ccc(OC(F)F)cc1 C1(N(C(CN(CC(C)(C)C)C)=O)C)CCCC(NC(c2nnn(C)n2)=O)C1 C1(C(N2C(CC(C)C)CC2)=O)CC2(CCC2)CN1C(C1CC(C)(O)C1)=O CCCCCCN(C(=O)CC1SCCS1)CCNC(C1CC1CCC)=O C(CC(C)(C)C(=O)N1CC(C)(NC(=O)CNC(=O)OCc2ccccc2)C1)SC C(=O)(C(O)C(C)c1ccccc1F)N(CCOCCOCCOC)C CCC(CC(=O)NCCC1CCCN1C(=O)CCC1=NNC(=O)CC1)C(C)(C)C C(CC(O)C(=O)N1CCCC(CC(=O)N(CC(=O)N(C)C)C)C1)SC C1(NC(CC=C)=O)CC2CCC1N2C(C1CC(=O)N(c2ccc(Br)cc2)C1)=O c1(C(N2C(C)CC(NC(Cn3c(C)ccn3)=O)C2)=O)c[nH]c(C#N)c1C c1(C(N(C)CC2CCCC(NC(=O)Cc3cn[nH]c3)C2)=O)cc2cn[nH]c2cn1 C#CCCCCCCC(=O)N1CCC(N(CC#C)C(c2conc2CC)=O)C1 Cc1cncc(CCC(=O)NC2CC(NC(c3ccc(CO)cn3)=O)CC2O)c1 c1(OC)ccc2nc(N3C4CCC3CC(Br)C4)sc2n1 C1(NC(C=C(CNC(CCCNC(C)=O)=O)C)=O)CCCC(F)C1 N=c1[nH][nH]cc1C(=O)NCC1CCC1C(=O)NC1(CF)CCCC1 Cc1cc(OC2CCN(C(C3CCCCN3)=O)C2)ccc1N1CCSCC1 C1(CNC(CC2CC(C)N(C(C3CC=CC3)=O)C2)=O)CN(C)CCN1C c1(C(=O)NC2CCN(C(C(CCC)O)=O)C23CC3)cccc2cc(O)ncc12 c1(OC)ccc(F)cc1C(N1CCC2(CC2NC(=O)C(F)C(F)(F)F)C1)=O c1(C(=O)NCC2N(C(C(C)NC(C)=O)=O)CCC2)cc2nccc(Cl)c2s1 C1(NC(CCc2nc(C)sc2)=O)COC2(CCN(C(=O)CC(C)C3CC3)C2)C1 CCCC(C)C(C(=O)Nc1cc(OC)cc(F)c1)N(C1(C)CC1)C C1(C(=O)NC2C3CN(C(COC(C)C)=O)C2C3)CC2(CCC(F)(F)CC2)CO1 C1(CN(C(=O)C(Cn2cncn2)NC(C2CCC2CC(N)=O)=O)C)COCCO1 c1(C(N2CCCN(C(C=CC)=O)CC2C)=O)cc(F)cc2nc(S)[nH]c12 c1(C(=O)NC2CC(N(C(=O)CCCN3CCCC3)C)C2)occc1F N1(C(c2n(C)ncc2)=O)CC2CS(=O)(=O)CC2(NC(=O)CCC2(C)CC2)C1 C(=O)(C1CCCc2c[nH]nc21)N(C(C)CNC(C1(CO)CC1(F)F)=O)C c1(NC(C)=O)cccc(CC(=O)NCCC(C)N(C(=O)C(C(C)C)N(C)C)C)c1 N1(C(C2CC(SC)C2)=O)CC(NC(=O)C(c2ccc(F)c(Cl)c2)(C)C)CC(C)C1 C(N=c1[nH]c(C)nc(C)c1F)C1(F)CC(NC(C2(COC)CC=CCC2)=O)C1 C#Cc1cncc(C(N2CCN(C(=O)CCn3cc(C)cn3)CC2C(C)C)=O)c1 CON=CC(=O)N1CCC(NC(=O)CCN2CCOCC2)C1 C(C)(C(=O)N(CC(O)CN(C)C(C1CC(C(C)C)C1)=O)C)NC(CC)=O c1(C(=O)NCCN(CC(C)O)C(C2C(C=C)C2)=O)cc2n(n1)CCC2 C1(C(=O)NCCC(C)CCNC(=O)CC(C)C)(CC)CNC(=O)C1 n1(C(C)C(=O)N(C2CN(C(C3(N(C)C)CC3)=O)CC2O)C)cnc2ccccc12 c1(C(N2CCCCC2C2CCCNC2)=O)ccc(OC(F)(F)F)cc1Cl c1(C(=O)NC2(CNC(CC(C)CN(C)C)=O)CC(F)(F)C2)ccc(F)c(F)c1 c1(CC(N2C(CNC(=O)CCOC3CC3)CCCCC2)=O)nc2c([nH]1)CCCC2 N1(C(CS(=O)(=O)NC)=O)CC2CCCC2(C(=O)NOCC)C1 C(=O)(C(C)(C#N)CC)NCC1CC(NC(CC2ON=C(CC)C2)=O)C1 c1(OC)ccc(C(=O)NC2(CO)CN(C(=O)C(F)C3CCC3)C2)nc1 C1(CC#C)CN(C(=O)CN(C(=O)C(C)COC)C(C)C)CCO1 N1(C(c2c(CC)ocn2)=O)CCC2(CCC2)C(NC(c2cc(CO)n(C)n2)=O)C1 N1(C(c2c(C)coc2)=O)CC(C)(C)CC1C(N1CCCC(F)C1)=O C1(NC(C2(C)CC(C)C2)=O)CC2(CCN(C(c3ccc(Br)c(N)c3)=O)C2)C1 C1(C)(NC(c2cc(C(=O)OC(C)(C)C)on2)=O)CCOCC1CO N1(C(c2ccn(COC)n2)=O)CC2CCCC(CNC(=O)C=CCO)C2C1 N1(C(C(CC)OCC)=O)CC2(CCN(C(=O)CC3CCC4(CCC4)CO3)CC2)C1 C1(NC(C2CCSC2)=O)CCC12CCN(C(C1CC1c1ccccc1)=O)CC2 C(=O)(C(C)(C)C(=O)NC1CCCN(C(=O)C=C2CCC(C)C2)C1)NC c1(CNC(c2c(C)nns2)=O)ccc2c(c1)CN(C(=O)C(C)O)C2 CC(C)(C#N)C(=O)NCC1CC(F)CN1C(c1ccc(C(F)F)cc1)=O c1(NC(c2nccs2)CC)cnc(-c2ccncc2)cn1 CC1CN(C(C2CC2C2CCCC2)=O)CCN1C(=O)Cc1ccc(Cl)s1 Cc1ccc(Cl)c(C(=O)NC2CC2NC(c2ccc(C(=O)N(C)C)nc2)=O)c1 N1(C(c2ccc(C)c(N)c2)=O)CCOCC(F)(CNC(=O)CN2CC=CC2)C1 CCC(CC)C(F)C(=O)NCC(C1CCC1)NC(C1(F)C(C)(C)C1(C)C)=O c1(C(C(=O)NC(C)CCCNC(C2(C3CC3)CCCO2)=O)(C)C)ccccc1F c1(CC(=O)NCC(=O)NCCCCOCCNC(C2C(C)C2)=O)cnc(O)[nH]1 N1(C(c2c(C)nc(C)o2)=O)CCC(NC(=O)C(C)(C)C2CCOC2)CC1C C12(C(=O)NC(CC=C)C(=O)Nc3cnc(F)nc3)CCCC1CCC2 C1(N(C(=O)CCC2CCN(C)CC2)C)CN(C(=O)Cc2cccn2C)CCC1O Cc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CCCCCc1cccs1 C=CCC(C(=O)N1CCC1CNC(C1(S(C)(=O)=O)CCOCC1)=O)C(C)(C)C c1(C(N2C(CNC(CN(CCC)C)=O)CC2)=O)csc(-c2cccs2)n1 c1(OC)cc(Cl)c(C)cc1C(=O)NCC1CC1CNC(c1occ2c1CCC2)=O c1(C(=O)NC2C(OC)CN(C(=O)CCC(C)SC)C2)c(C)nn(CCO)c1C c1(C(=O)NCC(CNC(c2cccc(CCC)c2)=O)O)cccc2nc(Cl)cn12 Cc1cc(C(N2CCC(C)C2CNC(c2sccc2C(C)C)=O)=O)cc(N)c1Cl c1(C(=O)OC)ccc2c(c1)C(C(=O)N(CCCNC(c1cnc[nH]1)=O)C)CO2 C1(C(=O)NCC2C(C)(C)C2(F)F)CC(C)(C)CCN1C(c1cn(C2CC2)cn1)=O c1(C(C(N2CCC(NC(c3nnn(C(C)(C)C)n3)=O)C2)=O)(F)F)ccc(F)cc1F C1(NC(C(CCC)N(C)C)=O)CC2C1CCN2C(=O)CC(=O)N(C)C C#CCC(C)(C)C(=O)NC(C)CNC(C1C=CCCC1)=O N1(C(C2OCC(C)(C)C2)=O)CCC2(CCCCC2NC(=O)CCc2cnn[nH]2)C1 Cc1cc(N(C)C)ccc1C(N1CC(CNC(=O)C(CO)c2ccccc2)C1)=O C1(NC(C=C(C)C)=O)Cc2ccccc2C1NC(c1cnc2c(n1)CCCC2)=O C(C(F)(F)CNC(=O)Cc1cc(C(F)(F)F)n(C)n1)(C1CC1)OC c1(C(C(=O)NCCCN(CCCCCC)C)O)cc(F)c(F)c(F)c1 C(=O)(C1=CCCOC1)N1C(CCNC(CCOCC(C)C)=O)CCC1 N1(C(C=C(C)Cl)=O)CCC2(CCOC2)C(CNC(=O)Cc2csc(SC)n2)C1 CC(C)C(C(=O)N(C1CCN(C(C2CC2Br)=O)CC1)C)c1ccn(C)n1 C1(C(=O)NCC(CNC(=O)Cc2cnccc2C(F)(F)F)O)CCCC1C1CC1 N1(C(C2CN(C(CC3CC(=C)C3)=O)CC2(C)C)=O)CCCC2(CCCC2)C1 CC1(C)CCN(C(c2ccon2)=O)C(C(=O)NC2CCN3CCC2C3)C1 c1(SC)ccc(Cl)c(C(N2CC3CCC3(CNC(=O)CC3CCC(=O)N3)C2)=O)c1 C1(CSC)CN(C(=O)CCC(=O)N(C)C)CCC1NC(=O)COC1CCOCC1 C1(C(=O)NC2C(O)CC2O)CN(C(=O)CC2CSC2)CC12CC2 N1(C(c2nc(C)cn2C)C(=O)NC)CCN(C(C)C)CC1C c1(C(N(CC(C)NC(=O)C(O)C(F)F)CC)=O)cc(S(C)(=O)=O)cnc1O C1(NC(CCc2c(C)noc2C)=O)CN(C(=O)C2=CSCS2)CC2(CCC2)C1 C12(NC(CCC3CC(OC)C3)=O)COC(CNC(C3CCC(C)C3)=O)(C1)C2 c1(OC)ccc(OC(=O)C(c2cccc(F)c2)OC)c(C)n1 C1(CNC(C2C(CC)C2)=O)CCN1C(=O)C(C)n1cncn1 c1(CN2C(C(=O)N=c3[nH][nH]cc3Br)CC3CC32)cccc2ccncc12 C1(=O)C#CC(OCC)OCC(=O)N(CCCC)C2CCN1C2.OC C1(CN(C)C(C2(C)CCC2)=O)CCCCN1C(C1CC1c1cnc[nH]1)=O Cc1cc2c(cc(C(=O)NCC(C)(C)CNC(c3ccoc3)=O)n2CC2CC2)s1 C1(CC=C)(NC(C2CC(O)C2)=O)CCN(c2nc(C(F)(F)F)ns2)CC1 C(C)(CO)(C(=O)NCCC(O)CNC(C1(CCO)CC1)=O)OC C(C)(N=c1[nH]cc(C#N)cc1C)C1(O)CN(C(c2cccc(COC)c2)=O)C1 c1(CNC(=NCCCCC)NCCNC(=O)NCCO)nccc2ncccc12 c1(C(=O)NCC(CC)NC(=O)Cc2cnn(CC)c2)ccc([N+](=O)[O-])c(C)c1 c1(CC(N)CC(=O)NCCOCc2ccccc2)cc(F)c(F)c(F)c1 C1(CCC)CN(C(=O)C(c2ccccc2Cl)OC)CCN1C(=O)CC(C)(C)OC c1(C(=O)NCC(C)N(C(c2c(C)cc[nH]2)=O)C)c(C)nc2ccccn12 C1(CNC(c2coc3c2COC3)=O)CC2COCC2N1C(=O)Cn1cnnc1 c1(CC)c(C(N2CC=CC(NC(=O)CNC(=O)CC(F)(F)F)C2)=O)nnn1CC C(=O)(CC(C(F)F)c1ccc(F)cc1Cl)N1C2C(NC(C(C(C)C)C)=O)C(C2)C1 C1(C(=O)NCC2CCC(N(C)C(C3(C)CCCCO3)=O)CC2)CCC2(CCC2)C1 C1(NC(C=C(C)Cl)=O)CCC2CN(C(=O)CSCC(c3ccccc3)=O)CC2C1 C1(CC(C)C)Oc2cc(Br)ccc2C1NC1CCC2(CCCC2)C1 CC1CCN(C(=O)C(CNC(=O)CC2COCCO2)CC2CC2)C(C)C1 N1(C(C(CCSC)O)=O)CC(C)CN(C(C2CC2(F)F)=O)C(C)C1 N1(C(CCc2onc(C)n2)=O)CCCCC(C(=O)NCCCCC(C)(F)F)C1 Cc1nn(CC(=O)N(CC(C)(C)CNC(C2SCCC2C)=O)C)c(C)c1C Cc1noc(C)c1C=CC(N1CCCCC1CCN(C(=O)CC1C=CCC1)C)=O Cn1cccc(C(=O)NCC(CC2CC2)C(=O)NCC2CCCC2(C)C)c1=O C12(C(=O)NC3C(SC)COC3)CCN(C(=O)C=CC3CC3)CCC1C2 n1(CC)nc(C(=O)NC(C)C(CO)NC(c2cccnn2)=O)c(Br)n1 c1(N(C(c2cccc(Br)n2)C(=O)NC(C)C)CCOCCCC)ccc(F)cc1 Cc1cc(C)c(CC(N2CCC(N(C(=O)C(F)=CCCF)C3CCC3)CC2)=O)s1 CC(C)(CC(F)F)C(=O)NCCC(O)C(N1CCc2sccc2C1)=O c1(C(=O)NCC(CO)NC(CCC2CCCN(C)C2)=O)c(O)ccc(Cl)c1F CC1CC(NC(=O)C=CC2CCCC2)CCN1C(C1CC2CCC1C2)=O N1(C(CN(C)CC)=O)CCC2(C1)CN(C(=O)CCC(C)c1ccccc1)CCO2 Cc1cncc(C)c1C(N1CCOC(c2cn(-c3ncc(Cl)nc3Cl)nn2)C1)=O N1(C(CCC(C)OC)=O)CC(NC(=O)CCCc2cccnc2)C2CCCCC12 CC(=Cn1ccnn1)C(=O)NCC(C)(C)CN(C)C(c1ccc(C)s1)=O N1(C(c2ccc(OC)s2)=O)CCCCC1C(N1CCOC(C2CC2)C1)=O Cc1nn(C)c(C)c1C(=O)NC(C)(C)C(=O)N(C)CC1COCCO1 C1(NC(CC2C(NC(C(C)c3cccs3)=O)CC2O)=O)CCCCC1N=[N+]=[N-] c1(C(=O)OCC)ncc(F)cc1NC(C1C2CC1N(C(=O)CC1CCCC1)C2)=O c1(CNC(C2COC2)=O)ccc(CNC(C2CCCC(F)(F)CC2)=O)c(F)c1 C1(C(=O)NCC2(OC)CCN(C(c3c(CC)nco3)=O)C2)C2CCCCCCC12 CC(C)CC(O)C(=O)N1CCCC(CNC(=O)CC2OCCC2(C)C)CC1 C1(CC(C)NC(C2CC3(CC3)CO2)=O)CCN(C(C2CC3C=CC2O3)=O)CC1 Cc1cn2c(CC(=O)NCC(CO)NC(c3c[nH]cc(Cl)c3=O)=O)csc2n1 c1(OC)c(-c2nc(CC(N)=O)no2)ccc(C)c1F N1(C(CN(C)C)=O)CCC(NC(C2CC2[N+](=O)[O-])=O)C(F)(F)CC1 c1(C(=O)NC2CN(C(CCCCSC)=O)CC(O)C2)c(C)cc(O)nc1C C(=O)(CC(O)CNC(C1CCCCC1CC(F)(F)F)=O)OCC S(=O)(=O)(c1ccc(NCCN=S(C)(C)=O)cc1Br)NC1CC(CC)(CC)C1 C1(C(N(C(C)C(C)(C)C)C)=O)CC2CC1CC2NC(=O)COCC(C)(C)C C(=O)(C1=CC2CCCCC12)N1C(CN(C)C(C2CN(CC(F)(F)F)C2)=O)CCC1 C1(NC(CN(C(=O)Cc2cn[nH]c2)CCOC)=O)CC(=O)NC1=O C1(C(=O)NCC2(CC(=O)NC(C3CCOCC3)C#C)CC2)CC2CC1CC2=O N1(C(C(c2[nH]c(=N)sc2)=O)=O)CC2CC(NC(=O)CCCc3cncs3)CC2C1 c1(C(=O)NCCN(CCC)C(C2C3(CC3)C23CC3)=O)ccc(C2CCCO2)nn1 c1(CC(=O)NC2(CN(C(=O)CCS(C)(=O)=O)C)CC2)cccs1 C1(NC(CCN(C(C(CC)(C)OC)=O)C)=O)CC2COCC2C1 N1(C(CC=C(C)C)=O)CC=CC1CNC(C1CCC(Cc2ccccc2)O1)=O CC1(C)C(C(N2CC=CC2CNC(=O)CCCc2nccs2)=O)C1C(F)F C1(NC(c2scc(OC)c2)=O)CC(NC(c2cccc(=O)n2C)=O)C12CCC2 c1(C(=O)NC2C3CN(C(CS(CC)=O)=O)CC32)cnc(OC)nc1C(F)(F)F c1(CNCC)cccc(CNc2nc(C)ns2)c1 c1(CNC(C=CCCC)=O)cccc(OC)c1F.C1C(OC)C(=O)N1C c1(C(N2CCC(CNC(c3c(C)ccn3C)=O)C2)=O)nc(C2CC2)ncc1Cl N1(C(C2(OC)CC(C)C2)=O)CCCC(NC(c2nnsc2SC)=O)C1 N1(C(c2c(C)cc(F)s2)=O)CCC(NC(c2cc(C(C)(C)C)ccn2)=O)C12CC2 CC1CN(C(c2cnccn2)=O)CC1NC(=O)CCOCCOCCCO c1(C(=O)NC23CC(CNC(C(C4CCOCC4)OC)=O)(C2)C3)cc(SC)c(C)o1 Cc1cnncc1C(=O)NCC(=O)NCC1(C#N)CC1 c1(C(N2CCC(N(C(C3CCCC(O)C3)=O)CC)C2)=O)cc[nH]c2nccc1-2 CC1OCCC1CC(=O)NC(C1CCCC1)CNC(C1CCCC1)=O c1(C(N2C(CCCNC(c3n(C)nnc3)=O)CCC2)=O)cc2ccc(F)cc2[nH]1 C1(C(N2CC(CC)N(C(C34CC(C)(C3)C4)=O)CC2)=O)CN=C2N=CNN2C1 C(=O)(CCCCCNC(=O)NC(C)C)N(c1c(C)n[nH]c1C)C c1(C(=O)NC2(CN(C(C(F)OC)=O)C)CC2)ccnnc1 C1(NC(=O)CC2CS(=O)(=O)C2)CN(C(=O)CC2(O)CCCCC2)C2(CCOC2)C1 c1(NC(C2CCCN(C(C34CCC(OC)C3C4)=O)C2)=O)n[nH]c2ccc(F)cc12 C1(CNC(CC2N(C(CC3(N(C)C)CCC3)=O)CC2)=O)CCCC2(CC2)C1 CCC(C)(O)C(=O)NC1C2CN(C(c3ccc(C4CCC4)nc3)=O)CC12 c1(C(=O)OC)ccc(C(CNC(c2ccc[nH]2)=O)NC(=O)C(C)CN(C)C)cc1 C12(C(N(C)CC34CC(C(C(C(C(C)C)O)=O)=O)(C3)C4)=O)C(=O)C3CCC1C2C3 C(=O)(C(C)CC(C)C(C)=O)N1C(CC(=O)Nc2cn(CCC)nc2)CCCC1 C1(CC)CCC(=O)N1C(=O)CCCc1nnc(-c2ccc(CN)cc2)o1 C1(C(=O)NCCCN(C(CN(CCC#C)C)=O)C)(CF)CCOCC1 C1(CSC)CCN(C(c2ccoc2C)C(=O)NCCCSC)C2(CC2)C1 CC1(C#CC(=O)N2CCC(CCC(=O)NC(CO)CCC3CC3)CC2)CCCO1 S(=O)(=O)(c1c[nH]c(=NCC2CCC2)cc1C)N1CC2C(OC)(CC2C(N)=O)C1 O=C1CC2(COC2)CN2N1CC1CCOC1CC2CCN(CC)S(=O)(=O)C1CC1 C(=O)(CC(O)CC(C)(C)C)NC(CNC(Cc1c(SCC)cccc1)=O)(C)CC c1(NC(N2C(CC#N)COCC2)=O)ccc2c(Cl)ccnc2n1 Cc1nc2cncc(C(N3CCC(C)C(CNC(=O)CCS(C)=O)C3)=O)c2[nH]1 c1(OC)cc(C(=O)Nc2c(Cl)ccnc2Br)cnc1-c1cnc(F)c(F)c1 CCCCCC(=O)N1CCN(CC2CCCN(C(C3CCCCO3)=O)C2)CC1 N1(C(c2c(OC)c(C)cs2)=O)CCC2(CCCN2C(=O)Cn2cc(Cl)cn2)C1 N1(C(c2cnnc(C3CC3)c2)=O)C2CCC1CC(NC(C1(F)CCOCC1)=O)C2 c1(C(=O)NC2CN(C(c3cscc3F)=O)CC2O)cccc2nc(O)ccc12 N1(CC(N2CCN(C(C3C(=O)NCCC3)=O)CC2CF)=O)CCCCCCC1=O c1(OC)ccc(S(N)(=O)=O)cc1NC(C1CNC(=O)C1(C)C)=O C(=O)(C(O)C(C)(C)C)NCCCN(C)C(c1c[nH]cc1-c1cccc(Br)c1)=O c1(C(=O)NC2CC(CNC(=O)CCCF)CC2O)cc(Cl)cc(Cl)c1 CC1CN(C(c2cc(O)nc(O)n2)=O)CC(C)N(C(=O)Cc2cc[nH]c(=N)c2)C1 C1(C(N(C)Cc2cn(CC)nn2)=O)CC(OC)CN1C(c1ccncc1NC)=O c1(N2CCN(CC)CC2)nc(=NC2CCC2N(C)C)[nH]c2c1CSC2 N1(C(C(CC(C)(C)C)OC)=O)CCCC12CCCN(C(=O)C=C(C)C(C)(C)C)C2 C1(NC(c2c(OCC)scc2)=O)CN(C(C2CN3CCC2CC3)=O)C(C)(C)C1 c1(CC)cc(Cl)ccc1NC(=O)C(O)C1CN(C(C2(C)CC2)=O)C1.C(C)(=O)OC C1(C(=O)NC(C2(CNC(c3ccc(C=C)cc3)=O)CC2)C)CCCC2(CCC2)O1 c1(-c2nc(C)c(NC(=O)C(O)CC(C)C)s2)cccc2c[nH]nc12 N1(C(C(C)=C(C)C)=O)CCN(C(=O)CCc2ccoc2)CC1CO C1(C(=O)NCC(CC(C)C)NC(=O)C(c2ccncc2)C)CCCCN1N=O c1(CC)nn(C)cc1C(N1CCC(N(CCO)C(c2cc(C(C)=O)cs2)=O)C1)=O C(=O)(C(C1=CCCCC1)N1CCCC(Nc2ccccc2)C1)NC(=O)C1CC1 C12(NC(C(C)c3cccs3)=O)CCCC1N(C(=O)CC1CCC(C(F)(F)F)O1)CC2 CC1CCC(C(N2CCC(CN=[N+]=[N-])C2)=O)N(C(c2ncccn2)=O)C1 c1(C(N2CCCCC(NC(C3N(CC)CCCC3)=O)C2)=O)cc(F)c(Cl)cc1Cl N1(C(C(CC)OCC)=O)C2CCC1C(C)C(NC(=O)Cc1cnccn1)C2 Cn1nc(C(=O)NC(Cn2cccn2)C(=O)NC2CCC(F)(F)CC2)cc1C#N c1(C(=O)NCCC2CCCN(CC3CCCCN3)C2)ccc(Br)cc1 C1(NC(CC2CC(=C)C2)=O)CN(C(=O)C(F)Cc2ccccc2)CC1N=[N+]=[N-] Cc1cc(C(=O)NC2C3CC2N(C(c2ccnc(O)c2)=O)C3C)ncc1F c1(C(C)C)ncc(C(=O)N(CCC(C)NC(=O)CC(=O)NC2CC2)C)s1 Cn1nnnc1SCC(N1CCC1CN(C(=O)C=C1CCCCC1)C1CC1)=O C1(C(=O)NCCOC2(C)CCC2)CC2CC2N1C(=O)C(c1ccccc1)O CC(C)(C)S(=O)(=O)CC(=O)NCCCCn1cc(-c2ccc(C#N)c(Cl)c2)nn1 c1(C(=O)NC(C)CNC(c2cnn3c2NCCC3)=O)cncc2c(F)cccc12 Cc1sc(C)c(C(=O)NCC2CC(O)CN2C(C2CCCN2C)=O)c1C#N c1(C(N2CC(CCOC)N(C(=O)C=CCO)CC2)=O)cccc2scnc12.C(C)(=O)O C=C(CNC(=O)C(C1CC1)C1CC1)CCNC(c1nocc1C1CC1)=O S(=O)(=O)(c1ccc(NC2CCC(O)CC2)c(Br)c1)NC(c1ccnn1C)COC c1(C(N(C)CCOCCNC(c2cnn(CC(F)F)c2)=O)=O)cccc(CF)c1 C(=O)(C1=CC(O)C(C(=O)Nc2cc(C)c(Br)nc2F)CCC1)OC C1(COC)(NC(c2csc(O)n2)=O)CCN(C(C2COC(C)C2)=O)CC1 O=C1CC(C(N2CCC(OCC(N3CCCCC3)=O)C2)=O)CC(=O)N1 c1(C(C(=O)NC(CC)C)N(C)Cc2ccc(F)cc2)cccc(OCCCC)c1 c1(N(CC#CC)C)nc(NCC2CC2C2CCCC2)nc2c1ncn2C c1(C(=O)NCC2N(C(C(C)N(C)C)=O)CCC2)cc(N)c(F)c(F)c1F C1(C(=O)NC2(CNC(CCC=C)=O)CCCC2)(N(C)C)COc2ccccc2C1 Cc1nc(Cl)c(NC(C2(C)CCN(C(=O)CCc3cnn(C)c3)C2)=O)cc1Br C1(C(N(C2CCN(CC(N3CCN(C)CC3)=O)C2)CC)=O)CCC2(CCC2)O1 N1(Cc2c(Cl)cc(C)cc2Cl)CCC2CN(C(c3c(C)cccc3Cl)=O)CCC12 n1(CC(=O)NC(C(=O)N(CC(C)SC)C)Cc2cn[nH]c2)cnc(C#N)n1 C1(CC(=O)NCC2N(C(C=CC(C)(C)SC)=O)CC2)CCCC(C2CC2)O1 c1(-n2c(C3(C)CC=CCO3)nc(Cc3cccc(F)c3)n2)cc(Cl)cc(Cl)c1 C1(NC(CC=C(C)C)=O)CCCC12CN(C(C1CC3(CCCC3)CO1)=O)C2 C1(NC(CN(C(=O)Cc2cnn(C)c2)CC#C)=O)COC2(CCC2)C1 C1(C)(C(=O)NCCN(CCC)C(c2cncc(F)c2)=O)CC(CC(C)C)C(=O)O1 C(CCN=c1[nH]nc(O)s1)N(C(c1c(C)cn(C)n1)=O)C C(=O)(C(F)C(F)(F)C(F)(F)F)NC(C)CNC(=O)C=Cc1cnc(C(C)(C)C)s1 c1(NC(c2n(CC)nnn2)c2nscc2Br)ccc(C(=O)OC)c(F)c1 C1(C(=O)NCCCC2OCCN(C(c3cc(C)oc3)=O)C2)OCC2CCCCC12 C1(C(N2CCC(NC(=O)CCc3ccc(Cl)s3)C2)=O)CC(=O)N(CCCF)C1 N(C(=NCCSCCOC)NCC(CSC)OC)C(c1cccc(Cl)c1)C(=O)OC C1(C(=O)NC(CC=C)CNC(C2CN(S(=O)(=O)CC)C2)=O)CN(C)C(=O)CCO1 C(=O)(CC(C)P(C)(C)=O)NC1C(C)CN(C(C2(C(C)(C)O)CC2)=O)C1 c1(C(C(=O)NC2C(CNC(C3(CC#C)CCC3)=O)C2)O)ccc(Br)cc1 C1(CC)CCN(C(=O)C(C)=C(C)C)C1C(=O)NOCCCC(F)(F)F c1(C(N2CC=CC(NC(C(C)CC3CCCCC3)=O)C2)=O)nc(Cl)cc(N)c1Cl C1(CNC(CSCC#C)=O)COCC1NC(=O)CCC1(C#N)CCC1 c1(C(=O)NCCOCCNC(C(C(COC)C)C)=O)cnc2ccoc2c1 c1(C(=O)NC2(CC=C)CCN(C(=O)C=NOC)C2)cc(F)c(F)cc1NC(N)=O N1(C(C(F)=CCC)=O)CCN(C(c2n[nH]c(C3CC3)c2Br)=O)CC1C(C)C C(=O)(CP(=O)(C(C)C)C(C)C)N(CCC(C(C)C)NC(C(C1CC1)OC)=O)C C(CC(C)(C)C)(C(=O)NC1CCC(OC)C1)NC(c1n(C=C)ncc1)=O C(=O)(C(C)(C)CCC#N)N1CCCC(NC(c2cc(SC)oc2C)=O)CC1 c1(NC(N(CCC#C)C)=O)ccccc1SC1CSC1(C)C c1(CNC(CSCC=C)=O)csc(CNC(c2cnoc2C2CCC2)=O)n1 CC(C)(CNC(=O)NC1CC2(C1)CC(CF)C2)C1=CCCC1 c1(CC(P(C)(C)=O)C(F)(F)F)cn(C2CCCc3cnccc32)nn1 c1(C(=O)NC(C(C)NC(c2c(OCC=C)cccc2)=O)C)ccc(C)n(C)c1=O C(=O)(C(C)(COC)OC)NC(CN(C(c1cc(C(F)F)cs1)=O)CC)C C(CCN=c1[nH]c(=N)[nH]c(=NCC23COCCN2C(=O)OC3)[nH]1)OCC c1(C(N2CCC(C(N(C)Cc3c(C)n[nH]c3)=O)(CF)C2)=O)ncn2c1CCC2 Cc1ccc(F)c(C(=O)NC(C)CNC(c2ccc(OCC(F)(F)F)o2)=O)c1 CC1(C(=O)NCNC(=O)CNC(c2nc(C3CC3)cs2)=O)CC1(Cl)Cl C1(C(=O)NCC(C)(C)OC(C)C)CN(C(C2CCCC(C)CC2)=O)CCC1(C)C N1(C(C2(CCCC)CCC2)=O)CCOCC(C(=O)NCCN(S(C)(=O)=O)C)C1 C1(C(=O)NCC2CC2(Cl)Cl)CCCCN(C(=O)C=CC2CCCC2)C1 c1(C(N(C2CCC(NC(CN(c3cnccn3)C)=O)C2)C)=O)cncc(O)c1 C1(C(N(CC(=O)OC)C)=O)(CC)CCCN(C(C2(SC)CCOC2)=O)C1 CC1CCC(C(=O)NCC2CC(O)C(O)C2)CN1C(C1CC1(F)Cl)=O N1(C(C(CC)CC)=O)CCN(C)CC1CNC(=O)C(c1ccc(Cl)cc1)CO C1(C(=O)NC(c2noc(C)n2)CC)CC(NC(=O)C(C#N)CC)CCO1 c1(C(=O)NC2CCC(N(C(C(CSC)C)=O)C)CC2)cc2cc(F)ccc2s1 C(CCS(=O)(=O)C(C)C)N(CC1CCCN(C(COCCC=C)=O)C1)CC N1(C(c2cc(NC(C)=O)ncc2)=O)CCN(CCc2ccccc2F)CC1C c1(NC(C2CC3CC3N2Cc2ccc(Cl)o2)=O)cc(F)c(F)cc1Br C1(C(=O)NCC(CC)NC(c2ccc(C(C)C)cn2)=O)CCS(=O)(=O)N1 c1(Cn2cc(C3(OC(=N)O)CC3)nn2)ccc(NC(CC2(C)CC2(F)Cl)=O)cc1 Cc1ncccc1C(=O)NCCOCCN(C(=O)C(C)OCCN(C)C)C N1(C(c2ccc(CCC)s2)=O)CCCC(O)(CNC(=O)Cc2cc(C)on2)CC1 Cc1cc(CC(=O)NC2CCN(Cc3sncc3Br)C2)cc(F)c1 N1(C(C2(CCC)CCC2)=O)CCC(C(F)CNC(=O)Cn2cc(C)cn2)CC1 c1(C(N(C)CC2CCCN(C(C(C)C)=O)C2)=O)c2c(cc3c1CCC3)CCC2 C1(C(=O)NCC2(NC(c3ncsc3Br)=O)CCC2)CC2CCC1O2 N1(C(CC(C)(C)C)=O)CCC(NC(c2cnn(CCF)c2)=O)C(CO)CC1 C=C(C)CC(C(=O)NC1CCC(C(=O)Nc2cnn(CC)c2C)C1)OC C(=O)(C1=CC(C)(CC)C1)NCCCC(Cc1ccccc1)NC(C(CCC)O)=O c1(NCc2ccnc(C)n2)[nH]c(=NCCCCn2cnnc2)nc2ncn(C)c12 c1(C(C)C)ccc(OCC(N2CCC(NC(=O)CC(C)CF)C2C2CC2)=O)cc1 C=CC(C)(O)CC(=O)NCC1CC(C)CCN1C(=O)Cc1sccc1C C1(CC(=O)N(C(C)CCNC(c2cnn[nH]2)=O)C)(CO)CCCCC1 c1(CNC2CC(NC(c3ncccc3Cl)=O)C2)cnn2c1CCCC2 c1(C(N2CC(C)N(C(=O)Cc3cc[nH]c(=N)c3)CC2)=O)ccc2nnnn2c1 Cc1ccccc1C1=NOC(C(N2CC=CC2CNC(C2(CF)CCC2)=O)=O)C1 N1(C(c2nc(OC)c(C)s2)=O)CCN(C(c2cscc2C)=O)C(CCO)C1 c1(C(=O)NC(C(N2C3CC(=C)C(C3)C2)=O)C2CC2)cccc2ccoc12 N1(C(CCOC(C)C)=O)CCC(CCNC(c2ccc(=N)[nH]n2)=O)CC1 Cc1cc(C(=O)NCCC(C)N(C)C(c2ncn(C(C)(C)C)n2)=O)n(C)n1 Cc1cccc(-c2cn(C(C)C(=O)NC(c3ccccn3)(C)C)nn2)c1 C(=O)(C1=CCCCO1)N1C(C(=O)NCC(C)C2CC2)CCCC1 N1(C(C(C)Cc2ccccc2)=O)CCC2(CCC2NC(C2CC(C)(C)C2)=O)CC1 c1(C(=O)NC23CC(C(N(C)Cc4cccnc4)=O)(C2)C3)cccc(=O)n1C N1(C(c2nnn(CC)c2C)=O)CC(CNC(=O)COc2ccon2)CC12CCC2 c1(SC)nccc(CN2CCCC(C(=O)NC(c3nccc(C)n3)C)C2)n1 c1(C(=O)NCC(C)(C2CC2)NC(COCCSC)=O)c(C)nsc1NC C(CNC(=O)C(c1cnn(C)c1)O)(CCCC)NC(COCC#C)=O c1(C(=O)OCC2CCN(C(=O)OC(C)(C)C)C2)ccc(O)c(O)c1 C1(CC(=O)NCCCCCN(C)C(c2cn(C3CC3)nn2)=O)CCCCC1(F)F C(CC(=O)Nc1ccc(C)cc1)(C(C)OC)NC(C(C)OCCC=C)=O C1(NC(C2CCC(=C)CC2)=O)CN(C(=O)C(C(C)C)NC=O)CC(C)(C)C1 N1(C(C(CC#C)O)=O)CCN(C(c2cnn(C)c2Cl)=O)CC1COC c1(C(c2n(CC(=C)C)nnn2)NC(C)CNC(=O)OC)ccc2occc2c1 c1(N(C(=O)CC2CC3COCC23)C)cccc2cccnc12 C1(NC(C(C)=C2CCCC2)=O)CN(CC2CCN(CC(C)C)C2)CC1C c1(C(=O)NCC2(OCC)CN(C(=O)C(C)OC3CCOC3)C2)nc(C)sc1C N1(C(COC)=O)CCCC(C(C)(C)C(=O)NCC2(N(C)C)CCC2)C1 c1(C(C(=O)NC2CN(C(C3(C)CC3)=O)C2)N(C)Cc2ccco2)cc(Cl)ccc1Cl N1(C(C2C=CCC2)=O)CC23CCCCC2(C1)CN(C(C1(C(F)F)CCCO1)=O)C3 C(=O)(C(CNC(=O)C(F)OC(F)(F)F)N(C)C)N(CC)Cc1ccoc1 CCC(C)(C(=O)NCCCN(CCO)C(C1CCC(C)(C)C1)=O)C(N)=O c1(C(N2C(CNC(C=CCOC)=O)C3CC3C2)=O)ccc(C)c(OC2CC2)c1 c1(OCC=C)cc(Cl)ccc1C(N1CC(CCNC(=O)CC2CCCC2O)C1)=O c1(C(=O)NCC2C(CNC(C(C)SC(C)C)=O)C2)cc(Cl)c(F)c(Cl)c1 CC1(C)CC(C)(CNC(=O)C2=CCCCO2)CN1C(c1ccc(C(F)(F)F)[nH]1)=O N1(C(c2cc(Cl)ccc2O)=O)CCCC2(C1)CN(C(c1cccnn1)=O)C2 Cc1[nH]c2ncccc2c1C(N1CC(N(C)C(C2CC(N(C)C)CCO2)=O)C1)=O C1(NC(=O)OC(C)(C)C)CC(NC(=O)NCc2cnc(C)c(C)c2)C12CCC2 N#CC1CCCCN1C(C1CCC(NC(c2cscc2Cl)=O)CC1)=O Cc1nc(C(N2CC=C(CNC(=O)CC(C)F)CC2)=O)ccc1Br Cc1ccnc(C(C)(C)C(=O)NC2CC(C)(NC(c3cn(C)c(O)n3)=O)C2)c1 C=CCCC(C(=O)Nc1ccc(N(C)C)nc1)NC(C1CC1C1(C)COC1)=O c1(C(=O)OC(C)(C)C)coc(C(C)(C)NC(=O)OC(C)(C)C)n1.CC1C(=O)N1 c1(C(N2CCC(CCNC(C(C)SCCCC)=O)C2)=O)ccc(Cl)c(OC)c1F N1(C(c2cc(C)cc(O)c2)=O)CC(C)(C)OCC1CNC(=O)CCC1CCOC1 c1(N2CCCC(OC)CC2)nc2cc[nH]c2c(=NC(C)Cc2ccccn2)[nH]1 n1(CCC)nc(C)cc1C(=O)NCC1CCN(C(=O)C(C)O)C1 Cc1nc2ccc(C(N3CC4(CCCCN4C(=O)C4=CCCC4)C3)=O)cc2s1 c1(OC)ccccc1C(C)CNC(=O)C(c1ccc(Br)cc1)F c1(C(N2C(CNC(CSCCCC)=O)C(C)(C)CC2)=O)ccc([N+](=O)[O-])cn1 N1(C(C(CCC)NC(N)=O)=O)CC2CC1CCN2C(=O)CCCCCN(C)C N1(C(CCCCN(C(C2CCN(C)C(=O)C2)=O)C)=O)CCCC(C2CCC2)C1 C1(C(=O)NC2CC(C)CN(C(c3csc(O)n3)=O)C2)CC2COCC(C1)C2 N1(CCO)CCCCC1C1C(NC(=O)CSCC(n2ccnc2)=O)C1 C1(C(=O)NC(C(C)SC)C)CC=CC(NC(=O)CCn2ccnc2)C1 C(C1CCCC1)=CC(=O)NCC1CC(CNC(C(C2CCCCC2)C)=O)C1 C(=O)(CCC(=O)N1CCC(CNC(c2cn(C(C)(C)C)nn2)=O)C1)OC CC(C(=O)NCC(C)(Cn1cccn1)NC(c1n[nH]c(CO)n1)=O)S(C)(=O)=O.CC C(=O)(C1CCCc2ccnn21)N1CC(NC(=O)CCOCC(F)F)C2(C1)CCC2 C1(NC(c2c(C)snn2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)C2(CCOC2)C1 Fc1ccc(Br)cc1CNc1nc(-c2cccc(I)c2)cs1 C(CCCCCF)N(C1(C(=O)O)CCOC1)C C(=O)(C1CCc2cccc(=O)n21)N1CCC(C)(NC(C2CCCCC2)=O)CC1 C1(NC(CN(C(=O)OC)C)=O)CC(F)(F)CC1NC(c1nc(C)n(C)c1C)=O c1(NC2C(NC(C(C)N(C)C)=O)CS(=O)(=O)C2)ncc([N+](=O)[O-])cc1Br c1(OC)ncc(C(N2CCCC2C(C)NC(=O)C(C)(C)OC)=O)cc1C(F)(F)F C1(CNC(c2c(CC)scc2)=O)CCN(C(c2cccc(C)n2)=O)CC1(F)F C1(C(C)(C)O)(CNC(C23CC(CO)(C2)C3)=O)CN(C(=O)C(C)CF)C1 c1(NC(C2(C)CCN(C(CCc3cccc(C)n3)=O)C2)=O)cc(Cl)ccc1I n1(CS(C)(=O)=O)c(N2CCC(c3ccccc3)CC2)nnc1C1CNC(=O)N1 C(CC(C)C)(C(=O)NCC(C(C)C)NC(c1cc(Cl)ccc1O)=O)OC C1(C(=O)NCCC(=O)Nc2c(F)cccc2Cl)C2Cc3ccc(Cl)cc3C12 CC1(C)CCCN(C(=O)CCCC2CC2)C1CNC(C1CCCOC1)=O C1(C2CCN(C(C3CC(=O)N(CC)C3)=O)C2)(NC(c2c(OCC)ccs2)=O)CC1 n1(CC#C)cnnc1C(=O)N(CC(=O)NC1CNC(=O)C1)C1CCC1 N1(C(C(CC)CC)=O)CCC(C(=O)NC2CC(C)(CO)C2)C(O)C1 N1(Cc2nn(C)c(Cl)c2[N+](=O)[O-])CC2COCC(C1)C(=O)N2 N1(C(C(C(C)C)NS(C)(=O)=O)=O)CCN(C)CC1CNC(c1cc(C(N)=O)co1)=O C(CCCC(=O)N(C1CCCC12CC2)C1CC1)NC(CC1ON=C(C)C1)=O C(CSc1nncn1-c1ccccc1)(C(=O)NC(C)CC(C)NC(C)=O)NC(C)=O C(=O)(C1CCCc2scnc21)NC1CC(F)(CNC(CCCC(CC)C)=O)C1 C1(C(N2CCC(N(CC(=O)NC(C)C)C)C2)=O)CCC(F)(F)CC1(C)C C(=O)(C(CC)CCCC)NC1CC(CCn2cc(C(=C)C)nn2)C1 C1(NC(C(C)(C)F)=O)COC2(CCN(C(c3cc(C#N)cs3)=O)C2)C1 C1(CCNC(CN(C(CC=CC)=O)CC(C)C)=O)CCCCC1O N#Cc1ccc(C(=O)NC(C2CCCCC2)C(=O)NCCc2cocn2)s1 Cn1[nH]c(C(=O)NC2CCCC2CNC(=O)CN2CCCC2CO)nc1=O N1(C(Cc2cccc(N)c2N)=O)CCCC(C2CC2NC(C2CCC(=O)N2)=O)C1 N(C1CCc2ccccc21)(C(CCC=C)C)CCOC1CCCC1 C#CCCCCCC(=O)NC(C)CNC(C12CCC(C(F)F)(CC1)C2)=O C12(CNC(CCCCSC)=O)CCCCC1N(C(=O)CCCNC(N)=O)CC2 C1(NC(Cn2ncc(C)cc2=O)=O)CCCC12CN(C(c1n[nH]c(C)c1O)=O)C2 C1(C)(NC(C2CC(=C)C2)=O)CCCN(C(=O)C=Cc2ccccn2)C1 N1(C(CN(CC)CC)=O)CCC(CCN(C)C(c2cnc(C(C)C)[nH]2)=O)CC1 C12(C(=O)NC(CN(C(=O)CC3(COC)CC3)CC)C)CC1COC2(C)C c1(C(N2CC(O)(C(C)NC(CS(CC)=O)=O)C2)=O)ccc(OC)c(N)n1 N1(C(C(C(C)C)(C)O)=O)CCS(=O)(=O)C(CCNC(=O)C2=CCC(C)CC2)C1 C1(NC(C(CCC)OCC)=O)CC2CCC1N2C(C1(C)CC1)=O c1(OCC)ccccc1OCC(N1CCCC(N(C(=O)Cc2ccon2)C)C1)=O C1(C(N(C2CCCCC2)CC#C)=O)CCCCC1CNC(C1(F)CC1)=O C(C(=O)NCCC(Cl)Cl)(C(C)(C)C)NC(CC(C)c1ccco1)=O N1(C(C(C)C2CCC2)=O)CCC(O)(CN(C(=O)Cn2ccc(Br)n2)C)C1 c1(C(N2CCCC(O)(CNC(c3nccs3)=O)C2)=O)c(F)cc(Br)cc1F c1(CC(=O)NC(C)(CNC(C2(C(F)(F)F)CCC2)=O)C2CCC2)cccnc1Cl N1(C(CN2CC(C)(C)C2)=O)CC(CNC(C2CCCCCC2)=O)CC1(C)C C(C(C)(C)C#CC(=O)NCC1(O)CCOCC1)NC(CC1ON=C(CC)C1)=O N1(C(c2cc(C)nn2C)=O)CCC2(CC1)COC(C)C2NC(C1CC1F)=O c1(CCC)nc(C)c(C(=O)NC2CCCCC2NC(c2ccc(F)cn2)=O)o1 c1(C(N2CCC(NC(C3CC(C(F)F)C3)=O)CC2)=O)cc2ccc(Cl)c(F)c2[nH]1 c1(C(=O)NC2CN(C(c3ccnnc3Cl)=O)C2)ccnc(Cl)c1Cl C(=O)(C(C)C(F)(F)F)NC1CC2(C(NC(c3c(C)cc(CNC)o3)=O)C2)C1 FC(F)CCN=c1cc(N2CC3CC2CC3(F)F)nc(C(F)(F)F)[nH]1 N1(C(c2cc(F)ccc2Cl)=O)CCC(N=c2ccc3nccn3[nH]2)C1 C1(CNC(C2(CC#C)CCCC2)=O)C2CCC(C2)N1C(c1cc(COC)cs1)=O C1(C#N)(C(N(CCCCNC(=O)CN(C2CCSC2)C)C)=O)CCCOC1 c1(CC)ccc(Cl)c(C(=O)NC(C)CCNC(=O)CNC(c2ccncc2)=O)c1 C1(CN(C(=O)C(C)(C)C2CCC2)C)CCCN1C(=O)CC1CCNC1=O C1(CNC(C(=O)NCC(n2cc([N+](=O)[O-])cn2)(C)C)=O)CCC(F)(F)C(=O)N1 C(=O)(C1=CCCC1(C)C)NC1CCCN(C(c2c(N)cn(C)n2)=O)CC1 c1(C(=O)NCCC2(CNC(C(C)(C)CO)=O)CC2)cc2ccnn2cn1 N1(CC(=O)NC2(C)CC(C(F)(F)F)C2)CC(C(F)(F)F)CCC1=O Cc1cc(CNC(c2cc(F)c[nH]2)=O)oc1C(=O)N(C)CC1CC1(F)F NC1CCc2cc(OCc3ccn(C4CC4)n3)ccc21 CCC(CC(C)C)C(=O)NC1COCC1C(=O)NCc1nnc(C2CC2)o1 C1(C2CCN(C(C3CNC(=O)CC3(C)C)=O)C2)(NC(c2c(CC)nco2)=O)CC1 c1(CC)cccc(C)c1NCc1ccc(N2CCC(C)CC2)c(F)c1 Cc1cc(C(N2CCCC2C=CC(N2CC(O)(C(F)(F)F)C2)=O)=O)cc(F)c1 C1(C)(C(=O)NC2CCN(C(c3cnc(C(C)=O)s3)=O)C2C)CCCCNC1=O C(=O)(CC(C)C(C)(C)C)N(CCCCCNC(c1ccn(C(C)C)n1)=O)C CC1(C)CCC(NC(=O)CC(F)(F)F)C(CNc2ccnc(C3CCC3)n2)C1 c1(OC(CC)C)cc(NC2CC(c3ccccc3)C2C)ccn1 c1(C(N2CC(CCCNC(C3N(CC)CC3)=O)OCC2)=O)cc([N+](=O)[O-])cn1C C#CC1CN(C(c2ccc(C(C)C)o2)=O)CCN1C(c1n[nH]c(CC)c1C)=O C(=O)(C1=CC2CCC=CCCC12)NCCCN(C(=O)CCF)C1CC1 c1(C(=O)NCCC(CNC(C=CC(C)C)=O)O)cc(F)ccc1O c1(C(=O)NCC2CCC(NC(c3ccc(Cl)nn3)=O)CC2)ccc2sncc2c1 Cc1ccc2c(c1)N(C(c1cc3ccncc3s1)C(=O)NCC(F)F)CC(C)O2 c1(C(N2CCC(C(C)NC(c3ccn(C(F)F)n3)=O)C2)=O)cc(O)nn1C c1(CC)cc(C)nc(C(=O)N(CCCCCNC(=O)C(n2cc(C)cn2)C)C)n1 CC1C(C(=O)NC2CC(C(=O)Nc3n[nH]c(-c4ccccn4)n3)C2)CCN1C c1(C(N2CC(C(NOCC(=O)OC)=O)OCC2)=O)ccc(C)c(OC)c1 N1(C(CN(CC(C)(C)C)C)=O)CCCC2(NC(=O)CC3CC=CC3)CCCC12 C1(COC)CC(O)CN1C(C1COCCN1C(=O)Cn1nc(C)oc1=O)=O c1(C(=O)NCC2(CNC(C(C(C)(C)C)N(C)C)=O)CC2)cncc2nc(O)[nH]c12 Cc1cc(C(=O)NC(C)CC(C)NC(=O)CCc2cnco2)cc(C)c1O Cn1ncc(CNC(=O)C(=O)NC2C3CC4C(C3)C24C(=O)O)c1S(C)(=O)=O N1(C(C2CCN(C(CC)=O)C2)=O)CC(S)CC1(C)C.C(=O)(C(CC)CC)OCCN C1(C)(CC)CC(NC(=O)C(C)(C)NC(=O)CCc2cnc(C)o2)C1 C1(C(=O)NC(CN(C)C(C2CNC(=O)C2)=O)(C)C)CC(C2CC2)C1 C=CC1(CC(N2CCC(CNC(=O)C=CC(C)CC)C(C)C2)=O)CCOCC1 C12(C(N(CCCNC(COCC(=O)NC)=O)C3CC3)=O)CCC(C(F)F)(CC1)C2 Cc1cc(=NCC(C(F)(F)F)n2cccn2)[nH]c(=NCC(C)C)[nH]1 c12ccc3cc(ccc3c1)OS(=O)(=O)O2.C=CCC(F)(F)C(=O)OC c1(OC)cc(Br)cc(CN2CCNCC2C(=O)Nc2nc(C)cs2)c1O N12CCCN(CC1C)C(=O)C(CCSC)N(C(C)C)CC2=O.CCOC c1(NC(C)=O)ccc(C(N2CCCC(NC(c3ccc(C)nc3)=O)C2)=O)c(Cl)c1 c1(C(=O)NC(C(C)NC(CC(CCC)O)=O)(C)C)ccc([N+](=O)[O-])cc1Br CC1(C(=O)NNC(=O)Cn2cnccc2=O)CC12CCOCC2 N1(C(c2ccc(C(C)(C)C)[nH]2)C(=O)Nc2ccccc2Cl)CC(CO)C(C)(C)C1 N1(C(C(CC)F)=O)CCN(C(=O)Cc2ccc(F)cc2C)C(c2cn[nH]c2)C1 N1(S(CCCCC)(=O)=O)CCC2(CCC2)CC1C(=O)OC C1(O)(C(=O)NCC(CC=C)NC(=O)C(F)=CC2CC2)CN2CCC1CC2 Cc1ccc(NC(=O)CCC(=O)N2CC(NC(=O)C(C)N3CCC3)C2)cc1C N1(C(C2OCC(C)C2)=O)CCn2ncc(CNC(C3CCSC(C)C3)=O)c2C1 C1(N(C(c2ccc(C)s2)=O)CC2CC2)CCN(C(c2nccn2C2CC2)=O)CC1 Cc1nc(CC(N2CC(CNC(=O)C(C(C)C)NS(C)(=O)=O)C(O)C2)=O)c(C)s1 c1(CC(N2CC(C)CC(CNC(C(CC)=CC)=O)C2)=O)coc2ccc(C)cc12 c1(NC(C(CCC)C)c2nnnn2C2CC2)ccc(CSCCC(N)=O)c(F)c1 C=CCC(C(=O)NC1(CC)CN(C(c2nnccc2C)=O)C1)NC(C)=O N=c1nc2c(C(=O)NC3CC(O)CN(C(=O)Cc4cn[nH]c4)C3)cccn2[nH]1 c1(C(N2C3CCC2CC(NC(C24CC5CC2C4C5)=O)C3)=O)cccc2occc12 C1(C(=O)OC2CC(C)OC2=O)COC2COCC2O1 C1(CC(=O)NCCNC(=O)Cc2cc(C(F)(F)F)co2)CCCOC1 c1(C(=O)OCC)[nH]c2nccnc2c1NCC.c1(C=O)nn(C)nc1Br CC(C)CC(C)C(=O)OC(c1ccc(Br)c(N(C)C)n1)=O CC1C(C(N2CCN(C(c3n[nH]cc3C(C)(C)C)=O)CC2)=O)CCN1C Cc1cn2ccc(C(=O)NCC(C(C)C)NC(=O)CNC(=O)C(F)(F)F)cc2n1 n1(CN2CCC(C#N)C2)ccc(=NC(=O)C2Cc3ccccc3O2)[nH]1 c1(-c2cc(C)no2)ccc(-c2nc(C(C)C)nn2C(C)C(C)C)cc1 Cc1nc(CN2CCC(NC(=O)C(C)OCC(C)C)C2)n[nH]1 C1(CC)(NC(=O)CCCC(C)=O)CCCN(C(=O)C(CC)N(CC)CC)C1 CN(NC(=O)NCCc1ccc(Br)c(Br)c1)c1ccccc1 c1(OC)ccc(Br)cc1C1CCCN1C(=O)C(=O)N1CCC1CC(C)C CC(C)CC(C)CC(C)NC(c1cccc(N2CCCC2=O)c1)=O C#CC1CN(C(C2CC2C2CCCC2)=O)CCN1C(c1cnn(C)c(=O)c1)=O c1(SCC)cccc(C(=O)NC(CNC(=O)CC2CCS(=O)(=O)C2)C(C)(C)C)c1 c1(C(=O)OC)coc(C(=O)NCCCCCN(C(=O)C(C2CC2)SC)C)c1 N1(C(C2CCC(C)(CC)O2)=O)CCC2(CCC2)C(CNC(c2cc(C)c[nH]2)=O)C1 C1(C)(C(N(C)CCNC(c2cnnn2Cc2ccccc2)=O)=O)CCCNC1=O c1(C(CC(=O)OC)NC(=O)C(C)(C)OC)ccc(OC(F)F)c(OC)c1 C1(CCOC)CN(C(=O)CC2CCCCN2C)CCN1C(=O)CC1(COC)CC1 c1(N2C(CC)CN(C(C3CN(C)C3)=O)CC2)nccc(S(C)(=O)=O)n1 C(=O)(CCC1=CCCCC1)N(C)CC1(O)CCN(C(CS(=O)(=O)NC)=O)C1 CCC(C)CCCC(=O)NC1CCCC(NC(c2cnn(C3CC3)c2)=O)C1 c1(CC(=O)NC(CC=C)CNC(C2(n3ccnn3)CC2)=O)ncccc1C n1(CCC)nc(C)cc1C(=O)NCC(C)(C)NC(=O)C(c1cncc(F)c1)C CC1CN(C(=O)C2=CC(C)(C)C2)CC(CCNC(c2cccc(C#N)c2)=O)O1 c1(C(N2CC(CC=C)(NC(=O)CC3(C)CC3)C2)=O)ccc(Cl)cc1Cl CC(C)C(C)(C)C(=O)NCc1cc(C(=O)NC(CC(C)N(C)C)=O)ccn1 CCC(F)(F)CC(=O)NCC1CN(C(C2CC(C)OC2C)=O)CC1C CC(C(C)(C)CN(C)C)NC(=O)NC(c1ccc(CSc2ccco2)nc1)=O C1(C(=O)NC2CC(CCNC(=O)Cn3cccc3)C2)CC2(C1)OCCO2 Cc1c(C(=O)NC2(C)CC(NC(C3CCC=CCCC3)=O)C2)cccc1O c1(NC(C2N(C(Cc3scc(C)c3)=O)CCC2(C)C)=O)ccc2ncccc2c1 c1(OCC(N2CC(CNC(C3(C=C)CC3)=O)C(O)C2)=O)cc(Br)ccc1F CC1=C(C)CC(C(=O)NCC(O)CC(=O)NCC2(CO)CCCO2)CC1 C1(CC=C)(NC(c2cc(C3CC3)oc2C2CC2)=O)CCN(C(C2CC2C)=O)CC1 c1(C(N2C(C(=O)Nc3cccc(OC)c3I)CC(C)C2)=O)cc(F)c(C)c(F)c1 c1(SC)ccc(C(=O)NCC(C2CCC2)NC(c2ccnn2CCF)=O)s1 CCC(C)C(O)C(=O)NC1(C(=O)NCC(=O)N2CCCO2)CC(F)C1 C1(NC(c2n[nH]c(C3CC3)c2Cl)=O)CCCN(C(c2cnccn2)=O)C1 N1(C(C(C)N(C)C(c2cccnn2)=O)=O)CC(O)(C(N)=O)C1 C(CN=c1[nH]c(NC(CC2CC2)C2CC2)nc2cc[nH]c12)(CC(C)C)OC C1(C(N(CCNC(C2(C(CC)=O)CC2)=O)C)=O)CC=CCC1 CS(=O)(=O)C1CC(C(=O)NCC2CCCN2C(C2CCC2)=O)C1 C1(NC(CCC)=O)CN(C(=O)CC2CCOC2=O)CCC12CCC2 c1(C(=O)NCC(CNC(C2(C(N)=O)CC2)=O)F)ccc(C#CC2CC2)cc1 Cc1cc(C)n(C)c(=O)c1CN(C(=O)C(=O)NCC1CCC=C1Br)C1CC1 Cc1cc(C(N2CCN(C3CCN(C(=O)C(C)C4CC4)C3)CC2)=O)oc1Br C1(C(N2CCC(C(F)F)(CNC(C3(Cl)CC3)=O)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC2CN(C(C3C(CC)C3)=O)CC2CC2CC2)cc(N)ccc1C CN1CCOC(CC(N2CC(CCc3cn(Cc4cccnc4)nn3)C2)=O)C1 Cc1cc(CO)oc1C(=O)NC1CC(CNC(c2cnccn2)=O)C1 N1(C(C2(C#C)CC2)=O)CCC2CN(C(c3ccc(F)c(SC)c3)=O)C2C1 c1(C(=O)NCC2C(NC(C(CC)NC(N)=O)=O)C2)oc(C)nc1C C(=O)(CC1=CCN(C)CC1)N1CCC(NC(c2c(C)cccc2O)=O)C1 C(=O)(C(Cc1cnc[nH]1)NC(=O)CCc1nc(=N)[nH][nH]1)N(C(C)CO)C C1(NC(C=C(c2nccc(C)c2)C)=O)CN(C(=O)CC(C)F)CC12CCOCC2 N1(CCNC(C(C2CC=CCC2)NC(c2cc(Cl)no2)=O)=O)CCC2CC12 c1(NC(C(CCC)OC)=O)ccc(NC(c2ccn(C(C)(C)C)c2)=O)cc1C N1(C(=O)C(F)C2CCOC2)CCN(C(c2ccc3c[nH]nc3n2)=O)C2(CC2)C1 C=C1CCCN(C(C)C(=O)NC(=O)NCC)CC1 n1(CC(=O)NC(CCCCNC(COC(C)=O)=O)C)nc(C(F)F)c2c1CCC2 C(=O)(CC(C(C)CC)NC(c1cccc(C)c1C)=O)NCc1n(CCC)cnc1 C(=O)(C1CCCc2nncn21)N1C(C)(C)C(NC(=O)C(F)=C2CCCC2)CC1 Cc1cccc(-c2csc(-n3c(-c4ccc(-c5n(CO)ccn5)s4)c(F)cn3)n2)c1 C(=O)(C(F)C(C)CNC(C1CC2(CC(=O)C2)C1)=O)NCCC(CCC)C1CC1 Cc1cncc(C)c1C(=O)NCC(c1cccc(Cl)c1)NC(=O)C(C)(C)C CCS(=O)(=O)c1ccccc1-c1cnc(NC(c2ccc(OC)nc2)=O)c(O)c1 CC1(C)CCC(CNC(C2CC=CCC2NC(C2(CO)CC(C)(C)C2)=O)=O)O1 C1(NC(c2cncc(Cl)c2)=O)CCNC2(CC2)C1 CCCC(CC)CCC(=O)N1CCC(C(N2CCCNC(=O)C2)=O)C1CC c1(CC)ccccc1C1CC1NC(=O)CC(C)(C)C N1(C(Cc2ccc(C(C)=O)s2)=O)CC(F)(F)CC1C(=O)NCCC1CCCO1 N1(Cc2c(NC)nccc2)CC2CC1CC2CNC(=O)C=C(C)C Cc1cc(Cl)cc2[nH]c(C(=O)N(C3CCN(C(c4csc(CO)n4)=O)C3)C)cc12 N1(C(c2c(C)nc(C(C)OC)s2)=O)C2CCC1CN(C(c1nc(O)c(C)s1)=O)C2 N1(C(=O)CSc2cccs2)CC(C2CCCN(C(C3CC34CC4)=O)C2)C1 C1(NC(c2cncc(OC)n2)=O)CCN(C(C2NC(=O)OC2(C)C)=O)CC1F c1(C(=O)NCCC2(CNC(C3(Cl)C(C)(C)C3)=O)CC2)ncn2c1CCC2 c1(C(C(=O)NCC(C)C)N(C)Cc2csc(CO)n2)cc2c(s1)CCOC2 C1(NC(c2n(CC(=C)C)nnn2)c2cncn2C)CC2CC3C(C2)C13 C1(NC(C2CC3(CC(C(N)=O)C3)C2)=O)CC2(CCC(NC(=O)CC3CC3)CC2)C1 CC1(C)CCCCC1CC(=O)NC1CC2C1CCN2C(c1cc([N+](=O)[O-])n[nH]1)=O C1(CC(C)NC(=O)CO)CCC(C2CC2)N1C(=O)CCc1ccoc1 C(=O)(CC(C(C)C)C(C)C)NCCNC(c1cncc(OCC)c1)=O c1(NC)ccc([N+](=O)[O-])c(C(=O)NCC2CN(C(=O)C=C(Cl)Cl)CC2(F)CO)c1 C1(C(N2CCC(C(F)(F)CO)C2)=O)CCN(c2ccncn2)C1 Cn1cnc(C(N2CC(NC(=O)C(O)CC3CC3)C2)=O)cc1=O C1(CNC(Cc2c(C)ocn2)=O)CCCC2CN(C(=O)CCCS(C)(=O)=O)CC12 C(=O)(N=c1cc(C2CC2)n(C)[nH]1)C1CN(C(CC(CC)O)=O)CC1C c1(C(=O)NC2CCC(NC(C(CC)(C)CO)=O)C2)nccn2ccnc12 Cc1cc(F)sc1C(N1CCC(N(C)C(C2CC(CCC(N)=O)C2)=O)C1)=O C1(CNC(C(C)N(C)C(c2ccnnc2)=O)=O)CCCC2CC12 C(CCCCCC(=O)NC1CCCC1N(C)C)NC(c1cc(OC)n[nH]1)=O.C(C)(=O)O CCCC(C(=O)N1CCC1C)NC(=O)C(C)(C)F N1(C(C(CCC)NC(C)=O)=O)CC2CCC(C(=O)Nc3ccccc3OC)(C2)C1 c1(OCC)cccc2[nH]c(C(N3C4CC3CN(C(C3CCC(C)O3)=O)C4)=O)cc12 N1(CC(=O)NCC2C(CNC(C3(C=C)CCC3)=O)C2)Cc2ccccc2C1=O C(=O)(CS(=O)C(F)(F)F)N(C(C)CN(C(=O)C1=NOCC1)C)C N1(C(C(C)=CC)=O)CC2(COC(CNC(=O)C(N3CCOCC3)OC)C2)C1 c1(OC)ncnc(NC(c2cc(-c3cncc(SC)c3)cnc2Cl)=O)c1OC c1(-c2c(C(N3C(C)CCC3C)=O)cc(Cl)cn2)nc2c(s1)CCC2 N1(C(CCCn2cc(CSC)nn2)=O)CC(C)C(O)C1 NS(=O)(=O)CCCCCC(=O)NCC1CN(C(=O)CCCc2cnn[nH]2)C1 c1(C(=O)NCC2C(NC(C(CC)O)=O)CCCC2)csc2ncnc(O)c12 FC1(F)CC1C1CCN(c2ncnc(C3CC3)c2Br)CC1 C(=O)(C(F)(CNC(=O)C(C)(C)C(F)(F)F)C(C)C)N1CC(CC)C(O)CC1 C(=O)(C(C)(CC)C(F)F)N(C1CCC(CNC(CCCC(=O)OCC)=O)CC1)C c1(C(c2n(CCCC)nnn2)N(C2CCC3CC23)C)ccc(CCSCC)cc1 N1(C(C2CN(C(C)=O)C2)=O)CCC(NC(=O)Cc2cnn(C(C)(C)C)c2)C1C c1(SC)ccsc1C(=O)NC(C)(C)CNC(=O)CC(C)C N1(C(Cn2cc(C(C)(C)OC)nn2)=O)CCCC(Cn2cc(CC(C)O)nn2)C1 CC(CC(C)(C)C)C(=O)NC1CC12CCN(C(c1ccc(Cl)cn1)=O)C2 C(CCCCCCCCC)(c1n(CC=C)nnn1)NCC(c1cccc(F)c1)(C)C CCCCC(C)C(=O)N1CCOC(CCCNC(c2sc(C)cc2Cl)=O)C1 c1(OC)ccc2ccc(=NCCOCCc3ccsc3)[nH]c2c1 N1(C(c2n(CC)ccc2)=O)CC(NC(=O)CCCc2ccsc2)CC(O)C1 N1(C(c2c(C)cccn2)=O)CC2(CCC(NC(C3CC3CN(C)C)=O)CC2)C1 CCCCCC(=O)NC1CC1CNC(=O)C(F)C(=O)OCC C1(O)(CNC(C2C3CCC23)=O)CCCN(C(c2ccccn2)=O)C1 c1(OC)ncccc1CNC(N1CCCC(C(C)(C)C)C1)=O N1(C(CC2CC3(CN(C(CC(CC)(C)C)=O)C3)C2)=O)CC2CC(C1)C2(C)C C=CCC(C(=O)NC1C=CCCC1C(=O)NCC=CCl)NC(C)=O CC1CCC(NC(=O)Cc2ccc(Cl)c(F)c2)CN1C(=O)CC1(C)CCCC1 C(=O)(C(C(C)C)C(C)C)NCC(CNC(Cc1nc(C(C)=O)sc1)=O)OC(C)=O Cc1cnccc1C(N1CC2C(CNC(c3cnc[nH]3)=O)C2C1)=O C1(C(N(CCC)CCNC(=O)CC2CCC3(CC3)CO2)=O)CCC2CC1C2(C)C N1(C(C(C(C)C)SC)=O)CC2(CCCC(CNC(=O)C(C)Cc3ccco3)O2)C1 c1(NC(CC(CC)NC(=O)COCC2CCCO2)=O)cc(OC)cc(F)c1 c1(OC)ccc(C(N2CCCN(C(C3CCCS3)=O)CC2)=O)cc1[N+](=O)[O-] C1(CCOC)(NC(C=CC=CCC)=O)CCN(C(C2(O)CC(C)(C)C2)=O)C1 C1(OC)CCC(CC(=O)NC2CN(C(=O)CN(C)C(N)=O)CC2C(F)(F)F)CC1 CCC(CC(=O)N(C)CCN(C)C(c1cnn(CC(F)(F)F)n1)=O)CC(C)C N1(C(C(C)(C)c2ccns2)=O)CC2CC(NC(=O)CC3CCCOC3)C1C2 c1(N(CC=O)CCNC(C2CCC(SCC)O2)C)cccc(C)c1C.OC N1(C(c2noc(CC)c2C)=O)CCN(C(c2cccc(F)c2)C)CC1C Cc1cc(F)ccc1C(N1CC(NC(C2CC2C#N)=O)C(C)(C)C1)=O C(=O)(CCCCCCCC1CC1)NC(C(C)C)(C)CNC(=O)CN(C)C1CC1 N1(C(C(C)=CC2CC2)=O)CCCC2(NC(=O)COc3cc(C)ccc3F)CC2C1 CCCCCC(CCCCC)C(=O)NCC1CN(C(=O)CC2=CCN(C)CC2)C1 C1(NC(c2ccc(C#C)o2)=O)CC2(C1)CC(C(=O)NCC1(O)CCC1)C2 C1N=C2C=C(C)NC(=NCc3ccccc31)N2.c1(CC)cc(CC)ccc1Cl c1(CC)nnc(C)o1.C1(C2(N(C(=O)C)C)CC2)CCCN1C(=O)CCn1ccnn1 N1(C(C(=O)NC(c2ccc(OC)cc2)C2CC2)=O)CCc2cncnc2CC1 CC1CC(C(=O)NCCC(C)(C)CNC(c2ccccc2C2CCOC2)=O)=NO1 c1(C(=O)NCC2CN(C(c3c(CC)n(C)nc3)=O)CC2C)cc(C)c(F)c(C)c1 c1(OCc2c(C(=O)Nc3scc(C(=O)NC)n3)nco2)cccc(C)c1 N1(C(C(Cn2ccnn2)NC(c2c(CC)cco2)=O)=O)CCCNC(=O)C1C N1(CCNC(c2c(CC)cno2)=O)CCCN(C(=O)CC2(C)CCCO2)CC1 C1(NC(C2(N(C(c3cnn(CC)c3C)=O)C3CC3)CCC2)=O)CCCC(O)CC1 c1(C(N2CCC(F)(CNC(=O)CC3CNC(=O)C3)C2)=O)cc(F)cc2nc[nH]c12 Cc1nc(C=CC(=O)NCC(C)(C)CNC(c2ncn(C(C)(C)C)n2)=O)[nH]c1C N1(CCC(=O)N(C(C)CNC(C2CCC2C(=O)OC(C)(C)C)=O)C2CC2)CCOCC1 N1(C(c2c(C(C)C)ccc(Br)c2)=O)CC2(CCCN2C(=O)C#CC2CC2)C1 C1(Nc2c(C)c(N3CCCOCC3)ncn2)CCN(CP(C)(C)=O)CC1 C1(SC)CC2CC(Cc3cnn(C)c3C(F)(F)F)C2C1 Cc1ccc(Cl)cc1C(=O)N(C1CN(C(C2(c3ccc(Cl)cc3)CCC2)=O)C1)C CN1CCC(C(=O)NCCc2ocnc2CNC(C2(CO)CCCO2)=O)C1 C1(NC(C2C(C(=O)NCC#C)C2)=O)CCOCC1NC(=O)CC1(C)CCCCC1 Cc1ccc2oc(C(N3CC4(CCN(C(=O)CN5CCCCC5)C4)C3)=O)cc2n1 C(=O)(C(F)(F)C(C)O)N1CC(CC(C)NC(c2c[nH]nc2Cl)=O)C1 C1(C(N(CC(O)CNC(C2CC2c2ccccc2)=O)C)=O)CC2C=CC1CC2 c1(CC(=O)NC2CCC(NC(C3(C#C)CCC3)=O)C2)c(C)cc(C)c(Br)c1C N1(C(c2ccn(CC)c2C)=O)CC2(CC(NC(C3CCS(=O)CC3)=O)CO2)C1 CCN=C(NCC(c1ccco1)N1CCCC1)N1CCC2C(C1)C2(F)F C(=O)(CC(C(F)(F)F)NC(c1cccc(OC)n1)=O)NCC(CC(=O)OC)O Cc1cccc(C)c1CNCC1(NC(=O)C(C)(CO)CO)COC1 Cc1cc(C(N2CCC(C)(C)C2CC(=O)NCCC2CC(F)C2)=O)nn1C N1(C(c2ccc(OC)cn2)=O)CCN(C(c2cncc(N)n2)=O)C2CCC12 N1(C(C(F)=CC)=O)CC(C)(C)CC1CNC(C1(c2cccc(Cl)c2F)CC1)=O C1(CNC(C(CC)N(C)C)=O)CCN(C(c2c(C)nn(C)c2C)=O)C12CCC2 C(=O)(C1=NOC(C2(O)COC2)C1)NC1CCC(NC(CC2(C=C)CCC2)=O)C1 Cc1ccc(Br)c(C(N2CCC(C(N3CCC(CO)C(O)C3)=O)C(O)C2)=O)c1F c1(-c2nc(CC)nn2-c2ccccc2OC)cc2scc(Br)c2[nH]1 N1(C(CCCCSC)=O)CC2CCC(C2)c2ccccc21 C1(C)(CNC(C(CC)=CC)=O)CN(C(c2cc(OC)nn2C)=O)C(C)(C)C1 C1(CC)COC(C)(C)CN1S(=O)(=O)CCc1cccc(F)c1 C1(COC)(NC(c2cnncc2C)=O)CCN(C(=O)CN(C)C)C1 C(=O)(CCCCC(F)F)N1CC2(CC(NC(c3cn(CCOC)nc3C)=O)C2)C1 c1(NC(C(=O)OCC)Cc2ccccc2)nc(-c2ccccc2)c2sccc2n1 C(=O)(CC(C)CNC(=O)CN(C)C(=O)C1CC1)NC.C1(CO)CCC1 Cc1ncc2n1CCC(C(=O)NC(C1CN(C(c3n[nH]c(=N)[nH]3)=O)CCO1)C)C2 C12(NC(CCc3c(C)ncs3)=O)CCOC(CNC(C3CCCSC3)=O)(C1)C2 Cc1ncncc1C(N1CC(F)CC1CC(=O)N(C1(CCO)CC1)C)=O N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CCCC(NC(=O)CCn2cc(Cl)cn2)C1 C(=O)(C(C(C)C)NC(C1CC(O)(CNC(c2cc(C(C)=O)on2)=O)C1)=O)OC N1(C(C=C(C)C(F)F)=O)CCC2(CCN(C(=O)C(C)(C)C(N)=O)C2)C1 CC(C)(C)CC1CC1C(=O)N(CCNC(C1(F)CC1)=O)CC1CC1 c1(C(=O)NCC(C2CCC2)NC(=O)CC2CCCC23CC3)cc(F)c(F)c(F)c1 c1(OC)ccc2ccccc2c1CCNC(c1cc(CN(C)C)on1)=O N1(CC(=O)NCC2CC2(Cl)Cl)CCCC(C(N2CCC2CO)=O)C1 C1(NC(C(CCC)C)=O)CN(C(c2cnncc2O)=O)CCC12CCOCC2 Cc1cc(CC(=O)NC2CC(C(C)NC(C3CCSCC3)=O)C2)n[nH]1 CC1(C)C2CCC1(C(N1CCC(C)(NC(c3ccn(CC(F)F)n3)=O)C1)=O)CC2 C1(NC(=O)NCC2N(C3(CC)CC3)CCC2)CCCCCC1 c1(C(=O)NC(C2CCN(C(CC(C)O)=O)CC2)C)ccn(CC(F)(F)F)c(=O)c1 c1(C(N2CCCC(NC(CS(C)(=O)=O)=O)CCC2)=O)ccnc2cc(F)cnc12 c1(CC(=O)NC2CCOCC2NC(c2ccc(Cl)nc2O)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NC2CCN(C(CCC(=C)C)=O)CC2CC)c(O)nnc2c1CCCC2 c1(C(=O)NCC(C)CNC(C2CC2Br)=O)nc(C(F)(F)F)n2c1CCCC2 C1(F)(C(=O)NC2CC(CCNC(C=CCCC=C(C)C)=O)C2)CC2(CCC2)C1 C1(C(N(CCC)CCO)=O)CN(C(=O)CC2CC3(CC3)C2)CC1C1CC1 N(C(=NCCCCl)NCCC1CCCCC1)C1CCC(CCC)CC1 Cc1nc2c(CC(=O)Nc3cc4n(n3)CCC4)cccc2o1 C(=O)(C(C)CCC(C)(C)C)N1CC2(N(C(C3CCC(CC)CC3)=O)CCC2)C1 c1(C(N2C(CN(C)C(c3coc(Cl)n3)=O)CCC2)=O)nn(C)cc1Cl N1(C(CCC(C)OC)=O)CCC(C(N2CCSCC2C)=O)(CC)CC1 C1(CC(=O)NC(C2CCOCC2)C#C)CC(NC(=O)C=CCCC)C1(C)C N1(C(c2c(CC)scc2)=O)CC2CCC1C2NC(=O)C(CO)OC C(C(CC(C)C)C(=O)NCC1(C(=O)NC(CCO)C2CCC2)CC=CC1)OC c1(C(=O)Nc2nn3ccc(C(=O)O)cc3c2)cccc(S(=O)(=O)C2CC2)c1 C1(O)(CNC(C=Cc2ccc(C(N(C)C)=O)cc2)=O)CCC(F)(F)CC1 C1(CCNC(C(C)=C2CCCC2)=O)CCN(C(=O)C(N2CCNC2=O)C)C1 N1(C(c2cnc(CC)s2)=O)CCN(C(C2CC(C(C)C)C2)=O)C2(CCC2)C1 N1(C(C(c2cnn(C)c2)C)=O)CCCC(O)(CNC(=O)CC=CC(C)(C)C)C1 c1(C(=O)NC2CC(NC(c3nccc(Cl)c3F)=O)C2)cc2cc(Br)ccc2s1 N1(C(C(CC#C)O)=O)CC(CC(=O)N(C2CCN(C)C2)C)CC1(C)C c1(-c2cc(C(N(CCNC(C3C(C)C3)=O)C)=O)no2)ccccc1Br N1(C(C(C(C)(C)C)NS(C)(=O)=O)=O)CC2CCN(C(C3CCC3)=O)C2C1 C1(CC)CN(C(=O)C(=Cc2c[nH]cn2)F)CCN1C(=O)C1=CCN(C)C1 c1(CC)cc(NC(=O)CC2CC(F)CN2C(=O)C(C)CN(C)C)cc(F)c1 C#CCC(C)(CC)C(=O)N1CC(O)(C(C)(C)CNC(=O)Cc2cccc(C)c2)C1 N1(CC)CCN(CC(=O)NC2CC(C)N(C(c3ccoc3Cl)=O)C2)CC1 N1(C(C(CCN(C)C)O)=O)CCC2CN(C(c3nocc3Cl)=O)CCC12 C1(N(C(C(CC)=CC)=O)C)CC2CCC(C1)N2C(C1CC(C(C)C)=NO1)=O CC(C)C(CCN(C(=O)C(C1CCCCC1)N(C)C)C)NC(=O)CC(C)(C)C C1(CNC(Cc2c(C)cccc2)=O)CN(C(=O)CC2CCSC2)C(C)(C)C1 N1(C(C(CC)COC)=O)CCN(C(=O)C2=NOCC2)C(C(C)(C)C)C1 N1(CC(=O)NCCC)CCC(CC(=O)NCC(c2cnn(C)c2)(C)O)C1 CCCS(=O)(=O)C(C)C(=O)N1CCN(C(=O)C=CC)CC1C(C)C N1(C(c2c(C)cccc2C)=O)CC(CNC(C2(C#N)CC2(C)C)=O)C2(CCC2)C1 N1(C(CC)=O)CCc2cc(CNC(=O)CC(C)N(C)C)ccc21.N12CCC1C2=O C(=O)(C1CCCc2ncccc21)N1C(CNC(C(C)CCO)=O)CC(F)(F)C1 Cc1[nH]nc2c1CCC(C(=O)NCC=C1CCN(C(=O)C(C)(C)C3CC3)CC1)C2 N1(C(C2N=C(C)SC2)=O)CCC2(CCN(C(=O)CC3CCCC(=O)N3)C2)C1 C1(N(C(C2CC(Cl)(Cl)C2)=O)CC)CCN(C(=O)CC2CCCCO2)CC1 CCCS(=O)(=O)CC(=O)NCC1CN(C)CCN1C(=O)CCCS(N)(=O)=O n1(CC(=O)NC(CC)CNC(C2COC(=O)N2)=O)cc(S(N)(=O)=O)cn1 C1(NC(c2[nH]cc(CC)c2)=O)CCC(C)(CNC(=O)C=Cc2sccc2C)CC1 c1(NC(=O)OCC)ccc(NC(=O)CNC(=O)NC(CSC)C(C)(C)C)c(F)c1 c1(CN(C)Cc2csc(-c3ccncc3)n2)nc(N(C)CCF)c2c(n1)COC2 N1(C(Cc2cc(C)on2)=O)CC2CC2(NC(=O)C(Cc2ccccc2)C2CC2)C1 c1(C(N(CCNC(C2CCCOC2C)=O)CC)=O)nccc2ncccc12 C(=O)(CC(C(F)(F)F)OC)NCC1CC(NC(C(C=C)OC)=O)CC1O c1(C(N2CC(CNC(CSCC#C)=O)C(O)C2)=O)ccc(N)c(Cl)c1 C1(CC(=O)NC(C2CCCCC2)C)CCCN1C(c1cc(C(F)(F)F)c[nH]1)=O N1(c2nn(CCN(C)C)c(=O)n2C)CCC2(CCCN2C(=O)OC(C)(C)C)C1 C12(C(=O)NCC(CNC(C(C)(C)SC)=O)OC)CCC(C#N)(CC1)CC2 CC(C)CCCC(C)C(=O)NCC1(CC(=O)N(C)CC2CC2C)CC1 c1(C(N2C3C(Nc4nc(CC)nc(C)c4)C(CC3)C2)=O)sc2cncn2c1C C1(CCN(C(C(=O)NCCC)C)C)CCN(C(=O)COC)C1 C1(=CC(=O)NCC(C)(CO)NC(c2cncnc2)=O)CN2CCC1CC2 C1(CNC(CCN(CCC)C)=O)CC(C(C)C)CCN1C(=O)C(CC)NC(C)=O O=S(CCc1nc(-c2c(F)ccc(F)c2Cl)no1)CC(F)(F)F c1(CC(=O)OC)nc(CNCC2CCCC2O)cs1 CC1(C)CCCOC1C(N1CCCC(CCNC(C2CCC=CCCC2)=O)C1)=O c1(OC(C)C)cc(C#N)ccc1CNC(=O)NC1(CF)CCCOCC1.C(C)(C)(C)O c1(CNC2C3CN(S(CC(=O)OCC)(=O)=O)CC32)cc2c(F)cccc2o1 C1(NC(C2C(NC(Cn3c(C)cc(C)n3)=O)CC2)=O)CCC(C2CC2)C1 C12(C(=O)OC3CCC(=O)NC3)CCC(CC1)OC2.c12ccccc1CN(C1CC1)C2=O Cc1coc(C(=O)N(C)CC2CCCN2C(=O)Cc2cccc(C(N)=O)c2)c1C N1(C(C(CC)C)=O)CCCC(CCCCNC(=O)Cc2ccc(C(C)=O)cc2)C1 C(=O)(C(O)C(C(C)C)OC)N1CC2C(CC(=O)NC3CCCC(C(=O)OC)C3)C2C1 Cc1cnc(NC2CCC(NC(=O)CC3CCCC3(F)F)CC2)nc1C c1(C(N2CC(O)(C(C(=O)NC(CCC)CC)F)C2)=O)cncc2[nH]ccc12 C(=O)(CC1CC(=O)c2ccccc21)N(C)CC1CCCN(C(C=CCC)=O)C1 c1(N2CCC(C#N)(NS(CC(C)C)(=O)=O)C2)ncnc2cccc(F)c12 c1(C(=O)NC(C2CCCN(C(=O)CNC(=O)C(C)(C)C)C2)C)cccc(Cl)c1Cl n1(C(C)C)ccnc1C(=O)NC1CCC(NC(C2CC(F)(CO)C2)=O)C1 N1(C(CC2CCCN(C(c3cnc(C)s3)=O)C2)=O)CCOC(C)(C)C1C N1(C(COCC(=C)C)=O)CC(O)CCC1C(N1CCOC(CC2CC2)C1)=O C1(CNC(CCCOCC=C)=O)CCC(C)(C)CN1C(c1cc(C#N)no1)=O C(=O)(CCCCN(C(=O)C(C)OC)C)NCC(C1CCCC1)OC CCCCN=C(NCc1ccc(C#N)cc1)N1CCC2(CC(C(F)F)=NO2)C1 CC(F)(F)C(Cl)CNC(=O)C(Cc1cn[nH]c1)NC(=O)COCCCF N1(C(=O)C(c2ccc(Cl)cc2F)O)CC2CCN(S(=O)(=O)c3nccs3)CC2C1 c1(C(C(=O)NCC2(F)CC(NC(=O)C=C3CCN(C)C3)C2)OC)ccccc1 c1(C(=O)NCC2(CNC(c3cnc(C(C)OC)s3)=O)CC2)ccc(O)c(F)c1F Nc1nc(Br)ccc1C(=O)NCC1CCCN1C(C12COCC1C2)=O Cn1ccnc1C(=O)NCc1n[nH]cc1C(=O)NCC1CC(CO)CO1 N1(C(C2CC(C#C)(O)C2)=O)CC2CCC2(CC(=O)N(CCC)CCN(C)C)C1 N1(C(C2(CC=C)CCC2)=O)CC(CNC(c2cc(CC)no2)=O)C(C)C1 c1(C(N(C)CCOc2cccc(F)c2)=O)cc(Cl)c(F)nn1 c1(OC)ccc(S(=O)(=O)N(C)C)c(NC(C2CC(=O)C2C(C)(C)C)=O)c1 N1(C(Cc2cc(C(C)C)no2)=O)CC2(CCCCN2C(=O)CN2CCSCC2)C1 N1(C(C(C2CCN(C(C3CCCN(C)C3)=O)CC2)C)=O)CCC2COCC2C1 N1(C(C2N(C(CNC(CCC)=O)=O)CC(C)C2)=O)CCC(O)C(O)C1 N1(C(C2N(C(C)=O)CCCC2)=O)CCCC2(NC(C3CCCC(C)O3)=O)CC2C1 c1(N2CCN(C(c3ccc(C)cc3O)=O)C3C2C3)ncc2[nH]ccc2n1 CCC(CC)(C(=O)NC1CN(C(=O)CC(C)(C)C)CC1c1ccccc1F)OC C(=O)(C1CC(=O)Nc2ccccc21)NCC(C)NC(c1ccc(C(F)F)cc1)=O CN1CC(C(=O)NCCOCCN(C)C(c2cnc(Cl)cn2)=O)C(C(F)(F)F)C1 S(=O)(=O)(c1cc2sc(C)nc2cc1Cl)NC1c2c(ccc(C)c2)OC1 c1(C(=O)NC2C(C)N(C(C3CCC3(F)F)=O)CC2)cc2c(s1)CCOC2 c1(C(C)OC)cc(S(=O)(=O)Oc2cccc(OC3CCNC3)c2)ccc1C C1(NC(C(CCC)NC(C)=O)=O)CCN(C(=O)CCN2CCCS2(=O)=O)C1(C)C Cc1nc2cccc(C(=O)NC(C)CC(C)NC(=O)CN3CC(C)(C)C3)n2n1 C1(C(=O)NCC(C)OC(F)F)CCC(C)N(C(=O)C(C)c2ccco2)C1 n1(CC)cc(CCNC(=O)C(c2cccs2)NC(C2CCC(=O)O2)=O)cn1 Cc1cc(CNC(=O)CCN(C(=O)C(C)CN(C)C)C2CC2)nn1C c1(C(N2C(C)CCC(CNC(CN(C)CC)=O)C2)=O)ccc(C)c2ccccc12 N1(C(C(CCC)(C)O)=O)CCCC2(NC(C3CCc4ccccc4C3)=O)CC2C1 c1(OC)ccnc(C(=O)NCC2CCN2C(C2CCC3CC3CC2)=O)c1OC Cc1cc(C(N2CCC(NC(=O)C(O)P(C)(C)=O)C2(C)C)=O)cc(=O)n1C CCCC(C)(CC)C(=O)NC1COCCN(C(C2CCCC2O)=O)C1 c1(OC)cc(NC(C2CCC(C)(C)OC2)=O)nc(C)c1 CC1(C)C2CCC1(C(=O)NCCNC(C1(C3CC3)CCOCC1)=O)CC2 c1(C(=O)NC(CCN(C(C2(CCOC)CCC2)=O)C)C)csc(C(F)F)n1 N1(C(N(C2C(C)OCC2)c2ccccc2)=O)CCc2nnc(N(C)C)cc2C1 C1(CCCNC(N(CCC)C)=O)CNCCO1 N1(C(Cc2nc(C(C)C)sc2)=O)CC(C)CCC1CNC(=O)CC1CS(=O)(=O)C1 C(=O)(C(C)(C)C(=O)NCC=CCC(=O)NCC(C)C(C)O)OC Cc1ncc(C(N2CC3C(NC(=O)C(C)N(C)C)C3C2)=O)cn1 Cn1ncc2cc(C(=O)NC3CC(NC(=O)C(O)CN4CCCC4)C3)sc12 c1(C(=O)NC2CC(C(=O)NCC3CCC(C)C3)CC2O)cnn(C)c1C#N C1(C(=O)NCC2(C)CCN(C(C=CC(C)(C)SC)=O)C2)CCCC12CCOCC2 C1(NC(C(C=CC)O)=O)C2CC3C1C3C2C(=O)NCC=CC=CC C1(C(=O)NCC(C)(C)CNC(=O)CC2CCCOCC2)CC2CCC1CC2 c1(C(C(C)C)NC(N2CC(c3ccc(C)cc3)(O)C2)=O)ccc(F)c(F)c1 C(=O)(C(CC(C)C)C(C)C)N1CC(CC=C)(C(N2CCC(C3CC3)C2)=O)C1 N1(C(C(c2cncnc2)C)=O)CC2CCC1C(CNC(c1cnc(N)cn1)=O)C2 C1(NC(C2COCCOC2)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 N1(NCc2c(OC(C)C(=O)O)cccc2)CC2CCCC(C(=O)O)(C1)C2(F)F c1(NCCC(C)C(F)F)cc(=NCC2CCSC2)[nH]cn1 N1(C(C(C)OC)=O)CCC(NC(c2cnn(-c3ccccc3)c2)=O)C1C(C)C N1(C(C(C)N(C)Cc2ccccc2)=O)CCC2(CCCN2C(=O)C2=NOCC2)C1 C(C(CO)(CO)NC(=O)CN1CCCC1C)N(C(c1cn(CC=C)nc1)=O)C Cc1nc(C(N2CCSCC2CCNC(C2OCC2(C)C)=O)=O)nn1C c1(CCC(=O)NC2CN(C(C=CCC)=O)CC(O)C2)c[nH]c2cc(C)ccc12 N1(C(C2CCCCC2)C)CCC(C(C)NCCC2CCCC2)C1 C1(C(=O)NC(CNC(C(CCC)c2ccccc2)=O)CC(C)C)CN(S(N)(=O)=O)C1 CC1CC2CN(C(=O)NC3CC3C3(C)COC3)CC2N1CCO c1(CC(N2CCC(O)(CNC(C3(F)CCCC3)=O)C2)=O)ccccc1OC(F)F N1(C(C2C(C=C)OCCC2)=O)CC(CNC(=O)CC(=O)NC2CC2)CC(C)(C)C1 N1(C(c2ccc(OC)cc2OC)=O)CC2(CCCC2NC(=O)CN(C)C2CC2)C1 CC1CCCN1CC(=O)NCCNC(C1CN(C(C2CCN2C(N)=O)=O)C1)=O c1(C(=O)OCC)cc(C)nn1CC(=O)NCC(Cc1ccco1)CO n1(CC(=O)N(C2CCCC(N)C2)C)c(SC(F)F)nc2ccccc12 N1(C(C(C)C#N)=O)CCN(CCNC(c2ccnn2CC2CCC2)=O)CC1 c1(C(=O)NCC(CC)NC(c2ccoc2)=O)cc2cc(OC)ccc2n1C N1(C(C)=O)CCCC1c1nc(CN(C(C)C(=O)O)C(c2ccccc2)C)no1 N1(C(CC2CC(C(=O)OCC)C2(C)C)=O)CCCCC(CNOCP(C)(C)=O)C1 CC1(C#CC(=O)NC2CN(C(=O)Cn3ccc(C(F)(F)F)n3)C(C)(C)C2)COC1 C1(CNC(=O)C=Cc2cc[nH]n2)CCC2CN(C(c3cn(CCO)nn3)=O)CC12 CCC(C)(C(=O)NCC1CN(C(=O)Cc2ccn(C(F)F)n2)CCN1C)C(N)=O c1(CC)ncccc1C(=O)NCc1nnn(C)c1C(N1CCC(CN(C)C)C1)=O C1(NC(CSC)=O)CN(C(c2cccnc2-n2nccn2)=O)CC1N=[N+]=[N-] N1(C(CCC=C)=O)CCN(C(=O)COc2cc(C)ccc2C)C(C)C1C c1(NC(C2CCC(NC(c3ccc(F)nc3)=O)C2)=O)cccc2[nH]ccc12 C1(CNC(C(C)Sc2nnnn2C2CC2)=O)CC2CCC1N(C(=O)C(C)(C)F)C2 c1(C(N2CCC(CC=C)(NC(=O)C(C)O)C2)=O)nc(Br)c2c(F)cccn12 C1(NC(c2nc(CNC(CN3C(C)CCC3)=O)oc2)=O)CCCCC12CC2 C1(N(C(CCNC(COC)=O)=O)C)CN(C(c2cnc(C(C)C)s2)=O)CC1F N1(C(C(n2c(C)ncc2)C)=O)CC(C2(NC(C3CC3C#N)=O)CC2)C1 O=C(CCCCN1CCCS1(=O)=O)NCc1ccccc1C1CCCC1 C1(F)(CNC(C2CCC(=O)N2)=O)CCCN(C(=O)Cc2ccncc2Cl)C1 N1(C(C2(N)C(C)(C)C2)=O)CCC(C)(O)C(O)C1 Cc1nc(C2CCC2)oc1C(=O)NCC1CC1NC(C12CCC(CC1)O2)=O N1(C(c2c(CC)ncs2)=O)CCN(C(=O)CCCC2CCCC(=O)N2)C(CC)C1 C12(C(=O)NC3CC(N(C)C)C3)CC(n3cc(C4CCCC4O)nn3)C1C2 Cc1cn2ccc(C(=O)NC3(CO)CN(C(C4CC5CCC5C4)=O)C3)cc2n1 c1(CC)oc(C)cc1C(=O)NC1CCC(N(C)C(c2cc(O)n(C)n2)=O)C1 c1(C(=O)NCc2c(C(=O)NC(C)CC3CCC3)nco2)cccnc1O c1(C(c2n(CC=C)nnn2)NCc2cnc(CC)s2)ccc2c(n1)CCC2 c1(C(=O)NC(C(C)(C)NC(CCCc2scc(C)n2)=O)C)cc(Cl)cc(C)c1C C1(C(N(C2CCN(C(CNC(C)=O)=O)C2)CCO)=O)CCC(NS(C)(=O)=O)CC1 c1(CNC(C(c2cnn(C)c2)NC(c2c(C)cccc2)C)=O)ncc(F)cc1F c1(C(=O)NC(CNC(CCCOCC=C)=O)CCOC)ccc(C)c([N+](=O)[O-])c1 c1(C(C)=O)cccc(C(=O)NC23CC(CNC(c4sncc4C)=O)(C2)C3)c1 Cc1cccc(C(C)C(=O)N2CC(OCCNC(c3nc(Cl)c(Cl)s3)=O)C2)c1 C1(C(=O)NC(C=C)C2CCC2)CC1C1CN(C(=O)CN=[N+]=[N-])C1 C(=O)(C1Cc2c(Cl)cccc21)OC.CCC1CC(=O)NCCC2CN(C2)C(=O)N1 c1(C2(C(=O)NCCC(=O)NCC=CCSC)CC2)ccncc1 Cn1nc2c(c1C(=O)NCc1ccc(Br)c(F)n1)CCCC2 CC1CN(C(=O)CC2CC(C(F)F)C2)CCC1N(C)C(c1cnc(C(F)F)s1)=O c1(OC(C(C=C)c2ccccc2)=O)ccc(Cl)cc1.C1(=O)C(=O)N(C2CC2)CC1=O.OC Cc1nn(CC(N2CC3C(NC(=O)C(C#N)C(C)C)C3C2)=O)cc1[N+](=O)[O-] Cc1ccc2ncc(C(=O)NCC3(F)CCN(C(=O)CCC4(C)CC4)C3)n2c1 C1(O)(CCNC(CC(CC)SC)=O)CCCN(C(c2ccc(N)cc2OC)=O)C1 C1(N(C)C(c2ccnn2CC#N)=O)CCC(NC(=O)CN2C(=O)CNC2=O)CC1 C(=O)(CC(C)(C(F)F)N(C)C)N(c1ncc(Br)cc1Cl)CC(C)C CCC(C#N)C(=O)NC1C=CCC(C(=O)NC2(CO)CC(F)C2)C1 c1(C(N(CCC)CCNC(=O)CC(C)(C)C)=O)cncc2c1CCNC2=O S(=O)(=O)(c1ccc(NC2CCOC2C2CC2)c(Br)c1)N(CCCCC)CCO Cc1cc(C(=O)NCC2CCN2CC=C(Cl)Cl)sc1C C1(NC(C(C)=C2CCCC2)=O)CC(F)CN(C(c2cnc(S)n2C)=O)C1 C(C(C(=O)N1CC(F)(CF)C1)n1cc(C2CC2)nn1)OCC.c12cc(no1)OC2 N1(C(COC2(C)CN(C(=O)CC3CCCOC3)C2)=O)CC23CCC2(COC3)C1 c1(C(N(C(C)C(=O)NC23CCCC2C3)CC)=O)ncn2ccccc12 CC(C)CC(C)C(=O)NC1CCCCC1CC(N1CC2CC1C2)=O N1(C(C(CC(C)C)C)=O)CC(C)CN(C(c2coc(S(C)(=O)=O)c2)=O)C(C)C1 CCC(CCC(=O)NCCC[Si](C)(C)C)NC(C1C2CCC(F)C12)=O Cc1nn(C)cc1CC(C)NC(c1ccc(OC(C)C)cc1)=O c1(C(=O)NC2(CC(=O)NCc3ccc(Cl)o3)CC2)cnc(CO)cn1 CC(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCN(C(C2CCN(C)C(=O)C2)=O)C1 c1(OC)ccc(F)cc1CC(=O)N(CC(O)CNC(C1CCCN1C(C)=O)=O)C c1(C(=O)NC2C(C)CCN(C(=O)CC3OCCC3C)C2)ccc2oc(=O)oc2c1 c1(C(=O)NC2CN(C(c3ncsc3C(F)(F)F)=O)C2)ncc2n1CCCC2 c1(C(N2CCN(C(C(C=C=C)C)=O)CC2)=O)ccnc2ccccc12 c1(C(N2CC(CCC=C)(C(=O)NC3CC(C)C3O)C2)=O)ccnc(C)c1 c1(NC(C2CC2CNC(C2(CCF)CC2)=O)=O)cc2c(C3CC3)cccc2[nH]1 Cn1cc(C=CC(=O)NCC(C)(C)C(=O)NCCn2ccnn2)cn1 c1(C(=O)NCC2(CNC(CC(C)C)=O)CC2)cc(F)cc([N+](=O)[O-])c1Br Cc1sc(C)c2sc(C(=O)NC(C)CC(C)NC(C3CCCN3C3CC3)=O)cc12 C(=O)(C(C)C(=O)OC)N1CC(CCNC(c2ccc(CSC(F)F)o2)=O)(OC)C1 C1(CC)CN(C(C2CN(C)C2)=O)CCC1NC(c1ncoc1-c1ccon1)=O c1(OC)ccccc1C(=O)NCC1(O)CCN(C(=O)CC2(C)CCOC2)C1 CC1(C)Oc2cc(C(=O)NC(CC(=O)c3ccsc3)C(=O)O)cnc2NC1=O C(CC(C(=O)NCC(C)SC)NC(c1nn(C)cc1Cl)=O)=CC c1(C(N2CCC(SC3(CC)CCC3)CC2)=O)ccc(C#N)cc1F C(=O)(C(CC1CCCC1)C(C)C)N1CC(CNC(Cc2c(C)n[nH]c2)=O)OCC1 C(N=c1[nH]c(=N)[nH]c(=NCC2CCCC(CO)CC2)[nH]1)c1ccc(F)c(C)c1F Cc1cncc(C(=O)NC2CCN(C(c3ccsn3)=O)CC2F)c1C C(=O)(CCS(=O)(=O)CC(C)C)N1CC2(CN(C(C(COC)OC)=O)C2)C(CO)C1 Cc1c(C(N2CCN(CCN(C)C(C3CCO3)=O)CC2)=O)cnn1CCC(C)C c1(OC)ccc(CNC2CCN(Cc3ccc(F)cc3O)CC2)c(C)c1C N1(C(C(C)(C)c2ccns2)=O)CC2(CCC2)OCC1C(=O)O C(=O)(C1CCCc2nccn21)N(CC(C)(C)CNC(c1ccc(F)cc1N)=O)C C1(C(N2CC3(CC(NC(C4(CCCC)CCC4)=O)C3)C2)=O)CC2(C1)CC21CCC1 Cc1nnc2c(C(N3CC=C(CNC(c4nsnc4O)=O)CC3)=O)cccn12 c1(C(N2C(CN(C(=O)CC3CCCN3C)C)CCC2)=O)ccc(-c2cccs2)o1 c1(CN2CC(C)CC(NC(=O)Nc3cc(C)cc(F)c3)C2)cccc2cc[nH]c12 c1(OC)cc(C(N2CCC(O)(CNC(c3ccnnc3)=O)C2)=O)ccc1F c1(C(N2CCC(C)(NC(C(C)SCCCCCC)=O)C2)=O)ccc(C)cc1CC Cc1cc(C(=O)NC(C)CC(C)NC(c2nnn3c2CSCC3)=O)cc(=O)n1C c1(OC)cc(C(=O)NC2CC(C)CN(C(c3ccc(O)c(Br)c3)=O)C2)ccc1Br C#CCCCCCC(=O)NC1CCCC1NC(=O)C(c1ccccc1Cl)(F)F O=C(CC(C(F)F)NC(=O)COCC1(O)CC(O)C1)NC1CCCC1 C(=O)(CCCC(=O)N(C)C)N1CC(C)C(NC(C2CCCN2c2nccs2)=O)C1 C1(C(=O)NC(C=C)C)CC2(CC2)CN1C(=O)COc1ccc(C)cc1 c1(C(C(=O)NC2CCCN(C(CN(CC)CC)=O)C2C)O)cccc2c1OCC2 c1(CC(=O)NC2CC(OCCOCc3cn[nH]c3)C2)ccc(C(F)F)cc1 c1(C(=O)NC(C2CCN(C(C(C)(C)OCC)=O)CC2)C)ccc2ccsc2c1 c1(C(=O)NC2(C)CN(C(C3C(CC)CCC3)=O)C2)cccc(Br)c1 Cn1nc(C(N2CC3CC2CC3NC(c2ccoc2Cl)=O)=O)ccc1=O c1(C(=O)NC(c2nocc2C(N2CCN(C)CC2)=O)C)ncccc1F CCCCCC(C)(C)C(=O)NC1CCOC(CNC(=O)C(C)CN(C)C)C1 c1(C(N(C2CCN(C(C3C4C5CCC(C5)C34)=O)C2)CC)=O)ccc2nc[nH]c2n1 c1(C(=O)OC)oc2ccccc2c1CNC(c1cc(Cl)ccc1F)(C)C(=O)O C1(C(N(C)CC2CN(C(C3CCC(CO)CC3)=O)CCO2)=O)CCC(N=[N+]=[N-])C1 c1(OC)ccc2cc(C(=O)NCC3(NC(C45CC(C)C4C5)=O)CC3)ncc2c1 c1(CNC(=O)NC(c2ccc(OCCCC)cc2)C)cc2ccncc2s1 CC1(C)C(C(=O)NCCC2NC(=O)NC2=O)CCN1C(c1n[nH]c(O)n1)=O CC1CCC(CNC(C2CCC(CF)C2)=O)N(C(=O)CN(C2CCCC2)C)C1 c1(C(N2CC(C(N)=O)(CNC(=O)C(c3cncn3C)O)C2)=O)cccn(O)c1=O N1(C(=O)CSCC(c2ccccc2)=O)CCCN(C(c2ccc(O)cc2)=O)CC1 c1(NC(C)CN2CCOCC2)[nH]c(=NCc2cc(C(N)=O)co2)nc2sccc12 C1(C(N(CC(C)(C)NC(=O)CCn2cnnn2)C)=O)CCC2(CC2)C1 N1(C(c2cnc(C)n2C)=O)CCN(C(C2C=CCC2)=O)C(C)C1 Cc1ccc(N2CCCC2)c(C(=O)NC(C)CNC(c2ccc(=O)oc2)=O)c1 CCCC(C)(O)C(=O)N1CCC(c2ccc(F)cc2)(NC(C2(F)CCCC2)=O)C1 N1(C(C2C(C=C)CC2)=O)CCC(NC(=O)CCCC)C12CCC2 N1(C(c2c[nH]c(=NC)o2)=O)CC(NC(c2ccc(C(C)(C)C)cc2)=O)CCC1C N1(C(C(CCCOC)C)=O)CC2CC1CCC2NC(=O)C=CC1(C)CCOCC1 c1(C(N2CCC(O)(CNC(=O)Cn3cnnn3)C2)=O)cccc2nc(O)ccc12 c1(NC(C2C(C(=O)NC(CCC)C(=O)N(C)C)C2)=O)cc(C)c(Br)cc1Cl c1(C(=O)NCCC2N(C(CNS(C)(=O)=O)=O)CCC2)cnc(O)n(C2CC2)c1=O c1(CC(=O)NC2(CNC(C(COC)O)=O)CC2)cccc(C)c1 C=CC(C)(CCOC)C(=O)NCC1CN(C(=O)Cc2cccs2)C2(CCC2)C1 C(C)(CNC(c1ncc(Br)cc1F)=O)(CC(C)C)NC(CSC)=O N1(C(C(COC)(C)O)=O)CC(C(=O)N(C)CC2CC2C)CC1(C)C CCC(O)C(F)(F)C(=O)NCC1CCCN1C(C1CC1C(N)=O)=O C(=O)(C1=C(C)CCCC1(C)C)NCC1N(C(C(CC)n2cncn2)=O)CCCC1C C(=O)(C1Cc2ccc(Cl)cc21)N(CC(C)NC(C(CC(=O)OCC)(C)C)=O)C c1(C(C)C)ccc(C(=O)NCC2CCN(C(C3(C)CCN(C)C3)=O)C2)nc1 N1(C(C(CC#C)C2CC2)=O)CCC2(CC(NC(C3(CC(=O)OC)CCC3)=O)C2)C1 c1(C(=O)NCC2(c3ccccc3)CC(NC(C3C(C)=C3)=O)C2)ccc(C)cc1 c1(SC)c(C(=O)NCC(C2CC2)N(C(=O)CC(C)O)C)ccc2c1OC(F)(F)O2 C1(N(C(c2c(C)ccs2)=O)C)CN(C(c2cc(C3CC3)oc2C2CC2)=O)CC1F CCCC(C)(C)CC(=O)N1CCC(F)(C(=O)Nc2cccc(CC)c2O)C1 C(=O)(C1=C(Cl)CCCC1)NC1(C(=O)NC(COC)C2CC2)CCCC1C c1(C(N)=O)ncn(CC(N2CC(CCNC(=O)Cn3ccnc3CC#N)C2)=O)n1 C1(NC(C)=O)CC(NC(C2CC(C(=O)OC(C)(C)C)C2(C)C)=O)C1(C)C CCCCC(C)C(=O)N1CCC(CN(C(c2cc(CO)on2)=O)C2CC2)C1 C(=O)(C1CCc2cccc(=O)n21)NCC=CCNC(CC1(C)OCCO1)=O N1(C(CC(CC)OC)=O)CCC2(NC(c3ccc(C(F)F)cc3Cl)=O)CCCC12 CC1CCc2[nH]c(=NCCCc3cnc[nH]3)[nH]c(=NCC(Cl)=CCl)c2C1 CC1(C)CCCc2c1n[nH]c2C(=O)NC(C)(CNC(C12CC(F)(C1)C2)=O)C1CC1 C1(C(=O)NCC(C)(CO)NC(CC(CC)SC)=O)CC(F)(F)C1(C)C Cc1ncc(Br)cc1C(=O)NC1CCN(C(C2CCCCC2)=O)CC1C C1(C(=O)NC(C)CCCNC(=O)C(=Cc2c[nH]cn2)F)CC1C1CCOCC1 C1(N(C(CSC)=O)CC2CC2)CCCN(C(=O)C(C(C)C)NC(N)=O)C1 n1(CC(=O)NCC(C)(CNC(c2cncc(C)c2)=O)OC)ccccc1=O c1(CC(=O)NCC(C)CNC(=O)Cn2cnc(C#N)n2)ccc(C(F)(F)F)cc1 CC1CC(CNC(c2csc(CO)n2)=O)CN1C(c1nn[nH]c1Cl)=O c1(C(N2C(C(=O)Nc3c(OCC)ncnc3)CC(F)C2)=O)cc(C)ccc1O C1(NC(c2c(C)cncn2)=O)CN(C(c2ccc(C(C)O)cc2)=O)CCC1O c1(C(=O)OC)cn2c(n1)CCC(c1nc(-c3ccc(Br)c(C)c3)no1)C2 c1(C(N2CC3(CN(C(C=CC)=O)C3)C2)=O)cc2ccc(Br)c(F)c2[nH]1 Cc1ccc(C#N)cc1C(=O)NCC1CC(NC(C2CC3CCC(C2)C3)=O)C1 CC(C)C(=O)C(=O)N(CC(=O)NCC(O)C1(Cl)CC1)C1CC1 S(=O)(=O)(c1ccc(NC(C)CC2CCC2)cc1Cl)C(CCCc1ccccn1)C.N C=C1CCC(C(=O)NC2CCCC2CNC(c2cnc(C(C)OC)s2)=O)CC1 C#Cc1ccc(CC(=O)NCCC(C)(C)CNC(c2c[nH]ccc2=O)=O)c(F)c1 Cc1cccc2oc(N3CC4CC(NC(=O)C5=NOC(C)C5)CC4C3)nc12 N1(C(C2CNC(=O)N2)=O)CCCCC(CNC(c2n[nH]cc2C2CCC2)=O)C1 O=C1CC(C(=O)N2CC(NC(c3ccccc3Cl)=O)CC2CO)=NN1 C1(C(=O)NCCc2c(C(=O)Nc3cc(C)no3)c[nH]n2)CCCCC(=O)N1 Cc1cc2ccccc2n1CC(=O)NC1CC2CCC(C1)N2CC1CC1 C1(C(=O)NCC=Cc2cccnc2)(CC)CCCN1C(C1CC(N(C)C)C1)=O CC1(Cn2cc(CC3CN(C(C4CCCCC4)=O)C3)nn2)CCCC1(F)F N1(C(c2nn(CC)c(O)c2)=O)CCN(C)C(C(=O)NCC(C)CC(=O)OC)C1 c12cc(C)c(cn1)c(=O)[nH]2.c1(N(CC(CC)(OC)OC)CC)ccnc(CO)n1 C1(NC(=O)COCCCF)CCCC1CC(=O)NCC1CCC(=O)O1 C1(CNC(C(C)OCC#C)=O)OCCC1C(=O)N(C)CCc1ccccn1 C1(c2ccc(OC)cc2)C(n2cc(COC(N)=O)nn2)CCC(=O)N1C CCCCC(C(=O)N1CCCC1(CNC(c1cnc(C)s1)=O)COC)C(C)C N1(C(C2N(C(Cc3cn(CC)nc3)=O)CC=C2)=O)CCCC(F)C1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NCC(CNC(CCC(C)(C)[N+](=O)[O-])=O)O c1(C(N2CC(CNC(c3cnc(C(C)=O)s3)=O)C2)=O)cccc2cncn12 C12=CN=C(SC)NC1=NC1CCCC1C(=O)N2.c1(COC)ccc(Br)cc1C CN1CCC(C(=O)NCC2CN(C(N)=O)C2)(NC(=O)CCC2CCOC2)C1 C1(C(=O)Nc2ccc(NC(CCOC)=O)cc2C)C2CSCC1CC(N)C2 N1(C(CSCC)=O)CC(OC)CC(NC=O)C1.c1(C2(C(=O)OC)CC2)ccccc1F Cc1c(C(N2CC3CC(C2)N(C(=O)C(C)C(C)(C)O)C3)=O)sc2ccc(Cl)cc12 c1(CC(=O)NC2C3CN(C(CCCCC)=O)C2C3)cnc2c(C)cccn12 c1(C(=O)NC(C(C)(C)NC(CSCC=C)=O)C)ccc(-c2cccs2)nc1C C1(C(=O)NCCCCCN(C)CC2CC2)CN(C)CCN1C(=O)C(=O)NC1CC1 C1(C(N2CCCN(C(C=Cc3c(C)n(C)nc3)=O)CC2)=O)CNC(=O)CC1(C)C C(CCCCCN(C)C(c1ncsc1Br)=O)NC(C1CCC(C)S1)=O Cc1cc(C(N2CC(=C(F)CNC(=O)Cc3cn[nH]c3)C2)=O)c(O)nc1C C=CC(O)(C(=O)NCC(CNC(c1ccc(Cl)cc1)=O)CO)C(F)(F)F C1(CNC(c2cnc(C(C)(C)C)o2)=O)(CO)CCN(C(=O)CC2CC(F)(F)C2)C1 C1(SC)CCCC1C(=O)NCC(c1ccccc1)NC(c1cnsc1C)=O c1(C(=O)NC2(CCNC(=O)OC(C)(C)C)CCOC2)nccc(N)c1Cl c1(C(C(=O)NCC(CN(C(C2SCCS2)=O)CC)(C)C)C)ccccc1OC c1(CC(N2CCCC(N(C(=O)COCC(F)F)C(C)OC)C2)=O)ccc(Cl)c(Cl)c1 S(=O)(=O)(c1nc[nH]c1Br)NC(CCC)(N)C(=O)O N1(C(c2c[nH]c(=NC)o2)=O)C(CNC(=O)CC2CC=CCC2)CC2CCCC12 CC1CCCC1(C(N1CCC1CN=[N+]=[N-])=O)NC(C1CC(=O)C1)=O c1(OC)ccc(CNC(C2(c3ccccc3)CC2(F)F)=O)cc1OC(F)F c1(C(C)C)ncccc1NC(C1CCC1NC(=O)C1=CCSC1)=O CC#CC1CCN(CCNC(=O)Cc2scnc2C)CC1 Cc1onc(CC(=O)NC2(C)CN(C(C3CCC3C(N)=O)=O)C2)c1C#N Cc1cc(Cl)c(Cl)cc1CN1CC2C(NC(c3cc[nH]n3)=O)C2C1 c1(C(C(=O)OC)NC(c2nc(=O)n(C3CC3)[nH]2)=O)ccc(F)c(C)c1 C=CC(CCC)CC(=O)NC(CCC(=O)NCC1CCCCCC1)C(C)C C1(CC(=O)NC2(CN(C(CCOCCCOC)=O)C)CC2)CC2C=CC1CC2 c1(NC(c2ncn(C(C)(C)C)c2)=O)cc(Cl)c(Br)cc1[N+](=O)[O-] CN1C(=O)c2ccccc2C1C(=O)N1CC2CC(NC(c3occc3F)=O)C1C2 C1(C(=O)NCC2N(C(CC(C(C)C)(F)F)=O)CCC2)CC12CCc1ccccc12 C12(C(=O)N(C)CCSC)CCC(CC1)C2.c1(C(=O)OC)n[nH]cc1CNC(=O)C1CC1 C1(O)(CC(=O)NCC=CCNC(C(C)CC2CCC2)=O)COC(C)(C)C1 C(C(C(=O)NCCC(C)(C)O)C(C)(C)C)NC(c1n(CC)ccc1)=O CCCCCC(C(=O)NCC(c1ccccc1)NC(=O)CCOCC)C(C)C c1(C(=O)NC2CCN(C(CCc3cc(C)on3)=O)CC2F)cc2cccnc2s1 Cc1ccc(C(=O)NCC2CC2)c(O)c1.C12(CCCO1)C(=O)NCC1(CC1)NC2=O C(CC(O)CNC(=O)CCOCCN(C)C(C1CN(C)C1)=O)OC C1(NC(C(C2CN(C(=O)CC3CC(C)(C)C3)C2)OC)=O)CC(C)(CO)C1 S(=O)(=O)(c1cn(C)nc1C)N1C(c2scc(C)n2)COCC1 c1(C(N2CC3C(C(N4CCC(N(C)C)C4)=O)(C3)C2)=O)ccc(Br)c(Cl)c1F c1(CNCC23C(CN(C(c4c(C)cc(Br)cn4)=O)C2)C3)cccc([N+](=O)[O-])c1 C1(C(=O)NCC2(CCC)CC2)CN(C(C23CSCC2C3)=O)CC1(C)C c1(C(C)(C)N(C(=O)CN2CCC(N3CC=CC3)C2)CC)cc(C)c(C)cc1C C(=O)(CC(C)C(F)F)NCC(CCCC)NC(C1CCCN(CC)C1)=O c1(C(=O)NC2C3CC2N(C(=O)Cc2cnnn2C2CC2)C3)cccn2nccc12 C12(C(N3CC(NC(C(C)CN4CCOCC4)=O)C3)=O)CCCCC1NC(=O)C2 Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)(C)CCNC(=O)C=C1CC1 C(=O)(C(COC)C(F)(F)F)NCCC1CC(NC(C(CCC)O)=O)C1 N1(C(CC2C=CC(NC(C=CC3(C)COC3)=O)C2)=O)CCCCC(CO)C1 Cc1cccc(C(C)C(=O)NC2C3CN(C(C4CC=CC4)=O)CC23)c1 N1(C(CSC(C)C)=O)CCN(C(C2CCCSC2C)=O)CC(C)C1 c1(C(=O)NCC2(CC(=O)OCC)CCCCC2)ccc2c(n1)OCC(=O)N2 c1(CC(=O)N(CCN(C(C2(C=C)CC2)=O)C(C)C)C)c(F)cccc1C#N C(=O)(C(=O)C(C)CC)NCCCCC(=O)NC1(CC=C)CCOC1 c12ccc-1c(C)n2.c1(C2N(C(CNC(C)=O)=O)CCC2)cccc(F)c1 c1(C(=O)OCC)ccc(=NCCNC2CCN(C)C(C(=O)O)CC2)[nH]c1 N1(CCCC=C(C)C)CCC2C(C1)NC(=O)CCN2C C1(C)(CC(=O)NC(C(C)NC(c2cnns2)=O)C)CCCO1 O=C(C1OCCn2ccnc21)NC1(CO)CCN(C(c2ccccn2)=O)C1 c1(C(=O)NCC2C3CN(C(c4n(C)nc(Cl)c4)=O)CC32)cnn2ccncc12 C1(OC)CCNC1=O.C1(C)(C(=O)OCCNS(=O)(=O)C2CC2)CCC(=O)C1 C1(NC(CC(=O)NCC)=O)CCOC12CCN(C(c1cc(Cl)ncc1F)=O)CC2 C1(NC(CC(CC)O)=O)CCCCN(C(=O)C(c2ccccc2)N(C)CC)C1 c1(C(=O)NC2C(CNc3nccc(OC)n3)CCCC2)c(Cl)c([N+](=O)[O-])nn1C N1(C(=O)C=Cc2cn[nH]c2)CCC2(CNC(C3(CF)CCC3)=O)CCCCC12 N1(CCC)CCCCC1c1nc(Oc2ccccc2)nn1-c1ccccc1SC C(C(C)(O)CC(=O)N1CCC(C(=O)NC2CCCC2C(N)=O)C1C(C)C)OC C1(NC(C2(C#C)CC2)=O)CN(C(c2c(Cl)csc2Cl)=O)CCC1C(F)(F)F CN1CCN(c2ccnc(C(N3CC4(CC(NCCN(C)C)C4)C3)=O)n2)CC1=O c1(C(N2CCC(CNC(C3(CN)C(C(=O)OC)C3)=O)CC2)=O)ccc(C)cc1F C12(CNC(C3N(C)CCOC3)=O)CC(C1)C(NC(=O)CN1C(=O)CCC1=O)CO2 Cc1cccn2c(C(N3CCN(C(=O)Cc4cnoc4)CC3C(C)C)=O)cnc12 c1(C(N2CCC(CN(C(=O)C(F)(F)CO)C)CC2)=O)ccc(F)c(N)c1 C(=O)(C(F)C(C)C(F)(F)F)NCC1(C)CCN(C(C(C)SCC)=O)C1 CN1CCCC(CNC(c2coc(CNC(C3CC3F)=O)n2)=O)C1 N1(C(C2N(C(C(CC)C#N)=O)CC(OC)C2)=O)Cc2cccc(C#N)c2C1 n1(CC)cnc(C(N2CC(C(C)NC(=O)CCn3ccc(C)n3)C2)=O)n1 C1(C(N2CCN(CCNC(C3(C4(O)CCC4)CC3)=O)CC2)=O)CC2C=CCC(C1)C2 C=CCCCCC(=O)N1CCC(CNC(C2CC23CCCCC3)=O)C1 C=CCC(C)(C)C(=O)NCCN1CCN(C(=O)CNC(c2n[nH]c(C)n2)=O)CC1 CCC(C)C(C(=O)NCCCN(C(C12CC(CC(C)O1)C2)=O)C(C)C)NC(C)=O c1(C(N2C(C(C)C)C(NC(=O)C=CCO)CC2)=O)cc(=O)c2ccccc2o1 c12nc(C)c(s1)c(=O)[nH]2.Cc1ncc(CC(=O)NC2CC(C(N)=O)C2)s1 Cc1c(C(N2CC(CC(C)NC(=O)C(C)CO)C2)=O)cnn1CC(F)F c1(C(N(C2CCC(NC(=O)C=C3CCC3)CC2)C)=O)cccc(C(F)F)c1 CC(C)C(C(C)NC(=O)CSc1nc[nH]n1)NC(=O)COc1ccc(Cl)cc1 C1(CCC)CN(C(=O)CC2CC3CC3C2)CCN1C(c1cc(C)ccc1C)=O C1(NC(c2ccn(C)c2)=O)CN(C(c2cncc(-n3ccnc3)n2)=O)CC12CCC2 N1(C(C(CCCC)O)=O)CC2CCC(C1)N2c1cc(C)nc(Cl)n1 C1(c2ncn(C)n2)CCCCN1C(=O)N(CC(c1ccc(Br)cc1)(C)C)CCO C1(NC(CC2CC(C(=O)OC)C2)=O)CCCCN(C(c2cc(C)co2)=O)C1 c1(C(N2C(COC)CN(C(=O)C(C)N(C)C)CC2)=O)cn(C)c(=O)c2cncn12 C1(NC(c2ncc(C)s2)=O)CC2(CCN(C(C3CCC(CO)CC3)=O)C2)C1 c1(CC(N2CCC(NC(C3CCCC3)=O)C2)=O)ccc2c(c1)CCCO2 C(C(C(C)(C)C)NC(=O)C(C1CC1)C1CC1)NC(c1c(C)[nH]cc1)=O Cc1c(C(=O)NC2CC2CNC(=O)CC2CCC2)[nH]ccc1=O N1(C(C2N(CC)CCC2)=O)CCC2(CC1)CC2C(=O)NCC1(O)CCC1 N1(C(C2N(C(c3c(C)noc3N)=O)C(C)C2)=O)CCN2CCCCC1C2 Cc1[nH]nc2c(C(N3CCC(NC(C4CCCOC4)=O)C(F)C3)=O)cccc12 C(CCCC(=O)NC1(C(=O)NCC2COC(C)(C)C2)CCOCC1)N(C)C N(C1CCCc2cccc(C)c21)C(=O)NC(COC(C)C)C C1(NC(C(CC)N(C)C)=O)CC(C)N(C(c2csc(Cl)c2OC)=O)C1 n1(CC)ccc2nc(N)ncc12.c1(NC(C2(N(C)C)COC2)=O)cnccc1C n1(CC)ccc2nc(N3CCC(NC(C4(C#N)CC4)=O)C(O)C3)ncc12 N1(C(CCC(CC)CC)=O)CC2(C1)CN(C(=O)Cc1sc(C)nc1C)CC2CO N1(C(=O)NC(C)C=CCc2ccccc2)CCCN(CC(O)C(F)(F)F)CC1 C(C(=O)NCC1COCCN1C(=O)C(=O)C(C)(C)C)(C(C)(C)C)N(C)C C(=O)(CCCCC(N)=O)NCC(C)CN(C)C(C1CC2CC1CC2O)=O N1(C(C2CC(C)CC(C)C2)=O)CCCC(O)(CNC(=O)CC2(O)CCC2)CC1 C1(C(=O)NC2CC(CNC(C3(C#C)CCCC3)=O)C2)CC1C1CC(F)(F)C1 C1(N(C)C)CCN(C(c2cnc(C(C)(C)C#N)s2)C(=O)NC2CC2)CC1 c1(-c2ccnc(N(CC(C)C)CCC#N)n2)nc2cncnc2nc1O c1(C(N2CCC(NC(c3nc(CC)sc3)=O)C(F)C2)=O)c(C)ccc(C)c1C c1(C(=O)NCC(CC(F)(F)F)NC(C(CSC)C)=O)nc2ccccc2[nH]c1=O C(C(O)C(F)(F)C(F)(F)F)NC(Cc1c(C)cc(Br)cc1)=O c1(OC)cc(C(=O)NC(C2CCN(C(c3ccccc3F)=O)C2)C)ccc1Cl C(=O)(CCCCCN=[N+]=[N-])NCCOCCNC(CC(C(=O)O)OC)=O.C(C)(C)(C)OCC N1(C(CCCCC#C)=O)CCCC12CCN(C(=O)C(CO)c1ccccc1)C2 N1(C(=O)COCCc2ccc(Cl)s2)CCN(C(C2CCCC2C(F)F)=O)CC1 c1(C(=O)NCC2CN(C(C(C)NC(N)=O)=O)CC2O)ccc2cc(O)ccc2n1 c1(CC)ccc(C(=O)NC2CCN(CCCNC(=O)C(O)C(F)(F)F)C2)c(C)n1 c1(OC)cc(Br)ccc1CN1CCC2(CC1)CC2C(=O)NCCN1CCCCC1 c1(C(=O)NCC2CN(C(C3C(C)=CCS3)=O)CC2O)cc(C)n(C2CC2)c1C c1(C2(C(=O)NCC3C(NC(c4coc(Cl)n4)=O)C3)CCC2)cccc(F)c1 C1(C)(NC(C2CC(NC(C(CC3CC3)OC)=O)C2)=O)CCC(C)C1 C1(NC(=O)CCF)CN(C(c2ccnc3ccsc23)=O)C2(CCCOC2)C1 c1(NC(CCC)CC)ncccc1S(=O)(=O)N(c1c(CN)cc(Br)cc1)C.N(C)C N1(C(c2ccc(OCC=C)cc2)=O)CCCN(C(=O)C=NOC)CC1C c1(CCC(=O)NCC2C(NC(C(C(C)C)(C)O)=O)C2)ccc2c(c1)CC(=O)N2 CC(C)(O)C(F)C(=O)NCCOCCCNC(C1CCS1(=O)=O)=O Cc1cn2ccc(C(N3CC(NC(c4cc(Cl)cnc4C)=O)C(C)C3)=O)cc2n1 c1(OC)ccc(C(N2CCC3(CC3NC(c3nccnc3C)=O)C2)=O)c(F)c1 C(CCC(=O)NO)NC(C(C1CCCN(C(=O)CC2NC(=O)NC2=O)C1)C)=O c1(C(C)CNC2CC(c3ccccc3)CO2)ccc(F)c(F)c1 c1(C(=O)OCC(c2ccccc2SC)NC(CC)COC)c(C)noc1C(F)F n1(CC)ncc(CN(C=O)CC2(CCF)CCC2)c1C n1(C(C)C)ccc(=NC(=O)C2(C)CCCN(C(c3ccc4c(c3)CC4)=O)C2)[nH]1 N1(C(C(C)SCC)=O)CCCCC1CCC1CCCN1C(c1n[nH]cc1CC)=O c1(C(=O)NC(CN(C(C(CCC#C)O)=O)C)C)cc(Br)cc(C)c1C c1(C(NOCCC=C)=O)ccc2c(n1)CN(C(C1CCC(OC)CC1)=O)CC2 c1(C(N(CCNC(Cn2c(C)nnn2)=O)C)=O)ccc(O)c(CO)c1 C(=O)(C(O)C(C)(C)C)NC(CC=C)CNC(c1cccc(CC=C(C)C)c1)=O c1(C(C(F)(F)F)OC(C=CCOC)=O)ccccc1F C(CCCCC(=O)N(C1CCCC(NC(c2cn(C)c(=O)n2C)=O)C1)C)OCC C1(NC(CC(CCC)O)=O)CN(C(c2cc(C(N)=O)cc(F)c2)=O)CCC1(C)C c1(CN2CCC(C(C(=O)OC)C)C(OC)C2)c(C)cc(C)nc1OC N1(C(C2C(=C)CC2)=O)CCC(C2CC2)C1CNC(c1ccc(C)c(Cl)c1F)=O C1(OCC)COCCC1Cc1nc(-c2ccn(C)n2)nn1-c1ccc(Br)nc1 c1(CC)cc(-c2nc(CN3CCCCCC3)nn2CC2CC2)c(C)o1 N1(C(CN(C(=O)C(CC)CC)c2snc(CCC)n2)=O)CCN(C(C)=O)CC1.CCS N1(C(CCn2ncc(C)c2)=O)CCC(c2ccc(Br)cn2)CC1 CC1CN(C(=O)COc2ccc(Cl)cc2)CC1CNC(C1C=CC=CC=C1)=O N1(C(C(CC#C)CC#C)=O)CCC2CN(C(=O)CCN(C)CC)CC2C1 CN=c1nc(N2CC3C4C=CC(C4)C3(C)C2)[nH]c(=NCC2(C)CC=CCC2)[nH]1 C1(CNC(c2c(CCC)occ2)=O)COCCN(C(c2cscc2C)=O)C1 Cc1ccc(C(=O)NCCCCC(C)NC(c2nncs2)=O)c(N=[N+]=[N-])c1 CC(C)CC(CCO)NC(Cc1nnnn1C)C1CC1 CCCCCCC(F)C(=O)NCCN1CCCN(C(=O)COc2nccs2)CC1 N1(c2cc(CCC)ncn2)CCC(O)(C(=O)N(CC(C2CCCC2)OC)C)CC1 c1(CN2CC3C(NC(c4cnc(C)nc4)=O)C3C2)ccc(Br)cc1O c1(C(CC(=O)O)NC(C(CC)NC(N)=O)=O)cccc(Br)c1 CCC(CC(C)C)C(=O)NCC1CCN(C(C23CC(COC)(CO2)C3)=O)C1(C)C N1(C(C(CCOC)NC(C(CC#C)O)=O)=O)CC2(COC(C)C2)C1 CC(C(CO)NC(=O)Cn1cncn1)NC(c1cc(-c2ccccn2)no1)=O N1(C(C(C)C2CCC2)=O)CC2CCCC1(CNC(c1ccn(C)c(=O)c1)=O)C2 c1(CC(=O)NCC(CNC(C2C(C)CN(C)C2)=O)(C)C)coc2cc(O)ccc12 C(=O)(C(C(CC)CC)OC)NCC(CNC(c1cc(CC)nnc1C)=O)(C)F C1(N(C(C2CC2(C)C)=O)CC)CCN(C(=O)CCc2ccc(O)nc2)CC1 n1(CC)ncc(I)c1C(=O)NC(c1ccc(Br)cc1)CC(=O)O c1(C(=O)NC23CC(CNC(COC(CC)(C)C)=O)(C2)C3)cnc(O)c(F)c1 C(C(CNC(C1CCCS(=O)(=O)C1)=O)C(F)(F)F)NC(CC(=O)OC)=O N1(C(C(C)n2ccnc2)=O)CC2CC(NC(=O)COCc3ccncc3)C(C2)C1 c1(CC(=O)OCC(=O)N(CCCC)C)c(C)n[nH]c1C Cc1ncc(NC(C2CCC(C)CN2C(C2CC3CC(=O)C2C3)=O)=O)cc1C#N C1(C(=O)NC2C(C(=O)NC(C(N)=O)c3ccco3)CCOC2)CCCC12CCC2 C(CC(C)C)(C(N)=O)NC(C1(COC)C=CCN1C(=O)CC1OCCO1)=O C(=O)(C#CC1CCOC1)NC(C)(C)CCCCNC(=O)CC1(C)CCOC1 C1(c2cccs2)(C(=O)NC(CN(C(=O)C(C(C)C)SC)CC)C)CCOCC1 C1(C(=O)OCC)C2CC1N(C(C1(C(C)C)CC1C(=O)O)=O)C2.C(C)(C)(C)O CCC(C)(C)C(=O)NCCCOC1CCN(C(c2cn(CC3CC3)nn2)=O)CC1 CCC(CCCC(=O)OC)NC(=O)C(CNC(=O)COc1ccccc1C)OC c1(C(=O)NCC=CCNC(C(C)OCc2ccc(C)cc2)=O)cc(N)c(Cl)cn1 C(=O)(C(C)(C)C(=O)NC)NC1CC(n2cc(C(CC)(C)O)nn2)C1 CC(C)CCCC(=O)N1CCCCC1C1(NC(=O)COc2ccccc2F)CC1 C(=O)(C(=O)N=S(C)(C)=O)OCC1C(C)(C)N(c2nc(OC(C)(C)C)ns2)CC1 c1(OC)ccc(SCSC(C)C(=O)Nn2cc(CCC3CCCC3)nn2)cc1 Cc1cc(CCC(=O)NCCCCNC(=O)C(=C2CCCCC2)F)cc(C)c1 C(=O)(CCCn1cc(C2(NC(C3(C(F)F)CC(O)C3)=O)CCC2)nn1)OC C1(C(=O)NCC(C)NC(=O)COC(F)F)CC2(C1)CC2F C1(N(c2ccc(C(=O)OC)c(Cl)c2)C(=O)CN(C)C)CCC12CCNCC2 C1(NC(C(c2cccc(C)c2)O)=O)CCC2CN(C(C3CCC(F)C3)=O)CC2C1 C1(NC(c2ccc(CC)c(Cl)c2)=O)CCC2(CCCN(C(=O)CC(F)(F)F)C2)C1 C=CCC(CNC(C1(c2ccccc2)CC1)=O)C(=O)NCC(C)OC C1(C(=O)NC2CCCC2N(C)C)(CC)CCN(C(=O)COCC(C)(C)C)CC1 CC(CC(F)F)CS(=O)(=O)NCc1cn(C(C)(C)C)c(=O)nc1O CC(O)C(F)(F)C(=O)NCC(C)(C)CNC(C1(F)CCCOC1)=O N1(S(CC(N2C3CCN(C=O)C3CCC2)=O)(=O)=O)CC2CC(C1)CS(=O)(=O)C2.CO N1(C(CC2(OCC)CCC2)=O)CCC2CC1CN2C(=O)CCCCCCSC c1(C(=O)NC2CN(C(CN(C(C)C)C)=O)CC2(C)C)cc2c(cc1N)CCCC2 C1(CC(=O)NCCCCSCC)CCCN(C(=O)CC(=O)OC(C)(C)C)CC1 C12(CNC(C3(CC=C)CCCN3C(=O)CCCC3CCC3)=O)COC(C1)C(O)C2 CC1(NC(=O)C=Cc2ccccc2)CCCCC1C(=O)NC1CCC(=O)NC1=O C(C)(C)(CCCCC(=O)NCC(C(C)C)NC(c1cnc(O)c(F)c1)=O)OC C(=O)(C1=CCCS1)N(C1CCC(NC(=O)Cc2cc(Cl)sc2Cl)C1)C CCCCC(C)CCC(=O)NC1CCCC(CNC(c2ocnc2C(C)C)=O)C1 C1(CCC)CN(C(c2cccc(=O)o2)=O)CC1NC(C1CC1C1CC1)=O N1(C(CSCC(=O)OC)=O)CCCC(O)(CNC(=O)CCc2ccccn2)CC1 c1(OC)ccnc(OC)c1C(N1CCC(NC(C2CCC(C(N)=O)O2)=O)CC1)=O Cc1nc(C#N)ccc1C(N1CCC(NC(C2CC23CC3)=O)C(C)(C)C1)=O c1(CC)cccc(C(=O)NC2CC3C(NC(c4cscc4C(F)F)=O)C3C2)c1F Cc1cc(CC(=O)NCc2ncoc2C2CN(C(c3sccc3Cl)=O)C2)no1 N12CC3=C(C1)CN(C3)C(=O)CNC(=O)C=CC2=O.c1(NC2CC2)nccs1 c1(C(=O)NCCCCC(C)NC(C2OCCN(C)C2=O)=O)ncn2c1CCCC2 c1(OCC(=O)NC2(C)CC(NC(c3csnn3)=O)C2)cc(F)ccc1F N1(C(CS(C)(=O)=O)=O)CC(CO)C2(C1)CN(C(c1cccc(CCO)c1)=O)C2 CCCS(=O)(=O)C(C)C(=O)NCC1CCCN1C(c1cc2nc(C)ccc2o1)=O CS(=O)c1ccc(C(N2CC(C)(C)C2CO)C(=O)NCc2ccco2)cc1 C(=O)(C(C)C(C)NC(=O)C(n1cc(-c2ncccc2F)nn1)C)OCC C1(CCP(C)(C)=O)CCN(c2nccc(C(F)F)n2)CC1 C(=O)(C(F)CC(C)(C)C)NCCCC1OCCN(C(c2n(C(C)C)ccc2)=O)C1 c1(C(C(c2cccc(F)c2Cl)C#N)=O)ccc2c(c1)OCC2 N1(C(c2c(C)scc2)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)C2CCC12 c1(NC(CC2CC(NC(c3nccc(C)c3)=O)C2)=O)cc(F)c(F)c(F)c1Br Cc1cc([N+](=O)[O-])c(C(N2CCC2CNC(=O)NCc2ccc[nH]2)=O)cc1F CN=c1nc(N2CC3CCC3(OC(C)C)C2)[nH]c(=NCC(F)F)[nH]1 CCCC(C(=O)N1CCC(N(C(c2ocnc2CC)=O)CC)CC1)C(C)C c1(OCCCOC(CC(C)n2ccnc2)=O)cccc(C2CCC2)c1 C12(CNC(c3nc(C)sc3C)=O)CN(C(=O)Cn3cccn3)CC1(C(F)(F)F)C2 C1(NC(C(C)N(C)C(C23CC(C)(CCO2)C3)=O)=O)CCCC(C2CC2)C1 C12(C(CNC(c3n[nH]cc3F)=O)NC(Cc3ccc(C)s3)=O)CCC(CC1)C2 N1(Cc2cccc(NC(=O)CCOC(F)(F)F)c2)CCS(=O)(=O)CC1 C(=O)(C#CC1CCC1)N1CC(OC)(CNC(=O)C(=O)NCC(F)F)C1 C1(NC(CCC(N)=O)=O)CN(C(c2snc(Cl)c2Cl)=O)CC(F)(F)C1 C1(CNC(C2(C)CCOC2)=O)CCCCN(C(=O)Cc2ccc(O)cc2)C1 C(CC(=O)N(C)CC1CCN(C)CC1)(C(C)(C)C)NC(C(CC1CCC1)OC)=O C1(C(CN)OCC)CC(F)(F)C1.C1C(OC)CC(=O)N1 c1(C(N(C(=O)OC(C)(C)C)CCN2CCCS2(=O)=O)=O)cccc(C(C)(C)C)n1 c1(C(N2C(CNC(C(CC=CC)C)=O)CC(F)C2)=O)nnc(O)nc1O N1(C(c2c(OC)nc(C)cc2)=O)CC2CCC1C1CN(Cc3ccccn3)CC21 C1(NC(C(CC=C)C)=O)CC2CCC1CN2C(=O)C1=CC(C)(C)C1 N1(C(CCc2ccc(C)c(F)c2)=O)CC(CO)C2(CCC2)C1 C1(C(=O)NC2CC(F)(CNC(CC3C(COC)C3)=O)C2)CCS(=O)(=O)C1 c1(C(=O)NCC(C)N(C(=O)CC(C)SC)CC)cnc(O)c(C(C)=NO)c1 c1(OC)cc(C(=O)NC(c2ccccc2)CNC(=O)C(C)(C)C#N)ccc1Br c1(C(N(CCCCCCNC(CC(CC)C)=O)C)=O)nc(C)ccc1C c1(OC)ccc(C(C)(C)CNCC2CCCCN2C2COC2)cc1 c1(CC(N2CCN(C(c3noc(C(C)CC)n3)=O)CC2)=O)cc(C)ccc1C C1(CC)CN(C(=O)CCC2CC2CC2CC2)CCN1C(=O)C(=O)NOC O=C(O)C#CC(=O)NC1CCC(CC(N2CCOCC2c2ccccc2)=O)CC1 Cc1cc(CCNC(c2ccccc2OC2CC2)=O)c(O)c(Br)c1 N1(C(C2(COC)CN(C(=O)C(C)c3ccco3)C2)=O)CCS(=O)(=O)CC1 N1(CC(=O)N(c2cn(CCCC)nn2)C(C)C)CC(Cc2ccc(C)s2)C(C)C1 n1(CCC(N2CC(C)(NC(c3c(C)cc(C)o3)=O)C2)=O)nc(O)c2c1CCCC2 N1(C2CN(C(c3c(C)n[nH]c3)=O)C2)CC(NC(C2CCC(=O)NC2)=O)CC1=O C#CC12CCN(C1)C2=O.C1(NC(=O)Cc2ncoc2C)C2CC3C1C3C2C(N)=O C=CC(C)(CCOC)C(=O)NC1CCCC(NC(=O)CCCC(=O)NCC)C1 c1(C(=O)NC(C)(CNC(=O)Cc2cnc[nH]2)C2CC2)cc2cnc(Cl)cc2s1 c1(-c2nc(CC)oc2)nc(Cc2cccs2)nn1C1COC(C)(C)C1 c1(C(=O)NC(CC)CN(C(=O)CCc2c(C)noc2Cl)C)nccc(Cl)c1C c1(N(CCC=C)C)nnc(N2CCC(C(=O)NCC=C)CC2)n1CCCNC N1(C(C(c2ccccc2F)OC)=O)CC=CC(NC(=O)C=C2CCN(C)CC2)C1 C(=O)(C1=C(F)CN(C(=O)C(C)CCCC(C)C)CC1)NCc1cnc(C)o1 N1(C(C2(CC=C)CCOC2)=O)CC(O)CC1C(=O)NC1CC(C)(CC)C1 Cc1nc(CCC(=O)NCC2(O)CN(C(=O)Cc3c(C)cnn3C)C2)oc1C N1(C(CCC(C)=O)=O)CCCC(F)(C(=O)N(C(C)C)Cc2ccoc2)C1 N1(C(CC)=O)CCCC(NC(c2ccnc(N(C)C)c2)=O)C1C C1(NC(c2c(C)occ2)=O)CCC(NC(c2cn(C(C)C)nc2C2CC2)=O)CC1 CCCS(=O)(=O)C(C)C(=O)NC(C)CCCCNC(c1scc2c1OCCO2)=O N1(C(c2nc(OC)oc2)=O)CCC2(C1)CN(C(c1c(C)n[nH]c1C)=O)CC(C)O2 C(c1cocn1)=CC(N1CC(CC(F)C(=O)N2CC(C3CCCCC3)C2)C1)=O c1(CNC(C2C(C)C(=O)C2)=O)ccccc1CN(C(=O)COC1CCC1)C C1(N(C(C(c2cccs2)SC)=O)C)CCCN(C(=O)CC2CC2)C1 N1(C(C2CCN(C(CCNC(C)=O)=O)CC2O)=O)CC(C)N(C)C(C)C1 C(=O)(C1=CCCSC1)NC1C(NC(=O)CCOc2ccc(F)c(Cl)c2)C1 N1(CCC)CCC(c2cn(C3CN(C(c4cc(C)co4)=O)CC3O)nn2)CC1 c1(C(C(=O)NCC)N(C)CC2CC23CC3(F)F)cc(CC)ccc1OC N1(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CC2(CC(NCc3cc(Cl)ccc3O)C2)C1 CCC(C#N)C(=O)NC1CCCC(CNC(=O)Cn2nccn2)C1 c1(OC)ccc(F)c(C(C(=O)NC2CCCCC2)N(C2CCCC2)C)n1 Cc1ccc(C=CC(N2CC(O)(CCNC(C3CC3C(F)(F)F)=O)C2)=O)o1 C1(C)(N(C)CC)CCN(C(=O)CC2CCCN(C(=O)C(C)C3CC3)C2)C1 C1(C(=O)NCCCCCNC(C(C)(C)c2cccs2)=O)CCCC(C2CC2)O1 c1(C(N2CCOCC(C(N3CCCNCC3)=O)C2)=O)ccc2cncnc2c1 C=CC1CN(C(c2ccc(F)cc2Cl)=O)CC1NC(=O)CN(CC(C)(C)C)C CC1CN(C(C2(S(C)(=O)=O)CC2)=O)CC1(C)CNC(=O)CCOc1cccnc1 C1(NC(C(CN(CC)CC)F)=O)CCN(C(=O)Cn2ncnn2)C(C)C1 C1(CNC(c2ncn(C(C)C)c2)=O)COCCN1C(c1cccc(Br)c1)=O Cc1cc(C(=O)NCCN(C(=O)CCc2cc(C)on2)CC(C)O)nc(O)n1 Nc1cc(C(=O)N(CCCNC(=O)CC2CC2C2CC2)C2CC2)ccc1Cl CC1CC1C1CC1COC(=O)C(F)CC1CCOC1 N1(C(C2C(C)C2)=O)CCOCC1CNC(C1(C(C)(C)O)CCC1)=O C1(N(C(CCCSC)=O)C)CCN(C(c2cnn(C)n2)=O)CC1C N1(C(CC2(OC)CN(C(C3CC4CCC3CC4)=O)C2)=O)CCCC(CO)(OC)C1 C1(NC(=O)CC2CC=CC2)CCCCC12CCN(C(c1c[nH]nc1C1CC1)=O)C2 CC1CC=C(C(=O)NCCC2(CNC(C3CCSC(C)C3)=O)CC2)CC1 c1(CCC(=O)NCC2(NC(COC(C)C)=O)CCCC2)ccccc1C(F)(F)F CC1CCC(NC(c2coc(C3CC3)n2)=O)CN1C(=O)CC1OCCO1 N1(C(c2c(C)ncc(C)c2)=O)CCOC2(CCN(C(=O)C(C)(O)C3CC3)CC2)C1 Cc1cc(C(N2CCOCC2CNC(=O)CSCC(C)C)=O)c(N)c(Cl)n1 c1(OC)c(F)ccc(F)c1C(N1CCN(C(C2CC2C2CCCC2)=O)C(C)C1)=O c1(CN(C(COC)C)C(C2CC(O)CN2C2CCN(C)CC2)=O)ccc(C)cc1 c1(OC)c(C)cc(C(N2CCC(NC(c3sccc3F)=O)C2)=O)cc1C c1(C(N2C(C)C(NC(C3CCCSC3)=O)CC2)=O)ccc2c(=O)ccoc2c1 N1(C(c2cc(CC)sn2)=O)CCCOC(CNC(c2nccnc2C(N)=O)=O)C1 C(=O)(CCCC(F)F)N1C(C(C)NC(C(n2ccc(C)n2)C)=O)CCC1 N1(C(C(CC)OC)=O)CCCC(C)(C)C1CNC(C1CC2C=CC1CC2)=O CC(C)C(CCNC(=O)CC(O)c1cnc[nH]1)NC(=O)CCCC1CC1 c1(C(=O)NC(C(=O)NC(CCC)C2CC2)c2ccco2)cnn2c1CCC2 c1(SCC)ccccc1CC(=O)N(CC(O)CN(C(=O)C(C1CC1)SC)C)C CCC(CCCC(=O)N1CC(O)C(N=[N+]=[N-])C1)NC(=O)CSC C1(C(=O)NCC(C)NC(=O)Cn2cc(P(C)(C)=O)cn2)C2CCC(C2)S1(=O)=O N1(C(c2cc(CNC(C(C=C)C)=O)oc2)=O)CC(F)(F)C1C1CC1 Cc1c(C(=O)NC2CCCN(C(=O)C3CC3)C2C)cccc1C(F)(F)F C1(CNC(CCN(C)C)=O)CN(C(=O)CN(C)C(c2ccsc2)=O)CCO1 c1(C(C(N2CCC(CNC(COC(CC)C)=O)C2)=O)C)ccc(F)cc1 C1(NC(C(=C(C)C2CC2)F)=O)CCC(NC(=O)Cc2ccc(C3CC3)cc2)CC1 C1(NC(c2ccc(Cl)cn2)=O)CC2CC1CN(C(C1CCOC1)=O)C2 N1(C(C(F)OC)=O)CC(NC(C2C=CC=CC=C2)=O)CC12CCCC2 c1(C(N2CC(CC)C(NC(=O)C(C)(C)COC(C)C)C2)=O)cc(Cl)c(F)cc1O c1(OC)ccc(C(=O)NCC(F)CNC(=O)C(C)OC)c(Br)n1 C(N=c1[nH]c2c(c(=NCc3ccc(C(N)=O)o3)[nH]1)COCC2)C1CC(C)OCC1 S(=O)(=O)(c1[nH]c(=NCCC(N)=O)ccc1Br)C(N1CCC(c2cccc(F)c2)C1)C N1(C(c2c(Cl)cn(C)n2)=O)CCC2(CCCN(C(=O)CCc3ncnn3C)C2)C1 c1(CCC(=O)OC)ccc(F)c(F)c1F.C12COC(C1)NC(=O)C2 C(=O)(CCN(OC)C(=O)Cc1cccc(C#N)c1)NC1C(OCC)COC1 N1(CC)CCCC(C(=O)NC2(CCC(N3CCCC3C3CC3)=O)CCOCC2)C1 CC(C(=O)NC(C)(C)CNC(c1cc2ccc(Cl)cc2o1)=O)C(C)C(C)(C)C c1(C(N2C(C3CCN(C(c4nc(O)n[nH]4)=O)C3)CCC2)=O)c(Cl)nsc1Cl C(=O)(C(C)(O)CC(C)C)NC(CCC)CC(N1CCC(CC)C(OC)C1)=O c1(-c2cc(OCC)c(OC)cc2OC)cccc2cc(C(=O)N(C)C)[nH]c12 Nc1cc(F)c(Cl)cc1C(=O)NCCCNC(C1(n2cnnn2)CC1)=O C1(C(N(C(c2ncc[nH]2)(C)C)C)=O)CCC(C2CCCCC2)CN1 c1(C(=O)NCC2CC3(CN(C(C(CC)O)=O)C3)C2)cc2cc(Cl)cnc2o1 c1(C(=O)NCC2(C)C(NC(C=CCC)=O)CCC2)cccc2nc(Cl)cn12 C1(NC(Cc2nc(C)sc2C)=O)CN(C(=O)C(C#N)=CC(C)C)CCC1O N1(c2nc(C)c(F)cn2)CCC2(CC1)CC(C(=O)N=c1cco[nH]1)CO2 Cc1cc(C(=O)NC(C2(CNC(C3(F)CCCOC3)=O)CC2)C)ccn1 C1(NC(c2cnc(OC)nc2)=O)CN(C(c2cn(C)cn2)=O)CCC1CO N1(C(CCC=CC)=O)CC(NC(=O)Cc2ccc3c(c2)CC3)CC(C)(C)C1 N1(C(c2cccc(SC)n2)=O)CCCC(C2CC2NC(C2CCCN(C)C2)=O)C1 c1(OC)cncc(C(=O)NCC=CCNC(=O)CCCc2csc(C)n2)c1C CCN=C(NCCCOC1CCOC1)N1CCC(C(O)C(F)(F)F)CC1 N1(C(Cc2nnc(C)o2)=O)CCCC2(CCCCC2NC(=O)C2=NOC(C)C2)C1 N1(C(C(C)C)=O)CCCCC1C1CCCN1C(c1c[nH]c(=O)c2ccnn12)=O C1(C(=O)NC2CN(C(CCC(C)(C)F)=O)C2)CC2(CCCCO2)C1 C=CC(CC)CC(=O)N(c1ncc(F)cn1)Cc1ccc(F)cc1 NS(=O)(=O)c1cc(C(c2ccc3noc(-c4ccccc4)c3c2)=O)c(F)cc1Cl CCC(C)(C)C(O)C(=O)N(CCC(C(C)C)NC(c1ccc(N)cc1C)=O)C C1(NC(Cc2nnc(C)o2)=O)CC2CC(NC(c3cncc(N)c3)=O)C1C2 c1(Nc2cccc(C(=O)Oc3ccc(OC)cc3)c2)cc(C)cc2cn(C)nc12 C1(C#N)(C(N2CC(CN(C(=O)CC3COC(C)(C)C3)C)OCC2)=O)CCOCC1 C(CC(CC)(CC)NC(c1ccc(-c2ccccc2)[nH]1)=O)NC(C(C=C)O)=O Cc1cn2c(n1)C(C(=O)N1CCC(C)(NC(=O)C(C(C)C)C(C)C)C1)CCC2 c1(C(CC)C)ccc(NS(=O)(=O)NN2CCN(C3(C(N)=O)CNC3)CC2)cc1 C1(C)(C(=O)NCC2(C)CCN(C(=O)CCCF)CC2)CC2CCC(C1)S2 c1(C(N(C2CCN(C(CCCC=C)=O)CC2)CC2CC2)=O)cn2c(n1)SCC2 N1(C(c2cnc(OC)s2)=O)CC2CCC2(CCNC(C2(C(N)=O)CC2)=O)C1 c1(C(=O)Nc2cccc(NC(C3CCC3(F)F)=O)c2)cccc(F)c1Br C1(C)(CNC(C2(CC#C)CC2)=O)CCN(C(=O)C(C)Oc2ccc(Cl)cc2)C1 C(=O)(CC(C)NC(C1CC1c1csc(Br)c1)=O)N(CC)CC C(CC(=O)NCc1cc(C)on1)(C(F)(F)F)NC(C(CCOC)C)=O CCCCC(O)C(=O)NC(CNC(=O)CCc1ccc(F)c(F)c1)CC(C)OC N(C(=NCCc1cccnc1OCC(F)F)NCCC(F)F)C(c1cccs1)C C=C1Cn2c(C(=O)NC(CN(C)C(C3CC4CCC3C4)=O)(CO)CO)nnc2S1 CC1CCCN(C(=O)C(=O)NC2CN(C(=O)Cc3c[nH]nc3O)CC2C(F)F)C1 c1(C(N2CCCC(NC(c3c(C)ncn3C)=O)C2)=O)ccc(N)c(F)c1Br C=C1CC2(C1)CC(C(=O)N(CCCOCCNC(c1cnc(O)cc1C)=O)C)C2 S(=O)(=O)(c1ccc(NCC23CCC(CC2)O3)c(C#N)c1)N(CCC)CC CC1CCN(C(=O)Cc2cc(Br)cs2)CC1CNC(C1OCCO1)=O Cc1cn2cccc(C(=O)N(C)CCN(C(=O)CCNC(=O)CO)C)c2n1 N1(C(COCCCCCC)=O)CC2CN(C(=O)Cc3cncs3)CC2(C)C1 N1(C(CC(CCC)(C)C)=O)CCC2(CNC(c3ncc(C)cn3)=O)CCCCC12 C1(C(N2C(C(N3CC(O)(CCC)C3)=O)C=CC2)=O)CSCC(=O)N1 CC(C)CC(C(=O)NC(C)C(C)(C)C(=O)NCC1CC(=O)N(C)C1=O)C(C)C CC1CC(NC(c2cnc3sccn23)=O)CCN1C(=O)CCc1cn[nH]c1 Cc1onc(Br)c1C(N1CCOC(CCCNC(c2cn[nH]c2)=O)C1)=O C1(C)(CNC(=NCC)NC2CCCC(SCC)C2)CCC(F)(F)CC1 c1(C(=O)NC(C)C(C)NC(=O)Cc2ccccc2O)cccnc1O c1(C(N(C2CCN(C(C3CCCN3C3CC3)=O)C2)CCC)=O)cc(F)c[nH]1 C1(C(N2CC(C)(NC(c3ccsc3)=O)C2)=O)COc2c(F)cc(F)cc2C1 Cc1ccnc(C(N2CCC2(C)CC(=O)NCC(C)(O)CCO)=O)c1N N1(C(C(=O)NCCCC(=O)OCC)C2CC(CC)C2)CCC2NC(=O)NCC2C1 c1(C(CN(C(=O)C(CNC(C2(O)CCCC2)=O)N(C)C)C)O)ccccc1 Cc1ncncc1C(N1CCC(NC(=O)COC2CCN(C)CC2)C1C)=O c1(C(N2C(C)CC(CNC(c3c(CC)[nH]cc3)=O)C2)=O)nc2n(c1Cl)CCCC2 c1(SCC(=O)NCC2(CO)CN(C(C(C)SC(C)C)=O)C2)ccc(F)c(F)c1 c1(C(=O)NCCCCC(C)NC(C(CC=C)CC=C)=O)cnc2c(c1)CCCC2 c1(OC)cc(C(N2CC(NC(=O)CCOC3CCC3)C(C)C2)=O)ncn1 c1(C(=O)NC(CC)(CNC(c2cc(C)ns2)=O)CC)c(C)cccc1Cl N1(C(C(C2CCC(=O)N2)C)=O)CC(C(=O)NOC2CCOC2)C(C2CC2)C1 C1(NC(CC2CC(=C)C2)=O)CCC(O)CN(C(c2ccn3nnnc3c2)=O)C1 CC1(CC(N2CCCC2CNC(=O)C(O)Cc2ccccc2)=O)CC1(F)F N1(C(c2c(CC)cno2)=O)CCN(C(=O)CC2CCCOCC2)CC1CCOC N1(C(C=C(C)Cl)=O)C2CCC1CN(C(c1nn(-c3ccc(F)cc3)cc1C)=O)C2 c1(C(=O)NCCOCCNC(C23C(C)(C)OC(CC2)C3)=O)ccc(Cl)c(N)c1Cl c1(OCC)cccc(CC(N2CCC(C)(NC(C3CCS3(=O)=O)=O)C2)=O)n1 C1(CC(N2C(C(N3C(C)(CC(=O)NC)CC3)=O)CCC2)=O)CCC(=O)C1C Cc1nc2cc(C(=O)NCC3CC(O)(CNC(=O)CN4CCCCC4)C3)[nH]c2s1 CN1CCN(C(C2CCC(NC(=O)CC3CCOC3)CC2)=O)CC1(C)C N1(C(C(CNC(CCCC=C)=O)N(C)C)=O)CCC(C)(C#N)C1 c1(C(CC)C)cc(C(N2CCC2CNC(c2ccnn2C(F)F)=O)=O)on1 c1(C(C)(C(=O)N2CCC(CNC(c3nc(Cl)cs3)=O)C2)N(C)C)ccccc1Cl N1(C(C=CS(C)=O)=O)CCC2(CCC(CNC(c3coc(CO)c3)=O)CC2)CC1 c1(C(=O)NCC2CCCCN2Cc2cccc(Cl)c2F)nccc2[nH]ccc12 c1(C(N2CC(CC(C)NC(c3n(CCOCC)ncc3)=O)C2)=O)ccncc1C Cc1cccc(C)c1CC(=O)NC1COCC1CNC(C12CC(C)(C1)C2)=O c1(C(=O)NCC2CC(C)N(C(=O)C3=CC(C)(C)C3)C2)ccc2occc2n1 N1(C(C2C(CCC)C2)=O)CCCCC2C1CCCN2C(c1ccco1)=O.C1CC1.O C1(CNC(CC2(C=C)CCC2)=O)CCCCN1C(C1(C)CCC1)=O C(=O)(C1=CCCN(C(C2CC(=C3CCC3)C2)=O)C1)N(CC(C)(C)OC)C c1(C(=O)OCC)ccc(CNC2CC2C(=O)NC(=O)CC2C(=O)NN=C2C)cc1 c1(C(c2nnnn2C)Nc2cc(C)c(Cl)cc2)ncc2ccccn12 C1(CC(=O)NCC(C)NC(C2(C=C)CCC2)=O)CC(C)(C)C(=O)N1 Cc1ccn(CC(=O)NCCCCC(CO)NC(=O)C(F)OC(F)(F)F)c(=O)c1 C#CCCC(C(=O)NCCC(C)(C)OCC)NC(=O)C=Cc1ccco1 c1(C(N2CC(NC(C#CC(C)C)=O)C(C)CC2)=O)cc(Cl)c(C)c(Br)c1 C(CCC(C)CC(=O)NCCC(C(C)C)NC(c1cn(C2CC2)cn1)=O)=C(C)C c1(C(=O)NCC2CN(C(=O)CCC=CBr)CCO2)cnc2ccccn12 c1(OCC)cnc(C(=O)N(CC(C)(C)CNC(=O)C(C)OCC)CC)cn1 c1(NC(C2C3(CN(C(CC(C)C)=O)C3)C2)=O)cn2nc(Cl)ccc2n1 C(C(C)C)(C(O)C(=O)N1CCCC(CC(N2CC(OC)CC23CCC3)=O)C1)OC CC1CCN(C(=O)C(C)Cn2ccnc2)CCN1C(=O)CC1(O)CCOC1 c1(CN2C(CCC(N3CCC(OC)CC3)=O)CCC2)cc(Br)cc(F)c1C c1(C(N2C(CC(=O)NC(CC)CO)CCC2)=O)cc(Cl)ccc1Br n1(CCSC)nnnc1C(c1n[nH]cc1C)NCC1CCCC1 N1(C(C(C(C)C)(C)C)=O)CCC2(CC1)CN(C(C1(C3CC3)CCCO1)=O)CCO2 c1(CCC)cc(C(=O)NCc2nocc2C(=O)NC(C)CC2CCCO2)no1 c1(CSC)noc(CCC(=O)N(C(C2CN(C(C3CCCO3)=O)C2)C)CCC)n1 CC1CCCN(C(=O)C(C)OCCOc2ccccc2)C1CNC(=O)C=CCF c1(C(=O)NC2CN(C(C(C(C)C)=O)=O)CC(F)(F)C2)cc2n[nH]cc2cc1Cl CCCCC(C(=O)N1CCCC1C(C)NC(c1cccc(C)n1)=O)N(C)C C1(C)(CNC(C2N(C(C)=O)CCC2)=O)CCN(C(C23CC(C#N)(C2)C3)=O)C1 N1(C(C2(C)C(C)C2)=O)CC(C2CCN(C(C3CCCC34CCC4)=O)CC2)C1 CC(CCNC(=O)CCc1cccnc1)CCNC(c1cnoc1C1CC1)=O C1=C(C)C(=O)NCC(=O)NC(C)(C)C1.C1(CC(=O)OC)(OC)CCC1 c1(NC(C2C=CCN(C(CSc3c(C)cccc3)=O)C2)=O)cccc(Cl)c1C c1(C(=O)NC(C)C(c2ccccc2)NC(=O)C=CBr)ccc2c(n1)NCCO2 C1(C(C)(C)CNC(=O)Cc2cccnc2)CCCCN1C(c1ccnc(O)c1)=O c1(C(=O)NC2C(C(N3CC(CC)OCC3)=O)CCC2)cc2[nH]ccc2cc1Cl CC1(C(=O)NCCN(C2CCCC2)C(=O)COCC2CCCOC2)CC(=O)C1 C1(NCc2c(C(=O)OC)ccs2)CCC(F)CC1.N12CCCC1CCCNCC2 c1(C(=O)NCCOCCCNC(C(C)CNC(N)=O)=O)ncnc2c1CCCC2 C1(C(=O)NC(CNC(CCC#C)=O)(C)C2CC2)CCC=CCCC1 c1(OC)cccc(NC(C2CC2NC(c2cc(Br)cc(F)c2O)=O)=O)c1C#N c1(N(C)CC2CCCN(C(=O)CC3CC3C3CC3)C2)ccc2ncnn2c1 N1(C(C(CC)C#N)=O)CC2OCCN(C(c3cccs3)=O)C2C1 C(=O)(CP(C)(C)=O)N1C(Cc2cn(CC(C)O)nn2)CCC1 O=C(CCCCNC(=O)COc1ccccc1)NCC(O)C1CC1 N1(C(C(C=C)O)=O)CC(OC)C(NC(=O)Cc2csc(-c3cccnc3)n2)C1 N1(C(c2cc(C)n(CC)c2C)=O)CC2CC1CN(C(c1scnc1Cl)=O)C2 C(CCCOC)(C(=O)NCc1cscc1C)NC(C(C(=O)OCC)F)=O C1(NC(=O)NCC2CCCOCC2)CC12CCOCC2 Cc1cc(S(N)(=O)=O)cc(C(=O)NC(C)CNC(=O)C(C2(O)CCCC2)F)c1C CCC(C)C(O)C(=O)NCC1=CCN(c2nnc(C)c(C)n2)CC1 c1(CCC(N2CC(NC(C3C(CC)CCCC3)=O)C2)=O)ccc(Br)c(Cl)c1 N1(C(C(CCOC)OC)=O)CC2(CC(C(=O)NCCS(C)(=N)=O)CO2)C1 C1(C(=O)NCc2c(Br)ccc(OC)n2)CC12CCN(Cc1cc(C)nn1C)CC2 c1(CC(C)NC(C2(N)CC(OC)C2)=O)ccccc1[N+](=O)[O-] C1(NC(CC(=C=C)C)=O)CCN(C(=O)C(C)NC(C)=O)CC(C)(C)C1 N1(C(CSC)=O)CCC2(CCC(NC(=O)COC3CCN(C)CC3)C2)CC1 C1(CC(N2CC(O)(CCNC(c3cc(OCC)n[nH]3)=O)C2)=O)CCN(C)CC1 C1(C(=O)Nc2c(C)cc(O)nc2)C2CCCC2CN1C(c1ccc(Cl)s1)=O CCCCS(=O)(=O)CC(=O)NC(CNC(=O)C(C)C(C)(C)C)CO C(=O)(C1=CCCC1(C)C)N(C1CCCC(N(C)C(c2ccc(Cl)cc2)=O)C1)C c1(C(N(C2CC(NC(C(COC)NC(C)=O)=O)C2)C)=O)ccc2oc(O)nc2c1 C1(NC(CC=CCC)=O)CCN(Cc2cn(-c3ncc(C)s3)nn2)CC1 N1(C(COC(CC)C)=O)C2CCC1CN(C(=O)CC1(C)CCOC1)CC2 Cc1ccc(F)c(C(N2CCSC(C)CC2)=O)c1O C(=O)(C(C)CC(N)=O)NCC(CC=C)NC(=O)COC1CCCCC1.c1(O)cn[nH]c1 N1(C(C(C=C)OC)=O)CC(C2CCCN(C(c3[nH]nnc3CC)=O)C2)C1 C1(C)(C(=O)NCCN(C)C(c2ccc(CO)c(F)c2)=O)CCNC(=O)C1 c1(CN2CC(C)(C(=O)NC(c3ccc(F)c(O)c3)=O)C2)nc(Cl)c(Cl)cc1Cl C1(C(=O)NCC(C)CNC(c2cc(C(F)(F)F)n[nH]2)=O)C(F)(F)C12CC2 N1(C(c2c(CC)ocn2)=O)CC(CNC(C2CCCC2C2CC2)=O)C2(CC2)C1 C1(CNC(c2cnn(CCF)c2)=O)CC2(CCC2)CN1C(=O)CCC(F)(F)F c1(C(N2CCC(CC=C)(NC(C3CCSC3)=O)C2)=O)c(C)nc(C2CC2)nc1O c1(SCCC2N(C(=O)OC(C)(C)C)CCOC2)nc(-c2ncccn2)ncc1F N1(C(C(C2CCC2)OC)=O)CCC2CN(C(c3nn(C)c(C)c3Cl)=O)C2C1 CC(C)CCC(=O)C(=O)NC(CC1CCC1)CC(=O)NOCC1(F)CCC1 C1(CNC(c2c(C)ccnn2)=O)CCCCN(C(c2cccc(C(N)=O)n2)=O)C1 CC1CN(C(=O)C(Cn2ccnn2)NC(=O)Cc2cnoc2)CCC1N(C)C c1(C(N2CC3C(CNCc4ccc(OCC)nc4)(C3)C2)=O)ccc(C#N)cc1C C1(NC(CNC(CC(C)C)=O)=O)CCC(NC(=O)C(C2CC2)N(C)C)CC1 c1(C(=O)NC(C(=O)NCC2OCC(C)C2)Cc2cn[nH]c2)cn(C)ccc1=O N1(C(C(C)N=[N+]=[N-])=O)CCCC12CCN(C(c1c[nH]nc1Cl)=O)CC2 N1(C(CCN(C(C(C)C)=O)C)=O)CCc2ncsc2C1 N1(C(C2(C(C)C)COC2)=O)C2CCC1CN(C(=O)CN1CCC(C)(C)C1)CC2 Cc1cc(C(=O)N(C2CCC(NC(c3nn[nH]n3)=O)CC2)C)cc([N+](=O)[O-])c1 C#Cc1cncc(C(=O)NC(C)(C(=O)NCc2conc2C2CC2)C2CCC2)c1.OCC c1(N(C)CC2CCN(C(=O)CC3(C)CCCO3)C2)nc2ccc(O)cc2s1 C1(C(N2CC(CNC(c3c(NC)nccc3)=O)C2)=O)CCCC(F)(F)CC1 c1(C(N(CC(C)(C)CNC(c2ccn(C)n2)=O)CC)=O)cc(C)c(Cl)s1 n1(CC)cc(C(N2CC3C(CNC(C4(C)CC(=O)N(C)C4)=O)C3C2)=O)cn1.CC N=c1nc(N2CCN(C(=O)C(N)=O)CC2)[nH]c(=NC2CCCC(N3CCC3)C2)[nH]1 Cc1noc(C)c1-c1cncc(F)c1.c12ccc(cc1)[nH]c2=O CC(C(C)(C)C(=O)NC1CCCOC1)NC(C1CN(C(=O)N(C)C)C1)=O C1(NC(C2N(S(C)(=O)=O)CCCC2)=O)CC2C3CCC(C3)C12 c1(CNC(c2cc(C)n(C)c2)=O)n[nH]c2c1CN(C(C1CC1C(N)=O)=O)CC2 C1(NC(C2N(C(CCCN(C)C)=O)CC=C2)=O)CC(C)(C)C12CC2 Cc1cc(C(=O)NCC2C=CCN2C(C2CC2c2ccco2)=O)c(F)c(Br)c1 C#Cc1ccccc1NC(=O)CC1CCCN1C(=O)Cc1ccc(OC)nc1 C1(CNC2(C(N3C(C(=O)OCC)CC(O)C3)=O)CCCCC2)Cc2nccn2C1 C1(CC(=O)NCC(CO)NC(=O)NCCc2csnc2Cl)CCC=N1 Cc1cc2ncnc(N3C4CCC3C(C)C(NC(C3(C)CC(C)C3)=O)C4)c2[nH]1 C1(CNC(C(C)OC)=O)CCC(NC(=O)Cc2coc(C)n2)CC1 C1(NC(C(CSC)c2ccccc2)=O)C2CC1CN(C(=O)CC(C)C)C2 N1(C(c2cc(Cl)ccc2Sc2ccccc2)=O)CC2CCCN2c2ccccc21 C=CCC(CC)C(=O)N1CCCOC(CNC(c2conc2C)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CC2CCC(NC(C(CCOC)(C)C)=O)(C1)C2 CC1(NC(C2OCCO2)=O)CCN(C(C2CCCN(C(=O)C3CC3)C2)=O)C1 c1(C(=O)NCCOCCCNC(C2(C(N)=O)CC2)=O)ccnc(CO)c1 Cc1nn(C)c(C)c1OCC(=O)NCC(O)CCNC(c1csc(S)n1)=O C1(NC(c2cocc2Br)=O)CN(C(=O)CCF)C2(CCCCCC2)C1 C1(C(=O)NC(c2ccccc2Cl)CO)CCCN(C(c2cc(Br)cs2)=O)CC1 c1(C(N(C(C)CNC(c2ccco2)=O)C)=O)cccc(Cl)c1O C(=O)(NNC(=O)CCCn1cc(C2CC2)nn1)NCC=CC(=O)OC C1(NC(COCCOC)=O)CC2CCCC(C1)N2C(=O)Cn1cc(Br)cn1 c1(C(=O)NC2CC(N(C(C3C(C)C3)=O)C)C2)cnn2c(N)ccnc12 N1(C(c2c(OC)nsc2)=O)CCCCC1C1CCCN(C(=O)CCCSC)C1 Cc1c(C(=O)O)cc(Cl)cc1S(=O)(=O)N(C)C(C1CCCCC1n1cccn1)=O C#CC1(NC(=O)CC2(C)CCN(C(=O)C(C)(O)C3CCC3)C2)CCC(C)CC1 C1(C(N(CC(C)O)CCNC(=O)CCCc2cccc(Cl)c2)=O)CCC(C)(C)C1 c1(NC(C2CC(OCc3ccccc3)C2)=O)cccnc1-c1cccnc1 c1(OCC(=O)N(C(CCNC(c2nc(C)[nH]n2)=O)C)C)ccc(Cl)cc1C(N)=O c1(C(N(CCN(C(c2c[nH]c(Br)c2)=O)CC)CC)=O)cc(O)n(CC)n1 c1(CC(N2CCSCC2)=O)cnn2c1CN(C(c1c(Br)ccc(F)c1F)=O)CC2 CCCCC(O)C(C)C(=O)NC(C)C(C(=O)N1CCC(=C(F)F)CC1)C(C)C c1(C(N2C(c3cn(C(CC=C)CC)nn3)CCC2)=O)nnccc1C C1(CNC(C2CC(CNC(COC(CC)C)=O)C2)=O)CC(C)(C)CO1 N1(C(C(C)(CC2CCC2)OC)=O)CCCC(CCNC(=O)C(C)(F)F)CC1 N1(C(C(CC=CCC)C)=O)CCCCCC(NC(=O)CCCC2CCCCC2)C1 C1(O)(C(N2C(C(NOC3(CCCC)CC(C)C3)=O)CC2)=O)CCOCC1 C1(C(N2C(CC(=O)NCCCn3cnnn3)CC2)=O)CC2(COCCO2)C1 CC(CC(C)(C)C)C(=O)NC(c1ccc(Cl)cc1)c1ccccc1C(F)(F)F CCCC(C)CCNC(=O)COC1CCN(C(=O)CC2CCOC2)C1 C1(CC#C)(C(=O)NCC2CC3CCC3C2)CCN(C(=O)CC(=O)NC)C1 c1(CC)nn(C)cc1C(=O)NCC1(NC(=O)C2=CCCO2)CCCC1 C1(C(N2CCCC2CNC(=O)C(C2(O)CN(CC)C2)F)=O)CC(=O)CC(=O)C1 c1(C(N(CCC(=O)N(CCCCC)C)CCO)=O)csc(=N)[nH]1 c1(NC(=O)OC)ccc2c(c1)CCN(C(C1CCCC13CC3)=O)C2C CC(C(C)C(=O)N(C1(C2CC2)CC1)C)NC(=O)C=Cc1cn(C)nn1 CC(C)(C)CC(O)CC(=O)NC1(CCCC(=O)NC(CO)C2(C)CC2)CCC1 N1(C(CN(C2CCCN(C)C2)C(C(CC)OC)=O)=O)CCOC(C2CC2)CC1 c1(C(N2CCC(N(C(=O)CC3(C4CC4)CC3)CC)C2)=O)nn2c(c1C)OCCC2 C1(NC(=O)COCC2CCC2)CCN(C(=O)C=Cc2ccsc2)CC1O C1(C(=O)Nc2c(C)c(CN(C)C)ccc2)C2CCC1(C)C2(C)C CC1(C)CC(NC(c2ncccc2Cl)=O)CN(C(c2ccccc2[N+](=O)[O-])=O)C1 S(=O)(=O)(c1ccsc1C(=O)NC(CNC(=O)C1=CCCCC1)C1CC1)N(C)C C1(NC(c2cccc(NC(C)=O)c2)=O)CC2(C1)CN(C(C1CCC(=O)O1)=O)C2 C1(CNC(c2c(CC)occ2)=O)CC(OC)CN1C(=O)CN(C)S(N)(=O)=O c1(C(N2CCC(Nc3nc(C)nc(O)c3C)CC2C)=O)ccc2ncncc2c1 c1(C(=O)OC)cc(N2CC3CCC3(OC)C2)nc(C(C)C)n1 c1(-c2nc(NC(C(C3CCC3)OC)=O)sc2)ccc(C)cc1 Cc1cc(NC(C2CCC=CCC2)=O)nc(Br)c1 C1(NC(c2cc(CSCC)on2)=O)CN(C(=O)C(C)(C)CC)Cc2ccnn2C1 C1(CC(=O)NC(C)(C)CF)CCCN1C(N)=O C(=O)(C1=CC2(CCN(C(=O)C(C)CC#N)C2)C1)N(c1cccc(C)c1C)C c1(N2CCCC(C)C2)cccc(S(=O)(=O)NC2CCC=C2Br)n1 N1(CC)CC(C)N(C(=O)CN(C(=O)CC2(OC)CCC2)C)CC1C N1(C(CC2CCN(C(C)=O)CC2)=O)CCC2C(NC(C3CC34CCC4)=O)C2C1 c1(OC)cccc(F)c1CN1CCOC(CC(=O)Nc2cnc[nH]2)C1 C1(NC(c2cc(COC)no2)=O)CC2CCC1CN2C(=O)CC(C)(C)C#N N1(C(CC(C)OC)=O)CC(OC)C(NC(=O)CSc2nncs2)C1 c1(C(N(CCNC(C(C)(C(C)C)NC(C)=O)=O)C)=O)oc(S(N)(=O)=O)cc1C c1(C(=O)NC)cc(C)[nH]c(=NCCCC(C)(C)NC(=O)CC(C)C2CC2)n1 C1(CNC(c2c(CC)ocn2)=O)C2CN(C(c3ccnc(OC(F)F)c3)=O)CC12 C(=O)(C(CCF)NC(=O)OC(C)(C)C)N(CC(c1ccc(F)cc1)(F)F)CC N1(CCNC(C(CC)N(C(=O)Cn2nccn2)C)=O)CCCOCC1 N1(C(C)C(N2CCCCC2)=O)CC2CC1CN2C(c1cc(C(N)=O)cs1)=O c1(CC(=O)N(CC(C)NC(C)=O)C)cccc(CSc2nnnn2CC(F)F)c1 CCCC(C)CN(C)C(C1(N(C)C(c2cc(C(C)C)[nH]n2)=O)CC1)=O c1(C(=O)NC2C(CNC(C(C(C)C)C3CCC3)=O)CC2)cc(F)ccc1F CCCCCCC(F)C(=O)NC(C)CNC(c1sc(CC)nc1C)=O n1(CC(=O)NC2C(CNC(C(C)c3cc[nH]n3)=O)CCC2)ncc(C#N)c1N c1(C(C)=O)cc(S(=O)(=O)NC(=O)C(C)(C)C(C)O)ccc1Cl N#Cc1cccc(F)c1CC(N1CC(NC(C2CCCO2)=O)CC(F)C1)=O n1(CC)ncc([N+](=O)[O-])c1C(=O)NCC(C1CCC1)NC(=O)Cc1csc(S)n1 S(=O)(=O)(c1ccc(N2CC3CC2CC3O)c(C#N)c1)NCC(CCC)O c1(C(=O)NCC(CC=C)NC(C2(F)CCOC2)=O)ccc(CCF)cc1 Cc1ccc(NC2CCOC(c3ccccc3)C2)nc1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NC(CNC(=O)C(C)(C)F)C C1(NC(C(C)O)=O)CCC2(CCN(C(c3cnsc3)=O)CC2)C1 C=C1Cn2c(C(=O)NC3CCCC(NC(C4CC(O)(C#N)C4)=O)C3)nnc2S1 C1(C(=O)NC2(CO)CCN(C(CNS(CC)(=O)=O)=O)C2)CC12CCC(C)(C)CC2 C1(C(=O)N)CCC(NC(=O)CCC(C2CC2)NC(=O)OCC)O1.c1(COC)ccsn1 CCC(CC(=O)N1CCCC1CC1CC1)NC(c1cc(C#N)cs1)=O c1(C(=O)NC2C3CCN(C(c4c(OC)nsc4)=O)C32)coc(S(=O)(=O)N(C)C)c1 C1(C(=O)NC(C)CCNC(c2nc(Cl)ccc2N)=O)CN2CCCCC2CO1 N1(C(Cc2c(C)nc[nH]2)=O)CC2CC(NC(=O)CCn3cnnn3)CC1C2 N(C1c2ccccc2CC1C)C(c1ccc(OC)nc1Br)=O C(c1ccccc1F)=CC(=O)NCC(CC)NC(c1cc[nH]c1C1CCCC1)=O C1(N(C(=O)CN(C)CCO)CC)CCCN(C(c2cc(OC)ccc2N)=O)CC1 N1(C(Cc2c(C)ccs2)=O)CCN(C(=O)CSC(C)C)C(C2CCCC2)C1 C1(N(C(C(F)=CC)=O)C)CCCCC1N(C)C(c1cncc(C(=O)OC)c1)=O c1(C(=O)NC(C2CC2C(=O)NC2CCOCC2F)C)ccc(C#N)s1 Cc1cc(C(=O)NCCC2CC(NC(=O)COC3(C)CCC3)C2)cc(F)c1 C12(C(N)=O)CCCC1(C(N1CC(NC(=O)CSCC3CCCO3)C1)=O)C2 CN1CCCC(CNC(=O)C=CCNC(C2C(C)(C)C2(C)C)=O)C1 Nc1cncnc1C(=O)NCCC1(C(=O)NCC2CC2Cl)CCC1 c1(C(N2CC(CO)C3(CCC3)C2)C(=O)NCCC#N)ccc2ncccc2n1 N1(C(C2(N(C(Cc3cnc(C)s3)=O)C3CC3)CCC2)=O)CCC12CCC2 CC(C(=O)NCCOCCNC(=O)CCSc1cccs1)N(C)C CN1CCCC1(C)C(N1CC2C(CNC(c3cncc(C4CC4)n3)=O)C2C1)=O c1(OC)ncc(C(=O)NCCN(C(=O)C(O)CCN(C)C)C)c(C(F)F)n1 C1(CNCC(=O)OCC)CC(C(=O)NN(C)C)=NO1 N1(C(CC2(OC)CCOCC2)=O)CCC2CN(C(=O)CCc3cnc(C)o3)C2C1 C1(CC)CCCN(C(=O)CN2CCOCC2)C1C(=O)NC(c1ccccc1C)C C1(OC)CC(O)CN(C(=O)C(CNC(=O)C(O)C(F)(F)F)N(C)C)C1 Cc1nc(N)cnc1C(=O)NC1CCOCC1NC(=O)CCn1cccn1 CC1CN(C(=O)CC2(C#N)CCCCC2)CCCN1C(C1CC(N(C)C)C1)=O c1(C(N2CCCC(C(=O)Nc3ccnn3CCO)C2)=O)cc([N+](=O)[O-])c(O)cc1O c1(CCC(=O)NC(C2CCOC2)CNC(C=C(CC)CC)=O)nc(C2CC2)no1 C(=O)(C(CCOCCO)NC(c1nncn1C)=O)N(C1(n2cnnn2)CC1)C c1(C(N2CCC(COC)(NC(=O)C=C(C)C(F)F)C2)=O)cc(C)n(C)c1C N1(C(C(C=C)OC)=O)CC(NC(C2CCCOCC2)=O)CC(C)C1 CC(N=c1[nH]nc(C(F)(F)F)s1)C1CCCN(C(C2CC2(F)F)=O)C1 C1(NC(Cc2ncc(C)[nH]2)=O)CCC2(CCCN(C(=O)CC3CC(=O)C3)C2)C1 c1(OC(=O)OC)ccc([N+](=O)[O-])c(C(=O)NC(CNCC=C)CC)c1 C1(NC(c2c(C)c[nH]n2)=O)C2CC(NC(=O)CC3CCCC3C)CC12 c1(C(C)C)ccc(CC(=O)NC2CC(NC(C34CC(C)C3C4)=O)C(O)C2)cc1F C(=O)(C(CCC(C)C)NC(C1CC(=O)C1)=O)NC(CCOCC)C C1(NC(CC2(CC(=O)OC)CC2)=O)CN(C(C2CCOC(C)(C)C2)=O)CC(C)(C)C1 C1(CNC(c2nn[nH]c2Cl)=O)CN(C(=O)Cc2cnsc2)CCO1 C1(C(=O)NCC#CCOC)CCN(C(c2cc(OC)cs2)=O)C1C(C)C c1(C(=O)NCC2CC(C(=O)NCC3CCCOC3)C2)cccc(F)c1F N1(C(c2ncc(-c3n(C)ncc3)nc2)=O)CCc2ccc(F)cc2C1 Cc1cc(F)c(N)cc1C(=O)NC(C(C)NC(c1ccc(Cl)c(F)c1)=O)C(C)C c1(C(C)C)nnc(N(CC(C)CNC(=O)C=CC2CCOC2)C)o1 C1(CNC(C)=O)CCCCN1C(=O)CC1CCCC(C2CC2)O1 C1(C)(NC(CCNC(=O)NC)=O)CCN(C(C2CCCCC2)=O)CC1 c1(C(N2CC(C)(NC(=O)Cc3ccsc3Br)C2)=O)cccn2nnnc12 N1(C(Cc2ccc(OCC)nc2OC)C)C(=O)NC(C2CCCO2)C1=O C1(CC)CCCCC1C(N1CCOCC1CNC(=O)CCNC(N)=O)=O C(=O)(CC1OCc2ccccc21)NC1CC(CNC(c2ccc(C)c(C)c2)=O)C1 Cn1cc(C(=O)NCC2CCCCN2C(c2ccnn2CC#N)=O)c(O)nc1=O C(=O)(C(C)(C)COCC)NCC1(CC(=O)N(CCCCC=C)C)CC1 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(N(C(C(CSC)OC)=O)C)C2(C1)CC2 S(=O)(=O)(c1ccc(NCCc2cc(Cl)ccc2Cl)nc1)N1C(COC)CCC1 S(=O)(=O)(c1ccc(F)c(F)c1)N1CC2C(NCc3c(O)ccc(C)c3)C(CC2)C1 C12(NC(c3ccoc3C(F)(F)F)=O)CCC(C1)N(C(C1CC=CCC1)=O)C2 CCC(C(=O)NCCN(C(=O)CCOc1cc(F)ccc1F)C1CC1)C(C)O c1(CNC(C)=O)ccoc1C(=O)NCC1CC(O)C1 N1(C(C(C)(N)C2CCCO2)=O)Cc2ccccc2C(C)(C)C1 c1(C(=O)NCC(c2ccccc2)NC(CCOC)=O)ccc(SC(F)(F)F)nc1 c1(OC)ccc2cc(C(=O)NC3CC(C)CN(C(C4CCCS4)=O)C3)ccc2c1 c1(OC)ccc(C(=O)NC2CC(NCc3c(C(F)(F)F)cccc3Cl)C2)c(O)c1 c1(CCNC(C(COC)NC(=O)C(C)CC2CC2)=O)cn(C)nc1C N1(C(C2C3(CC(NC(c4c(C)oc(CO)c4)=O)C3)C2)=O)CCC(C#N)CC1 CC(C)C(C(=O)NC12CC(CNC(=O)C(C)C#N)(C1)C2)Sc1ccccc1 c1(CNC(C(CC#C)NC(=O)CCC2CC2)=O)cc(C)ccc1F c1(CC(C(N2C(CNC(C(C)=C(CC)C)=O)CCC2)=O)C)cccc(Cl)c1 C1(C(=O)NCC2N(C(C3C(C)CC3)=O)CCC2)CC(C)(C)CO1 C1(N)CCCC2CN(C(=O)C3=CC(C)(C)C3)CC12.CCC(C)(C(=O)NC(C)(C)C)OC N1(C(C(C(CC)C)O)=O)CC2CCC1C(NC(c1[nH]ccc1C)=O)C2 CCC(C)CC(C)CC(C)C(=O)N1CCC(N2CCN(C(C)C)CC2)CC1 CCCC(C)CC(=O)N1CCN(C(c2cc(COC)cn2C)=O)CC1COC CC1=C(C(=O)N2CCC(NC(C3CCS(=O)CC3)=O)C(C(C)C)C2)CCC1 C=CCCC(C(=O)NCCC(C)F)NC(=O)CCC(CC)OC c1(N2CCC(N(C(C(C3CCOC3)OC)=O)CC)C2)nc(C)nc2c1cnn2C Cn1cc(C(F)=CC(N2CC(C)(NC(=O)C=CS(C)=O)C2)=O)cn1 CC1(C)CN(C(c2ccc(C(=O)Nc3ccccn3)c(Cl)c2)=O)CC1C(=O)O N1(C(COCCCC)=O)CCC(C)C(NC(=O)CCC23CCC(CC2)C3)C1C c1(CC(=O)NC2CN(C(CCCOCCC)=O)CC2C)ccc(CC)c(F)c1 N1(C(c2c(C)cc(F)cc2)=O)CC2CCCC2(NC(c2cnn(C)c2N)=O)C1 CC1(C)CC1(C)CNC(c1csc(O)n1)c1nnnn1C(C)(C)C C1(CNC(CCN(CCC)C)=O)CN(C(=O)C(N2CCOCC2)C)C2(CCC2)C1 c1(-c2cn(C(COCC)C(N3CCC(C)C3COC)=O)nn2)ncc(F)cn1 N1(C(CC2(C=C)CN(C(=O)CC(Cl)Cl)C2)=O)CCOCC(O)C1 c1(C(N2C(C)CN(C(CCCC#C)=O)C(C)C2)=O)c[nH]c2cccc(F)c12 C1(NC(CCCOC(C)=O)=O)CC2CCC1(NC(c1cc(C)n(CCO)n1)=O)C2 N1(c2n(CC(=C)C)c(-c3ccoc3C)nn2)CC(C)OC2(CCCOC2)C1 CS(C)(=O)=Nc1ccc(C(=O)NC2CCC(NC(c3sccc3C#N)=O)C2)cc1 c1(C(=O)NC2CCC(C)N(C(=O)COCCN(C)C)C2)ccc(P(C)(C)=O)cc1 c1(C(N(CC(C)NC(=O)C(O)CC2CCOCC2)C)=O)ccc(F)cc1N N1(C(C(CCC)O)=O)CC2(C1)CN(C(C1CN(C(C)C)CCO1)=O)CC2CO C(=O)(C(C)(C)CCCNCCCCOC)NC(CNC(C(CC#C)C)=O)(C)CO c1(C(=O)NC2CC(CNC(C=CCCC)=O)C2)cnc2sc(C)c(C)n12 Cn1cc([N+](=O)[O-])cc1C(N1CC2CCC(C1)C2NC(c1cscn1)=O)=O c12ccc(cc1)CC(=O)N2C.C(C)(CCNC(=O)C=C1CCC1)NC(=O)OCC C(CC(C)CC)(C(=O)NC(C)(C)CCN(C)C)NC(C1ON=C(CC)C1)=O c1(C(N2C(CC(=O)OCC)CCC2)C(=O)NCC(C)C)c(Cl)c(C)nn1C Cc1ccc(NC(C2CCOC2CNC(c2nonc2N)=O)=O)c(C)c1O CCCC(C)NC(=O)CSC.CCC(C)(c1nccs1)NC=O N1(C(C(C)SCCCC)=O)CCCC(NCCN(C)C(c2coc(CO)c2)=O)C1 Cc1ccc2c(CNC3CCCN(Cc4ccccc4)C3C)cc(=O)oc2c1 C(=O)(CC(C)CC(F)(F)F)N1CCC(N(CCC)C(C2(C)CC(C)C2)=O)C1 C1(N(C(c2sccc2Cl)=O)CC)CCCN(C(c2cc(Cl)cs2)=O)CC1 c1(C(N(CC(C)NC(=O)C(C)S(C)(=O)=O)CC)=O)nn2cccnc2c1Cl Cn1[nH]c(=NC(=O)NCC(C)(C)CN2CCCC2)c(=O)n(C)c1=O c1(CNC(CCC)CC)nc(O)c2c(C)c(CCCC)sc2n1 N1(C(c2ccc(CSC)cc2)C(=O)NCc2ccco2)CCOCCC1C1CC1 C1(C(=O)NC(C=C)C)CCC(c2ccccc2)CC1 C1(CCCNC(C(C)C2CCC2)=O)CCN(C(=O)C=Cc2cn[nH]c2)CC1 C(C)(c1cnn(C)c1)=CC(N1CC(CCNC(C(CC)C)=O)(OC)C1)=O c1(C(N2C(CC(=O)NCCCC(=O)OC)CC2)=O)nnc(O)nc1O c1(OC)cccc(CC(N2CCN(C(=O)C(CO)C(C)C)CC2C2CC2)=O)c1F CCC(CC1CC1)N=c1cc(C)[nH]c(=NCCC2CC(O)C2)[nH]1 C(=O)(C1=C(C)CCCC1)NCc1cn(CC(C)NC(C(CCC)C)=O)nn1 N1(C(c2c(C)cncc2)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)C2CCC12 O=S(=O)(c1cccs1)NCC1(O)CCCN(Cc2cc(Cl)ccc2Br)C1 N1(C(C2(CC)CCOC2)=O)CCN(C(=O)CCCOC)C(c2ccc(Cl)cc2)C1 c1(C(C)C)cc(=NC2CCN(C(C3(O)CCOC3)=O)CC23CCC3)[nH]c(Cl)n1 C1(C)(CNC(C(C)(C)NC(=O)NCC)=O)CN(C(=O)CC2C=CCC2)CC1(F)F Cc1cc(Br)cc(C)c1C(=O)NCC1CC(NC(=O)Nc2cccc(Cl)c2Cl)C1 Cc1nc(N(C2CCN(C(=O)C=C(Cl)Cl)CC2)C)ccc1[N+](=O)[O-].C1CCN1 Cc1nnc2n1CCCC2C(=O)Nc1cnc2n1CC(C(F)(F)F)CC2 N1(C(COCCCC#C)=O)CCN(C(=O)NC2CN(C3CCOC3)C2)CC(O)C1 N1(C(C2CN(C(C)=O)C2)=O)CCC(C)C1CNCc1ccc(N2CCCC2)nc1 CC1C(NC(c2ccc(-n3cncn3)nc2)=O)CCN1C(=O)CCC(F)F c1(C2C(C(=O)NCCC(C)NC(C3(c4nc[nH]n4)CC3)=O)C2)ccccn1 C(=O)(C1CCc2c[nH]nc21)NC(CC(C(=O)N(CC#CC)CC#C)F)(C)C C(=O)(C(C)(C)CN(C(=O)Cc1ccnn1C)C)NCCC1CC(C)C1 c1(C(=O)NCC(C2CCCC2)NC(=O)CC2(O)CCOC2)cc(Cl)c(Cl)s1 c1(C(N2CC(C(=O)N(C(C)(C)C)C3CC3)OCC2)=O)cccc2c1COC2 c1(CC(=O)N(CC(C)NC(=O)CCS(C)=O)CC)ccc(C)c(F)c1F c1(C(N2CC(C=C)C(NC(=O)CCc3cnco3)C2)=O)cncc2[nH]ccc12 Cc1cccc(C)c1OCC(=O)NC12CCCC1N(C(c1cnc(S)[nH]1)=O)CC2 CN1CC2(CCN(C(=O)CC3C4CN(C(=O)C(C)(C)CO)CC34)CC2)C1 C(=O)(CC(C)(C)CC(F)F)N1C2CC(CNC(C(C)OCCCC)=O)C1CC2 C1(NC(c2cnc3ncccn23)=O)CCC2CN(c3nnco3)CC2C1 Cc1cc(C(=O)NCC2(C)CCCN2C(C2(F)CCCCC2)=O)ncc1C(F)F CC1CCN(C(c2cnn(CCF)c2)=O)CCN1C(=O)C(F)CC(C)(C)C CCC(C)C(=O)C(=O)NC(C1CC(C)(C)C1)CNC(c1c[nH]nc1[N+](=O)[O-])=O N#Cc1cccc(S(=O)(=O)NCC(N2CC(O)C2)=O)c1 C1(CC(=O)NCC(C(=O)NCC(C)OCCO)O)CCC(=O)CC1 C12CCCCC1(C1CC1)CN(C(=O)OC(C)(C)C)CC1CC(C1)CNC(=O)N2 C1(C2(C)CC2)(C(N(CCCCNC(C(CC2CCC2)OC)=O)C)=O)CC1 c1(C(=O)NC(CNC(C(CC)O)=O)CC)c(C)cc(=O)n(C)c1C c1(CC(=O)NCCCN(C(=O)Cc2coc(-c3cccs3)n2)CC)cnc(C)[nH]1 C12(NC(=O)C=CC3CCCCC3)CCN(C(=O)Cc3c[nH]ccc3=O)CCC1C2 C=CC(C)(C)CC(=O)NC1C2CC1CN(C(C13CC(OC)C1C3)=O)C2 CN=c1[nH]cc(C(=O)NCCOC2CCN(C(=O)C3=NOCC3)C2)s1 CCCCS(=O)(=O)CC(=O)NC1CC1CNC(c1cc(OC)n(C)n1)=O C1(NC(CCOC2CN(C(C(C(=O)OC)C)=O)C2)=O)CCC(=O)N(C)C1 c1(C(=O)OC)c(NC(=O)C(C)(O)Cn2cc([N+](=O)[O-])cn2)sc(C)c1C C=CCC(CC=C)C(=O)N1CCC(NC(=O)CCCF)C(CO)C1 C(Cc1cn[nH]c1)(C(=O)NOCCCF)NC(c1ccoc1Cl)=O N1(C(C2CC(C#N)(OC)C2)=O)CCC(C)C(NC(=O)Cc2cnco2)C1C Cc1ccc2occ(CC(N3CCC4CN(C(C5CC5C)=O)CC4C3)=O)c2c1 N1(CCCNC(=O)CN(CCNC(c2cccnc2)=O)C2CC2)CCCC1=O N1(C(c2ccc(F)cc2F)C(=O)Nc2cccc(N(C)C)c2)CCOCC(N)C1 CC12COC(C(=O)NCC3(O)CN(C(=O)CCCn4cncn4)C3)(C1)C2 c1(OC)cccc2c1OC(C(=O)N(C1CCN(C(=O)C(C)C#N)CC1)CCO)C2 C(=O)(CCS(=O)(=O)N(C)C)NCCC1CC(NC(C=NOC)=O)C1 c1(OC)cc(NC(N2CCCC2CCNCCNS(C)(=O)=O)=O)cc(Br)c1 c1(C(N2C(CC(=O)NC(C)CC3CC3)CC2)=O)cn(C)c(=O)n1C c1(CC)nccn1C(C)CC(=O)NC1(CNC(=O)C(C)CC2CC2)CC1 c1(C(N2CC(CC(C)NC(=O)CC(O)C(C)C)C2)=O)ccc2cnccc2n1 CCC(CCCC(=O)NC1C=C(C)CCC1)NC(c1cc(COC)on1)=O c1(CC(=O)NCCN(C(c2ccc3nccn3c2)=O)CC)cc(F)c(N)cc1F Cc1nn2cccnc2c1C(=O)NC(CO)C(C)NC(=O)CN1CCCOC1=O C1(CNC(c2c(N(C)C)cccc2)=O)CCCN(C(=O)C2=CCCO2)CC1 CC1(C)C(CNC(=O)CCCc2ccc(Cl)cc2)CCN1C(=O)CC(O)C1CC1 N1(C(=O)COCc2nccs2)CCN(C(c2coc(O)n2)=O)C2(CCC2)C1 Cc1cc(OCCCn2nnnc2N(c2c(C)cccc2C)C)cc(C)c1 C1(NC(c2scc(C)n2)=O)CCC(=O)NC1C1CCCO1 C1(C(=O)NC2(C)CC(NC(C(Cc3ccc(C)cc3)C)=O)C2)CCOC(=O)CC1 Cc1c(C(N2CC3CC(NC(=O)C(F)C4CCC4)C2C3)=O)[nH]c2cc(F)ccc12 N1(C(c2c(C)cc(Br)o2)=O)CCC2(CNC(=O)CC3CC3)CCCC12 C(=O)(C1=C(C)OCCC1)N1C(CN(C(CC2CCC(C(C)=O)CC2)=O)C)CCC1 N1(C(C(c2cnn(C)c2)OC)=O)CCC2CCC(NC(=O)CC(C)C(F)F)C1C2 c1(C(=O)NCC2(OC)CN(C(=O)C(C)S(C)(=O)=O)C2)cc2cc(F)cc(C)c2[nH]1 C1(OC)CC(NC(=O)CC2CC3(CC3)CO2)N(C(=O)COCCOC)C1 c1(NC(C2CC2C(N2CCCCC(O)C2)=O)=O)cc(F)ccc1Br N1(C(C)(C)C)CCC(CNC(=O)NCC(O)Cn2cc(C(N)=O)nn2)C1 C1(CC#C)(C(=O)NC2CCC2CNC(=O)CN2CCCS2(=O)=O)CC=CCC1 N1(C(CNC(COC)=O)=O)CCN(C(=O)C=CC2CCCCC2)C(C)CC1C N1(C(CC(n2c(CC)ncc2)C)=O)CCC2(CC1)OCCC2NC(C12CC1C2)=O C(=O)(C(O)CC(C)(C)C)NCCCCCNC(C(C(C)C)SCC)=O C(C)(CCC(C)(C)O)(c1n(C(CC)(C)C)nnn1)NC1(CCO)CCOC1 C(=O)(CC(C)(C)NC(=O)C(C)C1(O)CCC1)NC(CCOCC)C c1(CC(=O)NC(C(=O)N2CC(n3cnnc3)C2)c2ccco2)cccnc1F c1(NC(CNC(CC(C)=O)=O)=O)cccc(Br)c1OC(F)F Cc1cccc(CC(=O)NC23CC2CN(C(C2C=CCCC2)=O)C3)c1 C(=O)(C(C#N)(CC)CC)NCC(CC(=O)Nc1c(CC)n(C)nc1)OC Cc1onc(C2CCCCC2)c1C(=O)NCCNC(=O)C(C1COC(C)(C)O1)O N1(C(=O)Cc2ccc(Cl)cc2)CCCC(NC(C2(C3CC3)CCCO2)=O)CC1 c1(C(C)(C)C(=O)NC2CC(CCn3cc(C4CCCC4)nn3)C2)cccnc1F S(=O)(=O)(c1c[nH]ccc1=NC1CCCOC1)N1Cc2c(cc(OC)c(OC)c2)C1 N1(C(C2N(C(c3cccc(C)c3N)=O)CCOC2C)=O)CCC(=C(F)F)CC1 Cc1ccc(CN(C(=O)C(C)(CNC(=O)CCC(N)=O)N(C)C)C)cc1 N1(C(CC2(C=C)CN(C(C3CC3C(N)=O)=O)C2)=O)CC2CCCCC12C N1(CC(=O)NC2(C)CC(NC(c3c(C)onc3)=O)C2)C(=O)NC(C)(C2CC2)C1=O C1(NC(C(N2CC(C)OC(C(F)(F)F)C2)=O)=O)CC2(C1)CC1CCC(C2)N1 C1(C(C(=O)NCCCC(=O)OC)N(CC(=O)NC(C)CC)C)CCC(C)CC1 c1(CC(N2CC(CNC(C(C(C)C)OC)=O)C2)=O)nn(C)c(=O)c2ccccc12 N1(C(c2nc(Cl)sc2Cl)=O)CCC2(CCCN(C(C3CC4CCC3O4)=O)C2)CC1 C1(C#N)(C(N(C)CCNC(=O)Cc2cc(C(F)(F)F)n(C)n2)=O)CCCOC1 c1(CN2CC3C(CNC(C(C)(C)O)=O)(C3)C2)c(F)c(F)cc(F)c1F C(=O)(C(O)C(F)(F)F)N1C(CNC(c2ccc(CCC)[nH]2)=O)(COC)CCC1 c1(C(N2C(CN(C(C3N=C(C)SC3)=O)C)COCC2)=O)ccc(=O)n(CCO)c1 N1(C(c2c(C)coc2C2CC2)=O)CC(NC(C2C(F)(F)C23CCC3)=O)C2(CC2)C1 Cn1cc(C(=O)NC2(C)CC(NC(C3CC4CCC4C3)=O)C2)ncc1=O c1(-c2cc(-n3c(-c4n(CC)ccn4)ncc3)[nH]n2)ccc(OCC(O)CO)cc1 C1(c2n(C(C(=O)OCC)C)nnn2)(NC(CC)C(C)C)CCCCC1 Cc1c(CN2CCCCC(Cc3nc(CO)no3)C2)cc(C#N)n1C C=CCCC(C(=O)NCC(C)(O)CCC)NC(=O)C(OCC)OCC CC(C)C(F)C(=O)N1CCC(C(O)CNC(c2ccc(OCCF)cc2)=O)CC1 N1(C(=O)CSC2CC2)CCCC2(CCN(C(c3csnn3)=O)C2)C1 c1(C(N2C3CC(NC(C4C(C=C)CC4)=O)CC2CC3)=O)ccc2nc(C)[nH]c2n1 N1(C(C(=O)NCC2CCN(C)C2)=O)CCc2cc(C#N)ccc2C1 C1(C(=O)NC2(C=O)CCN(C)C2)CC2(C1)CC21CC1.C1(O)(CO)CCNCC1 C1(CC(=O)N(C)CC#N)CCC(C(=O)Nc2ccncn2)CC1 c1(C(C)F)ccc(C(N2CC(N(C)C(c3ccc(C4CC4)o3)=O)C(O)C2)=O)cc1 N1(C(C(C)NC(C)=O)=O)CCOC(CCNC(c2cn(C(C)(C)C)nc2C)=O)C1 CCC(CC(F)(F)F)C(=O)NCC1CN(C(=O)CCNC(=O)CC(C)C)CC1O c1(C(N2C(C)CC(NC(C3C(C)(CC)C3)=O)C2)=O)cc(S(N)(=O)=O)co1 C1(O)(CNC(C2(C)CCCCO2)=O)CCCN(C(=O)CSc2ccncc2)C1 N1(C(C2C(C)N(C(=O)CCc3cncnc3)CC2)=O)C2CCCC1CN(C)C2 CC1(CNC(C2CCCCC2O)=O)CCCN1C(=O)CC1CCNC1=O C(=O)(C(C)C(C)n1cccn1)NC(CNC(COCc1onc(C)n1)=O)(C)C Cc1ccnc(NC(C2CCN(C(C34CCCC(CO3)C4)=O)C2)C)c1[N+](=O)[O-] Cc1cc(C(=O)NC2COCCC2NC(=O)C=Cc2cncn2C)cc(F)c1 CS(=O)(=O)C(C(=O)NCC1CCCC1NC(=O)Cc1ccsc1)C1CC1 c1(C(N2CCC(NC(C(CC=C)CC)=O)C23CC3)=O)ccc(=O)n2c1CCC2 c1(CC(C(=O)N(CC(CNC(CN2CC(CC)C2)=O)C)C)C)c(C)n[nH]c1C Cn1cc([N+](=O)[O-])c(=NC2CCN(C(C3CCC=CCC3)=O)CC2)[nH]1 C(=O)(C(CC)CCOC)N(C(CCNC(C1C(CC)CCCC1)=O)C)C N12CCC(F)(C1)C2=O.c1(CNC(C2CC(OC)C2)=O)ccn(C2CC2)n1.C(C)(=O)N c1(OC)nccc2c1CN(C(=O)C(=O)N(c1ccc(S(C)=O)cc1)C)CC2 n1(CC(=O)NCC2CC(OC)CN2C(c2ccon2)=O)sc2ccccc2c1=O C1(C(N(C(CC)CC(=O)NC2CCCCC2C)C)=O)CC2(C1)CC(C)C2 N1(CCc2nc(C)sc2)CCC2(CCCCN(C(c3cnon3)=O)C2)C1 c1(C(C)(F)F)ncc(Cl)c(-c2ccc(Nc3nccs3)cc2)n1 N1(C(C(C2CCN(C(C(C)(C)SC)=O)C2)C)=O)CCC(O)(CCO)CC1 N1(C(c2c(CC)nc[nH]2)=O)CC2(C1)CN(C(=O)Cc1cc(C)[nH]n1)C2 O=C(CC(O)C(Cl)(Cl)Cl)NCCCCNC(C1CC1C(F)(F)F)=O c1(CC(N2CC(NC(C=C(COC)C)=O)C(F)CC2)=O)coc2cc(Cl)ccc12 C1(C(=O)NC2CC(NC(C3(CC=C)CCC3)=O)C2)CC=CC(O)C1 CC1CN(C(=O)C=CC2CCC2)CC1NC(C1(C)CC2(CC2)C1)=O C1(C(C(=O)NCC(CNC(c2cc(C)n(C)c2)=O)OC)C)CCCCCC1 c1(NCC(C)NC(c2c(C)nccc2)=O)nc2c(cc1C#N)CCC(C)(C)C2 C1(NC(CCN(CCCCC)C)=O)CCCN(C(C2CC3CCC3C2)=O)C1 N1(C(CCCCC)=O)CCC(C2(NC(c3ccnc(Cl)c3F)=O)CC2)C1 CC1CCCCC1CC(N1CCCC1C1CCN(C(=O)CCC2(CO)CC2)C1)=O c1(C(=O)NCC(CC=C)NC(=O)C(C)N(C)C(C)=O)c(C)c[nH]c1CC(N)=O C1(CC2CCOCC2)C(=O)N1.C(CC=C=C)N.C1C(=O)N1.C#CCOC(C)=O.C C1(OCCC)CCCCC1C(=O)NC(C)CNC(=O)CCCCN(C)C c1(C(N2CCC(C)C2CNC(C2CCCCC2)=O)=O)cc2ccc(Br)cn2n1 C=CCC(CNC(c1ncccc1CC)=O)C(=O)NCCN(C)OC C1(C(=O)NC(CNC(C=CCNC(=O)OC(C)(C)C)=O)CO)CCCC2(CC2)C1 c1(C(=O)NCCC(C)N(C(=O)Cc2cccc(Cl)c2Cl)C)cnc2[nH]cncc1-2 CN=S(C)(=O)c1ccc(C(=O)NCCN(C(=O)CC2COCC(C)(C)O2)C)cc1 N1(C(CC2(CS(C)(=O)=O)CC2)=O)CC(F)(CNC(=O)C(F)C2CCOC2)C1 c1(C(=O)NCCC2(NC(=O)C(F)C3CCOC3)CC2)cccc2c1CCC2 S(=O)(=O)(CC(=O)NCCN(C(=O)C(C1CCCCC1)C)C1CCCC1)NC N1(C(C2C(OC)CN(C(C3CN4CCN3CC4)=O)C2)=O)CCC2(COC(=O)N2)C1 CC(CN(C)C(c1nccn1C)=O)C(=O)N1CC(N2CC(O)C2)C1 N1(C(C(C)NC(C)(C)C)=O)CC(C)(C)C(NC(=O)C=CCN(C)C)C(C)(C)C1 Cc1nc(C(N2CC(OCCNC(c3ccc(=O)oc3)=O)C2)=O)c(C)o1 N1(C(CN(C)C)=O)CC(OC)CC1CC(N1CCN(C(C2CSC2)=O)CC1)=O Cc1c(C(N2CCC(C)(NC(c3ccc(OCF)cc3)=O)CC2)=O)cncc1F c1(OC)cc(C(=O)N(C)CC2CCN(C(=O)CC(C)F)C2)ccc1F Cc1cc(N)cnc1C(=O)NCC(C)N(C)C(c1ccc(C(C)(C)C)s1)=O C12(NC(CC=C)=O)COCCC1CN(C(c1cc3ccnc(Cl)c3s1)=O)C2 C1(NC(=O)Cn2nnc(=O)[nH]2)CCCCN(C(=O)CSc2ccncc2)C1 Cc1ccc(Cl)c(C(N2CCN(C(=O)CCC(F)(F)F)CC2CF)=O)c1 c1(OC)ccc(C(N2CCC(C)(NC(=O)CN(C)S(N)(=O)=O)C2)=O)c(C)c1OC c1(C(C(=O)NCC(F)F)N(C(c2ccccn2)C)C)cn2c(F)cccc2n1 N1(C(CCC(=O)NC)=O)CCC2(NC(=O)CP(C)(C)=O)CCCC12 C(=O)(C(C)C(C)(C)c1ccccc1)NCC(C)N(C(c1c(C)nc[nH]1)=O)C C1(C(=O)NC2CCN(C(COC(C)(C)C)=O)CC2O)CC1C1CCCCC1 N1(C(Cc2cc(=N)[nH]cc2)=O)CC(NC(c2cnn3c2OCC3)=O)CC(O)C1 c1(C(=O)NC2(CCNC(C(C)OCC3CCCO3)=O)CC2)cc2occc2s1 c1(OCCC(=O)NCCC(C)N(C(=O)CC2CC3(CC3)C2)C)ccc(F)c(Cl)c1 C(=O)(C(F)(F)CCc1ccccc1)NCC1N(C(c2c(C)con2)=O)C2C(C1)C2 c1(OC)cc([N+](=O)[O-])c(-c2nc(CC3CCCCC3)no2)cc1OCCC#N N1(C(c2cc(C)on2)=O)CCCC(NC(C2CCC(C)(C)OC2)=O)C1C C1(CC)CN(C(=O)COc2ccc(F)cc2)CCC1NC(C1CNC(=O)N1)=O c1(C(C(=O)NCCCNC(C(C(C)SC)O)=O)(C)C)ccc(F)c(F)c1F N1(C(=O)CSC2CCCCO2)CCCC2C1CCN2C(c1cc(F)ccc1Br)=O N1(CCc2cc(C)n(C)n2)CCn2ncc(-c3ccccc3)c2C1 CC1(C(=O)NC2CC2NC(=O)C(O)Cc2ccccc2Cl)CCCCCC1 CCCCC(C(=O)NC1CN(C(=O)C(C)CC2CCCCC2)CCC1C)C(C)C c1(C(=O)NCC2C(NC(Cn3c(C)nnn3)=O)CCC2)cnn2c1CCCC2 N1(C(C(CC)(F)F)=O)CC(NC(=O)CCc2ccc(OC)cc2F)CC(C)(C)C1 c1(C(C)C)cccc(CC(N2CCC2CNC(C23CCCC2C3(F)F)=O)=O)c1 N1(C(C2C=CC(NC(=O)CCCC3CCCC3)C2)=O)CC2CCC(O)C(O)C12 N1(C(N2CCCC(C(C)NC(C3CC3C(N)=O)=O)C2)=O)Cc2ccccc2C1=O Nc1cncc(C(=O)NCC2C3CN(C(C4CCCC(O)C4)=O)CC23)c1 C(C(C(C)(C)C)NC(c1c(Cl)n[nH]c1C)=O)NC(C(C)(C)NC(=O)NCC)=O CCN=c1[nH]c(C(=O)NCC2CC(F)(CNC(C3CCN(CC)C3)=O)C2)cs1 c1(CC(=O)NC2(CNC(c3c(CC)c[nH]n3)=O)CCOC2)c[nH]c2ncccc12 N1(C(C(C)NC(CC)=O)=O)CC2N(C(=O)C(C)C(C)(C)C)CCC2(C)C1 c1(CC(=O)NCC(CC)NC(=O)CC2CCCOC2)cnnn1C C1(NC(CCC#CC)=O)CCN(C(=O)C#CC(C)C)C12CC2 C1(NC(C2CCCSS2)=O)CN(c2nnc(C3CCCC3)s2)C2(CCOCC2)C1 C#CC1(O)CC(C(N2CCCCC2CNC(c2oc(SC)cc2C)=O)=O)C1 c1(OC(C(C)Cc2cccnc2)=O)cccc(F)c1C#N C(=O)(C(CC(C)C)C(C)C)NCCC1CCN(C(C(C(=C)C)(C)C)=O)CC1(F)F CN1N=CC(CC(=O)NCC(CC2CC2)C(=O)NCC(F)(F)C(F)F)C1=O CC1(C)CCCCC1=CC(N1CCOC(CNC(C23CCC2C3)=O)C1)=O C1(CNC(CSCC(=O)OC)=O)CN(C(=O)C(C)(C)c2csc(C)c2)CCN1C C(=O)(CCCCC(N)=O)NCCC(C(=O)N(CC(C)SC)C)O Cc1nocc1CC(N1CCC1C(NC(C(=O)NC1CC1)=Cc1cccs1)=O)=O c1(C(=O)NC(CC=C)CNC(C2CC2CC)=O)cc([N+](=O)[O-])ncc1Br c1(C(N2CCC(C(C)NC(=O)Cc3cnoc3)C2)=O)cc2c(nc1O)CCCC2 O=C(CCCCO)O.C1C#CCNC(=O)C1.C(=O)(C(O)c1ccsc1)NC n1(CC)ncnc1C(=O)N(C)CC1CCCN1C(=O)CC1CCC2CC12 N1(C(C(CC)(C)O)=O)CC2(CCNC(=O)CC3CC(C)=NO3)CCC1CC2 C1(C(=O)NCC2CN3CCC2C3)(CC)CCN(C(=O)CC(C)(C)O)CC1 Cc1nocc1C(=O)NCC1(O)CN(C(=O)C(C)N(CC(F)(F)F)C)C1 C(=O)(C#CC1CCCOC1)NCCC1CC(OC)CN1C(C1CCC(=O)NC1)=O c1(NC(CCC)CCCNC(=O)CCOCCOCC)ncc2ncnc-2[nH]1 O=S(=O)(c1c[nH]ccc1=NC1CCCC(C(F)(F)F)C1)N(CCO)CC1CC1 C(=O)(C(C)C(O)C(C)C)N(CC1C2CN(C(C(SC)SC)=O)CC21)C1CC1 N1(C(c2cnn(C(C)C)n2)=O)CCCC(F)(CNC(=O)CCN(S(C)(=O)=O)C)C1 c1(OC)ncc(CNc2cn(C)c(C(=O)Nc3ccc(F)nc3F)n2)cc1Br C(=O)(C1CCc2cccc(O)c21)N1CC2(F)C(NC(C3CC(=C)C3)=O)(CCC2)C1 N1(C(CSCCN(C)C)=O)CCC(CNC(c2cc(C3CC3)on2)=O)C12CCC2 Cc1ccc2nc(C)c(COC(C3C(c4cccc(Br)c4)C3(C)C)=O)n2c1 n1(CCC(=O)NCC2CN(C(C(COCC)C)=O)C2)cnc2ccccc12 CCCC(CCC)C(=O)N1CCC(O)(CN(C(=O)Cn2ccnc2C)C)C1 Cn1cc(C(=O)NC(C)(CNC(c2cc(C(N)=O)cs2)=O)C2CCC2)ccc1=O c1(C(N(C2(C3CN(C(=O)CC4CCC5CC45)C3)CC2)C)=O)cc(Br)ccc1N c1(NC(C(C)C)C)cc(N)cc(C(N2CCCCCC2)=O)n1 C1(NC(c2cccc(OC)n2)=O)CCOC12CCN(C(=O)C(O)P(C)(C)=O)CC2 c1(CC)cnn(C)c1C(=O)N(CC(CC)NC(=O)CC(O)Cc1ccccc1)C Cc1cc(O)c(Cl)cc1C(N1CCCC1CNC(=O)Cc1cc[nH]c(=N)c1)=O CC(C)CC(C(=O)NCC1C2CC2CN1C(=O)Cc1ccc(Cl)c(F)c1)C(N)=O c1(C(N2CC(N(C(=O)CSCC(F)F)CC)C2)=O)cnc2c(C)cccc2c1 c1(C(N2C(CNC(CC(C)OC)=O)CCC2)=O)cn(C)nc1C(C)(C)C Cc1ccc(C(N2CCC(CC(=O)N(C)CCN3CCCCC3)C2)=O)n1C CC(C)C(C(=O)N1CCC(C(=O)NCCc2nccc(O)n2)O1)C1CCC1 c1(N2C(C(=O)NCCC(F)(F)F)CCC2)nccc(Br)n1 C1(C2CC2)(N(C(=O)C(O)C2CN(C(=O)CC3CC(=O)C3)C2)C)CC1 c1(C(N2CC=C(CNC(C(C)CC3CCC3)=O)CC2)=O)n[nH]c2c1CC(C)(C)C2 Cc1cn(C)cc1C(N1CC(NC(C2CCC(C(N)=O)N2C)=O)C(F)C1)=O CCCCC(=O)N1CSCC1C(=O)N(CC(C)O)CC.c1(NC(=O)COC)ccsn1 C1(C(=O)OC)CCC(C(=O)NC(C)CN(C(=O)CCCOC2CCOCC2)C)C1 C(=O)(N=c1[nH]cc(C(C)=O)nc1Cl)C1C(C)CN(C(C=CCCCCC)=O)C1 C(=O)(CC1=CCOCC1)NCC1C(C(N(C(CF)CF)C)=O)C1 c1(C(N2CC(C(C)NC(c3csc(O)n3)=O)OCC2)=O)cc2c(ncn2C)s1 C(=O)(C1=C(C)OCCS1)NCC(CC=C)C(=O)NC1COC(C)(C)C1 c1(C(=O)NCCNC(=O)C=C(Cl)Cl)ccc(F)cc1.C12C(C1(F)F)CC(=O)N2 C=CC1COCC1NC(=O)CN(C(c1ccccn1)=O)C(C)C Cc1cccc(C(=O)NCC(C2CCN(C(c3cc(C)n(C)n3)=O)CC2)F)c1C C1(CNC(Cc2cn(C)nn2)=O)CCN(C(=O)C(F)n2cccn2)CCC1(F)F C(=O)(C(C)(C(C)C)NC(=O)CO)NC1C2CC(NC(C3C(CC#C)C3)=O)CC21 C(=O)(C(C(C)CC)N(C)C(C1CCC(=O)O1)=O)N(C1(C#C)CC1)C C1(C(N2CCCC(N(C(=O)COc3cnn(C)c3)CC)C2)=O)CC(=O)OC1(C)C CC(F)(C(=O)N1CC(NC(=O)C(=O)NCC(F)F)C1)c1ccon1 C1(C(=O)NC2(CC)CCOC2)C2CC2CN1C(=O)CC1C(C)(C)C1(C)C C1(F)(CNC(=O)CCc2nc[nH]n2)CC(NC(c2cncnc2)=O)C1 c1(COC)nn(C)c2nc(C)c(-c3nn[nH]n3)c(C)c12.N12CC(OC)(C1)CC2=O C1(CCC(=O)NCC(C2CC2)OC)CN(C(C2CCC(C3CC3)C2)=O)C(C)(C)C1 c1(C(=O)NC(CC)CN(C)C(C2CCC2C(F)F)=O)cscc1SC N1(C(C2C(OCC)CC2)=O)CC(C)CN(C(=O)CCCn2ccnn2)CC1C O=C(C1Cc2ccccc21)NC1CCN(Cc2cc[nH]n2)CC1O c1(C(=O)NC2C(NC(C3C(=C)C3)=O)C2)cnc(OC)c(Br)c1 c1(CC)sc(C(N2CCCC2CCCNC(c2csc(O)n2)=O)=O)cc1C CCCCC(C(=O)NC1(c2ccccc2)CN(C(=O)COC(C)=O)C1)C(=O)O C(=O)(C1CCc2c[nH]nc21)NC1CCN(C(c2n(COC)ncc2)=O)CC(O)C1 c1(C(N2CC(C)(NC(c3cn(C(C)C)nn3)=O)C2)=O)ccc2c(c1)C(C)C(C)O2 C(C(C)NC(=O)CCNC(c1ccco1)=O)(C(C)C)NC(CN(C(C)=O)C)=O c1(C(N2CC3CC2C3CNC(=O)C(F)(F)CO)=O)ccc2n[nH]cc2n1 C=CCCCC(C1CC1)NC(C1CC1CNC(c1ccc(F)cn1)=O)=O C1(CO)CCN(C(c2cccc(C(N)=O)c2)=O)CC1C.C(=O)(C=CC=O)C(C)=O c1(NC(=O)CC2CCN(C(c3ccc([N+](=O)[O-])cc3)=O)C2)cccc2c1CCO2 N1(C(CNC(CCC)=O)=O)CCC(O)(CNC(c2cnccc2OCC)=O)CC1 c1(C(CCC2CCOCC2)NC(c2nnnn2CC)C2C(=C)C2)ncccn1 c1(OC)ncc(C)cc1NC(C1(SC)CCN(C(C2(C)CC3C=CC2C3)=O)C1)=O N1(C(c2cccc(CC)c2O)=O)CC2(CC(NC(=O)C(C)=CC3CC3)CO2)C1 c1(C(N2C(CCNC(C(C#C)(C)C)=O)COCC2)=O)cc2cccc(OC)c2[nH]1 n1(C(C(N2CCC(Cc3ncn(CC)c3)C2)=O)C)nc([N+](=O)[O-])cc1C N1(C(C2C(CCC)CCC2)=O)CCC2CCC(NC(=O)CCCCSC)C12 CC12C3C4C1C1C2C3C41C(=O)NC1CCN(CCNC(=O)Cc2ccco2)C1 C1(C(=O)NC2C(CNC(C=C(C)C3CC3)=O)CC2)CCCc2ccccc2C1 n1(C(C)(C)C)ncc2c1CCCC2NCc1cccc2ncccc12 C1(CNC(C2CC(CNC(=O)COC(=O)CO)C2)=O)Cc2nccn2C1 c1(CC)cnccc1C(N1CCC(CC)C1CNC(C1CC(C)=NO1)=O)=O C1(CC(F)F)C(=O)N1C.C(C(=O)NC1CC1)N(C(=O)COC1CCC1)C Cc1ncn(C)c1C(=O)NC(C1CCN(Cc2cn(C)nn2)CC1)C c1(C(=O)NC2CC(F)(CNC(c3c(C)c[nH]c3)=O)C2)oc(C2CC2)nc1C C1(C(=O)NC2CCC(NC(Cc3c(C)n[nH]c3)=O)C2)CC1C1(C)COC1 N1(C(c2c(CC)onc2)=O)CC2CCCC2(NC(c2ccc(O)c(CO)c2)=O)C1 C(CC1=CCCCC1)N(C(C1(CC=C)CN(C(C2CC(C3CC3)C2)=O)C1)=O)C c1(OC)ccc(F)cc1C(=O)NCC(C)NC(C12CC(C1)C(C(F)(F)F)O2)=O Cc1nc(C(N2CC(N(C(=O)COC3(C)CCCC3)C)C(F)C2)=O)sc1C c1(C(C)CC(=O)NCCN(C2CCCC2)C(C2CCCSS2)=O)ccc(F)cc1 C1(NC(c2occ(C)c2)=O)CN(c2nc(C(C)(C)C)ns2)C2CCCCC12 C#CC1CCCC1NC(=O)C(CN(C)C)NC(=O)CC(CC)OC C1(OC)CCCCC1C(N1CC(NC(=O)CC2(NC(C)=O)CC2)C(O)C1)=O C1(CC=C)(NC(=O)CCn2cncn2)CCN(C(C2CCS(=O)(=O)CC2)=O)CC1 C(C(C)(C)CC(=O)NCC1CC1CC(=O)N(CCO)Cc1ccccc1)OC N1(c2cccc(S(=O)(=O)N3CCC(F)C3)n2)CCCC2(C1)OCc1ccccc12 c1(CNC(c2cn(C)nn2)c2nnnn2CC2CC2)ccc(-c2cnccn2)cc1 c1(C(=O)OCC)c(C)[nH]c(C(=O)NC2CN(C(C3C=CCC3)=O)CC23CC3)c1C N1(C(CCCCC#C)=O)CC2(C(=O)NCC(C)CN(C)C)CC1CCO2 S(=O)(=O)(c1ccc(F)c(F)c1F)N(C)CC1CN(Cc2c(O)cccc2Br)C1 c1(CN2CCC(C(=O)Nc3onc(C)c3Br)C2)cc(Cl)cc(Cl)c1Cl C(=O)(C1=C(C)OCCS1)N(C1(C2CCCN2C(=O)C(C)C#N)CC1)CC C12(C(=O)Nc3c(COC)c[nH]n3)CC1CN(C(C1CC=CCC1C(F)(F)F)=O)C2 c1(OC)cnc(C(=O)NC(C2CN(C(=O)C=Cc3ccccn3)C2)C)cn1 C=C(C)CC(C)C(=O)NCCNC(=O)C(S(N)(=O)=O)c1ccccc1 CS(=O)c1ccccc1C(=O)NCC12CC1CN(C(c1ccnn1C1CC1)=O)C2 C(=O)(C(C)NC(c1ccco1)=O)NCCN(C(=O)C=C1CC1C(F)(F)F)CCC c1(C(=O)NCC(CO)NC(c2c(C)nsc2)=O)cnc2n1CCOC2 c1(CO)ccc(NC(c2cc(Cl)sc2Cl)c2nnnn2C2CC(F)(F)C2)cc1F C1(C(=O)NCCN(C(=O)Cc2csc(C)n2)CC)CCCCC(C)(C)C1 C12(CNC(c3cc(F)ccc3F)=O)CCC(CC1)N(C(=O)C(F)=CCCF)C2 N1(Cc2cn(CC)nc2)CCC2(CCN(C(=O)Cn3ccc(C)cc3=O)CC2)C1 C(=O)(CCCC(C)(F)F)N1CC(C(C(=O)NC2CCCCCC2CO)OC)C1 c1(OC)c(C(=O)NC2CCCCN(CC(c3ccccc3)O)C2)ccnc1F N1(C(CCOCC(C)(C)C)=O)CC(NC(=O)CCC2CCCOC2)CC(F)C1 N1(C(CC)=O)CCC(C)(CNC(=O)CCc2scnc2C)C1 c1(C(N(C2CCN(C(=O)Cc3occc3C)CC2)CC)=O)cc(C#N)ccc1Cl N1(c2cc(OC)nc(C)n2)CC2(CCC(NC(c3ncn(C)n3)=O)C2)C1 CCCC(CC)C(=O)NC(c1ccccc1F)CNC(c1cnc(S)[nH]1)=O C(=O)(C#CC1CCOC1)NCC1C(NC(C=CC(=O)OC(C)(C)C)=O)C1 C1(C(=O)NCCN(OC)C)CN(C(=O)C=Cc2nccs2)CC12CCC2 N1(CCNC(=O)Nc2ccc(Oc3ccccc3Cl)nc2)CC2CCC(C1)O2 c1(C(=O)OC)sccc1COC1CCOC1.C1CCN(C)C(=O)CO1 C1(CC(=O)NC2CCN(C(C=C3CCC(C)CC3)=O)C2)CCOCC1(C)C C(=O)(C(CO)C(F)(F)F)N(CCCC(=O)NCc1c(SC)csc1)C c1(CN2CCN(C(C)CC3(C(F)(F)F)CC3)C3C2C3)c2cc(Br)ccc2nn1C N1(C(C(C)(O)C2CC2)=O)CCC2(CCC2)C(NC(C2CCC(F)C2)=O)C1 c1(C(=O)NC2CCC(CNC(Cc3cc(OC)no3)=O)C2)cc(F)c(F)c(F)c1 C1(NC(COC2CN(C(C(C)(F)F)=O)C2)=O)CC2OCCCC12 CC(C)CC(O)C(C)C(=O)N(C)CC=CC(=O)NC1(C)CCC1 c1(OC)ccc(C(C)(C)C(=O)N2CCCC2c2n[nH]c(C)n2)cc1Br CC(C)(C)C(O)C(=O)N1CCC(CN(C(=O)CCC(F)F)Cc2cccnc2)C1 C(CCCCNC(c1[nH]nnc1C1CC1)=O)NC(=O)COC1CCCOC1 C(=O)(C(CO)C(F)(F)F)NC1(CC=C)CCN(C(C2CC3(C2)CC(C)(C)C3)=O)C1 C1(CC)CCCCC1C(=O)NCCCCNC(=O)C(C)(C)c1ccncc1 C1(C(=O)NC(C)C(C)(C)NC(c2ccc(O)nn2)=O)CCN(C2CC2)S1(=O)=O C(=O)(C(C)CCCc1ccccc1)N1CCC(C)(CNC(C=CCCC)=O)C1 C(C(CCN=c1[nH]c(=NCC2(OC)CC2)[nH]c2ccccc12)C(C)C)OC C(c1cc(Br)ccc1-n1cccn1)=NC(c1ccc(C)cc1)CC CCCCS(=O)(=O)CC(=O)NC1C2CC1N(C(=O)Cn1cc(C(F)(F)F)nn1)C2 c1(CN2CC3CC2CN3Cc2cccc(C(=O)O)c2F)ccc2nc(O)[nH]c2c1 c1(C(N2CCC(CCOC)(NC(=O)CSC)C2)=O)coc2ccc(Br)cc12 N1(C(COCC#C)=O)CCCC(C)(CNC(c2ncccc2C)=O)C1 C(=O)(CCCN(C)C)NCCC(C)NC(c1cccnn1)=O N1(C(C(C)NC=O)=O)CC2CCCCC2(CNC(c2c[nH]c(C#N)c2)=O)C1 N1(C(c2scc(C)c2)=O)CC(CCNC(=O)C=CC(=O)NC2CC2)C(C)C1 c1(C(=O)OCC2CCN(C(C3(CC)CC(=C)C3)=O)CC2)nc2cccnc2s1 C1(C(=O)NCC2N(C(C#CC(C)C)=O)CC=C2)CCc2cnn(C)c2C1 c1(CC)ccc(C)c(C(=O)NC2COCC2NC(C2(C)CCCC2(F)F)=O)c1 C1(C#N)(C(=O)NC(CCNC(Cc2cccc(OC(C)C)c2)=O)C)CC2(CC2)C1 C1(F)(C(N2CC(n3cc(-c4nncc(C)c4)nn3)C2)=O)CCS(=O)(=O)C1 C1(NC(CN(CCCCCC)C)=O)CCC(CNC(=O)CC(F)F)CC1 N1(C(c2cc(Br)cs2)C(=O)NC)CCC(c2cn(CCC(C)(C)C)nn2)CC1C CC1CN(C(C2CC(C)(C)C2)=O)CC2(CCN(C(=O)C(F)(F)c3nccs3)C2)O1 CS(=O)CCCC(=O)C=CCC(C)(C)N.C1(C)(C)CNC(=O)C1 CC1(C)CC(NC(C2(C)CCCNC2=O)=O)CCN(C(=O)COC2CCCC2)C1 CC(=O)CCN=C(NCC1(CO)CCCO1)N1CCN(c2ncc(F)cn2)CC1 CC(=O)CCCC(=O)NCCC1CC(NC(c2cn3c(n2)SCC3)=O)C1 C1(NC(c2cc(CCC)oc2C)=O)CN(C(C2CC(F)C2)=O)CC12CC2 N1(C(COC(CC)C)=O)CC2CC(C1)N(C(c1cnc(-c3cccs3)s1)=O)C2 N1(C(c2cocn2)=O)CCN(C(=O)Cc2cncnc2O)C2CCCCC2C1 N1(C(C(C)C)=O)CC(NC(C23CC(CN2C2CC2)C3)=O)CC12CCCCC2 N1(C(N(CC(C)(C)O)C(C)C)=O)CC2(COCS(=O)(=O)C2)C1 C(=O)(C(C)(CNC(=O)COc1ccsc1)CC)NCC1N(CC)CC1 N1(C(C(C)C)=O)CCCC2CN(C(c3cc(-n4ccnc4)ncn3)=O)CCC12 N1(c2ncnc(C)c2Br)CCc2sc(C(=O)NCCC3CCOCC3)cc2C1 N1(C(CC(CC=C)(C)C)=O)CC2CC3CC2C1C3NC(c1scc(C)c1C)=O c1(C(=O)NC2C(CNC(C(C)NC(CC)=O)=O)CC2)cnn2c1NCCC2 c1(N2CC3CN(c4ncc(COC)cn4)CC3C2)nc2c(cc1C#N)CCOC2 CC1OC2(C(=O)NC3CN(C(c4ccc5oncc5c4)=O)CC3O)CCC1CC2 N1(C(C2CCN(C(CC(C=C)CCC)=O)CC2(C)C)=O)CC(C)OC(C)(C)C1C Cc1ccc2nc(C(N3CCN(C(=O)Cc4occc4C)C(CO)C3)=O)cn2c1 C1(SCC)CCC(C(=O)NCCCCCCNC(c2nocc2C(C)C)=O)CC1 c1(OC(c2ccccc2)=O)cc(C)c(O)cn1.C(=O)(CC1N(C(C)=O)C1=O)OC C1(Nc2ccc(C3CCC(=O)N3)cc2)CCC2COCCC2C1 c1(C(C)C)ncc(Cl)c(C(=O)NCCCCNC(c2ncncc2F)=O)n1 c1(C(N2CC(CC(N3C(NC(N)=O)CC3)=O)C2)=O)cccc(CCO)c1 CC1CCCCCCN1C(=O)NC1CC2CC1CC2CO C1(C)(CC)CC(NC(c2cccc(C)c2)=O)CN1C(C1CCN(C)CC1)=O C1(NC(C2CCC(=C)CC2)=O)CCN(CCc2scnc2C)CC1C c1(C(N(CC)CC2CCN(C(=O)CC3C=CCCC3)CC2)=O)cnc(O)c(F)c1 Cc1cc(C#N)cc(C)c1C(=O)NC1CC(CCNC(=O)Cn2nccc2C)C1 N1(C(c2sc(C(=O)OC)c(C)c2)=O)CCCC2CN(C(C3CC(O)C3)=O)CCC12 C1(C#CC(=O)NCCOC2CN(C(c3cc(C(F)F)[nH]n3)=O)C2)(CC)CC1 C1(CCNC(COCCOC)=O)CN(C(=O)COc2ccsc2)CCCO1 c1(CCCNC(=O)NC(CCCC)CC)cccc2scnc12 N1(C(c2c(C)nn(C)c2)=O)CC2(CCCCN2C(C2(O)CCSCC2)=O)C1 c1(C(N2CC(CNC(c3cccc(SC(C)(C)C)c3)=O)C2)=O)cc(F)cc(F)c1 N1(C(c2c(OC)nsc2OC)=O)CCC(CNC(c2cc(C)[nH]n2)=O)C(F)(F)C1 C#CC1CN(C(C2CCN(C(c3cc(C)sc3C)=O)C2)=O)CCO1 c1(CC(=O)NCC2CN(C(=O)C(F)=CC3CC3)C2)cc(Cl)ccc1O c1(C(N(CCNC(C(N2CCNC2=O)C)=O)C2CC2)=O)ccc(O)c(CO)c1 C1(CNC(C=CC=CC)=O)CN(C(c2cc(F)c(F)cc2F)=O)CCC1(F)F CC1CC(CN2CCC2c2ccsc2)CN1.N1(C(=O)N)CCCC1 CC1(C)OCCC1NC(C1CC(CCNC(=O)CCN2CCCC2)C1)=O C12CCCN(C1)CCC(=O)Oc1c(cccc1)NC2=O.N1(CC)CC(O)CC1C O=C1NCC(C(=O)N(C2(C(=O)NC3(CCF)CCC3)CCC2)C2CC2)N1 C=C(C)CCCC(=O)N1CC(CC(N2CCC(OC)C2(C)C)=O)C2(CC2)C1 N1(c2ccnc(C(C)C)n2)CCC(NC(=O)C(C)NC(c2ccco2)=O)C(C)C1 C1(CN(C(C(C)NC(C)=O)=O)C)COCCN1C(=O)CN1C(=O)CNC1=O C(=O)(C(F)(CNC(=O)C(c1cnn(C)c1)=O)C(C)C)NCC(=C)Cl C(=O)(CCN(OC)C(=O)C1(F)CN(C(=O)C(OC)OC)C1)NCC Cc1cccc(COCc2nc(CNC(=O)CC(C)C)cs2)c1.C1(C)C(=O)O1 CC1(C)CN(C(=O)CC2(NC(N)=O)CC2)CC(C(=O)NCc2cccc(F)c2)O1 c1(CC(=O)NCCCNC(C2N(CCC)CCCC2)=O)cc(F)ccc1Cl CSC1=C(C(=O)N2CCC(O)(CNC(C3CCC(O)C3)=O)CC2)CCCC1 C1(N(C(CCC2CCC(NC(CC3ON=C(C)C3)=O)C2)=O)C)CCCCC1(C)C CC1CN(C(C23CCC(C2)C3(C)C)=O)CCN1C(c1cn2c(n1)CCC2)=O N(C(=NCC1CCC2(CCC2)O1)N(C)Cc1cc(Br)cn1C)C(C)C Cc1ccc(C=CC(N2CCN(C(=O)CC(C)(C)F)C(C3CC3)C2)=O)cc1 NS(=O)(=O)c1ccc(C(=O)NCC2CC2NC(=O)C=Cc2cscn2)c(C)c1 C(=O)(C(C(C)(C)C)OC)NCC(C(=O)NCc1c(OC)cccc1)O C1(CNC(c2cc(C)[nH]n2)=O)CCCC2(CN(C(=O)CN3CC4CC4C3)C2)O1 c1(CNC(C2CC(F)CN(C(c3sccc3Cl)=O)C2)=O)ccc(CO)cc1F N1(CC(=O)Nc2c(NC(N)=O)cccc2)CCCC(O)(CO)CC1 c1(C(=O)NC2CCCC(NC(c3ccc(C)nc3)=O)C2)ccc(Cl)c(O)c1 CC1(C)CCCN(C(C2CCC2C(C)(C)C)=O)C1C(=O)NC1(C)CCCC1(F)F C1(C(=O)NCCN(CCC)C(C2(C)CCCC2)=O)CCC(C(F)(F)F)O1 CC(C)C(CNC(=O)C(C)(C)C1(O)CCC1)C(=O)NC1(CCCCO)CC1 CCC(C)(CNC(c1cc(OC)ns1)=O)C(=O)NCCN(C)C1CC1 N1(C(CC2CCCN(C(C3(C#C)CC3)=O)CC2)=O)CCCCC(C)(C)C1 CC1CC2CN(C(c3ccc(=O)n(CCO)c3)=O)CC2N1C(=O)C(O)CF N1(C(C(CC)C(C)C)C(=O)NCCCOC)CC(C)(C)OC2CCCC12 C(=O)(C(C)CS(C)(=O)=O)NCC12N(C(C3(COC)CC3(F)F)=O)C(CC1)CC2 N1(CC(=O)NCCN(C(c2onc3ccccc23)=O)CC)C(=O)NC(C)(C)C1=O C1(NC(C2CC3(C2)CC3(F)F)=O)CCCN(C(c2cccnc2C(F)F)=O)CC1 N1(C(C(CC=C)(C)O)=O)CC2(C=C(C(=O)NCC(C)CC(F)(F)F)CO2)C1 C1(C)(CC(=O)NCC2CCN(C(C)=O)C2)CCN(C(=O)Cc2cnc(C)s2)C1 O=C1NCCN(C(C2CSCCN2C(C2CCC(O)CC2)=O)=O)C1CCO Cc1snc2sc(C(N3CC(C)(NC(=O)CC4COCCO4)C3)=O)cc12 C1(CNC(C2(C)CCCC2)=O)CN(Cc2cc(C(F)(F)F)cc(Cl)c2)CCC1O c1(CC)cccc(C(N2CC(O)CC2CNC(=O)CC(C)(C)SC)=O)c1 N1(C(CC(C(=O)OC)C)=O)CC(n2cc(C(C)(C)SC)nn2)C(S(C)(=O)=O)C1 c1(C(N2C(C)CC(NC(c3ccc(C4(C)CC4)cc3)=O)C2)=O)cc2n(n1)CCO2 c1(C(N2C(CNC(C(CC)=CC)=O)CC2)=O)ccc(F)c(C(F)(F)F)c1 C1(CC(=O)NCCC2CCN(C(c3cnco3)=O)C2)CCC2(CCC2)CO1 C=CC1(NC(=O)CC2C3CN(C(C45CCC(C4)C5)=O)CC23)CCCCC1 c1(C(=O)NC2CC(NC(C3(C)CC3(F)F)=O)C2)ccc(-c2cncnc2)cc1F C1(C(=O)NC(C)C(N2CCN(C)CC2)=O)CC(=O)N(C)C1c1cccs1 C=CC(CCC)CC(=O)NCC12CC(NC(=O)CCNC(=O)C=CCl)(C1)C(C)O2 O=C(C1=CCCCCC1)NCC(C1CCOC1)NC(=O)CC1(CO)CC1 C(C(C)(C)CCO)NC(C(C1CN(C(C2OCCC2C)=O)C1)OC)=O CN1CC(NC(=O)C(C2CC2)NC(=O)CC2CSCCO2)C2(CC2)C1 C1(NC(C2C(C=C)C2)=O)CN(C(=O)CCCc2nc(C3CC3)no2)CC1OC c1(C(N2CC(CNC(C(C)=C(C)C)=O)C(C)(C)C2)=O)cc2c(F)cc(Cl)cc2[nH]1 C1(C(=O)NCC(CC2CC2)CO)(CC)CCN(C(c2cscc2C)=O)CC1 c1(C(N2CCC(N(C(C3C(C=C)CC3)=O)C)CC2)=O)ccc(C)c(F)c1 N1(C(C(CCN(C)C)O)=O)CC(NC(=O)CCc2cnco2)CC(O)C1 C1(C(N2CC(OC)C(C(=O)NC34CCCC3C4)C2)=O)CC(C2CC2)=NO1 C=C(Cl)CC(C(=O)NCCc1cnn(C)c1)NC(=O)CC=CC(C)(C)C c1(C(N2CCOCC2CC(C)O)C(=O)NCC)cc(COC)ccc1OC C1(CNC(=O)C2CC2)CC(NC(=O)Cc2ccc(I)cc2)CC1O N1(C(CCNC(C)=O)=O)CCC2(CCN(C(c3cc(O)c4ccsc4c3)=O)C2)C1 C(=O)(C1COc2ccccc21)N(CC(c1ccccc1)O)CC(=O)NCC(F)F c1(N(C(=O)NCC(C)Oc2ccccc2Br)C)cccc(Br)c1Cl CCC(C)CC(C(=O)NC(CC1CC1)C(=O)NC)NC(c1cc(C)sc1C)=O c1(C(=O)NC2C(NC(C=CS(C)=O)=O)CCC2)ccc(C(F)(F)F)nc1N Cn1nccc1C=CC(N1CCCC1C1CCN(C(C2(C)CNC(=O)N2)=O)CC1)=O N1(C(c2c(C)scc2)=O)CC2ON=C(CNC(=O)C=CC3CCC3)C2C1 c1(C(=O)NCC(CN(C)C(C2CC(F)CN2C)=O)O)cnc2cc(O)ccc2c1 C12(C(=O)NC(C3CN(C(CC4CC(OC)C4)=O)C3)C)CCC(C(F)(F)F)(CC1)C2 c1(OC)ccc2cc(C(=O)NC(C)CC(C)NC(=O)CC(O)CN(C)C)[nH]c2c1 N1(CC(=O)NC(CNC(=O)C(F)(F)c2cscn2)CO)C(=O)CCC1=O c1(N(C)C)ccc(C(=O)NCC2(NC(=O)CN3CC4CC4C3)CCOC2)cc1 C=C(C)CC(C(=O)N1CCN(C(=O)C(c2cnn(C)c2)C)C(CC2CC2)C1)OC C1(CCNC(C(C)=CC)=O)(OC)CN(C(c2cnc(-c3ccncc3)s2)=O)C1 C1(C(N2CC(OC)C(F)C2)=O)CCCN(Cc2cc(O)cc(F)c2)CC1 Cc1c(C(N2CC(NC(=O)CSc3ncccn3)C(C#N)C2)=O)ccc(F)c1F c1(C(=O)NCC(CN(C)C(C2CCCN2C)=O)O)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NCCC2CCN(C(c3c(C)cncc3)=O)CC2)ccnc2[nH]cnc12 N1(CC(c2ccccc2)OC)CC2CCCN(C(c3csc4nccn34)=O)C2C1 N1(C(C(CCC#C)NC(c2coc(CO)c2)=O)=O)CCCC2(CCCO2)C1 N1(C(c2c(CC)c[nH]n2)=O)CCC(NC(=O)C(N2CCC(CC)CC2)=O)CC1C C1(NC(=NCC)NCCSc2cccc(C(F)(F)F)c2F)COc2nccn2C1 c1(C(=O)NC2CN(C(CN(C(C)=O)C)=O)CC(C)C2)cnn2ccn(C)c12 C1(COC)CCC(C(=O)NCCN(C)C(=O)C2CC2)C1 c1(NC2CCC(C(=O)O)(COC)CC2)cnc2c(c1)CNC2=O c1(SC)cccc(N2CC3CC(NC(C4(S(N)(=O)=O)CC4)=O)CC3C2)c1[N+](=O)[O-] C1(CNC(C(C)OCC)=O)CCCC2CN(C(=O)Cc3nc(C)no3)CC12 Cn1nc(C(=O)NC2CN(C(=O)C=Cc3cnc[nH]3)C(C)(C)C2)c2ccccc12 CC(C)(CC(=O)NCCN1CCCN(C(C2CCC23CCCO3)=O)CC1)C(F)F C=CCC(C)C(=O)N(CCCN(C)C(c1cccc(OC(C)C)n1)=O)C c1(C(=O)OC(C(=O)OCC=C)C(C)C)cc(C(C)C)nc2c1cnn2C(C)C C(=O)(CCCCCCCCCO)NC(C)CNC(C12CCC1C2)=O CCCCC(F)C(=O)N1CCN(C(=O)CNC(c2cc(SC)c(C)o2)=O)CC1 C(=O)(CC(C)C(=O)NC1CCCC1C(N1CC(C)(C)C1C1CC1)=O)OC c1(C(C)CC(=O)NCC2(NC(=O)CN3CCC(F)C3)CCCC2)ccc(F)cc1 C1(C(=O)NC2(CF)CN(C(Cc3ncc(C)[nH]3)=O)C2)CCOC(C)C1 c1(C(CC(=O)N2CC(NC(CCC(=O)OC)=O)C2)C)cccc(F)c1 c1(C(N2CC(C(C(=O)NC3CCNC3=O)OC)C2)=O)cnn2cccc2c1 N1(C(COCCCCC)=O)CCN(C(C2(SC)CCC2)=O)CC1CC1CC1 Cc1cc(=NC(=O)C2CC(F)CN(C(c3ccc4cnc(C)n4c3)=O)C2)[nH]n1C C(=O)(C(C)(C)F)NCCOCCN(C(C(C)OCCC=C)=O)C Cc1cc(=NC2CCN(C(c3cc(C(F)F)ncn3)=O)CC2C)[nH]c(C2CC2)n1 C1(F)(C(=O)NCC#CC(=O)Nc2cnn(C(F)F)c2)CC=CCC1 Cc1cc(CC(C)Nc2cc(NC(C)Cc3ccccc3F)ncn2)cc(C)c1 N1(C(CC(CC)SC)=O)CC2CC(CNC(c3cccc(OCCF)c3)=O)C2C1 C1(OC)CN(c2cc(SC)nc(C)n2)CCC1NC(c1cc(F)ccc1O)=O CC1CCc2c(C(=O)NC3CCN(C(C4CC4(Cl)Cl)=O)C3)csc2C1 C=CC(C)(CC)C(=O)N1CCCCC(CNC(=O)C(C)OCCC(C)C)C1 C1(NC(=O)C=Cc2ccco2)CCOC12CCN(C(=O)C=Cc1cccs1)CC2 C(=O)(CC(=O)NC)N(C1CCN(C(c2snnc2C(C)C)=O)C1)CCC C1(S(C)(=O)=O)(C(=O)NCC2CC(OC)CN2C(c2sncc2C)=O)CCCC1 c1(C(C)NC(CC2C(NC(C(CO)OC)=O)CCC2)=O)ccc(C)cn1 CCCCC(C)CCC(=O)NCCN1CCN(C(=O)CCCOC(C)C)CC1 C1(C(C)C)CCC(C(=O)NCC(C2(O)CN(C(C3CC(C)CO3)=O)C2)(C)C)CC1 c1(C(=O)NCC2N(C(C3CC(OC)C3)=O)CCC2)cccc(C)n1 C(=O)(CCS(N)(=O)=O)NC1CCN(C(c2c(OC)c(C)sc2)=O)C1 C1(c2nc(C(C)C)on2)CCCCN1C(=O)NC(CCO)c1ccco1 CC(C)(C#N)CCCC(=O)NC1CN(C(C23C=CC(CC2)C3)=O)CC1C1CC1 c1(C(N2CCN(C(c3ncc(C)cn3)=O)CC2CF)=O)ccc(C#N)cc1O C(=O)(C#CC1(C)CCCO1)NCCC(C(C)C)NC(c1ccc(CC)c(Cl)c1)=O c1(C(N2CC(C(=O)NC(C3CCOC3)C)SCC2)=O)cc(Br)cc(F)c1F C1(CCNC(c2n(C(C)C)cnc2)=O)CCCN(C(c2c(C)ncn2O)=O)CC1 C1(NC(C(CC2CCCCC2)OC)=O)CN(C(=O)C(C)C#N)CC1C c1(OCC(C(=O)N(CC)CCNC(C(CC)N(C)C)=O)(C)C)cccc(C#N)c1 c1(C(N(C2C3CN(C(C(C)NC=O)=O)CC32)C)=O)cc2nc[nH]c2cn1 C1(CNC(C(CC)O)=O)CCN(C(=O)CCCCNC(N)=O)CC1 N1(C(c2n(CCOC)cnn2)C(=O)NC2CCCCC2)CCC(C#N)CC1 CC1(C)C(NC(=O)C(=CC2CCCCC2)F)CC1CNC(c1cncc(Cl)c1)=O c1(OC)ccc(N)c(C(=O)NCC2CN(C(C3CC4CC4C3)=O)CC2C)c1 C(=O)(C1Cc2ccc(F)cc21)N(C1CCCN(C(c2c(CC)nc(C)s2)=O)C1)C c1(C(N2CC3C(NC(=O)Cn4ccnn4)C3C2)=O)ccc2sncc2c1 Cn1cnc(C(N2CCC(CNC(c3c(C(F)F)cnn3C)=O)C2)=O)cc1=O C1(CNC(c2ncn(C(C)(C)C)n2)=O)CC(C2CC2)C1 Cc1nn2c(c1CNC(=O)C(O)CC(F)(F)F)CN(C(=O)C(C)S(N)(=O)=O)CC2 c1(NC(C(c2ccccc2)C)C2CC2)nc(Br)nn1C C1(C(NOCC(=O)NC2CC(=C)C2)=O)CCOCC1(C)C C(C)(C)(CCC(=O)NCc1ccccc1O)NC(c1ccc(CC)cc1)=O c1(NC(C(CC)C)(C)c2nnnn2Cc2ccc(OC)cc2)c(C)cccc1F c1(NC(C(c2ccoc2)NC(Cc2c(C)n(C)cn2)=O)=O)ccc(O)cc1F c1(OC)cnc(CNC(C2CCN(CCCCC3CCOCC3)C2)=O)cn1 N1(C(C2(COC)C=CCC2)=O)CCC2(CC2C(=O)NC2(C)CCC3(CC2)CC3)C1 C1(CNC(CN(CCOC)C(C2OCCC2C)=O)=O)CCCC1C(C)C C1(C(=O)NC2CC(CCC(N)=O)C2)CN(C(C2CC3CCC2C3)=O)CC12CC2 c1(C(N2C(CCNC(c3n(C)nnc3)=O)CCC2)=O)cc(C#N)n(C)n1 N1(C(=O)CNc2ccc(Cl)cc2Cl)CCN(C(c2ncc[nH]c2=O)=O)CC(O)C1 Cn1[nH]c(=NC(=O)C2CC2NC(=O)Cc2cc(F)ccc2F)c2c(Cl)cccc12 C12(NC(=O)C(O)C3CC3)CCN(C(C3CCN(c4ccccn4)CC3)=O)CC1C2 N1(C(Cc2ccn(CC)n2)=O)CC(OC)C(OC)C1CNC(=O)C(O)C1CCC1 Cc1cc2ccc(C(=O)NC3CCCCC3N(C(=O)C(=O)NC(C)C)C)cn2c1 CC1Oc2c(C(=O)NCCNC(c3ccnc(C(C)(C)C)n3)=O)cccc2C1C C1(NC(C(CCCC)O)=O)CC2CN(C(=O)CC(O)c3ccccc3)CC2C1 C1(C(=O)NC2CCN(C(c3ccc(C(C)C)o3)=O)C2)C2CCN1CC2 c1(C(N2C(C)(CNC(C(CC#C)C)=O)CCC2)=O)cc(OC)ccc1[N+](=O)[O-] C(C)(C)(CCC(=O)NC1C=CCN(C(c2ccc(C(=O)N(C)C)cc2)=O)C1)OC c1(C(=O)NC2CCCCN(C(CC(C=C)CC)=O)C2)ccsc1S(N)(=O)=O c1(C(=O)OC)cncc(C(N2CC(F)(CNC(=O)C(C)Cc3ccco3)C2)=O)c1 C(=O)(CC(C)C(C)C)NCC1(O)CCN(C(c2n(CCOC)ncc2)=O)C1 N1(C(c2cc(CC)[nH]n2)=O)CCN(Cc2cc(F)c(I)c(F)c2)CC1C#N C1(NC(C(C)(C)OC(CCC)=O)=O)CCN(C(C2COCC2C(N)=O)=O)CC1 C1(NC(c2cc(C)nc(C)c2)=O)C(C)CN(C(c2cnc(O)o2)=O)CC1C c1(C(=O)NC2CCCN(C(C=NOC)=O)C2)ccc2nc(CO)[nH]c2c1 C(=O)(CCCC(F)(F)Br)NC1CCN(C(c2c(CC)non2)=O)C(C)C1 c1(C(=O)NCC(C(=O)NCCCN(C)C)CC2CCCC2)cn2ccnc2cn1 CC#CCCCC(=O)NCCN(CCCCCC)C(C1CCC=CCCC1)=O C1(CNC(c2onc(CC)n2)=O)CCN(C(C23CC2COC3(C)C)=O)C1(C)C C1(C(=O)NCC2CC(OCCO)C2)(OC)CCN(C(=O)CNC=O)C1 C1(C(=O)NC2(C(C)C)CC2)CC(=O)N(CCNC(=O)C(C)C2CCCO2)C1 C(=O)(C(C)(CC)C(N)=O)N1CCN(C(c2nc(COCC)sc2)=O)C(CF)C1 N1(C(c2ccnc(OC)n2)=O)CC(NC(=O)CCc2ccn(C)n2)CCC1C c1(NCC)ccccc1C(=O)NCC(=O)NCC1CCCN1C(c1cscn1)=O C1(CNC(C2(OC)CCSC2)=O)COCCN(C(=O)Cc2c(Cl)cnn2C)C1 C12(CNC(=O)CCCCO)CC(CO1)N(C(C1CC1Cc1ccc(F)cc1)=O)C2 C1(C)(C(N2C(CCC)(CCC)CCC2)=O)CC=C(C)CC1 Cc1cc(C(=O)NCC(C)(C)OCCNC(=O)CC2OCCC2C)cc(O)n1 N1(CCCNCc2cccc(OC(C)(C)C)c2)CCS(=O)(=O)CC1 C1(OC)CC(CO)N(C(C2CCN(C(=O)Cn3ncnn3)CC2)=O)C1 CN1C(=O)CN(CC(=O)NCCC2CCN(C(=O)Cc3ncc(Cl)s3)C2)C1=O C(=O)(C(O)CC(F)(F)F)N(C1CCN(C(C(C(C)C)C2CCC2)=O)CC1)C1CC1 c1(C(N(C2CCCCC2)C)=O)cccnc1.N1(CCN(C(C)C(=O)O)C)CCOCC1 C(=O)(C1=CCCCCC1)N1CCC(NC(=O)Cc2n[nH]cc2Br)C(O)C1 C(=O)(C(O)C(C)(C)C)N(C)CC1C(NC(CC2(OC)CCC2)=O)CCC1 C=CCC(C)(C)CC(=O)N(C1CN(C(=O)C(Cl)=CCl)CC1(C)C)C c1(COC(N2CC(C(=O)OCC)CC2C2CC2)=O)nc2c(s1)CC(C)(C)CC2 N(C1c2ccccc2CC1NC(=O)CCCC1CC1)C(C(C(C)O)N(C)C)=O Cc1cc(C(=O)NCC2C3CC2N(C(c2nn(C)cc2Cl)=O)C3)nc(C)c1 C1(C(=O)NC(CCC)C2CCCC2)CN(C(c2sc(C)nc2C)=O)CCO1 C(C(CC(C)C)C(=O)NC1CCCC1(C)N(C)C)NC(c1c(C)[nH]cc1)=O N1(C(C2C(C(C)C)CC2)=O)CCOC(CN(C(=O)COCC2(F)CC2)C)C1 N(C1c2ccccc2CC1NC(C1CCCC12CC2)=O)C(C(CCC)OC)=O c1(CC(=O)OC)nc(C)cn2cc(-c3ccc(C=O)o3)cc12 c1(SCC)cc(C(=O)NCC2CC2CNC(C2CCCC3(CC3)C2)=O)ccc1C N1(N2C(C)CCCC2)CCN(C(=O)CO)CC(C)(F)C1.n1(CC)cnc(C=O)c1 Cc1oc(-c2ccccc2)cc1CC(=O)NC1CN(CC=CCNC(N)=O)CCO1 c12cc(cc(F)c1)C(=O)N2.c1(NC(C2C(C(=O)OCC)C2)=O)cscc1C(C)C c1(C(N2CCSCC2)=O)ccc(C(N2CCCC2c2ccc(F)cc2)=O)nc1 CC1CC(c2nnnn2Cc2ccccc2)(NC2(C)CC2)CC(C)S1 C1(C)(CNC(=NCC(C)OC)NCC2CCOC2)CCCC(F)(F)C1 c1(CCC(=O)NCCN(C2CCCCC2)C(C2C(C#N)C2)=O)ccccc1F Cc1cccc(NC(=O)NCC(=O)NCCC2CCN(C(=O)CS(N)(=O)=O)C2)c1 N1(C(COCC)=O)CCC2CN(C(c3cnc(O)c(Cl)c3)=O)CC2C1 Cc1ccc(C(N2CCCCC2C(C)NC(=O)Cc2ccccc2C)=O)cc1C C(=O)(C1=CC2CCCC12)NCCC1CCCN(C(C2(C(C)C)COC2)=O)C1 N1(C(CCNCC)=O)CCN(C(=O)CN(c2ccccc2)C)C(CCOC)C1 C1(C(C)C)CCC(C)CC1CNC1CCNC1c1ccccc1 C1(NC(C(C)(C)C)=O)CC2(CCCN(C(c3ccnc(OCC4CC4)c3)=O)C2)C1 c1(CC)cc(C(N2CCOC(C(C)NC(C3CN(CC(C)C)C3)=O)C2)=O)nn1C c1(CC)cc(F)c(C(=O)NCCCN(C(=O)CCNC(=O)CO)CC)cc1F CC1(C)CN(C(=O)C(O)C(F)F)CCC1NC(c1ncn(-c2ccccc2)n1)=O CCC(F)(F)C(C)(C)C(=O)NCC(C)CNC(c1cnn2cc(C)cnc12)=O N1(C(CCCC=C)=O)CC2CCC(CNC(c3ccn(CC)n3)=O)C2C1 c1(C(=O)NC(CCOC)CNC(C2C(Cl)(Cl)C23CC3)=O)c(F)ccc(C)c1Cl N1(C(Cc2c(C)nc(S)s2)=O)CCCN(C(C2CCCCS2(=O)=O)=O)C(C)C1 N1(C(CCOCC#C)=O)CCC2(CCCN2C(c2ccnn2CCCC)=O)C1 C=CCCN=C(NCc1coc(C)c1)NCC1CCC(C)O1 CN1C2CCCC1CN(C(C1NCC3CCC1C3)=O)C2 c1(C(N2CC(NC(C(N3CCCCCC3)C)=O)C(C)C2)=O)csc(=NC2CC2)[nH]1 N1(C(c2ccnnc2)=O)CC2CCC(C1)N2C(c1c(O)cccc1F)=O C1(C2CCN(C(=O)Cc3cnsc3)C2)(NC(C(C)Cn2cccn2)=O)CC1 C1(NC(c2cc(C)c(C)nn2)=O)CCC2CC1CN2C(C1(C2CCC2)CC1)=O CCC(CCCC(=O)NC1CCOC12CCCC2)NC(c1cnn(C(C)C)n1)=O N#Cc1cc(C(=O)NC2CN(C(=O)CC3(N(C)C)CCOCC3)C2)cc(F)c1F c1(OCC(=O)NCC(CNC(c2nn[nH]c2Cl)=O)CO)ccccc1O N1(c2c(F)cnc(C)n2)CCC2(CCCCC2NC(C2(c3cccs3)CC2)=O)C1 N1(C(C2C(C)(C)C2(F)F)=O)CC(NC(=O)CCn2cc(Br)cn2)CC1(C)C c1(OC)ncccc1C(=O)NC(C(N1CC(N(C)OC)C1)=O)C1CCOC1 C#Cc1c[nH]ccc1=NC(=O)NC1CC1c1ccc(F)cc1 CC(C)CC(C(=O)N1CC(O)C1)NC(=O)CCn1cnnn1 C(CC(=O)N1CC(C(N)=O)(OC)C1)(C1CC1)NC(CC1CC(N(C)C)C1)=O CC(C)C(C(=O)N(CC(C)(C)NC(=O)CSC(C)(C)C)C)NC(c1cccs1)=O N1(C(c2ccc(SC)o2)=O)CCCCC1C.C1(C(=O)NCC(C)C)CCC1 Cc1cc(NC(=O)C(F)C(C)CNC(=O)Cc2cc[nH]n2)cnc1O C1(CCNC(c2cccc(OC)n2)=O)CC(F)(F)CN1C(C1C=CC=CC=C1)=O CC(C)CC(CNC(c1cccc(N(C)C)c1)=O)NC(C1CCCCC1O)=O N1(C(C(C)OCCOC)=O)CCC(F)(C(=O)NCCCCCCN(C)C)CC1 N1(CCNC(c2c(NC)nccc2)=O)CC(O)(C2CCCC2)C1 C(CC(O)CC(=O)N1CCOC(C(C)NC(=O)C=Cc2cc[nH]n2)C1)SC C(c1ccc2c(c1)OCO2)=CC(=O)NCCC(C)N(C(=O)C1=CCCOCC1)C c1(OC)ccc(C(N2CCCC(N(C)C(C3CC3CF)=O)CC2)=O)cc1Cl C(=O)(C(C)(C)CC(F)F)NCC(CC(=O)NCc1c(CC)nn(C)c1)C1CCC1 C1(C(N(C(CN(C(c2ncn(C(C)C)n2)=O)C)C)C)=O)CCC2(CCC2)C1 C1(CNC(CCOC)=O)CCCN1C(=O)CN(c1ccccc1)C Cc1nc2c(o1)CCCC2CC(=O)N1CCN(c2ncnn3cccc23)CC1C N1(C(C2N(C(C)=O)CCCC2)=O)CC2(C1)CN(C(C1COC(=O)C1)=O)C2 c1(N(C)CCF)nc2ccc(Cl)cc2c(=NC2COc3ccc(F)cc3C2)[nH]1 C(C(=O)N(C)CCNC(C1CCCN1C(=O)C(C)(C)C)=O)(C(C)C)NC(=O)OC C(=O)(C(F)C(C)(C)O)N(CCNC(C1CC(n2cccn2)C1)=O)CC.C(C)(=O)O N1(C(C2N(C)C(=O)OC2)=O)CC=C(CCNC(=O)CC2CCCOC2)CC1 C1(C(=O)NCC(C)(COC)CC)(CC)CCCN(C(C2CCC2)=O)C1 C(=O)(C#CC1CCOC1)NC1CCC(F)(CNC(c2ncc(CC)cn2)=O)C1 N1(C(C)C)CC(NC(C2C(C(=O)NC3CC(C)(O)C3)C2(C)C)=O)C(C)C1 N1(CC(=O)N(c2ccc(OC)c(C(F)(F)F)c2)C)C(=O)c2ccc(Br)cc2C1=O C(=O)(N=c1cc2ccccn2[nH]1)C1CN(C(CC(C)OC)=O)CC(C)(C)C1 c1(C(=O)NC2CCN(C(C34CC(C5CC5)(C3)C4)=O)C2)cc(C2CCCC2)n[nH]1 C(C(C)(C(N)=O)NC(=O)C(=O)NCC(=O)Nc1ccccc1Br)OC c1(C(=O)NCC2N(C(C=CC=CCC)=O)CC(O)C2)cccc2nccn12 C(=O)(C(C)CC(F)F)NCCOCC(=O)N(CC(C)O)CC C(=O)(C1CCc2c[nH]nc21)NC(CCC(N1CCN(C(=O)NC)CC1)=O)=O c1(CC)oc(C)cc1-c1nc(C(C)OC)nn1CCC(C)C Cc1nc(C(=O)N(C)C)ccc1-c1c(O)cccc1Cl N1(C(c2scc(C)c2)=O)CCCC(NC(=O)CC2CCCO2)C1C c1(N2CCCC(NC(c3ccc(CCC(=O)OC)cc3)=O)C2)ccc(C#N)nc1 C#CCC(C(=O)NC)NC(c1cnc(CNC(C2CCCC(F)C2)=O)nc1)=O c1(CCC)cc(C(=O)NCC2(OC)CN(C(=O)C(C(C)C)SC)C2)ccn1 c1(OC)ccc(C)c(NC(c2c(CNC(=O)C(C(C)C)OC)nnn2C)=O)c1 c1(CCCCCC)nc(-c2ccoc2Br)n(CCCO)n1 C1(C(C)C)CN(C(c2ccncc2F)=O)CCC1NC(c1cnn(CCF)c1)=O N1(C(c2c(CCC)nns2)=O)CCCC(CC)(NC(c2ccc(N)cc2F)=O)C1 N1(C(C(C)(O)c2ccccc2)=O)CC2CC2(NC(=O)Cn2ncnn2)C1 N1(C(CC(C)n2cccn2)=O)CC2(CCNC(C3CCCN3C)=O)CCC1CC2 C(=O)(CCCCC(=O)NCC1(C)CCC(NC(=O)CCCC(F)(F)F)C1)OC N1(C(c2nccc(C)c2)=O)CCCC(C)(C)C1C(N1CCC(C2CC2)C1)=O C(=O)(C#CC1CCOCC1)N1C2CC(CC(NC(CC3C(C)CC3)=O)C2)C1 c1(C(=O)NCC23CC(NC(C4CC(OCC)C4)=O)(C2)C3)c(C)n[nH]c1C C(=O)(CC(F)(F)C(C)C)NC1CCN(C(c2c(C)nc(=N)[nH]c2)=O)CC1C(C)C c1(OC)ccc2nc(SC)c(C#N)cc2c1.C1(C)(OC(C)=O)CNC1 c1(C(C)(C)C)ccccc1CNC(=NCC1CC=CC1)NC1CCCC1 CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc(C3CC3)no2)=O)C(C(F)(F)F)C1 c1(OC)cccc(C(C(=O)NC2CC(NC(=O)C(C)CF)C2)OC)c1 Cc1cc(C(N2CC(C)C2C(=O)NC2CCN(CCCO)C2)=O)nnc1C Cc1oc(C#N)cc1C(N1CC=CC(C(=O)NCCN2CCS(=O)(=O)CC2)C1)=O C1(C(=O)NCCCCN(C(Cc2cccc(OCC)n2)=O)C)OCCC12CCC2 c1(OCCC(N2CCC(N(C(CCC#C)=O)C)CC2)=O)cc(F)ccc1F Cc1c(Cl)ccnc1C(=O)N(C)CC1(NC(=O)COc2cccc(F)c2F)CC1 c1(C(N2C3C(C(N4CC(C)OCC4C)=O)C(C3)C2)=O)c[nH]c2cccc(Cl)c12 Cc1cc(O)ncc1C(c1nnnn1Cc1ccccc1)NC1(C)CC1(C)C CC1(C)CC(C#N)(CNC(=O)C(C2CC2)NC(c2nnsc2N)=O)C1 C1(CC)(NC(c2cn(C3CCC3)nn2)=O)CCN(C(=O)COCC(C)C)CC1 N1(C(c2ccc(C(C)(C)C)o2)=O)CC(NC(=O)Cn2cncn2)C2CC12 C(C)(CN=c1[nH]cnc(=N)[nH]1)NC(c1c(C)nc(COC)s1)=O C1(CC(=O)NCc2n(C(C)C)ncn2)CN(C(C2CC(=C3CC3)C2)=O)CC12CC2 C(C(CCCC)NC(C1(OCC)CCSCC1)=O)NC(C1(C(F)F)CC(=C)C1)=O C(CCN=C(NCCCOCCCO)NCC1CCCCO1)CS(C)(=O)=O c1(C(N2C(C)CC(NC(c3nc(C)nc(O)c3)=O)C2)=O)c(O)nnc2c1CCC2 c1(C(N2C(CNC(C(c3ccccc3)C)=O)CC2)=O)cnn(C(C)(C)C)c1 C(CN=C(NCC(=O)NC1CC(Cl)(Cl)C1)NC1CCS(=O)(=O)C1)SC CCC(C(=O)NCC(O)CNC(c1ocnc1C)=O)OC1CCCCC1 C12(C(=O)NC(CCOC)CNC(=O)C(O)CSC)C3CCC(CC13)C2(F)F Cc1cc(N)c(C(=O)NCCC2CCC(NC(=O)C3=C(Cl)CC3)C2)cc1C C#CCC1C(=O)N1.c1(NCC)nccn1C1CC1.C12(C)CN(C1)C(=O)C(=O)N2 Cn1cc2ccc(NC(C3CC(O)CCN3Cc3ccnc(O)c3)=O)cc2n1 N1(C(C2CC(NC(c3n[nH]cc3Br)=O)C2)=O)CCC(S(=O)(=O)c2ccccc2)CC1 C(=O)(CC(C)(C)C(=O)NCC1CCN(C(=O)CNC(N)=O)CC1C)OCC C(=O)(CS(=O)CC)NCC(CC)NC(c1cc(CC)[nH]n1)=O c1(NCc2c(C)nc(CCC)o2)nccc(=NCC2CC(O)C2(C)C)[nH]1 c1(OC)ccc(SCC2CC2)c(C(N2CCN(C(C)=O)C(CO)C2)=O)c1 c1(C(N(CC(C)C(=O)NC(c2csnn2)C)C)=O)ccc(N)c(F)n1 C(CC(CC)C(=O)N1CCC(C(N2CC=CC2CN(C)C)=O)CC1OC)=CC C1(NC(C2(COC)CN(C(=O)Cc3c[nH]nc3C)C2)=O)CC2CSCC2C1 c1(CC)ccc(C(N2CCCCC2COC)C(=O)NCCOCC2CC2)cc1 Cc1nnc(CC(=O)NCCC2CCC(NC(=O)Cc3nncn3C)C2)o1 c1(C(N2CCC(OCCN(C)C)C2)C(=O)NCC=C)csc(C#N)c1 C1(OC)CCCCN(CC(=O)NCC(C)(Cc2ccccc2)C(C)O)C1=O C1(N(C)C(C2C3CCC(F)(F)C23)=O)CN(C(C2SCCS2)=O)CC12CC2 c1(OC)cccc2cc(C(N3CCCC3CCCNC(C3CC3(F)F)=O)=O)oc12 C1(CNC(CC(C)C2CC2)=O)CN(C(=O)CNS(N)(=O)=O)CCCO1 CC1CCCN(C(C2CCCN(C(C(=O)O)c3ccsc3)C2)=O)C1 C1(NC(c2n(C)c(=O)ccc2)=O)CC2CCC1CN2C(c1ccc([N+](=O)[O-])o1)=O Cc1ccc(C)c(F)c1NC(c1cc(F)ccc1OCC(F)(F)F)=O C12(NC(C(CC)C)=O)COC(C1)C(NC(c1ccc(F)cc1OC(F)F)=O)C2 N1(C(CC2(N(C)C)CCCC2)=O)CCC(NC(C2CCCCC2F)=O)CC1 c1(C(=O)NCC2(O)CCN(C(C(C(=O)OC)C)=O)C2)ccc(OC)cc1F CCC(C)CCCCC(=O)N1CCC(Oc2ccc(NC(=O)C(C)C)c(C)n2)C1 c1(C(=O)NC(C)CCNC(=O)CC(c2ccc(N)cc2)C)cnc2n1CCC2 N1(C(CCN(C(C2CCC(=O)N2)=O)CC)=O)CCC(C(F)F)CC1 c1(C(=O)NCCCNC(C2CC2C(F)F)=O)cccnc1-c1ccccc1 c1(OC)cc(=NC(=O)C=CCC(C)(C)NC(=O)C(F)CC2CCOC2)[nH]n1C c1(C(=O)NCC2(NC(C(=O)NCC3CC3)=O)CC2)cnc(-c2cccnc2)s1 C(C(CC)(CC)C(N)=O)NC(C1C(NC(C2C(OC)CCCC2)=O)CCOC1)=O CCC(C(=O)N(C(C)(C(=O)NCCC1CCC(=O)N1)C1CC1)C)C(C)(C)CC C1(NC(C(CSC)O)=O)CC2(CCN(C(c3cccc(SC)c3)=O)CC2)C1 C1(C(=O)NCc2cnc(C(C)OC)s2)COCCN1CC(F)(F)F C1(NC(c2ccc(C)cc2)=O)CCCC12CCN(C(c1sc(Br)cc1Br)=O)CC2 C1(C(N2CC(NC(c3ccc(C4CC4)nc3)=O)C2)=O)C2CCCCC12 c1(OC)cc(N)cc(C(=O)NCC(C)(C)CNC(C2CC2CC(C)C)=O)c1OC c1(CC)ccc(C(C)C(=O)NCC(CO)NC(C2(OC)CS(=O)(=O)C2)=O)cc1 c1(C(=O)NCC(CCCC)NC(=O)C(C)OCC=C(C)C)cc(N)ccc1SC C12(CCN(C)C1)C(=O)N2.CC1CCC(C(=O)NCc2ccc(C(N)=O)o2)O1 C1(NC(c2ccc(OC(C)C)cc2)=O)CCCCN(Cc2cccc(Br)n2)C1 CS(=O)(=O)C1CCC(C(N2CCC(NC(=O)CC(F)(F)Cl)C2)=O)CC1 C1(CNC(c2c(COC)ccs2)=O)CCCN(C(C2(c3ccno3)CC2)=O)C1 c1(C(N2CCC(=CCNC(c3nncc(OC)c3)=O)CC2)=O)nnc(O)nc1O C1(N(C)C(c2ccn(CCF)n2)=O)CCCC(NC(=O)CC2CC2)C1 c1(C(N2CCC3C(NC(c4cc(CC)c(C)s4)=O)C32)=O)cc(N)cnc1Cl c1(C(N2CCC(OCCNC(C(C)OC)=O)C2)=O)ccc(C(F)F)nc1 c12ccc(cc1)SC1CC1N2.c1(C2CCCO2)ccc(C(c2ccccc2)=O)cc1 Cn1cc(C(=O)NCCn2ccc(C(N3CCC(CCO)C3)=O)c2)nn1 c1(C(=O)NCC2CN(C(C3N(C=O)CCC3)=O)C2)cc2ccccc2oc1=O c1(CCNC(CC2N(C(c3n(CC)ccc3)=O)CC2)=O)ccccc1F c1(CC)ccc(F)c(C(=O)NCC2CCCC(NC(c3[nH]ccc3C)=O)C2)c1F Cc1cc(C(=O)NCc2ccc(C(=O)NCC3CCCC3(F)F)cc2)c(C)n1C c1(C(=O)NCCOC2CN(C(C3CCC4CCC3O4)=O)C2)cccc2c1OCO2 C1(CNC(CCCCC#C)=O)CN(C(=O)CCCCOCC)CC(C)(C)O1 N1(C(c2ccc(SC)o2)=O)CCC2CCC(NC(=O)C(C3(O)CCCC3)F)C1C2 C1(CNC(c2ncc3ccsc3n2)=O)CC2(CCN(C(=O)C3CC3)CC2)C1 c1(OC)cnc(F)c(C(=O)NC2CC(F)CN(C(c3ccc(CSC)o3)=O)C2)c1 CN1CCN(C(=O)Cn2nc(O)ccc2=O)C(CNC(=O)Cc2cccn2C)C1 N1(C(CNC(=O)OC)=O)CCC(C2CC2)C1CNC(=O)C(C)S(C)(=O)=O N1(C(C2(C)SCCCS2)=O)CC(C2CN(C(C3COCCC3(F)F)=O)C2)C1 C1(NC(CCCOCCC)=O)CN(C(=O)Cn2cnc(C#N)n2)CCC1C CCCCC(C(=O)NCC(CC1CC1)OC)NC(C1CCC1CF)=O C1(C(=O)NCC(CC)NC(c2c(Cl)nn(C)c2Cl)=O)CCCNS1(=O)=O c1(OC)ccc2c(C(=O)NCC3CCN3C(=O)C3=CCSC3)ccnc2c1 Nc1ccc(Cl)cc1C(=O)NCC12CC(NC(c3c[nH]nc3C3CC3)=O)(C1)C2 C1(NC(CC(C)(C)SC)=O)CCN(C(c2ccc3cnnn3c2)=O)CC1(C)C N1(C(C2(CC)CC2)=O)CC2CC2(C(c2ccc(O)cc2)OC)C1 c1(C(=O)NC(C(C)NC(c2ccc(CC)o2)=O)C)cc2c(Cl)c(OC)ccc2[nH]1 c1(C(c2n(C(CC)(C)C)nnn2)NC2CCCS(=O)(=O)C2)cc2cccnc2o1 c1(CC)ccc2sc(CN(C)CCCCCN)nc2c1 C1(CC(=O)N(CCN(c2c(C(=O)OCC)cccn2)C)CC)CCCCCCC1 Cc1cc(C#N)cnc1C(=O)NCC1CC1CNC(C1CC12CCC2)=O CC#CCC(C(=O)NCCOc1cccnc1)NC(=O)OC(C)(C)C c1(C(=O)Nc2nc(C)cc(C)n2)ncn2cc(-c3cncn3C)sc12 C1(F)(C(N2CC(NCc3cn(C)nc3)OCC2)=O)CCCCC1(F)F CC1(C(=O)NC2CCN(c3ccnc(N4CCCC4)n3)C2)CCCCCC1 Cc1c(C(=O)NC(C)CNC(=O)COCc2cccnc2)cccc1O c1(C(N2CC(COC)(NC(=O)C(F)CC3CCC3)C2)=O)nc(C(C)C)ncc1Cl c1(C(=O)NC(C)CN(C)C(C2CCC(C#N)C2)=O)ccc2nc(O)cc(O)c2c1 C1(OC)CC(CNC(C2C=C(C)CS2)=O)N(C(=O)CN(C2CCCC2)C)C1 C1(C(N(CCC(N)=O)CC)=O)(CC)CCCN1C(c1cccnc1OC)=O C1(F)(C(=O)NC2C(CNC(c3cc(SC)oc3)=O)C2)C(C)(C)C1(C)C c1(N(CCCCCCCl)CC(F)(F)C2CCCC2)cc(Cl)ccc1Cl C1(C(N2C(C)(COC)CCC2)=O)CCC(C)(C)N(C(C2C=CCC2)=O)C1 N1(C(C)=O)CCC(CC(=O)N(CC(C)CNC(=O)CCC2CCC2)C)CC1 c1(C(N2CC(NC(C#CC(C)(C)C)=O)C(F)CC2)=O)ccc2cncn2c1 c1(C(N(C)CCOCCCNC(=O)CC2(CO)CC2)=O)cn(C(C)(C)C)nn1 C1(CC)CCCN(C(=O)NCCCN(C)C(c2ncoc2COC)=O)C1 C1(CC=C)(NC(c2cnc(OC)nc2)=O)CCN(C(=O)Cn2cnc(C#N)n2)C1 c1(C(N2CCC(=CCNC(CC(=O)N(C)C)=O)CC2)=O)cc(O)nc(C2CC2)n1 c1(OCC(=O)NC(C2CCCC2O)CNC(CC)=O)ccsc1Cl C1(NC(c2c(SC)scc2)=O)CC2CCC1N2C(=O)C(C)OC1CCCC1 C1(C(=O)NC(C=C)C2CC2)CC(N=[N+]=[N-])CN1C(c1c[nH]c(C)c1)=O N1(C(CCOCCOC)=O)CCC2(CC2)CC1C(N1CC(C)N(C)C(C)C1)=O CC(CC(=O)N1CCCC1(C)CNC(c1ccc(O)nc1Cl)=O)C(F)F C1(C(N2CC3C(CNC(c4ccon4)=O)C3C2)=O)(CC)CCNC1=O C1(C)(C(=O)NC(CC)CNC(=O)C(C)CC2CCC2)CCC(F)(F)C1 CCC(CC)CC(=O)NC1CC2CC(NC(C3(C(F)F)CCCCC3)=O)C1C2 Cc1ccc(C(C)C(=O)N2CC(CC(C)NC(c3ccsc3C(F)F)=O)C2)cc1 C(=O)(C1=CC2(CCOCC2)C1)N1C(C)(CC)CC(NC(=O)C(C)(F)F)C1 CCC(CC)(CCNC(C1CCCC(=O)N1)=O)NC(C1OCCCC1(C)C)=O C(C)(N=c1[nH]c(N2CCC(C3CCCC3)C2)nc2cc[nH]c12)c1nnc(C)s1 C1(CC)OCCC1NC(=O)CN(C(=O)C(CC)N1CCCC1=O)CCOC Cc1oc(C(=O)NC2CC(CCNC(=O)CCC3CCCO3)C2)cc1CO Cc1cncnc1N1CCCC(CCNC(C2(C(C)C)CC2)=O)C1 C(C(C)(C)CC(=O)NC1(C)CC2CCC1C2)NC(C(CC)COC)=O N12CC(C(O)C1)N(C)CC1(CC1)CC2=O.C(=O)(CCCc1ccncc1)OC CC#CCCCC(=O)NCCOCCN(C(=O)C(c1ccc(F)cc1)C1CC1)C c1(N2CCC(=CC)CC2)ccncc1[N+](=O)[O-].c1(C=O)cnn[nH]1 c1(C(=O)NC2CC(C)N(C(=O)C=CI)CC2)cc2n(n1)CCCO2 CC(C)(C)C(O)C(=O)N1CC2(CC(N3CCN(CC(F)F)CC3)C2)C1 CC1CC1C1CC1C(N1CCC(CNC(C23CC(C)(CO2)C3)=O)CC1)=O N1(C(c2cc(Cl)c(Cl)c(Cl)c2)=O)CCC2C1CCCN2C(C12CC(C1)C2)=O Cc1cc(O)ncc1C(=O)NCCN(C(=O)CC1COC2CC1C2)CC1CC1 n1(CC(=O)NC2CN(C(C3(CN(C)C)CC3)=O)CC2F)cnc([N+](=O)[O-])n1 C1(C(=O)NC(C(=O)OC)Cc2ccccc2Br)COC2(CCOCC2)O1 CC1(C)CC2(CC(C(=O)NC3CC(CNC(c4cccn4C4CC4)=O)C3)C2)C1 N1(C(Cc2ccc(C)s2)=O)CCCCC1CCCNC(=O)CSc1ccncc1 Cc1cccc(C)c1C(O)C(N1CCC(C2CCCN2C(=O)CC2CC2)CC1)=O C1(NC(c2c(C)cncc2C)=O)CN(C(=O)Cn2ccccc2=O)C2(CCC2)C1 c1(NC(N(CCC=C)Cc2ccccc2)=O)ccc2c(c1)OCCN2C N1(C(C2CN(CC(C)C)C2)=O)CC2CC2(NC(=O)CC(O)c2ccccc2)C1 c1(N2CCn3c(C)ncc3C2)[nH]c(=NC2CSC(C)C2)nc2c1ncn2C(C)C C1(C(N2CCCC(NC(=O)CN3CCC(O)CC3)CC2)=O)CC2(CCOCC2)C1 N1(C(C2(CCC)CCC2)=O)CC(CNC(c2cnc(=N)[nH]c2)=O)C(C)C1 N1(C(=O)Nc2cc(C)cc(N)c2)CC2(CC(S(C)(=O)=O)C2)C1 C1(NC(COCCOCC)=O)CCCC12CCN(C(c1nnn(C)c1N)=O)CC2 Cc1ccc(C2(C(=O)NCC(C)CCN(C(=O)Cc3ccnn3C)C)CC2)cc1 C(=O)(NNCC(F)F)N(C)CC1(c2ccccc2)CCOC1 C1(NC(C2(CCOC)CC2)=O)CCC2CC1CN2C(=O)C=Cc1nc(C)cs1 C1(NC(CC2N(CC)CCOC2)=O)CC(F)CN(C(=O)CC(F)(F)F)C1 C(=O)(C1=NNC(C(F)(F)F)C1)NC(Cc1cn(C)nc1)C(=O)O c1(N(C)CC2CCCN2CC2CCS(=O)(=O)C2(C)C)ncnc2c1CCC2 S(=O)(=O)(c1ccc(Br)cc1NCc1nc2ccccc2n1C)NC(CC)CO N1(C(c2c(COC)cco2)=O)CCC2CCN(c3ncc(C)cn3)CC2C1 c1(C(N2CCC(O)(CNC(c3c(C)coc3C)=O)C2)=O)cn2ccnc2s1 c1(NC2(CNC(C(CSC)C)=O)CC2)ncnc2c1cnn2C C=CC1(CC(=O)NC(C)CC(=O)OC)CN(C(=O)CC2CCCN(C)C2)C1 N1(C(=O)CC2CCCCO2)CCCCC1C1(C(N2CC(F)(F)C2)=O)CC1 N1(C(C(C)NC(c2ccc(CC3(CCN=[N+]=[N-])CC3)s2)=O)=O)CCOCC1CO Cc1[nH][nH]c(=NC(=O)C23CC2CN(C(=O)Cc2cccc(O)c2)C3)c1Cl C1(C(=O)O)(NCc2c(OCC)cccc2)CC2(CSC2)C1 c1(C(N2CC(N(C(C(C3CC3)SC)=O)C)C(O)C2)=O)cc(C)cc(F)c1N N1(CC(=O)NCCCN(C(=O)Cc2cccc(Br)n2)C)CCC(C)(O)C1 c1(CC(=O)NCC(CNC(C(COCC)C)=O)C)ccc(O)c([N+](=O)[O-])c1 CC1(C(=O)NC2CCC(NC(=O)CCSC(F)(F)F)CC2)CCC12CCC2 C1(C(N2CCC(C(=O)NC(CC#CC)CO)(OC)C2)=O)CC2CC(=O)C1C2 Cc1nc(C(=O)NC(CNC(=O)C(C)Oc2ccccn2)C2CCC2)cs1 C(C(=O)N1CCCC(CCNC(=O)C=C2CCC2)CC1)(c1ccccc1)=C(C)C N1(C(C(C)OCC)=O)CC(O)(Cc2cn(CC(N)=O)nn2)C1 N1(C(C2C(NC(C3C(OC)CCC3)=O)COC2)=O)CCN2C(=O)CCC2C1 CC(F)CC(=O)NCCCN(C1CCCC1)C(=O)CC1CC2CC2C1 Cc1c(NC(=O)CC2(C)CN(C(=O)COC3(C)CCC3)C2)ccc(Br)c1Cl N1(C(CC(C=C)CC)=O)CC(NC(C2CCC(=O)N(C)C2)=O)CC12CCOCC2 c1(C(=O)OC)cc(CC(=O)NCCN(C(=O)C(C)n2ccnc2)C(C)C)[nH]n1 Cc1c(C(=O)NCCC2CCN(C(c3cc4occc4s3)=O)C2)cccc1N Cn1cnc2ccc(C(N3CC(NC(=O)Cn4cccn4)C4CC34)=O)cc2c1=O C12(C(N(CC(C)(C)NC(c3cn(CC)nc3C)=O)C)=O)CCC(F)(CC1)C2 N1(C(CC(C)C2CC2)=O)CCCC2(CCN(C(c3cnc(F)c(F)c3)=O)C2)C1 C1(OC)CN(C(=O)C=CC2CCCN2C(=O)C(CC2CCC2)OC)CC12CC2 CC(C)C(F)(CNC(=O)CC(=O)N(C)C)C(=O)NC1(C2CC2)CCOC1 C(CC(F)F)(C(=O)NC(c1ccncc1)C)N(C(CCC(C)OCC)=O)C c1(C(=O)NCC(C)(C2CC2)NC(c2cc(COC)[nH]n2)=O)cnc(O)n(C)c1=O Cn1cc(CN2CC(O)(c3ccsc3)C2)c(C(F)F)n1 C1(NC(C(C=C)OC)=O)CCCCC12CCN(C(c1[nH]ccc(=O)c1C)=O)CC2 N1(C(c2cccc(N(C)C)c2)=O)CCCC(F)(CNC(C2CCCN2C=O)=O)C1 C12(NC(=O)CN3CC4CC4C3)CCCC1N(c1ccn3c(Br)cnc3n1)CCC2 C#CCCCCCCC(=O)N1CC(F)(F)CC1CNC(=O)CCCc1cc[nH]n1 c1(N(C2CCCC2)CCCC)ccc(CC)c(OC(c2cccc(SC)c2)=O)c1 c1(C(=O)NC2(C3CN(C(=O)C4=COCC4)C3)CC2)cncc2n[nH]cc12 c1(C(=O)NC(C)CN(C(=O)Cc2ccncc2Cl)C)oc2ccccc2c1CO c1(CC(=O)NCC(CCOC)NC(C2CCC(=O)NC2)=O)cc(C(C)C)n(C)n1 C=CCCC(C(=O)N1CC2(CCC2O)C1)NC(C1CCC1C(C)(C)C)=O C1(NC(C(CO)N(C)C)=O)CCCCN(C(=O)CCCc2ccc(F)cc2)C1 c1(C(=O)NC(C)C(C)NC(c2ccc(CO)c(F)c2)=O)c(O)cc(F)cc1F Cc1ncnc(C)c1C(=O)NCCC(C)NC(C1(CC(C)C)CCCC1)=O C1(NC(c2c(SC)cnn2C)=O)CC2CC(NC(=O)Cc3cn[nH]c3)C2C1 c1(N2CC3N(C(c4ccccc4F)=O)C(C3)C2)ncc2cn[nH]c2n1 N1(CC(=O)NCCN(C(CC2C(C)=NNC2=O)=O)C(C)C)CCc2sccc2C1 c1(NCCN(C(CC)=O)CC)ccc(S(=O)(=O)N2CCCC(C)(CO)C2)cc1F CC1(C)CC(=O)NCC1C(N1CC(NC(=O)OC(C)(C)C)CC1C(=O)O)=O c1(C(N2C(S(N3CCC(C#N)(OCC)C3)(=O)=O)CC2)=O)ccc2cc(O)ccc2c1 c1(CCC(=O)NC(C(C)NC(c2c(C)ccnn2)=O)CO)cc2ccccc2o1 c1(C(=O)NCC(c2ccccc2)N(C(CN(C(C)=O)C)=O)C)sc(C)cc1C N1(C(C2C(CC)CCN2C(=O)C=CCN2CCC2)=O)CCc2nc[nH]c2C1 CC1CN(C(C2CC2c2cc(F)cc(F)c2)=O)CCCN1C(C1OCCO1)=O N1(Cc2cnc(CCC)s2)C2CCCC1CC(C(=O)N(CC(C)C)CCOC)C2 C=CCC(CC(F)F)C(=O)NCC1CCC(C)(C)CN1C(=O)CC1CCC(=O)N1 C1(C(N2CC(NC(C=Cc3ncn(C)c3)=O)C2)=O)CCCC(F)(F)CC1 C(=O)(CCC(CC)CCC)N1CCC(C(=O)NC(C#C)CC2CC2)CC1 c1(C(=O)NCC(c2ccccc2)CNC(C=C=C(C)C)=O)cn2cccnc2n1 c1(N2CC(NC(C=C(C)C)=O)C(O)C2)ncnc2c(C)cccc12 C#CCCCCC(c1nnnn1C1CCOC1)Nc1ccc(OC(F)(F)F)cc1 CCCCCCC(O)CCC(=O)N(CC(O)CN(C(=O)C=CC=C(Cl)Cl)C)C N1(C(c2c(C)c(Br)sc2)=O)CCOCC(CNC(=O)C(C)C2CCC2)C1 n1(CC(=O)NC2CC(CNC(CCCCNC(C)=O)=O)C2)c(C)cc(C)nc1=O N#CCCCCC(=O)NC(CCOCCO)C(=O)NCC1(CO)CC=CC1 C1(NC(=O)OC(C)(C)C)CN(C(=O)N(C2CC2)Cc2ccsc2)CC1C(F)(F)F c1(OC)ncc(C)cc1CNC(=O)NC(C(F)(F)F)C1CCOCC1 C1(C(=O)NCC(C(C)C)=O)CCCN(C(c2cccc(CN)c2)=O)C1 N1(C(C=COCC)=O)CCCC2CCN(C(=O)CCc3ccc(Cl)s3)CC12 N1(C(C2CC(CCC)C2)=O)CCC1(C)CC(=O)N(C1CCOC1)CCC C1(CC(=O)NCC(=O)NCCSCCN(C)C)CCC2CC12 c1(SC)cc(C(N2CCC(C(C)(C)NC(=O)C=CC3CCOC3)C2)=O)co1 O=C(C(O)C(F)(F)F)NCC1CC2CCC1N2C(c1ccnc(CO)c1)=O N1(C(C=CC)=O)CCC(CCCNC(=O)COc2ccc(OC)cc2)CC1C c1(C(=O)NCCN2CC(O)CC(F)(F)C2)cc2ccc(-c3ccccc3)nc2[nH]1 C1(O)(CNC(C(C)Cc2cnco2)=O)CCN(C(C2CC3(CCC3O)C2)=O)CC1 c1(C(=O)NC2C(NC(Cc3cn(CC)nc3)=O)CCC2)cc(OC)ccc1F n1(C2CCCN(CC=C(C)c3ccsc3)C2)cc2ccccc2n1 C1(NC(CC(CCC)O)=O)CN(C(=O)Cc2ncc(Cl)s2)CC12CCOCC2 N1(CCC(N2CC(O)CC(NC(COC)=O)C2)=O)CCCc2ccccc21 c1(C(=O)NC(c2cc(Br)ccc2Br)C)c(F)cc(Br)cc1Br C12(CNC(CCC#C)=O)CCCCC1CN(C(=O)C(C)(C)C1CCC1)C2 Cc1nc2sccn2c1C(=O)NC1CCC(NC(c2ccc3cncn3c2)=O)C1 C(C(CC(F)(F)F)NC(=O)C(c1cscn1)N(C)C)NC(C(C)O)=O C1(NC(c2cncc(C)c2C)=O)CC2(CCN(C(c3cnc(S)[nH]3)=O)C2)C1 N1(C(C=NOC)=O)CCCCC(CNC(=O)C(C)S(C)(=O)=O)C1 c1(COC)ccccc1CC(N1CCCC1CN(C(=O)C(C)CC1CC1)CC)=O N1(C(C(COCC)C)=O)CCC2(CCCN(C(=O)Cc3c(C)noc3C)C2)C1 CC1=NOC(C)(C(=O)NC2CN(C(c3ccc(OCF)cc3)=O)CC2C)C1 CCC(O)C(C)(C)C(=O)NCCC1(NC(=O)CNC(c2ccc(Cl)cc2)=O)CC1 C(=O)(C(CC)CC(F)F)N1CC(C)(CNC(c2c(CCC)onc2C)=O)OCC1 C1(C(N2C(CNC(C3C(CCC)C3)=O)CC(OC)C2)=O)CC(=O)NC(C)C1 c1(C(=O)NCC2OCC(CNC(CN(C)C3CC3)=O)C2)cccc(N)c1 C(=O)(C(Cc1ccoc1)NC(C1CCOC1)=O)NCC(C1CCCC1)OC c1(NC(NC(C2CN3CCN2CC3)C)=S)nc(Cl)ccc1F c1(CC)cccnc1NC(C1(CC2CCCC(NC(=O)COC3CC3)C2)CC1)=O C=C(C)CCC(=O)N(C1CCCCC1)CCNC(=O)CC12COC(C)(C1)C2 C(=O)(CCC(C)(C)F)N1CC(C2(O)CN(C(C(C)CCOc3ccccc3)=O)C2)C1 Cc1c(Br)noc1C(=O)NC1CCCC1NC(=O)C(N1CCNC1=O)C C12(C(N3C4C(NC(CCc5ccc(OC)cc5)=O)C(C4)C3)=O)CCC(CC1F)C2 c1(-c2ncc(C(=O)Nc3ccc(OCC)nc3)nc2)ccc2c(CO)n[nH]c2c1 CCC1=NOC(C(=O)NC2(COC)CCN(C(c3sccc3OC(F)F)=O)C2)C1 C(C1c2ccsc2CCN1C(N)=O)NC(C1Cc2c(C)ncnc2CC1)=O N1(C(C(C)C2CC2)=O)CCC(N(CCO)CC2CC(C)(C)CO2)CC1 c1(NC(=O)NCC)ccc(S(=O)(=O)N2CCN(CC)C(C)(C)C2)c2ccncc12 c1(C(=O)NC(CCC#C)C(=O)OCC)oc2c(Cl)cc(Br)cc2c1C C1(NC(c2n(CC=C)ccn2)=O)CCN(C(c2ccsc2Cl)=O)C1C C1(O)(CCNC(C(=O)N(C)C)=O)CN(C(C2COCOC2)=O)C1 C1(CC)CN(C(C2OCC3CCCC23)=O)CCN1C(=O)C(O)C(C)C C(Cc1ccsc1)(C(=O)N(CCCNC(=O)Cc1ccc(C)o1)C1CC1)NC=O C1(CNC(C(CCC)CC)=O)CCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 CC1CN(C(=O)C(C)(C)C2(O)CCNC2)CCC(c2ccccc2)O1 c1(CCN(CCCOC)C(C)C)nc(-c2ccc(C)s2)no1 N1(C(COC(CC)C)=O)CC(C(C(=O)N)OC)C1.C1(OCCCCO)(CC)CCC1 CCC(O)C(C)(C)C(=O)NC(CO)C(C)NC(c1ccc(F)c(SC)c1)=O N1(C(=O)OCCC)CCC2(CCC(C(=O)NS(=O)(=O)CC)C2)CC1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2C(CNC(=O)CN(C)C(C)C)C2C1 c1(C(=O)OC)cncc(C(=O)NC2CC2CNC(c2ccc(C)c(N)c2)=O)c1C Cc1cc(N)c(C)nc1C(N1CCC(O)(C(C)NC(c2ccn(C)n2)=O)C1)=O N1(C(C(c2ccc(CC(C)C)cc2)C)=O)CCN(C(C2(C#N)CCC2)=O)CC1C c1(-c2nnc(CC(CC)C)n2CCC#N)cnc2[nH]ncc2c1 N1(C(COCCCC)=O)CCCC1(C)C(=O)NCCC1OCCC1C c1(OC)ncnc(OC)c1C(=O)NCCCCCCNC(C1COCCN1C)=O C1(NC(C(C)(C)SC)=O)COCCN(C(c2ccc(OC(C)(C)C)cn2)=O)C1 CCCCCC(C)CC(=O)N1CC(CNCc2cc(OC)nc(C)n2)C(C)C1 CN=c1cc(C(=O)NCC2(CNC(C3CCSC3)=O)CC23CCC3)cc[nH]1 Cc1c[nH]c(C(N2CCCC2(C)C(=O)NCCN2CCOCC2)=O)c1C Cc1ncc2n1CCOC2C(=O)NCCCCN(C)C(C12CCN(CC1)CC2)=O Cc1ncc(C(N2CC=CC2CNC(c2cn(C(C)(C)C)nn2)=O)=O)cn1 c1(C(=O)NC(C2CCN2C(=O)C(C2CCOCC2)F)C)cnoc1-c1cn[nH]c1 N1(C(C(C)C#N)=O)CC2(C1)C(NC(=O)Cc1cccc(F)c1)CCS2(=O)=O c1(C(=O)NC2CN(C(C(C(C)C)F)=O)CC(C)C2)c(Br)ccc(Cl)c1F N1(C(CCC(C)OCC)=O)CC=C(C(=O)Nc2ccc(C)c(O)c2)CC1 CC(C(=O)NC1CCCN(C(c2csc(-c3cnn(C)c3)n2)=O)CC1)S(N)(=O)=O CC(CC(=O)N1CC2CC(NC(C34CC(F)(C3)C4)=O)CC(C2)C1)CC(C)(C)C N1(C(=O)NCC(C)OCC=C)CCC(c2ccnn2C)C1 Cc1c[nH][nH]c1=NC(=O)C1CC(O)CN1C(c1ccc(Cl)nc1C#N)=O C(CN=C(NCCc1nnc2n1CCC2)NCC1CCCOC1)c1sccc1 c1(OC)ccc(CCC(N2CCN(c3nc(O)cs3)CC2)=O)cc1Br C(=O)(C(C)CN1CCCC1)NCCN(C(=O)CC1CC(C)(C)C1)CC CCCC(CC)C(=O)NC1(C)CC(NC(c2cscc2F)=O)C1 C(=O)(CCCC(F)(F)F)NCc1ccc(CC(C)NC(C(CC)O)=O)cc1 N1(C(c2c(C)n[nH]c2)=O)CCC2(CCC2)C(NC(=O)CC(C)c2cnn(C)c2)C1 CCCCC(CNC(=O)C(C)NS(C)(=O)=O)NC(=O)Cc1sc(C)nc1C N1(C(c2c(C)cno2)=O)C2CCC(C2)C1CNC(c1ncsc1C(F)(F)F)=O C(=O)(C(C#N)C(C)(C)C)N(C)CC1CCN(C(CN(CCC)C)=O)CC1 c1(C(=O)NC2CCCN(C(CC3CN(C)C3)=O)C2)ccc2nn[nH]c2n1 c1(C(=O)NCCCCn2cc(-c3c(OC)csc3)nn2)c(C)sc(C)c1C#N N1(C(c2nc(CC)oc2)=O)CCCCC1C1(NC(=O)CCc2cc(Cl)no2)CC1 c1(C(=O)NCC(C)(C)NC(c2ccc(C)c(O)c2)=O)cn2cccc(Cl)c2n1 Cc1ccc(CCC(N2CCC(CN(C(=O)CCC(C)(C)F)C)C2)=O)cc1C C1(NC(C2CC3(C2)CC3F)=O)CC2CN(C(C34CCC(O)(CC3)CC4)=O)CC2C1 CC(C)CCCC(=O)NC1(C)CCN(C(c2cnn(C(C)(C)C)c2Br)=O)C1 c1(C(N2C(CNC(C3=NOC(C)(C)C3)=O)CC2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] C1(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(C)C#N)CC)CCCC(C)(C)C1 C1(CC=C)(NC(c2csc(C(F)F)n2)=O)CCN(C(c2nn(C)cc2C)=O)CC1 C(CC(C)(C)C(=O)N1CCC(C)(CCNC(C2CC2C(C)C)=O)C1)OC c1(NCC(CCC)(C)C)nc(NCC2CCC3CC23)c2ccsc2n1 N1(C(c2c(C)nc(O)cc2)=O)CCN(C(=O)Cc2cnn(C(C)C)c2)C2CCC12 c1(C(=O)NC(C(C)NC(C(C)C(F)F)=O)(C)C)cccc2nc(C(F)F)sc12 N1(C(CCSCC)=O)CCCCC1C1CCCN(C(c2cc(OC)no2)=O)C1 c1(C(N2CCCC(N(C(CNC(CC)=O)=O)CC)CC2)=O)nccc2nn[nH]c12 C(CCC1CC1)(C(=O)N(C)CC1CCSC1)NC(c1cc(C)no1)=O C(=O)(C(C)(C)C(=O)N1CC=CC(NC(=O)Cn2cc(Cl)cn2)C1)NC N1(C(c2ccc3c(c2)CCCS3)=O)CC(S(=O)(=O)C2COC2)C1 C1(CN(C(COCCC#C)=O)CC)CCCN(C(=O)C(C#N)CC)CC1 C(=O)(C(CCC(C)(C)C)N(C)Cc1ccc(N(C)C)cc1)NCC c1(C(=O)NCC2N(C(CC)=O)CCCC2)cc(Cl)ccc1N.C12CCCC1C2 C(=O)(C1=CCN(C(C2CC3C(C2)C3(F)F)=O)CC1)NCC1(CN(C)C)CC1 CC(C(=O)N1CCCCC1C1CCN(C(c2c[nH]c(=O)cn2)=O)C1)C(C)(F)F N1(C(c2cc(C)ns2)C(=O)NCCC2CC2)CC(F)(F)CCC1C c1(OC)cc(C(N2CC(CNC(=O)Cc3cccs3)C2)=O)cc(F)c1F CP(C)(=O)C1CCC(NC(=O)C(=O)NCC(CCO)C(=O)O)C1 c1(C(N2CCC(CNC(C3(CC#C)CC=CCC3)=O)CC2)=O)n[nH]cc1[N+](=O)[O-] C#CCCCC(C)C(=O)NCC(C(C)(C)C)NC(c1cc(C)n(C(F)F)n1)=O C1(C(C2CC2c2cncs2)=O)(C(=O)O)CNC(=O)Cc2ccccc2C1=O C1(CCNC(=O)Cc2cnc[nH]2)CCCCN1C(=O)CCN(C1CCCCC1)C c1(CC(=O)N(CC(=O)NCCCC(=C)Cl)CC(C)C)ccc(C)nc1 C1(C(N2C(C(=O)OC)CC(OC)C2)=O)CCn2nncc2C1 C1(C)(C(=O)NC(C)CCCNC(c2ccn(C3CC3)n2)=O)CCCNS1(=O)=O CC(C)CCC(O)C(=O)NCC(CO)NC(c1cc2c(s1)CCCC2)=O C(=O)(C(CNC(=O)C(C)C(C)(C)C)CC(C)C)NC(CCC)C(=O)NC C(c1ccccn1)=CC(=O)NC1CC(C)(NC(=O)CC2OCCO2)C1 C=C(F)C1(CC(=O)NC2CC(C(=O)NCC(=O)NOC)C2(C)C)CCC1 c1(C(=O)NC(CCC)C(=O)N(C2CCC(C3CC3)C2)CC)cccc(F)c1C O=C(CCCc1cncs1)NCC(C1CCCC1)NC(=O)CN1CCCCC1 C(=O)(C(C(=O)NC1CC(N(N2CCN(CC(C)O)CC2)C)C1)OC)OC.C=O c1(C(=O)NC2(CO)CCN(C(CCCOC)=O)C2)cn2c(n1)CCCC2C O=C(C#CC1CCCOC1)NCCC1(O)CCN(C(=O)CCc2cccs2)C1 N1(C(C2CC(C)(CC)C2)=O)CC(O)CC1CNC(c1ccsc1C(F)F)=O C1(NC(=O)NC(CCc2ccccc2)C(=O)O)CCc2nccn2C1 C(=O)(C#CC1CCC1)NC(C1CC=CCC1)C(=O)NCCCNC(=O)OC c1(C(=O)NCCCCN(C(C=CCC)=O)C)ccnn1CCN(C)C N1(C(CN2C(C)CCC2)=O)CCC(C(=O)NCCCC2(C)CC2)C12CCC2 C1(CC=C)(NC(C2CC2C2CC2)=O)CCN(C(c2cc(OC)ncn2)=O)CC1 N1(C(C(=O)NC(Cc2cn(CC)nc2C)C2CC2)=O)Cc2ccc(C#N)cc2C1 Cc1cc(Br)ccc1C(N1CCCC(N(C)C(c2cn(C)cn2)=O)C1)=O C1(C(=O)OC)CS(=O)(=O)C2CN(C(=O)C#CC3CC(F)(F)C3)CC12 c1(C(N(C(CC)C)CC)=O)cn2ccc(Cl)cc2n1 C(CCC(=O)NC(c1ccccc1)CNC(=O)CCc1cccn1C)=CC(C)C c1(C(N2CCCC(CC=C)(NC(c3cc[nH]c3)=O)C2)=O)ccc2cccnc2c1 Cc1ccc(N2CCCS2(=O)=O)cc1C(N1CCC(CN=c2[nH]ncs2)C1)=O CCC(CCC(=O)N(C1CCOCC1C)C)NC(=O)C(=Cc1ccccc1)C C1(CNC(C(CCCC)C)=O)CC2(CCC2)CN1C(c1ccc(N)cc1Cl)=O c1(C(=O)Nc2ccc(C)cc2-c2cnn(C)c2)cc2n(c1)CCS(=O)(=O)C2 C1(C(=O)NCC(C)(C)NC(COC2CN(C(C)=O)C2)=O)(OC)CCC(C)C1 Cc1ccc(CNC(C2CCCN2C(=O)NS(=O)(=O)CC(F)F)=O)cc1 c1(CNC(C(C)N(C(=O)CC2CCCO2)CC)=O)csc(C)c1 c1(C(=O)NC2(CCCNC(COC)=O)CC2)n[nH]c2c1CC(C)CC2 N1(C(C2C=C(C)CS2)=O)CCC(F)(C(=O)NCC2(C)CCCC2O)C1 CC(C)(C)CC(O)C(=O)NCC(C(C)(C)C)NC(=O)CCc1ncc[nH]1 N1(C(C(CC=C)C)=O)CCC(CO)(CNC(=O)CC2CN(C(C)=O)C2)CC1 N1(C(C2C(C(=O)OC(C)(C)C)C2)=O)CCCCC1CNC(C1CC(O)C1)=O CC(=O)CCCC(=O)N1CCCC(NC(c2ccc(Cl)nc2N)=O)C1 C1(NC(C2C(C)(C)CCC2)=O)CCSC12CN(c1nc(C3CC3)nc(=N)[nH]1)C2 c1(NC(C(=O)NCc2c(CC)cccc2OC(F)F)=O)c[nH]c2ccc(Cl)cc12 c1(N(C(=O)CN2CCNCC2)CC2C(C)(C)NC2)ccccc1F N1(C(CCNC(=O)OC)=O)CCCC(C)C1C(=O)NC1CCC(C#N)CC1 CCCC(C(=O)N1CCCC1C(C)NC(C1(C(F)(F)F)CC1)=O)S(N)(=O)=O N1(C(CS(=O)(=O)NC)=O)CC(NC(c2cn(C)c(C)n2)=O)C(S(C)(=O)=O)C1 C1(C(N2CC3C(N(C)C(C4(C5CC5)CCC4)=O)C3C2)=O)CC(C)(C)OC1(C)C C1(NC(c2c(CC)nco2)=O)CC2CCC1C(NC(=O)CCOC)C2 C(=O)(C1=CCCC1C)NC(C(=O)NC(CCCC=C)C1CC1)C(C)C C1(N(C(CCC#C)=O)C)CN(C(c2ccc(C(F)F)cn2)=O)CC1F Fc1ccc2sc(CN3CCN(c4ccc(Br)cn4)CC3)nc2c1 Cc1ccc(CNC(c2cnc(-c3ccc(OC(C)(C)C)cc3)cn2)=O)c(F)c1 C(CN=C1NCC2(CCCCC2)C1)C1(COC)CCOC1 CC1(C)CN(C(=O)Cc2cnccn2)CC1CNC(C1CC1(C)C(F)F)=O c1(C(=O)NC(C2CCN(C(C3CCCC3)=O)C2)C)scc2c1OCCO2 c1(C(=O)NC2CN(C(C(N3CCC(C)CC3)=O)=O)CC2CO)n[nH]c2c1COC2 Cc1cc(C)n(Cc2ccc(C(=O)NCCCNC(C3CC3(F)Cl)=O)o2)n1 CC1OCCOC1C(=O)NCCOCCOCCNC(C1(F)CC=CC1)=O N1(C(c2scc(CNC(C(C)(CO)OC)=O)c2)=O)CC2(CCCO2)C1 C#CCC(CC#C)C(=O)N1CC(NC(=O)CCc2ccc(F)cc2)CC(C)(C)C1 C1(CNC(C2OCCN(C)C2)=O)CC12CCN(C(c1ocnc1C(F)F)=O)CC2 O=C1CC(C(=O)NC(C(=O)NCC2CC2CO)C2CC2)CC1=O Cc1cc(C(N2CCC2CC(=O)NCCN2CCC2)=O)c[nH]c1=N C12(CC(=O)NCC(C(C)C)SC)COC(C)(C1)C2.c12noc(n1)CCC(=O)NC2 C1(C)(CNC(C2ON=C(CC)C2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1 c1(OC)ccc(C(=O)NCCN(C(=O)C(N2CCNC2=O)C)CC(C)O)s1 Cc1cccc(N)c1C(=O)NCC1CCCCN1C(=O)CCC1CC(C)(C)CO1 CC1(COC(c2cnc(-c3ccsc3)s2)=O)CCCCC1 C12(CN3CC(n4cc(CNC(COC)=O)nn4)C(O)C3)CC1COC2(C)C N1(C(C2(CC)CN(C(=O)CC3(C)CCOC3)C2)=O)CCOC(C)(C)C1C Cc1cc(C(=O)NCC2(F)CN(C(c3ncccc3O)=O)C2)c(Cl)cc1F C1(CNC(CC(CC)C)=O)CN(C(=O)C(C2CCC(=O)N2)C)CCC1(C)C C1(C(N(CCCN(C)C(c2sccc2Br)=O)C)=O)C(C)(C)C1(F)F c1(CC(N2C(CN(C(C(COC)(C)C)=O)C)CCC2)=O)cc(Cl)ccc1Cl c1(C(=O)NCCN(C(=O)CN(C)C(N)=O)C(C)C)cn2c(n1)CCC(C)C2 C1(C(=O)NC(C2(C(=O)NC3CC34CCCC4)CC2)C)CCCCCN1C Cc1nn(C)c(N2CC(n3cc(NC(=O)C(O)CC(C)C)cn3)C2)c1Cl Cc1ccc(CC#N)c(N(C(=O)CCC(C)C)C(C)C(=O)OC(C)(C)C)c1 c1(OC)cc(C(N2CCOCC2Cn2cc(CC(CO)C3CC3)nn2)=O)sc1C c1(C(=O)NCC2N(C(c3c(C)n[nH]c3)=O)CC2)cc(Cl)ccc1N C1(NC(=O)CC2CSCCN2)CCN(c2cccc(Br)c2)CC1 c1(N2CCCC(OCCO)C2)nc2c(c(=NCc3nc(O)n[nH]3)[nH]1)COC2 N1(C(C2C(C)CC2C)=O)CCC(N(C)C(C2CC(Cl)(Cl)C2)=O)CC1 c1(NC(=O)NC(C(=O)OC)Cc2ncncc2OC)cccc(C(F)(F)F)c1C N1(C(Cc2cccc(C)c2)=O)CC(C(=O)NC2CCCCC2)CC(C)C1 c1(CNCCOC)ccc(C(=O)NC(C)(C)CCNC(C2(F)CC2C)=O)cc1 C1(CNC(C(C)(F)F)=O)C2CCC(C2)N1C(=O)CC(c1cccc(F)c1)O Cc1cc(CN(C)Cc2sc(Cl)cc2Cl)ccc1Br C1(C)(C(=O)NCCCN(C(c2cc(CCOC)on2)=O)CC)CCCNS1(=O)=O N1(C(C=Cc2n(C)ncc2)=O)CC2CCN(C(=O)C(O)P(C)(C)=O)CC12 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CN(C(=O)C(F)CN(CC)CC)CC2C1 N1(C(C=CCCC)=O)CC2(CCNC(C3(C(N)=O)CCC3)=O)CCC1CC2 c1(C(=O)NC(C)CCCNC(=O)Cc2cccc(O)c2)ncnc2c1OCCO2 C1(CC)CCCC1C(=O)NCCC1CC(NC(=O)COc2ccsc2)C1 c1(NC(C)=O)ccc(Br)cc1C(N1CCC2(CC2C(N2CCC(Br)CC2)=O)C1)=O C1(CNC(C2CCCC(C)CC2)=O)C2CCCC1N(C(=O)Cc1ccoc1)C2 C#CC1N(C(=O)Nc2cccc(NC(c3c(F)cccc3F)=O)c2)CC1(C)C C1(CNC(c2cccc(CC=C)c2)=O)CN(C(C2CCCC(=C)C2)=O)CC12CC2 c1(OC)ccc(CC(=O)NCC2(C(=O)NCC3COCCO3)CC2)c(OC)c1 C1(NC(COC)=O)CN(C(C2CCN(C)C2)=O)CC1n1cccn1 c1(CC(=O)NC2COCCC2NC(C2(n3cnnn3)CC2)=O)ccc(Cl)cc1F N1(C(CCOCC)=O)CC2CCCC2(NC(c2nc(C(C)C)ncc2NC)=O)C1 c1(CC(N2CCC(NC(C=C(CC)C)=O)C2CC)=O)cnc(Cl)cc1C C(c1cc(Br)ccc1F)=CC(=O)NC(c1nc(C(CC)C)[nH]n1)C C1(C)(CNC(C=C(CCC)C)=O)CC(F)(F)CN1C(=O)C(C(C)C)NC=O C1(F)(CNC(CN(C(C)=O)C)=O)CCN(C(=O)COC2(C)CCC2)C1 c1(CC)nc(C)oc1C(=O)NC1CCOCC1C(=O)NCCC1(C)CC1 N1(C(c2c(OC)ccs2)=O)Cc2ccccc2CC1CNC(C1CC(=C2CC2)C1)=O c1(C(=O)NCC(CCNC(c2c(CC)non2)=O)O)cc([N+](=O)[O-])cc(C)c1Cl c1(OC)cccc(C)c1C(N1CCN(C(=O)CNC(=O)C(C)CO)CC1)=O Cc1snnc1C(=O)N(C1CC1)CC1CCCN1C(c1ccsn1)=O C1(C(N2CCCC(CCO)C2)=O)CC(O)CN1C(=O)CCc1ccccc1F C1(NC(C=C(C)Cl)=O)C2CC3CN(C(=O)CCc4n[nH]c(=N)s4)C1C3C2 C(C(C)CC(=O)N1CCC1CNC(C1CCS(=O)(=O)C1)=O)OC CC(CC(=O)N1CCC(N(C)CCO)C1)C(C)(C)NC(C1COCC1(C)C)=O N1(C(C(C(C)C)SCC)=O)CCN(C(C2(C)CC2)=O)CC12CC2 N1(C(CCCC2(C)N=N2)=O)CCOCC(NC(C2(C(F)F)CCOCC2)=O)C1 c1(CN2CC3CC3(C(=O)N(C)Cc3ccc(C)o3)C2)cccc([N+](=O)[O-])c1 C#CCC(CC(F)F)C(=O)NCC(N1CC(F)(F)OCC1C)=O c1(N2C(C)CC(CNC(C(C(C)C)O)=O)C2)nc(Cl)nc2[nH]c(O)nc12 c1(C(C(=O)NCC(C)NC(=O)CCn2cc(Cl)cn2)O)cc(F)c(F)cc1F Cc1c(C(=O)N(C)CC2(NC(C3COC4(CCC4)C3)=O)CC2)cccc1F C1(CNC(=O)CCC2CC2)CN2CCCCC2CN1C(=O)CCn1cnnn1 CS(=O)c1c(N(C(N2CC(N3CC(C(=O)O)CC3=O)C2)=O)C2CC2)cccc1Cl c1(CN2CCC(N(C(C=Cc3cc(C)on3)=O)C)C2)c(F)cncc1F c1(C(=O)NC2CCN(C(c3ccc(COC)s3)=O)C2)n[nH]c2nccc(Cl)c12 c1(C(=O)NCC2N(C(c3n(CC)nnc3)=O)CCCC2)cccc2ncccc12 N1(C(C2CC(COC)C2)=O)CC(C2CCCN(C(C3CC4(CCC4)CO3)=O)C2)C1 C(=O)(C(C)C(O)C(C)CC)N(C(CC(=O)NCC)CC)Cc1cccc(CC)c1 c1(C(=O)NC2CCC(NC(C3CC(SC)C3)=O)C2)cccc2c(C)ccnc12 c1(C(=O)NCC2C(C)CN(C(=O)C(O)c3cnc[nH]3)C2)cc2ccncc2s1 CCS(=O)(=O)c1ccccc1C(=O)NC(CNC(c1ccc(F)cc1)=O)C(C)C C1(CNC(C(F)=C(C)C)=O)CC(C)N(C(C2CC(CF)C2)=O)C1 CC#CCCCC(=O)N1CCC(C(C)(C)C(=O)NCC(CC)C(C)(F)F)C1 N1(C(c2c(C)ccs2)=O)CCOCC1C1CCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 c1(C(=O)NCC(C)NC(c2ccc(OCC)nc2)=O)ccc(CC)c(OC)c1 CCCC(C(=O)N1CCCC1CCCNC(=O)C=C1CCCC1)N(C)C c1(CC)nc(C(=O)NCC2(C(=O)NCCC#CCO)CCCCC2)c(C)o1 N1(C(=O)C=CC2CCC2)CCC(C2CN(C(C3CC4(COCCO4)C3)=O)C2)CC1 c1(CN(C(CC2CCCO2)C(=O)NC2(C)CC2)C)ccc2ccccc2c1Br C1(C(=O)NC(c2ccc(N(C)C)cc2)C)CN(C(=O)C=C2CC2)CC1CC(C)(C)C c1(CC(=O)NC2CCN(C(=O)C(C3CCCCC3)F)C2)cccc(C2CC2)c1 c1(C(N2CCN(C(CCC#C)=O)C3C2CC3)=O)ccc2c(N(C)C)ncnc2c1 c1(NC(N2CCC23CCOC3)=O)cc(O)c2ccccc2n1 C(=O)(CS(=O)(=O)Cc1cccs1)NC(CCNC(c1c(CC)cncc1)=O)C c1(C(=O)NCC2C3CN(C(c4c(CC)[nH]nc4Cl)=O)CC32)c[nH]nc1S(N)(=O)=O c1(OC)cc(OC)c(C(N2CC3(C2)CN(C)C(=O)O3)=O)cc1OC c1(CC(N2C(CNC(C3CC(OC)(OC)C3)=O)CC2)=O)ccc(F)cc1C C12(C(=O)NCCN3CCN(C(c4c(C)n[nH]c4)=O)CC3)CCC(C1)C(C)O2 c1(NC(CN2CCC(C(=O)O)CC2)C2CC2)ccc2nc(C3CC3)oc2c1 O=C(C1=NOC2(CCCN(C(c3ccc(Cl)cc3F)=O)C2)C1)N(CCO)C1CC1 Cc1nc2cccc(C(=O)NC3CC3NC(c3nn(C)c4c3COCC4)=O)c2[nH]1 CCN=c1ccc(C(N2CCN(C(=O)CC3(CSC)CC3)C3CC23)=O)c[nH]1 Cn1cncc1C(O)C(=O)NCC1(F)CN(C(=O)C(F)=C2CCC2)C1 CC1CCCCC1(CNC(c1nc(C(F)(F)F)ccc1F)=O)NC(=O)C=CCO C(=O)(C1CCCc2cccnc21)N1C2CC(NC(c3cn(C)nc3)=O)CC1CC2 C(=O)(C(C)(C)C(=O)NCC1(F)CCN(C(C2CC2C(F)F)=O)CC1)OC C1(CC(=O)NCCCCCNC(=O)COC2CC(F)(F)C2)CC2(CC2)CO1 C(=O)(C1=CC2(CCN(C(=O)C=Cc3nccs3)C2)C1)NCC(CC(=O)NC)C Cn1cc(S(C)(=N)=O)c(COC(c2cc(Br)ccc2-n2cccn2)=O)n1 N(C1CCOc2c(Cl)cccc21)C(=O)NC1(CF)CCN(C(=O)OC(C)(C)C)C1 c1(OC)ccc(C(N2CCC(NC(c3cc(SC)cc(F)c3)=O)C2)=O)c(F)c1F CC(CC(=O)NC1CN(C(c2occ3c2CCC3)=O)CCC1C)CC(F)(F)F C(=O)(CC(C)(C)CC(=O)NC1CCC(NC(c2nnn3c2CCC3)=O)C1)OC c1(C(N2C(C)(C)C(C(=O)NCC(O)CO)CC2)=O)cnn2ccccc12 Cc1cccnc1C(=O)NC1CC(N(C)C)C1.C12CCC(C1)C(=O)NC2 C1(C(OC)O)CCCN(C(=O)CN2CCCC(Oc3ccccc3F)C2)C1 N1(C(c2c(C)noc2C)=O)CC(NC(=O)C(C)(C)c2cscc2Cl)CC(O)C1 Cc1ccc(C(=O)NC2(CNC(=O)C(c3cnn(C)c3)C)CCOC2)cc1C#N N1(C(C(C(C)C)=O)=O)CCC(C)(C(=O)NC2CCC(F)(F)CC2)CC1 C1(NC(CNC(=O)OC)=O)(CO)CCN(C(=O)Cc2cc(Cl)ccc2OC)CC1 C(CC(N)=O)(C(=O)N1CCC(C(C)(C)C)C1)NC(c1ccc(C(C)=O)[nH]1)=O N1(C(CC2(C)CC2)=O)CC2(C1)CN(C(c1cc3c(cc1Cl)OCO3)=O)CCO2 Cc1ccccc1CC1C(c2ccccc2)C(F)C(=O)N1C.c1(N)ccccc1 N1(C(C(C)(C)OC(C)=O)=O)CCCC(O)(CNC(=O)C(C)P(C)(C)=O)CC1 CC1CN(C(c2occ3c2CCOC3)=O)CC2(CCN(C(C34CC3C4)=O)C2)O1 Cc1nnc2n1CC(C(N1CC(C)(C)CC1CNC(c1ccon1)=O)=O)C2 C12(NC(c3ncc(F)cc3F)=O)CCC(C1)N(C(=O)CSCc1cccnc1)C2 C1(NC(CCCC=C)=O)CCC2(CCN(C(C3(Nc4ccncc4)CC3)=O)C2)C1 N1(C(C(C)C2CCC2)=O)CCC2CN(C(c3cnn4c3CCCN4)=O)CC12 c1(C(N(C)C)=O)cccc(CN2CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)c1 C(=O)(C1CCCc2scnc21)NC(CCCCNC(CSC)=O)C C1(CCC)CN(C(=O)C(C)OCCOC)CC1C(=O)NCC1CC2C(C1)C2(F)F Cc1c(C(N2CCC3(CC2)CC3C(=O)O)=O)oc2c1C(=O)CC(C)(C)C2 C1(NC(C2CC(OC)C2)=O)CCSC12CN(C(=O)CC(=O)OC(C)(C)C)C2 C1(C(=O)OC)CC2(COC(c3ccccn3)=O)CC1C2 c1(CNC(CC)=O)ccc(S(C)(=O)=O)cc1.C1CCCNC(=O)C1 C1(CC)CC(C(=O)N(C2CC2C2CC2)C)CCN1C(c1ccsc1C#N)=O C1(C(=O)NCC(=C)C)CCCN(Cc2ncccc2Br)C1 C1(C(N2CCC(C(=O)NC)C2)=O)CN(C(=O)Cn2ncnn2)CCN1C Cc1nc[nH]c1CC(=O)NC1COCC1CNC(c1cc(-c2ccco2)cs1)=O C1(NC(C(CC)OC)=O)CCN(C)C12CCCN(C(C1(CC)COC1)=O)C2 CC1(C)CN(N2CCCC(SC(F)F)C2)CC(C(N)=O)O1 N1(C(CCSCCC)=O)CC(NC(c2ncsc2Br)=O)C(C2CC2)C1 C1(C(=O)NC(c2ccc(F)c(F)c2)(C(=O)OC)C)CSC(c2cccs2)=N1 c1(CNC(c2c(CNC(CN(C)C)=O)c[nH]n2)=O)ccnc(C2CC2)c1 c1(CC)nc2ccccn2c1C(=O)N(O)Cc1cn(-c2ccc(F)c(F)c2)nn1 C(c1ccc(F)c(C)c1)=CC(=O)NC1CCN(C(CNC(CC)=O)=O)CC1CO c1(NC(C2(SC)CN(C(c3sc(O)nc3C)=O)C2)=O)ccc2ccncc2c1 C12(C(N3CC(NC(C4C(C)(C)CO4)=O)(CO)C3)=O)CCCN(CC1)C2 Cc1c(C(N2CCSCC2CCNC(=O)CN2CCSCC2)=O)nnn1C(C)C c1(C(N(CC(CC)NC(=O)C(C(C)C)N(C)C)C)=O)c[nH]nc1S(N)(=O)=O c1(C(=O)NCC(C2CC2)NC(=O)C(O)c2ccco2)csc2cncn12 S(=O)(=O)(c1ccc(O)c(C(F)(F)F)c1)N1C(C)(CC(C)C)CCC1 c1(CC)ncc(C(=O)NC2CC(CCC(=O)NC(c3nncn3C)CO)C2)s1 C12(C(=O)NCC3CN(C(C4C(C)CC4)=O)C(C)(C)C3)CC3CC1C2C3(F)F C1(NC(c2cc(C(C)C)[nH]n2)=O)(CF)CCN(C(=O)CC=CC(C)(C)C)C1 C1(NC(C2CC3(CC(F)C3)C2)=O)CCN(C(=O)Cn2ncnn2)CC1F CON(CC(C(=O)C(C)C(F)F)CCCCC)C(=O)CCC(C)C N1(C(C2(CCC)CCC2)=O)CC2CC(C(=O)NCCC#CCO)(C2)C1 c1(C(=O)NC(CCN(C(C(CC)C2CCC2)=O)C)C)c(C)noc1C(C)C C1(C(=O)NC2(C)CCN(C(CCC(=O)OCC)=O)C2)CCC2CCCCC2C1 C1(OC)CCC2(C(N3CSCC3C(=O)NCCC(C(C)C)OC)=O)CC12 C(=O)(C#CC1CCOCC1)NC(C1(C(N2CC3CCCC2C3CO)=O)CC1)C c1(C(C)(C)C)cc(CN2CCC(O)(C(=O)Nc3c(Br)ccnc3Br)C2)ccc1O C1(NC(C2C(C)CC(=O)N2)=O)CN(C(C2CC(=O)CO2)=O)CC2(CC2)C1 c1(N2CC(CC)C(CC(C)(C)C)C2)nc(=NCCC(N)=O)[nH]c2c1COC2 C1(CC(=O)NC(CC(C)NC(C2(C(N(C(C)C)C)=O)CC2)=O)C)CCS(=O)(=O)C1 N1(C(c2cncc(C)c2)=O)CCCN(C(c2ccnn2-c2ccccc2)=O)CC1 c1(CC(=O)NC2(CF)CCN(C(c3c(CC)ocn3)=O)C2)cc(Cl)cc(Cl)c1 N1(C(CNC=O)=O)CC(NC(c2cncn2C(F)(F)F)=O)C(C2CC2)C1 S(=O)(=O)(c1ccc(F)cc1)NCCNC(c1scc(C)n1)C c1(C(N(CCC(C)NC(c2cccc(C(F)F)c2)=O)C)=O)cnnc(C2CC2)c1 c1(C(N(C2CCN(C(C3CCC(=O)N3)=O)C2)CCC)=O)n[nH]c2c1CCC2 Cn1nc(CNC(=O)NC(c2ccccc2F)C(C)(C)C)nc1Br c1(COCC)nc(C)cc(=NC2CC3CN(C(c4csnn4)=O)CC23)[nH]1 C1(NC(C2(COC)CCC2)=O)CCC(C)N(C(=O)C2=COCCO2)C1 n1(CCC)cc(C(=O)NCCCC(C)NC(=O)CC(=O)Nc2nccs2)c(C)n1 C(=O)(C1CCc2snnc21)N1C(CNC(C2(C(=O)NC)CC2)=O)CC(O)C1 N1(C(C2C(C)=CCC=C2)=O)CCc2cccc(C(=O)NC(C)(C)CO)c2C1 C(CC(C(C)C)NC(c1ccc(C(=O)CF)cc1)=O)N(C(C(COC)O)=O)C C(C(N=[N+]=[N-])C(=O)N1CCC(CC(=O)N(CC(C)C)C)CC1)OCC CC1(NC(=O)C(O)C2CCCC2)CCC(NC(c2cccc(C(F)F)c2)=O)CC1 C(c1cnc(C)nc1O)=CC(=O)NCCNC(c1ccc(C(CC)(C)C)cc1)=O C1(NC(C=NOC)=O)CC(F)(F)CC1NC(=O)CCc1ccc(OC)c(Cl)c1 C1(NC(C(C)NC(N)=O)=O)CCCN(C(c2ccc(-c3ccccc3)s2)=O)CC1 N1(C(C(CC2CC2)OC)=O)CCN(CC(=O)Nc2ccccc2)CC1 C1(C(N2CCC3(CC3C(N3CC(CO)C(O)C3)=O)C2)=O)CCCC1C1CC1 c1(N(CC(C)O)CCC)ncc(S(=O)(=O)NCC2CCN(CC)C2)cc1Cl N1(C(c2cc(COC)no2)=O)CCOC(CCCNC(=O)C(C)N(C)C(C)=O)C1 c1(C(=O)NCC2(NC(c3ccc(Br)s3)=O)CCC2)ccc(OC(F)F)cc1 N1(C(C(CC)n2cncn2)=O)CC(C)N(C(=O)C=Cc2ccc(C)s2)CC1C C(=O)(C(C(C)(C)C)C1CCC1)NC(CNC(c1cc(C)on1)=O)(C)C c1(-c2ccccc2)nnc(C2CC2)n1-c1cccc(CSc2ccccc2Cl)c1 c1(C(=O)NC2(CO)CCCN(C(CCC(CC)OC)=O)C2)n[nH]c2c1COCC2 CC(C)(C)CCCCC(=O)N1CC(=O)NCC1C(N1CC(CCO)C1)=O c1(C(c2nnnn2CCSCS)CCc2csnn2)cn(-c2ccccc2)nn1 Cc1cccn2ncc(C(=O)NNC(=O)NCC3=CC4=NC=NC4=CC=NN3)c12 CC1(NC(C23CSCC2C3)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(C(=O)NC2CCC(NC(c3cc(=O)cc[nH]3)=O)C2)ccc(C(F)(F)F)cn1 N1(C(C(C)=C(CC)C)=O)CC2(CNC(C3CC3(C)COC)=O)CC1CO2 Cc1cc(F)c(CC(N2CCC(C(C)NC(=O)CC3CC3(Cl)Cl)CC2)=O)cc1F c1(N(CC(CN(C)C(c2cc(CC3CC3)on2)=O)O)C)cc(C(N)=O)nc(Cl)n1 c1(N(C(CC2CCN(C(C(CC)(C)O)=O)C2)=O)CC2CCCC2)ccc(O)c(F)c1 N1(C(CC2CCN(C)C2=O)=O)CCC2CN(C(c3ccc(Br)o3)=O)CC12 C1(C(=O)NN2CCCC2)CCCCC1n1cc(CC2(CO)CCC2)nn1 C1(C(=O)NC(CCOC)CNC(c2cncn2C)=O)Cc2cccnc2C1 CC1CC(c2ccc(F)cc2)CN1C(=O)CS(=O)(=O)N1CCNCC1 Cc1csc(C(=O)NC2CC2NC(=O)CSc2ccc(O)cc2)c1C CCCCC(O)C(C)C(=O)N1CCN(C(=O)C(COCC)N=[N+]=[N-])CC1C(C)C C1(CC)CN(C(=O)C(O)C(C)C)CCN1C(=O)CCCN(C)C(C)=O c1(O)cccc(C)c1.C(C)(C(=O)NCC1CC1CNC(=O)COCCC(C)C)OC CC1=NNC(=O)C1CC(=O)N(C)CC1CCCN1C(=O)CCC1CC1(F)F c1(C(C)(C)C)nc(NC2(C(=O)Nc3ccccn3)CCOCC2)cc(Cl)n1 C(=O)(C(C)(C)CNC(=O)C(C1CCN(C(c2c[nH][nH]c2=N)=O)C1)C)OC c1(C(N2CCCN(C(c3ccc(C)nn3)=O)CC2C)=O)sc2nnc(S)n2c1C C(=O)(C1CSc2ccccc21)NC1CC(CNC(C(=Cc2cccs2)C)=O)C1 C1(CC(N2CCC(NC(C3(N=[N+]=[N-])CC3)=O)C(F)C2)=O)CCC2(CCC2)CO1 C12(CCNC(=O)C(C3CCCCC3)O)CCC(CC1)N(C(=O)CN1CCCC1)C2 c1(C(=O)NCC2OCCCN(C(C3C(C#N)C3)=O)C2)cccc2ccoc12 C1(C(N2CC(O)(CNC(c3c(C)sc(Cl)n3)=O)C2)=O)OCC2CCCC12 C1(C(N2C(CNC(C(CCCOC)C)=O)CCCCC2)=O)CN=C2N=CNN2C1 C1(=O)C(C(C)(C)O)N1.C1(OCC)CC(CNC(C2CC(SC(C)(C)C)C2)=O)C1 C(c1nccs1)=CC(=O)NCC(C1CCOC1)NC(c1cc(C(F)F)on1)=O C1(CNC(CCC(=O)OC)=O)(CNC(=O)CCC(C)(C)C)CC2CCCC2C1 C(CC(CNC(=O)C(O)c1ccsc1)NC(=O)Cc1csc(C(C)C)n1)OC CCCCCCCCCCCCCC(=O)OC(C1C(c2ccncc2)C1(F)F)=O c1(C(=O)NCC2(O)CCN(C(c3cncc(O)c3)=O)C2)cc2c(Cl)cccc2[nH]1 C1(O)(CCNC(COC(CC)C)=O)CCN(C(c2ccnnc2C)=O)C1 N1(C(=O)N(C)C)CCC(C)C(Sc2ccc(C)cn2)C1 C#CC1(O)CCCN(C(c2cnn(Cc3cc(C)ccc3F)c2)=O)C1 C#CC1CCCN1C(=O)NC(=O)CCCSc1ccccc1 Cc1nc2ccc(C(=O)NC34CCN(C(=O)CN5CCOCC5)CC3C4)cn2n1 c1(N(CCCN(C)C)C)cc(N2CCC(CC3CCCO3)C2)nc(C(F)(F)F)n1 C1(CC(=O)NCCOC(C)=O)CCCCC1NC(=O)Cc1ccc(C)s1 c1(C(=O)NCC(CNC(c2c(C)ncs2)=O)O)cc2nc(Cl)ccc2s1 N1(C(C(C)C)=O)CC(NC(c2cc(F)c(O)c(Cl)c2)=O)C(C2CC2)C1 C1(C(N2CCC(OC)(CNC(C3CNC(=O)C3)=O)C2)=O)CC2CCC(C1)C2 C(c1c(C)coc1C)=CC(=O)NC1C(C)(CNC(C(COC)O)=O)CCC1 C1(COC(COc2cn(C)nc2)=O)CN2CC3CC2(CO1)C3.C(C)NC(=O)C1CC1 CCCCC(C(=O)N1CCCC1C1CCN(C(c2nocc2F)=O)CC1)N(C)C Cc1cnc(F)cc1C(C(=O)NC(C)(C)C)N(C1CCCCC1CO)S(C)(=O)=O c1(N(C)Cc2ccoc2)nc(N2CCCC(F)CC2)c2c(n1)CCOC2 c1(OC)ccc(NC(=O)C(=O)NC(C)C(C)C2CCC2)c(C#N)c1 N1(C(C2C(C(C)C)OCC2)=O)CC(C(=O)NCCCS(N)(=O)=O)C(F)C1 C12(C(=O)NCC(C)N(C(=O)Cc3ccccn3)C)CCC(C1)C2(C)C c1(CC)nncn1NC(=O)C(CCC(C)C)NC(c1ccccc1F)=O C(=O)(CCCC(=O)N(C)CC1C2CN(C(C3COCCO3)=O)CC12)NC(C)C CC1=C(C)CC(C)(C(N2CCC(CN(C)C(C3(CO)CCOCC3)=O)C2)=O)CC1 CC(C(=O)NCC(C1CC1)N(C)C(c1cnnc(O)c1)=O)C(F)F N1(C(CNC(CC)=O)=O)CCC(C(=O)NC2CC(CO)C23CCC3)=C(F)C1 Cc1nn(C)cc1C(C)C(=O)NC(C)CNC(C1(S(N)(=O)=O)CC1)=O C(CC[Si](C)(C)C)N(C(=O)CCC1CCN(C(=O)COCCF)C1)C C1(CCOC)(NC(c2cc(C)n(C)n2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1 CC(C)(C)C(CNC(C1(C#N)CC1)=O)NC(c1cnncc1O)=O C1(C(=O)NCCOCCOCCOC)(NC2CC2)CC1 C(CC(O)C(F)(F)F)NCONC(CCC1N(C(c2cc(C)[nH]c2)=O)CCC1)=O CC1CN(CC2CCCCC2)CCC1CN=[N+]=[N-] N1(C(Cc2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)CC1(C#N)CCCCC1 C1(CN(C(C2COCCN2CC)=O)CC)CCN(C(=O)CCCN(C)C)CC1 c1(-c2cn(CCN(C(COCP(C)(C)=O)=O)C3CC3)nn2)cccc(O)c1 N1(CC(N2CCC(C(C)NC(=O)CCc3cncs3)C2)=O)CC(=O)NC1=O N1(C(=O)N(c2cc(CN)oc2)CCO)CCN(C2CCOCC2)CC1 C12(C(N(CC(COC)O)C)=O)CC(CN(C(=O)CCS(N)(=O)=O)C1)C2 c1(OC)ccc(CNC(c2cnn(CCF)c2)C)c(F)c1Br c1(C(N2CCCC(C(C)NC(=O)C3=CCSC3)C2)=O)c(F)cc(F)cc1F c1(C(C(=O)NC2CCOC2)N(CCCOC)C2CC2)cc(C)c(Br)c(Cl)n1 N1(C(C(CCC)O)=O)CC2(C1)CN(C(C1(F)CCCCC1)=O)CC2CO c1(C(=O)OCCCCCCC=C)ccccc1S(=O)(=O)N(C)C C1(CNC(C(COC)C)=O)CCCCN(C(=O)C(C)SC(F)(F)F)C1 N1(C(CCC)=O)CC(NC(=O)C=Cc2ccc(C(N)=O)o2)CC12CCCC2 C(=O)(C1CCc2nnc(C)n21)NCC1(C2N(C(c3c(C)cc(O)cc3)=O)CCC2)CC1 Cc1cc(C)c(C(N2CCCC(N(C(=O)Cn3cccn3)C)CC2)=O)c(S)n1 C1(C(N2C(CN(C(C3CCCN3C)=O)CC)CCC2)=O)CCN(C)C(=O)C1 Cc1ccc(C(N2CC3C(CNC(=O)CCCCC(N)=O)C3C2)=O)c(O)c1C Cc1cn2c(CC(=O)NC3CC(N(C)C(c4ccc(F)cc4F)=O)C3)csc2n1 CN(C)S(=O)(=O)N(C)CC(=O)N(CC(O)CN(C)C(C1CCC2CC2CC1)=O)C c1(C2CC(C(N3C(CNC)CCC3)=O)C2)cccc(OC(F)(F)F)c1 c1(CN2CC3C(C(=O)NCCCOC)C3C2)cccc(OC)c1OC c1(COC(CC2C(OC)COCC2)=O)nc2cc(Cl)ccc2s1 Cc1cc(C#N)cnc1N(C1CCCN(C(C2(F)CCOC2C)=O)C1)C c1(C(N(C2CCCN(C(c3cc(C(C)(C)C)no3)=O)C2)C)=O)cc2c(s1)CCC2 c1(N2C(NC(CC(C)C)=O)CCC2)cnnc(-c2cn(CC(C)(C)O)nn2)c1 c1(C(=O)NC2C(CNC(C(N3C(CC)CCC3)=O)=O)CC2)cccc(CO)n1 c1(C(=O)NC(C(C)C)CNC(c2cn(C)ccc2=O)=O)cc(N)c(N)cc1F c1(C(C2CCC(N(C(=O)C(=O)Nc3cccc(Cl)c3)C)C2)=O)ccc(F)cc1 C(=O)(C(C#N)C(C)C)NCC(CCCC)NC(=O)C(=Cc1c[nH]cn1)F c1(C(=O)OC)ccc(C=CC(N2CC(C)(NC(C3COCCO3)=O)C2)=O)o1 CC#CCCCC1(C)c2nnnn2CCOc2ccc(cc2)CC(C)N1.CC c1(C(=O)Nc2c(OC)nc(F)cc2)cc(-c2cccc(F)c2)cc2c[nH]nc12 C1(NC(C2(CC=C)CCC2)=O)CC(=O)N(C2CN(C(=O)C(C)C(C)C)C2)C1 C1(CNC(c2ccnc(C)n2)=O)CC2(CC2)CN1C(=O)C(C1CCCCC1)F Cc1nn(CCO)cc1C(=O)NC1CC(C)N(C(=O)COc2ccc(F)cn2)C1 N1(C(CCCCOC)=O)CCC2(CC2NC(c2ccncc2F)=O)C1 CN1CCOCC1C(=O)NCCn1cc(C(=O)NCC2CC(F)C2)nn1 c1(C(=O)NC2CCN(C(C3(C)C(C)(C)C3)=O)C2)ccc(-n2cnnn2)cc1Cl C(=O)(C(C)(C)C1=CCSCC1)NCCC(C)NC(C1CC1C(F)(F)F)=O C1(NC(c2cnccc2Cl)=O)CCC12CCN(C(=O)CC1CCCCO1)CC2 C1(C(=O)NC2(C)CC(NC(C3C(C)(C)OC(=O)C3)=O)C2)CCCCN1S(N)(=O)=O C1(CC(=O)NCC2(CNC(c3ncc(N(C)C)nc3)=O)CC2)CCC(F)(F)CC1 c1(C(N2CCC(NC(C3(CF)CCC3)=O)C(F)C2)=O)cc(Cl)cc(Cl)c1Cl c1(OC)cc(CN2CC(O)CC2C(N2CCCCC2C(N)=O)=O)ccc1Br CC1(CNC(C2CC(F)(F)C2)=O)CCCN1C(c1cn(CC(F)(F)F)cn1)=O c1(C(=O)NCc2c(C)nccn2)ccc2c(n1)CN(C(C1(C)CCOC1)=O)CC2 CC1(C)CC(C(N2CCC(C(C)(C)C)C2)=O)CN(C(C2OCCC2(C)C)=O)C1 C1(C(=O)NCc2n(C)nnn2)CCCCC1(C)NC(=O)CC1CNC(=O)O1 C1(C(N2CCN(C(C)=O)CC2)=O)CC(C)(C)CN1C(N1CCC1C)=O CN1CCC(N(C(C2CC23CCOC3)C(=O)NC2CCOC2)C)CC1 N1(C(CNC(c2ccccc2F)=O)=O)CCN(C(C2CC3CC3C2)=O)CC12CC2 C1C(CC(C)(C)C)C(=O)N1C.c1(CNC(C=CCOCCOC)=O)ccco1 Cc1[nH]nc(C(=O)NC(C(=O)N(CCCC(C)O)C)C2CCOC2)c1C C=C=CC(C)C(=O)N(CCC(=O)NC)CC=C.C(C=C(C)C)N C1(C(=O)NC23CC(NC(=O)C4=CCCCO4)(C2)C3)CC2CCC(C1)C2O c1(NCC2CC(NC(C3N(C(C)C)CCCC3)=O)C2)nccc(C#N)n1 c1(CCn2cc(NC(N(CCC(=O)OC)C)=O)nn2)ccc(N(C)C)cc1 c1(OC)ccc(C(=O)NC(C)C(C)NC(=O)Cn2cc(CO)nn2)cc1 C(CS(=O)(=O)CC(=O)NCC(C)CN(C)C(C1CCCN1C)=O)OC C1(NC(c2cc(F)c[nH]2)=O)CCCCC12CCN(C(=O)C1=CCCC1)CC2 c1(NC(CC)CNC(C2CCCC2(C)C)=O)ccc(C#N)cc1[N+](=O)[O-] C(CC(=O)Nc1ccccc1Cl)(C(F)(F)F)NC(c1nn(C)c(O)c1)=O C=C(C)CC(C(=O)N(CC(C)(C)CNC(C1CCOC1C1CC1)=O)C)OC c1(-c2cc(NC(C)=O)ncc2)n[nH]c2c1CN(C(=O)Nc1cccc(Br)c1F)C2 c1(CCC(=O)NCC2C(NC(C3C(CC)C3)=O)C2)cnn(-c2ccccc2)c1 C1(CCNC(CCCC)=O)CC2CCC(C1)N2C(c1cnn(C)c1N)=O c1(C(N2CC(NC(CC(CC)OC)=O)CC3(C2)CC3)=O)cc2c(C)n[nH]c2cn1 C1(C(N(CCCNC(C2CCC(C)(C)C2)=O)CCO)=O)CCc2nnnn2CC1 c1(C(C)=O)cc(C(=O)NC(C2CCOC2)CNC(c2ncoc2C)=O)no1 c1(OC)ccc2[nH]cc(CN3CC4CC3CN4C(c3cc(C)nc(Cl)c3)=O)c2c1 O=C(CCC(=O)N1CCOCC1)NCC(CO)NC(c1cn(C2CC2)nn1)=O c1(C(N(C)CCNC(=O)C(c2ncc(Cl)n2C)(F)F)=O)cc(Cl)ccc1O c1(C(N(C)CC2COCCN2C(=O)CC2(CO)CC2)=O)cc(F)cc(Br)c1 S(=O)(=O)(c1cnn(C2CCCCC2)c1C)OCc1c(OC)cc(OC)cc1OC c1(CSCCNC(C(=O)Nc2c(C)cnnc2)=O)ccc(S(=O)(=O)N(C)C)cc1 Cc1cn2ccnc(C(N3CCC(NC(=O)CC(C)CC(C)(C)C)C3)=O)c2n1 C(CC(F)F)(C(=O)N1CCCC(N(C)C)C1)NC(c1nnn(CC)c1C)=O N1(C(c2c(C)nn(C)c2C)=O)CC2CCC(C1)N2C(=O)Cn1nc(C)c(Cl)c1C c1(C(N(CC(CC)NC(c2nccnc2C)=O)C)=O)ccc(F)c(Cl)c1 S(=O)(=O)(c1ccc(C(C)=O)cc1)N1CCCN(CCOC)C(=O)C1 C1(NC(CSCC(=O)OC)=O)CCC(CNC(=O)Cc2csc(SC)n2)CC1 Cc1ccc(-n2nc(Cc3ccccc3)nc2C(C)C(C)(F)F)c(C)c1 c1(CNC(C=NOC)=O)ccc(CCNC(=O)CC2CC2(Cl)Cl)cc1 N1(C(C=C=C(C)C)=O)CCC(C)(CNC(C2CCN2C)=O)CC1 c1(CN2CCC(C(=O)NCCc3cccnc3)C(O)C2)cc(O)c(O)c(O)c1 c1(C(=O)NCC2N(C(Cc3cnn(C)n3)=O)CCC2)ccc2cccnc2n1 N1(C(CSCC)=O)CCC2(CCN(C(=O)C(F)Br)CC2)C1 N1(C(C2(F)CCN(C(C(CC)(CC)CC)=O)C2)=O)C2CCC1CC1(C2)N=N1 c1(CN(C2CCN(C)C2)C(c2csc(Cl)c2)=O)cccc(N(C)C)c1 c1(CC)cc(C(N2CCC(F)(CNC(c3ccc(O)nc3)=O)CC2)=O)ccc1F c1(CN(CC)CC)ccc(C(=O)NC(=O)NCC(c2ccccc2C)(C)C)cc1 N1(Cc2ccc(F)c(O)c2)CCC(F)(CNC(C2N(S(C)(=O)=O)CCC2)=O)CC1 C(N=c1nc(N2CCCCC(SC)C2)c2c([nH]1)CSC2)c1cc(OCC)ns1 C12(C(=O)NCC(CC)NC(=O)C(F)CC3CCCC3)CCC(O)(CC1)CC2 C1(CC(=O)NCC(C)(C)NC(C(CCC)N(C)C)=O)OC(C)(C)OC1=O c1(C(=O)NCC2CC(NC(CCS(=O)(=O)NC)=O)C2)nccc2[nH]ccc12 N1(C(C(F)=CCC)=O)CC2(NC(=O)CCCc3cncs3)CCCC2(F)C1 C1(C2CN(C(=O)C(C)N=[N+]=[N-])C2)(NC(CC(=C)C)=O)CC1 Cn1[nH]c(=NC(=O)C2CCN(Cc3c(Br)cc(F)c(F)c3F)C2)cc1Cl N1(C(C2N(C(C)=O)CCC2)=O)CCN(C(c2ccnc(C(F)F)c2)=O)C(C)C1 N1(C(C(N)=O)=O)CCOC(CCNC(=O)CCC(=O)c2cccc(F)c2)C1 N1(C(CCOCCC)=O)CCOC(CNC(=O)C#CC2CC2)C1 c1(SC)ccc(C)c(C(=O)NC2CCCC2NC(C2CC23CC(F)(F)C3)=O)c1 N1(C(=O)CC2(C(=O)O)CC2)CCC2(C1)CN(C(C1(F)CCCC1)=O)C2 c1(C(N(CC(CN(C(c2c(C)scc2)=O)C)O)C)=O)nccc(Cl)c1F C(CC(=O)N1CCC(O)(Cn2cc(CCC3CCC3)nn2)C1)(C(F)F)N(C)C c1(C(=O)NCC2CCCCN2C(=O)CCn2ccnc2)ccc2c(c1)CCC=C2 c1(C(=O)NC2(CCO)CN(C(c3ccc[nH]3)=O)C2)cc2c(cc1Cl)NC(=O)CO2 C1(c2ccc(F)cc2)(C(N2C(CNC(c3ccon3)=O)C=CC2)=O)CCCCC1 C1(CCNC(C(C)(C)OCC)=O)CCC(C(C)C)CC1.C1COCCO1 c1(CN(C)C(=O)NC2(c3ccncc3F)CC2)ccc(Cl)cc1F C(CC(C(=O)N1CCC(CSC)C1)NC(=O)CC1CC1SC)OCC c1(OCC(N2CCC(C)(NC(=O)CCCn3ccnn3)C2)=O)cccc([N+](=O)[O-])c1 C(C)(C)(C(F)(F)F)n1cc(-c2c(CNC(CSC3C(C)CCC3)=O)ocn2)nn1 C1(Sc2ccccc2)C2CC3CN(C(=O)CCCNC(CCC(=C)C)=O)C1C3C2 c1(CN2CCC(CCC(C)(C)Nc3ccccc3)CC2)cnc2ccoc2c1 CC(C(=O)N(CCNC(=O)COc1cccc(F)c1)C1CC1)C1=CCCC1 c1(C(N2C(C)(C)C(CNC(=O)CSCC(F)F)CC2)=O)cc2nn[nH]c2cc1F c1(C(N(CCNC(C2CCC3CC23)=O)CC)=O)nccc2c1[nH]c1ccccc21 C(CN=c1ccnc(SC(F)F)[nH]1)c1ccc(CC(C)C)cc1 C1(NC(CC#C)CC)CCN(C(C=C)C(F)(F)F)CC1 c1(C(=O)NC2CC(CNC(C(c3ccc(C)s3)C)=O)C2)cccc(Cl)c1F c1(NCC2C(C)CN(C(=O)C=C(C3CC3)C3CC3)C2)nc2cccc(Br)c2o1 N1(C(=O)C=CBr)CCC2CCC(NC(C3(C4CC4)CC3)=O)C1C2 C(CS(=O)(=O)C(F)(F)F)NC(c1cccc(OC)c1)(c1n(CCC)nnn1)C1CC1 C(=O)(CC(O)C(C)C)NC(CCOCC)C(=O)NCc1cnn(C)c1O n1(CC)c(C)nn(CC(=O)N(C(C)CNC(=O)C(CCSC)N(C)C)C)c1=O C1(c2nnnn2C2(C)CC2)(NC(CSC)C)CC(C)(C)C(C)(C)C1 C1(C(=O)NCCN(C(=O)Cc2nn(C)cc2Cl)C)CCC(C)(F)CC1 c1(C(N2CC3(CN(C(C=Cc4n(C)cnc4)=O)C3)C2)=O)c(Cl)cccc1[N+](=O)[O-] N1(C(c2scc(C)n2)=O)CC(C)CC1C(=O)Nc1nc(C)cs1 CC(C)CC(O)CC(=O)N1CCN(C(C23CC(COC)(CO2)C3)=O)C(C)C1C c1(CC(=O)NCc2ccccc2CNC(C2(F)CCCC2)=O)ccc(Cl)cc1Cl Cc1nc2ccc(C(=O)NCCN(C(=O)Cn3cccn3)C)cc2s1 C(C)(CCC(=O)N(CCCCCNC(=O)CC(C)c1ccco1)C)SC C1(OC)CN(C(c2cc(C)n(C)c2C)=O)CCC1NC(c1cc(Cl)ncc1Cl)=O C1(C(=O)NCCC(C)N(C)C(C2CCCN2C)=O)CC12CCOCC2 c1(C(=O)NC2(CO)CN(C(C(C)CN(C)C)=O)C2)ccc(CC(C)(C)C)cc1 c1(C(=O)NC2CCN(C(CS(CCCC)(=O)=O)=O)C2)ccccc1C#CC1CC1 c1(CNC2CC(NC(c3c(C)nccc3F)=O)C2)cc2ccc(Br)cc2s1 C1(C(N2CC(F)(CNC(c3cc(C(F)(F)F)c[nH]3)=O)C2)=O)(OC)CCOC1 c1(C(=O)NC2CC(CNC(CSc3n(C)nnn3)=O)C2)ccc2cccnc2n1 C1(CN(C)C(C2CC2c2ccsc2)=O)CCCN1C(=O)CCc1cncs1 C1(C(=O)NC)CCCC1N(C)C(C1CCCN1C(=O)CCC1CCC(=O)C1)=O C12(CNC(C(CCCC)O)=O)CCC(CN(C(C3(C)CCCN3C(C)=O)=O)C1)C2 c1(C(N2C(CNC(C)=O)CCC2)C(=O)NCc2ccco2)ccc([N+](=O)[O-])cc1 N1(C(Cc2ccc(OC)nc2)=O)CC(NC(c2sc(C)cc2Cl)=O)CC2(CC2)C1 c1(OC)ccc2c(c1)CN(C(C1CCCN(Cc3ccc(Cl)cn3)C1)=O)CC2 C(=O)(C(O)CC(F)F)N1CCC(C(CNC(c2cc(C(C)(C)C)n[nH]2)=O)F)CC1 N1(C(c2nc(CCC)sc2)=O)CCC2(CC1)CC(NC(c1conc1C)=O)CO2 C#CC1(C(=O)NC(C)CN2CCCC2=O)CCN(C(=O)CC2CC(=O)C2)C1 c1(OC)cc(C(=O)O)ccc1CNC1CN(C)CC1(C)C C1(CNC(CC)=O)CC2(CC2)CN1C(=O)C(c1cccc(C#N)c1)C(C)C c1(C(N(CCCN(C(c2ccc(C)cc2)=O)C)C)=O)ccc2ncncc2c1 C1(CNC(C(C)CN(C)C)=O)CCN(C(c2cnn(C)c2F)=O)C12CC2 Cc1nn2cc(C(=O)NCC3C(C)CCN3C(=O)CCc3cncn3C)nc2s1 CC(C)C1CNC(=O)CCN(C(C2OCCC2C(F)(F)F)=O)C1 C1(NC(CC2CC(OCCCC)C2(C)C)=O)CC2(CCNCC2)CO1 Cc1cc(C(=O)NC(C)(CNC(=O)Cc2ccnnc2O)C2CC2)nn1C(F)F c1(C(=O)NC2CCN(C(C3CSCCS3)=O)C23CC3)c[nH]c2cc(Cl)ccc12 C1(NC(c2cncc(N(C)C)n2)=O)CCC2CC1CN2C(c1ccc(Cl)cn1)=O CCC(C)(CO)C(=O)NCC(C1CC1)N(C)C(C1(F)C(C)(C)C1(C)C)=O N1(C(C2(NC(N)=O)CC2)=O)CCC(CCNC(=O)C=Cc2cnc[nH]2)C(F)(F)C1 N#Cc1ccccc1OCC(=O)NC1CC(O)(CNC(=O)CC2CCCCO2)C1 c1(C(=O)NCC2C3CN(C(C4(C(CC)=O)CC4)=O)CC32)nc(Cl)ccc1Cl c1(C(=O)NCC(C)N(C(=O)CN2CCOCC2)CC)cccnc1C c1(C(=O)NCCN(OC)C(=O)C2CC(OC)C2)cccc2[nH]ccc12 N1(C(C(=O)NCc2n(C)ccc2)=O)CC(=O)NCC1C(N)=O C1(N(CC(CC)C)C(=O)N(C)C)CCN(C(=O)C(C)C2(O)CCC2)C1 N1(C(C(C)Sc2ccccn2)=O)CCCC(C(C)NC(=O)CNC(=O)C2CC2)C1 c1(C(N2CCC(C(C)C(=O)NCc3n[nH]cc3C3CC3)C2)=O)cc(O)nc(O)n1 N1(C(C2(OC)CS(=O)(=O)C2)=O)CCC2(C1)CN(C(=O)C=CC1CCCO1)CCO2 C1(NC(CCC(=C)C)=O)CN(C(c2cc(F)c(N)c(F)c2)=O)CC(C)(C)C1 c1(CC(=O)NCC2(F)CC(CNC(CCOC)=O)C2)ccccc1C C1(NC(C2(CC=C)CCC2)=O)CCC(NC(C2CCOCC2C)=O)CC1 c1(OCC)cnncc1C(=O)N(C)CCOCCNC(=O)CNC(N)=O C1(C)(C(=O)NC(CC)CNC(c2csc(-c3ccsc3)n2)=O)CCCOC1 c1(CC)ccc(C(=O)NC(C)(C)C(C)NC(=O)COC2CCOCC2)cn1 N1(C(c2cc(C)[nH]n2)=O)CC(F)CC1CN(C)C(C1CCN(S(C)(=O)=O)CC1)=O C(=O)(CC1COCc2ccccc21)NC(C)CNC(c1cc(Cl)cc(F)c1N)=O c1(C(=O)NC2CC(N(C(=O)CC(F)F)C)C2)ccc(F)c(F)c1N N1(C(C(C2CC=CCC2)NC(=O)CSC2CC2)=O)CCCC2(CC2)C1 CCC(CC(F)F)C(=O)N1CC(O)(C(C)NC(=O)CCn2ccnc2C(C)C)C1 N1(C(c2nc(CC)oc2C)=O)CCOCC(NC(=O)Cn2ncc(Br)n2)C1 c1(C(N(CCNC(C2CCCC2OC)=O)CC)=O)ccc2cccnc2c1O Cc1cc(C(=O)NC2COCCN(Cc3ccc(Cl)nc3Cl)C2)ccc1O CCC(CC)C(C(=O)NCC(CNC(C1NC(=O)OC1(C)C)=O)S(C)(=O)=O)OC Cc1ccc(C)c(C(=O)NCC(CNC(=O)C(C)Cn2ccnc2)S(C)(=O)=O)n1 C1(C2CN(C(C3CC3C(F)(F)F)=O)C2)(NC(C(c2cn(C)nc2)=O)=O)CC1 C(=O)(C1COc2ccc(F)cc21)NC1C(NC(C2(C(=O)OCC)CC2)=O)C1 O=C(CC1OCc2cc(Cl)ccc21)NCCNC(=O)C(c1cccc(Cl)c1)(F)F C(C(C)(C)NC(=O)C(=O)NC1CC1)NC(C=CC(=O)NC1C(C)C1)=O c1(OC)ccc(C(C)=CC(=O)NC2CCN(C(=O)C3CC3)CC23CC3)cc1 c1(C(=O)NCC2C(NC(=O)CC3CC3(Cl)Cl)C2)cc(C(F)F)cc(F)c1 c1(CC)ccc(CC(N2CCC(N(C(C3CCCCC3O)=O)CC)C2)=O)c(F)c1 C=CC(C)CC(=O)NCCOC(C)(C)CNC(C1CCC(O)C1)=O CS(=O)CCC(=O)N1CCC(CCCCCNC(=O)CC2(C)CCC2)CC1 c1(C(N(C2CCN(C(C3CC(N(C)C)C3)=O)C2)CCO)=O)ccc(Br)c(O)c1 c1(C(=O)NC2CN(C(C(c3ccc(F)cc3)OC)=O)CC2C)ccnc(F)c1N c1(C(=O)NC(C)CNC(=O)C(C)(C)Oc2ccccc2)cccc2nc(O)oc12 C(=O)(CCC(C)(C)C)N1CCC(CN(C(=O)Cc2ncns2)C)C1 c1(CNCCNc2c(OC)ccc(Cl)c2)cc2cc(Br)ccc2o1 C1(C(=O)NC2(CO)CC(C)C2)CCCC(NC(c2ccc(CO)cn2)=O)CC1 CCC(C)C(O)C(C)C(=O)NC(Cn1cccn1)C(=O)NC1(CCCCO)CC1 c1(CC)nc(C)[nH]c1C(=O)NCC(F)CNC(=O)C(CCSC)OC c1(C(=O)NCCCN(C(CCN(C(CC)CC)C)=O)C)ccccc1Br c1(C(=O)NCC2CCC(F)(CNC(=O)C(O)C3CC3)C2)cnc2c(c1)CCOC2 N1(C(CSCCC#N)=O)CCC2(CC1)CCN(C(=O)CCc1cc[nH]n1)CC2 c1(CC)ccc(C(=O)NCCc2n[nH]cc2C(=O)NCC2COCC2O)o1 C(=O)(C(O)CC[S+](C)C)N1C2(CN(C(C3C(C)OCCC3)=O)C2)CC1 c1(C(=O)NCCN(C(c2n(C)cnc2)=O)C2CC2)c[nH]c2cccc(Br)c12 Nc1cc(F)c(CC(N2CC3CCC(C2)N3C(C2CCCC(O)C2)=O)=O)cc1F N1(C(=O)NCCCCC(C)(F)F)CC(CO)Oc2ccccc21 C1(NC(=O)CC2CC(NC(c3cccc4[nH]ccc34)=O)C2)CC2(CNC(=O)O2)C1 c1(-c2nc(N3CCC(NC(CC(C=C)(C)C)=O)CC3)sn2)ccc([N+](=O)[O-])cc1 C(CNC(=O)C(C)(C)c1cncnc1)(CO)(CO)N(C)C(C1CNC(=O)N1)=O c1(C(N(CCNC(C2CCN(C3CCCCC3)C2)=O)CC)=O)oc(C)nc1C C1(NC(c2ccn(CC)n2)=O)CCCCC1NC(=O)C=CC(C)(C)C N1(C(C(C)(C)CO)=O)CC(CC(=O)NCc2ccc(C(=O)O)o2)C2(CC2)C1 C(=O)(C1CCCc2c[nH]nc21)NCC(CNC(C(C(CC)C)NC(C)=O)=O)O Cc1ccc(-n2nc(-c3ccc(C)o3)nc2C(=O)NC2CC2)cc1 c1(NC(C(c2ccccc2)NC(C2CC(F)C2)=O)=O)cncc(CO)c1 CS(=O)(=O)c1ccc(C(O)CNCC2CC3CNCC23)cc1 C1(OC)CC(NC(c2cnn(C(C)C)c2)=O)CN(C(c2cccc[n+]2[O-])=O)C1 C1(C(=O)NC2CCOCC2)CC1C1(C)COC1.CC1CC2(CCC2)NC1=O c1(NC(N(C2CC2CNc2ccc(C(F)(F)F)cc2I)C)=O)ccc(C#N)c(O)c1 CC(CCC(=O)N1CC(O)C1)NC(c1c[nH]cc1C1CC1)=O n1(CC(=O)NCCN(C(=O)CC#N)C(C)C)cc(CN2CCC2)nn1 c1(C(N2CC(NC(CSC)=O)C3C2C3)=O)c(C(F)(F)F)nn2ccccc12 C(=O)(C1=CCC(C)CC1)NCCCC1(NC(c2c(C)nc(COC)s2)=O)CC1 C(=O)(C(C(C)CC)NC(=O)C1=C(C)CC1)NC(CCC=C)CO c1(C(=O)NCCC2C(C)CCC2)cc(OC2CCCC2)cc(Br)c1 CS(=O)(=O)c1cncc(C(N2CC3C(C(=O)Nc4ncc(F)s4)C3C2)=O)c1 c1(CN2CCN(C(c3cnc(Cl)cc3I)=O)CC2)ccccc1[N+](=O)[O-] c1(C(=O)NC2C(C)N(C(C34CCCC3C4(F)F)=O)CC2)cc2nccn2c(O)n1 C(=O)(C1OC(=O)c2ccccc21)NC1CC(OC)CN(C(=O)CN(C)C(N)=O)C1 CC1c2ccccc2N(C(N2CCCC3(CCCNC3=O)C2)=O)C1C C1(C(N(C2CCN(CCC(=O)NC3CC3)C2)C)=O)CCN(Cc2cnc[nH]2)C1 N1(C(c2ccc(OC(C)C)nn2)=O)CCN(Cc2cc(F)cc(Br)c2)CC1C#N C1(C(=O)NC2CN(C(CCCCOC)=O)C(C)(C)C2)CC(c2ccccc2)=NO1 CC1CC(O)CCN(C(=O)C(Cc2cc[nH]n2)NC(c2cccc(=O)n2C)=O)C1 C(C(C)(C)C(=O)NC(c1ccccc1)C(=O)NCCCC(C)(F)F)OCC C1(F)(CNC(C(C)CCN(C)C)=O)CCN(C(=O)C(F)=CC2CC2)CC1 C(=O)(C(C(C)C)n1cc(Cl)cn1)NC(CC)CNC(c1ccc(C2CC2)o1)=O C1(C(=O)NCC(C)(CO)NC(CC=CC)=O)CCCCC12CCC2 C1(CC=C)(NC(c2cc(CF)on2)=O)CN(C(c2coc(-c3cnn(C)c3)n2)=O)C1 c1(C(N2CCC(C(F)(F)F)C2)=O)c[nH]c2cc(-c3cccnc3)cnc12 S(=O)(=O)(C1CCN(C(C2CCCN(C(C)C)C2)C(=O)NCC(F)F)CC1)NCC CC1(C)CC(CNC(=O)CC2CC(F)(F)C2)N(C(c2csnc2Br)=O)C1 C(c1cncn1C)=CC(N1C(C2(NC(CC3(OC)CCC3)=O)CC2)CCC1)=O N1(C(COCCCC(C)C)=O)CC2(CCN2C(=O)CCC2CCCO2)C1 C1(CCOC)CCCCN(C(c2nonc2N)=O)C1 N1(C(c2n(CC=C)ccc2)=O)CC(C2(NC(=O)CC3(O)CCCCCC3)CC2)C1 N1(C(CCC(=C)Cl)=O)CCCC2(NC(c3ccnn3C(CC)CC)=O)CC2C1 c1(CC(=O)N(CC(C)NC(=O)CCc2cncs2)C)ccc(C#N)c(F)c1 N1(CC#C)CCC(C(N2CCC(C)C2CNC(=O)C(F)=C2CCCC2)=O)CC1 N1(C(C(C)SCCCC)=O)CCC(NC(C2CCC(C3CC3)C2)=O)C(C)(C)C1 c1(NC(C2N(C(c3ncc(C#C)cc3C)=O)CC(O)C2)=O)ccc2nccn2c1 C1(CC=C)(NC(=O)CSc2cccs2)CCCN(C(C2CC2C(N)=O)=O)C1 C(=O)(C(C)C(=O)NCc1occc1C(=O)NC1CCN(C(N)=O)C1)OC N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)Cc2cncs2)CC1CCO Cc1cnc(NC2CCCCCCC2C(N)=O)c(S(=O)(=O)NCc2cnsc2)c1 C1(COC)CCCN(C2CCN(C(c3ccc(OC)cc3)C)CC2C)CC1 C1(CNC(C(C(C)C)SCC)=O)CN(C(=O)Cn2nc(C)oc2=O)CC(C)(C)O1 c1(C(=O)NCC(C2CC2)NC(C=C(CC)C)=O)ccc(C)c([N+](=O)[O-])c1 c1(CC(=O)N(C2CCCN(C(=O)CC3(O)CCC3)C2)C)cc2ccccc2s1 Cc1ccnc2ccc(C(=O)NC(C)CCCNC(=O)CCC(C)C)cc12 C1(CC)CCC(C(=O)NC2CCOCC2C(=O)NCCCCN2CCCC2)CC1 c1(OCC)ccc(C(=O)NC2CCN(C(c3c(Br)cncc3Br)=O)C2)cc1OC c1(C(N2CCN(C(c3cc(C)cc(N)c3)=O)CC2C)=O)cc(F)cc(C)c1C C(=O)(C=C1SCC(=O)N1C)NC1C(NC(CN(C)C)=O)COC1 C1(C)(CC)CC(NC(c2ccnc(N(C)C)c2)=O)CN1C(=O)CC1CCOCC1 C1(CCNC(c2cc(C(=O)OC)on2)=O)CN(C(C23CCC2C3)=O)CCS1(=O)=O N1(C(CC)=O)CCC(NC(C2CCC3(CC2)CC3)=O)C(CO)C1 C1(CCNC(CCn2ncc(C)c2)=O)CSCCN1C(=O)CSc1n[nH]c(C)n1 c1(NC(C2CCN(C(C3(C(F)(F)F)CCC3)=O)C2)=O)cc(F)c(O)cc1Cl C(=O)(C(C(C)C)S(=O)(=O)C1CCCCC1)N(CCC)CCNC(c1cnc[nH]1)=O N1(C(C2C(COC)C2)=O)CCC(CNC(c2ccc(C)cn2)=O)C(C)C1 N1(C(C(CCC)(C)CC)=O)CCCC2(CC(NC(C3CC4CCC3CC4)=O)C2)C1 N1(C(CC2(C)CC2F)=O)CCC(C2CN(C(=O)C3=CCCC3)C2)CC1 C(=O)(C(C)(C)C(C)O)NC1CCC(CC(=O)NC(c2c(C)noc2C)C)C1 c1(C(=O)NC(CC)(CNC(=O)Cc2nc(C)no2)CC)ccnc(OC)c1Br C1(C)(CC)CC(NC(c2cocn2)=O)CN1C(=O)Cc1cc(Br)ccc1F CC1(CNC(C2CCS2(=O)=O)=O)CCCN(C(c2ccc3c(c2)CC3)=O)C1 c1(C(N2CC(C)C(NC(=O)CC3CCN(C)CC3)C2)=O)nnc(Cl)cc1N C=CCCCCCNC(=O)C(CO)NC(c1ccoc1CC)=O Cc1cc(C(N2CC(NC(=O)CN(C)C)C3(CC3)C2)=O)nnc1C Cc1c(N2CC3CCOC3CC(C)(C)C2)nc2c(F)c(Br)cnc2c1Cl Cc1cc2nc(C(N3CC(=O)NC4(CC4)C3)=O)cc(=O)n2o1 C(=O)(C(O)CC(N)=O)NCC(CNC(=O)CCCn1cccn1)OC N1(C(C(C)N(C(CCC(C)SC)=O)C2CC2)=O)CC(CO)CC12CCC2 Cc1cc(C(N2CC3CC(C2)N3C(c2cc(O)ccc2F)=O)=O)cc(O)c1 N1(C(CNC(N)=O)=O)CCC(F)(F)C(CNC(=O)C=Cc2ccccc2)C1 C12(CCNC(C=CSC)=O)CCC1CN(C(c1ccc(C(F)(F)F)o1)=O)C2 N1(C(C2(CC)COC2)=O)CC2(C1)CN(C(=O)C(C)Sc1ccc(C)cc1)C2 C(=O)(C(CCS(C)=O)N(C)C)N1CCC(C)(NC(C=C(COC)C)=O)C1 C(C(C)(O)CC(=O)N(C1(C(=O)NCCC2CCCC23CC3)CC1)C)OC C(C(C)(C)C(=O)NC1CCCC(CN(C)C(C23CC(COC)(CO2)C3)=O)C1)OC C1(CNC(c2cc(OC)no2)=O)CC(F)CN1C(c1cnn(C(C)(C)C)c1C)=O c1(C(=O)NC(CC)(CNC(=O)C#CC2CCC2)CC)cc(F)c(F)cc1F N1(C(CCN(C(C)=O)C)=O)CCC(NC(=O)CC2(C)CC2)CC1C1CC1 C1(CNC(C2CN(C(C)C)C(=O)C2)=O)CC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 C1(CC(=O)NC(CC=CC)CO)CN(C(=O)CCCCC)CC1C c1(CCC)n[nH]cc1C(N1CC(N(C(=O)C(C)CC2CCC2)C)C1)=O N1(C(CC=CCNC(c2c(NC)cncc2)=O)=O)CC(C)OCC(C)(C)C1 C(=O)(CCNC(=O)C=CC(C)(C)C)N(C1CCOC1)CC#CC CCC(C)(CC(=O)O)NC(=O)CCn1cc(-c2cc(OC)cc(Cl)c2)nn1 N1(C(CNC(=O)NC)=O)CCN(C(=O)C(C)OCCC(C)C)C(CC2CC2)C1 Cc1cc(C(N2CC(NC(c3cccc(Br)c3)=O)C(C)C2)=O)c2c(C)noc2n1 Cc1nc2cc(Cl)ccc2cc1C(=O)NCC1CC(F)CN1C(=O)C1=CCSC1 CCC(CC)(CC(=O)OC)C(=O)N1CC(NC(=O)CCS(C)=O)C2(CC2)C1 c1(CC(N2CC(CCn3cc(-c4c(C)cnn4C)nn3)C2)=O)c(Cl)cccc1Br Cc1cccc2c1NCCC2C(=O)N1CCCC1CNC(=O)C=CC1CC1 CC1CCN(C(=O)CCCc2ccsc2)CC1CNC(C1COC(=O)C1)=O c1(C(=O)NC(C(=O)NC(CC)C)C2CC2)cnnn1C Cc1cncnc1C(=O)NCC(O)CN(C)C(c1nnc(S)n1C)=O C#CC1CCN(C(=NCCSCC)NCc2ccc(Cl)nc2C)C1 c12[nH]c(C)c(c1C)C(=O)N1CC(C1)CC(C)NC2=O.c1(CC)cccc(OC)n1 CC(N=c1[nH]c2ccccc2s1)C(=O)N1CC(C(=O)NCc2ccc(F)cc2)C1 C1(C(N2CC(C)C2)=O)(CO)CCCN(C(=O)CC2(c3ccccc3)CC2)C1 C(=O)(C1=CCCC1)N1CCC(CCNC(C2C(C)C2)=O)C1 c1(C(=O)NCCC(CNC(c2c(SCC)cncc2)=O)(C)C)nn(C)c(N)c1C c1(C(=O)NC2C3(CC(NC(CCCOC)=O)C3)C2)cnn2ccncc12 c1(OC)ncc(C(=O)NC2CCCN(C(C34CC(CO3)C4)=O)C2)nc1C c1(C(=O)NC2C(NC(c3cc(OC)ns3)=O)COCC2)noc2ncccc12 CCN=c1[nH]c2ccccc2s1.C1(C(=O)NCCOCCC2CC2)CC2CC2C1 Cc1c(NCC(C(F)F)c2ccccc2)ncnc1N1CCC(c2nccs2)C1 C1(C(N(CCCN(c2ccc3nnnn3n2)C)C)=O)CCc2nnc(O)cc2C1 N1(C(C(C)OCCC=C)=O)CCCCC1C1CCCN(C(c2cnc(C)cn2)=O)C1 N1(C(CC2(NC(C)=O)CC2)=O)CC2=C(C1)CN(C(=O)C=Cc1ccccc1)C2 CC1=CCC(C(N2CCCCC2C2CCN(C(c3ncnc(=N)[nH]3)=O)C2)=O)CC1 Cc1nn(CC(=O)NC2CCN(C(=O)Cc3cnn(C(F)F)c3)CC2)c(C)c1C CC(COc1ccccn1)N=c1[nH]c(=N)[nH]c(=NC2CC2C2(C)CCOCC2)[nH]1 C(C1CCCc2cccnc21)NCC(C1CCNCC1)C C1(CN(C(CC)C(=O)NC(C2(C(=O)N)CC2)C)CC)CC2C=CC1CC2 CC(C)(C)C(CNC(=O)C1=NOCC1)C(=O)NCC1CC2C=CC1O2 C(CN=c1[nH]cnc2c(F)c(F)ccc12)NC(C1ON=C(C(C)C)C1)=O C1(NC(c2n(C(C)C)cc(Br)c2)=O)CC2CC(NC(c3cn[nH]c3)=O)C2C1 c1(CC)cc(=NC(=O)C2=NOC(c3ccc(F)cc3Cc3ccccc3)C2)[nH][nH]1 N1(C(C(n2ncc(C)c2)C)=O)CCC2CCN(C(=O)CNC=O)CC12 c1(C(=O)NC2CCN(C(CC3NC(=O)OC3)=O)C23CC3)cncc2cnccc12 C1(CC(=O)NCC(CC)CO)CCC(NC(=O)CNc2cccnc2)CC1 C(=O)(C1CCc2c[nH]nc21)NCC(CCOC)NC(c1cnc(O)n1C)=O C1(C(N(CCN(C(c2c[nH]c(=NCC)s2)=O)C)C)=O)CC(C)(C)OC1(C)C c1(CC)nc(C)[nH]c1C(=O)NC1CCN(C(=O)C(c2cccnc2)OC)CC1 N1(C(c2nn(CC)c(O)c2)=O)CCCCC(CNC(=O)CCOCCN(C)C)C1 C12(C(N(C3CCC3)CC#C)=O)COCC1CN(C(C1CSC1)=O)C2 c1(C(C(=O)NC(CC)(C)CC)N(C)CCNC(C)=O)ccc(C(F)(F)F)c(F)c1 N1(CCC(=O)NC2C=CCN(C(CC(CCC)O)=O)C2)CCCc2ccccc21 C1(C(=O)NC(C(CO)NC(C(C)=C2CCCC2)=O)C)CC(C)CC(C)C1 c1(CC(N2CC(F)(CNC(C3CCC(C(=O)OC)C3)=O)C2)=O)cc(C)ccc1C N1(C(c2ccc(C#N)cc2)=O)Cc2ccc(O)cc2CC1C(=O)N1CCC1 CCC(C#N)C(=O)N1CCCC1CCNC(=O)CC1(C)CCCC1 c1(NC2C(CC(C)C)COC2)cc(F)c2oc(O)nc2c1 C1(CC(=O)NCCN(C(c2cccc(C#N)c2)=O)CC)CC2(CCOCC2)CO1 c1(NC(CC(=O)NCc2cccc(Br)c2Br)Cc2cccs2)cc(Br)nc(Br)c1 C1(NC(=O)COc2ccccc2)C2CC3C(C2)C13C(=O)NCCCC(F)F CN1CCC(O)(C2(C(N3CCC(CN(C(=O)C4=CCCCO4)C)C3)=O)CC2)CC1 Cc1nn(C)cc1C(N1CCC(C(N2CCC(O)(CN(C)C)C2)=O)C1)=O c1(C(=O)NC2C(NC(CSCC=C)=O)CCCC2)cnc(C)nc1OC c1(CNC(C2N(C(C(CN(C)C)(C)C)=O)CCC2)=O)cc(F)cc([N+](=O)[O-])c1 CC1CN(C(C2CC(=C3CC3)C2)=O)CC(CCNC(=O)Cn2ncccc2=O)O1 Cc1cccc([N+](=O)[O-])c1NCC1(F)CC(NC(=O)C=Cc2ccccc2F)C1 C=C(Br)CC(C)(C)C(=O)NCC1CCCCN1C(=O)C(C)=C(C)CC c1(C(=O)NCCc2ccc(CNC(CC(=C)C)=O)cc2)ccc2c(n1)CCCC2 c1(C(N2CC(C(C)NC(C3(c4ccnn4C)CC3)=O)C2)=O)c(F)cncc1Br Cc1cnc(C(=O)N(C)CCOCCN(C)CCC2CCCC2(F)F)c(C)c1 c1(C(=O)NCCCNC(C2(COC)CC2(F)F)=O)cc(SC)c(Cl)cc1Cl C1(C(=O)NC2(COC)CCCC2)CC12CCN(C(c1cn[nH]c1)=O)C2 Cc1ncc(CC(N2CC=CC2C(=O)NOCCF)=O)s1 C1(C(N(CCN(C(=O)CC2COCC(C)(C)O2)C)C)=O)CC(F)(F)C1(C)C C1(CC(=O)NC(CNC(CC=CCC)=O)(C)CO)CSc2ccccc2NC1=O c1(C(N2CCC(F)(CNC(CCC(C)N(C)C)=O)C2)=O)ccn2ncccc12 CC1CN(C(=O)C(F)n2cccn2)CCCN1C(=O)Cc1ccc(C#N)cc1F N#CCCCCCC(=O)NCC1CCN(C(C2CCCS2)=O)C1 C1(NC(c2n(CC)ccc2)=O)CCCCN(C(=O)C(C)OCCC(C)C)C1 N1(C(c2c(CC)n(C)nc2)=O)CCC(C)C(CC(=O)NCCCCC(C)C)C1 C1(NC(CCOCC)=O)CCC2(CCN(C(C3CCC3NC=O)=O)C2)C1.C(C)=O c1(NC(N(c2cccc(C(=O)NCC3CC3)c2)CC)=O)ncn2c1COCC2 C1(CC(=O)OC)COCCN(C(=O)NCC(C)(Cc2ccccc2)C(C)O)C1 C(CCC(C)CC(=O)NCC1(NC(=O)CC2CCC3(CC3)CO2)CCC1)=C(C)C c1(C(C)=O)[nH]c(C)c(C(N2C3CCC2(CNC(=O)COCC(C)C)CC3)=O)c1C S(=O)(=O)(c1ccc(NCC2CCC2)c(F)c1)N1CC(C(C)O)OCC1 C1(C(N(C2C(C)CCC2)C)=O)CC2(CC2)CN1C(=O)CCc1cnc[nH]1 C1(C(C)C)CC(CC(=O)NC2(CN(C)C(c3ccccc3F)=O)CC2)CCO1 C1(NC(C2C(C(=O)OCC)CCO2)=O)CCCN(C(c2ncncc2Cl)=O)C1 c1(C(=O)NC(CO)CCCCNC(c2ncsc2Cl)=O)cc2ccc(O)cc2[nH]1 C1(CC(N2CC(CCCCNC(CCOCCN(C)C)=O)C2)=O)CCCC1(F)F C1(NC(CC2C(CC)C2(F)F)=O)CN(C(c2c[nH]nc2OC)=O)CC12CCC2 c1(-c2cn(CC(CNC(C(C)NC=O)=O)(F)F)nn2)cccc(Cl)c1 C1(NC(Cc2cccc(C)c2)=O)CC2(C1)CC(C(=O)NC(C)(C)CN(C)C)C2 N1(C(c2ccn(C)c2)=O)CCOCC2(COCCN2C(c2ccc(Cl)nc2)=O)C1 c1(CC(N2CCN(C(CC(CC)C)=O)CC2CC)=O)ccc2c(c1)OC(F)(F)O2 C1(C(=O)NCC2C(NC(=O)Cc3ccc(F)c(Cl)c3)C2)CCc2nnc(O)n2C1 C1(CN(C(=O)Cc2ncc(Br)cn2)C)CCN(C(C2CC2F)=O)CC1 c1(C(N2CCCN(C(C(CC)COC)=O)C(C)C2)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(C)(C)OC)occc1SCc1cocn1.C1(=O)NCCN1 N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CCN(C(=O)C(C)O)CC1CC(F)(F)F N1(C(C=CC)=O)CCCC2(CCCN2C(c2ccc(Cl)c(OC)c2)=O)C1 C(=O)(C(C)(O)C1CCC1)NCCC(C)NC(c1cnc(Cl)s1)=O C1(OC)COc2cc(C(=O)NC3CCC(C)(C)CC3C)nn2C1 n1(CC(=O)NCC(=O)OC)[nH]cnc1=NCc1ccccc1CN=[N+]=[N-] C1(NC(CCCOC(C)(C)C)=O)CS(=O)(=O)CC1NC(C1CC2(CC2)C1)=O CC(C)C#CC(=O)NCC1CCC(NC(C2CCN2C2CCCC2)=O)CC1 N1(C(c2cnn(C)c2Cl)=O)CC(NC(c2c(F)cccc2Br)=O)C(C#N)C1 CCCCCCC(=O)NC(CNC(C1CCC(C(C)C)CC1)=O)C(C)C C1(NC(C(C2CCOC2)OCC)=O)CC(F)(CNC(=O)CC2CN(C)C2)C1 N1(CC(=O)Nc2ccc(CCC)cc2)CC2CCC(F)(C2)C1 CC1=C(C(=O)NC2CN(C(=O)C(C)Oc3cc(F)cc(F)c3)CC2C)CCCC1 C1(O)(CC(=O)NC(CC)(C)CCNC(=O)CN2C(=O)CCC2=O)COC(C)(C)C1 CCC(C#N)C(=O)N(CCCN(C(=O)CCc1ccc(Cl)s1)C)C N1(C(c2nc(OCC)oc2)=O)CC(CNC(=O)CSc2csc(=N)[nH]2)C(C)C1 N1(Cc2cc(OC)c(O)cc2)CCCC2(CCN(C(c3cnc(O)[nH]3)=O)C2)C1 N1(C(C(C)OCCCC)=O)CCC2(CCC(NC(=O)CCOC(C)C)CC2)CC1 C(=O)(C(C)(C)C(C)NC(=O)CC1(O)CCC1)NCC1C(C)C1 N1(C(c2c(C)occ2)=O)CCCCC(CNC(=O)CCNc2cncnc2)C1 c1(OCC)cc(F)ccc1NC(C1OCCC1NC(=O)Cn1ncn(C)c1=O)=O C1(NC(c2c(C)nc(C(C)OC)s2)=O)CN(C(=O)C=CSC)C(C)(C)C1 c1(C(=O)NCCN(C(=O)CN(C)C(N)=O)CC)cc2ccoc2cc1F C1(C(C)O)CN(C(=O)CN(C)C(C2CC23CC3)=O)CCO1 CC(F)CC(=O)NC(C)(C)CCN(C)C(C1CC=CCC1)=O C1(NC(C(CC=C)C)=O)C2COCC1CN(C(c1cc(C)[nH]n1)=O)C2 C12(CC(=O)NCC(C)CNC(=O)C(C)n3ccnn3)CCCN1CCC2 c1(CNCCNCCC(C)CO)ncccc1O C#CCC(C(=O)NOc1ccccc1)NC(=O)COC1CCC1.OC c1(C(=O)NCCC2OCCCN(C(CC(CC)C)=O)C2)cc(Cl)cc(C)c1OC CC(CCNC(=O)CCOC1CN(C(C2CCCCO2)=O)C1)C(C)(C)C N(C(=NCCCn1cccn1)NC1CC(CO)c2ccccc21)CCSC c1(OC)ccc(CC(=O)NC2CCN(C(c3cccnc3N)=O)CC2F)c(F)c1 C(=O)(C(CNC(=O)NC1(F)CC1)CC1CC1)N(C)Cc1ccccc1 Cc1ncc(C(N2CC(O)CCC2C(=O)NCC2CC3(CCC3)C2)=O)cc1C#N CC(N=c1[nH]c(=NC(C)CS(C)(=O)=O)[nH]c2c1COC2)C1CCC1 Cc1[nH]nc2c1CC(C(=O)NCCCC(C)(C)NC(=O)C(O)C(F)(F)F)CC2 Cn1ccc(C(=O)NCC2(NC(=O)C(c3ccccn3)O)CCCCC2)cc1=O N1(C(CSCC#C)=O)CCN(CC(=O)NCC2CC(CCC)C2)CC1 c1(OC)cccc(C(c2nnnn2C(C)(C)C)NC2(C)CCOC2)c1 N1(c2cc(N(C)C)[nH]c(=N)n2)CCC2CC(C(N3CCNC(=O)CC3)=O)C2C1 c1(CNC(C(CO)N(C)C)=O)cncc(C(=O)NC2CC(=O)N(C3CC3)C2)c1 C(=O)(C(C)CC1CC1)N(CCN(C(CC1C(OC)CC1)=O)CCOCCO)CC c1(C(N2CCN(CC3CC3)CC2)C(=O)NCC(C)C)ccnc(Cl)c1Br [N-]=[N+]=NCCCC(=O)NC1CCCCCC1NC(=O)Cn1cc(Cl)cn1 C1(NC(CCC=CC)=O)CCC2(CCN(C(c3ccnc(SCC)c3)=O)CC2)C1 C(=O)(C1=NOC(C)C1C)NC(CCC(=O)NC(CCOC)C)(C)C c1(C(=O)NC2(CCO)CN(C(=O)CC3CCOC3)C2)cccc2sncc12 Cc1scc(C(=O)NC2C3CC2N(C(c2cc(C(N)=O)c[nH]2)=O)C3)c1C c1(OC)ccc(Br)c(C(N2CCC(Cc3cn(CC(C)(C)C)nn3)CC2)=O)c1C C(=O)(C(C)CN(C)C(C1(c2ccno2)CC1)=O)N(C1CC(NC(C)=O)C1)C c1(CC(C2CC2)NC(CC=C(C)C)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)CC(F)F)NC1(C(=O)NC(CCC)CO)CCCCC1 N1(NC(NC(C2CCCCC2)C#C)=NCCCCl)CCc2cc(F)ccc21 c1(C(=O)NC2(C)CCN(C(C3C(COC)C3)=O)C2)cnc2cccnc2c1 C1(C(=O)Nc2ccc(OCC)nc2)CC2(CC2)CN1C(c1cc(I)ccc1Cl)=O N1(C(=O)CCN2CCCCC2)CC2(CCN(C(c3ccnc(Cl)c3F)=O)C2)C1 N1(C(c2c(C)onc2C2CC2)=O)C2CCC1CN(C(c1ccncc1F)=O)CC2 N1(C(C2CCC(CNC(c3ccc(SC)o3)=O)C2)=O)CCCCC(C)C1 C1(C(=O)NCCCNC(=O)COC(C)=O)(NC(C)=O)CCCCC1 c1(CNC(CC2(OCC)CCOCC2)=O)nc(C)cc(C)n1 S(=O)(=O)(c1c[nH]c(C(N2CC3CC2CN3C(=O)C(F)(F)CO)=O)c1)NCC S(=O)(=O)(c1cncc(Br)c1)N1C2CN(Cc3ccc(N(C)C)c(Br)c3)CC1C2 C1(C(=O)OC)CCN(C(=O)Nc2cccc(C3SCCS3)c2)C2(CC2)C1 C1(CC(=O)N(CC(=O)NCCCc2cnccn2)CCC)C(=O)NN=C1C C=CCC(F)(F)C(=O)N1CC(NC(=O)Cn2ccccc2=O)CC(C)C1 N1(C(c2c(C)cc(Cl)cc2)=O)CC2CN(C(C3CC(C)(C)OC3(C)C)=O)CC2C1 Cc1nc2ccc(C(=O)NC3CCN(C(c4ccc[nH]4)=O)C3C3CC3)cc2n1C C1(C(N2CCC(CN(C(=O)C=C3CCC3)C)CC2)=O)CC2(C1)CC(F)C2 N1(C(c2cc(C)c(-n3cncn3)cc2)=O)CCC(CNC(=O)C2CC2)C(F)(F)C1 c1(C(N(CC(C)NC(C2CC(n3cnnc3)C2)=O)C)=O)cc(C#N)on1 CCCCC(CNC(=O)CCNC(C1CCC1)=O)NC(=O)CC1CCC(=O)NC1 C1(CNC(CN2CC(C)(OC)C2)=O)CN(C(C2(C)COC2)=O)CC1(F)F c1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)ccnc(C(C)(F)F)c1 c1(CC(=O)NC2C(C)(CN(C(C(C)=C(C)C)=O)C)CCC2)cnn2c1CCCC2 Clc1cc(-n2cc(C3CCOC3)nn2)cc(Cl)c1Cl O(NC(=O)CC1(CNC(=O)CCOC2CCCC2)CC1)CCC=C CC1CCN(C(c2ncoc2C2CC2)=O)C(C)C1NC(=O)C=CC1CCCC1 CCC(O)(C(=O)N(C(CNC(c1ccc(C)nc1)=O)C1CC1)C)c1ccccc1 C(=O)(C(C)(C)S(C)(=O)=O)NCC1(C)CC(NC(C(C)Cc2ccccc2F)=O)C1 CCCCCCC(=O)NC1CC=CCC1C(=O)Nc1ccc(O)cc1 c1(CC(N2CC(CCNC(c3nc(OCC)oc3)=O)C2)=O)ccc(N(C)C)nc1 C1(NC(C(=O)NCc2ccc(C(=O)NCCOC)nc2)=O)C2CCC(C2)C1CN C1(NC(c2ccc(C)cn2)=O)CC(CNC(=O)Cc2cc(C)[nH]n2)C12CCC2 C1(CC(=O)Nc2cnc(C)s2)CCCCN1C(c1ccccc1-c1nn[nH]n1)=O C(=O)(C(C)(F)C(=O)NC(CNC(=O)CS(=O)(=O)Cc1cccs1)C(C)C)OC C12CCCCC1NC(=O)C=CCN(C)C2=O.C(=O)(CC1(CC2CCC2)CC1)OC N1(C(C2(CCNC(c3c(CC)[nH]cc3)=O)CC2)=O)Cc2ccnn2CC1C C12CCCN(CC1)C2=O.C1(C(=O)N(c2ccccc2)C(C)C)(OC)CCN(C)C1 c1(C(N2CCC(C)C(NC(=O)Cc3ccno3)C2)=O)c(N)cc(F)cc1F C(=O)(C1(C)CCCc2ccccc21)NC1C(NC(c2c(C)ccc(F)c2N)=O)C1 N(C1CCc2sc(Cl)cc21)C(c1c(C)n(-c2cnn(C)c2)nn1)=O C1(C(=O)NC(CO)C2CC2)CN(C(C2(O)CCCCC2)=O)CC12CCC2 C=CCCN=C(NCCC1CN(C(C)C)CCO1)N1CCC(CC)C1 S(=O)(=O)(c1ccc(C(=O)NCC2(F)CC(NC(=O)C3=COCCC3)C2)cn1)NC C1(N(C)C(c2cc(C(F)F)no2)=O)CN(C(c2cc(O)nn2C)=O)CC1(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)C(=O)N2)OC.n12c(C)cc(c1C)C=CC2 Cc1c(C(N2CCC(CC(=O)NC3CC(C)C3(C)C)C2)=O)sc2cccc(F)c12 C1(NC(CCCCCCSC)=O)CC2CCCC(C1)N2C(c1ncncc1F)=O c1(C(N(C(C)CNC(c2ccc(CC(N)=O)cc2)=O)CC)=O)cnc(=N)[nH]c1 CCCC(C)CCN=c1cc[nH]cc1S(=O)Cc1ccc(C(C)(C)C)cc1 n1(CCC(N2CC(C(N)=O)(CNC(=O)Cc3cc[nH]c3)C2)=O)cc[nH]c(=O)c1=O C1(C(=O)N(C)CCN(C(=O)C=CC(C)C)C2CC2)(OCC)CC(F)C1 c1(NC(C(CC2CCC2)NC(C(CCCOC)C)=O)=O)cccc([N+](=O)[O-])c1 n1(C(CNC(c2ccc(Br)s2)C)=O)ccc(=NC(=O)OC(C)(C)C)[nH]1 CC(C)C(C(=O)NCCNC(C1CSCCS1)=O)S(=O)(=O)C1CCCCC1 O=C(CCCCCN1CCOCC1)NCC#CCNC(c1cc(F)ccc1F)=O C(C)(c1ccccc1C)=CC(=O)N(C)CC1(NC(c2c(OC)scc2)=O)CC1 N1(C(c2c(CC=C)cccc2)=O)CC2CCCC(C1)N2C(C1CC(C)(C)CO1)=O CCCCCCC(C)C(=O)N1CC(NC(=O)C(F)(F)C(C)(C)O)C2CC2C1 C1(C(=O)NC2CC(CCNC(CCc3n(C)ncc3)=O)C2)CCc2nnnn2C1 C(CN=c1[nH]cnc2c1COC2)N(C(C1C(CC)OCC1)=O)CC S(=O)(=O)(CC(=O)NCC1(F)CC(CNC(=O)C(c2cccc(F)c2)C)C1)NC C1(CNC(CC2CC(C)C2)=O)CCC(NC(c2sccc2CC(N)=O)=O)CC1 C1(=CC(=O)NCCC(C)(C)NC(Cc2cc(C)on2)=O)CCN(C)CC1 N1(C(CCNC(c2cn(C(C)C)nn2)=O)=O)CCCC(CO)C1 c1(C(=O)NCC2CC(NC(C(C(CC)C)C)=O)C2)cc([N+](=O)[O-])cnc1C c1(C(=O)NCC(C(=O)NC(CN(CCC)CC)C)N(C)C)cc[nH]c(=NC)c1 c1(C(N2C(CNC(CC(C)C(F)F)=O)CC(F)(F)C2)=O)cc2ccc(F)cc2s1 Cc1cnc(Cl)[nH]c1=NC1CC2CN(C(C3(C)CS(=O)(=O)C3)=O)CC12 CN=S(C)(=O)c1cccc(NC(=O)Cn2cnc3ccsc3c2=O)c1 N1(C(c2cnn(CCCl)c2)C(=O)NCCCSC)CCC(C)(O)C(C)(O)C1 Cc1cc(C)c(C(N2CCSCC2C(=O)N(C)CC2CCOC2C)=O)s1 C(CN=C(NCc1cn(C(C)C)cn1)NCC1CC=CCO1)OCC C(=O)(CP(C)(C)=O)N(CC(CN(C(=O)CN1CC2CC2C1)C)O)C c1(C(N2C3C(NC(C(C(C)C)(C)C)=O)CC(C3)C2)=O)sc([N+](=O)[O-])cc1Cl C=CCC(C(=O)N1CCC(C)(NC(c2ccc(CN(C)C)nc2)=O)C1)NC(C)=O C1(CNC(C(C)C2CCC2)=O)CC2COCC2N1C(C1(C)CNC(=O)C1)=O c1(N2CCC(COC)C2)nc(N2CCN(C)C(=O)C2)c2ccccc2n1 c1(C(=O)NC2CCN(C(C(N3C(=O)CCC3=O)CC)=O)C2)sccc1S(N)(=O)=O n1(CC)ncc(C(N2CC(NC(=O)COC3CCCCC3)C(CO)C2)=O)c1C N1CCc2ccc(F)c(Br)c2C1.Cn1c(OC(F)F)ccc1C1COCCN1 Cc1cc(Br)c2c(c1)CN(C(C1C3CCOCC13)=O)CC2 c1(C(=O)NC(C(C)C)CNC(C2(O)CCC2)=O)cc(CO)ccc1Cl n1(CC)nc(C(=O)NCCCCCCNC(c2csc(C(C)=O)n2)=O)cc1C Cc1c(Br)ccc(S(=O)(=O)N2CCCN(C3CCNC3=O)CC2)c1F c1(CN2CCC(NC(=O)C3CC3)C2)cn2c(Br)cccc2n1 Cc1ccc(I)c(NC(C2CN(C(c3cccn3C(C)C)=O)CCS2)=O)c1 c1(COC(C2(Cc3ccc(Cl)cc3Cl)CC2)=O)cc2cc(F)ccc2o1 Cc1nc(N2CCC(CCNC(=O)C(N3CCCCCC3)C)CC2)c(C)c(Cl)n1 C1(CC(=O)NCC(C)OC(F)F)N(C(=O)C(=O)C(C)(C)C)CCC1(C)C Cc1cccc(CC(=O)NCC2CC(F)CN2C(=O)CC2(C)CCCCC2)c1F c1(N(C)CC2CCN(C(c3cccn(C)c3=O)=O)C2)cc(C(N)=O)nc(Cl)n1 C1(CC(=O)NCc2n(C)ncc2)CCCCN1C(=O)CCn1cccn1 C(=O)(C(CC)(CC)OC)N1C(CN(C(C=CCN(C)CC)=O)C)CCC1 C1(OCCNC(C2(F)CCCC2)=O)CCN(C(=O)Cc2ccc(O)cc2)CC1 c1(C(C)NC(C(C)(C)OCC)=O)ccc(OCCN(CC(C)O)C)cc1 C1(C(=O)NCC(CN(C(CCOCC)=O)C)(C)C)CC12CCC(F)(F)CC2 C1(NC(c2c(C)ccn2C)=O)CC2(CCC(NC(C3CC4CCC3C4)=O)CC2)C1 c1(OC)cccc2c1CCC2NC(=O)C(C)(C)OCC(C)C C1(NC(C(C=C)O)=O)CC(OC)CN(C(c2c(C(F)(F)F)n[nH]c2C)=O)C1 C1(C(=O)NC(CC(C)C)(C)CNC(=O)COCP(C)(C)=O)CC2(C1)CC1(CC1)C2 C1(NC(CC(CC)O)=O)CN(C(=O)COC(C)CC)CCC1C(F)(F)F CCCC(C(=O)NOCCCC(=O)OC)NC(c1c(Cl)cnn1C)=O c1(C(=O)NC2C(NC(c3nc(N(C)C)oc3)=O)CC2)cc(Cl)sc1Cl c1(N(CC(=O)NC2CC(NC(c3cc(O)no3)=O)C2)C)ccc(Br)cn1 c1(C(=O)OC(CCC)c2ccco2)c(C)nc(Cc2ccc(CC)cc2)nc1O N1(C(C2CCCN(C(C)(C)C)C2)=O)CCN(CC(N2CCCC2)=O)CC1(C)CC Cc1cc(C(N2CCC(CN(C)C(c3cc[nH]n3)=O)C2)=O)cc([N+](=O)[O-])c1Cl Cc1ccnc(C(=O)NC(CNC(=O)C(C)OCc2ccncc2)C(C)C)n1 C(CNC(c1cc(Br)sn1)=O)(C(C)(C)C)NC(C1(OC(C)C)CCC1)=O c1(C(N(C2CCCN(C(C3C(=C)C3)=O)C2)C)=O)cc2c(F)cc(F)cc2o1 C1(C(CNC(C(N)=O)=O)NC(=O)CCc2ccc(Cl)s2)CCCS1(=O)=O c1(C(=O)NCC(CC(C)C)NC(C2(CC)CCNC2=O)=O)c[nH]cc(F)c1=O N1(C(CCCCCC#C)=O)CC(CNC(=O)C(=O)NCC)CC12CCOCC2 C(=O)(C(O)CCC(F)(F)F)N1CCC(CN(C)C(C2CC3(CCO2)CC3)=O)C1 C(CCCC(C)NC(=O)Cn1nnnc1C1CC1)NC(C1C(C(=O)OC)C=C1)=O C(=O)(C(C(C)(C)C)C1CCC(F)(F)CC1)NCCN(C(=O)C(F)C(C)(C)O)CC Cc1cn2c(C(=O)NC(C3CCN(C(C4CCC(=O)C(C)C4)=O)C3)C)cnc2s1 N=c1nc2c(c[nH]1)CC(C(N1CCCN(C(c3ccsc3)=O)CC1CO)=O)CC2 N1(CC)C(=O)CCC1C(=O)NCC1(C(N)=O)CN(C(=O)Cc2ccc(Cl)cn2)C1 c1(SCC(=O)N(CCCNC(C2C(C=C)C2)=O)C(C)C)ccccc1O C(=O)(C#CC(C)(C)CNC(=O)CC1CCC(C#N)C1)NCc1c(C)nccn1 c1(C(N2CC3CC(NC(C4(Br)CCC4)=O)CC3C2)=O)cc2ncccn2n1 c1(OC)ccc(O)c(CNC(=O)NCC2CCCCCC2SC)c1 C1(C#N)(C(=O)NC(C2CCN(C(C3CC(=O)NC(=O)C3)=O)C2)C)CC2C=CC1C2 N1(C(C2(C)CC2F)=O)CCN(C(c2nc[nH]n2)=O)CC1 c1(OC)ncc(Cl)c(C(N2CCN(C(c3cnc(C)cn3)=O)C(C)C2)=O)c1Cl N1(C(CN(C(C)C)C)=O)CCCN(C(C2CCc3cnnn3C2)=O)C(C)C1 S(=O)(=O)(c1ccc(F)c(F)c1F)NC1CCC(C(N2CCCC(OC)CC2)=O)C1 C1(C(C)NC(N2CCC(C(C)O)CC2)=O)CCCC(NC(=O)OC(C)(C)C)O1 CC1CCCC(C(=O)N(C2CCCN(C(=O)Cc3cnoc3)C2)C)C1.C1CS1 C1(C)(C(=O)NCC(C)OC)CCCN1C(c1ccccc1-c1cn[nH]c1)=O S(=O)(=O)(c1ccc(Cl)cc1C(F)F)NC(c1ccc(Cl)c(F)c1)C c1(CN2CC(C(=O)OCC)(SC)C2)cc(F)c(C)cc1F N1(C(C(C(C)C)c2cncs2)=O)CC2(CCN2C(=O)C(C)O)C1 CC1(C)C=CC(NC(c2cc(CNC(=O)CCN3CCCCC3)cs2)=O)CC1 N1(C(C2(CC#C)CCOC2)=O)CC2CC(C1)N2C(=O)C(O)Cn1cncn1 C(=O)(C1CCCn2cnnc21)NC(CNC(Cn1ncc(C#C)c1)=O)C1CC1 N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2(CCCC2C(=O)NCCNC(C)=O)C1 CCC(CC(F)(F)F)C(=O)NCCC1CN(C(=O)CC2(C3CC3)CC2)CC(C)O1 C1(N(C(=O)CCC2CCCN(C)C2)C)CC2CCC(C1)N2CC1CCOC1 CC1OC(C)(C)OC1(C)C(=O)N(C)CCNC(=O)C=Cc1nnn(C)n1 CCS(=O)(=O)CC(=O)N1CCCCC(NC(=O)CCc2ccnc(C)n2)C1 C1(CNC(CC(CCC)O)=O)CN(C(=O)C=CC=C(Cl)Cl)CC2(CCC2)O1 N#CC1(C(=O)Nc2cccc(OCC3CCOC3)c2)CCOCC1 c1(C(N2CCC(NC(C=C(C)C(C)C)=O)CC2C2CC2)=O)ccn2ccnc2c1 Cn1cc(C(C(=O)N2CC(c3cc[nH]n3)C2)NC(=O)CC2CCCCC2)nn1 N1(C(C(C)NC(CC)=O)=O)CCC(CNC(c2ccc(Br)o2)=O)C1(C)C CCCC(C)(C)CC(=O)NC1CCCC(NC(=O)COCCSC)CC1 N1(C(C(C2CCCO2)NC(CC(=O)NCC)=O)=O)CCC(C)(CC(=O)OC)C1 N1(c2n(CCOCC=C)c(C(C3CCCO3)C)nn2)CCC2(CC1)CC2(F)F c1(C(=O)NCC2(C(=O)O)C(C)CCCC2)cn2c(n1)CCCC2 N1(C(C2(C(=O)OC)CCCNC2=O)=O)CCN(C(=O)CC(C)C)CC(O)C1 C(=O)(CCC(C)S(C)(=O)=O)NC1CCC2CN(C(COC(CC)(C)C)=O)CC21 C1(C(=O)CCSCC(=O)NCc2ccccc2)CC(F)(F)CCN1C1CC1 CC1CCCC(C(N2CCC(C3CCCN3C(=O)CC3CCCC3)C2)=O)CC1 c1(CC)n[nH]cc1CCCC(=O)NC(=O)O c1(C(=O)NCC2C(NC(CC(C(C)C)C)=O)CC2)sccc1S(=O)(=O)C(F)F C=CC1(CNC(C2CCN(C(=O)CC3CC(=O)C3)C2C)=O)CCCCC1 c1(-c2c(SC)cc(F)cc2)ccc2c(O)c(C(=O)NC(CO)CC(C)C)sc2c1 C#Cc1cc(C(=O)NC(CNC(=O)C(CC(C)C)OC)C2CCC2)cc(N)c1 c1(CNC(=O)Nc2c(OC)cc(OC)c(Cl)c2)ccc(S(N)(=O)=O)cc1 c1(CC(=O)NCC(CNC(C2CCCCC2)=O)OC)sc(C)cc1C C1(CN)COC(CNC(=O)NC(Cn2ccc(C)n2)CO)CO1 C1(CC)(NC(=O)COCC2CCCC2)CCCN(C(=O)C=CSC)C1 C1(NC(C2CC(N(C)C)C2)=O)CC2(C1)CN(C(=O)CCn1ccnn1)C2 C#CC1CCN(C(C2CC(NC(=O)C(C)Cn3cccn3)CCO2)=O)C1 C=CCCC(O)CNC(C1(CO)CCN(C(=O)CCCC2CC2)C1)=O c1(CC(C)C(=O)NCC2(NC(C3CCOCC3)=O)CCCC2)ccc(F)cc1 c1(NC(C2CC(N3CCCC3)C2)=O)ccc(NS(=O)(=O)C2CC2)c(C(F)(F)F)c1 N1(C(C(CCC)NC(=O)Cn2ccc(C)n2)=O)CC2(CC(N(C)C)C2)C1 C1(NC(C=CC(C)(C)C)=O)CN(C(c2ccc(C(C)(F)F)cc2)=O)CC1(C)C c1(C(C)=O)ncc(OC)nc1OC.C12CC1(Cl)C(=O)NCC1(CC1)CCNC2=O N1(C(COCC(=O)OC)=O)CCC(CO)C(NC(c2oc(Br)nc2C)=O)C1 CC(CC(C)(C)C)C(F)C(=O)N1CC(CCNC(=O)C=Cc2cocn2)C1 Cc1ccc(Cl)c(N=c2scc(-c3ccoc3)n2CCC(=O)NCC(C)C)c1Cl c1(CNC(C2CCN(C(C3CCC(=O)C3)=O)C2)=O)ccc(O)c(F)c1 c1(C(N2CCC(Oc3ccc(Cl)cc3)CC2)C(=O)NCCF)ccc(CO)cc1 C(=O)(C1=Cc2ccccc2C1)N.C1(OC)CN(C(=O)CCC2CC(OCC(=O)OC)C2)C1 C(CC(CNC(=O)CC(=O)N(C)CC)NC(=O)C=C(C)C(C)(C)C)OC.C(C)(C)(C)O c1(C(=O)NC2C(CNC(=O)COC3CCOCC3)C2)ccc(Br)c(F)c1 C(=O)(CCC(C(C)C)NC(C1CC(C)(C)CO1)=O)NCc1c(CC)c[nH]n1 O=C1NC(=O)C(CCNC(c2cccc(C(=O)NCc3cc(Cl)n[nH]3)n2)=O)N1 N1(C(C(C=C)O)=O)CCC2CN(C(=O)CSc3ccc(C=CC(N)=O)cc3)C2C1 C(=O)(C(F)C(=O)N1CCSCC1C(=O)NC1CN(CC)CC1C)OCC C(=O)(C(CC(=O)N1CCC(C)C(NC(C2COC(C)C2)=O)C1)C(C)=O)OCC CN1CCCC(C(=O)NCCn2cc(CC(=O)NC3CCC(CO)CC3)nn2)C1 N1(C(CCc2c(C)noc2Cl)=O)CCCC2(NC(c3csc(CO)n3)=O)CC2C1 Cc1cc(C(=O)NCc2cc(C(=O)NCCCC(=O)NO)no2)ccc1C#N C12(C(NOCC(N3CCC(C=C)C3)=O)=O)CC(C)(CCO1)C2 N1(C(C(C(C)C)NC(CC(C)C)=O)=O)CCC2CN(C(C3COCCOC3)=O)CC12 c1(OC)ccnc(C(N2CC(NC(C3CCCCO3)=O)CCC2C)=O)c1N CC1=C(C)CC(C)(C(=O)NCC2C=CC(NC(=O)C#CC3CCC3)C2)CC1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2CCN(C(=O)CCc3ncccn3)CC12 C1(NC(=O)CCC2CCCOC2)CN(C(c2ccco2)=O)CC1(F)F N1(C(CC(COC)C)=O)CCC(NC(c2ccc(C)cn2)=O)CC1C C1(NC(CC=CC)=O)CCC(C(=O)NCCN2CCC(O)CC2)CC1 CC(C)(F)CCC(=O)N1CC(CNC(=O)Cn2ccc(O)nc2=O)C(O)C1 C(=O)(C1CCCn2cnnc21)N1CCC2CN(C(c3c(OC)scc3)=O)CC21 C1(C(N2CCCC(NC(Cc3n(C)ncc3)=O)CC2)=O)CS(=O)(=O)CC12CCC2 N1(C(c2ccc(OCCC=C)cc2)=O)CC2(CC(NC(=O)CCOC3CC3)CO2)C1 c1(C(C(=O)NCCCN(C(c2c(CC)onc2)=O)CC)C)ccc(Cl)c(Cl)c1 O=C(CC(C(F)F)NC(C1CCNC(=O)C1)=O)NC12CCN(CC1)CC2 Cc1c(C(=O)NC2CC2CNC(C2CC3(CSC3)C2)=O)cnc2c(Cl)cccc12 CC1(C)C(NC(=O)CCC2(C)CCC(=O)N2)CCN1C(=O)CSc1ccc(F)cc1 c1(C(N2CCN(C(C3C(C)C3C)=O)CC2)=O)nnc(O)cc1O Cc1[nH]nc(C(=O)N(C)CCC2CCN(C(C3CC(F)C3)=O)CC2)c1C Nc1c(C(N2CC(CO)(NC(C3CCc4nccn4C3)=O)C2)=O)nc(O)nc1O N1(C(CSCC(=O)OC(C)(C)C)=O)CC2CC(C1)N(C(=O)CSC1CCCCO1)C2 C(=O)(C(C)C(C)c1ccc(Cl)cc1)NCCC(=C)CNC(C1(C)CCCCC1)=O N1(C(=O)OCC(F)(F)F)CCc2ccncc2C1C.Cc1cccc2c1NC2=O C1(CCNC(c2n[nH]c(C)c2O)=O)CN(c2nc(C3CC3)ns2)CCS1(=O)=O c1(C(=O)NCC(CC)NC(C2CC(=O)N(C)C2)=O)c(Br)c2ccccc2n1C C1(CNC(C(=O)NCCOC)=O)(CO)CCN(C(C2CCNC2=O)=O)C1 c1(C(=O)NC2CN(C(C3ON=C(CC)C3)=O)CC23CC3)c[nH]c2cccc(C)c12 N1(C(c2ccn(C)c2)=O)CCC(C2(NC(C3CCCC4CC34)=O)CC2)CC1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(CNC(c2ccc(C)o2)=O)CC(C)(C)C1 C1(CC(=O)N(C(C#C)C)CC)(NC(=O)CCNC(N)=O)CCC1 N1(C(C(C)(C)OC)=O)CCCC(O)(CCCNC(=O)C(C2CCOCC2)O)C1 CCS(=O)(=O)C=CC(=O)N1CC(CC(C)NC(c2csc3ccccc23)=O)C1 c1(C(C)C(=O)NC2CC(CNC(=O)CC3CCCSC3)C2)ccc2c(c1)OCO2 C(=O)(C(O)Cc1cn(CCO)nn1)NC1CC(OCC)C1 C(CC(C(C)C)NC(C1CCCS1)=O)NC(c1c(OCC)ccs1)=O C1(C(N2CC(CCNC(=O)CN(C)S(N)(=O)=O)(OC)C2)=O)CCN(C)C1=O N1(C(CC2C(C)(C)C2)=O)CCOCC2(COCCN2C(c2snc(Cl)c2Cl)=O)C1 c1(OCC=C)c(NC(=O)CCCCN2CCCC2)cccc1Cl C1(C(=O)NC2CC(O)C2)CCC(O)CN1C(C12CSCC1C2)=O c1(C(=O)OC)scc(-c2ccc(C)cc2)c1NC(=O)Cc1cc(C)no1 c1(C(N(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)=O)cnc(C(F)(F)F)cn1 c1(C(=O)OC)cnccc1CN1CC(OC)CC1C(=O)Nc1cccnc1C c1(C(C)C(=O)NCCN(C(c2c[nH]c(=N)o2)=O)C2CC2)ccc([N+](=O)[O-])cc1F Cc1nc(O)ccc1C(N1CCC(O)(C(C)NC(=O)CN(C)C(N)=O)C1)=O Nc1cc(C(N2CCC3(NC(c4cncc(F)c4)=O)CC3C2)=O)ncc1F c1(CNC2C(CC3(NC(C(C4CCCC4)SC)=O)CC3)C2)ccc(O)c(C)c1C C(CCCC(=O)NCC1CN(C(=O)C(=O)NCC(F)(F)F)C2CC12)SC N1(C(CCCN(C(C)C)C)=O)CCCC2(C1)CN(C(=O)CCS(C)=O)CCO2 c12nc(no1)CCC(=O)NC2.C1(C(=O)NC(CSCC)C)CC1(F)C(=O)OCC C1(O)(CNC(CCc2cn(C)nn2)=O)CCCN(C(C2(C)CC(F)C2)=O)CC1 N1(C(c2n(C=C)nnc2)=O)CCC2(C=C(C(=O)N3CC(=O)NCC3C(C)C)C2)C1 N1(C(C(CC)(C)O)=O)CC2CCC1C1CN(C(c3cccc(N)c3F)=O)CC21 c1(C(N2C(CCOC)CN(C(C3CCCOC3)=O)CC2)=O)nc2cnccc2s1 C1(C)(C(=O)NC23CN(C(C(C)C4CC4)=O)C(C2)C3)Oc2ccccc2NC1=O c1(OC)ccc(F)cc1CCC(=O)N(CCC(C)C)CCC(=O)O C12(NC(CNC(CCC)=O)=O)CCC(CNC(c3cnsc3)=O)(C1)OC2 c1(OC)c(F)ccc(F)c1C(N1C2CN(c3nccc(Br)n3)CC12)=O c1(-n2cc(C(N(CC(C)NC(CCC)=O)C)=O)nn2)ccccc1C C(C(C(C)C(C)C)NC(=O)CCc1nc[nH]n1)NC(C(c1ccc(CC)s1)=O)=O Cc1[nH]nc2ncc(NC(=O)C(C)(O)CCc3ccccc3)cc12 c1(C(N2CCCC(NC(C(C)(C)c3nccs3)=O)C2)=O)ccc(N)c(N)c1 CN1CC=C(CC(=O)NC2CCN(C(c3c(F)cc(O)cc3F)=O)CC2)CC1 c1(-c2ccc(C#N)cc2)cccc2ccc(C(=O)NCc3ncccc3Cl)nc12 C1(C(N2C(CNC(c3ncc[nH]c3=O)=O)CC(F)C2)=O)CCn2cncc2C1 C1(c2ccc(OC)cc2)NC(=O)N(C2CCCCC2C)C1=O C1(C(=O)OC(c2ccccc2)CC=C)CN(C(C)=O)CCO1 C1(NC(c2c(C)n(CCC#N)nc2)=O)CCN(C(C2OC(C)CC2C)=O)CC1C CC1CCC(NC(c2cc(O)nc(Cl)c2)=O)CN1C(=O)CC1C(C)(C)C1(C)C C1(NC(C=CCCC)=O)(COC2CCCC2)CCN(C(=O)C(C)(O)COC)C1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CC(NC(c2csc([N+](=O)[O-])c2)=O)C(O)C1 N1(C(C(CCC)C)=O)CC2CCC1CN2C(c1nc(-c2ccc(Cl)cc2)no1)C C1(C(N(CCCN(C)C(c2ccc(CSC(F)F)o2)=O)C)=O)CCCCS1 C#C[Si](C)(C)COCC(=O)NCC1CC12CCOC2 N1(C(=O)NCC2CC(F)C2)CCOC(Cn2cncn2)C1 C1(C(=O)NC(CC)CN(C)C(c2csc(C(C)(C)C)n2)=O)CN2CCN1CC2 C1(C(=O)NC2(C)CC(C(=O)NC(c3cncnc3)C)C2)CN(C)CCN1C CC1CC(CNC(=O)CCc2cc[nH]n2)CN1C(c1csc(S)n1)=O c1(OCC(=O)NCCC2CN(C(CC(C)(F)F)=O)C2)ccc(F)cc1Br C1(CC(C)NC(C2(CF)CC2)=O)CC2CCC(C1)N2C(c1cc(F)cnc1O)=O c1(OC)ccccc1C(=O)C(=O)NCCN(C(c1cnn(CCF)c1)=O)C(C)C N1(C(C(C)NC(c2ccccc2)=O)=O)CC2CCC1C2NC(C1CS(=O)(=O)C1)=O CC(CS(=O)Cc1nnn[nH]1)c1ccccc1.c1(C)ccccc1 N(C(=NCC(=O)N1CCCC1)N1CCC(n2cc(Cl)cn2)C1)Cc1n(C)ncc1 C1(NC(C(CC)OCC)=O)CC2CC(C1)N(C(=O)C(C#N)=CC(C)C)C2 N1(CC)CC2CCC1C(NC(=O)CC1CCCN1C(=O)CC1CC1(C)C)C2 CCCCC(C)C(=O)N1CC2C(N(C)C(C3CC4CCC(C3)S4)=O)C2C1 c1(C(N(C2CCCCN(C(=O)C(O)c3ccsc3)C2)C)=O)ncnc(O)c1Cl C1(O)(CCNC(=O)OC(C)(C)C)CCN(C(C2COC3CC2C3)=O)CC1 C(CCCCNC(=O)C(n1ccc(C(F)(F)F)n1)C)NC(C(C)OCC=C)=O O1NC(=O)CC(C)CN(C)C1.C(c1cnn(C)c1)=CC(N1C(CC=C)CCC1)=O c1(C(=O)NCC(CC)(C)NC(=O)C=C2CCN(C)CC2)csc([N+](=O)[O-])c1 c1(C(=O)NC(CCN(C(C(C(C)C)N(C)C)=O)C)C)cccc2nncn12 c1(C(=O)NCC2CC(NC(C(C)c3ccsn3)=O)C2)ccccc1-n1cccn1 C(C(CC(F)(F)F)NC(c1cc(F)cnc1O)=O)NC(=O)COCC1CCOC1 c1(C(N2C(CCNC(C3(C(F)F)CC3)=O)CC(OC)C2)=O)cc2oc(C)cc2[nH]1 N1(CC(COC)O)CCC(NC(=O)C(C)(C)c2cccs2)CC(C)(C)C1.C1=CC1 N1(C(C2N(CC)CCCC2)=O)CC(N(C)C(c2nnccc2C)=O)C2(CC2)C1 CS(=O)(=O)c1ccc(F)c(-c2noc(CCC(N3CCC(C4CCC4)C3)=O)n2)c1 S(=O)(=O)(c1ccc(N)c(F)c1)NCC.C(C(=O)N=c1cc[nH]cc1)C1(C)CC1(F)Cl c1(C(N2C(CNC(COC)=O)CC(O)C2)=O)ccc(N2CCCC2)c([N+](=O)[O-])c1 c1(OC)ccc(C(=O)NCCN(C(=O)C(O)P(C)(C)=O)CC(C)O)c(Cl)n1 O=C1CCC(CC(=O)NCC2CN(C(c3cscc3Cl)=O)CCO2)C(=O)N1 C1(C(=O)NCc2occ(C)c2)CCC=CC1NC(c1ccon1)=O C1(N(C(Cc2nc(COC)sc2)=O)C)CCN(C(=O)C#CC2CCC2)CC1C C1(NC(C)=O)OCCC1C.C1(N2C3CC(C3)C(F)C2=O)CCOC1C C1(C(N2CC(NC(c3c(C)sc(O)n3)=O)C(C)C2)=O)Cc2ccccc2C(=O)O1 C(=O)(CN=c1cc[nH]cc1)NC1C(C(=O)NC(C2(C)CC2)CO)CC1 c1(NCC(CCCCC)O)ccc(S(=O)(=O)NC2(c3ccc(F)cn3)CC2)cn1 C=CCC(C(=O)N1CC(C(N)=O)(CNC(c2cc(C3CCC3)no2)=O)C1)OC c1(SCCCNC(=O)CN(C(=O)COCC2CCOC2)CC)ccc(OC)cc1 CC(C)C(C)(CNC(=O)C(C)N(C(=O)CCC1CCOCC1)C)C(C)C C(=O)(C1=CC(O)CCC1)NC1(CC(N2CCC(C)CC2)=O)CCCCC1.C1(CC)CC1 c1(C(N2CC3CN(C(CSCC)=O)CC32)=O)c(F)ccc(Br)c1F c1(C(=O)NCC2C(C)CCN2C(=O)CO)ccc2c(n1)CCC2 C1(C(=O)NCc2nncs2)CCC(O)CN1C(c1cc(Cl)c[nH]1)=O N1(CC=C)CCN(C(=O)CCN(C(=O)C(C)C(=O)OCC)C2CC2)CC1 C1(CCC(=O)NCC2CCCN(C(C3C(C#N)C3)=O)C2)CCc2ccccc2C1 c1(CC(=O)NCC2(F)CCN(C(C3(CC)COC3)=O)C2)c(O)ncnc1O c1(CNC(CCOC(=O)COCC2CC2)=O)ccc2c(c1)OCCCO2 C(=O)(C(N=[N+]=[N-])C(C)C)NCC(C(=O)N(CC(C)OC)C)C N1(C(C(C(=O)OCC)F)=O)CCC2CCN(C(=O)C(C)O)CC12 C1(NC(CC(CC)OC)=O)(COC)CCCN(C(c2oc(C3CC3)nc2C)=O)C1 C1(C)(C(=O)NC2CC(CNC(c3c(SC)cccn3)=O)C2)CCN(C)CC1 c1(OCC#C)ccc(NC(=O)NC2CCCC(CC)CC2)cc1C C1(C#N)(C(N2C(COC)(CNC(C3CCN3CC)=O)CCC2)=O)CC2CC2C1 N1(CCCNC(C2C(C(C)C)OCC2)=O)CCN(C(c2cccnc2)=O)CC1 CC(C)(C)CC1CC1C(N1CCC1CC(=O)NCCF)=O c1(C(N2C(CCOC)CN(C(=O)C(C)CSC)CC2)=O)cc2ccccc2nn1 N1(C(C2C(CNC(CN3CCC(C)C3)=O)OCC2)=O)CCC(CN=[N+]=[N-])CC1 c1(OCC)ccc(Cl)nc1C(=O)NCC1CC(NC(=O)C(C)(O)C2CC2)CCO1 N1(C(C=CCOC)=O)CC(C2CCN(C(c3cccc(C(C)(C)C)c3)=O)C2)C1 C1(NC(Cn2c(C)nnn2)=O)CC2(C1)CC(C(=O)NC1(CCF)CCC1)C2 N1(C2CN(C(CC3CCC(C)(C)C3)=O)C2)CCN(C(=O)C(N)=O)CC1=O CC1(NC(c2cccc(COC(F)(F)F)c2)=O)CCN(C(C2CC(C)(F)C2)=O)C1 c1(C(N(CC(C)NC(COCC(=O)NC)=O)C)=O)ccc2oc(S)nc2c1 C(=O)(CC(C)C(C)C)NCCc1c(CNC(c2oc(CC)c(C)c2)=O)nco1 C=C(Cl)CC(C(=O)N(CC(C)(CC)OC)C)NC(C1CCCN1C)=O Cn1nc(C(=O)NC2CCC2NC(C2(C3CCCO3)CCC2)=O)ccc1=O Cc1ccc(N(C)C(C)C)c(C(=O)NC2CC(CNC(C3CC3(F)F)=O)CC2O)c1 CC1CN(C(=O)CC(C)n2cccc2)CCCN1C(=O)Cc1cnsc1 N1(CC)CCCC(C(N2CC3CC3(C(=O)NC3(C)CC(F)(F)C3)C2)=O)C1 C(=O)(C(CCC(=O)N(C)C)N1CC(C)OC(C)C1)Nc1c(C)cccc1 C(c1ccncc1)=CC(=O)N(C1CCCC(NC(=O)CCc2cn[nH]c2)C1)CC Cc1ccc2nc(N3CCCC(C4(NC(=O)CSS(C)(=O)=O)CC4)C3)sc2n1 C1(OC)CN(C)CC1C(N1CCC(CC(=O)NC2(C)CCOC2)C1)=O CC1(C(=O)NCC2CC3(CC3)CN2C(=O)C=Cc2cn[nH]c2)CCC(F)(F)C1 C1(NC(c2ccn(CC)n2)=O)CCC12CN(C(=O)Cc1ccc(CSC)cc1)C2 C1(C(N2C(C(C)NC(=O)COCC(F)(F)F)CCC2)=O)CC(=O)NC1(C)C c1(C(N2CC(C(C)(C)O)(CNC(c3cnc(C)[nH]3)=O)C2)=O)c([N+](=O)[O-])cnn1C Cc1cc(C(=O)N(CC(O)CN(C)C(c2cnc(C(C)O)s2)=O)C)ccc1N C(=O)(C1CSc2ccccc21)NC1C(NC(C=C(COC)C)=O)COC1 N1(CC)CCN(CC(N2CCC(N3CCCC3=O)C2)=O)C(=O)C1=O N1(C(C(C(CC)C)N(C)C)=O)CCC(C2CC2)(C(=O)NCc2ccncc2F)C1 c1(C(=O)NCc2ocnc2C(N2CCC(N3CCC3)C2)=O)cc(Cl)cnc1O c1(CNC2CC(NC(c3ncn(-c4ccccc4)n3)=O)C2)ccc(I)c(F)c1F c1(C(N(CC(C2CC2)OC)C)=O)ccc(CNC(=O)C(C)n2ccnn2)cc1 C1(C(N(C2CCN(C(=O)C3=C(C)CCOC3)CC2)CC)=O)CC12CCC(=O)CC2 c1(C(=O)Nc2c(OCC)cc(C#N)cc2)cncc2cnccc12 N1(C(CCCCCOCC)=O)CCN(C(=O)Cc2ccc(F)cc2)CC(CO)C1 C1(CNC(CCN(C(CC)CC)C)=O)COC(C)(C)CN1C(C1CC2CC2C1)=O c1(C(C(=O)NCCC(C)NC(C2COCC2C(F)(F)F)=O)O)ccccc1Cl CCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C(C)Oc2cccnc2)C1 c1(C(N2C(C)CN(C(C(C)=CC)=O)C(C)C2)=O)cc(O)nc2ccccc12 C1(CN(C(C2CC(CN(C)C)C2)=O)C)C2CN(C(c3cc(Cl)cn3C)=O)CC12 N1(C(CCOC)=O)CCCC(N(CCO)C(c2sccc2CN(C)C)=O)C1 N1(C(CCCNC(c2ccccc2C(F)(F)F)C)=O)CCC(C)(O)C1 Cc1cccc2[nH]c(C(=O)NC3CN(Cc4c[nH]c5ncccc45)CC3C)cc12 CC(C)(C)C(CNC(C1OCCCC1(C)C)=O)C(=O)NCc1ncc(Cl)cn1 n1(CC(C)NC(c2cnn(C3CC3)c2)=O)cc(CNC(C2CC(F)(F)C2)=O)nn1 C(c1ccc(SC)s1)=CC(=O)N(CC(C)NC(=O)CCn1cnnn1)CC C(=O)(CCC(N)=O)N(CC(=O)N(CCO)CCO)C(C)C Cc1cc([N+](=O)[O-])c(NC(=O)C(=O)NCC2(c3ccccc3)COC2)cc1Br N(C1CCCc2c1cnn2C)CNC(CCN1CCCC(N(C)C)C1)=O C1(C(=O)NC(CCOC)C(=O)N(C)Cc2cncs2)CC2OC1C1CC21 N1(C(C2N(C(C(CCC)=CCC)=O)C3C(O)CC2C3)=O)CCc2ccc(C)cc21 c1(C(=O)NC2C(c3ccccc3)(C)C2)ccc2c(c1)CCN(C(=O)C#CC(=O)O)C2 CCC(CCC(=O)NCc1cc(C)ncn1)NC(=O)C(C)NC(=O)NC N1(C(C2N(C(COCCC(C)C)=O)C(C)C2)=O)CCCC(O)(C2CC2)C1 c1(C(N2CCC(O)(C(C)NC(=O)C(F)=C(C)C)C2)=O)ccc(N)c(O)c1 C1(=O)C(C(C)C)C(C)N1.C(=O)(C(O)CN(C)C)NC1(C(=O)NCC#C)CC1 C(c1ccc2ncccc2c1)=CC(=O)NC1CCCC1NC(=O)CC1CCOC1 c1(C(=O)NC(CC)CNC(=O)CCCc2ccsc2)cccc(S(C)(=O)=O)c1 C=C(C)CC(C(=O)NC1CCC(Cn2cc(C(C)(C)F)nn2)CC1)NC(C)=O N1(C(C2N(C(C)=O)CSC2)=O)CCC(F)(C(=O)NCc2ccc(Br)s2)C1 c1(C(=O)NCC2CCCN(C(C(C)S)=O)C2)cc(F)ccc1F C1(NC(CC2CC(NC(C3CCN(C(C)C)C3)=O)C2)=O)C=CCCC1CO C(=O)(CC(C)n1cc(Br)cn1)NCC(CC)NC(=O)CCCC1CC1 c1(C(N2CC(CC(=O)O)Oc3c(Cl)cccc32)C)ccc(S(=O)(=O)C(F)(F)F)cc1 c1(C(=O)NC2COCC2NC(C2(C3CCCO3)CCC2)=O)cc2cccnc2[nH]1 c1(CC)ccc(C=CC(=O)NC(C)CN(C)C(c2ccnn2CC)=O)o1 n1(CC)nc(C)cc1C(=O)NCC1CCC1NC(=O)Cn1ncnn1 c1(C(N2CC(C)(C)C(NC(=O)C(Cl)=CCl)C2)=O)ccc2nn[nH]c2n1 CCC(CNC(=O)COC)(CC)C(=O)NC(c1cc(C)on1)C C#CCCN=C(NCc1ccc(C2CC2)cn1)NC(C)CCS(C)(=O)=O N1(c2n(CCCOCC)c(C3C4CC5C(C4)C35)nn2)CC2CS(=O)(=O)CC2(C)C1 CC1CN(S(=O)(=O)CCNC(=O)N(C)CCc2ccccc2)CC(C)O1 O=C(CS(=O)(=O)C1CC1)N1CCN(C(C2C=CCS2)=O)CC1 CC1CCN(c2nnc(-c3cnco3)n2CCC(=O)N(C)C)CC1C c1(C(=O)NC(C(C)C)C2CC2)ccc(CNC(=O)C(O)CN(C)C)cn1 C1(CNC(c2occ(C)c2)=O)CCN(C(=O)C(O)CC(C)C)C12CC2 N1(C(C=C(C)c2ccccc2)=O)CC2CC(C)N(C(C3CC3F)=O)C2C1 Cc1ccc2c(N(CC(Cl)Cl)C)nc(=NC3CCCC(C)C3)[nH]c2c1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CC2(NC(C3CC(C)(C)CO3)=O)COC1C2 S(=O)(=O)(c1ccccc1C#N)N1CC2CCN(C(C#CC)=O)C2CC1 c1(CC)cc(C(N2CCCC(N(C(=O)C=CSC)CCO)C2)=O)ccc1F N1(C(C(CC)(C)OC)=O)CC2CC(C1)C2NC(=O)C(CC(C)C)c1cccc(Br)c1 C(=O)(CC(C)(C)OC)NC(CC)CNC(C1(n2cc(Cl)cn2)CC1)=O C1(C(=O)NC(CNC(C(CC#C)O)=O)CO)CCCC2(CC2)C1 c1(C(=O)NCC(CNC(c2cc(COC)[nH]n2)=O)C)c(C)ccc(F)c1O c1(C(N2CCCCC(CNC(c3ccsn3)=O)C2)=O)cc2cccnc2o1 C1(NC(C(=O)NC2CCOCC2)=O)CCC2(CC1)CCN(C(c1cccs1)=O)CC2 O=C(CNCc1nc2ccccc2o1)NN=c1[nH]c(Cl)c(Cl)nc1Cl C12(NC(CCC(C)OC)=O)CCC(C1)N(C(=O)CNC(C1CCCC1)=O)C2 CC1CN(C(=O)CCSc2nnnn2C)CCN1C(=O)C(O)C(F)F N1(C(C23CC(C(=O)NC4CC(N=[N+]=[N-])C4)(C2)C3)=O)CCC(C2CCOC2)C1 c1(SCC2(C(=O)NC(C3(CSC)CC3)=O)CC2)ccc(F)cc1.C(CN1CC1)OC C12(NC(CCCOC)=O)CCC(F)(F)CC1CN(C(=O)C(C(C)(C)C)OC)C2 N1(C(C(n2ccc(C)n2)C)=O)CCC(C(N2CCC(C#N)C2)=O)C1C(C)C N1(CCNC(C(CSCC)NC(=O)CC(C)C2CC2)=O)CCCCC1=O N1(C(C(N)=O)=O)CCC(C(F)(F)F)C(CNC(c2cc(-c3ccoc3)on2)=O)C1 c1(C(=O)Nc2c(O)ccc(C)c2)n[nH]c2c1CN(Cc1ccccc1C(=O)O)C2 N1(C(c2c(CC)onc2)=O)CCC(N(CC(C)C)C(c2cc(C)c[nH]2)=O)CC1 C1(NCCCn2c(C(c3cncn3C(C)C)SC)nnn2)CCCN(O)C1=O c1(CSC)ccc(C(=O)N(C)CC2CCCC2NC(C23CC(F)(C2)C3)=O)o1 CC(C)(C)C(C#N)C(=O)NCCC(O)CNC(=O)Cn1cc([N+](=O)[O-])cn1 c1(C(N2CC=CC(NC(C(CCOC)C)=O)C2)=O)cc(C2CC2)cnc1Cl O=C1CCCC(C(N2CC=CC2C(=O)NC2CC2C(F)(F)F)=O)C1 C1(NC(C2CCS(=O)CC2)=O)CC(F)CN(C(=O)C=CC2CCC2)C1 C12(C(=O)Nc3cccc(C(N(CC(C)(C)C)C)=O)c3)CCC(CC1F)C2 N1(C(c2cscc2Br)=O)CCC(CNC(C2(F)CC=CC2)=O)CC1 N#Cc1ccc(CSCC(=O)NCCNC(=O)CNC(C2CCOCC2)=O)cc1 CCS(=O)(=O)CC(=O)NC1COCC1NC(C1CC2CCC2C1)=O c1(CC)oc2ccccc2c1C(=O)NCCOCC(c1ccc[nH]1)C.C(C(=O)N)O N1(C(C=CCCC(C)C)=O)CCC(C)C(N(C(=O)Cc2ccon2)C)C1 C1(NC(c2c(C)con2)c2nnnn2CSc2ccccc2)CC(C)OC(C)C1 N1(CCC(=O)NC2CC(CCC(=O)NC3CC(F)(CF)C3)C2)CCCCC1 N1(OC(C(C)=O)C)CCN(CC(c2ccccc2OC(F)(F)F)O)CC1.OC(F)(F)F c1(NC(CCC=C)(c2nnnn2CCC2(C)CC2)C2CC2)cnc2ncccn12 N1(C(C(F)(F)C2(OC)CCC2)=O)CC(NC(=O)C(C)c2ccco2)CC(F)C1 c1(OC(=O)NC(C)CN(C)CCc2ccccc2)ccc(Cl)c([N+](=O)[O-])c1 CC1=C(C)CC(C(N2CC(O)CC2C(N2CC3CC3C3CC23)=O)=O)CC1 Cc1ccccc1COCC(=O)NC(C1CCCN1C(c1cccnn1)=O)C C(=O)(CCCCCC#N)N1CC(CC(C)NC(C2(C)N(C)CC(OC)C2)=O)C1 CCC(CC(=O)NC1CN(C(c2ccsc2)=O)C2(CCOCC2)C1)CC(F)(F)F Cc1ncc(C(=O)NCC(C)(C)CNC(C2CC(CF)C2)=O)cn1 c1(C(N2CCN(CC3OCCC3F)CC2)=O)ccc([N+](=O)[O-])cc1 C1(NC(=O)C=Cc2cncnc2O)CN(C(=O)C(F)=C(C)C)C2(CCCOC2)C1 C1(NC(COC(C)=O)=O)CCCC1C(=O)NCC1(N2CCOCC2)CC1 c1(CC(=O)NCCC2CCN(C(=O)CC=C(Cl)Cl)CC2)ccc(F)cc1Cl C1(CC)(NC(=O)C(C)O)CN(C(=O)C(C)(F)c2ccccc2)C1 c1(OC)ccc2[nH]nc(C(N3CCC(C)C(NC(=O)C4=COCCO4)C3)=O)c2n1 N1(C(CNC(=O)OC)=O)CCC(NC(=O)CC(C)C(F)F)C(CO)C1 C1(CNC(c2n(C)nnn2)(C)Cc2nnnn2C(C)(C)C)CCCC(C)(C)O1 c1(C(CCN(C(=O)C(=O)NCC(CO)n2cccn2)CC)N(C)C)ccccc1 C(=O)(C1=NN(C)C(=O)CC1)NC(CC)(CNC(C1CC2CCCC2C1)=O)CC c1(C(=O)NC(c2c(C)c(F)ccc2)C)cc([N+](=O)[O-])c2n[nH]cc2c1 c1(CCC)ccccc1C(=O)NC1CCN(C(c2cc(CC)oc2C)=O)C1C C(CCC(C)(C)C(=O)Nc1ccc(NC(=O)CCc2n[nH]c(=N)s2)cc1C)OC N1(CC(=O)NC(C2CCCN(CC(=O)Nc3nncs3)C2)C)C(=O)CNC1=O C(=O)(C1CCCc2ccnn21)NC1(CF)CCN(C(C(C)C2CCCC2)=O)C1 C1(CN(C(=O)Cc2cocn2)C)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 CCCC(C)(CC)C(=O)N1CC(CC(C)NC(=O)C(C(C)CC)OC)C1 C#CC(C)(C)C(=O)N1CC(C(C(=O)NCc2ccc(CC)cc2)OC)C1 c1(NC(C(CC2CCC2)NC(C2CC3(CCC3)C2)=O)=O)ccc(CCF)cc1 c1(C(=O)NC2C(OC)CN(C(C3(F)CCOCC3)=O)C2)cnc([N+](=O)[O-])cc1C C1(NC(=O)CCc2nc[nH]n2)CC2(C1)CC(NC(c1csc(C(F)(F)F)n1)=O)C2 CC(C)CC(CNC(c1cc(=N)[nH][nH]1)=O)C(=O)N1CCCC1(C)C(C)(C)C C(c1cc(Cl)c2c(c1)OCCO2)=CC(=O)OCCCOCCN=[N+]=[N-] c1(C(C(N2CCCC(CN(C(CC)=O)C)C2)=O)C)ccc(OC)c(OC)c1 c1(OC)cccc(C(CN2CCC(NC(C)=O)CC2)NC2CC3CCC2O3)c1 N1(C(C2(C(=O)NC)CC2)=O)CCC2(NC(C34CC3COC4(C)C)=O)CCCC12 N1(C(C(C)N(CC=C)CC=C)=O)CCN(C(c2cccnc2)=O)CC1 Cc1cc(C(=O)Nc2cccc(-c3ncnn3C)c2)c([N+](=O)[O-])c(O)n1 N1(C(C2N=C(C)SC2)=O)CC(F)(F)CC1(C)CNC(c1cn(CCO)nn1)=O C(=O)(CCC(C)(C)O)N(C1CCN(C(=O)C(CC=C)c2ccccc2)C1)CCOC N1(C(c2c(OC)csc2)=O)CC(NC(=O)CCCCCc2cccs2)CC(O)C1 C1(CNC(C2(CNC(Cc3c(C)nsc3)=O)CCCCC2)=O)COCC(C)(C)O1 CCCCC(CC)C(=O)N(CC(O)CNC(c1cc(-c2csc(=N)[nH]2)c[nH]1)=O)C C1(NC(Cc2ccn(C)n2)=O)CCSC12CN(C(=O)CC1CCC(C)(C)C1)C2 C(=O)(C(F)(F)CC1CC1)N1CCC(NC(c2nc(CC(C)C)sc2)=O)C1 CC(c1ccccc1C)=CC(N1CC(CO)(NC(c2cccnn2)=O)C1)=O N1(CC(C)NC(=O)C(O)Cc2ccccn2)CCN(C(C2(O)CCC2)=O)CC1 Cc1cncc(NC(c2nnnn2CC2CC2)CC2CCCCO2)c1 C1(NC(c2n(C(C)C)ncc2)=O)CCC(N(C(=O)CC2CCN(C)C2)C)CC1 c1(C(C(=O)OCCO)C2CCCC2)ccccc1F.c1(C(C)OC)nocc1C=O N1(C(C2(OCC)CCOC2)=O)CC(CC(=O)Nc2cncc(C#N)c2)C2(CC2)C1 C=CCCC(C(=O)N(C)CCSC)NC(c1cocn1)=O C1(C(=O)Nc2c(O)cccc2Br)COC2(CCN(Cc3cnc(Cl)nc3)CC2)C1 CC1CN(C(=O)C(=O)N(C2CC2)C)CC(NC(C2CN(C(N)=O)C2)=O)O1 C1(NC(C(C)(C)CF)=O)CCC2(CC1)CN(C(c1n[nH]c3c1CCC3)=O)C2 c1(C(C)NC(c2n(CCCSC)nnn2)c2ccc(C(F)F)s2)cn(C)nc1C C(C(=O)NC1CCCC1CC(N1CCC2CCC12)=O)(C(C)C)OC c1(OC)nccc(C(=O)NC2CN(C(=O)C(C)OCC3CCCO3)C2)c1F N1(C(C=CCCC)=O)CC2OCC(NC(=O)C=Cc3ncc(C)[nH]3)C2C1 N1(C(C(CCCC)O)=O)CCC(C)(C)C(N)C1.C(CC(O)CO)N(C=O)C CCC(C)(CNC(c1ccc(O)cc1)=O)C(=O)NC1CCC(O)CC1 C1(c2ccccc2)(CNC(C=C(CC)CC)=O)CC(NC(=O)C(C)O)C1 c1(C(N(C2CCC(NC(COCCC#C)=O)C2)C)=O)ccc(P(C)(C)=O)cn1 n1(CC(=O)NCC2C(NC(C(CC)(C)OC)=O)C2)ccc2cc(F)ccc12 Cc1nc(C(C)(C)C)sc1C(N1CC=CC(NC(=O)Cn2cc(C#N)cn2)C1)=O c1(C(=O)NCC2(CCNC(CN(CCOC)C)=O)CC2)nccc2c1NCCC2 C1(NC(CC2OCC(C)(C)C2)=O)CC2CC(C1)N(c1nccc(C(C)(C)C)n1)C2 N1(C(c2ccc(C#N)o2)=O)CCC2(NC(C3CCS(=O)(=O)CC3)=O)CC2C1 Cc1nc2cc(Cl)cc(C(=O)NC3CN(C(c4ccoc4)=O)CC3C(F)F)c2[nH]1 c1(C(=O)NC(CC(C)NC(C2CC=C(C)CC2)=O)C)cc(O)nc2ncccc12 Cc1noc(C)c1CNC(=O)CCCCNC(=O)C(C)NC(=O)C1CC1 C1(CN=c2cc(C)nc[nH]2)CCC2(CCOCC2)CO1.c12ccc(N)cc1CN2C c1(C(=O)NCCCCC2(C(=O)OC)CCC2)c(OC)ccnc1O C(CN=C(NC(c1ccccc1)C)N1CCN(c2c(F)cccc2F)CC1)OC Cc1ccc(C2(SCCn3ccnn3)CC2)cc1.N12CC(C1)NCC1CC1C2=O C1(CC(=O)NCCOCCC(=O)NC(C)Cc2nc[nH]n2)CC=CCC1 C(C(C)C(=O)NCC1CC(c2ccccc2)C1)OC.C12(CCCC1)C(=O)NC2 Cc1cc[nH]c(=N)c1C(=O)NC1CC(NC(=O)COc2cccnc2)C1 CCC(C)(O)C(=O)NCC12CC1CN(C(c1ccc(OCOC)cc1)=O)C2 c1(CNC(C2(C#C)CN(C(=O)CCC3CCOC3)C2)=O)cnc(F)c(C)c1 N1(C(C(C)=CC)=O)CCCC2(CNC(c3cc(OC)cnn3)=O)CCCC12 Cc1c(Br)cnn1CC(=O)N(C(C)CCNC(c1ccc(N)cn1)=O)C c1(C(N2CCC(Cc3cn(CCc4scc(C)n4)nn3)C2)=O)ccc(Cl)cc1F c1(CC)[nH]nc(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)SC)c1[N+](=O)[O-] n1(CC)nc(C(N2CCC(NC(c3ncccc3OC)=O)CC2)=O)cc1C1CC1 c1(C(=O)NC2CCC(NC(C3CN(C)C3)=O)CC2)cc(S(N)(=O)=O)co1 C(=O)(C(C)(C)C(C)(C)C)NC1C2CN(C(C3CCCN(S(C)(=O)=O)C3)=O)C1C2 c1(C(N2CCC(C(CNC(C(CC)F)=O)C)CC2)=O)nnc2ccccc2c1N Cc1coc2ccc(C(=O)NCCOCC(=O)NCC3CCC(C)CO3)cc12 N1(C(C(CC)CN(C)C)=O)CCCC(N(C(=O)C=CC2CCOCC2)C)CC1 N1(C(C2(COC)CC2)=O)CCCCC(NC(=O)CC(C(F)F)c2ccccc2)C1 CCCS(=O)(=O)CC(=O)OCC(=O)Nc1ccc(Br)cc1F C1(C(C(C)N(C(C2CCC(C)C2)=O)C2CC2)=O)CC2C=CC1C2 c1(NC(C2(OC)CCN(C(=O)CC34CCCC3C4)C2)=O)cc(C)ccc1C C1(C)(CNC(CCC=CCC=C)=O)CCC(NC(C2COCCO2)=O)CC1 C1(NC(CC2(OC)CCCCC2)=O)CCN(C(=O)Cn2nnnc2C)CC1F N1(C(C(=O)OCC(=C)C)C(C)C2CCCC2)CC2CC1CCC2NC(=O)OC C1(C(F)F)(C(F)F)CCCN(c2cc(Cl)c(Br)cn2)C1 C1(C(=O)NCC(CC)NC(C2(N3CCCC3)CC2)=O)CCC2(CCC2)OC1 C(=O)(C(CC(N)=O)NC(C1(c2ccccc2)CC1)=O)N1CCC(=C)C1 N1(C(C(C)C2CCC2)=O)CCC(NC(C2(S(C)(=O)=O)CC2)=O)C(CO)CC1 CC(C(=O)N1CCCC1CCC(F)(F)F)C(C)(C)C Cc1ncc(Br)cc1NC(C1CC1C(=O)Nc1cnc(C#N)cn1)=O N1(C(C=CC(C)C)=O)C2CCC1CC(NC(=O)C(c1ccc(F)c(F)c1)O)C2 C(C(C(=O)N1CC(O)(C(N)=O)C1)C(C)C)NC(CC(CC)OC)=O c1(C(=O)NC(C(C)NC(C2CCC(N(C)C)C2)=O)C)ccnc2[nH]cnc12 c1(C(=O)NC(CC)CN(C(=O)COC2CC2(F)F)CC)cc2c(s1)CCOC2 C1(O)(CNC(C2CCCC2)=O)CCCN(C(=O)CCCn2ccnc2)C1 N1(C(c2c(C)c(I)nn2C)C(=O)NCCSC)CCC(O)CC1(C)C C1(CNC(C(C)n2cccn2)=O)CN(C(=O)CC(C)(C)CN(C)C)CC1(C)C CC1=C(C(=O)NCCCN(CCO)C(c2coc(C(C)(C)C)n2)=O)SCCO1 CC(C)(C)S(=O)(=O)CC(=O)NCC1CCC(NC(C2CC(F)C(=O)N2)=O)CC1 c1(C(N2CCC(C(C(=O)NCc3nc(C)oc3)C)C2)=O)oc(C)nc1CO N1(C(C(CC)=CC)=O)CCC2CN(C(=O)Cc3ccc(OC(C)C)cc3)CC2C1 C1(C(N(CCC#C)CCO)=O)CCN(C(C2CC=CCC2C)=O)C1CC CC1OCCC1(O)CNC(C1(CNC(=O)Cc2cn[nH]c2)CCCC1)=O c1(C(=O)NC2C=CC(C(=O)NCC3(F)CC(O)C3)C2)cnc(Cl)s1 N1(C(C(CC=CC)CC)=O)CC2CC(NC(c3n[nH]c(=N)s3)=O)C(C2)C1 c1(N2CCN(C=O)CC2)cc(C(F)(F)F)ncc1[N+](=O)[O-].CC1CCC(N)(N)C1 c1(CNC(C(Cc2cn[nH]c2)NC(C(c2ccc(=N)[nH]c2)C)=O)=O)ncc(Cl)cn1 CCC(C)CC(C(=O)N1CC2C(C(=O)OC)C2C1)NC(c1cc(C)[nH]n1)=O c1(C(=O)NC(CN(C)C(c2cc(C3CC3)[nH]n2)=O)(C)C)ccc(N)c(F)n1 c1(OC)cc(OC)c(C(C(=O)NC(C)(C)C)N(C)CCc2ccc(Cl)s2)cc1Br c1(C(N2CCCCC(NC(C3(C)ON=C(C)C3)=O)C2)=O)ncc2ccccn12 C1(CC(=O)NCC2C(C)(C)N(C(c3ccco3)=O)CC2)Cc2cc(F)ccc2O1 Cc1cccn2cc(C(N3CC4CCCC(C3)N4C(=O)C3=CCCC3C)=O)cc12 Cc1cc(C(=O)NCC2CCC(NC(C3Cc4nccn4C3)=O)C2)cc(N)c1O c1(C(=O)NC2C(C)(C)CN(C(=O)CN3CC(=O)NC3=O)C2)cnc2sccc2c1 C1(C(=O)NCC(C)NC(c2ccc(F)c(N)c2)=O)C(C)OC(C)C1C CCCC(C)(C)CN=c1[nH]c(=NC2CCCCC2CC)[nH]c2c1SCC2 O=C1CC(CC(=O)N(C2CCCN(C(C3(F)CCCCC3)=O)C2)CCF)CCCN1 c1(C(=O)NCC(C)N(C(C(C)Cn2ccnc2)=O)C)cn(C)nc1-c1ccoc1 N#Cc1cnn2cc(C(=O)NC3CN(C(C4CC4F)=O)C3)cnc12 C1(=CC(=O)NCC2CCC2NC(C2CC2[N+](=O)[O-])=O)CCCCCC1(F)F c1(NCC(C2CCC2)OC)nccc(=NCC2CCC=CCC2)[nH]1 CC(C)(C)CC(O)C(=O)NCCC1CSCCN1C(c1ccc(N)cn1)=O c1(C(=O)NC2C(CNC(CCC#C)=O)C2)cc(F)cc2c(Br)cccc12 c1(C(N2CC(C)CC(NC(C(C(CC)C)O)=O)C2)=O)ccc2ccoc2c1 c1(C(=O)NC(CCNC(C2(C(=O)NC)CCC2)=O)C)cc(-c2ccco2)on1 N(C(=NCc1ccc(Cl)nc1)NCC(=O)N(C)OC)C(CC)C.C(C)(C)SCC C1(CNC(CC(C)O)=O)CCCCC1C(=O)NCCNC(C1CCCC1)=O n1(CC)cc(C(N2CC(Nc3nccc(C)n3)CC2C)=O)c(C(C)C)n1 N1(C(C2CCN(C(CC(CC)O)=O)CC2O)=O)CCN(CC)C(C)(C)C1 C=C(C)CC(C(=O)NCC1(CCNC(=O)C(CC(C)C)N(C)C)CC1)NC(C)=O N1(C(=O)Cc2cccc(Cl)c2)CCC2C(CCN2C(c2c(F)ccc(F)c2O)=O)C1 C(CCC(=O)NC(C1CCN(C(=O)Cc2cnn(C)c2)C1)(C)C)NS(C)(=O)=O C1(NC(C(C2CCN(C(c3csnn3)=O)CC2)C)=O)CC2CC1CC21CC1 c1(CC(=O)N(CCOCCN(C(=O)Cn2nnc(=N)[nH]2)C)C)ccsc1Br c1(C(=O)OC)c(CO)nc2sccn12.C123CCC(CO1)(C2)CNC(=O)C1(CC1)S3 C(=O)(C(C)(C)C(C)(C)O)NCC1C(NC(c2cn(CC)nc2C)=O)CC1 CC(C)C(C(C)NC(=O)C=Cc1ccccn1)NC(c1ncncc1Cl)=O N1(C(C2CC(=O)OC2)=O)CCCC2(CNC(c3cnoc3)=O)CCCC12 CC1(C)CC(CC(=O)NC2CCC(C(=O)NC3(C)CCOC3C3CC3)C2)CO1 Cc1cncc(C(=O)NC(CC2CCC2)C(=O)NCCCNC(=O)C(C)C)c1 N1(C(CCC=C(C)C)=O)CC(CC(=O)NC(c2nn[nH]n2)C2CC2)CC1(C)C CCC(CC)C(C)C(=O)N(C)CC1COCCN1C(c1ccc(S(C)(=O)=O)o1)=O C(=O)(CCCCCF)NC1CCN(C(c2scc(OCC)c2)=O)C1 CC1(C)COC(CC(=O)N(C2CCCC2)CCNC(=O)C=Cc2cncs2)C1 c1(-c2cc(OC)c(O)cc2)n[nH]c2c1CN(C(=O)C(C)N(C)C)CC2 N(C(=NCCC=CC)NC1CCOC(C)C1)CC1(OCC)CCCOC1 C(=O)(CCCCCn1cc(C2CCN(C)C2)nn1)N(CC(=O)OC)C(C)C c1(C(=O)OC)ccc(C)c(S(=O)(=O)NCCc2nnc3n2CC(C)CC3)c1 C(=O)(CCS(C)(=O)=O)N1CC(N(C(c2c(C)nc(CC(F)(F)F)s2)=O)C)C(O)C1 N1(C(C(c2ccccc2)N(CC)CC)=O)CC2CC1C2CNC(=O)C(C)C(F)F n1(CC)nc(C(=O)NC(C)CCNC(=O)C(O)C(C)(C)C)c(Cl)c1Br CC1(C)CCCC(NC(N2CCOCC2c2ncno2)=O)C1 C1(NC(CN(C(=O)Cc2cnn(C)c2C)CC#C)=O)CCn2nnnc2C1 N1(C(C2N(C(C3CCCO3)=O)CCC(CC)C2)=O)CCc2nc(C)[nH]c2C1 C1(NC(CC2CC(COC)C2)=O)CC2CCC(C1)N2C(c1cnc(OC)nc1)=O C12(NC(CCCC#C)=O)CCOCC1CN(C(c1noc3ccc(Cl)cc13)=O)C2 CCC(C)CC(=O)NC1CC(NC(=O)CN2CSCCSC2)C1 N1(C(c2c(CC)[nH]cc2)=O)CCC(COC)(NC(=O)CNS(=O)(=O)NC)C1 Cc1cc(C)n(CC(=O)NC2CC(C)(CNC(C3(F)CCOC3)=O)C2)n1 C1(C(=O)NC(c2cc[nH]c2)CNC(C2C(OCC)CC2)=O)CCN(C(C)=O)C1 C1(NC(c2n(CC)nnc2C)=O)CN(C(C2(n3cnnn3)CC2)=O)CCC1CO C1(C(=O)NCC2(F)CCN(C(c3c(C)nn(C)c3Cl)=O)C2)CCc2cncn2C1 C1(CNC(CSC)=O)N(C(C2(c3cccc(C)c3)CC2)=O)CCC1(C)C N1(C(C=CC)=O)CCC2CCC(NC(c3ccc(F)cc3[N+](=O)[O-])=O)C1C2 n1(CC(=O)NC2C(CNC(C(CCSC)O)=O)COC2)cc([N+](=O)[O-])ccc1=O C=CC(CC)CC(=O)NC1(CCNC(=O)CSS(C)(=O)=O)CCCC1 c1(C(=O)NC(C(C(C)C)C)CNC(C23CC(CO2)C3)=O)ccnc2c1CCC2 N1(C(C(C)O)=O)CCC(C2(O)CCN(C(c3cc(Br)ccc3N)=O)C2)CC1 O=C(N1CC2OC(=O)OC2CN1)NCc1ccc(Br)c(F)c1F c1(CC)nncn1CCNC(=O)CCOCCN(C(=O)C(c1ccn(C)n1)C)C C1(C(N(CC=C)Cc2ccco2)=O)CCC(n2cc(-c3csnc3C)nn2)C1 c12cccc(C)c1S2.C1(CC)CCCCN1CCC(c1ccccc1)OC(=N)O C1(C(=O)NCc2cc(OC)ncc2)CCCCN(C(C2CCC(C)(C)OC2)=O)C1 C1(CC(=O)NC2(CC=C)CN(C(=O)CN(CC)CC)C2)CCN(C)C1=O CCCN(CCO)N1CC(S(=O)(=O)N2CCCCC2)C1 CON1CC(C(=O)NC(C)(CNC(c2cn(C)nn2)=O)C2CC2)CC1=O c1(C(=O)NC(CCCNC(C(C)Cn2ccnc2)=O)C)ccc(S(C)=O)cc1 C(C)(N=c1[nH]c2c(c(=NCC3CC34CCC4)[nH]1)CCCCC2)c1nnc(C)o1 C1(C(=O)Nc2ccc(CC)nc2)C(C2CC2)CCN1C(=O)Cc1ncoc1C c1(CC(=O)NCCN2CCN(C(c3c(C)ccs3)=O)CC2)ccccc1S(C)=O Cn1ccc2c(S(=O)(=O)N3CCC(COc4ccccc4Br)C3)cccc12 C1(CC(=O)NC(CCN(C(c2c(C)noc2C)=O)C)C)CCCNC(=O)C1 C1(NC(c2n(C)ccn2)=O)CCC2(CC1)CN(C(C1CC1C1CCC1)=O)C2 c1(CNC(c2cc(C)nn2C)c2n(CCOC)nnn2)cnc2ncccn12 c1(CCCC(=O)N(CCCNC(c2cccs2)=O)C(C)C)csc2ccccc12 C1(C(N2CC3(CN(C(C=CCC)=O)C3)C2)=O)CCc2ccc(F)cc2O1 c1(NC23CC(CNC(=O)OC(C)(C)C)(C2)C3)sc2cccnc2c1N CC1CCN(C(c2ccncn2)=O)CC1N=c1ccnc(C2CCCC2)[nH]1 n1(CC(=O)NCC(CC)NC(=O)CCCn2cccc2)nc(C)n(C)c1=O c1(CNC(CC2CC(C)C2)=O)ncoc1C1CN(C(=O)C(C)NC=O)C1 C(C(=O)N1CCC(NCC(c2cncc(C)n2)(C)C)CC1)(C(C)C)NC(C)=O Cc1cccc(C)c1S(=O)(=O)CCN1CCCCCC1c1cc(C(=O)O)cc(F)c1 C1(C(C)C)CN(C(=O)COCP(C)(C)=O)CCN1C(=O)Cc1nccn1C n1(CC)nccc1C=CC(=O)NCCC(C)CCNC(C1(CSC)CC1)=O CC1CN(C(C2CCCCS2)=O)CCN1C(=O)COC1CCCOC1 C1(O)(C(=O)NCCN(C(=O)CSc2nccn2C)C)CCOC1 N1(C(C(CC)(C)CC)=O)CC2CCC1C(NC(c1ccc(C)c(C(C)=O)c1)=O)C2 CC1CC(C)(C(=O)NCC(=O)NCC(=O)NCC2CC23CCC3)C1 Cc1ncc2c(n1)CCC(C(=O)N(C)CCNC(c1coc(S(C)(=O)=O)c1)=O)C2 N1(C(CC2CCN(C)CC2)=O)CC2(CCCC2NC(=O)C=CC2CCOCC2)C1 c1(NC(C2CN(C(=O)NC3CCC(C)C3)CC(F)(F)C2)=O)coc2ccccc12 c1(C(N(CC(CNC(c2nc(CC)oc2)=O)C)C)=O)cc(Cl)c(F)c(Cl)c1 N1(C(C(C)SC)=O)CC2CCCC(C1)N2CC1CN(C(C)C)CCS1(=O)=O c1(C(N2CC(O)(CNC(c3cc(F)ccc3Cl)=O)C2)=O)cc(F)cc2nn[nH]c12 N1(C(CCOCC#C)=O)CCC2(CCCN2C(c2cccc(CC)c2O)=O)C1 n1(CC)cnc2c(NC(C)CN3CCOCC3)nc(N3CC4C(C3)C4(F)F)nc12 C1(C)(NC(C)=O)CCN(C(=O)CC2C=CC(NC(c3cccc(CO)c3)=O)C2)C1 C1(OC)CC(CNC(c2cc(CO)c(C)o2)=O)N(C(=O)CC2C=CCC2)C1 N12CC3CCCC1C3(CO)CC(C)CN(C(=O)OC(C)(C)C)CCCC2=O C1(C(N2CCC(OCc3onc(CC)n3)C2)=O)CCN(C)CC1 Cc1cc(N)cnc1C(=O)NCC(C)(C(C)C)NC(=O)CC1OCCC1(C)C C(CCCCN(C)C(C12CC(F)(C1)C2)=O)NC(C1C(C)C1C)=O c1(C(N2CCC(NC(C(C)(C)CC3CC3)=O)C2)=O)cn2cc(Cl)cnc2n1 CC1CN(C(=O)CCC2CCCCN2C(=O)C=CC(F)F)CC1O c1(C(N2CCC(COC)C2)=O)cc(N2CCCC2)nc(Cl)c1 c1(NC(N(C)Cc2ccc(F)cn2)=O)nccc(N2CCCCC2)n1 c1(NCC(=O)NCC2CCN(C(C(OC)OC)=O)CC2O)ccc2ccoc2c1 C1(COC)CN(C(c2cc(C)ccc2I)=O)CCN1C(c1cc(C)c(Br)s1)=O N1(CCn2cncn2)CCCC(C(N2CCCNC2)C)C1 c1(C(=O)NCC2OCC(CNC(C(CSC)C)=O)C2)ccc(C(C)(C)C)cn1 N1(C(C(C)Oc2ccccc2)=O)CCN(C(c2ccc(F)c(CO)c2)=O)C2CC12 N1(C(Cc2cnc(C)[nH]2)=O)CCCC(CCNC(c2c[nH]cc(Cl)c2=O)=O)CC1 CCCCC(C)(F)C(=O)NC(c1cccc(C)c1)CNC(=O)CCc1nccs1 N1(C(CN2CC(C)(C)C2)=O)C(CNC(C23CCC(CC2)OC3)=O)CC2CCCC12 C1(CNC(Cc2nnc(C)o2)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1C Fc1cc(CNCCc2cccs2)c2nncn2c1 c1(C(=O)NCC2CCCCN(C(=O)C(F)CC3CCC3)C2)cccc([N+](=O)[O-])c1 Cc1cc(C(N2CC=CC2C(=O)NCCCc2ncn(C)n2)=O)cs1 c1(CC(=O)NC2CN(C(c3cc(C)n(C)c3C)=O)CC2O)cccc([N+](=O)[O-])c1 C(CNC1C(C)C1)(C(C)(C)C)NC(=O)CCN(CCCO)C(C1CSCCS1)=O C(=O)(CC(CC(=O)O)C(C)(C)C)NCc1nc(C)cc(C)n1 C=CCCCC(C)N=c1[nH]c(=NCCCn2cccn2)[nH]c2cccc(F)c12 C(C(COC)CC(=O)NCCC1CCN(C(=O)Cc2ccsc2C)CC1)OC C(=O)(C(CC(C)C)C(C)C)N(CCCNC(CC(C(F)(F)F)OC)=O)C c1(C(=O)NCCN(C(c2c(C)c(C3CC3)on2)=O)C2CC2)cccc2c1COC2 CC1CC(=O)CCC1C(=O)NC1CC2(C1)CC(C(N1CCCC1CN(C)C)=O)C2 C1(C(N2C(CCNC(CC3CC(=C)C3)=O)COCC2)=O)CCCCC(=O)N1 C1(C2(O)CN(C(C3CC(F)(CO)C3)=O)C2)(CNC(=O)Cc2ccc(Cl)cn2)CC1 C(=O)(C(C)C(C)C)NC(CN(C(CCNS(CC)(=O)=O)=O)C)(C)C c1(C(=O)Nc2cnc(OC)nc2)ccc(-c2cccc3ncnn23)c2cc[nH]c12 N1(C(C)=O)CCC2(CC1)OC1(C)CC2(NC(=O)CCCc2ccc(C)c(C)c2)C1 C1(C(N2CC(NC(C3(C)CC3(Cl)Cl)=O)C(CO)C2)=O)CC2C(C1)C2(C)C N1(C(c2c[nH]c(=NC)s2)=O)CCC(O)(CNC(c2ccnnc2S)=O)CC1 c1(CC)ccc([N+](=O)[O-])cc1C(N1CCCC(C(C)NC(=O)C2=CCC2)C1)=O c1(CCNC(C2C(=C)C2)=O)ccc(CNC(c2sccc2OC)=O)cc1 N1(C(Cc2ccn(C)n2)=O)CCCC(CCCCNC(=O)Cc2ccoc2)C1 N1(C(C=CC(C)C)=O)CCC2C(C(=O)NCC34CCCC3OCC4)C2C1 C1(C(N2CC(C)(NC(Cn3c(C)cnc3)=O)C2)=O)CCn2ccnc2C1 N1(C(C2=C(C)OCC2)=O)CCC(NC(=O)C=CC2(C)CCOCC2)C2(CCC2)C1 C12(NC(c3cc(Cl)cnn3)=O)CCOCC1CN(C(=O)C=Cc1ccco1)C2 C1(NC(c2nnc(C(C)C)s2)=O)C(C)CCN(C(C2CCC(=O)N(C)C2)=O)C1C c1(COC)nc(C)cc(=NC(C)C2CN(C(c3ccc(Cl)cc3)=O)CCO2)[nH]1 C1(NC(c2c(C)nc(CCC)o2)=O)CN(C(c2[nH]ncc2C#N)=O)CC12CCC2 c1(OC)cc(C(=O)NCC(C2CCOC2)NC(c2cnn(CCF)c2)=O)sn1 c1(NC(C2C(NC(c3ccc(F)nc3)=O)C2)=O)ccnc(Cl)c1 c1(C(N(CC(CNC(C(CC)CC2CCCC2)=O)O)C)=O)cccc2sncc12 CCC(CCO)N=c1nc2c(ncn2C(C)C)c(NC(CC)CCO)[nH]1 c1(C(=O)NCC2C(NC(COCCCOC)=O)C2)[nH]c(=N)ccc1C c1(C(=O)NCC2N(C(C(CC)CC)=O)CC(O)C2O)cnc2c(ccn2C)c1 O=C(C1=CS(=O)CCC1)NC1(CF)CCN(C(c2cccn3ncnc23)=O)C1 c1(C(N(CCNC(C(C(C)C)OC)=O)C)=O)cc2c(F)cc(F)cc2[nH]1 Cc1oc(CO)cc1C(N1CCCCC1C(=O)N(CC(C)CO)C)=O N1(C(C(CCC)NC(C)=O)=O)C2CCCC1CC(NC(c1cc(C#N)c[nH]1)=O)C2 C(CC(O)C(=O)NCc1ncccc1CNC(=O)CCn1cccn1)SC N1(C(c2cc(CC)on2)=O)CCC(CNC(=O)C(C)Cc2ccccc2)C12CC2 C1(O)(CNC(c2cn(CC=C)nn2)=O)CCCN(C(C2CCC3(CC2)CC3)=O)C1 C(=O)(CCC1=CCc2ccccc21)NC1CC(N(C(C(CCC)C#N)=O)C)C1 N1(C(Cc2cnc(C)s2)=O)CCN(C(=O)CN(C)C(N)=O)CC1c1cccnc1 C(=O)(C(C)C(F)(F)F)NC1C=CC(CC(=O)NC2(c3nc(C)on3)CC2)C1 C1(CNC(C(C)NC(=O)C(C)(C)C)=O)CCN(C(c2ccns2)=O)CCC1(F)F C(=O)(CCN(OC)C(=O)C(C)C1CCN(C(=O)CCNC(C)=O)C1)OC c1(C(C)C)cnc(O)c(C(=O)NCCCN(C(=O)C(C)(C)COCC(F)F)C)c1 N1(C(C(CC)NC(C)=O)=O)CC2=C(C1)CN(C(C1CCCCN1N=O)=O)C2 N1(C(C=CCOC)=O)CC(CNC(c2cccc(C)c2C)=O)CCC1C N1(C(C(C)Oc2cccc(F)c2)=O)CC(n2cc(C3CCCOC3)nn2)C(C)C1 C1(C(=O)NCc2cnc[nH]2)COCCC12CCN(C(C1CCCS1)=O)CC2 N1(C(c2cc(OCC)no2)=O)CCCC(C)C1CNC(c1ccn2ccsc12)=O Cc1ccc(C(=O)NC(CNC(=O)CC2(C)CCCC2)C(C)C(C)C)c(=O)n1C Cc1ccc(Cl)c(O)c1C(N1CC2CC2(NC(=O)C(N)=O)C1)=O C1(CCC)CN(C(c2cncc(OC)c2)=O)CC1NC(=O)Cc1nocc1C C1(C(N2C(CNC(CC3(C(=O)OC)CCCC3)=O)CC2)=O)CCS(=O)(=O)C1(C)C Cc1cc(=NCC2(C3(CNC(C4CCOCC4)=O)CC3)N=N2)c([N+](=O)[O-])c(C)[nH]1 N1(C(C2C(C(C)C)C2)=O)CCN(C2CCN(C(c3cncc(N)n3)=O)C2)CC1 Cc1nc(C(=O)NC(CC(N)=O)c2cn(CC3C(CO)C3(C)C)nn2)[nH]c1C C(=O)(CCC(N)=O)N(C1CCN(C(=O)C(=Cc2ccncc2)C)CC1)CC c1(C(=O)NS(=O)(=O)CCC2CN(CCO)C2)c[nH]c(=O)cn1 N1(C(CCOC)=O)CCN(C(=O)CC2CCC(OC)CC2)CC1c1nccn1C c1(C(N(CC(CN(C(c2ccc(C(C)=O)o2)=O)C)O)C)=O)cc(=O)cc[nH]1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC(NC(CC(CCCC)O)=O)CC1 N1(CCCOC)CC(NC(=O)C(=O)N2CC(c3ccc[n+]([O-])c3)C2)CC1=O C1(C(N(CC)CC2CCN(C(=O)C(C)CO)CC2)=O)CC2CC1CC2O C1(CC(=O)N(C2CN(C(c3cc(Cl)sc3Cl)=O)C2)C)CCCC2CCCCC12 c1(CC)cc(C(N2CC3CC3(CNC(c3ncccc3C(F)F)=O)C2)=O)ccn1 CC1OCCC1(C)C(=O)NCC1(C(=O)NCC(c2ccccc2)C)CCC1 CC1CC(NC(c2csc(CO)n2)=O)CCN1C(C1(C)CC1)=O N1(C(c2nnn(COCC)c2N)=O)CCCN(C(C2CC2(C)CC)=O)CCC1 N1(C(CCCNC(C)=O)=O)CCC(CNC(C2CCCC3CCCC23)=O)C1(C)C c1(C(=O)NCC2CCN(C(C=CCC)=O)CC2C)cc(Cl)cc(Cl)c1OC(F)F C1(C(N(CCNC(CCc2ccc(C)cc2)=O)C)=O)CC(c2ccncc2)=NO1 CCC(CC(=O)NCC(CC)N(C)C(C1CC(N(C)C)C1)=O)C1CCC1 Cc1cc(S(N)(=O)=O)sc1C(N1CCCCCC(NC(=O)C(F)C(C)C)C1)=O C1(CNC(c2cnc(CC(C)C)[nH]2)=O)CCCN(C(C2CC(C(F)F)C2)=O)C1 C(=O)(C1=C(Cl)CCCC1)NCCCCCCN(C(c1c(CC)cc(C)cc1)=O)C N1(C(C=CC)=O)CCN(C(=O)CC(F)(F)F)CC1CS(C)(=O)=O c1(C(=O)O)cc2n(n1)CCN(CC1CCc3cc(Br)ccc3O1)C2 N1(C(CCC#C)=O)CC(C)OC2(CCN(C(c3cc(O)cc(Cl)c3)=O)CC2)C1 C(CCCC(=O)NCCc1ocnc1CNC(=O)C(C1CC1)C1CC1)OC N1(C(CC#N)=O)CCCC(C2CCCCN2C(c2cn(C3CCOC3)nn2)=O)C1 C1(NC(C=CSC)=O)CCC2(CC1)CC2NC(=O)C=CC1CCOCC1 c1(C(=O)NCCN(CCC)C(C2CCSC(C)C2)=O)[nH]nc2ncccc12 CCC(CNC(=O)OC(C)(C)C)(C(=O)OC)NCCN1CCCCC1 C1(NC(c2cc(C)on2)=O)CCCN(C(=O)CC2CCOCC2)CCC1 S(=O)(=O)(c1cc(F)c(F)cc1F)N1C2CN(C(c3cc(C)cc(C)c3)=O)CC21 c1(C(N(C2CC(NC(C3(C)SCCCS3)=O)C2)C)=O)ncc2[nH]ncc2n1 C=C(C)CC(C(=O)N1CC2CC2(NC(=O)Cn2cc(C(C)=O)nn2)C1)OC C(=O)(C(O)CCCCC)N(CCOCCN(C(CCCCCC)=O)C)C C1(C(=O)NCC2(CNC(C(C(CC)C)OC)=O)CC2)CC12CCCCCC2 CCCCCCC(=O)N1CCC(COC)(NC(c2cnc(C(N)=O)cn2)=O)C1 C1(C(=O)NCCCCC(C)NC(CCCCC=CC)=O)COC2(CCC2)CO1 Cc1cnn(C(C)C(N2CC(c3ccccc3)(NC(=O)CCC3CCC3)C2)=O)c1 O=C(CC1OCCc2ccccc21)N1CCN(C(c2ccnnc2)=O)C2(CC2)C1 C1(C(=O)NCC2N(C(C3(c4cccc(F)c4)CC3)=O)CCC2)CCCS(=O)(=O)N1 c1(SCC(=O)NC(CN(C(C2C(C)C2)=O)C)(C)C)ccc(S(N)(=O)=O)cc1 C1(NC(C2CC3CC3C2)=O)CCCC12CN(C(c1csc(Cl)c1Cl)=O)C2 C1(NC(C(C)Oc2cccnc2)=O)CCCC(NC(c2cncc(N)c2)=O)CC1 C(=O)(C1CCCc2c[nH]nc21)NCC1CC(O)(CNC(C(CCCCC)F)=O)C1 C1(c2onc(C)n2)CCCN(C(=O)Nc2ccccc2C(C)C)C1 N1(C(c2nnc(C3CC3)s2)=O)CCN2C(=O)N(CC(F)(F)F)CC2C1 CCC(CCCC(=O)NC(CO)CCC(C)C)NC(C1(CCOC)CCC1)=O C1(NC(CC(C)n2ccnc2)=O)CCCCN(C(=O)CP(C)(C)=O)CC1 c1(OC)cccc2c(C(=O)NC(CNC(=O)C3=CCOC3)C(C)(C)C)c(C)[nH]c12 c1(C(=O)NCC2COC(CNC(C3CN(C4COC4)C3)=O)C2)n[nH]cc1[N+](=O)[O-] CCC(C)(C)C(=O)C(=O)N1CC2CC1CN(C(=O)COC1CCOC1)C2 C(=O)(C1=CCCC1)N(c1ccccc1)C(CNC(Cc1nc(COC)sc1)=O)C1CC1 c1(NC(C(N2CCC(CNC(N(CC)CC)=O)CC2)=O)=O)cc2cccnc2[nH]1 C1(C(N2CC(CC=C)(NC(=O)CC(C)OC)C2)=O)CCC(NC(N)=O)CC1 C1(C(=O)NC2CC(NC(=O)C=Cc3cc[nH]n3)C(O)C2)CCCC2(CC2)C1 N1(C(=O)Cc2cc(Br)cs2)CC2CCC1CN2C(C1CC(O)C1)=O c1(C(=O)NCC(c2ncc[nH]2)C)ccc(CNC(C2CCSC2)=O)nc1 C1(C(C(=O)NC(Cc2ccc(C)cc2)C(=O)O)NC(C)=O)CCCCCC1 N1(C(C=CCC)=O)CCCC(C(C)(O)CNC(c2ccsc2Cl)=O)C1 c1(OC)ccc(SCC(N2CCCC2C(C)CNC(C2(C)CCCS2)=O)=O)cc1 N1(C(c2ccn(CCC)n2)=O)CC(C(=O)NCC2CC23CCCCC3)CC1(C)C C1(NC(=O)NCCNC2(C3CCCO3)CCCC2)CC12CCSCC2 C1(CNC(C(C)(C2(C)CC2)OC)=O)CCCC(NC(=O)C(F)=CC2CC2)C1 CC1CCC(CC(=O)N(CCCN(C)C(c2cnn(C)n2)=O)C)O1 N1(C2CCN(C(C3C(=C)C3)=O)C2)CCN(C(=O)C(CC)n2ccnc2)CC1 C1(O)(C(N2CCC(CCCC)C2)=O)CCN(CC=Cc2ccco2)CC1 N1(C(C(N2CCN(C)CC2)C)=O)CCC(C(F)(F)F)C(NC(C2(CF)CC2)=O)C1 c1(CN(C2COC2)CC#C)ccc(NC(C2CCN(C(=O)NC)C2)=O)cc1 C=CC(C)CC(=O)N1CCOC(CCCNC(c2ccc(CC)[nH]2)=O)C1 c1(N2CCC(=CCNC(c3c(Cl)nc(N(C)C)s3)=O)CC2)ccc2nnnn2n1 c1(C(=O)NC(CC)CN(C(=O)C=C2CCOCC2)CC)cn(C)c(C)n1 C=C(C)CC(C)C(=O)NCC(C)(C)CN(C)C(c1csc(C(C)(C)C)n1)=O c1(C(=O)NCCOC2N(C(CNC(CCC)=O)=O)CC2)ccsc1-n1cnnn1 c1(C(=O)NCC(C)N(C(=O)CC2CSCCS2)CC)cnc(C)nc1C1CC1 C(N=c1cc(-c2cccs2)nc[nH]1)C1CCC(CNC(C(CC)C(C)O)=O)CC1 n1(CC)ncc(C(=O)NCC2C(C)CCN2C(c2ccc(C(C)=O)cn2)=O)c1C c1(C(N2C(C)CC(CNC(C3CCC(CC)O3)=O)C2)=O)cc(C)c(O)nn1 N1(C(CSC)=O)CCC2(CCC2)C(CNC(C2CC2C2CCCCC2)=O)C1 c1(OCC)ccccc1NC(c1nnnn1CCCF)(C)CSC1(C)CCCO1 CC1CN(C(=O)CC2COC(C)(C)C2)CCC1NC(=O)CCCc1cnn[nH]1 c1(N2CCC(NC(CCn3c(C)csc3=O)=O)C(O)C2)nn(C)cc1[N+](=O)[O-] c1(CC(=O)NCC(CNC(C(C2CC2)SC)=O)C)ccc(C(N)=O)nc1 c1(NC(=O)C(c2cccs2)NC(C2CC(CF)C2)=O)cncc(C(N)=O)c1 N1(C(c2cnc(C)[nH]2)=O)CCC(F)(F)C(CNC(=O)CN2CCCNC2=O)C1 C1(C)(C(N(C)CC2OCCN(C(CN3CC(CC)C3)=O)C2)=O)CCCS1(=O)=O n1(CC)ncc(Cl)c1C(N1CCC(CCNC(c2cnc(O)n2CC)=O)C1)=O CCCC(C)CCCC(=O)N1CC(O)(C(C)(C)CNC(=O)C(C)SC)C1 Cc1nc(C(=O)NCC2(F)CCN(C(C3(C(N)=O)CCC3)=O)C2)cc(O)n1 N=c1[nH]c(=NCc2ncccc2N)[nH]c(=NC2CCN(C3CC3)C3(CCC3)C2)[nH]1 N12C3CCC1CC(C3)C2=O.C1(C(=O)NCc2nc(C)c(C)[nH]2)(CC)CCCOC1 c1(C(=O)NCC(C)(CO)NC(C(CC)n2cncn2)=O)ccc2n[nH]cc2n1 N(C(=NCCN1CCC(C)(C)CC1)NC(C)C(C)COC)C(COC)C N1(C(CC(C(C)C)O)=O)CCCN(C(=O)CCNC(c2cnccn2)=O)C(C)C1 C(=O)(C1NCCOc2ccccc21)Nc1c(NC(C)=O)ccc(N=[N+]=[N-])c1 C1(C(=O)NCC(=O)N(C(C)CCO)C2CCCC2)C2CCC1(c1ccn(C)n1)C2 Cc1cc2c(s1)CCN(C(=O)NC(c1c(C)nn(C)c1C)c1ccccc1)C2 N1(C(c2n(CC)nnc2)C(=O)NCCC2CC2)C(CO)CC2CCCCC12 CC1CN(C(=O)C(F)n2ccnc2)CC1NC(c1csc(C(N)=O)n1)=O N1(C2C(=O)N2)CC(OC)(CNC(CSCCOC)=O)C1.c1nccn1C.C1CC1 C1(C(=O)NCCN(C(C2CC(c3cccc(Cl)c3)(O)C2)=O)CC)OC2CCC1CC2 N1(C(C(C)O)=O)CC(C)(NC(c2ccoc2I)=O)C1 C(C)(N=c1[nH]c(N2CCCN(C)CCC2)nc2ccsc12)C1CCCC(CC)C1 Cc1ncccc1CNC(c1nnn(C2CC2)c1C(F)(F)F)=O N1(C(c2n(C=C)nnc2)=O)CCC2(CC1)CC2CNC(=O)CCCSC c1(C(N(C(CC)CNC(c2cn(CCOC)nn2)=O)C)=O)cnc2ccccn12 C1(CNC(CC(c2ccccc2Cl)C)=O)CCN(C(=O)CN(C)C2CC2)CC1C C1(C(=O)NCC(C)(C)C2(O)CCC2)CC12CCC(F)(F)CC2 N1(C(C(CCC)OC)=O)CCCN(C(=O)COc2cccnc2)CC1C(C)C C(N=c1[nH]c(C)cc(=NC2CCC3CC2CO3)[nH]1)C1CCN(CC)C1 C(CCF)(C(=O)OC(C)(C)C)NC(N1CCC(C(C)(C)C)(C(=O)OCC)C1)=O C1(CC)CCCC1(C)C(N1CCN(CCCNC(=O)C2CC2)CC1)=O N1(C(C2CC=C(C)CC2)=O)CCC(C)C(N(C)C(C2(C)CCN(C)CC2)=O)C1 CP(C)(=O)CCC(=O)NCc1cc(C(=O)Nc2ccc(Cl)cc2O)co1 C1(C(N2C(C(N)=O)CCC2)=O)(CNC(c2cc[nH]n2)=O)CC12CCC2 C(=O)(CCCC(=O)C1CC1)N1CCC(NC(=O)C(N2CCCC2)C2CC2)CC1 O=C(CC(C1CC1)NC(c1c[nH]cc1C1CC1)=O)NC1CCOC1=O C(C(C)(O)CC(=O)N1CCC(C(=O)NCCC(F)(F)CO)(C(C)C)C1)OC C#Cc1cccc(C(=O)NCCCOCCNC(C2(CC3CC3)CCOC2)=O)c1 c1(OC)c(Br)cc(F)c(OS(=O)(=O)c2cn(C)c(C)n2)c1[N+](=O)[O-] C1(NC(c2nc(CC)sc2)=O)CN(C(=O)COCC2CCCC2)C2CC12 Cc1nc2c(CCC(N3CCC(CNC(=O)CCOC(C)C)C3)=O)cccc2o1 C12(C(=O)NCCC(C#C)C)C(NC(=O)C(CO)OC)C3CC1C2C3 C(CCCCCC(=O)NCC1CCSC(C)C1)NC(CCCOCC)=O C(Cc1ccoc1)(C(=O)NCCC(C)C)NC(C=CC)=O c1(C(=O)NC(CN(C(CC(CC)C2CC2)=O)C)C)cc(S(C)(=O)=O)ccc1OC N1(C(c2c(CC)cno2)=O)CCCC(F)(CNC(C2CC(F)(CO)C2)=O)C1 c1(C(N2C(C(C)(C)NC(C(C)C(F)F)=O)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(=O)NC2(CC=C)CCN(C(C3CCN(C)C(=O)C3)=O)C2)cnc(Cl)cc1N CC1=C(C(=O)NC2CCCC2CC(=O)NC(CC(C)C)C(=O)N(C)C)SCCO1 N1(CC(=O)NCC2C(O)C(O)CN2C(C2CCC(=O)O2)=O)CCCCS1(=O)=O C1(C(N(C2CC(NC(C(C)NC(N)=O)=O)C2)C)=O)CCCC2(CCC2)C1 c1(C(=O)NC2(CC(=O)N(CCOC)C)CCC2)ccc(C)cc1O C=CC(CC)C(=O)N1CCCC(CCCCNC(C2CC(=O)N(C)C2)=O)C1 C1(N2CC(N(CCCOCCCO)C(=O)Nc3ccccc3)C2)CCOCC1 CCCN=C(NCc1ccc(SC)cc1)NC1CC(C)N(Cc2ccccc2)C1 C1(NC(C(C=C)CC)=O)CN(C(=O)C(c2ccccc2F)O)CC1C=C N#Cc1cc(NCC2CC23CCC3)nc(Cl)c1 CC(C)(C)C(CC(=O)N1CC(O)C(F)C1)NC(C1CCCC(CF)C1)=O Cc1ccc(C(=O)NC2CC3CCC2N3C(=O)CC(C)c2cnn(C)c2)nc1C Cc1cccc(C)c1OCC(N1CC(NC(=O)CCc2ncco2)C(F)C1)=O c1(C(C2CCOCC2)=O)ccnc2ccncc12.N12CC(C3(CC3)C1)C2=O C1(C(=O)NC2CCCN(C)C2)CC2CN(C(=O)COC3CCOC3)CC2C1 c1(C(=O)NCC2CCC(NC(c3c(CC)nn[nH]3)=O)C2)cnc(C2CC2)nc1O c1(C(N2CCN(C(c3c(CC)c[nH]n3)=O)CC(O)C2)=O)ccn2c(C)ncc2c1 Cc1cc(C)c(NC(C2(NC(=O)CCCn3ccnc3)CCC2)=O)cn1 O=C(CC1OCc2ncccc21)NCCSCC(O)CO c1(C(=O)NC2CCC(NC(C(Cc3c(C)nc[nH]3)O)=O)C2)csc([N+](=O)[O-])c1 CCC(C#N)C(=O)N1CCC1CNC(=O)C=CCO C1(CNC(=O)Cc2ccc(F)s2)CCN(c2ncccn2)CC1O c1(C(N(C)CC2(O)CCN(C(C(C)OCC#C)=O)C2)=O)cccc2nncn12 C(C(O)CC(=O)NCc1nocc1C(=O)N(C1CC=CC1)C)N(C)C Cc1cc(C(C)C)nc(N(C2CCN(C(C3CC(C)(C)C3)=O)CC2)CCO)n1 N1(C(c2c(Cl)cn(C)n2)=O)CC(C)(C)OCC1CNC(=O)CC1CSCCS1 c1(C(N2CCCC(C(=O)NC(C(=O)OC)C(=O)O)CC2)=O)ccc2cnoc2c1 c1(CN2CC(C(=O)N(C3CC3)Cc3ccccc3)OCC2)c(F)ccc(F)c1F N1(C(C2CCC2(F)F)=O)CCC(F)(C(N2CCN(CCO)CC2)=O)C1 c1(C(=O)OC)[nH]c(=NC2CC23CC(NC(C2OCC2(C)C)=O)C3)sc1C c1(C(=O)NCC2CCCCN(C(=O)Cc3cnns3)C2)cccn2cncc12 C1(C2CCN(C(=O)CC3CCOCC3)C2)(NC(c2cnnc(Cl)c2)=O)CC1 C(=O)(CC(C(F)(F)F)N1CCOCC1)NC1(CO)CN(C(CCCC(C)C)=O)C1 N1(c2nc(OC)c(Br)cn2)CCC2(CC1)CC(NC(=O)CS(C)(=O)=O)CO2 C(=O)(C1=CC2CCCCCC12)NC(C(c1ccc(OC)cc1)OC)C C1(C(N2CC(NC(c3c(C)con3)=O)CC3(C2)CC3)=O)Cc2cc(Cl)ccc2O1 C1(NC(C2CCN(C3CC3)C2=O)=O)CCC(C(=O)NCc2ccccc2O)CC1 Cc1csc2c(C(N3CCC3CNC(=O)C(C3(O)CCCC3)F)=O)cccc12 C1(NC(COCCCC(C)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CCC1C C1(CC(=O)NC(CC)CNC(=O)CNC(C2CC2C)=O)CCCCC1 C1(OC)CCC(CNC2CCCN2C(=O)COc2ccccc2)CC1 CC(C)(C(=O)NCC1CCCO1)C1CCN(C(C2CCSCC2)=O)C1 N1(C(C(=O)NCc2ccn(C)n2)=O)CCC(N)CC1 N#Cc1c[nH]cnc1=NCC1CCCCC1NC(C1CC2(C1)CC(F)(F)C2)=O C1(C(=O)NCCCCN(C(=O)C(F)(F)C2(O)CCC2)C)COCCO1 c1(C(=O)NC(C)(C)CCC(=O)NCC2CCCSC2)cc2cc[nH]c2cn1 C1(NC(c2ncn(C)c2)=O)CC2CC(C1)N(C(=O)CC1NC(=O)NC1=O)C2 c1(-c2nc(CC(CC)C)nn2CCC(C)C)cc(C)ccc1Br C(C(C)(C)C(C)(C)C)NC(CC1CN(C(COCCNC(C)=O)=O)C1)=O c1(C(C(=O)OCc2cccc(OC(F)F)c2)=O)cc2ccccc2s1 O=C(C1CCc2cc(O)cc(=O)n21)N1CCC(C(F)(F)F)OC(C2CCCC2)C1 c12nc(Br)ccc1OC2=O.N1(CC)CC(O)(CC(C)C)C1 C=C(Cl)C(C)(C)C(=O)NCC1CCN(C(=O)C(C)Oc2cccc(C)c2)C(C)C1 C1(OC)CC2(C1)CN(C(=O)CN(C)C(C1(C)CCNC1=O)=O)C2 C(C(COC)C(=O)NCCN(C(=O)CC1CCCOCC1)C)OC c1(CC)ccc(C(=O)N(C)Cc2cccc(Br)c2)c(OC)c1 C1(CN(CCO)CC)CCCCN1C(=O)Cc1cnn(C)c1C N1(C(C2CN(C(COC(CC)(C)C)=O)CC2F)=O)CC(C)=CC(C)C1.C(C)(=O)O c1(C2C(NC(=O)CCCC3N=N3)C2)cccc2ccccc12 N1(C(CCc2c(C)nccc2)=O)CCC2(CC1)CC2C(=O)NC1CCC1(C)C C1(N(C(c2nc(OCC)oc2)=O)C)CCC(NC(=O)CCC(=O)N(C)C)CC1 CCC(CC)CC(F)C(=O)NC1CC(N2CCNC2=O)C1 c1(C(=O)NCC(CO)NC(c2ccc(OC(F)(F)F)nc2)=O)c[nH]cc(F)c1=O C1(C(=O)NCC(C)OCC=C)CC=CCC1NC(=O)COc1ccn(C)n1 C(C)(C(=O)NCCN1CCC(NC(C2CCS2(=O)=O)=O)CC1)(C(C)C)OC c1(C(N2CCCC2CO)=O)ccc2c(c1)CCN(Cc1cccc3c1OCO3)C2 C(=O)(C(C)CC)N(CCC)Cc1sccc1C CCCC(CNC(C1CCN(C(=O)C=Cc2cc[nH]c2)C1)=O)OC C(=O)(C(C)(O)C1CC1)NCC(=O)NCC(=O)N(C)Cc1ncco1 c1(OCC)cc(Cl)ccc1C(N1C2CCC1(CNC(C1CC3CC3C1)=O)CC2)=O c1(OC)nscc1C(N1CCCC1CC(=O)NC1CC1C(F)(F)F)=O N1(C(CC(C)OC)=O)CC(CO)C2(CCN(C(c3csc(CO)n3)=O)CC2)C1 N1(C(C(C)(c2cccs2)N(C)C)=O)CCC(F)(CNC(=O)C#CC(C)(C)O)CC1 C1(C(=O)Nc2cncc(F)c2)(NC(Cc2c(C)non2)=O)CCCC1C c1(C(c2n(CCC)nnn2)NC(C2(C)COC2)C)cnn(C(C)C)c1C(F)(F)F C(=O)(C(C)(F)C(=O)OCC)N1CCC(N(CCC)C(C2CNC(=O)O2)=O)C1 Cc1csc(=O)n1CCCC(N1CCCCC1C1CCCN(CC(C)O)C1)=O C(=O)(CCCS(N)(=O)=O)N1CCC(NC(C(Cn2ccc(C)n2)C)=O)C1C1CC1 N1(C(CC)=O)CCc2[nH]nc(CNC(=O)CSc3cc(Cl)cc(Cl)c3)c2C1 C1(C)(CNC(CC=C)C)CCCNC1=O.c12cc(cs1)COCC2=O CCS(=O)(=O)CC(=O)N1CCC(C)(N(C(=O)C(c2ccccn2)C)CC(F)(F)F)C1 CCC(CC(=O)NC1CC(C(=O)NC2COCCN(C)C2)C1)C(C)(C)C N1(C(C(C)OCCCC)=O)CCC(CNC(c2cn(CCC3CC3)nn2)=O)CC1 c1(CNC(CC2CC(CC)C2)=O)n[nH]cc1C(=O)N(C(CO)C(C)C)C N1(C(C(CC(C)C)N(C(C(COC)(C)OC)=O)C)=O)CCc2ncsc2C1 c1(C(N2CCCC(NC(=O)Cc3ccns3)C(F)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(NC(C2(F)CC2)=O)ccc(C2CCN(Cc3ccnnc3)CC2)cc1 N1(C(CCC=CCC=C)=O)CC(NC(=O)C(=O)N(c2ccccc2)CC#N)C(C)C1 CC1CC(C(=O)N(CC(=O)NCC(O)Cn2cccn2)CC2CC2)CN1C c1(OC)cc(=NC(=O)C(C)(C2CC2)N(C)C(C2C3CCCOC23)=O)[nH]n1C c1(NC2CC(C)C(C)(C)CC2)ccc(S(=O)(=O)NC2CCCCC2)cn1 CC1(C(N2CCCC2CNC(=O)C(F)(F)c2csc(Cl)c2)=O)CCNC1=O CCCC(C)(C)CC(=O)NCC1CCN1C(C1CCC2(CCC2)OC1)=O c1(C(=O)OC)cccc(N(CCNC(c2ccc(C)cn2)=O)CCN(C)C)c1 N1(C(C2CCCN2C(=O)CCn2cccc2)=O)CCCC(OC(F)F)C1 c1(C(=O)NCC2CCCC(NC(=O)CSC(F)F)C2)ccc2nc[nH]c2c1 C1(NC(C2CCOCC2)=O)COCC1CNC(C1CC1F)=O C1(C(=O)OC(C(CC#C)C2CNC2)=O)CC(C)(C)CN1C S(=O)(=O)(c1ccc(Br)s1)NCC(c1cccc(C)n1)C(=O)OC c1(C(=O)NCC2CC2F)cccnc1.C12CCN(C1)C(=O)C(=O)NC(=O)CS2 c12ccc(cc1)S(=O)(=O)N2.C1(CC)CCCCCN1C(=O)N(C(C)C(C)(C)O)C C(=O)(C1CCc2cccc(O)c21)NC(C)CNC(c1ccc(CNC(N)=O)o1)=O CCCC(C)C(c1nnnn1CC)NCCc1noc(CC)n1 C(=O)(C(F)(F)C(O)CC)N1CCC(Nc2scc(CNC(CCCCC)=O)n2)C1 N1(C(c2c3[nH]c(=N)oc3ccc2)=O)CCC2(CCC(NC(=O)CSC3CC3)C2)C1 CCC1=C(C(=O)N2CCN(C(=O)C=Cc3ccncc3)C3CC23)CCCO1 C(CN=c1[nH]nc(C2CC2)s1)=CCNC(c1cnc(Cl)c(C2CC2)c1)=O c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(C(C)C)NC(N)=O)C(C)C)c(C)n1 CCC(C)(C)CCCC(=O)NCC1CCN(C(c2cc(Cl)n[nH]c2=N)=O)CC1C CC(C)CC(O)C(=O)N1CC(c2ccccc2COCc2ccccc2)C(C)C1 c1(C(=O)NCC(C(C)(C)C)NC(CC=CCC)=O)ccc(CC)cc1N Cc1cccc(Br)c1C(=O)NC(CNC(=O)C(C)(C)n1cnnn1)C(C)C C1(CNC(c2ccn(CC)n2)=O)CC2(CC2)CN1C(=O)CCC(=O)c1cccs1 Cc1c(CN2CC(CC(=O)Nc3cccc(-c4cccnc4)c3)C2)ccnc1Cl c1(CCOCC(=O)NC2(CNC(C=CC=CC)=O)CCOC2)ccc(Cl)cc1 CCC(C)C1CS(=O)(=O)N1.c1(NC(=O)OC2CCCCC2C)ccc(OC)cc1 C12(NC(C3CCN(C(C(C(CC)C)=O)=O)C3(C)C)=O)CC3CC(CC1C3)C2 C1(N(C(=O)C(F)CC2CN(C(=O)CC3(C)CCC3)C2)C)CCC(O)CC1 C(CCN=C(NCc1ccc(F)c(F)c1)N1CCC(C)(F)C1)SC c1(C(=O)NCc2nccc(SC)c2)ccc(Cl)cc1C C1(CC(=O)NCC2CCC(NC(c3cc(-c4ccoc4)[nH]n3)=O)C2)CC2(CC2)C1 c1(C(N(C)CC2CCCN(C(C3C(C)C3C)=O)C2)=O)cn(CCO)c(=O)nc1O C(C(C)(CO)CO)N(C)C(C1CCOC1CNC(C1COCCN1C1CC1)=O)=O C(CC(C(=O)N1CC(CO)CC1CO)NC(=O)CC1(O)CCC1)N(C)C CC(C)CC(C)C(=O)N1CCCCC1C1CCN(C(=O)CC2CCCOCC2)C1 Cc1cc(N)c(C(=O)NC(C)CCNC(C2CC2[N+](=O)[O-])=O)c(F)c1 C1(NC(c2c(CCC)nco2)=O)CC2CCCC(C1)N2C(=O)C(C)C(O)C(C)C C(=O)(C1=NN(CC(C)C)C(=O)CC1)NC(C1CCCN1C(=O)CCCN=[N+]=[N-])C C1(NC(C=CC=CCC)=O)CC2CC(C1)N(C(C1CCCN1CCC(C)C)=O)C2 N1(C(C(CCNC(=O)CCc2ccnn2C)OC)=O)CCOCC(O)C1 c1(C(=O)NCC(CNC(C(CC)O)=O)O)cncc(NC(=O)CC)c1 C1(C)(CC(=O)N(C)CCOCC2CC2)CCN(C(=O)CCC(N)=O)CC1 Cc1cccc(C(C)NC(=O)C(O)CNC(C2(Cl)CC2)=O)n1 C1(OC)CCCCC1C(=O)NC(Cn1ccnn1)C(=O)NCCCO CON1CC(C(N2CC(C)(C(=O)NC3(CCO)CCCC3)C2)=O)CC1=O N(C(=NCCC1(N(C)C)CCCCC1)NCF)C(C)C1CC1.c12nc(n[nH]1)C2 c1(CC(C)NC(=O)C(C)(C)CO)ccc(CNC(c2cccnc2CN)=O)cc1 c1(NC)ccc(C)cc1C(=O)NC(C1CC1C(=O)Nc1cnc(C)nc1)C C(C)(C(C)CCC)NC(CCN(C(CCC)=O)CC1CC1)=O c1(C(N(C(C)CNC(c2cccnc2)=O)CC)=O)cnc(N(C)C)o1 c1(OC(C)C(=O)NCC2CC(NC(=O)C=C3CCCCC3)C2)cccc(F)c1 N1(C(C2(C3N(C(C4OCCC(C)C4)=O)CCC3)CC2)=O)CCC2(CCC2)CC1 C1(C(=O)NCC(CNC(Cc2nc(C)oc2)=O)F)CCc2c(n[nH]c2C)C1 CCCC(C(=O)NCC(C)N(C)C(c1ccccc1N(S(C)(=O)=O)C)=O)N(C)C C1(CC=C)(C(N2CCCC(C(C)NC(=O)CS(=O)(=O)NCC)C2)=O)CCOCC1 C(=O)(C1(C)CCc2ccccc21)N1C(CNC(CN(C(C)=O)C)=O)C(C)(C)CCC1 N1(C(C2CC(CC)OCC2)=O)CCCC(O)(CNC(c2nc(C)oc2C)=O)CC1 N1(C(c2nc(C)c(C)s2)=O)CCCc2ccc(OC(F)F)cc2C1 c1(CC)c[nH]c2ccc(C(=O)OC)cc12.c12cnccc1CN1C(CC1)C(=O)N2 C1(CC(=O)NCCCN(CCC)C(c2cnc[nH]2)=O)CCCC1C c1(C(=O)NC2(CC(=O)NC(CC)C(C)C)CC2)ccncc1N Cn1cc2c(n1)CC(C(N1CC(NC(=O)COC3CC3)C3(CC3)C1)=O)NC2=O CCC(C)CCCCC(=O)NCC(C1CC1)NC(c1cc(C)oc1C)=O c1(OC)ccc(C(C(=O)NCC(F)F)N2CCC2C(C)C)c(Br)c1O C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NCCC(CNC(c1c(C)n(C)nn1)=O)O N1(C(CC(C)F)=O)CC2(NC(c3ccc(=O)n(C)c3)=O)CCC1C2 C(=O)(C1CCCn2ncnc21)N1CC(C(C)NC(C2CC3(C2)CC(O)C3)=O)C1 C1(CNC(=O)Cc2cncnc2)CC2(CCN(C(c3cnccc3Cl)=O)C2)CO1 c1(C(N(CCCNC(c2ncoc2C2CC2)=O)CC)=O)cnn2c1NCC(C)C2 c1(C(=O)NC(C(C)(C)C)CNC(c2ccccn2)=O)n[nH]c2c1CS(=O)(=O)CC2 C1(CNC(CC2C(C)CCC2)=O)COCCN(C(c2ncc(C(F)F)s2)=O)C1 N1(CC)CC(C(=O)NC2C=CCN(C(=O)CN3CCS(=O)CC3)C2)CCC1=O N(C1CCOc2c(Br)cccc21)C(=O)Nc1cc(NC(=O)OCC)c(C)cc1 N1(C(CC2CC(=O)N2)=O)CCc2cc(NC(C3CC(O)C3)=O)ccc21 O(P(=O)(COCC)C(C)(c1ccccc1)NC(=O)NCCc1ccccc1)CC c1(CC)oc(C(=O)NCC2C3CC=CCC23)cc1C C1(CC=C)(NC(c2ccc(CF)cc2)=O)CCN(C(C2C=CCCC2)=O)C1 c1(C(N2CCC(N(C(=O)C(C)(C)O)C)C2)=O)ccc2c(c1)S(=O)(=O)NC=N2 CC(C)(C)C(O)C(=O)NCC1(NC(=O)CSCCN(C)C)CCCCC1 N1(C(C(C)(C)OC)=O)CCCC(NC(c2cc(C)nn2C)=O)C1 C(=O)(C#CC1(C)CC1)NC1CCC(NC(c2c(OCC(C)C)nccc2)=O)CC1 c1(C(=O)NCC(CCCC)NC(=O)C(O)CCN(C)C)cc(N)ccc1CC Cn1ccc(=O)c(C(N2CC(NC(=O)CNC(=O)CN(C)C)C3CC23)=O)c1 c1(CC(=O)NC2CNOC2)ccc(Cl)nc1 C1(CNC(C(CC)OC)=O)Cc2ccccc2CN1C(=O)COC1CCCOC1 c1(C(=O)OC)cc(NC2(CO)CN(C(=O)C(C)NC(C3CCC3)=O)C2)oc1C N1(C(Cc2c(C)con2)=O)CCC(CNC(=O)C(C)C(C)C)C12CCC2 C=CC(C(=O)N(C(C)CC(=O)Nc1ccccc1)C)c1ccccc1.C1(=O)CO1 c1(CC)conc1C(=O)NCC(C)(CC)NC(c1sccc1C(C)=O)=O C=CCCC(C)(C)C(=O)NC1CCCC1CNC(=O)CCCC(=C)C N1(CCn2c(C)cc(C)n2)C2CCC1CN(C(C1CCOC1)=O)CC2 C1(N2CCN(c3c(C)nccc3)CC2)CCCCN(C(C2CCC(C)C2)=O)C1 C1(C)(C(N2CC(NC(c3n(CC)c(O)nc3)=O)C(O)C2)=O)CCCCC1(F)F C1(NC(CCS(C)=O)=O)CN(C(c2cc(C(F)F)cs2)=O)CCC1(C)C N1(C(CSCC)=O)CC2CCOC2(CNC(c2cn(C)nc2-c2ccoc2)=O)C1 C(=O)(C(C)(C)CN(C)C)NCC1(OC)CN(C(c2cc(Cl)n[nH]2)=O)C1.C(C)(C)(C)O C1(c2ccn(CC)n2)CC12CCN(C(=O)COC(C)CC(C)C)CC2 Cc1ccoc1CNC(=O)N(CC(C)C(C)C)C C1(CCC)CCC(F)(C(=O)NCCN(C(=O)CNC(=O)CN(C)C)CCOC)C1 c1(OC)ccc(C(F)(F)C(=O)NCC2CCCN2C(C2(O)CCCC2)=O)cn1 C(=O)(C(O)C(F)(F)F)N(CC(CNC(c1n[nH]c(C)c1Br)=O)C)C C(CSC1CC1)(C(C)C)NC(=O)NC(CC)C N1(C(=O)Cc2ccc(Cl)nc2)CCN(C(C23CCCC2CC3)=O)CC12CC2 c1(CNC(=O)NCC(=O)NCCC2(NC(c3cscc3F)=O)CC2)ccncc1 CC(CC(=O)NC1CC(CO)C1)C(C)(C)NC(C1CC1(F)Cl)=O N1(C(CC(=C=C)C)=O)CCCCCC(NC(=O)Cc2nnc3n2CCOC3)C1 c1(C(=O)OC)ccnc(Cl)c1OC.C12CCCC(C1)N2C(C1(SCC)CC1)=O C(=O)(C#CC1CCOC1)N(CCCC(=O)NC1CC2(CCCC2)C1)C C1(CC)CN(C(=O)C(=O)C2CCCC2)CCC1NC(c1ccc(=O)n(C2CC2)c1)=O c1(C(N2CCC(NC(c3c(OC)cccc3)=O)C2)=O)cc2cccnc2s1 N1(C(CCC(C)SC)=O)CCN(c2cc(CC3CC3)ncn2)CC(C)(F)C1 c1(C(N2CC(NC(C=C)=O)C(C)C2)=O)nc(Cl)ccc1F CC1(C)CC(NC(C2CC(CF)C2)=O)CN1C(=O)CCc1ncc[nH]1 N1(C(C(C2(O)CCC2)NC(c2cn(CC=C)nc2)=O)=O)CCN(CCO)C(C)C1 N1(C(C(COC)N(C)C)=O)CCOCC(CNC(=O)CCc2cc(C)on2)C1 C1(NC(c2ccc(CC)s2)=O)CCN(C(c2ccc(N)cc2C)=O)C(C)C1 N1(C(CC=CCC)=O)CCC(C(C)(C)NC(=O)Cc2cc(C3CCCC3)[nH]n2)C1 C1(CC)CCC(C(=O)NCC2(OC)CCN(C(=O)C(C(C)C)C3CCC3)C2)CC1 C12(C(=O)NCCOCCCNC(c3c(C)[nH]cc3)=O)CC1COC2(C)C C(C)(C)(C(=O)N1CC(O)(CC)C1)OCC N1(C(c2cn(CCC)nc2C)=O)CCN(C(=O)C(O)COC)C(C)C1 c1(C(=O)NCCn2cc(CCN(C(=O)C(O)c3cnc[nH]3)C)nn2)c(Cl)cnn1C CN(CC1CCN(S(C)(=O)=O)CC1)N1CCOC(c2ccc(C#N)cc2)C1 c1(SCCC=C)ccc(C(=O)NCC(C)(O)CNC(=O)C(C)O)cc1 N1(C(C2(SC)CCC2)=O)CCC(CCNC(=O)Cc2csc(Br)n2)C1 C1(NC(C2(C)CCOCC2)c2n(CC=C)nnn2)CCS(=O)(=O)CC1 N1(C(c2c(C)nco2)=O)CCOCCC1C(N1CCC(CO)C(C)C1)=O C1(NC(C(C2CCC2)NC(C(C)NC(CC)=O)=O)=O)CNC(=O)C1(C)C C1(C(=O)NC(CC)COC)(CNC(=O)CSC(C)(C)C)CC2(CC2)C1 C(=O)(CC1=CCN(C(c2cnc(C3CC3)o2)=O)CC1)NC(c1nc(C)[nH]n1)CO c1(OC)cc(CNCc2cc(Br)c(C)cc2O)ccc1S(C)(=O)=O CC(C)(C(=O)NCC(C)(C)C#CC(=O)NC1(C(C)(F)F)CC1)C(F)(F)F c1(C(=O)NCCCNC(C(C)N2CCCC2)=O)nc(=O)n(C)[nH]1 C1(OC)CNCCC1CNC(c1cnc(N2CCNCC2)s1)=O C(=O)(C1=CC2CCC1C2)N1CC(NC(c2ccc(C(N)=O)[nH]2)=O)C1 c1(C(=O)NCC2N(CC(=O)NC3CCC4CC34)CCCC2)cccn2cncc12 CN1CCN(c2ncc(Cl)c(O)n2)C(CNC(C2CCCS(=O)(=O)C2)=O)C1 c1(C(N(CCNC(CN2C(C)CCC2C)=O)C)=O)cc(Cl)c(F)cc1F C1(C(N2C(C)(CC)CC2)=O)CN(C(C2COCC(C)O2)=O)CCC1O c1(C(N2CC(NC(c3ccoc3)=O)CC(C)C2)=O)n[nH]c2ccc(C(F)(F)F)cc12 C(=O)(C1CCc2ccc(Cl)nc21)N1CCC(CNC(c2ncc(F)cc2F)=O)C1 c1(SCC(N2CCC(CNC(c3cscn3)=O)CC2)=O)ccc2c(c1)CCC2 C(=O)(CCCCCC#N)NC(CNC(COc1c(C)ccc(Cl)c1)=O)C C1(C)(CNC(c2nc(CC)oc2)=O)CCCN1C(=O)C(CO)NC(=O)C(F)(F)F N1(C(c2sc(CC)c(C)c2)=O)CCOC(C)(CNC(=O)Cc2ccc(C)nc2)C1 Cc1cc(C(=O)NCC2CC(CNC(=O)CNc3ccccc3)C2)c(Cl)cc1N c1(C(=O)NC2(CO)CCN(C(C3N(CC)CC3)=O)C2)cc(=O)c(Br)c[nH]1 CCC(CC)(CC)C(=O)NC1CCN(C(=O)C=C(C)C(F)F)CCC1CO C1(NC(C=CC(=O)OCC)=O)CC2CCC(C1)N2C(C1C2CCCOC12)=O C(=O)(C(O)CCC(C)C)NCC12C(CN(C(c3c(C)cn(C)n3)=O)C1)CC2 c1(OC)ccc(C=CC(=O)N(CC(C)(C)CNC(=O)C(C)CS(C)=O)C)nc1 c1(C(=O)NCC(CC=C)NC(c2cnc(N(C)C)cn2)=O)cc2cccn2cn1 C1(OC2CCOC2C(=O)NCCOC2(CCCC)CC2)COC2(C1)CN(COCC)C2 C(=O)(CC(C)C(F)(F)F)NCCC1N(C(Cc2c(C)cccn2)=O)CCOC1 C(=O)(CCCCC(=O)c1cccc(OC(F)(F)F)c1)NC1(C)CCOC1=O C1(NC(C2C(C)C2)=O)CC2(CCN(C(=O)Cc3cc(Cl)cc4c3OCC4)CC2)C1 CC1OCCN(C(C2CCN(C3COC3)C2)=O)C1C(N1CCCNC(=O)C1)=O N1(c2ncnc3[nH]cc(CC)c32)CCCC12CCN(C(=O)CSCCN(C)C)C2 C1(C(N(C2CCN(C(CC(=C)Br)=O)CC2)CCC)=O)CCn2c(O)nnc2C1 N1(C(C2(CC)CC2(F)F)=O)CCC2CCC(NC(C3CCCCCC3)=O)C1C2 c1(C(N(C2CCCN(C(=O)CCS(=O)(=O)NC)C2)CC)=O)csc2nccn12 C=CC1(CC(=O)NCc2ccc(Cl)o2)CN(C(c2cccnc2OC)=O)C1 c1(C(N2CCC(CCNC(C3CN(CC)C(=O)C3)=O)CC2)=O)cc2c[nH]nc2s1 C(C(C(=O)N1CC=CCO1)NC(=O)CC#N)N(C)C c1(C(=O)OC)nn(C)cc1-c1cn(C2CC(NC(c3cnsn3)=O)C2)nn1 N1(C(c2c(CC)nccn2)=O)CCC(C(=O)NC(C)CN2CCOCC2)=C(F)C1 c1(C(=O)NC(C)CF)ccccc1N1CCCS1(=O)=O N1(C(c2cc(CC)on2)=O)CCN(C(c2csc3cncn23)=O)C(CCOC)C1 c1(NC(C2(C)CCN(CCCCCC)C2)=O)ccc(OC)cc1C c1(C(=O)NC(C2CCN(C(C3CCS3(=O)=O)=O)C2)(C)C)ccc2oc(=N)[nH]c2c1 C1(OC)CC(CO)N(C(=O)C=Cc2ccc(Br)o2)C1.c1(C(=O)N)nocc1C CC(C)CC(C(=O)NCCC(N1CCCC1C1(C)CC1)=O)C(C)C c1(OC)c(C(N2CCC(CNC(=O)CC3CCCCC3)C2)=O)oc2ccccc12 N1(C(CCCOCCOC)=O)CC2CCCC2C1C(=O)NCC(C)O c1(C(N2CCC(C(=O)NCCCC)C2)C(=O)NC2(C)CC2)cc(Cl)c(F)c(Cl)c1 C(CC(C)(C)C)(C(=O)NCCC1CC(NC(c2ccnc(OC)c2F)=O)C1)OC N1(C(c2cc(OCC)no2)=O)CCCC2(NC(=O)C(C)(C)CC)CCCC12 c1(C(=O)NC2CN(C(C3C(C)(C)C3)=O)CC2N=[N+]=[N-])cc2c(s1)CCCCCC2 C(C)(CCC(=O)NCc1ccc(C(N2CCC(C3(C)N=N3)C2)=O)o1)OC c1(C(=O)NCC2(C)N(C(C3CC(C)N(C)CC3)=O)CCC2)ccc2c(c1)CCN2 c1(N(CCOCCCOC)C)nc(NC2CCCC2C)nc2c1CCC2 Cn1ncc2c(C(=O)NCC(C3CCCC3)NC(C3(O)CCSC3)=O)ncnc12 N1(C(C(C=C)CC)=O)CC(C)(C)CC1CO.C(=O)(CC)NC(CCC)C1CC1 C1(OC)CCN(C(C2CCCN2C(C2(O)CCOCC2)=O)=O)C1C(C)C Cn1cc(C(N2CC(CCNC(=O)C(C)(C)C(N)=O)C2)=O)c(=O)c(Br)c1 Cc1ccc(C(N2CCN(C(C3CC3F)=O)CC2c2cccnc2)=O)c(=O)n1C C1(c2nnnn2C2CCC2)(NCc2cc(C)nc(Cl)c2)CC2CCC(C1)O2 CC(C)CS(=O)(=O)CC(=O)NC1CCN(C(C2CCCS2(=O)=O)=O)C1 N1(C(=O)CC2CCCCC2O)CC2CC(C1)N(C(c1cnc3[nH]ncc3c1)=O)C2 C1(C(=O)OC)CCN(CCO)C(=O)C1.N12CC(C1)N(C)CC=CC2=O c1(OCC)ccc(CC(C)C(=O)NCC(C)(C)NC(C2CCC2(C)C)=O)cc1 c1(NC(C2CCN(C(C3OCCC(NC)C3)=O)CC2)=O)ccc2occc2c1 N1(C(=O)OC(C)(C)C)CCCC(O)(C(F)(F)C(=O)NCC2CCCN2C2CC2)C1 c1(C(=O)NC2(C3N(C(CC(C)C)=O)CCCC3)CC2)cccc2nncn12 CCC(C(=O)NCCN(C(c1csc(Cl)c1OC)=O)C(C)C)C(C)C c1(CC2CN(C(C3CC(C(F)(F)F)C3)=O)C2)ccccc1[N+](=O)[O-] N1(CCNC(C(C)CC2CCCCC2)=O)C(=O)CNC1=O c1(C(=O)NC(CN(C(C(CC)c2cccnc2)=O)C)C)noc(C)c1C(=O)OC CC1=C(C(=O)N(C2CCN(C(C3CC(O)C3)=O)C2)CCO)CCCO1 C(=O)(C(F)CC(CC)CC)N(CCN(C(C(C1CCCC1)OCC)=O)C)C C=CCCCCC(=O)NC1COCC1C(=O)NC1CCC=CCCC1 c1(CCC(=O)NC(CC)(CNC(=O)CCC(C)SC)CC)cnc2n1CCCC2 c12cc(nn1C)S2.N1(C(COC)=O)CC(=Cc2cccs2)CC1=O C1(C(N2C(CC)(CO)CCC2)=O)CC(N(C)C)CN(C(=O)Sc2ccccc2)C1 C1(CC)CC(CC(=O)NC2CCCC2NC(=O)C=CCO)CCO1 C1(C(=O)NCC#CCNC(CNC(=O)NC)=O)CC(C(C)=O)C1(C)C C(=O)(C1CCc2cc(Cl)ccc21)NCC1C2CN(C(C(CCCCC)O)=O)C1C2 C(C1CCc2ncnn21)N1C(CNC(c2cn3c(n2)CCC3)=O)CCC1 C1(F)(CNC(C2N(CC)CC2)=O)CC(CNC(c2c[nH]c(Br)c2)=O)C1 c1(OCC)ccc(-c2nc(C(c3cnccc3C)C)n(Cc3ccsc3)n2)cc1 c1(C(N2CCCC(COC)(NC(=O)CC(C)F)C2)=O)cnn2cccc2c1 CC1CCN(C(=O)CN2CC(F)(F)C2)CC1CNC(=O)C=CCC1CCCCC1 CC(N=c1nc(-c2ccccc2)nc(N(C)Cc2cccnn2)[nH]1)c1ccoc1 N1(C(c2n(C)c(O)nc2)=O)CC2(C1)CN(C(=O)CCCCO)C2 C1(C(N(C2CCOC2)OC(=N)O)=O)CCCN(CC2CCN(CC(N)=O)CC2)C1 c1(C(N2C(C)CC(C(=O)NC(c3ccncc3)C)CC2)=O)ccc2cc[nH]c2c1 c1(NC23CC(C(=O)OC)C(C2)C3)ccc(C(C)(C)C)cc1Br C(C(C)C(C)C(=O)NC1CCC(CNC(C2(CF)COC2)=O)CC1)OC N1(C(CSC(C)=O)=O)CCC2C1CCCN2C(=O)C(O)CC c1(C(C(=O)NCC2CCN(C(C=CC(C)C)=O)C2)O)ccc(O)c([N+](=O)[O-])c1 c1(C(CC)C)nc(C)cc(=NC2C3CC2CN(C(c2ccc(F)c(Cl)n2)=O)C3)[nH]1 Cc1cnc(O)c(NC(C2CCC3(CC3)N2C(=O)CN(C)C2CC2)=O)c1 Cc1cc(F)cnc1C(N1CCC(C)C(CNC(C2CC(F)(F)C2)=O)C1)=O C=CC(C)(C)C(=O)N(C)CC1CCN(C(=O)C(C)c2ncco2)C1 N1(C(C(CCCC)O)=O)C2CCC1C(F)C(NC(c1nccnc1N)=O)C2 N1(C(CCC#C)=O)CCCC(C(=O)NCC(=O)NC(C(=O)N(CC)CC)C(C)C)C1 C1(Cl)(C(=O)NCC(C)(C)CNC(C2CN(CC(F)(F)F)C2)=O)CC12CCOCC2 N1(C(c2c(C)oc(C(C)(C)C)c2)=O)C2CCC1CC(NC(c1n[nH]cc1Cl)=O)C2 C#CCC(C)C(=O)NCCc1ccc(NC(c2cscc2C)=O)cc1 Cc1ccc(-n2ncc(-c3nc(CCN)no3)c2C)cc1 N1(C(C=Cc2c(C)ccs2)=O)CCN(C(C2CCCN2C)=O)CC2(CC2)C1 c1(C(N2C(CN(C(=O)C(F)n3cccn3)CC)CCC2)=O)cc(F)cc(N)c1F C1(NC(c2n(C=C)nnc2)=O)CN(C(c2cnoc2CC)=O)C2CCCC12 C1(NC(C(CC)n2cccn2)=O)C(C)CCN(C(=O)Cc2ccc(C)nc2Cl)C1C C1(C(N(C2(C(=O)NC3CCC(C)C3)CCC2)C2CC2)=O)CCN(C)C1=O C1(NC(=O)C(=Cc2cccnc2)F)CC(O)CN(C(c2c[nH]nc2F)=O)C1 c1(C(=O)NC2C(NC(C(C)OC)=O)CCCC2)cc(F)c(Cl)cc1Cl c1(C(N2CCN(C(c3cnc(C)s3)=O)C(CO)C2)=O)cccc([N+](=O)[O-])c1Br c1(OC)cc(CCNC(C2(C)CN(Cc3ccccc3)C2)=O)cc(Cl)c1 C(C(C)(CO)NC(=O)C(C)CC1CCC1)NC(COCCCN(C)C)=O C(=O)(C(O)C(F)F)NC(C1CCN(C(c2cccc(N)n2)=O)C1)(C)C Cc1ccnc2c(N3CCN(C=O)CC3)cnn12.C12CC3CC1C2C3 C12(C(=O)NC3(CC)CC(C)(C)C3)C(NC(c3ccc(C)cc3C)=O)C3CC1C2C3 C1(C(=O)NCCC2(OC)CCCCC2)CCC2(CN(C(C3CCC(=O)O3)=O)C2)O1 c1(CNC(C(=O)NC(C)C)=O)nnc2n1CCN(C(=O)CNS(=O)(=O)N(C)C)C2 c1(OC)cc(=O)n(C)cc1C(=O)NCCCN(C(=O)C(F)CC1CC1)C c1(C(N2CCC(NC(c3c(CC)n(C)nc3)=O)CC2)=O)c(F)ccc(Br)c1C c1(CCCN2C(C)(c3cccc(OC)c3)CC(CN)C2)cc(C#N)ccc1C C1(C(=O)NC2C(C)(C)CN(C(C3CC3(F)F)=O)C2)CNC(=O)CC12CCOC2 c1(C(=O)NC2CCCC2NC(C2CC(n3ccnn3)C2)=O)coc2c1COC2 C1(F)(CNC(C2(C#C)CC2)=O)CCCN(C(=O)CCC(=O)Nc2nccs2)C1 CC1CCn2c(C(=O)NC3CN(C(c4ccccc4CO)=O)CC3O)cnc2C1 Cc1cn2c(n1)C(C)CC(C(N1CCN(C(c3c[nH]nc3F)=O)CC1C)=O)C2 C1(C(=O)NCC2C(C)C2C)CC2CC1CN(C(=O)C#CC1CCC1)C2 C1(C(NOCCC)=O)CCC(CNC(=O)C=CC2CCOC2)O1 N1(C(C(C)=CCC)=O)CCCC(CC(=O)NCCCC(F)(F)F)CC1 Cc1noc(CCNC(C2(C)CC2)=O)n1.C1(C(=O)N)COCC1C(N)=O C(=O)(C1COc2ccc(F)cc21)NCC1(O)CN(C(CCc2nc(=N)[nH][nH]2)=O)C1 c1(COC)n[nH]c(=NCCCC(C)NC(=O)C(c2cccc(Cl)c2Cl)O)s1 c1(CC(=O)NC(C(=O)NCCC=CC)CC2CCCC2)ccc(F)nc1 N1(C(COCC(=O)NC2CCOCC2)=O)CC(C)(COCCSC)CC1(C)C CC1CN(C(c2cn(CCN(C)C)nn2)=O)CCN1C(C1CCN1C1CCCC1)=O C12(NC(c3c(C)con3)=O)CCCC1N(C(c1cc(Cl)sc1Cl)=O)CC2 CC(C)CC(C(=O)NCCc1cnnn1C)ONC(C1(C)CC=CCC1)=O N1(C(CCN(C)CC)=O)CC(NC(c2ccc(N3CCCC3=O)cc2)=O)CC1C C(=O)(C(C(=O)NC1CC(C)(NC(c2ccc(C)cn2)=O)C1)OC)OCC N1(C(c2cn(CCC(F)(F)Cl)nn2)C)CCOC(C)(CO)C1 c1(C(=O)NC(C2C=CCC2)=O)ccc(CCN(C(c2n[nH]cc2Cl)=O)C2CC2)cc1 C1(OC)CN(C(=O)Cc2cn[nH]c2)CC1NC(c1c(C(F)(F)F)cnn1C)=O Cc1cccc(C(=O)NCCC(=O)NCCC(O)C2CC2)c1 N1(C(c2cc(SC)oc2C)=O)CC=C(CNC(c2cncc(C(N)=O)n2)=O)CC1 C(=O)(CCS(N)(=O)=O)NCCN(C(=O)C=CSC)CC N1(C(C(C(C)C)SCC)=O)CC(CO)C2(C1)CN(C(c1nn(C)c(C)c1Cl)=O)C2 C#Cc1cncc(C(=O)NC2CCCCC2NC(=O)CCc2nc(C)c(C)[nH]2)c1 C1(CCNC(C(C)NC(COC)=O)=O)CCCCN1C(c1cc(C)c[nH]1)=O C(=O)(C(F)(F)C(C)(C)O)N1CC(C(=O)NC(C)C(C)(C)CO)CC(C)C1 Cc1cc(C(=O)NC2CC3CC(C2)N(C(=O)C(=O)NC2CC2)C3)ccc1C#N C1(CNC(C2(c3c(C)ccc(C)c3)CC2)=O)CC2COCC2N1C(=O)C(C)C#N c1(C(C)C)nc(Cl)cc(=NC2CCC(NC(=O)CC3CCCC(=O)N3)CC2)[nH]1 C1(NC(CC2C3CN(C(C(CC#C)C4CC4)=O)CC32)=O)CC2(CCCO2)C1 N1(C(c2cccc(SC)c2)=O)CC2CCC(C1)N2Cc1ccnc(F)c1 Cc1cc(C#N)ccc1C(N1CC(C)(CNC(=O)CCCCN(C)C)C1)=O CC(C)(F)C(C)(F)C(=O)N1CC(NC(C23CC(CC(F)F)(C2)C3)=O)CC(O)C1 c1(C(N)=O)ccccc1CCC(=O)NCCCC1CCCN1C(=O)CC N1(C(C2N(C(C)C)CCC2)=O)C(CC(=O)NCCCC(F)F)C2CCCC12 c1(CC(C(=O)NC(CCC=C)C(=O)O)(C)C)cc(OC)c(OC)cc1OC c1(C(N2CCN(C3CN(C(CS(CC)=O)=O)C3)CC2)=O)cc2c(s1)CN(C)CC2 N1(C(CNC(C)=O)=O)CC2(CCC2NC(=O)C(c2ccc(F)cc2)F)C1 C1CC(O)C(=O)N2CC(C2)NC(=O)C2(CC2)NC(=O)N1.N1(C(C)(C)C)CCCC1 c1(C(=O)NC(C)CCNC(=O)CNS(N)(=O)=O)cncc(Cl)c1Cl c1(C(=O)NCC(CO)NC(CCC(CC)C)=O)sc2ncccc2c1N N1(C(c2ccc(OCCN(C)C)c(F)c2)C(=O)NC)CCC(P(C)(C)=O)C1 C(N=c1[nH]c(Cl)ncc1F)c1ccc(CNC(C(C(C)C)F)=O)cc1 C1(c2nc(NCC3(C)CC=CCC3)[nH]n2)CCCN(C(C2CC(CC)C2)=O)C1 c1(CCC(=O)NC2CN(CCn3cc(CO)nn3)CC2F)ccc2c(c1)CCO2 C(=O)(CC(C)(C)CC(F)F)NC(C1(O)CCN(C(C2CC2C(C)(F)F)=O)CC1)C c1(C(=O)NC(CNC(C(C)c2ncco2)=O)C)sccc1Cl C(=O)(C(CCOC)NC(c1cnc(C)o1)=O)N(CC(C(=O)NC)O)C C1(C(=O)NCC2CCCS2)CCN(C(=O)CCOCC2CC2)C1 C1(NC2(c3n(C4(C)CC4)nnn3)CC(NC(C)(C)C)C2)CCCC(C2CC2)C1 Cc1ccc(CCC(=O)NC(C2CCCC2)CNC(=O)CC2(C(F)(F)F)CC2)s1 N1(C(C(C)C)=O)CCC2(CC1)CC(NC(C1CC1(C)C(C)C)=O)CCO2 C1(O)(C(=O)NCC=CCNC(Cc2c(CC)noc2CC)=O)CCCC(C)CC1 c1(C(=O)NCCC2N(C(C=CSC)=O)CCC2)ccc(Br)c(C)n1 C(CC(C(=O)NCc1cccc(Cl)n1)NC(c1cc(C2CC2)no1)=O)SC C(=O)(C(F)CC(C)(C)NC(c1cn(C)cn1)=O)N(C1CCCN1C1CC1)C N1(c2c(C)cccc2)C(=S)NC(c2csc(C#N)c2)C2=C1CCNC2=O C1(N(C(=O)NC(c2nccn2C)C)C2CC2)CCc2nc[nH]c2C1 CN1CCC(NC(=O)C(C2CCNCC2)O)C1c1cccnc1 c1(-c2n(CCN(C)C)nc(C3CC3(C)C)n2)cc2c(C(F)(F)F)nn(C)c2s1 c1(C(=O)NCC2N(C(c3c(CC)occ3C)=O)CCC2)ncnc2c1CCC2 c1(C(N(C(C)C(N2CC(C)(C#N)C2)=O)CC)=O)ccnc2cc[nH]c12 NS(=O)(=O)c1cc(C(=O)NCC2C=CCN2C(=O)Cc2cc[nH]c(=N)c2)co1 N1(C(C(C2CN(C(c3cnn(CCF)c3)=O)C2)OC)=O)CCCC(CCO)CC1 c1(C(C(=O)NC(CNC(C=CC=CCC)=O)C)O)cccc(C)n1 c1(C(N2CCCCC2)C(=O)NC(CN2CCC(C)(CN)C2)=O)cc(O)ccc1Cl C1(NC(CSCC=C)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CC1CO Cc1nc(C(N2CCC(NC(=O)Cn3cc(C#N)cn3)C(CO)C2)=O)c(C)n1C C(=O)(C1CCCn2nccc21)N1CCN(C(COc2ccc(C)cc2F)=O)CC1 N1(C(C(C)(C)O)=O)CC2CC1CN2CC1CCCS(=O)(=O)C1 C1(NC(CN(c2ncccn2)C)=O)CCCCN(C(c2cccc(F)c2Cl)=O)C1 c1(C(N2CCC3(CC2)CSC3)C(=O)NCCOCC)cc2nc(Cl)ccc2s1 N1(C(c2cc(OC)nc(Cl)c2)=O)CC2CCN(C(C3C(C)(C)OC3(C)C)=O)C2C1 C[Si](C)(C)C1(CNC(=O)NC(C2(CC3CCCO3)SCC2)C2CC2)CC1 C1(CNC(C2N(C(N)=O)CCC2)=O)CCN(C(C2(CCO)CC2)=O)CCC1(F)F c1(C(=O)NC23CC(CNC(c4nc(CO)sc4)=O)(C2)C3)ccc2sncc2c1 c1(C(=O)NC2CCC(N(C)C(C3CC3(F)F)=O)CC2)cc2ccnc(Cl)c2[nH]1 c1(CC(=O)NCC(C2CCCCC2)NC(C2C(OCC)C2C)=O)ncc(C)[nH]1 c1(N2CC3C(C(N4Cc5c(nn(C)c5N)C4)=O)C3C2)ncnc2c(F)cccc12 c1(C(N2C(CNC(=O)C3CC3)CCC2)=O)cccc(C2(O)COC2)c1 c1(C(=O)NC2C(CC)CN(C(=O)C(F)=CC3CC3)CC2)cn(C)c2ccccc12 Cc1noc(C)c1CCNC(=O)C(CN(C)C)NC(=O)C(C)(C)C1CCC1 C1(C(=O)NCC2N(C(c3cc(C)sc3)=O)CCC2)CCCCCS1(=O)=O N1(C(c2c(C)cco2)=O)CCC2(NC(c3cccc(OC(F)F)n3)=O)CCCC12 N1(C(c2cc(=N)[nH]cc2)=O)CCC(CNC(c2scnc2Cl)=O)C12CC2 N1(C(CNC(c2c(C)c(C)cc(C)c2C)=O)=O)CCCC2(CC1)CNC(=O)O2 N1(C(c2c(C)cc(=N)[nH]c2)=O)CC(C)CN(C(=O)CC23COCC(C2)C3)C(C)C1 C1(C(=O)NC(C)(CNC(=O)CCC(F)F)C2CC2)CC2CCC1CC2 C(CCS(C)(=O)=O)NC(CC(C1CC1)NC(Cc1cc(C)sc1)=O)=O Cc1oc(C2CC2)cc1C(=O)NCC1CCCC(NC(=O)Cn2cc(Cl)cn2)C1 C1(CNC(CCCOCC=C)=O)C(CC)CCN1C(c1ncncc1N)=O C(CCC)(C(=O)N1CCC(NC(=O)CN2CC3CC3C2)C1)=CCC CN1CCN(C(c2ccc(C(F)F)nc2O)=O)CC1CNC(c1ccoc1Br)=O C(CO)(C(F)(F)F)NC(C(CC1CCOCC1)NC(c1cc(=N)[nH][nH]1)=O)=O C1(N(C(c2c(CC)ocn2)=O)C)CCCN(C(=O)Cc2ccccc2O)CC1 C(=O)(CC(F)(F)C(F)F)NC(CC(C)NC(C=C(C)Cl)=O)C CCCC(C(=O)NCc1ccnc(C(=O)Nc2cccc(CC)c2)c1)C(C)C N(C1CCCn2ncnc21)C(c1cc(CNC(C2SCCS2)=O)cs1)=O c1(C(=O)NC2CCN(C(=O)CC3=CCCC3)CC2O)ccc2[nH]nc(O)c2c1 CC(CC(F)(F)F)N(C(=O)CCC1CC(NC(=O)CCc2cscn2)C1)C Cc1[nH]c(=N)nc(O)c1CC(N1CCC(NC(c2cc(Br)no2)=O)C12CC2)=O C1(C(=O)NCC=CCNC(=O)CCC2CCC(O)CC2)CC2(C1)CC2(F)F c1(C(=O)NCC2(C(=O)NC(C3(OC)CCC3)C)CCCC2)cc(C#N)n(C)n1 C1(=CC(=O)NCC(C)NC(c2ccc3c(c2)OCC3)=O)CCCCCC1(F)F c1(C(=O)NCCC(C)NC(CCSCC)=O)ccc(OC(C)=O)cc1Cl c1(CC(=O)NCC2CCN(C(c3n(CCC)ccc3)=O)C2)ccc(Cl)nc1 C(=O)(C(O)C1=CCCCC1)NCC1N(C(C(C=C)(F)F)=O)C2C(C1)C2 S(=O)(=O)(CCC(=O)c1c[nH]nn1)N1C(CN(C)C(=O)Nc2ccccc2)CCC1 N1(C(C2(OC)CCOC2)=O)CC2(C1)CN(C(c1ccnnc1)=O)C2 N1(C(c2cn(CCC)nn2)=O)CC(CNC(c2cncn2C)=O)CCC1C N1(C(C2ON=C(CC)C2)=O)CCc2ccc(C(=O)NCCC(C)(O)CC)nc2C1 C(=O)(C1=CCCN(C(c2cnc(C(C)C)o2)=O)C1)N1CCC(SC)C1 C(C)(C(C)C(=O)N1CCN(C(C)C)CC1)NC(c1cnc(CC)s1)=O S(=O)(=O)(CCCN=c1[nH]c2c(c(=NCCS(=O)(=O)N(C)C)[nH]1)COC2)NC C1(C(=O)NC2CC(CCNC(c3cc(C)n(C(F)F)n3)=O)C2)CC(S(N)(=O)=O)C1 c1(C(=O)NCCC(C(C)C)NC(=O)CCCC(N)=O)cc(F)cc2ccncc12 N1(C(c2ccc(OC)nc2C)=O)CCC2CN(C(=O)C(C)O)CCC12 c1(C(=O)NC2CCN(C(C(CC)CC(C)C)=O)C2)cccc2cccc(C)c12 c1(CN(C(CCN(C(c2nc(C)sc2)=O)C)=O)C)cccc(O)n1 C1(C(N(CCNC(C2CCN(C(C)=O)C2)=O)CC)=O)CN(C)C(=O)N1 N1(S(CCNS(CC)(=O)=O)(=O)=O)CCN(C(C2CCCC2(C)C)=O)C(C)C1 N1(Cc2scc(CC)n2)C2CCC1CC(NC(=O)COC1CCCC(C)C1)C2 c1(N(CC(C2CC2)OC)C)cc(=NCCC(=O)OC)[nH]cn1 C(=O)(C1=CCCN(Cc2cc(F)c(O)cc2F)C1)Nc1cc(OC)cc(Br)n1 C1(C)(C(=O)NC(CCC)c2nn[nH]n2)C=CCN1C(c1cnc(C2CC2)o1)=O c1(OC)ccc(C)cc1NC(=O)C(=O)NC1CC1CSc1nccn1C CC1CCCN(C(=O)C(=O)NC2CC(NC(C3(C)CCCOC3)=O)C2)C1 CC(C#N)CN=c1nc2sccc2c(NCC2(C)CC2(F)F)[nH]1 C(=O)(C#CC1(C)CCCO1)N1C(CC(=O)NC2C(N(C)C)CCC2)C2CCCC21 c1(OC)cccc(-c2ncccc2C(N2CCC(c3c(C)noc3C)C2)=O)c1 C1(CNC(CCCc2c(C)ccs2)=O)(NC(C2CC2C2CC2)=O)CCOCC1 C1(COC)(CNC2(CCC(=O)OC)CC2(F)F)CCC(=O)N1 N1(C(C(CC)O)=O)CCc2sccc2C1CNC(c1ccc[n+]([O-])c1)=O c1(C(N2C(CNC(C(C(CC)O)C)=O)C3CCC2C3)=O)ccnc2[nH]cnc12 CCCC(O)CC(=O)NC1CCN(C(=O)C2CC2)CC1NC(=O)NC c1(SC)cccc(C(=O)NC(CNC(=O)C2=CCC2C)CO)c1[N+](=O)[O-] CN1CCC(F)(C(=O)NC2CCC(NC(=O)CNc3ccccn3)C2)CC1 N1(C(c2c(CC)nco2)=O)CC(O)CC1CNC(C1CCC1C(C)(C)C)=O c1(C(=O)NCC2(O)CN(C(=O)C=C(Cl)Cl)C2)coc2c1CS(=O)(=O)C2 c1(OCC(=O)NCCN(C(=O)CCc2ccccc2Cl)CCOC)ccccc1C c1(C(N2C(CNC(c3csnc3C3CC3)=O)CC(OC)C2)=O)ccc(C)cc1C C1(C2CC2)(CNC(C(CC)(C)O)=O)CCN(C(c2cnc(O)nc2O)=O)C1 N1(C(Cn2c(C)ncc2)=O)CCN2CCN(C(c3cc(C(F)F)no3)=O)CC2C1 N1(C(c2c(OC)ccs2)=O)CCN(C(=O)CC(C)(C)C2CC2)CCC1C C12(C(=O)NCC3C(NC(C(C)CC(F)F)=O)C3)CC3CC(C1)CC(C)(C3)C2 C(=O)(C(C)C(C)(F)F)NC1C(NC(CS(N2CCC(C)CC2)(=O)=O)=O)COC1 c1(C(N(CCC(=O)NCCc2cc[nH]n2)CC=C)=O)cncc(OC)n1 c1(C(=O)NC2C(OC)CN(C(C3CC(SC)C3)=O)C2)cnc(O)c2cccnc12 CCCC(CC(C)C)C(=O)N(C1CCC(NC(=O)C(C)SC(C)C)CC1)C C(=O)(C(C(F)(F)F)OC(C)=O)NCCN(C(=O)CC1CC1C1CC1)CC N1(C(C2C(C)(Br)C2)=O)CCC2(CCOC2)C(CNC(c2c[nH]cc(Cl)c2=O)=O)C1 C1(C(N2CCC(OCCNC(C(c3cc(C)sc3)(F)F)=O)C2)=O)CC(N=[N+]=[N-])C1 C1(O)(CCNC(CCNS(CC)(=O)=O)=O)CCN(C(=O)C(C)(F)CC)C1 C1(CC(=O)NC2CCC(F)C2)CC2(C1)CN(C(=O)Cc1csnn1)C2 C(CS(=O)(=O)CC(=O)NCCC1(CNC(=O)Cc2cccn2C)CC1)N(C)C C(=O)(CCCCCCC(=O)O)NC(C1CC(OC)C12CCCC2)=O C(=O)(C(C)(C=C)CCOC)NCC(CNC(C(C=C)(C)C)=O)O Cn1cc(CNCC2(C(F)(F)F)CC(O)C2)c2cc(Br)ccc12 c1(C(=O)NCC2C(NC(C3CC(C)CC(C)(C)C3)=O)C2)cccc(C=C(F)F)c1 C(=O)(CC(C(C)(C)C)NC(=O)CC1CCCO1)NC(C(=O)OC)C N1(C(CCC(CC)C)=O)Cc2ccc(CNC(=O)C(C)N(C)C(C)=O)cc2C1 c1(OC)cc(C(N2CCC3(C2)CN(C(c2onc(C)c2C)=O)C3)=O)c(C)cc1O C1(C(=O)NC(CNC(CN(C)CC)=O)(C)CC)CCc2nc(O)[nH]c2C1 CC1(C(=O)O)CCCC1NC(=O)NCc1ccc(NS(C)(=O)=O)cc1 C1(NC(c2c(CNC(c3ccc(C#C)cc3)=O)c[nH]n2)=O)CCn2ncnc2C1 N1(C(c2cccc(SC)n2)=O)CC2CCC(N(C)C(c3ccnnc3O)=O)C2C1 c1(COCC(=O)NCCN(CC(=O)NC(F)(F)C(F)(F)F)CC)cccc(C)c1 N1(Cc2c(-c3c(C)ccnc3)cccc2)CC2(CC2)n2nccc21 C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)NCCCN(C(CC1CC(CC)C1)=O)C CCC(O)C(C)(C)C(=O)N1CCC(CO)(NC(c2ccc(O)c(C(C)=O)c2)=O)C1 c1(CC)cccc(C(=O)NC2CC(NC(=O)C(F)CC3CC3)C2)n1 c1(C(=O)NC(C2CCNCC2)C)cc2cc[nH]c2cn1 CCC(C)(F)C(=O)N1CC(OCCN(c2cc(C)sc2C)C(=O)OCC)C1 N1(C(C=NOC)=O)CC(NC(=O)CSCc2ccncc2)CCC1C C12=NNC(=NC(=O)N1C1CCCCC1)S2.N1(CC)CCC1CF CN1CC2CCC(C1)N2C(=O)C(C)(C)CNC(=O)CC1CCCC1O C1(C(C(=O)NCC(=C)C)N(C(C)C)CC)CCCC1(C)C Cc1n[nH]c(=NCCC(C)(C)NC(C2CC(OC(F)(F)F)C2)=O)s1 CC(CN=c1cc(Cl)nc(C2CCC2)[nH]1)NC(C1(C)CC(O)CN1C)=O N1(C(=O)NCCC=CCCC)CCC(CN(C)C)CC1 CC#CCCCC(=O)NCC(CNC(c1ccccc1CN(C)C)=O)OC CP(C)(=O)c1ccc(C(N2CC3(C2)CN(C(=O)CC2CCC4CC24)C3)=O)nc1 c1(C(=O)NCC(CC)(C)NC(=O)CC2CCC(C3CC3)O2)cnn2c1CCC2 c1(C(=O)NCC2C3CN(C(COCC#C)=O)CC32)cc(S(C)(=O)=O)oc1C CC1=C(C(=O)NC2CCCCC2NC(C2CC(C(C)C)=NO2)=O)CCCO1 C1(NC(C(CCOC)C)=O)CCCC2CN(c3cc(C#N)nc(C)n3)CC12 C(c1cccc(OC)c1OC(F)F)=CC(N1CCC(CNC(C(CC)C)=O)C1)=O N1(Cc2c3n[nH]c(C)c3ccc2)Cc2ccc(NC(c3nc(Br)cs3)=O)cc2C1 c1(CC(=O)NCC(CC)NC(c2ccc(C)cc2O)=O)c(F)c(F)cc(F)c1F C1(C(=O)NCC2C(NC(c3nnc(C(C)(C)C)s3)=O)CC2)CCC(F)(F)CC1 N1(C(c2c(Cl)cn(CCC)n2)=O)CCC2C(CCN2C(=O)C=CC(C)C)C1 c1(C(N(C2CC2c2sccc2C)CC)=O)ccc(OCC(F)F)cc1[N+](=O)[O-] C1(NC(C(CC=C)OC)=O)C2CCC(C2)C1C(=O)N(C(C)CC(F)(F)F)C c1(C(=O)OC)c(N=[N+]=[N-])cnnc1N1CCCC(N2CCCS2(=O)=O)CC1 c1(CC(=O)N(CCNC(C=Cc2occ(C)n2)=O)C2CC2)ccc2ncsc2c1 Cn1nc(C2Cc3ccccc32)nc1-c1cc(CC2CC2)on1 CC(C)(C#N)CCC(=O)NCCC1CC(NC(C2CCCCN2C(N)=O)=O)C1 Cn1cnc2nc(N3CCC(c4nncs4)CC3)[nH]c(=NC3CCOCC3F)c12 Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NC12CC(C1)N(C(=O)CC(F)(F)C(F)F)C2 c1(C(C(F)(F)F)NC(C(C)=C2CCCC2)=O)ccccc1C#N c1(C(=O)NCCC2(NC(C3=C(C)OCC3)=O)CCC2)ccc(S(N)(=O)=O)cc1 C1(NC(c2c(C)nncc2)=O)(CO)CCCN(C(C2(C#N)CCCO2)=O)C1 C=CCC(CC(=O)NCC(C)CC(=O)OC)NC(C1(CCC)CC(=O)C1)=O c1(CCC(=O)NCC(C)N(C(C(C(C)C)CO)=O)C)cc2ccccc2o1 c1(N(CC(CC)OC)C)nc(=NCC(C(C)C)OCC)[nH]c2cc[nH]c12 c1(OCC(=O)NC2C(NC(C(C)c3cccs3)=O)C2)ccccc1C(F)F c1(C(N2CC(OC(C3(C)C(C(=O)OCC)CC3)=O)C2C)=O)c(C)noc1C1CC1 C12(C(=O)NC)COCC1CN(C(=O)CN(C)C(=O)C1CC1)C2.C1CCN1 c1(C(=O)NC(C)CN(C)C(c2ccn(C3CC3)n2)=O)ccc(N)cc1F c1(C(C(=O)Nc2ccc(Cl)cc2)N(C)C)n[nH]c2c(F)cccc12 S(=O)(=O)(c1ccccc1Br)N1CC(N(S(CC)(=O)=O)C)C1 c1(C(C)NC(=O)NCC2CN(C)C(=O)O2)ccc2cc(Br)ccc2c1 CC(C)C(C)(O)C(=O)NC(CNC(c1cc(-c2cccs2)on1)=O)CO c1(CC(N2C3CC(CC(NC(COC)=O)C3)C2)=O)coc2cc(C(C)C)ccc12 C1(C(N2CC(C)C(CCNC(=O)CCn3cccc3)C2)=O)CC2CCC1CC2 N1(CC)CCOCC1CC(=O)NCCC(C)N(C(=O)Cc1cnns1)C CC1CC2CN(C(=O)C3=NN(C)C(=O)CC3)CC2N1C(c1ccncc1)=O N1(C(C2(CF)CCN(C(C3C4CC5C(C4)C35)=O)C2)=O)CC2CCC(C1)C2O c1(NC(CN(C)CC2CCN(C(=O)CC3CCC(=O)O3)C2)=O)ccc(F)cc1Cl CC1CC2CN(C(C3CCC(C)(C)OC3)=O)CC2N1C(=O)C(F)C(C)(F)F c1(OC)c(COCCn2c(N(N3CCN(C)C(=O)C3)C)nnc2C)cc(F)cc1F N1(C(CCCC2CC2)=O)CCC2(C=C(C(=O)NC(CC3ON=C(CC)C3)=O)C2)C1 C1(OC)CC(CO)N(C(=O)CC(CNC(=O)C(C)C(C)C)C2CCC2)C1 C(CCC(=O)NCC(C)NC(C1CC1(C)C(C)C)=O)OCC(C)C CC1CN(C(c2c[nH]nc2[N+](=O)[O-])=O)CCCN1C(C1OC2CCC1CC2)=O c1(NCCCC=C)ncccc1S(=O)(=O)NC(c1cccc(F)c1C)C C1(C(=O)NCC2(NC(C3CN4CCC3C4)=O)CC(C)(C)C2)CC2CC1CC2=O N=c1[nH]c(=NCCc2cc(Br)no2)[nH]c(=NC2CC3CSCC3C2)[nH]1 C1(C(=O)NCC=CC(=O)N(C2CCCCCC2)C)CCCCC1CO c1(NCc2cc(C)c(C)[nH]2)c(C)cccc1[N+](=O)[O-] c1(C(N2CCCSCC2)C(N2CCC(n3ccnc3)CC2)=O)ccccc1F c1(C(N2CC(CC(C)NC(C3(C(C)C)CCCO3)=O)C2)=O)cc(Cl)c(N)cc1F C1(NC(=O)CCc2cnoc2)CC2CC(NC(=O)Cc3nnc(O)s3)CC12 N1(C(CCN(C(COCCCCC)=O)CC)=O)CCCN(C)C(=O)C1 C1(NC(=O)Cn2ccnn2)CC2CC1CN(C(c1nn[nH]c1Cl)=O)C2 N1(C(C2CN(C(C(C)N(C)C)=O)C3(C2)CCC3)=O)CC2CCC(C1)C(=O)N2 N#CC1(C(=O)NC2CC(F)(CNC(C3CCOC3)=O)C2)CC12CCOCC2 c1(CC(=O)NC2CC(CNC(C3(C(C)=O)CC3)=O)C(O)C2)nc2ccccc2[nH]1 C(=O)(C(O)CC(C)C)NCC(C(=O)NC(CCOC)C)(C)C Cc1ncc(C(N2CC=CC2(C)C(=O)NCCCCN2CCC2)=O)n1C Cc1csc(C=CC(=O)NCCC(O)CNC(=O)C(Cc2ccsc2)NC=O)n1 c1(C(N2CCN(C)CC2CNC(c2ccc(=O)oc2)=O)=O)ccn2nccc2n1 N1(C(c2cccc(CC)c2N)=O)CC(C)(C)OCC1CNC(=O)Cn1cnnn1 CCC(O)C(C)C(=O)N1CC(C)C(C)(CNC(=O)CSCc2c(C)noc2C)C1 c1cccc(O)c1.c1(CC(=O)NC(C2CN(C(C3CC3)=O)C2)C)ccoc1C CC1=NOC(=O)C1CCC(=O)NC(C)CC(C)NC(c1cccc(C)n1)=O c1(C(=O)OC)nc(NC(C2CCC2CN)=O)cnc1OC(C)(C)C c1(C(N(CC(C)N(C(C(CC)n2ccnc2)=O)C)C)=O)cc(S(N)(=O)=O)cs1 C1(CCCNC(C2CC2CF)=O)(CNC(C(C)=CC)=O)CCCC1 c1(NC2(C(F)F)CC(NC(c3ccc(OC)nn3)=O)C2)nc(OC)cc(C)n1 c1(C(=O)NC2C(CC)CN(C(c3ccoc3C)=O)CC2)ccc(C)c(F)c1N N1(C(CCOCc2c(C)ncs2)=O)CC(CNC(=O)CCN(C)CCO)C(O)C1 N1(C(c2ncc(C)nc2)=O)CC2(CNC(c3c[nH]nc3C(F)F)=O)CC1CCO2 C(=O)(C(CO)C(C)C)N1C(CN(C(c2ccc(OC)cc2)=O)C)CCC1 N1(C(C(Cc2cn[nH]c2)NC(C2C=CC=CC=C2)=O)=O)CCC(C2CCCC2)C1 c1(C(=O)NCC(=O)NCC2C=CCN2C(=O)CC2CC2(Cl)Cl)ccc(CO)cc1F C(=O)(CC1=CCN(C(C2(Cl)CCC2)=O)CC1)NCC(CC(=O)OC)O C(CC(C(C)(C)C)N(C(CC(C)SC1CC1)=O)C)NC(=O)Cc1cccc(N)c1 c1(C(=O)OC)ccc(Br)cc1OC.C12(CCC1)CC(=O)O2 N12CCc3ccccc3C1CN1C(=CC=C([N+](=O)[O-])C=NC(CCF)C1=O)C2=O c1(C(=O)NCCC2N(C(C3CC(=O)NC3)=O)CCC2)cc2c(cn1)COCC2 C1(C(=O)NCC2CCCN(C(COCCCCC)=O)C2)CC2(C1)CC1(CC1)C2 Cc1c(CC(=O)NC2CCCC(NC(=O)CCn3ccccc3=O)C2)ncn1C c1(C(N(C2CCN(C(=O)Cc3sc(O)nc3O)C2)C)=O)cc(F)c(CO)c(F)c1 C1(CNC(c2c(C)cco2)=O)COCCN1C(c1cc[n+]([O-])cc1)=O C1(C(C(N2C(CC(=O)N(CC(C)(C)C)C)CCC2)=O)=O)CCCCCC1 C12(NC(=O)OC(C)(C)C)CC(C(F)(F)F)C1CN(C(=O)CCc1nc(O)n[nH]1)C2 C1(CC(=O)N(CCCC)CCOC)C2CCC(C2)N1C(=O)CC1(CSC)CC1 C1(OC)(CNC(=O)C(F)C(C)C)CCN(C(c2sccc2SC)=O)C1 c1(C(N2CC(CNC(CCSC)=O)C3C2C3)=O)cc(Cl)c2c(c1)OCO2 C1(C2(C(N(CC(CNC(COCC(C)C)=O)O)C)=O)CC2)CCCCO1 CCC(CC(C)C)C(=O)NC(C)(C)CN(C)C(c1cnnn1CC)=O C(=O)(CC(C)C(=O)c1ccccc1)N1CC(CC(C)NC(C2(C)CCCC2)=O)C1 C1(CNC(c2nc(CCC)sc2)=O)CCC12CCN(C(=O)C(F)(F)C(C)O)CC2 C(=O)(C1=C(C2CC2C)N(C)C(=S)NC1c1cc(C)n(C)n1)OC CCC(C(=O)OC)C(=O)NCC1(NC(c2cc(C(C)C)on2)=O)CCC1 c1(NC(N(C)Cc2ccc(N3CCOC3=O)cc2)=O)cn(C)c(=O)nc1O C1(C(C)(C)C)(CNC(c2ccc(O)nc2)=O)CCN(C(=O)C=CC2CCOC2)C1 N1(C(CCN(C(=O)CN2CCCC2=O)CC)=O)CCC(C)(C2CC2)C1 C1(C(N(C)CC2CCN(C(=O)CC3(N(C)C)CC(O)C3)C2)=O)CN2CCN1CC2 c1(C2C(CNC(=O)Cc3cccc(Cl)c3)C2)ccc([N+](=O)[O-])cc1 C#Cc1cnc(C(=O)NCC2N(C(=O)OCC)CC2(C)C)c(C)c1.C(C)(C)(C)O Cc1sc2ccccc2c1C(N1CCC(CN(C)C(C2(C(N)=O)CC2)=O)C1)=O CC1CN(C(=O)C2=COCCO2)CCC1NC(c1cc(CO)ccn1)=O CCN=C(NCCCN(S(C)(=O)=O)CC(C)C)NCC1(N2CCCCC2)CCCC1 CC1(CCNC(=O)C2=CCCO2)CCN(C(C2CCCOC2)=O)C1 S(=O)(=O)(c1ccccc1S(=O)(=O)Nc1ccc2c(c1)CCCO2)NC N1(C(N(CC(N2CC=CCC2)C)C)=O)CCCC(CO)(NC(=O)OC(C)(C)C)C1 CCC(CCCO)NC(=O)C(N1CCCCC1COCC(C)(C)C)=O N1(C(CCC(=O)NCCC)=O)C2CCC1CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 Cc1nc2ncccc2cc1CCC(=O)NNC(=O)c1coc(-c2cccs2)n1 c1(C(=O)NC)ccc(C(=O)NCC2(O)CC(NC(C3(C#N)CCCO3)=O)C2)cc1 C12(C(=O)NC(C(C)C)C(C)NC(=O)C=CC(=O)NC3CC3)CCC(CC1)CC2 Cn1c(C(=O)NCC2(C(N3CC(C#N)(CCF)C3)=O)CC2)cc[n+]1[O-] c1(C(=O)NC2CCC(NC(c3snc(C)c3N)=O)C2)c(C)cncc1C N1(C(=O)CCn2ccnn2)CCCC(C2CCN(C(C3CC34CC4)=O)C2)C1 c1(C(=O)Nc2c(C)c(Cl)ccc2)n[nH]c2c1CN(C(=O)C(C1(O)CCCC1)F)C2 c12c[nH]c3cc(NC(C#C)CC4CCCO4)c(cc3c1=O)C(=O)OC2.O(C)OC CC(CCCc1ccccc1)C(=O)N1CCCC(C)(NC(c2ncn(C)n2)=O)C1 C(c1cnccn1)=CC(=O)OCC(c1nnc(C)s1)=O c1(NC(CC2(O)CCN(C(c3nc(C)oc3)=O)CC2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC2CC(C(=O)Nc3ccn(C(C)(C)C)n3)C2)cnn2cc[nH]c12 N1(C(C2(CNC(C3C(=O)NCC3)=O)CCCC2)=O)CC2C=CC1CC2 C1(OCCNC(=O)CC2CCCO2)CCN(C(=O)Cc2cc(C3CC3)no2)CC1 Cc1ccn2ncc(C(=O)NCC3CCCCC3NC(c3ccn(C)c3)=O)c2c1 CC(C)(O)C(F)CNC(=O)CC1(C)CCN1C(C1CC=CCO1)=O N1(c2ncnc(=N)[nH]2)CCC2CCC(C1)N2C(=O)CN1CCNC(=O)C1 C1(Nc2ncc(C(=O)OCC)cn2)CN(C(=O)COC(C)=O)CCC12CCC2 c1(C(N2CC(NC(=O)Cc3c[nH]nc3O)C(CO)CC2)=O)cc(F)c(F)cc1F N1(C(C(C(C)C)F)=O)CC(C)(C)CC1CC(=O)Nc1cccc(NC=O)c1 N1(C(C2(C)CC(=C)C2)=O)CC2(CCC2NC(=O)C(C2CCCCC2)O)C1 C=C(C)CC(C)C(=O)NC(CNC(c1cccc(C)c1Cl)=O)C1CC1 c1(NC(c2ccc(O)cc2)=O)ccc(NC(c2cc(Br)c[nH]2)=O)nc1 C1(C(=O)NCC(C(C)C)NC(c2c[nH]c(=NCC)s2)=O)CCc2cncn2C1 CC1=CC(C)CN(C(=O)CC(CC2CC2)NC(=O)Cn2c(O)nnc2O)C1 c1(C(=O)NC(C)(CNC(=O)Cc2ccnc(Br)c2)CO)cc2n(n1)CCC2 c1(CC)nc2sc(C)cn2c1NC(C1CCN(C(=O)COC(C)=O)C1)=O C1(OC)CN(C(=O)CCC(N)=O)CCC1NC(C1(CO)CCC1)=O N1(C(C=C(C)c2ccco2)=O)CC2(CCC2)CC1C(=O)NC1CNC(=O)C12CC2 C1(C(=O)NCCC(C)NC(=O)CC2C=NN(C)C2=O)(CSC)CC(F)(F)C1 N1(C(c2c(C(=O)OC)scc2)=O)CCC(C2CCCN(C(=O)CSC3CC3)C2)C1 Cn1ncc(C(=O)N(CCNC(c2cc(Br)no2)=O)CCOCCO)n1 C12(C(N(CCCCCNC(C3CC34CC(O)C4)=O)C)=O)CCC(CC1)C2(C)C C1(C(=O)NCC2(F)CC(CNC(=O)CCF)C2)CN2CCN1CC2 N1(C(CC=C)=O)CCC(N(C(=O)CN2CC(NC(C)=O)CC2=O)CC)CC1 C1(NC(=O)CC2CC=CC2)CC2CN(C(=O)Cc3ccnc(F)c3F)CC12 C=CC(CC)CC(=O)N1CCC(C)C(CNC(C23CC4CC2C3C4)=O)C1 Cc1nc(CC(N2C(C(=O)Nc3ccccc3Br)CC3CC23)=O)c(C)s1 c1(C(=O)NCC2N(C(C3C(C(C)O)C3)=O)CC(F)C2)cccc(=O)n1C CCC(C(=O)N1CCC(NC(c2cnc(S)n2C)=O)C(F)C1)C(C)C c1(C(CC)C)nc(N2CC3(CN(C(c4cc5sccc5[nH]4)=O)C3)C2)cc(C)n1 N1(C(CC2(C)CCN(C(c3c(C)cnn3C)=O)C2)=O)CCCC(C)C1CO CC(CS(C)=O)C(=O)NCCNC(=O)Cc1csc(NC2(NS(C)(=O)=O)CC2)n1 c1(C(=O)NCC2C(NC(C3(C)CNC(=O)C3)=O)CC2)cc([N+](=O)[O-])c(Cl)cc1Cl Cc1c(C)c(C)c(C(=O)NC2CCCC(NC(C3CC3C)=O)C2)c(C)c1C N1(C(C2(OC)CC2)=O)CCC(OCCCNC(=O)Cn2cncn2)CC1 C1(N(C(C=CSC)=O)C)CCCC(NC(=O)C(C)NC(=O)NC2CCCC2)C1 c1(CC)ncc(C(=O)N(C)CC2(NC(=O)CSCCOC)CC2)[nH]1 C(CC(F)(F)F)N(C(=O)CC1CN(C(C2CC(F)(CF)C2)=O)C1)C CC1CN(C(C2OCCCO2)=O)CCCN1C(C1CN(C)CCN(C)C1)=O c1(OC)ccccc1C(=O)NCC1(CCNC(C2CC(n3cnnc3)C2)=O)CC1 CC(CC(=O)N(C1CCN(C(=O)CC=CC(C)(C)C)C1)C)c1ccncc1 N1(C(C2(CCC)CC2)=O)CCC2(CC1)CC(NC(c1cn(C3CC3)nc1C)=O)C2 C1(NC(C2CCCCC2)=O)CCCN(C(=O)C(O)C(F)(F)F)CCC1 C1(NC(c2ccc(Cl)c(-n3nnnc3C3CC3)c2)=O)CCCNC12CCC2 C1(C2CCN(C(C=NOC)=O)C2)CCCN(C(=O)CC2(C)CC2)C1 C12(C)CCCN(C1)C(=O)C1CCN(C1C)C2=O.C1(CC)CC2(CSC2)C1 CC(C)C(C)C(=O)NCc1cnn(C)c1C(=O)N(C1CC1)CC1CC1 c1(CNC(=O)NC2CCCC(N(C)C)C2)nnc2ccccn12 N1(C(c2cnc(CC)nc2)=O)CCCC2(CNC(C3C=CCS3)=O)CCCC12 Cc1ccnc(C(=O)NC2CC3(C2)CC3C(=O)N(C)Cc2cocn2)c1F c1(C(NCP(OCC)(C)=O)=O)cnc(CNC(=O)CC2CC3(CC3)CO2)nc1O C1(NC(C(CNC(C=Cc2c(C)cccc2)=O)O)=O)CC2(CCCCC2)C1 CC1CCCCC1C(=O)N(C)CC1(O)CN(C(=O)CS(=O)(=O)N(C)C)C1 Cc1nc(C(=O)NCC(C(C)(C)C)NC(=O)CC2(O)CCCOC2)nn1C C(CC(=O)NC(C)C(=O)NCCF)N(C(=O)C(C)C1(O)CCC1)CC C1(COC(C)(C)C)CCC(C(=O)NC2CCN(C(=O)CC3CCOC3)C2)CC1 c1(OC)ccc2c(C(=O)NC3(C)CN(C(c4cc(=O)cc[nH]4)=O)C3)ccnc2c1 C(=O)(CC(C(F)(F)F)NC(=O)COCC1CC1)N(C)CC1CCSC1 C1(C(N2CC(O)(CN(C(c3cc(CC)on3)=O)C)C2)=O)CC(OC)C(OC)C1 N1(CCCC=C)CC2CCN(C(c3ccc(C(C)CC)cc3)=O)CCC2C1 C(CC(C)(C)C(=O)NC1(CC(=O)NCC2(C)CCCOC2)CC1)OC N1(C(C(CN)C2CCC2)=O)CCC(C(C)O)CC1 C(=O)(CCC(CC)CC)NCCCC(CCC)NC(=O)CCc1nc(C)c(C)o1 C1(C(=O)NCC(C)NC(c2cccc(-c3ccc(O)nn3)c2)=O)OCCOC1C CCC(O)C(C)(C)C(=O)NCC1(F)CC(NC(c2cccc(SC)c2)=O)C1 c1(C(N(CCNC(CCn2ncn(C)c2=O)=O)C2CC2)=O)cnc2nccn2c1 N1(C(C=Cc2cnc(C)s2)=O)CCC(NC(C2CCCC(=O)N2C)=O)C(C)C1 N1(C(CCCC)=O)CCC(C(F)CNC(C2(CC)CC(C)(C)C2)=O)CC1 c1(C(=O)NCCN(C(=O)C(C)C(C)C)CC)cncc2n[nH]cc12 C(=O)(CN1C(=O)C(F)(F)c2cc([N+](=O)[O-])ccc21)N(c1cccc(C2CCN2CCN)c1)C CN1CC2(CC2)CC1C(=O)NC(C(N1CCC(O)(C(F)F)C1)=O)C1CCCO1 c1(NC(C)=O)ccc(F)c(N(C2CCNCCC2C)C(c2ccc(F)cn2)=O)c1 c1(NC(C2CCN(Cc3ccc(CO)o3)CC2O)=O)cccc2c(I)n[nH]c12 N1(C(C(C)NCC(C)(C2CC2)OCC)=O)CC(C)C1 CC1OCCC1CC(N1CC(C)(NC(=O)NCC(=O)N(C)C)C1)=O c1(C(N(CC(CC)NC(c2csc(NC(C)=O)n2)=O)C)=O)cnc(C)[nH]1 C#CC1(NC(C23CSCC2C3(F)F)=O)CCC(C)(C)CC1 c1(C(N2C(CN(C(C3C(CC)C3)=O)C)CCCC2)=O)cc2c(=O)[nH]ccn2n1 C1(NC(c2c(C)cnc(F)c2)=O)CN(C(=O)C(CC)CO)C2CCCCC12 Cc1nccnc1C(=O)NCC1CCC(N(C(=O)C=Cc2cnc[nH]2)C)CC1 Cc1c(C(=O)NC2CN(C(=O)C(=O)NCC3CC3)CC2C(F)(F)F)nnn1C C(CCCCC(=O)N(C(C)CNC(=O)Cc1sccc1Br)C)SC CC(C)(CF)C(=O)NCCC1CCN(C(c2ncc(C(F)(F)F)s2)=O)C1 C1(C(C(=O)NCC2CC2)N(C)Cc2ccncc2F)CC2C(C1)C2(F)F.C1(C)CC1 c1(C(c2n(CCCSC)nnn2)NCCc2ncccc2C)ccc(Cl)cc1F c1(CNC(CCC2OCC(C)(C)C2)=O)ccc2c(c1)CN(C(=O)CO)C2 C1(OC)CN(C)CC1NC(=O)C(c1ccnn1C)NC(c1nonc1N)=O c1(C(=O)NC(C)CNC(=O)C(C)(O)C2CCOCC2)noc2cc(Cl)ccc12 C(=O)(CCC(=O)c1cccnc1)NC12CC(NC(CNC(CN(C)C)=O)=O)(C1)C2 C=C(C)C(CC(=O)NC1CN(C(c2cnc(C)s2)=O)CCC1C)OCC Cc1cc([N+](=O)[O-])c[nH]c1=NCC12CCCCC1OCC2 N1(C(C2N(C(C(CC#C)C3CC3)=O)CCC=C2)=O)CCC2CCCC2C1 C1(NC(C(N2CCCCC2)C)=O)(CO)CCN(C(c2cccc(CO)n2)=O)C1 N1(C(C(CCC)CC2CCCCC2)=O)CCC2(CC1)CN(C(=O)C=CCOC)C2 C1(NC(C2C(OC)CCC2)=O)(CNC(C2CC=C(C)CC2)=O)CC2CCC1CC2 n1(C(C)C)c(O)nc(N2CCC(CNC(c3ccc(Cl)nn3)=O)CC2)cc1=O N1(C(C2SC3C=CC2CC3)=O)CCc2cc(O)c(Br)cc2C1 CCC(C)(C(=O)N1CC(O)(C(C)NC(=O)Cn2ncnn2)C1)OC C(c1ccc(F)c(F)c1)=CC(=O)NCCCC(CCC)NC(c1cc(C)no1)=O C1(C(N(C2(C)CC2)CC#C)=O)CC12CC(NC(=O)CN(C)CC)C2 CC1CC(C(=O)N2CCC23CN(C(C2COCCN2C)=O)C3)=NO1 CCC(C(=O)N1CCC(CCC(=O)N(CCCCCC2CC2)C(C)C)CC1)C(C)C C(=O)(C(CCF)NC(=O)C(C)C1CCC1)NCC(=O)OCCCC.OCC C1(CC(=O)N(C2C(OC)COC2)C)N(C(=O)CNc2ccccn2)CCC1(C)C CON1CCC(C(N2CC3CC(NC(c4cnnn4C4CC4)=O)C2C3)=O)CC1 C(=O)(C(C)CC(C)CC)N1CCC(CNC(CC=CC=C)=O)C12CC2 c1(C(N(C)CC2CCN(C(CC(C=C)CC)=O)CC2)=O)cc2occc2n1C N1(C(c2c(C)noc2)=O)CCN(C(=O)CCc2cccnc2Cl)CC1C(C)C C#Cc1ccc(C(N2CCC(CC=C)(NC(=O)C(CC)OC)CC2)=O)cc1 c1(CN2C(C)(C(=O)NC(CC(C)C)c3ccccc3)CC2)cccnc1O C(=O)NNc1c(F)cccc1Br.C1(CC)CCC1(C)CS(=O)(=O)Cc1ccccn1 c1(OC)cccc(CC(=O)NCC2CC(CNC(C3(O)CCC3)=O)CO2)c1Cl c1(C(=O)NCC2N(C(c3scc(C)c3)=O)CC=C2)ccc(C)cc1F N1(C(c2ccc(OC)s2)=O)CCC2CCC(NC(=O)CC3CCC4CC4C3)C1C2 N1(C(CC2(C)CN(Cc3ccc(Br)o3)C2)=O)CCC2(CC1)OC(=O)NC2=O C(=O)(C(O)C(C)(C)C)NC1CCN(C(CC(C)SC)=O)C1 C(=O)(CC(C)C(F)F)N1CC(c2c(CNC(c3nccc(OC)c3)=O)nco2)C1 c1(OC)cc2cc(c1Br)NC1CC(C1)NC2=O.c1(OC)cccnn1 C(N=c1nc2c(ncn2C(C)C)c(NCc2ncc[nH]2)[nH]1)c1cc(C)cc(C)n1 N#Cc1cnn2ccc(N(CCC(F)(F)F)CC3NC(=O)NC3)nc12 Cc1cc(C(N2CC(NC(c3cccc(=O)o3)=O)CC(O)C2)=O)ccc1F N1(C(=O)NC(C(c2ccc(F)cc2)OC)C)CCCC2CC1C2(C)C N1(C(CCc2onc(C)n2)=O)CCC2CCC12CNC(c1cccnc1N)=O c1(C(C(=O)N(CCC(=O)NCCOCCC=C)C)C)ccnn1C C1(O)(C(=O)NCC2(NC(c3ccn(C)n3)=O)CC2)CCCC(C)(C)C1 C1(CNC(c2cc(OC)nn2C)=O)CC2COCC2N1C(=O)CCOC(C)=O CC1CCc2ncc(C(=O)NC3CN(C(C4CC(C)(C)C4)=O)CCC4CC34)n2C1 N1(C(CC2(NC(c3cc(C)c(F)cc3)=O)CCC2)=O)CCC2CN(C)CC2C1 c1(OC(C)C)cccc(C(=O)NCC(O)CNC(=O)C2=CCCOC2)c1F C(=O)(C1=Cc2ccccc2OC=C1)N(C)CCNC(c1csc2cnccc12)=O Fc1ccc2c(-c3ccccc3C3CC3c3c[nH]c4ncccc34)c[nH]c2c1 CC(C)(C)CC(O)C(=O)N1CC(C)(C)C1C1CCN(C(c2cc[nH]n2)=O)CC1 N1(C(CC2CCC(C)CC2)=O)CC2CN(C(=O)CN(C3CCCC3)C)CC2C1 C1(C(=O)NC(C2CCN(C(=O)C=C(C)C(C)(C)C)C2)C)(OCC)CCOCC1 CC(C(=O)NCCCCCN(C)C(c1ccccc1CC(C)(C)C)=O)C(C)(C)C c1(C(C)(C)C(=O)NCC2(CCNC(=O)Cc3ccon3)CC2)ccc(Cl)nc1 c1(CC)nc(C)c(C(=O)NC(C2(O)CN(C(c3ccc(CN(C)C)o3)=O)C2)C)s1 C(=O)(C1CCCn2nccc21)C(C)CC1CN(C(c2ccc(O)c(O)c2)=O)C1 C(CC(C(=O)N(CC(CO)(CO)NC(C12CCCCC1C2)=O)C)NC=O)SC N1(C(CC=CCCCCC)=O)CCN(C(=O)C(c2ccc(F)cc2)=O)C(CC)C1 C1(N(C(CCNC(C2CCN(CC)C2)=O)=O)C)C2CC3C(C2)C13 N1(C(=O)NCCC=CCCC)CC(CN(C)C)C(O)C1 CC1(C)C2CN(C(=NCCCC3CC3)NCC3CCS(=O)(=O)C3)CC12 c1(OC)cc(Br)c(CN2CC3CC2CN3C(=O)Nc2ccc(SC)cc2)cc1O N1(C(CC=CCc2nc(=N)[nH]cc2)=O)CCCC(n2cc(C3(O)CC3)nn2)CC1 C#CCCCCCC(=O)N(C(C)C(N1CC2(CCC2)C1)=O)C c1(CC)n[nH]c(=NC2CC(CNC(=O)CCc3c(F)cccc3F)C2)s1 c1(C(=O)NCC(C2CCOC2)NC(Cc2scc(CC)n2)=O)cn(C)nc1CC C1(C)(CNC(COCC)=O)CCCC1NC(=O)C(C)NC(=O)OC N1(C(c2cc(C)c(C)s2)=O)CC(C)CN(C(=O)CN2CCC(C)C2)CC1C N1(C(CNS(CC)(=O)=O)=O)CCC(NC(=O)C(=CC2CCCC2)C)CC1 C12CCN(C(C)C1)C2=O.N1(CC)CCC(NC(C2CC2C(=O)OC)=O)C1=O C1(NC(=O)COc2ccc(F)cc2)CN(C(C2CCO2)=O)CC1n1ccnn1 N1(C(c2nccc(OC)c2)=O)CCN(C(=O)C2=C(C)CC2)CC1C1CCC1 C1(C(=O)NCC2N(CC)CCC2)C2CC3C(C2NC(c2ccc(C#N)n2C)=O)C13 N1(C(CCC2N(C)CCC2)=O)CCC(C2CCN(C(=O)C=CBr)C2)C1 N1(C(c2cccnc2OCC2CC2)=O)CCN(C(C2CCOCC2)=O)C(C2CC2)C1 c1(CCC(=O)OC)ccc(CNC2CN(C(=O)COC3COC3)CC2C)cc1 O=S(=O)(c1ccn(C2CCCC2)n1)NC1(CCCl)CCC1 c1(CC(=O)NC(C)C(C)NC(c2cccn2C2CC2)=O)ncn(C2CCCC2)n1 CC(C(=O)NCCCN(C)C(c1cn(C)nc1-c1ccccc1)=O)P(C)(C)=O N1(C(CCN(C(=O)CCOCC2CC2)C)=O)CCOC(C)(C)CC1 N1(C(c2ccc(CO)o2)=O)CCC2C(CCCN2C(=O)CC(F)F)C1 C1(O)(CN(C(c2cc(C)nn2C)=O)C)CCN(C(C2CCCCC2F)=O)CC1 N1(C(Cc2n(C)nnc2)=O)CCC2C(CCCN2C(c2ccc(C#N)cc2)=O)C1 C1(C(N2CCN(C(c3c(C#C)cnn3C)=O)CC2)=O)CC2CC1CC2(F)F S(=O)(=O)(c1cnc(Cl)nc1)NCC1CCC(NC(c2cc(I)cnc2Cl)=O)CC1 c1(C(=O)NC2CN(C(CC(C)(O)C(F)(F)F)=O)C2)c(N)nn2ccccc12 c1(C(=O)NCCN(C(=O)C(C)SC2CCC2)CC)nnn2c1COCC2 C1(NC(C(C)C)=O)CCCCC1NC(=O)COC1CCSCC1 N1(C(c2cscn2)=O)CC2(CCN(C(=O)C(c3ccc(F)cc3)(F)F)C2)C1 N1C(=NCC(F)F)NC1.O(N(CC)C(=O)CNC1CCC(OC)C1(C)C)CC Cc1cccc(C(=O)NC2(CNC(C3CC3C)=O)COC2)c1O N1(C(Cn2ccc(C)cc2=O)=O)CCN(C(c2cnc(F)cc2C)=O)CCC1C C1(C(N2CC(C=C)C(NC(=O)C(CCC)OC)C2)=O)CCc2ccccc2O1 CC1(C)COC(C(=O)NCC(=O)NC2C=CCCC2)C1 C1(CCC#C)CCCN1C(c1nc(CC(=O)OCC)co1)C(=O)NCC(C)C c1(CC(=O)OC)ccc(OC(=O)CCc2ccnc(Br)c2)cn1 N1(C(c2scc(CNC(CC(C)CCC)=O)c2)=O)CC2CCOC2C1 c1(CC(=O)NC2CN(C(c3n(CCC)ncc3)=O)C(C)C2)c(OC)cccc1C c1(C(=O)NC2(CNC(c3cc(C)c(Cl)cc3)=O)COC2)c(Br)cc(F)c(Cl)c1F Cn1nc(C(=O)NCC2CCCCCN2C(C2C3CCCOC23)=O)c(Cl)c1Cl C=CCCC(CC(C)C)C(=O)N(C1CC1)Cc1cn(C)nc1C(C)C C#Cc1cccc(C(=O)NCC2CC2CNC(=O)C=Cc2ccc(Cl)cc2)c1C N1(C(c2ccc(S)cc2)=O)CC2CC1CN2Cc1c(Cl)cccc1Cl C1(OC)CC(CNC(=O)COC2(C)CCC2)N(C(=O)CC2CNC(=O)O2)C1 CC1(C)OCC(C(=O)N(CCNC(C2CCCC2(C)C)=O)Cc2ccccc2)O1 C(=O)(C1=CCCCC1)NCCCN(C1(CN(C)C(C2CCOCC2)=O)CC1)C C1(N(C(=O)CSCc2ccccc2)C)CN(C(=O)Cc2cncn2C)CC1O c1(C(N(CCOCCC(=O)NC(CC#C)C)C)=O)ccnc(O)c1 C1(C(=O)NCC2CC(NC(C(C)n3cnnn3)=O)C2)CCC(C)CC1 c1(C(=O)NCC2(O)CCN(C(C(C)(C3CC3)NC(C)=O)=O)C2)cccc(F)c1C N#CC1(C(=O)NCCn2cnc(C(=O)Nc3cc(=O)cc[nH]3)c2)CCOC1 c1(C(C)(C)C)nc(=NC(=O)C(=O)NCc2noc(C3CCC3)n2)s[nH]1 C1(C(=O)NCC(C)N(C)C(c2c(N)cnn2C)=O)CC2C=CC1C2 C1(c2nnnn2C2CCCCC2)(Nc2c(CC)cccc2)CCC(C)(C)CC1C N1(C(CC=C(C)C)=O)CCCC2(NC(=O)CN(C)S(N)(=O)=O)CCCC12 C12(C(=O)NC(C3CCN(C(c4cc(Cl)n(C)n4)=O)C3)C)CCN(CC1)C2 C=CCC(Cc1ccccc1)C(=O)NC(C)(CNC(=O)CCP(C)(C)=O)CC N1(C(C2CCN(CCC)CC2)=O)CCN(C(=O)C2=CCCC2)C(C2CC2)C1 C1(NC(C2C(CC)C2)=O)CCC2(CCCN2C(=O)Cc2ccc(F)cc2)CC1 N1(C(CC(C)CF)=O)CCN(C(=O)C=Cc2c(F)ccc(Cl)c2F)CC2(CC2)C1 Cc1cc(C(F)(F)F)c(C#N)c(N2CCN(Cc3cc(Br)cc(C)c3N)CC2)n1 CC1(C)CCC(C(N2CCC(C)(CNC(C3(C(F)(F)F)CCC3)=O)C2)=O)OC1 N1(C(CCN(CCCO)C(C2C(CC)CC2)=O)=O)CCC(F)(F)C(C)C1 N1(C(c2nc(C)oc2)=O)CCC2(CCCC2C(N2CCOCC2)=O)C1 C1(CNC(C=CCC)=O)CCCC2(CN(C(=O)CC3CC=CCN3C)C2)O1 c1(C(N2C3CC(CNC(c4cc(OC)ns4)=O)(OC3)C2)=O)cccc2ccnn12 C1(NC(CNC(CC)=O)=O)CCC(N(C)C(c2cc(C3(C)COC3)no2)=O)C1 Cn1c(C(=O)NC(CO)C(=O)NCc2cn[nH]c2)cnc1Cl c1(C(=O)NC2C3CN(C(C(C)(C)C(F)F)=O)CC32)csc2ncnc(O)c12 [N-]=[N+]=Nc1ccc(Cl)cc1C(=O)NCCCc1ccc(N(C)C)nc1 Cc1nn2cc(C(N3CCCC(CNC(=O)CSc4nncs4)CC3)=O)nc2s1 Cc1ccc(F)c(CC2(O)CCN(Cc3nn[nH]n3)C2)c1Cl C1(C(C)NC(CSCC(C)=O)=O)CCN(C(=O)Cc2nc(O)n[nH]2)C1 N1(C(=O)Cc2cscc2F)CCCC2(CCN(C(=O)CC3CC34CC4)C2)C1 CCC(CC)CC(=O)NCC1CCC(C)N(C(=O)C(c2ccccc2C)C)C1 CCCC(CCC)CC(=O)NC1CC2CN(C(c3cc(C4CC4)nn3C)=O)CC12 C1(OC)CN(C(c2cnoc2C(C)C)=O)CC1NC(C1CCCCO1)=O c1(NC(CCNC(C=Cc2cccc(C)c2)=O)C)ncnc2cc(F)c(F)cc12 c1(C(N2CCC(Cc3cn(-c4ncccn4)nn3)C2)=O)cnc2ccccc2c1 N1(C(CC(=O)OC(C)(C)C)=O)CCN(C(N2CC(c3cnc(C)[nH]3)C2)=O)CC1 c1(C(=O)NCC(=O)NC2CC2C(=O)NCC2CC2)cccc(Br)n1 C1(CC(C)NC(c2cc(Br)c[nH]2)=O)CCN(C(c2cn(C)c(O)n2)=O)CC1 CCC(CCC(=O)NC1(C2CN(C(C3CCCCC(=O)N3C)=O)C2)CC1)OC CC1(NC(=O)CCN2CCOC2=O)CCN(C(=O)CC2CC(=O)NC2=O)CC1 c1(C(N2CCC(F)(CNC(c3coc(Cl)c3)=O)C2)=O)coc2ccc(Cl)cc12 C1(C)(OC)CC(NC(=O)CC2(O)CCN(C(c3ccc(F)nc3)=O)CC2)C1(C)C C(C(=O)NC(C)(CNC(=O)C(O)Cc1ccccc1)C1CCC1)(C(C)C)SC c1(C(N2CCC(OC)(CNC(=O)Cc3cc(C)on3)C2)=O)ccc(F)cc1O c1(C(=O)NCCC(C(C)C)NC(C(F)=CC)=O)ccc(C(F)(F)F)cc1N N1(C(N2CCCC(N(C)C(=O)OC(C)(C)C)C2)=O)CCC2(CCC(C)(O)CC2)C1 C(=O)(CC(F)(F)F)NC1C=CC(CC(=O)NCC(C)OC)C1 N1(C(COC)=O)CCC(C2CCC2)(CNC(c2nnc(S)n2C)=O)CC1 N1(C(C(CCC)O)=O)CCN(C(C2(F)CCOCC2)=O)CC1CC1CC1 C(c1nc(CNC(CC(C)C)c2nnnn2C2CC(F)(F)C2)co1)=C(C)C N1(C(CCCCCOC)=O)CCOC2(CCN(C(=O)C(C)(C)CC(C)C)CC2)C1 Cc1cc(S(=O)(=O)N2CCCC(C)(C(N3CCOC(C)C3)=O)C2)ccc1Br C1(C(N2CC(C(C(=O)OC)OC)C2)=O)C2CCC(C2)C1C(F)F C1(n2cc(C(=O)OC)nn2)CC(O)C1(C)C.S1(=O)(=O)CCC2(CC2(F)F)N1 N1(C(C2(CCC=C)CC2)=O)CCC(CCNC(=O)C(N2CCCCCC2)C)CC1 N1(C(c2c(N)n(CCO)nc2)=O)CCN(C(=O)CC=C(Cl)Cl)C2CCCCC2C1 C1(C(C)NC(=O)CCC2CC2)CCCCN1C(=O)COCC1CCOCC1 C1(OCC)CC2CN(C(=O)C(CC(C)C)NC(=O)CC3(C#N)CC3)CC12 C1(N(C(C2(C)CC2)=O)CCO)CCN(C(=O)C=C2CCC(C(C)(C)C)CC2)CC1 C(C(=O)NCC1=CCCOC1)(C(C)C)NC(C(COC)C)=O c1(C(=O)NCC2C(NC(C3(CCOC)CCCC3)=O)C2)cc(C)ccc1O N1(C(c2c(NC)ccc(F)c2)=O)CCC2CC1CN(C(=O)CCC=C(C)C)C2 C1(NC(=O)CC2C=CCCC2)CCC2(CC1)CN(C(=O)C(=O)NCC(F)F)C2 c1(CC(=O)NCCCCCCNC(C2(C(CC)(F)F)CC2)=O)nnc2n1CCOC2 C1(NC(C2N(C(Cn3ncc(C)c3)=O)CC=CC2)=O)CN(C)CCC1O N1(C(=O)Nc2nc(-c3cnc[nH]3)cs2)CCCOC(CCCO)C1 S(=O)(=O)(c1ccc(NCCCS(N)(=O)=O)cc1Cl)N1C(CC)CCCC1 C1(C(N2C3C(NC(=O)CC4CCS(=O)(=O)C4)C(C3)C2)=O)CC12CCOCC2 C=CC1CCCCN1C(=O)COC1CC(NC(c2ccccc2SCC)=O)C1 C=CC(C)C(C)C(=O)NC1CN(C(c2cc(-c3nn(C)cc3CC)n[nH]2)=O)C1 c1(C(N2CC(COC)N(C(c3nccn3C)=O)CC2)=O)ccc2c(c1)COCO2 c1(C(=O)NCC(C)(C)CNC(=O)C(CC(F)F)C2CCC2)ccc(N)cc1F CC(F)(F)CCCC(=O)NCC1CC(NC(=O)C(F)(F)c2cnccn2)CC1O C1(CNC(c2cc(COC)on2)=O)CN(C(C2(OC)CCCC2)=O)CCO1 O=C(N=c1ccn(C2CN(Cc3ccc(I)c(F)c3)C2)[nH]1)c1c(F)ccnc1Cl c1(CC(N2CCC(N(c3c(C(=O)OC)ccnn3)C)C2)=O)nc(F)c(F)cc1F C1(C(=O)NCC23CC(NC(C4CC4(F)F)=O)(C2)C3)C2Cc3ccc(Br)cc3C12 C1(NC(C(c2ccccc2)OCC)=O)CCN(c2ncc(F)cn2)C12CCC2 N1(CCCC)CC2CCC1C(NC(=O)C(C)Oc1ccc(OC)cc1)C2 CS(=O)(=O)c1cccc(C(N2CC(NC(c3ccnc(Br)c3)=O)CC(F)C2)=O)c1 N1(C(c2nc(C(C)C)oc2)=O)CC(C2CN(C(C3SC4C=CC3C4)=O)C2)C1 CC(C(=O)N1CCC(O)(CNC(C2CCC3(CCC3)C2)=O)CC1)C1=CCCC1 Cc1nn(C(F)F)c(C)c1S(=O)(=O)N(C)CC1CCCCO1 C1(CN(C(=O)C(O)Cc2cnn(C)c2)C)COCCN1C(=O)CC1(C(F)F)CC1 C1(C(=O)NC2C(NC(c3ccc(F)c(Cl)c3F)=O)C2)CCc2cc(F)ccc2O1 C1(NC(CC#C)=O)CCc2nc(NC(c3cc(F)cc(Cl)c3)=O)sc2C1 c1(NC(COCCOCC#C)=O)cccc(CN(C(=O)C(C)CF)C)c1 CCC(C)(COC)CNC(C12CC1CCN2C(=O)CNC(C1CC1C)=O)=O C1(NC(c2c(C)ncs2)=O)CC2(C1)CN(C(C1CCC(F)(F)CO1)=O)C2 C12N(CC13CCCC3)C(=O)C1C(CCC)CN(C1)C2=O.C(C(O)CO)OC c1(CC(=O)N(CCC(C)NC(=O)Cn2ncnn2)C)csc2ccccc12 C1(C(N(CC(=O)N(C)C)CCC)=O)CN(C(=O)Cc2cnoc2)CC1(F)F Cn1ncc(C(N2CC(O)(C(=O)NCCCNS(=O)(=O)C(F)F)C2)=O)c1F N1(C(c2c(C)scc2)=O)CCC2CN(C(c3cnc4n3CCS4)=O)C2C1 c1(C(C)C)nc2c([nH]1)CC(C(=O)NCCN(C)C(c1nnn(C)n1)=O)CC2 c1(C(N(C(CNC(c2cnc(C)nc2C)=O)C)C)=O)scc2c1OCCO2 c1(C(=O)NCC(CC)NC(=O)CC2CCCS2(=O)=O)cccc2ncnc(O)c12 CC1(C)CC(NC(C2CC3CC2C2CC32)=O)CN(C(c2ccnc(Cl)c2)=O)C1 c1(C(=O)NC2CCC(NC(c3ccc(C)cn3)=O)C2)ccc2ccccc2c1O O=C(CCCC(F)F)Nc1cccc(NCCO)c1.c1(N2CC2=O)ccccc1 C(=O)(C1Cc2ccccc21)NCC1N(C(c2cc(C(=O)OCC)no2)=O)CCC1 c1(C(=O)NC23CC(CNC(C4(F)C(C)C4)=O)(OC2)C3)cc(S(C)(=O)=O)ccc1O c1(C(N2CC(CCNC(=O)CC3CCCC3)(OC)C2)=O)cn(C)c(=O)n1C c1(C(CO)Nc2cccc(C(=O)NCCCC(C)C)c2)cccc(Cl)c1Cl C1(CNC(CCSC)=O)C2CCC(C2)N1C(c1ncccc1C(F)F)=O c1(C(=O)NCC2C(NC(c3c(SC)csc3)=O)C2)cc2c(nc1O)CCCCC2 c1(OCC(N2C(CNC(=O)CSCC(F)(F)F)C=CC2)=O)ccc(F)cc1O C1(CNC(c2snc(O)c2Cl)=O)CCCC(CNC(=O)C(F)(F)C2CC2)C1 CC1CC(C(=O)N2CCC(C)(C)C2CNC(C2C3CC4C(C3=O)C24)=O)=NO1 c1(C(=O)NC2CCN(C(c3ccon3)=O)C2)cnn2cc[nH]c12 c1(C(=O)NC(C(C)NC(C2(C(F)(F)F)CCCC2)=O)C)cc(F)c(F)cc1N C1(C(=O)NC(COC(C)=O)CO)CC(C)CN1C(c1cc(C(C)C)[nH]n1)=O CC1CCN(C(c2c[nH]c(=N)s2)=O)CCN1C(c1ccc(CN(C)C)o1)=O N1(C(CCC(CC)C)=O)CC(C)(C)OCC1CNC(c1cc(C)c(Cl)c(C)c1)=O c1(NC(C2CC(NC(c3c(C)nn(C)c3)=O)C2)=O)cccc(Cl)c1C c1(C(=O)NC2CC2c2ccco2)ccc(-c2ccccc2F)cc1 C1(C(N2CCN(C(CC)=O)CC2)=O)(C(=O)OC(C)(C)C)CC2(CC2)C1 Cc1cc(C(F)F)nn1CC(=O)NC(CNC(c1ccc(C(N)=O)o1)=O)CC(C)C C1(C(=O)NC2CC2)CCCN(C(=O)CN2CCC2)CC1.C(=O)(CC(F)F)N(CC)CC CCC(C(=O)N(CC(=O)NC1CCN(C(C)=O)C1)CC)C(C)C n1(CC)cnc2ccccc12.Cc1noc(C2CN(C=O)C2)n1 c1(C(=O)NCCCCNC(C2CN(C(C)C)C2)=O)cnn(C2CC2)c1 C(c1cncn1C)=CC(=O)NCC1CC(NC(CN(c2cnn(C)c2)CC)=O)C1 c1(CC)ccc2ccccc2c1CCNC(c1cn[nH]c1)=O C1(CNC(Cn2c(C)cc(C)n2)=O)CCCCCN1C(=O)C(F)CC1CCC1 N1(C(C2(OC)CCCC2)=O)CC2C(N(C(=O)C=C3CCC(C)C3)C)C2C1 c1(C(=O)NC2CN(C(c3n(CC)ncc3)=O)CC2SC)nn(C)c(Cl)c1Cl c1(NC=O)nc(CC(=O)N(C2CCN(C(C3CC3C(F)F)=O)C2)CCO)cs1 C#CC1(C(=O)NCCCCC(=O)OC)CCN(OC(C2CCOC2)=O)C1 C12CCCC(C1)C(=O)N2.C1(OCCC(=O)NC(c2cccnc2)C)CCCOC1 C(C(C)(C(=O)N1CC(CO)(NC(C2(c3cc[nH]n3)CC2)=O)C1)OC)OC N1(C(C(C)(C)C#N)=O)Cc2ccc(CNC(=O)C=CSc3nc[nH]n3)cc2C1 CCCCC(C(=O)N1CCCC(CO)CC1)NC(c1cc(=N)[nH][nH]1)=O CN=c1[nH]c(=NCCc2ccncc2Br)[nH]c(=NC2CC3CSCC3C2)[nH]1 c1(C(=O)NC(CCOC)CNC(C2CC=CCC2)=O)cnn2ccc(OC)cc12 c1(CNC(=O)COC(c2csc3ccccc23)=O)cn2cnnc2cn1 c1(C(=O)NC2C(NC(=O)C=Cc3cn[nH]c3)C2)ncc2n1CCCC2 C(=O)(CCCCCC#N)NC(C(C)NC(c1cc(C)nc(C)n1)=O)CO Cc1nc(CO)sc1C(=O)NCCCCCC1CCN(C(=O)CC#N)CC1 N1(C(c2n(CCN(C)C)ncc2)=O)CCCC(c2cn(C3CCCC3)nn2)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCN(C(=O)CNC(C2CCC23CCC3)=O)CC1 S(=O)(=O)(c1ccc(-c2ccc(O)c(C=O)c2)o1)N.C1(N(C)C)CNCCC1CO C12(C(=O)NC(CC=C)CNC(=O)C(C)Oc3cccc(Cl)c3)CCN(CC1)CC2 c1(N2CC3C(CNC(C4CC(CC)(CC)C4)=O)C3C2)ncnc2cc(Br)ccc12 N1(C(C(CCC)CCC)=O)CCC2(CO)CN(C(=O)C(=O)NC(C)C)CC2C1 C=C(Cl)CCC(=O)NC1(C(=O)N(CCN2CC=CC2)CC)CC(CO)C1 c1(OC)ccc(Br)c(CN2CC3CC(C2)N3C(c2cc(O)ccc2C)=O)c1F c1(C(N2C(CC)C(C(N3CC(N4CC(O)C4)C3)=O)CC2)=O)cccc2occc12 CCCCC(CC)CC(=O)NC1CCCN(C(=O)CSCc2ccccn2)CC1 C1(CN(C(CCSC)=O)C)CN(C(=O)C(F)(F)Cc2ccccc2)CCO1 c1(C(=O)NC(C2(O)CN(C(c3nc(CC)sc3)=O)C2)C)cc(CO)oc1C C12(C(=O)NC3(CC=C)CC3)C(NC(=O)CC3CCOC3)C3CC1C2C3 C(N=c1nc(N2CC(C)=C(C)C2)c2sccc2[nH]1)c1c(N(C)CC)cccc1 c1(C(=O)OC(N(C)C)=O)ccccc1CN1CC2CC2C1 CCCC(C)(O)C(=O)NCCOCCOCCNC(=O)CSc1cnn(C)c1 C(CCCC(=O)N1CC(O)CC1C(N1CC(c2ccccc2O)C1)=O)NC(N)=O C1(NC(c2cnco2)=O)CCCC2CN(C(c3cnn(C4CCC4)n3)=O)CC12 Cc1c(Br)cc(C(=O)NCCCCNC(C2(C)CC(C)C2)=O)c(=O)n1C CCCCCCC(C1(N2CC(CNC(CSCC3CC(SC)C3)=O)C2)CC1)=O C(=O)(CC(C)C(C)(C)NC(N1CC(C)C(CN)CC1C)=O)OC N1(C(CSC)=O)CCC2(CC1)CN(C(c1ccc(Cl)c(Cl)c1)=O)c1ccccc12 C(=O)(CS(=O)CCC(F)(F)F)NC1CCN(C(C2C(CC)N(C)CC2)=O)CC1 c1(CNC(CC2C(C)C2)=O)ccc(CNC(C2CCCOCC2)=O)cc1 N1(C(c2n(CC)ncc2Cl)=O)CCCC(O)(CNC(=O)C(O)CSC)C1 N1(C(c2c(C)scc2)=O)CCC12CN(C(C1CNC(=O)CC1C)=O)C2 N1(C(C2(CC)CN(C(=O)CN(C)C(C)C)C2)=O)CC2(CCOC(=O)N2)C1 C(CCC(=O)NC1(C(=O)NOCCF)CCSC1)OCCOC C1(C(N(CCCCN(C(Cc2cc(C)no2)=O)C)C)=O)CCCC(CF)C1 N1(C(CC2(OC)CC2)=O)CCC(O)(C(C)NC(=O)Cc2cc(C3CC3)no2)CC1 c1(C(N2CCC23CN(C(c2cscn2)=O)C3)=O)cnc(Cl)cc1Cl c1(C(N2CC(NCc3cc(C)n(C)n3)C(C)C2)=O)ccc2c(n1)NC(=O)CC2 Cc1ccc2ncc(C(N3CCC4CN(C(c5cnn(C)n5)=O)CCC34)=O)n2c1 N1(C(=O)C(F)OC(F)(F)F)CC2(C(=O)NCC3CCCSC3)CC1CO2 c1(C(=O)NC2CCC(NC(=O)CSc3ccccc3Cl)C2)cccc2nncn12 CCC(CC)CCC(=O)N1CCC(C)(CNC(=O)C(O)P(C)(C)=O)C1 Cc1ccc(C(=O)NCC2CCCCC2NC(C2OCCCO2)=O)c(Br)c1 c1(CC(=O)NCC(CO)NC(C2CCC=CCCC2)=O)ccc2cnccc2c1 C(=O)(CCC(=O)N(C)CCN(C)C(c1c[nH]nc1Cc1ccccc1)=O)N(C)C c1(CC(=O)NC(CC)CNC(=O)C(F)CC2CC2)cc(C(F)(F)F)n(C)n1 N1(C(c2cc(OC)ns2)=O)CCC(NC(=O)Cc2cccc(Cl)c2OC)C(C)C1 N1(C(CN2CC(C)(C)C2)=O)CCCC(NC(C2CC2C(C)(C)C)=O)CC1 C(=O)(CC(C(F)F)NC(=O)C#CC(C)(C)O)NCCCCNC(CC(C)C)=O C1(C(=O)NCCCN(C(=O)C2=C(Cl)CC2)C2CC2)CC2CCC(C1)C2O c1(C(N2CC(NC(c3c(CC)n(CC)nc3)=O)C(C)C2)=O)cc2n(n1)CCOC2 c1(C(=O)NC(CC)CNC(C2(C)CCOC2)=O)nc(Br)c2n1CCCC2 C=CCCCCCCCCC(=O)NC(CNC(C1CCCN1N=O)=O)CCCC c1(NC(C(CC)C)=O)cc(C(=O)Nc2cccc(CN3CCCC3)c2)ncc1Br N1(C(c2c(OC)cccc2F)=O)CCN(C(=O)CC2CCCN(C)C2)CC12CC2 c1(NC(C2CN(C(=O)C=Cc3cccc(Cl)c3)C2)=O)cnc2ccc(Br)cn12 N1(C(Cn2c(C)ccn2)=O)CC2CCC1CC2NC(c1ccncc1Cl)=O c1(C(C)=O)cc(C(=O)NCC(C)(C)NC(=O)CC2CC2(Cl)Cl)co1 N1(C(C2CCC(C(C)C)CC2)=O)C2CCC1CN(C(C1CC13CC3)=O)CC2 C1(C(=O)NCC2CC(F)(CNC(CCC=CCC=C)=O)C2)COCCN1C C(=O)(C(CCC(=O)N(C)C)N1CCCC(N2CCOCC2)C1)NCC(=C)C CC(CC(C)(C)C#N)Nc1c(C(N)=O)c(C(F)(F)F)nn1C C1(CC)CCCC1(C)C(=O)NCC1(O)CN(C(C2COCC(C)O2)=O)C1 N1(C(CCCNC(=O)OCC)=O)CCC(N(C(C2(F)CC=CCC2)=O)CC)CC1 c1(C(=O)NCC2CC2CNC(c2ncncc2F)=O)c(F)cccc1Br c1(C(=O)NCCOCCCN(C(=O)Cc2cc[nH]c2)C)cccc2nnn(C)c12 c1(CCC(=O)NCC2(CNC(c3cc(C(N)=O)n[nH]3)=O)CCC2)cccc(F)c1 C1(O)(CN(C)C(C2(O)CCCC2)=O)CN(C(C2CSCCS2)=O)C1 N1(C(C(=O)NCCCSCC)c2nccs2)CCOC(CC2CC2)C1 C1(NC(c2c(C)oc(CNC(=O)C(C)CC3CCC3)n2)=O)CCCCC1(C)C C1(CSC2CN(C(=O)Nc3cnc(C4CC4)o3)C2)CCCC12CC2 N1(C(CNC(=O)NC2C(C)C2)=O)CCOC2(C1)CN(C(c1cc(O)n(C)n1)=O)C2 FCCN=C(NCc1cc(Cl)ncc1Cl)NCC1CC2(CCC2)C1 c1(OC)cccc(C(C)CNCCCc2ccccc2F)c1 Cc1cc(C(=O)NC2(C)CC(NC(=O)CC34CCC(CC3)CC4)C2)nc(C)c1 c1(C(N(CCC)CCNC(c2ccc(C3CC3C)o2)=O)=O)ccc2ncccc2c1 c1(-c2nc(C(CC(C)C)CS(C)(=O)=O)on2)cccc2ccncc12 C12(C(N3CCC(CNC(c4n(CC)ccc4)=O)(CO)C3)=O)CCC(C)(CC1)OC2 C1(C(N2C(CC#N)CN(C(=O)C(O)CCl)CC2)=O)CCC2CNCCC2C1 c1(C(=O)NCC(C2CCOC2)NC(c2cnc(C3CC3)[nH]2)=O)ccc(OCF)nc1 CCCC(C(=O)NC12CC(CNC(=O)C(C(=O)OC(C)(C)C)N(C)C)(C1)C2)OC c1(C(N2CC(CNC(CCC)=O)C(C(F)(F)F)C2)=O)c(S(C)(=O)=O)cnn1C C12CN(CCO1)C(=O)CC1(CC1)CC1C(C1)NC2=O.c1(SCO)ccccc1 CCC(F)(F)CC(=O)N(C1CCCCC1NC(C1C(Cl)(Cl)C12CC2)=O)C c1(CCC)cc(C(=O)NCC2(CNC(=O)CCC(C)N(C)C)CC2)cc(O)n1 N1(C(CN(C(CSCC=C)=O)C2CC2)=O)CC(F)(F)C(F)(F)C1 c1(CN2CCCC(C(N3CCS(=O)(=O)CC3)=O)CC2)cc2c(s1)CCCCC2 C(C(C)CC(=O)NCc1cc(C(=O)NC(CO)CCC2CC2)n(C)n1)OC C(=O)(C(F)C(C)(F)F)N(CCCNC(C1CC12CCC2)=O)C(C)C N1(C(C2OCCN(C)C2)=O)CCC(C)(C)C1C(=O)NOCCC1CC1 N1(CC(N2C(CN(C(=O)Cc3ccc(Cl)cn3)CC)CCC2)=O)CC(=O)NC1=O N1(C(C2(CC)CCOCC2)=O)CCC2(CC(NC(c3sc(C)c(C)c3C)=O)C2)C1 CCCCC(C)CCC(=O)N1CC2CC1CN(C(c1cnn(CCO)c1N)=O)C2 C1(NC(C(C)N(C)C)=O)C(C)CCN(C(c2cc3ncccc3[nH]2)=O)C1C c1(OC)cc(OC)cc(C(N2CC(NC(c3ccc(F)o3)=O)C(C)C2)=O)c1 c1(C(N2C(CNC(CCC=C)=O)C(CC)CC2)=O)cc(Cl)cnc1O N1(C(c2c(C)cc(F)s2)=O)CCC(CO)(NC(c2ccc(O)nc2)=O)CC1 N1(C(C2(F)CCN(C(C(C)OCCOC)=O)C2)=O)CC2CCCC(C1)N2C c1(N2C(CNC(CCC(C)OC)=O)C(C3CC3)CC2)nc(C)nc2n[nH]cc12 C#Cc1ccc(C(=O)NCC(C(C)(C)C)NC(C2(CC)CC2)=O)o1 C1(C(N2CC(C(C(=O)O)OC)C2)=O)CC(=O)N(c2cccc(C(F)(F)F)c2)C1 C(=O)(CCCCCCCC(=O)N(CCCNC(=O)CC1(C)CCCCC1)C)OC C(=O)(C#CC1(C)CCCO1)NCC1(C)CN(C(c2nc[nH]c2C(F)(F)F)=O)CCO1 C(=O)(C(=O)C=Cc1cccs1)NCC(C)N(C)C(c1ccnn1C)=O C1(C(N(C(C)C)CC)=O)CCC(n2cc(C3CCN(C)C3)nn2)C1 c1(CCN(C(=O)C(=O)N(C)C)CCNC(C2C(C)C2C)=O)ccccc1 C1(CCCC)CN(C(C2CC(C(F)F)(OC)C2)=O)CCN1C(=O)C(C)N(C)C CC1CC(C(N2CC(CNC(c3cn(C)c(=O)cn3)=O)C2)=O)CC(C)C1 C#CCCN=C(NCC1(C)CC=CC1)NC1COC2CC1C2 c1(CC(N2CCC(N(C(=O)C(F)n3cccn3)C)CC2)=O)cnn2c1CCCC2 N#Cc1cc(NC(C2CC23CCN(Cc2cn[nH]c2)C3)=O)ccc1F c1(C(=O)NCC(CO)NC(CC(CCC)CCC)=O)c(C)ccc2ncccc12 C1(C(N(CCNC(CCN(C(C)=O)C)=O)C)=O)Cc2cc(C)ccc2O1 c1(C(N2CC(CC(=O)NCCC(C)CO)OCC2)=O)ccc(C#N)cn1 CCC(CC(=O)NCC(C)(C)CNC(C1(N(C)C)CC1)=O)C1CC1 O=C(CC1C(=O)Nc2ccc(F)cc21)N1CC(C2(NC(c3cnc[nH]3)=O)CC2)C1 C1(NC(COC2CC(NC(C3CC(OC)(OC)C3)=O)C2)=O)CNC(=O)C12CC2 c1(C2C(OCC)CC2O)ccc(S(=O)(=O)NC2(CO)COC3(CCC3)C2)c(Cl)c1 C(=O)(CC(C)(C)C(=O)N1CC(C)C1C(N1CC2COC(=O)C2C1)=O)OC c1(C(=O)NCCCNC(C2CCC2)=O)cccnc1-c1ccccc1 N=c1[nH]c2ncc(C(=O)NCC#CCNC(c3ccc4sccc4c3)=O)cc2s1 N1(C(c2scc(COC)c2)C(=O)NC2(C)CC2)CCCN(C)CC1C N1(C(c2cn(CC=C)nn2)=O)CCC(NC(=O)C(C)(C)CC)C(O)C1 C1(NC(C(CC)N(COC)CC)=O)C2CC3CN(C(=O)C(C)=C(C)C)C1C3C2 CC1(C)CC2(CN(C(C3CN(C(=O)C(C4CCOCC4)F)C(C)(C)C3)=O)C2)C1 S(=O)(=O)(c1ccc(NC2C=CCCC2)cc1Br)N1CCCC(C)(CCC)C1 Cc1c(CC(=O)N(CC(C)NC(C2CC3CC3C2)=O)C)nc(Br)n1C Cc1nc2cccc(C(N3CCCCC(NC(=O)C(C)C(C)O)C3)=O)n2n1 c1(CNCCC(C)N(C)C)cc(Br)ccc1Br C1(NC(C=CC=CC)=O)CCC12CCN(C(c1c(F)ccc(Br)c1F)=O)CC2 c1(CNC(=O)CCC(=O)NC(C23C(CN(C(C)=O)C2)C3)=O)cc(Cl)ccc1I.NCC N#CCCCC(C(=O)NCCCF)N1CC2CCCC(C1)N2CC(=O)NCCS c1(C(=O)NCCN(C(=O)Cc2cccnc2Br)CC)c[nH]c2cc(C)ccc12 N1(C(CCC=CC(C)C)=O)CCC2(CC1)C(N(C(=O)CC(C)(C)O)C)CS2(=O)=O CC1CN(C(C2CN(C)CC(C)O2)=O)CC1(C)C(=O)NCCCc1cnn(C)c1 Cc1cnc(CNC2CCCCC2C(=O)Nc2ncc(Br)cc2C(F)F)cc1Br N1(C(C(CC)(F)F)=O)CCC(CNC(=O)Cc2ccc(C)o2)C(C)C1 N(C(=NCCCCc1ccccc1)NCc1ccnn1C)C1CC(OC)C1 c1(C(=O)NC2(C)CCN(C(C(C(C)SC)O)=O)CC2)cnnc2ccccc12 Nc1cccn(CC(=O)N(c2cccc(F)c2)C2CCC2)c1=O Cc1[nH]cc(C(=O)NC2CC(F)(F)CC2NC(=O)C(N)=O)c(=O)c1Cl c1(C(CCSC)NCC(=O)OC(C)=O)ccc(Br)cc1 N1(C(C(C)(C)C#N)=O)CC(C2CCCCN(C(c3ccc4sncc4c3)=O)C2)C1 c1(CC)cc(C)ccc1C(=O)NCC(CNC(c1ccccc1CC#N)=O)OC c1(C(N(CCNC(=O)C(C)(O)C2CC2)CC)=O)snnc1C(C)C c1(C(c2n(CC(=C)C)nnn2)NCCc2ccc(Cl)s2)ccc(OCCC)nc1 C#CCCN=C(NCC(C=C)OC(=N)O)N1CCC(OC)C1.c1(NCCCl)ccc(O)cc1 CCC(C)C(CNC(=O)C(F)CC1CN(C(=O)Cn2ncn(C)c2=O)C1)CO c1(OCC)cc(C(N2CSCC2C(=O)NCc2cc(Cl)no2)=O)on1 c1(C(=O)NC2CC(CNC(Cc3c(C)ncs3)=O)C2)cnc(C(F)F)nc1 N1(C(COCC(=O)NC)=O)CCN(C(=O)Cc2ccc(SCC)cc2)C(C)C1C c1(SC)cn(C)nc1C(=O)NC1CCC(CNC(c2nc(C3CC3)cs2)=O)C1 C1(O)(CNC(c2c(SC)scc2)=O)CCN(C(C2(C)CC(C)C2)=O)C1 c1(CCC(=O)NC(C)CC2CN(C(=O)CCC3CC3(Cl)Cl)C2)cn(C)cn1 c1(CC(=O)N(C(CN(C(CC2(COC)CCCC2)=O)C)C)C)nncnc1O c1(OCC)cccc(C(=O)NCC(C(C)(C)C)NC(=O)OC(C)(C)C)c1[N+](=O)[O-] C=CCC(C(=O)N1CCC1CNC(c1cnc(CC)[nH]1)=O)NC(C)=O C1(C(=O)NCc2cn(C3C(C(=O)O)C3)nn2)COCCN1CC(F)F Cc1cc(C(=O)NCCc2n[nH]cc2C(=O)NC(C)CCC2CC2)ncc1N CC(C)CC(C)CC(=O)NC1C2CC1N(C(=O)Cn1cccn1)C2 c1(C(N2CCC(NC(C=NOC)=O)C2)=O)ccc(C)c(F)c1 C1(NC(CSCC(N)=O)=O)COCC1CNC(=O)COCC1CCCOC1 N1(CC)CCOCC1C(=O)NCCn1cc(C(=O)NCC(CC2CC2)OC)cn1 Cc1cccc(O)c1C(N1CC2(CCC2NC(c2cnn(C)c2)=O)C1)=O CC(CCC(=O)N1CCC(NC(=O)C2CC2)C1)NC(=O)CC12CCCC1C2 c1(CNC(C(C)Oc2ccccc2Cl)=O)cncc2n[nH]cc12 c1(NC(C)C)ccc(C(=O)NCCCCCNC(=O)CC2(O)CCC2)cn1 n1(CC(=O)NC(CCN(C(C(C(CC)O)(C)C)=O)C)C)ccc(=O)c([N+](=O)[O-])c1 c1(OC)ccc(NC(C2CCCN2C(c2ccnc(Br)c2)=O)=O)cc1S(N)(=O)=O N1(C(C(CC2CCC2)OC)=O)CC(N(C)C(c2cc[nH]c2)=O)C(C)(C)C1 c1(C(C(=O)NCCCC)N(C(C#C)C2CCC2)C)cc(Cl)c(Cl)s1 c12sccc1SC2.C1(N(C(C=CC=CC)=O)C(C)=O)CCOC1 CN1CCN(C(c2n[nH]c(O)n2)=O)CC1C(=O)NCC1CC(F)(F)CO1 C(=O)(CC(CNC(=O)NCCCC1CCOC1)CC(C)C)OC C1(F)(C(N2CC(CC)C(NC(=O)CCC3CCOC3)C2)=O)C(C)(C)C1(C)C N1(C(CSCC(CNC(C(C)N2CCCC2)=O)(C)O)=O)CCOCC1 N1(C(CCNC(=O)NC)=O)CC2CC1CN(C(C1CN=C3N=CNN3C1)=O)C2 N1(C(CC2C(C)CCC2)=O)CC(C2CCN(C(C3(O)CCCCC3)=O)CC2)C1 C1(CNC(NC(CCC=C(C)C)C)=NCC2CC2)COC(C)(C)CO1 N1(C(c2n(C(C)C)ncc2)=O)C(CNC(=O)CNC(N)=O)CC2COCC12 Cc1nn(C)cc1C(O)C(=O)NCC(C)(C)NC(=O)CC1CCCCN1C C1(N(C(=O)CCc2cccc(Cl)c2)C)CN(C(=O)CC2CC2(Cl)Cl)CC12CC2 C1(CC)(NC(c2ncn(C)c2C)=O)CCCN(C(=O)CC2(O)CCCOC2)C1 CC(CC(=O)NCC12CCCC1CCC2)C(C)(C)NC(C1CCCN1C1CC1)=O c1(OC)ccc(Cl)c(C(=O)N(C2CCCN(C(=O)CC(C)OC)C2)C)c1F Cc1cnn2cc(C(N3CCCC4(NC(=O)CC5CC=CC5)CC4C3)=O)cnc12 C(=O)(N1CCC(C(=O)NOCC2CCCO2)O1)n1ccc(CC)n1 C(CCS(C)(=O)=O)(C(=O)OC(C)(C)C)NC(=O)ONC(CCO)C(F)(F)F c1(OCC(=O)N(C)CCNC(=O)CCC#N)ccc2c(c1)CCC(=O)N2 C(=O)(CCCC(=O)OC)N1CCC(N(C(=O)C(C)CC2CCCO2)CCC)CC1 c1(CC(=O)N(C2CCN(C(C3CC(C)(C)O3)=O)C2)C)nccc2ccccc12 C1(C(=O)NCC(=O)NC)CC(F)CCN1C(c1ccsc1C)=O N1(C(CC=C)=O)CCC2(CC1)CCN(C(=O)C(C)CN1CCOCC1)CC2C C1(NC(C2(C=C)CC2)=O)CC2CCC1C(NC(=O)C(C)Cc1cccc(Cl)c1)C2 c1(C(=O)NC(CC)CNC(=O)OC(C)(C)C)cc(CN(C)C)on1 C1(C(=O)NCC=CC(=O)NCCC2CCOC2)CCC2CC12 N1(C(c2c(C)cn(C)c2)=O)CCC(C)C(NC(c2ccncc2Cl)=O)C1C c1(OC)nc(C(F)(F)F)c(C(=O)N(C2CCN(C(=O)CSC3CC3)C2)C)s1 C(CCCCC(=O)N(C1CCCN(C(C2(C)CC(OC)C2)=O)CC1)C)OC N1(C(c2ccc(C(C)C)nc2)=O)CCC(C2CC2NC(=O)C=C(Cl)Cl)CC1 Cc1cc2occ(CC(N3CC(O)(C(C)NC(C4CC4(Cl)Cl)=O)C3)=O)c2cc1C Cc1cc2ccccc2cc1C(=O)NC1CN(C(=O)C(C)c2ccon2)CC1C C(C)(CNC(=O)C(=Cc1ccccc1)C)(C(C)C)NC(CCCN(C(C)=O)C)=O N1(C(CCC(=O)NCCC)=O)CCOCC(C)(CNC(=O)C(C)c2ccsc2)C1 N1(C(C(CNC(C(CC)C(=O)OC)=O)C)=O)CCc2cncnc2C1 Cc1cc(-c2nccn2CC2C=CC=NC2=O)sc1-c1ccccc1C(N)=O N1(C(Cc2cc(C)[nH]n2)=O)CC(N(C(=O)CCc2cc[nH]n2)C)C(F)C1 c1(C(c2nnnn2CSc2ccccc2)NC(C)CCCO)nnc2n1CCC2 C1(NC(C2CC(C)(NC(COCC(=O)OC)=O)C2)=O)CC2(C1)CC(CO)C2 C1(CC(=O)N(CCC)C2CC2)CN(C(c2[nH]ccc2COC)=O)CCC1C C(C)(CCC(=O)NC(C)(CC)CCNC(C1(OC)CCC1)=O)N.C(COC)O C1(CN(C)C(c2ccc(Br)nc2)=O)CN(C(C2CC2C2CC2)=O)CCO1 C1(OC)(CNC(C2CCCCN2C(C)=O)=O)CCN(C(=O)C=CC2CC2)CC1 C1(C(N2CCC(CNC(=O)C(c3ccccc3)F)C2)=O)CCC(F)CC1 N1(C(=O)Cc2nccs2)CCCN(C(c2cn(CCF)nn2)=O)C(CO)C1 S(=O)(=O)(c1cc(F)cc(F)c1)N1C(C(=O)N(C2(CC)COC2)C2CC2)CC2CC21 C(=O)(CC(O)CCC)NC1(CC=C)CCN(C(=O)Nc2ccccc2F)C1 N1(C(C2CCN(CCC#C)CC2)=O)CCC(C)N(C(=O)Cc2cccnc2)CC1 O(NC(=O)C(C(C)O)NC(=O)CC1CC1COC)CC=C C(N=c1nc(N(C)CC2COC(=O)N2)c2[nH]ccc2[nH]1)c1scc(C)n1 c1(C(=O)NC2CN(C(C(CC=C)C(C)C)=O)CC23CC3)cccc2c1CNC2=O C(=O)(CC(C(F)F)NC(C1CSCN1C(C)=O)=O)N(CCCC)CCO C1(CC=C)(NC(C2CC(C(F)(F)F)C2)=O)CCCN(C(C2CCC3(C2)N=N3)=O)C1 C(=O)(CCCCCN(C)C(C1CN(C2CCC2)C1)=O)NC(C)Cc1ncon1 c1(C(=O)NC(CCCCNC(CCC=C=C)=O)C)ccn(CCO)c(=O)c1 C1(C(N2C(C(C)C)CN(C(=O)CC3CC3(C)C)CC2)=O)CCc2ccccc2N1 c1(C(=O)OC)cc(N(C)CC2CCCCN2C(=O)C2=CCCC2)cc(C#N)c1 C1(NC(C(C)(C)N(C)C)=O)CN(C(C2CCC=CCC2)=O)C2CCCCC12 S(=O)(=O)(c1ccc(N2CC3CC2CS3)c(Br)c1)N1CCCC(C(C)C)C1 c1(CNC(C2(C(C)C)CC2)=O)ccc(CCNC(C2(C)CS(=O)(=O)C2)=O)cc1 c1(CNC(c2cnc(-c3ccncc3F)cn2)=O)ccccc1F CCCC(C#N)C(=O)NC1CC(CCC(=O)NC2CCCCCC2F)C1 C(CC(=O)NCC(C)(C)C1CCCC1)N(C(=O)C(C)N1CCCC1)CC C1(C(=O)NCCC2CCCCCC2)C2CC2CN1C(=O)C=CC(F)(F)F c1(CC)oc2ccccc2c1CC(=O)NCC1CCN(C(=O)C=CSC)CC1C c1(C(=O)NC2C(OC)CN(C(C3CCOC(=O)N3)=O)C2)cc(C)cc(F)c1 N1(C(CC2CC(=C)C2)=O)CC(NC(=O)C(=O)NCC(F)F)CC1C c1(C(=O)OC)cnc(N2CCN(C(=O)C(c3cnn(C)c3)O)CC2C)nc1C c1(C(N(CCC2N(C(C(COCC)C)=O)CCCC2)C)=O)n[nH]c2ccccc12 c1(C(=O)NCC(CC=C)NC(c2ccc(CCC)s2)=O)ccc2c(c1)OCC2 C1(C(N2CCC(CNC(=O)CC3CCC(C4CC4)O3)CC2)=O)(CC)CC(F)(F)C1 N1(C(C(C)Sc2ccccn2)=O)C2CCC1C(NC(=O)CCc1ccc(Cl)s1)C2 N1(C(CCOC)=O)CCN(C(C2CCC(F)(F)C2)=O)C(C2CCC2)C1 Cc1cnc(C)c(NC(C2CN(C(=O)C(C(C)C)N(C)C(C)=O)CC23CC3)=O)c1 C1(C(N2C(CNC(C(C)n3ccnc3)=O)CC(O)C2)=O)CC12CCSCC2 Cc1n[nH]c(C)c1CC(=O)NC1(CNC(C2CC23CC3)=O)CCOC1 C1(C(C)NC(c2c(C)n[nH]c2)=O)CCCN(C(C2(C)CSC2)=O)C1 c1(C(=O)NC(CCOC)CNC(c2c(C)n[nH]c2C)=O)cnc2cc[nH]c2c1 Cc1ccc(F)cc1CCNC(=O)COc1cccc(F)c1 C(CC(=O)N1CCC(CNC2CCC(C)(C)CO2)CC1)(C(N)=O)NC(C)=O c1(C(=O)NCC=CCNC(CC2(OC)CCCCC2)=O)occ2c1CCC2 CN1C(=O)NCC12CN(C(C1CN(C(C3(C)COCCO3)=O)CC13CCC3)=O)C2 c1(CC)cc[nH]c1C(=O)NCc1nocc1C(=O)N(C1CCCC1C)C C1(NC(C(C)O)=O)CCOC12CCN(C(=O)Cc1cncn1C1CC1)CC2 C1(CCNC(CC(=O)NCC)=O)CN(C(c2cncc(C)n2)=O)CCO1 c1(C(N(C(CNC(C2CCOCC2)=O)C2CC2)C)=O)ccc(C2CC2C)o1 C1(CC)CN(C(=O)C=CCN(C)CC)CCC1CNC(C1CCCC1O)=O C1(NC(c2c(Cl)cn(C)n2)=O)CN(C(C2CC(C)(C)O2)=O)CCC1CO C(=O)(C(C(C)(C)C)N1CCCCC1=O)NCC1N(C(CCC=C(C)C)=O)CC1 C#CCCN=C(NCCC(C)(C)S(C)(=O)=O)NC1Cc2ccccc21 N1(C(c2ccnn2C)C(=O)NC)CCCC2(C1)OCc1ccccc12 Cc1noc(C)c1C(C)(C)C(=O)OCCn1ccnc1C CC1(C)NC(=O)CC1C(=O)NC1COCC1NC(C1(CC2CC2)CCC1)=O c1(NC(C2CN(C(C(F)=CCC)=O)CC2F)=O)ccc2ccncc2c1 c1(OC)nc(C)ncc1C(=O)NCC1C2CC1N(C(C1CCCC(C)(C)C1)=O)C2 N1(C(C2CCC(C)C2)=O)CCCC(N(CCO)Cc2cnon2)C1 N1(C(C2(F)CN(C(CC(C)F)=O)C2)=O)CCC2(CCOCC2)C1 n1(CC)ccc(C(=O)NC2CCC(C)(CNC(=O)CCN3CCC(O)CC3)C2)c1C c1(C(N2CCC(N3CCN(C(C(C)C(F)F)=O)CC3)C2)=O)cc(S(N)(=O)=O)cs1 c1(N2CCC(C)(CSC)CC2)nc2ccc(Cl)cc2c(=NCCCN(C)C)[nH]1 Cc1ccn(CC(N2CC(NC(C3CN(S(C)(=O)=O)C3)=O)CC2CO)=O)c(=O)c1 C1(NC(Cc2c(C)scc2)=O)CC(C(=O)NCC(F)(F)C(C)C)C1(C)C N1(c2nc(SC)nc(C)c2)CC2CC(NC(c3ncc(Cl)s3)=O)CC2C1 C12(NC(CNS(NC)(=O)=O)=O)CCOCC1CN(C(c1sccc1C(F)F)=O)C2 N1(C(C2C(CCOC)C2)=O)CCC(C=CC(=O)NCC(O)CN2CCC2)CC1 O(NC(=O)C(CN=[N+]=[N-])NC(C12CCCC1C2(F)F)=O)CC#C Cc1nc2ncnn2cc1C(N1CC(C)N(C(c2ccc(C#N)[nH]2)=O)CC1C)=O c1(C(N(C2CCN(c3nnc(C(F)F)s3)C2)CC)=O)ccc(C)nc1Cl c1(CN2CC(NC(c3ccc(C)c(O)c3)=O)C(O)C2)ccc2ncnn2c1 N(C(=NCCCc1cccc(F)c1)NCCF)C1CCCN(CC)C1 C(C)(C)(CCCC(=O)Nc1cncc(CO)c1)NC(CN1CCC(C)C1)=O CCCS(=O)(=O)CC(=O)NC1CCN(C(C2(c3ccno3)CC2)=O)C12CCC2 c1(C(C)NC(CC(C)NC(C2N(CC)CCC2)=O)=O)ccc(F)cc1 n1(CC=C)nnnc1C(c1cc(C(=O)OC)co1)NCC(C)COC C(=O)(C(O)CC(F)(F)F)NC1C(SC)CN(C(c2ccnnc2)=O)C1 C1(N(C(C(CC)F)=O)CC(C)C)CCN(C(c2cc(-c3cccs3)on2)=O)CC1 C1(COC)(CNC(=O)CC2CCN2C(=O)CC2(C#N)CC2)CCCCO1 c1(C)ccnc(O)c1.c1(CCNC(c2nnnn2C2CC2)COCC)noc(=O)n1C C=CCC(C)(O)C(=O)NC1CCC(CC(=O)NC2CCC3CC23)C1 c1(C(C(=O)NCC2CC(NC(c3nc(OCC)oc3)=O)C2)(C)F)ccccc1F N1(C(CCCc2cc(C)no2)=O)CC(NC(C2CC3(CCOC3)C2)=O)C2(CC2)C1 C1(CCC)CCC(CN(C(c2cc(O)ncn2)=O)CC)CC1 C(=O)(C1COc2ccc(Cl)cc21)N(CC(C)(C)NC(C(S(CCC)(=O)=O)C)=O)C N1(c2ncc(C(=O)OCC)s2)CCOCC(C(=O)NCC2CCCC(F)(F)C2)C1 c1(NC(CC)CSC)[nH]c(=NC2CC2C(C)C)nc2c1ncn2C(C)C C(=O)(C1=COCC1)NCC(CCOC)NC(=O)C(C)SCc1ccccc1F C1(CNC(CCP(C)(C)=O)=O)CCN(C(c2ccc(CO)nc2)=O)CCC1(F)F c1(N2CC(C(C)NC(N3CC(C)C=C(C)C3)=O)C2)ccc([N+](=O)[O-])cc1 O=C(C(O)C1CCc2ccccc21)N1CCOC(C(F)F)CC1 CCCCC(CCC)CN=c1nc(N2CCC(O)CC2)c2c([nH]1)CCCCC2 N1(C(C2(CC)CCOCC2)=O)CC(NC(=O)C(CO)OC)C2(CC2)C1 C(C(O)CC(C)(C)CO)NC1C(c2n(C)cnc2)C1 c1(C(=O)NCC2(O)CC(NC(CC(CC)C3CC3)=O)C2)cnc2cnccc2c1 c1(C(=O)NC2C3CN(C(c4c(N)cnc(Cl)c4)=O)CC32)ccc(O)c([N+](=O)[O-])c1 Cc1nn(C)c(C)c1C(=O)NCC1(CC(N2CCCC(C#N)C2)=O)CC1 O(NC(=O)C(C(C)CC)NC(=O)C(CC(C)C)OC)CC=C N1(C(COCCCC)=O)CCC(NC(c2ccccc2OC)=O)C(F)C1 CC1C(NC(C2(CF)CCC2)=O)CCN1C(C1CCN1Cc1ccccc1)=O C(=O)(C1=CC(C)(CC)C1)NC1(CNC(C2C(CCCC)CCC2)=O)CC1 CCCCC(CO)NC(=O)CCN(C(=O)CC1CCC(=O)C1)C1CC1 c1(C(=O)NC(CC)(CNC(=O)C(C)C(C)COC)CC)ccc2c(c1)NC(=O)C2 N1(C(C(C)(C)OC)=O)C2CCC1(CNC(=O)C(C)(C)c1ccno1)CC2 c1(C(N(C(CC)CO)CC)=O)coc(CNC(=O)Cc2cccnc2)n1 C1(CNC(C(n2ncc(C)c2)C)=O)(NC(c2c(C)noc2C)=O)CC2CCC1C2 N1(C(=O)NC(C#C)Cc2ccc(F)cc2)CCC(O)(CCCO)CC1 c1(C2(C(=O)Nc3ccc(CC)cn3)CC2)ccccc1C#N N1(C(CCCC#CC)=O)CCC2C(CCN2C(c2cc(Cl)n(C)n2)=O)C1 Cc1cc2c(CC(=O)NCC(F)CNC(=O)Cn3cc(C(F)F)cn3)csc2s1 C1(Cc2cc(C)[nH]n2)CCN(NCC(CN2CCCC2)C(=O)O)C1(C)C C(=O)(C1COc2ccc(Cl)cc21)NCC1(C(=O)NCCC2CCC3CC23)CC1 CC(O)(CC(F)F)C(=O)N1CCN(CCNC(=O)C(N)=O)CC1 C1(NC(=O)NCc2cccc(C(C(C)C)(OC)OC)c2)CCOC12CCOC2 C(CCCC(C)(C)NC(=O)Cc1cnoc1)NC(C(C)c1ccco1)=O c1(C(=O)Nc2ccc(CCO)cc2)cnc2nc(Cl)ccc2c1 C(=O)(C(C(C)C)NC(=O)OC(C)(C)C)NCCCNC(c1c(CC)cco1)=O c1(NCCC2(CSC)CC2)ncccc1S(=O)(=O)N1CC(C)C(C)C1 C1(NC(C2CN3CCN2CC3)=O)CN(C(=O)COc2cccnc2)CC12CCC2 c1(C(=O)OC)ccc(OC)cc1Br.C12C3CC3CN1C(=O)N2 c1(C(=O)NCCOCCN(C)C(c2csc(O)n2)=O)nccc2nn[nH]c12 C1(NC(C(CC)(F)F)=O)CC2CCCC(C1)N2C(c1ncncc1C#N)=O C(=O)(CC(F)(F)Br)NCCOCCN(C(=O)C=CC=C(Cl)Cl)C C1(C)(C(=O)NCCCC(C)NC(c2c(C)ncn2O)=O)CCS(=O)(=O)CC1 C1(NC(C(C)N2CCC2)=O)CCC2(CC1)CC2NC(c1cc(CO)on1)=O N1(C(CC=CC=C)=O)CC=C(CNC(=O)C(C)c2cccs2)CC1 c1(C(N(CC(C)N(C)C(c2cnc(O)o2)=O)C)=O)n[nH]c2c1CS(=O)(=O)CC2 C1(C)(NC(c2c(COC)noc2)=O)CCN(C(=O)C(c2ccc(C)cc2)(F)F)C1 c1(C(=O)NC(C(C)C)C(C2CCCCC2)NC(C2CCC2)=O)ncc(F)cc1F C1(C(=O)NC2CCN(C(C(c3ccc(F)cc3)=O)=O)C2)CCC12CCOCC2 c1(C(=O)NC2CC(F)(CNC(CCOCCN(C)C)=O)C2)c(F)cccc1F N1(C(C2N(CC)CCC2)=O)CC(F)CC1C(N1CCC(C(C)(C)O)C1)=O c1ccc2c(c1)CCC2.Cc1[nH]c(C)c(C(=O)OCC2CCC2CC(=O)O)c1C c1(C(N(C)CC2(C)C(NC(c3c(C#C)c[nH]n3)=O)CCC2)=O)cc(C)nc(O)n1 c1(NC(N2CCN(c3c(C)n[nH]c3C)CC2)=O)ccn2cc(Br)nc2n1 C1(C(N(C)CCNC(c2cnsn2)=O)=O)CCC(c2nc[nH]n2)CC1 O=C(C1=NOCC1)NC1CN(C(c2cccc(C(F)(F)F)c2)=O)CC1O CC1CN(CC(=O)Nc2noc3c2CC(C(C)(C)C)CC3)Cc2cccc(Br)c2O1 CC1CCCn2c(CC(=O)NCCNC(=O)Cc3ccccc3)cnc21 C12(CC(=O)NC3(CNC(CC4C(C)(C)C4)=O)CCOCC3)CCCCC1C2(F)F c1(NC(C2CCCN2C(c2ccc3ccccc3n2)=O)=O)cc(F)c(F)c(Br)c1 C1(C(=O)NCC(CC=C)NC(C)=O)CCC(NC(=O)CCC(=O)NC)CC1 C1(C(=O)NCCC(CC)(O)CC)CC(N=[N+]=[N-])CN1C(=O)CC1CC(C)=NO1 C#CC1(C(=O)NC2(C=C)CCCCC2)CCN(C(=O)Cc2cnoc2)C1 C1(C(=O)NCC(CNC(COc2cn(C)nc2)=O)O)C(F)(F)C12CCC2 C=CC1(C(=O)NCc2c[nH]nc2C2CC2)CCN(C(c2cnc(N)cn2)=O)C1 C1(NCc2ccc(CC(C)C)cc2)CCS(=O)(=O)CC1 Cc1cc(C)c(C(=O)NC2CC2CNC(=O)C(C)Cc2ccco2)s1 C(CO)(CCCCNC(=O)C(C)(C)F)NC(c1cccc(SCC)c1)=O N1(C(C(C)=C(CC)C)=O)CCC(C)(C)C1CNC(=O)Cc1nn(C)cc1Cl C12(C(=O)NCC(CNC(CCn3c(C)ncc3)=O)O)CCOC(C)(C1)C2 c1(C(=O)NCC(CC=C)NC(c2cc(C(F)(F)F)n[nH]2)=O)oc(CO)nc1C C(CC(C)C(=O)NCc1nc(CNC(=O)CC2C(O)C(O)CO2)cs1)=CCC c1(S)ccc(C(=O)O)s1.C1C(O)CN1.C(CC(C)C)OCC c1(C(=O)NCC(N(C(C(CC)CC)=O)C)C2CC2)ccc2c(c1)NC(=O)CN2C N1(C(CC(CC2CC2)NC(CCSCCC)=O)=O)CCCC(C)CC1 N1(C(C=C(C)C(F)F)=O)CC(NC(=O)C(c2cccc(C)c2)C)CC(C)C1 Cc1cc(C(N2CCC(C(C)NC(c3cocn3)=O)CC2)=O)cc(Br)c1C C1(CNC(c2cccc(C)n2)=O)CC(C)(C)CN1c1cc(-n2ccnc2)ncn1 C1(C(=O)NC2CC3CN(C(C=Cc4ncc(C)[nH]4)=O)C2C3)CCCCC(F)(F)C1 CC(=O)CC(C)(C)CC(=O)N1CCC2(CC1)CC2NC(=O)C(C)CO C#CC1(C)CCCN(C(C2(SC)CN(C(c3cnn(CCF)c3)=O)C2)=O)C1 c1(C(=O)NC2C(NC(COCP(C)(C)=O)=O)COCC2)cnc(O)c2ccccc12 Cc1cnn(C)c1S(=O)(=O)N1CCN(C(=O)CSc2ncc(Cl)cc2Cl)CC1 c1(NC(C2CCC(NC(c3scc(C)c3Cl)=O)C2)=O)cc(Br)c(O)cc1Br c1(C(=O)NC23CCN(C(C4(O)CCC4)=O)CC2C3)cccc2scnc12 CC(C)C(CC(=O)NCC12CCC(CC1)N(C(c1cnc(S)[nH]1)=O)C2)C(C)C CCCC(CC)CCC(=O)N1CCCN(C(=O)Cc2cscn2)C(CO)C1 C1(NC(C(C)NC(C)=O)=O)COC2(C1)CN(C(C1CN(C3COC3)C1)=O)C2 c1(CC(=O)NCC2CC(NC(C3C(C)OCC3)=O)C2)ccc(F)c(Br)c1 c1(NC2CCN(C(C3CC3F)=O)CC23CCC3)nc(Cl)nc2sccc12 C12CC3(C1)CC(C3)CNC2=O.CCCCCC(=O)NCCC1(C(=O)N(C)C)CC1 Cn1c(O)ncc(C(N2CC(CNC(=O)CNC(c3cccs3)=O)C2)=O)c1=O C(=O)(C(CC)C(=O)NC1CC(N(C)C(c2ccc(OC)s2)=O)C1)OCC Cc1cc(C(=O)NC(CNC(c2cc(CF)on2)=O)C(C)(C)C)[nH]c1C n1(C(=O)N(CCO)C2CC2)ncn2nccc2c1=O CC1CCN(CC(=O)NCCOCCN(C)C(c2csc(Cl)c2Cl)=O)CC1 N1(C(CCn2cc(C3C(C)C3)nn2)=O)CCCC(CCNS(C)(=O)=O)C1 c1(OC)ccc2c(c1)CC(=O)N(CCC(=O)CCCCS(N)(=O)=O)N2.S(C)(=O)(=O)N c1(OC)cc(C(=O)Nc2nc(C(=O)Nc3cccnc3C#N)cs2)c(F)cn1 C(C(C(=O)N1CCC(N2CC(O)C2)C1)NC(=O)CCc1cncn1C)N(C)C Cc1ccc(C(c2ccccc2)NC(=O)NCC(N)C(F)(F)F)cc1 C(=O)(CS(=O)(=O)CCOC)NC1CCN(C(CC2(C=C)CC2)=O)CC1C C=CCC(C(=O)N1CC(C)C1C(=O)NC(C)C(C)C)OC C(=O)(C(C(C)(C)C)c1ccccc1)N(Cc1nn(C)c(F)c1)C1CC1 CC1=C(C(=O)NCC#CCNC(c2ccc(C)c(N(C)C)c2)=O)CCCO1 C(=O)(C(CO)C(C)(C)C)NC(CCC)CCCNC(c1cc(C)c(Cl)s1)=O Cc1nc(N(C)C)sc1C(=O)NCC1(NC(=O)Cc2cncn2C)CCOC1 c1(N(C(CNC(C2(CSC)CC2)=O)C)C)nc(C)nc(O)c1C c1(C(=O)NCCCC(CCC)NC(=O)C(C(C)C)SC)ccc2c(c1)C=CCC2 C(=O)(C1=C(Cl)CCCC1)NC(C)CCN(C)C(c1ccccc1C(C)(C)C)=O CC(C)C(CCN(C)C(C1CC1(F)F)=O)NC(c1c(Cl)cnn1C1CCCC1)=O C1(NC(c2cn(CC=C)nc2)=O)CCCC1(C)CNC(=O)C=Cc1sccc1C N1(C(C(CC)n2nccc2C)=O)CCCC(C)(NC(c2cc(C(C)C)[nH]n2)=O)C1 NS(=O)(=O)CCC(=O)NCCCNC(c1c[nH]nc1Cn1ccnn1)=O C1(C(=O)NCC(CC)n2cccn2)CN(C(=O)Cc2csnc2C)CC12CC2 c1(C(C)=O)ccsc1C(=O)N(CCC(C)NC(=O)CC1CCCCO1)C c1(CC(N2C(CNC(C3C4COCC34)=O)CCC2)=O)cc2ccccc2c(=O)o1 C1(NC(C(COC)C)=O)CCSC12CN(C(=O)C=Cc1ccccc1OC)C2 c1(N2CCC(COC)(CO)C2)nc(=NC(C)C2CCCCC2)[nH]c2ccsc12 N1(C(CNC(CC(C)C)=O)=O)CC(F)CC1CN(C(=O)CC1CC2CC2C1)C CC1(NC(c2ccnc(C3CC3)c2)=O)CCC(NC(C2CC(F)(CF)C2)=O)CC1 C1(C(N2CC(C(C)NC(c3cn[nH]c3)=O)OCC2)=O)CCC2(CC1)CC2 c1(CC)nc(C(=O)NC(C)Cn2cc(CCCCC3CCCCC3)nn2)cs1 n12cc(nn1)CNC(=O)C2.C(CCOCC(=O)NCCSC1CC1)OC C1(NC(CCC(CC)NC(C2CC=C(C)CC2)=O)=O)CCCCC1N=[N+]=[N-] C1(NC(C(CNC(COC2(C)CCC2)=O)CC2CC2)=O)CC2(C1)CC(C)(C)C2 C(=O)(CC(C)CC(=O)NC1(CC(=O)NCc2nccn2C2CC2)CCC1)OC C(N=c1[nH]c(C(C)C)ncc1Br)C1CN(C(C(COCC)N=[N+]=[N-])=O)C(C)C1 C(CCCC(C)NC(=O)C(C)CCO)NC(C1(C)CC(=C)C1)=O c1(CCNC(CCN(C(C(COCC)C)=O)C)=O)ccccc1F C12(C(=O)NC3C(C)CN(C(=O)Cc4ccsn4)C3)CCCCN1CCC2 c1(C(N(C(C)C(=O)NCc2ccc(O)nn2)C)=O)ccnc2cc[nH]c12 N1(C(C(C)OCCC(C)C)=O)CCN(C(=O)C=CC2CCCO2)CC(C)(C)C1 C1(C(=O)NCC2(F)CC(NC(c3c(OC)n[nH]c3)=O)C2)CN=C2N=CNN2C1 N#Cc1ccc(N2CCCC(NC(c3cc(OC(F)F)cc(F)c3)=O)C2)cn1 C(=O)(CS(=O)(=O)C1CC1)N1C(CCCNC(c2c(C(N)=O)nccn2)=O)CCC1 c1(C(N(CCC(=O)N(C(C(=O)OCC)C)C)C2CC2)=O)cnc(N)cn1 c1(C(C(=O)NCC(CO)NC(=O)Cc2ccoc2)NC(N)=O)cc(F)cc(F)c1 c1(C(=O)NC(CNC(C2(C(F)F)CC(=C)C2)=O)CCOC)cccc(C=C(F)F)c1 N1(C(C2CC2)CS)CCN(S(C)(=O)=O)CCC1C.C1(CC(C)N)C2CC3C(C2=O)C13 C1(CC)(CNC(C2CN(C(C3(NC(C)C)CCC3)=O)C2)=O)CCOC1 C(=O)(C#CC1CCCOC1)N1CCCC(NC(c2cc(N)c(Cl)cn2)=O)(CO)C1 N1(C(CCC(CC)OC)=O)CCCC12CCN(C(c1cnn(C)n1)=O)C2 C1(OC)CCC(N=c2[nH]c(=NCc3c(C)coc3C)[nH]c3c2CC(C)CC3)CC1 N1(C(C)C)C(C)CCC1C.N1CC(O)(C(C)NC(=O)Cc2ccoc2)C1 N1(C(=O)CN2CCCS2(=O)=O)CC2C3CCC(C2C1)N(CCn1cccn1)C3 C(C(=O)N1CC2C(CNC(=O)CN3CCOCC3)C2C1)(C(C)(C)C)SC C1(C)(C(N2CCC(N(C)C)CC2)=O)CN(C(C2C3CC4C(C3)C24)=O)C(C)(C)C1 c1(CCNC(=O)NC2(CO)CCC(C)C2)ncc(Cl)c(O)n1 N1(C(C2CC23CC3(F)F)=O)CCn2c(CNC(C3(O)COC3)=O)nnc2C1 C(=O)(CCS(=O)(=O)C(F)(F)F)NC1(C2CN(C(C3N(C)CCOC3)=O)C2)CC1 C1(CS(C)(=O)=O)(C(N(C)Cc2ccnc(OC(F)(F)F)c2)=O)CC(F)(F)C1 C1(C(=O)NCC(C)NC(C2CC(C)(C)CN2C)=O)Cc2ccccc2N1C C1(c2nnnn2CCCN2CCOCC2)(NCc2cnc[nH]2)CC2CC2C1 C(C)(C)(CCCC(=O)N(C1CC(CO)C1)C)NC(CC1N(C)CCC1)=O CN(CCCC(=O)NCC1(O)CCN(C(C2(C3CCC3)CC2(F)F)=O)C1)N=O N1(C(C(CC)C)=O)CC2(CCN(C(C3(c4cccc(C)c4)CCC3)=O)CC2)C1 C1(C(=O)NCCC(N)=O)(CC)CCCN1C(C1CCCN1C)=O c1(CNC(=O)C(=O)NCC2COCCN2Cc2ccccc2)cc(O)cc(Br)c1 C1(CC(=O)NCCCN2CCN(C(CCCC#N)=O)CC2)CCCCCCC1 C(=O)(C(CC(C)C)C(N)=O)N1CCC(CC=C)(NC(c2ncc(F)cn2)=O)CC1 c1(C(N2CCCCCC(NC(CC=C(C)C)=O)C2)=O)[nH]nc2c1CCCC2(C)C c1(C(=O)NC(CCNC(C2(CC(=O)OC)CC2)=O)C)cccc(OC)c1Br c1(C(=O)NCC2CN(C(C(COCC)(C)C)=O)CC2C)cc(C)cc(Cl)c1N N1(C(=O)Cc2csnn2)CC2(C1)CN(C(c1ccoc1C1CC1)=O)C2 Cc1cc(F)ccc1C(=O)NC1CC(C)N(C(C2CCC(C(C)(C)O)CC2)=O)C1 CC1(CNC(C23CSCC2C3)=O)CCCN(C(c2ccc(O)nc2)=O)C1 N1(CCN(C)C)CCCN(C(C2CCC3(CCC3)C2)=O)CC1 N1(C(CCCC2(NC(c3n[nH]cc3Cl)=O)CCC2)=O)CC2(CCC2)C1 Cc1ccc(C=CC(N2CCCC(C)(C)C2CNC(C2CC23CC3)=O)=O)cc1Cl C(=O)(C1=CCC(NC(=O)C(C)NC(=O)CC)C1)NCC1(C#C)CCC1 c1(C(=O)NCC(CC(C)C)NC(C2CC(O)C2)=O)ccc2occc2n1 CCCC(C)(O)CC(=O)NCC1(F)CC(NC(c2cc(Cl)ncc2O)=O)C1 C(=O)(C(F)C(C)(C)O)NCCCOCCNC(C(C)(C)C1(O)CCOC1)=O C1(C)(NC(C2(NC(c3c(CC)ocn3)=O)CC2)=O)CCCC1(C)C c1(N2CC3C(CNC(C=C(C)C)=O)(C3)C2)nc(C)nc2n[nH]cc12 N1(C(COCCN(C(=O)CCOC2CCC2)C)=O)CCN(C2(C)CC2)CC1 C1(C(=O)NC2C(NC(c3nc(C)n(C)n3)=O)C2)OCC2COCCC12 C1(C(N2C(C(=O)NCC3CC34CCC4)CC2)=O)CC2CC1CC2=O c1(COCC)nc(C(=O)NC2CCC(CCNC(C34CC(C)(C3)C4)=O)C2)cs1 C1(CC)CCC(C)CN1C(=O)CCCN(C(=O)Cc1cccn1C)C c1(C(=O)NC2CC(C)N(C(c3cnc(O)s3)=O)CC2)cccc(S(C)(=O)=O)c1 c1(C(=O)OC(C(C)C)C(=O)Nc2ccccc2Cl)nnc2n1CCC2 c1(C(=O)NC2CCN(C(=O)COCC3CCCO3)C2)c(Cl)cc(F)cc1Br C1(C)(NC(=O)Nc2n(C)ccn2)CCCN(C(=O)C(CO)Nc2ccccc2)C1 CCCCCCC(C)C(=O)N1CCCC1CN(C(=O)CCN(S(C)(=O)=O)C)CC N1(C(C=C(C)CNC(c2cnc(S)nc2)=O)=O)CCC(C)OC(C)C1 N1(C(C2CC(OC)C2)=O)CC2(COC(CNC(c3ccsn3)=O)C2)C1 c1(C(c2nc(-c3cnn(C)c3)n(-c3nccn3C)n2)C)ccc2ccccc2c1 c1(-c2c(C#N)cccc2)ccc2c(c1)OCCO2.OS(=O)(=O)C(Cl)Cl Cc1cc(C)c(C(=O)NCC(C)(O)CNC(=O)C(O)CCN(C)C)c(N)c1 C1(CC(=O)NCC(CC)(CC)OC)CC2(C1)CN(C(=O)Cc1ccn(C)c1)C2 n1(-c2ccc(C)cc2)cc(C#CCNC(c2cc(Cl)cc(Br)c2F)=O)nn1 Cc1ccc(C(=O)NCCc2ccc(C(=O)NCc3ccncc3)cc2)c(O)n1 c1(CC)ccc2occ(C(=O)NC3CCC(NC(=O)CCn4ccnn4)C3)c2c1 N1(C(COCCCOC)=O)CC2CCC1C2NC(=O)Cn1ccc([N+](=O)[O-])n1 c1(C(CC(=O)NC(CSC)OC)OC)cc(Cl)ccc1C c1(CC(=O)N(CCCCN(C)C(c2cc(Cl)cs2)=O)C)nc(C2CC2)cs1 c1(OCC(=O)NC(C)(C)CNc2cccc(C(F)(F)F)c2)cc(F)cc(Cl)c1 c1(C(N2C3CN(Cc4cc(Br)cc(Br)c4F)CC23)=O)cc2n[nH]cc2cc1Cl C1(C(c2ccc(-c3n(CCC)nc(C)n3)cc2)=O)Cc2ccc(Br)cc2C(=O)O1 C1(N(C)C(c2ccn(-c3ccccc3)n2)=O)CCC(NC(c2cc[nH]c2)=O)CC1 C1(OC)C2CC3CC1CC(C(N1CC(NC(C4CCCC4C)=O)C(O)C1)=O)(C3)C2 N1(C(C2CC3CC2C2CC32)C(=O)NCCC2(C)CC2)CC(C)(C)OC2(CCOC2)C1 C(=O)(CC(C)(C)O)NCc1cc(C(=O)NCC(CCC)OC)on1 O=C1CN(c2ccncc2F)CCN1Cc1cnccc1C1CC1 CC(C(C)(C)C(=O)NCC1CCCOC1)NC(C1COCCC1C)=O N1(C(CCN(CC)CC)=O)C2CCC(C2)C1CC(=O)NCC(C)CC(=O)OC C(c1ccc(OC)cc1)=CC(=O)NCC(CCCC)NC(=O)CCC(C)OC C1(NC(c2c(CC)nns2)=O)(CNC(=O)Cc2sc(S)nc2C)CC2CCC1C2 N1(CC)CC2(CN(C(=O)C(c3cnn(C)c3)NC(=O)CC3CCCOCC3)C2)C1 N1(C(=O)CC2C3CCCC3N2C(=O)CC2CC=CCC2)CCc2n[nH]cc2C1.CN CC(CC(F)F)C(=O)NCC(c1ccccc1F)NC(c1n[nH]cc1F)=O c1(OCC)c(C(=O)N(C(C)C)CC)cc(Cl)cc1C CN1CCC(C)(C(=O)OCC2(C(C)(C)C)CCN(C(=O)OC(C)(C)C)C2)C1=O c1(OC)ccnc(C(=O)NC2CN(C3CN(C(=O)C=CC(C)C)C3)C(=O)C2)c1O C1(CNC(c2c(Cl)cn(C)n2)=O)CC2(C1)CN(C(=O)COC1CC(F)(F)C1)C2 c1(C(=O)NCC(CNC(c2c(C(C)C)onc2)=O)O)nccc2cccnc12 C(=O)(C1=NOC(C)C1)N1C(C(=O)NCC2(C#C)CCC2)CC(O)C1 C1(OC)CN(C(=O)C(C)SC(C)C)CCC1NC(c1ccc(C(N)=O)[nH]1)=O C1(NC(c2cnc(OC)nc2C)=O)CN(C(=O)C(C)C2CC2)CC(C)(C)C1 c1(C(=O)NCC2OCCN(C(CSc3c(C)noc3C)=O)C2)cc2[nH]ccc2s1 C(C(C)CC(=O)NCCOCC1CCCC1)NC(Cc1onc(C)n1)=O CCC1=NOC(CC(=O)NCC2CCCCN2C(c2cc(C(=O)OC)sn2)=O)C1 C(=O)(CC(O)c1ccccc1)NCCCN(C(=O)CC1COCC1O)CC c1(C(N(CC(C)NC(=O)C(C)CCCOC)CC)=O)ccc2nc(C)sc2c1 C1(NC(CN(CC)CC)=O)COCCN(C(C23CC(CSC)(C2)OC3C)=O)C1 N1(C(C=CC=CCC)=O)CCCC1C1CCCCN1C(=O)CNS(=O)(=O)N(C)C c1(OC)cc(OC)c(C(=O)NC2CCCCN(C(C3CCC(C)(C)O3)=O)C2)cn1 C1(NC(c2cc(C)c(C)nn2)=O)COC2(C1)CN(C(c1ccc(Br)o1)=O)C2 C1(C(=O)OCC(=C)OCOC)CC(N=[N+]=[N-])C1 C1(CNC(C(C)SC)=O)CN(C(=O)CCC(C)(C)F)CCC12CCC2 Cn1ccc(CCC(=O)NC2CC(NC(=O)C=CC(F)(F)F)C2)c1 N1(C(C2C(OCC)C2)=O)CCCC2CN(C(=O)CSc3nccn3C)CC12 N1(C(C=CC)=O)CCc2ccccc2C1CNC(c1sc(Br)cc1F)=O C(=O)(C1=CCC(C)CC1)N1CC(CCNC(c2c(C)nc(C(C)(C)C)s2)=O)C1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2CCCC(NC(C3C4COCC34)=O)C2C1 C1(C(=O)NCc2cc(C)cc(O)c2)N(C(=O)Cn2cccn2)CCCC1(C)C N(C1c2ccccc2CC1NC(C1CCCC(F)C1)=O)C(C1(F)CC1)=O N1(C(CC2(CSC)CC2)=O)CCC2CCC(C1)N2C(=O)C(c1nc(C)cs1)C C1(CCCC)CCC(C(=O)NC(c2ccc(F)cc2)C(C)N)CC1 CC(C(=O)NC1(CCNC(=O)COCC2CCCOC2)CCC1)C(F)F C1(NCc2cccc(OC(c3ccccc3)CC)c2)CCCC2(CCCCC2)C1 N1(C(c2c(OCC)n[nH]c2)=O)CC2CS(=O)(=O)CC2(NC(=O)C2=CCCCC2)C1 c1(-c2cn(C(C)CNC(=O)CCCN3CCCC3)nn2)sccc1O N1(C(C(=O)N(C)CC2(O)CCCC2)=O)CCC2(CCOC2=O)C1 C1(NC(CC2(N(C(C=CCOC)=O)CC)CC2)=O)C=CCCCC1 C1(CCOC)CCCN(c2nnc(C3CC3)n2CCc2ccccc2)C1.C(COC)S N1(C(=O)CN2CCNCC2)CCCN(C2CCOCC2)CC1 c1(N2C(C(C)NC(C(CC)CC3CCCC3)=O)CCC2)[nH]c(=O)n(C)c(=O)c1C#N CCC(C(=O)NCCC(C)(C)C(=O)NCC1(O)CCCC1C)C(C)(C)CC c1(OCC)ccc(C(=O)NCCCC(CO)NC(=O)C(O)C2CCCC2)cc1 C1(N(C(=O)Cc2scnc2C)CC)CCCN(C(c2csc(S)n2)=O)C1 N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCC(O)(CCNC(C2CCC3(CC3)C2)=O)C1 N(C(=NCCC1CCN(C(N)=O)C1)NC1CCOCC1)CCc1cn(C)nc1 N1(C(C2(CC)CCCC2)=O)CCC2(CCC2)C(CNC(C2C=CC=CC=C2)=O)C1 c1(NC(C)=O)cccc(CC(=O)NC2CCC2NC(c2cc(C)c(C)[nH]2)=O)c1 n1(CC)cnc2c(NC(C)Cn3cccn3)[nH]c(=NC(C)C3CC3)nc12 N1(C(C2(COC)CC2)=O)CCC(O)C(C(=O)NCc2ccc(=O)oc2)C1 Cc1c(C(N2CCCC(C)(NC(=O)CN(C3CCCC3)C)C2)=O)cccc1Cl c1(CNC(C(=O)N(C(C)C(C)(C)C)Cc2ccccn2)=O)cccc(Br)n1 CC1c2cccc(F)c2CCN1C(c1sc(Cl)cc1Br)=O C1(C(=O)NCC(C)N(C)C)CN(C(=O)COC2CCCCCC2)CC12CC2 c1(CC(=O)NC2CC(CO)N(C(=O)C(C3CCSCC3)=O)C2)ccc(F)cc1F C1(NC(c2cc(C(C)C)no2)=O)CC=C(C(=O)NCC2CC2(F)F)C1 C(=O)(C(F)CCC(C)(C)C)NCC12CCN(C(CN(CCOC)C)=O)C1CCC2 c1(C(=O)NC2CNC2)cnn2cccc(-c3ccnc4[nH]ccc34)c12 C(=O)(CC(O)C(C)C)NC1CCN(C(CNS(CCCC)(=O)=O)=O)C1C1CC1 Cc1cc(C(N2CC=C(C(=O)N3CC(n4cc(C)cn4)C3)C2)=O)nc(C)c1 C(=O)(C(CC1CCCC1)NSCC(=O)OC(C)C)NCCOC=C c1(OC)ccc(CC(=O)NCCC2(O)CN(C(=O)Cn3cc(Br)cn3)C2)cn1 C(=O)(C(C(=O)N(CCNC(c1n[nH]c(C)c1[N+](=O)[O-])=O)CC)C(C)C)OCC c1(CNC(C(C)(C)CCl)c2nnnn2C2CCCCC2)nc2ccc(Cl)cc2[nH]1 Cn1nc(-c2ccsc2)cc1CNC(c1cnn(C2C=CCCC2)c1)=O N1(C(=O)C2=COCC2)CCC2CCN(C(=O)CC3CCC4CC34)CC2C1 c1(OCC)c(-c2cnc(OC)cc2C(=O)NCC2CCSCC2)ccc(F)c1F C1(CNC(c2cccc3nncn23)=O)CCCC12CCN(c1nnc(O)s1)CC2 c1(C(N2CCC(C)C2)C(=O)NCCSC)ccc(C(F)(F)F)o1 c1(C(=O)NC2C(NC(=O)Cc3ccc(C4CC4)s3)COCC2)cc(F)ccc1Cl N1(C(c2c(SC)ccs2)=O)CCC(F)(CNC(=O)C(F)C2CC2)CC1 c1(C(=O)NCc2ccc[n+]([O-])c2)cnn2c1NCC2 N1(C(c2c(SC)cn(C)n2)=O)CCC(CNC(=O)CCOCCN(C)C)C(C)C1 CC1CCC(NC(=O)C(C2CCCCC2)N(C)C)CN1C(C1C2CC3C(C2=O)C13)=O c1(C(=O)NC(C)(C)C)coc2c1COC2.CC1CCN2C1CNC(=O)CCC2=O c1(C(N(C2CCC(CNC(CC(=C)C)=O)CC2)C)=O)cc(Cl)c(C)cc1[N+](=O)[O-] C1(NC(C(C)=CC)=O)CCC2CCN(C(c3cccc4c3C(=O)NC4)=O)C1C2 Cc1cc(C(=O)NC2CCCC2NC(C2CN3CCC2CC3)=O)ccc1O CCC(C)(CC(=O)N1C2CCCC1CN(C(=O)C=Cc1cscn1)C2)C=O c1(C(N2CCC(C)(NC(C=CSC)=O)C2)=O)c(Br)cncc1[N+](=O)[O-] N1(Cc2cccc(C(=O)OC)c2F)CCC2(CC1)OCc1ccccc12 c1(N2CCC(CC)(CC)C2)nc(=NCCc2ccncc2)[nH]c2c1CCCCC2 c1(C(CCC)n2cccn2)cccc(Sc2nnc(C)n2-c2cccnc2)c1 N1(C(C2(COCC)CC2)=O)CC(OC)CC(NC(C2(O)CCSCC2)=O)C1 C1(NC(CCCCOC)=O)CC12CCN(C(c1cc([N+](=O)[O-])n(C)n1)=O)CC2 C1(C(C)C)CC(O)CN1N(C)Cc1nncn1C(C)C c1(C(N2CCN(C(c3n[nH]cc3Br)=O)CC2)=O)cccn(CC(F)(F)F)c1=O C1(C(=O)NCC(CO)NC(c2cnc(C(C)(C)C)s2)=O)C(F)(F)C12CCC2 CCC(CC(C)C)C(=O)N1CCC(C(=O)NCC(O)CC(F)(F)F)O1 c1(-c2nc(NC(c3c(C)cc(OC)nc3)=O)sc2)nccn2nc(C)cc12 C=C1CCCN(C(=O)CN(C2CCC2)C(C2CC=CCO2)=O)C1 C1(NC(c2ccnnc2)=O)CCCCC12CCN(C(=O)COCC(F)(F)F)C2 c1(C(=O)NC(C)CC(C)NC(c2ccco2)=O)cc(Cl)ccc1OC(F)F Cc1cnc(NC(=O)Nc2ccc(OC(C)C)cc2)nc1Br c1(SC)nc2ncnc(N(CCCNC(C3NC(=O)CC3(C)C)=O)C)c2s1 c1(C(=O)NCC(CC)N(C(C(C)NC(CC)=O)=O)C)c(C)nc(C)nc1C N1(C(CCS(C)=O)=O)CCCOC(CNC(c2ccc(F)c(N)c2)=O)C1 N1(C(C(F)OC)=O)CCCC(CCNC(=O)CSc2nncs2)C1 N1(C(CCCCC(=O)OC)=O)CC(C2CCN(C(C3CC3(C)C)=O)CC2)C1 C1(NC(C=CCN(CC)CC)=O)CN(C(=O)CC2CC(N(C)C)C2)C(C)(C)C1 C1(NC(C(C)(C)C#N)=O)CC(NC(=O)Cn2nnnc2-c2ccsc2)C12CCC2 C12(C(=O)NCC3(C)CCN(C(C(C)OC)=O)CC3)CC(CO)(C1)OC21COC1 CC1CC=C(C(=O)NCC2=CCN(C(c3ccoc3Cl)=O)CC2)CC1 S(=O)(=O)(c1cc(C(N)=O)ccc1F)CSCCNCC(CCC)CCO c1(N2CC=C(C#N)CC2)nc(NCC2CC23CCCCC3)c2ccsc2n1 N1(C(C(CN(C)C)NC(CCC(C)OCC)=O)=O)CCOC(C#N)C1 C(=O)(C(F)(CNC(c1nc(C2CC2)oc1C)=O)C(C)C)N(CC(C(C)C)OC)C N1(C(c2cc(OC)no2)=O)CCCN(C(=O)CC(c2ccccc2)N(C)C)CC1 S(=O)(=O)(c1cccc(N2CCC(N3CCCC3)C2)n1)N(C)CC1CCCS1 C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NCCC1CC(NC(c2c(C)ocn2)=O)C1 N1(C(c2n(CC)ncc2)=O)CCC2(CCCN2C(c2nccc(Cl)c2F)=O)CC1 C(N=c1[nH]c2c(c(=NCC(C(C)C)OC)[nH]1)CCCCC2)c1c(CC)cccc1 C1(C(=O)NC(CCCC)CO)CN(C(C2CCC2C(=O)OC)=O)CC1(C)C C(CCCCCCO)CNC(CC1(N(C(=O)CCc2ccoc2)C)CC1)=O n1(CC)nc(C(=O)NCC2(C)CCC(NC(=O)CCN3CCOCC3)C2)cc1C C(=O)(C1=CCCCC1)N1CC(NC(C2CCCCN2C2CC2)=O)C1 N1(C(CCSC)=O)CCC(C(C)CNC(c2cc(Cl)nn2C)=O)CC1 c1(C2CN(C(CCN(C(C=CC(CC)C)=O)CC)=O)C2)ncc(C)cn1 C(=O)(CC(C(F)F)NC(=O)NCC(=Cc1ccccc1)F)OC CC1CCC(O)(C(=O)NCC2CC(O)(CNC(C3CCCCO3)=O)C2)CC1 N1(C(c2cc(CC)on2)=O)CCCC2(CO)CCCC12.C(C)(C)(C)NC(=O)O C(=O)(CCCCC(F)F)NC1CN(C(Cc2c(C)noc2)=O)C(C)CC1 N1(C(c2c(CC)csc2)=O)CC2(CCC2NC(c2cc(C(F)F)no2)=O)C1 C(=O)(C(C)CC(C)C(C)=O)NCC(C(=O)N1CC(=CCC)C1)OC CCCC(C(=O)NC1CCN(CC(O)COc2ccccc2C)CC1O)C(C)C c1(NC(C(CC)NC(=O)C(=Cc2cn[nH]c2)C)=O)ccc2c(c1)OCO2 CC(C)(CC(=O)N1CCC(C)(CNC(C2(CC(=O)OC)CC2)=O)C1)CC(F)F C(CNC(c1sccc1C#N)=O)(CC(F)(F)F)NC(CN1CCC(C)CC1)=O c1(CC)onc(C(N2CCCC2C2CCN(C(c3c[nH]c(Br)c3)=O)C2)=O)c1C c1(CCNC(CC2N(C)CC=CC2)=O)c(F)cc(Br)cc1F c1(C(N2CC(O)CC(NC(C(CCC)OCC)=O)C2)=O)nc(C)c(C)nc1C c1(C(=O)NCC(CC)(CC)NC(=O)C(C)CO)cncc2ncccc12 Cc1cccc(C(C)C(=O)NC2CC(CNC(=O)CCc3cncc(O)c3)C2)c1 Cc1nc2cc(C(=O)NC3CCC3NC(c3n[nH]c4c3CCC4)=O)ccc2s1 C(=O)(C1=CCCCO1)NCCCC(C)NC(c1ccc(C(=O)OC)n1C)=O C1(CCNC(CC2(OC)CCC2)=O)CCN(C(=O)Cc2cncnc2O)C(C)C1 CC(C)(C)C(O)CNC(C1CC(=O)CN1C(C1COCC1C(N)=O)=O)=O Cc1cc(C(C)(C)C)ccc1NC1CC(F)CN(C(=O)OC(C)(C)C)C1 C1(N(C(c2cnccn2)=O)CC)CCCN(C(=O)C(C)n2cnnn2)C1 c12cccnc1NC(=O)CS2.c1(NC(CCC)=O)ccc(-c2nn[nH]n2)cc1 Cc1ccn(CC(=O)NC2(CC(=O)NC3CSC3)CCC2)n1 C1(NC(c2cnc(CCCC)s2)=O)CC2CC(C1)N(C(C1(C3CC3)CCC1)=O)C2 N1(C(c2c(C)c[nH]n2)=O)CC(NC(c2cc3occc3[nH]2)=O)CC(F)C1 Cn1nccc1C=CC(=O)NC(C1(NC(N)=O)CC1)=O C(=O)(CC(C)CC(C)C)N(C1CN(C(c2ccc(C)c(C)n2)=O)CC12CC2)C C(=O)(CCCC(=O)NC(C)C)NCC(C1CC1)NC(c1nncc(C)c1)=O c1(C(=O)NC2CC(OC)CN(C(COCCOC)=O)C2)cnc2ncc(Cl)cn12 C1(NC(=O)OC(C)(C)C)CCC(C(N2CCCC(NC(=O)C3=CCC3)C2)=O)CC1 N1(C(=O)C=Cc2ncc[nH]2)CCCCC1CNC(C1(CC2CC2)CCC1)=O