SMILES O=C(CC(=O)NCC(C1CCC1)NC(C1CCNC1=O)=O)Nc1ccccc1 C12(C(=O)NCCCC(C)NC(c3ccc(OC)cc3)=O)CCCC1C2(F)F c12ccc(cc1)CC(=O)NC(C)(C)CN(C)C(=O)C2C.N(CCO)(CC)CC C1(NC(Cc2nc(C)sc2)=O)CCC2(CC1)CN(C(=O)COCCCF)CCO2 C1(C(N(C(CC)C)CC(N2CCOC(C)(CC)C2)=O)=O)CCc2cc(C)ccc2O1 C1(C(=O)Nc2cc(C)sc2)CCCCC1(C)NC(=O)Cc1ccc[nH]1 C=CCC(CC=C)C(=O)NC(C)C(C)NC(c1cn(C)nc1C(C)C)=O c1(SC)ccc(F)c(C(N2CC3CCC3(C(N3CCC(C)C(O)C3)=O)C2)=O)c1 S(=O)(=O)(c1cccnc1)NCC(=O)NC(CNC(c1c(CC)ncnc1)=O)CO [N-]=[N+]=NCC(C(=O)N1OC2CCC1C2)NC(=O)CC1CCC(=O)N1 N1(C(C(C=CC)O)=O)CCN(C(CNC(c2ccsn2)=O)C(F)(F)F)CC1 C(=O)(CCCCCC(C)(C)C)NCC1CN(C(C(CCC)O)=O)CC1O c1(N(C)C)ccccc1NC(C1COCCN1C(=O)CSCC(N)=O)=O C(N=c1[nH]c(=NC(C)c2c(F)cccc2Br)c2ccccc2[nH]1)c1cnc(C)[nH]1 C1(NC(CCCCCCC)=O)COC2(CCCN(C(c3cnn(C)n3)=O)C2)C1 N1(C(C=CC=CCC)=O)CCC(CCC(=O)NC2(C(O)CO)CC2)CC1 n1(CC)cnc2c(NC3CCN(C(C)C)C3)nc(N3CC4COCC4C3)nc12 Cc1ccc(F)cc1NC(=O)CN1CC(CCC(=O)O)CCC1C N1(C(C(C)NC(c2cccs2)=O)=O)CC2CCN(C(C3CC=CC3)=O)C2C1 CC1(NC(=O)CC2CCCS2(=O)=O)CCCN(C(c2cnn(CC3CC3)c2)=O)C1 C(=O)(C1=CCCCC1)NCC1(C(=O)NC2CCN(CC)C2)CC(=C)C1 CC1=C(C)CN(C(C2CCCCN2C(=O)Cn2c(O)nnc2O)=O)C1 c1(OCC)ccc(C2CN(C(c3ccc(C(F)(F)F)o3)=O)CC2N)cc1 c1(C(=O)NC2C(CNC(C(C)c3ccsc3)=O)CC2)cccc2sccc12 n1(CC)c(C)cc(C(=O)NC2CC2NC(=O)CN2C(=O)CCC2=O)c1C C=CC1CN(C(=O)C=Cc2ccn(C)c2)CC1NC(=O)CC12CCCC1C2 c1(CC(N2CCN(C(C=CC=CC)=O)CC2CO)=O)c[nH]c2cc(Br)ccc12 C(CCCCCCc1ccccc1)N(C)C(c1ccc(C(F)(F)F)cc1)=O C1(NC(CCC=C)=O)CCCCC12CCN(C(C1CCCC(F)C1)=O)C2 c1(C(=O)NCCCCCNC(c2cc(C)cc(F)c2)=O)cccc(F)c1C#N C1(C(=O)NC(c2ccc(C)o2)c2ccccc2)NC(=O)CC1C(F)(F)F C(=O)(CCNC(=O)NCC(C)(C)c1cncs1)NCC CC(CCc1cncs1)NCC(O)CO c1(OC)cc(CC(N2CC(NC(c3cnn(CCO)c3)=O)CC2C)=O)ccc1O C(=O)(C1=CCC(C)(C)CC1)N(CCCCCC(=O)NC(CCN(CC)CC)C)C C(CCN(C)C(C1(c2cc[nH]n2)CC1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O CC(C)C(O)C(C)(C)C(=O)N(C1(C(=O)NCC(C2CC2)N(C)C)CC1)C c1(CC(=O)NCC2(NC(=O)CN3CCS(=O)CC3)CCC2)c(F)cc(F)cc1F Cc1cccc2sc(NC(=O)C(=O)NC3CCC3(C)C)nc12 c1(C(N(CC(CO)(CO)NC(C(C(C)(C)C)SC)=O)C)=O)nn(C)cc1[N+](=O)[O-] Cc1coc(C)c1C(N1CC2CC1C2NC(=O)C(C)Oc1ccccc1)=O C(=O)(CCC(C)CCCC)NC(CC=CC)C(=O)NCC(C)C(F)F N1(Cc2c(OC)cc(C)cc2)CCCc2cc(OC(F)(F)F)ccc21 N1(C(CC(CC)CN(C)C)=O)CCCN(C(c2cnnc(C)c2)=O)C(C)C1 N1(C(c2c(NCC)ccc(C(=O)OC)c2)=O)CC2CCC1C(Cc1ccsc1)C2 C(=O)(C(O)Cc1cnc[nH]1)NCCOCCCN(C)C(C1COCCO1)=O C(CNC(=O)CCCOCC)(C(C)(C)C)NC(c1ccc(CCC)[nH]1)=O C(=O)(C(F)CCC(C)C)N1CC(NC(C(C(=O)OCC)(C)C)=O)C(SC)C1 c1(OC)cccc2c1OC(CNC(=O)Nc1cc(Cl)c3c(c1)OCCO3)C2 NS(=O)(=O)c1ccc(NC(C23CC2CN(Cc2ccnc(O)c2)C3)=O)cc1 C1(C(=O)NCC2OCCN(C(CCOCCOC)=O)C2)CCOC(C)(C)C1 C(N=C(NCC1CCCS1)NC(c1snnc1C)C)c1cc(C)on1 C(=O)(CS(=O)(=O)CCO)N1CCCCC(CNC(CC(C=C)C)=O)C1 c1(C(=O)OCC)c(Cl)n[nH]c1COC(c1csc(Cl)c1)=O N1(C(c2ccn(CC(=O)NOCCOCCSC)c2)=O)CC=CC(OC)C1 C1(CC(=O)N(CC#C)CC2CC(C#N)C2)CC(F)CN1C(=O)Cc1ccc(C)o1 c1(OC)cc(C)c(CNC2CN(C(=O)C(c3ccccc3)SC)CC2C)c(O)c1 C12(C(N3C(C)CNCCC3)=O)CC3CC(C1)CC(n1cncn1)(C3)C2 C(CCC)(C(=O)NC1CCC(C(=O)NCC2C=CCC2)C1)=CCC CC1CN(C)CC1NC(=O)C=CC(C)(C)NC(=O)COc1cccnc1 N1(C(C(CO)N(C)C)=O)CC2CCC(N)C2C1 CC1CCN(C(c2ccc(C#N)[nH]2)=O)CCN1C(=O)CSCc1ccc(Cl)s1 N1(C(CC(C)(F)F)=O)CCCC2(CC(NC(C3CCS(=O)CC3)=O)CO2)C1 N1(CC)CCCN(C(c2cnc(C(C)O)s2)C(=O)NC2(C)CC2)CC1 C1(CNC(=O)Cc2nnc(O)s2)CCC12CCN(C(C1CC1(F)F)=O)CC2 C1(C(=O)NCC(CC)N2CCCC2)CCN(C(C2CC(C)(C)CO2)=O)CC1 c1(-c2cn(C(=O)N(C3CCC3)C3CCC3)nn2)ccc(C2CCC2)nc1 c1(C(=O)NCC2CN(C(CSCCOC)=O)CC2(C)C)cccc(Cl)c1[N+](=O)[O-] C(C)(CCC(=O)N1CCCCC1CC(=O)NCC1(CC)CCCC1)OCC N1(C(c2ccc(CC)nc2)=O)CCCC(COC)(NC(=O)COCC(C)C)C1 CC1CCN(C(c2cc[nH]n2)=O)CC1CNC(=O)C=C1CN2CCC1CC2 c1(OC)ccc(Cl)c(C(N2CCC(NC(=O)C=C(C)c3cccs3)C2C)=O)n1 C12(NC(=O)C(O)C(F)(F)F)CCOCC1CN(C(=O)CCc1ccc(Cl)cc1)C2 Cc1ncccc1C(N1CCC2C(NC(=O)C(C)Cc3ccc(F)cc3)C12)=O N1(C(C)=O)CC(C(=O)O)C2(CCN(C(C3(C(=O)OC(C)(C)C)COC3)=O)CC2)C1 N1(C(C2CC(C)NC(=O)C2)=O)CC2(CCN(C(C3CC3(C)C)=O)C2)C1 c1(CCC)cnnc(C(=O)NC2CN(C(C3CCC(=O)N3C)=O)CC2O)c1 Cc1cc(F)cc(C(N2CCCCC(NC(=O)C(C3CCCCC3)F)C2)=O)c1C Cc1coc(C)c1CNC(=O)C(C1(C)CC1)NC(C1CC1(C)C(F)F)=O C(=O)(C1=C2CCCN=C2NN1)NCC(c1ccccc1)NC(C(C(C)C)(C)O)=O N1(C(=O)OCC(C2CC2)OCC)CCOCC1.C1(=O)CO1 C12(CNC(C(CC(=O)OC)C)=O)CCC(CC1)N(S(C)(=O)=O)C2 c1(OC)nc(NC2CCN(C(c3ccnc(O)c3)=O)CC2C)ncc1C C1(NC(c2c(C)occ2)=O)(CF)CCN(C(=O)CNC(=O)CCC2CCCC2)C1 c1(Cn2cc(C(=O)NCC3CC(C)OCC3)nn2)csc2ccccc12 c1(C(=O)NC(C(C)C)(C)CNC(C2CCC3(CC3)C2)=O)ccn2ccnc2c1 c1(C(c2nnnn2C)Nc2ccc(N(C)C)nc2)ccc(Cl)cc1OC(F)F C12(CNC(C3C4(CC4)C34CC4)=O)CCCC1N(C(=O)C1=C(Cl)CCOC1)CCC2 C12(CNC(C(C)(C)OC)=O)COCCN1CCN(C(=O)C(c1ccc(C)s1)C)C2 CC1CCOC(C(=O)NCC2CCCN(CC(=O)NC3CCCC3)C2)C1 c1(C(=O)NC(C(C)NC(=O)CC(=O)NC2CC2)(C)C)cccc(F)c1N N1(C(C23CCCC(C)(OC2)C3)=O)CC2CCC(N=c3cnc(F)c[nH]3)CC2C1 C1(NC(c2cc(C)[nH]n2)=O)CN(C(=O)C(c2cccc(Cl)c2)(F)F)CC(C)(C)C1 C1(C(C)(C)C)(CNC(c2cnc[nH]2)=O)CCN(C(C2CC2c2ccccc2)=O)C1 C1(C(=O)NC2(CC(=O)NCc3ccc(CO)o3)CC2)CC(O)C(F)C1 CN1CC(C(N2CC(N3CCN(C(C45CCC4C5)=O)CC3)C2)=O)S(=O)(=O)CC1 N1(C(CN(c2ncccn2)C)=O)CCN(C)CC1CNC(C1CCCSC1)=O Cc1cn[nH]c(=NC(=O)c2ncc(-c3cnn(CCN4CCC4)c3)cn2)c1 C1(F)(NC(=O)C=CCNC2(C3CCCO3)CC2)CCCCC1 c1(CC(C(=O)N(c2cnccn2)C)NC(=O)OC(C)(C)C)ccc(O)cc1 c1(C(c2nnnn2C2CC2)CCNSCCOC(C)=O)conc1-c1ccccc1.C N1(C(c2nc(=N)[nH]cc2)=O)CCC2(C=C(C(=O)NC3CCCOC34CCC4)C2)C1 N1(C(CCOCCNC(C(CC)(C)O)=O)=O)CCC(C)(C)C1C c1(C(C(=O)NC(CCN(C(=O)C=C(C)C(F)F)CC)C)N(C)CC)cccnc1 Cc1sc(O)nc1C(=O)N(C(C)C(=O)N(C(CO)CC(C)C)C)C1CC1 N1(C(c2c(C)[nH]nc2C(C)C)=O)CCN(C(C2CCCCS2)=O)CC(O)C1 C1(C(=O)NC(CNC(C(C)(C)OC)=O)(C)C(C)C)CCc2cnnn2C1 c1(C(=O)NC(CCOC)CNC(C2CC(F)(CF)C2)=O)ccc[n+]([O-])c1 C(=O)(CC(CC)C1CCC1)OCC(COC)(C)NC(=O)NCC1(O)CCOCC1 C1(C)(CCC)CCN1C(=O)CONC(=O)CN1CCC(OC)C1 c1(OC)ccc(F)c(N)c1C(=O)NCC1CCC(F)(CNC(C2(CF)CC2)=O)C1 N1(C(c2cc(C)[nH]n2)C(=O)NCCCC)Cc2ccc(OC)cc2CC1C Cc1nc(C2CCOC2)sc1C(N1CCC(CNC(=O)C(F)=CCCF)CC1)=O c1(N2Cc3c(nc(N(C)C)s3)CC2)nc(N2CCC(O)CC2)c2c(ncn2C)n1 Cc1cc(C(=O)NCC2CC(NC(=O)C3=CSCCO3)C2(C)C)c(N)cc1F c1(C(N2CC(NC(c3cc(C)cc(F)c3)=O)C(C)C2)=O)cc2nc(C)ccc2o1 Cc1cnc(C(=O)N(CC(C)(C)NC(C2CC2c2ccnn2C)=O)C)c(C)c1 CCC(C(C)CN(C)C)NC(=O)Cn1cc(CNC(c2cc(O)n(C)n2)=O)nn1 C1(CCNC(C(COCC)NC(c2cn(CC)cn2)=O)=O)CC(C)(C)CO1 Cc1cccc(OC(C)CN2C(=O)CN(CC3=CCCOC3)C2=O)c1C C12(OC)CCC(C(N3CC(N(C)Cc4cn(CCCN(C)C)nn4)C3)=O)(CC1)C2 C=CCC(C)(C)CCNC(=O)CCCC1CCCCN1C(C1CC(C)(F)C1)=O N1(C(C(C)O)=O)CC2(CCC2)CC1CNC(=O)CN1C(=O)CNC1=O C#CCC(C)(C)C(c1nnnn1CCC1(C)CC1)Nc1cnc(C)nc1C N1(C(C2(OCC)CCOCC2)=O)CCC(NC(=O)CCCOCC)CC(C)(C)C1 Cc1cc2[nH]cc(CCNC(C3CS(=O)(=O)CC3N3CCOCC3)=O)c(=O)n2n1 c1(C(=O)NCCCOCCNC(C(CC=CC)C)=O)cc(C2CC2)n(C)c1C c1(C(=O)NCCC(CNC(C2CCN(C)C2=O)=O)O)ccc2nnc(O)n2c1 c1(C(=O)NC(C2CCCN(C(=O)CCCC3CC3)C2)C)c(Br)cc(F)c(F)c1F c1(OC)cc(C(F)(F)F)ccc1CN1CC(C)CC1C(=O)Nc1cnc(Cl)cn1 c1(C(C(=O)N2CC(CC(C)NC(C3CS(=O)(=O)C3)=O)C2)(C)O)ccc(F)cc1 C(=O)(C1=CCC(C)CC1)N(CC(=O)NCc1ncoc1C1CC1)CC#C N1(C(c2n(CC)nnc2)=O)CCCCC1CNC(C1CCCN1C=O)=O N1(C(C(CC#C)(C)C)=O)CC2CCC1CC2NC(c1ncn(C)n1)=O C(=O)(CS(=O)(=O)c1ccccc1F)N1C(C)CC2(CCC2)C1 Cn1ccc2cccc(C(N3CC4(CNC(c5cscc5Cl)=O)CC3CO4)=O)c12 N1(C(C(CC(F)F)NC(c2c(CC)ncs2)=O)=O)CCCC2(CCCO2)C1 c1(NC(CC(C)NC(=O)NC)=O)cccc(CNCc2n(CC)ncc2)c1 Cc1nn(C)cc1C(O)C(=O)NCc1ccc(NC(=O)COCCN(C)C)cc1 C1(CNC(C2C(NC(CN3CC(C)(C)C3)=O)CC2)=O)OC2CCC1CC2 C(c1cccc(Br)c1)=CC(=O)NCCCN(C)C(c1cnc(O)o1)=O c1(C(=O)NC(CCCC)CNC(=O)CNC(=O)OC)sccc1S(N)(=O)=O C=CCCC(C(=O)N(CCCN(C(C1CC1CCC)=O)CC)C)c1ccccc1 c1(C(=O)NC2CN(c3nc(CC)nc(C#N)c3)C(C)C2)cc2c(Cl)nccc2o1 C1(NC(=O)NC(C(C)C)C)COC2(C(=O)Nc3ccc(F)cc3)CC1C2 Cc1sc(-c2nc[nH]n2)nc1C(N1CCC1CNC(=O)C=Cc1cn[nH]c1)=O N1(C(C(C)OCCOCC)=O)CCC(COC)(NC(=O)CN2CCOC2=O)C1 c1(N2CCCC(CSC)CC2)ccc(S(=O)(=O)N(C2CCCC2)C)c(Br)c1 CC1CN(C(C2CC23CC3)=O)CCCN1C(=O)CCCc1ccc(Br)cn1 N1(C(CCC)=O)CCC(NC(=O)COC(C)(C)C)CC1C.CSCC C(=O)(C1=CCCC(C)(C)C1)NCC1C(OCC)CN(C(C2(C)CCN(C)C2)=O)C1 C(=O)(C(C)CC(=O)OC)NC1CCC(CCC(N2C(C#C)CC2)=O)C1 c1(CCC(=O)NCC(=C)CCNC(=O)CN2CCC(C)C2)cccc(C(N)=O)c1 CC1(C)CCC(CNC(c2ccoc2CNC(=O)Cc2cnoc2)=O)C1 C1(NC(CCc2scc(C)n2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)C1(C)C c1(C2(NC(C3(C)COC(=O)N3)=O)CC2)ccc(Cl)c(Br)c1 c1(C(=O)NCC(CC)NC(c2ccc(C)c(C#N)c2)=O)cc(F)cc2cc[nH]c12 CCCCC(C(=O)NC1CN(C(C2CCC(=O)N2)=O)CC1C)c1ccccc1.C1CC1 c1(CC)nc(=N)[nH]c(=NC(C)CN(C)C(C2CC(=O)N(CC)C2)=O)[nH]1 N1(C(Cc2c(C)nccc2)=O)CCCC(C)C1CNC(=O)CC12CC(C1)C2 c1(NCCCC(C)NC(c2c(CC)ocn2)=O)cc2nnc(C(C)C)n2cn1 c1(CC(=O)N(C2CCN(C(=O)CSCC(C)C)CC2)CCC)cccnc1O CC1(C)CC(CC(=O)NCCOCCNC(c2c(CO)cccc2F)=O)CCO1 CCC(CC)(CO)C(=O)NCC1(NC(=O)Cc2sccc2Cl)CCCCCC1 N1(C2C(=O)CCC2)CCN(C(=O)C(N2CCC(N3CCCNC3=O)C2)=O)CC1 c1(CC)c(C)nc2ncnn2c1NC1CS(=O)(=O)CC1NC(=O)Cc1ccoc1 C=CC(C)CC(=O)NCC1CCCN1C(c1ccccc1OC(F)F)=O N1(C(C(C)(C)C)=O)CCCC2C1CCCN2C(=O)Cn1cc(C(=O)N(C)C)nn1 CC1(C#CC(=O)N2CC(C3CN(C(C4CCCS4)=O)CCO3)C2)CC1 c1(C(=O)NCc2ccc(-n3cncn3)cc2)cc(C2CCN2)ccc1Br c1(CNC(C(CC)F)=O)ncccc1CNC(c1c[nH]nc1OC)=O C1(C)(CCNC(C)=O)CCN(C(=O)CNc2ncccc2Br)C1 N1(C(c2cc(C)[nH]n2)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC1C N1(C(CN2CC(C)(OC)C2)=O)CC2(CC(NC(=O)CC(=O)N(C)C)CO2)C1 c1(OC)ccc(F)cc1C(=O)NC1CCCC(NC(=O)C(C)OC2CCCC2)C1 C1(C(=O)NC(CO)CCO)CC2(CCN1C(c1ccnc3cc[nH]c13)=O)CC2 c1(C(=O)NCC2N(C(CC(CC)OC)=O)CC(O)C2)n[nH]c2c1CCCC2 C1(C)(C(N2CCCC(N(C(=O)CCF)C)CC2)=O)CC(C(F)(F)F)=NO1 N(C(=NCCC(C)C)NC1CCN(CC(N)=O)CC1)C1CC(OCC)C1SC N#CC(CCc1ccccc1)C(=O)N1CCCC(CNC(c2cnccn2)=O)C1 C(C)(C(=O)N1CC(C2CC2n2cc(-c3cnsc3)nn2)C1)(OC)OC N1(C(CCC2(C)CN(C(C(CCC)(C)C)=O)C2)=O)CCOCC(F)(F)C1 C1(NC(c2sccc2Cl)=O)CCN(C(=O)Cc2ccnc(F)c2F)CC1F N1(C(c2c(C)ccs2)=O)CC2CCCC1(CNC(=O)CC1CCNC(=O)C1)C2 N1(C(C(C)OCCOC)=O)CCN(C(c2ncn(C(C)C)n2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc(NCc2ncnc3sccc23)cc1Cl)NCCC(=O)NC c1(C(=O)NC(C2CCOC2)CC)cc2c(s1)CCC2 c1(CC(=O)N(CC(C)(C)NC(C2CC2(F)F)=O)C)csc(Br)n1 CCCCC(C)CCC(=O)NCC#CC(N1CC2CCC(C1)C2C#N)=O c1(NC(C(COCC)NC(C2CCNC(=O)C2)=O)=O)c(Br)cc(C)cc1[N+](=O)[O-] C1(CC)CN(C(C2COCCO2)=O)CCN1C(=O)Cc1csc(Br)n1 O=C(C1=CCCCC1)NCC1CN(C(c2cn(CC3CCOC3)nn2)=O)CC1O N1(C(C(C2CCC(C)(C)CC2)C)=O)CCC2CN(C(=O)CCC(=O)N(C)C)CC12 C(C(C)C)(C(O)C(=O)N(C1CN(C(c2ccc(F)cc2C)=O)CCC1O)C)OC C(C(O)CCNC(C1CC2(CC2)C1)=O)NC(=O)CSc1nncs1 N1(C(CC2(OC)CC2)=O)CC2CCC1C(CNC(=O)C(C)C1(O)CCC1)C2 N1(C(c2cc(CC)[nH]n2)=O)CC2CCC1(CNC(=O)CC1NC(=O)NC1=O)CC2 c1(CC)noc(CC)c1CC(N1CCC(NC(=O)CC(C)CF)C1)=O N1(C(CSCC#C)=O)CCOCC(CNC(=O)C(c2c(F)cccc2F)C)C1 n1(CC)cnc2nc(=NCc3cccnc3)[nH]c(NCCc3nnc(C)n3C)c12 N1(C(C2C3(CC(OCC)C3)C2)=O)CCC2(CCC2NC(=O)C=C2CCCC2)CC1 C1(C(N(C(CO)C2CC2)C)=O)CC(F)(F)CN1C(=O)COCCF c1(COC(=O)COC(C2CN(C(=O)NCC3COCCO3)C2)=O)ccccc1 C(CCCC(=O)NC1(CO)CCN(C(=O)C=Cc2cn[nH]c2)C1)OCC c1(C(N(C2CN(C(c3cc(F)cc(F)c3)=O)C2)C)=O)ncc(Cl)cc1Cl N1(C(C2(C)CCC(=O)N2)=O)CC(C2(NC(c3cncc(C#N)c3)=O)CC2)C1 C(=O)(CC(C(C)C)NC(=O)OC(C)(C)C)NC(CNC(COCC=C)=O)C(C)C Cc1cccc(C(=O)NC2CCCN(C(C3COCOC3)=O)C2)c1F C=CCC(C(=O)N1CCC(C(=O)N(C)C(c2cccs2)C)CC1)OC N1(C(c2cnc(CC)[nH]2)=O)CCC(NC(c2nncn2C2CC2)=O)C(O)C1 N1(C(CN(C2CCC2)C)=O)CC2CC(NC(=O)CCC3CCCCO3)C(C2)C1 C1(C(N2CC(O)(C(C)NC(CSCC(C)C)=O)C2)=O)CC(C)CCC1C(C)C N#Cc1ccc(CC(=O)NC2CS(=O)(=O)CC2NC(c2ccncc2)=O)cn1 C1(CNC(CC=CCC)=O)CCCCN(C(c2nc(Cl)c(Cl)s2)=O)CC1 c1(CNC(CCc2cc(C)on2)=O)ncccc1CNC(=O)C(C)C#N C(=O)(C1=NNC(=O)CC1)N1C(CCCNC(CC(C)SC)=O)CCC1 c1(CC(=O)NCCC(CNC(C2C(C)C2)=O)O)c[nH]c2cccc(F)c12 CC(C)C(C(=O)NCC(CC(F)(F)F)NC(=O)CC1CC(=O)C1)C(C)C N1(C(C2CC(CCC)C2)=O)CC(CNC(c2cc(C)n(CC)n2)=O)CC1(C)C N1(C(CN(C(=O)CC(O)CC)c2ccc(C(C)=O)cc2)=O)CCC2CCCC2C1 Cc1cc(C(N2CCC(C)C2C(=O)NCC(C)(C)C2CCCC2)=O)c(O)nn1 CC1(C)CC(NC(c2cccc(C#N)c2)=O)CN1C(=O)CC1CC=CC1 Cc1ccncc1C(N1CCCC1CC(=O)NCCn1ccc(=O)cc1)=O c1(CNC(=O)C(N2CCC(CCO)C2)=O)cc(F)c(O)c(F)c1 N1(c2nc(=N)[nH]o2)CCCCC1c1ncc(C(F)(F)F)cn1 c1(C(N2CC(NC(=O)C(C)NC(N)=O)CC(C)C2)=O)c([N+](=O)[O-])cnn1C C1(NC(C2CCC(=C3CCC3)CC2)=O)CN(C(=O)COc2cn[nH]c2)CCC1CO c1(C(N(C2CCN(C(=O)Cn3cccc3)C2)CCC)=O)cnc(OC)nc1 Cc1ccnc(C)c1C(C)(C)NC(N1CCC1Cc1c(Br)cnn1C(C)C)=O C(=O)(CC(CC(N)=O)CC(C)C)NCC(CC(C)C)NC(c1cc(C)nn1C)=O C=CCCCC(C(=O)NCCOCCC)NC(c1cnc(O)c(C)c1)=O N1(C(C(CC=CCC)C)=O)CCOC(C(=O)NCC(O)CC(C)(C)C)CC1 C1(COC)(NC(c2ccnc(C)n2)=O)CCN(C(C2CCCO2)=O)CC1 c1(C(N2CC(N(C)C(C3CCC3(C)C)=O)C2)=O)cncc(P(C)(C)=O)c1 C(N(C)N1CCC(N(C)C(=O)OC(C)(C)C)CC1)C1CC(NC(CC)CC)C1 C1(C(=O)NCC2(c3ccncc3)CC2)CC2CC(F)(F)CC(C1)C2(F)F N1(C(C(c2cccc(Br)c2)C)=O)CC2(CCCN(C(C3(C)C=CCC3)=O)C2)C1 C(=O)(C1=CC2C=CC1C2)N1CCC(C(=O)NCCN=[N+]=[N-])(CC)CC1 c1(OC)oc(C)nc1C(=O)NC1CC1CNC(c1ccc(CS(C)(=O)=O)o1)=O Cc1ncc(F)c(NCCCN2CCN(C(c3[nH]nnc3C)=O)CC2)n1 C1(NC(=O)OC(C)(C)C)CC1C1CCN(C(c2cc(Cl)cc[n+]2[O-])=O)CC1 c1(-c2cn(C3CCN(C(c4ccc(CSC)o4)=O)CC3)nn2)ncc(Br)c(O)n1 c1(NC2(CC(N3CCOC4CC34)=O)CCC2)ncnc2cc[nH]c12 C1(C(=O)NCCCCC#CC)CC12CCN(C(C1(N(C)C)CCC1)=O)C2 N1(C(C2CCC(=C)CC2)=O)CC2CCCC2(NC(c2cnncc2C)=O)C1 N1(C(C(=O)N2CCCC2)CCC2CCOCC2)CCC(O)(c2ccc(Br)cc2)CC1 c1(OC)ccc(O)c(NC(C2(F)CCN(C(c3c(Cl)cccc3Br)=O)CC2)=O)c1 C(C)(C)(CCC(=O)NC(Cc1ccc(Cl)cc1Cl)CC(C)C)OCC c1(CC(N2CC(N(C(c3nc(OCC)sn3)=O)CCO)C2)=O)cccc(OC)n1 C1(C(=O)NCC(C)C(=O)NCC2CC2)CCCC(C)(C)C1 N1(C(c2ccc(F)cc2Cl)=O)CCCC2C1CCN2S(=O)(=O)c1cccc(Br)n1 N1(C(c2ccc(OC)nn2)=O)CC(NC(c2cc(C(F)(F)F)n[nH]2)=O)CC(F)C1 c1(CNCC(F)(F)N(c2ccccc2)C)cc(F)cc(Br)c1F c1(C(N2CC(N(C(=O)CNC(c3ccccn3)=O)C)C2)=O)ccc2cc[nH]c2c1 C1(OCC(=O)NC(CCC)C)CCN(C(=O)CCOC(C)C)C1 N1(C(C2NCC(N=[N+]=[N-])C2)=O)CCC2C(F)(F)C2(c2ccccc2)C1 c1(C(COCC(=O)NCC2(NC(c3cnn(C4CC4)c3)=O)CC2)F)ccccc1 N1(C(CCCC(N)=O)=O)C2CCC1CC(CNC(c1ccnn1C1CC1)=O)C2 CC1CN(C(c2ccc3c(c2)CC3)=O)CC(C)CN1C(=O)C1=CC2CCCC12 c1(C(=O)O)cccc(Nc2cccc(C3CCCN(C4CC4)C3)c2)c1 C(C(O)C(=O)NCCCC(=O)OC(C1CC=CCC1)C)SC CP(C)(=O)C(CC(=O)N1CCCC1c1ccccn1)c1ccccc1 c1(CC)cc(C(N2CCN(C(=O)CC3CNC(=O)C3)CC2)=O)c(C)o1 C1(NC(C(c2ccnn2C)NC(c2cccc(C)c2)=O)=O)CCC(C2CC2)CC1 c1(C(=O)NCCC2CN(C(C(CN(C)C)O)=O)C2)ccc(F)c(Cl)c1F C1(C)(CCNC(c2nc(C)sc2)=O)CCN(C(=O)CCCC#N)C1 C1(c2n(CCCOC)nnn2)(Nc2cc(F)cc(Br)c2)C2CCC(C2)C1(C)C c1(C(=O)NC2CC3CC(NC(c4ccccn4)=O)C2C3)cc2nc(=O)ccn2[nH]1 Cn1cc(C=CC(N2CCC(O)(CCNC(=O)CN3CCS(=O)CC3)C2)=O)nn1 c1(CC)cc(C(=O)NCCC2(OC)CN(C(C34CC(C)C3C4)=O)C2)sc1C c1(C(=O)NC(C2CCCN2C(=O)C=C2CCC2)(C)C)n[nH]cc1F C(c1cc(Cl)cc(Cl)c1)=CC(N1CCCC(CNC(CC(C)SC)=O)C1)=O c1(C(=O)NC2(CCO)CCC2)conc1CNC(=O)OCCCl NC(=O)CCCCC(=O)NC1CCN(C(c2n[nH]c(C3CC3)n2)=O)CCC1CO C1(NC(C(C)CCN(C)C)=O)CCCCC12CCN(C(C1CCCOCC1)=O)C2 CC1CN(C(=O)C2=CCCCCC2)CCN(C(c2cccn3ccnc23)=O)C1 c1(C(=O)NC(C)CNC(C2CCC(C#N)CC2)=O)ccc2scc(Br)c2c1 N1(C(c2n[nH]c(C)c2Cl)C(=O)NCC2CCCO2)CCCC2NC(=O)CC12 C1(C(N2CCC(C(=O)OC)C2C)=O)CC(F)CCN1C(=O)C(c1ccccc1)F C(=O)(C(F)CCC(C)C)N1CC2(CN(C(C3N(C(CCC)=O)CCCC3)=O)C2)C1 C1(CC)C(C(=O)Nc2conc2C)CCN1C(=O)Cc1ccns1 c1(C(N2C3(CN(Cc4c(OC)c(Cl)ccc4)C3)CC2)=O)ccc(C#N)cc1C CC1CCN(C(=O)CN2CCCCC2)C1C(=O)NC1(C2CCCCO2)CC1 C1(CNC(c2c(C)nn(C(C)(C)C)c2)=O)CN(C(=O)CCC2CC2C)CCC1C c1(C(N2CCCCC(NC(C3C(C)CCO3)=O)C2)=O)cn2cccnc2n1 Cc1ccc(O)c(C(N2CCOC(CCCNC(=O)CC(C)N(C)C)C2)=O)c1 c1(NCC(CC)(C)CO)[nH]c(=NCCCOCCN(C)C)nc2c1ncn2CC C1(OC)CCCC(NCC2(C(F)(F)F)CCCCCC2)CC1 CC(C)CC(C)(CNC(=O)Cc1cnns1)NC(=O)CCOCC(F)F C=C(C)C1OCCC1C(=O)NCCC1COCCN1C(=O)CCNC(C)=O c1(C(=O)NC2(CC(N3C(COC)CC3)=O)CCC2)sccc1CSC C(=O)(C(Cc1ccoc1)NC(N)=O)NCCN(C(C(C)N1CCCC1)=O)C c1(C(=O)NC2CC(c3ccc(Cl)cc3)(O)C2)cc(Br)c2c(c1)OCCO2 n1(CC(=O)NC(CNC(C2N(CC)CCCC2)=O)(C)C)cnc2c1CCCC2 C(C)(C)(CC(=O)NCC1(O)CCCOC1)N(C(C(CC)NC(N)=O)=O)C c1(C(=O)NCC(CC)NC(=O)COCP(C)(C)=O)ncc(C#N)cc1C N1(C(c2c(Cl)cccc2Cl)C(=O)OC)CCn2cc(Br)cc2C1 C1(OC)CC(NC(=O)C(=O)NC(C)CNC(N)=O)N(c2ncccc2C)C1 Cc1cc(CCC(=O)NCC2CC(C)(CNC(=O)CCNC(N)=O)C2)c(C)s1 C1(C(N2CC3C(NC(c4ccc(O)c(F)c4)=O)C(C3)C2)=O)CCC2CCCCN12 N1(C(C2C(=C)CC2)=O)CC(OC)CC1CNC(c1ccnn1C1CCCCC1)=O C(=O)(CC(C)C(C)(C)C)N(C1(c2ccccc2)CN(c2cnc(F)cn2)C1)CC N1(C(C)C)CCCC1C(=O)NC1CN(C(c2cnn(CC3CC3)c2)=O)C1 C(=O)(C(C1=NOCC1)N(C1(C(=O)OC)CC1)C)NCCCC(=O)OCC Cc1ccc(Br)c(C(=O)NC2CC(NC(=O)C(O)C(F)F)C2)c1 C=C=CC(C)C(=O)N1CC(CNC(=O)CCc2cnc(C)s2)(OC)C1 c1(C(=O)NCC(CNC(C2(C)CC3CC3C2)=O)O)ccc(S(N)(=O)=O)o1 N1(C(C(C)(C)C2(O)CC2)=O)CCCC(CCNC(c2cocc2C(N)=O)=O)C1 c1(N(CC(F)(F)Br)C)nc2cccnc2c(=NCC2CC2(C)C)[nH]1 C1(C(=O)NC(CC)CN(C(=O)CC2CCN(C)C2=O)C)CC2CC(=O)C1O2 CCC(CCCO)N=c1cc(C)nc(N2CCOC3(CCSC3)C2)[nH]1 c1(CNC(c2n(CCOC)nnn2)c2cc(C(=O)OC)cs2)ccnc(F)c1 CC1(CNC(C2CC(C3CC3)C2)=O)COCCN(C(=O)Cc2cc[nH]c(=N)c2)C1 c1(CC(=O)NCC2C(NC(c3cn(CCCC)nn3)=O)CC2)nc(C)sc1C c1(CNC(=O)CC2CCCN(C(=O)CC3CCOC3=O)C2)cccc(O)c1F N1(C(c2c[nH]nc2[N+](=O)[O-])=O)CC2CN(C(=O)CC3CC4(CC4)C3)CC2C1 C(CC(C(C)C)NC(=O)C(C)(C)C1(O)CCOC1)NC(c1c(C)scc1)=O C1(NC(c2ccc(CCC)s2)=O)CCCCC1NC(=O)CC(O)CC c1(OC)ccc(C(C)NC(=O)NC2CC3(CC(OC)C3)C2)cc1OC(F)F C1(C(N(C2CCN(C(C=CCOCCOC)=O)C2)CC)=O)COC2COCC2O1 c1(C(=O)NCC(C)N(C(=O)C=C2CCCC2)CC)cc2ccc(F)cc2o1 CN1CCn2nc(C(=O)NC3CC3NC(=O)Cc3cc(Cl)ccc3O)cc2C1 C12(CNC(c3csc(Cl)c3)=O)CCC(CNC(C3CC4C=CC3O4)=O)(CC1)CO2 c1(OCC)ccc(C(=O)NC2CC2NC(c2ccc(CCO)cc2)=O)cc1 C1(NC(C(C)OCCOCC)=O)CCN(C(=O)CC2(CC(=O)OC)CC2)C12CCC2 C(=O)(CCC(C)(C)C#N)N1CC2C(CCNC(c3cc(OC)ncn3)=O)(CC2)C1 C1(C(N2CC3C(NC(c4[nH]ccc(=N)n4)=O)C3C2)=O)Cc2cccnc2C1 c1(CC)nc(O)c(C(=O)N(C(C)CNC(=O)Cc2ccc(Cl)c(C)c2)C)cc1C C(=O)(C(=O)CCC(C)(C)C)N1CCC(C(=O)OCc2c(OC)c(Cl)ccc2Cl)C1 C1(C)(NC(C2CC(C)(CC)C2)=O)CCN(c2nc(Cl)ncc2C(F)(F)F)CC1 C1(CC(=O)NCC2(C(N(C)Cc3ccco3)=O)CC2)CSCCO1 C1(NC(CN2C(C)CCC2C)=O)CCSC12CN(C(c1ccc(Cl)nc1O)=O)C2 N1(C(c2cnc(OC)c(C)c2)C(=O)NCCC)CC(C)c2ccc(OC)cc21 C1(C(=O)NCC2C(NC(CCCC#CC)=O)C2)CN2CCCN1CC2 N1(C(C(C)C2CC2)=O)CC(NC(c2coc(-c3ccccc3)n2)=O)C(C(F)F)C1 c1(C(=O)NCCn2ncc(C(N3CCN(C(C#C)C)CC3)=O)c2)cnc(C=C)cn1 CCC(C)(CO)C(=O)NC1CC(CNC(=O)C(C)C(O)CC)C1 C1(C(N(CCCCC)C)=O)CCCCC1CNC(=O)C(=Cc1ccco1)C S(=O)(=O)(c1cccc(CNC(=O)C(=O)Nc2ccc3c(c2)NC(=O)C3)c1)NC C(=O)(C1Cc2c(Cl)cccc21)NC1CCN(C(C(CCC)OCC)=O)C1C C(=O)(C(C)C(C)C)NC(c1cccnc1)C(N1CC(O)(CCC)C1)=O C1(C(N2CCCCC(N(C(=O)CCC3CCCC3)C)C2)=O)CCCCCC1(F)F C12(C(N3CCCN(C(=O)CC4CCC5(CCC5)O4)CC3)=O)CC3CC(CC(C3)C1)C2 Cc1cccc(OCC(N2CCC(CNC(c3cncc(Cl)c3C)=O)C2)=O)c1C C(CC(=O)N1CC(CC23CC(C2)C3)C1)NC(C1C(C)C1)=O.C12CCC1C(=O)N2 c1(C(N2CC3CN(C(N4CC(c5ccccc5)C4)=O)C3C2)=O)cn2ncccc2n1 CCC(CC)CC(F)C(=O)N(C)CC1(O)CCN(C(=O)C(C)N(C)C)CC1 c1(C(C)C)ccc(C(N2CCCC2C(C)NC(C2CC23CCCC3)=O)=O)nc1 C(=O)(C1CCCc2nccn21)N1CCC(CCNC(C(N)=O)=O)C1 N1(C(C(CCOC)OC)=O)CCC(C(=O)Nc2cn(CCF)nc2C)(CC)CC1 C#CCCC(O)C(=O)NCC(O)CCNC(c1sc(C)cc1C)=O CC1(C)OB(C2CNC2)OC1C(N1CCC12CCS(=O)(=O)C2)=O N1(C(C(c2ccccc2)OCC)=O)CCCC(N(C(=O)CCc2cncs2)C)C1 N1(C(C(CC=C)(C)C)=O)CCC2C1CCCN2C(=O)C(Cl)=CCl c1(OCCCC(=O)NCC2CC(NC(C3C(C)CC3)=O)C2)ccc(F)cc1F N1(C(C2C(c3ccn(C)n3)C2)=O)CCCC(CO)(NC(=O)Cc2ccco2)C1 c1(C(=O)NC(CN(C(COC(CC)(C)C)=O)CC)C)ccc2nccn2c1 N1(C(CCCC)=O)CCCC2CN(C(c3cc(F)ccc3F)=O)CCC12 C1(NC(CC2ON=C(CC)C2)=O)CC2CC1N(C(c1ccoc1CC(N)=O)=O)C2 C1(C(=O)NCCN(C(C(C=C)(F)F)=O)C)CCc2c(cnn2C)C1 N1(CCCNC(=O)NC2CC(C(CC)CC)OCC2)C(C)(C)CCCC1(C)C O=C(CNC1CCN(c2ccc(Cl)c(Cl)c2)CC1)NN=c1ccc(Cl)n[nH]1 C1(N(C(=O)C(C)O)CC)CCN(C(C2(C#N)CCCO2)=O)CC1 C(=O)(CCCCC(N)=O)N1CC(NC(c2c(N(C)C)cncc2)=O)C(CO)CC1 C12(NC(c3ncc(Br)cc3F)=O)CCN(C(=O)CCCc3ncco3)CC1C2 C1(C(=O)NC(C#C)C(C)C)(CC)CCN(C(=O)CC2CCCC2)C1 C1(CC)CN(C(=O)C(c2ccccc2C)(C)C)CC1NC(=O)C(CC)OC Cc1nc(C(=O)Nc2ccc(N(C)C(C3C4CNC3C4)=O)cc2)nc(C)c1Br c1(OC(C)C(=O)NCCOc2cc[nH]c(=N)c2)ccc(Br)cc1F C1(NC(c2c(C)cns2)=O)CCCCN(c2nc(Cl)ncc2Cl)C1 C1(C(=O)NC(C#CCC)(C)C)C2CCCC2CN1C(=O)CCC(=O)NCC c1(N2CC(NC(c3cc(C)[nH]c3)=O)CC3(C2)CC3)cc(C)c([N+](=O)[O-])cn1 C1(C)(NC(CSCCN(C)C)=O)CCN(C(=O)C(F)(F)CN2CCCC2)C1 Fc1ccc(I)c(NCc2ccc(OCc3ccccc3F)cc2)c1 C1(NC(C2CC3(CC(OC)C3)C2)=O)CC2CC1CN(C(=O)Cc1n[nH]c(C)n1)C2 c1(C(=O)NC2CC(CNC(=O)C=C3CCCC3)C2)cc2ccsc2[nH]1 C1(C(=O)NC2CC(F)C(=O)N2)CC2(CCN(C(=O)C3=CC4C=CC3C4)C2)C1 S(=O)(=O)(c1ccc(N(C)CCO)c2cnccc12)N1C(CN)CC(O)C1 C1(C(N2CCC(O)(C(C)C)C2)=O)COC2(C1)CN(C(=O)CCCn1cncn1)C2 CC1(C2CCN(C(C3CCCN(C(c4cccc5[nH]ccc45)=O)CC3)=O)C2)CC1 Cc1nc(C)c(C(N2CCC2CNC(c2cncc(-n3ccnn3)c2)=O)=O)o1 CN1CCC(C(=O)OC2(CSC3CC3)CCOCC2)C1=O N1(C(c2ccc(CC)[nH]2)=O)C(C(=O)NC(CO)CC(C)C)CCC1C C1(C(N(C)CC2CN(C(=O)C(c3csc(=N)[nH]3)=O)C2)=O)Cc2cccnc2C1 N1(C(C=C(CC)C)=O)CC2CCC(C1)N2C(C1CC(OC)(OC)C1)=O C(=O)(CCCS(N)(=O)=O)N1CC2C(CNC(C(c3cccc(F)c3)(C)O)=O)(C2)C1 C#CCC(C(=O)OC)NC(=O)CNC(=O)CC(CC)SC C1(O)(C(N2CC(NC(C(=O)NC(C)C)=O)C2)=O)CC(C)(C)C1 C1(C(N(C)CC2CCN(C(c3cc(C(N)=O)c[nH]3)=O)C2)=O)CCCNS1(=O)=O N1(CC)CC(Nc2cc(NC3CC4CC4C3)nc(C)n2)CCC1=O Cc1sc(C(N2CCCC(O)(CCNC(c3cc(O)cs3)=O)C2)=O)c(C)c1C C1(CC(=O)NC2C(CNC(C3CC(SC)C3)=O)CCC2)CCC(C)CC1 N1(C(c2c(C)nc(C)[nH]2)=O)CCCN(C(C2CC(F)(CF)C2)=O)CC1C Cc1oc2cc(C(=O)NC3CN(C(c4cc(C(C)(C)C)n(C)n4)=O)C3)[nH]c2c1C C#CCCC(O)C(=O)NCC(CC)NC(=O)C(c1ccc(Br)cc1C)(C)C N1(C(C=CCCCCC)=O)CC(NC(=O)C(C(C)C)n2ccnc2)CC1(C)C C1(OCC)CC(C)N(C(c2cn(C)ccc2=O)=O)C(C)C1 C(C)(C(=O)NCCC1CN(C(C2(CCF)CCC2)=O)C1)(C(C)C)NC(C)=O c1(OC)ccc(S(=O)(=O)Cc2ccnn2C2CCCC2)cc1Cl C=CCC(CC(=O)N1CCCC1C(O)CO)NC(c1n[nH]cc1CC)=O C1(NC(C2C(C(C)(F)F)C2)=O)CCN(C(c2cc(N)cnc2Cl)=O)C12CCC2 Cc1c[nH]cc(C(N2CC=CC(NC(c3c(Cl)n[nH]c3C3CC3)=O)C2)=O)c1=O C1(C(=O)NC2CN(CCC)C(=O)C2)CCN(C(c2cnn(C)c2Cl)=O)C12CCC2 Cc1nc(C(=O)NCC(C2CC2)NC(c2cccc(CF)c2)=O)nn1C C(=O)(CC(C)(C)CN(C)C)N1CC(NC(C(C)OC)=O)C(c2ccccc2)C1 C(=O)(CC(O)C(C)CC)N(CCOCCCNC(c1cc(COC)oc1C)=O)C C(=O)(C(CNC(=O)C(C(C)C)NC(C)=O)CC1CC1)NCC(C(=O)NC)O C1(NC(C2(CCC)CC2)=O)CN(C(C2CCOC2)=O)C2(CCCCC2)C1 c1(NC(C(CCNC(C2CC2C(F)F)=O)OC)=O)ccc(O)cc1Cl N1(C(c2[nH]cc(C(C)=O)c2)=O)CCCC(CNC(c2onc(Br)c2C)=O)C1 O=C1CC(CC(=O)NCC(O)CNC(C2(Oc3ccccc3)CC2)=O)CC(=O)N1 Cn1nnc2cc(C(=O)NC3CCCC(NC(C4CNC(=O)C4)=O)C3)ccc12 C1(C(=O)NC(CCC=C)CO)CN(C(c2ccc(CC)cc2)=O)CC1(C)C N1(C(c2ccn(C)c2)=O)CCC(=O)NC2CN(C(=O)CC3=CCCCC3)CCC12 c1(CCC(=O)NC2(C)CCN(C(=O)C(F)=CCCF)C2)cccc(F)c1F C=C=CC(C)C(=O)N1CCOCC1CNC(=O)CCc1cnn(C)c1C C1(C(=O)NCCc2ncn(C)n2)CC2(CCC2)CN1C(=O)CCC(CF)CF N1(C(=O)COc2nncs2)CCCN(C(=O)COCC2CCOC2)CCC1 C1(CC=C)(NC(c2ccnn2C2CC2)=O)CCN(C(C2(n3ccnn3)CC2)=O)C1 c1(CNc2[nH]c(=NCCS(CC)(=O)=O)[nH]c(=N)n2)ccc2nsnc2c1 CCCC(C)(C)CC(=O)N(CC(=O)NCc1cnco1)OC C(=O)(C1=CCCSC1)NCC(C(=O)NC(CO)CCC1CC1)OC C(C)(C(F)(F)F)(c1ccc(NC(C)=O)cc1)NC1CN(CC)C(=O)C1 N1(C(C(CNC(CCCCCC=C)=O)C(C)C)=O)CCC12CCC(O)CC2 CC1C2CCC(C2)C1C(=O)NCC1(NC(C2CSCCS2)=O)CC1 C1(C(N2CCCC(CNC(c3cc(CF)on3)=O)C2)=O)COCC2(CCC2)O1 Cc1cc(-c2nnc(N(C)C(C)C3CC3)n2CC(=O)OC(C)(C)C)cc(Br)c1 N(C(=NCCCF)N1CCC(OC)C1)C(C#C)CC c1(OC)ccc(N(C(=O)C(C2CCN(C(=O)CCN(C)C)C2)C)C)c(C)c1 N1(C(C2C(NC(Cn3ncc(C#N)c3)=O)CC=CC2)=O)CC2CCC(CO)(C2)C1 C(CCCC(=O)NCC(F)CNC(=O)C(C)(C)Cc1ccc(O)cc1)NC(C)=O Cc1[nH]nc2c(C(N3CC(N(C)C(C4CNC(=O)CC4(C)C)=O)C3)=O)cccc12 C1(C)(CNC(C2C(C)(C)COC2)=O)CCCN(C(C2(C(C)(C)O)CC2)=O)C1 N1(C(CC)=O)C2CCC1C(C)C(NC(c1cccc3[nH]cc(Cl)c13)=O)C2 N1(C(C(CC)C2CC2)=O)CCC2(CCC2)C(NC(=O)COc2cccc(C)c2)C1 CCCCC(C)C(=O)NCC(O)CNC(=O)C(=Cc1ccc(C)cc1)C Cc1cc(C(=O)NCC2(F)CN(C(c3ccc4c(c3)NCC4)=O)C2)cn(C)c1=O c1(C(=O)NCC(c2ccc(OC)cc2)N)ccc(Br)cc1OC(F)F C(=O)(CS(=O)(=O)CCO)NC1CC(CCNC(c2c(C)csc2Cl)=O)C1 C1(C(N2CCCC(CCNC(CCNC(C)=O)=O)C2)=O)CCc2nccn2CC1 c1(C(N(CCCNC(C2CC3C=CC2C3)=O)C(C)C)=O)cccc(F)c1N N1(C(C(CC)CCOC)=O)CC(NC(=O)Cc2cc(C3CC3)on2)CC2(CC2)C1 C1(OCCCNC(C=CCOC)=O)CCN(C(=O)OC(C)(C)C)CC1 C1(NC(CCC=CC)=O)CC(OC)CN(C(C2CCCCN2CC(F)F)=O)C1 Cc1ccc(Br)cc1C(N1CC2C(NC(=O)C(C)S)C2C1)=O N1(CC)CCN(CCC(=O)NCC2CC2NC(=O)CCn2ccnn2)CC1 c1(C(=O)NCC2CC(F)(F)CN2C(=O)CC2CC=CC2)ccn2nnnc2c1 c1(C(=O)NC(COC)CC(=O)NCCC2CCCC23CC3)ncc2ccccn12 C12(NC(C(C)(C)CC3CC3)=O)CCCC1CS(=O)(=O)C2 c1(CC)cccnc1C(N1CC(CNC(c2snnc2C)=O)C(C)C1)=O c1(CC)nc(N2CCCC(C)(CNC(=O)C(F)n3cccn3)C2)c(C#N)cc1C S(=O)(=O)(CCCCCl)N1CCC(C(F)(F)F)(OC)CC1.C1C(=O)N1C(C)=O O=C(C1=CCCCCC1)NCC1CC1CNC(c1ccc(C2CC2)cc1)=O C1(C(C)NC(=O)C(O)C2CCC2)CN(C(=O)CC2CS(=O)(=O)C2)CCO1 CCC(O)C(F)(F)C(=O)NCC1(CCCNC(C2(OC)CC2)=O)CCCC1 c1(C(=O)NCC(CC(C)C)NC(c2ccc[nH]2)=O)c[nH]c2nccc(Cl)c12 N1(C(CC2N(C(C(CC)C(F)(F)F)=O)CC(O)C2)=O)CC2CCC(C1)C(=O)N2 Cc1ccc(CC(=O)NCC(CC(F)(F)F)NC(=O)CC(C)F)cc1F N1(C(Cc2c(C)n[nH]c2)=O)CCC(F)(C(=O)NCCC2CC(C)(C)CO2)C1 c1(C(N2CCC(O)(CN(C(CCCOC)=O)C)CC2)=O)n[nH]c2c1CCSC2 C1(COC)(CNC(=O)C(C)(C)C2CCCCC2)CCCN1C(=O)C(CO)N(C)C CC1COC2(C1)CN(C(C1CN(C(=O)C(F)(F)CO)CC1(F)F)=O)C2 C=C1CCC(C(=O)NC(C(=O)NCC2CNC(=O)C2)C(C)OC)CC1 Cc1nc2c(C(=O)NC3CCC(C)N(C(=O)CCC(=O)N(C)C)C3)cccc2o1 c1(OC)ccc(CCC(=O)NCC2(CNC(c3cnnc(O)c3)=O)CC2)cc1Cl CC1(C(=O)NCCC2CC2C2CC2)CCN(C(=O)Cc2cc[nH]c2)C1 C1(C2(O)CCC2)(C(=O)NCCNC(C2CCCS(=O)(=O)C2)=O)CC1 C(=O)(C#CC1(C)CCCO1)NCCCC(C)NC(Cc1nc(CC)sc1)=O c1(C(=O)NC2CC(C)(NC(c3cnn(C(C)C)c3N)=O)C2)cnc2ncccn12 N1(C(C2CCCC(C)(C)C2)=O)CCC2(CC1)CC2NC(=O)Cc1cccnc1O N1(C(C2(S(C)(=O)=O)CC2)=O)CC2(CCN(C(=O)C(c3ccc(F)c(Cl)c3)O)C2)C1 C1(C(N2CC(CNC(CCC3CCCN(C)C3)=O)C2)=O)OCCN(C)C1=O C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(C23CC(CO2)C3)=O)CC1F C1(NC(C2CCN(C)C2=O)=O)CCC2(CC1)CN(C(C1C3COCC13)=O)CCO2 c1(CCC(=O)NC(C)CNC(C2(c3ccccc3)CC2(C)C)=O)ccc(Cl)cc1 N1(C(C(CCC)NC(C)=O)=O)CC2CCC2(NC(C2CC(OCC)C2)=O)C1 C(C(CCN=C(NCC1(OC)CCOCC1)NC(C1(OC)CCC1)C)OC)OC N1(C(C2CC(NC(CCC(C)OC)=O)C(O)C2)=O)CCC12CCN(C)C2 N1(Cc2c(-c3ccccc3)nccc2)CC(c2cccs2)CC(c2ccccc2)C1 C1(C(N2CC(CC(C)NC(=O)Cc3scnc3C)C2)=O)(COC)CCCO1.C1CC1 C1(CNC(C(C)(C)CC2CC2)=O)C(O)C(O)CN1C(c1ccc2c(c1)CC2)=O Cc1cc(=O)oc(C)c1C(=O)NCC1(O)CCCN(C(C2OCCC2C(C)C)=O)C1 C=C(C)CN=C(NCc1cc2sccc2s1)N(C)Cc1nnnn1CC(=C)C Cn1nc(Cl)c(C(=O)NCC(C2CCOC2)NC(=O)C(C)(C)C#N)c1Cl N1(C(CC(CC)O)=O)CC2CCN(C(=O)C(F)Cl)C2C1 Cn1cnc2c1C(C(=O)NC1CC(NC(=O)CCP(C)(C)=O)C1)CC(=O)N2 Cc1cc(C(=O)NCC(CO)NC(=O)Cc2nnn(C(C)(C)C)n2)cnc1C c1(CC)cc(C(=O)N(C)CCOCCC(=O)N2CC(CC(C)C)C2)c(C)o1 C=C1CCN(C(=O)CCn2ccc(C)n2)C(C(N2CC(=O)NCC2CC)=O)C1 CC(C)CC(CNC(=O)CC(C)(C)O)NC(C1CCN(c2nccn2C)C1)=O CCC(C(=O)N1CCCN(C(=O)CN(C)Cc2ccc(Cl)s2)CC1)C(C)O CC1=CC(NC(c2oc(CNC(=O)Cc3ccccn3)nc2C)=O)CCC1 c1(C(C(N2CCC(N(C(=O)CC3CC3)CC)C2)=O)C)c(F)cccc1F N1(C(C2CCC(C(C)C)CC2)=O)CCC(NC(=O)C=CC2CCCO2)C(C)(C)C1 N1(Cc2onc(-c3ccc(OC)cc3)n2)CCc2c(O)ncnc2C1.c1ccccc1 CC(C)C(CN(C)C)C(=O)NC(C)CNC(=O)C(C)NC(c1ncccc1F)=O C1(NC(c2cc(CNC(c3c(OC)scc3)=O)[nH]n2)=O)CN(C)CCC1O c1(C(C(=O)N(C)CCNC(c2csc(C3CC3)n2)=O)O)ccccc1Br Cc1cc2cnccc2n1CCNC(=O)NCc1ccnc2cc[nH]c12 c1(C(=O)NCC2CN(C(C3(CC(C)C)CC3)=O)C2)cc(C#N)ccc1N c1(NC(=O)NC(C2CCCN(C(C)=O)C2)C)nnc2ccc(OC(F)F)nn12 c1(CC(=O)NCC(CN(C(C2(CCC)CCC2)=O)CC)(C)C)ccc(F)cn1 C1(NC(c2ccn3ccsc23)=O)CCN(C(=O)CCc2cnc[nH]2)CC1O C1(C(=O)NC2CC(NC(CCc3n[nH]c(=N)s3)=O)C2)CCC2(CCOCC2)O1 N1(C(C2C(CC)CCO2)=O)CC(CNC(=O)CN2CCOCC2=O)CC12CCC2 C1(CC(=O)NCCC2(OC)CCC2)C2CCCC2N1C(=O)COCCCC(C)C c1(C(=O)NC(CC=C)CNC(=O)CC(C)C2CC2)cc2cc(Cl)ccc2n1C c1(C(C(=O)NCC)N(CC(C)C#N)CC2CCCC2)oc(C(=O)OC)cc1Br c1(C(N(C2CCC(NC(C(CC#C)O)=O)CC2)C)=O)cnc(O)cc1C C(=O)(C1CCc2cccnc21)NCCN(C(c1c(CC)[nH]cc1)=O)CC C1(C(N2CCC(C(C)NC(c3nncs3)=O)CC2)=O)CCC(C)(C)CC1 CC#CCCCC(=O)N1CC2(NC(c3ccc(CCC)cc3)=O)CC1C2 C1(C(N2CC(NC(CCNC(=O)NC)=O)C2)=O)CCS(=O)(=O)C1 C1(COC(C(=O)N(CCNC(C2(CCOC)CCCC2)=O)C)C)CCCCCC1 C1(F)(CNC(C=CC(C)(C)SC)=O)CC(NC(C2CCC(N(C)C)C2)=O)C1 Oc1ccc(CNCc2ccc(-c3cncc(O)c3)nc2)cc1 CCCC(C(=O)NC(C)(CNC(=O)CN(C)C)C1CC1)NC(c1ccccc1)=O c1(C(=O)NC2(CNC(c3nc(C)oc3C)=O)CC2)ccc2c(c1Cl)OC(F)(F)O2 C1(C(=O)NCCCNC(c2ccco2)=O)CCn2c(O)nnc2C1 N1(C(c2cc(C)on2)=O)CC(NC(C2COC(=O)N2C)=O)C(n2ccnn2)C1 c1(C(=O)OCC)cc(C(N2CCC(n3cncn3)C2)=O)cs1.C1(=O)CC2(CC2)CN1 c1(OCC(=O)OC)c(C)cc(COC(c2cc(Cl)ccc2C(C)(C)C)=O)cc1C c1(-c2nc(C(C3(C)CC3)C)nn2-c2ccc(Br)c(F)c2)ccc2cncn2c1 CC1C(=O)N(C)CCN1C(=O)C(C)N(C(=O)C=Cc1ccsc1)C1CC1 c1(C(=O)NCC(c2ccsc2)C)cc(-c2ccccc2)n2cnc(C(N)=O)c2n1 C1(NC(C(COC)C)=O)CCN(C(c2ccc(OC)cc2C)=O)CC1OC C1(NC(c2ncc(Br)cc2F)=O)CC2CC1N(C(=O)CC13CC(C1)C3)C2 C=CCCCCCCC(=O)NC1CN(C(c2ccc(C#N)[nH]2)=O)CC1O c1(OC(c2cn(C(C(N3C(CC)OCC3)=O)C)nn2)C)cccc(C(F)(F)F)c1 c1(C(C(N2CC(OCCNC(CC3C(C)CCO3)=O)C2)=O)=O)ccccc1[N+](=O)[O-] CC1CCCC(CC(=O)NCC23CC2CN(C(=O)C(C2CCOCC2)F)C3)O1 N1(C(c2c(C#C)c[nH]n2)=O)CCC2CC2(C(=O)NC2CC(C)(C)C23CCC3)CC1 Cc1cc(=NC2C=CCCCC2)[nH]c(N2CCC(COCCC(C)C)CC2)n1 C12(Cn3cc(C4(N(C)C)CCC4)nn3)CCC(CC1)N2C(C1CC(O)C12CCC2)=O CCCC(C(=O)NCCC1(OC)CN(C(=O)C(CC)N(C2CCCC2)C)C1)OC C1(NC(c2c(NC)snc2C)=O)CC(NC(=O)CCC=C(C)C)C12CCC2 N1(C(c2c(C)[nH]nc2Cl)=O)CC(C)(C)OC2(C1)CN(C(c1sncc1Br)=O)C2 c1(C(=O)NCC2(O)CN(C(c3cn(CCN(C)C)nc3)=O)C2)cnn2c1CCC2 N1(C(CC2CN(Cc3ccc(NC(C)C)c(Br)c3)C2)=O)CCN(C)C(=O)C1C N1(C(c2c(C)[nH]c(=NCC)s2)=O)CCCC2(C1)CN(C(=O)C(N)=O)C2 C1(CNC(C=C(CNC(C(CC)NC(N)=O)=O)C)=O)CC(O)C(O)C1 C(=O)(C(O)CC(C)(C)C)N1CC2(CC(CNC(C3OCCN(C)C3)=O)C2)C1 C(=O)(CC(C)(C)C(F)(F)F)N1CC(COC)C1.C12(CCOCC1)CC(=O)NC2=O.C CC1NC(=O)CCC1NC(N1CC(O)(CN2CCCC2)C1)=O N1(C(C2C(OC)C2)=O)CC(NC(=O)CCCS(C)(=O)=O)CC(F)(F)C1 C(C(CC1CC1)C(=O)N1CCC(c2nn[nH]n2)C1)NC(c1scc(C)c1)=O C1(NC(=O)C=Cc2cocn2)CN(C(=O)Cc2cncc(O)c2)C2(CCC2)C1 Cc1cc(C(N2CC3CN(S(=O)(=O)c4cccs4)CC3C2)=O)ccc1[N+](=O)[O-] N1(C(c2ccc(C)cc2)=O)CCC(C)N(C(C2CCCC(F)C2)=O)CC1 Cc1nc2c(NC(=O)C(=O)NCCc3nc(C(F)(F)F)cs3)cccc2o1 C(CC(C(=O)NC(CO)C1(C)CC1)NC(=O)Cc1cc(C)[nH]n1)OC C=C(C)CCCC(=O)N(CCCCN(C)C(c1ccc(C(=O)NC2CC2)s1)=O)C C(=O)(CS(=O)(=O)CC(C)C)NCC(CNC(c1c(C)cc(O)nc1C)=O)F c1(OC(C(C)C)C(=O)NC2CCN(C(c3ccco3)=O)C2C)c(F)cccc1F CCCCC(C)C(=O)N(C1CCN(C(=O)CC)C1)Cc1cncc(Cl)c1 C(=O)(C1=C(C)OCCC1)N1C(C)(CC)CC(NC(=O)CC=CC(C)(C)C)C1 c1(C(=O)NC(C2CCOC2)C)cnc(NC(C2(C)CSC2)=O)s1 C1(C)(NC(C(CC2CC2)NC(c2c(OC)csc2)=O)=O)CC(O)(CO)C1 N1(C(C2(C)CC(C#N)C2)=O)CCC(C2CC2)(CNC(C2CCCCNC2=O)=O)C1 c1(C(=O)NCC2(NC(CC(C(C)C)OCC)=O)CC2)cc2ccccc2cc1O c1(CSC)ccc(C(=O)NCCCCCNC(=O)C(F)CN(C)C)cc1OC c1(C(=O)NCC2(O)CC(NC(C(COC)(C)O)=O)C2)cccc2c1OCC2 CCC(O)C(=O)NCc1cc(CCNC2CC2)cs1 c1(OC)ccn2c(C(=O)NCCNC(c3cccc(C(C)C)n3)=O)cnc2c1 Cn1nc(C(=O)NCC(CC(=O)NCCCc2ccccc2)C2CCC2)cc1Cl c1(COC(c2ccncc2)=O)ccc(OC(F)(F)F)c(Cl)c1.CC1CNC1 CCC(CC(F)F)C(=O)NCC1COCC1NC(=O)CCOc1ccccc1 C1(C(N(C(CC#C)C)C)=O)CC=CC(NC(c2cncc(O)c2)=O)C1 C1(NC(C2(N(C)C)CCCC2)=O)CC2CCC(C1)N2C(=O)C(F)=CCCF c1(C(=O)NCC2C(CNC(CCNS(CC)(=O)=O)=O)C2)c[nH]c2nccc(Cl)c12 c1(C(=O)NC2(C)CC(NC(CCC3CCC(C)O3)=O)C2)coc2c1CCCC2 Cc1cc(C(=O)NC23CC(C2)N(C(c2cccc(C)c2Cl)=O)C3)n2nccc2n1 C1(NC(C2(OC)CC2)=O)CC(OC)CN(C(=O)C=Cc2ccncn2)C1 C1(C(=O)NCCC2CCN(C(c3cnn[nH]3)=O)CC2)C2Cc3ccc(Cl)cc3C12 N1(C(Cc2ccc(C)cc2)=O)CCC(NC(C2CNC(=O)N2)=O)C12CC2 C(C(CC)C(C)C)(c1nnnn1C1(C)CC1)N1CCC1.c1(OCC)ccccc1 C(=O)(CS(=O)C(F)(F)F)NC12CN(C(CCCC=C)=O)C(CC1)C2 C1(F)(C(=O)Nc2c(OCC)scc2)CCN(C(=O)C(CSC)CC)CC1 C1(C(=O)NC2CN(C(C3CCC(F)C3)=O)C2)CCC(O)CC1 C(C#CC(=O)NCC1CC1(C)C)NC(CN(C(C)C)C)=O CCC(C)(O)CNC(=O)CCC1CCN(C(C2CCC2C(C)(C)C)=O)C1 CC(C)CCC(C(=O)N1CCCCC(C)C1)NC(c1cccc(F)c1O)=O C1(CC(=O)NCC2(O)CCN(c3ncc(C(=O)O)[nH]3)CC2)CCCC2(CC2)C1 CC1=CCC(NC(c2ncoc2C(=O)NCC2(c3ccccc3)CC2)=O)CC1 c1(NC23C(CN(C(CNC(N)=O)=O)C2)C3)ncc2cc(Br)ccc2n1 C1(CCS(=O)(=O)NC)NC(=O)CCN(CC2C(C)C2C2CC2)C1=O c1(N(C)C)cncc(C(N2CC(O)(CCNC(C3CC3c3ccco3)=O)C2)=O)n1 C#CCCN=C(NCc1cc([N+](=O)[O-])ccc1N(C)C)N1CCC(C(C)C)C1 N1(C2CN(C(C(n3cc(Cl)cn3)C)=O)C2)CCN(C(C2COC(=O)N2)=O)CC1 c1(NC(C(CCC)C)=O)ccc(NCC(=O)OC(C)(C)C)cc1NC(C)=O C1(C(=O)NCCC2(CC(=O)O)CCCC2)CNCC1C1CCCC1 C1(OC)CN(C(c2nnn(C)c2C)=O)CC1NC(C1CCCN1CCC(C)C)=O c1(N2CCC(C=C)CC2)nc2c(c(=NCC3CCN(CC(C)C)CC3)[nH]1)CCC2 N1(C(c2cn(CCC)nn2)=O)CC2CCCN(C(=O)CC3CCC=CCC3)C2C1 N1(C(C2(NC(=O)C(O)C3CC3)CCSC2)=O)Cc2cccc(F)c2C1 CC1(c2cccc(C(F)(F)F)c2)CCCN1C(=O)NCc1cc(C(F)F)cs1 C(CCC(F)(F)F)N(C(=O)CCCc1sccc1Br)C c1(C(=O)NCC(=O)N(C)CC)cc(S(=O)(=O)NC(N)=O)ccc1Cl CC1CC2(CC(C(N3C(C(=O)NC4CCC45CCCC5)CCC34CC4)=O)C2)C1 n1(CC(=O)NCC)ccc(=NC(=O)C2CC2)nc1O.c12ccc(cc1)[nH]c2=O C1(C(N(CC(C)(C)C(=O)NCC2CC3(CCC3)C2)C)=O)CC2CCC(C1)C2 c1(C(=O)NC2C3CN(C(C(C)SCC)=O)CC2C3)cn(C)c2c(Cl)cccc12 N1(C(Cc2ccc(C)cc2)=O)CC(NC(=O)C#CC2CCCO2)C(S(C)(=O)=O)C1 N1(C(CC2CCN(OC)CC2)=O)CC(NC(=O)C(C)(Cl)Cl)CC12CCOCC2 C(=O)(CCC(C(C)C)NC(=O)C(C)c1cccs1)N1CC(OCC)C1 CC1(C)OC(C(N2CC3(C2)CN(C(c2ccc(S(N)(=O)=O)s2)=O)C3)=O)C(C)(C)O1 O=C1CN(C(C2(c3cccs3)CC2)=O)Cc2cc(Br)cnc2N1 C1(NCC(c2cc(F)cc(F)c2)OC)CCSC(C)(C)C1 c1(C(=O)NC(CN(C(C(C2CCCCC2)OC)=O)C)C)nncn1C Cn1ncc(S(=O)(=O)N2CC3CCCC3(NC(=O)OCc3ccccc3)C2)n1 N1(C(C)=O)CC(F)CC1C(=O)NCCOc1cccnc1C(F)(F)F CC(C)CCCC(C)CNC(=O)CC12CCC1CN(C(c1cc(Cl)cs1)=O)C2 N1(C(C(CCC)=CCC)=O)CCN(C(=O)Cn2cnnn2)CC1c1ncc[nH]1 CCC(CC)CC(F)C(=O)N1CCC(C(=O)NCCC2CCN(C)C2)(CC)C1 c1(C(N2CC(N(C(c3cc(CC)no3)=O)C)C2)=O)cnc(SC)n1C c1(-c2c(C)cco2)nc(C2CC(O)C2)n(-c2ccccc2F)n1 CCC(CC)C(=O)N1CC(CC(C)NC(C2(c3ccc(F)cc3)CCC2)=O)C1 c1(NCC)cncc(C(=O)N(CCCCNC(=O)CN2CC3CCC2C3)C)c1 C(C(C)(CC(C)C)NC(c1cnc(OCC)s1)=O)NC(C=CC)=O CCC(C)(C)C(O)C(=O)NCC1CCN1C(c1cc(C(C)(C)C)n(C)n1)=O c1(C(=O)NCC(CCNC(c2n(CC#C)ccc2)=O)(C)C)n[nH]c2c1CC1CC21 c1(OC)c(CNC2C(N)CC2O)cccc1C C1(F)(CNC(c2cccc(F)c2Br)=O)CCCN(C(C2CCC2)=O)C1 c1(C(N2C(CC(=O)Nc3ccc(OC)cc3)COCC2)=O)cnn2ccncc12 N1(Cc2c(C)nn[nH]2)CC2CN(C(=O)OCOc3ccccc3)CC2C1 CC1CC(C(=O)N(CCCNC(C2(CO)CC2)=O)CCO)CCC1=O c1(C(=O)NCC(CC)N(C(=O)CC2CCC(=O)N2)C)ccc(C2CC2C)o1 c1(C(N(C2CCN(C(C3ON=C(CC)C3)=O)CC2)C)=O)c[nH]c(=N)cc1C c1(C(C(=O)N(CCC(=O)OCC)C2CC2)N)ccncc1OC c12cc(cc(O)c1)C(=O)NC1CN(C1)C2=O.C1(CC(=O)OC)CCC(=O)N1CC C1(NC(C(CC)C(C)C)=O)COC2(CCN(C(=O)CCc3cnn(C)n3)CC2)C1 N1(C(c2ccn(CCNC(CC)=O)c2)=O)CCC(C)(C2CC2)C1 CONC(=O)C(=O)N(CC(C)NC(=O)CC(C)CN(C)C)C c1(CC(=O)NCC(CNC(C2CN(C)C(=O)C2)=O)O)ccc(F)c(Br)c1 C1(NC(C(C)Cn2cccn2)=O)CCC(C(=O)NCc2nncs2)CC1 N1(C(=O)C=C2CN3CCC2CC3)CCC2CCCN(C(c3ccsc3)=O)C2C1 C1(NC(C(NOC)=O)=O)COC2(CCN(C(C34CSCC3C4)=O)C2)C1 Cc1cnc2c(C(N3CCC(C4CC4)(NC(=O)CCCN(C)C)C3)=O)cnn2c1 CC(=O)C(C)(C)CC(=O)NCC1CC(C)N(C(c2ccc(C(F)F)o2)=O)C1 c1(C(C(=O)NCCCC2CC2)N(CCC)CCC)ccc(Cl)cc1C(F)F Cc1cc(Br)cc(C)c1C(N1CCN(S(=O)(=O)C2CC2)C(CC#N)C1)=O c1(C(=O)NC2CCN(C(CCNC(=O)OC)=O)CC2F)cc2cncn2c(O)n1 c1(N2CCC(CC=C)C2)ncc(S(=O)(=O)N(C2CCCC2)C)cc1Cl C(CCC(C)(C)C(=O)NC1CCN(CCCNC(c2ncccc2Cl)=O)C1)OC C1(C(=O)NCCCCN(C)C(C2(C)CC2(Cl)Cl)=O)CCCCN1N=O N1(C(C=Cc2ccc(OC)cc2C)=O)CCN(C(C2CC(O)C2)=O)C(C)CC1C C=CCC(C)C(=O)N(C1CCN(C(c2nscc2C)=O)CC1)CCOC N#Cc1cc(F)ccc1C(N1CCC2(C1)CN(C(c1ncccc1Cl)=O)C2)=O n1(CC)nnc(C)c1CNC(=O)CN(CCOC)C(c1cnco1)=O C1(CCNC(c2ccc(CC)[nH]2)=O)CC2CCC(C1)N2C(=O)CNS(=O)(=O)CC C1(C)(CC)CCC(C(=O)NCC2(COC)CN(C(=O)C(c3cnn(C)c3)=O)C2)O1 C1(CNC(CSCCC#N)=O)CC2CCC(C1)N2C(C1CCC=CCC1)=O c1(CCN(c2cc(-c3cccs3)sn2)C)ccc(Cl)cc1 C12(CNC(C3(CC(C)C)CCC3)=O)CC(CN1C(=O)CCC1CCN(C)CC1)C2 c1(C(=O)NCC2(OC)CN(C(C3CCOC(=O)N3)=O)C2)scc(C)c1C c1(OC)ccc(CC(N2CCC2C(=O)NC2CCS(=O)(=O)C2)=O)cc1 c1(C(C)CC(=O)N2CCC(NC(=O)C(C)(C)N3CCCCC3)C2)ccccc1F Cc1c(C(=O)NCC2CCN2C(=O)CCn2cccn2)nn2ccccc12 c1(CNC(N2CC(C)(C(=O)OC)OCC2)=O)ccc(F)c(F)c1F c1(N2CC3(CCC(CO)CC3)C2)nccn2nc3c(c12)CCCC3 N#Cc1cc(C(N2CC3CC(NC(c4cc(Cl)cs4)=O)C2C3)=O)c(N)nc1O C=CC1CN(C(C2CC(O)C2)=O)CC1NC(c1cccc(OCC=C(C)C)c1)=O c1(C(=O)NCC(CCNC(CNS(NC)(=O)=O)=O)O)c(F)ccc(F)c1F c1(C(N(CC(O)CNC(C2CCCO2)=O)C)=O)ccnn2ccnc12 N1(C(C(C)OCC)=O)CCOC(C(C)(C)CNC(=O)CN(C)C(N)=O)C1 c1(CC)cccc(C(N2CCC(C)C2C(=O)NC(c2ccc(O)nc2)C)=O)c1 N1(C(C(C)N(C(C2CC(C(C)(C)O)C2)=O)CC)=O)CCC(F)(CO)C1 C1(NC(c2ccc(CC)c(C)c2)=O)CC2CCC1CN2C(C1CC1C1CC1)=O C1(CNC(Cc2c(C)ccs2)=O)CCN(C(C2CCC(C(F)(F)F)O2)=O)C12CC2 Nc1ccc(C(=O)NCC2COCC2NC(=O)Cc2cccc(Cl)c2)nc1N C1(C(=O)NCC2CCN(C(C(C)=C(C)C)=O)C2(C)C)CCC(N=[N+]=[N-])CC1 N1(c2ccc(OC(C)C)c(C)c2)CCC(F)(F)C(C(=O)NC(CO)CO)C1 c1(C(=O)NCCCCCCNC(c2n(C=C)ncc2)=O)ccc2[nH]ccc2c1F C12(CCNC(c3c(C)nn(C)c3)=O)CCC1CN(C(c1ccc(CO)cc1)=O)C2 Cc1cc2nc[nH]c(=NCC3(O)CN(C(c4ccc(F)c(C(N)=O)c4)=O)C3)c2[nH]1 CCC(CCCC(=O)N1CCOC(C)C1)OC(=O)CN1CCC(OC)C1 C1(C(=O)NC2C(NC(CCCCC)=O)CC(F)(F)C2)CCCCCC(=O)N1 N1(C(c2c(COC)cc[nH]2)=O)CCCN(CCNC(C2CCN(OC)CC2)=O)CC1 C1(C)(NC(C(CN(C(c2cc(C)sc2)=O)C)C)=O)CC2(CCC2)C1 CCCCC(O)C(=O)NCc1nc(C(=O)NOC2CCCCC2)c(C)o1 N1(C(C(CNC(C(C)=CCC)=O)C)=O)CCCN(CCC)CC1 CC1CN(C(=O)CSCc2csc(=N)[nH]2)CC1NC(=O)CN1CCCCCC1 C(c1ccoc1)=CC(=O)NCC(O)C(=O)NCC=CCl CC(CC(=O)N1CCC1CNC(c1scnc1C(F)F)=O)N(C)C n1(NC(C(n2cc(-c3c(OC)ccc(C)c3)nn2)C)=O)cnc2c(N)ncnc12 c1(C2(C(=O)NC(CC)CNC(c3cnc[nH]3)=O)CC2)ccccc1C CC(C)CCCC(=O)NCc1cn(C2CCN(C(C3COC(=O)N3)=O)CC2)nn1 N1(C(C2(CC)CCOCC2)=O)CC2CN(C(c3c(Br)cnn3C)=O)CC12 c1(C(=O)NCCCCCNC(C(C)C(F)(F)F)=O)ccc2c(n1)CCOC2 C1(C)(C(=O)NCC=CCC(=O)NC(c2n(CC)ccn2)C)CCCCO1 C1(C(=O)NCC(CCNC(C2(SCC)CC2)=O)O)CCS(=O)(=O)C1 CCCCC(CC)C(=O)NCC1(O)CCN(C(C2(N(C)C)CCCCC2)=O)CC1 c1(C(=O)NCC(CC=C)(C)C)n[nH]c2c1CN(C(C1CCCC1C1CC1)=O)C2 C#Cc1cnc(C(=O)NC2C=CCN(C(=O)Cc3ncoc3C)C2)c(C)c1 c1(C(=O)NCCOC2CCN(C(CCC(C)N(C)C)=O)C2)cc(C#N)ccc1F C12CCCN(CC1)C(=O)C(C)C1(CC1)NC(=O)NC2.CN(S(N)(=O)=O)C(C)(C)C n1(CC)nc(C(=O)NN(C)CCOC2CCCCC2)cc1O.c12cc(on1)C2 N#Cc1cccc(CNc2csc(-c3ncccc3Cl)n2)n1 Cc1ncc(C(=O)NC(c2ccc(F)cc2F)CNC(=O)C(C)(F)F)c(=N)[nH]1 N1(C(CN(CCCCCC)C)=O)CC2(C1)CN(C(=O)C1=COCCO1)CC2CO c1(CC(=O)OC)ccc(CN2CCC(C(N3CC(O)C(F)C3)=O)CC2)cc1 c1(NCc2nc(C)sc2)cc(Cl)ccc1C1CCCCC1 C1(CNC(C2C(C(=O)OC)C=C2)=O)CCN(C(C2OCCC2C)=O)CC1 C1(NC(c2c(C)nsc2C)=O)CCN(C(=O)Cc2cn[nH]c2)C1(C)C c1(C(=O)NCC(CCCC)NC(=O)CS(N)(=O)=O)cc2c(cc1N)OCO2 c1(CN2CCN(S(CC3CCC(C)(CC)O3)(=O)=O)CC2)cnc(O)c([N+](=O)[O-])c1 CCC(C)(COC)C(=O)NC(CNC(=O)C(C)Sc1ccc(N)cc1)C(C)(C)C c1(C(N2CCC(N(c3nn4cc(C)nc4s3)C)C2)=O)ccc2c(c1)NC(=O)CO2 CN1CCN(C(=O)CC2C3CCCC3N2C(=O)CCC2CCOC2)CC1CO c12cc(C)c(Cl)cc1OC2=O.C1(OC)CCC(C(F)(F)F)CC1 N1(C(C(C)N(C2CC2)C)=O)CC(C(F)(F)F)C(CNC(C2CNC(=O)O2)=O)C1 C12(NC(CC=CC=C)=O)CCOCC1CN(C(c1ccnc(C(F)(F)F)c1)=O)C2 c1(C(N2C(CNC(=O)COCCCF)CCC2)=O)ccc(C(F)(F)F)c(Cl)c1 N1CCC(O)C(F)(F)C1.Cc1cc(OCC#N)ccc1-c1cccnc1C=O C1(N(C(C(c2ccc(C)cc2)F)=O)C)CCN(C(=O)CC2CCC2)CC1C N1(C(CNC(C)=O)=O)CCCC2(CNC(c3cc(C(C)=O)c(C)o3)=O)CCCC12 c1(C(=O)NCC2N(C(c3c(C)nn[nH]3)=O)CC2)cc2cc(Br)cc(F)c2o1 N1(C(CC(=O)OCC)=O)CC(NC(c2oc(CO)nc2C)=O)CCCC1C Cc1nc2cc(C(N3CC=CC(NC(c4cnc(S)nc4)=O)C3)=O)ccc2n1C Cc1c(C(N2CCC(C(C)NC(=O)COC3CCCCC3)CC2)=O)ncn1C C1(CNC(c2n(CC)ncn2)=O)CCN(C(C2CCCO2)=O)CCC1(F)F c1(C(=O)NCC(CC=C)NC(C2CC(C)C2)=O)c[nH]c2c(F)c(Cl)ccc2c1=O N1(C(c2nccc(OC)c2)=O)CCN(C(C2CCCC23CC3)=O)CCC1C N1(C(N2CCN(c3ccccc3OCC(F)(F)F)CC2)=O)CC2CC1CC2O c1(C(N(C2CCN(C(=O)CCc3cscn3)CC2)CC#C)=O)cccc(C)c1C N1(C(C(CCC)CNC(=O)CC2CC(F)C2)=O)CCC2(CNC(=O)O2)C1 c1(OC)cc(OC)c(C(=O)NC2CCC(N(C)C(C3CC(O)C3)=O)CC2)c(F)c1 C1(CC(=O)NCCN2CCOCC2)CCCCC1NC(c1ccc(C(F)F)o1)=O CN1CCC(C(=O)NC2CN(C(c3nccs3)=O)CC(C)(C)C2)c2ccccc21 N1(C(c2ncc(OC)cn2)C(=O)NCCCOC)CCOCC12CC2 CC1CC(NC(c2ccc(O)nn2)=O)CN(C(=O)C=C2CN3CCC2CC3)C1 CC(C)CCCC(=O)N1CCC(O)(CNC(=O)Cn2ncccc2=O)C1 c1(C(=O)Nc2cc(OCCOC)ncc2)ccc(Cl)cc1F C(=O)(C1=C(F)CN(C(C2(C)C=CCC2)=O)CC1)NC1CN(C)C(CO)C1 C1(NC(N)=O)CN(C(=O)C(C2CCCO2)NC(=O)C(=O)NCC2CC2)C1 Cc1cnc(C(N2CCC(=CCNC(C3CC(N(C)C)C3)=O)CC2)=O)c(C)c1 C=CCCC(=O)N.C1(=O)C(C)N(C)CN(C)CCN1CC CC(C)(F)C(C)(F)C(=O)NC1CCN(c2cc(Cl)ncn2)C1 C(=O)(C1=C2CCCN=C2NN1)N1C(NC(C(C)(C)OC)=O)CC(OCC)C1 n1(CC)nc(C(=O)NCC2CCCCC2NC(=O)CCC(F)F)c(Br)n1 C1(NC(c2cc[nH]c2)=O)CN(C(c2ccccc2N2CCCCC2)=O)CCC1O C1(C)(CNC(Cc2c(C)occ2)=O)CN(C(=O)C(C)OCC2CCCO2)CCO1 c1(C(NS(NCCN(C(C)=O)C)(=O)=O)=O)ccc2c(c1)cc(C)n2C C1(NC(CC(C)(C)O)=O)CCN(C(C2CC3CCC2CC3)=O)C12CCC2 C1(C2CN(C(=O)CC3OCCO3)C2)(NC(=O)C(C2(O)CCCC2)F)CC1 C1(CCNC(Cc2cnn(C)n2)=O)CCCCN1C(=O)Cn1nnc(C2CC2)n1 CC1CN(CCNC(N2CCCC2Cn2cccn2)=O)Cc2ccccc2O1 C1(CN(C(C2N(C(C)C)CCC2)=O)C)CN(C(=O)C(C)CC2CCCC2)CCO1 N1(C(C(=O)N(CC(C)C)C(c2ccoc2)=O)C)CCC(CC(=O)NC2CC2)C1 C(=O)(CS(=O)c1cc(Br)ccc1C)NC1(c2ccc(OC)c([N+](=O)[O-])c2)CC1 CC(O)(CNC(=O)C=C1CCCCC1)CNC(c1csc(Br)n1)=O C#Cc1cnn(C)c1C(=O)NCC=CCNC(c1sccc1SC(F)F)=O C1(C(C)=O)CC=CCC1C(N1C(C(=O)NCC(N2CCCC2)C)CC2CC12)=O C(=O)(C(CC(C)CC)NC(=O)C1=C(C)OCCS1)NC(C(=O)NCCC)CC N1(C(C(F)=CCC)=O)C2CCC1CC(N(C(=O)C(F)C(F)(F)F)CC)C2 c1(NCCSCc2c(C(=O)OC)csc2)ccc(Cl)cn1 C(C(C)(C)CC(=O)N1CCCCC1C(C)(C)NC(C1CCCC(=O)N1)=O)OC N#CCCCC(=O)NCc1ccnc(C(=O)N(CCO)Cc2cccs2)c1 N1(C(=O)OC)CCc2cc(C(=O)NC(C)(C)C(C)NC(c3cocn3)=O)ccc21 C(=O)(CC(O)CCCC)NCCOCCN(C(C1CCCCC1)C#C)CC N1(C(COC(CC)C)=O)Cc2occ(C(=O)NC3CCN(C(C)C)CC3)c2C1 N1(C(c2n(OC)cnc2C)=O)CCC2(C1)CN(C(C1CC(C)CC(C)C1)=O)C2 CCCC(C)CCN=c1nc2scnc2c(N(CC(C)C#N)C)[nH]1 c1(OC)cc(O)c(COC(=O)C(F)(F)c2csc(Cl)n2)cc1Cl c1(CCC(=O)N2CCC2CO)nc(-c2ccncc2)cs1.N12CCCC1CC2=O N1(C(C=CCOC)=O)CC(C)CCC1CNC(c1cn(-c2ccccc2)nn1)=O C1(C)(CNC(C2(C)CSC2)=O)CN(C(C2(C(C)(C)O)CCC2)=O)CCO1 c1(C(=O)OCC)cc(Cl)cc(Cl)c1S(=O)(=O)N1CCCCC1c1ccc(F)nc1 CCC(C(=O)OC)C(=O)NCC=CC(N1CCSC(C)CC1)=O C1(NC(c2cc(OC)nn2C)=O)CC2CC(C1)N(C(=O)CC(O)CC(C)C)C2 C1(C(=O)NCCC(C)(C)NC(Cc2ccc(C)o2)=O)CCC2(CCC2)OC1 CCCCC(CNC(=O)CCc1cccc(O)n1)NC(C)=O c1(C(N2CCC(c3ccccc3)(NC(CC=C)=O)C2)=O)cc(C)c(Cl)cc1OC C1(C#N)(C(N2CCCCC(NC(CC3CCC(C)CC3)=O)C2)=O)CC12CCCC2 O=C(CCCCn1ccnn1)NCC(O)CCNC(C1CCSCC1)=O C1(C2CN(C(=O)CC3CCC(F)(F)C3)C2)(NC(CC2C(=O)NC(=N)S2)=O)CC1 N1(C(C2(F)CN(Cc3ccc(OC)nc3)C2)=O)CCN(C)C(C)(C)C1 C1(C(=O)NC2CCC(N(C(=O)CC3CSCCO3)C)C2)CCCCC1O C1(N(C(=O)CN2CC(=O)NC2=O)C)CC2CCC(C1)N2C(C1CC(=O)C1(C)C)=O O=C(CCC1=CCCCC1)NC1(Cc2cc(F)ccc2F)CCC1 c1(C(N2C(CNC(CCN(c3ccncc3)C)=O)CC2)=O)cccc(=O)n1C c1(C(=O)NCCCC2N(C(CCOC)=O)CCCC2)cccc2[nH]nc(O)c12 C=C(C)C(C)(C)C(=O)N1CCCC(CCCCNC(=O)CCC2CCCO2)C1 C1(CC(=O)NCc2cc(C(=O)NCCCCC3CC3C)cs2)(CC=C)CCCC1 C12(C(=O)NCCNC(C)=O)CCCC1CCN2C(C1CC(C(C)C)=NO1)=O CN=c1[nH]c(=NCc2ccnc(C#N)c2)[nH]c(=NCC(C)(C)CO)[nH]1 C(=O)(C1CCCc2nncn21)N1C(CNC(c2cnc(C)nc2C)=O)COCC1 C(=O)(CCCCCCC(=O)Nc1cn(C)c(C(=O)Nc2cccc(O)n2)n1)OC Cc1ccc(C(N2CC3CC(NC(C4CCC4)=O)C2C3)=O)cc1S(C)(=O)=O CCCCCCCCN=c1[nH]c(C)cc(=NC2CCN(C3CCN(C)C3)CC2)[nH]1 CC1CN(C(c2cc(C3CCC3)nn2C)=O)CCN1C(c1ns[nH]c1=O)=O C(=O)(C(C)C(C)(C)C)N(C(CN1CCCC(C(=O)OC)C1)=O)CC(C)C N1(C(CCOC(C)=O)=O)CCC(C(=O)NC23CCN(CC2)CC3)C(C)C1 c1(CN(C2CCN(C(=O)CCF)CC2)Cc2ccccc2)cc(F)c(F)cc1Cl C1(O)(C(=O)OCC)CCN(C(CCC=C(C)C)C(=O)NC2CCC2)CC1 N1(C(C(N2CCC(C)C2)=O)=O)CC2CCN(C(C3C=CC=CC=C3)=O)C2C1 N1(C(c2c(NC)ccc(F)c2)=O)CC(C)N(C(c2coc(C(N)=O)c2)=O)CC1C c1(CC)cn2c(C(N3CCN(C(c4ccnn4C)=O)CC3CF)=O)cccc2n1 C1(CNC(C)=O)CN(C(c2cc(Br)cc(N)c2C)=O)CCC12CCOC2 C#CCCC(C(=O)NCc1cc(C)ccc1F)NC(c1ccc(O)cc1F)=O C1(C(N2CCC(NC(C3CCC(CC)O3)=O)C2)=O)CCOCC1(C)C c1(CCC(=O)O)ccc(S(=O)(=O)N2CCC(CNC(c3n[nH]cc3I)=O)C2)cc1 c1(C(=O)NC2C3CN(Cc4ncc(C)o4)CC32)cccc2c1C1CCC2CC1 O=S(=O)(c1ccc(Br)cc1NCC1CCCC1O)NCc1cc(Br)ccc1F c1(OC)ccc(C(N2CC(NC(C3CC3CF)=O)C(C)(C)C2)=O)c(F)c1Cl Cc1ccc(F)c(C(=O)NCC2(C)CCN(C(C3(S(C)(=O)=O)CCC3)=O)C2)c1F N1(C(c2cncc(C)n2)=O)C2CCC1CN(CC(C)O)C2 C=CCC(C(=O)NCC1COCCN1C(c1ccc(C(C)=O)cc1)=O)C(C)C c1(C2(C)CC2)cccc(C(=O)NC2CC2CNC(=O)CC(O)CC2CC2)c1 C(C(=O)Nn1cccn1)NC(c1ncc(CC)cn1)=O Cc1cc(=O)n(CCC(N2CCC(NC(=O)C(F)=C3CCC3)C(CO)C2)=O)cn1 CC1(C)NC(=O)N(CCC(=O)NC2CCOCC2NC(=O)CC#N)C1=O N(C(=NCC(C)(C)c1c(C)nn(C)c1C)N1CCC2(CCCN(C)C2)C1)C(C)C c1(C(=O)NCC2C(NC(c3ccc(CC)c(F)c3)=O)C2)ccc(N)cc1[N+](=O)[O-] c1(C(N(CCCCCNC(C2(C)CC2(Cl)Cl)=O)C)=O)ccc(F)cc1 S(=O)(=O)(c1ccc(Cl)nc1C)N1CCN(c2ccc(C)nc2C)CC1 C(=O)(C1=CC2CCCC12)NC1CN(C(CCOc2cccc(C)c2)=O)CC(C)C1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(C(CC)n2cncn2)=O)C(C)C1 C1(NC(=O)C=Cc2cc[nH]n2)CC2C(O)C(O)CC12.C12CC(C1)NC(=O)CO2 C(C(C)(O)CC(=O)NCC=CCNC(CC=NC(=O)OC1CC1)=O)OC C1(NC(c2sccc2F)=O)COC2(CCN(C(=O)OCCCCl)C2)C1 c1(C(=O)NC2C(CNC(C3N(C(C)=O)CSC3)=O)COC2)cc(C)nn1C C(CC(C)(C)CC(=O)N1CCC(C)(CC(=O)Nc2cc(C)cc(C)c2)C1)OC Cc1sc(O)nc1C(=O)NC1(C)CN(C(=O)C(C)n2cncn2)C1 N1(C(C(CC)CC)=O)CCC2(CC1)COC(CNC(=O)CCS(C)=O)C2 c1(CCC(C)C)ccccc1C(=O)NCC1CC(F)(CNC(=O)CNC=O)C1 C(=O)(n1cc(CN2CCC(NC(c3cc(Br)ccc3I)=O)C2)cn1)OC(C)(C)C c1(CCC)ccc(C(=O)NC2CCCC2CN(C(=O)C(c2ccccc2)C)C)[nH]1 N1(CC)CCC(CNC(c2cc(CNC(C3CC3Cl)=O)no2)=O)C1 c1(C(=O)NCCCC(=O)NC(C2CCCCO2)CC)ccc(CO)cc1 N1(C(C(CCC)C)=O)CCCC2CN(C(c3csc4c3CCC(C)C4)=O)CC12 CN1CC(C(=O)Nc2cccc(OCCO)c2[N+](=O)[O-])c2ccccc21 C(CCCC(=O)N(C)CC1CCSC1)NC(C1C(CCOC)C1)=O c1(CC(N2CCC(O)(CNC(CN(C)C(N)=O)=O)C2)=O)cc(Cl)c2c(c1)OCO2 CCCC(C(=O)OC)C(=O)N1C(CNC(c2cnc(S)n2C)=O)CC2CCCC12 CCCCCCCC(=O)NCC12CC1CN(C(C1CC3CC3C1)=O)C2 c1(C(N2CC(C=C)C(NC(=O)Cc3cn(C)nn3)C2)=O)cccc2ccncc12 c1(C(=O)OCC)cn(C(C)C)[nH]c1=NC(=O)N1CCn2c(C3CC3)nnc2C1 N1(C(c2c(C)nns2)=O)CC2(CC(C(=O)NCc3ncccn3)CO2)C1 C1(O)(CN(C(CCOCCOC)=O)C)CCN(C(=O)CC2CCC(O)C2)CC1 CC(c1ccco1)=CC(=O)OC(C)(C)C.N12CCN(CC1)C(=O)OCCC2 N1(CCN(C)C)CCCN1C(OC(F)F)=O C1(F)(C(=O)NC(CN(C(c2ccc(C)c(Cl)c2)=O)C)C)CC12CCCCC2 c1(CC2CCC(C)(C)C2)nc(C(C2CC2)SC)n(-c2ccnc(C(F)(F)F)c2)n1 N1(C(C2(OC)CCCC2)=O)CCOC2(C1)CN(C(C1CCCC3CCCN13)=O)C2 C(c1cccc(Cl)c1)=C(C)C(=O)N(CC(C)(C)NC(C1CCCS1)=O)C CCCCC(CCCC)C(=O)NCC(C(C)(C)C)NC(c1cncc(CO)c1)=O c1(SC)ccc(C(=O)NC(CC)C(=O)NC(C2CSC2)C)o1 c1(NCCC=C=C)[nH]c(=NCc2cc(C)c(F)c(C)c2)nc2ncn(CC)c12 c1(C(N2C(CC#C)CCCC2)C(=O)NCCOC)ccc2ccc(Br)c(F)c2n1 C1(C(=O)NCCC2(NC(C=CCC)=O)CCC2)CCc2nnc(C)n2C1 N1(C(c2c(CC)onc2)=O)CCC(NC(=O)C=CC2CCCCC2)CC1 c1(C(N(CCNC(c2c(C)ccn2C)=O)CC)=O)cc2ccc(Cl)cn2c1 CCCCCC(F)C(=O)NC(C)C(=O)NC1CC1.c12nc(C)c(o1)C(=O)NC2 N1(C(Cc2cccc(OC)c2)=O)CCN(C(c2ccc(CF)cc2)=O)C(C)C1C c1(NC(c2c(C)c[nH]c2)=O)ccccc1N1CCN(C)CC1 c1(C(=O)NC(C(=O)N(C)Cc2cncs2)C2CCC2)ccn2ccccc12 c1(CNC(c2ccccn2)C)cnn(C2CC2)n1 c1(NC(C2(COC)C=CCN2C(C2CC(OC)C2)=O)=O)ccc(OC)cc1O c1(CCC)nc(C(=O)N(C)CCNC(=O)C(COCc2ccccc2)OC)cs1 C(=O)(CCS(C)(=O)=O)NCCN(C(C(C)C)=O)C1CC1 C(=O)(CCCC(F)(F)F)N1CCCC(N(C(C(C)SC(F)(F)F)=O)C)C1 N1(C(CCN(C(C(C)S(CC)=CC)=O)C2CC2)=O)CCC(CO)C12CCC2 C(C(=O)N1CC(=O)NC(C)C1)(C(C)(C)O)NC(C1C(OC(C)=O)C1)=O C(CCCCCC(=O)N1CCCC1(C)C1CCC1)NC(c1cnc(C)s1)=O c1(-c2c(CC)ccs2)ccc2occ(CC(=O)Nc3nc(C)c(Cl)cc3Cl)c2c1 Cc1cc(C(=O)NC2(CNCc3ccc(Br)c(F)c3)COC2)cc(C)c1Cl CC1N(C(=O)CCc2ncc(-c3ccc(F)cc3)o2)CCC1(F)F N1(C(C2C(CC)N(C(c3cc[n+]([O-])cc3)=O)CCC2)=O)CCC2CCCCC2C1 C(CC(C(=O)Nc1cccc(F)c1)NC(c1snnc1C)=O)OC C1(Cc2nnc(N3CCC(OCCCC)CC3)n2CCC#N)CCCCNC1=O c1(C(=O)NCC2(O)CC(C(N(CC(CC)O)C)=O)C2)cccc(C)n1 C(=O)(C(C)(C)C1=CCN(C(=O)C2=CC3C=CC2C3)C1)NC1C(C)CC1 n1(CC)cnc2c(NCC(=C)F)[nH]c(=NCC(C(C)(C)C)SC)nc12 c1(OC(C)C(N2CCN(C(c3ccc(Cl)s3)=O)CC2)=O)cccc(Br)c1 C1(C(=O)NCc2c[nH]ccc2=O)CC2(CC2)CN1C(C1CC2C(C1)C2(F)F)=O C1(NC(CC(CNC(CC(COC)(C)O)=O)(C)C)=O)CCCCN(C)C1=O c1(OC)cc(Br)cnc1C(C(=O)NC1CCC1)N(C)CC1CC2CCC1C2 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCC2CN(C(c3cncc(Cl)c3Cl)=O)CC2C1 c1(C(=O)OCC(C(=O)OCC)C)cccc(S(=O)(=O)CF)c1 c1(C(=O)NC(C)CNC(=O)CCc2nc[nH]n2)cccn(O)c1=O C1(NC(Cc2c(C)ocn2)=O)CCN(C(=O)CSc2ccc(O)cc2)CC1F C=Cn1nccc1C(=O)NCC12CC(NC(C3CCC=CCC3)=O)(C1)C2 C1(N(C(CCOC(C)=O)=O)C)CCCN(C(=O)C(O)Cn2cncn2)C1 Cc1nn(C)c(C)c1CC(=O)NCC1(CN(C(=O)Cn2ccccc2=O)C)CC1 Cc1ccc(CNC(c2cn(CCNC(C3CCC4CC34)=O)nn2)=O)cc1O C1(NC(C2=CN=C(N(C)C)CC2)=O)COC2CN(C(=O)CC3(C)OCCO3)CC12 CCC(C)C(O)C(=O)NC1C2CC1N(C(c1cccc(F)c1C(F)(F)F)=O)C2 C1(NC(c2ccccn2)=O)CC2CCC1N2C(c1ccnnc1O)=O c1(CC)ccnc(C(C(=O)NCCN2CCCCC2)N(C2CCCC2C#N)C)c1 C1(NC(C(C)c2cc[nH]n2)=O)CCC2(CC1)CN(C(c1ccc(Cl)nc1N)=O)C2 c1(C(=O)NCCC(C)NC(=O)CN(C2CCCCC2O)C)cc(Cl)ncc1Cl c1(C(=O)NC2CN(C(CS(CC)=O)=O)C(C)(C)C2)cnc(O)n(C)c1=O N1(C(C)=O)CS(=O)(=O)CC1C(N1CCN(C(c2cc(O)ncn2)=O)CC1)=O c1(C(N2CC(C(=O)OC)OC(CC)C2)C(=O)NCC=C)ccc(OC)c(C)n1 c1(C(=O)NCC(C)(O)CNC(c2cn[nH]c2)=O)cc2cccnc2[nH]1 N1(C(CCC=C=C)=O)CCC2(CC1)CC(NC(c1cn(C)nc1C(C)(F)F)=O)C2 C1(NC(C2CN(C(CCC3C(C)(C)C3)=O)CC2F)=O)CC1C1CCCCC1 N1(c2cc(C)ncn2)CC2(C1)C(NC(=O)CC1CC3CC3C1)CCS2(=O)=O C(=O)(CCC(C(C)C)NC(=O)CC1COCC(C)O1)NCCN1CC=C(C)CC1 n1(C(c2cccnc2)C)nc(-c2ccn(C)n2)nc1CCC1CCC1 C1(CN(C)C(C2C3COCC23)=O)CC(O)CN1C(=O)CN1CCC(F)CC1 C1(C(=O)NC(C)CCCCO)CN(C(=O)C=CC(=O)N(C)C)CC(C)(C)C1 c1(C(=O)NC(CNC(C(C)c2ccsn2)=O)C)c[nH]c2cccnc2c1=O c1(CC)cc(C(=O)NCC2CCC(C(=O)NCC(C3CC3)N(C)C)O2)n[nH]1 C1(NC(c2cc3[nH]cc(Br)c3nn2)C)Nc2ccccc2C1(C)C c1(C(=O)NCC=CCNC(C2COC(=O)O2)=O)cc(Cl)c2n[nH]cc2c1 C(=O)(CCC(=O)N1CC(CNC(=O)C(C)NC(=O)NC)CC1C)NC N1(C(Cn2c(C)cc(C)n2)=O)CC(O)CCC1C(=O)NCC(=C1CCCCC1)F c1(OC)ncc(NC(c2csc(-c3csc(C)c3C)n2)=O)cn1 CC#CCCCC(=O)N(C)CCNC(c1cc(Br)c(Cl)cn1)=O C1(C(=O)NC(C)CCNC(=O)CC2CNC(=O)C2)Cc2cscc2C1 c1(C(N2CCCC(NC(c3cc(C)c(Cl)s3)=O)C2)=O)ccc(F)c(Cl)c1F Cc1cc(C(N2CCC(NC(c3cn(C)ccc3=O)=O)C(O)C2)=O)c(C)c(C)c1 C(=O)(CCC(C)(C)OC)NC1CC(C(=O)NCCOCC(=C)C)C1(C)C c1(C(N2CCC(CNC(C3N(C)CCOC3)=O)CC2)=O)ncc([N+](=O)[O-])n1C C1(CC=C)(NC(C2CC(=O)N2)=O)CCN(C(C2CCCCC2OC(F)(F)F)=O)C1 c1(N2CCCCC(CNC(=O)C(F)CC3CCCCC3)C2)ncnc2sccc12 c1(C(C)NC(C2C3CN(C(C(CC)O)=O)C2C3)=O)ccc(S(C)(=O)=O)cc1 c1(C(=O)NCCCCCNC(C2C(C3C(C)C3)C2)=O)cnn2ccc(Cl)c(F)c12 c1(NCC(=O)N(c2ccc(Br)cc2)C)ccc(N)c(OC(F)(F)F)c1 c1(C(N2C(CC)CN(C(c3cn(CC)nn3)=O)CC2)=O)ccc2sncc2c1 N1(C(CCC(C)OC)=O)CC(C(N2CCC(N3CCCC3)C2)=O)CC(C)(C)C1 c1(CCN(CC(=O)NC(C)C(C)(F)F)C)ccccc1OCc1ccccc1 c1(C(=O)NC(C)(CC2CCCC2)CO)cncc(C(F)(F)F)n1 C1(C(=O)NC(CNC(CC=C=C)=O)(C)C)CCCC2(C1)NC(=O)NC2=O n1(CCC(=O)NC2(C)CN(C(CCC(C)OC)=O)C2)c(=O)oc2ccccc12 N1(C(CC2(C)CC2(Cl)Cl)=O)CCC2CCC(NC(C3CCCC3O)=O)C1C2 CCCS(=O)(=O)C(C)C(=O)NCc1ccc(CNC(C2CC(O)C2)=O)cc1 c1(C(=O)NC2(CF)CCN(C(c3c(NC)cccc3)=O)C2)cccc2oncc12 C1(NC(C(C)O)=O)CN(C(=O)CCc2cnoc2)CC12CCOCC2 Cc1cc(C(=O)NC(C)CCCCNC(c2ccns2)=O)c(Cl)cc1F C1(N(C(C(C=C)O)=O)C)CCCC(NC(c2ccnc(OC3CC3)c2)=O)C1 c1(CN2CC3C(C(=O)NCC4CCN(C)CC4)C3C2)cc(Cl)ccc1Br N(C(=NCC(F)F)N1CCC(C)(OC)C1)Cc1nc(CC)sc1 CN1C(=O)CC(C(=O)NCC(C)(CO)NC(c2ccc3c(c2)NCC3)=O)NC1=O N#Cc1cc(C(=O)NCC(C2CCOC2)NC(=O)CNC(c2ccco2)=O)co1 c1(CC)ccc(C(N2CC3C(NC(=O)CNc4ccccc4Cl)C3C2)=O)c(C)n1 c1(C(CN2CCC(NC(=O)OC(C)(C)C)CC2)=O)cc(Br)nc(Br)c1 c1(CNC(CC2(C)CC2(Cl)Cl)=O)cc(O)nc(CNC(c2ccc(F)cc2)=O)n1 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCOCC(NC(c2cnn(C3CC3)n2)=O)C1 C1(NC(C(C2CCCC2)OCCC=C)=O)CCN(C(C)COC)C1 N1(C(CCNC(c2cccc(NC)c2)=O)=O)CCC(N=[N+]=[N-])C1 C1(C(=O)NC(CCN(C(=O)CCc2cccc(O)n2)C)(C)C)CC2C=CC1CC2 Cc1scc(C(=O)NCC(C)(C)CNC(=O)CC23COCC(C2)C3)c1C CC1(C)CCCCC1C(=O)NCC(O)C(N1CCC(F)C(F)C1)=O CC(CNC(c1ccc(Cl)nc1O)=O)CN=c1cc(Cl)nc(C2CCC2)[nH]1 N1(C(Cn2ncn(C)c2=O)=O)CCN(C(c2sccc2SC(F)F)=O)CC1CO CCCC(F)C(=O)NCCC(O)CNC(c1ccc(C(C)C)s1)=O CC1(C)CCOC(C(N2CCCC(NC(c3cc(CC4CC4)on3)=O)CC2)=O)C1 C1(CC(=O)NCc2onc(C)n2)CCCN(C(C2CCC(C(N)=O)O2)=O)CC1 c1(C(N2C3C(CNC(C(C)OC)=O)C(C3)C2)=O)c(F)cccc1Br Cc1nc(N2CCOCC(C(=O)NCCc3ccncn3)C2)c2ccccc2n1 c1(NC(C(c2nc(Cc3ccccc3Cl)no2)C)=O)ccnc(CO)c1 Cc1ccnc(NC(=O)CCCCCc2ccc(F)cc2)c1Br c1(C(=O)NCC(C)CNC(C2CCC(O)C2)=O)cc([N+](=O)[O-])ccc1Cl c1(CC)nc(C)ncc1C(N1CCC(F)C(NC(=O)Cc2cnccc2Cl)C1)=O C1(C)(CNC(CCc2ncn(C)c2)=O)CCN(C(=O)CC(F)(F)F)C1 Cc1nc2ccccc2c(C(N2CC(CNC(c3cnsc3)=O)C(C)C2)=O)c1C C1(C)(C(c2nnnn2C2COC2)NC(CC)COC)CCCCCC1 c1(C(N2CCC(CNC(C=C(C)C3CC3)=O)C(C)C2)=O)cccn2nccc12 Cc1cc(F)c(Cl)cc1NC(C1CC2CC2N1C(c1ccc2c(c1)CCC2)=O)=O c1(C(N2CCC(CC(=O)NCc3scc(C)n3)C2)=O)cccc(I)c1Cl C1(NC(CS(=O)(=O)NC)=O)CN(C(C23CCC(CC2)CO3)=O)CCC1C(F)(F)F C1(NC(c2ccsc2)=O)C2CCC1N(C(c1ccc(-c3nnc(S)o3)cc1)=O)C2 N1(C(c2cn(CC)nc2C2CC2)=O)CCC2(CCC2)C(CNC(C2(F)CC2)=O)C1 c1(CC(N2CCC(NC(C3(CO)CCCO3)=O)CC2)=O)n[nH]c2cc(Cl)ccc12 N1(C(CC2(CNC(c3c(C)ccs3)=O)CC2)=O)CCC2CC1C(=O)N2C c1(C(C(=O)NC(C)CCNC(=O)COCCF)O)ccccc1OCC1CCC1 C1(C(=O)NC2CCN(C(C3CC(OC)C3)=O)CC2)CCCC(C)(C)C1 C(=O)(CCCCC)N(CC(C)NC(c1c(CC)ocn1)=O)C c1(C(=O)NCCN(C(=O)C#CC2CCOCC2)C(C)C)cncc(P(C)(C)=O)c1 CCC(O)C(C)(C)C(=O)N(CCC(C)NC(=O)C(=O)NCC(F)(F)F)C N1(C(c2n[nH]c(C)c2C)C(=O)NCC(C)C)CC(C)OC(C)(C(F)F)C1 C=CCC(C(=O)N1CC(O)(CNC(c2cc(C(C)(C)C)c[nH]2)=O)C1)C(C)(C)C S(=O)(=O)(CC(=O)NCC1CCC(CNC(c2ccoc2Cl)=O)CC1)NCC CC(CCC(=O)N(CCC(O)CO)C)NC(=O)CC1CCCC(=O)C1 c1(CNC(C2CC(C)(F)C2)=O)cc(C(=O)NC2CC=CCC2)ccn1 C1(NC(Cc2n(C)nnc2)=O)CC2(CCCCN2C(=O)CS(=O)(=O)C2CC2)C1 CC1CC(NC(c2coc(NS(N)(=O)=O)n2)=O)CCN1C(=O)COC(F)(F)F O=C(NNC(=O)c1ccc(CCCOCc2ccccc2)s1)C1CCS1 CC1Cc2cccnc2N(C(c2noc3cc(Br)ccc23)=O)C1 C1(C(NOC)=O)(C(=O)N(C(C)CO)C)CCN(CC(c2cccc(O)c2)O)CC1 CCCC(F)C(=O)NC(CO)C(=O)NC1C2CCCCC12 C(=O)(CCC(F)(F)F)N1CCC(C(C)Nc2nccc(OCCC)n2)C1 c1(N(C(C)CNC(C2CCCC23CCC3)=O)C)nc2ccc(Br)cc2s1 C1(CNC(CCCCOC)=O)CCN(C(=O)C(c2ncccc2C)(F)F)CC1O N1(C(C=CCN(C)C)=O)CCC(NC(C2(C3CCCO3)CCC2)=O)C(CO)C1 N1(C(C(C=C=C)C)=O)CCC(C2CN(C(C3CC(C)(CC)C3)=O)C2)CC1 c1(C(N2CC(CCCNC(C=CCC)=O)OCC2)=O)cc(O)cc(F)c1 c1(-c2c(C)nn(CC)c2C)ccc2nc(C(=O)NC(CO)CO)sc2c1 CC(C)(C(=O)NCC(C1CCCCC1)NC(=O)CN(C)C1CC1)C(N)=O N1(C(c2scc(NC(C)=O)c2)=O)CC(C)CN(C(c2csc(Cl)n2)=O)CC1C C1(CC(=O)NCC(CO)NC(=O)C(C)(C)c2ccccn2)(OC)CCCCC1 CC(CC(=O)NCC1CCCCN1C(C1CCC(C)(C)O1)=O)C(F)(F)F N1(C(c2ccc(C(C)=O)cc2)=O)CCCCC(NC(C2CCC=CCCC2)=O)C1 c1(C(=O)Nc2cccc(C(=O)O)c2)c(F)cc(O)cc1F C1(C2(O)CCN(C(C3CCCS3(=O)=O)=O)CC2)(NC(=O)COCC2CCC2)CC1 N1(CC(=O)NCCC(N2CCC(NC(=O)CCF)C2)=O)CCCC1CO N1(C(=O)CCc2cnc[nH]2)CC2CN(Cc3cc(O)ccc3F)C2C1 c1(CN2CC3CCN(C(c4ccc(C)cn4)=O)C3C2)c[nH]c2cc(F)c(F)cc12 c1(OCC)ccc(C(=O)ON2CC(c3[nH]nc4c3COC4)C2)cc1OCC c1(CNC(C(CC)(C)C(F)F)=O)n[nH]c2c1CN(C(C1CCC(=O)N1C)=O)CC2 CCC(CC(=O)NC(CNC(c1cc(C2CC2)ccn1)=O)C1CC1)C1CCC1 CCC(CCNC(=O)C(C)C(CC)CC)C(=O)N(C)OC C(=O)(CC(C)CC(C)C)NC1CCN(C(c2ncn(CC)n2)=O)CC1O N1(C(C(C)(O)c2ccncc2)=O)CCC(CO)(Cc2ccccc2)C1 N1(C(CCC=CC)=O)CC(=O)NCC1C(=O)N(CCO)CC1CC1 Cc1ncc(C(=O)NCC2(CCNC(=O)Cn3ccc(C(F)F)n3)CC2)c(=N)[nH]1 C1(NC(C(C=C)(C)C)=O)C2CC3C1C3C2C(=O)NOCCCCF C1(OCC(=O)NCC(C)NC(=O)CCc2cnc(C3CC3)o2)CCN(C=O)C1 CC1CC(NC(=O)C(C)(C)C(F)F)CN(C(C2CCNC(=O)C2)=O)C1 C1(NC(c2ncc(CC)cn2)=O)C2CCN(C(=O)CCCOC(C)(C)C)CC12 c1(C(=O)NC2C(SC)CN(C(=O)Cn3cnnc3O)C2)c(C(C)C)cccc1F C12(CNC(c3onc(C)n3)=O)CCCC1N(c1ccnc(C#N)n1)CCC2 c1(C(=O)NC2C(NC(Cn3c(C)cc(C)n3)=O)CC2)cncc2cc(Cl)ccc12 C(=O)(C(C)(C)C(F)(F)F)N1C2CC(CNC(C=CSC)=O)C1CC2 c1(C(=O)NCC2(OC)CCN(C(c3cc(C)[nH]n3)=O)C2)cc(C(=O)OC)ccc1C N1(C(CC(CC)C)=O)CCC2(CC1)CCN(C(C1CC1c1nc[nH]n1)=O)C2 N1(C(C2=C(C)CCCC2)=O)CCC2(C1)CN(C(=O)C(C)Cn1ccnc1)CCO2 C(CCS(=O)(=O)c1ccc(F)cc1)N1CCC(C)(CC)C1 C1(NC(CCCC#C)=O)CCN(C(=O)CC(C)NC(N)=O)C12CCCC2 CCC(C)C(O)C(=O)N(CCCCNC(C1CC1F)=O)C N=c1nc(CC(=O)NCC2(F)CC(NC(C3CC34CC4)=O)C2)[nH][nH]1 C1(OC)CCN(C(=O)CCc2ccc(C(F)F)cc2)C1(C)C.C(=O)O CC1C2C(CCN2C(C2CCS(=O)(=O)N2C)=O)CN1C(=O)CNC(c1ccon1)=O Cc1noc2cc(C(=O)NCCCCN(C(=O)C=Cc3nccs3)C)ccc12 c1(NC(C(=O)NCC(CC=C)NC(=O)C(C)(CC)CC)=O)ccc(N=[N+]=[N-])cc1 Cc1nc(C)c(C(N2CCN(C(c3cccnc3S)=O)C(C(F)F)C2)=O)nc1C C1(C)(CCC(=O)N(C2CCC(NC(=O)C(=O)NC3CC3)CC2)C)CCC(=O)N1 c1(C(=O)NCC(CN(C(CN(CC)CC)=O)C)C)cc2c(s1)CCOC2 C1(NC(C(N(C(C(COC)C)=O)C)C2CC2)=O)CCC2(CCC2)C1 c1(-c2c(C)n(C)nc2)ccc2nc(C(=O)NCCOCC3CC3)sc2c1 n1(CCN(C(C)C(=O)NCc2cccs2)C)cc(CO)nn1 C1(O)(CCNC(C(C)=CCC)=O)CCCN(C(=O)Cn2c(C)csc2=O)C1 CC1(C)CCN(C(C2CCC(F)CC2)=O)CC1CNC(=O)COC(F)F Cc1ccc(OCC2CC2)c2c1CCC2.C(C(=O)O)OCC O=C1CC2C(C(=O)NCC3CCCN3C(=O)CCC3CCCCCC3)C2C1 CC1(C)C2CN(C(C3(C#N)CC3)=O)C(C(=O)Nc3cc(F)c(Br)c(F)c3)C12 N1(C(Cc2c(C)noc2)=O)CCC(NC(=O)C(F)(F)CO)C(CO)C1 C(=O)(C1=Cc2cc(F)ccc2OC1)N1CCC(NC(c2nnn(C)n2)=O)C1(C)C CCC(C(=O)NCCCNC(C12CCCC1C2)=O)Oc1ccccc1 CC1CCN(C(C2OCCN(C)C2=O)=O)CC1NC(C1CC(F)(F)C1(C)C)=O Cc1onc(C(=O)NCC2CCCN2C(C2CS(=O)(=O)CC23CC3)=O)c1[N+](=O)[O-] c1(NC(C)=O)cccc(C(=O)NCC2CC(NC(C3(C4CC4)CCCC3)=O)C2)c1 c1(C(=O)NC2CCOc3ccccc3C2)cc2n(c(=O)c1)CCS2 Cc1ccc(C(N2CC(COC(C)(C)C)(NC(=O)C=CCO)C2)=O)cc1CO C(=O)(C1=CCCCCC1)N(C1CC2CCC(C1)N2C(=O)Cn1ccnn1)C c1(C(=O)NCCC(C(C)C)NC(=O)C2CC2)c(Br)cccc1Br c1(N2CCC(C(N=c3n(C)[nH]cn3)=O)(F)CC2)ncnc2c1ncn2C C1(CNC(CCN(CCC)C)=O)(CNC(=O)COCC(C)C)CCCCC1 Cc1cncc(C(=O)NCC(C)(CO)NC(=O)CSCCC(C)C)n1 C(=O)(C1OCCn2ccnc21)N1CC2C(NC(=O)CCc3ccc(Cl)cc3)C2C1 N1(C(CCCc2cc(C)no2)=O)CCN(C(=O)C=Cc2cocn2)C(CO)C1 CC1C(NC(=O)C(O)C2CC2)CC2CCC1N2C(c1cc2ccccc2o1)=O c1(C(=O)NCC2C(NC(c3c(C)nc(C4CC4)[nH]3)=O)C2)c[nH]c2cccc(Cl)c12 N1(C(CCCN(C(C)=O)C)=O)CC2CC1CN(C(=O)Cc1ccc(C)cc1Cl)C2 C1(NC(c2ccc(CC)[nH]2)=O)CC12CC(NC(=O)CC(C)(F)F)C2 C1(NC(C(C)SC(C)C)=O)CC(C)(NC(C)(C)C)C1.C12CCN1C(=O)C2.C(=O)(O)N C1(C(N2CC3C(CO)C3C2)=O)CC12CN(Cc1ccc(Br)[nH]1)C2 c1(C(N(C2CC(O)CN(C(=O)CC(C)(C)C#N)C2)C)=O)cc2ccccc2n1C CC1CN(C)C(C)CC1NC(c1cc(CNC(c2csc(Cl)n2)=O)ccn1)=O C12(C(N(C)CC3(C)CCCO3)=O)C(NC(c3nnc(O)nc3O)=O)C3CC1C2C3 C1(C2CCN(C)CC2)(NC2(C(N3CCC(C)(NC(CSC)=O)C3)=O)CCC2)CC1 c1(C(=O)NCCCN(C(c2cnn(C)c2SC)=O)CC)c(Cl)nn(C)c1C CC1(C)CCCCC1=CC(=O)NCC1CC1NC(=O)CC(=O)N(C)C c1(C(=O)NC(CNC(C(Cc2c(C)nc[nH]2)O)=O)CC(C)C)csc2nccn12 CCC(C)CC(C)C(=O)N1CC(NC(=O)Cn2c(C)cc(O)cc2=O)CC1C C1(CCNC(CCSC)=O)CCCCN1C(=O)C(C)Sc1ccccn1 C#Cc1ccc(C(=O)NC(CNC(=O)Cc2cnc(C(F)(F)F)s2)C(C)C)cn1 N1(C(CCSC)=O)CCC(NC(=O)CCc2cncnc2O)CC1C1CC1 c1(-c2scc(NCc3n(C)ncn3)n2)ccc(C#N)nc1 c1(C(N2CC3CN(C(c4c(C)c[nH]c4)=O)C3C2)=O)cccc2c1CCN2C C(C(C)C(C)C(=O)N1CC(CNC(c2ncccc2OC(F)F)=O)(OC)C1)OC C1(C(N2CCCC(O)CC2)=O)COC2CN(S(=O)(=O)CC3CC3)CC12 c1(CCCC)nc(C(=O)NC(CNC(C2CC2C)=O)CCOC)cs1 N1(C(C(n2ccc(Br)n2)C)=O)CC(NC(C2(CC3CCC3)CC2)=O)C(O)C1 Cc1c(C(=O)N(C)CC2CCN(C(=O)C3CC3)C2)[nH]c2ccc(C(N)=O)cc12 N1(C(c2ccc(CC)nc2)=O)CC2(C)CC1(C(=O)NCCCn1cnnn1)C2 N1(S(c2nc(C)n(C)c2)(=O)=O)CCC2(CC1)CC2(C)C(=O)Nc1ccccc1Cl c1(C(N2CC(NC(c3scc(C)n3)=O)C3(C2)CC3)=O)cccc2cc(Br)cnc12 Cc1ccc(CC(=O)NCC(c2ccccc2)NC(=O)C(C)(O)C2CC2)c(F)c1 c1(C(=O)NCCC(CNC(c2c(CC)c[nH]c2)=O)O)[nH]cnc1C#N N1(C(COC)=O)CC(CO)C2(C1)CN(C(=O)C(F)CCC(C)C)C2 Cc1cc(=NCCc2nc(O)n[nH]2)[nH]c(N2CCN(c3nnc(C)n3C)CC2)n1 Cn1c(O)nc(N2CC(n3cccn3)CC2C(N2CCCC(O)C2)=O)cc1=O Cn1cc(Cl)c(C(=O)NCc2nc(CNC(C3CC4(C3)CC4F)=O)cs2)n1 C1(C(N(C)CC2COCCN2C(c2csc(Cl)n2)=O)=O)CCCC12CCC2 c1(C(=O)NCC23CC(NC(C4CC(=C)C4)=O)(C2)C(C)O3)cccc2ncsc12 n1(CCNC2(F)CCN(C(=O)OC(C)(C)C)C2)c(O)nc2ccccc2c1=O C12(C(=O)NC(C(C)NC(=O)C#CC(=O)N(C)C)(C)C)CCCC1OCC2 C(=O)(C1=CCC(C)(C)CC1)NCC1CC2N(C(C(CCCCC)O)=O)C(CC2)C1 Cc1nc2cccc(C(N3CCC(C)(NC(C4COCCC4(F)F)=O)C3)=O)n2n1 Cc1cc(=NCc2cncs2)[nH]c(NC(C)CS(=O)(=O)CC(C)C)n1 CCC(CC(=O)NCC(C)(CNC(=O)C=Cc1ccccc1F)OC)CC(C)C c1(C(=O)NCC2N(C(CCN(C)CC)=O)C3C(C2)C3)cccn2c(C)nnc12 C12CN(C3(CCOCC3)C1)C2=O.n1(CC)nc(C)c2cc(-c3nnn(C)n3)sc12 N1(C(C(C2CCC(F)(F)CC2)OCC)=O)CCCC2(CCC2NC(=O)C(N)=O)C1 N1(C(c2ccnc(OC)n2)=O)CCC(C2(NC(=O)C(F)CC(C)C)CCC2)CC1 c1(N2CCN(C(C3C(C)C3)=O)CC2)ncnc2ccc(C(F)(F)F)cc12 N#Cc1cc(NC(C2CCCC(NCc3cc(Br)c(Br)s3)C2)=O)cc(F)c1 c1(C(=O)NCCC2(NC(c3c(N)ccc(OC)c3)=O)CC2)cc(S(C)(=O)=O)co1 Cc1ccnc(C)c1C(=O)NCC(F)CNC(c1cc(F)cs1)=O C1(C(C)C)OCCC1NCc1cn(CCCc2cnn(C)c2)nn1 CC(CC(C)(C)C)C(=O)N1CCC(CNC(=O)Cn2ncnn2)C(O)C1 C1(NC(N(CCN(C)C)Cc2nc(C(F)(F)F)cs2)=O)CC(=O)C1(C)C c1(OCCC(=O)NC(C2(CNC(C=C(CCC)C)=O)CC2)C)ccccc1[N+](=O)[O-] C1(NC(CC(C(C)OC)NC(=O)CN2CCOCC2=O)=O)CC2CCC(C1)N2C C1(NC(CC=CCC)=O)C2CC3C(C2)C13C(=O)NCCc1ncc[nH]1 N(C1CN(C(=O)CC2CCC23CCC3)Cc2ccccc21)C(C=COCC)=O C12(CNC(c3cc(C)no3)=O)CCCC1CCN2C(=O)COc1ccsn1 CC1(C)CC(C(=O)NC23CC(CNC(C45CSCC4C5)=O)(C2)C3)C(C)(C)O1 C1(NC(CCC(=O)NCCC)=O)CN(CCc2cccnc2C)CCC1C C(=O)(C(C)C(O)CC(C)C)N1C(C(N2CC(N(OC)C)C2)=O)CCOCC1 C(=O)(C(C)CC(N)=O)NC(c1nocc1C(=O)NCC1CC2(CC2)C(=O)O1)C N1(c2ncc(C(=O)OC)cc2Cl)CCN(C(c2ncsc2C)=O)CCC1C CC1CCN(C(c2cc(Cl)cc(Cl)n2)=O)CC1NC(c1cc(C2CC2)on1)=O c1(N2CCCC(NC(CC(CC)O)=O)CC2)ncnc2sc3c(c12)CCCC3 C(C(=O)NCc1ccccc1C)(C(C)CC)N(C(C(=O)NCC)=O)C C(=O)(CC1CCc2ccccc21)NC1(CN(C)C(C2Cc3nccn3C2)=O)CC1 N12CCC(CC(O)C1)C2=O.c1(C(=O)NCC(C2CC2)OC)ccc(CO)cc1F C(CCC(=O)NCCCSCCO)N(C)C(C1CC1F)=O N1(C(C(n2c(C)ccn2)C)=O)CCCC(C)(C)C1C(=O)NC1CCCC1C(C)C N1(C(CNC(CNC(c2c(C(=O)OC)nccc2)=O)=O)=O)CCC(O)C12CCC2 c1(CNC(C2CCCN(Cc3ccnc(Cl)c3Cl)CC2)=O)ccc(F)c(Br)c1 c1(N2CC3(N(Cc4c(C)ccc(C#N)c4)CC3)C2)ncc2cc(F)cc(Br)c2n1 C12(CNC(C3CCN(C(C(CO)NC(N)=O)=O)C3)=O)CCC(CC1)OC2 C12(CNC(COCC)=O)CCCC(CN1C(=O)COc1nn(C)cc1Br)C2 Cc1ccsc1C=CC(N1CCCC1CN(C)C(c1cnc(C2CC2)[nH]1)=O)=O C1(C(N2CCN(C(CCN(C)CC)=O)C(C3CCC3)C2)=O)C2CCC1(C)C2(C)C N1(C(C(c2ccc(C)s2)C)=O)CC(NC(=O)CCSC2CC2)CC1(C)C Cc1[nH]c2ccc(C(=O)NCc3cn(C4CC4)cn3)cc2c1C c1(NCCCOCC(C)C)ccc(C(F)(F)F)cc1S(=O)(=O)NCC1(C)CCC1 C1(C2(O)CCC2)(C(N2CCC(CC(=O)Nc3ccc(OCF)nc3)CC2)=O)CC1 C1(C(=O)NCC(C2CCCN2C(c2ncoc2C)=O)(C)C)(CC)CC(C)(C)C1 C1(C(=O)NCC(C)N(C(=O)CC2CC3CCC2C3)C)Cc2ccccc2O1 C1(C(=O)NCc2csc(C)n2)(NC(c2ccc(OC)o2)=O)CCCC1C N1(C(C2CCN(Cc3c(C)ncc(Cl)c3)CC2O)=O)CCC2COCC2C1 N1(C(Cc2nc(CC)sc2)=O)CCC(CO)C(NC(c2sccc2Cl)=O)C1 Cc1cc(C(N2CC(O)CC2CNC(C2CC23CC3)=O)=O)nn1CCO N1(C(c2cnn(C(C)C)c2Cl)=O)CCCCC(N(C)C(C2CC(F)C(=O)N2)=O)C1 C12(NC(CC(CC)C3CCC3)=O)CCCN(C(C3CC(O)C3)=O)CC1C2 c1(C(N2C(CN(C(=O)C3=CCCCC3)C)CCCC2)=O)cc2n(n1)CCCC2O c1(CN2C3CC(NC(CCNC(C(C)(C)C)=O)=O)C2CC3)ccc(F)c(C#N)c1 C(=O)(CCC(=O)c1cccs1)N(CCNC(=O)CCC1CC(C)C1)CC C1(NC(C=CCCC)=O)C2CC3C(C2)C13C(=O)NCc1ccc(O)cc1C C1(C(N(CCNC(C(CC)(C)O)=O)C)=O)CCc2ncsc2C1 c1(N2CC(=C(CNC(CCC(C)OC)=O)F)C2)ncnc2sc(C(F)(F)F)nc12 C1(NC(CC(CC)(C)C)=O)CN(C(C2CC3(C)CCC2(C)O3)=O)C2(CCCOC2)C1 CCCC(C(N)=O)NC(c1conc1C(C)NC(c1cnc(OC)s1)=O)=O c1(C(=O)NC2CN(C(c3cn(C)nn3)=O)CC2(C)C)ccc2nn[nH]c2c1O C1(C)(CNC(CC2(CC=C)CCCC2)=O)CCCN1C(=O)CN1CCC(C)(O)C1 CC1Cc2cccc(C(=O)NC34CCCCC3CN(C(c3ccsc3)=O)C4)c2O1 C1(F)(C(N2CC(CCNC(CCCN=[N+]=[N-])=O)OCC2)=O)CC12CCCCC2 Cc1ncnc(C)c1CC(N1CCC(CN(C)C(C2COCCC2(F)F)=O)C1)=O C1(CNC(CSCCOC)=O)CN(C(=O)CC(C)C)CC1O C(=O)(C(C(C)(C)O)NC(C)=O)NCC1(NC(COc2c(OC)scc2)=O)CCC1 c1(CC)ccc(C(=O)NC(C)CNC(=O)C(F)(F)C(F)F)cc1F c1(SCC(=O)NCC(C)(C(C)C)NC(C(CC)F)=O)ccc(F)c(F)c1 c1(C(=O)Nc2ccc(Sc3ccc(Cl)cc3)cc2)cccc(C#CCO)c1 CCCCCCCC(=O)NC(CCC(C)C)C(=O)NC1CCC2CC1CO2 C1(C(N2CCC(NC(c3n(C)cnc3)=O)C23CC3)=O)CCCC12CCOCC2 S(=O)(=O)(c1ccc(C(=O)NC(C(=O)N(CCNC(C)=O)C)C)cc1)NCC CC1(C)C(CNC(c2cnco2)=O)CCN1C(=O)CCC1CC1(Cl)Cl C#Cc1cncc(C(=O)NCC2(C)CCN(C(=O)CC3CCCOCC3)C2)c1 CC(C)CC(C)CC(=O)NCC1CC2(CC2)CN1C(c1cc2n(c1)CCOC2)=O Cn1ncc(CNC(=O)C(C)(C2CCC2)NC(=O)C2=C(Cl)CC2)c1O C(=O)(C1=NOC2(CCC2)C1)N1CC(OCCC(=O)NC2CC2O)C1 C=Cn1nccc1C(N1CC(C(=O)NCCNC(C2CC(C)CO2)=O)C1)=O c1(C(N2CCC(NC(CCCC#CC)=O)C(C)(C)C2)=O)ccc2c(c1)OCCN2 N1(C(c2ccc3nc(NC)sc3c2)=O)CCCC2CN(C(=O)C=C3CC3)CCC12 C1(C(N(C(C)C(F)F)C)=O)CCCN1C(C1(C)C=CCC1)=O C1(NC(N(CCOC)CCN(C)C)=O)CCC1 c1(NC(=O)CC2CCN(CC(O)CC3(C(F)(F)F)CC3)C2)nccc(Cl)c1F c1(OCCN(C)C)ccccc1CNC(C1CCN(C(=O)CCC#N)CC1)=O CC1CN(C(=O)CCNC2CC2)CC1NC(c1cc(-c2ccccc2)cs1)=O C1(NC(C(C)C)=O)CC2(CCC(CNC(c3cnn(C)c3C(F)F)=O)OC2)C1 C1(OC)CN(C(C2CC2c2ccsc2)=O)CC1NC(=O)CC1OCCCO1 C(=O)(C(C)(O)C(F)(F)F)N1CCC(F)(C(=O)NCc2ncc(C)cn2)CC1 N1(C(CCS(C)=O)=O)CC2C3CCC(C2C1)N(C(c1ccc(F)c(N)c1)=O)C3 n1(C(C)C)cccc1C(=O)N(C1CCN(C(C2(C(=O)N(C)C)CCC2)=O)C1)CCO C1(NC(C(CN(CC)CC)F)=O)CC2(CCC(CNC(=O)C(C)(C)CO)OC2)C1 CC(C)(C(=O)N1CC2CC(NC(c3ccc(O)nc3)=O)CC2C1)C(F)(F)F c1(C(=O)NC2CCN(C(CCc3onc(C)n3)=O)C2)cc(F)c(O)c(F)c1 CCC(O)C(F)(F)C(=O)N1CCN(C)C(CNC(=O)Cc2ccc(F)cc2C)C1 C1(C(=O)NC(CCNC(c2n(CCC)ncc2)=O)C)CCCCN1CCC C(=O)(CCCCC(C)CC)NC1C(NC(c2ccc(C#C)c(OC)c2)=O)CC1 CC(C(=O)NCC1(F)CCCN(C(=O)C(C)(C)n2cccn2)C1)S(C)(=O)=O c1(CC)cc(C(N2CCC(CN(C)C(c3ccc(C)o3)=O)C2)=O)ncn1 N1(C(C2(C)C(C)C2)=O)CC2(CC(C(=O)Nc3ccccc3SC(N)=O)CO2)C1 C(=O)(CC(C)(C)CC(F)F)NC1CCCN(C(COc2c(C)cccc2)=O)CC1 C1(C(N(CC=CC(=O)NC2CCN(CC)C2)C)=O)OCCOC1C c1(-c2onc(CCCCSC)n2)cc(=O)c2cc(Br)ccc2[nH]1 n1(CC)nnnc1C(c1nnc(C)s1)NCc1ccc(Cl)s1 C1(=CCO)CCN(CC(c2ccns2)NC(=O)CCc2ncc(C(C)(C)C)o2)CC1 N1(C(C2(C)CCCCC2(F)F)=O)CC2(C1)CN(C(C1CC(O)C1)=O)CC2CO N1(C(Cc2c(C)noc2C)=O)CCC2(CCCN2C(c2ccc(O)c(N)n2)=O)C1 C1(CC)CN(C(=O)CCc2cc(C)[nH]n2)CC1C(=O)NCC(C)C(=O)NC Cc1cnccc1-c1ccc(C(=O)OC(C)C(=O)NC(c2ccc(F)cc2)C)s1 c1(NCCc2cc(CC)no2)cc(C(C)(C)O)ncn1 N1(C(c2cc(C)oc2C)=O)CC2(CCCC(CNC(=O)CSc3nc[nH]n3)O2)C1 c1(CC23C(NCC4NC(=O)CC(C)C4)CN(CC2)C3)cn2ccnc2cn1 CCCCCC(CC)C(=O)N1CCCCC1CNC(c1nc(C)no1)=O N1(C(CS(=O)(=O)NC)=O)CC2(CC2)CC1CC(=O)NCc1ocnc1C CN1CCCC(C(=O)NC2COCC2NC(c2nccc(CC#N)n2)=O)C1 c1(N2C(C)CN(C3CC3)CC2)nccc(=NCc2c(N)cccc2Cl)[nH]1 C1(NC(C(C)CF)=O)CCN(C(=O)CN2CCCCCC2=O)CC12CCC2 C(CC1CC1)(CC(=O)Nc1c(O)ncnc1O)NC(c1c(OC)nn(C)c1)=O C1(C(=O)NCCCOCC=C)N(C(=O)CC(CC)CC)CC12CCCC2 N1(C(CCN(CC)CC)=O)CCC2(CCCCC2NC(c2cnco2)=O)C1 CC(F)(F)CCC(=O)NCCC(Cc1ccccc1)NC(=O)C=Cc1ccco1 C1(C(N2CC(OCCO)C2)=O)CCN(C(=O)C2CC3(CCC3O)C2)O1 C1(C)(CC)CC(C(=O)N(CCC(N2CCC(c3nn[nH]n3)C2)=O)CCCO)C1 C1(CC)CN(C(=O)CC2CCCC3(CC3)C2)CCN1C(c1ccnn1C(C)C)=O c1(CCC)ccccc1C(=O)NC1CCCC1CNC(=O)C=Cc1nccs1 N1(C(C(CC)CC)=O)CC2CC(C(N3CC4CC3CC4O)=O)CC2C1 c1(C(N2CC(NC(=O)Cc3csc(S)n3)CC(OC)C2)=O)nc2cnccc2s1 N1(C(CCC(C)SC)=O)CCC(C)N(C(=O)CSC(=N)N)CC1 Cc1nn(C)c2c(NC3CCNC(=O)CC3)nc(=NCC3(C#N)CCCC3)[nH]c12 C(=O)(CCCCCCC(=O)N1CC2CCN(C(C3CC4C=CC3C4)=O)CC12)OC CC#CCCCC(=O)N1CCC1CC(=O)NC(COC)CO C=CC1CN(C(c2cccc(C)c2N)=O)CC1NC(C1CCCC1C(F)(F)F)=O N1(C(CCC(=C)C)=O)CCCC(NC(=O)CCC(=O)N(C)C)C(F)C1 N1(C(C(C)n2cccn2)=O)CCc2sc(CNC(=O)CN=S(C)(C)=O)nc2C1 c1(C2N(C(=O)CC3CCN(Cc4ccc(F)cc4)C3)CCC2)cc(F)ccc1F Cc1ccc(CCC(=O)NC(C)CNC(=O)CC2OCCC2C)cc1C N1(C(c2cnc(CC)[nH]2)=O)CCCC1C1CCCN1C(c1oc(C)cc1C)=O C1(C(C(=O)NCC)N(CCC(C)CC)Cc2cn(C)cn2)CCCC1C(=O)OC C1(C(N(CCC(N2C(CCC(C)O)CC2)=O)CC2CC2)=O)CC2(CCC2)C1 C(=O)(CCCCC(N)=O)NC1C2(CCN(C(CCCCCSC)=O)C2)C1 c1(NC(c2n(CC)nnn2)C2CC2(Br)Br)cnn(-c2ccc(C)cc2)c1C C1(CNC(c2cnc(CC)[nH]2)=O)N(C(=O)CC2CCC(C)CO2)CCCC1(C)C Cc1cc(C(=O)NC2CC(N(C(=O)CC(C)c3cnn(C)c3)C)C2)sc1Cl C1(NC(C(Cc2cc(OC)cc(OC)c2)N)=O)CC2CC1C1CCCC21 N1(C(c2ccc(C(C)=O)o2)=O)CCc2c(OC)ccc(OC)c2C1 CC1CCN(CCC(N2CCCC(CNC(=O)CC3NC(=O)NC3=O)C2)=O)CC1 C#CCCCCCCC(=O)NC(C1CCN(C(C2(CCOCC)CCC2)=O)C1)C C1(C(CC(N(CCC)CCOc2nc(C)cc(O)n2)=O)(C)O)CCOC(C)(C)C1 N1(C(CCN(CC)CC)=O)CCC(C(=O)NCC2(O)CCC(C)(C)C2)C(O)C1 C(=O)(C1=NOC(C)C1C)NC(CCSCC)C(=O)Nc1cc(C)c(F)c(C)c1 c1(NC(CC2(O)CN(C(C(=C)F)=O)C2)=O)ccc(C(F)(F)F)cc1O C1(S(C)(=O)=O)(C(=O)NCCN(C(c2cc(C)ns2)=O)C)CCCCC1 c1(C(N2CCC(=CCNC(CCn3c(C)ncc3)=O)CC2)=O)cc(Cl)nnc1Cl CC(O)C(C)C(=O)NC1CC(F)(CNC(c2cc(-c3ccc(Cl)cc3)ns2)=O)C1 C(=O)(C1=CCN(C)C1)NC(C1CC=CCC1)C(=O)NCCCCCCOC n1(CC)nc(C(F)(F)F)c(C(N2CCC(c3cccnc3)OC(C)C2)=O)c1C(F)F CCCCC(CC)NC(=O)C(F)CC1CN(C(=O)CNc2cccnc2)C1 Cc1nn(C)c(-n2ccnc2C)c1C(=O)NCCC1CCN(C(=O)C(C)O)C1 CC1CC(NC(=O)CCCc2ccccn2)CCN1CCc1ccc(Br)cc1F c1(C(N2CCN(C(C3CCCCNC3=O)=O)CC2)=O)n[nH]c2c1COC2 CC(CC(=O)N1CCCc2ccnn21)NC(=O)CC1CC1C1CC1 Nc1cc(C(N2CCCC2CNC(c2ccncc2Cl)=O)=O)cc(F)c1 N1(C(CONC(C=CC=CC)=O)=O)CCC(O)C12CCC2 C(=O)(CCCCC1CC1)N1CCC(CCNC(=O)C(O)C2CCC2)C1 S(=O)(=O)(c1ccc(C(=O)O)cc1F)NC1CN(C(c2ccc(C)nc2Br)=O)C1 c1(C(N(C2CCCC3CC23)C)=O)cc(Cl)c([N+](=O)[O-])cc1F Cc1cc(C(=O)NCCN(C)C(C2CN(C)CC(=O)N2)=O)cnc1OC(F)F c1(C(C)C)cc(C(c2nnnn2C)NCCCN2CCCC2=O)no1 O=C1CCN(C(=O)Nc2ccc3c(c2)CC3)CC1c1ccccc1 C(C(C(=O)OC(C)(C)C)NC(=O)Nc1cnn(C2CCOCC2)c1)OC CCC(C)C(C(=O)N1CCN(C(C)CNC(c2cc(C)c(C)cn2)=O)CC1)OC C1(CCNC(c2cnc(N(C)C)s2)=O)CCc2ccccc2C1 c1(C(=O)NC2C3CN(C(C4C(C(=O)OCC)C4)=O)C2C3)cc(OC)cc[n+]1[O-] C12(C(=O)NCCCc3cccc(N)c3O)CCCN(C(C34CC(C)(C3)C4)=O)CC1C2 N(C(=NCCSC)NCC(N1CCCC1)=O)C(C)Cc1ccccc1 C1(C)(C(=O)NC2CC(CC(=O)Nc3cc(C)no3)C2)CC(F)(F)C1 O=S(=O)(c1ccc(Br)cc1NC1(CO)CCOCC1)N1CCCC(CCO)C1 CC(C)C(CCNC(=O)C(=O)NCC1CCCCC1N)N1CCCC1 C1(NC(=NCCOC(C)C)NC(c2ccccc2Cl)C)CCc2ccccc2C1 N1(C(c2c(OC)nsc2)=O)CCCC(O)(CN(C)C(C2CC2(F)F)=O)C1 CC(C)C(C)C(C)CC(=O)N1CCC(C)(NC(c2nccnc2Cl)=O)CC1 N1(C(C(=O)NCC)=O)CCN(C)CC1CNC(c1cc(C(N)=O)cc(Cl)c1)=O Cc1nc(CCNC(=O)C(C)N(C(=O)C=CCO)C)[nH]c1C C1(C(=O)NCCCOc2ccc(C)cc2)CC(N=c2[nH]cnc3cc[nH]c23)C1 C1(C(=O)Nc2ccc(OCCC)cc2)CCc2cnn(CC)c2C1 N(C1CCOc2ccc(Br)cc21)C(C1CC(O)CN1C(=O)Cc1cc[nH]n1)=O N1(C(Cc2ccc(C)cc2)=O)CCC(O)C(C(=O)NCCc2cn(C)nc2C)C1 c1(C(=O)NC2C(NC(CN3CCC(C)C3)=O)CS(=O)(=O)C2)cnc2ccoc2c1 N1(C(C(C(CC)(C)C)O)=O)CCC2(CCCCN(C(=O)C(C)NC(C)=O)C2)C1 C1(CNC(C(c2ccccc2)C)=O)CC(NC(=O)CCc2ccn(C)n2)CC1O c1(C(N2CC(C(C)C)N(C(C3CCCCN3C)=O)CC2)=O)cc2c([nH]1)CCOC2 N1(CC2CCN(c3c(OC)cccc3)C2)CC(N)CC(O)C1 C1(C2C(C(N(C(CC3CCC3)CF)C)=O)C2)CCCNC1 c1(N(C)CC2OCCN(C(C(n3ncc(C)c3)C)=O)C2)ncnc2scnc12 C1(C(=O)OCC)CCN(C(C2C(CC)CCN2C(=O)OC(C)(C)C)=O)CC1CO CC1(C(=O)NC2CC2NC(c2c(F)cccc2Br)=O)Cc2ccccc2N1 CCCC(CC(C)C)C(=O)NC1C=CCN(C(C2(N(C)C)CCCC2)=O)C1 C1(NC(C(C)OCCOC)=O)CCCC(NC(=O)C(c2cc(C)ccn2)(C)C)C1 C(=O)(CCC(=O)N(CCCOCCNC(=O)C(c1ncccc1F)(F)F)C)NC C(=O)(C(C)CS(C)(=O)=O)N(C1CN(c2cc(C)nc(C3CC3)n2)C1)C N1(C(C(n2cc(C(OCC)OCC)nn2)C)=O)CCC2CC12C C1(CNC(Cc2ccc(C(C)=O)s2)=O)CC2CCC1N2C(=O)C(F)OC C(=O)(C1Cc2ccccc21)N1CCCC(NC(C=Cc2ccc(C)o2)=O)C1 CC1(C)CC(C(=O)N2CC(NC(C3CC(n4ccnc4)C3)=O)C3(CC3)C2)=NO1 N#CCCCCCC(=O)NCCC1CCCN1C(C1CC2CC2C1)=O C(CCC(C(=O)NC1(CF)CCCC1)NC(=O)CCCN=[N+]=[N-])OC C(=O)(CCC(C)CC)N(C1CCC1NC(c1nc(CC(=O)OCC)oc1)=O)CC C1(C(=O)NCC2CCCCN2C(c2cc(CN(C)C)c[nH]2)=O)(CC)CCNC1=O c1(OC)cnccc1C(N1CC2CC1(CNC(=O)CC1CC(C(F)F)C1)C2)=O c1(C(=O)NC23C(CN(C(C4(C#C)CC4)=O)C2)C3)ccc(N=S(C)(C)=O)cc1 C1(C(N(C)CC2CCCC2)=O)CCN(C(C2(N)CC2)=O)CCO1 Cc1[nH]nc(C(=O)NCC2C3CN(C(=O)C(C)C4CC4)CC23)c1C(F)(F)F N1(C(C(C2CCCOC2)OC)=O)CCC(C)(CNC(c2ccc(C)nc2C)=O)CC1 O(C=C(C#N)C(=O)NCC(O)CNC(=O)CC1CCS(=O)(=O)C1)CC c1(OC)ncc(NC(c2ccc(C(=O)NC3CC3C(C)C)o2)=O)cc1C CCC(C(=O)NCC1CCCCN1C(c1cnc(C)nc1O)=O)C(C)C N1(C(CCNC(=O)OCC)=O)CC(OC)CC(NC(C2(C)CC(C)(C)C2)=O)C1 C(=O)(CS(=O)(=O)C(C)C)NC12CC(NC(C34CCC(CC)(OC3)C4)=O)(C1)C2 S(=O)(=O)(c1nc(N2CCC(Cc3nccs3)CC2)ccc1Br)N(CCOC)C N1(C(Cc2cc(C)no2)=O)CCN(C(=O)C=CCOc2ccccc2)CC(C)C1 Cc1c(C(=O)NC(C)CCCNC(=O)C(C)(C)c2cncs2)nc2sccn12 Cc1ccnc2c(S(=O)(=O)N3CCCC4(CC4)C(F)(F)C3)cccc12 c12ccn(n1)CCC(=O)NCC2C.c1(COC(C)C)ccccc1 CCC(C#N)C(=O)NCC(CO)NC(c1ccnn1CCN(C)C)=O S(=O)(=O)(c1ccc(C)c(C(=O)NC23CC(C2)N(C(c2cnsc2)=O)C3)c1)NCC c1(C(=O)NCC(C)NC(C(C)OCC)=O)cnc2c(F)cccc2c1C1CC1 N1(C(C2C(CC)CCC2)=O)CCC(CC2CCN(C(=O)CC3CC3)CC2)CC1 c1(CN(C(C(CC)N(CC)CC(C2C=C2C)=O)=O)CC)cccc(CN(C)C)c1 C1(NC(C(C)OC)=O)C=CCN(C(c2cccnc2-n2ccnc2)=O)C1 c1(C(N2C(CNC(CC(=O)N(C)C)=O)COCC2)=O)c(F)cccc1Cl N1(C(Cc2cc(OC)no2)=O)CC(NC(=O)CCN2CCOCC2)C2(CCC2)C1 C1(NC(c2nc(COC)oc2)=O)CN(C(=O)Cn2nnc(C(C)(C)C)n2)CC1O C1(C(F)(F)F)(OC)CC(C(N2CCC(N(C(=O)C=Cc3cocn3)C)C2)=O)C1 N1(C(c2scc(CC)c2)C(=O)NC2CC2)CCCc2ccc(NC(C)=O)cc2C1 Cn1cc(C(N2CCCC2C2CCN(C(c3cccnc3O)=O)C2)=O)ccc1=O N1(C(c2n[nH]cc2Br)=O)CCN(C(=O)CN2CC=CC2)C(C2CCCC2)C1 CC(C)C(C(=O)NCC12CC(NC(=O)C(F)CC3CC3)(CO1)C2)n1cncn1 C1(c2nnnn2CC2CCOC2)(NCc2onc(C(C)(C)C)n2)CC2CC2C1 N1(C(CCC#CC)=O)CCC(C)CC1C(=O)NC(CCOC)C(C)C C1(CNC(C(C)SC)=O)CC(O)(CNC(=O)Cc2cnn(C)c2)C1 c1(CC(C(=O)NC2CC2)NC(c2ccc[nH]2)=O)cccc(Cl)c1.C12CN(C1)C2=O C1(C)(NC(C=CCC)=O)CCCN(C(=O)CCc2cc(Br)ccc2F)C1 C1(C(=O)NC2C(NC(=O)CNC(c3cscn3)=O)C2)CC12CC(F)(F)C2 CCCCCC(=O)NCC(=O)NC1CN(C(=O)C(CC)SC)CC1C.N1(C)CCC1 Cn1ncc(Br)c1C(=O)NCC1CCN(C(c2cc(=O)cco2)=O)C1 C1(C(=O)Nc2cc(CCC)no2)CC(F)(F)CN1C(c1ccc(F)cc1C)=O O=C(CC(F)(F)Cl)NC1CCC(NC(C2(C(F)(F)F)CC=CCO2)=O)C1 N1(c2ncc(C)s2)CCN(C)C(c2ccccc2)C1.N12CCC(O)(C1)C2=O N1(C(c2ccc(C)cc2)=O)CCC(CNC(=O)C=CCN(C)C)C(C)C1 CC1CN(C(c2coc(N(C)C)n2)=O)CC1C(N1CCC1c1cccnc1)=O.C(O)(=O)N.C=O N1(C(C(C)Cc2cnc[nH]2)=O)CC2CCCC1C2CNC(=O)CCF C1(OC)CCC2(C(N3CCCC3CN(C)C(C3CCC(=O)N3)=O)=O)CC12 c1ccc(S(=O)(=O)N2CCN(C3CC3)CC2C)c(Cl)c1.CC1COCCC1C Cn1cc2c(n1)CCN(C(=O)CNC(=O)CCc1cn[nH]c1)C2 CC(C)C(CCNC(C1CC1(C)C)=O)NC(c1cc(=O)n(-c2ccccc2)[nH]1)=O C1(NC(c2c(OC)nsc2OC)=O)CS(=O)(=O)CC1NC(=O)CNS(C)(=O)=O c1(CN(CC(C(OCC)OCC)O)C)cc(S(=O)(=O)N2CCOCC2)ccc1C N1(C(C(C(C)C)O)=O)CCC12CN(C(=O)Nc1c(F)cccc1F)C2 CN1CC2(CCN(C(C3C4CC3N(Cc3cscc3Br)C4)=O)CC2)C1 C(CC(O)CNC(=O)COCC(F)(F)F)NC(COC)=O.C1(C)CN1 N1(C(CNC(=O)C2CC2)=O)CC2CC(NC(C3(n4ccnn4)CC3)=O)C1C2 c1(OCC)cc(C(=O)NC2CCC(C)(CNC(=O)C(F)F)C2)ccn1 C(=O)(C(C(C)C(F)(F)F)OC(c1cc(C)c(Cl)cc1C)=O)OC Cc1ccccc1C=CC(=O)NC1C2CN(C(=O)C=Cc3cccc(Cl)c3)CC12 CCC(C)CCC(=O)N1CC(OCCC(=O)NC(CO)C(=O)N(C)C)C1 c1(C(N2CC3C(NC(=O)CCc4ccsc4)C3C2)=O)cnc2ncccn12 C(=O)(CC(C(F)F)c1ccccc1F)N1C(c2cc(COC)on2)COCC1 C1(C(N2CC(O)(C(=O)NC)C2)=O)CC(NC(C2(C(=O)N(C)C)CC2)=O)CCO1 c1(C2C(C(N3C(c4ccc(C)cc4)C(=O)NCC3)=O)C2)c[nH]c2ncccc12 c1(C(=O)NC2C(C)CN(C(=O)CC3OCCO3)C2)cccn2nnnc12 C1(C(=O)NC2CC2)CN(C(=O)C(CCc2ccsc2)N2CCCC2)CCO1 C1(C(N2CC(=O)NCC2)=O)CC2CC1CC2NC(=O)CC1CCSC1 C1(C(=O)NCC2C(C(=O)OC)CC2)CC(F)(CNC(CN2CCCC2)=O)C1 C12(C(=O)NCC3C4CN(C(c5c(OC)nsc5)=O)CC43)CCCC1C2(F)F C1(NC(C2CC23CC3)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)CCC1CO CC1(CC(N2CCC(NC(=O)COC(F)(F)F)C2)=O)CCOCC1 N(C1CCCNc2ccccc21)C(C1(C(CC2CC2)=O)CCSCC1)=O C1(COC)CCC(NC(=O)C(Cc2cn[nH]c2)NC(c2nsnc2O)=O)CC1 Cc1ccc(C(=O)NCC(CC(C)C)NC(C2C(C)CC2C)=O)c(F)c1F c1(C(=O)NC(CN(C)C(c2ccc(C(F)F)s2)=O)(C)C)ncccc1N C(c1ccc(C)c(C)c1)=CC(=O)NCC1C2N(C(C(C)SCC)=O)C(CC2)C1 n1(C(C)C)cnnc1SCC(N1CC(NC(=O)Cc2coc(C(F)F)n2)C1)=O c1(C(=O)NC(C(C)NC(c2cocn2)=O)C)ccc(N2CCCS2(=O)=O)cc1 C1(C2CCN(C(=O)C(F)CC(C)C)C2)(NC(Cc2cc(OC)no2)=O)CC1 C1(CC)CN(C(=O)Cn2nnnc2C)CCN1C(=O)CC(=O)OC C(=O)(CC1=NNC(=O)C1)NC1CN(C(C(C)(C)SC)=O)CC12CC2 C(=O)(C(C)(C)S(C)(=O)=O)NCC(CNC(C(C)(C)Cc1cnn[nH]1)=O)O Cc1cc(CNC(=O)C=CC(C)NC(=O)CCN2CCOC2=O)co1 C12(C(N(CCC)CCNC(=O)C(O)CCN(C)C)=O)COC(CF)(C1)C2 N1(CC)CCC(C(=O)NC(CN(C)C)C(N2CC(C)(C)C2COC)=O)CC1 CC1CN(C(c2nnsc2C(F)F)=O)CCC1N(C(=O)C(Cl)=CCl)C C1(C(=O)NC2CC(C)(NC(c3c(Br)ccc(C)n3)=O)C2)OCC2CCCCC12 N1(C(c2cn(CC)nn2)=O)CCN(C(=O)CC(C)(C)O)C(CC(F)(F)F)C1 c1(C(N(C)CC2N(C(C(C)NS(C)(=O)=O)=O)CCCC2)=O)ccc(N)cc1O c1(C(C)=O)cccc(OCC(=O)NCC(C2CC2)NC(c2cc(O)n(C)n2)=O)c1 Cc1cnc2cc(C(=O)NCCC(C(C)C)NC(=O)CC3C=CCC3)ccn12 C1(CC)CN(C(=O)CC2CCCCN2C)CCN1C(=O)CN1CCC(O)CC1 CC1CCC(C(=O)CCC(=O)N2CCC2CNC(=O)C=Cc2cncs2)CC1 CCCCCC(O)C(=O)NC1CC2CC(C1)N(C(c1cc[nH]c(=N)c1)=O)C2 C(=O)(C(C(C)(C)C)c1ccccc1)NCC1CN(C(c2ccc(COC)s2)=O)C1 C1(CCC(=O)N2CCCC2)CCC(=O)N1.C12CCN(C1)C(=O)C2.CC(C)NC c1(C(=O)NCC2(C)N(C(C(CC=C)C)=O)CCC2)ccc2nc(C)sc2c1 c1(C(=O)NCCC(C)NC(C=C(CC)CC)=O)sc(C)c(Br)c1OC C1(C#N)(CCN(S(=O)(=O)CC2COC3(CCCC3)O2)C)CCS(=O)(=O)CC1 C12(COC)CC(CNC(=O)CCn3ccnc3)(CN1C(=O)C(C)CC1CCCO1)C2 c1(C(=O)NC2CCCC(N(C(c3ccc(SC)o3)=O)C)C2)cc(N)c(Cl)c(O)n1 C1(C(N2CCC3CN(C(c4[nH]cc(C)c4)=O)CC32)=O)Cc2ccc(F)cc2C1 c1(C(N(CCC(=O)NC(C)CC2CCC2)CC=C)=O)coc(COC)n1 N1(C(C(=O)NCC=C)C)CCC(NC(=O)Cc2cc(O)nc(O)n2)CC(C)(C)C1 C(=O)(C1CCc2cccc(F)c21)NCC(CNC(c1scc(C)c1)=O)O c1(OC)ccc(C2CC2)cc1CNC(c1nnc2n1CCC2)C c1(C(=O)NCC2C(NC(c3c(COC)cccc3)=O)C2)cc(OC)c(C2CC2)nn1 C1(CNC(c2cc(C)[nH]n2)=O)CC(C)N(C(=O)C=Cc2ccsc2C(F)(F)F)C1 c1(OCC(N2CCC(CNC(C(C)c3ccco3)=O)C2)=O)ccc(F)cc1Cl Cc1cc(C(=O)NC2(C(N3CC4CC=CC3C4)=O)CC2(C)C)nc(C)n1 c1(NCC(CNC(CC(n2ccc(C)n2)C)=O)O)nc(Cl)nc2sccc12 N1(C(Cc2c(CC)cccc2)=O)CCC2(CC1)CN(c1nccc(C)n1)CCO2 c1(OC)cc(NC(C2CCCCC23CCC3)c2nnnn2C)ccc1S(N)(=O)=O n1(-c2ccccc2)nc(C2CSC2)nc1C1CC1 Cc1nc(C(N2CCCC2CN(C(=O)CCCOC2CCOCC2)C)=O)sc1C c1(CNC2CC3(CC(NCc4ccc(C)cc4O)C3)C2)c(Cl)cc(Br)cc1Cl c1(CNC2C(C(=O)Nc3cccc(CC)c3)C2)cccc(OC)c1Br C1(CCNC(c2c(C)c[nH]c2)=O)CCCCN1C(c1cc(O)nn1C)=O Cc1cc(C(=O)NC2CN(C(=O)CCn3cccn3)CC23CC3)ccc1Br c1(N(CC)CC)ccc(C(N2CC3C(CNC(C4CC(C)C4)=O)C3C2)=O)cc1 C1(NC(Cn2nnc(C)n2)=O)COC2(C1)CN(C(C1CCC13CCC3)=O)C2 N1(C(CC=C)=O)CCc2ccc(C(=O)NC3CCCCC3OC)nc2C1 N1(C(C=C(C)Cl)=O)CCCCCC(NC(C2CCCN2c2ccccc2)=O)C1 C1(CCOC)CN(C(c2cc(O)nc(Cl)c2)=O)CCN1C(=O)CC(C)(C)C#N C(=O)(C1=NN(C2CC2)C(=O)CC1)NCC(CNC(C(C(C)C)OC)=O)CO C1(C(N(CCCCNC(c2c(C)coc2)=O)C)=O)CCc2ncsc2C1 c1(Cn2cc(CC=C)nn2)cccc(CNC(C2COCC2CS(N)(=O)=O)=O)c1 C12(C(N(CCCNC(C(C)NC(=O)C(C)(C)C)=O)CC)=O)CCCC1(C(N)=O)C2 c1(CCC(=O)NCC2N(C(CC(C)SC)=O)CC=C2)ccccc1[N+](=O)[O-] c1(C(=O)NCC2C(NC(C3N(N=O)CCC3)=O)COC2)ccc(C(F)F)c(F)c1 c1(C(=O)NC(CCCC)CNC(c2ccc(Cl)c(N)c2)=O)nnn2c1CCCC2 N(C1CCc2ccccc21)C(=O)CC1CCCN(CSc2cccc(Br)c2F)C1 Cc1cc(OC(C)C(=O)NC(C)CNC(C2CC(C)(F)C2)=O)ccc1Cl C1(CC)(NC(=O)Cc2cc(C(C)C)no2)CCN(C(C2C(OC)C2)=O)CC1 C1(C2CCCCC2)(C(=O)NCC2CN(C(C(CSC)OC)=O)CC2O)CC1 Cc1cn2cc(C(N3CC4(CCCC4NC(=O)C(C)OCC4CC4)C3)=O)nc2s1 C1(CNC(=O)Cc2ccoc2)C2CCC(C2)N1C(c1cncc2nc[nH]c12)=O N1(CC(=O)NCC(C)(C2CC2)OC)CCN(C(C2(CO)CCCO2)=O)CC1 N1(C(C(F)=C(C)C)=O)CC2C(C(N3CCCC3C(=O)N(C)C)=O)C2C1 c1(C(N2CC(N(C)C(C3CC(c4ccccc4)O3)=O)C2)=O)c(Cl)cccc1Cl C1(C(N2CC(NC(C3(CC=C)CCOCC3)=O)C(O)C2)=O)CC2(CCC2)CO1 c1(C(=O)OC)cc(C)nnc1NC1CC(CNC(=O)CN2CCS(=O)(=O)CC2)C1 c1(C(c2nnnn2C2(C)CC2)NC(C=C)C)cn(C)cn1 CC1(F)CCC(C(=O)NC2(C)CC(NC(c3ccncc3)=O)C2)CC1 N1(C(C(CCC)O)=O)C2CCC1(c1cn(CCOc3cnn(C)c3Br)nn1)CC2 c1(C(=O)NC(C)CC(C)NC(=O)Cc2cnsc2)cnc2c(c1)COCC2 C1(CC)CN(C(c2ncoc2CC)=O)CCC1NC(=O)C(C1CCCO1)C1CC1 c1(C(=O)NCC(CO)NC(C(CC#C)C2CC2)=O)c(C)[nH]c2ccc(F)cc12 N1(c2nc(C)nc(O)c2)CC2CCC1CN2C(c1ccc(F)nc1F)=O c1(C(C(=O)NC2C(NC(CC3(OCC)CC3)=O)CCC2)O)cccc2c1OCC2 C1(C)(CNC(Cc2c(C)cco2)=O)CCN(C(=O)C(F)F)C1 c1(C(N(C(C)CNC(=O)CCC2CCCN2C)C)=O)ccc(S(=O)(=O)N(C)C)o1 C1(CC(N)=O)(NC(=O)C(N)=O)CCN(C(c2cc([N+](=O)[O-])sn2)=O)CC1 C1(C(N(CCCCNC(c2scc(C)c2)=O)C)=O)NC(=O)CC1C(F)(F)F c1(NC(=O)CCC2CCCN2C(c2ccccc2CO)=O)cc(O)ccc1Cl C(CCCCNC(=O)CCCC1(NC(=O)CC2CCCO2)CCC1)N(C)C c1(C(=O)NCCN(CC)Cc2nn[nH]n2)ccc(NC(=O)OC)c(F)c1F C1(C(=O)NC2C(CNC(CC3CC(N(C)C)C3)=O)CCCC2)CN2CCC1CC2 N1(C(CC2N(CC)CCOC2)=O)CCN(C(C2CCC(=O)N2)=O)C2CCCC12 c1(OC)cc(C(=O)NC2CC(O)(CNC(C3CCCOC3)=O)C2)c(C)cc1O c1(C(=O)NC(C)C(C)NC(c2c(C#N)cnn2C)=O)cnc2ccccn2c1=O c1(SC(C(=O)NCC(CC)NC(c2nocc2Br)=O)C)ccccn1 CCCCC(C(=O)N1CCOC(C(=O)NCC(=O)OCC2CC2)CC1)C(C)C C(=O)(C(C)(C)CC(F)(F)F)NCC1(CNC(C(C)n2ccnc2)=O)CCC1 C(=O)(CC(C)CC(F)(F)F)N1CCC(CC)(NC(=O)C(CN(C)C)C(C)C)CC1 CCCCCC(CC)C(=O)NCCC(C)N(C(=O)COCc1ccc(C)cc1)C C1(NC(C2(COC)CCC2)=O)CCCCC1CNC(=O)Cc1c(C)cnn1C C(=O)(C(C)C(C)O)N(CCOCCCNC(c1cc(C(C)C)no1)=O)C N1(CC)CCN(CC(N2CCC(NC(=O)C(CC(C)C)OC)CC2)=O)C(=O)C1=O CCC(CC(=O)N1CCC1CC1CC1)NC(c1ccn(C)c1C)=O C(=O)(C1=CC2(CCN(C(=O)CCCC(CC)CC)C2)C1)NCC(C=C)(C)C c1(CC)cc(C(N2CCC(CC)C2C(N2CC(O)(C(=O)OC)C2)=O)=O)c(C)o1 c1(C(=O)NCC(CNC(=O)C2=CCSC2)O)nccc2c(Cl)cccc12 c1(C(=O)NCCCCCCNC(C(P(C)(C)=O)O)=O)coc2ccccc12 C1(C)(CNC(C(C2CCOCC2)OC)=O)CCCN1C(c1cccc(CO)c1)=O C=CC(C)CN=C(NCc1cccs1)NC1CC2CCC1OC2 Cc1cncc(CCNC(=O)C(O)CCNC(C2(CO)CC(C)(C)C2)=O)n1 c1(CN2C(C(=O)NC(c3ccc(Br)cc3)C)CC3CC32)c(O)cc(Br)cc1F c1(CC(=O)NCC2CC(F)CN2C(C2CC23CC3)=O)cnn2c1CCCC2 C1(CNC(c2cnc(CC)o2)=O)CCCCN(C(=O)C#CC2CC2)C1 c1(C(=O)NCC(C)C)ccc(C(=O)NCC2CCN2C(=O)C2=CCSC2)cn1 Cc1cc(F)sc1C(N1CCCC1(C(N1CCC(CN=[N+]=[N-])C1)=O)C(C)C)=O CCC(C)(CO)C(=O)N1CCOC(CC(=O)NC2CC3(CCCC3)C2)C1 C1(C#N)(C(N2CC(CC(C)NC(CCN(C(C)=O)C)=O)C2)=O)CC2CCC1C2 C12(C(=O)NCC(C(C)C)NC(c3c(C)cccn3)=O)CC(C)(C1)OC2C C(=O)(C(F)C(F)(F)F)N(C1CCN(C(c2cc(COC)sc2)=O)C1)C Cc1cnsc1C(=O)NCC1(O)CC(C(=O)NC(C)CCc2cn[nH]c2)C1 N1(C(=O)OC(C)(C)C)CC2CC1CN2C(C1(S(C)(=O)=O)CC1)=O C1(CNC(c2ccn(CC)n2)=O)CN(C(C2CC(OC(F)F)C2)=O)CCO1 c1(C(=O)Nc2cccc(C3CCCCC3)c2)cc(Cl)c2ncccc2c1F C1(C(=O)OC)CCCC1NC(=O)N(C)Cc1ccnn1C C(CCC(C)CC(=O)N(C(CNC(C1C=CC=CC=C1)=O)C1CC1)C)=C(C)C C1(OC)CC(CCNC(=O)Cc2ccoc2C)N(C(C2CC3CC3C2)=O)C1 C(C(O)C(=O)NC(Cc1cc[nH]n1)C(=O)NCC(=C1CCCCC1)F)=CC c1(C(=O)NCC(CC=C)NC(=O)C(C)=CC)ccc(Br)c(CC)c1 C1(OCC(=O)NCC)CCN(C(=O)Cn2nc(C)cc2C(F)F)C(C)C1 c1(CC(N2CC(NC(CCNC(=O)C=CCl)=O)C(O)C2)=O)c(F)cccc1Cl C(=O)(CCCCCCC(=O)N1CCCC(NC(=O)Cn2cnnc2O)C1C)OC C1(CCC)CN(C(=O)C=C2CCC2)CC1NC(=O)C(C1CCC1)OC C1(NC(=O)C(c2ccccc2)F)CCCCC12CCN(C(=O)CC1CC=CC1)C2 c1(C(=O)NCC2(NC(C(C)n3ccnn3)=O)CCOCC2)cc2[nH]ccc2s1 c1(OC)ccc(N)c(CC(N2CCC(NC(=O)COCC(C)C)C2)=O)c1 c1(N(C)C)ccc(C(N2CCC2Cn2ccnn2)=O)cc1 C(CC(=O)NCc1ccc(O)nc1)(C(F)(F)F)NC(C(CCC)C#N)=O C1(C(=O)NC(CN(C(c2cc(C(C)C)on2)=O)CC)C)CN(CC)CCO1 C1(C(=O)NC(c2ccsc2)C)CCN(C(c2cnnc(O)c2)=O)C(C)(C)C1 N1(CCC(=O)N(CCN(C(C2CC(OC)C2)=O)CC)CC)CCOCC1=O c1(N2C(C)CC(CNC(c3ccc(OC)cc3)=O)C2)ncc2ccnc-2[nH]1 CC(C)C(C)CCNC(=O)CC1CCN1C(=O)C(C)SC(C)C C=C(Cl)C(C)(C)C(=O)N1CCN(C(c2cc(OC)ns2)=O)C(C(=O)NCC2CC2)C1 c1(N2CCC(CNC(CCc3cc(C)no3)=O)CC2)ncnc2scc(C)c12 N1(C(C2(NC(CCSCCC)=O)CSC2)=O)CC(C)CCC1C C1(CNC(c2ncccc2O)=O)(NC(C2C(Cl)(Cl)C23CC3)=O)CCCCCC1 C=CCCC(C(=O)NC1CCCC1CN(C)C)NC(c1cncc(NC)c1)=O C1(NC(CCCOc2cccc(C)c2)=O)CCCN(C(=O)CC2CC2C)CC1 C1(CNC(c2cnc(C)[nH]2)=O)CC(NC(=O)CC2CC2C(F)(F)F)C1(C)C O=C1NCC2(CCN(C(=O)NC3CCc4ccc(F)cc4O3)CC2)O1 Cc1cc(Cl)c(C(=O)NC2C3CN(C(C4CCCC(=O)N4C)=O)CC23)cc1N c1(C(=O)NC2CCN(C(C3C(=C)C3)=O)C2C2CC2)cc(C)sc1S(N)(=O)=O N1(C(C(C(=O)OC)C)=O)CCC(C(=O)NCCCOCCOCCO)(CO)CC1 N1(CC(N2C(CC(N3CCC(N(C)CC)C3)=O)CCC2)=O)CCCCC1C c1(CC(C(=O)NCCC2CCN(C(=O)Cc3cccnc3)C2)O)ccccc1Cl N1(C(c2ccnc(F)c2OC)C(=O)NC(C(=O)OC)C)CCC2CN(C)CC2C1 C1(NC(C(CC=CCC)C)=O)CC2CCCC(C1)N2C(c1cn(C)nn1)=O C1(COCC(=O)NCCOCCNC(COCC(=C)C)=O)CCOC1 c1(C(=O)NC(C)Cc2ccc(CNC(c3cnco3)=O)cc2)nccc(Cl)c1F Cn1nccc1C(F)=CC(=O)NC1(CNC(C2(C(C)(F)F)CC2)=O)CC1 C#CC1(C(N2CC=CC2)=O)CCN(C(=O)CC(CC)C2CCC2)CC1 c1(-n2c(C(C3(C)CCCS3)NCCC(N3CCC(C)C3)=O)nnn2)ccc(F)cc1 c1(C(=O)NCCOCCCN(C(C2CC(C)OC2C)=O)C)occ2c1CCOC2 n1(CC)ccc(C(=O)NC2CCCCC2NC(c2occc2COC)=O)c1C c1(CC(=O)NCC(C)NC(=O)CCC2CC2(Cl)Cl)ccc(O)nc1 n1(CC(CC)O)cc(C#CCNC(=O)CN2CCCNC2=O)nn1 N1(C(c2c(CC)scc2)=O)CC(NC(C2(CC)COC2)=O)CC(O)C1 c1(C(N2CCS(=O)(=O)C(CCNC(C3CC3C)=O)C2)=O)nccn2c(Br)cnc12 c1(CNC(C2CCN(CSc3ccccc3C3CC3)CC2)=O)ccc(O)c(F)c1 c1(NC(C2(c3ccccc3I)CC2)=O)cc(F)ccc1CO C(=O)(CC1=CCCC1)N1CCC(OC(C(=O)OC)C2CC2C(=O)OC)CC1 C12(C(=O)NC(C)CNC(c3cccc(OC(F)(F)F)c3)=O)CCC(C)(CC1)C2 C12(C(=O)NCc3c(C(=O)NCCCC=CC)con3)CCC(CC1)CO2 c1(C(N2C(C)(C(=O)NC3CCN(C(C)=O)C3)CC(O)C2)=O)ccn2nccc2c1 CC(C)C(C(=O)NC1(CNC(=O)CCN2C(=O)CCC2=O)CCOC1)NC(N)=O c1(C(=O)NC2C(OCC)CCOC2)ccc(N(C)C)c(Br)c1 N1(C(C(N2CCCCC2=O)C)=O)CCCC(CN(C)C(C2(C)C=CCC2)=O)C1 C1(C(N(CC(=O)N(C(C)CCO)C)C)=O)CC2CCC2C1 CC(C)(C)CCCCC(=O)NCC1(F)CCN(C(C2CC(C#N)C2)=O)C1 C1(C(=O)Nc2cccc(NC(CCCN=[N+]=[N-])=O)c2)CCN2CCOCC12 N1(C(=O)NCCCC2CCCCO2)CC2C(c3ccc(Br)cc3)(CCS2(=O)=O)C1 N1(C(C2C(C(C)C)OCC2)=O)CC2(C(N3CC(O)C(C4CC4)C3)=O)CCC1CC2 c1(SCC)ccccc1NC(c1cn(CC)nc1C)C(=O)NC(C)C(CC)CC C(C(C)C(C)(C)C)(c1nnnn1-c1ccc(C)cc1Cl)Nc1cccc(CC)c1 c1(OCCCOC)ccc(CN2CCCCC2C(=O)O)cc1 c1(SC)ccc(NC(N2CCC(C(F)(F)F)(CO)C2)=O)cc1[N+](=O)[O-] C1(NC(COCC)=O)CC2CCC1N2C(C1(F)CCCOC1)=O c1(C(N)=O)ccc(C(=O)NC23CC(CNC(C4CC4(Cl)Cl)=O)(C2)C3)o1 C1(C(N2CCC(C(C)C(N3CC(F)C(F)C3)=O)C2)=O)C2CCC(C2)C1C C(=O)(C(CC(F)F)NC(=O)CC1CC2(CC2)CO1)NC(C(C)C)CCO C(=O)(CCC(C)OC)NCC(C1CCC1)NC(CNC(CC)=O)=O c1(C(N2CC(CO)(NC(C3(F)CCC3)=O)C2)=O)ccc(=O)n(-c2ccccc2)c1 C(=O)(CCCCC(=O)NC)NC(C(C)NC(CC=CC=C)=O)CO C12(CNC(C(CCOC)(C)C)=O)CCCCC1N(C(C1CCSC(C)C1)=O)CC2 c1(CC)cc(OC)ccc1C(=O)NCCC(C)NC(c1cnc(OC)s1)=O N1(C(COCC(C)C)=O)CCCC1CC(=O)NC1C=CCC1 C=C(C)c1cn(C(C)C(c2ccccc2)NC(c2cc(C)ncn2)=O)nn1 C1(C2CCCN(C(c3ccc(N)c(C)c3C)=O)C2)(NC(c2cnc(C)[nH]2)=O)CC1 c1(OC)cc(C(=O)N(C(C)CCNC(=O)C(C)=C2CC2)C)c(Br)cc1C N1(C(CCNC(C2C(C)C2)=O)=O)CCCC(O)(CCNC(=O)C=CC2CCC2)C1 c1(C(N2CC(CNC(c3coc(Cl)n3)=O)C3(C2)CC3)=O)cnn2c(Cl)cccc12 CC1CC(NC(c2cccc(Cl)c2C(F)(F)F)=O)CN(C(C2CC(C#N)C2)=O)C1 C1(C(=O)NC(C2(O)CN(C(C3CC4(CCC4)CO3)=O)C2)C)CCC(=C(F)F)CC1 C1Cc2c(O)cccc2N1C(=O)OCCN1CC(C)OC(C)(C)C1.C(C)(C)(C)O CCCCC(C(=O)N1CCC1CC(N1CCC(OC)CC1)=O)C(C)C.C1(C)(C(=O)NC=O)CC1 C(=O)(C(C(=O)OC)OC)N(CC)CC.C1C(C)(C)CS1.C12CCC1CNC2=O N1(C(C(c2c(C)n[nH]c2C)C)=O)CC2=C(C1)CN(C(=O)C1=CCCOCC1)C2 N1(C(c2ccc(C)c(F)c2)=O)CC2C=CC1C(C(=O)NC1CNC(=O)C1(C)C)C2 C(=O)(C1=CC(O)C(O)C(O)C1)N1CC2C(C)(C)C2C1C(=O)Nc1ncccc1Br C1(C(=O)NC2CCN(C(C(C)CC(N)=O)=O)C2(C)C)CN(CP(C)(C)=O)C1 N1(C(=O)CCOCC2CCCO2)CCCCC(C2CN(C(=O)C(O)C3CC3)C2)C1 c1(CN(CC(CC(=O)NC(C)C)C)C)[nH]c2ccccc2c1C C1(NC(c2cc(OC)nn2C)=O)CC(F)(F)CC1NC(=O)Cc1cccc(Cl)c1 c1(CC(=O)NCC(CC)NC(c2ccsc2C)=O)c(C)ncnc1C N1(C(c2cc(C)ncn2)=O)C2CCC(C2)C1CC(=O)NCC1(F)CCCCC1 c1(C(=O)NCC2OCCN(C(Cc3ncc(CC)[nH]3)=O)C2)c(C)ncn(C)c1=O C1(C(=O)NCCNC(=O)OC)C2CCN(C(c3cnncc3C)=O)CC12 N1(CC(=O)NC2(C)CC(NC(C3(c4ccnc(Cl)c4)CC3)=O)C2)CCCNC1=O C1(C)(C(=O)NC2COCCN(C(C3C(C)(Br)C3)=O)C2)CCCNS1(=O)=O c1(OC)ccc2c(c1)C(C(=O)OCC(C1OCCOC1C)=O)CO2 c1(C(=O)NCCC(CC)(CC)NC(=O)C=C(C)C(C)C)ccc2c(c1)CC(C)O2 c1(C(=O)OCC)c[nH]c(=NC(C)C2CCN(C(c3cc(CF)on3)=O)CC2)cn1 Cc1ccc(Cl)c(F)c1C(=O)NC1CCN(C(c2ccc(N)c(N)n2)=O)CC1F c1(C(=O)NCC2(O)CC(NC(C3COCCOC3)=O)C2)cc(F)ccc1O C1(COC)(NC(c2cccc(C3CCCOC3)c2)=O)CCN(C(C)=O)C1 C(C(C(C)C)OCC)N(C(CCN(CC=C)C(C1CCC1C(C)(C)C)=O)=O)C n1(CC(=O)NCC2CN(C(C(C)OCCC=C)=O)C2)cc(Br)ccc1=O c1(C(=O)NCC2C(NC(c3ccc(CCC)[nH]3)=O)C2)cnn(CC)c1C C1(NC(=O)COC2CCC2)CC2CCC(C1)N2C(c1cn2c(n1)SCC2)=O C1(CC)(NC(=O)CCc2cn(C)nc2C)CCCN(C(=O)C(C(C)C)N(C)C)C1 c1(-c2cnc(OC)c(C)c2)cccc2c(C(=O)Nc3ccc(C#N)nc3)[nH]nc12 N1(C(c2c(CC)occ2)=O)CCCN(C(=O)C(O)CSC)CC1CO CC1(C(=O)NCC2CC2NC(c2cc(Cl)c[nH]2)=O)CCC(F)(F)CC1 c1(CC(=O)NC2CC(NC(C(C)(C)n3cnnn3)=O)CC2O)c[nH]c(=N)nc1O c1(CC)cc(CC(N2CCCC2C(C)NC(=O)C(C)=C2CC2)=O)n(C)n1 c1(C(N2CC(N(C(CC(C)OC)=O)C)C3(C2)CC3)=O)[nH]c2ccccc2c1C#N n1(CC)c(O)nc2ccc(C(=O)N(C)Cc3cccc(C#N)c3)cc12 C1(CC(=O)OC)CCC(NC(=O)CN(C(=O)Cn2cc(C)cn2)CC2CC2)C1 C(=O)(C(CC(C)C)C(N)=O)NCC1=CCCN(C(CCc2ccc(C)o2)=O)C1 C(C(C)NC(c1cnc(C2CC2)[nH]1)=O)(C(C)C)NC(c1cnc(SC)s1)=O N1(C(c2nc(NC(=O)CCc3ncc[nH]3)sc2)=O)CCC2(CC1)CC(CO)C2 C(=O)(CCCCC(C)(C)C)N1CC(C)N(C(=O)C=CC(N2CCOCC2)=O)CC1 c1(CC)c(C(N2CC(CNC(=O)CSCCC#N)CC2C)=O)oc2ccccc12 C1(NC(=O)C=CCF)CC(F)CN(C(c2cncc(-n3cnnn3)c2)=O)C1 C1(NC(c2nnn(C)n2)=O)CC2CC1CN2C(=O)CCc1cn[nH]c1 c1(C(=O)NC(C)C(C)(C)NC(=O)C(O)C2CC2)cc(Cl)c(C(F)F)cc1F N1(C(Cc2ccn(C)n2)=O)CCC(CC(N)=O)(NC(c2cc(C#N)cs2)=O)CC1 c1(NS(CSCC(=O)NCC(=O)N(C)C)(=O)=O)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] N1(C(CCCC(C)(C)C)=O)CCCC(C2CC2NC(C2CC23CCSCC3)=O)C1 C1(C(=O)NCCCC(=O)NCCCOC=C)CCC(C)(C)C1 C1(N(C)C(c2ccnc(S)c2)=O)CCCC(CNC(=O)CCc2cncs2)C1 N1(C2CCCN(C(C(C)OCC3CC3)=O)C2)CCN(C(=O)CP(C)(C)=O)CC1=O N1(C(c2c(COC)cc[nH]2)=O)CCCC2(C1)CN(C(C1(C)CC=CCO1)=O)CCO2 O=S(=O)(c1ccc(NCC2=CCCOC2)c(Cl)c1)N1C2CCCC1CC1(CC1)C2 c1(N2CCC(Br)=C(C)C2)nc2c(c(=NCCS(=O)(=O)C(C)(C)C)[nH]1)CCC2 c1(CC)cscc1C(N1CCC(n2cc(C3CCOC3)nn2)C1)=O N1(CCCC(=O)NC(CC)CNC(C2CCS2(=O)=O)=O)C(=O)CN(C)C1=O c1(C(=O)NC2C(N=[N+]=[N-])CN(C(C3(F)CCC3)=O)C2)ccc2c(c1)C(=O)NCC2 CCC(CC(=O)N1CCOCC1CNC(c1cc2c[nH]nc2s1)=O)C(F)F Cc1nc(C(=O)NCCCCCCn2cc(CNC=O)nn2)sc1C N1(CCOC)CC(C(=O)NC2CN(C(c3cnns3)=O)CC2SC)CCC1=O N1(C(COCCCN=[N+]=[N-])=O)CCN(C(=O)CS(=O)(=O)c2cccs2)C(CO)C1 C1(N(C(C2C(CC)CCCN2C(=O)CC2(O)CCOC2)=O)C)CCCC(C)(C)C1 C1(NC(C(C2CCC2)OC)=O)CCC(NC(=O)CCc2ccccc2)C1 Cc1ncccc1CC(=O)NC1(c2cn(C3CC(F)(F)CO3)nn2)CCCOC1 c1(-c2cn(CC3CCN(C(CN(CCC)C)=O)C3)nn2)ccc(Cl)c(C)c1Cl C(C(C(=O)NCCCOCCO)NC(C)=O)OC.C1(=O)C(C)N1 C1(CNC(c2ncccc2F)=O)CCCC(NC(c2ccnn2CC2CC2)=O)C1 N1(CC)N=C(C(=O)N2CCC(NC(C3CN(CC(C)C)C3)=O)CC2C)CCC1=O CN1CCN(C(=O)Nc2ccc(Br)cc2I)c2cc(F)ccc21 C1(CNC(c2nc(Cl)c(Cl)s2)=O)CC2(C1)CN(C(C1CC1F)=O)C2 C12(NC(c3cccc(N4CCCNC4=O)c3)=O)CC1CN(C(c1cscn1)=O)C2 Cn1nc(O)cc1C(=O)NCC1(O)CN(C(C2(C(C)(F)F)CC2)=O)C1 N1(C(C(=O)NC(C2CCC(F)CC2)CC)=O)CCOCC(n2ccnc2C)C1 c1(C(=O)NC2CCC(NC(c3c(CC)ocn3)=O)C2)sc(C(F)(F)F)nc1C C1(NC(=O)CC2C=CCC2)CC(NC(c2cc(-c3ccccc3)no2)=O)CC1O C1(C(=O)NC2C(NC(=O)CCCF)CCC2)CCn2nnnc2C1 C1(NC(CCC=C)=O)CCC2CN(C(C3CC(CC)=NO3)=O)CCC2C1 C1(NC(CN(C(C)C)C)=O)CCN(C(C2CCOC(=O)N2)=O)C1C1CC1 N1(C(C(CCCC)F)=O)CCC2C(CCN2C(=O)CCC(C)SC)C1 c1(C(=O)NCCCCCCN(C)C(c2cnc(O)c(F)c2)=O)sc(C#N)cc1Cl C=C(C)CC(C(=O)NCCCCCCCC)NC(C1COC(=O)N1)=O CCCCCC(O)C(C)C(=O)N(C(c1ccccc1)C)Cc1occc1C C12(CNC(COCC#C)=O)CC1CN(C(=O)C(Cc1ccsc1)NC=O)C2 CC(F)(F)C(F)C(=O)NCC1(C(=O)NCCCCCO)CC12CCC2 N1(C(c2cnc(OC)nc2)=O)CCN(C(=O)CC2COCC2O)C(CC(F)F)C1 N1(C(c2ccc(CC)o2)=O)CCCC1C1CCCCN1C(=O)CCc1cnc[nH]1 c1(CC(N2C(C(C)NC(C3(C=C)CCC3)=O)CCC2)=O)n[nH]c2ccccc12 N1(C(c2cn(C)nc2C2CCCC2)=O)CC2CN(C(=O)C(O)C(F)(F)F)CCC12 Cc1cc(C(=O)NCC2(O)CCN(C(=O)CCC3CCCOC3)CC2)cc(C)c1 N1(C(C2N(C(C(CC)=CC)=O)CCC=C2)=O)CCC(F)(F)C(O)C1 C1(C(=O)NCCCCNC(c2cnc(OC)s2)=O)CCc2nc(C)[nH]c2C1 N#Cc1ccsc1C(N1CCCC(N2CCN(C(C3CC4(CC4)C3)=O)CC2)C1)=O C(=O)(N=S(C)(=O)C1CC(O)C1)C1(COC)CC(F)(F)C1 C12(NC(C(c3c(C)nn(C)c3)C)=O)CCCC1CN(C(=O)CC1OCCCO1)C2 C(=O)(CCC(F)(F)Cn1cc(C(C)(O)CC)nn1)NCC1C(CC=C)CCCC1 CCN=c1[nH]cc(C(=O)NC(C2CCOC2)CNC(=O)CNC(=O)CN(C)C)s1 CC(C)CCC(F)C(=O)NC(Cc1cc[nH]n1)C(=O)NOCC(=O)N(C)C c1(NC)ccc(F)cc1C(N1CCC12CN(C(=O)C=C(C)C)C2)=O C(C)(CNC(=O)CC1CCOC1C)(CNC(c1cc(C(C)(C)C)on1)=O)OC c1(OC)cc(C(=O)NCc2nc(CNC(C3(O)CC4(CCC4)C3)=O)cs2)c(F)cn1 c1(C(=O)NC(CC#C)(C)C(=O)N2CCN(C(=O)NC)CC2)ccn2cncc2c1 c1(C(=O)NCC(=O)NC2(CC(F)F)CCC2)ccc2c(c1)CNC2=O c1(CNC2CN(C(c3cccc(O)c3)=O)CC2F)ccc(Br)c(Cl)c1 N#CC1(C(N2CC3CC3(NC(=O)COc3ccccc3C(N)=O)C2)=O)CCCC1 c1(CCC)noc(CCCC(=O)NC(C)C(C)(C)NC(C2CC2CC)=O)n1 C(=O)(C1=CC2(CCOC2)C1)NCC(C(=O)NCC1(CC)CCCCO1)C(C)C c1(C(=O)NC(CC)C(=O)OC)ccc(NC(c2nc(C3CC3)cs2)=O)nc1 CCCC(CNC(c1cc(C)cc(Br)c1)=O)C(=O)NC(c1cc(C)ccc1C)C C(CCCCC(F)(F)F)SC.C1(CC)(CO)CCCN1 CC1ON=C(C(=O)NC2COCCC2NC(c2cccnc2S)=O)C1C C1(C(N2C(C(C)(C)C)CNC(=O)C2)=O)Cc2ccccc2C1=O Cc1ccc(F)cc1C(=O)NCC1CC(C)N(C(=O)Cc2cccc(C)c2O)C1 c1(C(N2C(CCCNC(c3nc(OC)c(C)s3)=O)CCC2)=O)ccc(C)cc1O C=CCC(CC(C)C)C(=O)N(CCCN(C(=O)C(C#N)(CC)CC)C)C CC1CN(C(c2scnc2C(F)F)=O)CCC1CNC(C12CSC(C1)C2)=O N1(C(CSCC#C)=O)CCN(C(=O)C(C)OCCNCC(F)(F)F)CC1CCO N1(C(COCC)=O)CCCN(C(=O)CCc2ccccc2C(F)(F)F)CCC1 C1(C(=O)NC2CCN(C(CC3OCC(C)(C)C3)=O)CC2F)CCN2CCOCC12 Cc1nc(O)nc(C)c1CC(N1CC(NC(c2ccc(F)cc2)=O)C2CC12)=O C1(CC(=O)NCC2C3CN(C(=O)C4=CCCC4)CC23)CCC12CCC2 c1(CC)ccccc1C(N1CCOCC1CCNC(=O)CC1CCCN(C)C1)=O c1(C(=O)NC(C(C)NC(C2C(CC)C2)=O)(C)C)ccc(C)nc1N c1(C(N2CCN(C(c3cc(C)n(C(C)C)n3)=O)CC2)=O)ncc(Br)cc1O c1(-c2c[nH]nn2)csc2nc(C)cn12.N1(CC)CCC(C(=O)N2CC(O)CO2)CC1C C1(C)(C(=O)NCC(CN(C(c2c(C(C)C)[nH]cc2)=O)C)C)CS(=O)(=O)C1 N1(C(C2CCCN(C(c3cc(CC)ncc3)=O)C2)=O)CCc2nc[nH]c2C1 C1(NC(C(C2CN(C(=O)CC3CCC(OC)CC3)C2)OC)=O)CS(=O)(=O)C1(C)C c1(C(=O)NC2C=CCN(C(Cc3cnc(C)s3)=O)C2)ccc2oc(S)nc2c1 Cc1cc(C(=O)NCC2CC3CCC2N3C(=O)CC(C)(C)C2CC2)nc(C)c1 C12(C(=O)NC3C(C)N(C(=O)CCCSc4ccccc4)CC3)CCCC1C2(F)F c1(C(C)(C)C)cc(CNCC(O)CO)ccc1O.C12(CCC1)CC(=O)N2 N1(C(C)(C)C)CCCOC(CCOC(N2CCCC2NC(=O)OC2CC2)=O)C1 CC(CCC(C)(C)C)NC(=O)CN1CCN(C(C2COCCN2C)=O)CC1 CCC(C)C(O)C(=O)N1CC(F)(CNC(=O)CCCCSC)C1 Cc1nc(Cl)c(C)c(=NCCC(C)NC(=O)CNC(=O)CC2CCCC2)[nH]1 N1(C(C(C(C)C)SC)=O)CCC2(CCN(C(c3sc(CO)nc3C)=O)CC2)C1 N1(C(C2C(c3cn(-c4c(OC)ccnc4)nn3)CCC2)=O)CCn2nccc21 C1(C(=O)NC2CC(NC(CSCC(N)=O)=O)C2)CCN(C2CCCCC2)C1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC(F)(C(=O)NC(CN(C)C)CCO)C1 CCCCC(O)C(C)C(=O)NC(CCC(=O)Nc1ccccc1F)C(C)C c1(C(=O)NC(CCNC(c2cnn(CCC)c2C)=O)C)cccc(O)c1[N+](=O)[O-] C=CCC(CNC(c1cnc(O)cc1C)=O)C(=O)N(C(C)CC(F)(F)F)C CN1CC(NC(=O)CC2(NC(C3CCC4(CC3)CC4)=O)CC2)CC12CCC2 N1(C(c2nc(=N)[nH]cc2)=O)CCc2nc(O)cc(C(N3CC(O)CC3CF)=O)c2C1 N1(C(c2c(CNC(COC3(C#C)COC3)=O)ccs2)=O)CCC2(CC1)CC2CO O(C1CCOc2ccc(OC)cc21)C(C1C(C(=O)OC)C=C1)=O n1(CC)nc(C(C)C)cc1C(=O)NCCCC(CO)NC(=O)CC(C)COC c1(C(=O)NC2CCCC(NC(C=CC=CC)=O)CC2)c(C)nc(C2CC2)nc1C CC1(C(N2CC(CCn3cc(C(C4CCOC4)C)nn3)C2)=O)COC(=O)C1 C1(NC(C(CSC)O)=O)CC1C1CCN(C(C2(C#N)CCOCC2)=O)CC1 C#CC(CNC(=O)C(C)C(C)NC(c1cc[nH]c1C(C)C)=O)C(C)C N1(C(CCCC#CC)=O)CCN(C(c2cc(CS(C)(=O)=O)on2)=O)CC(O)C1 Nc1cnc(Cl)c(C(N2CCN(C3CN(C(=O)CC4CC45CC5)C3)CC2)=O)c1 c1(NCC(CCCC)NC(C23CCCCC2C3)=O)c(F)cc([N+](=O)[O-])cc1F c1(C(=O)NCC(C)(C)OCCNC(C(CCC)OCC)=O)n[nH]c2c1CCC2 C1(NC(COCC)=O)CS(=O)(=O)C12CCN(C(c1ccccc1SC)=O)CC2 Cc1cc(O)c(C(C)C)cc1C(=O)N(CC(C)NC(=O)COCCCC(C)C)C C(C)(C(C)C(=O)NC1CCC(CCO)CC1)NC(CCCOC(C)=O)=O Cc1n[nH]c(=NC(C)C2CN(C(=O)CCCc3cnn[nH]3)CCO2)s1 Cc1ccc(C=CC(=O)NC2CC(NC(c3cc(N)ccc3F)=O)C2)c(C)c1 c1(C(=O)Nc2c(C(=O)OC)ccc(Br)n2)cc2ccccc2c(Cl)n1 c1(NC(C2C(C(C)=O)CC2)=O)ccc(C(=O)NCC23CCCCC2C3)cc1C c1(N(C(=O)C(C)Sc2nncs2)CCCC)cn(C2CC(O)C2)nn1 Cc1cccc(OCC(=O)NC(C)C(C(C)C)NC(=O)COc2ccsn2)c1 c1(OC)nc(Cl)cnc1NC(=O)Cc1csc(NC(C2CC2C(=O)C2CC2)=O)n1 c1(CNS(NCCC(=O)N(c2ccccc2)CC)(=O)=O)c(F)cc(Br)c(Br)c1F CC1(O)CCC(C(=O)NCC2CN(Cc3ccc(C#N)s3)CCO2)CC1 N1(C(c2cc(C)c(O)c(N)c2)=O)CC(NC(C2CC2C)=O)CC2(CCOCC2)C1 N1(C(C2C(COC)CC2)=O)CCC(C)C(CNC(c2occc2COC)=O)C1 c1(N(C2CCC(CCC)CC2)C)nc(=NC2CSCC2SC)[nH]c2cccnc12 c1(OC)ccc(C(=O)NCC23CC(C(=O)O)(CCO2)C3)c(N)c1 C1(CNC(Cc2nc(=N)[nH][nH]2)=O)CN(C(c2ncccc2Cl)=O)CCCO1 C1(C)(c2ccc(OC)cc2)NC(=O)N(C(C#N)CSc2ccc(C)cc2)C1=O C1(C)(CNC(C(C)CO)=O)CCCN(C(=O)CCc2ccccc2C(F)(F)F)C1 C1(CC(=O)NCC(CCCC)NC(=O)C=C2CCCCC2)CCC2(CC1)CC2 CCC(N=c1nc(N(C)Cc2cn(C)nn2)c2cccc(F)c2[nH]1)C1CC1 c1(C(=O)NCCC(CNC(c2sccc2CO)=O)OC)ccc(C)cn1 C1(CNC(=O)CC(=O)Nc2nccs2)CN(C(C2CCCC2)=O)C2CC12 N1(C(=O)OC(C)(C)C)CCN(C(=O)N(C2CC2)Cc2cccs2)C(CC#N)C1 c1(OC)cc(F)c(F)cc1CNC12CCC(C(=O)Nc3ccsc3)(CC1)CC2 c1(C(=O)NC2CC3CN(C(C(C=C=C)C)=O)C2C3)cnc2c(c1)CCCO2 Cc1oc2ncc(C(=O)NC3(CNC(C4(CN(C)C)CC4)=O)CC3)cc2c1C N1(C(C(C)(C2CC2)OC)=O)CCCCC(CNC(=O)Cc2ccc(O)c(F)c2)C1 C1(C(=O)OC)(COC)CN(C(=O)C(c2ccccc2)NC(=O)C=C2CCC2)C1 c1(CC)nc(=NC(=O)N2CCCC2c2cc(OC)c(OC)cc2OC)[nH]n1C N1(C(CCn2ccc(C)n2)=O)CCC(NC(c2ccnnc2S)=O)C(O)C1 C1(C(N(CCC(=O)NC(c2csnn2)C)CC#C)=O)CCC(C)=C(C)C1 CC1CCN(S(=O)(=O)CC(=O)NCC2(CCNC(c3ccc[nH]3)=O)CC2)CC1 N1(C(c2c(C)noc2)=O)CCCC2(CC(NC(c3sc(C4CC4)nc3C)=O)C2)C1 S(=O)(=O)(c1cccs1)NCC(=O)NC1CN(C(CN(CCOC)C)=O)C2C1C2 Cc1ncc(Br)c(C(N2CCC(NC(=O)CC3CCCOC3)C2(C)C)=O)n1 c1(OC)cccc2c1C(C(=O)NC1CCCN(C(c3[nH]ncc3C#N)=O)C1)CC2 C1(C(C(=O)NC(c2cncnc2)C)F)CCN(C(c2nc(Cl)cs2)=O)C1 c1(C(=O)NC2C=CCN(C(C3(C#N)CC(=O)C3)=O)C2)ccn2nncc2c1 c1(C(=O)NC(CC(C)NC(c2c(C)cccc2F)=O)C)ncccc1S(C)(=O)=O C=C(C)CCC(=O)N1CCC(NCc2ccc(Oc3cc(C)ccn3)cc2)CC1 C1(NC(c2cn(C(C)(C)C)nn2)=O)CC2CC(C1)N(C(c1cc[n+]([O-])cc1)=O)C2 c1(N(C(CNC(CC(n2ccc(C)n2)C)=O)C)C)c([N+](=O)[O-])c(C)nn1C(C)C CCCC(O)CC(=O)NC(C1CCN(C(=O)CC2CSCCS2)CC1)(C)C Cc1cc(Br)ccc1CC(N1CCC(NC(C2CCOC(=O)CC2)=O)C1)=O N#CC1(NC(c2cc3c(s2)CSC3)=O)CCN(C(=O)CC2CCCCO2)C1 N1(C(C(CCC)C)=O)CC(C2CN(C(c3cnn(C=O)c3)=O)C2)C1.C(C)(C)(C)O C(C1CCCN1C(c1ccc(=N)[nH]c1)=O)=CC(=O)NCC1(N(C)C)CCC1 c1(C2CC(Nc3cc(N4C(CC)CCCC4)ncn3)C2)nnc2c(Cl)cccn12 C(=O)(C#CC1CCOC1)NCCC1N(C(c2c(C(C)(C)C)cccc2)=O)CCC1 C=Cn1nccc1C(=O)NCc1ncc(C(=O)N(CC(C)O)C(C)C)cn1 CC(O)(Cc1ccccc1)C(=O)NCCN(C(=O)CSC1CCCOC1)C1CC1 c1(NC2C(CC)CN(C(C3CCCN(C(N)=O)C3)=O)CC2)nc(C)nc(C)c1F C(=O)(C(C)(COC)OC)NC(CN(C(c1nc(CCCCC)sc1)=O)C)CC C(=O)(CC1=Cc2ccccc2C1)NCC1(CNC(CC2CCC(C)(C)O2)=O)CC1 c1(C(=O)NCC2(NC(C(CCCC)F)=O)CCOC2)cc(C#N)ccc1C C1(NC(N2CC(c3ccccc3)C2)=O)CC(=O)N(c2ccccc2)C1 C12(C(=O)NC3C(CC(=O)N(CCN=[N+]=[N-])CC)CCC3)CCC(CC1)CC2 c1(C(=O)NC(CCCC)CO)c(-c2ccnc(OC(C)C)c2OC)cncc1F c1(C(N(CC(C(C)C)OC)C)=O)ccc(F)c(SC)c1 C(C)(c1ccc(F)cc1F)=CC(=O)N(CC(CNC(CCCCC=C)=O)O)C C12(NC(COCc3cc(C)on3)=O)CCN(C(C3(C#N)CC3)=O)CC1C2 C1(NC(C(C)CNCCC(=O)O)=O)CS(=O)(=O)C12CCOCC2 c1(C(=O)NCC2CCN(C(Cc3cc(C)[nH]n3)=O)C2)cc(F)ccc1Br N1(C(Cc2n[nH]c(=N)s2)=O)CCN(C(=O)C=CCO)CC1c1cccnc1 C(=O)(C1CCc2c[nH]nc21)N1CC(NC(c2cnc(-c3cccs3)s2)=O)(CO)C1 C(CS(=O)(=O)CC(=O)NC(C1CN(C(C2(C)CCC(=O)C2)=O)CCO1)C)OC c1(CC(=O)N(C2CCN(C(=O)CCc3cncnc3)C2)C)ccc(O)nc1 C1(C(C)NC(=O)CCF)CN(C(C2CCN(c3ccncc3)C2)=O)CCO1 C1(C)(CC)CC(NC(=O)CC2CCCCC2NC(c2cc(C)nn2C)=O)CCO1 c1(C(=O)NC(CCC(=O)OC(C)C(C)Cc2ccccc2)=O)cccc(O)c1F N1(C(c2cc(C)cc(C)n2)=O)Cc2ccccc2CC1CNC(c1cocn1)=O C1(C(N(CCCN(C)C)CC)=O)COCCC1NC(=O)CC1C=NN(C)C1=O c1(COC)cc(C(=O)NCCCCNC(=O)CC2C(C)C2(F)F)n[nH]1 C#CCC(C)(CC)C(=O)NCc1nc(C2CCN(C(=O)C(C)CSC)CC2)n[nH]1 CC(C)P(=O)(CC(=O)N1CCC1CNC(=O)C(C)(C)CC#N)C(C)C C1(Nc2ccc(OC)c(C(F)(F)F)c2)CCC2CN(C(=O)OC)CCC2C1 c1(C(=O)NC(C(C(C)C)NC(=O)C2=CC(C)(C)C2)C)cnc2[nH]cncc1-2 c1(C(N2CCCCC2)=O)nc(-c2cncc(F)c2)n(-c2ccc(F)nc2)n1 N1(C(C2N(CC)CCC2)=O)CCCC(NC(C2(c3ccccc3)CCCC2)=O)C1 c1(C(N2C3CN(C(C4C5COCC45)=O)CC2C3)=O)ccnc2c1OCO2 c1(C(=O)NC(C2CCCN(C(=O)COCC(F)F)C2)C)cc2c(ncn2C)s1 c1(C2C(C(=O)NC3CC(N(C(CC(=O)NCC#C)=O)C)C3)C2)ccccc1Cl N1(C(C2C(CC)C2)=O)CCC(C)(C)C(CNC(C2(C3CCC3)CC2)=O)C1 C1(CNC(C2OCCN(C(C)=O)C2)=O)CN(C(c2cnsc2)=O)CC12CCC2 N1(C(c2c(NCC)scn2)=O)CCCC(C)(CNC(=O)C(C)CC(N)=O)C1 N1(C(c2nnn(C)c2N)=O)CC(NC(C2CC(CC3CC3)C2)=O)CC2(CCC2)C1 CC1C(NC(=O)C(c2ccc(Cl)cc2)C)CCN1C(C1(C#N)CC=CC1)=O C1(C2CCCN(C(=O)C3=CCCC3C)C2)(NC(CC=C(C)C)=O)CC1 C1(C(=O)NC2CCC(NC(C3CC(SC)C3)=O)C2)COCCN1C c1(CC)c(OC)cccc1C(=O)NCC1CCCCN(C(=O)COC(C)(C)C)C1 C(C(C(C)(C)C)NC(c1cccnc1N)=O)NC(C1N(CCC)CCC1)=O CCCS(=O)(=O)CC(=O)N1CC(NC(c2csc(COC)n2)=O)CCC1C n1(CC(C)C(=O)NCC2(O)CCC(C)(C)C2)ccc2ccccc12 C1(CN2CC(CNC(CC=C)=O)(CO)C2)CCSC1(C)C c1(C(N(CC(C)C)Cc2ccc(Br)o2)=O)coc2c1CN(C(=O)OC(C)(C)C)C2 N1(C(C(COC)OC)=O)CCC(CNC(c2c(OC)noc2C)=O)C(C)C1 C(CC(C)C)(C(=O)NCCCC1CCCC1)NC(c1c(CC)ccs1)=O c1(C(=O)NCC(CCNC(c2c(C)nn[nH]2)=O)O)c[nH]cc(C)c1=O Cc1cc(=O)n(C)nc1C(=O)NCCN(CC(C)O)C(c1ccc(COC)o1)=O N1(C(Cc2onc(C)n2)=O)CC(NC(=O)Nc2ccc(F)c(F)c2)CC(F)C1 C1(C(N2C(CNC(c3c(C)coc3)=O)CCC2)=O)CCN(CC(C)C)CC1 C(=O)(CCC(F)(F)Cn1cc(CCC(C)(C)C(N)=O)nn1)NC(c1nncs1)C c1(C(C(C)OC(C2(Br)CC23CCC3)=O)=O)ccc2c(c1)CCC2 C1(C(=O)NCC2(F)CCN(C(C3C(OC)CCC3)=O)CC2)Cc2cc(F)ccc2O1 S(=O)(=O)(c1ccc(NC(c2cc(Br)ccn2)C)cc1Br)NC(CC)(C)C CCN=c1ccc(C(=O)NC2CCC(NC(C3CN(C)CC(C)O3)=O)CC2)c[nH]1 CC(C)C(F)C(=O)N(CCNC(c1coc(C(N)=O)c1)=O)CCOCCO c1(CN=C(NCC2N(C)CCC2)NCC2CCC2)csc(S(N)(=O)=O)c1 C1(O)(C(N(CC(C)NC(C(CC=C)C)=O)C)=O)CCCC(C)CC1 N1(C(CCC(C)OCC)=O)CCN(C(=O)CC(c2ccccc2OC)C)CC1C Cc1ccc(Cl)c(F)c1C(=O)NCC12CC(C1)C(NC(=O)C=CCO)CO2 CC(CCCCNC(C1(F)CC=CC1)=O)NC(=O)COc1cncc(Cl)n1 CC1CCN(C(=O)C=CC2CCCN2C)C1C(=O)NC1CCN(C(N)=O)C1 N1(C(C)C)CC(C(=O)NC2(CO)CN(c3ccc(C#N)nc3)C2)CCC1=O C1(NC(C=CCOC)=O)CN(C(=O)COCc2ncnn2C)C(C)(COC)C1 N1(C(C(=CC2CCCC2)C)=O)CCC(O)(C(C)NC(=O)CC(=O)NC2CC2)C1 C(=O)(C(S(C)(=O)=O)C1CC1)NCCCC1N(C(C(C)=C2CCCC2)=O)CCC1 C1(NC(C2C(C)CC2)=O)C(C(=O)NCCc2cnn(C)c2)C1(C)C c1(CC(=O)NCCOC2CN(C(CCOCC#C)=O)C2)c(C)ncnc1C.OCC C(CCCC(=O)NC1CCOCC1NC(C12CCCC(CO1)C2)=O)(OC)OC c1(C(=O)OC)cccc(CNC(N2CCCC(CC(=O)OC(C)C)C2)=O)n1 C(CN=c1cc(CC2CC2)nc[nH]1)(C1CCCOC1)NC(C1(CO)CC1)=O c1(C(=O)NCCC2CCCN(C(=O)C(F)(F)CF)C2)cccc2c1CCO2 C1(NC(CC2C=NN(C)C2=O)=O)CC2(CCCCN2C(C2CCC2)=O)C1 N1(C(C(C)(C)OC)=O)CCCC(C2CN(Cc3ccc(F)c(Br)c3)C2)C1 C(=O)(C1=C(Cl)CCCC1)NC1C(NC(Cc2scc(C(C)=O)c2)=O)COC1 C1(C(=O)NCC2N(C(c3n[nH]c(C)c3C)=O)CCOC2)C2CCC3C(C2)CC13 c1(OC)ccc2ccc(C(=O)NC3CN(C(C4CC4(C)Br)=O)C3)cc2c1 c1(C(=O)NC(CNC(C2C(C(C)C)C2)=O)(C)CO)cc(O)cnc1Cl C1(CC)CN(C(=O)C(C)(C)C(F)F)CCN1C(c1cc(C(C)(C)C)[nH]c1C)=O C1(CNC(N(CCn2ccc(=O)cc2)CC)=O)CNC(=O)CC12CCC2 N1(c2nc(N(C)CC3CCCC3O)cc(C)n2)CCC2(CCC(=O)N(C)C2)CC1 N1(C(CNC(=O)OCC=C)=O)CC(NC(c2ccc(=O)n(CC)c2)=O)C12CCC2 C(CC(=O)NCC(F)CO)(C(F)F)NC(C(C)OCCCC=C)=O C1(NC(c2[nH]nnc2-c2ccccc2)=O)CCCN(C(=O)CC2CC3CC3C2)C1 N1(C(C(C)Sc2ccccn2)=O)CCC(N=c2nc(N(C)C)[nH][nH]2)C(C)C1 C1(CNC(C2(NC(C)=O)CCC2)=O)CCN(C(C2CCCC2C(F)F)=O)C1 CCC(C)(C)C(O)C(=O)NC1CC(NC(c2coc(C3CCOCC3)n2)=O)C1 c1(OC)ccccc1C(C)N(C(C)C(N1CCC(C(=O)OC)C1)=O)C c1(C(N(CCNC(C2(C)CC=CCO2)=O)CC)=O)cc(F)c(Br)cc1OC CC(C(CO)NC(=O)C(O)COCc1ccccc1)NC(=O)CN1CCOC1=O C1(C(=O)NC2(C3CN(C(=O)C4=CCSC4)C3)CC2)CCCC2(CCCCC2)C1 Cc1cncc(C(=O)NC2CC3CC(NC(c4cc[nH]n4)=O)C2C3)c1C CN1CCCC(CCc2cn(CCC(=O)NC3CSCN3C)nn2)C1 c1(CC(=O)OC)cccc2c1OCCN(S(=O)(=O)CC1(C#N)CCOCC1)C2 C(C(N=c1[nH]nc(-c2ccc(Br)cc2)o1)C(C)C)NC(CCNC(C)=O)=O CC1Cn2nccc2CN1C(c1ccc(CNC(C2CC2(F)Cl)=O)cc1)=O CCC(O)C(C)C(=O)NCC1(O)CCN(C(C2(C)CCN(C)C2=O)=O)C1 c1(CC)ccccc1N(C(=O)C(C)CCSC)CCc1cn(C(=O)NCCO)nn1 N1(C(c2ccc(C(C)C)nc2)=O)CCCC2CN(C(=O)CN(C)C(C)C)CC12 n1(CC(=O)NCCN(C(=O)CCN2CCOCC2)CC)nc(Cl)ccc1=O c1(NCC(C)(C2CC2)NC(C=CCC)=O)nc2ccccc2cc1[N+](=O)[O-].SCC c1(OC)c(C(=O)NCCC2(CNC(C3COC(C)C3)=O)CC2)cc(Cl)cc1C N1(C(C(C)c2ccsc2)=O)CCN(C(C2(F)CCCC2)=O)CC1C1CCC1 Cc1ccc(O)c(C(=O)NCCCC(O)C(=O)N2C(CO)CC2C)c1 C1(C(N(C2CN(C(C=CC(=O)N(C)C)=O)C2)C)=O)C(C(F)(F)F)C1[N+](=O)[O-] C1(C(=O)NC2CCCCC2NC(=O)C2CC2)Cc2ccncc2C1 C1(N(C)C(c2ncccc2C2CC2)=O)CCN(C(=O)CNC(N)=O)C12CC2 C1(CC2(NC(N(CCOC)C)=O)CC2)CCC2C(CC1)C2(F)F c1(CN=C(NCCCO)NCC(C2CC2)C2CC2)c(Cl)oc2ccccc12.C1(N)CC1 c1(C(=O)NC2CN(C(CCS(=O)(=O)NC)=O)CC(O)C2)ccc2ccn(C)c2c1 C(=O)(CCCCCCCCCC)N1CCC(CC=C)(NC(C2CC2(C)Br)=O)C1 CN1CCN(C(C2CCC(=O)O2)=O)C(CNC(=O)C=C2CCN(C)CC2)C1 c1(C(=O)NCC2CN(C(C(C(C)C)c3ccncc3)=O)C2)cc2c(s1)CCCC2 CC(C)CC(C(=O)NCCCC1CCCCO1)ONC(c1ccc(O)cc1)=O Cc1cccc2cc(C(=O)NC3CN(c4ncc(Cl)c(O)n4)CC3(C)C)oc12 N1(C(c2ccc(Cl)cn2)C(=O)NC(C)(C)C)CCCc2oc(Br)cc2C1 N1(C(c2n(C)c(S)nc2)=O)CCN(C(=O)CN2CCCOC2=O)CC1CC1CC1 c1(NC(C2CN(Cc3cnco3)CCC2O)=O)nccc(Br)c1Cl c1(C(=O)NC(C2OCCN(C(c3c(CC)ncs3)=O)C2)C)cc(F)c(F)cc1F c1(C(=O)NCCNC(c2ccc(N(C(C)C)CCO)cc2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC2C(C(N(C3(C)CC3)CC)=O)CCO2)cc(=O)cc[nH]1 c1(C(N(C2COCC2O)CC)=O)cn2c(n1)CCN(C(=O)C(C)(C)CSC)CC2 c1(CSC)noc(CNC(=O)C(C)N(C(=O)CCCN2CCCC2)C)n1 CC1CCC(NC(=O)CN2CSCCSC2)CN1C(C1(C2CCC2)CC1)=O C1(NC2(COC)CCOC2)CCOCC1C(=O)NCCC(=O)NC(C)(C)C N1(C(C(COC)C)=O)CC2CC(C1)N(C(=O)CCc1cc(Cl)sc1Cl)C2 CC(C)C(C(=O)N=c1cc(CS(C)(=O)=O)o[nH]1)Nc1ccc(C#N)cc1 N1(C(CC(COC)C)=O)CCC2(CC2C(=O)NC2CC(CN(C)C)C2)C1 CCC(F)(F)CC(=O)N1CC(O)CC1CNC(c1ccc(C(C)C)s1)=O C1(NC(CNC(C(CC)C)=O)=O)CCC(C)N(C(c2cc3c(s2)CCC3)=O)C1 N1(C(c2cc(OC)n(C)n2)=O)CCC(NC(=O)C=Cc2ccc[nH]2)C(C)C1 c1(C(N2CCC(C(C)(C)NC(C34COC(N3)CO4)=O)C2)=O)ccc(OC)c(O)c1 CCCCCCC(C)CC(=O)N1CCC(C(C)NC(c2ccc(F)cc2N)=O)C1 c1(C(=O)NC(C(C)NC(=O)CCC2CCC2)CO)ccc(C#N)cn1 C1(C(N(CCC#N)C(C)C)=O)CCCN(c2nc(-c3ccccc3)cs2)C1 C1(C(=O)NC(c2cnc(C)s2)CC)C2CC2CN1C(c1cncc(OC)c1)=O C1(CC(=O)N(CCNC(=O)CC2CC3CC3C2)CC2CC2)(OC)CCCC1 c1(NC(C)=O)ccccc1CCC(N1CCC2C(NC(c3cnc(Cl)s3)=O)C12)=O N1(C(CC2CC(=C)C2)=O)CCC(CNC(C2CCCN2C2CC2)=O)C1(C)C c1(NCCC2(C)CCOCC2)nccc(=NCC2(c3ccccc3)CCCO2)[nH]1 c1(C2(C(=O)NCCCNC(=O)C(F)Cc3ccccc3)CCC2)ccc(Cl)cc1 N1(C(C(C)CC2CC2)=O)CC2(COC(CNC(=O)CCn3cncn3)C2)C1 c1(NC2CCN(C(c3nc(NC(C)=O)sc3)=O)C2)c([N+](=O)[O-])ccc(F)c1C N1(C(C2(C)CC2)=O)CCC2(C=C(C(=O)NC3COCC3F)C2)C1 N1(Cc2ncc(C)o2)CCN(c2cc(NCCCc3ccc(C)s3)ncn2)CC1 C(C)(CC(C)N=c1[nH]nc(C)s1)NC(CCc1cncc(C)c1)=O C(C1CCC(C)CC1)=C(C)C(=O)NC1CCC1NC(=O)Cc1coc(C)n1 C1(C)(C(=O)NCC(CC)NC(=O)CNS(=O)(=O)NC)CCC(=O)NC1 C1(CN(C(=O)C(C)(C)CF)C)COCCN1C(c1[nH]nnc1-c1ccnn1C)=O N1(CC(=O)NC(C(C)NC(CCCCC)=O)CO)CCc2sccc2C1 Cc1nc2cc(Cl)ccc2cc1C(=O)NCCCNC(=O)C=C1CCC(C)CC1 CC(N=c1nc(N2CC3C(C2)C3(C)C)c2c([nH]1)CCC2)c1ccncc1Br N1(C(CSCCC)=O)CCC(NC(C2(Cl)CCCCC2)=O)C(OC)C1 C#Cc1ccc(N(C(=O)COC(=O)CNc2cccc(F)c2F)C)cc1 c1(-c2cc(OC)c(F)cc2)ccc2nnc(C(N3CCCC(C)(O)CC3)=O)n2c1 C1(O)(C(N2CC(NC(C3N(CC)CCC3)=O)(CO)C2)=O)CCC(C)(C)CC1 Cc1cc(C#N)cc(C(N2CCCC(N(C(=O)CN3CCNC(=O)C3)C)C2)=O)n1 CC1(C)CC(O)(CN2CCOC(C(=O)OCC(C3COCCO3)=O)C2)CO1 C(=O)(NNC(=O)Nc1nnnn1C)NCCC(C)F CC(C(=O)NC1CCCCC1NC(=O)C(N1CCNC1=O)C)C(F)(F)C(F)F c1(C(=O)NCc2c(C)ncs2)ccc2occc2c1 C(=O)(C(O)CC(C)C)N(CCN1CCCCC1)CC.C12CCC(CC1)C(=O)N2 C12(NC(C3CCN(C(C45C(=O)C6CC4C5C6)=O)C34CC4)=O)CCCN(CC1)C2 c1(C(=O)NC(CNC(C2OCCN(C(C)=O)C2)=O)C2CC2)cc(N)c(C)c(N)c1 c1(OCC)ncc(C(=O)NC2CCN(C(=O)Cc3c(O)ncnc3O)C2)cc1Cl C1(C(=O)NC2(CNC(C3(CC(C)=O)CC3)=O)CCCC2)NC(=O)OC1C C(=O)(C(=O)N=S(C)(C)=O)NCC1CC(Cc2cn(CC3(C)CCCC3)nn2)C1 Cc1cc(C(=O)NC2CC(NC(C3CS(=O)(=O)C3)=O)CC2O)cnc1O C1(CNC(C2(OC)CCC2)=O)CN(C(=O)COc2ccsn2)CCC1(F)F CCCC(CC)CCC(=O)N1CC(NC(c2cnc(N)c(Br)c2)=O)CC1(C)C N1(C(C(CC#C)C)=O)CC2CCCC2(NC(c2cnn(CCF)c2)=O)C1 O=C1CCC(CCNC(c2cccc(-c3ccc(O)nc3)c2)=O)C(=O)N1 c1(C(=O)NCC(C(=O)NCC(C(=O)NC)O)(C)C)c(C)cccc1O C(c1cccs1)=C(C)C(=O)NC1CC1CNC(=O)CC(C)F CC1(C)OC(C)(C)c2nc(N(CCOCF)C3CC3)c(C#N)cc21 c1(C(N2CC(OCCOC(CCC3(C)CC3)=O)C2)=O)c(F)cncc1F c1(C(N)=O)cc(C(=O)NCC(O)CNC(=O)CN2CCCS2(=O)=O)cc(F)c1 C1(NC(c2cnc(CC(C)C)s2)=O)CC2CC(C1)N(C(=O)CCS(C)(=O)=O)C2 CS(=O)c1ccccc1-c1cnc(C(=O)Nc2ccnc(C#N)c2)nc1 N1(C(c2cnc(CC)[nH]2)=O)C2CCC1C(CNC(C1(C(F)F)CCCCC1)=O)C2 C1(CC#C)(C(N2CCC(C)(CCNC(C34CSCC3C4)=O)C2)=O)CC=CCC1 C1(c2n(CC=C)nnn2)(NC2CC2c2cnn(C)c2C)CCOCC1OC C(=O)(CC(O)CC(C)(C)C)NC1COCCN(C(c2c(OC)nccn2)=O)C1 C1(C(=O)NC(C)CNC(C2CCCO2)=O)CCCC2(CC2)C1 N1(C(CC2C(C)C2)=O)CCCC(NC(C2(F)CC2c2ccccc2)=O)C1 c1(NC(C(n2c(C)cc(C)n2)C)=O)cc(C#N)ccc1Cn1cncn1 c1(CC(=O)N(CCN(CC(CN(C)C)O)C)C)nc2ccccc2s1 N(C(=NCCC(C)(C)O)NC1CCN(C(=O)NC2CCC2)CC1)CC(C)C1CC1 N1(C(=O)NC(CC)CCCO)CCCC(C(=O)NCCNC(c2cnn[nH]2)=O)CC1 c1(CN(C(C2C(=C)C2)=O)CCNC(=O)C(O)Cc2cnc[nH]2)cccc(Cl)c1 CC(F)(CC1CCCC1)C(=O)NC1CC(NC(c2ccccc2O)=O)C1 CC1(C)CNC1=O.C(CCCCCC1CC1)NC(=O)Cc1csc(Br)c1 CC1CC(C#N)(C(=O)NCC(C)NC(c2ncsc2C2CC2)=O)C1 C(=O)(N1CCC(C(=O)NC2CCCCN(C)C2)O1)c1n(CC)nc(C)c1 C1(NC(C(=O)N(C)C)=O)C2CC3CN(C(=O)CN4CC(=O)NC4=O)C1C3C2 C1(=C(C(=O)N(C(C(N2CC(CC(=O)OC)C2)=O)C)C2CC2)F)CCCCC1 c1(N2CC(CC)NC(=O)C2)nc(NC2CC3C(C2)C3(F)F)nc2c1COCC2 c1(C(=O)NC2CC3(C(NC(C(CC)C(F)(F)F)=O)C3)C2)cncc2ncn(C)c12 C1(NC(c2ccsc2Cl)=O)CCCC12CCN(C(=O)CSCc1ncc[nH]1)C2 N1(C(CC2(C=C)CC2)=O)CCCN(C(c2ncc(N)nc2C)=O)C(CO)C1 c1(NC(C2CCC(NS(=O)(=O)CCCl)C2)=O)cccc(N2CCCCC2)c1 C=CC(CCC)CC(=O)N1CCCC(CCNC(=O)CNC(C)=O)CC1 C(CN=c1c(Br)c[nH]cc1[N+](=O)[O-])n1cc(C(=O)NC(C=C)C(=O)O)nn1 c1(C(N2CC(CNC(C(C)SCCCC)=O)N(C)CC2)=O)ccn2ncccc12 C12(NC(c3ncc(Br)cc3F)=O)CCCC1N(C(=O)C=CC1CC1)CCC2 c1(C(=O)NCC2C(CNC(CS(C)(=O)=O)=O)C2)n[nH]c2nccc(Cl)c12 C=CCC(CC(C)C)C(=O)NCC(O)CNC(=O)CCOCC(F)(F)F C1(C(=O)NC2CC(NC(c3cccc(CF)c3)=O)C2)CCn2nncc2C1 C(=O)(C(C)CC(C)C(C)=O)N1CCC(CC=C)(NC(=O)CSC2CCC2)C1 n1(CCN(C=O)OC)cc(NC(=O)NC2CC2)c(N2CCC(C(=O)OC)C2)c1.C(C)C N1(CC(c2ccccc2)NC(C)CC2CCC2)CCCC1=O N1(C(CNC(CCC)=O)=O)CCCC(NC(c2cncc([N+](=O)[O-])c2)=O)C(F)C1 C1(C)(CC)CCC(C(N2CCC(CCNC(C3CC(C(F)(F)F)C3)=O)CC2)=O)O1 N1(Cc2oc(C)c(Br)c2)CCC2CN(C(C3CCN(C)CC3)=O)CCC12 c1(CC)ccc(F)c(C(=O)NCC2CCCCCN2C(=O)C(=O)NCC(F)F)c1 N1(C(C2CC(N3CC(O)C3)C2)=O)CCCC(CCCCNC(c2ccon2)=O)C1 C#CC1CN(C(c2ccccc2SC)C(=O)NCC(C)C)CCO1 c1(C(N2CC3N(C(CC(C)SC)=O)C(CC3)C2)=O)cnc2c(F)c(F)ccc2c1 Cc1cnc(NCC(CO)N(C)C)c(S(=O)(=O)N)c1.C1(N)CCCCC1(C)C c1(C(=O)OC)ccccc1C(N1CC(C)(NC(C2NC(=O)CC2C)=O)C1)=O c1(C(=O)NC2CCCN(C(CCC=CCC=C)=O)CC2)cccc2ccsc12 N1(C(c2c(C)ccnc2)=O)CCCC(O)(CNC(=O)C(F)c2ccco2)C1 c1(CCNC(COCCC=C)=O)n[nH]cc1C(=O)NC(C)CCN(C)C C1(NC(=O)CC2ON=C(CC)C2)CC2CC1CN2C(C1CCCC(=O)N1)=O N1(C(CN(CC(C)C)C(c2cccc(CO)n2)=O)=O)CC2(CCC2O)C1 C1(F)(C(=O)NC(c2ccc(Cl)cc2)C(N)=O)CCCN(C(=O)CNC(N)=O)C1 c1(C(=O)NCCC2CCN(C(C(COC)(F)F)=O)C2)n[nH]c2c1CC1CC21 C1(C(C)C)CC(C(=O)NC(C2CCCN2C(C2CC23CC(O)C3)=O)(C)C)CCO1 N1(C(CCCCC)=O)CCN(C(c2cnc(C)s2)=O)C(c2ccccc2OC)C1 c1(CNC(c2cccc(C)c2N)=O)ccc2c(c1)CCC2NC(C12CCC1C2)=O C12(CC(N3CCC(C4CCCCN4c4nnc(O)s4)C3)=O)COC(CF)(C1)C2 CC(C)CCC(=O)N(C(=O)CSS(C)(=O)=O)C.C12CCC(C1)NC(=O)C2 c1(N2CCC(CCC)C2)nc2cccc(F)c2c(=NCC(C)c2ncc(C)s2)[nH]1 N1(C(C(C)n2cccn2)=O)CCC(C)(NC(=O)C=CC2CCCN2C)CC1 C1(NC(C(c2cn(C)nn2)N(C(CC)CC)C)=O)CC12CCOCC2 Cc1onc(Cl)c1C(N1CCN(C2CCN(C(=O)CCCCCl)C2)CC1)=O c1(NC(C)=O)ccc(Cl)c(C(N2CCN(C(c3cc(Cl)ncn3)=O)C3CC23)=O)c1 C1(C)(C(=O)NCC(C)CNC(c2ncc(C(F)(F)F)cc2N)=O)CCC(F)(F)C1 Cc1cc(CNC2CCC(NC(c3ccc(C#N)cc3)=O)C2)ccc1Cl N1(C(C2CC(C)(C)C(=O)NC2)=O)CCN(C(=O)Cc2ncc(Cl)s2)C2(CCC2)C1 Cc1nc(CC(=O)NC(C)CCCCNC(=O)COCCO)c(C)s1 c1(C(=O)NC2CC3(C2)CC(C(=O)Nc2cccnc2F)C3)cn2ccccc2n1 C12C(C)CCCN1C(=O)COC2=O.CCCC(C)(CC)NC(=O)OC(C)(C)C c1(C(=O)NCC(C2CCCCC2)NC(=O)CC2(C(F)(F)F)CC2)ncncc1Cl c1(C(N(C2CCC(NC(=O)C=Cc3cnccn3)C2)C)=O)nc2cnccc2s1 N1(C(C2(NC(=O)Cc3ccccn3)CCC2)=O)CCSC2CCCC12 N1(C(CCC=C)=O)CCC(C2CCN(C(=O)Cc3cc(C(F)(F)F)nn3C)C2)C1 N1(C(C2(C)N(C(c3cncc(C)n3)=O)CC(O)C2)=O)CC2CC3CC2C1C3 c1(OC)ccc(C(=O)NCC23CC2CN(C(C2CC(C(C)(C)C)C2)=O)C3)c(Cl)c1 N1(C(CC2CN(C(C)=O)C2)=O)CCOCC1CC(=O)NC1CCCC1C(C)C c1(OC)ccc2c(c1)C(CCNCN(C)S(=O)(=O)N1CCC(C#N)C1)=CC2 O=S(=O)(CC1Cc2ccccc21)NCCC12CCC(CC1)NC2 Cc1cc(NC(=O)CC2CCC(NC(c3nnn(C)c3N)=O)CC2)cnc1O c1(C(=O)NC2(CCCNC(C3C(C)(CC)C3)=O)CC2)nc(Cl)cs1 Cc1cccn2nc(C(N3CCC4(CCN(C(=O)CCCCC#N)C4)C3)=O)cc12 C=CCC(C(=O)NCCNC(=O)C(C1CCC(CC)CC1)C1CCCC1)C(C)C c1(N2Cc3c(nc(C)s3)CC2)[nH]c(=NCC2CC(O)CCO2)nc2c1ncn2C C1(CNC(=O)Cn2ccnn2)CCN(C(c2ccn3nccc3n2)=O)C12CCC2 CC(C)CC(CC(C)C)C(=O)N(C)CCN(C(=O)Cc1cc(F)ccc1Cl)C C1(C)(NC(Cn2ccc(C)c2)=O)CCCCC1C(=O)N(C1CCCC1C#N)C c1(C(=O)NCCCNC(C(c2c(C)cncc2)C)=O)cnn2c1OCC(C)C2 N1(C(CSC)=O)CC(C2CN(C(C3CCCC(NC(=O)OC(C)(C)C)C3)=O)C2)C1 C1(c2n(CC(=C)C)nnn2)(NCc2nccn2C)CCN(CC)C1 N1(C(CC2C=NN(C)C2=O)=O)CC2(NC(c3n[nH]cc3Cl)=O)CCC1CC2 N1(C(C(C)CNC(=O)Cc2cncnc2)=O)CC2C(C(N)=O)C2C1 C1(C(N2C(C(C)(C)NC(COCCOCC#C)=O)CCC2)=O)CC12CCOCC2 c1(C(N(CCNC(=O)C(C)CSC)CC)=O)cncc2c(Cl)cccc12 C(C(C)(C(C)C)NC(=O)COc1cccnc1)NC(C(N1C(CC)CCC1)=O)=O c1(CCC(=O)NC(CNC(C2(C(=O)OC)C(=C)CC2)=O)(C)C)c(C)noc1C c1(C(=O)NCCC(=C)CNC(C2CCCCO2)=O)cc(Cl)ccc1Cl C1(c2nnnn2C2CCCC2)(CNS(Cc2cc(C)ns2)(=O)=O)CCC(=O)NC1 C1(C(N2CC(NC(Cc3c(C)cc(O)cc3)=O)C2)=O)CCOC2(CCOCC2)C1 n1(CCC(N2CC(CC(C)NC(C(c3cccs3)OC)=O)C2)=O)ncn(C)c1=O Cc1ccc(CC(=O)NC2(C)CC(NC(c3ccn(CC(F)F)n3)=O)C2)c(C)c1 C(CNC(=O)C(=O)NC1CNCC1(C)C)(CC(C)(C)C)OC N1(C(C(C)OCCCC)=O)CCCC(N(C(=O)Cc2scnc2C)CC)C1 N1(C(c2ccc(CC(=O)NC)cc2)=O)CCCC2(CC1)CC2(F)F C1(CCN(C(=O)NCc2n[nH]c(C)c2Br)C)CCCCC12OCCO2 N1(C(C=C(C)C2CC2)=O)CC(NC(=O)CC=CC(C)(C)C)CC12CCOC2 C(CCCCC(=O)NCC1CC(C)CN(C(c2c(C)noc2C)=O)C1)=CC Cn1nc(CNC(C2CC=CC(O)C2)=O)cc1C(N1CCC(N2CCCC2)C1)=O c1(CC)ccccc1OCC.N12C3CN(CC13)S(=O)(=O)Cc1ccc(s1)C(=O)C2=O C12(NC(C(C(C)C)SCC)=O)CCC(CN(C(c3cnsn3)=O)C1)C2 C(=O)(C1=C(c2ccccc2)SCCO1)NC1CC(NC(CCCC#C)=O)CC1O c1(CC(=O)OC)ccnc(NC(CNC(=O)CN2CC(C)(OC)C2)C(C)C)n1 CC1(C(=O)NCCOCC(=O)NCc2nc(=O)o[nH]2)CNC(=O)C1 C12(C(N(C3CC(C(=O)NCCC(C(=O)OC)O)C3)C)=O)CCC(C)(C1)OC2 N1(C(=O)CCN(C(=O)Cc2ccc[nH]2)CCO)CCn2ncnc2C1 C1(F)(CNC(c2cscc2F)=O)CCN(C(C2CCC3(CCC3)O2)=O)CC1 C1(NC(C2C(C)(C)C2)=O)CCN(C(c2cc(O)nc(Br)c2)=O)C12CC2 C(CCCC(=O)N1CCC1NC(=O)C(C1CCCCC1)C)N(C(C)C)C c1(C(=O)OC)sc2ccncc2c1NC(=O)C(=O)NCCN1CCOCC1C C12(CNC(CN(C(=O)CCC(C)(C)C)CCCN(C)CC)=O)CCCC(C)(C1)OC2 c1(CCC(=O)N(C(CN(C(C2CCN(CC)C2)=O)C)C)C)ccc2c(c1)CCO2 c1(NC(CCN(C2CC2C=O)C)=O)ccc2c[nH]nc2c1.N1(CC#N)CCNC(=O)C1 N1(C(c2ccc(OCC(=O)OC)nc2)C(=O)NC(C)C)CC(=O)N(C)C(=O)C1 c1(SCC(=O)NC(CCCNC(CCC(C)OCC)=O)C)ccc2c(c1)CCC2 c1(C(N(CCC(C(C)C)NC(CC(CCC)C)=O)C)=O)ccc2cnoc2c1 C(C(C(=O)NCC1CCC1C(=O)OC)NC(=O)CCC=C(C)C)OCC C1(COC)(NC(=O)C(O)COCC(C)C)CCN(C(=O)C(C)OCC)C1 c1(C(N2CCN(Cc3ccc(OC)c(Br)c3)C3C2C3)=O)ccn2cncc2c1 C1(C)(CC(=O)NCC(Cn2cc(C3(F)CCOCC3)nn2)OC)CCSCC1 CC(CC(C)(C)C)C(=O)N1CCCCCC1C(N1CC(n2cnnn2)C1)=O C12(C(N3CCC(O)(C(C)C)C3)=O)CCCC1CCN2C(=O)CC(C)(C)C#N C1(NC(C(=O)NC2CCN(Cc3ccccc3)C2=O)=O)CCS(=O)(=O)CC1 c1(SC)cccc(C(=O)NC2(C)CCN(C(C3CC3C)=O)C2)c1Cl c1(C(=O)NCC2(NC(C(CC)n3ccnc3)=O)CCOC2)cc(Cl)ccc1OC c1(OC)ccc(CC(=O)NCC(C)CN(C(=O)C=CC2CCOCC2)C)cc1F c1(N2C(C)CCN(C(c3cnn(C)n3)=O)CC2)nc2ccc(Cl)cc2s1 c1(C(=O)NC(C2CCCCC2)CC)cc(Cl)cc(Cl)n1 c1(C(N(CCNC(c2cn(C)nc2)=O)CCN2CCCCCC2)=O)ccc(O)cn1 CC1CN(C(=O)CC(C(F)F)NC(=O)Cc2ccn(C)n2)CCN(C)C1 C1(C(=O)NCCC2(O)CCN(C(c3scc(C)c3Cl)=O)C2)CCc2cnnn2C1 C1(C#C)(NC(CC2CN(C(CCOCC#C)=O)C(C)C2)=O)CC2CCCC12 c1(CC(N2CC(NC(c3c(C)c[nH]n3)=O)C2)=O)c[nH]c2cccnc12 C1(NC(c2c(CNC(Cn3c(C)ncc3)=O)cc[nH]2)=O)CNC(=O)C(C)(C)C1 C1(CCNC(c2cc(C)sc2)=O)CCCCN1C(=O)CC(C)N(C)C C(=O)(C(C)(C)CCCNC(c1cnn(C)n1)=O)N(C(C=C)C1CC1)C C1(C(N2CCC(F)(CNC(CCCOCC)=O)C2)=O)CCc2ccccc2C1 c1(C(C)C)nc(C(C)(C)C)cc(=NCC2(NC(C3CCCN3)=O)CC2)[nH]1 Cc1cccc(C)c1C(O)C(=O)NCC(C)N(C(=O)C(F)(F)c1ncccn1)C C1(C(N2CC(C)C(CNC(C3(C)CCCOC3)=O)CC2)=O)CCc2cncn2C1 C#CC1(O)CCCN(C(C2(C3CC3)CN(C(=O)C(O)C=CC)C2)=O)C1 C1(c2cn(C)nc2)(C(F)(F)F)CCN(Cc2cnc(Br)c(N)n2)CC1 C1(C)(NC(c2c(CNC(C(COC)OC)=O)ocn2)=O)CC(C)(C)OC1=O N1(c2cc(CC)nc(CC)n2)CCC2C(CCCN2C(c2ccn(CC)n2)=O)C1 C(CC(C(=O)N)OC)OC.C(C(F)C(=O)N(C)C)C1(CCCCSC)CC1 c1(C(=O)NCCC2CCCN(C(c3cnnc(O)c3)=O)C2)cc(Cl)c(Cl)cc1O C1(CN(C)C(c2cccc(C(C)(F)F)n2)=O)CCN(C(=O)CCc2cscn2)C1 CNS(=O)(=O)N1CCC(C(=O)NCc2cn(CC3CCCN3C(C)=O)nn2)C1 Cc1cnc2n1C(C(=O)N1C3CCC1CC(NC(=O)CC(F)(F)Cl)C3)CCC2 CCC(O)(CC)CCN=C(NC1CCn2ccnc2C1)N(C)CCOC C1(C)(OC(=O)NCC(CC)(CC)Nc2cccc(C(F)(F)F)c2)CCS(=O)(=O)C1 C1(NC(C(C)c2cc[nH]n2)=O)C=CC(C(=O)NC2COC(C(F)F)C2)C1 C1(C2CCCN(C(=O)CCc3ccc(O)nn3)C2)(NC(CC(C)F)=O)CC1 C1(N(C)C)(C(=O)NCCNC(=O)C(N2CCC(O)CC2)=O)CCCSC1 N1(C(c2nc(C)co2)C(=O)Nc2ccc(OC)cc2)CCC2CCCCCC2C1 c1(CC(=O)N(CCCCn2cc(C(=O)NC)nn2)CC2CCOC2)c(Br)cnn1C N1(C(Cc2c(C)cc(F)cc2)=O)CCC2CCN(C(=O)CS(=O)(=O)CCO)C2C1 N1(CC(=O)NCCC(C)N(C(=O)C2=CSCCO2)C)CCc2sccc2C1 c1(C(=O)NCCC2CCCN(c3ncncc3I)CC2)ccc2[nH]ccc2n1 CC1(C)Cc2ccc(NC(N3CCN(c4cc5cccnc5s4)CC3)=O)cc2C1 N1(C(CSCC=C)=O)CC(C2CCCN(C(c3ccnc4cc[nH]c34)=O)C2)C1 c1(C(=O)NCC(CC)NC(C2CCOC(=O)CC2)=O)ccc2n[nH]cc2c1C Cc1cnc(CCN(C)C(=O)NCC(C2CCCOC2)(C)O)s1 c1(C(=O)NCC2CCCN2C(=O)CCc2cnc[nH]2)cccnc1-n1nccn1 n1(CC)nc(C)c(C(=O)NCc2ccc(CNC(C3C(C)=NO3)=O)c(F)c2)c1C C1(O)(CNC(C(C)=C2CCC2)=O)CCN(C(=O)C(C)(O)C2CCC2)C1 N1(C(COc2cc(C)on2)=O)CCC2CCC(NC(C3CCC(C)(C)C3)=O)C1C2 c1(C(N(C2CCCN(C(Cc3c(C)n[nH]c3)=O)C2)C)=O)c(C)nn(C)c1C C(=O)(C1(C)CCc2ccccc21)NC1CN(C(c2c(CC)nc[nH]2)=O)CC(C)C1 c1(OC)ccc(OC)c(C(=O)NC2CCC(NC(=O)C(F)(F)C3CC3)CC2)c1N C1(NC(C2CCC(NC(c3c(C)n(C)nc3)=O)C2)=O)CC(C)CCC1O c1(C(=O)NC(COC)C)nsc2cc(-c3ccc(I)cc3)ccc12 C(CC(C)C(=O)NCCCCC(=O)NCc1ccccc1CO)=CC N1(C(C(c2cncc(Cl)c2)(C)C)=O)CCC2CN(Cc3ccc(F)cc3N)CC12 C1(NC(Cn2ccc(C)n2)=O)CCN(C(=O)Cc2nnc(C)n2C)C1(C)C C(CCC(C)(C)C(=O)Nc1ccccc1O)NC(c1[nH]cc(C)c1C)=O c1(OC)cc(OC(C)F)cc(CNc2cc(C(=O)OCC3CC3)ccc2C)c1 C(C(O)C(=O)N1CC(CC(=O)N(C2CCCC2C)C)(OC)C1)OC N#Cc1c[nH]c(=NC2CN(C(C34CCC(CC3)C4)=O)C2)c2sccc12 c1(C(N2CCC(NC(c3c(C)cc(SC)o3)=O)C23CC3)=O)cnc2n1CCCC2 N1(C(C2C(C)(C)CC2)=O)CC2CC(N=c3[nH]c4ccccc4o3)C2C1 CCC(CC(=O)NC1(C)CCN(C(=O)C(C(F)(F)F)OC(C)=O)C1)C(C)(C)C c1(C(N(C2CC3CCC(C2)N3C(C2CC2(F)F)=O)C)=O)ccnc2ccccc12 c1(C(=O)NC(C)CNC(=O)CC2CC2C2CC2)cc(Br)c(C(F)F)s1 C(=O)(CCCC(C)C)NCC(C1(O)CCN(C(c2c(C)nn(C)c2)=O)C1)C N1(C(C(c2cc(C)sc2)(C)C)=O)CCCCC(NC(=O)C(C)(C)C2CCOC2)C1 C1(C(=O)NC2CCN(CCNC(C=CS(C)=O)=O)CC2)(OC)CCCCCCC1 n1(CC=C)nnnc1C(c1cn[nH]c1)NCc1csc(Cc2ccccc2)n1 N1(C(COCCC#C)=O)CC2CC1CN(C(c1cn(C)c(=O)cc1OC)=O)C2 CCC(C)C(=O)NCCOCC(=O)NC(COC)C(=O)OC C1(NC(c2cc(CCNC(c3cn(C)nc3)=O)on2)=O)CCC(F)(F)C1 n1(CC(=C)C)nc(C2CCC2)nc1CCc1ncc(F)cn1 c1(OCCC)c2cc(cc1Br)CN1CCCC1CO2.C(C(F)(F)F)SC C1(C(C)NC(c2cnc(C)[nH]2)=O)CCN(C(c2scnc2C(C)(C)C)=O)CC1 c1(NC(C23CC(NC(C4CN(C)C(=O)CC4)=O)(C2)C3)=O)cccc(C#N)c1F C1(NC(CCC)=O)CCC2(CC1)CC2NC(=O)Cc1c(C)noc1C C1(NC(CC2CCCN(C(C3C(CC)N(C)CC3)=O)C2)=O)CCC2CCCC1O2 c1(CCCCCOC(C(C2CC(F)(F)C2)OC)=O)ccc(F)cc1 C1(CC)C(NC(=O)COCC(C)C)CCCN1C(C1CC12CCCC2)=O C1(CNC(CCCCSC)=O)CN(C(c2ccc(C)o2)=O)CCC12CCC2 C1(C)(C)C(=O)NC2CC(C2)C(F)C1=O.C1CCC(C(N)=O)O1.CNC c1(CNCC(c2c(OC)cccc2)(F)F)ccc(Br)cc1OC(F)F C1(N(CC(C)(C)OCC)C)CCN(C(=O)CC2CCCC2)CC1 N1(C(CCCCC=C)=O)CCC2(CCOCC2)C(NC(=O)C(CC)(CC)CO)C1 Cc1nc(C(=O)NCc2ncoc2CCNC(=O)C(C(C)C)N(C)C)sc1C C1(C(=O)NC)CCCC1NC(=O)CNC(C1CCC(OC(C)=O)C1)=O c1(CCC(=O)NC(CN(C(c2cn(CC=C)nc2)=O)C)C)ccc2c(c1)CCO2 c1(C(N2CCN(CC(C)NC(CSCCCC)=O)CC2)=O)cnc2n1CCS2 C=CCC(CC(=O)NCc1cn(C)nn1)NC(c1ncccc1Cl)=O c1(CC(N2CCN(C(c3n(C)c(O)nc3)=O)CC2)=O)cn2ccccc2n1 C1(C(N2CC(CCO)(NC(C=CC3N(C)CCC3)=O)C2)=O)CCn2cncc2C1 c1(C(=O)NCCN(C(=O)CC2CN(C)C2)CCOC)ccc2oc(C)nc2c1 N1(C(c2cc(CCC)on2)=O)CCN(C(=O)Cc2cncc(OC)c2)C2CC12 N1(CC23C(C(=O)OC)(CC2)C(C)C(C)CO3)CCC=C(c2cncnc2C)C1 c1(-c2cn(C(C(=O)OCC)C)nn2)ccc(NC(=O)CCc2ccc(C)[nH]2)cc1 C1(C(=O)NCC=CC(=O)NCc2cn(CCC)nn2)CNC(=O)CC1C c1(C2(C(N3CCC(N(C(=O)CC4OCCCO4)CC)C3)=O)CCC2)ccccc1 c1(CC(=O)NCC2N(C(C=CC)=O)CCC2C)nc2ccccc2[nH]1 N1(C(c2c(CC)nn(C)c2)C(=O)NC(C)C)CC2(C)CCC2(C)C1 Cc1nc2c(C(=O)NCC(C)CNC(c3c(C)ccc(C)c3N)=O)ccnc2[nH]1 N1(C(CCN(C(C)=O)C)=O)CC2CCC1CN(C(=O)C(C)(C)O)C2 c1(C(=O)NCC(=O)NCC(CC)NC(=O)C(F)(F)CC2CC2)ccc(F)cc1 c1(C(N2CC(F)(C(=O)Nc3cn(C(C)C)nn3)C2)=O)ccc(I)c(Br)c1 C1(C(=O)OCc2nnc(OCC3CCOC3)s2)C2CCCOC12 C1(CNC(c2ccncc2F)=O)CN(C(C2SCCS2)=O)CCC1(F)F c1(OC)cccc2c1OC(C(=O)NCCCCC1CN(C(C3CCOC3(C)C)=O)C1)C2 c1(C(N(C(CNC(C(C(=C)C)(C)C)=O)C)C)=O)ncc2ccccc2c1N C#CCC(C(=O)N1CSCC1C(=O)NCC(CC)n1cccn1)C1CC1 c1(C(=O)NC2CC(NC(C3(C=C)CCCCC3)=O)C2)cc2c(s1)CC(C)CC2C C12(C(=O)NCC(CO)NC(c3scc(C)c3)=O)CC(C1)C(c1ccccc1)O2 C1(C)(CNC(CC2CN(C(C)=O)C2)=O)CCN(C(=O)CC2CSCCO2)C1 C=CCC(C)(O)C(=O)NCC(CNC(=O)CCC(C)(F)F)OC c1(CCC)cc(C(=O)N(C)CCOCCNC(=O)C(C)NC(C)(C)CC)ccn1 CC(C)(C(=O)NCC1CCC(C(=O)NC(C2CCCCO2)(C)C)CC1)C(F)(F)F CCCC(C)(C)CC(=O)N1CCC(N(CCO)C(c2cc(C(C)C)no2)=O)C1 c1(C(N(CC(CC)NC(c2c(Cl)n[nH]c2C)=O)C)=O)cc(F)cc(F)c1 c1(C(=O)NC(c2cn(CC3CCOC3)nn2)CCC)ncccn1 CCC(O)C(C)(C)C(=O)NCC1(OC)CN(C(C2CCC(=O)N2CC)=O)C1 CC1(C)CCCC(NC(=O)C2=NOC(CNC(=O)C=CCN3CCCC3)C2)C1 c1(N(CC(C)C)C)ccc(C(=O)NC2CCC(CNC(=O)CSC3CCC3)C2)[nH]1 Cc1ccc2nc(C(=O)NC(C)(CNC(C3SCCS3)=O)C3CC3)cn2c1 C1(CNC(C2CCC(CC)O2)=O)CC(O)CN1C(=O)CSCc1csc(=N)[nH]1 CC(C)C(COCC)C(=O)NCCOCCOCCNC(=O)CC1C(C)(C)C1(C)C c1(C(N2CCC(N(C)C(C3CCOC3)=O)CC2)=O)c(F)cc(OC(F)F)cc1F C1(C(=O)NCc2c(CO)cn(C)n2)CCN(C(=O)C(C)(C)C#N)CCO1 c1(C(=O)NCCN(C(c2cc[nH]c2)=O)CC)cccc2[nH]c(C)cc12 C1(NC(C(C=C=C)C)=O)CCN(C(c2csc(Cl)c2)=O)C1(C)C N1(C(c2ccc(C(N)=O)[nH]2)=O)CCOCC1CC(=O)NOCC1CCCCCC1 c1(NCC(C(C)(C)F)(C)F)ccc2sncc2c1 c1(C(c2n(CCCSC)nnn2)NCCC2CCC(=O)N2)cn(C)nc1Br C(=O)(C(C)C(C)NC(c1cc[nH]c1CCC)=O)NC(CCCC)C C1(C(=O)NC2CCC(NC(c3nc(C)oc3)=O)CC2)COC2(CO)CC1C2 N1(C(CC2CN(C)C2)=O)CCc2c(CNC(=O)CCc3ccsc3)cccc2C1 c1(CC(=O)NC2CN(C(c3c(C)cc[nH]3)=O)CC2F)coc2ccccc12 C(=O)(CCCCCCCC)NC(CNC(C(CC=C)(C)O)=O)CC=C N1(C(c2c(N)ccc(OC)c2)=O)CC2CCCC(NC(=O)Cc3cnsc3)C2C1 C1(NC(C=C(C)C(C)C)=O)COC2(C1)CN(C(c1coc(Cl)n1)=O)C2 C(=O)(C1CSc2ccccc21)N1C2CC(NC(=O)Cc3cnc[nH]3)C(CC2)C1 C1(C(O)F)CCN(N2CCN(c3nccc(N4CCCCCC4)n3)CC2)C1 c1(C(N2C(CNC(C3CCCS3)=O)CC(C)(C)C2)=O)cc(O)c2sccc2c1 C1(CC(=O)NC(C(=O)NC(C)CCc2cn[nH]c2)CO)CC2(CC2)CO1 CC(CNC(c1cnc(=N)[nH]c1)=O)C(F)C(=O)N(C1CC1C)C c1(NC(C(C(C)NC(c2c(C)snc2)=O)C)=O)cnc2[nH]cnc2c1 c1(C(=O)NCC(CC)NC(C2(c3ccc(F)cc3)CCC2)=O)cc2c(s1)CCC2 C(=O)(CC(=O)NCC(c1ccccc1)CNC(C1CCC(F)C1)=O)NCC c1(CC(=O)NC(CCNC(C(C=CCCC)O)=O)(C)C)cc(C(N)=O)ccc1N N1(C(C2N(C)CCC2)=O)CC2CCC1C1CN(C(c3c(Cl)cccc3Cl)=O)CC21 N1(C(CS(C(C)C)(=O)=O)=O)C2CCC1C1CC1(NC(C1CC1F)=O)C2 CC1CC=C(C(=O)NCCCN(CCCNC(=O)C=CCCC(F)(F)F)C)CC1 CC(C)C(F)C(=O)NC(C)(CN(C(=O)C(C)(F)c1ccon1)C1CC1)C1CCC1 c1(CC)[nH]nc(C(N2CCC(NC(=O)CN3CCSCC3)C2C)=O)c1Br Cc1conc1CC(=O)NCC1(NC(=O)Cn2cnc(C(F)(F)F)c2)CC1 C12(CNC(c3cc(C)[nH]n3)=O)CN(C(C3(CC4CC4)CC3)=O)CC(F)(C1)C2 CN1CCN(C(C2(C3CC3)CC=CC2)=O)CC1CNC(C1CCOCC1)=O Cc1cccc2c1CN(C(c1cncc(CNC(=O)C(C)(C)C(F)F)c1)=O)C2 C#Cc1cc(C(=O)NCC2(NC(c3oc(CO)nc3C)=O)CC2)ccc1C Cc1cc(=NC(=O)C2CCCC2NCc2cc(Br)ccc2C)[nH][nH]1 C(=O)(CCCCCC#N)N(CCCCCC(=O)N1C(CCC=C)CCC1)C N1(C(c2nc(OC)c(C)s2)=O)CC(NC(=O)CCc2cc(C)[nH]n2)C2CC2C1 C=CCC(CNC(=O)CC1CC1C1CC1)C(=O)NCCc1cocn1 C1(NC(C2(C(=O)NC)CC2)=O)CN(C(=O)C(C)SC)CC1c1ccnn1C c1(OCC(=O)NCC2CCC(NC(C3C(C)C3C)=O)C2)cccc(Cl)c1Cl C(=O)(CC(C)N(C)C)NC1C(C(=O)NC(C(=O)OCC)C2CC2)CC1 CP(C)(=O)c1c[nH]ccc1=NC(=O)N1CCCC2(CCCCN2)C1 C1(C(=O)NC2CCCCCCC2)(CC)CCCN(C(c2nocc2COC)=O)C1 C1(N(C)C)Cc2ccccc2N(C(=O)NC2CCCC2c2ccccc2F)C1 c1(CC(N2CCC(N(C(=O)CC3CC(OC(C)(C)C)C3)CC)C2)=O)cccnc1 c1(OC(C)C(=O)NCC(C)(C)CN(C)C(c2ocnc2C2CC2)=O)ccccn1 N1(C(C2N(C(CC(CC)C(F)F)=O)CC23CCCC3)=O)CCC2(CCCCO2)C1 Cc1ccc(C=CCC(=O)NC2CC2NC(c2onc(C)c2C)=O)cc1 C1(C(=O)NCCOCC#C)CCN(C(c2ccncc2NC)=O)CCO1 c1(C(=O)NCC(CO)NC(C2CC(C)C2)=O)cc(Br)c(O)cc1F C1(NC(C(C(CC)C)N)=O)COC2(CCN(C(=O)CCc3ccc(C)nn3)C2)C1 Cc1nn(C)cc1C1=NOC(C(N2CCN(C(=O)CCF)CC2CO)=O)C1 C12(CNC(C3COCCO3)=O)CCC(CC1NC(c1ccc(Br)o1)=O)C2 CC(CC(=O)NC1CC(NC(C2(C#N)CCCO2)=O)C1)CC(F)(F)F Cc1cc(Cl)cc(Cl)c1OCC(=O)NC1CCCCCN(C(C2(SC)CC2)=O)C1 N12CCC(C(F)C1)C2=O.CC1CCOC1CCN(C)C C1(n2cc(CC=C)nn2)CC2CCC1(NC(=O)Cc1cc(Br)cs1)C2 N1(C(CCC#C)=O)CCC2(CC1)CC2CNC(c1ccc(CSCCC)o1)=O n1(CCOC)cc(C(=O)NCC(C)CN(C(=O)CN(C)CCO)C)c(C)n1 n1(CCNC(=O)CCC2CC(NC(=O)CC3CCCCO3)C2)cc(CO)nn1 C(=O)(C(F)C(C)C)N1CC(OCCC(=O)NC(C=C)CO)C1 N1(C(C(C(C)C)N(C)C)=O)CCOCC2(COCCN2C(c2ccoc2)=O)C1 c1(C(N2CCC(C)(NC(C(CC)OCC)=O)C2)=O)nc(C)n(C)c1C C1(NC(C2C(C)CCC2)=O)CN(c2nnc(C3CC3)o2)CC2(CC2)C1 C#CC1C(C(=O)NCCN(C2CCCOC2)C(=O)CN(C)C(C)=O)C1(C)C N1(c2ccnc(C)n2)CCN(C(c2ccc(-c3ccc(O)nc3)o2)=O)CC(O)C1 CC(C)CC(F)(F)C(=O)NCCN(C(=O)Cc1ccc(C(F)(F)F)cc1)C(C)C c1(OC)c(F)ccc(F)c1C(=O)NCCNC(c1cn2cc(C)nc2s1)=O N1(C(C=Cc2c(C)nsc2)=O)CC2CC1CN2C(=O)C(C)C1(O)CCC1 CC1(C)CN(C(c2cccc[n+]2[O-])=O)C(CNC(C2CC(F)C(=O)N2)=O)CO1 c1(OC)ccc(Br)cc1C(=O)NCC1CCCCN1C(c1nccnc1Cl)=O C12(NC(C3N(C(CCC)=O)CCC3)=O)CC1CN(C(=O)CCSCC(C)C)C2 CC(C)CCN=C(NCCN1CCCS1(=O)=O)NCC(C1CCCCC1)F N1(C(c2cnc(CC)[nH]2)=O)CC(NC(c2cc(C(C)=O)cs2)=O)CCC1C C1(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)C(C)C)CCc2cnn(C)c2C1 C1(N(CC#C)C(c2occc2C)=O)CCN(C(c2ccnc(COC)c2)=O)CC1 C(=O)(C1CCc2cccc(F)c21)N(CCCN(C(C(C(CC)(C)C)O)=O)C)C CC1CNc2c(C(N3CCN(C(C4CC5(C4)CC(O)C5)=O)CC3)=O)cnn2C1 c1(OC)cccc(C(N2CC(C(=O)NC34CCCC3OCC4)(OC)C2)=O)c1C C(=O)(C(C)=Cn1ccnn1)NC(CC)CN(C)C(c1cncc(C(C)(C)C)c1)=O c1(C(=O)NCCOCCNC(C(C)NC(N)=O)=O)nocc1C(C)C CCCC(C(O)C(=O)NCCCn1cnnc1)NC(C1CN(C)C(=O)N1)=O C1(NC(CCC(CC)C)=O)CCCC12CN(C(c1cc(C)c(Cl)cn1)=O)C2 C1(CNC(CNC(N)=O)=O)CCC2(CC1)CCN(C(C1CC=CCO1)=O)CC2 c1(SCCC)cccc(C(N2CCC(F)(CNC(C3CCCCS3)=O)C2)=O)c1 c1(CN=C(NC2CCN(CC(F)(F)F)C2)NC2CCC2)cc2n(n1)CCOC2 C1(C(=O)NC(COCC)C(N2CCOC(C#N)C2)=O)CC(=O)NC(=O)C1 C(=O)(CCCCC(C)C)NC1CCC(C(=O)NC(CCCC)C(C)O)C1 C(C(C(C)(C)C)NC(C1(C)CC(C)(C)C1)=O)NC(c1cnc(C)[nH]1)=O Cc1csc2c(C(N3CC4CC(NC(c5ccco5)=O)CC4C3)=O)ncnc12 C#CCC(CC(F)F)C(=O)NCc1ccsc1C(=O)NC1CCCC1C(=O)OC CC1(C)CCCN(C(=O)CNC=O)C1CNC(=O)CC1(C(F)(F)F)CC1 c1(NC(C2N(C(c3ccn(C)c3C(F)F)=O)CCC2)=O)nc(Cl)c2c[nH]nc2n1 c1(NC(C(c2cccs2)NC(C(CCOC)OC)=O)=O)cnc(C)c(C#N)c1 CC(C)C(O)C(=O)N1CCCCC1CC1CCC1 C(=O)(CCCC(=O)N(C)C)N(CC(C)NC(C1CN(C)CCN1C)=O)C CC(C)CC(=O)C(=O)NCC1(C(=O)NC(C2CCOCC2)C)CCC1 C1(C(=O)NC2(CF)CCN(C(=O)C=C(Cl)Cl)C2)CCc2nncn2C1 c1(C(N2C(C)CCC2C(=O)NCC2CCS(=O)(=O)C2)=O)c(F)cc(Br)cc1Br C1(CNC(=O)CC2C3CN(C(=O)CCc4cccnc4)CC23)CC(F)(F)CO1 c1(OC)ccc(C(=O)N(C2CCN(C(=O)C(F)(F)C(C)O)CC2)C)cc1C C1(C(=O)NCCCN(C(C(c2scc(C)n2)C)=O)C(C)C)CC(C)CC(=O)N1 c1(C(=O)NC(CC)CNC(c2csc(CC(F)(F)F)n2)=O)ccc(O)c(C)c1 c1(C(N(C(CNC(C2N(C(CCC)=O)CCC2)=O)C)C)=O)ccc(CSC)cc1 N1(C(c2ccc(OC)nc2)=O)CC(NC(=O)C2=NOC(C)C2C)CC(C)(C)C1 N1(Cc2c(Cl)nc(C)nc2Cl)CCC2C1CCCN2C(=O)Cc1ccc(Cl)cc1 c1(C(=O)NCC(CC2CN(C(CCC(C)OC)=O)C2)(C)C)ccc2cccnc2n1 C1(C)(C(=O)NCCOC2CN(C(C(CC(C)C)(F)F)=O)C2)Cc2ccccc2N1 c1(C(=O)NC2CC(NC(c3cc(C)[nH]n3)=O)C2)n[nH]c(C(C)C)c1Br N1(C(CCC(=O)NC)=O)CCC(CNC(=O)CCC(C)SC)C12CC2 N1(C(C)C(=O)NC2CC(CNC(c3coc(Br)c3)=O)C2)CCCCCC1 c1(C(=O)NCCC(C)NC(C2C(=C)CC2)=O)ccn(C2CCCCC2)n1 N1(C(C23CCC(OC)C2C3)=O)CC2(C1)CN(C(=O)CCCn1nc(C)cc1C)C2 C12(CNC(COCC(C)C)=O)CC1CN(C(C1CCOC1C(F)(F)F)=O)C2 C1(CNC(c2cc(F)cs2)=O)COCCN(C(C2C=CCCC2)=O)C1 C(=O)(C(C)(C)C(C)(C)O)NC(COC)CC(=O)NC(C)C(=O)OC C(=O)(CC(C(F)(F)F)C1CC1)NC1C(C)N(C(c2cc3cccnn3c2)=O)CC1 c1(OC)ccc(C(=O)NCC(C2CCN(C(C3CCCCO3)=O)CC2)F)cc1F c1(C(N2CCC(CCNC(=O)COC3CCC3)C2)=O)ccc2c(n1)CCCC2 C1(C(=O)NC2C(C(=O)NCCC(C)(C)O)OCC2)CC2CCC2C1 c1(C(=O)NC2CCN(C(C=CCN(C)CC)=O)C2)ccc(NC)c(F)c1 c1(CNC(=O)NC2CCC(CC(=O)OC)C2)cccc2c1OCO2 c1(NC(N2CCCC(C(=O)NC3(C4CC4)CC3)C2)=O)ccc(F)cc1 CCC(C)CC(C(=O)NCC(F)F)NC(=O)C1=CCCOC1 c1(C(N2CCCC(CC)(NC(C34CC(F)(C3)C4)=O)C2)=O)cccc2c1CC(=O)N2 C=C(Cl)C(C)(C)C(=O)NCCOCc1ccc(CN2CC(C)CC(C)C2)cc1 CP1(=O)CCN(CCc2nc(-c3cocn3)no2)CC1 N1(CC)C(=O)CCC1C(=O)NCC1COCCN1C(=O)CCNC(N)=O C1(C(C)NC(=O)Cn2cnc(=N)[nH]2)CCN(C(=O)Cc2nnc(O)s2)C1 C1(C(C)C)CN(C(=O)C(C)O)CCN1C(=O)CSc1nn(C(C)C)c(=S)s1 c1(C(=O)NC2C3CN(C(=O)CCC4CCCO4)CC23)cnc2n1CCS2 c1(C(N2C(C)CC(NC(=O)C3=CC4CCC3C4)CC2)=O)cccn2c(O)nnc12 N1(C(C=Cc2ncc(C)[nH]2)=O)CCC(CNC(=O)CC=C(Cl)Cl)C(C)C1 c1(C(=O)OCCNC(c2cnn[nH]2)=O)ccc(S(=O)(=O)N2CCCCC2)cc1 C1(COC)CN(C(c2scc(C)c2C)=O)CCN1C(C1CC1C)=O Cn1ccc(C(=O)NCC2(O)CC(NC(C3CCC3(F)F)=O)C2)n1 c1(C(=O)NCC2OCC(CNC(c3cnsc3)=O)C2)sc([N+](=O)[O-])cc1Cl O=C(C(CO)c1ccccc1)N1CC(CO)(NC(C2(C3CC3)CC2)=O)C1 c1(CNC(c2n[nH]cc2NC(c2c(O)cccc2O)=O)=O)ccc(Br)c(F)c1F c1(OC)ccc2c(c1)CCC(C(=O)NC1CC(NC(c3cnc(C)[nH]3)=O)C1)C2 N1(C(=O)OC)CCC2NCCC2C1.C12CCC(C1)C(=O)NC2 C(=O)(CCC(C)O)N(CCCNC(=O)CCOCC(F)F)CC N1(C(c2nc(C)n(C)n2)=O)CC(C2CCCN(C(=O)C3=C(Cl)CCOC3)C2)C1 Cc1cc(S(=O)(=O)N2CCC3C2CCCN3C(c2cnc(O)[nH]2)=O)c(C)cc1Cl S(=O)(=O)(c1ccc(Br)nc1)N1C(CCC)(Cc2ccccc2)CCC1 C1(C(=O)NCC2C3CN(C(CNC(=O)NC)=O)CC32)CCOC2(CCCC2)C1 N1(C(C(C)Sc2ncccn2)=O)C2CCC1CC(NC(C1CCC(C)(C)OC1)=O)C2 c1(OCC)ccc(C(=O)NCc2ccsc2OC)c(OC)c1 N1(c2cc(NCCCCN(C)C)nc(C)n2)CCCN2c3ccccc3CC2C1 CCC(CC)CCC(=O)N1CCC(CNC(C2CCCC3(CCC3)O2)=O)CC1 CCC(CC(F)(F)F)C(=O)N1CCCCC(NC(c2cc3c(s2)CCC3)=O)C1 N1(C(c2cncc(C(C)C)c2)=O)CC(CNC(=O)COC2CCCC2)C2(CC2)C1 N1(C(C2(OC)CCOC2)=O)CCOC2(C1)CN(C(=O)C(C)NC(C)(C)C)C2 C1(C)(C(N(CCC(C(C)C)NC(c2c(O)cccc2Cl)=O)C)=O)CCOC(C)C1 Cc1nc2ncc(C(=O)NC(C)CC(C)NC(C3CCC=CCC3)=O)cc2o1 CP(C)(=O)CC(=O)NC1CCC(CC(N2CCCCC2CCCO)=O)CC1 c1(NCCOCCN(C)C(C2CCCC2)=O)ccnc2cnnn12 C12(CNC(CCCC)=O)CC(CCO1)N(C(c1ccc(OC)nn1)=O)C2 CC1CC(CC(=O)NC2CC(CNC(C3Cc4cscc4C3)=O)C2)CC(C)(C)C1 N1(c2c(C)cnc(C)n2)CCC2CCC(NC(C3(O)CCCC3)=O)C1C2 Cc1nc2c(C(=O)NCCCCNC(c3c[nH]c(Br)c3)=O)cccc2o1 CC1=C(C(=O)NCC(O)CNC(=O)C=Cc2ncccc2C)C(=O)OC1(C)C N1(C(C(CC#C)O)=O)CCCC(O)(CNC(c2cc(Br)ncc2OC)=O)C1 N1(C(C=CCC)=O)CCN(C(C2(C)CCCN2C(=O)OC(C)(C)C)=O)CC1(C)C CC1CCCCN1CC(=O)NCCOCCC(=O)NC1CCCCC1N(C)C c1(CC(=O)N(C(C=C)C)C)noc(C2CCC2)n1 n1(CC)nc(C(=O)NC23CC(NC(c4ccc(CN=[N+]=[N-])o4)=O)(C2)C3)cc1C C1(C(=O)OC)CN(C(c2ccc(Br)cc2)=O)CC12CN(C(c1nc[nH]n1)=O)C2 C#Cc1cccc(C(=O)NC(C)(C)CCNC(=O)C(S(C)(=O)=O)C2CC2)c1 c1(CC(=O)N(C2CCN(C(C(CC)n3ccnc3)=O)C2)C)cnn(C)c1C(F)F N1(C(C2C3CCCC23)C(=O)NCCC#N)CCC(OCc2ccccc2)CC1 C(=O)(C1(C)NC(=O)c2ccccc21)NC(C)CCCNC(=O)C=C1CCC1 C(=O)(CCN(CCC(=O)O)C(=O)Cc1ccco1)NCCCN(C)C N1(C(CC(C(=O)O)c2cccs2)=O)CCc2nnc(Cl)cc2C1 C(C1(O)CCCc2ccccc21)NCC(N)Cc1ccncc1 n1(-c2cccc(C)c2)cc(S(=O)(=O)CC(N2CCOCC2)c2ccccc2)cn1 C1(NC(c2n(C3(C)CC3)nnn2)(C)CCc2ccccc2)CCOC(C)(C)C1 c1(SCC(=O)NCC(CNC(CC(=C)Br)=O)OC)ccc(OC)cc1 c1(CC(=O)NC(CN(C(C23CCC2C3)=O)CC)C)ccc2c(c1)OCO2 c1(C(=O)NC(c2c(C(NOCC(CC)C)=O)con2)C)cc(OCC)cc(F)c1 C(=O)(C(CC(F)F)N(C)C(c1nnn(C)c1C)=O)N1CCC(OCC)C1 c1(NC(CC2N(Cc3c(OC)ccc(Br)c3F)CCC2)=O)cnc2ccoc2c1 n1(CC)nc(C)c(C(=O)NCC2(CNC(=O)CCn3c(C)csc3=O)CC2)c1Cl C1(C(=O)NC(C=C)CO)C2C(CN1C(C1CCCOC1)=O)C2(C)C c1(NCC)cncc(C(=O)NC(C2CCN(C(C3C4CCCC34)=O)C2)C)c1 c1(C(N(CCC)CCNC(C2CCOC2C)=O)=O)nccc(N)c1Cl CC1(C)CN(C(=O)Cc2cscn2)CC1CNC(c1c[nH]nc1Br)=O C(=O)(C1COc2ccc(F)cc21)N1CCC(NC(CC(C)(F)F)=O)C12CCC2 C1(NC(CC=C)=O)CC(O)CN(C(c2cscc2C2CC2)=O)C1 C(CC(C)C)(C(=O)NC(C)Cc1ccn(C)n1)NC(Cc1cc(C)sc1)=O N1(c2ncc(C)cn2)CCCC2C1CCN2C(c1ccc2nc(O)sc2c1)=O N1(C(C2C=C(C)CS2)=O)CCCC(F)(CNC(=O)Cc2n[nH]c(C)n2)CC1 C1(O)(CNC(CC(CC)CC)=O)CCCN(C(=O)C#CC2(C)COC2)CC1 N1(C(CC2CCCN(C(c3c(CC)c[nH]n3)=O)CC2)=O)CC(=O)NCC12CC2 C(=O)(C1CCCc2ccnn21)N1CCC(N(C(c2[nH]cc(CN(C)C)c2)=O)C)C1 N1(C(C2CN(CCOC)C(=O)C2)=O)CC(NC(=O)C=C(C)C2CC2)CC1(C)C C1(C(=O)NCC(c2cccc(C)c2)NC(c2scnc2Cl)=O)CCC(F)(F)CC1 C1(C(=O)NCC(C)C)C(F)(CC)C2CCCCN2N1C(CCF)C(=O)OCC N1(C(C(CNC(CS(CC)=O)=O)(C)C)=O)CCC2C(C(N)=O)C2C1 C(=O)(CN=c1cc[nH]cc1)NCC(C)N(C)C(C1CC1c1cn[nH]c1)=O c1(C(N(C2CCN(C(=O)CCN3CCOC3=O)C2)CCC)=O)sccc1F Cc1c(C(=O)OCC2CC3(CCCCC3)CCO2)oc2c(Cl)cccc12 c1(C(N(CCC(=O)NCC2(F)CCOC2)CC#C)=O)ccc(F)c(F)c1 C1(NC(CC(CC)C2CCC2)=O)C2CC1CN(C(=O)C=Cc1cccc(Br)c1)C2 Cc1cc(C(=O)NC2CC(NC(=O)C3=CCCOC3)C2)cnc1C(F)(F)F c1(C(N(C2C(C)CCN(C(c3cnccc3Cl)=O)C2)C)=O)cnc2nccn2c1 C(=O)(C(C)CC(=O)N(C(C)CNC(=O)C(O)Cc1cnc[nH]1)C)OC CC1(C(=O)NC2CCC2C(=O)NCC2(CO)CCCCC2)CCOCC1 C1(C(=O)NC(C(=O)NCCS(CC)(=O)=O)C)CC2CC(=O)C1O2 c1(N2CCC(C(C)(C)NC(c3cnc4n3CCS4)=O)CC2)ccccc1[N+](=O)[O-] Cc1ccc(Cl)cc1C(N1CCC(NC(=O)Cc2cccc(Br)c2F)C1)=O N1(C(c2ccc(C(C)=O)cn2)=O)CCCCCC1C(=O)NOCC(=O)N(C)C N1(C(c2ccc(C)cn2)=O)CCC(CO)C(NC(=O)C(C)(C)c2cccnc2)C1 Cc1ccc(C(C)(C)C(=O)NCC(CO)NC(C2CCC(C)(C)CC2)=O)c(C)c1 C1(C(CCC(=O)NC2C(c3cc(C)[nH]n3)C2)=O)CCC(C(F)(F)F)CC1 Cn1cc(C#N)cc(CNC(=O)C(=O)NCCCCC(C)(F)F)c1=O CC1(F)CN(C(=O)CC2(O)CCCCC2)CCN(C(c2cncc(O)c2)=O)C1 C1(C(=O)NCC=CCNC(C(C)(C)OCC(F)(F)F)=O)CC2COCCN2C1 Cc1ccc2cc(C(=O)NC3CC(C)N3)ccc2c1 C1(CC(C)NC(C2(C)CC2Br)=O)CC2CCC(C1)N2C(=O)CCc1csc(=N)[nH]1 c1(CC)ccnc(C(=O)NCC2CCCN2C(=O)CNC(c2cnccn2)=O)c1 N1(CCNC(c2c(C)cc(C)s2)=O)CCCN(C(C2CC2CN(C)C)=O)CC1 C1(NC(CSCCN(CC)CC)=O)CCN(C(=O)CCS(C)=O)CC1F c1(CCC(=O)NCCC2CN(C(C3(O)CCSCC3)=O)C2)ccnc(Cl)c1F CC1=C(C(=O)N(CCC(C(C)(C)C)NC(c2ccc[nH]2)=O)C)C(C)(C)CCC1 N1(C(C=CCOC)=O)C2CCC1C(CNC(=O)CC(c1ccc(F)c(F)c1)C)C2 N1(C(C2(NC(CCSCC)=O)CCC2)=O)CCCC2C1CCN2C C1(OC)CCC2(C(N3CCN(CC(=O)NCCNS(N)(=O)=O)CC3)=O)CC12 c1(CNC(=O)Nc2nccc(-c3ccccc3F)n2)ccc(Cl)c(Cl)c1 c1(CC)ccccc1OC(=O)NC12CC(NC(=O)CCC(=O)NCCCF)(C1)C2 CN1CCCCC1C(=O)NCC1CC(NC(=O)C(C)(C)N2CCOCC2)CCO1 c1(C)cc2c(Cl)nccc2o1.c12ccc(cc1)CNC(=O)C(=O)NC2C.C1CC1 N1(C(c2c(C)nn(C)c2)=O)C2CCCC1CN(C(c1nc(Cl)sc1C(C)C)=O)C2 CC1(C)CC(CNC(c2cnsn2)=O)CN(C(=O)CCC2CC2(F)F)C1 c1(C2(C(=O)NC(CC3CN(C(CC(=O)OCC)=O)C3)C)CC2)ccc(F)cc1C C1(C(=O)NCc2cncc(C(N)=O)c2)CC2(C1)CN(C(C1CCCCC1F)=O)C2 N1(C(CC2C(CC)C2(F)F)=O)CC2C(CNC(=O)C(C)(C)C3CCCCC3)C2C1 c1(C(C2CN(C(c3cnnn3-c3ncccc3Cl)=O)C2)=O)ccc(O)c(F)c1 C(C)(CCN=c1cc(C)nc(N2CCOC3(CCOCC3)C2)[nH]1)S(C)(=O)=O C(CN=c1[nH]c(=NC2CC(Nc3ccccn3)C2)[nH]c2c1COC2)OCC(=C)C Cc1c(O)ccc(C(N2CC3CC2CN3c2ncnn3cccc23)=O)c1C C=CC(C)(O)CC(=O)NC(CCCC)C(=O)NCC1OCC2CCC1C2 C(C(COC)CC(=O)N1CCC(CN(C(=O)C=Cc2cncc(C)c2)C)C1)OC c1(C(N(CC(CN(C(CC)=O)C)O)C)=O)cnn(CC2CC2)c1 C1(CC(=O)NC2CCCC2CNC(C2CC(SC)C2)=O)(SC)CCOCC1 Cc1cc(Cl)ccc1CC(N1CC(C)(NC(C2CCOC2C)=O)C1)=O CC(C)(C(=O)NCC#CC(=O)NCCCCCF)C(F)(F)F C(Cc1cccs1)(CC(=O)NC1CCCCC1O)NC(=O)C=Cc1ccco1 C1(C)(CNC(c2c(C)nn[nH]2)=O)CC(F)(F)CN1C(c1ccc2n[nH]cc2c1)=O N1(C(CC2(OC)CCC2)=O)CC2(CCC(NC(=O)CC3CCCC3C)CC2)C1 c1(OC)cn2c(cc1=O)CN(C(=O)CC1(OC)CN(C)C1)CC2 c1(C(=O)NC2(CC)CCCN(C(C=CC(CC)C)=O)C2)cnn2c1CCCC2 c1(C(N(CC2CCN(C(C=CCCC)=O)CC2)CC)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)C(C)(C)O)N(CCC(C)NC(c1c(OCCC)cccn1)=O)C N1(C(n2cc(CC)nn2)C(=O)NCCOCC)CCN(C(=O)OC)C2(CCC2)C1 C(=O)(C(O)CC(F)(F)F)NCc1ccc(C(=O)NCCCCC(=O)OC)s1 c1(C(N2CCC(C)(NC(CC(CCC)C)=O)C2)=O)cc(F)c(F)c(F)c1F c1(-n2c(NC(N(C)Cc3ccccc3Cl)=O)ccn2)cccc2ccccc12 c1(C(N2CC(CC)N(C(=O)C=CCOC)CC2)=O)cnc2ccnn2c1C c1(CC(=O)OC)ccnc(NC(=O)Cc2scnc2C)c1 C(N=c1nc2c(ncn2C)c(NCc2cc(Br)ccc2F)[nH]1)c1nc(C)c(C)[nH]1 CCCCC(CC)CC(=O)N1CCN(C(=O)CC2CCCC2O)CC12CCC2 C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(CCCN=[N+]=[N-])=O)(CO)C1 C12(C(=O)NC(C)CC3CN(C(=O)CN(C4CCCC4O)C)C3)CCN(CC1)C2 N1(C(=O)C(C2CCCCC2)O)CCCC2(CCN(C(C3CCOC3)=O)C2)C1 C12(NC(C3C4CC(=O)OC4C3)=O)CCC(CC1)N(C(=O)CCC1CC(N(C)C)C1)C2 C1(C(C)C)CN(C(=O)CCC2CCC(=O)C2)CC1C(N1CCC1CN=[N+]=[N-])=O n1(C(C(=O)N(CCC)CCc2nn[nH]n2)C)cnc2sccc2c1=O N1(C(C(C)OCCC(C)C)=O)CCOCC(NC(C2COCCN2C)=O)C1 C(=O)(CC(=O)N1CC(C(C(=O)NCC(F)Cl)OC)C1)OC C1(C(N(CCN(CC(=O)NCCOCCNC(C)=O)C(C)=O)C)=O)C(C)C1C C#CC1CCN(C(=O)CCC2CCCCN2C(=O)CC(C)N(C)C)CC1 C1(C2CCC2)(NC(c2nnnn2CCCSC)(COCCOC)C)CC1 c1(C(=O)NC(CNC(CC2(OC)CC2)=O)CC(C)C)nc(Cl)ccc1N N1(C(Cn2nc(C)oc2=O)=O)CC(N=[N+]=[N-])CC1C(=O)NCC1CC(C)C1 C1(CC(N2CCN(C(C3C(C=C)C3)=O)CC2)=O)CCC2(CCOCC2)CO1 N1(C(CCc2nc(=N)[nH][nH]2)=O)CC(O)C(O)C1CNC(=O)CN1CCSCC1 C12(C(=O)NCC=CCNC(CCCCNC(N)=O)=O)CC1Cc1c[nH]nc12 N1(C(C(CO)NC(C(C)C)=O)=O)CC2CCCN(C(=O)CN(C)C(C)C)C2C1 C1(C(N2CC(CCNC(COCc3n(C)ncn3)=O)C2)=O)CS(=O)(=O)CC(=O)N1 C(=O)(C1=CCCSC1)N1CC(N(C)C)C(CNC(c2cnn(C)c2N)=O)C1 c1(C(N2C(C)(CNC(C3(CC)CCCCC3)=O)CCC2)=O)cc(C)cc(Cl)c1N C1(NC(CCNC(N)=O)=O)CCCC(C(=O)Nc2ccc(CO)c(F)c2)CC1 Cc1ccc(C(N2CCC(CNC(c3ccc(C(F)(F)F)s3)=O)C2)=O)nc1 c1(CC=C)ccc(C(=O)NCC(C)N(C)C(C2CC(C)(O)C2)=O)cc1 C1(C(=O)NC2CC(F)(CNC(CCC(C)(C)C)=O)C2)CC2CCC(C1)C2O C1(CCC(=O)NCC2CC(F)(F)C2)CCN(C(C2(C(N)=O)CC2)=O)C1 C(CCC1CC1)(C(=O)NCC12CC(C1)C2)NC(c1ccnc(Cl)n1)=O CC(C)CCCC(=O)N1CC2(C(N3CCC(CO)C(O)C3)=O)CC1CO2 c1(C(N2C(C)C3CC2C3NC(=O)CCc2ccn(C)n2)=O)ccc2n[nH]cc2n1 C(=O)(C1=CSCCO1)N(C1CCCN(C(c2c(C)ocn2)=O)C1)CCO C1(C(N2CCC(O)(CCNC(CNS(NC)(=O)=O)=O)C2)=O)CCCCC(=O)N1 C1(C(N2CC(F)(F)CC2CNC(C2(O)COC2)=O)=O)CCCC2CCCCC12 C1(NC(c2c(C)ocn2)=O)CC2(C1)CC2C(=O)N(C1CC(CO)C1)C c1(C(=O)NCCC2(NC(CC=CC=C)=O)CCCC2)c(Cl)cc(CO)cc1Cl Cc1cc(C(N2CCC(NC(=O)C(c3cccc(Br)c3)O)C(F)C2)=O)ccc1O c1(C(=O)NCC(C2CC2)NC(C(C=CC)O)=O)ncc(N)nc1C C1(NC(COCCC#C)=O)CN(C(=O)CCC(=O)c2ccc(CC)cc2)C2CC12 C1(NC(CCc2ncc(C)[nH]2)=O)CCCCC12CCN(C(=O)C(Cl)=CCl)CC2 CC(=Cn1ccnn1)C(=O)N1CCCC1C(C)NC(c1cc(C)n(C(C)C)c1)=O c1(OC)cccc2cc(C(=O)NCc3ccccc3O)c(=O)oc12 c12ccc3cc(n(C)c3c1)NC2=O.CCC(F)(F)CC(=O)N1CCCC1CC c1(C(C2CC2)NC(C(=C)CO)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CC(CCNCC(C)(C)C1CCOC1)CC(C)(C)C N1(C(C2N(C(c3cc(OC)ncn3)=O)CC3CC32)=O)CC2CN(C)CC2C1 N1(C(C(C)C2CC2)=O)CCN(C(=O)CCOC2CC2)CC(O)C1 Cc1nc(-c2cn(CC3CCCC3NC(=O)CSn3cccn3)nn2)ccc1F N1(C(CC2C(C)(C)OCCO2)=O)CC2CCC(C1)C(NC(c1cnco1)=O)C2 C12(NC(=O)CCc3cnc[nH]3)CC1CN(C(=O)CNC(=O)C(=O)O)C2 n1(CC(=O)NC2C3CCN(C(C4OCCN(CC=CC)C4)=O)C32)cc([N+](=O)[O-])cn1 CCCCCCCCC(=O)NC(c1ccccc1)C(N1CCCC(CO)(CO)C1)=O C1(C(N(CC(C)N(C(=O)Cc2ccno2)C)C)=O)CCS(=O)(=O)N1 C1(CC(=O)N(CCCNC(=O)CCNC(N)=O)CC)CCC(=O)C1 Cc1c(CC(N2CCOC(C3CN(C(=O)CCC4CC4(C)C)C3)C2)=O)cnn1C c1(CC=C)ccccc1C(=O)NC(C)CN(C(c1csnn1)=O)CC c1(C(=O)NCC=CCNC(C2(C)N(C(C)=O)CCC2)=O)cc2cncn2c(O)n1 c1(C(=O)NCC(O)CNC(C2COC(=O)C2)=O)ccc2c(c1)CCCS2 Cc1cc(C)n2ncc(C(=O)NC(C)Cn3cc(-c4cnsc4)nn3)c2n1 c1(C(=O)NCC(C)(C)NC(Cc2cncc(C)c2)=O)cc(F)c(C)cc1Cl C1(CNC(CN2CC(=O)N(C)C2=O)=O)CC2CCC1N(C(c1sccc1F)=O)C2 C1(N(C(c2c(CC)nccn2)=O)C)CCCCN(C(=O)CNC=O)C1 N1(C(CCn2c(C(C)C)ncc2)=O)CCCC12CCN(C(C1CCCO1)=O)CC2 C(=O)(C(O)CC(C)(C)C)NCCC(C)N(C)C(C1CC(C(F)(F)F)C1)=O C(N=c1cc(Cl)c(O)n[nH]1)C1CN(C(c2n[nH]c3c2CCC3)=O)CC12CCC2 C1(NC(C(CCC)C)=O)CC2CN(C(C3CCCCN3N=O)=O)CC2C1 c1(C(N2CCCC(C)(NC(C(CC(C)C)F)=O)C2)=O)cc(S(C)(=O)=O)co1 C12(NC(=O)C3=CCOC3)CCCC1CN(C(c1cnc3[nH]cncc1-3)=O)C2 CN1CCC(CC(=O)NCc2ccccc2CN(C)C(C2SCCCS2)=O)CC1 C1(C)(C(=O)NCC(=C)CCNC(c2cn(-c3ccccc3)nn2)=O)CC(C)=NO1 C1(NC(CCC(=O)OC)=O)CN(C(c2cnn(CCF)c2)=O)C2(CCCOC2)C1 C#Cc1ccc(C(=O)NC(C)CN(C(=O)C(C)n2cnnn2)CC)c(F)c1 C1(CC)CCCCC1C(=O)NCC1CCCCC1NC(=O)C(CO)N(C)C C1(NC(c2cccc(CC)c2)=O)CCN(C(=O)CCCCSC)CC1OC N1(C(c2c(C)cn(C)c2)=O)CC2CCC2(NC(c2ncc(Cl)cc2O)=O)C1 C1(NC(=O)CCc2cncs2)CCCC12CN(C(=O)Cn1nnc(=O)[nH]1)C2 N1(C(C(COC)OC)=O)CC2CCN(C(=O)C(C)c3ccco3)CC12 CC1c2c[nH]nc2CCC1C(=O)N(CC(O)CNC(=O)CC1CC(F)(F)C1)C C(=O)(C(C)CC(C)(C)C)NCC1ON=C(C(=O)N(C)Cc2cc(C)ncc2)C1 c1(C(=O)NC(CCCC)(C)C)nccc2n[nH]cc12 c1(CN2CC(C(=O)Nc3ccc(OC)cn3)OCC2)cc(F)c(Cl)c(Cl)c1 CC1(C#CC(=O)N2CC(CCCCNC(=O)C3=CCOCC3)C2)CC1 CC1CC2CN(C(=O)C(O)C3CCC3)CC2N1C(=O)CSCC(F)F N1(C(C2CC(=O)OC2)=O)CCC(n2cc(CCNCCO)nn2)CC1 c1(OC)ccc(C(N2CC(NC(C3CC(=C4CCC4)C3)=O)CC2CO)=O)c(C)n1 CN1CCC(N(C(=O)CN(CCOC2CCC(=O)NC2)N)C)CC1 c1(C(=O)NC2(C)CCN(C(=O)CC3CCCCC3)C2)ccc(S(C)(=O)=O)s1 C1(C(C(=O)NC2CC(C)(NC(C)=O)C2)N(C)C)CCC(F)(F)CC1 C(CCCCC(=O)NC1(C)CC(OC)CN1C(c1cc(C)n(C)c1C)=O)OCC N1(C(c2c(C)con2)=O)CCC2C(CCCN2C(=O)C(=O)C(C)(C)C)C1 C(=O)(CCC(=O)NN(C)C)NC1(COC)CN(C(C2(n3nccn3)CC2)=O)C1 c1(CC)ccc(OC)cc1C(=O)NC1CCC1CNC(c1ccc(C)cc1N)=O c1(C(N2C(CC(=O)Nc3nccc(Cl)c3Cl)CCC2)=O)ncc([N+](=O)[O-])cc1I C(=O)(C1CCCc2ccnn21)NC1CCN(C(C(CC)N(C)C)=O)CC1 c1(C(N2CC(C(N3CCCC(C(=O)NC)C3)=O)(CCl)C2)=O)cccc2cc[nH]c12 N1(c2ccc(C)cc2)N=C(C(=O)NCCCn2cccn2)CCC1=O n1(CC(=O)NCc2cnccc2Cl)ccc(=NCc2cc[nH]n2)nc1O C12(C(=O)NC3CN(C(CC(c4ccc(Cl)cc4)N(C)C)=O)C3)CC(C1)S(=O)(=O)C2 N1(C(c2cn(C)nc2C2CCC2)=O)CCN(C(C2CC2CF)=O)C(C2CC2)C1 C1(C(N2CCC(N(C(=O)CCCc3csc(=N)[nH]3)CC)C2)=O)CCC=CO1 C1(CNC(CC(COC)C)=O)CN(C(=O)C(F)(F)C(C)(C)O)CC2(CCC2)O1 C1(CNC(CC2(COC)CCOC2)=O)CCN(C(=O)C(=Cc2cccs2)C)CC1 N1(C(C2CCC(F)C2)=O)CCC2(CCCN(Cc3cc(C4CC4)[nH]n3)C2)CC1 N1(C(C2C3CN(C(=O)C=CCN4CCC4)CC32)=O)CC2(CO)CCC1CC2 C(=O)(CCCCC(C)(C)C)N(c1cccc2nc[nH]c12)C1C(C)CCNCC1 C1(N(C)C(c2cn(CC(N)=O)nn2)=O)CCCC(NC(=O)CNC=O)C1 C12CCCCN1C(=O)N(C1CC1)CC2(C)C.c1noc(N(C)C)n1.C(=O)(C)OC C12(CNC(=O)CCn3ccnn3)CC(CNC(c3nc(C4CC4)cs3)=O)(CO1)C2 c1(C(=O)NC(C)CNC(=O)Cn2cccc2)sc(=N)[nH]c1-c1ccccc1 N(C(=NCCN1CC=CC1)NCc1ccccc1)CC(C)(C)Sc1ncn(C)n1 N1(C(CCCSC)=O)CCC2(C=C(C(=O)NCC3CC(C(C)(C)C)C3)C2)C1 N#Cc1ccc(Cl)c(C(N2CCN(CCCNC(C3C4COCC34)=O)CC2)=O)c1 C(C)(CCC#N)(c1nnnn1C1CC1)NC(=O)NCC(C(C)C)OC O(NC(=O)CCN(C(c1ccnn1C)=O)C1CC1)C(CC)CC c1(C(N(C2CCCN(C(c3cc(N)c(F)cn3)=O)C2)CC)=O)cc(C)c(F)cn1 C=CC(C)C(C)C(=O)N(C)CC1(NC(=O)CCCCCNC(=O)OC)CC1 N1(C(=O)Cc2cnc(C3CC3)[nH]2)CCN(C(C2CC23CCCC3)=O)C(CCO)C1 N1(C(C2OCCN(CC)C2)=O)CC2CC1CN(C(=O)CC1CCCO1)C2 N1(c2nc(CC)c(C)cc2C#N)CCC2(COC(CNC(=O)CC(C)(C)O)C2)C1 Cc1ccc2c(=NCC3C4CN(C(=O)CCOCC(F)(F)F)CC34)[nH]cnc2c1 C(=O)(C(O)CCNC(=O)CCc1ccncc1)NC(CN(CC)CC)C Cn1nnc2cc(C(N3CCN(C(=O)CSC4CC4)C(C(F)F)C3)=O)cnc12 c1(C(N2CC3C(NC(C(CCC)OC)=O)(C3)C2)=O)cnc(OCC(F)F)c(Cl)c1 C(CCCCCCC)N(C(c1cc(C2CC2)[nH]n1)C(=O)NCCOCC)CC1CC1 C(=O)(C1CCCn2cnnc21)NC1CC(O)(CNC(c2c[nH]cc(C)c2=O)=O)C1 C1(C(N2CC=CC2)=O)N(C(c2sccc2Cl)=O)CC12CCCC2 c1(NC(C2COCCN2C(=O)Cc2cc(Br)cs2)=O)ccc2c(c1)OCCO2 c1(C(=O)NC2CN(C(C(CCC#C)O)=O)CC2SC)cc(Cl)cc2ccncc12 c1(C(C(=O)NC2CCC2)N(CC(=O)NC)C)ccn(C)c1 C(=O)(C1=CCCCC1F)NCCC1CC(NC(=O)CC2CCC(F)(F)CC2)C1 c1(C(C)C)ccc(C(N2CCC(F)(C(=O)NCCC(F)(F)F)C2)=O)c(Cl)n1 C(=O)(C(C)(C)CN(C)C)NCC1(OC)CN(C(=O)CCc2nccn2C)C1 c1(CC)cc(C(N2CCC(CCNC(c3ncccc3Cl)=O)C2)=O)ccn1 c1(NC(CN2CCC(OC)C2)=O)nnc2n1CCNC2 c1(C(=O)NC2CC(C)(NC(=O)CO)C2)ccccc1-c1ncnn1C1CCCC1 CC1CCCC(C(=O)NCC(N2CCN(C(=O)C=Cc3nccs3)CC2)C)C1 c1(NC2C(NCc3cccc(OC)n3)CCC2C(=O)O)ccc(C(C)C)nc1C c1(C(=O)NCCC(C)N(C(=O)CCCCC(N)=O)C)ccc2[nH]ccc(=O)c2c1 C(=O)(C1CCCc2ncc(C)n21)NC1(CCCNC(C(S(CCC)(=O)=O)C)=O)CC1 C1(C(O)C(N)=O)CC(=O)N1.c1(CNC(CC2(SC)CCC2)=O)cccc(C2CC2)c1 CC1CN(C2CC2)CC1(c1nnnn1CC(F)F)NCc1csc(Cl)c1 c1(NCCCCCCC)[nH]c(=NC2CCCN(CC)C2)nc2c1cnn2C n1(CC)ncc2c1CC(C(=O)NCC1CCCN1C(c1cn(C)[nH]c1=N)=O)CC2 N1(C(C2CN3CCN2CC3)=O)CC(F)(F)CC1CNC(C1(C(=O)C2CC2)CC1)=O C#CCC(C(=O)NCc1nonc1C)NC(C1COCC1(C)C)=O C1(C)(NC(C2CCC(=C)CC2)=O)CCCN(C(C2(SC)CCOC2)=O)C1 c1(C(CC(=O)NC(C(CO)NC(C(CC)O)=O)C)NC(C)=O)ccccc1C C1(NC(C2CCC(C)C2)=O)CN(C(c2cccnc2S)=O)C2(CCOCC2)C1 c1(CC(=O)NC(CC)CNC(=O)C(N2CCOC2=O)C)cc(C)cc(F)c1 N1(C(CN2CC(=O)NCC2)=O)CCC2C(C(=O)NC3CCOCC3O)C2C1 c1(C(=O)NC2CCN(C(CC(C=C)C)=O)CC2(C)C)cc2c(s1)CCC(C)(C)C2 C1(CNCc2cnc(CC)[nH]2)CCN(C(=O)Nc2ccc(F)c(C)c2)C(C)C1 N1(CCCc2cccc(C)c2)C(C(=O)O)CCC12CC2 C1(C(N(C2CCCN(C(=O)CC(C)(C)C#N)C2)CC)=O)Cc2c(C)cccc2O1 c1(OC)ccc(C(N2CCCCC2c2cn(C3CCC3)nn2)=O)c2c1C(=O)NC2 c1(OC)c(C(=O)NC(=O)Cc2nnc(O)n2-c2ccccc2)cccc1Cl c1(C(N2CCCC2)=O)cc(C(CC(CO)NC(c2cccnc2)=O)=O)n[nH]1 CCCCCC(F)C(=O)NCC1CC(F)(CNC(C2CC3CCC(C2)O3)=O)C1 CC(C)(C(=O)NCC(CO)NC(=O)C(C1(O)CCCC1)F)N1CCOCC1 c1(C(=O)NCCCC(=O)NC2CCN(CCOC)CC2C)cccc(C#N)c1C N1(CCNC(CC2C(C)CCCC2)=O)CCCC2(CC(O)C2)C1 C#CC1(C(N2CCC(CN(C)C)C2)=O)CCN(C(=O)C=CC2CCCN2C)C1 c1(C(N2CCC(CNC(=O)C=CCF)CC2)=O)cccc(OCC2CCCO2)c1 Cc1[nH]cc(C(=O)NC2CC2NC(=O)Cc2c(Cl)cccc2Cl)c(=O)c1Cl C1(C(N(CC(C(C)C)C)C)=O)CN(C(c2cc(CO)[nH]n2)=O)CCC1(C)C C12(CC(=O)NCC(CNC(=O)CC3CCOC3)O)CNC(=O)C(C1)C2 O=C(CCCCc1cccc(O)c1)NCCC1CCN(C(C23CC(O)C2C3)=O)C1 C1(C(=O)NCCC(CN(C)C)O)CCC(CNC(c2cnn(C)c2N)=O)CC1 N1(C(c2cncc(N)n2)=O)CCCC(NC(C2(O)CC2)=O)CC1 N1(C(CN(C)C(c2ncccc2Br)=O)=O)CCCC2(CC2)C1 N1(C(C(CC)F)=O)CC2CC1(CNC(=O)CSc1cccc(OC)c1)C2 C(=O)(C(CC)C(C)(C)CC)N1C(C)(C(N2CC(C=C)C2)=O)CCC1 CC1(C)C(C(N2CCC(O)CC2)=O)CCN1C(=O)CCOC1COC1 N1(C(CCN(C(CCC)C)C)=O)CCN(C(=O)CC2(C)CCCC2)CC1C(C)C c1(-c2cncc(C#CC)c2)cccc2sc(C(=O)Nc3cnc(C)c(C)c3)cc12 c1(OC)cccc(C(=O)NCC(C2CCC2)NC(c2cc(CO)n(C)n2)=O)c1C Cn1cncc1C(N1CCC(OCC2CCCOC2)C1)=O N1(C(C(C)(F)F)=O)CCC(O)C(NC(=O)C(O)CCn2cncn2)C1 c1(C(=O)NCC2C(NC(c3cc(C)nn3C)=O)CCC2)cc2c(cn1)COCC2 c1(C(N2CCC(C(C)C(=O)N(C)CC3(C)CCCC3)CC2)=O)cn(C)ccc1=O c1(OCC)c(C(F)(F)F)csc1NC(c1cnoc1C1CCOCC1)=O C(C(C)(C)C(=O)NOC(CO)C(C)C)N(C(=O)CN1CC2CCC1C2)C1CC1.CO O=C(C1CCc2snnc21)NC1CCCC1NC(c1cnc2cccnn12)=O O=C(CC1=CCN(C(c2ccsn2)=O)CC1)NC1CC(CO)C12CCC2 N#Cc1cc(C(N2CCC(CNC(=O)CC3CCC3(F)F)C2)=O)ccc1F CC(C)CC(F)C(=O)N1CC(C)(NC(c2ccc(Br)cc2N)=O)C1 C1(CNC(c2c(C)coc2)=O)CCC2(CN(C(C3CCCC4(CCC4)O3)=O)C2)O1 C12(C(CNC(C3C4CC5C(C4)C35)=O)NC(c3c(C)csn3)=O)CCC(CC1)C2 c1(C(=O)NCC(C)N(C(C(C)OC2COC2)=O)C)csc(Cl)c1Cl c1(CC(N2CC(NC(C(CCC)OC)=O)C(OC)C2)=O)ccc2oc(C)nc2c1 C1CCN(N(C)C(C2CCC2CC(C)C)=O)CC1.n1(CC)cc(C)cn1 c1(C(=O)NC(CC(C)C)CNC(c2cc(F)nc(F)c2)=O)ccnc2[nH]c(O)nc12 C1(NC(COc2c(CC)cccc2)=O)CCN(C(C2CCC(O)CC2)=O)C(C)C1 c1(CC)nn(C)c(Cl)c1C(=O)NC(CO)C(C)NC(=O)CC1COC(C)(C)C1 N1(C(CN(C)C)=O)CC2CCCC2(NC(c2ccc(N(C)C)nn2)=O)C1 C1(C(=O)NCCC)(NC(=O)CC2CCC3CC23)CCN(C)C1 C1(CNC(Cc2cncc(C)c2)=O)COCCC1(F)F.C12C3CN(CC13)C2=O c1(CC)cc(NC(=O)C(C(C)C)NC(=O)CCCC2(OC)CCC2)ccc1C N1(C(c2c(C)noc2)=O)CCCC(NC(=O)CN2CCS(=O)(=O)CC2)C1C c1(OC)cc(C(=O)NC(Cc2ccoc2)C(=O)N2CCC(CC3CC3)C2)ncn1 c1(C(N2C(C)C(NC(=O)CC3CC3(C)C)CC2)=O)ncc2ccccc2c1O c1(CC)nnc(CNC(C2C(C)CN2C(=O)Cc2ccc(C)o2)=O)o1 N1(Cc2c(C(=O)NCc3ccc(C#N)o3)cccc2)C(=O)c2ccccc2C1=O c1(C(N2CCC(NC(Cc3nc(C)sc3)=O)CC2C)=O)cccc2c[nH]nc12 C1(O)(C(N)=O)CCCN(C(C2C3CN(C(c4nc[nH]c4[N+](=O)[O-])=O)CC23)=O)C1 C1(NC(c2n(C=C)ncc2)=O)CN(C(=O)CC2CC(O)C2(C)C)CC2(CC2)C1 C(=O)(C(C)(C)CC(=O)NC1CC(c2cn(-c3cccc(Cl)n3)nn2)C1)OCC c1(C(=O)NC2CC(CO)N(C(c3ccnc(C4CC4)n3)=O)C2)cn2c(n1)SCC2 C1(C(=O)NCC2(NC(c3cc(C)on3)=O)CCCCC2C)CCCCN(C)C1=O N1(C(c2cc(Cl)cs2)C(=O)NCC(C)C)CCCC2(CC=CCC2)C1 Cc1nc2ncnn2cc1C(=O)NC1CCCN(C(=O)C2=CCC2)CC1 N1(C(CC2(C(N(CC(=C)C)C)=O)CC2)=O)CCC(OCC(=O)OC)C1 C(=O)(C1CCc2ccccc21)N(CC(=O)NCC1(C)CC(F)C1)CC#C c1(C(N2CCC(N(C(=O)C(=Cc3cccs3)C)CC)C2)=O)cc(SC)ccc1C c1(C(C)C)ncc(Br)c(C(=O)NCCN(C(C2CC2F)=O)CC2CC2)n1 C1(N(C(CC2CCC(C)O2)=O)CC2CC2)CCN(C(=O)C=CCN2CCC2)CC1 C1(NC(C2C(=C)C2)=O)CC2(C1)CC(C(=O)N(C(C)COC)C)C2 N(C(=NCCC(O)C(F)(F)F)NC1CCOCC1)Cc1c(O)ccc(Cl)c1 C(CC(C)C(=O)N(C(CNC(=O)COCc1ccc(F)cc1)C1CC1)C)=CC C1(C(N2CC(CN3CCN(C(=O)CC4(O)CCCC4)CC3)C2)=O)CC2(C1)CC2F CC1(C)CC(C(=O)NC2CC2NC(=O)C=C2CCC2)CNC1=O c1ccc(-n2nnnc2C2CN(C3CCSCC3)C2)cc1 S(=O)(=O)(c1cccs1)N1CCC(CNC(=O)NC2CC(CN)C(O)C2)C1 FC(F)(F)C(F)(F)CCn1cc(CCCOC2CCOCC2)nn1 Cc1nc(=N)[nH]cc1C(=O)NCC(C)CNC(c1nnn(C)c1C(F)(F)F)=O C1(C(=O)NCC#CCNC(COC)=O)(OC)CC(C)C1 Cc1cc(CCC(=O)NC(C2CCCN2C(=O)CC2CC(F)(F)C2)(C)C)n(C)n1 c1(OC)cc(C)c(CN(C)C(C2CCCN(c3ccc(Cl)nn3)C2)=O)cc1OC N1(C(c2n(C)ccc2)=O)CCC2(CCN(C(c3cc(Cl)c4c(c3)OCO4)=O)C2)C1 C1(NC(C2(COC)CC2)=O)CCC(NC(=O)C(C)(CC2CCC2)C2CCC2)CC1 c1(SC)nc(C)cc(=NCC(CC(C)C)NC(c2c(Cl)cnn2C)=O)[nH]1 CC(O)CCCC(=O)NC1CCC(CNC(c2cccc(C(F)F)c2F)=O)CC1 C1(C(=O)NCC2CC(O)CN2C(=O)CN2CC3CC3C2)Cc2nccn2C1 N1(C(C2CCC(NC(C)=O)CC2)=O)CC2CC1CN2C(c1ccc(C)s1)C C(=O)(C1Cc2ccc(Cl)cc21)N1CC(NC(CC=CCC)=O)CC1(COC)CC C#CCCCC(C)C(=O)N1CC(C)(C(=O)NC(c2ccccc2)CC)C1 C(=O)(C1=CCCN(C(c2ccc(C(F)F)o2)=O)C1)NCC1CC[Si](C)(C)C1 C1(CC)CN(Cc2cccnc2C#N)CCN1C(=O)Cc1ccccc1 CC(C)CS(=O)(=O)CC(=O)NCC12CC(C1)C(NC(=O)CC1CC1(C)C)CO2 c1(OCC)cc(NC(=O)CC2CCC(C3CC3)O2)[nH]c(=NCC(C)C2CC2)n1 CC(CN=c1[nH]c(=NCc2cscc2Cl)[nH]c2c1CCCCC2)S(C)(=O)=O C1(C(=O)NC(CC)CNC(c2cnn(CCOC)c2)=O)(COC)CCOCC1 CON1CC(C(N2CCC2C(N2CCCC2C2CCOC2)=O)=O)CC1=O Cc1cc(C(=O)NC2CC(F)CN(Cc3cccc(Cl)n3)C2)cc2[nH]ccc12 Cc1cc(C(N2CCN(C)C(CNC(=O)CN3CCCCC3=O)C2)=O)nc(O)n1 C1(C(N2CC(OCCNC(=O)CCCC3CCCC3)C2)=O)CCn2nncc2C1 CN1CCN(CC(=O)NC2CCOC2CNC(C2CC(=O)NC(=O)C2)=O)CC1=O N1(CC(CC)(C)N=c2[nH]nc(C3CC3)o2)CCCC(C2(CC(=O)OC)CC2)C1 c1(C(=O)Nc2cnn(C3CCCCC3)c2)ccc(OCC2CCCCO2)cc1 C1(NC(CSCCC)=O)CCC(C)(CNC(c2cn(CC(N)=O)nn2)=O)C1 N1(CC(=O)NCC(=C)C)CCCC(CO)CC1.c12ccccc1CNC(=O)CC2C c1(C(N(C2CCCC2)CCCNC(CC(CC)C)=O)=O)cccc2c1CCCC2 C1(C#N)(C(=O)NC2C(C(=O)NCC=C(C)C)OCC2)CCCOC1 C(=O)(CCCF)NC1CC(CCNC(C(C)NC(C2CCC2)=O)=O)C1 c1(C(C)C)cc(C(=O)NC2(c3nnnn3C)CCC2CC(F)(F)F)nn1C C(CC(C)C)(C(=O)NCC(O)CNC(c1ccc([N+](=O)[O-])s1)=O)OC c1(C(C)(F)F)cccc(C(=O)NCCNC(C2CC3CCC2C3)=O)c1 c1(CC(=O)NC2CC(NCc3ccc(Cl)nc3)C2)cc(O)nnc1O c1(C(=O)NC(C2N(C(C(CC)SC)=O)CCC2)(C)C)cnn(C(C)C)c1C c12ccccc1CS(=O)(=O)NC2.C1(CCC)CNCC1C(=O)NCCOC C1(C(=O)NCC2(OC(C)C)CCC2)CC(C)N1C(C1CC(CC2CC2)C1)=O C1(C)(NC(c2cn(CC=C)nn2)=O)CCCCCC1.c12ccc(nc1)C(=O)NC2 Cc1nccc(=NCC(C)CC(C)O)[nH]1.c1(O)ccc(Br)cc1 N1(CC)CC(N(Cc2ncc(-c3ccccc3)nc2O)CC)CC12CCCCC2 C1(CCNC(c2c(C)nco2)=O)COCCN1C(=O)C(C)CN(C)C c1(N2CCC(C)C(NC(=O)C=Cc3ccccc3F)C2)cc(=O)n(C)c(=O)n1C c12cccc(c1OC)C1CCN2C1.C1(NC(=O)NCC)CC(C(C)=O)C1(C)C CCC(C)(CCC(C)C)C(=O)NCCOCCCNC(c1cnn(C(C)C)c1)=O c1(OCCC(=O)NCC(C)CNC(=O)CO)ccc(F)cc1F N1(C(CC(=C)C)=O)CCC(C2(NC(c3cc(C)cc(O)c3)=O)CCC2)CC1 N1(C(CC2N(C)CCC2)=O)CCC2(C1)CN(C(c1cc3ccsc3s1)=O)CCO2 N1(C(c2ccccc2Nc2cnn(C3CCOCC3)c2)=O)CC2CC2(O)C1 c1(NCCC(C)C2CCCC2)ncccc1S(=O)(=O)NC(c1sccc1Cl)C C#CC1(C(N2CCC(NC(=O)C(C)=CC)C(C)C2)=O)CCCCC1 CC1(F)CN(C(c2cc(=O)cc[nH]2)=O)CCN(C(C2CCC3(CCC3)C2)=O)C1 O=C1CC2C(C(=O)NCC3(C(=O)NC4CC5C=CC4CC5)CCCCC3)CC2O1 N1(C(C2N(C(CCC)=O)CCCC2)=O)CCC2(C1)CN(C(=O)CSCCC#N)C2 C(c1ccccc1)=CCC(=O)NC(C(=O)NCC1(CC(=O)OC)CC1)c1cccs1 c1(C(=O)NCCCN(C(C(C2CCCC2)OC)=O)C)cccc2ccccc12 C1(CC)CC1N=c1[nH]c(=NCC(CO)Oc2ccc(Cl)cc2)[nH]c2ncn(C)c12 C(=O)(C1=COCCO1)N1CCC(N(C(c2ccc(C(=O)OC)[nH]2)=O)C)CC1 C1(C(N(C2CCN(C(C(C(C)C)(C)C)=O)CC2)C)=O)CN(S(=O)(=O)N(C)C)C1 C1(NC2(c3n(C(C)CC4CC4)nnn3)COCCOC2)CCC2COCCC2O1 c1(OC)ccc(C(N2CC(NC(=O)CCn3ccccc3=O)C(C)C2)=O)cc1O c1(CC(=O)NC2(CC(=O)NC(C3CSC3)C)CCC2)cncnc1O c1(C(C(=O)NC2C3CN(C(c4c(C)cc(C)o4)=O)CC32)C)c(C)nn(C)c1C c1(OC)ccc(CCC(=O)NC2CC(C)N(C(c3cc(C)c(C)[nH]3)=O)C2)cc1Cl N1(C(C(CCC)C)=O)C2CCC1CC(CC(C)NC(=O)Cc1cnccn1)C2 C=CC(C)N=c1[nH]c(=NCC2CCN(C3CCCC3)C2)[nH]c2c1COCC2 C1(O)(C(C(=O)N(C2CCC2O)C)NC(CCCOC(C)C)=O)CCCCC1 c1(CC(=O)NCCC(CC)(C)NC(=O)CCc2cnoc2)cc(C)cc(C)c1 N1(C(C(CCC)F)=O)CC(C)N(C(=O)C(C)C2CCC2)C(C)C1 N1(C(c2c(C)nsc2C)=O)CC2CCC(C1)N2C(C1CCC2(CCC2)CO1)=O c1(CC)oc(C)cc1C(=O)NCc1ccc(C(N2CCCC(CF)C2)=O)o1 C(CC(F)(F)F)SCC(=O)NC(CN(C(CCC)=O)CC)CC S(=O)(=O)(c1ccc(Br)cc1F)N1C2CCCN(C(C(CC)NC)=O)C2CC1 N1(C(c2c(CC)c(C)sc2)=O)CC(CO)C2(C1)CN(C(=O)CCOCC(C)C)C2 N1(C(C(CCCOC)NC(C2C3CCC(F)C23)=O)=O)CCc2c(nnn2C)C1 N1(C(C(CC)NC(C)=O)=O)CCC(CCOC)(NC(C2CC23CC3)=O)CC1 C(CC(N)=O)(C(=O)NCC(CO)NC(=O)C(F)=CCCF)NC(CC(C)C)=O C(=O)(CS(C)(=O)=O)NC(CNC(c1nc(C)oc1)=O)CO C1(C#CC(=O)NCC2CCC2NC(=O)CC(c2ccccc2OC)C)(CC)CC1 S(=O)(=O)(c1ccc(Br)cc1Nc1ccc(C)cc1)N1CCC(COCC)CC1C Cc1c(C(N2CC(O)(C(C)CNC(C3CN(C)C(=O)N3)=O)C2)=O)ccn1C(C)C C1(O)(CN(C(C(COC)OC)=O)C)CCN(C(=O)Cc2cc[nH]c2)CC1 C(=O)(C(O)CC(C)(C)C)NC1C(NC(C23C(C(=O)OC)C(CC2)C3)=O)CC1 c1(C(=O)NC2(N(C(=O)C(CN(C)C)N(C)C)CC)CC2)ccc(C)nc1C CC1=C(C(=O)N(C2CCN(C(=O)CC(C)C(F)F)CC2)C)COCC1 N1(C(=O)NCCc2nc(C(N)=O)on2)c2ccccc2CCC2CCCCC12 C(C)(CC(C)N=c1[nH]nc(-c2ccon2)s1)NC(C(CCSC)O)=O N1(C(C)=O)CCC(CC(=O)NC(C2CCN(C(C3CCCCN3C)=O)C2)C)CC1 CC1CC(NC(=O)C=CC(N)=O)CCN1C(c1ccc(F)cc1Cl)=O c1(N(C(=O)COc2ccn(C)n2)C)ccc(NC(=O)Cn2cccc2)cc1 C1(NC(Cc2nnc(C)s2)=O)CCN(C(c2ccc(OC(C)C)nn2)=O)C12CC2 C1(NC(CN(C(=O)OC(C)(C)C)CC2CC2)=O)CCOC12CCOC2 c1(CC(N2CCC(NC(CNC(C)=O)=O)C2)=O)c(C)[nH]c2ccccc12 c1(CC)cccc(C(N2CCN(C(c3cc(C)c(F)cn3)=O)C(C)C2)=O)c1F C1(C(=O)OC)(C(=O)Nc2csc(Cl)c2)CCN(C(=O)C(F)CC2CCOC2)C1 C1(NC(C2C(=C)C2)=O)CCN(C(c2csc(=NCC)[nH]2)=O)CC1C C1(C(=O)NC(C(C)NC(c2ccns2)=O)CO)COC(C)(C)CO1 C1(CNC(Cn2c(C)c(Br)cn2)=O)CC(C(C)(C)C)CCN1C(=O)C1CC1 C(=O)(C1CCc2nccn21)N1C2CC(NC(Cn3c(=O)ccc(C)c3)=O)(C2)C1 N1(C(C2N(CC)CCOC2)=O)Cc2[nH]nc(C(=O)NCc3cscc3C)c2C1 C1(CCC)COCCN1C(=O)NCc1csc(-c2cccs2)n1 C1(C(=O)NC(C2CCN(C(C=C(C)C(C)(C)C)=O)CC2)C)CNC(=O)CC1C C1(=CC(=O)NCC(C)N(C(C2CCC(C)CC2)=O)CC)CC2CCC(C1)N2C CCCCCCCCCC(=O)NCCCN(c1ncc(Br)c(COC)n1)C1CC1 C(C(O)CC(F)(F)F)NC(C1(C2N(C(CCCC#C)=O)CCC2)CC1)=O c1(C(N2CC3CN(C(c4cnn(C)n4)=O)C3CC2)=O)ccc2c(c1)NC(=O)CN2 N1(C(CCC(C)N(C)C)=O)CC2CCOC2(CNC(C2CCCCC2)=O)C1 Cc1cc(C(=O)NC2CCN(C(c3ccc(C#N)cc3)=O)C2)ncc1S(N)(=O)=O c1(C(N2CC(C(C(=O)C(CO)c3ccccc3)C)C2)=O)ccccc1S(C)=O c1(C(N2CCCC(CN(C(Cn3c(C)ccn3)=O)C)C2)=O)cc2sccc2cn1 c1(OC)ccc(CC(=O)NCC(C2CC2)N(C)C(c2ccsn2)=O)c(C)c1 C=C(CNC(=O)C(Cn1cccn1)NC(=O)CC1OCCCO1)C(F)(F)F C1(CC(=O)OC)CCCCN1C(=O)CC1C2CNCC12 C1(C(N2CCCC(N(C(C3N(C)CCCC3)=O)C)C2)=O)CC(=O)C12CCCC2 C1(C(N2CCCC(N(C(=O)CC(F)(F)F)C)C2)=O)CCC([N+](=O)[O-])CC1 c1(C(=O)NCC(C)CNC(=O)CCCCN(C)C)c(Br)nc2n1CCOC2 N1(C(C(c2cccc(C#N)c2)C)=O)CC(NC(c2n[nH]cc2Cl)=O)CC2(CC2)C1 c1(C(N(CCCCNC(C2CCCC23CC3)=O)C)=O)cnc2ccc(F)cn12 C(=O)(CCCc1cccs1)N1CC(CC(C)NC(=O)C=C2CCC2)C1 Cc1nc(CC(C)C)c(C(=O)NCCCCNC(=O)COc2ccc(O)cc2)s1 C1(CNC(CC=C)=O)CN(C(c2c[nH]cc2Br)=O)CCC12CCC2 N1(C(C)=O)CCCN(C(C23CC2CN(Cc2ccc([N+](=O)[O-])[nH]2)C3)=O)CC1 N1(C(C(C(C)C)OC)=O)CC2(CCCN(C(=O)C3=NOC(C4(O)COC4)C3)C2)C1 C1(CCN(C(C)C)C(CC(O)Cn2cccn2)=O)CCCC1 c1(C(N(CC(CN(C(CCOCC)=O)C)O)C)=O)cc2ccccc2nn1 C(C)(C)(CCCCC(=O)N1CCC(NC(C2(CC3CC3)CCC2)=O)CC1)OC N1(C(C(c2cnn(C)c2)OC)=O)C2CCC1CN(C(=O)C(C)CCN(C)C)CC2 C12(C(=O)NCC3(O)CN(C(C4(CN(C)C)CCCC4)=O)C3)CCN(CC1)CC2 N1(C(C2(C=C)CCC2)=O)CCCOC(CCNC(c2cc(SC)ccc2O)=O)C1 Cc1c(C(=O)NC23CC(NC(=O)NC4(C(F)(F)F)CCC4)(C2)C3)cccc1Br C(=O)(CCCC1CC1)NC(CNC(C(C)n1cccc1)=O)C N1(C(=O)NC2C(C)(CC)C2)CCC2(C=CCO2)C1 N1(C(=O)Cc2ccc(Cl)cc2)CCCCC1C1CCN(C(=O)C(O)CC2CC2)C1 c1(-c2nc(CO)nn2Cc2ccc(OC)cc2F)ccc([N+](=O)[O-])nc1 Cc1cc(=O)n(C)nc1C(N1CCC(NC(=O)C(F)C(C)C)C(F)C1)=O c1(C(=O)NCC2CCN(C(C(CCOC)C)=O)C2)cc(Cl)cc(C)c1N c1(CC)ncc2c(n1)CC1CCC2N1C(c1cc2ccccc2[nH]1)=O Cc1cc(C=CC(=O)NCCN(C(C2CCCCC(=O)N2)=O)C(C)C)ccc1F N1(C(c2cc(-c3n(C)cnc3)[nH]n2)=O)CCCC1(C)C(N1CCCC1(C)CO)=O N1(C(C2N(C)CCC2)=O)C2CCC1CC(NC(=O)CSCc1csc(=N)[nH]1)C2 c1(C(N2CC(CCNC(c3cccc(C)n3)=O)C2)=O)cc(C)nc2onc(C)c12 N1(C(C2CC3(CC(=C)C3)C2)=O)CCC2(C1)CN(C(c1cccnc1CC)=O)C2 C(=O)(C(CCC1CCC1)NC(C12CC(C#N)(C1)C2)=O)NCC(COCC)C C1(NC(C2=C(C)OCCS2)=O)CCC2(CC1)CN(C(C1(C)CC1(F)F)=O)CCO2 c1(NC(N)=O)ccccc1C(=O)NC1CC(CNC(C2CCNC2=O)=O)CC1O c1(-c2cn(C(CNC(c3c(CC)cco3)=O)C)nn2)ccc(OC)cc1OC N1(C(c2ccnn2CCOC)C(=O)NCCCC(=O)OCC)CCN(C=O)CC1 c1(C(C)(C)C)nc(=NC2CC3CN(C(c4ccc5nccnc5n4)=O)CC23)s[nH]1 CP(C)(=O)C(CC(=O)NCCNc1cccc2ccncc12)P(C)(C)=O c1(C(=O)NCCn2cc(CCC(C)=O)nn2)cc(C)nc2ccc(C)cc12 CC1COCCC1N(C)C(C1(C)C=CCN1C(=O)Cc1cn[nH]c1)=O C1(NC(C2CN(CC)C(=O)C2)=O)CCCCN(C(C2CC3(CC3)C2)=O)C1 C1(SCCc2ccnc(NC3C(OCCC)COCC3)n2)Cc2nccnc2C1 c1(OC)c(COC2CCCN(C(c3cc(OC)cc(F)c3)=O)C2)cccc1F c1(C(=O)NCCN2CCN(C(C3CCCO3)=O)CC2)cc2ncccc2s1 N1(C(C(C)OCCOC)=O)CC(C)(C)CCC1CNC(c1nc(C)nn1C)=O N1(C(C2N(C)CSC2)=O)CC(C2CCCCN(C(c3occc3C3CC3)=O)C2)C1 Cn1nc(C(F)F)c(C(N2CCOCC2CC2CCCO2)=O)c1C#N c1(C(=O)NCC2(F)CCC(NC(CC(C)O)=O)C2)cc([N+](=O)[O-])cnc1N N1(C(c2c(CC)c(N(C)C)ccc2)=O)CCC(CNC(=O)C(F)CC)C(F)(F)C1 Cc1ccc(Br)cc1CC(=O)Nc1cccnc1N1CCCCC1 C1(C(N2CCC(CN(C(c3c(C)ccnc3)=O)C)C2)=O)OC2CCC1CC2 N1(C(C(F)OC)=O)CC(CNC(C2CCCOC2)=O)OC(C)(C)C1 C1(NC(Cc2cc(C)on2)=O)CN(C(=O)CC2CCCNC(=O)C2)CC1(C)C N1(C(COCCC(C)C)=O)CCOCC1CNC(c1cnccc1C(F)(F)F)=O c1(C(=O)NCC2(CCNC(C3C(C)OCCC3)=O)CC2)cc2c(s1)CCCCC2 Cc1ccc(C(=O)NC2CCN(C(=O)CCn3ncn(C)c3=O)CC2)c(F)c1 N1(C(c2cnc(C3CC3)s2)=O)CCC2(CCC2)C(CNC(C2(C(F)F)CC2)=O)C1 Cc1ccc(Cl)c(C(N2CCCCCC(NC(c3cc(O)ncn3)=O)C2)=O)c1O c1(CCC(=O)NC2CC(C)(NC(C(CC)C#N)=O)C2)ccc2ccccc2c1 C=CC1(NC(C2C3CN(C(C4CN(C5CCC5)C4)=O)CC23)=O)CCCC1 c1(C(=O)NC2(C)CCCN(C(=O)Cc3nnc(S)nc3O)C2)cccc2c1CCO2 c1(C(=O)NC2C(CO)CCN(C(CCCCC#C)=O)C2)c(O)cc(Cl)cc1Cl N1(C(C2CCC(N(C)C)CC2)=O)CC(NC(C2(F)CCOC2)=O)CC(F)C1 Cn1nc(NCc2cccc3ccc(Br)nc23)c2cc(Br)ccc12 Cc1nc(C2CC2)sc1CC(=O)N(C)CCNC(C1CC2CC2C1)=O CC1=NOC(CC(N2CC(O)(C(C)NC(=O)CCc3cnn(C)c3)C2)=O)C1 c1(OC)c(C(N2CC(CCNC(=O)COc3ccccc3)C2)=O)cnn1C c1(C(=O)NCCCCCCNC(C(C=C)(F)F)=O)c(C)cccc1N C(=O)(C1OCCc2ccccc21)N1CCN(CCNC(CC(CC)(C)C)=O)CC1 n1(CCNC2CCN(C(C3N(C(CC)=O)CCC3)=O)C2)ccc2ccccc12 Cc1cnc(C(=O)NC2CCC(NC(c3ccc(C(N)=O)o3)=O)CC2)cc1Cl c1(C(=O)Nc2cc(O)nc(-c3ccccc3)n2)cc2n(c1)CCNC2 Cc1cc2sc(C(=O)NCC3CN(C(=O)CCCc4ncco4)CCO3)cc2s1 N1(C(c2c(CC)n(C)nn2)=O)CCN(C(C2(C)CCN(C)C2=O)=O)C(COC)C1 c1(OC)ccc(S(N)(=O)=O)cc1C(=O)NCCCCNC(=O)C(C)OCCN(C)C CC(CC1CCC1)C(=O)NCC=CC(N1CCC1CN=[N+]=[N-])=O N1(C(CCC2(NC(C3(OC)CCSC3)=O)CCCC2)=O)CCCCC(F)(F)C1 C1(NC(CN2C(C)CCC2)=O)CCN(C(=O)CC2CCC(=O)NC2)CCC1CO C1(C(=O)NC(c2ccccc2OC)CC)C2CC(F)C(C2)N1C(c1ccnnc1)=O c1(C(=O)NCC(Cn2cc(C(C)O)nn2)OC)cc(C(F)(F)F)cc(F)c1 C(c1ccc(F)c(C)c1)=CC(=O)N(CCC(C(C)C)NC(C(CC=C)CC)=O)C N1(C(CCCCC#C)=O)CCCC(C2CN(C(c3csc4nccn34)=O)C2)C1 c1(C(=O)NCC2N(C(CCOCC)=O)CCCC2C)c(C)nc(C2CC2)nc1S c1(C(=O)NC(C(=O)NC)C)cc2c(s1)C1(CCN(CCN=[N+]=[N-])CC1)OCC2 N1(C(c2csc(C)c2C)=O)CC2CC(NC(=O)CCCN3CCCC3)C(C2)C1 c1(NCC2C(C(F)(F)F)CN(C(C(COC)(C)O)=O)C2)nc(C)ccc1C#N C(=O)(C(F)C(C)CNC(=O)Cc1c(C)cnn1C)NCC(C#C)OC N1(C(c2n(CCC)ncc2)=O)CC(CNC(C2CC(CCO)C2)=O)CC(C)(C)C1 C1(NC(CCc2[nH]c(=N)sc2)=O)CC2CC(C1)N(C(c1ccc(Cl)c(F)c1)=O)C2 C(CCCCC(=O)NC(c1ncc(C)s1)C)N(C(C(C(C)C)SC)=O)C C1(CSc2nc(NC(N3CC(C)(CS(C)(=O)=O)C3)=O)[nH]n2)CC(=O)NC(=O)C1 C1(NC(C2(C#N)CC(C)C2)=O)CN(C(=O)CC2CCC(=O)NC2)CC2(CCC2)C1 c1(OC)cc(Br)c(C(=O)NC2CN(Cc3cc4ccccc4o3)C2)cc1O C(=O)(C1=COCC1)NC(C1CN(C(c2ncoc2-c2cccc(Br)c2)=O)C1)C CCC(=O)N1CC(NC(C(C)(C)O)c2ccccc2)CO1 c1(OCC)ccc(C(=O)NCC23CC2CN(C(=O)CCC(N)=O)C3)c2ccccc12 c1(C(N(CC(CNC(C=Cc2c(C)ccs2)=O)C)C)=O)c(F)ccc2ccoc12 CC1(C)CCC(CCNC(c2ncc(Br)s2)c2nnnn2C2(C)CC2)C1 c1(NC(C2N(C(c3c(SC)nccc3)=O)CC2)=O)cc(F)cc(F)c1Cl c1(OCCCN(CCC)C(C2CC23CCOC3)=O)ccc(F)cc1 C1(C(=O)NCC(C)(C)NC(c2cc3cnccc3o2)=O)CCCC2CCCN12 C1(NC(C(C)N(CC(F)(F)F)C)=O)CC12CCN(C(=O)CS(N)(=O)=O)CC2 C12(NC(C(C)NC(CC)=O)=O)CCCC1(F)CN(C(c1c[nH]cc1CC)=O)C2 N1(C(c2cc(CC)[nH]n2)=O)CCCCC(C(=O)NC(C)(CC)CC)C1 c1(CNC(=O)NCC2(C)CN(C)C(=O)C2)nc2ccccc2[nH]1 CCCC(C(=O)OC)C(=O)N(C1CCN(C(=O)C(c2ccccc2C)(F)F)C1)C C(C(CC1CCCC1)C(=O)NCCNC(C=NC(C)=O)=O)N(C)CC c1(C(=O)NC2(CF)CCN(C(Cc3c(C)cnn3C)=O)C2)cc(S(C)(=O)=O)cs1 C12(CNC(CC3(C)CC3F)=O)CCC(CC1)N2C(=O)Cc1cc(C2CC2)nn1C Cc1cc(F)cc(C)c1C(N1CC(NC(c2cn(C)nc2C2CC2)=O)C1)=O Cn1nnc2c(C(N3CC(NC(c4cc(N)c(N)cc4F)=O)C3)=O)ccnc12 c1(OC)cc(C(=O)OCc2nc(OC)cc(C(F)F)n2)cc(C2CC2)c1 c1(OC)ccc(OC(C(=O)NCC2(NC(=O)C(C)OC)CC2)CC2CCC2)c(F)c1 c1(CN(CCCNC(c2ccc(C)s2)=O)C(C)=O)ccc(F)cc1 Cc1nc(=N)[nH]cc1C(N1CCC(CNC(c2sccc2C)=O)C(C)C1)=O c1(C(N2CC3C(NC(c4ccc(C)cc4N)=O)C3C2)=O)cnc(O)n(C)c1=O c1(N2CC(C)=C(C)CC2)nc2cc[nH]c2c(=NC2CCC3(CCC3)C2)[nH]1 C(=O)(C(O)CCS(C)=O)NCCN(C(CC(C)C(F)F)=O)C N#Cc1cnc(N2CC(N3CCN(C(c4ns[nH]c4=O)=O)CC3)C2)c(Br)c1 N1(C(c2c(F)cc(C)c(F)c2)=O)CCOC2(CCCN(C(C3CC(C)C3)=O)C2)C1 Cc1ccc(F)c(C(=O)NCCC2CC(F)(F)CN2C(=O)C(C)CF)c1 N1(C(CC)=O)C(C)CC2CN(C(=O)CCC3(C)CC3(F)F)CC12 C1(NC(=O)NC(c2nc3c(s2)CCCC3)C)CCCCC12CCC2 c1(CNC(=O)Nc2n(C)nc(C(C)=O)c2I)cc2ccccc2nc1C c1(C(N(CC(CNC(C2(CCCC)CC2)=O)C)C)=O)nnc(O)c2ccccc12 C(=O)(CC(F)(F)C(C)C)OCCCc1ccc(OC)cc1 N1(C(c2c(COC)cc[nH]2)=O)CCCC1C1CCCN1C(=O)CCCC Cc1cc(C(N2CC(O)(C(C)NC(=O)C(C)(C)CF)C2)=O)cnn1 Cc1cnc(C(=O)NC(Cc2cn(Cc3ccccn3)nn2)CC(=O)O)c(C)c1 C12(CNC(C(C)c3cccs3)=O)CC(CCO1)N(C(c1ccc([N+](=O)[O-])o1)=O)C2 N(C1CCc2ccccc21)C(C(C1(C)CC1)NC(C1C(C(C)(F)F)C1)=O)=O N1(C(c2ccc(SC)s2)=O)CCCC(C)C1CCNC(c1ccc(CO)cn1)=O c1(C(=O)NC2CCN(C(C3(CCOC)CCCC3)=O)C2)c[nH]c2cc(F)ccc12 Cn1cc(S(=O)(=O)NCC(=O)NC2(c3ccc(Br)cc3)CNC2)cn1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(NC(=O)CC(C)C)C2 C1(NC(c2cn(C(C)C)nc2)=O)(CO)CCN(C(C2CC2Cl)=O)C1 c1(C(=O)NC(c2cccc(Cl)c2)CNC(C(CC)F)=O)oc(CC(C)C)nc1C N1(C(Cc2c(OC)nccc2)=O)CCC2C(CCCN2C(C2CCOC2=O)=O)C1 C(=O)(N=c1[nH]n(C)cc1C(C)C)N1CCC(NC(c2n(C(C)C)ncc2)=O)C1(C)C c1(C(=O)NC(CC(C)C)CNC(C2CCC3CC23)=O)cccc(F)c1Br c1(C(=O)[NH+](CC2C(CNC(C(CC#C)O)=O)C2)[O-])c(C)nc(C2CC2)nc1O.C1CC1 S(=O)(=O)(c1c(C)cc(C(F)(F)F)cc1C)N1C(c2ncc(C)o2)CCCC1 C1(C(N2C(C)C(NC(=O)CN3CCC(CO)CC3)CC2)=O)CCC(F)(F)CC1 N1(C(c2c(OC)cncn2)=O)CCC(C(=O)NC2(C)CC=CC2)C12CC2 C1(C(=O)NCCNC(CC=C)CNC(=O)C=CC(=O)NC)CCCC12CCC2 N1(CC(=O)NCC2CCN(c3ccc(F)cc3)C2)CCC(F)(F)CC1 C=CCCCC(C(=O)NCC(F)(F)COC)NC(C12CCCC1C2(F)F)=O C1(C)(C(=O)NCCCN(C(c2c(OC)ccc(CO)c2)=O)C)CCC(=O)N(C)C1 C1(CNC(CCC(C)(F)F)=O)CN(C(=O)C(F)C(F)(F)F)CC1(F)F C1(CNC(c2cnc(-c3cccnc3)s2)=O)CN(C(C2CCO2)=O)CC1(F)F c1(CC)nc(C)n(C)c1C(=O)NC1CCCC1NC(=O)CCP(C)(C)=O Cc1ccc(Br)c(NC(C2(C)CCCN2C(c2cc[nH]c2)=O)=O)c1F C1(C)(C(=O)NC2CN(C(CCCc3ccc(C)cc3)=O)CC2O)CCC(O)CC1 Cc1cccn2c(CC(=O)NCC3CCCN(C(C4CCCSS4)=O)C3)cnc12 C1(NC(CN(C2CCC2)C)=O)CCC(CNC(=O)Cc2ncsc2Cl)CC1 C1(CC(=O)NCC(CC)C)C(C(=O)Nc2ccccc2)CC1O CC1(C)CC(CNC(=O)CC2CCC(F)(F)C2)N(C(=O)CC2OCCCO2)C1 C1(NC(C2C3CCN(C(C4CCCSC4)=O)CC23)=O)CCCCCC1F C1(C(N2C(C)(CC(=O)Nc3cc(C4CC4)ncn3)CC2)=O)CC2C=CC1C2 CCCC(O)CC(=O)NC1(COC)CN(C(=O)C(C(C)C)n2cnc(C)c2)C1 C1(C(N2CC(NC(C3(S(N)(=O)=O)CC3)=O)C(C(F)F)C2)=O)(OCC)CCCCC1 C(=O)(C(CC(N)=O)NC(C12CCCCC1C2)=O)NCC1(CC)CC1 C1(C(=O)NC(C=C)CO)(NC(=O)CC(C)C2CC2)CC(F)C1 c1(CSC)cccc(C(=O)NCC2CC(C)N(C(c3coc(C(C)=O)n3)=O)C2)c1 CC1(C)CN(C(c2sc(C#N)cc2Cl)=O)CCC1NC(C1CCCOC1)=O N1(C(CSCc2nnc(C)s2)=O)CCC2(NC(=O)CSC3CCOC3=O)CCCC12 C1(NC(C2COC3COCC23)=O)CCCCN(C(c2csc(O)n2)=O)C1 C1(CN(C)C)CCC(C(=O)NC2CN(C(c3cscn3)=O)C2)O1 C(CN=c1nc(N2CCCC(c3cnc[nH]3)C2)c2ncccc2[nH]1)C1C(F)(F)C1 c1(C(=O)NCC2(c3nccs3)CC2)ccc(-n2cncn2)cc1Cl c1(C(C(=O)NCCOCC(C)C)NC(C=CC(CC)C)=O)c(C)cccc1Br CC1CN(C(=O)CSCCC(F)(F)F)CC1CC(N1CC(O)(C(=O)C2CC2)C1)=O c1(CNC(=O)NC2(C)CCCOC2)ncc(Br)c(Cl)c1Br N1(C(C(C)CBr)=O)CCC(CCNC(=O)CN2C(=O)CSC2=S)CC1 c1(C(=O)NCC(C2CC2)NC(=O)CCc2ncccn2)cncc(C2CC2)c1 n1(CCC(=O)Nc2nnc(C(=O)OC)s2)c(O)nc2ccccc2c1=O C1(C(N2CCC(C3CCCO3)C2)=O)(NC(C2CC2[N+](=O)[O-])=O)CCCC1 C1(CC)CN(C(=O)C(C)(CC(F)(F)F)c2ccccc2)c2ccccc2O1 CC(CCC(=O)NCCNC(C1CCc2nccn2C1)=O)S(C)(=O)=O N12CCOC(C1)C2=O.C(C(C)S(C)(=O)=O)NC(c1nc(COC)oc1)=O c1(C(=O)NC2CC(C)N(C(=O)CCS(C)(=O)=O)CC2)cc(S(N)(=O)=O)co1 Cc1cn(C)nc1C(N1CCN(CC(=O)NC2(C(N)=O)CC2)CC1)=O N1(C(c2nc(C)sc2Br)=O)CCC(NC(=O)Cc2cc[nH]c2)CC1C C1(OC)CN(C(C2CCSCC2)=O)CC1C(=O)NC1(C)CC=CC1 Cc1c(C(=O)NCC2(CNC(c3nn[nH]c3Cl)=O)CC2)nn(C)c1N c1(CCNC(CCC(=O)OCCOC(C)(C)C)=O)cc(F)ccc1F N1(C(CCC#CC)=O)CCCC(C2CCCN(C(c3ccc(CC)s3)=O)C2)C1 CCCCCCC(C)C(=O)N1CC(CNC(c2cc(COC)[nH]n2)=O)C(O)C1 C12(C(=O)NC(c3ncccn3)C)COCC1CN(C(c1ccc(Cl)o1)=O)C2 c1(C(N2CC(F)(CNC(C3CC(=C)C3)=O)C2)=O)cc2cccc(Cl)c2nc1C C1(c2nnnn2C(C)C)(Nc2c(C)c(F)ccc2)CCC2(CCNC2=O)C1 C1(N(C(C(C)OCCN(C)C)=O)C)CC2CC1N(C(C1CC3(C1)OCCO3)=O)C2 C1(NC(c2ccc(OC)nc2)=O)CCN(CCn2ccc(=O)cc2C)C(C)C1 C(=O)(C(C(C)(C)C)OC)NC1C(C(N2CCCC(CC)C2)=O)CCCC1 C(c1cnccn1)=CC(=O)N(C(C)CN(C(=O)CCCc1cncs1)C)C c1(NCC2CC2)ccc(OC)nc1.c1(COCC(=O)NCC(CC)N)ccnn1C N1(C(c2cnc(OCC)nc2)=O)CCCC(O)(CNC(c2nn(C)cc2N)=O)C1 O(C1CCCc2ccccc21)CCNC(=O)C(=O)NCC1(CS(N)(=O)=O)COC1 c1(C(C(=O)NCC)OC)ccccc1CC.C1(=O)CN1C(C)=O CCCCCCCCCC(=O)NC1CCN(Cc2ccc(OC)nc2)CC1O C(=O)(CCCC(=O)NC1CC2CC(C1)N(C(c1ccc3cnsc3c1)=O)C2)NC C1(CC)CN(C(c2ccnc(OC(C)C)c2)=O)CCC1NC(=O)OCC c1(C(N2C3CC(CC(NC(CCCCC=C)=O)C3)C2)=O)cccc2c1CCCC2 CC(C)CC(=O)NCCC(C)(C)NC(=O)C(C)OCC(=O)OCc1ccccc1 C1(C(N2CC3(CCCC3)C2c2ccccc2)=O)CCC2(CCNCC2)CC1 c1(NC(c2cscn2)C)ccc(S(=O)(=O)NC(C2(C)OCCO2)C)c(Cl)c1 N1(C(C2CC(C)(C)C2)=O)CC(NC(C2(O)CC(F)(F)C2)=O)CC12CCCCCC2 Cc1cc(C(=O)NC23CC(C(=O)N(CCC(C)C)CC(C)C)(C2)C3)cc(F)c1 N1(C(C(CCCC)NC(C2CC3(CCC3)C2)=O)=O)CCC2(CCCCO2)C1 N1(Cc2cccc(CC)c2)CCCC2(CCN(C(c3c(O)cccc3Br)=O)CC2)C1 C(C)(C(C)(C)C(=O)N(C1CC(CO)C1)C)NC(C(C)C)=O CC1=C(C(=O)Nc2ccc(N3CCC(C(=O)N(C)C)CC3)nc2)SCCO1 C1(C(N(C(C)CNC(c2cncc(-n3cnnn3)c2)=O)C)=O)OCCOC1(C)C C1(=CC(=O)NCC2C(NC(c3occ(C)c3C)=O)C2)CCOc2ccccc21 CCCC(C(=O)N1CC(CC(C)(C)CNC(=O)C=C(CC)CC)C1)OC C(CCF)(C(=O)NCCC(=O)NO)NC(CCc1n(C)ccn1)=O Cc1cc(C(=O)NCC2CC2CNC(=O)CN2CCC(C)C2)c2ncccc2c1 N1(C(CCC2(NC(C3N(C)C(=O)OC3)=O)CCCC2)=O)CCN(C)C2(CC2)C1 c1(C(=O)NC2(C)CC(NC(C3(C)CC4CCC3C4)=O)C2)cc(O)c2ccoc2c1 N1(C(C(F)OC)=O)CCC2(CC1)CN(C(C1CCC3(CC3)C1)=O)CCO2 c1(C(=O)NCCCN(C(C(CC)n2cncn2)=O)CC)nn2c(c1C)CCCC2 C1(O)(C(C)NC(C2C3COCC23)=O)CCN(C(=O)C(F)(F)c2ccncc2)CC1 CC(C)(CCC(=O)NCC1CCC1NC(C1(CN2CCCC2)CC=CC1)=O)OC N1(C(CCCN(C)C)=O)CC(C(C)(C)C)CC(CNC(=O)C(C)(C)CCF)C1 C12(CCC)CN(Cc3nc(-c4ccccc4)co3)CC(CO)(C1)C2 C1(C(=O)O)CCOC(C)(CNC(C23CC(C2)C(C(F)(F)F)O3)=O)C1 C(=O)(C(=O)C(C)(C)C)NCCNC(c1oc(C)c(Br)c1)=O CC12CCN(C(C3CN(S(=O)(=O)F)C3)=O)CC1C2(Cl)Cl N1(C(C2(CC)COC2)=O)CCN(C(c2ccc(OC)cn2)=O)CC(C)C1 C1(NC(CC=CCNC(C2N(C)CCOC2)=O)=O)Cc2ccccc2C1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCN(C(c2ccc(N)c(C)c2Cl)=O)C(C)C1 Cc1cnc(CNC(C2(NC(=O)Cn3ccc(C)n3)CC2)=O)c(C)c1 N1(C(C(C)SC)=O)CCCCC1C(=O)NCC1CCC(C)CC1 Cc1cc2cccc(CNC(C3CCC4(CN(CC5CCCO5)C4)O3)=O)c2[nH]1 C1(CC=C)(NC(=O)C(F)C(F)(F)F)CCCN(c2cc(CC)nc(Cl)n2)C1 c1(C(=O)NC2CN(C(c3c(OC)csc3)=O)CC(O)C2)ccnc2cc[nH]c12 Cc1ccc(OCc2cc(Br)cc(I)c2)c(-c2ccc(C(N)=O)cc2)c1 c1(CC)cc(CC(N2CCCC2c2cn(CC3CCCC3OC)nn2)=O)no1 C12(CNC(=O)C=CC3CCC3)CN(C(C3CC4C=CC3O4)=O)CC1(C(F)(F)F)C2 C1(NC(=O)CC2CCCC2)CC2CCC1N2C(c1cnn(CCF)c1)=O N1(C(C2CC(C)=C(C)CC2)=O)CC2CCN(C(=O)C=C3CCOCC3)C2C1 c1(C(N(CCC(C)NC(c2c(CC)ccs2)=O)C)=O)ncc(CC)cn1 C1(NC(CC2(O)CCN(C)CC2)=O)CCC2CN(C(=O)CSCC(N)=O)CC2C1 c1(OC)cc(C(=O)NCC(C)CNC(C2C(C)C2(F)F)=O)cc(Cl)c1OC C1(CNC(=NCCC(=O)NC)NCCCC(=O)N(C)C)CSc2ccccc2O1 c1(C(N(C(CNC(c2c(CC)[nH]nc2Cl)=O)C)C)=O)cc2c(cnn2C)nc1O C(=O)(CCCCCCCC(=O)Nc1cc(F)c(Br)cc1C)OC CC(F)(F)C(F)C(=O)N1CCCCC(CCC(=O)NCCOC2CCOC2)C1 c1(CN2CC(CC)N(C(c3nc(C(=O)O)cs3)=O)CC2)c(F)cccc1[N+](=O)[O-] N1(C(c2ccns2)=O)Cc2cccn2CC(C(N2CCc3c(O)n[nH]c3C2)=O)C1 C(c1cnccn1)=CC(=O)NC1CC1N.c1(C(N2CCOCC2)=O)ccc(C=O)o1 C1(N(C(C=CSC)=O)C)CCN(C(=O)C(N2CCCCCC2)C)CC12CC2 c1(C(=O)NCC(CC=C)NC(C2OCCC2C)=O)csc2ccccc12 Cc1cncnc1C(=O)NCC1CC1NC(=O)Cn1cccnc1=O c1(C(=O)NC2C3(CCC(NC(C=CCC)=O)CC3)C2)c[nH]c2nccc(Cl)c12 C1(N(C(=O)CN2CCSCC2)C)CN(C(c2cncc(N)c2)=O)CC1O C(N=c1cc(N)c(Br)c[nH]1)C1CCC(CCCC)O1 c1(C(=O)NC2(OC)CN(C(C(C(=O)OC)OC)=O)C2)cc(OC)cc2c1CCC2 N1(C(C(C=C)O)=O)CCC(N2CCC(NC(=O)CSC3CCS(=O)(=O)C3)C2)CC1 N1(C(=O)NCCN(CC)Cc2cccc(Br)c2)CCCC2(C1)CC2(F)F C(=O)(CS(=O)(=O)CCO)N(CC(CN(C(c1cc(OC)cc(Cl)c1)=O)C)O)C C(=O)(C(C)Cc1ccncc1)NC(CN(C(COCCOCC)=O)C)(C)C N#CC1(C(=O)NC2(CC(N3CCCCC3CCCO)=O)CC2)CC=CC1 C1(CNC(=O)CC2C=CCC2)(NC(c2cccc(=O)o2)=O)CCC(F)(F)CC1 c1(NC(C(C2CN(C(=O)Cc3c[nH]nc3O)C2)OC)=O)cnn(C)c(=O)c1 c1(C(N2CC(NC(c3ccc(CC)[nH]3)=O)C(F)C2)=O)cc2cccnn2n1 N1(C(C2CCCN(C(c3cc(OC)ncc3)=O)C2)=O)CC2CCCC(C2)C1 c1(C(N2C(C)CC(NC(=O)CC3=CCCCC3)C2)=O)ccc2c(c1)NC(=O)CCN2 C1(C(N2CCCC(CCC(=O)NCC3CC3Cl)C2)=O)C2CCCCCCC12 C(CO)(CCCCNC(C1CC1c1cnc[nH]1)=O)NC(C(CN(C)C)(C)C)=O N1(C(C2CC(C)(CC)C2)=O)CCCC(NC(C2(C)CCCCO2)=O)CC1 c1(C(=O)NCC(C)N(C)C(c2ccc(C3CC3)nc2)=O)cc(C2CC2)n(C)n1 C1(C(=O)NC2CN(C(=O)C(C)=CC(C)(C)C)CC2SC)(OCC)CCSCC1 c1(C(=O)NCC2CCCC2NC(C2CC23CCC3)=O)cccc2nccn12 N1(C(C(N2CCCC(C)C2)=O)=O)CCN(C(=O)Cc2cnsc2)CC1CS(C)(=O)=O c1(OC)nc(Cl)ccc1C(=O)N(C)CCNC(c1cc(-n2ccnc2)ccn1)=O C1(CCNC(CCC(CC)C)=O)CCN(C(=O)CCCCC(N)=O)CC1(F)F C1(CN(C)CCOCCN(c2ncc(C3CC3)o2)C)CCS(=O)(=O)CC1 c1(C(N2CCC(N(C)Cc3ncc(OC)nc3)C2)=O)n[nH]c2ccc(Br)cc12 c1(CC(=O)NC2(CN(C(C(C)OCC)=O)C)CC2)cncc(O)c1 N1(C(C2(C(C)C)CCN(C(=O)CC(C)N(C)C)C2)=O)CCC2CC1C(=O)O2 c1(C(=O)NC2CC3CN(C(CC(C=C)C)=O)C2C3)c(F)ccc(OCC)c1F c1(C(=O)NC(C2C(C(=O)NC3(C(C)C)CC3)C2)C)cc(O)n(C)n1 C1(NC(c2c(C)nco2)=O)CCCCC1CNC(c1ccnn1CC#N)=O c1(CC(N2CCC(NC(C(COC)(F)F)=O)C2)=O)c[nH]c2cccc(C)c12 C(=O)(C1=NN(C)C(=O)CC1)N(C)CC1CCN(C(=O)CC23CCCN2CCC3)C1 C(=O)(C#Cc1ccccc1C)NCc1cccc(CSC)c1 Cn1nccc1CC(N1CCC(NC(=O)CCNC(=O)Nc2ccoc2)C1)=O N1(C(C2CCCN(C(CC3N(C)CCC3)=O)CC2)=O)CC2(CCC(=O)N2)C1 c1(OC)cc(N2CC(CO)(CNC(c3cccc(C)c3F)=O)C2)ccc1[N+](=O)[O-] C(CN1CCCC1)(C(=O)NCCCF)N(C(=O)CCNC1CC1)C C1(NC(Cc2ccc(C)cc2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC1C(C)C c1(CC)cc(C)c(C(=O)NCCCN(C(c2cc(C(F)F)cs2)=O)C2CC2)o1 C1(c2nn[nH]n2)(CCN(CCC)C=O)CCOC1.C(C)(C)(C)S.C1(=O)NCCO1 c1(C(c2nc(-c3nnc4n3CCCC4)no2)OC)cn(C)c(=O)c2ccccc12 C(=O)(CC(C)(O)c1ccccc1)N1CCC(NC(C(c2cn(C)nc2)=O)=O)C1 CC(C)C#CC(=O)NC(c1ccccc1F)CNC(c1cc(C(N)=O)cs1)=O N1(C(C(COCC)C)=O)CC2CC(C(=O)NC3(CN(C)C)CCCC3)(C2)C1 C1(CNCC(C)(C)c2cncs2)N(C(=O)OC(C)(C)C)CCCC1(C)C C(=O)(C(O)P(C)(C)=O)N(C)CC1CCN(C(=O)C(c2cc(F)cc(Cl)c2)=O)C1 CCC(C(=O)N1CC(OC)C(NC(C2CNC(=O)C2)=O)C1)C(C)(C)CC c1(CC(=O)NCC(CNC(CC(C)OC)=O)F)ccc(Cl)c(F)c1 c1(CC(C)NC(CC2CCN(C(Cn3nnc(C)n3)=O)C2)=O)ccc(Br)cc1 C1(CC)CC(C(=O)NC2CC(c3ccc(OC)cc3)C2)CCN1 CCCCCCC(=O)NC1CN(C(=O)COCc2ccnn2C)C2CC12 C1(NC(CCOc2c(C)cccc2)=O)CCN(C(=O)CN2CCOCC2)CC1C c1(Cc2nc(COCCC)n(-c3ccc(F)cc3)n2)cc2ccccc2o1 N1(Cc2scc(C(=O)OC)n2)CCN(N2CCOC(C3(O)CC3)C2)CC1 CCCCC(C)C(=O)N1CCC(NC(c2cn(C)nc2C2CCCCC2)=O)C1 C1(S(C)(=O)=O)(C(=O)NCCCCCCNC(CC2(OC)CCOC2)=O)CCC1 CC(C)(C#N)CCC(=O)N1CCC2(CC1)CC2NC(=O)Cc1cncnc1 c1(C(N2C(CC)CN(C(=O)C(C)(F)c3ccon3)CC2)=O)nc2ncccn2n1 N1(C(=O)NC(C2CCOCC2)CCO)CCCC2(C1)C(O)CC2O C1(C(=O)NC2CN(C(CNC(CC(C)(C)C)=O)=O)CC2O)CCOC(C)(C)C1 c1(C(N2CCCC(CN(C(c3ccc(C)[nH]3)=O)CC)C2)=O)cccc(=O)n1C N1(C(c2ccc(SC)s2)=O)CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C(C2CC2)C1 N1(CC(N2CC(C(C(=O)NCC(C)O)(C)C)(O)C2)=O)CCCCC1C c1(OC)ccccc1C(C)CCNC(=O)NC1CN(C)C1 C12(NC(c3nn(-c4ccccc4F)ccc3=O)=O)CCC(C1)C(F)(F)C2 CN=c1cc(C(N2CC(NC(=O)C(=Cc3ccccn3)C)CC(C)C2)=O)cc[nH]1 C1(C(N2CC(c3cn(CC(=O)OC)nn3)C2)=O)CC12CCSCC2 c1(C(N2CCCC(C(=O)OCC)(CC)C2)=O)ccn2ncc(CC)c2n1 c1(OC)ccc(C(C)C(=O)NCC(CNC(=O)C(C)(C)C#N)OC)cc1 Cc1ccc(C(=O)NCC2(F)CC(NC(c3occc3C)=O)C2)c(Cl)c1 c1(CNC(c2cccc(CNC(Cn3c(C)ncc3)=O)n2)=O)cc(F)ccc1O c1(OC)cccc2c1C(C(=O)N1CCN(C)C(C(F)(F)F)C1)CC2 N1(C(C2C=CC(=O)N=N2)=O)CC2(CC(N3CCNC4(CC4)C3)C2)C1 c1(NC(CC2CCC(C)N(C(=O)C(N)=NOCC#N)C2)=O)ccc2c(c1)CCC2 C1(CNC(=O)OC(C)(C)C)CCN(Cc2csc(-c3ncccn3)n2)CC(O)C1 Cc1noc(C)c1CNC(=O)COC1CCN(C(c2ccc(=N)[nH]n2)=O)C1 c1(COC(C2CC(CNC(=O)OC(C)(C)C)C(O)C2)=O)ncc(Br)cc1F c1(NC2CCC3CN(C(C(CCCOC)C)=O)CC32)ncnc2c(Br)cccc12 Cc1nc(CC(=O)NCC(C)(C2CC2)NC(=O)CC2CC2(C)C)cs1 c1(CC)ncc(C(=O)NCC2C(C)CCN2C(c2csnc2Cl)=O)c(C)n1 c1(-c2cc(C)oc2)csc(=Nc2cccc(Cl)c2C)n1Cc1nc2ccccc2o1 N1(C(C(CCC)(C)C)=O)CCC(C)N(C(=O)C=Cc2cncs2)CC1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(C)C(NC(=O)Cc2cnnn2C)C1 c1(C(=O)NCC2N(C(c3occ(C(N)=O)c3)=O)CC2)cc(C(F)(F)F)cnc1O C(=O)(C(C(C)C#N)N(CCS(C)=O)C)NCC C(=O)(NN1CCCOC1=O)C1C(N)C1.C12(CCC1)C(=O)NO2 C1(NCC(C(=O)NCC(=O)NC2CCN(S(C)(=O)=O)C2)(C)C)CC2(CCOC2)C1 n1(CC)nnc2c1C(C(=O)N(C1CC(O)C1)C(C)=O)CN(C(=O)C=CC1CC1)C2 C1(CNC(C(CC#C)C)=O)CN(C(c2ccnc(Cl)c2OC)=O)C(C)(C)C1 N1(C(C(C)OCC(C)C)=O)CCC(CNC(=O)CS(N)(=O)=O)C(C)C1 C1(C)(C(=O)NCCCNC(C2N(C(C(C)(C)C)=O)CSC2)=O)CCC(F)(F)CC1 CCCC(C(=O)NCC(N1CCC(OCCOC)CC1)C(C)C)N(C)C c1(C(=O)NCC(C2CCCC2)NC(C2C(OC)CCC2)=O)cc(C)nnc1O c1(N2C3CN(C(c4c(CC)non4)=O)CC2CC3)cccc(OC)c1[N+](=O)[O-] N1(C(CC2CCC(=O)N2)=O)CC(NC(C2Cc3nccnc3C2)=O)C2(CCC2)C1 C1(C(=O)NCC(CC)N(C)C)COCCN1C(c1cnc(Cl)s1)=O C1(C(=O)NC(CNC(C2(c3ccccc3)CC2)=O)C2CCC2)CCNC1=O N1(C(c2c(SC)ccs2)=O)CCN(C(=O)COCc2cccc(C)c2)C(C)C1 C(=O)(C(C)SC1CCC1)N(C(C)CNC(=O)CC1CCCO1)CC c1(C(C)NC(=O)NC2CCC3CC3C2)cc2c(cc1Br)OCCO2 CC1=C(C(=O)NC(CCC2CCC2)C(N2CC(=O)NC3(CC3)C2)=O)COCC1 C1(N(C(CC)=O)C)COCC1C(=O)NC1CC1CNC(=O)Cn1ccnc1C CC(C)(CNC(=O)Cc1ccccc1)CNC(=O)COC1CCOC1.C1(=O)CCN1 C1(CNC(Cc2c(C)nsc2)=O)CN(C(=O)CC2CC2c2ccoc2)CCC1C CC1(C)C(=O)N1.C1(C(=O)OCC=CCS(C)(=O)=O)CC(=C2CCC2)C1 C1(=O)C(CC2CCC2)N1.NS(=O)(=O)NCc1cncs1.C1(C(=O)N)CCN1 C1(C(C)(C)C)CCCCC1NCCNC(=O)NC1COC1 c1(C(N2CC(C)C(O)C2)=O)ccc2nccc(C3=CCN(C)CC3)c2c1 C1(C(N(c2c(CC)cccc2)C)=O)CC(C)CN(C(=O)C=Cc2ccco2)C1 CCC(CC(=O)N1CC(CO)CC1CO)C(C)C C(CC(F)(F)F)N(C(=O)C(C1CCOCC1)NC(=O)CNC(=O)OC(C)(C)C)C C1(NC(CC(C(C)C)O)=O)CC2CCC1N(C(c1cc(F)cc(Cl)c1)=O)C2 c1(C2(F)C(C(=O)N(c3ccccn3)c3cnsc3)C2)ccccc1 N1(C(CCCSC)=O)CC(F)CC1C(=O)NC(C(C)C)c1nc[nH]n1 N1(C(c2c(C)n(C)nc2)=O)CC2CCCC(C1)N2C(C1(CO)CCCO1)=O C1(NC(c2ncc(OCC)nc2)=O)CN(C(C2CCC(C)O2)=O)CC1C1CC1 CC1CN(C(=O)CC2CCCCN2C(c2ccc[nH]2)=O)CCCO1 Cc1ccc(C(=O)NC2CC(n3cc(-c4ccc5c(c4)CC5)nn3)C2)c(I)c1 N1(C(CN(C(C(C)C)=O)C)=O)CC(NC(=O)C(C)(C)CC#N)CC12CCC2 N1(C(c2cc(CC)nnc2C)=O)CC2CCCC2(NC(=O)CN2CCOCC2)C1 CCCCCCCCCCCC(=O)N1CC2(CC(C(=O)NCC3CC34CC4)C2)C1 C1(CNC(c2ccn(CCC)n2)=O)(NC(=O)CC2CCCCN2C)CCCCC1 N1(C(C=CC(=O)OCC)=O)CC(NC(=O)CSc2cn[nH]c2)C2CCCCC12 c1(C(=O)NC2CC(CNC(C(CCC)OCC)=O)C2)ccc2sccc2c1 C1(NC(=O)NC(c2c(-c3onc(C)n3)cccc2)C)CCCC23OCCC2CC13 c1(C(=O)NC(CCCNC(Cc2ccn(CC)n2)=O)C)ncccc1C c1(C(c2n(CC)nnn2)NCCC2CCCO2)cc(Br)ccc1OC c1(CC(=O)NCc2c(C(=O)NC(CN(CCC)C)(C)C)con2)cn(C)nc1C N1(C(C(CC#C)C)=O)CC2CCCC2(CNC(=O)C(CC)=CC)C1 C(CCS(C)(=O)=O)NC(c1ccc(C(F)(F)F)cc1)(c1n(CC)nnn1)C c1(CC(=O)NCCCCNC(c2c(C)ncnc2)=O)cn2cc(Cl)ccc2n1 N1(CC(N2CCOCC(NC(Cc3nnc(C)o3)=O)C2)=O)C(=O)C(=O)N(C)C1=O CC(c1ccccc1)=CC(=O)N(C(CNC(c1cnc(O)c(F)c1)=O)C1CC1)C C1(C(C)NC(c2ncn(CC)n2)=O)CCCCN1C(c1ccccc1F)=O C12(C(=O)NC(CCCNC(C3CCC(C)CC3)=O)C)CCC(O)(CC1)CC2 C1(CC(=O)NCCCCC2N(C(c3n(CC)ncc3)=O)CCC2)CCC12CCC2 C12(NC(c3cc(CNC(c4ncn(C)c4)=O)no3)=O)CCN(CC1)C2 CC1CN(C(c2nn[nH]c2C(F)(F)F)=O)CC1CNC(=O)COC1CCCOC1 C(=O)(C1CCCc2ccnn21)N1C(C)CC(NC(C(CC)O)=O)C1 CCC(C)(CC)C(=O)N(C1CC1)CC1CCCN1C(c1n[nH]c2c1CCC2)=O c1(C(=O)NC2CCN(C(=O)COCCF)C2)ccc2cc([N+](=O)[O-])ccc2n1 C1(C(N2CCC(N(C(c3c(CC)oc(C)c3)=O)C)CC2)=O)CCCC(F)(F)CC1 N1(C(C2CCC3CCC2N3C(=O)C(F)=CC2CC2)=O)CC2C3CCC(O3)C2C1 c1(OC)ccc(C)c(C(=O)NC2CN(C(=O)C3=CSCS3)CC2C)c1 c1(C(=O)OC)cc2[nH]c(C(N3CC4=C(C3)CN(C(=O)C3=C(Cl)CC3)C4)=O)cc2s1 c1(C(N(C(C(N2C(CNC(C)=O)CCC2)=O)(C)C2CC2)C)=O)oc(C)cc1C c1(C(N(C2CCN(C(C(C)NC(=O)NC)=O)C2)C)=O)ccc(C)cn1 C1(CNC(c2c(C)ncs2)=O)CCCCCN1C(c1ncn(C(C)(C)C)n1)=O C(=O)(C1Cc2ccccc21)N1CCC(N2CCN(C(CC(C)F)=O)CC2)CC1 c1(C(=O)NCCC(C)N(C(=O)CC2(C3CC3)CC2)C)oc2ccccc2c1Cl C1(C2(NC(CN(C3CCC3)C)=O)CC2)CCCN1C(=O)Cn1cnnn1 C1(NC(c2ccc(C(C)(C)C)cc2)=O)C2CCC1N(C(=O)C=Cc1ccco1)C2 N1(C(CC(CC)SC)=O)C2CCC1CC(NC(=O)CCCC1CCCO1)C2 c1(-c2cn(C3C(OC)CN(C(c4cnsc4C)=O)C3)nn2)c(Cl)cccc1Cl c1(C(=O)NCCCCc2ccc(OC)cc2)cnc(Cl)c(Cl)c1 N1(C(C2C(C)(C(C)C)C2)=O)CCCC2(C1)CN(C(C1SCCS1)=O)CCO2 c1(C(=O)NC(c2cn(CCN3CCCC3)nn2)C)cc2ccnc(Cl)c2o1 C1(C2CCCN(C(c3cnc(Cl)c(Cl)c3)=O)C2)(NC(CC(COC)C)=O)CC1 Cn1nc(Br)c(C(=O)NC2CC(CNC(=O)CNC(N)=O)C23CCC3)c1N N1(CC)CCCC1C(N1CC(C(C(=O)NC2CC(O)C2OC)OC)C1)=O C(CC(C)(C)C(=O)N1CCCC(CN(C)C(C2CCS(=O)(=O)N2C)=O)C1)OC c1(-c2nc(CC)[nH]n2)cccc(C(=O)NC2CC2NC(=O)CC(C)(C)C)c1 C1(C(N(C)Cc2onc(CC)n2)=O)CN(C(c2cnnn2C2CC2)=O)CC1(F)F C12(NC(c3c(C)cc(C(F)F)o3)=O)CCCC1N(c1ncc(F)cn1)CCC2 c1(N2CCC(CNC(C(C)C3CC3)=O)CC2C)c[n+]([O-])ccc1[N+](=O)[O-] C(N=c1[nH]c(=NCC(C)CN(C)C)[nH]c2ccsc12)c1cccc(COC)c1 C(C(=O)NCC(C(C)C)NC(c1cc(C(F)(F)F)n(C)n1)=O)(C(C)C)SC Nc1nc(Cl)ccc1C(N1CCOC(CCNC(c2cc(C3CC3)on2)=O)C1)=O c1(C(N2CC3(CC(CNC(C(C=C)(C)C)=O)C3)C2)=O)ccc2c(c1)CCCN2 c1(C(=O)NC2COCCN(C(C(C)OC)=O)C2)nc2c(cc1Cl)OCCO2 c1(C(N(CCCCNC(C(C(=O)NC)(C)C)=O)C)=O)cccc2c1OCCO2 C(=O)(C1=CCCOCC1)N1CCC(CCNC(c2c(C)nc(C)s2)=O)C1 Cc1nnc2ccc(-c3cccc4cc(C(N5CC(F)CC5C#N)=O)[nH]c34)cn12 C(=O)(CCCCC(C)(C)C)NC(C(C)NC(c1c(O)ccc(OC)c1)=O)C c1(C(=O)NCC2CN(C(C(CCC#C)O)=O)C2)cc2c(C)cc(OC)cc2[nH]1 C#Cc1ccc(C(=O)NC2CCC(CCC(=O)NC3CC4CCCC4C3)C2)cn1 C1(CC(=O)N(C(CC)CC)CCO)CCCN(C(C2CCOC(C)(C)C2)=O)CC1 C(=O)(C(C)(C)CC(F)F)NCC1(C)C(C)CN(C(c2ccc(SC)o2)=O)C1 C#CCC(C)(C)CNC(C12CC1CN(C(C1CC(N(C)C)C1)=O)C2)=O C1(CNC(c2ccc(C)nn2)=O)CC2(CCC2)CN1C(C1CCCCC1O)=O C1(C(=O)NCCN(C(=O)CC2COCCO2)C)CCC(c2nc[nH]n2)CC1 C(CC(CC)C(=O)NCC1CCOC1C(=O)N(CC(F)F)CCO)=CC C1(NC(CCCOCC=C)=O)CCN(C(=O)C(C)Oc2cccc(C)c2)CC1F N1(C(COCCCOC)=O)CCC(CCNC(=O)Cn2ccc(C(F)(F)F)n2)C1 c1(OCC)ccc(Cl)nc1C(=O)NC1CC1NC(=O)CC1CC=CC1 N1(C(C2(C(C)NC(c3cc(=O)n(C)cn3)=O)CC2)=O)CCCC2OCCC12 C(=O)(C(C)S(C)(=O)=O)N(C(C)CCNC(=O)CNC(c1ccccc1)=O)C C1(C2CCCC2)(C(N2CCC(N(C(COCCCCC)=O)C)C2)=O)CCNC1=O N1(C(c2c(CC)ncs2)=O)CCC2CN(c3ncncc3F)CC2C1 C(=O)(Nn1cnnc1)c1ccn(C2CN(C(C3C=CC3C(Cl)Cl)=O)C2)c1 C#CCC(CC(=O)N(C)Cc1cccc(F)c1)NC(=O)C(C)C(C)C c1(C(N2C(CNC(=O)C(C)(C)c3cccs3)CC(OC)C2)=O)cc(C)cc(N)c1 c1(C(=O)OC)cc2c(s1)CN(CCC(C)P(C)(C)=O)CC2 c1(C(N2CCC(NC(c3cnc(C)o3)=O)CC2C)=O)cccc([N+](=O)[O-])c1N c1(C(N2CC(CC)C(NC(=O)C(C)(C)OC)CC2)=O)cc(F)c(Cl)cc1Cl N1(C(c2cc(CC)[nH]n2)=O)CCN(C(c2oc(C(C)C)nc2C)=O)CCC1C C=CC(C)(CCOC)C(=O)N1CCC1CNC(c1c(N)cccc1Cl)=O C1(CC=C)(NC(=O)CCC=CBr)CCCN(C(c2cccc(C)c2)=O)C1 C(C)(C(=O)N1CC(CCCCNC(=O)CCC2CC(C)C2)C1)N(C(C)=O)C S(=O)(=O)(c1ccc(-c2cncc(F)c2)o1)NC(c1c(C)cno1)=O CS(=O)(=O)c1cccnc1NC1CS(=O)(=O)CC1NC(=O)Cn1ncnn1 N1(C(C2C(COC)C2)=O)CCCC1C1(NC(=O)C(C)OC)CC1 C1(C2CC2)(CNC(C=CC(CC)=CC)=O)CCN(C(=O)C2=CCCCO2)C1 N1(C(CC(=O)N(C)C)=O)CC(NC(=O)CC2NC(=O)NC2=O)CC(F)C1 CC(C)(CF)C(=O)NCCCC1(CNC(=O)C(C)(C)C)CCCC1.C(=O)(N)OCC C(=O)(C#CC1CCOC1)N(CC(C)O)CCNC(C(C=C)OC)=O CN1CCCC1C(N1CC=CC1Cn1cc(C2(Cc3ccccc3)CC2)nn1)=O N1(C(C(c2ccccc2)C)=O)C2COCC1CC(NC(=O)Cn1cnnn1)C2 c1(OC)cccc(C(CN)NC(=O)CCOC)c1 c1(C(N2CCCC(NC(C(C#C)(C)C)=O)C2)=O)ccc2c(=O)cc[nH]c2c1 c1(C(N(C2CN(C(C(C3CC3)OCC)=O)C2)C)=O)ccc2c(c1)C(=O)OC2(C)C CP(C)(=O)CC(=O)NCC1CN(C(=O)CCc2cncs2)C1 C(C)(CCC(=O)NC1CC(Nc2cc(Nc3ccccn3)ncn2)C1)OC C1(CNC(C2CC(C#C)(O)C2)=O)C(C2CC2)CCN1C(=O)C1=CCCS1 C1(C(=O)NCC(C(C)C)OC)CCC2(CC2)N1C(c1cn(C)nc1C)=O N1(C(C(=O)N(CCCCCC)C)=O)CCOC(Cn2cc(C)cn2)C1 C12(CNC(CC3ON=C(C)C3)=O)CC(CO1)N(c1ccc(C(F)(F)F)cn1)C2 N1(C(C(C2CC2)NC(C(C)OCC2CCC2)=O)=O)CC2(CCC(C)OC2)C1 CCCC(C(=O)NC1CCC(NC(=O)NC)CC1)c1cnccn1 S(=O)(=O)(c1cc(C(N2CCCC(NC(C3(C)CCNC3=O)=O)C2C)=O)co1)NC C(=O)(C(C)(C)CC(F)(F)F)N1CCC(F)(CNC(C2N(C(C)C)CCCC2)=O)C1 c1(CNC(CC2(CC)CC2)=O)ccccc1CNC(c1cncc(OC)n1)=O C1(CCC(=O)NC2(C(=O)OC)CC2)CCCN(C(=O)CC2(O)CCC2)C1 C(=O)(CCC(=O)N1CCCC(NC(C2(c3occc3C)CC2)=O)C1)NCC C=CC1(O)CN(C(c2n[nH]cc2CNC(=O)C(CO)OC)=O)C1 C(=O)(C(C)(F)C(F)(F)F)N(CCCCN(C(CS(=O)(=O)N(CC)CC)=O)C)C c1(OCC(=O)NOCC2CC2)cc(F)cc(F)c1.c12cccnc1COC2=O Cc1oncc1C(=O)OC(C)C(=O)N1CC(n2ccc(CC3CC3)n2)C1 CCC(C)(CO)C(=O)N(CCC(=O)NC1(C)CCCC1(C)C)OC C(=O)(C1=CSCCO1)NCC=O.C1(Cc2cn(CC)nn2)CC(=O)N(C2CCCC2)C1 c1(C(N(CCNC(C2(CC(C)C)CC2)=O)CC2CC2)=O)cc2ccc(Cl)cc2o1 C=CC(C)(O)CC(=O)N1CCN(C(=O)CNC(C2CC2[N+](=O)[O-])=O)CC1 N1(C(c2ccc(NC(=O)OC)cc2)=O)CC(C2CN(C(=O)C(F)=C3CCC3)C2)C1 C1(NC(CC2CCC(C)(C)C2)=O)CCN(C(=O)CC(=O)NC)CC(O)C1.CCC1=CCC1 N1(C(C)=O)CCN(C(=O)NCCNc2cccc(C)c2Br)C(C)C1 C1(NC(C(CC)C)=O)CC2CC1N(C(c1ccc(OC)cc1C(F)F)=O)C2 N1(C(C(C=C)O)=O)CCC(C2CC2NC(c2ccccc2CC=C)=O)CC1 c1(C(=O)NC2CCCN(C(c3ccc(C)c(O)n3)=O)C2)ccc(S(N)(=O)=O)cc1 c1(OC)cccnc1C(=O)NC(C)(CNC(=O)C(C)NC(C)=O)C1CC1 c1(N2CCC(C)C2)nc(N(C)CC2CCC(C3CC3)O2)nc2cc[nH]c12 C1(C(=O)NCC(CCC)C)CN(C(c2ncccn2)=O)CC1(C)C C(=O)(C(C1=NOCC1)N1CCC(N2CCCOC2=O)CC1)NC(c1ccccc1)C CC(=O)CCCC(C)C(=O)N1CCC(C(=O)NCCC2CC(C)C2)C(O)C1 C123CC(CO1)(C2)NC(=O)COCC(=O)NC3.C1(CCN(CC)CC)CCC1 N1(C(Cc2ccc(OC)nc2)=O)CC2CC(NC(=O)C3=NOCC3)C2C1 c1(C(=O)NC2CC(NC(C3(C#N)CC(C)C3)=O)C2)nccc2ccn(C)c12 Cc1ccc(CC(=O)NC2(C)CCCN(C(=O)CC(C)C(F)F)C2)c(Cl)c1 c1(C(N2CCC(C(C)NC(=O)C=CC3CC3)CC2)=O)cnc(F)c(Cl)c1 CC(C)(C)CC(O)CC(=O)NC(C(N1CCCCC(C)(F)C1)=O)C1CCC1 N1(C(CC)=O)CCCC2(CNC(c3cc(OC)ccc3F)=O)CCCCC12 CCCCC(C(=O)NC1(C)CN(C(C2CC(OC)C2)=O)C1)N(C)C C1(CC)(CNC(=O)CC(C)N(C)C)CCCN(C(c2cnnc(C)c2C)=O)C1 c1(C(N(C)CC2(O)CN(C(c3n[nH]cc3Cl)=O)C2)=O)ccc2c[nH]nc2n1 N1(C(CCNC(C)=O)=O)CCCCC(NCc2cc(Cl)ccc2C)C1 c1(C(=O)NCC(C)(C)NC(C2CC(CO)CO2)=O)ccc(CNS(C)(=O)=O)o1 c1(NCC)ccc(Cl)cc1C(=O)N(CC(C)CNC(=O)C=Cc1cc[nH]n1)C CCC(C)(C)CC(=O)NCC1CCN1C(=O)CC1CCCCO1 C(=O)(C(CN(C)C)C(C)C)N1CC(N(C(Cc2c(C)ncs2)=O)C)C1 C1(O)(CN(C(=O)CCNC(=O)C2CC2)C)CCCN(C(c2cnnc(O)c2)=O)C1 C1(NC(C2CN(C(C(C3CC3)OC)=O)C(C)(C)C2)=O)CCCC(C2CC2)C1 C1(CC(NOCC(=C)Cl)=O)C2CCC(C2)N1C(C1CC(F)C1)=O C(=O)(CCCC(=C)C)N1CCC(C)(CC(=O)NC(C#C)(C)C2CCOC2)C1 C1(CC(C)N(C(CSCC(C)C)=O)C(C)C)CN(C(=O)C(C)C)C1 C#Cc1ccc(C(=O)NCC2CCCCCN2C(=O)CN2CCCC2=O)cc1 C1(NC(C2CCC(C)(C)OC2)=O)CCC2CC1CN2C(c1cc(N)ccc1O)=O c1(CN(C(C2CC(C)(C(=O)OC)C2)=O)C)ccc(C)nc1 N1(C(CCCOCCOC)=O)CCC(CF)(NC(=O)CCc2ccsc2)C1 N1(CC)CCN(CCC(=O)NCC2(O)CN(C(C3CC3(Cl)Cl)=O)C2)CC1 CS(=O)(=O)C1(C(=O)NCC2CC(O)(CNC(=O)Cc3cscn3)C2)CCCC1 c1(CNC(C2ON=C(C)C2)=O)cnc2cc(C)nn2c1.C12(CCCCCC1)NC2 C(=O)(CCCC(C)(C)C)N1CC2C(CC(=O)NCCNOC)(CC2)C1 C1(N(C(CCN(C(c2ccc(C(C)=O)o2)=O)CC)=O)C)COCC1NC c1(C(N(CC(=O)NC(C)CC2CCOC2)C)=O)cccc2[nH]ccc12 c1(C(=O)NC)ccc(NC(=O)C(c2cc(Cl)ccc2F)C)c(Cl)c1 c1(C(=O)NCC(C(C)C)NC(=O)CC2CC2C2CC2)cc2cccn2c(O)n1 C1(CN(C(=O)CCc2cncs2)C)C2CN(C(=O)Cn3cc(Cl)cn3)CC12 N1(C(COCC#C)=O)CCC(C(=O)NCCCC(C)O)(C(C)C)C1 CCCCC(C(=O)N1CCC(NC(c2ccnc(Cl)c2)=O)C1C)ON=C(C)C c1(C(C(=O)NCCCC2CC2)N(C)CC2CCC(=O)N2)nccc(C(F)(F)F)n1 N1(c2cc(SC)ncn2)CCC2(CCCC2C(N2CCc3cccnc3C2)=O)C1 Cc1ncsc1CCNC(C1(NC(=O)C=CCF)CC(F)C1)=O c1(C(=O)OC)ccc(O)c(NC(=O)C=CC(C)NC(=O)C#CC(C)(C)C)c1 C#Cc1ccnc(C(=O)NC(CC#CC)C(=O)N2CCCOC(C)C2)c1 C1(CC(C)C(=O)N)CC2CCC(C1)N2C(=O)C1=COCCC1.C1(CC=O)CCOC1 C(=O)(N=c1[nH][nH]c2c1CCCC2)C1(C)CN(Cc2cc(F)cc(C)c2O)C1 N1(CCC)CCCC(C(N2CC(N(C(=O)CSc3cccc(CC)c3)C)C2)=O)C1 C1(C(N(CCCNC(CCC(C)(F)F)=O)C2CC2)=O)CCCN2CCCCC12 c1(OC)cc(C(=O)N(CC(C)NC(=O)CC2CCCCC2O)C)ccc1O CCC(F)(F)C(C)(C)C(=O)N1CC(N(C)C(c2cc3cccn3cn2)=O)C(F)C1 C1(NC(c2c(C)coc2)=O)CCC2CN(c3ncncc3Cl)CC2C1 C12(CNC(C=C(CC)C)=O)CCCC1CN(C(=O)C=CCO)C2 n1(CCC(=O)NCC2(O)CC2)cc(C(C2CCC2)O)nn1 c1(C(=O)OC(C(=O)OC)C2CCOC2)cc2[nH]nc(C)c2cn1 N1(C(c2c(CC)scc2)=O)CC(OC)CC(NC(=O)C(n2nc(C)cc2C)C)C1 c1(Nc2ccc(NS(C)(=O)=O)c(Cl)c2)ncc2c(ncn2C)n1 C1(CCO)(NC(CN(C)C(N)=O)=O)CN(C(=O)CCc2cscn2)C1 CN(CC(=O)OCc1ccc(F)cc1)N1CCC(OCCO)C1 C12(C(N3CCN(CC#C)CC3)=O)COCC1CN(C1CCCCC1C)C2 C1(O)(C(C)NC(c2ccc(F)s2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 N1(C(C#CC(C)(C)O)=O)CCC2CN(C(c3ccc4nncn4c3)=O)CC2C1 c1(OC)ccc(C(O)CC(=O)N(C)CCNC(C2CC23CC(O)C3)=O)cc1 C1(C(N2CCC(CCNC(c3cccc(OC)c3)=O)C2)=O)(OC)CCCCCC1 C1C2CC3CC(C2)CC1C3.c1(CC(N2CC(NC=O)C2)=O)ccc(O)nc1 O=C(CCCc1cnn[nH]1)NCC1CC1CNC(C1CC1c1cccnc1)=O N1(C(CC#C)CO)CCC(NC(C2(NS(=O)(=O)CCCOC)CCC2)=O)CC1 C1(CCCC)CN(C(=O)C=NOC)CCN1C(c1ccc(F)c(N)c1)=O C(CC(C)(C)C(=O)NC(C)CCC)NC(C=C(CC)CC)=O C(N=c1[nH]c(N(CCCCN2CCCC2)C)nc2ccsc12)C1N(C)CCC1 C1(F)(CNC(C2CNC(=O)N2)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 N1(C(C2(C)CCC(=O)C2)=O)CC2C3CCC(C2C1)N(C(c1cscc1F)=O)C3 N1(C(C)=O)CC(O)CC1C(N1CCCC1C(C)NC(C1(N(C)C)CCC1)=O)=O Cc1cc(C(N)=O)cc(C(=O)N(CCCNC(=O)Cc2cncc(C#N)c2)C)c1 C(c1ccccc1)=CC1(C(=O)NCC(CNC(=O)Cc2cccnc2)OC)CC1 C1(NC(CCC)=O)CN(C(=O)C=Cc2cc(C)ccc2OC)CC12CCC2 C(=O)(CC(C)CCC=C(C)C)NCC(C)N(C(=O)CCc1cc(C)on1)CC C(=O)(CCS(=O)(=O)c1ccc(C)cc1)NCCC(=C)CNC(C1CNC(=O)C1)=O CC1CCN(C(=O)CCS(C)=O)C(C)C1NC(=O)CCCn1ccnc1 Cc1[nH]nc2c1CN(C(C1CCCN1C(=O)Cc1cccc(F)c1Cl)=O)CC2 c1(NC)cnncc1C(=O)NC(C)C(=O)NC1CC2(CCC2)C1 C1(C2(C(N(CCC)CCC)=O)CC2)CCNC(=O)C1 CCC1=C(C(=O)NCCCCC(=O)NCC(CC)n2cccn2)CCCO1 C1(C(=O)N(CCNC(C2CC2C(F)(F)F)=O)CCOCCO)CCCO1.COC C1(C(=O)NC2CC(C)SC2)C2CCCC2CN1C(=O)C(C(C)O)N(C)C N1(C(CC2CCN(C)CC2)=O)CC2CC3CC2C1C3NC(C1CCC(F)(F)C1)=O C1(C(N2C(CNC(CCCOCCOCC)=O)COCC2)=O)CC(C2CC2)=NO1 c1(C(N(C2CC(NC(=O)C(c3cnn(C)c3)O)C2)C)=O)cnn(C)c1C1CC1 CCC(C)C(C(=O)N(C)Cc1ccco1)N(C)C(c1ccncc1O)=O C12(C(N3C4(C(NOCCCC)=O)CC(C3)C4)=O)CCN(CC1)CC2 N1(C(C2C(OCC)C2)=O)CCC(C)(C)C(CNC(c2n[nH]c(C)c2Cl)=O)C1 CCCCN=C(NCCN(c1cc(Cl)ccc1C)C)NC(C)CC(C)(C)C Cc1cc(C(=O)NC2CCC(C(=O)Nc3sc(C)cc3C#N)OC2)cc(C)c1O C12(CC(=O)NC3(C)CC(NC(CCN(CC)CC)=O)C3)COC(C)(C1)C2 C1(CNC(CC(C=C)C)=O)CC2CN(C(=O)CCCN(C)C)CC12 N1(C(C(C)(C)SC)=O)CCC2CN(C(C34CCCC3C4Br)=O)CC2C1 CN1CCCCC1CC(=O)NC1CC2(C1)CC2C(=O)NCCS(C)(=O)=O C(=O)(CCCCCC(C)(C)C)N(C1CC(NC(C=CC(CC)C)=O)C1)C N1(C(C2CC(C#N)(OC)C2)=O)CCC2(CCCN(C(=O)CCCCC(C)O)C2)C1 C1(c2n(CC)nnn2)(NCC2CC2(C)C)CC(C)OC(C)C1 C=C=CCCC(=O)N1CC(C(N2CCN(C(c3c(C)cnn3CC)=O)CC2)=O)C1 C(C(C)C(F)C(=O)NC(C1CSC1)C)NC(c1cc(CCC)on1)=O N=c1[nH]c(O)ncc1-c1cn(C2CC(C(N3CCCC(C(F)F)C3)=O)C2)nn1 C1(NC(C(CC)O)=O)CCCCN(C(=O)C=Cc2cnn(C)c2C)C1 CC(C)(CC(=O)NC1CCN(C2CCN(C(=O)Cc3cn[nH]c3)C2)CC1)C(F)F O=C(CC(C(F)F)n1ccnc1)N(c1ncc(C2CCOCC2)s1)C1CC1 C12(CNC(CCC#C)=O)CC(CO1)N(C(C1CC1Br)=O)C2 c1(C2(C)NC(=O)N(CC3COC4(COC4)C3)C2=O)ccc2ccccc2c1 Cc1ccc(C(C)C)c(NC(C2CC2C(=O)NCc2ccncc2Cl)=O)c1 C1(C)(CNC(C(C)(N(C(c2n(CC)ncc2)=O)C)C2CC2)=O)CC2CC2C1 C(CN=c1[nH]cnc(NCCC2=CCCCCC2)c1C)c1c(OC)cccc1 C(CCNC(=O)Nc1cccc(Br)c1O)(C(F)(F)F)OC c1(CNC(COC(CNC(C=CC(C)C)=O)(C)C)=O)nccn1C C(CCO)(C(F)F)NC(C1(CNC(c2cc(CCC)[nH]n2)=O)CC(=C)C1)=O c1(NCC(CCCC)NC(c2ncc[nH]2)=O)ccnc2nc(C)nn12 c1(C(=O)NC(CCC=C)C2CC2)oc(CNC(=O)C#CC(C)C)cc1C S(=O)(=O)(c1ccc(F)c(F)c1)NC1CCCN(Cc2cc(C)[nH]n2)C1 C1(C=C)(C(=O)NC(CC=C)C(=O)OCC)CCN(C(c2ccc(CC)o2)=O)C1 C(=O)(C(CC(=O)NCCN(C(=O)C(C)Cc1ccncc1)CC)C(C)=O)OCC C1(NC(C(COC)O)=O)(CO)CCN(c2ncccn2)CC1 C=CC(C)(O)C(=O)N1CCC(O)(CNC(=O)C(C)Oc2ccc(Cl)cc2)C1 N1(S(=O)(=O)CCn2cccn2)CC2(C1)CC2(F)Br C1(N(C)C)CCC(C(=O)NC2CCCC2CNC(=O)CCOC2COC2)CC1 C12(C(N(C(CCNC(CC=CCC)=O)C)C)=O)CCC(N=[N+]=[N-])C1C2 N1(C(CC2C=NN(C)C2=O)=O)CCN(C(C2(C3CC3)CC2)=O)CC(C)(C)C1 Cc1ccc(C(=O)NCC2(C)CCN(C(c3cc(C#N)on3)=O)CC2)c(F)c1Cl Cc1nnc2n1CCC(N(CC(=O)N(c1nnnn1CC(C)C)C1CC1)C)C2 C(C(=O)N(C(CC)CO)C)(C1(C)CC1)NC(C=CCCC)=O N1(C(C2(C3CC3)CC2)=O)CCC(C2CCN(C(c3ccncc3)=O)CC2)C1 N1(c2cc(NCC3CCCc4nccn43)nc(COC)n2)CCC2(CCOC2)C1 C12(NC(C(CSC)OC)=O)CCC(C1)N(C(=O)Cc1cnn(C(C)(C)C)c1)C2 C1(CN(C)Cc2sccc2Cl)CCCN1C(c1sccc1C(F)F)=O C#CC1(C(=O)NCC(CCOC)NC(=O)CCc2csc(=N)[nH]2)CCCC1 N1(C(c2c(OC)cccn2)=O)C2CCC1C1CC1(NC(c1cncc(Cl)c1)=O)C2 C12CCC(=O)N(C1)C2.c1(C(C(=O)N(C2CCNOC2)C)N(C)C)ccc(Cl)cc1 C1(C(c2n(CCOC)nnn2)NCC(C)CC(C)C)COc2cc(F)ccc2C1 CC(C(=O)NCC(CO)NC(c1cnc(C(F)F)s1)=O)C(C)(C)C Cc1ccc(Cl)c(F)c1C(=O)NCC1(F)CCN(C(=O)CCCn2ccnc2)C1 c1(CC)nn(C)c(Cl)c1C(N1CC2(C1)CN(C(=O)CC1CCCCO1)C2)=O N1(Cc2n(C)nnn2)CCC2(CC1)OCCC2NC(=O)C1=COCCO1 C1(C(C)C)CCCC1NC(=O)CCN(C(=O)CN(C)C)C.C1(C)CC1 C=CCC(C)(C)C(=O)NC(C)(CNC(=O)C(C)(C)NS(C)(=O)=O)C1CC1 C1(C)(CNC(C(CC(C)C)F)=O)COCCN(C(=O)COc2ccccn2)C1 N1(C(C(C)C2CCOC2)=O)CCN(CCSc2ccccc2O)CC1 c12ccncc1OC2.C(=O)(C(C1CC1)NC(C1CC(CC)C1)=O)NCC c1(C(=O)NC(CNC(c2c(C)nncc2)=O)C)cn2ccc(CO)cc2n1 N1(C(C(=O)NC)=O)CCCC1CNC(=O)Cn1ccnc1C C12(C)CCCN(C1)C2.C1(c2cn(C(C)CSC)nn2)(C(=O)OC)CCCO1 c1(OC)ncc(C(N2CCCC(O)(CNC(=O)CC(Cl)Cl)C2)=O)c(C)n1 N1(C(c2n(CCCC)ncc2)=O)CC(CNC(=O)CCCNC(N)=O)CCC1C O(NC(=O)C(C)(CO)NC(=O)CN1CCSCC1)CCC N1(C(c2cn(C(C)(C)C)nc2)=O)CCC2(CCCN2C(=O)C2=CCOC2)CC1 CCC(C(=O)N(C1(CC2CC2)CCC1)C1CC1)N(C)C.c1(C=O)nc[nH]n1 c1(C(=O)OC(c2ncc(C)o2)C)[nH]c2ccc(Br)cc2c1F C1(C(=O)NCC2N(C(C(C(C)C)c3ccncc3)=O)CC2)CC2(CCC2)CO1 c1(C(=O)NC(C(=O)NC(CC)C2CCC2)CCSC)cccc(C)c1O CC1CC2(CCOCC2)CN1C(=O)C(=O)NCC1(C(=O)O)CCCO1 n1(CC(N2C(COC)CC2)=O)cc(CNC(C2CCCC2C)=O)nn1 N1(C(c2cn(CC=C)nc2)=O)CCN(C(=O)C(C)CN(C)C)C(CC)C1 c1(C(=O)NCC2(C(N)=O)CN(C(c3c(CC)ccs3)=O)C2)cnc(C(C)C)n1C c1(C(=O)NCC(C(C)C)NC(=O)C=CSc2nc[nH]n2)ccn2ccnc2n1 C(CC(C)C)(C(=O)NCC(CO)C1CCC1)N(C(c1c(C)nc(CC)o1)=O)C Cc1ccc(C)c(C(=O)NCC2CN(C(=O)CN3CCN(C)CC3)CCC2C)c1 [N-]=[N+]=NCCCC(O)CCNc1ccccc1OCC1CCCCC1 CCC(C)C(C(=O)NC1(C)CCSC1)NC(C1CN(C2COC2)C1)=O N1(C(c2c(CC)onc2)=O)CCC(CC)CC1C(=O)NC(COC)C1CC1 C(C)(CCCC(=O)NCC(C1CC1)SC)NC(c1cccc(CC)n1)=O c1(NC(c2cn(C(C)C)nc2)C)ccc(S(=O)(=O)N2CC=C(Br)CC2)c(Br)c1 c1(C(N2CC(C)OC(CCNC(=O)Cn3nccn3)C2)=O)cccn2nnnc12 c1(OCC)cnc(C(=O)NCc2ccc(CNC(=O)CCF)cc2)c(Cl)c1 CC(C(F)(F)CO)NC1CCCC(CS)C1.C1(C(=O)OC(C)(C)C)CCN(C=O)C1 c1(CC)nc(=N)[nH]cc1C(=O)NCC(C1CC1)N(C)C(c1nc(O)sc1C)=O N1(C(CCCCC)=O)CCc2nc[nH]c2C12CCN(C(=O)CC(C)CN(C)C)C2 Cc1cc(F)cc(C)c1C(=O)NC(C(C)NC(c1ncoc1C)=O)C(C)C N1(C(c2ccc(SC)s2)=O)CCCC2(CCC(NC(C3CCCC3)=O)C2)C1 C(CCCCCC(=O)Nc1cc(C)c(F)cc1F)NC(C1CC=C(C)CC1)=O C(=O)(C=CS(F)(F)(F)(F)F)NC(C)CNC(C1CCCCS1)=O N1(C(C)=O)CC=CC1C(=O)N(C(C)(C)C1(C(F)(F)F)CC1)Cc1ccncc1 CCCCCCC(F)C(=O)NCC1(NC(=O)CN2CCCCC2=O)CCCCC1 C1(CN(C)C(c2ccc(CS(C)(=O)=O)o2)=O)CN(C(C2C=CCCC2)=O)CCO1 N1(C(c2c(CC)cno2)=O)CCC(F)(CNC(c2sc(C)cc2C)=O)CC1 c1(CC(=O)NCCC2CCCN(C(C(C)SC)=O)C2)cc(Cl)ccc1Cl Cc1cc(C#N)cnc1N1CCCC2(NC(c3ccc(F)c(Cl)n3)=O)CC2C1 c1(C(C(N2CCC(N(C(=O)C(Cl)=CCl)CC)C2)=O)C)cccc(O)c1 Cc1cc(NC(=O)Nc2cc(C#N)nc(C3CC3)n2)cc(C)c1C c1(C(N2CC(NC(C3CCCN(CCC)C3)=O)C(C)C2)=O)c(C)ncn(C)c1=O O=C(CCCCCc1cccs1)NCC(C1CC1)NC(c1ccnnc1Cl)=O C1(NC(C2N(CCC)CCC2)=O)C2CC(NC(c3csc(C)n3)=O)CC12 c1(C(=O)NCC(C)NC(C2C3(CC3)C23CC3)=O)cnn(C)c1-n1c(C)ccc1C N1(C(C(CC)n2cncn2)=O)CCCN(C(=O)CC(C2CC2)SC)CC1 C1(CNC(C2CCCC23CC3)=O)CC2CCC(C1)N2C(=O)Cn1ncccc1=O c1(C(=O)NCC(C)NC(=O)C=CS(C)=O)ccc(Br)cc1C(F)(F)F C1(NC(COC(CNC(C(C)N2CCCC2)=O)(C)C)=O)CCCCC1O CC(CC#N)C(=O)NOCC(=O)NC(c1ccc(F)cc1)C Cc1nn(-c2ccccc2F)cc1NC(N1CCCC1C(C)(F)F)=O CCCCCCC(C)(CCC)C(=O)NC(CNC(c1cccc(C#N)c1)=O)CC Cc1ccc(C(=O)NCC2CCN(C(c3ccc(F)cc3Cl)=O)C2(C)C)nc1C c1(C(=O)NCC2CCCN2C(=O)CCC2CCC2)cc(Br)c(Cl)s1 c1(C(N2CC(NC(CSCCN(CC)CC)=O)C2)=O)nccc(C)n1 CCCCCCCn1ccnc1-c1ncccc1CSc1ccccc1 Cc1c(Br)cnc(O)c1C(=O)Nc1ncnc2c1CCC2 C1(SC)CN(C(C2(c3ccncc3)CC2)=O)CC1NC(c1cc(F)n[nH]1)=O N1(C(c2n[nH]c(C)c2O)=O)CCC(NC(=O)CCCN=[N+]=[N-])CC1C1CC1 N1(C(c2c(COC)cco2)=O)CCCC1(C)C(=O)NC(CF)C(F)(F)F CCCCCCCC(=O)N(C)CC1CCCN1C(=O)C(S(C)(=O)=O)C1CC1 c1(SC)cccc(F)c1C(=O)NC1CCC1CNC(C1CCC1)=O S(=O)(=O)(c1cc(C)ccc1C)N1CCC(NC(N2C(C#C)CC2)=O)C1 c1(CN(C(C(=O)Nc2cccc(CC)c2OC)=O)C)cc2ccccc2[nH]1 C12(C(N3CCC(O)(CCNC(C4(CO)CC4)=O)CC3)=O)CCC(C1)S(=O)(=O)CC2 c1(N2C(C(CC)NC(C3CCC(F)C3)=O)CCC2)ncnc2c1cnn2C CCC(C)(CCNC(=O)CN1CCCC1)NC(=O)C=Cc1cn(C)cn1 C1(C(N2CC(CCO)(CC)C2)=O)CC2(CC(NC(=O)Cn3cnnc3)C2)C1 C(=O)(N=c1[nH]n(CC)cc1C#N)c1cc2cnn(Cc3ccc(CC)o3)c2cc1C c1(NC(CCC2N(C(C(=C)C(F)(F)F)=O)CCC2)=O)c[nH]c2cc(Br)ccc12 C1(C(N2C3CC(NC(c4scc(C(N)=O)c4)=O)(C3)C2)=O)CCC2(CCC2)CO1 C1(CC)C(NC(=O)C(C)Oc2cccc(F)c2)CCN1C(=O)CCOC1CC1 c1(OC)cccc(C(C)C(=O)OC(C)Cn2cc(C3(C)CCCO3)nn2)c1 C1(C(=O)NCC(COCC)C)CC2C=CC1N(C(c1cnc(O)c(C)c1)=O)C2 N1(C(c2ccnc(OC)n2)=O)CCC2CCN(C(c3ccc(F)cc3)=O)CC2C1 C=C(C)CCC(C(=O)NC1CN(C(=O)OC)C1)N(C)CC1(OC)CCOC1 c1(NC(c2cccc(-c3ccc(C(C)=O)s3)c2)=O)ccsc1C#N N#Cc1ccc(NC(=O)NC2CN(C(C3CC3C3CC3)=O)CC2O)cc1 N1(C(CSC)=O)CC(C)(C)OCC1CNC(=O)C(C1CCCC1)N(C)C(C)C Cc1cc(C(=O)N(CCCCN(C)C(C2C=CCC2)=O)C)c2ncccc2c1 c1(C(=O)NC(C2CCCC2)CNC(C2CSCCS2)=O)c(F)ccc(F)c1O N1(C(c2n(C)cnc2)=O)CC2CCN(C(=O)Cc3ccc(Cl)nc3)CC(C2)C1 Cc1cc(F)cc(C)c1C(=O)N(C1CN(C(c2ccccc2)=O)CC1C)C CC1CCOCCN1C(=O)CC1(NC(c2cnc(Cl)n2C)=O)CCC1 C1(CC(=O)NCCC(=C)CNC(=O)CCc2cscn2)CCCCC1(F)F Cc1c(C(=O)NCC2CN(C(=O)CN3CCCC3)C2)sc2cc(F)ccc12 CC(CCCO)N=c1nc(N2CCN3CC(F)CC3C2)c2ncccc2[nH]1 C1(C(C)(C)C)CN(C(=O)C(C2CCCCC2)F)CCN1C(c1ccc(N)cn1)=O C=CCC(CC(F)F)C(=O)NCC1CCC1NC(c1cc(C)sn1)=O N1(CC(C2CC2)OCC)CCCC(C)(CNC(c2cscc2C)=O)C1 N1(C(c2cnc(OC)s2)=O)CC2(CC(C(=O)NC3CCn4ncnc4C3)CO2)C1 c1(C(=O)NCCCN(C(=O)C(O)C(C)(C)C)CC)ccc(OC(F)F)cc1F C1(CNC(COCC)=O)CCC12CN(C(=O)C=Cc1ccc(Br)o1)C2 C(=O)(C1=CSCCO1)NCC(C)(C(C)C)NC(CNC(c1c(C)cccc1)=O)=O c1(COCC)nc(C)cc(=NCC2CN(C(C3(S(N)(=O)=O)CC3)=O)CC2C)[nH]1 C(c1c[nH]c(=N)c(C)c1)=CC(=O)N(CCNC(C1(C(=O)OC)CC1C)=O)C c1(C(N2CC(C)(C)C(NC(=O)CC=C(Cl)Cl)CC2)=O)cc2cccc(Cl)c2[nH]1 C1(NC(C2CCC(OC)CC2)=O)CC2CN(C(c3ccsc3C)=O)CC2C1 c1(SCC(=O)NCC2C(NC(c3c(C)cc(CC)o3)=O)C2)cc(Cl)ccc1Cl C(=O)(CC(C)CN1CC(n2ccnn2)C(C)C1)OC C1(CNC(c2cc3cnn(C)c3nc2)=O)CC2(CCOCC2)CN1C(=O)C=CCO N1(C(c2c(C)cco2)=O)CC2CCCC(NC(c3cc[nH]c3C)=O)C2C1 N1(C(C2(CC#C)CC2)=O)CCC2(CC(NC(=O)C(c3ccc(Cl)c(F)c3)O)C2)C1 C1(NC(c2c(C)ncnc2)=O)CCCC12CN(C(=O)C(C)SC(F)(F)F)C2 C1(C)(CNC(C2C(C(C)C)N(C(c3ncn(C(C)C)n3)=O)CC2)=O)CCC(=O)N1C N1(C(C(C2CC2)OCC)=O)CC(NC(c2csc(C(C)C)n2)=O)CC(F)C1 C1(CCC)(NC(C2CCS(=O)CC2)=O)CCCN(C(=O)C(C)C2(O)CCC2)C1 c1(C(N2CCC(N(C(=O)Cn3nc(C)cc3C)CC)C2)=O)cc2ccccn2c1 N1(C(Cc2c(C)non2)=O)CC2(CCN(Cc3ccccc3CCBr)C2)C1 C1(NC(CCC=C)=O)CCN(C(=O)CC(C)N2CCCC2=O)C12CCC2 N1(C(=O)C(O)C2CC2)CC(F)(F)CC1CNC(C1(c2ccccc2)CCOC1)=O C(C(C)(C)C(=O)N1CCC(CC(N2CC(O)C(F)C2)=O)C1)OC(C)C N1(C(C2ON=C(C)C2)=O)CCOC2(C1)CN(C(=O)C(C)n1ccnn1)C2 n1(CC(N)=O)cc(C(N2CCC2CNC(C2CC(C(F)(F)F)C2)=O)=O)nn1 c1(C(=O)NCC2CCN(Cc3ccc(N(C)C)nc3)C2)ccc(F)c(O)c1F N1(C(CCn2c(C)cc(C)n2)=O)CCC(NC(c2cc(Cl)n[nH]2)=O)C12CC2 C1(NC(C(C)OC(c2ccc(-c3ccccc3)[nH]2)=O)=O)CCS(=O)(=O)C1 Cc1cc(C)n(CC(N2CC3C(C(=O)NCCC4CCOC4)C3C2)=O)n1 c1(C(N2CC(NC(CC3CC(=C)C3)=O)C(SC)C2)=O)c(C)cc(F)cc1Br N1(C(=O)C=CC2CCCO2)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C2(CC2)C1 c1(C(N2C(C)(CC(=O)NC(COC)CCO)CC2)=O)cnc(S)nc1 C(CNC(=O)Cn1cc(C)cn1)(CCCC)NC(COCCCCC)=O c1(C(c2n(C(C)C)nnn2)Nc2cnn(-c3ccccc3)c2)ccc(Cl)cc1Br c1(C(N(CCCCN(C(C2(CC)CCCC2O)=O)C)C)=O)cc(C)cc(O)c1 Cc1cc(Cl)c(C(=O)NC2CCCN(C(=O)C(C)(C)C3CCOC3)CC2)cc1F C(=O)(CC(F)(F)C(F)(F)F)N1CC2CC(NC(C=CCC)=O)CC2C1 N1(C(CC2CC(=C)C2)=O)CC(C)CCC1CNC(c1ccc(C(C)=O)nc1N)=O CC1CN(C(c2c[nH]c(Br)c2)=O)CCC1NC(=O)COC1CC=CC1 Cc1ccc(C)c(C(N2CCN(C(=O)C(O)CCN(C)C)CC2CC2CC2)=O)n1 C1(C(=O)NCc2ncn(C)c2)CN(C(=O)CC#N)CCN1 CC1=NOC(=O)C1CCC(=O)NCC1CC1NC(c1cnc(CC(C)C)[nH]1)=O C1(NC(c2cc(C)n(C)n2)=O)CCCCN(C(C2CC(OC(C)(C)C)C2)=O)C1 CC1CC(=O)NCCN1C(=O)CC(C)(C)N(C(=O)CCC1CCOC1)C Cc1cn2ccc(C(=O)NC3CCCC3NC(=O)C(C3CC3)N(C)C)cc2n1 C(C(CN=c1ccn2ccnc2[nH]1)C(F)(F)F)NC(c1cn(C)c(=O)n1C)=O C1(CNC(CC(C)SC)=O)CCCC1C(=O)NC(C)C C1(C(F)(F)C(=O)NC(C)CNC(c2nnn(C)c2N)=O)(OC)CCCCC1 c1(C(CN2CCC2C2CCCC2)N(C(C)C)CC)nscc1C c1(C2C(C(=O)OCC3(C)CCC3)C2)nc2ccccc2s1.C1(=O)CO1 c1(C(C)C(=O)NC2(CO)CCN(C(=O)C(=O)N(C)C)C2)cccc([N+](=O)[O-])c1 CC1=C(C(=O)NC2CCC(CNC(=O)CCC(=O)N(C)C(C)C)CC2)CCC1 c1(C(=O)NCC(c2ccc(C)cc2)C)nccc2c1[nH]c1ccccc21 C(=O)(C1=C(C)OCC1)NCCC(CNC(C(CC)n1cncn1)=O)O c1(C(=O)NC23CC(NC(C4(SC)CC(O)C4)=O)(C2)C3)coc2c1C(=O)NCCC2 C1(C)(C(N2CC(NC(c3ccc(C(CC)=O)cc3)=O)C2)=O)CCCS1(=O)=O c1(CC(=O)NCCC2(OCCC(=O)NC3CC(N(C)C)C3)CC2)ccccc1F c1(CNC(C=C(COC)C)=O)csc(CNC(=O)C(CO)N(C)C)n1 N1(C(c2c(C)snc2)=O)CCc2ccccc2C1CNC(c1ncccc1F)=O CN1CCN(C)C(CNC(C2(NC(c3cnns3)=O)CC(CO)C2)=O)C1 C(=O)(CCCC(=O)NCC(=O)Nc1ccccc1F)NCC(CNC)O C1(C(=O)NCCOC2CCN(C(=O)CSc3cn[nH]c3)C2)CC2CCCCC2O1 Cn1nc(O)cc1C(=O)NC(C)CCCCNC(=O)C(c1ccccc1)C1CC1 c1(N2CCC(CCOC)(NC(c3cc(Cl)no3)=O)C2)[nH]cnc2nc(Cl)cc1-2 N1(C(CCCC#C)=O)CCC(C(=O)NCC2CCOC2=O)C12CC2 Cc1cc(C#N)ccc1C(N1CC(C)N(C(C2C=CCS2)=O)C(C)C1)=O C1(C(=O)NCc2c(C)nns2)CCC(C2CC2)N1C(c1cc(C(C)C)on1)=O C=CC(CCC)CC(=O)NC1CCC12CN(C(c1cccnc1N(C)C)=O)C2 C1(C(=O)NC2CCC(N(C)C)C2)CCCC1NC(=O)Cc1ccccc1 N#Cc1cccc(C(=O)NC2(C(=O)NCC3(O)CC(O)C3)CSC2)n1 N1(C(C(C(=O)OCC)(C)C)=O)CCCC2(CC(NC(C3CCC=CO3)=O)C2)C1 N1(C(CC)=O)CC2(CC(C(N3CCC(O)CC34CC4)=O)CO2)C1 CC(CCc1cnn(C)c1O)N=c1cc[nH]cc1S(=O)(=O)N1CCC(C)(CO)C1 N1(C(C(C)=C(CC)C)=O)CCCC(F)(CNC(=O)CCCN=[N+]=[N-])CC1 N1(C(CC(C)(C)C#N)=O)CC2(C)CN(C(C3CCC3n3cccn3)=O)CC2(C)C1 C1(NC(C2C(C(=O)OC)C2)=O)CCCN(C(c2ncc(C)cc2F)=O)CC1 C1(C(N2C(C(C)O)CC2)=O)C(NC(=O)Cc2cnoc2)C1(C)C N1(C(C2N(C=O)CCC2)=O)C2CCC1CN(C(C1(CC(F)F)CCC1)=O)C2 N1(C(C(C)(CO)NC(=O)CCc2cnn[nH]2)=O)CCCC(CO)CC1 c1(C(C(=O)NCC2CCCCC2)N(C2CCCC2C#N)C)nc(C2CC2)n(C)n1 c1(C(C(N2CCC(C(C)(C)NC(C3CCOCC3)=O)C2)=O)O)ccc(F)c(F)c1 C=C(C)CC(C(=O)N(C1CCC(NC(C2CC2C#N)=O)CC1)C)OC C12(CNC(C3C(NC(=O)Cc4cccc(O)c4)CC3)=O)COC(C1)C(O)C2 C(C(C)(C)CC(=O)NC1CC1c1cncs1)NC(C1(C)CC(C)C1)=O C(=O)(CS(=O)(=O)CC)NC(C(=O)NC(CC#C)C)CC c1(C(N2CC(CC(C)NC(=O)C3=CCS(=O)(=O)C3)C2)=O)c[nH]c2nc(Cl)ccc12 C1(C(N2CC(C)(NC(c3ncc(CC)cn3)=O)C2)=O)CC2COCC2C1 CN1CCOCC1C(=O)N(CCNC(C1(C)CC=CC1)=O)CCc1ccccc1 C1(CCOCC#C)CCCN(C(=O)CN(CCCC)C)CC1.C1(=O)CN1C1CC1 CCC(N=c1[nH]c(=NC(C)c2ccc(F)cc2)[nH]c2c(F)cc(F)cc12)C(C)C C1(OC)CCC(F)(F)CC1.C12(CCN(C(c3c[nH]cc3C)=O)C1)C(=O)N2 Cc1[nH]c(C(C)(C)C)cc1C(=O)NC(C)C(C(C)C)NC(=O)CC1CC1 C1(C)(NC(CN(C(=O)C=Cc2cc[nH]n2)CC#C)=O)CC(O)(CO)C1 C(=O)(C(CC(C)C)C(C)C)NC1CCC(NC(COCCC=C)=O)C1 N1(C(c2cc(C)nc(O)c2)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)CC(C)C1 c1(C(N(C2CN(C(c3cccc(I)c3)=O)CC2F)C)=O)ccccc1C#N N1(C(C(CSC)O)=O)CCC(C(N2CCCC2C(O)CO)=O)C(C)C1 n1(CC)cnc2c(NCCc3cn[nH]c3)[nH]c(=NC(C)C(C)COC)nc12 N1(C(C(F)=CCC)=O)CCCC1(C)CNC(=O)CC1(c2ccccc2)CCCO1 C1(c2cn(C)nc2)CN(C(=O)C=CCO)CC1NC(C1(C#N)CC1)=O Cc1nc(C)c(C(N2CCCC(C(C)NC(=O)CCc3cnn[nH]3)C2)=O)o1 C1(NC(CCOC)=O)C(C)CCN(C(c2ncc(Cl)cc2Cl)=O)C1C N1(C(C(C)Cc2cccc(O)c2)=O)CCN(C(=O)C=CBr)C2CCCC12 C1(CC)CN(C(C2(CCF)CC2)=O)CCN1C(=O)CC1CC=CCC1 c1(C(=O)NCC(CN(C(CC(=C)I)=O)C)O)ccc(=O)oc1 Clc1cc2c(Br)ccnc2n1CCNc1ncc(Br)cc1Cl C1(NC(CC2(OC)CN(C(=O)C(C)CC3CC3)C2)=O)CN(C)CC1C C1(NC(c2c(CC)non2)=O)CC2(C1)CC(CNC(c1ccc(C)cc1O)=O)C2 C=CC(F)(F)C(=O)NC1COCCC1C(=O)N(CC(C)(CO)CO)C CC(C)CC(O)CC(=O)NC(C(=O)NC1C2CCCOC12)C(C)O CC1c2c(F)cccc2CCN1C(=O)Cc1cc2ccccc2nc1O CCCC(C(=O)NCCCN(C(C1CCCN1C(=O)OCC)=O)C1CC1)N(C)C C1(CCC(C)C)CCCN(N2CCC(N3CCS(=O)(=O)CC3)CC2)C1 n1(CC)ccc(C(=O)NCC2(CCNC(=O)C(C)C(F)F)CC2)cc1=O Cc1ncncc1C(N1CCC(NC(c2ccnc(-c3ncc[nH]3)c2)=O)C1C)=O c1(OC(c2cccc(NCCN3CC3)n2)C)ccn2ccnc2n1 N1(CCOC)CC(C(=O)N(C)CCOCCNC(=O)CC2CC=CC2)CC1=O c1(NCC(N2CCCC2)C)cc(S(=O)(=O)N(C)CC2CCCOC2)ccc1C#N C#Cc1ccnc(C(N2C(C(N3CCCC(F)CC3)=O)CCC2C(C)C)=O)c1 c1(OC)ccc(C(N2CCC(O)(C(C)NC(c3ccoc3C3CC3)=O)C2)=O)cn1 c1(OC)cc(CNC(C2(NC(c3ncncc3Cl)=O)CCCC2)=O)n(C)n1 C=CC(CCC)CC(=O)N1CCCC1C(=O)NCc1ccnc(SC2CCC2)c1 C1(CNC(c2cc(CC)oc2C)=O)CC2(CC2)CN1C(=O)C(c1ccccn1)C N(C(=NCc1ccc2c(c1)ncn2C)N1CCC(O)C1)CC(=O)NC(C)C CCCCCC(C)NC(C1CN(C(=O)Cc2cnc(C)s2)CC1CC)=O CCCC(O)C(=O)NCCC(C)NC(COCCC(=O)NC(C)(C)C)=O c1(C(=O)NC(C2CCN(C(C3C(OC)C3)=O)CC2)(C)C)cccc(C(=O)OC)c1C c1(C(N(CCOC)CCNC(=O)C2=CCC2)=O)cn2ccccc2n1 c1(C(=O)NCC2CCC(CNC(c3ccoc3Br)=O)CC2)coc2c1CSC2 S(=O)(=O)(c1cccs1)NCC(=O)NC(CNC(=O)CC1(C(F)F)CC1)C1CC1 C1(C(=O)NCC2COCCN(C(c3ccc(=N)[nH]n3)=O)C2)CN2CCCC2CO1 c1(C(=O)OC)cnc(NC(C2CCN2CCS(N)(=O)=O)=O)nc1C C(CS(=O)(=O)CC(=O)N1CCC(O)(CCNC(=O)C(c2cncnc2)C)C1)OC N1(C(c2c(C)nc(O)cc2)=O)CC(O)(C2(CNC(=O)CCc3ccco3)CC2)C1 C#CCCCCCCC(=O)NC1(C(=O)NC(C)C(C)C)CCC(C)(C)C1 n1(-c2c(C)ccc(OCC)c2)c(-c2sccc2C)csc1=Nc1sc(C)nc1C C(=O)(C(C)S(=O)(=O)C1CCOCC1)N1CC2(CC(NC(C(CC)(C)C)=O)C2)C1 C1(N(C)C(c2nocc2Cl)=O)CCCN(C(C2CC(O)(C(F)(F)F)C2)=O)C1 C1([Si](C)(C)C)(CNC(CN(CCC)C(c2cncc(OC)n2)=O)=O)CC1 C1(C#N)(C(=O)NC2(CNC(C(CCOC)C)=O)CCOC2)CCOCC1 C1(CNC(c2ccc(C(C)C)cc2)=O)CN(C(C2CCCC2C)=O)CCC1(C)C Cc1ccc(NC(=O)CCN2CCN(CCn3cc(CCO)nn3)CC2)c(F)c1 CC1(C2CCCN(C(=O)CCCCCNC(C3CCC4CC3CO4)=O)C2)CC1 O=S(=O)(c1ccc(NCC2(Br)CC2(F)F)c(F)c1)NC1CCn2ncnc2C1 N1(C(C(CC)C)=O)CCCC(C)(CNC(c2nc(C3CC3)ncc2Cl)=O)C1 c1(SC)cccc(C(=O)NC2CCN2C(=O)COC2CCN(C)CC2)c1Cl C1(CNC(CCCCCSC)=O)CN(C(c2cncc(O)c2)=O)CC2(CCC2)O1 c1(C(=O)NCCN(C(CCCC#C)=O)CC(C)O)nc2cc(F)ccc2s1 Cn1ncc2cc(CN3CC4CN(C(c5ccc(F)cn5)=O)CC34)ccc12 c1(CC)cc(C(=O)NC2N(C(CN3C(CC)CC3)=O)CCCCC2)c(C)nn1 c1(CC(=O)NC2C(NC(C=C(C)c3cnn(C)c3)=O)C2)ccc2nc(O)[nH]c2c1 CCCC(C)C(=O)NCc1nc(CNC(=O)C(C)OCCOC)cs1 C1(C(=O)NOCC2CCOC2)CN(C(=O)CC2CCSC2)CC12CCC2 c1(C(N(CC(CC)NC(=O)C(C)NC(C)=O)CC)=O)n[nH]c2c1CCOC2 c1(C(N2CCC(O)CC2)=O)ccc2c(c1)CN(C(c1cnn3c1CCC3)=O)C2 N1(C(c2cn(C)nn2)=O)CC2CC1CCN2C(c1nccn2ccnc12)=O CC(C(C)(C)O)NC(=O)CN(C1CC(C#N)C1)C(=O)Cc1ccoc1 C(=O)(C1CCCc2nncn21)N(C(CCNC(C1(OC)CC1)=O)C)C C12(NC(c3cn(CCC)nc3)=O)CCC(C(=O)OC(C)(C)C)(CC1)C2 c1(CC(N2CCC(OCCNC(C3C(OC)(OC)CC3)=O)C2)=O)ccc(C)cc1 c1(C(N2CCC(CC(C)NC(C(=O)NCC)=O)CC2)=O)c(F)cc(F)cc1F c1(-n2cc(C3N(C(Cc4c(C)cccc4)=O)CCOC3)nn2)ccc(Cl)cc1F c1(OC)ncc(C(=O)N(C(C(F)(F)F)C2CC2)C)cc1C C#Cc1ccc(C(=O)NC(C)(C)C(C)NC(C2CN(C(C)C)C2)=O)cc1Cl c1(OC)cc(C(=O)NC2CC(CNC(c3cncc(C)n3)=O)C2)ccn1 CC1(C)CCC(C(N2CC=C(CNC(=O)C(O)Cc3cnc[nH]3)CC2)=O)OC1 c1(C(=O)NCCN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC)cnc(C(C)C)nc1C N1(C(C2(CC)CCN(C(c3c(CC)oc(C)c3)=O)C2)=O)CC(C2CC2)(OC)C1 c1(CCC(=O)NCCN(C(=O)C(O)C(C)C)CCOC)ccnc(Br)c1 N1(C(CC2CCC(=O)NC2)=O)CCN(C(=O)C(=O)NC2CC2)C(CF)C1 C1(C(=O)NCCC2CCCN(c3nc(C(C)(C)C)ns3)C2)(OC)CS(=O)(=O)C1 c1(C(N2CCN(C(CC(C)(C)O)=O)CC2CO)=O)nc[nH]c2ncc(Br)c1-2 C#Cc1ccc(Br)c(C(=O)NC2CN(C(=O)C3=CC4CCC3C4)C2)c1 c1(C(CNC(C(=O)NCCOCC)Cc2csc(Br)c2)C)cc(Cl)ccc1Cl n1(CC(=O)NCC2(F)CCC(NC(C=CSC)=O)C2)ccc(=O)c(O)c1C C1(C2CN(C(=O)CN3CCCCC3)C2)(NC(C2C(C#N)C2)=O)CC1 N1(C(CCC(=C)Br)=O)CCN(C(=O)CC(C(F)F)n2cccn2)C2(CCC2)C1 C1(N(C)C)CCC(NC(=O)C(CO)NC(=O)C=CCNC(N)=O)C1 CC1C(NC(C2CC(N=[N+]=[N-])C2)=O)CCN1C(=O)CCn1ccc(=N)[nH]1 C1(CNCC)CCCN(C(C2CC(OC)CN2C(c2[nH]cc(C)c2C)=O)=O)C1 C1(CN(C2CCCCC2)C(=O)OC(C)(C)C)CCCC1(C)C C12(CNC(C(CC)OC3CCCC3)=O)CC1CN(C(C1CCN1C)=O)C2 C=C(C)CC(C)C(=O)NC1CCCCC1NC(=O)CCN(S(C)(=O)=O)C C1(NC(C2(CC3CC3)CCC2)=O)CCOCC1C(=O)NCCC(F)F C1(CC)OCCC1C(=O)NCCCN(C1CCCC1)C(c1cc(Cl)n[nH]1)=O CC1CCc2[nH]c(=NCCC(F)(F)Cl)[nH]c(=NCC3CCC4(CC4)CO3)c2C1 Cc1cc(C(=O)NCC2CCCN2C(=O)C(C)C2(O)CCC2)nn1C(C)C1CC1 c1(C(=O)NC(C2CCCN2CC(O)COC)CC)cc(C(C)C)[nH]c1C(C)C C(CC(C)C(=O)NC(C)CCC(=O)N1CC(c2nncs2)C1)OC c1(C(=O)NCC2N(C(=O)COCC3(C)CCC3)CC2)cc(C2(O)COC2)on1 C(=O)(CCCCC(F)(F)F)NC(C1CCN(C(=O)C#CC2(O)COC2)CC1)C Cc1ccc(C(C)C(=O)N(CC(C)O)CCNC(=O)C2=CCOC2)cc1 C(N=c1[nH]c(=NC(CF)CF)[nH]c2ccsc12)c1nc2ccc(C)cn2c1.C1CCC1 N1(OC)CC2CC(N3CC(F)C3)CC1C2.c12cccc(c1C)C(=O)NC2 C1(CC(C)C(=O)NC(CCO)C2CCCC2)CCC(F)(F)CC1 C1(NC(C(C)c2cc[nH]n2)=O)CCC(NC(=O)CC=C(Cl)Cl)CC1 N1(Cc2c(C)cccc2Cl)CC2(CN(C(c3ccccc3Br)=O)CC2CO)C1 C1(C2CC2)(NC(CCCC)=O)CCN(C(=O)C(CC)C(C)C)C1 c1(C(CNC(=O)NC(c2ncc(C)s2)C)(C)O)ccc(F)c(C(F)(F)F)c1 C(=O)(C(C)CS(C)(=O)=O)N(C1CN(C(C(N2CCOC2=O)C)=O)CC1O)CCO C1(C#N)(C(=O)NC2CCCN(C(CCSCCCC)=O)C2)CC12CCCC2 c1(C(=O)NC(C)CC(C)NC(c2ccc(F)o2)=O)ccc(-c2cnn(C)c2)cc1 c1(C(=O)NCCC(CCNC(C2C(C)OC(=O)N2)=O)C)ccc(S(N)(=O)=O)o1 c1(C(=O)NC2CCC(CNC(CCCNC(C)=O)=O)C2)cc2n(n1)CCO2 N1(C(CC2(N(C)C)COC2)=O)CCC2(CC2NC(C2CC2F)=O)C1 C1(CCNC(CCNC(=O)NC)=O)COCCN1C(C1COC(=O)O1)=O C1(C)(C(=O)NC2CC(C)(CNC(C3(Br)CC3)=O)C2)CCC(=O)C1 C(C(C)(O)CC(=O)NCC1(NC(c2cc(=O)cc(Cl)[nH]2)=O)CCOC1)OC c1(C(=O)NC2CC(CNC(C(CC#C)C)=O)C2)cc(OC)c(OC)cc1[N+](=O)[O-] Cc1[nH]nc2c1CCC(C(=O)NC1CCC(NC(c3csnn3)=O)C1)C2 CC1(CNC(C2CCCC2)=O)CCC(NC(c2ccc(C(F)(F)F)nc2)=O)C1 C1(NC(c2cc(C)sn2)=O)C=CCC(C(=O)NC(c2cn[nH]c2)C)C1 C=CC1(NC(=O)COC2CN(C(c3c[nH]nc3C3CC3)=O)C2)CCC1 C1(C)(C(=O)OC)CCCN(CC(=O)C2CC2C2CCCCC2)C1 C=Cc1cncc(C(c2nnnn2CC(F)F)NCCC(C)CCC)c1 C(=O)(C(CNC(=O)CN1CCC(n2ccnc2)C(C)C1)C(C)C)OCCC C1(CNC(C(c2cccs2)SC)=O)CN(C(=O)Cc2cc(Cl)cs2)CCC1C c1(C(N2C(CNC(C=CCCC)=O)CCCC2)=O)ccc(C)n(C)c1=O c1(-c2nc(OC)c(Br)cn2)n[nH]c2c1CN(C(C1(C(=O)N(C)C)CC1)=O)C2 C1(CNC(C(CC)n2cncn2)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1(F)F c1(C(=O)NCC(C)(O)CNC(c2csc(S(C)(=O)=O)c2)=O)cccc2occc12 Cc1ccc(C(=O)NCC(O)CCNC(=O)Cc2cnn(C)c2)nc1C Cn1c(CCC(=O)NCC#CCNC(C2(C)CCCC2O)=O)nnc1S N1(C(c2ccn(CC)n2)=O)CC(C)CCC1CNC(=O)CCSc1nnnn1C C1(NC(C(CCN(C)C)NC(=O)C(F)C2CCC2)=O)CCC2CC1CO2 CCCCC(CC(=O)N(CC(C)(C)C)C)NC(c1coc(CC)n1)=O C1(CCC(=O)NCC(C)NC(=O)C(C)NS(C)(=O)=O)CCCCN1C C(=O)(CN=c1cc[nH]cc1)N1C(C(=O)NCC(C2CCC2)OC)CC2(CCC2)C1 O=C(CN=c1ccc(Cl)n[nH]1)NC1CC(O)CN(C(=O)C(C2(O)CCCC2)F)C1 c1(C(N2CC3C(NC(COCC)=O)C(C3)C2)=O)cnc2ccnn2c1 C1(CNC(C2N(S(CC)(=O)=O)CCC2)=O)CN(C(C2(n3cccn3)CC2)=O)CCO1 C(=O)(C1Cc2ccc(Cl)cc21)NCCN(C)C(c1c[nH]cc(F)c1=O)=O C(=O)(C(C)(O)C(C)(C)C)NCC(CC=C)NC(c1cc(CC)cc(Cl)c1)=O CC1(C)CCCN(C(=O)CC2COCCO2)C1C(=O)NCC12CCCC1OCC2 CC1(C)CCC(n2cc(CC3CCNC3=O)nn2)CN1C(C1(CC2CC2)CC1)=O N1(C(C=CC)=O)CCC2CC(NC(=O)CC(C)(O)C(F)(F)F)CCC2C1 C1(OCC(=O)NC(CC(C)NC(C2CN(C(N)=O)C2)=O)C)CCC(F)(F)CC1 C1(CC(=O)N(CCCN(C(c2cc(CN(C)C)on2)=O)C)C)OCCOC1(C)C C(=O)(C(C1=CCC2CC2C1)NC(N1CCCC1Cc1ccncc1)=O)OC N1(C(c2cc(C)nc(O)c2)=O)CC2CCCC(Nc3cc(Cl)ncn3)C2C1 n1(CC)nnc(C)c1C(=O)NCCOCCNC(C1(C)CC1(F)Cl)=O CCCC(C(=O)N1CC(Cc2cn(CC3CCCC3)nn2)C1)c1cccc(Cl)c1 N1(C(CC2CC(CC)C2)=O)C2CCC1CN(C(C1C3CCCC13)=O)C2 c1(C(=O)NC(C(C)NC(c2cc(C)nc(O)c2)=O)(C)C)coc2ccccc12 C(C(C)(C(C)C)NC(=O)C(C)CC1CCCCC1)NC(C(C1CCCC1)OC)=O CC(CC(=O)N1CCC(F)(F)C(CNC(c2cc[nH]n2)=O)C1)C(F)(F)F N1(C(C)=O)CCC2(CC1)CCN(C(c1cccc(Cc3ccccc3C)c1)=O)C2 C1(C)(C(N2CC(NC(c3c(C)nn(C)c3)=O)C(C(F)F)C2)=O)CCCCC1(F)F N1(C(CSCC#C)=O)CC(O)(C(F)C(=O)NCC(=O)N(C)O)C1 O=S(=O)(c1ccc(OC(F)F)c(F)c1)N(C1CC2CNC1C2)CCc1cnco1 C(CCCN=c1[nH]c(Cl)ncc1Br)NC(c1sc2c(c1)C(C)CC(C)C2)=O C1(CC#N)CN(C(=O)C(Cl)(Cl)Cl)CCN1Cc1ccc(N2CCOCC2)cc1 C1(N(C(=O)CCN2CCCC2)C)CN(C(=O)C=Cc2nccs2)CC1F C1(C#N)(CCCCCNC(=O)OC(C)(C)C)CCN(C(=O)CO)CC1 C1(CCN(C(=O)CC2CC(F)C2)C)CCCCN1C(c1snc(Cl)c1Cl)=O c1(CC)cccc(F)c1C(=O)NC(C1CCCN1C(C1CC=CC1)=O)C c1(C(N2CCCCC(NC(C(C)(Cl)Cl)=O)C2)=O)cc(Cl)cc2ccncc12 c1(C(N2CCC(C)C2C(=O)NC2CC(=C3CC3)C2)=O)cc([N+](=O)[O-])c[nH]1 N1(C(c2c(CNC(C(C=C)CC)=O)ocn2)=O)CC2CC3CC2C1C3 N1(C(CCCOC)=O)CC(NC(c2nc(Br)sc2C2CC2)=O)CC1C c1(C(N2C(CNC(C(C)CC3CC3)=O)CC2)=O)cnnc2ccccc12 C=CCC(C)(C)CCNC(=O)C(C1CCCO1)NC(=O)CCOC1COC1 Cc1ccc(N)cc1S(=O)(=O)NCc1cc2cc(F)ccc2o1 C1(C(=O)NC2CCCC(CN(C(=O)C(N)=O)C)C2)CC(=O)C12CCCC2 c1(C(N2CCN(C(=O)C3=COCC3)CC2CO)=O)cccc2nc(O)oc12 C1(NC(CC2(C=C)CC2)=O)CCCN(C(=O)CCOc2cc(F)cc(F)c2)CC1 c1(NC(c2nc(CNC(C(CC(=C)C)OC)=O)oc2C)=O)cc(C)c(F)cc1C c1(C(=O)NC(C2CN(C(=O)C3CC3)CCO2)C)nnn2ccccc12 N1(CC(=O)NC2(CO)CCCN(C(=O)CSC(F)F)C2)CCc2ccccc21 C1(CNC(C(c2ccc(Br)cc2)OC)=O)(CNC(C)=O)CC12CCC2 N1(C(CCC#C)=O)CCC(C2CN(C(c3cncc4nc(O)[nH]c34)=O)C2)CC1 C1(CCOC)(C(=O)NCC2CN(C(=O)CC34CC(C3)C4)C2)CCC1 c1(C(=O)NC(c2ccccc2Cl)C)ccc2c(-c3cccc(F)c3)n[nH]c2c1 N1(C(COC)=O)CC=CC1(C)C(=O)NCC(O)C(=O)OC N1(C(C(CN)C2CCCCC2)=O)CCC(C2CNCCO2)CC1 C1(O)(CNC(C2CCN(C(N)=O)CC2)=O)CCN(C(=O)CSC2CC2)CC1 c1(C(=O)NCC(CC)NC(=O)C(C)OC(C)(C)C)nc(C)c(C)s1 c1(OC)ccc(C=CC(=O)NCCNC(=O)C(F)CC(C)(C)CCC)cc1OC Cc1n[nH]c(C)c1C(=O)NC(C1CCN(C(=O)CNC(C2CCC2)=O)C1)C C1(C(N2CC(C)(c3cn(CC(C)(C)C)nn3)C2)=O)(OC)CCC(F)(F)CC1 c1(OC)cccc(CNC(C)(CSc2cn(CCOC3CC3)nn2)C(=O)O)c1 c1(C(=O)NC(C(=O)NC2C(C(=O)OC)C2)C2CC2)cc(Br)cnc1O C1(C(c2cn(CC(=O)O)nn2)C)CCCN(C(C2CC23CC(F)(F)C3)=O)CC1 Cc1ccc(O)cc1C(N1CCCC(NC(c2ccoc2Cl)=O)C1C)=O C1(NC(CC(C)C2CC2)=O)CC2CN(C(=O)CC3CN4CCC3CC4)CC2C1 c1(NCC(=O)N(C)CCc2nnc(C(F)(F)F)s2)nn(C)cc1Cl C1(C(N2CCC23CN(C(=O)COC(C)C)C3)=O)(OCC)CCC(C)(C)CC1 N1(C(C(C=C=C)C)=O)CCN(C(=O)CCC2(COC)CC2)CC1CS(C)(=O)=O C1(C(=O)NCC(CNC(c2c(CC)csc2)=O)C)COc2cccc(OC)c2C1 c1(NC(=O)NCC2(C)CCCN2Cc2ccccc2)c(Cl)cccc1I c1(C(N2C(CNC(C(=O)N(C)C)=O)CC3(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 c1(C(=O)NC(CNC(c2ccc(C)s2)=O)C(C)C)cccc(C(N)=O)c1C C(CCCCCN(C)C(c1cc(C(F)F)ccn1)=O)NC(C1CCC(C)C1)=O N1(C(CSCC=C)=O)CCC(C2CN(C(c3cnc4c(C)cccn34)=O)C2)CC1 C1(C(N(CC(C)(C)NC(CN2CCN(C)CC2)=O)C)=O)CCCC1S(C)(=O)=O n1(CC(=O)NCCC(C)N(C(C(CC(C)C)C)=O)C)nnc2ccccc12 O=C(CS(=O)(=O)CC1CCCO1)NCC(O)CCNC(c1ccoc1Cl)=O C1(NC(C(C2CCC2)OC)=O)CCCCCC1C(N1CCOCC1CO)=O Cn1cncc1CCC(=O)NC(C1CCN(C(C2CNC(=O)C2)=O)C1)(C)C Cc1cc(F)c(NC(C2CCCN2Cc2cnc(C3CC3)s2)=O)cc1F C1(C(N(c2nc(CC3CCCOC3)cs2)C)=O)CC2C(C1)C2(F)F C1(NC(=O)CC23COCC(C2)C3)CN(C(c2csc(C(F)(F)F)c2)=O)CC12CC2 N1(C(=O)CCC(=O)N2CC(Cc3cccs3)C2)CCCc2ccccc21 c1(Nc2[nH]nc(CSC)n2)c(C)nn(CC(F)F)c1C C1(CNC(CC2(OCC)CCC2)=O)CN(C(c2cnncc2NC)=O)CCC1(C)C C(C)(CN=C(NCCSc1ccccc1)NCc1n[nH]cc1Br)c1ncc(C)s1 c1(C2CCC(NC(C3CNCC3C(F)(F)F)=O)C2)ccc(Cl)cc1 NC(=O)CCC(=O)NCc1cccc(NC(C2CCS(=O)(=O)N2)=O)c1 c1(CC(=O)NC(C2CCN(C)C2)C)ccccc1F.C1(=O)C(CO)N1 N1(C(CCC=C)=O)CC2(C1)CN(C(C1(c3ccsc3)CC1)=O)C2 C1(NC(C2(CC(C)C)COC2)=O)CCCC2CN(C(C3CCCC34CC4)=O)CC12 c1(C(N2CCCC(NCCOc3ccc(C)cc3C)C2)=O)n[nH]c(C)c1[N+](=O)[O-] N1(C(C2CC(C)=C(C)CC2)=O)CCCC2(CCN(C(=O)C(F)(F)C3CC3)CC2)C1 c1(CC(=O)NCC2N(C(C(C)OCC)=O)CCC2C)ccc2c(c1)CCCC2 C=C(C)CCC(=O)NC1CCCC1NC(=O)C(C12CCC(CC1)C2)OC C(=O)(C(CCCOC)N1CCCC(n2cc(Cn3cccn3)nn2)C1)NC c1(C(=O)NCC(CCNC(c2nnc(O)nc2O)=O)O)coc2cc(O)ccc12 C(=O)(CCC(F)(F)F)NCC1(C(C)NC(=O)C2=NOCC2)CC1 c1(CC)ccccc1CC(=O)NCC1CCN(C(=O)C(c2cc(Br)co2)=O)C1 N12CCN(CC1)CC1CC(C1)C2=O.c1(C(C)NC=O)ccc(N(C)C)nc1.CO c1(C2C(CC(=O)NCC(C(=O)O)NC(=O)OC)C2)cccc(OC)c1 N1(C(CCOCCN(C)C)=O)CC2CN(C(C3(O)CCOC3)=O)CCC12 N1(CC(=O)NCC(C(C)C)NC(C(CC)(C)O)=O)C(=O)c2ccccc2S1(=O)=O CC(F)CN=c1[nH]c(N(CCCS(N)(=O)=O)C)nc2c1CCCC2 C1(NC(C2CCC(NS(C)(=O)=O)C2)=O)CC2CC1N(C(c1cnc[nH]c1=N)=O)C2 Cc1nc(C2CC2)sc1C1C(C(=O)OCC(=O)Cc2ccccn2)C(C(F)(F)F)C1 N1(C(COC(CC)C)=O)CCC(CF)(NC(=O)COCc2cccc(Cl)c2)C1 C=CC1(C(N2CCCC(CC)C2)=O)CCN(C(c2ccc(OC)o2)=O)C1 Cc1nc(CNC(=O)CCCN(C(=O)C(C)c2cc[nH]n2)C)c(C)s1 c1(CC)cc(C(N2CCN(C(c3cnnn3C)=O)C3CC23)=O)cc(O)n1 c1(C(=O)NCC=CCNC(CCNC(=O)OC)=O)cc(C)n(C2CCC2)n1 c1(C(=O)NCCC2CCCN(C(CC3(C)CC3(Cl)Cl)=O)C2)cccc(Cl)c1O c1(C(=O)NCC(C)CC2CCCO2)ccc2nncn2n1 Cc1c(C(=O)N(CC(C)O)CCNC(c2ccc(C#N)[nH]2)=O)nn2c1CCCC2 c1(C(=O)NCC2CC(NC(C(C)(C)C3CC3)=O)C2)ccc(N)c([N+](=O)[O-])c1 N(C(=NCC1CC(=O)N(CCSC)C1)N(C)Cc1nnnn1CC1CC1)C(CC)C N1(C(CS(C)(=O)=O)=O)CCOCC2(COCCN2C(c2ccc(O)nc2Cl)=O)C1 N1(C(C(CCF)NC(CNC(C(C)(C)C)=O)=O)=O)CC(=O)NC2(CC2)C1 C1(CC2CC2)CC=CC(c2csc(N(c3[nH]cnc3C#N)C(=O)OC(C)(C)C)n2)C1 N1(C(Cc2ccc(C(N)=O)cc2)=O)CCC2(NC(=O)CSC(F)(F)F)CC2C1 c1(CCNC(=O)NCc2snc(C(C)C)n2)ccc(F)c(C(F)(F)F)c1 c1(N(CCOC)C(C)=O)ccccc1.c1(C2CNC(=O)O2)ccccc1 c1(C(=O)NC2CC3CC(NC(C4(CC(C)C)CCC4)=O)C2C3)c(N)cccc1Cl Cc1cc(Cl)ccc1C(N1CCC(CNC(=O)CC2CCC(O)C2)C(C)C1)=O Cc1nc2ncnn2c(C(=O)NC(CN(c2cnc(O)n2C)C)C)c1C N1(CC(N2C(CNC(CCC(=C)Cl)=O)CC(OC)C2)=O)CCCCS1(=O)=O N1(C(CC(C)(C)C2CCCCC2)=O)CCOCC(n2cc(C3(CO)CC3)nn2)C1 N1(C(COC(CC)C)=O)CCC(CNC(C2CCC(O)CC2)=O)C1(C)C C1(n2c(-c3cccnn3)nc(CCC(C)C)n2)CCS(=O)(=O)CC1 N1(COC(C)(C)C)CCc2cc(NCc3cc(Br)cnc3OC(F)F)ccc21 C1(COC)CCCCN1C(=O)CC(=O)N1CC(N2CCS(=O)CC2)C1 Cn1cc2ccc(CN3CC4(CC4C(=O)NCC4CNCCO4)C3)cc2n1 c1(C(=O)NC2CC(CNC(C(C)N3CCC3)=O)C2)c(F)c(F)cc(F)c1F C1(c2n(C(C)C)nnn2)(NC(C2CCCCC2)c2ccccn2)CCC(C#N)C1 C1(NC(c2cnc(CC)o2)=O)CCC2(CCN(C(=O)C(C)(C)O)C2)C1 C12(C(N3C(CNC(CCOCC#C)=O)C(CC)CC3)=O)CC3CC1C2C3(F)F CC(C)CC(C)(C)C(=O)N1CCCC(C(=O)NC2CCC(N(C)C)CC2)C1 N1(CC(=O)NCC2CN(C(C(N)c3ccoc3)=O)C2)C(=O)CSC1=S C1(NC(c2ccc(C)o2)=O)C2CCC1N(C(=O)Cc1cc(C)n(C)n1)C2 c1(NC(C(=O)NC(c2ncc(C)[nH]2)C2CC2)=O)cc(Cl)ccc1OCC(F)(F)F C(=O)(C(S(=O)(=O)NCC1(c2ccccc2)CC1(C)C)C1CC1)OC N1(C(=O)COCC2CCC2)CC2(CC2)CC1CNC(C1(CCF)CCC1)=O N1(C(c2onc(C)c2C)=O)CC2CN(C(=O)C3=CSCS3)CC2C1 N1(C(c2cnn(C)n2)=O)Cc2ccnn2CC(NC(c2cc(Cl)sc2Cl)=O)C1 c1(C(=O)NCCC2CCCN2C(=O)CCC2CCC2)c(F)ccc(O)c1F N1(C(C2C(C)(CC)C2)=O)CCCC(C(N2CCC(C(=O)NC)CC2)=O)C1 N1(CC)CC(C)C1CNC(C(N)=O)C1CC1 c1(CC)ccc(C)cc1C(N1CCC(O)C(NC(C2CC(C(F)(F)F)C2)=O)C1)=O c1(SCC(=O)N(C2CCN(C(C3CC3C3CCCO3)=O)C2)CC)cccc(C)c1 c1(CC)c(C(=O)NCC(O)CNC(C2(C)CCCNC2=O)=O)cccc1C c1(C(C(=O)NC2(NC(=O)OC(C)(C)C)CC2)N(C)C)ccc(F)c2[nH]ncc12 C1(CC)CCN(C(=O)CC2CCCOCC2)C(C(N2CCCC(OC)C2)=O)C1 Cc1cccc(F)c1C(N1CCC(NC(c2nccn2C)=O)C(F)C1)=O C1(NC(COC)=O)CCCN(C(c2ccc(OC(F)F)cc2OC)=O)CC1 C1(NC(C(=O)OC)C)CCN(C(=O)C(CC)OC)CC1(C)OC(N)=O CCCC(C(=O)N1CCC(C(=O)NCC2CC2Cl)C1C)N(C)C Cc1nn2c(c1C(=O)N(CC(C)C(c1c(F)ccc3occc13)=O)C1CC1)CCCC2 C(=O)(C(CC)C(C)(C)CC)N1CCCC(F)(C(=O)NCC=C=C)C1 c1(CNC(c2nnnn2CCC(=O)OCC)CCC)cccc(Br)c1OC CC(C)CC(CNC(=O)Cn1ccnc1)C(=O)NCCS(C)(=N)=O C1(CNC(COCC)=O)CN(C(=O)C(C)(Cl)Cl)CCC12CCOCC2 N1(CC(C(=O)N(C(C)(C)C)CCF)OC(NCC)=O)CCC(C)CC1 C(=O)(C(C)CC(F)(F)F)N(C1CCC(N)CC1)C(C1CC1c1cccs1)=O.CO C#CC1(C(=O)N(CC(C)C(F)(F)F)C)CCN(C(=O)C(CO)C(C)(C)C)CC1 CC1(CNC(=O)C=CCF)CCN(C(C2(c3cncnc3)CCCC2)=O)CC1 c1(C(N2CCN(CC(C3(C)CC(F)C3)=O)CC2)=O)ccc(-n2ccnc2SCC)cc1.CO CCCC(C(=O)NC1(C(=O)N(C2CCCC2C#N)C)CC1(C)C)OCC N1(C(C(C)(Cl)Cl)=O)C2CCC1CN(C(=O)COCc1ccncc1)C2 Cc1ccc(C(N2CCC(O)C(NC(=O)Cc3cccc(F)c3)C2)=O)c(O)c1 CC1CCN(c2ccc(C(=O)NC(Cc3ccncn3)C(=O)O)cc2)CC1 CC1(C)CC(NC(=O)C(Cc2ccoc2)NC(C2CCS(=O)CC2)=O)C(C)(C)O1 C(=O)(CC1=CCCCC1)NCC1OCC(C(N(C)Cc2nccs2)=O)C1 CCCCCC(F)C(=O)NC(CC(=O)NC1CC2CC1OC(=O)N2)C(F)(F)F S(=O)(=O)(CCC(=O)N1CCN(C(C2C(F)(F)C23CCC3)=O)C(CCO)C1)N(C)C C(=O)(C(F)C(=O)NCC(C)(C1CC1)NC(=O)C=Cc1cn(C)cn1)OCC CC1CCC(CNC(c2ncc(F)cn2)=O)CN1C(=O)CC1CCC2(CC1)CC2 N1(C(c2c(C)nco2)=O)CC(C(=O)NCCN2C(=O)CCC2=O)C(C)(C)C1 c1(C(N2C(CNC)CCCC2)=O)cc(S(=O)(=O)NC)oc1C C1(C(=O)NC(CCC)(C)C)COC2(C1)CN(C(=O)CCc1cncs1)C2 C(=O)(CCC[N+](=O)[O-])N1CC(OCC)C(CNC(=O)C(C2CC(F)(F)C2)O)C1 c1(C(N(C2C(N(C(C(CCC)O)=O)C)CCCC2)C)=O)ncc([N+](=O)[O-])cc1C c1(NC(C2CN(C(C3CC3C3CC3)=O)CC2C)=O)c(C(F)(F)F)cc(F)cc1Br c1(OC)cc(OC)[nH]c(=NCC(C2CCCC2)NC(c2cnco2)=O)n1 Cc1cnn(CC(=O)NC2C3CCC2N(C(c2coc(C(F)F)c2)=O)C3)c(=O)c1 C(=O)(C(C(C)c1ccccc1F)NC(c1cncnc1-c1ccccc1)=O)OC C1(N2CC(O)(CC)C2)CCC(=O)N(C)CC1 c1(C(N2CC3CC2C3C(F)(F)F)C(=O)NC(C(=O)OC)C)cc(OC)ccc1C c1(C(=O)NC(C2CCN(C(C(COC)N(C)C)=O)CC2)C)cc(N)cc(C)c1F N1(CC(N2CCC(NC(c3cnnc(Cl)c3)=O)(CF)C2)=O)CCc2ccccc21 C(=O)(C(F)C(C)C(F)(F)F)NC1(CC=C)CN(C(c2c(C)nn(CC)c2Cl)=O)C1 c1(OC)cc(C)c(CN2CC(C(=O)Nc3cc(F)c(Br)c(F)c3)C2)c(O)c1 Cc1nn(CCF)cc1NC(C1CCCC(NC(C2C(C(C)C)C2(C)C)=O)C1)=O Cc1ccncc1C(=O)NC1CCC1NC(C1CNC(=O)N1C)=O Cc1ccc(C(C)OC(C2CCC2)=O)cc1[N+](=O)[O-] C1(CCC)CN(C(=O)CCN2CCN(C)CC2)CC1NC(c1cscn1)=O c1(OC)ccc(C(c2nnnn2C)NCc2cc(Cl)cc(Cl)c2)c(Cl)c1OC C(CC(C(=O)NCC1CCN(C(C2CCS(=O)(=O)N2)=O)CC1)NC=O)SC C1(CC)C(C(=O)NCC(C)(C)CNC(c2c[nH]c(=S)cn2)=O)CCN1C Cc1cc(=O)c(C(N2CCCC(N(C)C(C3CCOC3(C)C)=O)C2)=O)c[nH]1 c1(C(C(N2CCC(C3CCCN3C(=O)Cn3cc(Cl)cn3)C2)=O)F)ccccc1 C1(CC)(OC)CN(C(=O)CN(C2CCC2)C(c2c[nH]cc2C2CC2)=O)C1 c1(C(N2C3CC(NC(c4c(CC)nccc4)=O)(C3)C2)=O)cc2cc(C)ccc2s1 C(C(=O)NCC1(CNC(=O)C(F)(F)c2cnccn2)CC1)(C(C)C)SC C1(NC(Cc2nc(C)oc2)=O)CCN(C(c2cncc(Cl)c2Cl)=O)CC1O O=C1CCC(C(=O)NCC2(O)CN(C(=O)C=C3CCC3)C2)CN1 C#CC1C(C(N2CCC(N(C(=O)Cc3sc(S)nc3C)CC)C2)=O)C1(C)C CCC(CC)C(C)C(=O)N1CC(OCC(=O)NC2CCCCC2C#N)C1 C1(CNC(C2C(C(C)C)C2)=O)CCN(C(=O)Cn2cc(C3CC3)cn2)CC1(F)F c1(CN(C(CCN(C(C(=CC2CCCC2)C)=O)C)=O)C)ccc(O)cc1 CN=c1[nH]cc(C(=O)NC(C(=O)NC2CCCC3CC23)C2CCC2)s1 Cc1c(F)ccc(C(=O)NCC(O)CNC(=O)COc2ccsn2)c1C C=CCCCC(C(=O)N(C(C)CO)C)NC(=O)CCn1cncn1 N1(C(C(COC)O)=O)CC2(CNC(c3csc(O)n3)=O)CC1CO2 c1(Cc2c(NC(N(C(CF)CF)C)=O)cco2)ccc(C#N)cc1 N1(C(c2c(=O)cc(C)[nH]c2)=O)Cc2occ(C(N3CCOC(C4CC4)C3)=O)c2C1 CN1CCC(N(C(=O)N(C)C)CNc2c[nH]nc2-c2ccc(Br)s2)CC1 C(=O)(CCN=C(NCc1ccc(C2CC2)cn1)NC1CCCC1(F)F)N(C)C c1(C(=O)NCC2(O)CC(CNC(C3CC(OC)C3)=O)C2)cc2n(n1)CCCO2 c1(NC(=O)NC2CCCC(F)C2)cccc(Cc2cccc(Br)c2)n1 CC1(NC(=O)C=Cc2ccco2)CC(C(=O)NC(CO)C2CCC2)C1 C(=O)(C1CCCc2cccnc21)N(C(C)C)CCN(C(=O)C(O)CC(N)=O)C CCCCCC(O)C(=O)NC(C1(CNC(=O)COC2(C)CCC2)CC1)C CC(C)CC(C)C(=O)N1CCCC1CN(C)C(C1(C)CCCO1)=O CCCC(C)C(CO)NC(c1cc[nH]c(=N)c1)=O C1(C(=O)NC(c2scc(C)n2)C)CC2CCCC2N1C(c1cc(F)cnc1O)=O Cn1nc(C(=O)NCC2CCC(NC(c3ncc(Cl)s3)=O)C2)cc1C#N C(CCN=C(NCCC1CC1)NCCSc1cccs1)=CC=C N1(C(CCC(=C)C)=O)CCC2(CC1)CN(C(=O)C(CCC)=CC)C2C(C)C Cc1ccc(C(C)C(=O)NCCCCC2(Nc3ncncc3OCF)CC2)cc1 c1(C(N2CC(O)(CNC(c3cccc(Cl)c3Cl)=O)C2)=O)c[nH]c2ccc(Br)cc12 Cc1ccc([N+](=O)[O-])c(C(N2CCC2CNC(C2OCCCO2)=O)=O)c1 C1(CNC(COC(CC)(C)C)=O)CN(C(C2(C)CC2C)=O)CCN1C c1(CC)ncc(C(=O)N(C2CCCCC2NC(c2cc(CCO)on2)=O)C)cn1 CC(CC(=O)N1CC(CC(C)(C)CNC(=O)CN2C(=O)CCC2=O)C1)C(C)(C)C C(=O)(C(C)CC(C)C)NCC(C1CC1)NC(c1ccc(OCCC)cc1)=O N1(C(c2cn(C)c(=O)cc2)=O)CCCCC12CC(NC(=O)C=CC(N)=O)C2 c1(C(N2CC3CC(NC(=O)C=CC(F)(F)F)CC3C2)=O)cccc(C#CCO)c1 c1(C(N2CC(SC)C(NC(=O)C(C)=C3CCC3)C2)=O)cc(S(N)(=O)=O)cn1C C1(C(=O)NCC2CCC(NC(c3c(C)ocn3)=O)C2)CCCCN1CC(F)F N1(C(CSCC=C)=O)CC(NC(C2(c3cccc(F)c3)CCC2)=O)C(C)(C)C1 c1(NC(c2ccnn2C)CC)cc(N2CCC(Cn3cccn3)C2)nc(C)n1 N1(C(C2(CC)CC2(F)F)=O)CCC(CF)(NC(C2CC3CC2C3)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(F)(C(=O)Nc2c(CC)csc2)C1 C(N=c1nc(N2CCC(OC)C(C)C2)c2c([nH]1)CCOC2)C1CC(COC)C1 C1(CNC(C2CC(=O)NC2)=O)CN(C(=O)CCN2CCC2)C2(CCOCC2)C1 n1(C(C)C)ccnc1C(=O)NCC1(CNC(C2(C)CCC2)=O)CC1 Cc1n[nH]c(C)c1CCC(N1CCOC(CC(=O)NCCCCCN(C)C)C1)=O c1(NCC(C)NC(=O)COC(F)(F)F)nc[nH]c2ncc(C(N)=O)c1-2 Cc1oc2c(F)c(F)c(F)c(F)c2c1C(=O)NCCC(C)NC(c1ccoc1)=O C1(C(=O)NCC(CCC)NC(C2(C(C)C)CC2)=O)CCC(F)(F)C1 C1(CN(C(=O)C(CCN(C)C)NC(=O)OC(C)(C)C)C)CCC(F)(F)C1 C1(C(C)NC(=O)COC(F)F)CCCN(C(c2cc[nH]c(=N)c2)=O)C1 C1(NC(C(CC)OC)=O)CC(CNC(C2(CC3CC3)CCCO2)=O)CC1O C1(CNC(c2cc(C)c(Br)cn2)=O)C2CCC1CN(C(=O)CCC(N)=O)C2 c1(OC)nccc(Br)c1C(=O)NCCN(C(=O)CNC(C1CCCC1)=O)C C1(NC(c2ccc3occc3n2)=O)CC12CCN(C(C1CCNC1=O)=O)CC2 N1(C(CC2CN(C)C2)=O)CCC(O)C(N(C(=O)Cn2cc(C(=O)OC)cn2)C)C1 C(=O)(C1c2c[nH]nc2CN1C(c1ncc(C)cc1C)=O)Nc1c(CC)cccn1 C1(C2CN(C(c3ccc(F)c(O)c3)=O)C2)(NC(C2CC(C)OC2)=O)CC1 C=CCN=C(NCC1(OC)CCCS(=O)(=O)C1)NCC1(SC)CC2CCCC12 C1(C)(CC)CC(NC(=O)CCn2nc(C)nc2C)CN1C(c1[nH]c(C)nc1C)=O C(CCCCN=c1[nH]c2c(c(=NCCCn3cc(Br)cn3)[nH]1)COC2)C1C(CC)C1 c1(NC(C2(C)CC2C(F)(F)F)=O)nc(C2CC2)sc1Br N1(C(c2ccc(OCCO)cc2)=O)CC2(C1)CN(C(=O)C(F)(F)C1CC1)C2 C(CNC(c1cc(Cl)c(Cl)n1C)=O)(CC(F)(F)F)NC(CC(COC)C)=O C1(C(N2CC(OC(C)C)C2)=O)CC2(CC(NC(=O)C(C)n3ccnc3)C2)C1 C(c1ccccc1)=CC(C(=O)NC1CC(NC(C2(OC)CCCC2)=O)C1)C N1(C(C(C(C)C)F)=O)CC2(CCC2)CC1C(=O)NC12CC(C1)C2 C(=O)(CCCCC(C)=O)N(CC(=O)NCC1CC2CCCC2C1)CCC c1(C(N2CC3(C)CC2(CNC(=O)CCC(N)=O)C3)=O)cnn2cc[nH]c(=O)c12 CC(C)(F)CCC(=O)N1CCCCC(CCC(=O)NCCc2csnn2)C1 Cc1cc(C=CC(=O)NC(C)(CNC(=O)C(C)(C)CF)CO)ccc1F C(C)(C(=O)N1OC2CCC1C2)C1CCCCN(C(c2c(OC)cncc2)=O)C1 c1(C(N2CC(CNC(c3cn(C)nn3)=O)C(C(F)(F)F)C2)=O)cc(N)cc(Cl)c1 C1(OC)CN(C(C2CN(C(C3CC4C=CC3O4)=O)CC2OC)=O)CC1(C)C N1(CC(=O)N(C)CC2CN(C(=O)CCCc3cccs3)C2)CCCS1(=O)=O C(=O)(C(O)CC(F)(F)F)N1CC(CC)C(C(=O)N(CCCC(O)CO)C)C1 C=C=C(C)CC(=O)NC(CC=C)C(=O)NC(c1nncn1C)C Cn1ncc(C#N)c1C(=O)NCC(C1CCCCC1)NC(c1ccncc1)=O N1(C(C(CC)OCC)=O)CC(NC(=O)CCc2cn(C)nc2C)C(S(C)(=O)=O)C1 C=C(Br)CCC(=O)N1CCCC1C(N1CCC(C(=O)OCC)C1C)=O C1(NC(=O)Cn2nnc(=O)[nH]2)CN(C(c2ccc(F)cc2)=O)CC1C(F)F CCCCC(O)C(=O)N(CC(C)(C)NC(C1Cc2ccccc2O1)=O)C CC1(O)CN(C(=O)C2=CCC(NC(=O)Cc3ccoc3)C2)CCC1O C(=O)(CCCCC(=O)NC1CCCC(CNC(=O)CCNC(N)=O)C1)N(C)C N1(C(CN(C(C(C)C)=O)C)=O)CCC(C(=O)NC2CC2(Cl)Cl)C(O)C1 c1(C(=O)NC2CCC2NC(=O)C(F)(F)F)cnn(C2CCCC2)n1 C#CC12CC(CN1C(C1CCC(C3CC3)N1C(=O)CNc1ccccn1)=O)C2 Cc1cccc2nc(N3CCC(C)(CNC(C4CCOC4C)=O)CC3)oc12 C1(CN(C(c2n(CC#C)ccn2)C(=O)NCCOC)C)CCCN(C)C1=O N1(C(CCCOCC)=O)CCC2CN(C(c3nc[nH]c4ncnc3-4)=O)CC2C1 C(=O)(CC(C)P(C)(C)=O)NC1CCN(C(c2c(C)nccn2)=O)CC1C(N)=O c1(C(=O)NCC(CCCC)NC(=O)Cn2nccc2C)ccc(O)c(C)c1 Cc1ncc(NC(C2CC2C(=O)NC(c2ccc(Cl)c(Cl)c2)CO)=O)cc1F c1(CNC(C(CCC#C)O)=O)ccc2c(c1)CN(C(c1cnc(O)n1CC)=O)C2 C1(NC(c2nn(CC)c(C)c2)=O)CCCCN(C(C2C(C)C2(F)F)=O)C1 C(=O)(C(F)CCC(C)C)N(CCCNC(CCCCN(C(C)=O)C)=O)C c1(N2CCCC(NC(c3c(CC)oc(C)c3)=O)CC2)ncnc2cnn(C)c12 C1(C(N(CC(C)NC(C(CC=C)(F)F)=O)C)=O)CC2OC(C)(C)OC2C1 N1(C(OC)=O)CCN(C(C2C3CN(C4CCOC4=O)CC23)=O)CC1 N1(C(C(CCOC)C)=O)CC(C2(NC(=O)CC=C(Cl)Cl)CC2)C1 c1(OCCC)c(Cl)cc(C(N2CCN(C(C3CC4CC4N3)=O)CC2C)=O)cc1Cl c1(C(N(CC(C)NC(c2ccc(=O)n(C)n2)=O)CC)=O)snc2ccccc12 C1(C(N2CCC(CN(C)CC)C2)=O)C2CC1N(C(=O)CC1CCC(C)CC1)C2 C(C)(C(=O)N(C)OC1CCCC1)N(C(C(C)CN1CCOCC1)=O)C C(=O)(C1CSc2ccccc21)NC1CCN(C(CC2(C=C)CC2)=O)C1 C1(CNC(C2(C(C)C)N(C(C3CC(OC)C3)=O)CCC2)=O)CC12CCOCC2 c1(OC)ccc(C(N2CCC2CNC(=O)Cc2csc(S)n2)=O)cn1 CC1CCc2c(C(=O)NC3CN(C(=O)C=C4CC4)C4(CCC4)C3)csc2C1 N1(CC(=O)N)CCC(F)CC1.Cc1c[nH]cc1CN1CC(=C(C)C#N)C1 C#CC(CNC(=O)CC1CC(NC(c2ccoc2C)=O)C1)C(C)C CC(C)C(C)C(C)CC(=O)N1CCN(c2ccc(S(=O)(=O)N(C)C)cn2)CC1 c1(C(=O)NCC2(NC(C3CCC(=O)O3)=O)CCCC2)c(O)cc(Cl)cc1Cl C(CCC(=O)Nc1cc(C)cc(O)c1)(C(C)C)NC(c1ccc(C#C)nc1)=O CCCCCC(C)(CC)C(=O)NCC1CCN(C(c2ccc(Cl)cc2Cl)=O)C1 C1(C(=O)NCC(CC=C)(C)C)N(C(=O)CC(C)COC)CC12CCCC2 N1(C(C#CCNC(C(C)=C2CCC2)=O)=O)CCC(CC(C)O)CC1 C1(OC)(OC)CCC1C(=O)NC1CCC(NC(=O)Cc2cccs2)C1 c1(C(N2CCCC(C(C)NC(=O)C=Cc3cc[nH]c3)C2)=O)n[nH]c2c1CCCC2 N1(C(C(C)OCC=C)=O)CCCC2CN(C(c3nc(CC)no3)C)CCC12 C12(C(=O)NC3CC(C)(NC(=O)CN4CC=CC4)C3)C(=O)C3CCC1C2C3 c1(C(N2CC(NC(CC3C(C)(C)C3)=O)C2)=O)ccc(F)c2c1OCC2 N1(C(CC(=O)NC)=O)CCC2(CCCC2CNC(C2CC2(Cl)Cl)=O)CC1 CC(C)(F)CCC(=O)NC(C)(CNC(C12CC(F)(C1)C2)=O)Cn1cccn1 N1(C(c2ccc(C)cn2)=O)CC2CC(C1)N2C(C1CCC(C2CCCO2)C1)=O c1(C(=O)OC)sc2ccc(Br)cc2c1N(CCC(C)OC)C N1(C(CC(=C)C)=O)CCC(C2CCOCC2)(CO)C1.C(C)(C(=O)O)=CC(=O)N C1(C(=O)NC2CN(C(c3ccc[n+]([O-])c3)=O)CCC2F)CCS(=O)(=O)C12CCC2 N1(C(c2cc(OC)no2)=O)CC2CC1CN2C(C1CC(=C(F)F)C1)=O C(=O)(CCCn1ccnc1)OCCC(=C)C C(N=c1ccc(NCc2cc(Cl)c(Cl)cc2O)c[nH]1)c1cc(C(=O)OC)no1 C1(C(=O)NC(CC)CNC(=O)CC2CCCOCC2)CCOC2(CCC2)C1 C1(C(=O)NCCN(C(Cc2c(C)c(F)ccc2)=O)C)CCN2CCCC2C1 c1(C(N(C2CCN(C(=O)CC(O)C(C)C)C2)CCC)=O)ncnc(C)c1OC C(CCCCCNC(c1cn(CCF)nn1)=O)NC(C1C(OC(C)=O)C1)=O c1(C(=O)NCC2C(NC(c3cc(F)cnc3O)=O)C2)c(O)nnc2c1CCCC2 N1(C(C2(C#C)CC2)=O)CC(C)CN(C(c2ccc(-c3ccncc3)o2)=O)CC1C C(=O)(C(CCS(C)(=O)=O)OC)NC1CCCN(C(c2c(CC)nccn2)=O)CC1 C1(C(C)C)CN(C(c2ccncc2)=O)CC1C(=O)NC(C)CN1CCOCC1 C1(C(=O)NCC2CC2CO)(CNC(COCCC(C)C)=O)CC(C)(C)C1 N1(C(c2c(CC)onc2)=O)CCCCC1C1(NC(c2c(C)n[nH]c2C)=O)CC1 CCCCCCC(CC)NC(=O)CC1(O)CCN(C(=O)CC(C)(C)C#N)C1 c1(-c2c(C(=O)NCC3(NC(C4CC4(F)F)=O)CCOC3)nco2)ccc(Cl)cc1 c1(C(N)=O)cccc(CCC(=O)N2CC(n3cc(C4(C5CC5)CC4)nn3)C2)c1 N1(C(C2(C3CCOCC3)CC2)=O)CCC(CNC(c2cnc(O)o2)=O)C(F)(F)C1 C(CC(=O)NCCc1ncc[nH]1)(C(C)C)NC(C1(C=C)CCCC1)=O C(=O)(CCCCCCNC(=O)Cc1ccccc1C)N1CC(CC)OC(C)C1 C(=O)(CC1=CCCCC1)NC(c1cn(C)nn1)C(=O)NCC1CCC(F)C1 C1(NC(C2ON=C(C(C)C)C2)=O)CN(C(C2CCS(=O)(=O)N2)=O)CC2(CC2)C1 C(=O)(CCC(C)O)NC1(CO)CN(C(c2c(CC)ocn2)=O)C1 CC(C)CCC(O)C(=O)N1CCOC(CC(=O)NCC(C)C#N)C1 Cc1ccc(NC2(c3nnnn3C)CC2(C)C(C)C)cc1Br CC(O)CCC(=O)NC1CCCCC1NC(=O)COCc1ccnc(O)c1 c1(CC)cc(=NC2CN(C(c3cc(N(C)C)ccn3)=O)CC2C)[nH]c(Cl)n1 c1(OC)cccc(C(O)C(N2CCC(N(C(=O)Cn3cnnc3O)C)C2)=O)c1 C1(C(=O)NC(C2CCCCC2)CNC(=O)C(C)(C)N(C)C)(CC)CC1(F)F N1(C(CC(C)C2CCCCC2)=O)CCC(CO)(NC(c2cscc2Cl)=O)C1 C1(NC(C(C2CC2)SC)=O)CCC(C(=O)N(C2COCC2O)C)C1 c1(CN2C(C(=O)NCc3cn[nH]c3)CC(=C)C2)cc(C)c([N+](=O)[O-])cn1 C1(CC)CC(C(=O)NC(C)(C)CN(C)C(c2oc(C)cc2C)=O)CCO1 c1(C(=O)NCCC2(O)CCN(C(C(C)CF)=O)C2)cnn2c1OCC(C)(C)C2 c1(C(=O)NC(C(C)NC(=O)COC2CC=CC2)(C)C)ccc2c(c1)NC(=O)CN2 C(CC(=O)O)(C(=O)OC(C)=O)NC(c1ccc(C(F)(F)F)cc1F)C N1(C(CCC=C)=O)CCC(N2CCN(C(C3CCCO3)=O)CC2)CC1 C(c1cc(Cl)c2c(c1)OCO2)=CC(N1C(C(CC)O)CCC1)=O N1(C(CC(C)N(C)C)=O)CCCCC1CNC(=O)C(C)(C)n1cncn1 CN1N=C(C(=O)NCC2CCC(NC(=O)CC3CC4(CC4)C3)C2)CCC1=O C=C=CC(C)C(=O)NC(c1ccccc1F)CNC(c1ccon1)=O c1(C(=O)OC)cc(CSC2(c3ccc(OC(F)(F)F)cc3)CCC2)cc(C)c1 c1(NC(=O)NC(CCC)CCO)ccc2c(c1)CCOC2 C1(C(=O)NCC(C)(C)CN(C)C(c2nc(C)sc2C)=O)(COC)CCCOC1 c1(OC)ccc(C(=O)NCC2CCN(C(c3nn(C)cc3Cl)=O)C2(C)C)c(C)n1 c1(OCC(=O)NC2CC(C)N(C(=O)CNC=O)C2)ccc(Cl)c(F)c1 c1(C(N2CC(CO)C(C)(C)C2)C(=O)NCCCSC)ccc(F)cc1I O=C1NCc2cccc(C(N3CCCCC3CC(O)C(F)(F)F)=O)c2O1 N1(C(C2C(C)(C)CC2)=O)CCC2(CCC(CNC(=O)C3=NOCC3)O2)CC1 c1(C(N(CC(=O)NCC2C=CCOC2)CC)=O)ccnc(O)c1 Cc1c(Br)c(C(N2CC(NC(=O)CCc3nnc(S)n3C)C2)=O)nn1C C1(CNC(=NCC)NCc2cc(Cl)nc(=N)[nH]2)CC1C1CCCC1 c1(C(=O)NC2CCN(C(c3c(Cl)cn(C)n3)=O)C2)cc(F)cc(F)c1N c1(NC(CCSCCNC(C=CCSC)=O)=O)cccc(Cl)c1C N1(C(Cc2cnc(C)o2)=O)CCCC(N(c2ncc(Br)cn2)C)C1 Cc1ccn(CC(=O)NC2CC3CC2N(C(=O)CC(C)n2ccnc2)C3)c(=O)c1 N1(C(c2ccc(C#C)o2)=O)CCCC2CCN(C(=O)CC3(O)CCC3)CC12 CC1CCN(C(=O)OC(C)(C)C)C=C1C(=O)N1CC(=O)NC(C)C1 C(=O)(C(C)(C)CSCC(F)F)NCC1CC(N(C(=O)CC2CC(F)C2)C)C1 c1(CC)ccnc(C(=O)NC(CNC(=O)C(c2cscn2)N(C)C)CO)c1 Cc1cc(CC(=O)NC2(CCC(=O)NC3CNC(=O)O3)CCC2)no1 c1(C(=O)NCCCNC(C2C(C(=O)OCC)C2)=O)ccc(CN(C)C)cc1 CCC(COC)(CC)C(=O)NCc1c[nH]nc1C(N1CCC(CO)C(O)C1)=O CC1CCOCCN1C(C1CCOCCN1C(=O)CCN1CCOCC1)=O c1(CNC(COC(CNC(C2(CSC)CC2)=O)(C)C)=O)oc(C)nc1C N1(CC(=O)N(c2ccccc2O)C)Cc2c(Br)cccc2C1=O C1(CNC(c2nc(OC)oc2)=O)CCCCC1NC(c1cnsn1)=O Cc1cc(C(=O)NC2CCC(CNC(C3(C)CC(C#N)C3)=O)C2)c(C(F)(F)F)o1 N1(C(C2CN(CCC)C(=O)C2)=O)C2CCC1C(C)C(NC(=O)C(C)S(C)(=O)=O)C2 C(CCCCC(=O)N1CCC(CC)C1CNC(C1CCCC(=O)CC1)=O)=CC C1(NC(=O)COCC(F)F)C=CCN(C(c2cccc(Br)c2)=O)C1 n1(CCC)nc(C)cc1C(C(=O)Nc1ccccc1C)N(C)Cc1nc(C)cs1 O(N1CCC(CC(=O)NCCNC(C2(Cl)CC2(C)C)=O)CC1)CC C(=O)(C(N)C(C)CCC)C(=O)CCCCC(C)C.C=CCCCCNCC c1(OCCNCCCNC(C2N(C)CC(C)(C)C2)=O)ncc([N+](=O)[O-])cc1F c1(C(=O)NCCC(C)N(C)C(C2CN3CCN2CC3)=O)cn(C)c2ncccc12 N1(C(C2CCCOC2)=O)CCCCCC(N=c2ncc3c(Br)cccc3[nH]2)C1 N(C(=NCCCC(=O)OC)NCc1cc(Cl)c(Cl)s1)C(CC)CC C1(C(=O)NC(CC(=O)NC)C2CC2)CC2(C1)CN(C(=O)CC1CC(C)=NO1)C2 CC(C)(C(=O)NCCC1(NC(c2cnc(-c3ccccc3)[nH]2)=O)CC1)C(N)=O c1(NC2CN(C(c3nccc(OC)c3OC)=O)C2)c(Cl)cc([N+](=O)[O-])cc1Cl Cc1ccnc(C)c1C(=O)NCC1CN(C(C2CCCC(C)(C)C2)=O)CCCO1 n1(CC)cccc1C(=O)NC1CC(N(C(=O)COC)C)C1 c1(OC)c(C(=O)NC2CCCCC2NC(c2nc(Cl)cs2)=O)nc(O)nc1O CC(O)(CC(=O)OCc1nc(C(F)(F)F)nc(=N)[nH]1)CC(=O)O CC(C)CC(C(=O)NCCCN1CCCC1C)NC(=O)C1=NOCC1 C1(CCNC(C(CC)N(C)C)=O)CCCN(C(c2ncoc2-c2cccs2)=O)C1 C1(C(N2C(CN(C(=O)CCCC(F)F)CC)CCCC2)=O)CCCNS1(=O)=O N1(C(C2CN(C(C)(C)C)C(=O)C2)=O)CC2CCN(C(=O)Cc3cncnc3)CC12 Cc1[nH]c(=N)sc1C(=O)NCCOC(C)(C)CNC(C1CCCCCC1)=O CC1(CNC(C2CCC(C)(F)CC2)=O)CCCN(C(C2(C)C=CCCC2)=O)C1 C(=O)(CC1=CCOCC1)NC(CSC)(C)C(=O)NCC1CC1Cl c1(SCc2cnc(CC)s2)cc(C(=O)NC2CC(C(=O)OC)C2)nn1C c1(OC)ccn2c(C(=O)NCC3(C)CCCN3C(C3CCCC3)=O)cnc2c1 Cc1ccc(F)cc1CC(=O)N(C1CN(C(c2csc(C3CC3)n2)=O)C1)C C1(C(N(C(C)CNC(=O)C(F)(F)c2cnn(C)c2)C)=O)CCC(=O)C(C)C1(C)C N1(C(c2c(C(=O)OC)coc2)=O)CCCC(CO)(NC(c2ccc(SC)o2)=O)C1 CCC(CN1CCOCC1)N=c1nc(N(C)Cc2cscn2)c2c([nH]1)CCCC2 C(=O)(CCC(=O)c1ccc(F)cc1)N1C(CNC(c2cnc(Cl)s2)=O)C=CC1 N1(C(C(=O)NCCSC)C2CC2(C)C)CCOC(C#N)C1.c12ccc(cc1)[nH]c2=O c1(Cc2cnns2)cn(C2CCCc3cccnc32)nn1.N12CCC(C1)NC(=O)C2 Cc1nc2cc(C(N3CCCC(NC(=O)C(Cl)=CCl)C(F)C3)=O)ccc2s1 N1(C(CC2C(C)CN(C(C3CC4CCC4C3)=O)C2)=O)CC2CSCC2C1 C(C(C)(C1CC1)NC(=O)Cc1cscn1)NC(C1(CCOC)CC1)=O N1(C(c2nnc(C(C)(C)C)s2)=O)CCC2CN(C(=O)CC3(CO)CC3)CC2CC1 N1(C(Cc2nc(COC)sc2)=O)CCC(N(C(=O)CC(F)F)C)C(C)C1 C=C=CC(C)C(=O)NC(CC=CC)C(=O)NCC(=O)NC(C)CC.C(C)=O CCC(CC(=O)NCCC1(O)CCN(C(=O)C(CO)NC(N)=O)C1)OC C#CCC(C)(CC)C(=O)N1CCC(CNC(c2cc(C)c(C)[nH]2)=O)CC1 c1(C(N2C(C)CC(CCNC(C3CN(C)C3)=O)CC2)=O)cc2cc(Cl)cnc2[nH]1 c1(C(C(N2CC(CNC(c3n(C(C)C)cnc3)=O)C2)=O)C2CC2)ccc(Cl)cc1 C1(CNC(c2cnco2)=O)CCCCCN1C(c1ncc(Br)cc1F)=O CCC(COC)C(=O)N(C(CNC(c1cc(-c2ccccn2)no1)=O)C1CC1)C c1(CNC(=O)C(c2ccc(O)cc2)O)ccc(-c2cccc(Cl)c2)cn1 C(CC(O)C(=O)NC1CCCC(NC(=O)Cc2csc(C(=O)OC)c2)C1)OC CCC(C)C(C(=O)NCc1cc(C(=O)NC(C2CCCCC2)C)cs1)N(C)C c1(NC2CCC(NC(N3CC(C(=O)OC)C3)=O)C2)cccc(Br)c1F c1(NC(N2C(COC)(CO)CCC2)=O)ccnc2ccnn12 c1(C(C(=O)NC(CC=C)CNC(c2cccnc2N)=O)C)cc(F)cc(F)c1 c1(CCC(=O)NC(C(=O)NCCCCO)C2CCOC2)ccccc1 O=C(CC1=NNC(=O)C1)N(CCCNC(=O)C(F)C(F)(F)F)Cc1ccccc1 N1(C(C(CO)N(C)C)=O)CCN(C(=O)C=CC2CCOC2)CC(C)(C)C1 c1(OC)c(CNCc2ccc(OCCO)cc2)ccnc1F O=S(=O)(NC(CSCC1CCC=CCCC1)C(F)(F)F)N1CCOCC1 C(=O)(C1=CCCC1)N(CCCNC(c1cnc(-c2ccccc2)[nH]1)=O)C C(=O)(CCCC(=O)C1CC1)N1CC2C(CN(C(=O)CCOC3CC3)C)C2C1 CC(C)(C)C(=O)C(=O)NC1COCCC1NC(c1csc(Cl)c1)=O C1(CCc2c(C(=O)OC)cccc2)(OC)CCN(C(=O)COCC(F)F)CC1 c1(C(=O)OC)ncc[nH]c1=NNC(=O)NCC1(O)CCN(C(=O)OC(C)(C)C)C1 c1(N(CC(COC)(C)C)C)nc2ccsc2c(=NCC(C2CCC2)OC)[nH]1 N#Cc1ccc(C(N2CC3CC3(C(=O)Nc3cccc(Cl)c3O)C2)=O)cc1F C1(NC(C(N2CCCCC2)C)=O)CCC(CCC(=O)NC(CN2CCC2)CO)C1 N1(C(C(=O)NC(c2ccccn2)C2CC2)=O)CCCC(C(F)(F)F)C1 C1(C(=O)NCC=CCC(=O)N(CC(=O)NC2CC2)C)CCC(O)CN1C C1(CC)C(NC(C2CC(O)C2)=O)CCN1C(=O)CCc1ccc(C)nc1 c1(C(N(C(CNC(=O)Cc2cncc(O)c2)C2CC2)C)=O)cc2c[nH]nc2s1 c1(C(=O)NCC(CC)(CC)NC(C2COCCN2C)=O)cc(OC)ccc1OC Cc1cc(=NCC2CN3CCN2CC3)[nH]c(N2CC3CCC(C2)O3)n1 C(C)(c1ccc(OC)cc1)=CC(=O)NC(CC)CN(C)C(C1CC2CCC1O2)=O C1(C(=O)NC2C(NC(CN(C)C3CC3)=O)CC2)CCCOCC1 CCCC(C)CCCC(=O)NCC(C)N(C)C(c1cnc(OC)cn1)=O N1(C(C2CCCSC2)C(=O)N(c2ccccc2)C2(C)CC2)CCC(F)(F)C(O)C1 Cc1cc(C(=O)NCC2(O)CN(C(c3cc(F)n(C)n3)=O)C2)nn1C(C)C1CC1 CCCC(C)CC(C(=O)Nc1cccc([N+](=O)[O-])c1)N1CCC12CCCCC2 N1(C(C=CC(=O)N(CCNC(C)=O)CC)=O)CCCC(C(=O)NC2CC2)C1 c1(CC(=O)NCC(N(C)C(c2ccc(F)cc2Cl)=O)C2CC2)ccc(O)c(O)c1 C1(C(=O)NCCC(C)NC(CC(C)c2ccccc2)=O)CCC(OC(F)F)CC1 N1(C(C23CCC(OC)C2C3)=O)CC2CC1CCC2NC(=O)CCC(C)C Cc1cc(C(=O)NCC2CC(NC(C3CC(F)C(=O)N3)=O)C2(C)C)cc(F)c1 c1(OC)ccc(C(=O)N(C)CC2CCCN2C(=O)Cc2ccc(C)nc2)nc1Cl C(=O)(C1=CC2(CCOC2)C1)N1CC2(OCC(NC(c3cn(C(C)C)nc3)=O)C2)C1 C1(C(N2C(C)(C)C(NC(=O)COCC3CCCC3)CC2)=O)CC2OC(=O)OC2C1 CCCC(C)(C)CNC(c1csc(-c2nc(C)no2)c1)c1nnnn1C C1(C(N2CCC(NC(CC(CCC)O)=O)C(F)C2)=O)CCc2n[nH]c(C)c2C1 Cc1nc(N2CC(O)(C(C)NC(C3CCS(=O)(=O)N3C)=O)C2)cc(SC(C)C)n1 N1(C(C2(NC(C(C)S(C)(=O)=O)=O)CCOCC2)=O)CCCC(C2CCC2)C1 C1(CCC)CN(C(=O)CNC(=O)NCC)CC1NC(C1NC(=O)OC1C)=O c1(OC)cc(C(N2CCC(NC(c3cc(F)n[nH]3)=O)C(F)C2)=O)cnc1OC N1(CC(N2CCN(C(c3ccc(CC)s3)=O)CC2)=O)C(=O)CN(C)C1=O CC1(O)CCCN(C(C23CCC(NC(=O)C=Cc4cc[nH]c4)(CC2)C3)=O)C1 Cc1cc(C(=O)NC2(CCNC(=O)C#CC(C)C)CCCC2)ccn1 C1(C(=O)NC(C2CCCOC2)COC)CC2C=CC1C2.c12cn(nn1)C2 N1(C(c2[nH]cc(CC)c2)=O)CCN(C(C2(C(C)(F)F)CC2)=O)CC1C(C1CC1)C CC1(C)CC(n2nc(-c3cc[nH]n3)nc2-c2cc(Cl)cnn2)CCO1 C(CC1CCc2ccccc21)NC(c1cc(N2CCC(OC)CC2)ncc1)=O c1(CNC(NC(COCC)CC)=NCC2CCOC2)ccc(Cl)c(O)c1 c1(CNC2C(C(=O)NCC(=C)C)C2)c(Cl)ccc(C)c1F n1(CC)c(C(N2CCCC2CO)=O)cnc1O.c1(C2C(=O)N2)cncc(F)c1 CN1CCCC(C(C)(C)C(=O)N2CC(CN(C(=O)C(C)(C)CF)C)C2)C1 C(=O)(C(C)C(O)C(C)C)N(CC(=O)NCCN1CCCNC1=O)CCOC N1(CC)CC(CNC(=O)C(Cn2cncn2)NC(=O)Cn2ccnc2)CC1=O CC1(C)CC(F)(F)CCC1CNC(=O)Nc1nc(C2Cc3ccccc3C2)cs1 C(C)(C)(C=CC(=O)NCCOC(C)(C)CNC(=O)C(C)c1ccco1)SC C1(C)(C(N(CCCC(=O)OC)C)=O)CC(O)CN1C(=O)CCCC1CC1 C#Cc1ccc(NC(=O)CC2CCCC2NC(C2CCC(=O)N2)=O)c(C)c1 C1(C(N(CC(C)NC(c2cc(C(C)C)[nH]n2)=O)C)=O)CC12CCCCCC2 C1(C(=O)NCCCC=CC)CCOCC1NC(C1CCO1)=O C(CC(C(=O)N(CC1=CCCOC1)C)NC(=O)Cn1ccc(C)c1)=CC CC(CC(C)NC(=O)C=CCO)NC(=O)CCc1cccs1 CC1CN(C(c2cc(Br)c[nH]2)=O)CC(CCNC(=O)CC2CC(C)(C)C2)O1 CCCCN=C(NCC1=CCCCCC1)NCCOCC(C)(C)O C=CCC(CNC(c1c(C)cccc1C)=O)C(=O)NC1COCC1F c1(C(N2CC(N(C)C(C3C=CCC3)=O)C3(C2)CC3)=O)cc2ccc(F)cc2o1 C1(C(=O)NC2C=CCC(C(=O)NCc3ncsn3)C2)(CC)CNC(=O)C1 C1(CNC(C=C(CC)C)=O)COCCN1C(=O)C(C1CC1)SC C1(C(=O)NCC(CNC(=O)C=Cc2ccsc2)F)CCCC1C1CC1 c1(C2C(C(=O)NCC3CCN(C(c4ccc(COC)[nH]4)=O)C3)C2)ccccc1F C1(OC)=C(C)c2c(cc(F)cc2)C1(C)NC(=O)NCC1CC(C)(O)C1OC C1(CCNC(=O)CCc2cc[nH]n2)(OC)CN(C(c2csc(C)c2)=O)C1 C1(C(=O)NC(CCC)CO)(CC)CCN(C(=O)C(C2CC2)OC)CC1 N1(C(C(C)OC)=O)CC2CCOC2(CNC(=O)CC(C2CCC2)C2CCC2)C1 c1(CCC(=O)N(C2CC(NC(C(C(C)C)SC)=O)C2)C)cc(C)nc(C)c1 N1(C(CCCC#C)=O)CCOC2(CCC(NC(=O)C3=CC(O)CCC3)CC2)C1 C1(O)(C(=O)NC(CNC(c2cc(C(F)F)cs2)=O)C2CC2)CCSC1 c1(OC)ncc(Br)c(OC)c1C(=O)NCC1CCN(C)C(C)C1 C(=O)(CCC(C)NC(c1cccc(COC)n1)=O)N(CC(CC)(F)F)C C1(C(N2CCCC2Cc2cccnc2)=O)NCC12CC2(F)F c1(C(N(CCNC(=O)CCCSC(C)(C)C)CC)=O)cc(C)oc1C C(CC(C)C)(C(=O)NC(C1CCCN1C(c1oc(C)cc1C)=O)C)OC C1(CNC(c2c(C)n(C(C)C)nc2)=O)CN(C(=O)Cc2ccccc2)CCN1C C(=O)(C(C)C(O)C(C)C)NCC1(NC(c2cccc(C)c2Cl)=O)CCCCC1 CCC(CCCC(=O)N1CCC(C)(CCO)C1)NC(c1ccc(COC)o1)=O C=CC(C(F)(F)F)NC(c1ccc(CNC(C2CC23CC3)=O)cc1)=O Cc1cc(C)c(C(=O)NC2CCN(C(c3nc(=O)cc(N)[nH]3)=O)C(C)C2)c(C)c1 c1(C(=O)NC(C(=O)N(C)Cc2ncc(C)o2)CC2CCC2)ccn2ccccc12 C1(C(Cn2cc(C(CC)O)nn2)F)CCNCC1.C(=O)CCC(C)c1nn[nH]n1 N1(C(C2CCC(C)CC2)=O)CCCC(C2CN(C(c3ccc(N)c(Cl)n3)=O)C2)C1 C1(C(=O)NCCc2c(C)n(C)nc2)C2CCC3(COC(=O)C13)O2 C1(NC(C2(O)CC(C)(C)C2)=O)CN(C(c2cccs2)=O)CC(F)(F)C1 CC(C(F)(F)C(F)(F)F)=CC(=O)NCC1(C(=O)Nc2cnc[nH]2)CCCCC1 CCCCC(O)C(=O)NC(Cc1cccs1)CC(=O)NCc1ccc(Cl)cn1 CC1CN(C(=O)CCNS(C)(=O)=O)CC2(CCN(C(C3(C)CC(F)(F)C3)=O)C2)O1 CC(C)(C(=O)NC1C2CN(C(c3sccc3C3CC3)=O)CC12)C(F)F CCC(F)(F)C(=O)N1CCC(C(C)NC(C2CCSCC2)=O)C1 C(=O)(C(C(C)OC)NC(c1n[nH]c(C(C)CC)n1)=O)OCC C1(N(C(C(C2CCCC2)OCC)=O)C)CN(C(=O)Cc2ccccc2Cl)CC1O c1(OC)ccc(Cn2nc(-c3cnn(C)c3)nc2C(O)CCS(C)=O)cc1 CC1(C)CN(C(C2CCOC2C2CC2)=O)CCC1C(=O)NC1CCCCCCC1 CCC(C(=O)NC(Cc1ccco1)C(=O)NCC1CCOC(C)(C)C1)C(C)C S(=O)(=O)(c1ccc(NCCF)c2cnccc12)NC(C)CCC1CCCO1 C1(O)(CCNC(c2nc(CC)oc2)=O)CCCN(C(=O)CCOCC(F)F)C1 N1(C(C(C=C)c2ccccc2)=O)CC2CC1C2CNC(=O)C=CC1CCCCC1 N1(C(c2ccccc2F)=O)CCCC2(CCCN2C(=O)CNC(C2(C)C(C)C2)=O)C1 C(C)(CCC(=O)NC1CCC(NC(=O)CSC2CCCCO2)CC1)SC CCC(CC(=O)NCc1occc1C)N(C(=O)CC1CCC(C)(C)C1)C c1(NC(CC(CCSC)O)=O)ccc2cnn(CCCO)c2c1 N1(C(C(CC)Nc2ccccc2)=O)CCN(C)C(CNC(=O)CCC(C)C)C1 C1(NC(c2cc(CC)[nH]n2)=O)CCCN(C(c2conc2CC)=O)C1CC N1(C(c2ccc(N(CCC)C)nc2)=O)CC(NC(c2ccns2)=O)CC(C)C1 C(=O)(C1CCc2c[nH]nc21)N1C(CC(=O)NCCC(CC)N(C)C)COCC1 Cc1cnc(C(=O)Nc2ccc(C(F)C(F)(F)F)cn2)c(C)c1 C(=O)(C1CCc2cccc(OC)c21)N1CCCC(N(C)Cc2ccc(C#C)s2)C1 c1(CC)nc(CNC(=O)CC2CCN2C(=O)CC2CC2)n[nH]1 N1(C(C(C)N(C)C)=O)CC2CCOC2(CNC(=O)CCc2nc[nH]n2)C1 N1(C(Cc2c(C)noc2C)C(=O)NC2CCCC2)CC2CCCCC2(CO)C1 C1(NC(C(C)CC2CC2)=O)CC2CN(C(=O)Cn3ccccc3=O)CCN2C1=O C(C)(C)(C(=O)N(CCC(=O)NC1CC(CCO)C1)OC)OCCC C(=O)(CCC(=O)N(C)C)NCC(CC)N(C(Cc1c(CC)con1)=O)C N1(C(c2n[nH]c(C)c2Cl)=O)CCC2(C=C(C(=O)N3CC(OCC(N)=O)C3)C2)C1 Cc1cc(S(=O)(=O)N2CCOCC2c2ccc(Br)cc2)cc(Br)c1C N1(C(CC(=C)Br)=O)CCC(CNC(=O)Cc2c(C)ncnc2C)C(O)C1 c1(C(=O)OC)ccc2c(c1)CC(C)(C)C2NCC1COCC1C c1(C(C(=O)NCCC)N(CC(=O)OC)CC#N)cc(OC)c(Br)c(C(C)C)c1 C=C(C)C1OCCC1C(=O)N(CCC(N1CCCC1CN=[N+]=[N-])=O)C(C)C c1(NC(Cc2ccc(C)cc2)=O)cc(Cl)ccc1C#N.C12CC(C1)CC(=O)N2CCl c1(C(=O)NCCN(CC)Cc2ccn(CC(C)C)n2)cccc(-n2cnnc2)c1 Cc1sc(C(F)(F)F)nc1C(=O)NC1CCC(CCNC(c2ncn(C)n2)=O)C1 c1(CC)nc(C)c(C(=O)NC2CCCC2(C)CNC(=O)C(C)NC=O)o1 C1(NC(C(CCSC)(C)C)=O)CC2CC(C1)CN(C(C1CC3(CCO1)CC3)=O)C2 N1(C(c2cn(CCC)nn2)C(=O)NCCOC)CCOCC1C1CCCO1 c1(C(N2C(COC)(CNC(=O)C(F)(F)CC3CC3)CCC2)=O)ccc(C#N)cn1 C1(C(=O)NCC(CNC(c2cnc(C)nc2)=O)OCC)CCC(C(N)=O)CC1 Cc1cnccc1CNC(C1CCC(C2CC2)N1C(=O)CCc1cnccn1)=O C#Cc1c[nH]nc1C(=O)NCC1(CC)CCCN1C(=O)C(COC)COC C(=O)(C1Cc2c(Cl)cccc21)N1C(CO)CC(NC(C(COC)(F)F)=O)C1 c1(OC)cccc(C(=O)NC23CCC(NC(C4CNC(=O)C4)=O)(CC2)C3)c1F.CN N1(C(C(C)OCC(F)(F)F)=O)CCC(N(C(=O)C=Cc2ccsc2)CCO)C1 CCN=c1cc(-c2nc(C(c3ccn(C)n3)C)n(CC3(C)CC3)n2)cc[nH]1 Cc1c(F)cc(C(N2CCC23CN(C(=O)Cn2cc(Br)cn2)C3)=O)cc1F N1(C(C2CN(C)C(=O)N2)=O)CCCC2CN(C(=O)CCN3CCCC3)CCC12 C1(C(=O)NCCOCCC(=O)Nc2cncc(C(N)=O)c2)(COC)CCCCC1 C(=O)(CCCCN(C)C)NC(CC)CNC(=O)C(C)NC(=O)NC c1(NCC(c2ccc(Cl)cc2)C)ncc(S(=O)(=O)NC2CC(CO)C2)cc1Cl C(=O)(CCC(=O)NC1CCC(NC(=O)CCC(=O)c2ccccc2N)C1)NC C1(CC)(NC(c2cc(OC)nc(C)c2)=O)CCCN(C(C2CCC(=O)O2)=O)C1 C1(OC)(CNC(=O)C=C(C)C2CC2)CCN(C(c2nonc2C(C)C)=O)C1 C=CCCC(C(=O)NCC(C)(C)C=C)NC(=O)CCCOC N1(C(C2C(C=C)OCC2)=O)CCC(C2CN(C(=O)CC3CCC3(C)C)C2)CC1 N1(C(C2(C)CCC(O)CC2)=O)CCCCC12CC(NC(=O)CC1(O)CCOC1)C2 C1(CNC(c2ccnc(C)c2C)=O)CCCC2CN(C(C3CCCC3F)=O)CC12 C1(C)(C(=O)NCC2N(C(C(C)N(CC(F)(F)F)C)=O)CC2)CCCOC1 Cc1cc(C)n2nc(C(N3CC(CO)(NC(=O)CCCC(F)(F)F)C3)=O)cc2n1 N1(C(CCNS(CC)(=O)=O)=O)CCC2CCC(C1)N2C(c1nnc(S)n1C)=O c1(C(N2CCC(O)(C(C)C)C2)=O)ccc2ccsc2c1.C12(CC1)C(=O)N2 CCC(F)(C(=O)OC)C(=O)NCC(C)(C1CC1)NC(=O)CCCNC(C)=O C#CCC(C)(C(=O)NC1(CO)CC2(CCC2)C1)NC(=O)CCC(F)(F)F CC(C)S(=O)(=O)CC(=O)N1CCCC1CC(=O)NCCNC(=O)C(C)(C)C C1(O)(COC)CN(C(=O)CN(C(C2CN(C(C)=O)CCO2)=O)C2CC2)C1 C1(C(N(C2CCCN(C(CC3CCC(C)CC3)=O)C2)C)=O)CC(S(C)(=O)=O)C1 C1(C(=O)NC(CC#CC)C)CCOCCN1C(C1CCC(CC)CC1)=O C1(NC(C2(C#N)C(C)C2)=O)C2CCC1CN(C(C1CC(F)(CF)C1)=O)C2 c1(SCC(CC=C)NC(CNC(C=C)=O)=O)cc(Br)ccc1S(C)(=O)=O C12C=CCN1C2=O.C1(C(N(C)C)=O)CCN(C(=O)COC(C)(C)C)C1 c1(CC)cc(CC(=O)N(CCCNC(=O)C=CCCC(C)C)CC2CC2)n(C)n1 c1(C(C)=O)ccc(NC(c2conc2C(C)NC(c2cnsn2)=O)=O)cn1 N1(C(c2ncc(OC)cn2)=O)CC(NC(=O)C(C)(O)C2CCC2)CC2(CC2)C1 C1(C(C)C)N(C(=O)C(C)(F)F)CC12CCN(C(=O)CN1CC(=O)N(C)C1=O)CC2 c1(C(=O)NCC2N(C(c3n(C)nc(Br)c3)=O)CCC2)cc(N)c(F)c(F)c1Cl c1(C(=O)NCC(C(C)C)C(=O)N(C2CC(C)C2)C)cccn2nccc12 c1(C(=O)NC)cc2c3c(ccc2[nH]1)N(C(c1cnccn1)=O)CC3 c1(C(=O)NCCCN(C(C(CC)SC)=O)CC)ccc2nc(C)c(=O)n(C)c2c1 C1(CNC(c2n(CC=C)nnn2)c2cn(C(C)C)nn2)CC2(CC2)C(=O)O1 C1(NC(=O)C=CCF)C2CCN(C(=O)C(C3CCCCC3)=O)C12 C1(CC)CN(C(=O)C(C)COC)CCC1NC(=O)CCc1conc1C C1(NC(C2OCCN(CC)C2)=O)CN(C(=O)CCOCC(C)(C)C)CC1C1CC1 c1(CC(N2CCC(NC(CCC(C)(F)F)=O)C2(C)C)=O)n[nH]c2c1CCCC2 N1(C(CCc2cnc(C)s2)=O)CC(C(C)(C)C)CC(CNC(C2CCO2)=O)C1 c1(CNC(C2(C)CC(=C)C2)=O)cccc(CN(C)C(C2CC2[N+](=O)[O-])=O)c1 C(=O)(C1=CCC(C)(C)CC1)N1CCCC(CC=C)(NC(=O)CCC(N)=O)C1 c1(C(N2C3C(NC(COC)=O)CC(C3)C2)=O)cc2n(n1)CC(F)C2 C(=O)(C(=O)N=S(C)(C)=O)NC1CC(OC)CN(C(c2ccc3c(n2)NCC3)=O)C1 C1(CC(=O)NCCCOC=C)CC2(C1)CN(C(c1ccc(Cl)c(Cl)n1)=O)C2 C(CC(C(N)=O)NC(c1cc(-c2ccccc2)ncn1)=O)OC Cc1ccc(C=CC(=O)N(C2CCC(NC(C3(C)CCC3)=O)C2)C)cc1 c1(C(N2CC3CC(NC(CC(CCC)C)=O)C3C2)=O)ccc(Cl)c(F)c1F C12(CNC(CC(C)OC)=O)CCCC1N(C(=O)CCOc1cccc(F)c1)CC2 c1(CC)oc(C(=O)NCCC(C)N(C(=O)CC2CC3(CC3)CO2)C)cc1C C1(NC(C(CC2CC(F)(F)C2)SCC(=C)C)=O)CC2CC(CO)CC12 Cc1cc(=O)c(C(=O)NC2CN(C(=O)CC3CCCC3)CCC2F)cn1C1CC1 CC1C(=O)N(CC(=O)NC2(CNC(c3csc(S)n3)=O)CCOC2)C(=O)C1C CC1CCC(C)N1Cc1cn(C(NOCC2(c3ccon3)CC2)=O)nn1 Cc1cc(F)cc(C(=O)NCC2(F)CCN(C(=O)C=C3CCN(C)C3)CC2)c1N c1(CNC2C(CC=C)CCC2)cc2ccccc2s1 N1(C(=O)Nc2ccoc2C(F)(F)F)CCN(c2ncccc2Cl)CC1 c1(COC)cc(C)n(-c2ccc(NC(=O)CC(C)c3cnn(C)c3)cc2)n1 N1(CC(=O)O)CCC(O)(C(=O)NCC(c2ccc(Br)cc2)O)CC1 C(=O)(CCCCC(F)F)N1CCC(NC(C2C(C(C)C)CCC2)=O)C(O)C1 C#CCCCCC(=O)N1CCC(C(C)C(=O)NCC(CCC)CCC)C1 Cc1nc(CNC(=O)CCNC(=O)CNC(=O)C#CC(C)C)oc1C C1(CNC(C2(C(C)C)CC2)=O)C=CCN1C(=O)C(C)CO Cc1c(C(=O)NC2CN(C(c3ccncn3)=O)C(C)(C)C2)sc2ccc(F)cc12 C1(C#N)(C(N2CC(F)(CNC(CCCc3cc(C)no3)=O)C2)=O)CCCCC1 C(C(C)(C)CC(C)O)NC(C=CC(C)NC(C1CC(O)(CC#C)C1)=O)=O C1(C(=O)NC2(C(F)F)CC(NC(=O)CC3(n4cncn4)CC3)C2)CCCOCC1 C1(CNC(C2(CCC)CC2)=O)CN(C(=O)CCc2nnc(S)n2C)CCC1C C1(NC(C(CC)CN(C)C)=O)CC2CCC(C1)N2C(=O)CCN1CCCCC1 N1(C(c2ccc(SC)cc2)=O)CC2(C1)CN(C(=O)CCN1CCC(F)C1)CCO2.CN Cc1cc(C2CCCN2C(=O)C(=O)Nc2cccc(F)n2)cc(C)c1 C1(NC(CCCC(C)OC)=O)CCCC12CCN(C(=O)Cc1ncoc1C)CC2 C1(NC(CSCC(C)C)=O)CCN(C(=O)COCCCF)C(C)C1 c1(CC(=O)NC(CCNC(c2c(C)nc(C)[nH]2)=O)C)ccccc1S(C)=O N1(C(CC2C(NC(C3C(C)(C)C3C#N)=O)CCC2)=O)CC2(CCC2O)C1 C12(CC(=O)NCC(C3CC3)NC(C3CC(OC)C(OC)C3)=O)CCCN1CCC2 N1(C(CC(=O)OCC)=O)CCCC2(CNC(=O)CSCC(N)=O)CCCC12 C12(C(=O)NCC(c3ccccc3)NC(C(CC)N(C)C)=O)CCC(O)(CC1)CC2 C1(NC(CCOCC)=O)CN(C(=O)Cc2c(C)n[nH]c2C)CC1n1ccnn1 C1(c2n(-c3cccc(C)c3)nc(C3CN(C)CCO3)n2)CC2CC1CC2(F)F C1(CNC(CC(=C)C)=O)CCC2(CCC2)C1NC(c1ncccc1OC(F)F)=O C#Cc1cc(C(=O)NC2COC3(C2)CN(C(C2CCN(C)C2)=O)C3)ccc1C c1(C(=O)NC2CCCC(C(=O)NC(c3nc(=O)o[nH]3)C)C2)ccc2c[nH]nc2c1 CC(C)C(CNC(c1ccc(C#N)o1)=O)C(=O)N1Cc2c[nH]nc2C1 c1(C(=O)NC(CNC(C2=CC(C)(C)C2)=O)C2CCC2)cc(F)cc(Br)c1O C1(CCNC(C(C)CN(C)C)=O)CCN(C(C2(C(F)(F)F)CNC(=O)C2)=O)CC1 c1(NC(C(C2CC(C(N(C)C)=O)C2)F)=O)cc(F)ccc1O c1(C(N2C(CNC(C3C(CC)CCO3)=O)CC(C)(C)C2)=O)nccn2nccc12 Cc1cc(C)c(C(N2CC(C(C)NC(c3ncccc3C)=O)C2)=O)o1 C(=O)(CC(C)(C)O)N1C(CNC(C2C(C)CCC2)=O)CC1 c1(NCC2(c3cccc(F)c3)C(C)(C)C2)ccc(S(=O)(=O)N2CC(OC)C2)cc1Cl C1(O)(CN(C(c2c(C)nsc2)=O)C)CCN(C(c2ccc(C(C)C)cn2)=O)C1 c1(NC(N2CC(CO)C3(CCC3)C2)=O)cc(Br)c2c(c1)OCCO2 CC1CC2CN(C(=O)CCC(F)(F)Cn3cc(-c4cc[nH]n4)nn3)CCN2C1 c1(C(=O)NCCC2CCCCN2C(c2cccs2)=O)cc(Br)ccc1O C1(C(N2CCC(N(C)C(c3nnc(C)s3)=O)C2)=O)(COCCOC)CCCCC1 N1(C(C(CC)F)=O)CC(NC(=O)CC2(OCc3ccccc3)CC2)C(C)C1 N1(C(c2n[nH]c(C)c2C)=O)CC(C)(C)OCC1CNC(C1(S(C)(=O)=O)CCC1)=O C1(CCOC)(NC(=O)CC2CCCC(C)C2)CCN(C(c2nn(C)cc2C)=O)C1 C(c1ncco1)=CC(N1CC(NC(C2(C(C)(F)F)CCC2)=O)C1)=O C1(N(C(C2CCN(C)C2=O)=O)C)CCCN(C(c2cncn2C)=O)CC1 CC(CN(C)C(C1(C)CCC(=O)NC1)=O)C(=O)NOCCCC1CC1 N1(C(C=CC(C)C)=O)CCC(C(N2CCC(O)C(C)C2)=O)C(F)C1 Cc1ccnc(O)c1CN1CCC1NC(=O)C(O)C(C)c1ccccc1F Cc1cc(C)c(C(=O)NCC2CC2CNC(c2cccc(C)c2N)=O)c(C)n1 CC(N=[N+]=[N-])C(=O)NC(Cn1cccn1)C(=O)N(CCCCO)C C(C)(C(=O)NC1CC(CNC(=O)CNC(=O)CCSC(F)(F)F)C1)SCC N1(C(C(=O)Nc2ccn(C(F)F)n2)=O)CCCC(c2nnc(Br)o2)C1 c1(CC)ccc(C(=O)NCC(C(C)C)NC(=O)C(C)CCSC)cc1.N(CC)(CC)C Cc1cc(-c2ccc(CNCCCn3ccnc3)cc2F)ccc1CC(=O)OC c1(NC(C)=O)cc(C(=O)NCC2CCCC(NC(c3cocn3)=O)C2)ccn1 c1(N2CCC(=C(C)C)C2)nc(=NC(C)c2cnn(C(C)C)c2)[nH]c2c1SCC2 c1(NC(C2(C(F)(F)F)CCCNCC2)=O)cccn2nnnc12 C1(C)(CNC(CC2C(CC)C2)=O)CCCN(C(=O)C(Cl)=CCl)C1 C(CC)(CCC(=O)NC(C)CCSC)NC(c1c(CC)non1)=O CP(C)(=O)CN1CCCC(NC(=O)NC(Cc2ccccc2)C(O)C(F)(F)F)C1 CC1(C2CN(C(C3C=CC(NC(c4ccc(C#N)cn4)=O)C3)=O)C2)CC1 S(=O)(=O)(c1cnccc1N(CC(c1ccc(C)s1)O)C)NCc1ncc(CC)s1 C(CCCCC(=O)N1CCOCC1CNC(=O)CCC1CCCN1C)OC CCC(C)C(=O)C(=O)N(CC(C)C(=O)N1CCC(OCCF)C1)C [N-]=[N+]=NC1(C(N2CCCC2(C)C2CC2)=O)CCN(C(=O)C#CC2CCC2)C1 CC1CC=C(C(=O)NC2(C3CC3)CCN(C(C3CC(C)(O)C3)=O)C2)CC1 C(CCNC(c1ccoc1Cl)=O)(C(C)C)NC(CC=CCC)=O S(=O)(=O)(c1cccc(C(=O)NCCC(F)(F)C(=O)O)c1)NC(CCC#C)C c1(OC)cc(C(=O)N(C)CC2CCCC2NC(C23CSCC2C3)=O)ccn1 Cc1ccc(C=CCN2CCC(C(C(=O)Nc3ccn(C4CC4)n3)C)C2)cc1 c1(C(N(C(CC)CNC(=O)C(C)C2CCCO2)C)=O)ccn(C)c1C c1(C(=O)NCC(CN(C)C(C2CC2c2ccco2)=O)(C)C)cn(C)[nH]c1=N C1(C(=O)NCC23CC(CNC(C4C(C)(C)C4)=O)(OC2)C3)CCc2nccn2CC1 N1(C(CC2CCN(C(c3c(C)csc3)=O)C2)=O)CCC2(CC1)CCN(C)CC2 C1(NC(C2(C(=O)OCC)CCC2)=O)CC=CCC1C(=O)NCc1cn(C)nc1C O=C1CCCN1C1CCN(CCC(N2CCNCC2)=O)C1 c1(CC(N2CCCC(O)(CCNC(C3C(C)C3)=O)C2)=O)ccc2[nH]ccc2c1 C1(CCNC(c2c(CC)nn[nH]2)=O)CSCCN1C(=O)C(F)CC1CCCC1 c1(CC)conc1CC(=O)N(CC(C)O)CCNC(=O)Cc1nonc1C N1(C(c2ccc(N(C)C)cc2)=O)CC2OCCN(C(c3ccns3)=O)C2C1 c1(C(=O)NC2CN(C(c3ccnc(O)c3)=O)CC2F)ccnc2c1CCO2 c1(C(=O)NCC(CC=C)NC(=O)Cc2nnc(C)o2)cncc(S(C)(=O)=O)c1 N1(C(CN2CCC(C)CC2)=O)CCC(C2CCN(C(C34CC(C)(CO3)C4)=O)C2)C1 CC1(CC(=O)NCCN(C(C2SCCS2)=O)Cc2ccc(F)cc2)CCS(=O)(=O)N1 Cc1nc(C(N2CCN(C3CCN(C(c4cnc(S)nc4)=O)C3)CC2)=O)cn1C C1(N(C(C(=O)N(CCC)C(C)C)C)CC)CCCN(C2CCC2)CC1 c1(C(=O)NCC(=C)CCNC(=O)C(C2CC2)OCC)cnc(OCC(F)F)cn1 c1(CC)c(C(N2CCCC(NC(=O)C=Cc3ccccn3)C2)=O)cccc1F C(=O)(CCC=CBr)NC1C(CNC(CC(=O)OCC)=O)C1 C1(C(=O)NCC2N(C(CC(=O)N(C)C)=O)CC=C2)C2CCC(CC2)C1C(F)(F)F N1(C(C=CCOC)=O)CC2CCCC(NC(=O)CC3(CO)CCC3)C2C1 c1(OC)cccc(Cl)c1C(N1CCC(CNC(c2cc(N)ccc2SC)=O)C1)=O N1(Cc2cn(C(C)C)nc2)CCC2(NC(c3ccoc3)=O)CCCC12 C1(CNC(=O)CSc2cccc[n+]2[O-])CC2CCC1N(C(c1cc[nH]n1)=O)C2 N1(C(c2c(NC)nccc2)=O)C(C)C2CC1C2NC(C1(NC(C)C)CC1)=O O=C(C1=CCCCC1)NCC1C2CC1N(C(c1ccc(F)c(Br)c1)=O)C2 C12(CNc3cc(C)nc(C)n3)CCCC1CCN2C(=O)COC1CC(F)(F)C1 c1(CNC(C2(CNC(=O)CCc3ccoc3)CCOCC2)=O)ccc(F)cc1O c1(C(N2CC(NC(C3(SC)CC3)=O)C3C(C2)C3)=O)c(C)cc([N+](=O)[O-])cc1C C(C(C(=O)N1CCC(C)(CNC(C23CCC(CC2F)C3)=O)C1)C(F)(F)F)OC C(=O)(C(CNC(c1ccc(O)cc1F)=O)C(C)(C)C)NC(C=C)CO C12(C(=O)NCC3CN(C(c4ccc(Cl)o4)=O)CC3O)C3C4C1C1C2C3C41CO N1(C(C2C(C)CCO2)=O)CCCC2(CCC2NC(c2cc(C3(C)CC3)on2)=O)C1 c1(C(=O)NC(C(=O)NCC)C2CC2)cc(C(=O)OC)cc(Br)c1 CC1(C)CC(C(=O)NC2CCC(NC(=O)CCc3cc[nH]n3)CC2)C1C(F)(F)F c1(C(N2CCC(C)C2CNC(c2ccnnc2Cl)=O)=O)ccc(F)cc1N N1(C(C=C(C)C(C)C)=O)CCCC(C2CC2NC(=O)C(c2cncn2C)O)C1 CC1=C(C(=O)N2CCC(C)(C)C2CNC(c2cccc(C(C)C)c2)=O)CCCO1 c1(C(N2CC3C(CNC(C(C)NC(N)=O)=O)(C3)C2)=O)csc2cncn12 c1(C(=O)NCC(C(N2CC(CC)OCC2)=O)O)cnn2c1OCC2 N1(C(C2(C)CC2(F)F)=O)CC2(CCN2C(C2(F)CC=CCC2)=O)C1 N1(C(COCCCC#C)=O)CC2CC(C(=O)NC(CCF)C(=O)OC)C(C2)C1 N1(C(CSCCC#N)=O)CC2CC(NC(c3cc(C(N)=O)cs3)=O)CC2C1 N1(C(C2CCN2C(c2ccc(C3CC3)cn2)C2CC2)=O)CC(O)C2(CCCC2)C1 Cc1cc(C)c(C=CC(=O)NC23CC(NC(C4CCS(=O)(=O)N4)=O)(C2)C3)c(C)c1 c1(C(=O)NC2CN(C(CCCOCC)=O)C(C)C2)cnc2cc(C)ccn2c1=O N1(C(C=C2CCC(C)C2)=O)CC2C(N(C(=O)COC(F)F)C)C2C1 C(=O)(CS(=O)c1cccc2occc12)NC(C#C)C C=CCCC(C)(C)C(=O)NC(CNC(=O)CCCC(C)(F)F)CC=C N1(C(c2cnc(COC)s2)=O)CCC(C)C(CNC(c2cnn(C(C)C)n2)=O)C1 C(C)(CNC(c1cn(C2CCC2O)nn1)=O)(C(C)C)NC(Cc1cnc(C)[nH]1)=O C#Cc1cnc(C(N2CCN(C)CC2C(=O)Nc2cc(C)cc(Cl)c2)=O)c(C)c1 CCCCC#CC(C)(C)NC(c1ccc(C2CCCN2)[nH]1)=O C1(C(N(C2C3CN(C(C4(CC5CC5)CCC4)=O)CC23)C)=O)CC12CCOC2 c1(OC)ccn2ncc(C(N3CC(O)(CNC(=O)CC4C=CCCC4)C3)=O)c2c1 c1(NCC2N(c3c(C)cnc(C(=O)OC)n3)CC(F)(F)C2)cc(Cl)cc(Cl)c1Br CCCCC(F)(F)C(=O)N1CCC(C(=O)NNCP(C)(C)=O)O1 c1(C(N2CC3C(CCNC(CC#N)=O)(CC3)C2)=O)cc2cc(Cl)ccc2o1 N1(CC(=O)NC2CCC(CNC(=O)CSC(F)(F)F)C2)CCOCC1=O C1(=CCNC(CCc2scc(C)n2)=O)CCN(C(=O)Cc2occc2C)CC1 C1(C(=O)NCC2CC(NC(CNC(=O)OCC=C)=O)C2)CCC(F)(F)C1 c1(CC(C(=O)NCCC2CN(C(COCC#C)=O)C2)O)ccc(C(F)(F)F)cc1 c1(NC(C2N(C(C3CN(CCOC)C(=O)C3)=O)CCSC2)=O)cc(C)cc(C)c1 c1(C(=O)NCC2CC(NC(C3C(OC)CCC3)=O)C2)ccc(Cl)c(O)c1 C(=O)(CS(=O)(=O)CCO)N(C1CCN(C(c2cnc3ccsc3c2)=O)C1)C N1(C(C=C(C)Cl)=O)CC(CNC(=O)C(C)Cc2ccc(Cl)c(Cl)c2)C2(CC2)C1 c1(C(=O)NCC2(O)CN(C(CN(C(C(C)C)=O)C)=O)C2)ccc(C(C)(C)C)cc1 c12cc(F)ccc1NC1CCN(C1)C2=O.C(CC)(CC)OCC(=O)NC C(=O)(Nn1cccn1)C1CN(C(CC(CC)OC)=O)CC1F C1(CNC(=O)CCCF)CC2(CC2)CN1C(=O)CCC1CCCO1 c12ccccc1C(OC)c1cn-2nn1.C1(C(COC)C2CCC2)CCCCCC1 N1(C(C2CCCC(C)CC2)=O)CC2CCC1CN2C(C1CC(OC(F)(F)F)C1)=O C(=O)(CC(C)CC(C)C)NC1C(OC)CN(C(c2cnc(C(C)C)nc2)=O)C1 c1(C(=O)NCC(CO)NC(CNS(CCC)(=O)=O)=O)cncc(C(C)C)c1 N1(C(c2ccc(C)cn2)C(=O)Nc2ccccc2)CCOC(C2CC2)CC1 N1(C(N(C2(C#N)COC2)C)=O)CCN(CC(c2ccc(F)cc2)C2CC2)CC1 N1(C(CC2CC(=O)OC2)=O)CCCC(CC(=O)NCC2CCC(=O)O2)C1 CCCS(=O)(=O)CC(=O)NCC1CCN(C(C2(CF)CC(=O)C2)=O)C1 c1(CNC(C(CC)NC(=O)C(C)NC(N)=O)=O)ccc(Br)cn1 c1(-n2c(C(C)(C)OCCC(C)C)nc(C(C)C)n2)cc(Cl)nc(Cl)c1 N12CCCOC(C1)CNC(=O)C1(CC1(F)F)CCNC(OC)C2=O.CCOC Cc1[nH]nc(C(=O)NC(C)C(=O)NCc2ncc(CO)o2)c1C c1(C(N(CC(CNC(C2(NC(C)=O)CCCC2)=O)(C)C)C)=O)cccc(C#N)c1 c1(C(C)NC(=O)OC(C)(C)C)ccc(OCCC(N2CC(F)(CSC)C2)=O)nc1 C(=O)(C(F)(F)C(C)(C)O)NC1C(CC)CN(C(=O)CN(C)C(=O)C2CC2)CC1 C(=O)(C(C)(C)C(C)NC(=O)COCCCF)N1CCCC(OC(C)C)C1 c1(CC)cc(C(N2CC3C(N(C)C(C4OCCOC4C)=O)C3C2)=O)cc(C)c1 Cc1ccc2c(c1)CC(C(=O)NCC(C1CC1)NC(c1sccc1C(F)F)=O)S2 C12(NC(C3N(C(c4cccc(CC#N)c4)=O)CC3)=O)CCCC1OCC2 Cc1conc1CC(=O)NC1CC(C)(NC(c2cc(C3CC3)no2)=O)C1 C1(C)(C(=O)NC2CCC(N(C)C(c3ccnc(OC(F)F)c3)=O)C2)CCCCCC1 N1(CC(=O)NCC#N)C(CNC(c2cn(CCC3CC3)nn2)=O)CC2COCC12 C12(C(=O)NC(c3ncc[nH]3)CC)CCC(CN(C(=O)C(C(C)C)SC)C1)C2 CC(=O)CCCCC(=O)NCC=CC(N1CCC(O)C1(C)C)=O N1(C(Cc2cc(C)n(C)n2)=O)C2CCC1CN(C(C1CCN(C3CC3)CC1)=O)C2 C(C(=O)NC1CC(CC(=O)O)C1)(C(C)(C)C)n1cc(-c2n(C)cnc2)nn1 c1(NC(C(Cc2cc[nH]n2)NC(C2CCCOC2)=O)=O)cccc(C2CC2)c1 C=CC1(CC(=O)NC2CC(N(C)C(c3cnccc3C)=O)C2)CCCCC1 N1(C(CS(CC)(=O)=O)=O)CC2CCC1C(C(=O)Nc1c(C(N)=O)cccc1F)C2 N#CC1(F)CCN(C(c2cnc(C3CCCO3)s2)C(=O)NC2CC2)C1 CCC(CCCC(=O)N1CC2CC(C1)N(C)C2)NC(=O)C(F)n1ccnc1 C1(CNC(COC(C)C)=O)CC2(CCN(C(=O)CC3CCC4CC4C3)C2)CO1 c1(C(N2C3CCN(C(c4c(C)coc4)=O)C(C3)C2)=O)ccnc2c(F)cccc12 c1(C(N2CCC(NC(=O)NCc3n[nH]c(C)c3C)CC2)=O)[nH]nc2ncccc12 C(=O)(CCCCN=[N+]=[N-])N1CC(C(=O)NC2CN(C)C(C)(C)C2)OCC1 C1(C(=O)NCCNC(C=CC(c2ccc(C(C)C)cc2)C)=O)CC(S(C)(=O)=O)C1 N1(C(CC2N(C)CCOC2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)CC(CO)C1 c1(C(N2CCC(CCNC(C(C3CC3)OCC)=O)CC2)=O)cncc2[nH]ccc12 CCCCCCCC(=O)N1CC(C(=O)NCC(C2CCC2)OC)C(C)(C)C1 Cc1[nH]nc2ncc(C(N3CCOC(CNC(C4CC(N(C)C)C4)=O)C3)=O)cc12 Cc1[nH]nc(NS(C)(=O)=O)c1-c1nc(-c2cccc(OC(F)F)c2)no1 c1(CN(CC#C)C(=O)NC(Cc2ccccc2)C(=O)O)sccc1Br C=CCN=c1[nH]c(C(N2CC3(C2)SCCC3NC(=O)C(F)C(F)(F)F)=O)cs1 CCCCCC(=O)NCC1CC(NC(=O)C(C)CC=Cc2ccccc2)CC1O c1(C(=O)NCC2(CN(C(=O)CCCCC3CC3)C)CC2)cc(C#N)no1 c1(C(=O)NCC2CN(C(c3ccc(OCC)cc3)=O)CC2C)cccn(C)c1=O C(CCC(C)C)(C(=O)NC(C)CC1(O)CCC1)NC(C1CC(CC)C1)=O C(CCCCNC(c1coc(Br)c1)=O)NC(CN(C)C1CC1)=O c1(OC)cc(C(=O)NC2CCC2CNC(=O)C(C)Sc2ccccn2)on1 N1(C(c2cn(CCC)nn2)C(=O)NC2CC2)CCc2ccccc2C1CC N1(C(CCC#CC)=O)CC(C)(C)OC2(C1)CN(C(=O)CCc1cnco1)C2 Cc1cnccc1C(=O)NC1CCC(CNC(=O)CC2CCC3CC23)CC1 N(C(=NCCCCl)NC1CCN(CC2CC2)CC1)C(C)COC1CCOC1 c1(C(N(C(=O)CN(C2CCCC(C)C2)C)CC)=O)cc(Br)ccc1[N+](=O)[O-] C1(CNC(CN(C(c2cc(C#N)cs2)=O)CC)=O)COCC(=O)N1C N1(c2n(CCCOC)c(-c3cccs3)nn2)CCN(C2CCOCC2)C(=O)C1 N1(C(c2c(C(C)C)onc2)=O)CCC2CCN(C(c3cc(C(N)=O)c[nH]3)=O)C2C1 N1(C(CC2CN(C(c3c(NC)cccc3)=O)C(C)C2)=O)CCc2nc(O)[nH]c2C1 N1(C(c2ccc(CCC)[nH]2)=O)CCCC(O)(CNC(=O)Cc2cn(C)nc2C)C1 c1(C(N2C(CNC(CCCC#C)=O)CC(O)C2)=O)cc(C(F)(F)F)cc(F)c1 c1(C(=O)NC2CN(C(C3C=CCC3)=O)CCC2CO)ccc2cccc(O)c2c1 C1(NC(Cn2cc(C)c(C(F)(F)F)n2)=O)CN(C(C2CSCN2C)=O)CCC1C C(=O)(CC1=CSC2=NCCN12)NC1C(C)CCN(C(=O)C(C2CCCCC2)O)C1 Cc1cnc2n1CC(C(=O)OC(C)(C)C)CC2.N12CC(C(F)(F)C1)NC2=O CC(C)C(C(=O)NCC1(C(N)=O)CN(C(C2CC(C)CO2)=O)C1)NC(N)=O Cc1cc2n[nH]c(C)c2cc1CNC(c1cc(C)n(C(C)(C)C)n1)=O c1(CC)ccc(O)c(C(=O)NCC(O)CN(C)C(C2CCC(=O)N2)=O)c1 c1(C(=O)NCCCN(C(=O)COc2ccc(Cl)cc2)C)cccc2nc(O)oc12 C1(OC)CC(CNC(=O)Cc2csc(SC)n2)N(C(=O)C(C)OCC(F)(F)F)C1 c1(C(=O)NCC2CCN2C(c2cc3cc[nH]c3cn2)=O)nncc2ccccc12 c1(C(=O)NC2C(NC(Cc3c(C)nc[nH]3)=O)CCOC2)ccc(P(C)(C)=O)s1 c1(C(=O)NC23COC(CNC(C4CCCSC4)=O)(C2)C3)cc(F)c(F)cc1F N#Cc1ccncc1C(=O)NC(C(=O)NOCC1CCOC1)C1CCCC1 C1(C(=O)NCC(CNC(C2(O)CCC(C)CC2)=O)(C)O)CC2(C1)CS(=O)(=O)C2 C1(C(=O)NCc2ccc(COC)cc2)(NC(c2c(CC)nn[nH]2)=O)CCSCC1 c1(SC(C(=O)NCC(C2CCC(C)CC2)(C)O)C)ccc(C#N)cc1 C(=O)(C(F)C(F)(F)F)Nc1cccc(C(=O)NCC2CCC(OC(F)(F)F)C2)c1F C1(C(=O)N(CC(C)(C)CNC(C2CCOC2C)=O)C)(OC)CCS(=O)(=O)C1 C1(C(=O)NCC(=C)Cl)CC2CC1CN(C(c1ccc(COCC)cc1)=O)C2 c1(OC)ccc(CN2CCC3(CC3C(=O)Nc3c[nH]nc3Cl)C2)c(OC(C)C)c1 CC1C(C)SCCN1c1cc(NCC(=O)N(C)C2CC2)nc(C(=O)O)n1 C(=O)(C(CC(C)C)ONC(c1c[nH]c(C#N)c1C)=O)NC(COC)C C12(CC(=O)NC3CCCC34CC4)CCC1CN(C(C1CC1Cl)=O)C2 c1(C(N(C)CC2CCCN2C(=O)C=CCO)=O)ccc2cc(Cl)ccc2c1 C1(N(C)C(C2(C)CC3(CCC3)C2)=O)CN(C(=O)C(N)=O)CC12CC2 C(CC(C)C)(C(N)=O)NC(C1(CC=C)CCN(C(=O)Cc2occc2C)C1)=O C=CC(C)(O)C(=O)NN(C(=O)CCOC(C)C)C.C12CCC(CC1)CC2 O=C(C(O)CC(F)(F)F)NCc1cc[nH]c1C(=O)NCC1Cc2nccn2C1 C(=O)(C1CCC(=O)c2cccn21)NC1CCCN(C(c2c(C)scc2)=O)C1 C(C)(CNC(=O)CCc1ccn(C)n1)(CNC(=O)C(=Cc1cocn1)C)OC N1(C(C2(C)C=CCC2)=O)C(C(=O)Nc2cncc(C#N)c2)C2CC(O)C1C2 C(CC(C)(C)O)NC(CCN(C(c1cnn(C)c1)=O)CC)=O C(=O)(CC(O)CC(C)(C)C)NC(CNC(c1cn(CC=C)nn1)=O)(CC)CC c1(CC)cc(C(N2CCCC2CC(=O)NCC2(O)CN(C)C2)=O)c(C)o1 N1(C(C(C)OCCCC)=O)CCN(C(=O)CCc2nc(O)n[nH]2)CC1CCOC c1(C(=O)NC2CC(CNC(C3(F)CCCC3)=O)C2)n[nH]c2ccc(F)cc12 C1(SC)CN(C(C2CCC(=O)NC2)=O)CC1NC(=O)C=Cc1ccccc1 c1(Nc2ccn(C(C)C)n2)ncccc1S(=O)(=O)N1CC(C)N(CCO)C(C)C1 N1(C(CCC(=O)OC)=O)CCCC2(C1)CN(Cc1cccc(F)c1Cl)CCO2 C1(C)(CC)CC(NC(=O)CSCC(C)C)CN1C(c1cnsc1C)=O O=C(CCCCCn1cnnn1)NC1CC(NC(c2ccc(Br)s2)=O)C1 c1(OC)cc(C(=O)NCCN(CC(C)O)C(C2CC=CCC2)=O)c(N)c(C)c1 n1(CC)nc(C(=O)NC2C3CC2N(C(=O)CC2CC(C(C)(C)C)C2)C3)ccc1=O c1(C(=O)NCCC(C)NC(c2cc(C3CCCC3)n(C)n2)=O)cn2c(n1)CCC2 C(=O)(CC(C)C(F)(F)F)NC1CCN(C(C)C)C1.C12CCC(CC1)N(CC)C2=O CCC(COC)C(=O)NCC1(CNC(c2nc(C)sc2C)=O)CC12CCC2 C1(CC(=O)NC(CC(=O)NCc2n(CCC)ncn2)C2CC2)CCCN(C)C1 N1(C(CNC(C)=O)=O)CC2COCC2(C(=O)NCC2C(CO)C2(C)C)C1 c1(C(=O)NCCCC(=O)NCC2NC(=O)NC2=O)ccc2[nH]ccc2c1 c1(OC)cncc(C=CC(=O)NCCN(C(C2CNC(=O)CC2(C)C)=O)CC)c1 C1(CC(=O)N(CCNC(C(C)OC)=O)C2CC2)CCCNC(=O)C1 Cc1cc(C(=O)NC(C)(CNC(=O)C(C2CCOCC2)C)CO)c(C)cn1 c1(C(N2C(CCCNC(C3C(CC)C3)=O)CCC2)=O)cnc(O)c2ncccc12 c1(-c2nc(C)nn2C(c2ccc(F)c(F)c2)c2ccccc2)scc2c1OCCO2 c1(C(C(=O)NC(C2CN(C(C(C#C)(C)C)=O)C2)C)C)ccc2ccccc2c1 C1(NC(c2ccc3ccnn3c2)=O)CCC2(CC1)CN(c1ncncc1Cl)C2 N(C1c2ccccc2OCC1O)C(=O)NC(c1nccn1C)CC C(=O)(CCCC(N)=O)NCC(CO)NC(c1ccc(CSC)cc1)=O N1(C(C)CNC(=O)C2=NOCC2)CCN(C(=O)C(F)=CCCF)CC1 C1(CNC(C2CC2F)=O)CCC2(CC1)CCN(C(c1c[nH]cc(Cl)c1=O)=O)CC2 N1(C(C(C)C2CCOC2)=O)CCOC2(CCN(C(c3cc(O)cc(O)n3)=O)C2)C1 Cc1cc(=NC(=O)C(=O)N2CC(NC(=O)C(C)CC(F)F)C(C3CC3)C2)[nH]o1 N1(C(c2c(C)cc(C)c(N)c2)=O)CCC2(CCCCC2CN)C1 C#CCC(CC(F)F)C(=O)N1CC(C(N2CCC(O)(CC)C2)=O)C2(CC2)C1 C=C(C)CC(C)C(=O)NCC(C)(C)CN(C)C(c1ccc(O)cc1F)=O CC(C(=O)N1CCC(C(=O)NC2CCCCC2N=[N+]=[N-])O1)c1ccn(C)n1 c1(C(N2CC(NC(CN3CC(C)C3)=O)C2)=O)cnc2c(F)ccc(F)c2c1 C1(CNC(C2C(C)CCS2)=O)CCC2(CC1)CC(NC(c1cc(O)n(C)n1)=O)C2 c1(CNC2C(Nc3nc(C)nc(N(C)C)c3)CCCC2)cc(C)c2ccccc2n1 c1(C(=O)NC(C(C)NC(=O)CN(C2CCSC2)C)(C)C)nccc(Cl)c1O Cn1cc(OCC(=O)NC2CCC(NC(=O)Cc3c[nH]nc3O)C2)cn1 Cc1nc(-c2cnn(Cc3ccccc3)c2)ccc1NC(c1cncnc1C)=O C1(C)(N(C)C)CCN(C(=O)CC2C(NC(=O)COC3CCOC3)C2)CC1 CC1(C)Cc2cc(C(=O)NC3CC(F)(CNC(=O)C=CC(F)(F)F)C3)sc2C1 c1(CC(=O)NC2CN(C(CC3CCC(C)C3)=O)C2)ccc(C(F)(F)F)nc1 N1(C(c2nc[nH]n2)=O)CCCCC1C(N1CCC(OCC2CC2)CC1)=O c1(C(=O)NC(C)(C)CCNC(=O)CC2CCCO2)ccc(Cl)c(C#N)c1 CC1c2cc(F)cc(Cl)c2CCN1N1CCCC(n2cccn2)C1 C12(CC)CC1CN(C(C1C(O)CCN1C(=O)C(C)OCC(C)C)=O)C2 C1(N(C)C(c2ccc(O)cc2)=O)C2CN(C(=O)CCn3ccnn3)CC12 c1(OC)nc(C)ncc1C(=O)NC1(C2CN(C(C3COC(C)C3)=O)C2)CC1 CC(C)C(O)CC(=O)N1CC2CC(C(N3CCCC3CO)=O)(C2)C1 N1(C(CN(C(C)=O)C)=O)CC(O)CC1CNC(=O)CC1NC(=O)NC1=O CCCC(C)(C)CC(=O)NCC1CCC2(CN(C(=O)CC3C=CCCC3)C2)O1 N1(C(C(CC)OCC)=O)CC(CNC(c2cc3occc3n2C)=O)CC12CCC2 CC(C)C(O)CCN=c1[nH]c(=NC(C)c2ccsc2)c2[nH]ccc2[nH]1 CCC(C)(CCNC(=O)OC(C)(C)C)NC(=O)NC(c1ccsc1Cl)=O C1(C(C(N2CCC(CCNC(C=CS(C)=O)=O)CC2)=O)O)CCCCCCC1 C(=O)(C1=CCCCC1C)N(C)CC1N(C(c2cnc(CC(C)C)[nH]2)=O)CCC1 c1(CC(=O)NC(CC)CN(C(=O)C(C)S(N)(=O)=O)CC)ccc2nn[nH]c2c1 n1(CCCC)cc(C(=O)NC2CCC(NC(=O)C(O)c3cscn3)CC2)c(C)n1 C(=O)(CC(C)CNC(=O)C(Cc1cc[nH]n1)NC(=O)CC1CSC1)NC c1(CN2CCCC(NC(c3ccn(C)n3)=O)(CO)C2)cccc2cccnc12 CC1(C(=O)NC2(C3CCCN3C(c3cncc(CO)c3)=O)CC2)CC=CCC1 N1(C(C=CC=CCC)=O)CC(C)(NC(=O)CC2CCCN2C(C)=O)C1 N1(C(c2ccc(C(N)=O)s2)=O)CCC2CN(C(c3cc4cscc4s3)=O)C2C1 C1(C)(C(=O)NCC(C(C)(C)C)NC(C(N2CCCC(O)C2)C)=O)CC2CCC1C2 N1(C(c2cc(C)n(C)c2)=O)CC(C)N(C(c2nnn(C(C)C)c2C)=O)CC1C Cn1ncc(Cl)c1C(N1CCCC1c1ccccc1Br)C(=O)NC1CC1 C=C1CC(C)(C(=O)NC2CC(NC(=O)CC(C)SC)C2)C1 c1(C(N2CC(O)(c3cc[nH]n3)C2)=O)ccccc1OC1CC1 N1(C(c2c(C)nns2)=O)CCN(C(=O)Cc2ccco2)CC1CC(C)(C)C CC1CCOC(C(=O)NC2CC(NC(c3cnn(CC4CCCCO4)c3)=O)C2)C1 C(=O)(C(CCSC)NC(=O)CC1CCCC1)N.CCC(CN1CCCC1)OC c1(-c2ccc(C(N3CCC(F)(C(N)=O)CC3)=O)nn2)ccc2occc2c1 C1(C(=O)NCC2(OCC)CC2)N(C(=O)C(O)CC(C)C)CC12CCCC2 c1(NCCC(=O)NC2(CN(C(=O)Cc3cc[nH]c3)C)CC2)ccccn1 N1(C(c2cnco2)=O)CCC2(CCCN2S(=O)(=O)CCC(F)(F)F)CC1 Cn1ncc2c(O)cc(C(N3C4CCC3CN(C(=O)Cc3csnn3)C4)=O)cc12 C1(F)(C(N(CCOc2cccc(C)c2)C)=O)CCCN(C(=O)CN2CCCC2)C1 C1(C(=O)NC2CC(CNC(=O)Cc3cncnc3)C2)CC2CCCC(C1)C2(F)F c1(C(N2CC(O)(CCNC(c3c[nH]nc3Br)=O)C2)=O)ccc2nc[nH]c2c1 C(=O)(CCCCCn1cc(Cc2ccc(F)cc2)nn1)N(C(C(=O)OC)C)C C1(CNC(CSCCOC)=O)CN(C(c2cnc(C)nc2O)=O)CC12CC2 c1(OC)cc2[nH]c(C(N3CCC(C(=O)O)C3)=O)cc2c(OC)c1Cl C(=O)(CC(C(C)C)OCC)NC(CC=C)CNC(C1CC(=O)N(CC(C)C)C1)=O C1(NC(=O)CCF)CCCC(NC(=O)CCn2cc[nH]c(=O)c2=O)CC1 N(C1CCSc2ccc(Cl)cc21)CCCC(C(=O)OC)(C)C C1(O)(CNC(C(CC)C)=O)CC2CCC(C1)N2C(=O)C(C)(C)CN(C)C n1(CC)cc(Cl)c(C(=O)NC2CC(O)(CNC(=O)C(C)CSC)C2)n1 C1(NC(c2nn(C)c(C3CC3)c2)=O)CCN(C(C2(CCF)CC2)=O)CC1CO C1(NC(c2c(CCC)nns2)=O)CC(O)CN(C(c2onc(C)c2C)=O)C1 c1(CC)ccccc1OCC(=O)NC(C)(CC)CCNC(=O)CCCF C1(C(N(C)CC2(O)CN(C(C(C)OC3CCCCC3)=O)C2)=O)Cc2nccn2C1 c1(OC)c(CO)n[nH]c1C(c1noc(-c2ccccc2)n1)C c1(CC(=O)NCC23CC2CN(C(C2CCC4(CCC4)O2)=O)C3)ncc(F)cc1F N1(C(c2cnn(CC)n2)=O)CCC(C2CC(NC(=O)CCCNC(C)=O)C2)C1 C(N=c1[nH]c2c(c(=NCc3nnc(C(F)F)o3)[nH]1)COCC2)C1CCCC(O)C1 C1(C(=O)OC(C)(C)C)CC(C)N1OC.C(=O)(CN1CC(=O)NCC2C(C2)C1)OC C1(NC(c2c(CC)occ2)=O)CN(C(=O)Cc2ncn(C)c2C)CC1F N1(C(C2(CC#C)CCCOC2)=O)CCCC2(C1)CN(C(c1cnco1)=O)CCO2 Cc1c[nH]cc(C(=O)NC2(CCCNC(c3csc(Br)n3)=O)CC2)c1=O Cn1nc(C(=O)NC(Cn2cncn2)C(=O)NCCc2cccnc2)cc1C#N N1(C(CCc2cnn(C)n2)=O)CC2CCC(C1)N2C(c1ccc(C2CC2)s1)=O CCC(C)(COC)C(=O)N1CCCC(N(C(=O)C=CCN2CCCC2)C)CC1 C1(CNC(C=CC)=O)COC(C)(C)CN1C(c1cc(C)cc(C(C)(C)C)c1O)=O C=CCC(C(=O)NCC(CC(C)C)NC(c1cccc(C(F)F)c1)=O)N(C)C N1(C(C=CCC)=O)CCC(C)C1CNC(C1(CCN(C)C)CC1)=O C=CC(CC)CC(=O)NCCn1cnc(C(N2CCOC(C(C)(C)C)C2)=O)c1 FC1(F)CCC2(CC1)CC(Nc1cc(CNC3CC3)ccn1)CCO2 C1(NC(c2ccc(OC)nn2)=O)CC(NC(C2CCC3CCC2O3)=O)C12CCC2 C(=O)(C(CCC1CCCC1)N1CCCC1CC1CCCCC1)NCCC#N C1(C(N2CCC(CN(C(=O)CCN3CCCCCC3)C)C2)=O)CC(C)(C)CN1C c1(C(N2C(C(=O)NC(CC=CC)CO)CCC2)=O)cn2c(n1)CCC2 c1(CN2CC(NC(c3c(CC)noc3C)=O)C3C2C3)ccc(OC)c(Br)c1 N1(C(CCc2c(C(C)=O)c(C)[nH]c2)=O)CC2CCC(C1)N2C(C1CC1C(N)=O)=O N1(C(c2cccnn2)=O)CCC(F)(C(N2CCC(O)(CO)C2)=O)CC1 N1(C(C(CCC)N(C)C)=O)CC(CNC(=O)C(=O)Nc2ccccc2)C(C)(C)C1 C12(NC(CCCC)=O)CC1CN(C(C1(c3ccccc3)CC1(F)F)=O)C2 C(CN=c1[nH]nc(O)s1)N(C(=O)CCc1nccs1)C C1(C)(CC)C=C(C(=O)N2CCOCC(NC(=O)CCn3cncn3)C2)C1 N1(C(CCCCSC)=O)CCC2(CCC2)C(CNC(C2CC=C(C)CC2)=O)C1 c1(C(=O)NC2CC(C)N(C(=O)Cc3cncn3C)CC2)cncc2n[nH]cc12 C1(C(=O)NCCc2c(CNC(Cc3cc(C)[nH]n3)=O)nco2)(CO)CCC(C)C1 C1(C(=O)NC(CC)CC(=O)OC)CCCCC1(C)NC(=O)C(O)CC1CCCC1 C(C(C)(C)C(=O)NCC=CBr)NC(CC(C)C1CCCO1)=O C1(OC)CC2(C1)CC(C(=O)NC1CN(C(=O)CCCN(C)C)C3CC13)C2 c1(OC(C)C)cc(C(N2CCN(C3CN(C(C4(C)CC4F)=O)C3)CC2)=O)ccn1 c1(C(=O)NCC2CN(C(C3OCCCO3)=O)CC23CC3)c[nH]c2ncccc12 c1(C(=O)NC2CC(NC(C3CNC(=O)N3)=O)C2)cnc2c(Br)cccn12 c1(C(=O)NCC2C(CNC(c3cn(C(C)(C)C)nn3)=O)C2)cc(N)c(F)cn1 C1(C(=O)NCCc2c(C)noc2C)CCN(C(=O)C(C)CCN(C)C)CC1O C(CCCC(=O)NN1CCCC1C(=O)NC(C)(CO)C(F)(F)F)N(C)C CCC(C)(C)CCCC(=O)N1CC2CC2(CNC(=O)CCCc2nncn2C)C1 N1(C(c2cnn(C)c2Cl)=O)CC2OCC(C(N3CCC(C(C)(C)O)C3)=O)C2C1 N1(C(C2CC(CC3CC3)C2)=O)CC2(C(=O)NC3CCCC(O)CC3)CCC1CC2 c1(OC)ccnc2c1CCC2NC(=O)C(=O)C=Cc1cccs1 C(=O)(C(C)(CSC)NC)NCC1(O)CN(C(C2(CC=C)CC2)=O)C1 C1(N(C(C)(C)C(=O)NC)C(c2ccc(Cl)c(I)c2)=O)COC2(CCNCC2)C1 C(=O)(CC1=CCCC1)NCC1CCC(F)(CN(C(C2C(CN(C)C)C2)=O)C2CC2)C1 N1(C(C(C2CCCCC2)N(C)C)=O)CC2COCC2(NCC=CCl)C1 c1(N2CCC(CNC(=O)CC3CCCCO3)C2)c(Br)cccc1[N+](=O)[O-] c1(C(=O)NC2C(NC(CC3CC(=O)NCC3)=O)CC2)cc(C(F)(F)F)cnc1O C1(NC(CCC#C)=O)CC12CCN(C(c1noc(C)c1C)=O)C2 N1(CC)CCN(c2cc(N(C)Cc3ccc(SC)cc3)nc(SC)n2)CC1(C)C n1(CC)nccc1C(=O)NC1C=CC(C(=O)N(C2CCC3CC23)C)C1 c1(C(C(=O)NCCC)N(C2CC(n3cccn3)C2)C)ccc(S(C)(=O)=O)o1 N1(c2nc(N(CC(CCC)C)C)nc3c2SCC3)CCN(C)c2ccc(C)cc21 CCC(CCC(=O)NC(C)(C(=O)NOC1CCC1)C1CCC1)OC N1(C(c2c(CC)ccs2)=O)CCN(C(c2cc(C(F)F)cs2)=O)C(C)CC1C C(=O)(C(C)C(=O)N1CC(NC(C2CC(C)(F)C2)=O)C(C)C1)OC C1(NC(C(COC(C)C)(C)C)=O)CCC(C)(C)N(C(=O)CN2CC3CC3C2)C1 C1(C(F)(F)F)(C(N(CCN(C(C)C)C(c2cncc(N)n2)=O)C)=O)CC=CCO1 Cc1ccc2c(c1)C(CCNC(=O)NC1CC(C)OC1=O)C(=O)N2 C(=O)(C#CC1(C)CC1)NCC(C)N(C(=O)Cc1csc(C2CC2)n1)C C(CCCC(C)NC(=O)C(c1cnn(C)c1)C1CC1)NC(C(COC)C)=O Cc1ccc2c(C(=O)NCC(CC(C)C)NC(=O)Cc3ncc(C)s3)coc2c1 c1(N2CCC(NC(c3cn(CCOC)nc3)=O)C(O)C2)ccnc2nc(C)nn12 c1(NC(C2(C)CCN(C(C3C(C)C3C)=O)C2)=O)cccc(N=[N+]=[N-])c1 C1(C(=O)NCc2c(C3CCN(C(CSC)=O)C3)n[nH]c2)CC(=O)N(OC)C1 n1(CC(=O)NCC(CNC(C2(CC#C)CC2)=O)O)cc(Br)c(C)n1 CC1=C(C(=O)NCCC(C)NC(=O)Cc2sccc2Br)SCCO1 N1(C(C)=O)CCC2C(CCN2CC(c2cc(Br)ccc2Br)=O)C1 C1(C#CC(=O)NC(CNC(c2cnc3cc[nH]c3c2)=O)CCOC)(CC)COC1 N1(C(c2cc(C)oc2)=O)CCC(C)(CNC(C2(C)CCCCC2C)=O)CC1 CC(C(=O)NCCCN(C(=O)CN1CCC(=O)NC1=O)CCO)C(C)C(C)(C)C CCCC(C)(O)C(=O)NCCCCCCNC(C1C2C3CCC(C3)C12)=O Cc1nc(C)c(C(=O)NCCOCC(C)C(=O)Nc2ccncc2)o1 c1(C(=O)NC(C2CCCCCC2)CC)ccc(-n2cc(CCOC)nn2)cc1C c1(C(=O)NCCC(CNC(c2ncn(CC)n2)=O)O)c(C)nc2sccn12 c1(C(=O)NC2(C3CCCN3C(c3ccc(Cl)s3)=O)CC2)cccc2oc(O)nc12 C(c1cnc(O)nc1O)=CC(=O)NCC1(NC(c2c(C)[nH]c(C#N)c2)=O)CCC1 C12(CNC(c3cnsc3)=O)CCC(CC1)N2C(C1CC2(C1)CC(O)C2)=O c1(C(=O)NNC(=O)NCC2(COC)CC3CCCC3C2)cccc2ccccc12 N1(C(c2ccccc2F)C)CCC(C2(NC(=O)Cc3cccs3)CC2)CC1 C1(C(=O)NCC2(CC)CCCO2)CC2(CCN(C(=O)CC3(O)CCCCC3)C2)C1 C1(C(CNC(=NC)NC(C)CF)C)CCN(C(=O)OC(C)(C)C)CC1 N1(C(=O)CSC2(c3ccon3)CCC2)CCCN(C(=O)Cn2cc(Cl)cn2)CC1 c1(C(N2CCC(NC(=O)CS(=O)(=O)CCO)C2C2CC2)=O)cc2cc(F)ccc2o1 C1(OC)CC(NC(=O)Cc2cc(C(F)(F)F)nn2C)CN(C(C2SCCS2)=O)C1 n1(C2(C(=O)NC(C)CCNC(C3CC3(C)C(F)(F)F)=O)CC2)cc(Cl)cn1 C1(C(=O)NC(C)CNC(C2CCN(C)C2)=O)CC(=O)C12CCC2 c1(CC(=O)NC2C3CCN(C(C(C)n4ccnc4)=O)C32)ccc2c[nH]nc2c1 N1(C(c2c(C)ccs2)=O)CCCC2C1CCCN2C(=O)C=Cc1cn(C)cn1 C1(=CC(N2C3C(NC(CC(C)OC)=O)C(C3)C2)=O)CCCCCC1(F)F C1(C(=O)NCCn2c(C)cnn2)CN(C(=O)C(C)c2ccsc2)CC1C(C)C c1(OCC)c(NC(N(C2(C)CCOCC2)C)=O)cc(Cl)cc1CC c1(C(C(N2C(CO)CC(NC(C(C)(C3CC3)OC)=O)C2)=O)C)nc(F)ccc1Cl C1(C(=O)NC(c2ccccc2)C#C)CSCN1C(c1cnsc1C)=O c1(OC)c(CNC(=O)C(c2ccc(O)c(C)c2)O)cccc1C(C)(C)C N1(C(c2c(C)n[nH]c2C)=O)CC(C)(C(=O)NCCP(C)(C)=O)CC1(C)C c1(CC)ccc(C(N2CCC(CNC(C3CC(C)C3)=O)C(C)C2)=O)cc1N c1(C(F)F)ccc(N2CCN(Cc3ccc(-c4ccccc4)s3)CC2)nc1 CCCCC(C)C(=O)NCc1c[nH]nc1C(=O)N(C)Cc1scnc1C CC1(C)CN(C(C2CC2C2CC2)=O)C(CNC(c2cc(N)cc(F)c2)=O)CO1 C1(NC(CC2(N(C)C)CC2)=O)C=CC(CC(=O)NCC(n2cccn2)C)C1 CCC(C(=O)NC(C)C(C(=O)NCC(C)(F)C(C)(C)F)C(C)C)C(C)(C)CC c1(C(N2C3CCC(NC(c4c(C)nc(CC)o4)=O)(C3)C2)=O)cc(S(N)(=O)=O)cs1 C(=O)(CC(CCCCC)CCCCC)N(CCNC(CCCC#C)=O)C1CC1 C1(CC)(NC(=O)Cc2ccnc(OC)c2)CCN(C(c2ccccn2)=O)CC1 c1(C(N(C(C)C(=O)N(C)CCC2CN(C)C2)C)=O)ccc(F)cn1 c1(OC)nc(=NC2CCC3CN(C(=O)CS(=O)(=O)C4CC4)CC23)[nH]c2[nH]cnc12 c1(Cn2c(C(c3ncc[nH]3)NC(COC)C3(C)CC3)nnn2)ccc(F)cc1 c1(CCC)[nH]ccc1C(=O)NCC1CCOC1C(=O)NCC(CC)n1cccn1 N1(C(C)C)CC(NC(=O)C(C)(C)CNC(C2CCC(=O)C2)=O)C(C)C1 C(=O)(C1=CC(O)C(NC(C2CCCC2O)=O)C1)NC1C(C#C)CCC1 CC1CN(C(=O)NC2CNCCN2C2CCCCC2)C(=O)N1 C(=O)(C(F)C(F)(F)F)NCC1N(C(C(C(C)C)NC(COC)=O)=O)CCCC1 C1(NC(CC2(CSC)CC2)=O)CC(O)CN(C(C23CC(C)(C2)C3)=O)C1 c12c(C)nn(c1C)CN(C)ONC(=O)C2.c1(N(C)C)nc(CC2CCCO2)cs1 C(=O)(C(C)(C)CCSC)NC(CC(=O)NC(CC)CC(C)O)COC Cc1nnc2cc(N3CCC=C(CNC(c4cccc(F)c4F)=O)C3)ncn12 CCCC(CNC(=O)CSCCC#N)C(=O)NCCCc1nccs1 Cc1nc(N)cnc1C(=O)NCCCN(C)C(C1(C)CCCO1)=O C=CCC(CC(C)C)C(=O)NC(Cc1cc[nH]n1)C(=O)NC1CC(O)C1 N1(C(c2nc(C)n(C)n2)=O)CCN(C(C2COCC2(C)C)=O)CC1CC(C)(C)C Cc1nn(C(C)(C)C)c(C)c1S(=O)(=O)NCC1CCN(C2CC2)CC1 C1(CC)C(C(=O)NCc2cc(C)nn2C)CCCN1C(=O)C(O)CN(C)C C1(n2c(C(C(C3CC(F)(F)C3)OC)NCCCCOC)nnn2)CCCCCC1 N1(C(CS(CC)=O)=O)CC2CN(C(c3cccnc3C3CC3)=O)CC2(C)C1 c1(C(=O)NCC2(CO)CCN(C(C(CCC)OC)=O)C2)c(C)nn(C)c1OC Cc1cc(C(=O)NCC2CCCC2NC(=O)CCc2nc(C(C)C)no2)ncn1 N1(C(CC)=O)CCN(S(=O)(=O)NCCCOc2cc(Cl)cc(Br)c2)CC1 C(=O)(C1=Cc2cc(F)ccc2OC1)N1CCC2(CN(C(C3C(=O)NCC3)=O)C2)C1 c1(C(N(C(CC)CC(=O)NCC23CCC(CC2)O3)C)=O)cccc(O)c1F C1(NC(CCNC(=O)NC)=O)CC2CCC1(C(=O)N(C)Cc1cccc(C)n1)C2 Cc1cc(O)ccc1CC(=O)NC1(C)CCN(C(c2cnn(C)c2)=O)C1 N1(C(c2c(C)occc2=O)=O)c2ccc(Cl)cc2N(C)C(=O)C1(C)C C#CC1CC(NC(=O)C(=O)NC(c2ccco2)C)C1 N1(C(C(CC)SC)=O)CC(O)CC1CNC(=O)C(=O)NC(C)C C1(C(=O)NC(CC)C(=O)NCC2CC3(CCO2)CC3)CC2(CCO1)CC2 c1(OC)ccccc1C(C)NC(=O)C(=O)NC(C1CCCO1)COC c1(C(=O)NCC2OCCN(C(c3onc(C)c3C)=O)C2)ccc2occ(C)c2c1 C1(C(=O)NCc2ccncc2F)CN(Cc2cc(F)cc(I)c2)CCC1(F)F C1(C(N(C(C)CNC(=O)CCC(=O)c2cnn(C)c2)C)=O)CNC(=O)CC1(C)C c1(C(=O)NC2(C)CC3(CC3)C(NC(=O)OC(C)(C)C)CC2)cccc2ccsc12 N1(C(CCCC=C)=O)CCCC(F)(CNC(C2CCC3(CCC3)O2)=O)CC1 C1(NC(C2C(C)CCC2)=O)CC2(C1)CN(C(=O)Cc1nnc(S)n1C)C2 C1(C(=O)NCC(C(=O)NCCCC(F)F)N(C)C)CCN(C)C1=O c1(C(N(C)CC=CC(=O)NC2CCC3(CC3)C2)=O)ncccc1C c1(C(=O)NC(C2CN(C(C3OCCOC3(C)C)=O)C2)C)ccnc2[nH]nnc12 N1(C(CC#C)=O)CCN(C(c2cc(C)nc(C)n2)=O)CC1C Cn1c(-c2ccc(Cl)cc2)nnc1CC(C1CCCCC1)=O C1(NC(CCCCOC)=O)CC2CN(C(=O)CN(C3CCC3)C)CC2C1 c1(NCC(CC)CC(F)(F)F)cc(=NC(C)Cc2ccncc2)[nH]c(C)n1 C(=O)(C1=CCC(NC(=O)CC2CCCCCC2)C1)NC(c1ccsc1)C C1(C(=O)NC2C(C)NC(=O)CC2)CN(C(c2ccsc2C#N)=O)CC(C)(C)C1 c1(-c2cn(C3CCN(C(CC4(C)CCC4)=O)C3)nn2)cncc(C(=O)O)n1 C(=O)(C1=CC2CCC(C1)C2)N1C(C)CC(CC(=O)N(CCF)C2CC2)C1 c1(CNC(C2C(C(N3CC(N(C)CC)C3)=O)CCO2)=O)ccc[n+]([O-])c1 C1(C(=O)NC2C(C(C)(C)C)N(C(=O)CC=C(Cl)Cl)CC2)CCc2ncnn2C1 c1(C(N2C3C(NC(CCCCCC)=O)(CCC3)CC2)=O)ccc2c(c1)C(=O)NC2 C(CS(=O)(=O)CC(=O)NC1CCCN(C(=O)C=Cc2ncc(C)[nH]2)CC1F)OC C1(CNC(C(CC(C)C)(C)C)=O)CCCC2CN(C(=O)C(C)(C)OC(C)C)CC12 CC(CO)C(=O)NC(CNC(=O)CCOC1CCCC1)CO C(=O)(N=c1[nH]oc2cc(Br)ccc12)C1N(C(Cc2cn(C)nc2)=O)CC2(CC2)C1 C(CCO)(C(C)(C)C)NC(C1(N(C(C2COCC(C)O2)=O)C)CC1)=O c1(C(=O)NC2CCN(CCNC(C(C)=C(CC)C)=O)CC2)cccc(F)c1F CCCC(CC)C(=O)NCc1cc(C(=O)NCC(CO)C2CCC2)cs1 C1(F)(C(=O)NCCC(C)(C)C)CCCN(C(C2(C)COC2)=O)C1 C1(C)(CNC(C(CC)O)=O)CCCN(C(=O)C(c2ccc(Cl)cc2)=O)C1 N1(C(CC(C=C)(C)C)=O)CCC(O)(C2CCN(C(=O)C=Cc3ccoc3)CC2)C1 Cc1ccc2nc(C)c(C(=O)NCC34CCCCN3CC(N)C4)n2c1 C(C)(C)(CCC(=O)NCCCCCC(=O)NC1C2CCC(F)(F)C12)OC Cc1cc2c(CNC3CC(n4cc(C(C)(C)C(N)=O)nn4)C3)cccc2s1 C1(C(N(CCCNC(=O)COC(C)(C)CC)CCC)=O)CCCN1C=O C1(NC(C(C(C)C)CNC(c2sccc2CO)=O)=O)CCC2CCCC1O2 Cc1ccc2c(c1)C=C(C(=O)NC1CCC(CCC(C)C)C1)CO2 Cn1c(C(=O)NC(C2CCN(C(C3(CCO)CC3)=O)C2)(C)C)nnc1S C(C(C)C)(C(O)C(=O)N1CC2CCN(C(=O)CC3CCCSC3)CC12)OC C1(NC(C2(CC)CC(F)(F)C2)=O)CC2(NC(=O)CCc3cccnc3)COC1C2 N1(C(CNC(CC=O)=O)=O)CCCC(OCCSCC)C1C.CCN O=C(C#CC1CCCO1)NCC1CCC(NC(=O)C(F)CC2CCCC2)CC1 c1(CC)cc(F)ccc1CC(=O)NCC1COCCN1C(=O)C=CC1CCOC1 N1(C(C(C)O)=O)CCC12CCN(C(C1(Cc3cccc(F)c3)CCC1)=O)CC2 c1(C(N(CCC(C)NC(c2ccn(CCC)n2)=O)C)=O)cnc2n1CCC(C)C2 N1(C(C(c2ccnn2C)C)=O)CC2(C1)CN(C(C1(F)CCN(C)CC1)=O)CCO2 N1(C(C(CC)(C)C)=O)C2CCCC1CN(C(=O)CC1CN(C)C1)C2 C(=O)(C1CCc2ccccc21)N1CC(C(C)NC(C23CCC2CC3)=O)C1 N1(CCC)CCCCC1C(N1CCC(=CCNC(C2CCC(F)CC2)=O)CC1)=O c1(CNC(c2ccc(C)cc2)C(=O)O)ccc2cc(F)ccc2n1 c1(C(N2CC(C)(NC(c3c(F)cc(O)cc3F)=O)C2)=O)cncc(S(C)(=O)=O)c1 c1(C(C)=O)ccc(NC(C2CCCN2C(c2ccc(O)nc2Cl)=O)=O)cc1Cl N1(C(=O)CC=C(Cl)Cl)CCC2(CCCN2C(=O)COCc2ccccc2)C1 C(CC(=O)N1CC(CO)CC(C)(C)C1)(C(F)(F)F)NC(c1c(CC)cccc1)=O C1(Cn2cc(CC3N(C(c4c(C)nsc4N)=O)CCC3)nn2)CCCCNC1=O N1(C(c2cnc[nH]2)=O)CCCC2(CCCN(Cc3c(C4CC4)cccc3F)C2)C1 CCC(O)C(C)(C)C(=O)N(CC(C)N(C)C(c1ncccc1F)=O)C n1(CC(=O)NC(CC=C)CNC(=O)Cc2cc[nH]c2)cc(C(F)(F)F)ccc1=O C1(CNC(C2C(=C)C2)=O)CCN(C(c2ccc(OC)c(N)n2)=O)C1(C)C c1(C(=O)NC2CN(C(C(C)(C)c3cnsc3)=O)C2)ccc2cccc(Cl)c2n1 C(c1cccnc1)=C(C)C(=O)NCCC1(O)CCN(C(C2CCCCN2C)=O)C1 Cc1nn(C(C)C)cc1C(N1CC(NC(C2SCCCS2)=O)C(C(F)F)C1)=O C1(CNC(c2c(CC)scc2)=O)CN(C(=O)Cc2ccccc2O)C2CC12 C1(C(=O)NC(c2nc(CC)on2)C)CN(C(C2(NC3CC3)CCC2)=O)CCN1C c1(C(=O)NCC(CNC(C(C)OCCN(C)C)=O)(C)F)cccc(F)c1F c1(C(=O)NC(CNC(C(C(C)C)C)=O)CC(C)C)ccc2occc2n1 C1(C(=O)NC(c2ncc[nH]2)CC)(NC(=O)CCNC(N)=O)CC1C c1(CNC(CCSCC)=O)cc(C(=O)NCC2CC2C2CC2)n[nH]1 CC1=C(C(=O)N2CCN(C(=O)C=C(Cl)Cl)CC(O)C2)CCC(C)(C)C1 c1(C(N(C2CCN(C(c3c(NC)cccc3)=O)C2)C)=O)cc(C2CC2)ccc1F C#CCC1CC(=O)N2CCC(C)(CC2)N1.c1(C(=O)NC)cnc(OC)cn1 CC1=NOC2(C1)CC(C(N1CC(O)(C(C)NC(C3CC(C)CO3)=O)C1)=O)C2 N1(C(C2(C(C)=O)CC2)=O)CCC2(CCN(Cc3cc(C(F)F)no3)C2)C1 CC(N)(C(=O)Nc1ccc(CCCO)cc1)C(F)(F)F CC1=CCC(C(=O)NCC2(CO)CCN(C(=O)Cn3cc(CO)nn3)C2)CC1 C1(C2CC2)(NC(C(CC)C(C)O)=O)CCN(C(=O)CCOc2cccc(C)c2)C1 CC(C)(C)CC(O)C(=O)N1CCN(C(=O)CS(=O)(=O)N2CCCCC2)C(CO)C1 c1(CC(C)NC(C2(n3cc(-c4ccccc4Cl)nn3)CC2)=O)cccc(F)c1 C1(C(=O)NCc2c(C(C)C)scn2)CN(C(=O)C=CSc2nc[nH]n2)CCN1C CCC(O)C(C)(C)C(=O)NCCN(CC(C)O)C(=O)C=C1CCCC1 c1(OC)ccc(C)c(NC(C2C3CN(C(=O)C(CC(C)C)OC)CC23)=O)c1 N1(C(c2c(N)ccc(F)c2)=O)CCC2CN(C(=O)Cc3ccc(Cl)cn3)CC2C1 N(C(=S)NCCC)CC(C)C.S(C)(=O)(=O)N Cc1cc(C)nc(SCC(=O)NCC2CCN2C(C23CC(F)(C2)C3)=O)n1 c1(C(=O)NC(CC)CNC(CCC)=O)cccc2ncccc12 C12(C(=O)NCC(C(=O)NC)(C)C)CCN(C(=O)C(C3CCCCC3)C)CCC1C2 C(C(O)CC(C)(C)C)NC(c1cc(CNC(CN(C(C)=O)C)=O)nn1C)=O C(=O)(CC1=CCCCC1)N1CC(C)(NC(Cc2c(NC(C)=O)cccc2)=O)C1 C(=O)(C1=NOC2COCC12)N(CCC(C)NC(=O)C1=Cc2ccccc2C1)C C1(NC(c2n(C)nc(C)c2Cl)=O)CCC2(CCN(C(=O)C(C(C)C)C(C)C)C2)C1 N1(C(c2ccc(N(C)C)cc2F)=O)CCN(C(=O)CCCC2CC2)CC(C)(C)C1 N1(C(=O)OC(C)(C)C)CC(CNC(C2CCOCC23CCC3)=O)OCC1(C)C C1(NC(C2=C(C)OCC2)=O)CC2CCC1N(C(=O)C(C1CCOCC1)F)C2 c1(C(=O)OC)ccc2n1CCCN2C(c1sccc1Cl)C(=O)NC1CCOC1 Cc1nc(-c2cccc(F)c2)sc1C(=O)NC1CC(NC(C2CCC(O)C2)=O)C1 C1(C2CCN(C(c3cc[nH]c3)=O)C2)(NC(C(Cn2ccc(C)n2)C)=O)CC1 C1(NC(C(CC)NC(C)=O)=O)CCN(C(c2ccn(CC)c2C)=O)CC1O N1(C(CCC=CC)=O)CCC(O)(CNC(=O)C(O)C(C)CC)CC1 N1(C(C2(CCC)CCNC2=O)=O)CCCC(NC(=O)CCC2(C#N)CCC2)CC1 N1(C(CC2N(C(c3c(C#N)ccs3)=O)CC2)=O)CCCC(C#N)C1 c1(C(N2CCC(C(N3CC(N(CC=C)C)C3)=O)(CC)C2)=O)ccc2nccn2c1 c1(C(N(C)Cc2ccnn2CCc2ccccc2)=O)cn(C)c2ccc(Cl)cc12 C(=O)(C(F)C(C)CNC(c1cn(CC)nn1)=O)NCCCC=CC C1(C(=O)NC(C)(CNC(=O)Cn2ccnn2)C2CC2)CCc2nncn2C1 C(=O)(C#CC1CC(F)(F)C1)NC(C1CCN(C(c2ccnn2CC#N)=O)C1)C CC(C)CCC(F)C(=O)N1CCC(C)CC1C(=O)Nc1ccc(F)c(O)c1 C(=O)(C(C)C(CC)CC)NCC1ON=C(C(=O)N(C2CCCCC2)CCC)C1 c1(N(C2CCN(Cc3ccc(=N)[nH]c3)C2)C)ccc(Br)cc1 C1(C(=O)NC2(CNC(C(C)=C3CCC3)=O)CCOCC2)CCOC(C)(CC)C1 C1(C(=O)NC(C)C(CO)NC(c2cocn2)=O)CCC12CCOCC2 CC(c1cccc(Cl)c1)=CC(=O)NC(C)CCCCNC(c1sccc1F)=O C1(C(=O)NC(CC)CN(C(=O)Cn2nccc2C)C)Cc2cc(C)ccc2S1 c1(N2CCC(C)(NC(=O)CCc3cnc[nH]3)CC2)ncnc2sc([N+](=O)[O-])cc12 c1(C(N2CC3CN(C(=O)Nc4ccc(F)c(F)c4)C3C2)=O)ccc(B(O)O)cc1 N1(C(C)=O)CCC(NC(=O)Nc2cnc(N3CCCCC3)nc2)C(C(C)C)C1 C1(CNC(C(=Cc2ccccn2)C)=O)CCN(C(c2ncsc2C)=O)C(C)C1 c1(C(CC)N(C2CC2)NCC)cccc(-c2ncccc2OC)c1 C=C(C)C(C)(C)C(=O)NCC1C(C)CCN1C(=O)CC1CC(=O)NC(=O)C1 C1(CNC(C23CC(CC)(OC2)C3)=O)CC(C)CN(C(C2CC3CC3C2)=O)C1 c1(C(N2CCCC(N(C(CCCCC=C)=O)CC)C2)=O)nc(Cl)c(=O)[nH]c1N c1(-c2cnc(OC)c(C)c2)ccc2ncc(C(=O)Nc3nc(O)cs3)c(=O)n2c1 CC1(C)CCN(C(c2sccc2C#N)=O)CC1CNC(C12COCC(C1)C2)=O C(=O)(CN=c1[nH]c(N2CCC3CC3C2)nc2cccnc12)NC(C)C N1(C(c2ccc(CC)s2)=O)CCC(CCNC(=O)Cn2cnnn2)CC1C c1(CC(=O)NC(C)C(C)(F)F)ccc2c(c1)OCCO2 c1(N2C3CC(NC(c4nc(CC)sc4)=O)CC2CC3)nc(Cl)nc(CC)c1C#N C1(C)(C(=O)NCC(CN(C)C(C23CC(CC(F)F)(C2)C3)=O)O)CC2CCC1O2 c1(C(=O)NC2(CCNC(C=CCCC)=O)CC2)ccnc2ncc(C)cc12 C(CN=c1[nH]c(Cl)ncc1F)C1CCC(NC(CCn2c(C)cc(C)n2)=O)C1 C1(C(=O)OC)C(C(=O)NC2CC(CCNC(=O)CCSC)C2)C1(F)F C1(NC(=O)COCC(F)F)CCC(C(=O)Nc2cnncc2Cl)CC1 Cc1[nH]c(C(=O)NCC2CC2NC(C2(c3ccn(C)n3)CC2)=O)c(C)c1[N+](=O)[O-] C(=O)(C1Cc2ccc(Cl)cc21)NCC1(F)CC(NC(C2CCC(CC)CC2)=O)C1 N1(C(CCN(C(C(C(=O)OCC)(F)F)=O)C)=O)CC(C2=NOC(C)C2)C1 C(CCC(C)(C)NC(C1(NC(=O)CCCNC(C)=O)CCC1)=O)OC C1(C(=O)NC(C)CO)CC2(CCN(C(c3ccc4ncnn4c3)=O)CC2)C1 N1(C(C(C)=C(CC)C)=O)C(C)CN(C(=O)CCc2cnc[nH]2)CC1C c1(C(N2CCCCC(NC(CC(=O)NC3CC3)=O)C2)=O)c(F)ccc(Cl)c1F c1(-c2cc(C)oc2)csc(=Nc2cnn(C)c2)n1C1CCN(C)C1C C12(CNC(=O)OC(C)(C)C)CC(CCC(=O)N(c3cccc(C)c3)C)(CCO1)C2 C(=O)(C(C)(Cl)Cl)N(CCN(C(C(C1CCOCC1)OC)=O)C(C)C)C c1(C(=O)NC(CCN(C)C(C2CCC2C(F)(F)F)=O)C)cccc2c1CCCC2 N1(C(CSCCC)=O)CCC(F)(CNC(=O)Cc2nc(C3CC3)n[nH]2)CC1 C1(NC(C2CCCN2C(=O)CC2CCOCC2)=O)C=CCCC1CO CC1=NN(C)C(=O)C1CC(=O)NCCC1COCCN1C(C1CC(C)(O)C1)=O S(=O)(=O)(c1cnc(N2CCCCC(C3CC3)C2)c(Cl)c1)NC1CCN(C(C)=O)C1 CCC(C)(C#N)C(=O)NC1CC(CC(=O)NC(C2CC3CC3C2)=O)C1 Cc1ncnc(O)c1CC(=O)NCC1C(NC(=O)C(C)SCC2CCCO2)C1 c1(C(N(C2CN(C(C(C=C)O)=O)CC2(C)C)C)=O)ncnc2cc[nH]c12 c1(OCCC(=O)NC2CC(CNC(c3c(C)coc3C)=O)C2)ccc(Cl)c(F)c1 CC1CC(C(=O)NCC2CC(NC(c3sc(F)cc3Cl)=O)C2)=NO1 n1(CCCC)nnnc1C(c1ccco1)NC1CC(COC)C1 Cc1c[nH]c(C(=O)NC(C(=O)NCC2(n3cccn3)CC2)c2ccco2)c1 CC(C)(C)C(O)C(=O)NCc1ccsc1C(=O)NC1CC(F)C1 C1(CC(=O)NC(CNC(C2(C=C)CCC2)=O)C2CCC2)(N(C)C)CCCCC1 CCC(O)C(C)C(=O)N(C1CCC(CNC(C2OCCN(C)C2=O)=O)CC1)C c1(C(=O)NCC2CCC(NC(c3n(CC)ccn3)=O)C2)ccc(=O)oc1 c1(C(=O)NC2CC23CC(NC(C2(CF)CC2(F)F)=O)C3)cccc2nncn12 c1(C(N2CC(CNC(CC)=O)C(F)(F)CC2)=O)ccc2nnn(C(C)(C)C)c2c1 n1(CCC)cc(Cl)c(C(=O)NCC(C(C)(C)C)NC(c2[nH]cnc2CC)=O)n1 C1(CNC(c2cnc(C3CC3)nc2)=O)CC(O)CN1C(=O)CCn1cccc1 C(=O)(C(C)(C)C(F)(F)F)NCC1C=CC(NC(CCOCC)=O)C1 CCC(C)(CC)C(=O)NCC(C)(C)CN(C)C(c1cn(C)c(O)n1)=O Cc1c(C(=O)N(CCCNC(C23CCC(C2)C(C)O3)=O)CCO)nn(C)c1N N1(C(C2CC2C2(O)COC2)=O)CCN(C(C2(c3c(C)c[nH]n3)CC2)=O)CC1 CC1(C)CN(C(=O)Cc2cncs2)CC1CNC(c1ccc(O)cc1)=O C1(CNC(C(C(C)C)N(C)C)=O)CC2(CCN(C(c3sc(F)cc3Cl)=O)C2)CO1 C(CCC(C)CC(=O)NC1(CCNC(c2cc3c(C)[nH]nc3s2)=O)CC1)=C(C)C C1(CNC(c2nc(COC)sc2)=O)CCC(NC(=O)Cc2cccs2)CC1 Cc1cc(-c2cn(CCNC(=O)C(C3CCCN(C)C3)(C)C)nn2)ccc1C#N C(C(=O)NCc1ocnc1C(=O)N(C(CO)CC(C)C)C)(C(C)C)OC c1(OC)nc(C)ccc1C(=O)N(C)CC1CN(C(C2C3CC4C(C3)C24)=O)CCO1 CON(CCC(=O)NC1CCCC(O)CC1)C(=O)CC1CCOC1(C)C N1(C(Cc2cn(CC)nn2)=O)CCC(C)(CNC(c2nc(C)ccc2F)=O)CC1 C(C(CC(C)C)C(=O)NCCC1(O)CCN(C(c2oc(CO)cc2C)=O)C1)OC N1(C(C(C)NS(C)(=O)=O)=O)CCC(C)(CNC(C2(C#N)CC3CC3C2)=O)CC1 C1(NC(C2C(NC(CCSCCC)=O)C3CCC2C3)=O)CC2(C1)CC21CCC1 c1(N(C)CCN2CCOCC2)nc2c(c(=NC3CC4(C3)C(F)(F)C43CC3)[nH]1)CSC2 C1(CC(=O)NCC2OCC(CNC(c3c(C)oc(Cl)n3)=O)C2)COCC(C)(C)O1 C1(CN(C)C(C2CCOC2)=O)CCCCN1C(c1c(Br)nnn1C)=O C1(C(=O)NC2CC(C)(NC(CC(=C)C)=O)C2)NC(=O)OC1C N1(C(c2cnc(C)s2)=O)CC2(C1)CN(C(C13CC=CCN1CCC3)=O)CC2CO C1(SC)CCCC1C(=O)NCCOC1CN(c2nc(C(F)(F)F)ns2)C1 C1(C(C)C)CC(C(=O)N2CCCC(C)(CNC(=O)C(c3ccnn3C)O)C2)=NO1 Cc1cccc2c(CCC(=O)N3CC(CNC(=O)C(C)C(C)C)C3)c[nH]c12 c1(COC)nc(NC2(CCNC(=O)CC(C)(C)O)CCC2)cc(O)n1 N1(C(c2cc(C#N)[nH]c2)=O)CCN(C(C2CCCCCCC2)=O)C(CF)C1 C1(NC(C(CC)(COC)CC)=O)CC2CC(C1)CN(C(C1CC(C)C1)=O)C2 c1(C(=O)NCC2C(C)CN(C(=O)C(=O)NCC(F)(F)F)C2)c2c(nn1C)CCC2 Cc1cccnc1C(F)(F)C(=O)NCC1CCC1NC(c1cc[nH]n1)=O C1(CC(=O)N(CC(CC)NC(=O)Cn2cccc2C(=O)OC)C)CCCC1C N1(Cc2cncc(C)n2)CCC(NC(=O)CCc2ccc(N(C)C)nc2)C(O)C1 C1(NC(C2=C(C)OCCS2)=O)CCC(N=c2ccc(C#N)n[nH]2)CC1 C1(O)(C(=O)NC2CN(C(CCc3c(C)cccc3)=O)C2)CCCC(C)CC1 C1(CN(C(=O)COc2ccc(O)cc2)C)CC(F)CN1C(C1CC=CCC1)=O C(CCCCC(=O)NC1CC2CC1N(C(=O)CCc1nncn1C)C2)OCC C(=O)(C(F)CCC(C)C)N1CCC(C(CO)NC(C(CC2CC2)OC)=O)CC1 C1(OC)CN(S(=O)(=O)CCCl)CCC1NC(C1CC2CC2C1)=O c1(C(C)NCC2CC3OCCC3O2)ccc(Cl)cc1C(F)(F)F CN1CCCCC(C(N2CCC(O)(CNC(C3C4CNC(=O)C34)=O)CC2)=O)C1 N1(C(C2C(C)(CC)C2)=O)CC2CC1C2NC(=O)CC(C)(C)c1ccccc1 CC(C)(CO)C(=O)NCC1CC(O)CN1C(c1cc(C2(C)CC2)on1)=O C1(CNC(c2ccc(-c3cccc(Cl)c3)s2)=O)CCCN(C(C2C3CCC23)=O)C1 c1(OCCC(N2CCC(NC(C(C)(C)O)=O)C(O)C2)=O)cccc2ccccc12 C(=O)(C1CCCn2cnnc21)N1CCC(C)(CNC(COC(CC)CC)=O)C1 C#CCCC(O)C(=O)N1CCN(C(=O)C2=CCCC2)CC1c1cccc(OC)c1 N1(C(C2C(C(N)=O)C2)=O)CC2(CCC(NC(=O)Cc3ccc(F)cc3F)CC2)C1 C12(C)CCC(C1)NC(=O)C(=O)NC2.CCC(F)(F)C1CC1.C1C(=O)N1 C1(C(=O)NCCC2(CO)CCC2)CC2(CCN(C(=O)C(O)CN3CCCC3)C2)C1 Cc1c(C(=O)NCCC2(NC(C3CC3F)=O)CCC2)cnn1C(C)C c1(C(=O)NC2CCC(NC(C=CC(CC)C)=O)CC2)nc(Br)cnc1N Cn1cc(C(=O)NCCCCCNC(=O)Cc2ccccc2C(F)(F)F)c(Cl)n1 C1(C(=O)NC(C(=O)OC)C2CC2)CCN(C(C2CCC(C)C2)=O)C1 N1(C(c2cncc(Br)c2)=O)CCCCC2(CCN(C(c3ccncn3)=O)C2)C1 N1(C(CCC=C(C)C)=O)CCN(C(c2ccc(O)nc2C)=O)C(CC(F)F)C1 c1(C(=O)NC2CC(NC(C(C=CCCC)O)=O)C2)ccc2nnnn2c1 c1(C(C(=O)N(CC(C)NC(C=CC(CC)=CC)=O)C)OC)ccccc1Br C1(C(=O)Nc2cnc(C)nc2)CCC(C)(C)N(C(c2[nH]ccc2C)=O)C1 C1(C)(C(=O)NC2(CC=C)CCCC2)CCN(C(c2c[nH]ccc2=O)=O)C1 C1(CNC(Cn2nnc(C)n2)=O)CN(C(C2(CCF)CC2)=O)CCN1C C(=O)(C(CNC(c1nnc(S)n1C)=O)C(C)C)NC(c1ncc[nH]1)CC C(=O)(C(C)(C)CC=C)NCC(CNC(C(CC#C)O)=O)C C12(CC(=O)NCC3N(C(C4C(C(C)=O)C4)=O)CCC3C)CCC(CC1)OC2 Cc1nc2ccccc2nc1C(=O)NC1CCC1NC(=O)C(c1cncnc1)C c1(OCC)ccc(CC(C)C(=O)N(CC(O)CNC(c2cnns2)=O)C)cc1 c1(SC)cc(NCC(C)N(C(=O)CC2CCCS(=O)(=O)C2)C)nc(SC)n1 C12(NC(CSCCC)=O)CCOCC1CN(C(=O)Cn1cc(C)ccc1=O)C2 C1(OCC)CN(C(C2CCN2C)=O)CC1CNC(C1CCN1C)=O CN=c1nc(N2CCC(CN(C)C(=O)OC(C)(C)C)C2)[nH]c(=NCCOC)[nH]1 C1(CNC(C2CCC(C)O2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)C12CC2 Cc1ncc(N)cc1CN1CCC(C(N)=O)CC1.N12CC(CC1CO)NC(=O)C2 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CC2(C1)CN(C(c1cscc1C)=O)CC(C)(C)O2 CCC(CC)CCC(=O)N1CCC(O)(CCNC(C2CN(C3CCOC3)C2)=O)C1 c1(NC(C2CCN(C(c3ccc(=O)oc3)=O)CC2)=O)nccc(C(F)F)c1F C1(C(N2CCC(N(CC#C)C(c3cc(OC)ns3)=O)C2)=O)CCC(F)CC1 CCN=c1[nH]c(C)c(C(N2CCN(C)CC2CNC(C2CC2CN(C)C)=O)=O)s1 N1(c2snc(C(C)C)n2)C2CCCC1CN(C(c1ccco1)=O)C2 c1(OC)ccc(COCCCN(C)C(C2CN(C(=O)OC(C)(C)C)C2)=O)cc1 C1(c2n(CCC)nnn2)(NCCC(C)CO)CC2CCC1CC2 N1(C(COCCC=C)=O)CCCC(O)(CNC(C2(F)CCS(=O)(=O)C2)=O)C1 c1(C(=O)NCCOc2c(C)cccc2Br)cccc([N+](=O)[O-])c1N C(=O)(C(C)(F)C(=O)N1CCC(CC(=O)NCCOc2cccnc2)C1)OC C(=O)(C(CN=[N+]=[N-])NC(C1CCC1)=O)NC(c1ccnn1C)C N1(C(C(COC)O)=O)CCN(CCCCCNC(=O)C(O)CCSC)CC1 C1(NCC2(n3cc(CNCc4cnc(OC)nc4)nn3)CC2)CCCCC1(F)F c1(OC)ccc(C(=O)CCC(=O)NC2CCN(C(=O)CC34CC(C3)C4)C2)cc1F C1(C(=O)NC(C2(O)CCN(C(c3[nH]nnc3C3CC3)=O)C2)C)CC2CCC1CC2 c1(C(N2CC(=C(CNC(C(CCSC)(C)C)=O)F)C2)=O)ncc(Cl)c(N)c1Cl N(C(=NCC(C)N(C)C)NCc1ccc(N2CCCC2)nc1)C1C(C)C1 c1(C(=O)NC(CNC(Cc2cn(CC)nc2)=O)CC(C)C)c(C)ccc(Cl)c1N C(=O)(CS(=O)(=O)C1CC1)NC1COCCN(C(c2ccn(CC)n2)=O)C1 C1(CC(N2CCC(F)(CF)C2)=O)CC(F)(F)CN1C(=O)Cc1ccoc1 CC(CN(C)C)CCC(=O)NCCn1cc(C(=O)NCC(O)CCO)nn1 C#CCCN(O)C(=O)N1CCNC1=O.C1(CC)CC1 C1(C(N(C2CN(C(CSCCC)=O)C2)C)=O)CCc2ccccc2O1 N1(C(CNC(N)=O)=O)CCC(c2cccc(F)c2)(NC(C2CC(F)(CO)C2)=O)C1 Cc1noc(C)c1SCC(=O)NCC1(F)CN(C(=O)C=Cc2cncs2)C1 C1(C(=O)NCC2(O)CN(C(CC(COC)C)=O)C2)CN2CCCN1CC2 N1(C(C=CC)=O)CC2CCC(C(=O)N(C)CC3COCCO3)(C2)C1 c1(C(N(C2CN(C(CSCC#C)=O)CC2F)C)=O)n[nH]c2cc(Cl)ccc12 c1(C(=O)O)ccccc1S(=O)(=O)NC1CCSc2sccc21 Cc1ncc2n1CCC(C(=O)NC1CC(F)CN(C(C3CC(C)(C)C3)=O)C1)C2 C(CC(=O)NCC1(CCNC(=O)C(C)(C)c2cccnc2)CC1)(C(F)(F)F)OC n1(CC)ccnc1C(N1CCC1C(N1CCC1CC1CC1)=O)=O NS(=O)(=O)c1sccc1C(=O)NC1CN(C(=O)CC2OCCCO2)CCC1F c1(C(N2CCC3CN(C(=O)COc4cccnc4)C3C2)=O)ccc2sncc2c1 C1(CC(=O)NC(C=C)CO)CC(C)N(C(=O)CN2C(=O)CCC2=O)C1 C1(C(N2CCC(F)(CNC(=O)C=CC3CCCC3)CC2)=O)CCC2CCCCN12 N1(C(c2c(OCC)cc(Cl)cc2)=O)CCCC2CN(C(c3cc(C)c[nH]3)=O)CC12 CN1CCCC(C(=O)N(C)CC2(O)CCN(C(=O)CC3(C(F)(F)F)CCC3)C2)C1 Cc1nscc1CC(=O)N(CC(=O)NCC(C(=O)CC(C)n1ccnc1)=O)C c1(C(N2C(CNC(=O)CSC(F)(F)F)CC2)=O)cccc2c1CCOC2 c1(CC)cc(C)[nH]c(=NCCC2CC(C)N(C(c3ccc(CC)o3)=O)C2)n1 c1(C(N2C(C)CCC(c3cn(C4CC4)nn3)C2)=O)ccc2cnccc2n1 c1(OC)cccc(C(=O)NCCN(C(=O)C(=O)NC2(n3cnnn3)CC2)C)c1 c1(C(=O)NCC(C2CCOC2)NC(COCCCC#C)=O)csc(CC)n1 C1(C(N(C2CCCN(C(c3cccc(=O)o3)=O)C2)C)=O)CC(C2CC2)C1 N1(C(C(C)NC(C)=O)=O)CCCN(C(c2csc(Cl)n2)=O)C(C)C1 C#Cc1ccc(C(=O)NCC(CC(C)C)NC(=O)C=Cc2cn[nH]c2)nc1 CC(C)C(CNC(=O)CC1C2CCCC2N1C(c1ccsn1)=O)C(C)C O(NC(=O)C(C)(C)CCNC(C1CCC(OC)CC1)=O)CCCC C1(NC(c2c(C)nc[nH]2)=O)(CNC(=O)C(F)(F)Sc2cnn(C)c2)CCCCC1 c1(C(=O)NCC(CNC(c2nccc(C)n2)=O)CO)cc2c(s1)CN(C)CC2 c1(C(=O)NC23CN(C(C4(SC)CC4)=O)C(C2)C3)ccc(C)n(C)c1=O C1(NC(CC2CC(OC)C2(C)C)=O)CCN(C(c2ccc(Br)o2)=O)CCC1CO S(=O)(=O)(c1cccnc1Cl)N1CC2(N(C(COc3c(C)cccc3)=O)CC2)C1 c1(CN(C(=O)CNC(=O)COC2(C)CCC2)C)n[nH]c2c1CCC2 c1(OCCCC(=O)NCCN(C(c2cnc(=N)[nH]c2)=O)CC)ccccc1Cl N1(C(CC(CC)C2CCC2)=O)CCOC(C(=O)NCCCCCN=[N+]=[N-])CC1 C1(C2CCCN(C(c3scnc3Cl)=O)C2)N(CCC2CC2(Cl)Cl)CC12CCC2 n1(CCC(=O)NCCC2CCN(C(c3n(CC=C)ccc3)=O)C2)c(C)ccc1C C(=O)(C(=O)C(C)(C)C)NC1(CC=C)CCN(C(C2CCCC(O)C2)=O)C1 c1(C(N2CCN(CCCNC(c3cccnc3)=O)CC2)=O)c(Br)cc(O)cc1Br N1(C(=O)Nc2ccccc2)CCC(COCc2ccco2)C1 c1(C(N(CC(=O)NCC(O)COC(C)C)CCC)=O)sccc1CC c1(OC)cc2ncccc2cc1-c1csc(C(N2CCNCC2C(N)=O)=O)c1 C(C(C)(C)CCNC(c1ccnc(C)c1)=O)NC(CCN(CCCCC)C)=O N1(C(C(C(=O)OCC)F)=O)CCC(NC(c2oc(CO)cc2C)=O)CC(C)(C)C1 C1(NC(=O)CCc2ncc[nH]2)CCCC12CCN(C(c1nnc(O)nc1O)=O)C2 c1(C(C#C)NC(=O)NC2CC2CNC(=O)OC(C)(C)C)cccnc1 C1(n2cnnn2)(C(N(CC(CN(C(c2nc(C)oc2)=O)C)O)C)=O)CCCCC1 c1(OC)ccc2nc(C)c(C(=O)NC3CCCN(C(=O)Cn4ncnn4)C3)n2n1 Cc1nn(C)cc1CC(=O)NCCOCCCNC(C1CC1Cl)=O Cc1nnc(CCNCC2CCN(C(=O)C(C)N(C)C(C3CCOCC3)=O)C2)s1 CC1CCCCC1(C)C(N1CCC(CO)(CF)C1)=O.N12CCC(C1)NC2=O.C(CF)O C1(CC(=O)NC(C2C(C(N3CC(SC)C3)=O)C2)C)CCCCN1C C1(NC(CCCOCCC)=O)CC12CC(CCC)C2.N12CCC(CC1)C2=O C#CC12CCC(C(N3CCC(C)(CN(C(=O)C=CC4CC4)CC)CC3)=O)(CC1)CC2 N1(C(C(CCCOC)(C)C)=O)CCN(C(C2CCCN2C=O)=O)CC12CCC2 CS(=O)c1ccc(CC(=O)NC2CCCCC2NC(=O)CCC(N)=O)cc1 Cc1cnc(NC(c2cccc(F)c2F)C)c(S(=O)(=O)NC2(CCC(C)C)CC2)c1 c1(C(=O)NCC2(C)OCCN(Cc3nc(C)[nH]n3)C2)cnc2ccc(C)cn12 C1(CNC(C=CSC)=O)CCC2CN(C(=O)C=Cc3cncn3C)CC12 N1(C(=O)Nc2ccn(-c3ccc(CC)cc3)n2)CCn2c(Br)cnc2C1 C1(CNC(C2CC2(Cl)Cl)=O)CN(C(c2nocc2C2CC2)=O)CCO1 c1(NC(C2CCN(C(c3ccc(Cl)o3)=O)C2)=O)cccc(F)c1F Cc1cccc(-c2ccc(NC(c3ccccc3N3CCOCC3)=O)cn2)c1F c1(C(N2CCC(C(C)NC(C(C3CC3)OCC)=O)CC2)=O)ccc(OC)cc1C C1(NC(c2nccc(C#C)c2)=O)CC12CCN(C(C1CCOC(=O)CC1)=O)CC2 C1(NC(=O)NCc2cc(Br)no2)CCOC2(CCCCC2)C1 C1(C(=O)Nc2c(C)n(CC3CCCC3)nn2)COCCN(c2ncns2)C1 CN=c1cc[nH]c(-c2nccn2CC(N2CCN(CC(N3CCCC3)=O)CC2)C)n1 c1(C(=O)NC2(CNC(CCOc3c(C)cccc3)=O)CC2)cc2n(c1)CCCC2 c1(CC(=O)OCCSCC=C)c(F)cc(CC)cc1S(N)(=O)=O Cc1cc(C(=O)N(C)CCN(C(=O)CCN2CCC(C)CC2)C)oc1C c1(-c2cncc(C(=O)Nc3ccncn3)c2)cc(N2CCOCC2)c(F)c(F)c1 C1(CC(=O)NC)CN(C(C)=O)CCN1C(c1cc[nH]n1)=O.C12=CC=C(C=N1)C2 c1(C(N2CCCC(CCC)CC2)C(=O)NCC)cccc2c[nH]nc12 C=CCCCC(C(=O)Nc1cnc2c(c1)CCC2)NC(=O)CN(CC)CC Cc1coc(-c2ccccc2)c1C(=O)NCCCNC(=O)CCc1cc(Cl)no1 Cc1cc(CCC(=O)NC(C)C(C)NC(c2cccc(O)n2)=O)ccc1Cl c1(C(=O)NC2C(NC(CC3(OCC)CCC3)=O)CCC2)cnn(C)c1C(C)C C(=O)(CCC(C)(C)O)NC(C1CCN(C(C(C)OCC)=O)CC1)C c1(NC(=O)CCOC2CC(NC(C34CCCC3C4)=O)C2)cccc(O)n1 C(=O)(CCS(=O)(=O)CC(C)C)Nc1cc(-c2cn(CC3CN(CC)C3)nn2)cn1C C(C)(CCC(=O)N1CCC1C(N1CC(c2noc(C)n2)C1)=O)SC Cc1ccc(CCC(=O)NCC23CC(NC(=O)COc4cnn(C)c4)(C2)C3)o1 C1(C(N2CCC(F)(C(=O)NCC3(C#N)CC3)C2)=O)C2CC3C(C2=O)C13 C1(NC(CS(=O)(=O)NC)=O)CN(C(=O)C(O)C(C(C)C)OC)C2CCCC12 CC(C)CC(=O)NC1CCC(Cn2cc(Cn3cncn3)nn2)C1 c1(C(N2CCC(NC(C3CC(C)NC(=O)C3)=O)C2)=O)cc2ncccn2n1 Cc1cc(C(N2CC(C(=O)NCC3(C)CC(F)(F)C3)CC2(C)C)=O)ccc1C#N c1(-c2cc(C(=O)NCCCOCCNC(C(C)CO)=O)n[nH]2)ccc(F)cc1 C1(C(=O)NC2(CNC(c3nn(CC)nc3C)=O)CC2)CCOC(=O)CC1 O=C(CN=c1ccc(Cl)n[nH]1)NC(CNC(C12CC3CC(C(=O)N1)C2C3)=O)CO C(CCCCC(=O)N1CC(O)(c2cn(-c3ccccc3)nn2)C1)SC(=N)N C1(NC(C(C2CC2)SC)=O)CN(C(=O)CC2CN(C)C2)CC12CC2 C1(C(N2CCN(S(=O)(=O)c3ccc(Br)cn3)CC2)=O)C2CC3CC(C2)CC1C3 N1(Cc2n(C)nnc2)CCOC2(CCN(C(C3CCCCC3)=O)CC2)C1 c1(C(=O)NC)ccc(C(=O)NC2CCC(CNC(c3cc(C)cs3)=O)C2)cc1 C(=O)(CN=c1cc[nH]cc1)NC(CN(C)C)C(=O)NCCc1nncs1 c1(C(=O)NCC(CNC(CCc2ccc(SC)cc2)=O)O)cc2cccnn2n1 C(=O)(C1=CCC2CCC1N2C(=O)C(O)c1ccsc1)N1CC(C)N(C)CC1 c1(OC)ccc2[nH]c(=NC(C)CCC3CCC3)nc(N3CC(C)C(F)(F)C3)c2c1 N1(C(C(CC)Sc2ccccc2)=O)CC(N(C(=O)COCCOC)C)C(C)(C)C1 C12(NC(=O)CC(C)CC)CCOC(CF)(C1)C2.N(S(N)(=O)=O)CC(=O)NCCOC C1(CC(N2CCC(C)C2CNC(=O)CC2COC(=O)C2)=O)CCCC(C)(C)C1 c1(C(=O)NCC(C(C)C)NC(C(C)OCC#C)=O)cc(Cl)c(Cl)c(Cl)c1 C(N=c1cc(C2CC2)nco1)C1CCN(C(C(C)=C2CCOC2)=O)C1(C)C C1(NC(CC=C=C)=O)C2CN(C(c3cc(Br)n(C)c3)=O)CC12 N1(C(c2occ(C)c2)=O)CCN(C)C(CNC(=O)C(F)Cc2ccccc2)C1 CC1CCN(C(=O)C(=O)NC2CCC2CNC(C2(C)CCCS2)=O)CC1 Cc1cnc(CNC(C2CC2C(=O)NCc2ccc(Cl)s2)=O)cc1Br c1(C(=O)OC)cscc1C(=O)NCC(C(C)C)NC(C1(OC)CCC1)=O Cc1cnn(C)c1CC(=O)NC1CCN(C(c2cnncc2O)=O)C1 C1(NC(CCC=C(C)C)=O)CN(C(c2nn(C)cc2Cl)=O)CC1C1CC1 c1(C(=O)NC(C)CNC(c2cn(C)cn2)=O)cn(C)c2cc(Br)ccc12 C1(NC(CCC(C)SC)=O)CCN(C(c2sc(C)nc2C)=O)CCC1(F)F N1(C(=O)OC(C)(C)C)CC2(C1)SCCC2Nc1nccc2occc12 CN1N=C(C(=O)NCC(O)CCNC(c2cc(C#N)n(C)n2)=O)CCC1=O Cc1ccc(C=CC(N2CCCC2CN(C)C(c2nc(C)ncc2Cl)=O)=O)cc1 C(CC(N)C(=O)NC(C)CN1CCOCC1)SC C(C)(CCC(F)(F)F)NC(C=CCC1(NC(C=C=C(C)C)=O)CCC1)=O C1(OC)CC(C(=O)NC2CC2CNC(=O)CNC(=O)CC2CCCC2)C1 C1(CC(=O)NC(CCCC=C)C)CCCN(C(c2cc(C)sc2C)=O)CC1 N1(C(C(C#N)=C2CCCC2)=O)CC2C(CNC(C3CC34CC4)=O)C2C1 c1(C(N(CC(C)N(C(c2c(C)cc(CC)o2)=O)C)C)=O)ccc(F)cc1F C1(C(=O)NCC2(CO)CCN(C)C2)CCCC(NC(C2CCC(=O)NC2)=O)CC1 N1(C(Cn2ncc(C)c2)=O)CCCC(C)(C)C1CNC(=O)CCC1CCC(=O)C1 c12cc(ccn1)CNC2=O.C(CC)(C(=O)NC(C)Cc1csc(COC)n1)=CC n1(CC)cc(C(=O)NCC(C2CC2)NC(=O)CCCNS(C)(=O)=O)cn1 c1(CNC(N2CC(C)C(c3ccccc3)C2)=O)nc2ccncc2n1C C1(c2cc(C3(N)CC3C(F)(F)F)on2)CCN(C(=O)C(F)Cc2ccccc2)CC1 O=S(=O)(C(F)(F)F)N1CCC(CCNC2CC3CC2C3)C1 C1(C(=O)NC(C(=O)NC)CC)CC2CC2N1C(C1CC(OC)(OC)C1)=O C1(C)(Cn2c(C(C3(CF)CC3)NCc3nc(C)on3)nnn2)C(C)(C)C1(C)C c1(C(N2CCN(C(=O)CO)CC2)C(=O)NC2COC2)ccc(Cl)cc1Cl Cc1cnc2cccc(C(=O)NC3CCC34CN(C(c3cccc(Cl)c3)=O)C4)n12 C(=O)(C1CCOc2ccc(Cl)cc21)NC1C(F)CCN(C(CSC(C)C)=O)C1 N1(CC)CCCC(CNC(=O)CCNc2ccc(N(c3ccccn3)C)cc2)C1 C(=O)(CCC(=O)NCCC1CCC(NC(=O)Cn2nccn2)C1)NCCC C(=O)(C1=CC2CC(C1)CC2O)N(C1CCN(C(c2cc3cccnc3[nH]2)=O)C1)C C(CC(=O)N(C)CC1(NC(=O)Cc2cnoc2)CC1)CCN(CC)CC C1(CNC(C2CCS(=O)(=O)C2)=O)COCCN(C(=O)CCF)C1 C1(CNC2(c3nnnn3C3CCOC3)CC(OC)C2)CCN(C(=O)NC)CC1 N1(C(C=CC(C)C)=O)CCN(C(=O)CN2CCC(C)C2)C(CC(F)(F)F)C1 C1(NC(C(=O)NCC(CNC(=O)OC(C)(C)C)O)=O)CSc2ccccc2N1 S(=O)(=O)(c1ccc(O)cc1)NC(C)C(=O)Nc1cccc(F)c1C#N C1(NC(CCC(C)(C)C)n2nnnc2C(CC(C)C)SC)CC2(COCCO2)C1 Cc1cc(O)ccc1CC(=O)NCC1CN(C(C2COCCC2(F)F)=O)C1 CCCC(C(=O)NC(C)COc1cccc(Br)c1)c1ccccc1 C(=O)(CCCCN=c1nc2sccc2c(NCc2cnn(C3CCC3)n2)[nH]1)NC C(N=c1[nH]c2c(c(=NCCOCCF)[nH]1)COC2)c1c(S(=O)(=O)NC)cccc1 c1(C(N(CC(C)C(N2CCCC(CC=CCO)C2)=O)C)=O)c[nH]ccc1=O c1(OC)nccc2c(C(=O)Nc3cc(Br)c(C(=O)OC)cc3C)csc12 CCC(C)C(C(=O)N(CC(C)CNC(=O)CCCC1CCCO1)C)N(C)C C1(C(=O)NC(CC(=O)NC)C)C(C)OCCN1C(=O)CC1CCCC2CC12 c1(CC(=O)NC2CC3(CN(C(C4(C(=O)NC)CC4)=O)C3)C2)ccc2occc2c1 c1(OC)c(C)nc[nH]c1=NCC1(CNC(C2CCCC(O)C2)=O)CC1 c1(N2CCCC(CC)(CC)C2)nc(=NCc2cccc(C)c2Br)[nH]c2c1SCC2 C1(NC(C(C=CC)O)=O)CCN(C(C2CCC(C)(O)CC2)=O)C(C)C1 CN1CC(NC(C2(N(C(C3CCCC3)=O)C3CC3)CCC2)=O)C(C)(C)C1 CC(C)CCCN(C)C(C1CCCC1NC(=O)C(C)OC(C)(C)C)=O C(=O)(C(C)(C)CC(C)(C)C)NCC12CC(NC(c3c(Br)ccc(C)c3)=O)(C1)C2 c1(CC)ccccc1C(CNC(=O)CC1(O)CC1)NC(=O)CN(C1CCOC1)C N1(C(C(C)(C)n2ccnn2)=O)CCCC(CCNC(C2CC(CCO)C2)=O)CC1 Cc1cc(F)cc(C)c1C(=O)NCCC(C)(C)NC(c1cc(O)nc(Cl)c1)=O N1(C(CC=CC)=O)CCOCC1CC(N1CCC(C(C)C)CC1)=O C1(C(N(CC(C)N(C)C(c2csc(C(F)F)c2)=O)C)=O)CC2(CCOC2)C1 c1(NC(=O)NCC23COCC(C2)C3)cccc(S(=O)(=O)C(F)(F)F)c1 C(CC(N)=O)(C(=O)N1CCCC(F)CC1)NC(C1CC(=C)C1)=O c1(C(N2C(C3CCN(C(C(C)C(C)O)=O)CC3)CCC2)=O)cc2c(ncn2C)[nH]1 Cc1ccc(C2CC2C(=O)NCCOC(C)(C)CNC(C2CCC(F)C2)=O)cn1 C(N(C)N1CC2(CC(F)C2)C1)c1n(C)ncc1Br C(c1ccc(F)c(Cl)c1)=CC(=O)NCC1CC(NC(c2ccoc2)=O)C1 c1(CC)[nH][nH]c2ncnc(=NC(CCNC(=O)CC(C)(C)O)C(C)C(C)C)c1-2 Cc1[nH]c(=N)nc(O)c1CCC(N1CC(CNC(=O)Cc2cn[nH]c2)C(O)C1)=O C1(NC(=O)C=Cc2ccc(Cl)cc2)CN(C(=O)C2=CCOC2)CC12CCC2 C=C1CCN(C(=O)C(C(=O)OCC)OC)C(C(=O)NCC(C)CC2CCC2)C1 C1(C(N(C(C(C)C)C)C)=O)CN(C(c2cc(Cl)cn2C)=O)CCN1C C1(C(=O)NC(C2CCOC2)C#C)CC2CCC1CNC2 c1(CN2CC(CC(=O)Nc3c(-n4c(C)ncc4)nccc3)C2)cc(F)ncc1C Cc1cc(NC(c2csc(CNC(=O)C(C)(F)F)c2)=O)cc(CO)c1 C1(C(=O)NCC2(CC(=O)OC)CC2)(CC)CCN(C(=O)C(O)Cn2cncn2)CC1 C1(C(N2CCC(C3N(C(c4c(CC)non4)=O)CCC3)C2)=O)CCC(F)(F)CC1 c1(OC)ccc(C(N2CC(NC(c3nc(C)n(C)c3C)=O)CC(O)C2)=O)nc1Cl C1(C)(C(N2CC(CCO)(CNC(CC=C)=O)C2)=O)Oc2ccccc2NC1=O c1(NC2CC(F)(CNC(=O)CC3CCC4CC34)C2)cc(=O)n2ccccc2n1 C(=O)(C(F)(CNC(c1cnc(C)c(C)c1)=O)C(C)C)N1CCC(OCCC)CC1 c1(CC(=O)NCC(C2CC2)NC(CCCOCCOC)=O)cccc(CSC)c1 C1(C(N2CC(NC(C(C)OCCCC)=O)C2)=O)CCCC2CC12 n1(CC(=O)N(C2CC(=C)C2)C)cc(CNC(=O)C=CC)nn1 Cc1c(CN2CCC(O)C2C(=O)Nc2cc(O)ccc2Cl)cccc1O C1(C(=O)NCc2cncc(OC)c2)(NC(CN(CC)CC)=O)CCN(C)C1 C(=O)(C(CCC(N)=O)N(C)C)N1CCN(C(c2c(C)oc(Cl)n2)=O)CC1C1CC1 c1(C(=O)NCCN(C(c2cnc(C(C)=O)s2)=O)C)ccc2ccccc2n1 N1(C(C(c2ccc(OC)cc2)C)=O)CCN(C(c2cnn[nH]2)=O)C(C2CCC2)C1 c1(C(=O)NCCC2CCN(C(CSCCC)=O)C2)cccc(F)c1Br CC1CC(C)N(C(c2cn(C(C)(C)C)nn2)=O)CCN1C(=O)CO c1(C(N2CC(CC)N(C)CC2)C(=O)NC2CC(F)(F)C2)cn2cc(C)ccc2n1 C1(C)(C(=O)NC(C)C)CCCN1C(=O)CCc1nncn1C.n1(C2CC2)cccn1 C1(CC(=O)N(CCCNC(c2ccc(OC)cc2)=O)CC)COC(C)(C)CO1 Cc1cc(Cl)ccc1C(=O)NCC#CCNC(c1ccncc1Br)=O Cc1nn2c(c1CNC(=O)Cc1cccs1)CN(C(=O)Cn1cccc1)CC2 CCC(C)C(O)CC(=O)N1CC(C(=O)NCC(=O)N(C)O)C(F)(F)C1 N1(C(COCCC(C)C)=O)CCC2CCCC12CNC(c1cnnc(O)c1)=O N1(C(CN(C(CN2CC(C)(OC)C2)=O)CCO)=O)CCC2C(C(N)=O)C2C1 Cc1ccc(C(=O)NCc2c(C)[nH]c(C(=O)NC(C#N)C(N)=O)c2C)cc1Br C1(C(=O)NC2CCN(C(c3cc(CF)on3)=O)C2)CN2CCC1CC2 Cc1c(C(N2CC3CC(NC(=O)C4=CCOCC4)C2C3)=O)ccc2cncn12 c1(C(=O)OCC)ccc(CC(N2CC(F)CC(NC(C)=O)C2)=O)cc1F C(N=C(NC(C)C)N1CCCC(C2(C)OCCO2)C1)C1(OC)CCCS(=O)(=O)C1 C1(C(N(CCC(=O)N(CC2CC2)CC2CC2)CC=C)=O)CC12CCOC2 C12(CNC(C3(SC)CCC3)=O)CCCC1N(C(C1(C)CCN(C)C1=O)=O)CCC2 Cc1[nH]c(C(=O)OC(C)(C)C)c(C)c1C(N1CCC(NC(N)=O)C(O)C1)=O Cc1cc(C(N2CCCC2C2CCOC2)=O)ccc1O.N12CC(C1)OCC2=O N1(C(C(CC(C)C)OC)C(=O)NCC2(C)CC2)CCC2(CC1)C(=O)NCCN2C C=CCC(C)(C(=O)N1CC(F)(CNC(=O)C(C2CCOCC2)O)C1)N(C)C N1(C(C2(CC#C)CC2)=O)CCN(C(c2onc(Br)c2C)=O)C(C)C1 c1(C(=O)NCC(CC=C)NC(C2CC(Cl)(Cl)C2)=O)ccnc2c1CCC2 C(=O)(C(C)C(CC)CC)N1CCCC(NC(c2c(O)ncc(CC)c2)=O)C1 C1(OCC=C)CCN(C(c2cc(CNC(c3[nH]c(C)nc3CC)=O)cs2)=O)CC1 C(=O)(CCCC(=O)N1CCCC1c1nc(C(=O)NC(C2CCOC2)C)cs1)OC Cc1ccc(CC(N2CC(NC(c3ccc(C)c(C)c3)=O)C3CC23)=O)cc1C c1(NC(C2(C)CN(C(c3ccc4ncnn4c3)=O)C2)=O)cccc([N+](=O)[O-])c1Br N1(C(C2CC(CC)OCC2)=O)CCN(C(c2c(C(C)C)cnn2C)=O)CC12CC2 C(=O)(CCS(C)(=O)=O)N1C(C(C)(C)C)C(NC(C2CC(CCC(N)=O)C2)=O)CC1 C1(C(=O)NCCNC(CCCNC(=O)OCC)=O)CC(O)CN1c1ccnn1C c1(NC(C2C3CN(C(CCOC)=O)C2C3)=O)cc(C(F)(F)F)ccc1CO C(=O)(C(CC(F)F)c1ccccc1)N(CC(C)NC(=O)Cc1ccsc1)CC C(CS(=O)(=O)CC(=O)NC1CC1NC(c1ccc(C)c(C(=O)OC)c1)=O)OC c1(C(=O)OCC)[nH]c(C)c(C(=O)NCCn2ccnc2)c1C.N12CCCC1(C)C2=O c1(CC)c(C(=O)NCC(F)CNC(c2nccn2CC)=O)oc2ccccc12 C12(NC(C(n3ccc(C)n3)C)=O)CCC(CC1)N(C(C1CC(OC(F)F)C1)=O)C2 c1(C(=O)NCC(N(C(CCCC=C)=O)C)C2CC2)ccc(Cl)c2c1OCCO2 Cc1oc(C(C)C)cc1C(=O)NCC1CC(NC(=O)C(c2cccs2)N(C)C)C1 C(=O)(CC(C)(C)CNC(=O)Cn1cccnc1=O)NC(C)(C)Cc1cccnc1 c1(OC)cc(C(N2CCC2C(=O)O)=O)ccc1N1CCCCC1=O Cc1cc(NC(C2CC2CF)=O)ccc1NC(C1(C)CCCO1)=O c1(NC(C2N(C(CCN(C)C)=O)CC3(CC3)C2)=O)ccc2nc(Cl)sc2c1 C1(C(=O)NC(c2ccc(SC)cc2)C)(CC)CCN(C(=O)C(CSC)OC)CC1 N1(C(CCC=C=C)=O)CCCN(C(c2cccc3cc[nH]c23)=O)C(C(C)C)C1 c1(N2CCN(C(C)=O)CC2)nc2ccsc2c(=NCCC2CCC(C)CC2)[nH]1 c1(C(=O)NCC2CC(NC(CC3C(C)OCC3)=O)C2)cncc(C(F)F)c1 C(C(C(=O)NC(C)CCc1cn[nH]c1)C(C)(C)C)NC(C1(OC)CCCCC1)=O c1(C(C(F)(F)F)NC(Cc2c(Cl)cc(C)c(F)c2)=O)cccc2ccccc12 CC1(CNC(C2(CCc3ccccc3)CC2)=O)CCN(CCC(F)(F)F)CC1 C1(C(N(C)CCN(C)C(C2(C#N)CC2(C)C)=O)=O)CC(c2ccc(F)cc2)=NO1 CCC(CN(C)C)CC(=O)NCCC1(C)CCN(C(c2cc(C(C)C)on2)=O)C1 c1(C(=O)NC(CN(C(c2c(C)noc2C)=O)CC)C)ccc(CO)cc1OC C(CC(F)F)(C(=O)N1CC2(C=CCO2)C1)NC(=O)Cc1cccc(O)c1 c1(CNC(C(c2ccc(C)s2)N(CCC)C2CC2)=O)ccc(Cl)s1 n1(C(C)C)nccc1CNC(=O)CC1(N(C(=O)CC2CCCO2)C)CC1 c1(C(=O)NCC2(F)CC(NC(CC(C)SC)=O)C2)ccc(F)cc1C(F)F N1(C(CN(C)CCO)=O)CC(C)(C)C1C1CCN(C(c2cnc(O)o2)=O)CC1 CCC(C)CC(C(=O)NC1CC2(CCCCO2)C1)NC(c1ncncc1C)=O c1(-n2cc(C3CCN(C(C4CC(CC)OCC4)=O)C3)nn2)ccc(C)c(Cl)c1 C1(NC(COCCC)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1O C1(CNC(C(CC)n2cncn2)=O)CN(C(=O)C(C)n2cccn2)C2(CCC2)C1 c1(C(=O)NC(CC)(C)CNC(=O)CCC2CCC2)nc(C(C)C)oc1C C1(C(=O)NCC(C2CC2)SC)CCC(=O)CC1(C)C C(=O)(C1=CCCSC1)NC(CCC)CNC(C1CCCCC1COCC)=O N1(C(c2onc(C)c2C)=O)C2CCC1C(F)C(NC(C1CCNC1=O)=O)C2 N1(C(CC(CNC(C2N(CCC)CCC2)=O)C)=O)CC(F)(C2CC2)C1 C1(NC(C(C)(C)SC)=O)CCC(NC(=O)Cc2ncc(Cl)s2)CC1 C=C(CNC(=O)Cc1nonc1C)CCNC(C1(CCOC)CC1)=O N1(C(c2n(CC)nnc2)=O)CC(NC(c2cccc(Cl)c2O)=O)CCC1C O=C(CS(=O)(=O)CCO)N1C2CCC1(CNC(C1Cc3cccnc3C1)=O)CC2 Cc1cc(=NC(=O)C(=O)NC2CCN(C(C3COC(=O)N3)=O)C23CC3)[nH]o1 c1(C(N2C3CN(C(C=C(COC)C)=O)C(C3)C2)=O)coc2ccc(Br)cc12 C(=O)(CC(C)C(=O)NC(C)C(C)(C)C(=O)N(C1CCOC1)CCF)OC c1(N2C(CNC(C(CC)(F)F)=O)C(C)CC2)ncc(Br)cc1[N+](=O)[O-] C1(NC(=O)Cn2cnnc2O)CN(C(=O)C=CCF)CC1n1cccn1 CC(F)(F)CCCC(=O)NCC1CCN(C(c2cccn(C)c2=O)=O)C1 c1(C(=O)NCCCCN2CCCC(C)C2)cnc2ncn(C)c2n1 C=CC(C)C(C)C(=O)N1CC2CC(C1)C2NC(c1ccnc(C2CC2)n1)=O c1(CC(=O)NCC2CCN(C(CSC(C)C)=O)CC2C)cncc2ccccc12 CCC(C(=O)Nc1cccnc1)NC(=O)C(c1cnn(C)c1)C c1(CNC(CNS(NC)(=O)=O)=O)cnc(C)cc1C C1(N(C(=O)CC=C(Cl)Cl)C)CCCN(C(C2(O)CC2(C)C)=O)CC1 C(CCCCCN(C(=O)C(C)CC)C)NC(CC=CCC)=O C1(C(=O)OCC2COCCO2)CCc2ccccc2O1 N1(C(C(F)=CC)=O)CCC(N(C(c2ccc(C3CC3)o2)=O)CC)CC1 C1(C(C)C)CCN(C(=O)NCc2c[nH]cc2C2CC2)C1 c1(C(=O)NC2CC(C)(C)N(C(=O)Cn3ccnn3)C2)cccc2sccc12 c1(CN(CCN(CCC)CC)CC)ccc(C(=O)NC2(C(=O)OC)CCC2)cc1 c1(CC(=O)N(C(CNC(CCNS(CC)(=O)=O)=O)C)C)ccccc1O Cc1c(C(N2CC=CC2C(N2CCOC3(CC3)C2)=O)=O)cc(F)cc1Br CC(C)CC(C(N)=O)NC(c1n[nH]cc1CNC(=O)C(C)CC1CC1)=O C1(C(c2cccs2)N(C)C(=O)OC(C)(C)C)CC2C=CC1N(C(C1CCC1)=O)C2 CC1(CNC(=O)C(c2ccc(F)cc2)F)CCCN1C(=O)CSc1ccccn1 C(CNC(=O)CNC(c1cccnc1)=O)(C(C)(C)C)NC(C(F)=CC)=O N12CCCC(CC1)C2.C(=O)(CC(=O)N(C)C)NC(c1cnoc1C1CC1)C C1(C(=O)NC(C=C)C2CCC2)CCN(C(=O)C(N2CCOCC2)C)C1C CCC(C)(C)C(=O)C(=O)N1CCC2(CC2NC(c2ccc(CO)s2)=O)C1 c1(N(c2ccccn2)C)ccc(NC(=O)C(N2CCOC3CC23)=O)cc1 CN1CC2(CCN(C(C3(F)CCN(C(C4CC4C(C)(F)F)=O)CC3)=O)CC2)C1 c1(C(N2CC3C(CNC(c4cccc(CF)c4)=O)(C3)C2)=O)ccccc1[N+](=O)[O-] C1(C)(NC(C(N2CCN(C)CC2)C)=O)CCN(C(=O)C2=CCOC2)C1 N1(C(C2CN(C)C(=O)N2)=O)C2CCC(C2)C1CC(=O)NCCc1csnn1 c1(C(=O)NC(CNC(C=CCOCCOC)=O)(CC)CC)cc(O)nc(Cl)c1 N1(C(C2CC(N(C)C)C2)=O)CCOC2CN(C(=O)CN3C(=O)CCC3=O)CC12 CCS(=O)(=O)CC(=O)N1CCC(NC(c2c[nH]cc(Cl)c2=O)=O)C1 c1(C(N2C(CNC(c3ccnc(C)n3)=O)CCC2)=O)cccc2cc[nH]c12 c1(CCC(=O)NC2CC(F)(CNC(C(C)SCCCC)=O)C2)ccc(C)nc1 c1(N2CCC(CNC(C(N3CCOCC3)C)=O)C2)nc(Cl)ncc1C(N)=O CC(O)C(C)C(=O)NCc1cc(C(=O)Nc2cccc(CCF)c2)co1 c1(C(N(C(C)C)CCNC(c2ccc(N)c(N)n2)=O)=O)ccc(F)c(Cl)c1F C1(CCCC)(C(=O)NC(CN(C(=O)C(C)C2CCOC2)CC)CC)CCC1 CC(C(=O)N1CCC(C(N)=O)C1)(C1CCC1)NC(c1cc[nH]n1)=O Cc1ccc2c(C(=O)NC3(CNC(c4c(C)noc4C)=O)CC3)csc2c1 Cc1ccc(N(C)C(C2CN(C(=O)COCCC(C)C)CC2C)=O)cc1C c1(C(=O)NC(C)C(C)NC(=O)CCc2nc[nH]n2)cc(-c2ccco2)no1 C1(C(=O)OC)CCCC1NC1CN(C(c2ccc(CN3CCCC3)o2)=O)C1 C1(NC(c2c(CC)nc[nH]2)=O)CC2CN(C(=O)C(C)N(C)C(C)=O)CC12 C1(CNC(C2C(=C)CC2)=O)(CNC(C2CCC2(OC)OC)=O)CCCC1 S(=O)(=O)(c1ccc(Br)c(F)c1)NCc1cccc(C(N2CC(C)OC(C)C2)=O)c1 CCC(C(=O)NCC1(NC(c2cc(Cl)ccc2OC)=O)CCCCC1)C(C)O c1(C(=O)N(CC2N(CC(=O)NC3CC=CC3)CCC2)C2CC2)cnc2ccncc2c1 C(=O)(CC(O)C(Cl)(Cl)Cl)N1CC(NC(C2N(C)CC(F)C2)=O)(CO)C1 C(=O)(CCCCCOCC)N1C(C)(CC(=O)NCC(C(=O)OCC)C)CC1 c1(C(N2CCC(NC(c3cnc4n3CCCC4)=O)CC2)=O)ccn2nccc2n1 N1(C(C2CCN(C(C)=O)C2)=O)CC(CNC(=O)C(C)(C)C(C)C)CC(C)(C)C1 C(=O)(C(C(C)C)c1cnc(C)s1)NC(CNC(CC1(C=C)CCC1)=O)CO CC1(C(=O)NCC2CCCN2C(C2(C)C=CCC2)=O)CCNC(=O)C1 N1(C(C(n2cc(-c3c(Cl)ccc(OC)c3)nn2)C)=O)CCn2c(O)nnc2C1 N1(C(CCOC(C)C)=O)CC(CNC(C2CCCCC2)=O)CC1C N1(C(C(C)NC(N)=O)=O)CCN(C(=O)CCc2nnc(S)n2C)CC1CO C(C)(C)(CC(=O)NCC1CCCCO1)N(C(CC(C)n1cccc1)=O)C N1(C(CN(c2ccncc2)C)=O)CCC2CCC(NC(c3cocn3)=O)C12 N1(C(c2c(CC)cccc2)=O)CC2CCC(C1)C(NC(C1CCCOC1)=O)C2 C(=O)(CCC(O)C(C)(C)C)N1CCC(CNC(CN(C)C(N)=O)=O)C12CC2 N1(C(c2ccc(OC)c(F)c2)=O)CCC(N(C(=O)CC(C)SC)C)C2(CC2)C1 CC(C)(C)CCC(=O)N1CCC(CNC(c2coc3c2COC3)=O)C12CC2 C(N=c1[nH]c2c(C)cccc2o1)C1(CNC(C(C(C)C)OCC)=O)CCC1 Cc1cccc(S(=O)(=O)N(C2(CO)CC2)CC2CC3(CCNCC3)C2)c1 c1(C(=O)NCCC(C)NC(=O)CC2(C)CCS(=O)(=O)N2)ccnc2ncccc12 c1(C(=O)NC(C2(O)CN(C(C3ON=C(CC)C3)=O)C2)C)c(F)cc(Cl)cc1F C1(C(N2CC(OCCC(=O)NCc3c(CC)nn[nH]3)C2)=O)CCOC(C)C1 C1(CNC(CCC(=O)N(C(C)C)C)=O)CCCCN(C(C2(C#N)CCCO2)=O)C1 N1(C(C(=O)C2CC2)=O)CCN(c2ccc(I)cn2)CC1 C1(CC#C)(C(=O)NCC(C2(O)CN(C(=O)Cn3cnnc3)C2)F)CCCC1 c1(C(=O)NC(CN(C(=O)CC2(C)CC2(Cl)Cl)C)(C)C)ccc(NC(N)=O)cc1F Cc1nnnn1CC(=O)N(CCNC(=O)CN1CCCC1C)CCN(C)C c1(-c2cn(CC3N(C(C(C)NC(N)=O)=O)CC=C3)nn2)ccc(F)cc1F N1(C(C(c2cccnc2)C)=O)CCC2(C1)CN(C(C1CC(S(C)(=O)=O)C1)=O)C2 N1(C(CCCC(=O)NCC)=O)CCC2(NC(=O)C=CS(C)(=O)=O)CCCC12 c1(C(=O)OC)cc(Br)c(F)cc1NC(C1C2CC1N(c1ccnc(OC)n1)C2)=O Cc1cc(=O)oc(C)c1C(N1CCC(O)C(NC(c2ccncc2Br)=O)C1)=O C1(C(=O)NC2C(C(=O)NC(C#CC)(C)C)CCC=C2)CN2CCN1CC2 CCCC(C)(CCCNC(=O)NCC(C1CCCCC1)O)C1OCCO1 C1(CNC(C(C)S(C)(=O)=O)=O)CC2(CCC2)CN1C(c1ccoc1Br)=O C1(NC(c2cc(C(C)=O)oc2)=O)COCCN(C(=O)C(C)(C)c2cnco2)C1 CC(O)(CC(F)(F)F)C(=O)NC1CC2(C1)CN(C(=O)CC1CCC1)C2 O=C(CS(=O)CCC(F)(F)F)NCC1C2CN(C(c3cc[nH]c(=N)c3)=O)CC12 C(=O)(C(=O)C(C)(C)C)NC1CC2(C(C(=O)Nc3c(COC)cccc3)C2)C1 c1(C(N2CC(CC)N(C(=O)CCc3nccn3C)CC2)=O)c(C)nc(O)nc1C C(CCN(C)C)(C(=O)NC1CN(C2CC2)C1)NC(CCNC(=O)NC)=O CCCC(C)CCCC(=O)N(C1CCN(C(C2CCOCC2)=O)C1)CCO C1(C(=O)NCCCN(C(=O)C(C)CF)C(C)C)COc2c(F)cc(F)cc2C1 N1(C(C(N2CCOCC2)C)=O)CCC2(CC1)CN(C(C13CC1COC3(C)C)=O)C2 c1(CC(=O)NCC2CC(NC(c3c(CC)[nH]cc3)=O)C2)cccc(C)c1C C1(C2CCCCC2)CC1.CC(C)C(C)C(CNC(=O)C1CC1)NC(=O)OC(C)(C)C C1(S(=O)(=O)c2ccccc2)(C(=O)NCC(C)NC(c2cccc(CO)n2)=O)CC1 N1(C(c2cc(CC)ncc2)=O)CCC(NC(c2cc(=O)n(C)o2)=O)C(F)C1 N1(C(CCCCN(C)C(C23CCCC2C3)=O)=O)CCCC(C2(C)CC2)C1 N(C(=NCCOCC(F)(F)F)NC1CCCC(C)C1)CC1CCC(=C)CC1 C(=O)(C(O)C(C(C)C)OC)N(C(C(=O)N(C1CCCC1)CC)C)C1CC1 N1(C(C(CNC(C2COC(=O)N2)=O)OC)=O)CC2CCC2(C)C1 N1(Cc2ccc(C(=O)OC)cc2)CC(O)Cc2cc(Br)ccc21 N(C(=NCCC(=O)N1CCCCC1)NC1(Cc2ccccc2)CC1)CC(CCC)C N1(c2ccc(OCC)cc2O)C(=O)NC(CC)C2=C1C(C)NC2=O C1(NC(CC2CCCC(C)(C)C2)=O)C2CC3CN(C(=O)Cn4cccn4)C1C3C2 Cc1cc(F)c(Br)cc1NC(C1CC2CC2N1C(c1cc(F)ccc1Cl)=O)=O c1(N(C(C)=O)CC)cc2cc(OC(c3ccccc3[N+](=O)[O-])=O)ccc2[nH]1 N1(C(CCCCOC)=O)CCC(CNC(=O)Cc2cc(OC)cc(F)c2)C(C)C1 N1(C(CC(C)N(C)C)=O)CCC2(NC(=O)CCc3ccsc3)CCCC12 C1(C(N(CCCCC=C)C)=O)CCCN(C(=O)CCCNC(=O)OC)C1 C1(N(C2CCS(=O)C2)CC(=O)OC)CCCN(C(=O)OC(C)(C)C)CC1 C1(F)(CNC(=O)CCOCC(F)F)CCC(NC(c2ccnc(O)c2)=O)C1 CCC(C)C(C(=O)N(CCCN(C)C(c1cc2n(n1)CCO2)=O)C)N(C)C c1(CCNC(=O)NC(c2cc3ccccc3o2)C)c[nH]c2c(Br)cccc12 N1(C(C2CN(C(=O)NC)C2)=O)CCCC(C)(N(C(C2CCCC(C)(C)C2)=O)C2CC2)C1 Cc1cn(C)nc1CNC(=O)COC(C)(C)CNC(C1CCCC1F)=O c1(NC(CSc2nc(C)[nH]n2)=O)ccc(F)c(CO)c1 C1(C(=O)NC(CNC(c2cnc(C)o2)=O)(C)C)C2CCN(CC2)S1(=O)=O Cn1cc(C(N)=O)cc1C(=O)NC1CC(n2cc(C3CCCC(F)C3)nn2)C1 C1(CNC(C(CC=C)C)=O)C(O)C(O)CN1C(=O)CC1CC2(CCC2)C1 c1(OC)ccc(C(=O)CN(C2CC2(C)C)CC#N)c(OC)c1 CCCC(C(=O)N1CCN(C(=O)C(C)(C)C(C)C)CC1CF)S(N)(=O)=O C1(C(=O)OC(C)(C)C)CC2(CCC2)CO1.C12CCC(CC1)CC(O)C(=O)N2 c1(-c2ccc(CNC(COc3c(CC)cccc3)=O)o2)nnc2cnccn12 C1(C)(C(N(CCC)CCNC(=O)C=CS(C)=O)=O)Cc2ccccc2C1 C(C)(CCC(=O)NCCN(C(c1c(C2CCCC2)noc1C)=O)C1CC1)OC c1(CC)ccc(F)c(C(=O)NCC(CC)NC(=O)C(CC)N(C)C)c1 C(CCCC(=O)NC1(C(=O)N(CC(C2CCCC2)O)C)CCSC1)OC c1(CC)nc(=N)[nH]c(=NCC2CCC3(CCC3)C2NC(=O)CCc2cscn2)[nH]1 C1(CC#C)(C(=O)NC2CC(NC(c3cc(C(N)=O)co3)=O)C2)CCCOC1 c12ccc(c(N3CCNC3=O)c1)S(=O)(=O)O2.c1(OC)ccc(O)nn1 N1(C(C(=O)N(CCCNC(c2c(C)coc2)=O)C)C)CCN(C)CC1 CN1CCC12CN(C(=O)C(c1cn(C)nn1)NC(c1coc(C3CC3)c1)=O)C2 C1(C(=O)NCCCC(C)(C)NC(C(CN(CC)CC)F)=O)CCn2nncc2C1 CC1c2ccccc2OC1C(=O)NCCCCN(CCCNC(C1CC1F)=O)C c1(C(C(N2CCC(F)(C(=O)OC)C2)=O)N(C2COC2)C)cc(C#N)n(C)c1 Cc1cc(F)cc(C(N2C(CNC(c3ccncn3)=O)CC3COCC23)=O)c1N C(c1ccc(C(N)=O)o1)=CC(=O)NCC(O)CNC(=O)C=C1CCSCC1 Cc1ncc(CNC(C2(NC(=O)C(C)C3CCCC3)CCSC2)=O)n1C C1(NC(C2(O)C(OCC)COCC2)=O)CC(OC)C12CCOCC2 c1(OC)ccccc1SCNC(=O)C(c1cnc(N(C)C)cn1)N1CCC(C)C1 C#CC1(C(N2CC(C(F)(F)F)C(CNC(=O)CCC)C2)=O)CC(=O)C1 c1(C(N(CCNC(Cc2c(C)ocn2)=O)C)=O)c(-c2ccccc2Cl)noc1C c1(C(=O)NCCC(C)NC(c2csc([N+](=O)[O-])c2)=O)cn2ccc(CO)cc2n1 N1(C(CSc2cc(C)no2)=O)CCC(OC2CN(C(=O)C=C3CC3)C2)CC1 c1(C(N2CCC(NC(C(CCCC)CC)=O)C23CC3)=O)cc(C)nc2ccnn12 N1(c2n(C)ncc2[N+](=O)[O-])CC2CCC(C1)N2C(=O)Cn1ccc(O)nc1=O C1(C(=O)NC2CCN(C(CCC(C)OC)=O)C(C)C2)CCn2ncnc2C1 C(=O)(C(CC(C)C)NC(C)(C)C)NC(C(c1ncc(C)n1C)N(CCCF)C)=O CCCCC(C)N=c1[nH]c(=NCCC2CCN(C(C)=O)C2)[nH]c2c1CCCCC2 CCC(C)(C)CC(=O)NC1(c2nnnn2CCC2CC2)CCC2CC12 C(=O)(C1=COCCO1)NC1(CC=C)CCN(C(C2CCC(CO)CC2)=O)C1 C1(C(=O)OC)CCC(C(=O)NCC(O)CNC(=O)CC2CCCCC2O)CC1 CC#CCCCC(=O)NC1CCC(C)N(C(=O)CCn2cnccc2=O)C1 CC1=NOC(C(N2CCC(CC(=O)NC3CC3(C)C(F)F)C2)=O)C1 CCC(C)(C(=O)N1CC=CC(C(=O)NC(C)CSC(F)F)C1)OC CC(C(F)C(=O)NCCCCCCNC(c1ncc2[nH]ncc2n1)=O)C(F)(F)F CC(C)CC(CC(=O)NCC1(C2(O)CCC2)CC1)NC(=O)CC1CC(=O)NC1=O c1(C)ccccc1C(=O)NC1COCC1OC.C1(C)(CC=O)CCN1OC N1(C(c2cc(C#N)on2)=O)CC(NC(=O)CC2CC2(Cl)Cl)CC(F)C1 Cc1cc(NC(c2csc(COC(C)C)n2)=O)c(C)s1.C12CC(C1)CNC2=O c1(C(=O)NC(C2CCOC2=O)CC)ccc2nnnn2c1 N1(C(C2CC(C)C2)=O)CCC2(CCCCN(C(C34CCC(C)(CC3)OC4)=O)C2)C1 C1(CNC(CC(CCC)O)=O)CCC(C)(C)CN1C(=O)CC1(O)CCOCC1 c1(C(=O)NC(CC)CNC(=O)C2=CCCS2)c(C)n(C)n(C2CCCCC2)c1=O C#CCCCCN=C(NC(C)Cc1ccsc1)NC1CCOCC1 C(N=c1[nH]cncc1I)C1C(C)CCCN1C(=O)CC1CCC2CC2C1 C(N=c1[nH]c2c(c(=NCCNC(=O)C(C)C)[nH]1)CCCCC2)c1cnc(C)[nH]1 c1(C(=O)NCC(CC=C)NC(c2nn[nH]c2Cl)=O)cc2cc(F)cc(F)c2[nH]1 N1(C(c2cc(C)oc2)=O)CCC(N(CCO)Cc2oc(CO)nc2C)CC1 CCC(C)(CCNC(=O)C(O)C(C)C)NC(C1CCCS1(=O)=O)=O C1(C)(NC(C(C2CCOCC2)C)=O)CCCCC1C(=O)NC1CCCC1CF c1(C(N2CC(CCNC(C(C)CC(N)=O)=O)OCCC2)=O)cccc(C#N)c1F N1(C(=O)C=Cc2ccccn2)CCC2CCCC12C(N1CCC2(CCC2)CC1)=O C1(CNC(c2c(C(C)C)nns2)=O)CC2(CC2)CN1C(=O)CC(O)C(C)C c1(NC(C2(C)CCCCC2)c2n(CC)nnn2)ccc2c(c1)OCCOC(=O)N2 c1(CCNC(C(C=CC)O)=O)ncc(-c2cn(C3COCC3OC)nn2)cc1C C1(C(=O)NCc2nc(CNC(C(CSC)C)=O)sc2)CCC2(CCC2)CC1 C1(F)(C(N(CCCCO)C(C)C)=O)CCN(C(=O)C(C)N=[N+]=[N-])C1 N1(CN(C)CC2OCCOC2(C)C)C(=O)CCN(CCC=Cc2ccccc2)C1=O C12(NC(c3nnc(C)s3)=O)CCCC1N(C(c1cc(C(C)C)no1)=O)CC2 c1(OCC)cccc(CNC(=O)C(C)(C)C)c1.C12CC1C(=O)O2 c1(C(=O)NC(C(=O)NC(C)(C)C)(C)C)cccc(OCC(F)(F)F)c1 c1(C(N(CCN(C(=O)C=Cc2nc(C)cs2)CC)CC)=O)cccc2nn[nH]c12 c1(-c2onc(-c3cccc(C)c3)n2)cc2scc(Cl)c2[nH]1 N1(C(C(C)(C)S(C)(=O)=O)=O)CCC2CN(C(C3CCSC3)=O)CC2CC1 C(=O)(C(C)CCC(C)(C)C)N1CCC(NC(C=C(CC)C)=O)CC1 CCCCCCCCOCC(=O)NCC1CCCC1NC(c1cnc(S)n1C)=O C1(C2CCCO2)(C(=O)NCC(CNC(COc2cn(C)nc2)=O)O)CCCO1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(O)(C(C)NC(c2nc(C)n(C)n2)=O)C1 C1(C)(CC)C=C(C(=O)N(CCN(C(=O)C(C)(O)C2CC2)C)C(C)C)C1 C1(C(=O)NCC(c2cccnc2)O)(NC(C(C)O)=O)CCc2cc(Br)ccc2C1 Cc1noc(C)c1S(=O)(=O)NC(c1ccsc1)CNC(C1(C(F)F)CCOCC1)=O c1(OC(C)C)c(C(=O)NCC2CCN2C(=O)CC(C)O)cccc1N c1(C(=O)NCC2CCC(NC(C(C3CCC3)OCC)=O)C2)ncc(C)nc1OC N1(C(C2(CC=C)COC2)=O)CC(C2CCCN(C(c3cc(C)ccc3F)=O)C2)C1 C12(CNC(CCCSC)=O)COC(CNC(C3CCC(C)(C)O3)=O)(C1)C2 C1(C)(C(=O)NCC(c2ccccc2)N(C)C(c2nccs2)=O)C=CCC1 Cc1nc(CO)ncc1C(=O)NC(C)CC(C)NC(=O)CCC(C)O C1(C(=O)NCCCCCCC)CCCC(NC(C23CC(C(=O)OC)(C2)C3)=O)CC1 CC1CCC(C(N2CC(NC(=O)Cn3cc(Cl)cn3)C3CC23)=O)CC1 N1(C(c2ccn(C(C)C)n2)=O)CC2COCCC2(NC(=O)CC2CC(F)(F)C2)C1 c1(CC(N2CCN(C3CN(C(CCC=C(C)C)=O)C3)CC2)=O)cn2ccsc2n1 N1(C(C=C(CC)CC)=O)CCN(C(=O)Cn2cc(C3CC3)cn2)C2CC12 c1(C(=O)NCC2C(NC(CC)=O)CCC2)ccc(=O)n(C)n1 C1(CNC(c2nc(C)sc2)=O)CC2CN(C(=O)C(C)OC3CCCCCC3)CC12 CCCC(F)(F)C(=O)N1CCOCC(C(=O)NC(c2nn[nH]n2)CC)C1 C1(C(=O)NCC(CNC(c2nc(C)oc2C)=O)F)CC(C)OC(C)C1 N1(C(C=CCC)=O)CCC(C(=O)N(C)Cc2cccc(C)n2)(OC)C1 C1(SCC(C2CCCOC2)OC)CC2OC(C)(C)OC2C1 C1(CC(=O)N(C(=O)Cc2csc(NC=O)n2)CC)C(=O)NN=C1C c1(C(N2CCCC2c2ccnn2CC)C(=O)NCC(=C)C)cncc(C(=C)C)c1 c1(C(N2CCC(N3CCN(C(C(C)(C)C)=O)CC3)CC2)=O)cc(Cl)c(Cl)cc1F CC1CC=C(C(=O)NC(C)CCCCNC(=O)C2=CCCC2(C)C)CC1 c1(CCC(=O)NC(C(N2CC(OCC)C2)=O)C2CCCC2)ccccc1 c1(C(N(C)CC2N(C(C=CCCC)=O)CCOC2)=O)c(Br)ccc2c1OCO2 c1(C(=O)NCC(C)(C)OCC(=O)NC(CCC)CO)cc(N)cc(F)c1 c1(CC(C(=O)OCC)NC(c2ccc(C3CC3)s2)=O)c[nH]c2c(C)cccc12 C1(C(N(CCCNC(c2cc[nH]n2)=O)CCO)=O)OCCO1 CC1CC(C(=O)NC2CC3C(NC(C4CC(=C5CCC5)C4)=O)C3C2)CC(C)C1 C(N=c1[nH]c(=NC(C)C2CCC2)[nH]c2c(F)cccc12)c1c(C)c(F)c(F)cc1 c1(C(=O)NCCCC(C)NC(C2CCC(C)(CC)O2)=O)cc(C)nc(N(C)C)n1 C(=O)(C(C)C(F)(F)F)NC(C1CCCCC1)CNC(Cc1nc(C)sc1)=O C1(NC(C(C)Sc2ccccn2)=O)CCN(c2ccncc2C#N)CC1(C)C Cc1ccc(CC(=O)NC23CC(NC(=O)C(F)C(C)(C)O)(C2)C3)cc1C N1(C(C=Cc2nc(C)sc2)=O)CCC(CNC(c2cc(C(F)F)[nH]n2)=O)CC1C c1(C(=O)NC2(C3N(C(CCC=CC)=O)CCC3)CC2)cn(C)c(C)n1 N1(C(C(CC)C)=O)CC(C2CCCCN(C(c3nc(Cl)sc3C)=O)C2)C1 C1(CNC(c2c(C(N)=O)nccn2)=O)CCCC12CCN(C(C1CC1F)=O)CC2 N1(C(C(CC(N)=O)O)=O)CCC2CN(C(=O)CSC(F)(F)F)C2C1 C12(C(=O)NCC3(CN(C(C(CC)(C)O)=O)C)CC3)CCOC(C)(C1)C2 CCC(CC(=O)N1CCOCC(NC(c2cc(C(C)C)nnc2C)=O)C1)C(F)F C#CCCCC(C)C(=O)N1CC2CC(C1)N(C(=O)CN1CCCC1=O)C2 c1(OC)cc(C(C(=O)NC2CCOC2)N2CCC2C2CCC2)ccc1Br C12(C(N(C)Cc3cnco3)=O)CC1CCN2C(=O)CCC1(N(C)C)CCCC1 c1(C(=O)NC(CC=C)CNC(C2CCN(C)C2)=O)ccccc1CNCCO N1(C(C2(C(=O)OCC)CC2)=O)CCC(CNc2ncc(CC)cn2)C(C)C1 c1(C(=O)NCCCCCNC(CSC(C)(C)C)=O)cc2cnccc2[nH]1 N1(CC(C)(C)NC(C(c2n(C)ncc2)CO)=O)CCN(C(=O)C(=O)N(C)C)CC1 N1(C(COc2cc(C)on2)=O)CCCN(C(C2CC2c2ccncc2)=O)CCC1 Cc1cc(CO)oc1C(=O)NCC1CN(C(=O)Cc2ccco2)CC1C Cc1cc(C)c(C(=O)NCc2ocnc2C(=O)N(C2CC(F)(F)C2)C)o1 N#Cc1cccc(CN2CCC(F)(C(N3CCC(O)C(O)C3)=O)C2)c1Cl c1(C(=O)NCC2CC(O)(CNC(C3CC3F)=O)C2)cc(Cl)ccc1Br c1(C(=O)NCCN(C(=O)CN(C)C(N)=O)CCC)cc2c(cc1N)OCO2 C1(CNC(c2c(OC)ccs2)=O)CC2CN(C(c3cnc(C)[nH]3)=O)CC12 CCC(CCCC(=O)NCC(=O)OC)NC(c1ccsn1)=O c1(C(=O)NCCNC(C2CCC(=O)C2)=O)ncncc1Br N1(c2ccc(C#N)cn2)CCC(F)(F)C(C(=O)NCCN2C(=O)CNC2=O)C1 O=C(CC1=CCN(C(=O)CC2(O)CCCC2)CC1)N(CCCO)CCO c1(N2CCC3CN(Cc4c(C)cc(O)cc4C)CC32)ncnc2ccccc12 CCC(C)C(=O)C(=O)NCC(O)CC(=O)N1CCN(CC)CC1 C=CCC(Cc1ccccc1)C(=O)OCCC(=O)NC(=O)Nc1ccccc1 CCC(C)(C)CC(=O)NCCCCN(C(=O)C(C)OCc1ccc(F)cc1)C C(CCCCCNC(=O)Cc1ccsc1)NC(C1(NC(C)=O)CCC1)=O CCC(C)(C)C(O)C(=O)NCCCNC(c1ccc(N(C)C)nc1)=O c1(-c2ccc(C(N3CCN(CC(F)(F)CO)CC3)=O)s2)cc(Cl)cc(Cl)c1 C1(CC#C)(C(=O)NCCOC2CN(C(c3nc(Cl)cs3)=O)C2)CC=CCC1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCC2(CN(C(C3(SC)CC3)=O)C2)CC1 c1(NC(C2CN(C(c3scc(C)c3)=O)C2)=O)n[nH]c2ccc(Cl)cc12 Cc1nc[nH]c1CC(=O)NC(C)(CNC(c1ccoc1CC(N)=O)=O)CO Cc1cccc(CC(=O)NCC2CCN2C(=O)C(C)SC(C)C)c1Br C1(NC(c2[nH]cc(C)c2)=O)CN(C(=O)CSc2nncs2)CC(C)(C)C1 c1(-c2cn(CC(=O)NC3(C#N)CCC3)nn2)cccc(C2CCCC2)c1 N1(C(C(CC)F)=O)CCOC(CCCNC(c2coc(-c3ccsc3)c2)=O)C1 c1(-c2ccnc(C)c2F)cn2cc(C(N3Cc4ccc(O)cc4C3)=O)ccc2n1 N1(Cc2c(CCC)cccc2)CC2(CN(C(=O)CCc3scnc3C)CCO2)C1 c1(OC)cc(C)cc(CN2CCC3(CN(C(=O)Cc4c(C)nn(C)c4C)C3)C2)c1O C(=O)(CC(C)(C)C(C)=O)NC1(C(=O)NC2CC3CC(OC)C3C2)CC(CO)C1 N1(C(C(C)N2N3CCCC3C2=O)=O)CCC=C(F)C1.CCOC N1(CC2CS(=O)(=O)CC2O)CC2CC3(CCCCN3)C2C1 C1(O)(CN(C(C(CN(C)C)N(C)C)=O)C)CCN(C(C2(N(C)C)CC2)=O)C1 C(CC(C(=O)NCC1=NOCC1)N(C)C)N(C)C C(=O)(C(C)(C)CC(=O)OC)NCC=CCNC(C1CC(C(=O)NC)NC(=O)C1)=O c1(OCC)cnc(C(=O)NC(C)C(C)NC(c2cc(C3CC3)ccn2)=O)c(Cl)c1 Cc1cc(C(N2CCCC3C2CCCN3N=O)=O)c2ccc(C(F)(F)F)cc2n1 N1(C(c2c(C)csc2)=O)CCC(C)(CC(=O)NCc2cccc(Cl)n2)C1 C1(C)(C(N(CCCCCC)CCO)=O)CC12CCN(c1ncccc1C#N)CC2 N1(C(CCCOC)=O)CCC2(CC2)CC1C(=O)NCC1(C)C=CCCC1 C1(NC(c2snc(OC)c2Br)=O)CCC2CCN(C(C3CC3C)=O)C1C2 C1(C(=O)NC(c2cccc(N(C)C)c2)C)CC2(C1)OCCO2 C1(C(C)C)CN(C(=O)C(C(C)O)N(C)C)CCN1C(=O)C(C)OCC1CCCO1 C1(C(F)(F)C(=O)N2CCC(CCN(C(=O)C3CC3)C3CC3)C2)(OC)CCCC1 C(CN(C)C(C12CCC(CC1)C2)=O)(CO)(CO)NC(COCCCC(C)C)=O CC1CC(C(N2CCC(CN(C(=O)C3=CCCOC3)C)CC2)=O)Cc2nn[nH]c21 N1(N2C(C=O)CC2)CC(C2(OC3C(CC)CCCC3)CC2)C1.C(=O)CCCC#N C(=O)(C1OCCc2cc(O)ccc21)N1C2CC(NC(c3n[nH]cc3Cl)=O)C2CC1 Cn1cccc1C(=O)N(C1CC1)CC1CCCN1C(c1csc(C(N)=O)n1)=O C(=O)(C1=CCCOCC1)NCCC1(OC)CN(C(c2nc(C)ccc2F)=O)C1 C(=O)(CCCN=[N+]=[N-])N1C(CCC(=O)NC(C(N)=O)CO)CCC1 C1(C(=O)NCc2c(C(=O)NCC(C(C)C)(C)O)cco2)CC2C(C1)C2(C)C c1(C(N2CCN(C(CCSCC)=O)CC2CO)=O)ccc2[nH]nc(Cl)c2c1 CC1(C(=O)NC2CC(CNC(=O)C=CC(F)(F)F)C2)CCCS1(=O)=O CCC(C)CCC(=O)N1CCC(N(C(=O)CCc2ccc(C(F)F)cc2)C)C1 CCC(C)(O)C(=O)NCCCCCCNC(c1nnn(C)n1)=O c1(OC)n[nH]cc1C(=O)NC1CC(CCNC(=O)CC2CC2(Cl)Cl)C1 c1(OCCOC)ccc(C(=O)NCC2CCCCN2C(=O)CCC(C)SC)nn1 Cc1nccnc1C(N1CCOCC1c1cn(Cc2ccc(F)cn2)nn1)=O c1(C(=O)NC2CC(NC(C(C)CN(C)C)=O)C2)ccnc2c(F)cccc12 C(=O)(CC(CC)C(C)C)N1CCC(CCNC(c2cncc(C#C)c2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC2(CNC(=O)CCc3ccncc3)CCC1C2 C1(CNC(CCCN(C)C)=O)(NC(C2CCCN2C)=O)CC(F)(F)C1 C1(CNC(c2n[nH]c3c2CCCCC3)=O)CCCC2(CN(C(=O)CCF)C2)O1 Cn1cnc2nc(NCC(Cl)=C)nc(N3C4C=CCC3CC4)c12.N N1(C(C2CCC(=C)CC2)=O)CCC2CN(C(C3CSCCS3)=O)CC12 c1(CNC(CNC=O)=O)ccc(C(=O)NCc2ccns2)nc1 C1(C(C)C)N(C(=O)C(=O)N(N2CCOC(CC(F)(F)F)C2)C)CC12CCC2 c1(C(=O)NCC(C)N(C(C(C)OCCCC)=O)C)ccnc2c1CCO2 C1(CNC(c2[nH]nc3cnccc23)=O)CN(C(=O)CC2CCCC2)C2(CCC2)C1 n1(C2(C(=O)OC)CCOCC2)cc(C#N)c(=NC(=O)c2cc(Br)c(F)cc2Br)[nH]1 c1(C(N2CC(F)(CNC(C3C(C)CN(C)C3)=O)C2)=O)nccc2ncccc12 C(N=c1[nH]c(N2CCCC(C(C)(C)C)C2)nc2c1COCC2)c1n(CC)ccn1 c1(C(=O)NCC(CO)NC(C(c2cn(CC)nc2)(F)F)=O)cc(C)c(C)s1 C1(NC(c2n(C)cnc2)=O)CN(C(c2cscc2C#N)=O)CC12CCOCC2 C1(C(=O)NCc2occ(C(=O)NCC(C)C3CCC3)c2)C2CCC(=O)C12 CC(C(=O)NC1CCN(Cc2csc(C(C)(C)C)n2)C(C)C1)C(C)(C)C c1(OC)cc(C(N2CC(CC(C)NC(=O)C(CC)Oc3ccccc3)C2)=O)sn1 c1(C(=O)NCC(CN(C)C(C2CCC2C(N)=O)=O)(C)C)cc(C(F)F)ccc1F Cc1ccc(C(C)C)c(C(=O)NCCCCNC(=O)C(F)n2cccn2)c1 c1(OC)ccc(CC(=O)NCC2CC(O)CN2C(=O)CC2CC3CC3C2)cc1F O=C(C#CC1CCCOC1)NC1(C2CN(C(C3CCCO3)=O)C2)CC1 CN1CCN(C(=O)CCF)C(CNC(C2CC(F)(F)C2(C)C)=O)C1 CC1CC1(C(N1CC(C(=O)N(C)C)C1)=O)NC(=O)CC1CCOC1 CCCCC(CNC(C1(O)CCSC1)=O)NC(=O)C(C)COC(c1ccco1)=O C(C(C(=O)N1CCCCC1CCCO)C(C)(C)C)NC(C(C)=C1CC1)=O N1(C(C2CCCN(C(c3ccnc(O)c3)=O)C2)=O)CCC(C2=NOCC2)C1 c1(OC)ccc(F)c(C(=O)NCC2CC2NC(c2ncc(Br)cn2)=O)c1 C1(C(C)C)(NC(CCOCCN(C(CSC)=O)C)=O)CCCO1 C12(C(=O)NCC3(F)CCC(NC(c4ccc(C(C)C)s4)=O)C3)CCC(F)(CC1)C2 c1(C(=O)NCc2cccc(CNC(C(CCC#C)O)=O)c2)cc(S(N)(=O)=O)c[nH]1 C1(C(=O)NCC2(NC(CCNC(=O)OC)=O)CCOC2)OCCC1(C)C C12(C(=O)O)CC1CCCN2C(c1cccc(-c2cn(-c3cncc(F)c3)nn2)c1)=O CC1(NC(=O)CN2CCCCC2)CCN(C(=O)Cn2ccc(C3CC3)n2)C1 C1(C(=O)NCc2cscc2C)(CC)CCN(C(=O)CCC2CCCC2)CC1 c1(C(=O)NC2CCC(COC)C2)cc(CNC(=O)C(O)C(C)C)nn1C c1(OC)ccc(CC(=O)N(CC(C)N(C(=O)C=C2CCSCC2)C)C)cc1O CCC(CCOC)C(=O)N(C)CC1CCN(C(c2occc2F)=O)C1 C1(C(=O)NC(CCNC(c2cncc(C)n2)=O)C)CC2(CCOCC2)C1 C1(C(=O)NC2COCCN(C(C(CCC)C(C)C)=O)C2)CNC(=O)CC12CCC2 c1(CC)cnn2ccc(C(N3CC4CCN(C(=O)C(F)=C5CCC5)C4C3)=O)nc12 Cc1cc(C)c(C(N2CCCN(c3nc(C(C)C)ncc3Br)CC2)=O)cn1 C1(CNC(Cc2ccc(SC)cc2)=O)CCCCN(C(=O)CC2CC(C)(C)C2)C1 c1(OC)cnc(C(=O)NCC(O)CNC(=O)CC2(C)CCCC2)nc1 C1(C(N(C)CCn2ccnc2)=O)CCN(C(=O)C(=O)NCC(F)F)C1C1CC1 c1(CSC)noc(CN2CCC(NC(=O)N(S(C)(=O)=O)C)C2)n1 Cc1conc1CC(=O)NC(C)(CNC(=O)Cn1cnnc1)C1CC1 CCCCC(C(=O)N1CCC(C(=O)NCC(CC)CC)C1(C)C)C(C)C Fc1ccccc1-c1cscc1CNc1nc(C2CCC2)no1 c1(CNC(=O)NCc2n(C)cc(Br)c2Br)c(Br)c2ccccc2n1C CCCC(C)(CCC)C(=O)N1CC(C2CC2C(=O)NCC(C)C#N)C1 N1(C(=O)C=CC2CC2)CCC2(C1)CN(C(c1cc3n(n1)CC(F)C3)=O)C2 N1(C(C2C(C(C)C)CCC2)=O)CCC(CNC(c2coc(Cl)c2)=O)CC1 c1(OCC(=O)N(CCC(C)NC(=O)CN2CSCC2=O)C)cccc(CO)c1 c1(C(N(CC(CNC(CCC=CCC=C)=O)O)C)=O)cc(O)nc(CC)n1 C1(NC(=O)CCCCCF)CC12CCC(NC(C1(C3CCOCC3)CC1)=O)CC2 Cc1cc(-c2cc(O)ncc2Br)cc(C)c1F C(=O)(CCCC(=O)NC1C2CCC1N(C(=O)C(C)(C)c1cccs1)C2)N(C)C c1(CC(=O)Nc2ccsn2)cccc2c1OCO2.C1(C2CCC2)C(=O)N1 c1(C2C(C(N(C(C)C)CCCCCN3CCOC3=O)=O)C2)ccc(N)cc1 C1(CNC(CCC(C)c2ccccc2)=O)N(C(=O)Cc2cc[nH]n2)CCC1(C)C N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC1(C)CCN(C(c2cncc(CO)c2)=O)C1 Cc1c(C#N)sc2ccc(NC3C4CCC(C4)N3C(=O)OC(C)(C)C)cc12 N1(C(C=C(CC)C)=O)CCN(C(C2CCN(C)C2)=O)CC1c1cccc(Cl)c1 CC(c1ccccc1)=CC(=O)NCC(C)NC(C1CCCO1)=O N1(C(C2ON=C(C(C)C)C2)=O)CCn2nc(CNC(=O)Cc3cncs3)cc2C1 c1(N(C2CNCC2C#N)C(c2ccc(C)nc2F)=O)ncc2[nH]cc(I)c2n1 C(=O)(C(CC(N)=O)NC(=O)CCc1ccc(Br)c(C)c1)OCC=C C1(NC(c2cnn(CC)c2C)=O)CCN(C(=O)CC2(C3CC3)CC2)CC1F c1(C(=O)NCC(N2CCN(C(CC(C)OC)=O)CC2)C)cccc2c(C)n[nH]c12 C(=O)(CC(C(F)(F)F)NC(C1CC2(CCC2)C1)=O)N(C(c1cc(C)on1)C)C c1(C2C(C)C2)cn(C)nc1NC(C1CC(Cn2cc(C3(C4CC4)CC3)nn2)C1)=O c1(C(N(C2CCCC2)CCCC)=O)[nH]ccc1CNC(c1coc(CO)c1)=O C(=O)(C1Cc2ccccc21)NC(CNC(C(C)C1CCC1)=O)(C)Cn1cccn1 C(CCCCNC(=O)COCCOCc1ccccn1)NC(CN1CC(C)C1)=O c1(C(N2C(C)CC(NC(COCCSC)=O)C2)=O)nccn2ccnc12 N1(C(c2ccc(CSCCC)o2)=O)CCOCC1CNC(C1CCC1(C)C)=O C1(CC=C)N(C(=O)CCn2cc(-c3cc(N)n(C)n3)nn2)CCC1(C)C N1(C(CCN(C)CC)=O)CCCC2(C1)CN(C(C1CCCN1C1CC1)=O)C2 c1(CC)ccc(C(=O)NCC(C)N(C(=O)Cc2ccon2)C)c(C)n1 c1(C(=O)NC2C(NC(C(C)(C3CCOCC3)OC)=O)COC2)n[nH]c(C)c1Cl c1(C(N2C(C(=O)NC(c3cccnc3)C(C)C)COCC2)=O)ccc([N+](=O)[O-])nc1 N1(C(c2nc(CC)sc2N)=O)CCC(NC(c2ccc(Cl)[nH]2)=O)C(C(C)C)C1 c1(NC(C(N)CC2CCS(=O)(=O)C2)=O)ccc2c(c1)CCC2N CC1CCN(C(c2cnccc2Cl)=O)CC1NC(C1(C(F)(F)F)CCC1)=O C1(NC(CC(C)SC)=O)CCN(CCC2CC3CCC2C3)CC1 c1(C(=O)NCC2N(C(C3N(C=O)CCC3)=O)CCC2)ccc2nnnn2c1 N1(C(=O)C=C(C)COC)CC=CC(OOC(CN(C)CC)C2CCC2)C1 c1(OCC)ccccc1OCCC(N1CC2CC2(NC(c2cnn(C)n2)=O)C1)=O N1(C(C(c2ccc(OC)cc2)=O)=O)CCN(C(C2CC(C)C2)=O)C2COCC12 N1(C(c2cc(OC)c(-c3nnc(C)o3)cc2)=O)CCC2CCCC2C1 N1(C(CN(C(COC)=O)C)=O)CCN(C(c2[nH]cnc2C)=O)C2CCCCC2C1 C1(C(=O)NC(CCC=C)C(C)C)CCN(C(=O)CC(C)C=C)CC1 c1(CC)ccc(C(=O)NC(C)C(=O)N2CC(c3nncs3)C2)o1 CC(C)(CCF)C(=O)N1CCC(CCC(F)(F)F)C1 C1(CC(=O)OCC2CC(=O)NCC2)CC2(CCOCC2)CO1 N1(C(C(CC=CC)C)=O)CC2CCC2(CNC(=O)C(C)(C)OCC(F)(F)F)C1 C1(C(=O)NCC(C)C(=O)NCC2COCCN2C)CC(=O)NC(=O)N1 CC(C)CC(C)(CNC(=O)CSC1CCCCO1)NC(=O)C=Cc1c[nH]cn1 C=C=CCCC(=O)NC1CCOCC1C(=O)NCC1(C)CC(O)C1 CC1CCc2ncc(C(=O)NC3CC3CNC(c3sccc3C#N)=O)n2C1 C1(N(C(=O)COCCOCCO)C)CCCCN(C(C2CCS(=O)(=O)N2)=O)C1 n1(CC(=O)NC(C(C)NC(C2CCCCC(=O)N2)=O)CO)ncc2ncccc12 C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC12C(CN(C(c3c(C)ncnc3)=O)C1)C2 N1(C(C2C(C(=O)OCC)CC2)=O)CC(NC(=O)Cc2cncnc2)C(C)(C)C1 c1(C(=O)NC2C(C)(C)C(Nc3ccncn3)C2)cn2cc[nH]c(=O)c2n1 C1(NC(C(C)(CO)OC)=O)CCN(C(=O)Cc2cc(C3CC3)no2)CC(C)(C)C1 CC1=NC(C)(CNC(=O)C(=O)NCc2ccccc2NS(C)(=O)=O)CS1 c1(C(N2CC(NC(CCOCC)=O)(CF)C2)=O)cccc2ccnn12 c1(OC)ccc(CC(=O)N(CCCNC(=O)C(F)(F)c2cccnc2)C)cc1O C12(C(=O)NCCCC3CC(C)C3)CCN(C(c3ccn(C(C)C)c3)=O)CCC1C2 C1(C2CC2)(C(N2CC(C(C)NC(CCCCC)=O)OCC2)=O)CC=CC1 C(=O)(C1COc2ccc(Cl)cc21)N(CCCNC(=O)CC1CC(C)(C)OC1=O)C CC(O)CCN=c1[nH]c2c(c(=NCC3(CO)CC34CCOCC4)[nH]1)COC2 C(=O)(C1=CCC2CCC1N2C(=O)CCC1CCOC1)NCCc1c(C)nc[nH]1 C(CCCCCC(=O)NC(C(=O)N(C)C)C(C)C)NC(CCC(=C)Cl)=O CCCCCCC(C)C(=O)NC1CC2CC1N(C(=O)C(=O)NC1CC1)C2 N1(C(C(C)OCCC#C)=O)CCC2(C1)CN(C(c1cc(C(F)F)no1)=O)CCO2 C12(NC(CCCC#CC)=O)CCCC1N(C(C1CN(c3ncc(F)cn3)C1)=O)CC2 CCC(O)C(F)(F)C(=O)N1CCCOC(CCNC(=O)CCN2CCCC2=O)C1 C1(C(=O)NC2CCOCC2NC(c2ccc(C(=O)OC)s2)=O)(OC)CCOCC1 N1(C(CC(=O)OC)=O)CCCCC1CCNC(c1c(C)ccn1C)=O CCC(CC(F)(F)F)C(=O)N(C)CCNC(c1ccc(OC)c(C(C)C)c1)=O C1(C(=O)NC2(C)CC(NC(C(C)NC(CC)=O)=O)C2)CCN(C)C1CC CC(C)C(C(=O)NCC1CCC(NC(c2cncn2C)=O)CC1)NC(N)=O C1(C(N(CC(=O)OC)CC)=O)CCCC2(CC2)C1.c1(SCCC)ncn(C)n1 C(N=c1[nH]c2c(c(=NCCOC(F)F)[nH]1)COC2)c1ccc(SC)nc1 C1(NC(c2c(C)csn2)=O)CCN(C(=O)Cc2ccsn2)C1c1ccccc1 C1(N(C(Cc2c(C)n[nH]c2)=O)C)CN(C(=O)CCC(=O)c2cccs2)CCC1C CC1(C)C(CNC(=O)CC2(c3ccccc3)CC2)CCN1C(=O)Cc1cnns1 C1(n2c(-c3c(C)n(CO)nn3)nc(-c3cccc(CO)c3)n2)CCCC(C)(C)C1 CN1CC2CCCC(CC1=O)N2C(c1cc(Cl)ncc1Cl)C(=O)NC(C)(C)C c1(C(=O)NC(CN(C(c2c(OC)ccc(O)c2)=O)C)C)cccc2c1OCCO2 c1(C(=O)NC(CC)CNC(=O)CC2CC2CC)c(F)ccc(C)c1Cl c1(C(=O)NCC(C)CN(C(=O)CC2CC3(CC3)C2)C)ccc2c(c1)COB2O CC1(C)CCC(O)(CNC(C2(c3ccccc3)CC2)=O)CC1 C1(C(=O)NC2(CNC(=O)C(F)=C3CCC3)CCOC2)CCC1(F)F C1(S(C)(=O)=O)(C(N(C2CCCN(C(=O)C(C)(CC)CC)C2)CC)=O)CCC1 C1(CCNC(c2cnc(OCC)s2)=O)CN(C(=O)CC2(C)CC2)CCS1(=O)=O C1(C(N(C2CN(C(C(CC=CCC)C)=O)C2)CC)=O)CCCC1C1CC1 C1(C(C)C)CC(C)(C)CN1C(=O)C=Cc1ccc(SC)s1.C1(C(=O)OC)CC1C c1(C(N2CC(CNC(CSCC#C)=O)N(C)CC2)=O)c(F)c(F)c(F)c(F)c1F C1(CNC(CC(CC)SC)=O)COCCN(C(c2cnc(NC3CC3)s2)=O)C1 C1(CCCC)CN(C(=O)COCc2nc[nH]n2)CCN1C(c1cnc(C#N)s1)=O [N-]=[N+]=NC1CC(C(=O)NCCOC2CCCC2)N(C(C23CCCC2C3)=O)C1 C1(CC=C)(NC(C2CCCC2C)=O)CCN(C(=O)C(C)NC(=O)CC)CC1 N1(C(c2c(OC)n[nH]c2)=O)CC2(CCOCC2)CC1CNC(C1CC1C(C)C)=O Cc1cc(C(N2CC3CC3(CNC(=O)C=CC3CCOCC3)C2)=O)c(N)cc1F Cc1cc(NCC(=O)NC2CC(NC(=O)CSc3ncc[nH]3)C2)ccc1C(N)=O C(CC(C)C(=O)NC1CC2(C1)CC2C(N1CCC2CC12C)=O)=CCC N1(C(=O)NC(C(=O)NC(CC)C)C)CCC(F)(c2cccnc2)CC1 C1(COC)CN(C(=O)NCCC2(C)CC2(F)F)C1(C)C C1(C(N2CC(C(=O)NC3COCC3C)(CC)C2)=O)CC2(C1)CC(O)C2 C(c1ccc(C)c(Cl)c1)=CC(NOCc1cccc(CNC(C=NOC)=O)c1)=N N1(C(c2ccc(F)cc2Br)C(=O)NCC=C)CC(=O)N(C)CC1CC C1(C(F)(F)F)(NCC(COC)C(C)C)CCC(C)(C)CC1 C12(C(=O)NCC(CNC(c3cn(CC(C)C)nc3)=O)CO)C=CC(C1)OC2 C(c1cccnc1)=CC(=O)NC1CCC(N(C(=O)C=CC(F)(F)F)C)C1 C(=O)(CC(C)C(=O)NC(C)(C)C(=O)NOCC(O)C(C)(C)C)OC c1(C(=O)NCC2(COC)CN(C(C3CCN(C)C3)=O)C2)cnc2sc(C)c(C)n12 Cc1nnc2n1CC(C(=O)N(C)CCNC(=O)COCP(C)(C)=O)C2 c1(CN(C(c2cc(C#N)cs2)C(=O)NCCCF)CC)ccc(S(N)(=O)=O)cc1 N1(C(C(C)Cc2cnco2)=O)CCN(C(c2ccoc2CC(N)=O)=O)CC1CO Cc1ccc(CN=C(NCc2cccs2)NC2CCCC(F)C2)cc1 C1(C(N2CCC(N(C(=O)CCC3CC3(C)C)C)C2)=O)CCC(F)(F)CC1 C1(C(=O)NCC(C(=O)NCC=C)C)CN(C(=O)OC(C)(C)C)CCO1 n1(CC)ccnc1C(=O)NCCCCCNC(=O)C(Cc1ccccc1)C1CC1 C=CCC(C)(CC)C(=O)NCCOCCCNC(c1ccnn1CC1CCC1)=O N1(Cc2ncn(C)c2)CCCCC1NC(=O)CC(C)(C)C c1(C(N2CCC(C(=O)NCc3ccccc3F)C2)=O)ccc2ccsc2c1 C(=O)(C#CC1CCCCC1)NC(C(=O)OCC1CC(OCC)C1)CC(C)CC c1(CC)cc(C(N2CCN(C(=O)COCCOCC)C(C(F)F)C2)=O)ccc1C Cc1ccc(C(=O)NC23CC(C2)N(C(=O)CCC2CCC(O)CC2)C3)cc1N C1(C(=O)NCC2(O)CC(NC(c3c(C)nc(CC)o3)=O)C2)CNC(=O)CC1(C)C C(=O)(CCC(=O)C(C)(C)C)N(CC(=O)NC(C#C)CC1CC1)C1CCC1 c1(C(N2CCC(N(C(=O)CCN3CCCC3)CC)C2)=O)cc(F)cc2nn[nH]c12 Cc1noc(C)c1CNC(c1cc(NC(=O)NC2COCC2C(N)=O)ccn1)=O C1(C(=O)NC2CC(CNC(C(CC)N(CC)CC)=O)C2)CC2OC1C1CC21 N1(C(CNC(=O)Cn2cccn2)=O)CCN(C(=O)CCc2cccc(F)c2)CC1 c1(NCC(CC)(C)OC)[nH]c(=NCCc2cc(C)c(O)c(C)c2)nc2sccc12 N1(C(CCCN(C)C)=O)CCCCC1C1CCCN(C(=O)Cc2n[nH]c(=N)s2)C1 Cc1cccc2cccc(C(=O)NC(C)(CNC(=O)CC3CC(F)C3)CO)c12 C1(NC(C2C(C(C)C)OCC2)=O)CCCCCC1C(=O)N1CCCO1 c1(C(C)(C)C(N2CCN(C(c3ccc(S)cc3)=O)C3CC23)=O)ccc(C#N)nc1 C(c1nc2ccccc2o1)=CC(=O)NC(C)CCN(C(=O)C(CO)C(C)(C)C)C C1(C(=O)NCC2CCN2C(=O)COCCF)CCN(C2CCCCC2)CC1 c1(C(N2CCC(C)(CCNC(C3N(C)C(=O)OC3)=O)C2)=O)ccc2ccoc2c1 c1(NC(CC(C=C)CC)=O)cc(CC(c2cn(CC)nn2)=O)cc(CCO)c1O N1(C(C(C)=C2CCC2)=O)CCC2(CCCN2C(=O)C=Cc2ccco2)C1 CC1C2CCC(C2)C1C(=O)N(CCCn1cc(CCCCCO)nn1)C.O C1(C(N(CCNC(c2cnc(C)[nH]2)=O)C2CC2)=O)Cc2nn[nH]c2C(C)C1 C12CCN(C1)C2=O.c1(C(C)(C)NC(CN(S(CC)(=O)=O)C)=O)cncnc1 N1(C(C(c2ccccc2F)OC)=O)CC2(CCN2C(=O)C(C)(C)C(C)C)C1 N1(C(C2C(C)OCC2)=O)CCC(NC(c2ccc(-n3cnnn3)cc2)=O)C1(C)C C1(C(=O)NC(c2nocc2C(=O)NCCS(C)(=N)=O)C)CC(=O)C1(C)C C(=O)(CCCC(C)(C)C)NC1C(CC)CN(C(c2ncoc2C2CC2)=O)CC1 c1(C(N2C(CNC(=O)Cn3ccnn3)CCC2)=O)ccc(C2CC2)cc1Cl C1(CNCc2c(F)ccc(C)c2Br)(CO)COCC2COCCN12 C1(C(N2CC(NC(=O)C(F)(F)CC3CC3)CC(F)C2)=O)Cc2cc(Cl)ccc2O1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(C)C(CNc2ncc3c(n2)COC3)C1 c1(CC)ncc(NC(=O)C(O)C2CN(C(C3(N(C)C)CC3)=O)C2)cn1 C1(C(C)C)(CNC(c2c(CO)c[nH]n2)=O)CNC(=O)C1.C12(CCC1)CC(=O)NC2 C(=O)(CC(O)CNC(C12CC1CCN2C(=O)CCn1cnc(=N)[nH]1)=O)OC c1(NC(C)=O)ccc(S(=O)(=O)NC(C)CN(C(C)C)C2CC2)c(Br)c1 CC1=NC(C)(CNC(=O)C(Cn2cncn2)NC(c2cccnn2)=O)CS1 C1(CNC(CNC(=O)OC)=O)N(C(C2CCCN2C(C)=O)=O)CCCC1(C)C C12(CNC(COC)=O)CC(CNC(C3(CC(C)C)CCNC3=O)=O)(CO1)C2 C=C(Cl)CC(C(=O)N1CCC(C(C)CC)CC1)NC(c1nn(CC)nc1C)=O c1(C(=O)NC2(C)CCN(CC(N)=O)CC2)nccc(Br)c1C#N N1(C(c2c(C)noc2)=O)CCN(C(C2CCS(=O)CC2)=O)C2(CC2)C1 O=C(C1=CC2C=CC(C1)C2)NC1(CF)CCN(C(=O)C(O)Cc2cnc[nH]2)C1 N1(C(Cc2cc(SC)c(C)cc2)=O)CCC2(CO)CN(C(=O)C=CCF)CC2C1 C(=O)(C(F)CC(C)(C)NC(=O)CCc1ncnn1C)N(CCCSC)C C(C(C)(C(=O)NCCC1CCN(C)C1=O)OC)OC.C1=CCNC1=O C(=O)(C(C)CC1CC1)NC(C(=O)N(CC(=O)OC)CC1CC1)C1CCC1 C1(CN(C(c2[nH]c(COC)nc2C)=O)CC)CCCCN1C(=O)C(CSC)OC C12(NC(c3c(C)cc(F)s3)=O)CCN(C(c3coc(C(C)C)n3)=O)CCC1C2 c1(OC)cnc(C(=O)NCC23CC(CO2)N(C(C2C4COCC24)=O)C3)c(F)c1 CCCC(CC)CCC(=O)NC1CC(F)(CNC(=O)Cc2ccn(C)n2)C1 c1(COC(C2(CN(CCN(CC)CC)C)CC2)CC)c[nH]c2cc(C)ccc12 Cc1cc(C(C)(C)C)oc1C(=O)NNC(=O)NCCC1(C)CCOCC1 C1(CC(N2C(CNC(C3CC3C3CCC3)=O)CCCC2)=O)CCCCC1(F)F c1(C(N2CCC(N(C(=O)Cc3csc(Cl)c3)C)C2)=O)cn(C2CC2)nc1C(F)F C1(CNC(C)=O)CCN(CC(=O)C2CC2c2ccccc2)C1 c1(CCC(=O)NCCCCCc2cn(C3CCN(C)C3)nn2)ccncc1Br N(C1CCCc2nccnc21)C(Cc1c(S(C)(=O)=O)csc1)=O C12(CC)CC(C(=O)NCC(O)CNC(=O)C=Cc3ccn(C)c3)(CO1)C2 CC(C)C(C)CC(=O)N1CCOCC1CNC(c1cn[nH]c1)=O Cc1ccc(S(=O)(=O)N(C)C)cc1C(=O)NC(C1CCCO1)CO CC(CCCNC(c1coc(C2CC2)n1)=O)NC(=O)CCn1cc(Cl)cn1 O(N1CCN(c2ccc(C(=O)NCCOCCC#N)cn2)CC1)CC CC1CN(C(C2CC(C)(C)C2)=O)CCCN1C(C1(CO)CC(F)(F)C1)=O N1(C(C)=O)CCC(N=c2nc(N3CCCC3)[nH]c(N3CC(F)(F)C(F)(F)C3)n2)C1 c1(CC(=O)N(C)CCN(C)C(c2ncn(C)n2)=O)c[nH]c2cccc(Cl)c12 N1(CCCCNC2CCN(C(=O)CCn3cncn3)C2)CCN(CC(F)F)CC1 CCCC(O)CC(=O)NCCC12CCC(C1)N(C(c1cc(C3CC3)on1)=O)C2 C(N=c1[nH]cc([N+](=O)[O-])c(O)n1)C1CCCN(C(CC2C(C)=NOC2=O)=O)C1 C1(CNC2CCN(c3n(C)ccn3)C2)CCC(n2cc(C3CC3CO)nn2)CC1 c1(C(N2C(C(=O)NCCc3n(C)cnc3)CCC2)=O)ccc(F)c(F)c1 C1(CC)OCCC1C(=O)N(C1CCCCC1)CCNC(=O)COC1CC1 c1(-n2cc(CCCNC(CN(C3CCC3)C)=O)nn2)ccc(S(C)(=O)=O)cc1C CC(C(=O)NCC1CC(NC(c2ccncc2N)=O)C1)C(F)F CC(C)C(C)(O)CNC(C1(NC(=O)CCc2ccn(C)n2)CCSC1)=O c1(C(=O)OCc2coc(Br)n2)cccc2ccc(O)nc12 C1(NC(c2c(OC)cccc2C)=O)CC2(CCN(C(=O)CSCC3CC3)C2)C1 C(C(CNC(=O)CCCCc1cn(C(C)C(=O)O)nn1)C(C)C)OC N(C1CCc2c(F)cccc21)C(c1ccccn1)C c1(OC)cnc(Cl)[nH]c1=NC(=O)c1sc(=NCc2ccccc2[N+](=O)[O-])[nH]c1C c1(CNC(C2CC(NC(=O)COCC(F)(F)F)C2)=O)c(F)cccc1F C1(C(N2CC(F)(CNC(C3(CC)CC3(F)F)=O)C2)=O)CC2CCC1O2 CCC(C)C(C(=O)NC1(CCO)CN(C(c2cc(SC)ccc2Cl)=O)C1)OC C1(NC(c2c(SC)nccn2)=O)(CNC(=O)CC2CCCC2)CCCCC1C O=C(C1=CC(O)C(NC(=O)C2=C(Cl)CCOC2)C1)NCC(C1CCCCCC1)O N1(C(CC2CCCN(C(c3c(C)ccnc3O)=O)C2)=O)CCC2(CCN(C)C2)C1 c1(C(=O)NCC2C(C(=O)Nc3c(CC)nsc3)CCCC2)cccc(O)c1F C1(NC(c2c(-c3nc(C)sc3)c[nH]c2)=O)CCN(C(=O)C2=CC(C)CC2)CC1O c1(C(=O)NC2CN(C(C3CC(=C)C3)=O)C2)ncc(C)cc1C(F)(F)F N1(CCC(N2CCC(OCCOC)C2)=O)C(=O)c2ccccc2S1(=O)=O c1(CN2CCC(NC(c3cnc(C)[nH]3)=O)C(F)C2)ccc2cn(C)nc2c1 c1(NC(=O)C(=O)NC2CN(C(=O)OC(C)(C)C)C2)ccccc1.CCSCC C=CC1COCCN1C(=O)C(CC1CC1)NC(=O)CNC(=O)CCC C1(COC)CN(C(C2(C(=O)NC3CC3)CCC2)=O)CCN1C(=O)C=CS(C)=O C(=O)(C(C)C(C)c1ccccc1Cl)N(CCC)CCNC(c1cnnn1C)=O c1(C(NNC(=O)C2CC(=O)N(c3ccccc3)N2)=O)n[nH]c2ccccc12 c1(C(=O)NCC(CNC(C2CCC(=O)N2)=O)O)cc2nccc(C(F)(F)F)n2n1 N1(C(C(CCOC)OC)=O)CCC(C(N2CC(N3CCCC3)C2)=O)C12CC2 C1(C(F)(F)C(=O)NC2CCC2CNC(=O)CC2CC2C2CC2)(OC)CCCC1 c1(OCC(=O)NCC(N(C(c2ncc(C)nc2)=O)C)C2CC2)c(C)occc1=O c1(C(N2CCCC(O)(CNC(c3c(CC)cno3)=O)C2)=O)cc(C)c(F)cc1Cl C1(C(CNC(c2cc(CC)no2)=O)O)CCN(C(=O)CCSCC(=O)OC)CC1 c1(CC(=O)NCC2CN(C(C3N(N=O)CCCC3)=O)C2)ccc2[nH]ccc2c1 c1(CC)nc(C(N2CCC(CCNC(c3occc3Br)=O)C2)=O)c(N)s1 N#Cc1ccc(C(N2CC(F)(F)CC2CCNC(=O)C2=CCCOC2)=O)c(F)c1 C1(NC(COc2cccc(C#C)c2)=O)(CO)CC2CCC1CC2.c1(C(=O)N)ccns1 c1(C(=O)NC(C2CCN(C(CSC)=O)C2)C)cc2c(C)c(Cl)ccc2[nH]1 CCCCCCC(C)CC(=O)N(C1CCN(C(c2cc3c([nH]2)CCCC3)=O)C1)C C1(C(=O)NC2CCN(C(c3cccc(C)n3)=O)C2C)Cc2nnsc2S1 CC(O)C(C)CNC(=O)C(c1ccccc1)NC(=O)CCc1cn[nH]c1 c1(OC)ccc(C(=O)NC2COCCC2NC(=O)C(C)C(C)C)c2[nH]ncc12 C1(OCC)CC2CN(C(=O)C(C)N(C)C(C3CCCN3C)=O)CC12 C(=O)(C1=CC(O)C(NC(C2CS(=O)C2)=O)C1)NCCN(C)CCO C1(n2cc(COC(=N)O)nn2)CCCN(C(=O)CC(C)n2ccnc2)CC1 C1(C(=O)NCC2CN(C(C3C(C)C3)=O)C2)CC12CCOc1ccc(Cl)cc12 N1(CC(N2CCC3CC(COC)C3C2)=O)CCn2c(Cl)ccc2C1C N1(C(Cc2c(C)nc[nH]2)=O)CC2CC(NC(c3c[nH]nc3OC(C)C)=O)C(C2)C1 n1(C(CC)C)nnnc1C(c1cc(C(=O)OC)cs1)NCc1conc1C1CC1 C1(CNC(CC(C)c2cnn(C)c2)=O)Cc2ccccc2CN1C(C1(CO)CC1)=O N1(C(C2CN(CC)C(=O)N2)=O)CCC2CCN(C(c3cnc(C)nc3C)=O)CC12 c1(C(=O)NCCCN(C(C=C(CCC)C)=O)C(C)C)c(C(C)C)cccc1C CC1CN(C(c2cnns2)=O)CC1NC(C1C2CCCC12)=O C12CC(=NO1)C1CCN(CC1)C2.c1(OC)ccc(-c2nc(C(=O)OC)cs2)cc1 CC1(C)CCCN(C(=O)Cc2cc[nH]n2)C1CNC(=O)Cc1c(F)cccc1Cl c1(C(=O)NC2(c3cc(C)no3)CCCCC2)cncc2n[nH]c(N)c12 c1(OC)cccc(C=CC(=O)N(C2CN(C(=O)CCC3(C)CC3)CC2O)C)c1 C(=O)(CC(C)C(C)(C)C)Nc1c(OC)noc1C1CC1.C12CCCN(C1)C2 C1(C(=O)NCC(c2ncn(C)c2)O)CCN(C(C2CCCOCC2)=O)CC1 Cc1c(C(N2CCN(C(C3CN(C(N)=O)C3)=O)CC2C)=O)cncc1F c1(CC)cccc(C)c1C(=O)NCC12CC(NC(=O)C(C)CSC)(C1)C(C)O2 CC(CCC(=O)N(CCNC(=O)Cc1ccc(Br)nc1)C1CC1)N(C)C N1(C(CN2CCN(C)C(=O)C2)=O)CCC(C2(C)CC2)C1 C1(NC(C23OCC(C(C)C)(C2)C3)=O)CC2CN(C(C3CC34CCCC4)=O)CC2C1 c1(C(N(C2CC(NC(=O)CCOc3cccnc3)C2)C)=O)cnn(C)c1Cl c1(N(C)C)cc(C(=O)NC2CCCC2(C)NC(=O)CC2CC(C)(C)CO2)ccn1 C(c1cccc(Br)c1)=CC(=O)NC12CC(NC(=O)CC3CCCCO3)(C1)C2 Cc1nc(Br)sc1C(=O)N(C)CCOCCCNC(=O)C(C)C(C)C Cc1nc(CO)sc1C(=O)NC1(C)CCN(C(=O)C(=CC2CCCCC2)F)C1 N1(C(c2cnn(C)n2)=O)CC2CN(C(c3occ4c3CCC4)=O)CCC2(CO)C1 CON(C)C(=O)CCCCCNC(c1cc(Cl)ccc1C)=O n1(C(C)C)ncc(C(=O)N(C)CC2CCCN2C(=O)C=CC(C)(C)C)n1 N1(C(C(C)N(CCC)C(c2ccc3n[nH]cc3c2)=O)=O)CCN2CC(C)CC2C1.C Fc1ccccc1OCCSCCC(c1ccccc1)C1CCC1 c1(CC(=O)NC2C(CNC(C(C)OCOC)=O)CCC2)cccc(C(F)(F)F)c1 N1(C(C(C)CO)=O)CCC(NC(c2ccn3c(O)nnc3c2)=O)C2(CCC2)C1 N1(C(CC=CC(C)(C)C)=O)CC2(C(=O)NCC(O)C(C)(C)O)CC1CO2 N1(C(c2c(C)cco2)=O)CCCC(C(C)NC(c2ccc(C(C)C)o2)=O)C1 C1(NC(C(C)SCCCC)=O)CC(O)CN(C(c2cc(Cl)ccc2C)=O)C1 c1(C(CNC(C)=O)OC(c2ccc(CC(C)C)s2)=O)ccc(F)cc1F c1(NC(C2(CC)CCC2)=O)cc2nncn2cn1.N12CCC(=CC1=O)CC2 C1(CNC(c2csnn2)=O)CN(C(=O)CC(C(F)F)n2cccn2)C2(CCC2)C1 n1(CCCN(C)C)cc(CN(C)C(C2CCC(C(=O)O)C2)=O)nn1 c1(C(C(=O)NCC2CCOC2)N(C(C)C)CC)ccsc1C CC(C)(CC(F)C(=O)Nc1ccc(Cl)cc1O)NC(C1CC(=O)C1(C)C)=O c1(OC)ccc(C(N2CCOC(C(N3CCC(C(C)(C)O)CC3)=O)C2)=O)cc1 c1(CC(=O)NC2CCN(C(c3cc(C(F)(F)F)ccn3)=O)C2)cccc(Cl)c1 CN1CC(NC(=O)C(CNC(c2ncccc2O)=O)CC2CC2)CC1(C)C C1(C(N(C(=O)CN2CCN(c3ccnnc3)CC2)C2CC2)=O)CC(C2CC2)=NO1 CC1(C)CC(NC(C2(CO)CCC2)=O)CCN(C(=O)Cc2nc(C3CC3)cs2)C1 C1(CC=C)(NC(C2(CC3CC3)CCCO2)=O)CN(C(=O)C(C)N2CCCC2)C1 O=C1COc2ccc(C(=O)Nc3nnc(-c4cc(Cl)ccc4F)o3)cc2N1 c1(C(=O)NC2C(CNC(CCc3cnn(C)n3)=O)C2)cnc2cc[nH]c2c1 N1(C(CCCNC(=O)CC(F)(F)F)=O)CC2CN(C(=O)CC3=CCCC3)CC2C1 c1(C(=O)NC(C)CCCCNC(c2ccnc(C3CC3)c2)=O)cccc(Cl)c1F c1(C(N(CC(C)NC(=O)Cc2ccn(C(F)F)n2)CC)=O)cc(OC)ncn1 C1(F)(CNC(c2c(C)snc2)=O)CCCN(C(=O)CCNS(C)(=O)=O)C1 CCCC(CCC)C(=O)NC(CC(=O)NCC1(CC)CCC1)C1CC1 c1(CN2CCOCC(NC(=O)Cc3ccc([N+](=O)[O-])o3)C2)c(Cl)ccc(F)c1Cl C1(C(N(CCCCCNC(C=C(CC)CC)=O)C)=O)CCN(C)C1CC c1(C(C(=O)OCC)(F)F)n[nH]c(=NC(=O)N2CC3(C2)CN(C(C)=O)C3)s1 N1(C(C(CCC)C)=O)CCC(NC(=O)CCc2nnc(C)o2)C(F)C1 c1(SC)c(N2CCC(N(C(CC)=O)C)C2)cc(Br)cc1F.C12CCN(CC1)C2 C1(CC)(NC(=O)CC(C)(C)C)CCN(C(C2CCNC2=O)=O)CC1 N1(C(C2CN(C(C)=O)C2)=O)CCCC2(NC(C3CC3c3cc(C)[nH]n3)=O)CC2C1 c1(OC)c(CCN=C(NCC(=O)N(C)C)NC2CCCCC2)cc(Cl)cc1Cl C12(NC(C(=O)NCC)=O)CCC(CN(C(=O)C(C)Oc3ccc(Cl)cc3)C1)C2 N1(C(c2n(COC)ncc2C)C(=O)NCCSC)CC(C)OCC1C(C)C C1(NC(C2CCC(C)O2)=O)CCN(C(C2(C)CCC2)=O)CC1(C)C C1(NC(C(C)NC(N)=O)=O)CCC2CN(c3cc(O)nc(=O)n3C)CCC2C1 C1(C2CCC2)(CNC(C=CCNC(C2(CC=C)CC2)=O)=O)CC1 C1(NC(C=CCC)=O)CCN(C(c2ccc(C(C)(C)C)o2)=O)C(C2CC2)C1 C(=O)(C#CC(C)C)NCC(CN(C(c1ccc(-c2ccc(C)o2)s1)=O)C)O c1(C(=O)NCCN(CCC)C(c2cccc[n+]2[O-])=O)cccc2cccnc12 C1(OC)(CNC(=O)NC(C)CC(=O)N2CCCCC2)CCSCC1 C1(CC(=O)N(CCC(=O)OC)C)CCCC1NC(=O)C(C)NCCN(C)C C1(CC)C(c2ccccc2)CCN1C(C1CC1C1CC1)C(=O)NC CC(N=c1[nH]c2c(c(=NCC3CC34CCC(O)CC4)[nH]1)CSC2)c1cnn(C)c1 C1(NC(C(C)CNC(=O)C=C2CCOCC2)=O)CC1C1CCC1 N1(C(CC2N(C)CCCC2)=O)CC2CCC(C1)N2C(=O)C(O)C1CCC1 c1(C(=O)NC2C(NC(C(CN(C)C)(C)C)=O)C2)cccc(N=S2(=O)CCCC2)c1 c1(C(N(c2ccccc2F)CC)=O)cc[nH]c2nccc1-2 C(=O)(C(=O)N=S(C)(C)=O)NC1CN(C(c2ccc(CN(C)C)o2)=O)CC(O)C1 c1(NC(=O)NC(CC)(C)C)cccc(CO)c1OCCN1CCC(F)C1 C1(CNC(C2(F)C(C)C2)=O)COC(C)(C)CN1C(c1nccc(Cl)c1O)=O N1(C(c2cc(CSC)oc2)=O)CCCC(N(C(=O)C(C)C2CCC2)C)C1 CC1CCN(C(C2(C3CC3)CN(C(=O)C(C)C3CC3)C2)=O)CCS1 N1(C(C2(C)CC3CCC2C3)=O)CC2CC(NC(=O)C3=CS(=O)CCC3)CC1C2 Cc1nccc(C(N2CCC(CO)C(c3ccccc3)C2)=O)c1C c1(C(=O)NCCC2CCC(NC(CCC#C)=O)C2)c(N)c(F)cc(F)c1F S(=O)(=O)(c1ccc(C(N2CCCN3CCCC23)=O)cc1)N(C(C)CO)CC O=C(CC(C(F)(F)F)NC(c1ccc(Cl)cc1)=O)NCc1cccnc1F c1(CC(c2cn(CNC(C(C)OCC3CCCO3)=O)nn2)(C)O)ccc(Cl)cc1 C(=O)(C1(C)CCOc2ccccc21)NCC1CN(C(CSCC#C)=O)CC12CC2 c1(C(=O)NC2C3CN(C(c4c(OC)cc(N)cc4)=O)C2C3)nccn2cnnc12 N1(C(c2c(CC)cno2)=O)C(C)CC2CN(C(C3CCC(OC)C3)=O)CC12 c1(CC(=O)NCC2COCC2NC(c2cc(CF)on2)=O)cc2ccccc2o1 c1(COC)cccc(-c2cn(C3(C(=O)NCC4CC4(C)C)CC3)nn2)c1 N1(c2cccc(CN3CC(=O)NC3=O)c2)CC2CC1CN2C(c1ccoc1)=O N1(C(C(CC=C)CC)=O)CC2=C(C1)CN(C(=O)CN1CC(C)(C)C1)C2 c1(CNC(C(=O)N(CCOC)Cc2cnn(C)c2)=O)nc2cccc(C)c2n1C CC1(NC(C2CC2(C)Br)=O)CCN(C(C2CC(n3ccnn3)C2)=O)C1 CC1(C)CC(C(=O)NCC2CCCN2C(=O)C=C2CC2)C(C)(C)O1 CC(C)(C)CC(C)(C)C(=O)N1C2CC1CN(C(=O)C(C1CCCO1)C1CC1)C2 C1(C(=O)NCC2N(C(c3ccc(C(N)=O)[nH]3)=O)CCC2)CC12CCC1(CC1)CC2 c1(C(N2CC(C)C(NC(C3(C(N)=O)CCC3)=O)C2)=O)cc(F)cc(Br)c1 C1(NC(c2cc(C)c(C)o2)=O)CC(F)CN(C(=O)CN2CCCS2(=O)=O)C1 C1(NC(C)=O)COCCN(C(=O)CN(C2CN(C)CCN2C)CC2CCOCC2)C1 N1(C(C(c2nc3ccccc3[nH]2)C)=O)CC2(CC(CNC(=O)C(O)CF)CO2)C1 C1(C)(C(=O)NC(C)C(=O)N(CC(O)C2CCC2)C)CC(=O)N(C)C1 C(=O)(C1=C(C)OCCC1)NC(CN(C(=O)CCC1CC(F)(F)C1)CC)C C1(C(N)=O)CCN(S(=O)(=O)NCCCOc2ccc(S(N)(=O)=O)cc2)CC1 N1(C(=O)OC(C)(C)C)CCCC1(CCF)C(N1CCC(CO)CC1)=O c1(NC(CC2(C)CCN(C(C3CC(NC)C3)=O)C2)=O)cc(OC)cc([N+](=O)[O-])c1 C(C)(C(=O)NC1CCC1NC(c1ccc(-c2ccncc2)s1)=O)(C1CC1)OC c1(C(=O)NCC2C(NC(CC(C)(C)O)=O)CCC2)coc2c1C(O)CCC2 C1(C2CCN(C(c3ccc(C4CC4)nc3)=O)C2)(NC(CCCSC)=O)CC1 c1(C(N2CCC(F)(NS(CC)(=O)=O)C2)=O)c(Cl)cc(F)cc1Cl N1(C(c2c(OC)ccs2)=O)CCC2C(C1)CN2C(C1CCC(F)CC1)=O NS(=O)(=O)c1cnc(NC(=O)NCc2sccc2S(C)(=O)=O)nc1 c1(C(=O)NC2C(NC(Cc3n(C)ncc3)=O)CCC2)ncccc1Br c1(C(N2C3C(NC(=O)CSC(F)(F)F)C(CC3)C2)=O)cccc2c1C1CCC2O1 Cc1c(C(=O)NCC(C)(C(C)C)NC(=O)C=Cc2cncn2C)noc1C1CC1 N1(C(c2c(C)scc2)=O)CCCC(CCNC(c2ccc(CC3CC3)cc2)=O)C1 C1(C(COC)NC(CCC)=O)CCN(C(=O)C(COC)N(C)C)CC1 N(C(=NCC(C)(C)F)NC1CCOCC1)C(C)Cc1ccccn1 N1(C(C(C)=C2CC2)=O)CCC(C(F)(F)F)C(NC(=O)C=CC2CC2)C1 c1(C(C)C)cc(CNC(c2ccc(C(F)(F)F)s2)C(=O)O)no1 CC(CC(=O)c1ccc(F)cc1)C(=O)NCCn1[nH]nnc1=N N1(C(CCN(C)CC)=O)CCOC(CCNC(c2ncncc2F)=O)C1 CCS(=O)(=O)CC(=O)NCc1cnn(C)c1C(N1CCCCC1C(C)C)=O c1(C(=O)NC2CN(C(CCCCC=C)=O)CC3C2C3)sc2cccc(F)c2c1Cl c1(C(N2CC(C)(CNC(=O)C(O)C(F)(F)F)OCC2)=O)ccc2cccnc2c1 c1(C(=O)NCC2(NC(c3cc(Br)c[nH]3)=O)CC2)ccc2n[nH]cc2c1Cl C1(CNC(C2C(OCC)C2)=O)C(C)CCN1C(=O)CCOC(C)C.OCC c1(C(N2CCC(CCNC(=O)C(F)=C3CCC3)CC2)=O)cc(O)nc(C2CC2)n1 CCS(=O)(=O)CC(=O)N1CC2(CCN2C(c2ccn(C3CC3(F)F)n2)=O)C1 CC1C(NC(c2cn(CC(F)(F)F)cn2)=O)CCCN1c1nnc(C(F)F)s1 c1(C(N2C(C3(O)CN(C(C(COC(C)=O)C)=O)C3)CCC2)=O)ccc(F)cc1F N(C1CCC(C)(C)c2ccccc21)Cc1ncc(C(=O)OC)cn1 c1(CC(=O)N(CCCNC(=O)C(N)=O)C)ccc2oc3ccccc3c2c1 C(CCC(C)C)(C(=O)NCCCCCOC)NC(CCCCCC)=O C1(C2(O)CN(C(C3CCC(F)(F)CC3)=O)C2)(CNC(Cc2c(C)scc2)=O)CC1 c1(C(=O)NCCCC2N(C(C(CC)C#N)=O)CCCC2)cc(C(C)C)ccc1C C1(c2ccc(OC)cc2)C(C(=O)NC2COCCC2NC(=O)CO)CC(=O)N1C CC1CN(C(C(=O)Nc2ccc(F)cc2)C2CC2)CC(c2cccc(CN)c2)O1 c1(C(=O)NCC#CCNC(C(c2cccc(Cl)c2)CC)=O)noc(C2CC2)c1C C(=O)(C1=NOC(C)C1C)NC1C(CC)N(C(c2ccc(C)c(C)c2)=O)CCC1 C(C(=O)NOCCOC)(C(C)C)NC(C1ON=C(CC)C1)=O C1(NC(c2ccsn2)=O)CN(C(c2cn3ncccc3n2)=O)CCC12CCC2 c1(NC(C2(CNC(CC(CC)C)=O)CC2)=O)ccn2nccc2c1 CC1OC2CCC1(NC(c1sccc1CNC(c1cc(O)cc(=O)o1)=O)=O)C2 C=C1CC2CCC(C1)N2C(=O)C(O)CCCNC(=O)C(F)(F)C(O)CC C1(C(N2CCC(CCNC(C(c3ccccn3)C)=O)CC2)=O)COC2COCC12 c1(C(=O)NCC2CN(C(C3CC(C(C)(C)C)C3)=O)C2)cccc(Br)c1Cl CC1(C(=O)NC2C=CC(CC(N3CC(F)(CO)C3)=O)C2)CCC(=O)NC1 c1(OC)cccc(F)c1C(=O)NC1C2CN(C(=O)CSc3nc[nH]n3)CC12 C#CCC(C)(C)C(=O)NC1CCC1NC(c1ccn(C)c(=O)c1)=O C12(C(=O)NCc3c(C)n[nH]c3)CC(CCO1)N(C(c1cc(C(N)=O)co1)=O)C2 c1(SC)ccc(O)c(C(=O)NCC(C)(C2CC2)NC(C2CS(=O)(=O)C2)=O)c1 Cn1cnc2c(NCC(C)(C)N(C)C)[nH]c(=NCc3cnn(C(F)F)c3)nc12 C1(C(=O)NC(CCOC)CO)CC(F)(F)CN1C(=O)CN(C1CCCC1)C N1(C(C2(C)COC2)=O)CCC2(CC1)C(NC(C1CCCC3CC13)=O)CS2(=O)=O c1(C(=O)NC(C)CNC(=O)Cc2ccc(N)cc2)coc2c(F)cc(F)cc12 c1(OC)cnc(C(=O)NCC2CCN2C(=O)C(Cc2cnc[nH]2)NC(C)=O)nc1 c1(C(c2n(CCOC)nnn2)NC2C=CCC2)ccc(Br)c(C(F)(F)F)c1 C1(C2CC2)(c2n[nH]c(=N)s2)CCN(C)C1.CC(C)(C)OC(=O)N.C12CC1C(=O)NC2 n1(CC(=O)NCCC(C)N(C(C=CC(C)C)=O)C)ccc(-c2ccccc2)n1 Cc1cc(C(=O)NCCC2CCC(NC(c3ccc4c(c3)CC4)=O)C2)cc(C)n1 C(=O)(N=c1cc(C)o[nH]1)NC(Cc1cccc(C(=O)OC)c1)C(=O)OC(C)C C1(NC(c2cccc(OC)n2)=O)CN(C(=O)C=C(Cl)Cl)CC2CC12 C1(CNC(c2c(CC)cco2)=O)CC(C(=O)NCC2CCOCC2)=NO1 N1(C(Cc2c(C)cco2)=O)CCC(C2(NC(=O)C(c3cnn(C)c3)OC)CC2)C1 CC1(C)CCCCC1CC(N1CCN(C(=O)Cc2csc(S)n2)C(CCO)C1)=O c1(C(N2CC(NC(c3c(C)onc3)=O)C3(C2)CC3)=O)c[nH]c2c(C)cccc12 c1(C(c2n(CCSC)nnn2)NC(c2nnc(CO)s2)C)sc(=O)n(C)c1Cl c1(C(N)=O)ccc(F)c(CO)c1.C12CCN(C(=O)CN3CC=CC3)CC1C(=O)N2 C1(CC(=O)NC(CNC(=O)CCc2ccco2)CO)CCC(F)(F)CC1 c1(-c2c(C(=O)NC(CC)CNC(C3CC(C)C3)=O)cccc2)ccc(OC)cc1 c1(C(=O)NC2C(OC)CN(C(=O)CC(=O)NCC(F)(F)F)C2)cc(F)cnc1O CC1CCCC(O)(C(N2CC(O)(CN(C(=O)C(c3cccn3C)=O)C)C2)=O)CC1 C=CC(C)(O)CC(=O)NC(C)C=CC(=O)Nc1cc(OC)cc(F)c1 c1(C(N2CC(CCNC(CCSC)=O)C2)=O)cnc(C2CC2)nc1 C1(OCC)CCCC(NC(=O)CC2(OC)CN(C(=O)COCC(C)(C)C)C2)C1 C1(C(=O)NCC(C2CC2)NC(c2ccnc(OC)n2)=O)CC2C(C1)C2(C)C n1(CC(C)NC(c2cc[nH]c2C2CC2)=O)cc(CNC(C2CC23CC3)=O)nn1 N1(C(C(CC)C#N)=O)CC(NC(=O)C2=CCCS2)CC(F)C1 C1(NC(C(C)=CC)=O)CC12CCN(C(C1(COC)CCC1)=O)CC2 N1(C(c2c(OC)cc(C)cc2)=O)CCC2(CCN(C(=O)C3=CCCC3C)C2)C1 N1(C(C=C(C)C(C)(C)C)=O)CC(F)(F)CC1(C)CNC(c1c(C)nnn1C)=O c1(C=O)cc2c(F)ccc(Cl)c2[nH]1.N12CCN(CC(F)F)C(C1)C1CC(CC2=O)CC1 CN1CC=C(CC(=O)N2CC(NC(=O)CCc3cccs3)CC23CCCC3)CC1 N1(C(C2CC(=C)C2)=O)CCC(OCCNC(C2CN(C)C2)=O)C1 C1(CC)C(NC(=O)Cc2cccnc2)CCCN1C(=O)C(F)CC1CCOC1 c1(C(N2C(CNC(CCCC=C)=O)CC(OC)C2)=O)ncnc(OC)c1F C(=O)(C1=CCCC1(C)C)N(C)CC1CN(C(Cc2cccc(SC)c2)=O)C1 N1(C(C(C)CF)=O)C2CCC1CN(C(C13CC1COC3(C)C)=O)C2 Cc1cc(C(=O)NCCCCC(C)NC(C2CNC(=O)CC2C)=O)cnc1F CCC(C)(CNC(C1CN(C(C2C3CC(=O)CC23)=O)CC1F)=O)C(N)=O c1(C(=O)NCC2CCCN(C(c3cc(C)c(C)nn3)=O)C2)n[nH]c2c1CCSC2 N1(C(COC(CC)CC)=O)CCOCC(NC(=O)CCN2CCCC2)C1 C1(CNC(c2n(CCC)ccc2)=O)CC(C)N(C(=O)C(C(C)C)NS(N)(=O)=O)C1 C1(CC(=O)N(C2CCCN(C(C(C)(C)CF)=O)C2)CCF)CCOCC1(C)C CN=c1ccc(C(=O)NC2CC(C)N(C(=O)Cc3cnc(C)o3)C2)c[nH]1 c1(CC)oc(CN2CCN(c3n(C4C(C(=O)OC)C4)nnn3)CC2)cc1C(=O)O C1(CNC(CCCCOCCC=C)=O)CC(C)(C)CN1C(=O)CC(C)(C)C C(=O)(C#CC1CCOCC1)N1CCC(C)(CCNC(C(C)CC(F)F)=O)CC1 c1(C(=O)NC2C(CNC(C3C(=O)NCC3)=O)CC2)coc2c(Cl)cccc12 Cc1cnc2n1C(C)CCC2C(=O)N(C)CCNC(C1CCC(N)CC1)=O C1(C)(CNC(CC2(N(C(c3c(C)ccs3)=O)C)CC2)=O)CNC(=O)O1 C(=O)(CCCCN1C(=O)CCC1=O)NCC1C(NC(C(C)=CC2CC2)=O)C1 C1(CNC(Cc2cc(C)ns2)=O)CCC2(CN(C(=O)C(N3CCCC(C)C3)=O)C2)O1 c1(OC)cc(CN2CCC(NC(=O)C(C)(C)Br)C(F)C2)c(OC)cc1C C(C(CO)C(F)(F)F)NC(c1nc(C)n(-c2ncccn2)n1)=O N(C(=NCCOc1ncccn1)NCC(N1CCSCC1)(C)C)CC(=C)C Cc1cc(-c2csc(Cc3cc(O)ncn3)n2)c[nH]c1=N c1(C(=O)NC2CC(NC(C3(SCC)CC3)=O)C2)ccc(N2CCCC2)cc1 C1(OC)CC2CC(C(N3CCCN(CCNC(c4coc(C)c4)=O)CC3)=O)CC12 CC1CN2CCN1C(C(=O)N(CC(O)CNC(=O)C(F)(F)C1CC1)C)C2 c1(C(CC)CO)nnc(N(CCF)CCOC)n1CC(C)C N1(C(C(CC(=C)C)C)=O)CCc2ccccc2C1CNC(=O)C#CC1CC1 C=CCCCCC(=O)N1CCCC(F)(CNC(=O)C(C)C2CCCC2)C1 c1(C(C2C(C)C2C(=O)NCCNC(=O)OC(C)(C)C)=O)ccc(Br)cc1F n1(CCC)nc(C)c(C(N2CC3CC3(CNC(=O)C=C3CCN(C)C3)C2)=O)c1C c1(C2N(C(c3nc(C(C)(C)C)[nH]n3)=O)CCC2)cccc(Cl)c1 C(C(=O)NNC(=O)NC1(c2nc(C3CCC3)no2)CC1)c1ccc(C)o1 n1(C(C)C)cc([N+](=O)[O-])c(=NC2CCC(NC(=O)CCC[N+](=O)[O-])CC2)[nH]1 CC(Cn1ccnc1)C(=O)NCC1CCN1C(=O)N.C1(C)(OC(C)(C)C)CCOC1 Cc1nn(C)c(Cl)c1CC(=O)NCCC1CC(NC(C2(C)CC=CC2)=O)C1 CC(C)CC(C)C(=O)N(CC(C)(C)CNC(C1OCCCC1(C)C)=O)C C1(NC(c2c(CC)ocn2)=O)(CNC(c2cc(C)co2)=O)CCCCC1C C(C(=O)Nn1nnc2c1CCCC2)C1(N(C(c2cn(CC=C)nn2)=O)C)CC1 C(C(C)(C(=O)NCC(C)(C)CN(C(=O)CC=C(Cl)Cl)C)OC)OC N1(C(CC(CC)O)=O)CC2(CCN(C(c3cnn(C)c3C3CC3)=O)C2)C1 c1(CCC(=O)NCCNC(c2c(C)n(C(C)C)cc2)=O)cc2ccccc2[nH]1 c1(OC)cc(C(=O)NCC23CC2CN(C(=O)COC2CCOC2)C3)cc(F)c1F n1(CC(C)O)cc(C(=O)NC2CC(C)(CNC(C3(Cl)CC3)=O)C2)ccc1=O c1(C(N(CC(CC)NC(C2CC2CC(C)C)=O)CC)=O)cn2ncnc2nc1C C1(NC(CC)=O)CCC2(CCN(C(=O)C(=O)Nc3ccc(SCC)cc3)CC2)C1 C1(CCCC)CCC(C(=O)Nc2nccc(-c3cncc(OCC)c3)n2)CC1 C1(CNC(C(C(C)O)N(C)C)=O)N(C(c2ccoc2Cl)=O)CCCC1(C)C c1(CNC(C2N(C(C(C)Oc3ccccn3)=O)CC2)=O)ccccc1O N#Cc1ccc(F)c(C(N2CCC(NC(=O)C(F)n3cccn3)C(F)C2)=O)c1 N1(C(c2cccn(C)c2=O)=O)CC2(CCN(C(c3c(O)ccc(F)c3F)=O)C2)C1 c1(C(=O)NC2CN(C(C3(C)CCCOC3)=O)C2)ccc(N)c2c1CCCC2 CC1CN(C(=O)CC2CCCCN2C)CCN1C(=O)CNC(N)=O N1(C(c2cc(SC)n(C)n2)=O)CCN(C(=O)CCCC(N)=O)C(C)C1C C1(CC(=O)N(C(C)CNC(=O)Cn2ccccc2=O)C)CC2CC(=O)C1C2 c1(OC)nc(C)cc(C)c1CNCC1CCCCC(O)C1.c12ccc(cc1)NC2 c1(C(=O)NCC(CN(C(C(CCOC)C)=O)C)O)cc(C)c(C)c(S(N)(=O)=O)c1 c1(N(c2nc3cc(Br)ccc3o2)C)ccnc(S(N)(=O)=O)c1 n1(CCC)cc(CNC(C2C(C(=O)OC)C2)=O)nn1.C12(CC1)C(=O)NC2 CC1CCCCN(C(c2ccc(CO)c(-n3cc(-c4ccns4)nn3)c2)=O)C1 Cc1ccn(CCC(=O)NCc2occc2C(=O)NCCC2CCN(C)C2)n1 N1(C(C=CC(=O)OCC(C)C)=O)CC(NC(=O)CC(F)(F)F)CC2(CC2)C1 N1(C(c2c(CCC)nns2)=O)CCC(C2CN(C(C3(C)CCC(C)C3)=O)C2)CC1 c1(C(=O)NCC(C)NC(c2cnc(C(F)F)nc2)=O)ccc2ncccc2c1F c1(C(=O)NCC(C)NC(c2ccc(-c3cccc(Cl)c3)cn2)=O)ccc[n+]([O-])c1 N#CC1(NC(N2CC(C(F)Cn3cc(-c4cc[nH]n4)nn3)C2)=O)CC12CCCC2 C1(CNC(CCCOC(C)=O)=O)CN(C(c2nonc2N)=O)CCCO1 Cc1cc(C(N2CCN(C(C3CCN(C)C3=O)=O)CC2c2ncc[nH]2)=O)c(C)n1C c1(NC(c2c(C)cco2)=O)ccc(C(C)Nc2cnc(F)cn2)cc1 Cc1c(F)cc(NC(C2CCC(NC(c3ccc(CO)cc3)=O)CC2)=O)cc1Br C(=O)(CCC(c1ccc(OC)cc1)NC(=O)C=C(C)I)OC c1(C(=O)OC)c(C(N2CC3C(CNC(C4(CCO)CC4)=O)C3C2)=O)cnn1C.CC n1(CC(C)C)cc(CC(=O)NCC(O)CN(C(=O)C(F)C2CCC2)C)cn1 c1(C(=O)NCCCCCNC(C2C3CCC2CC3)=O)ccc(Br)c(F)c1 C#CCCCCCC(=O)NC1CCC(O)CN(C(=O)C(CC(C)(C)C)OC)C1 C1(C(N2CC(OCC)C2)=O)CC=CC(NC(C2CC23CCOC3)=O)C1 N1(C(C)=O)CC2CC(C1)N(C(c1cc(C(F)(F)F)c(Br)cc1F)=O)C2 S(=O)(=O)(c1cc(OC)ccc1NC(=O)N=c1ccn(C(F)(F)F)[nH]1)OCC Cc1nc(C2CCC2)cs1.c12occc1-c1nc(no1)N2C1CCC1.c1ccco1 C1(C(=O)NCC2OCCN(C(CCN(C(C)=O)C)=O)C2)CCCC(F)(F)C1 N1(Cc2c(OC)ccc(Br)c2)CCC(N=[N+]=[N-])(c2nc(C(N)=O)no2)C1 c1(CC(=O)NCC2CC(OC)CN2C(c2ccc(N)cc2F)=O)cc(F)cc(F)c1 C(=O)(C(C)CO)N(CC(=O)N(C)CCn1ccnc1)CC CCC(C)C(CC(=O)N1CCCC1CC(C)C)NC(=O)C(C1CCOCC1)=O C1(N(C(CN(c2ccccc2)C(C)=O)=O)C)C2CN(C(c3cnc(Cl)[nH]3)=O)CC12 C1(C)(CC)CCC(NC(=O)C(O)c2ccco2)CC1.c12ccc([nH]1)C(=O)NOC2 C(=O)(C#CC1CCCO1)N(CC(CNC(Cc1c(C)nn(C)c1C)=O)C)C C1(CNC(C2CC(OCC)C2)=O)CN(C(c2ccn(CCF)n2)=O)CCO1 c1(C(N(CCC(C)NC(c2cnn(C)n2)=O)C)=O)ccc2nonc2c1 O=C1CC2(CCC2)C(C(N2CCC(CO)(NC(c3ccco3)=O)CC2)=O)CN1 N1(CC(=O)NC(C)C)CCC(CCNC(=O)C(C)SCCO)C1 C1(NC(c2cc(C)no2)=O)CC2CCC1CN2C(=O)C(O)Cn1cncn1 c1(C(N2CCC(O)(c3cccc(F)c3)C2)C(=O)NCCC)cccn2ccnc12 N1(C(C(C2CCOC2)NC(C(CCN(C)C)O)=O)=O)CC(CO)CC(C)(C)C1 c1(C(=O)OC)nc(NC(c2cccc(NC(=O)NC(C)=O)c2)=O)sc1C c1(C(=O)NCC2CCC(NC(=O)Cc3cccs3)CC2)cnc2n1CCCC2 C(=O)(C1=C(C)N(C)c2nnnn2C1)NCC1CC(OC)CN1C(C1CC1(F)F)=O c1(C(=O)NC(C2CCN(C(C3(CCOC)CCC3)=O)C2)C)c(C)noc1C1CC1 C1(C)(C(N2CCC(C(C#C)C)CC2)=O)CN(C(=O)C(O)C(C)CC)C(C)(C)C1 C(CO)(C(C)NC(=O)CCc1ccc(Cl)s1)NC(C1(CC=C)CC1)=O Cc1nc(CCC(=O)NC2(C)CC(NC(=O)CC(C)(C)F)C2)oc1C CS(=O)(=O)CC(=O)NC1CN(C(C2CC2c2ccccc2)=O)C1 C1(N(C(CN(CCCCCC)C)=O)C)CCCCN(C(=O)C(C)C(C)(F)F)C1 c1(C(=O)NCC(C2CCC2)NC(=O)CCc2cc(Cl)no2)n[nH]c2c1CC1CC21 C=CC(C)(O)CC(=O)N1CCOCC1CC(=O)NCCC(=O)N(C)C1CC1 C1(C(=O)NC23C(CN(C(c4ccc(C(C)C)o4)=O)C2)C3)CCc2n[nH]cc2C1 c1(OCC2(C3CCN(C(CCS(=O)(=O)NC)=O)C3)CC2)ccc(S(C)(=O)=O)cc1 C(=O)(C(C)(C)N(C)C)NCC(CC)NC(c1ccnn1C1CCC1)=O C12(NC(C(C)=C3CC3)=O)CC(CNC(=O)CCc3nc(C)c(C)[nH]3)(C1)OC2(C)C C12(CC(N3C(C)CCC(NC(C4C(C)C4)=O)C3)=O)CCCCC1C2(F)F c1(C(=O)NCC(C)N(C(c2onc(CC)n2)=O)C)ccc(F)cc1 C1(C(=O)NCC2(NC(C34CC(F)(C3)C4)=O)CCCC2)CCc2nncn2C1 C12(C(N3C4CC(CNC(c5ccc(Cl)s5)=O)(OC4)C3)=O)CCOC1CCOC2 c1(C(=O)NCCN(CC(C)O)C(c2cc(F)ccc2Cl)=O)cccn2cncc12 C1N=C(N2CCC(c3ccccn3)C2)NC2CC12.Cn1ccc(CN2CCCC2)c1 C1(C)(C(=O)NC2CC(C)(NC(Cc3c(C)noc3Cl)=O)C2)CCN(C)CC1 c1(C(N2CC(C)(CCC(=O)NC(C)C(F)F)C2)=O)cc2ncccc2[nH]1 C1(C(N2CCCC(CN(C)C(c3ccn(C)c(=O)c3)=O)C2)=O)CCCCC(=O)N1 N1(C(C=CCC)=O)CC(O)(C2(CNC(C34CCOC3CCOC4)=O)CC2)C1 c1(C(=O)NC(CNC(C)=O)C(C)C)ccc(CC2CC(=O)NC2=O)cc1 N1(C(C2(C)CC(=C)C2)=O)CCC(C2(NC(c3cc(C(C)(C)C)no3)=O)CC2)C1 C1(N(C)CC)(CC)CCN(C(CNC)Cc2ccccc2)C1 C1(C(=O)NCc2conc2CNC(C2CC3CC3C2)=O)CC12CCCCC2 c1(C(CNC(c2c(CC)[nH]cc2)=O)NC(=O)CC2CC2)ccc(N(C)C)cc1 CCCCC(C(=O)NCCN1CCCCC1C)NC(=O)C(C)OC c1(C(=O)OC)ccn(CCC(=O)NC2(CNC(=O)CO)CCC2)n1 N1(C(c2c(C)c[nH]n2)=O)CCC(CO)C(NC(=O)CN2CC(C)C2)C1 CCC(CC)(C(=O)NCC1CC(NC(=O)CCn2ccnn2)C1(C)C)OC N12CCSCC1C2=O.C(=O)(CCCSc1ccccc1)OCC(C)C CC(=O)C(C)(C)CC(=O)N1CCC2CCCC12C(=O)NOCC(O)CO C1(C(N2C(CNC(c3c(C)cc(C#N)s3)=O)CCC2)=O)CCn2nccc2C1 CC1(C)CC(NC(=O)CC2(O)CCCCC2)CN(C(c2cccc(Cl)c2F)=O)C1 c1(C(=O)NCC(CC)(C)NC(=O)COc2ccccc2F)cnn2ccncc12 C(C(CC(F)(F)F)NC(=O)CC(C)(C)CC)NC(CC1(C=C)CC1)=O CC(CCCCCO)NC(C1(NC(=O)C(F)n2ccnc2)CCC(C)(C)C1)=O CC1(C(=O)NC2C=CCN(C(=O)CCOC3CCOCC3)C2)CCNC1=O c1(C(N(C)CC)=O)ccc(C(N2CC(C)C2c2ccccc2)=O)cc1 N1(CC(C)NC(=O)CC2CC2(Cl)Cl)CCN(C(=O)C(c2cccnc2)C)CC1 N1(C(c2n(CC(C)C)ncc2)=O)CCCC(CO)(NC(=O)C(F)C2CCC2)C1 C#Cc1ccc(C(=O)NC(C2CN(C(=O)CN(C)CCO)CCO2)C)c(C)c1 c1(CCC(=O)NC(CN(C(C)C(=O)N(C)C)CC)=O)cccc(CSC)c1 C1(CC)(NC(=O)C(C)CCO)CCCN(C(=O)C(C)NC(=O)NC)C1 C1(NC(c2c(C)nc(CC)o2)=O)CCN(C(c2cnc(C)n2C)=O)C12CCC2 N1(C(C(C2CN(C(C(=O)NCC)=O)C2)OC)=O)CCC(CC2CC2)C1 c1(CC2(C(N(C3CCS(=O)(=O)C3)CCC)=O)CCC2)ccccc1F Cc1cncc(C(N2CCC2(C)C(N2CC3CC2CO3)=O)=O)n1 N1(C(Cc2c(OC)ccc(C)c2)=O)CCC2(CCCC2NC(c2cc[nH]n2)=O)C1 N1(C(c2c(NC)cccc2)=O)CCCC2(CCCCC2NC(C2CC23CC3)=O)C1 c1(NC(C2NCCN(C(CCC)=O)C2)=O)cc(C(=O)OC)nc(Cl)c1 c1(OC)ccc2nc(C)c(C(=O)NC3C4CN(C(=O)CCC5CC5)CC34)n2n1 C1(C(F)(F)C(=O)NCCCCNC(=O)C(F)C2CCC2)(OC)CCCCC1 C1(C(=O)NCc2c(F)ccc(C)c2)CC2CC1CN(C(C1CCOC1(C)C)=O)C2 N1(C(C(C)(C)NC(C)=O)=O)CC2C(C(=O)NCc3cc(C)no3)C2C1 C(=O)(C(C)(C)C(=O)NCCN(CC(C)O)C(=O)COC1(C)CCCC1)NC c1(OCC)cc(NCc2ccc(N(C)C)nc2)cc(C(=O)O)c1OCC C=C(CNC(N1CC(c2ccncn2)C1)=O)CC(F)(F)F N1(c2cc(NC3CCCC(C=C)C3)nc(C)n2)CCCN(C)C(=O)C1 CC1CN(C(=O)CC2(n3cccn3)CC2)C(C)CN1C(c1cc(O)cc(=O)o1)=O c1(N2CCC(N(C)C(C3CCC(C)(C)C3)=O)CC2)nc2ncc(Cl)cc2o1 CC1CCC(C(=O)NCCC(C)(C)NC(c2ccc(-c3ccco3)s2)=O)C1 N1(C(C2C(NC(c3ccc(Br)c(F)c3)=O)CCCC2)=O)CCn2ncnc2C1 C1(C(N2CCC(C)C2CNC(C23CSC(C2)C3)=O)=O)Cc2ccccc2C1 Cc1nc(N)cnc1C(=O)N(C)CCNC(=O)Cc1cccc(OC(F)F)c1 c1(C(=O)NCCN(C(C=CC=CC)=O)CC2CCCC2)cn(C2CC2)nn1 c1(C(N2CCC(N(C(c3cc(Cl)n(C)n3)=O)CC)C2)=O)cncc(O)c1Cl C1(C#N)(C(N2CC(SC)C(n3cc(-c4ccncc4Cl)nn3)C2)=O)CCOCC1 c1(C(=O)NCCCN(C(C(C=C=C)C)=O)C(C)C)cnc(O)c(OC)c1 c1(OC)nc(C(N2CC3C(NC(C4(N(C)C)CCC4)=O)C3C2)=O)sc1C N1(C(CCc2cnc(C)s2)=O)CC2(CC(NC(=O)C(C)(C)F)CO2)C1 c1(C(N(CCN(C(CCOC)=O)C)C)=O)ccc2c(c1)C(=O)CCS2(=O)=O CC(CCc1ccco1)N=c1[nH]c2c(c(=NC3CCOC(C)(C)C3)[nH]1)COC2 Cc1cc(CC(=O)Nc2ccc(C(c3nn[nH]n3)C)cc2)cc(C)c1 c1(-n2cc(CN(C(C(CCC)F)=O)C)nn2)ccc(OC)cc1OC C1(CS(N2CC(C(N)=O)CC(C)C2)(=O)=O)CCC2(CC1)CC2(F)F C1(CNC(c2ncc(C(F)F)s2)=O)C2CN(C(C3CC(C(F)(F)F)C3)=O)CC12 CCCC(O)(CCC)CC(=O)N(CCNC(c1cc(C)c(C)cc1C)=O)C1CC1 c1(-c2c(OC)cncc2)cccc2ccc(C(=O)Nc3c(C)cc(Br)cc3Br)nc12 c1(OC)ncc(CCNC(=O)CCn2cc(-c3cnccc3Cl)nn2)cc1C C(CCC(C)CC(=O)N1CCC(NC(=O)C(C)C2CC2)C1)=C(C)C Cc1ccc(C(N2CCC(O)C2C(N2CCC(C)(F)CC2)=O)=O)c(O)c1 C(=O)(C(O)CC(N)=O)N1CC(CC=C)(NC(=O)C(CC)NC(C)=O)C1 N1(C(=O)NCC(c2ccc(C(F)(F)F)cc2)C(F)F)CCCC(F)(F)CC1 c1(C(=O)NCCC2CCN(C(=O)C(F)F)C2)nncc2ccccc12 N1(CC(N2CCC(O)(CNC(Cn3cnc(C#N)n3)=O)C2)=O)CCCNS1(=O)=O C#CCC(CC(=O)OC)NC(=O)C(N)Cc1ccsc1.c1ccccc1 C(=O)(C(CC)n1cncn1)N(CC(=O)NCCSCCOC)CC#C C12(C(=O)NC3CCC(CNC(c4c(C)nn(C)c4N)=O)C3)CCCCC1C2(F)F n1(CC)nccc1C(N1CSCC1C(=O)Nc1cnn(CCO)c1)=O C1(CCC=C)(C(=O)NC(CC2CC2)CO)CN(C(c2cc(COC)[nH]n2)=O)C1 C(=O)(C(CC(F)F)NC(C1(C)CC(O)C1)=O)NC(c1cncc(CO)c1)=O C=CC(C)(C)CC(=O)N(C1CN(C(c2cc(Cl)c[nH]2)=O)CC1(C)C)C CC(CCNC(C1(NC(c2csc(=N)[nH]2)=O)CCCC1)=O)C(F)(F)F N1(C(c2nn[nH]c2Cl)=O)CCC2C(C1)CN2C(c1cnc2[nH]ncc2c1)=O c1(C(N2CC(CCNC(C3CC34CCC4)=O)(OC)C2)=O)ccc(F)c(Cl)c1F C1(CC(=O)NCC(C)NC(C2CCC(C3OCCO3)CC2)=O)CCC(=O)NC1 c1(OCC(=O)NCC(C2CCC2)NC(=O)C2=CCSC2)ccc(F)cc1Cl c1(C(=O)NC2CCN(C(CC3C(=O)NC(=N)S3)=O)C2)ncnc(O)c1Cl c1(CC)ccc(Cn2cc(CN(O)C(=O)c3ncoc3-c3cccs3)nn2)cc1 Cc1cc(C(N2CCN(C(=O)C=C3CCSCC3)CC2CCO)=O)c(C)cn1 N1(C(C(C)OCCC(C)C)=O)CCC(C2CC2)(CNC(c2ccco2)=O)C1 N1(C(c2n(C)ccn2)=O)CCC2(CC1)COC(C(=O)Nc1cnn(CCO)c1)C2 CC#CCCCC(=O)NC1CCC(C)N(C(c2ccc(C(C)(F)F)cc2)=O)C1 N1(C(CCCN(C)C)=O)CCC(CF)(NC(=O)CCSc2cccc(Cl)c2)C1 C1(C(F)F)(CNC(CSC(C)C)=O)CCN(C(=O)C(C)Sc2ccncc2)C1 Cc1nc(C(N2CCC(NC(=O)CC3CC(C)C3)C(O)C2)=O)ccc1[N+](=O)[O-] C1(NC(C(C(=O)OCC)F)=O)CCCCCC1NC(c1c[nH]nc1CC)=O c1(C(=O)NC(C2N(C(CCC(=O)OC)=O)CCC2)C)coc2cc(C)c(C)cc12 CP(C)(=O)c1ccc(CN2CCCC3C(C(=O)O)C23)nc1 C1(C(=O)NCc2n(CCC)ccn2)CCC(O)CN1C(C1CC2(CC2)CN1C)=O N1(C(C2CCN(C(c3cnc(CC)s3)=O)C2)=O)CCC(C)(F)C1 c1(CC)ccc(C(N2CC(C(C)NC(c3ccoc3C(F)(F)F)=O)C2)=O)c(C)n1 CC(C)CC(C)CNC(=O)C(CNC(C1CC1(F)F)=O)N(C)C C(=O)(C(O)CCS(C)=O)N(CCOC)CCNC(c1cnn(CCO)c1C)=O c1(NC(c2cc(C)nn2C)=O)ncc(-c2ccc(F)nc2)cc1O c1(CC)cc(O)c(C)cc1C.C1(C(c2nnnn2C)(CC)N(C)C)CCS(=O)(=O)C1 c1(C(=O)NC2CC(NC(CC(=C)C)=O)C(O)C2)cc(C)nc2[nH]nc(O)c12 C=CC1(C(=O)N(CC(C)O)CCNC(=O)CSc2c(C)n[nH]c2C)CCOCC1 N1(C(CSCC(N)=O)=O)CC2(CCC(NC(=O)CC(=O)Nc3nccs3)O2)C1 C1(C(N2C(CCCC)CCC2)=O)CN(C(C2COCCN2C)=O)CC1C N1(Cc2ccc(OCC)c(OC3CCCC3)c2)CCC2(O)CCCCC2(O)C1 N1(C(Cc2cccc(OC)c2)=O)CCN(C(=O)C(C)(C)C(=O)N(C)C)CC(O)C1 c1(C(N2C3CC(NC(C4CCC(CC)CC4)=O)C2CC3)=O)cc2ncccc2o1 c1(C(=O)NCC2CCCCN(C(COCC=C)=O)C2)nccn2cc(C)nc12 C1(CNC(=O)C(N2CCCCC2C2(O)CC2)=O)CCc2ccccc2C1 Cc1ccc(-c2ccc(-c3cnccc3C)cc2)cc1N c1(C(C(=O)N(CCCN(C(=O)CCc2cn[nH]c2)C)C)(C)O)ccc(Cl)cc1 CCCCS(=O)(=O)CNC1(c2nnnn2CCOCC2CC2)CCOC1 C1(NC(C2(CC=C)CN(C(C34CC(F)(C3)C4)=O)C2)=O)CCCCCCC1 C(C(=O)NCCC1CCC(=O)N1)(C(C)C)NC(C(C)NC(COC)=O)=O C1(C#N)(c2cn(-c3ccc(NC(CC4CCC(C)C4)=O)nc3)nn2)CCOCC1 N1(C(C(CC)C)=O)CCN(C(c2cncc(COC)c2)=O)C(CF)C1 CC1CN(C(c2csnc2Cl)=O)CCCN1C(C1CCCN1C)=O C1(CNC(COCCSC)=O)CCC2(CN(C(=O)CC3=NNC(=O)C3)C2)O1 C(C)(CC(=O)NCCc1nccn1C)NC(CC=C(C)C)=O C(=O)(CCCOc1cccnc1)NC(CNC(C1(C(C)(C)C)CCC1)=O)CO N1(C(C(CC)C(C)O)=O)CCc2cc(CNC(=O)CCCC(C)C)ccc2C1 CCCCCS(=O)(=O)CC(=O)NCC1CCC1NC(=O)Cc1ccco1 N1(C(C2(COC)COC2)=O)CC2(CC=CC2)C1C(C)C N1(C(C23CN(C(CCc4n(CC)ccn4)=O)C(C2)CO3)=O)CC(=O)NC(=O)C1C C1(CN(C(=O)CC2(C)CC2(F)F)C)CCC(NC(=O)C(=C2CCCCC2)F)CC1 c1(N2CCC(C)(CSC)C2)nc(=NCC2(CCO)CC2)[nH]c2ccc(Cl)cc12 Cc1cc(CNCC2(C(=O)O)CCSC2)cc(F)c1 C(C(C)(O)CC(=O)NCCC(C)NC(=O)C=CSCc1ccco1)OC C(C(CC(C)C)NC(C12CC(F)(C1)C2)=O)NC(C(C)NC(C)=O)=O Cc1ccc(C)c(CC(N2CCCCC(NC(c3sccc3C)=O)C2)=O)c1 N1(C(CNC=O)=O)CCCC(C2CN(C(c3cc4c(cc3Cl)OCCO4)=O)C2)C1 C1(NC(C(n2ncc(C)c2)C)=O)C2CC1CN(C(c1ccc(C(C)(C)C)s1)=O)C2 c1(CCC(=O)NCC2(NC(CCCN(CCC)CCC)=O)CCC2)nc(C)c(C)[nH]1 N#Cc1ccc(O)c(C(=O)NC2COCC2NC(C23CC=CCN2CCC3)=O)c1 C1(NC(C(=O)Nc2cnccn2)C2CC2)CC(C)OC1=O.CC(C)CCN1CC1=O C(=O)(C(C)(C)CC(=O)c1cccc(CO)c1)OC1CC(SC)C(O)C1 c1(NC(C2N(C(c3c(OC)ccnc3)=O)CSC2)=O)cnc2ccnn2c1 c1(CNC(c2n(CC=C)nnn2)C2CC23CCC3)c(F)ccc(C)c1F C1(C(=O)NC(CC(=O)OC)C)CC(C(C)C)CCN1C(=O)CCNC(=O)CO C#CC1(N(C)C)CN(C(=O)C(C2CCN(C(=O)Cc3cc(C)nn3C)C2)F)C1 C1(NC(c2c(CC)cccn2)c2nnnn2C)CC2(CCC(C(=O)OC)CC2)C1 C1(NC(c2cn(CC)nn2)=O)C2CC1N(C(=O)CCc1csc(=N)[nH]1)C2 CN=c1cc(C(N2CCCC(NC(=O)C(O)CC(C)C)C2)=O)cc[nH]1 C1(C(N2CCC(NC(CCSC)=O)CC(O)C2)=O)CCc2nnn(C)c2C1 CCCCCC(F)C(=O)NCC(C1CC1)NC(c1cc2cccnn2n1)=O C=C1CCN(C(=O)CC(C)C)C(C(=O)NC(C(C)C)c2nc[nH]n2)C1 c1(C(C)C(=O)N(CCCNC(C2(C)CCNC2=O)=O)C)ccc(F)c(F)c1 CCCC(CNC(C1CC(=O)C1(C)C)=O)C(=O)NC1CCCC1N=[N+]=[N-] c1(OCC(=O)NCCC(CNC(CC(=C=C)C)=O)O)cc(C)ccc1F c1(CC)ccc(C(=O)NC2(CNC(C3CC(CF)C3)=O)CC2)cc1 C1(C(=O)OC)CCCC1(C)C(=O)NNC(=O)NCc1cnccc1C C(CC(CC)C(=O)NCc1ccc(C(N2CC3CCC3(CO)C2)=O)cc1)=CC Cc1ocnc1CCNC(C1CCCN1C(c1cc[nH]n1)=O)=O Cn1cnc(C=CC(N2CC(C(=O)NCCNC(c3ocnc3CO)=O)C2)=O)c1 c1(OC)cccc(C(=O)NCC2COCC2NC(=O)CC23CCCC2C3)c1O c1(SC)ccc(F)c(C)c1-c1ccc(C(=O)Nc2nonc2C(N)=O)c(C)c1F C1(F)(CNC(C(=CC2CCCC2)C)=O)CCN(C(C2CCC(C)(C)OC2)=O)CC1 CC(CC(=O)N1CCCC1C(N1CCC2(CCC2)C1)=O)C(F)F C(CCN=c1[nH]c2c(cc1C#N)CN(C)CC2)NC(C(C)OCCOCC)=O C(=O)(C1=CCS(=O)(=O)C1)NC1CN(C(C(C)(C)C2CCOC2)=O)CC(F)C1 C1(COC)(NC(=O)CC2CC2)CCN(C(C2(C)CC(C)=NO2)=O)CC1 C12(NC(CCCSC)=O)COCCC1CN(C(c1ccccc1C(N)=O)=O)C2 c1(C(=O)NCc2nc(CNC(C=CCOC)=O)sc2)cccn2nccc12 C1(C(=O)NC(C(=O)OCC)CO)CN(Cc2cc(F)cnc2Cl)CC(F)(F)C1 N1(C(CCCN(C(C(CC=C)CC)=O)C)=O)CCC2(CC1)CSC2 C1(NC(=O)CC2CC(F)(F)C2)CN(C(c2cn3c(n2)CCCC3)=O)C2(CCC2)C1 CC(C)(C)C(C(=O)NCCNC(c1ccc(Cl)c(N)c1)=O)C(O)C(F)(F)F C1(NC(C2CC(C)(C)N(C(=O)CCc3csnn3)C2)=O)CC2CCCCCC12 C(=O)(C(C)C(C)(C)C)NC12CC(NC(c3c(COC)cccc3)=O)(C1)C2 N1(C(CC)=O)Cc2nccn2CC(NC(c2c(C)cc(OC)cc2F)=O)C1 Cc1oc(Br)cc1C(=O)NC1COCC1CNC(C1CCCCCC1)=O Fc1ccc2c(c1)C(NC1CCCC1c1ccccc1)CCC2 C1(C(=O)NCCCNC(C2C(C=C)CC2)=O)CC(=O)c2ccccc2C1 N1(C(c2cc(C)cc(C)n2)=O)CC2OCC(NC(c3c(C)nn(C)c3F)=O)C2C1 c1(C(=O)NCC=CCNC(C(CCC)OCC)=O)ccc2c(=O)n(C)cnc2c1 c1(C2(C(=O)NC3CCCC(NC(C=CC)=O)C3)CC2)ccc(OC)cc1F O=C(CC(O)CNC(C12CSCC1C2)=O)N1CCC(OCCF)C1 c1(OCCC#C)ccc(C(=O)NCCCC(C)(C)NC(=O)CC2CC2C)cc1 Cc1cc(C(N2CCN(C)C(C(N3CCOCC(C(C)C)C3)=O)C2)=O)ncc1N C(=O)(C(F)C(C)(C)O)N1CCC(CC=C)(NC(=O)CCc2cn(C)nn2)C1 C1(C)(CN(C(Cn2c(C)ncc2)=O)C)CCCC1NC(c1cc(C(F)F)cs1)=O Cn1cc(Cl)c(C(=O)NC(CC2CCCC2)C(=O)NCc2ccoc2)n1 Cc1ccc(C(CNC(=O)CCc2cccc(C)n2)NC(=O)C#CC2CC2)cc1 N1(CC(=O)NCC2C(CCC)C2)CCN(C(c2coc(CCC)n2)=O)CC1 Cc1nn(CCN2CCN(C(=O)C(C)C)CC2)c(C)c1C1CCCCC1 C1(C2CCCN(C(C3(CC(C)C)CCC3)=O)C2)(NC(C(F)OC)=O)CC1 N1(C(C2(OC)CCSCC2)=O)CC2(CCC2NC(c2ccc(Cl)cc2)=O)C1 C1(NC(C2CCOC2C2CC2)=O)CN(C(C2(c3ccccc3)CC2)=O)CCC1F C1(S(N)(=O)=O)(C(=O)NCC(=C)CCNC(C2CCCN2CC)=O)CCCC1 CN(C)S(=O)(=O)N1CCC(CNS(=O)(=O)CCC(F)F)c2ccccc21 C1(C(=O)NC(CC(=O)NC)C)CC2CCC(C1)N2C(=O)CC1CCCC2CC12 C1(CC(=O)NCCNC(CCC=C)=O)Cc2ccccc2C1=O N1(CCNC(=O)NC2C(C)CNCC2)C(C)CCCC1C c1(C(CNC(c2ncsc2C)=O)NC(C(C)OCC=C)=O)ccc(C)cc1 c1(C(=O)NC23CC(NC(c4c(C)nns4)=O)(C2)C3)cc2c(O)cccc2[nH]1 N1(C(C(C=C)C)=O)CC2CC(C(N3CC4CCC=CC34)=O)C(C2)C1 C#CCC(C(=O)N1CC(CCO)C1)NC(=O)CCOCC1CC1 Cc1cc(O)c(F)cc1NC(C1C=CCN(C(=O)C(C)(C)C(F)(F)F)C1)=O c1(CNC2(c3n(CCOC)cnn3)CCC2)csc2ccc(F)cc12 C(CO)(CC(F)(F)F)NC(CC1(OC)CN(C(=O)Cc2cnc(C)s2)C1)=O C1(C(=O)NCCOC(C)(C)CNC(c2ccsc2Cl)=O)CC2C=CC1C2 C(=O)(C(O)CC(F)(F)F)N1CCC2C(N(C(=O)C(C)(C)NC(N)=O)C)C(C)(C)C21 c1(NC(C2C(NC(=O)OC(C)(C)C)C=CCC2)=O)ccc(C#N)cn1 c1(C(N(C)CC2(NC(C3CCCCC3F)=O)CC2)=O)nnn2c1C(=O)NCC2 N1(S(CC=C)(=O)=O)CCc2ccc(NC(=O)CCCC(F)(F)F)cc2C1 Cc1nocc1C(=O)N(CCC(=O)NCCCC(F)F)C(C)C C(CS(=O)(=O)N=S(C)(C)=O)NC(c1n(C(CC)C)nnn1)c1n[nH]cc1C C1(CNC(Cn2c(C)c(Cl)cn2)=O)CC2(CO1)CN(C(=O)CCCCCC#N)C2 c1(C(N2CCN(C(CC(C)CF)=O)C(C3CCC3)C2)=O)nc2ccccn2c1F N1(C(=O)CC2COCCN2)CCC2(CC=CCO2)C1 C=CC1(C(=O)NCC2CCC2CO)CCN(C(=O)CS(=O)(=O)NCC)C1 C1(C)(COC)CCCC1NC(C1CCCC(NC(=O)Cc2ncoc2C)C1)=O N1(C(C2N(C)C(=O)NC2)=O)C2CCC1CC(N(C)C(c1cccs1)=O)C2 N1(C(C(N2CC(CS(=O)(=O)NC)C2)=O)=O)CCC(C2CCNC2)C1 c1(C(=O)NC2(CCO)CN(C(=O)C(O)Cc3ccccn3)C2)ncc[nH]c1=O N1(C(C2C(OC)CCC2)=O)CCCC(CO)(NC(=O)Cc2ccn(C(C)C)n2)C1 Cc1nc(N2CCOCC(CNC(=O)CCC3CCCO3)C2)cc(C#N)n1 N1(C(CCCN(C(C)=O)C)=O)CCN(CC(=O)NC2CCOC(C)C2)CC1 C1(C(N)=O)(CC)CCN(N2CCC(C(c3ccccn3)O)CC2)CC1 C1(NC(Cc2cn(CC)nc2C)=O)CCN(C(=O)CSc2nncs2)C(C)C1 N1(C(CSCCC)=O)CCN(Cc2cn(C3C4CC5C(C4)C35)nn2)C(C)C1 N1(C(COc2ccn(C)n2)=O)CC2(CCCN(C(=O)C(C)(C)n3ccnn3)C2)C1 C1(C(=O)NCCCCCSC)CN(C(=O)CCc2nc[nH]n2)CC12CC2 C1(CNC(c2c(OC)cncn2)=O)CN(C(=O)C(C)(C)C(C)O)CCN1C N1(C(CC#N)=O)CCC2(CC1)OCCC2NC(=O)Cc1c(F)cc(F)cc1F C1(CNC(C2CC(O)(CNC(COc3cc(C)on3)=O)C2)=O)CC12CCOCC2 C1(C2(O)CCC2)(C(=O)NCC(CC(C)C)NC(C(CC)N2CCCC2=O)=O)CC1 Cc1cc(O)c(Cl)cc1C(=O)NCC1(NC(=O)C(O)C2CCCC2)CCCC1 CC1CC(NC(c2cn3ccc(C4CC4)cc3n2)=O)c2ncnn21 Nc1c(C(=O)NCC2CCN(C(=O)C(F)=CC3CC3)C2)cnc2ccnn12 C1(CC(=O)NCc2ccc(CC)s2)N(C(=O)C(c2ccc(C)o2)C)CCC1(C)C c1(C(C(=O)NCCCC)N(c2ccccc2OC)CCC)cc(OC)cc(C)c1 C(=O)(C(C)CC(C)(F)F)NC(CC=C)CNC(c1c(C)nn(C2CC2)c1Cl)=O N(C(=NC)N1CCC(C)(C#N)CC1)N(CCN(c1ccccc1)CC)C N1(C(CC2CN(C(C)=O)C2)=O)CC2CCCC2C1C(N1CCOC2CCC12)=O N1(C(C2(OC)CCCC2)=O)CC2(CCCC2NC(C23CCCC2C3(F)F)=O)C1 C(=O)(CCCCCNC(C1CCCC1C1CC1)=O)NC(c1ncccn1)CC C#CC(CC(C)(C)C)NC(=O)CC1(C)CCN(C(=O)CCc2nncs2)C1 c1(CC(=O)OCc2c(C)noc2C)ccc2c(c1)CCOC2 N1(C(c2nncc(CCC)c2)=O)CC(O)CCC1C(=O)NCC1CC(OC)C1 c1(OC)cc(C(=O)NCC(F)CNC(c2ccoc2C)=O)cc(Cl)c1OC c1(C(N2CCC(OC)(CNC(C3CNC(=O)C3)=O)C2)=O)ccnc(Cl)c1O c1(OC)ncc(C(=O)NC2CCCCCC2NC(=O)C(O)CN(C)C)cc1C S(=O)(=O)(c1ccc(-c2ccc(Cl)c(Cl)c2)cc1)NCC(=O)OC CCCC(C(=O)OC)C(=O)NC1CC(C(=O)NCC(C)C2CC2)C1(C)C C#Cc1nc(C(=O)NC2CC(CNC(=O)Cn3nccc3C)C2)cs1 c1(C(N2CC(CC(C)NC(C(C(C)(C)C)OC)=O)C2)=O)c(F)c(C)cc(N)c1F c1(C(=O)NCCCCCCN(C(C2CC(SC)C2)=O)C)ccc(C#N)cc1O CC1CN(C(=O)Cc2ccncc2Cl)CC(C)CN1C(c1cscc1F)=O C(N=c1[nH]c2cc(Cl)ccc2s1)C1(NC(C(CC)n2ccnc2)=O)CC1 N1(C(CN(C)C)=O)CCC2OCCN(C(=O)COCCCF)C2C1 N1(C(c2nc(OC)c(C)s2)=O)CCCC1C1CCCCN1C(=O)Cc1cnc[nH]1 n1(CCC(=O)NCC(c2ccc(F)cc2[N+](=O)[O-])C)cnc2c(N)ncnc12 c1(C(=O)NCC2CN(C(c3cc(C(CC)C)no3)=O)C2)ccccc1SCCO c1(C(=O)NCC2(CNC(CC3COCC(C)(C)O3)=O)CC2)cc2cccnc2[nH]1 Cc1cc(C(=O)NCC(CNC(C2CCC(N(C)C)CC2)=O)OC(N)=O)sc1C N1(C(CN(C)C)=O)CCN(C(=O)COCC2CCOC2)CC1c1ccccc1Cl c1(N(C)Cc2nc(C(C)(C)C)cs2)ccc(S(=O)(=O)NC2CCC=CCC2)cc1Cl C1(C(=O)NCC2(C)CCN(C(Cc3c(C)ccnc3)=O)C2)CC2COCC(C1)C2 C(CC(=O)NCC(O)CN(C)C(C1CC1C(F)(F)F)=O)SC Cc1cc(O)ccc1CC(N1CC=CC1CNC(=O)Cc1c(Br)cnn1C)=O C12(C(N3CC(C)(C(=O)NCCO)C3)=O)OCCCC1C2(F)F.c12ccccc1S2 c1(CC(=O)NC(C2CC(NC(=O)C(C3CCC3)C3CCC3)C2)C)ccccc1C C1(NC(CC(CC)O)=O)CC1C1CCCN(C(C2CN(C(C)C)CCO2)=O)C1 Cc1cccc2cc(C(=O)NC(C)CN(C)C(c3ccc(CN(C)C)s3)=O)sc12 c1(OC)ccc(C(=O)NC(C2CN(C(C3(F)CCOC3)=O)CCO2)C)cc1F N1(C(Cc2cc(C)[nH]n2)=O)CC2(CCN2C(C2CCN(CC(C)C)C2)=O)C1 C1(C(N2CC(N(C(Cc3cc(C)no3)=O)C)C2)=O)OCC2COCCC12 Cn1nc(O)cc1C(N1CC2C(C1)N2C(c1cccc(C2CC2)c1)=O)=O CC1CC(C(=O)NCCCc2ccco2)N(C(=O)Cc2cn(C)cn2)C1 C12(C(=O)NC(c3ncnn3C)C)CCC(CC1NC(=O)CCc1ccn(C)c1)C2 S(=O)(=O)(c1ccc(NCc2cn(C3CC3)nn2)c(F)c1)NC(CC(=O)NC)C Cc1nnc2n1CCC(C(=O)N(CCCCNC(=O)CC1(O)CCOC1)C)C2 CC1(C2CCCN(C(C3CCCCCN3C(=O)CCC3CCC(=O)C3)=O)C2)CC1 C1(C)(NC(C(c2cccnc2F)(C)C)=O)CCCN(C(C2(CC(F)F)CC2)=O)C1 CC(O)(CC(=O)NC1(CNC(=O)C=Cc2cocn2)CCOCC1)C1CC1 c1(C(=O)NCC(C)NC(c2c(C)ncn2C)=O)ccc(-c2cccs2)cc1F c1(C(N2CC3CC(NC(C4CCCSC4)=O)C3C2)=O)coc2cc(O)ccc12 Cc1cc(C)c(C(N2CCN(C(c3cc4n(n3)CC(F)C4)=O)CC2C)=O)c(C)c1 CCCCC(O)C(=O)N(CCCOCCN(C(=O)CC1(C)CC(F)(F)C1)C)C c1(CC)[nH]c(-c2ccccc2)cc1C(=O)NCC(C1(O)CCOC1)O c1(CCC(N2CC(C(C(=O)NCC(C)N(C)C)C)C2)=O)cn(C)cn1 c1(C(=O)NC2C=CC(C(=O)NCc3ncc(Cl)cn3)C2)cc(O)cc(O)c1 C1(NC(C2N(C(C(C(=O)OCC)OC)=O)CCOCC2)=O)CCCCC1N=[N+]=[N-] C1(N(C)C)C=CC(C(=O)NCC(C2CCCC2)NC(=O)CCCc2cncs2)C1 c1(NC(C23CC(NC(CC#C)=O)(C2)C3)=O)cc(F)c(Cl)cc1Cl N1(c2n(CCOCC=C)c(CCc3ccc(C)cc3)nn2)CCC(C2CCC2)C1 c1(OC)ncccc1C(=O)NC1CC(C)(NC(=O)Cc2cncn2C)C1 c1(C(N2CCC(CNC(c3nc(C)[nH]n3)=O)C2)=O)cc(Br)c(C)cc1F S(=O)(=O)(c1ccc(NC(C)Cc2ccc(Cl)s2)c(C#N)c1)N(C(C)CO)C C(=O)(CCCCCN(C)C(C1(SC2CC2)CCC1)=O)NC1CCCC(C)C1 CCCCC(O)C(C)C(=O)NC(CCC1CCC1)C(=O)NC(C1CCCO1)CO n1(CC=C)cc(C(=O)N(CCCN(C)C(c2ccoc2C)=O)C)cn1 C1(CNC(c2c(C)noc2)=O)CN(C(=O)Cc2cnn(C(C)C)c2)C(C)(C)C1 Cc1sncc1C(N1CCC1(C)C(N1CC(N(CC(C)C)C)C1)=O)=O Cc1ccc(C(CNC(c2ncc(C)cn2)=O)NC(=O)Cc2ccc(C)s2)cc1 C1(C(C(=O)NCCCCCC)N(C)Cc2ncc(OCC)cn2)CCC2(CC2)C1 Cc1c(Cl)ccc(C(N2CC(CNC(c3cc(C(C)C)cnc3O)=O)C2)=O)c1N C(=O)(CCN=c1[nH]c(N2CCCC(C3CCC3)CC2)nc(=N)[nH]1)NC(CC)C C(C)(C)(CC(=O)N1CC(NC(c2cscc2OC)=O)C2CC12)OC Cc1cc(Cl)c(-c2nc(-c3nccs3)nn2CC(C)(C)CO)s1 C1(NC(C(C)C)=O)CCCCC12CCCN(C(=O)COc1cncc(Cl)n1)C2 N1(C(c2c(C)onc2)=O)CCC2(CC1)COC(CNC(=O)C(C)(O)CC(C)C)C2 C(=O)(CCC(C(C)C)NC(=O)COCC(C)C)N(C1CCCCC1)CC=C O=C(CC1=CCCCC1)NCCNC(=O)CNc1ccc(O)cc1 c1(CN(C(=O)NCC(C2CCC2)OC)C)c(F)cc(Br)cc1F c1(C(N(C(C(=O)NCC2CCN(C(C)=O)C2)CO)C)=O)cc(C#N)n(C)n1 c1(CN(C(C2CC(NC(C3C(OCC)CC3)=O)C2)=O)C)cnccc1C C1(NC(c2cnc(OCC)s2)=O)CN(C(C2(N(C)C)CC2)=O)CCC1O C1(C)(CCNC(c2c(C(C)C)n[nH]c2)=O)CCN(C(C2CCC2)=O)C1 C#CCCCCCCC(=O)N(C)CCNC(c1c(C)sc(C)c1C#N)=O N1(C(CC(C)OC)=O)CCC(CNC(c2[nH]ccc2C)=O)CC1C c1(NC(N2C(CC(=O)OCCC(C)C)CC2)=O)ccc2n[nH]cc2c1 C1(C(C(=O)N(C2CN(C(=O)CC(c3cccs3)C3CC3)C2)C)O)CCCCCC1 c1(COC(C)(C)C)ccc(C(=O)NC2CC(CNC(C3CCC(SCC)C3)=O)C2)o1 c1(C(C(=O)NCCC)N(C2CCCC2C)CCOC)cc(Cl)c(C)c(C)c1Cl C1(NC(=NCC)NCc2nn(C)c(Cl)c2Br)CCN(c2ccc(OC)cc2)C1=O c1(C(=O)OC)ccc(C(=O)NC(C)CCCNC(=O)C=CC(C)C)o1 N1(C(C=CC(C)N)=O)CCC2(CC(O)c3ccccc3O2)C1 c1(OC)ccc(CNC(=O)C(Cc2ccc(C)cc2)NC(=O)OC(C)(C)C)nc1 C1(C(=O)NC(C)CCC(=O)OCCCCOCCOC)C2CN(CCC)CC12.OC c1(SC)ccc(CC(=O)NCC23CC(NC(=O)C(O)CCSC)(CO2)C3)cn1 N1(C(CCN(C)CCO)=O)C2CCC1CC(CNC(=O)C1=CCCOCC1)C2 c1(OCC)ccc(C(=O)NC2CN(C(C3(CCF)CC3)=O)CC2C)cc1 CS(C)(=O)=Nc1cccc(C(N2CCCCCC(N)C2)=O)c1 CC(O)CC(=O)N1CCCC1C(=O)NC(c1ccccc1)CN(C)C C1(C(=O)OCC)CC(NC(=O)CCc2c(C)c[nH]c2C)CCO1 c1(C(N2CCC(C)(NC(CC(COC)C)=O)C2)=O)cc(Br)c(F)cc1N N1(C(C(C)CC2CCCC2)=O)CC(NC(=O)CC2CCN(C)CC2)CC(C)(C)C1 c1(CC)ncccc1C(=O)NCc1cc(C(=O)NCc2ccc(Cl)cc2)n[nH]1 CC1=C(C(=O)NCC(CO)NC(=O)COCc2nccn2C)S(=O)(=O)CCO1 c1(-n2cc(CN3C(C)C(C(=O)O)CCC3)nn2)ccc2c(c1)CCN2 N1(C(Cn2ncc(P(C)(C)=O)c2)=O)CC2(CC(O)C(O)CO2)C1 C1(NC(c2cc(C3CC3)n[nH]2)=O)CCC2CC1CN2C(=O)CC(C1CC1)C1CC1 C1(C(N(CCNC(C2N(C(=O)OCC)CSC2)=O)C)=O)CN2CCN1C(C)C2 C1(CC(=O)NC2CC(CNC(CCC(=C)Cl)=O)C2)CCOC(C)(C)C1 c1(C(=O)NC)ccc(CC(=O)N(CC(C)C)Cc2ccnc(Br)c2)cc1 N1(C(C(CSC)(C)C)=O)CC(NC(c2ccc(=O)n(C)c2)=O)CC2(CCC2)C1 c1(C(=O)OC2CCCCN(C(=O)OC(C)(C)C)C2)cnc2ncnn2c1O C1(CNC(CNC(=O)OC)=O)CC2(CCN(C(=O)Cc3ccsn3)CC2)C1 c1(OC)ccc(C)c(C(=O)NC2CCCCC2N(C(=O)C(F)C(C)(C)O)C)c1 CCC(CNC(c1cnnc(C)c1)=O)(CC)NC(C1CC1(C)Br)=O CCC(O)C(F)(F)C(=O)N1CC2CCC1C(NC(=O)C(CC)SC)C2 C1(CNC(C=CC(=O)OC)C)CC2(CCCCC2)CO1 CC1Cc2c(F)cc(Br)cc2C1NC(C1CCCC(F)(F)C1)=O N1(C(C2CCCCO2)C(=O)NCc2ccc(F)cc2)CCCC(O)(CO)C1 CCC(CO)(C(=O)N1CCC(C)(CCNC(C23CCC(OC)C2C3)=O)C1)OC C1(N(C(=O)CN2CCC(C)(O)C2)C)CN(C(=O)CC(C)(C)C2CC2)CCC1O CC1(C)C(CNC(c2cc[n+]([O-])cc2)=O)CCN1C(c1ccoc1C1CC1)=O N1(C(c2scc(C(=O)OC)c2)=O)CCOC2CN(C(=O)CCCC(C)=O)CC12 c1(OC)ccc2c(c1)CC(C(=O)NC1CC1NC(=O)C=C1CC1)CO2 c1(C(=O)NCC(C)NC(c2cc(C(F)F)ccn2)=O)cc(F)ccc1C(F)(F)F O=C1CCC(C(=O)NCCN2CCN(c3ccccc3OC(F)F)CC2)CC1.OC N1(C(CC2(C(C3CCC3)=O)CC2)=O)CCN(C(c2cccc(F)c2)=O)C(C2CC2)C1 CP(C)(=O)C(CCC(N1CCC(c2ccon2)C1)=O)c1ccon1 c1(C(=O)NCC(C)N(C(c2nc(C)ccc2C)=O)CC)cc2cccc(C)c2[nH]1 c1(NCc2c(C)noc2)ccc(C2CCC2)cc1 N#Cc1nc(Cl)ccc1NC(=O)CC1CC(CNS(=O)(=O)CC2CCC2)C1 CC(C)C(C#N)C(=O)N1CC(S(C)=O)CC1c1n[nH]c(NS(=O)(=O)c2cccs2)n1 C1(CNC(C2(CC)CCOC2)=O)CCCN(C(=O)C=CC=C(C)C)CC1 C(CN=c1ccnc(NCc2ccc(-c3ccc(C)cc3)o2)[nH]1)OCC=C C1(NC(C2C(OCC)CC2)=O)CC2CC1N(C(=O)CC1CC(C(=O)OC)C1)C2 N1(C(CN(CC)CC)=O)CCN(C(c2cc(C)sc2C)=O)C(C2CC2)C1 C(=O)(CC(C(F)(F)F)n1cccn1)NC(CCN(C(C=C(C)C)=O)C)C(C)C N(C1CCc2c(F)cccc21)CC(N1CCc2sccc2C1)C CCC(CCC(=O)NOCCCF)NC(c1sccc1C)=O C(C)(CN=c1nc2c(cnn2C)c(NCCCOCCCO)[nH]1)OCCSC C1(NC(CCOC)=O)CN(C(=O)C(O)CC2CC2)C(C)(C)C1 c1(C(NC(=O)OC(C)(C)C)CCl)ccc(S(=O)(=O)N2CCC(CS(N)(=O)=O)C2)cc1 N1(C(CC=C=C)=O)CC2(CCN(C(C3Cc4ccccc4S3(=O)=O)=O)CC2)C1 C1(C#N)(NC(c2ccc(C)s2)=O)CCN(Cc2ccc(Cl)c(F)c2)C1 N1(C(c2ccc(CC)c(F)c2)=O)CCC(C)(C)C(NC(=O)C=Cc2cscn2)C1 C#CCCCC(=O)N(CCNC(C1CC(O)CN1C(=O)C(C)C)=O)CC1CC1 C#CCC(C)(C)C(=O)NC(CCCNC(C1CCOC1CC)=O)c1ccccc1 c1(CC(=O)N(CCC(=O)N(CCCN(C)C)CCC)CC)ccncc1 N1(C(C2(CCNC(Cc3nc(C)[nH]n3)=O)CC2)=O)CCCC(C)C1 N1(c2ccc(COC)cn2)CCC2C(CCCN2C(=O)C(C)OCCC(C)C)C1 c1(C(=O)NCC2CCN(C(C)=O)CC2)c(C)nn(-c2ccc(F)cc2)c1C Nc1c(C(=O)NCCC2CN(C(C34CCC3C4)=O)CCO2)ccnc1Cl C=C(Cl)CC(C(=O)NC(C)CC(C)C(F)F)NC(c1nnccc1C)=O N1(C(c2cc(C)c(Cl)s2)=O)CCCC(C)(NC(=O)CCC2C(=O)ON=C2C)C1 C12(NC(CC(C)SC)=O)CCCC1N(c1nc(Cl)nc3[nH]ccc13)CCC2 c1(C(=O)NC2C(CNC(C(CC#C)C)=O)CCC2)n[nH]c2c(C)cccc12 c1(N2CCC(CN(C(=O)CCc3cccc(F)c3)C)CC2)cnc(C#N)c(C#N)n1 C1(OC)COCCC1CC(=O)NCCCCCN(C)C(c1oc(C)nc1C)=O N1(C(CCc2ccc(C)o2)=O)CC2CC1CCN2C(C1CCC(C)O1)=O c1(N2C(C)CC(NC(=O)C3=CCC3)C2)cc(=O)n2cc(Cl)ccc2n1 Cc1cc(C(N2CCC(NC(c3cccn(C)c3=O)=O)CC2C)=O)c(Cl)cc1N N1(C(CCN(C(C)=O)C)=O)CCCC1C1CCCCN1C(=O)C=Cc1ccoc1 CCCCCCC(=O)NC1(CF)CCN(C(=O)CCC(=O)CC)C1 C1(CNC(C2(C(C)NC(=O)CN3CC4CC4C3)CC2)=O)CC2(CCC2)CO1 C12(CC(=O)N(C3C(C)C3)C)CCC1CN(C(c1nccs1)=O)C2 C1(CC(=O)N(C2CN(C(C=C(C)C(F)F)=O)CC2(C)C)C)Cc2ccccc2O1 N1(C(c2cc(C)[nH]n2)=O)CCCN(C(C2CCCCNC2=O)=O)CC1 c1(OC)ccc(F)cc1C(=O)C(=O)N(C1CCCN(C(=O)CCCC2CC2)C1)C c1(C(=O)NCC2OCCC(NC(C3(C)CC(C)C3)=O)C2)ccnc2ccsc12 C(=O)(CCC(O)C(C)(C)C)NCC(=C1CN(C(c2n(C(C)C)ccc2)=O)C1)F c1(CC(=O)OCC)cccnc1C(F)(F)F.C12(CCOC1)CCNC(=O)N2 C1(C(CC)C)CCN(C(c2cncc(Cl)n2)=O)CC1 N1(C(c2c(CCC)n[nH]c2)=O)CC=CC1(C)C(=O)NCCSCCO C1(C(=O)NCC(=C)CC)CN(C(=O)Cc2cc(C)nn2C)CCN1C N1(C(C(CC)(C)O)=O)CC2CCC1C(CNC(=O)CCCc1csc(=N)[nH]1)C2 C1(C)(C(=O)NC(c2ccc(Cl)cc2)CC)CCCN(C(C2CC(O)CCN2)=O)C1 C1(N(C(C(C)=CC)=O)C)CC2CCC(C1)N2C(=O)Cc1cc(Cl)ccc1Cl c1(-c2c(NCc3cnc(C)s3)ccs2)cncnc1O C(=O)(NNC(=O)C12CC(n3cc(-c4csc(C(C)(F)F)n4)nn3)C1C2)N(C)C C(=O)(CC(C(C)C)c1ccccc1)NC(CNC(C(C)OCCOC)=O)(C)C Cc1cc(C(=O)NC2CCCC(NC(c3c(C)ncnc3C)=O)C2)ccc1O C1(C2CCN(C(c3cc(C(F)F)[nH]n3)=O)C2)(NC(C2CC23CCCCC3)=O)CC1 C(=O)(C(C)(C)CCNC(C1CCC=CCCC1)=O)N1CCCCC(C(C)(C)C)C1 N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C)CC1C(N1CCC(C)C1(C)C)=O c1(C(CNC(=O)CSC2CC2)NC(C2N(CC)CCC2)=O)ccc(F)cc1 c1(OC)cc(OC)cc(C(C)(C)C(=O)NCC2(F)CC(NC(C3CC3C)=O)C2)c1 CC(CS(C)=O)N=c1nc(N2CCC3(CCC3)S(=O)(=O)CC2)c2c([nH]1)CCCC2 c1(N(CCCC=C)C)nc2ccsc2c(=NCCC(C)c2ccccc2)[nH]1 Cc1cc(C(N2CC3(CNC(=O)CC4CC(F)(F)C4)CC2CO3)=O)ncc1N C(=O)(C1=CCCCCC1)NC1C(C)CN(C(=O)C(c2ccc(Cl)cc2)CO)C1 C1(C(N2CCC(O)(CNC(c3cccc(N)n3)=O)C2)=O)CC12CCSCC2 C(C(C)C(=O)NCCCOCCN(C(=O)Cc1n[nH]c(C)n1)C)OC N1(C(C2CCC(=C)CC2)=O)CC(NC(C2(C)CCOCC2)=O)C(C2CC2)C1 C#CCCN=C(NCc1ccc2nc(C)[nH]c2c1)NCC(F)C(F)(F)F S(=O)(=O)(c1cccc(F)c1)NCC(=O)NCC1N(C(C23CC(C)C2C3)=O)CCC1 CC(O)C(N)C(=O)N1CCCCC1NC(=O)C(F)(F)F.n12cc(nn1)C2 O(N(C)C(=O)CNC(=O)C(F)CC1(OC(C2CC2CC(C)(C)C)=O)CC1)CC C1(C(NOCCCC)=O)CCC(NC(=O)C(C)N(CC(F)(F)F)C)CC1 c1(-c2cn(C(C)C)nn2)nc(-c2cccc(Cl)n2)nn1CCCCO N1(CCCNC(CCc2cn(C)nn2)=O)CCN(C(C2CCSC2)=O)CC1 CON1CC(C(N2CCN(C(=O)CCCn3cncn3)CC2CO)=O)CC1=O C1(OCC)(CNC(=O)CCC2(N(C)C)CCCC2)CN(C(=O)C(C)C#N)C1 N1(C(C2(C#C)CC2)=O)CC2CCC1C(CNC(=O)C(C)CC(F)(F)F)C2 C1(C(=O)NCCC2ON=C(C)C2)CC(=O)CN1C(C1CCS1(=O)=O)=O N1(C(c2c(C)nc(CO)s2)=O)CC(CNC(c2cn(C(F)F)cn2)=O)C(C)(C)C1 C(C1=CCN(C(c2cc(N)ccc2C)=O)CC1)NC(CCN(C(C)=O)C)=O c1(CN2CCC(N(C(c3cc(C)c(C)nc3)=O)C)C2)c(Br)ccc2c1OCO2 c1(CS(=O)(=O)NC(CCC(C)C)C(=O)O)ccc2c(c1)C(=O)N(C)C2 Cc1cccc2c(C(N3CCCOC(CNC(C4(O)CC4(C)C)=O)C3)=O)coc12 N1(C(C(C)NC(C)=O)=O)CCC2(CC1)CC2(C)C(N1CC(O)C(N=[N+]=[N-])C1)=O N1(C(c2c(COC)cc[nH]2)=O)CCCC(C2CN(C(C3(CF)CC3(F)F)=O)C2)C1 c1(CNC(=O)C(C2CCCCN2)O)cc2occc2s1 c1(N(C)CCn2cc(CN(C)S(N)(=O)=O)nn2)cccc(OC(F)F)n1 C1(C)(NC(C2N(C(C3C(=C)C3C(=O)OC)=O)CCC2)=O)C(C)(C)C1(C)C c1(C(N)=O)cccc(C(=O)NC2CCOC(c3cccc(F)c3)C2)n1 C1(C(=O)NC(C#C)(C)C)COCCN(C(c2ccc(F)cc2)CC)C1 c1(CC=C)cccc(S(=O)(=O)NC2CCNC(C(=O)OC)C2)c1 c1(C(=O)NCC=CCNC(c2ccc(N)c(C)c2C)=O)cc2cccc(F)c2o1 C1(CNC(=O)OC(C)(C)C)CC(C)(C)CCC1C(=O)NCC(C1CCOCC1)O c1(OC)ccc(F)c(C(N2CCC(CF)(NC(=O)C(F)C(F)(F)F)C2)=O)c1 c1(CC)cc(Cl)c(Cl)c(Cl)c1-n1nc(C(C)O)nc1CO N1(C(c2c(CC)ncnc2)=O)CCC(C)C(C(=O)NC2CCCCC2C#N)C1 C#CC1CN(C(C2C3(CC3)C23CC3)=O)CCN1C(=O)C(CCC)N(C)C C(=O)(C1=C(Cl)CCC1)NC1CCN(CCCNC(C2(OC)CC(CF)C2)=O)C1 c1(C(N2C(C)CCS(=O)CC2)C(=O)NC2CCCC2)cccc2c1OC(C)(C)C2 Cc1ccc(C(=O)NC(C)CN(C(=O)CC2CCC(C)CO2)C)c(F)c1F C(=O)(C(CCC(N)=O)N1CCCC1OC)N1CCC(Cc2ccc(OC)s2)CC1 CC(N=C(NCC(=O)NC1CCCSC1)NCC1CC1)C1CCC1 CCC(CC)C(C)C(=O)N1CC2(C1)CN(C(c1c(C)nn(C(C)C)c1C)=O)C2 CC(C)(C)CC(O)CNC(c1ccoc1CNC(C1(C)CC(C)(C)C1)=O)=O C12(NC(C(CC)=CC)=O)CCCCC1N(C(=O)Cn1ccc(=O)n(C)c1=O)CC2 C1(C(N(CCNC(c2cc(C(F)F)ccn2)=O)C2CC2)=O)CC12CCOC2 c1(C(=O)NCC(C2CC2)NC(CN(C(C)=O)C)=O)cc(=O)c2ccc(O)cc2o1 C1(CNC(C(C)(C)C)=O)CCN(C(c2nonc2N)=O)CC1(F)F c1(C(=O)NC(c2cn(CC(C)(F)C(C)(C)F)nn2)CCC)ccc(C)c(C)c1Cl c1(C(N2CC(C)C(CNC(=O)Cc3nnc(O)s3)C2)=O)csc2ccc(F)cc12 c1(C(=O)NC2C3CCN(C(C4CCC(C(N)=O)C4)=O)C32)cnc2ncccn12 c1(C(N2CCC(CNC(=O)C3=CCSC3)C2)=O)cnc2c(c1)OCC(=O)N2 c1(C(N(C)CC2(CNC(=O)CC3(C)CC3(F)Cl)CC2)=O)ccc(C(N)=O)c(Cl)c1 c1(CC)c(C(N2CCCC(CNC(C3(C(N)=O)CCC3)=O)C2)=O)nnn1C C1(C(=O)NC2CCCCC2)C2CCCC1CN(C(=O)Cn1cc([N+](=O)[O-])cn1)C2 n1(CC(N2CC=CC(NC(C(CC(C)C)(F)F)=O)C2)=O)ccc2c(N)cccc12 Cc1cc(CNCC2(O)CCCN(C(=O)C(c3cccs3)C3CC3)C2)ncc1F C1(CNC(CCN(CCCO)C)=O)CCN(CCCC2CCCC2)C1 C1(NC(CC)=O)CC(C)CN(C(c2csc(-c3csc(C)n3)c2)=O)C1 C1(CNC(C2(CC#C)CCCCO2)=O)C(O)C(O)CN1C(C1CC(C)(C)C1)=O c1(C(=O)NC2(CNC(C(CSC)OC)=O)CCOCC2)cc(C)nc(O)c1 c1(C(=O)NCC2C(NC(CSCCC#N)=O)CCCC2)cccc2c1CCOC2 N1(CC)CC(C(=O)NC2CC3C(NC(C4CCC(=O)N4C(C)C)=O)C3C2)CC1=O C(=O)(C=CS(F)(F)(F)(F)F)NCC1(O)CCN(C(c2cccc(C(C)C)n2)=O)C1 C1(CNC(C2CC(C)=C(C)CC2)=O)CC(N=c2[nH]nc(C(F)(F)F)s2)C1 C1(NC(=O)CCCc2cccnc2)CCCC12CCN(C(=O)C(F)F)C2 C1(NC(C2CC(C)(C)C2)=O)CCN(C(C2(C)CCCS2)=O)CC12CCC2 N#CC1(C(=O)NC2CC(CCNC(C3CC3(F)Cl)=O)C2)CCCC(=O)C1 C(C1(O)CCCc2ccccc21)NC(C(=O)Nc1c(O)cc(C)cc1C)=O N1(C(CCCNC(C)=O)=O)CCOCC1CC(N1CCSC(C(C)C)C1)=O O(C1CCc2c(Br)cccc21)C(c1nn(CC)nc1Br)=O N1(C(=O)C2=CCCOC2)CCC2(CCN(C(c3cc4ncccc4[nH]3)=O)C2)C1 C(=O)(C1CCCc2nc[nH]c21)NC1CC(C)(C)CN(C(c2csc(S)n2)=O)C1 C1(C(=O)OC)CCC(NC(N2CCC2CC2CCCC2)=O)C1 N1(C(=O)CC2C=CCCC2)CC2OCCN(C(=O)Cn3ccc(Br)n3)C2C1 c1(C(=O)NC(C2CCCN(Cc3cscn3)C2)C)cccc(F)c1F C1(C(=O)NCC2CC(CNC(C(C)NC(C)=O)=O)C2)CCCC2(CC2)C1 CC1(C#CC(=O)NCC(O)CC(=O)NCC(N2CCOCC2)=O)COC1 N1(C(C(c2ccccc2)SC)=O)CC(CNC(c2cnc(C(C)O)s2)=O)(OC)C1 C1(CC#C)(C(N2CCC(CN(C(=O)CN(C)C3CC3)C3CC3)C2)=O)CCCC1 C1(C(=O)NCC(c2ccccc2)CNC(=O)CC2CCCC2)C(Cl)(Cl)C12CC2 C=CCN=C(NCC(C)C(=O)OC(C)(C)C)NCC1(CC2CC2)CC1 C1(C(=O)NC2CC3(C(C(N4CCCC(C(=O)OC)C4)=O)C3)C2)CCCCCCC1 C(=O)(CC1=NN(C)C(=O)C1)NCC(C(=O)NCC(CC)CC(C)C)OC C1(F)(CCNC(CCCC(=O)NC)=O)COCCN(C(C2CC(=O)C2C)=O)C1 C(=O)(N1CCC(C(N2CCC(NC(=O)OC(C)(C)C)C2C)=O)O1)NC(C)(C)C N1(C(c2c(NC)snc2C)=O)CC2CCN(C(=O)C(F)(F)c3nccs3)C2C1 C=CC(CC(=O)N(C)CCOCCN(C)C(C)=O)c1ccccc1 CCCCC(CNC(=O)C(C)=C1CCCC1)NC(C1(C)CCCCO1)=O c1(COC)cc(NC(C2CCC2NC(=O)C(CO)N(C)C)=O)cc(O)c1 c1(C(N(CCNC(c2ccnc(O)c2)=O)CC)=O)ccc(N)cc1C(C)(C)C Cc1ccc(C(C)NC(C2CC(=O)CN2C(C2CC(C)N(C)C2)=O)=O)cc1 C1(CC)CN(C(c2cc(CNC(=O)Cc3cccn3C)on2)=O)CCO1 CCCCCCCCCC(CC)C(=O)N(CCC(C)C)CC(F)F Fc1cccc(C(CN2CCCC2)NCc2ncoc2C(F)F)c1 C(=O)(C(F)(F)CCn1cc(-c2nccs2)nn1)NCC(C(=O)OCC)O c1(C(N2CCC(C(CNC(C=CCC)=O)(C)O)CC2)=O)ccc(C)c(OC)c1 c1(C(N(C2CC(NC(C3(N4CCCC4)CC3)=O)C2)C)=O)cn(C2COC2)nn1 CC(C)S(=O)(=O)c1ccccc1NC(=O)Nc1cnc(S(C)(=O)=O)nc1 C(C)(C(C)C(=O)NCC1CCC(C)C1)NC(c1c(CC)ocn1)=O N1(C(C2N(C(C(CC(C)C)N(C)C)=O)CC2)=O)CCOCC(C)(C)C1 C1(CNC(C2(NC(CSCCOC)=O)CC(CF)C2)=O)CCN(C)CC1 C(C(CC(C)C)NC(=O)CNc1ccccc1)n1cc(-c2cnc(CC)o2)nn1 C#Cc1ccc(C(=O)NC2CCN(C(c3cc(C)c(Cl)cn3)=O)CC2C)c(C)c1 C1(C(=O)OC)CCCCN1C(C(=O)NCCCSC)c1csnn1 c1(NC(C(=O)NCC(C)OCC=C)=O)ccccc1-n1nc(C)cc1C c1(C2(C)C(C(=O)NC(c3ccc(O)cc3)CC)C2)ccc(F)c(F)c1 Cc1cnc2n1C(C(=O)NCC1CC(NC(=O)CC3CC3C3CC3)C1)CCC2 C(=O)(C(F)(F)CC)NC(CCC)CNC(=O)C(O)CN1CCCC1 C1(C)(C(N2CC(C)(C)C(Nc3ncncc3I)C2)=O)CCCCCNC1=O CC(C(=O)NCC1CCCCC1NC(=O)CCC(C)(C)O)C(F)(F)F CC(=O)CCCC(=O)NC12CC1CN(C(=O)Cc1coc(C)n1)C2 N1(C(C(n2cc(CC(C(=O)OC)C)nn2)C)=O)CCCN(C(N)=O)CC1 c1(C(=O)NCC(C)(CC)NC(C(CC)C(C)(F)F)=O)cc2ccccc2cc1Cl C1(CNC(=O)Nc2ccn(C3CCC3)n2)CCC(N2CCCCC2)CC1 C1(NC(C(C)OCC2CC2)=O)CCC2(CC1)CC(NC(=O)C(C)C(C)(C)C)C2 c1(NC(C)=O)ccc(C(=O)NC(C)CCNC(=O)CC2CC=CCN2C)cc1 n1(CC(=O)NCC2C(NC(C(C)C#N)=O)CCC2)ccc2nc(O)nc(O)c12 c1(CC(N2CC(C)(NC(C3CCC(CC)O3)=O)C2)=O)cc(F)ccc1Br Cc1ccc(F)cc1C(=O)NCC1(NC(c2ccnn2C2CCC2)=O)CC1 OCCCCCCCCCCCCCCN1CCCC(Cn2cccn2)C1 C1(C(=O)NC(C=C)C)CC2CCC(C1)N2C(=O)CN(C)C1CC1 c1(NC(C(C2(C)CC2)NC(c2c(CC)ncnc2)=O)=O)ccc(O)c(C)c1 C1(COC(=O)NCC)CN(C(=O)CC2(C(F)(F)F)CC2)CCO1 c1(C(N2CC3C(NC(C4CCC5(CCC5)O4)=O)C(C3)C2)=O)occ2c1CCCC2 CC(O)C(C)(C)C(=O)N1CCCC2(CNC(=O)CCC(F)(F)F)CC12 C(=O)(CS(=O)(=O)C(C)C)N1CCC(OCCCNC(c2cnc(CC)[nH]2)=O)CC1 C1(CNC(c2cc(C)nnc2O)=O)CC2(CCC2)CN1C(=O)Cc1csnn1 c1(CC(CNC(C=CC)=O)NC(=O)C=CI)ccccc1 CCC(CC)C(C(=O)N1CC2CC2C1C(=O)Nc1cccc(O)c1)OC c1(C(=O)NCc2scc(C(=O)NCCCC(CC)CC)c2)cc2ccccn2n1 c1(OC)ccc(CN2CCN(C(c3c[nH]cc3C)=O)CC2C)cc1Br C(=O)(CCCC(C)=O)NC(C1CC=CCC1)C(=O)NC(CC=C)CC c1(C(=O)NC2C(NC(C=Cc3cn(C)nc3)=O)COC2)c(F)ccc(F)c1O C(C(=O)NNC(=O)CNCCCCC(C)(F)F)c1ccc(OC)cc1 C12(NC(=O)CCc3ccccc3Cl)CCC(CN=c3[nH]cncc3Cl)(CC1)OC2 C1(CNC(c2c(CCC)onc2C)=O)CN(C)CCN1C(C1CCC(=O)NC1)=O N1(C(CNC(C2COC(=O)O2)=O)=O)CCN(C(c2nc(C(F)(F)F)cs2)=O)CC1 C1(C(N2C(C)CC(N(C(C)(C)C)C)C2C)=O)CCc2nnn(C)c2C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1(CCCNC(C(C)NS(C)(=O)=O)=O)CC1 C1(C(N2CC(CC)N(C(=O)C=CCO)CC2)=O)CCc2nn(C)cc2C1 Cc1c[nH]cc(C(=O)NCC(C2CC2)NC(C2(C)CC(C)(C)C2)=O)c1=O Cc1nc(Cl)cc(=NCC(C2CC2)NC(C2CCCN(C)C2)=O)[nH]1 N1(C(C(CC=CC)C)=O)CC(NC(c2cnn(CCF)c2)=O)CC12CCC2 C1(CC)CCC(C(=O)NC(C(=O)N2CC(OC)C2)c2cccs2)O1 N1(C(c2ccc(Cl)o2)=O)CCC2(CCC(NC(C3(CO)CCC3)=O)C2)CC1 C1(C(=O)NC(CNC(CC2(C(=O)OC)CCCC2)=O)CO)(C(F)F)CCCCC1 c1(N(C2CCC2O)CC)nc(N(C)C)c2cc(C(=O)OC)ccc2n1 c1(NC(c2c(NCc3cnc(C)[nH]3)nc(Cl)cc2)=O)cc(Br)c(F)cc1F CC1(C)CCC=C(C(=O)NC2CN(C(C3(F)CC=CC3)=O)CC2F)C1 CC(C)(CC(=O)N1CCCC1c1ccc(Br)cc1)C(=O)O.c1ccc(Cl)nc1 N1(C(C(C(=O)OCC)OC)=O)CCC2(CC(NC(=O)CCCSC)C2)C1 N1(C(C2(C)CC2)=O)CCOC2(C1)CN(C(=O)CCC1CC1(F)F)C2 c1(C2C(C)C2)nc(-c2cc(Br)sc2Cl)n(C(c2ccncc2)C)n1.C1CCC1 c1(C(=O)NCCCN(C(=O)CCOCCN(C)C)CCC)c(C)nsc1N C1(CC(=O)NCC(N2CCOCC2)C)C(NC(c2csc(F)c2)=O)CC1O C(=O)(C(=O)NC1CC1)N(C)CCOCCN(C(=O)C=CC1CC1)C CC(C)C(C(=O)NC(CNC(=O)CCn1cnnn1)C1CC1)NS(N)(=O)=O N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(C(=O)NCC(C)(O)CO)OC(C)C1 N1(C(c2n(C=C)ncc2)=O)CCC2CN(C(=O)CCc3cccc(O)n3)CC2C1 c1(C(N(CC(CNC(C(C)OCCOC)=O)C)C)=O)cccc(N)c1O C1(CNC(Cn2cc(COC(C)C)nn2)=O)OCCC1(C)C Cc1nc(C(=O)N(CCC(=O)NCC23CCC(CC2)CC3)C(C)C)ccc1C#N c1(NC(c2n(CC(=C)C)nnn2)c2cc(COC)no2)cc(F)ccc1SC N1(c2nc(OC)nc(C)c2)CCC2(COC(NC(C3CCCN3C3CC3)=O)C2)C1 C1(OC)CC2CC1CN(C(=O)CC1N(C(c3cc(C)[nH]n3)=O)CCC1(C)C)C2 CCCCC(C)C(=O)NCC(O)CC(=O)Nc1ccc(C)c(OC)c1 c1(COC)cc(C(N2CCC(O)(CN(C)C(c3csnc3C)=O)C2)=O)ccc1F CC(C)(C)C#CC(=O)NCc1ncoc1CCNC(=O)C(C)(C)c1cncnc1 C#CCC(C)C(=O)NC1CC(CNC(=O)C(C)OCc2ccccc2C)C1 C(CC(C)(C)C)(c1ccc(C)cc1)CC1N(C(=O)NC(C)=O)CC1 c1(C(=O)NCC2(C(C)(C)C)CCN(C(C(CC#C)O)=O)C2)ccc(CO)cc1OC C(=O)(C1SCCc2ccccc21)N1CCC(NC(c2cnc3c(c2)COC3)=O)C1 c1(C(=O)NC2C(OC)CN(C(C3CCC(C)(C)OC3)=O)C2)cc2c(s1)CCOC2 C1(NC(CC2(C)CC2)=O)CCCCN(C(=O)CCC2(C#N)CCC2)C1 Cc1ccc(=O)n(CC(=O)NC2CC3CC2N(C(C2CC(CC(F)F)C2)=O)C3)c1 Cc1nn(C)c(C(=O)NC2CCCCN(C(=O)CC3CCCCO3)C2)c1Cl c1(C(=O)NC2CN(C(COCCC)=O)CC2C)cc(C)n(-c2cccnc2)c1C CN1CC(O)(CNC(=O)CCNC(c2ccccc2)=O)C1 N1(C(CCc2n(C)ccc2)=O)CC(C(=O)NCc2ccccc2)C2(CCC2)C1 n1(CCC)cc(C(=O)N(CC(=O)NCc2n[nH]cc2C)CCC)cn1 c1(-c2n(CCOC)nc(Cc3cc(=O)c(OC)co3)n2)cc(F)c(Br)cc1Cl C(=O)(CC(C)CF)N1CC(O)(CNC(c2c(COC)ccs2)=O)C1 C1(CC(C)NC(c2csnn2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1 Cc1nc(C)c(C(=O)NC2CCCC2NC(c2ncc3ccccn23)=O)c(C)n1 C=CCCCCC(=O)NCC1(F)CC(CNC(C2(F)CC=CCC2)=O)C1 C1(CC(=O)NCC(COC)NC(c2cc(OC(C)C)cs2)=O)CCC(C)C1 c1(C(=O)NC2CCC(NC(c3scc(C)c3)=O)C2)cnc(Cl)cc1Cl C1(CNC(CCN(CC)Cc2cccc(Cl)c2)=O)CC2(CO1)CN(C(C)=O)C2 C(=O)(C1=CCC(C)(C)CC1)NC1CCN(C(CCCCC)=O)CC1F C1(C(=O)NCC(CC)N(C)C)CCCN(C(=O)C(SC)SC)C1 CC(CNC(c1ccc(C2CC2)s1)=O)(CO)NC(=O)C(c1ccccc1)=O C(=O)(C(O)CC(C)C)N1CC(CNC(CC(CC)C)=O)C1 c1(C(N(CCC)CCNC(=O)CC(C)C2CC2)=O)cc(Br)cn1CC N1(C(C(C2CCC2)OC)=O)CC2(CCCC(CNC(=O)Cn3cc(Cl)cn3)O2)C1 C1(C)(CC)NC(=O)C2=C1N(C1CC1C)C(=S)NC2c1cc(OC)cc(Br)c1 C1(C#N)(C(N2CCC(C)(CNC(=O)CC3COCCO3)C2)=O)CCS(=O)(=O)CC1 CC1CC(=O)NC(C(=O)NC(C)(C)C=CC(=O)N(C2COC(C)(C)C2)C)C1 c1(C(N2CC(CC(C)NC(C3CCC4CC34)=O)C2)=O)c(N)cccc1[N+](=O)[O-] N1(CC(=O)NCCN(C)C(C2CCOC(C)(C)C2)=O)CCOc2ccc(Cl)cc21 c1(C(N2C(C)(CNC(c3sc(F)cc3Cl)=O)CCC2)=O)cnn2ccc(O)nc12 N1(C(CNC(=O)NC)=O)CCC2CCN(C(c3nc(C4CC4)sc3C)=O)CC12 C1(NC(CCCCCC)=O)CCN(C(c2nccc(Cl)c2C)=O)CC(C)(C)C1 c1(C(=O)Nc2c(C(=O)OC)c(F)c(C)cc2)cccc([N+](=O)[O-])c1Cl N1(C(C(c2ccccc2)OC)=O)CCC(N2CCOC2=O)CC1 c1(CC(=O)NC(C(=O)N(C2CC(OC)C2)C)CC2CCC2)ccc(C)cc1 c1(C(N2CCN(C(c3cn(C)nc3O)=O)C(CCO)C2)=O)ccc(F)c(O)c1F C1(O)(CC(=O)N(CC(C)O)CCNC(c2nc(=N)cc[nH]2)=O)CCCCCC1 c1(OC)ccc2c(c1)CN(Cc1ccc(N)c(SC)c1)CC(C)(C)O2 c1(CC(CSC)NC(c2cncs2)C)nnnn1Cc1ccco1 C1(C(=O)NCCc2n(C)ncn2)CC(NC(C2CC(O)C2)=O)C1(C)C C(=O)(C(O)(C(F)(F)F)c1ccccc1)N(CC(C)NC(=O)C(F)CC1CCC1)C c1(OC)ccc(CC(=O)NCC2(O)CCN(C(=O)C3=CCCC3C)CC2)cc1F c1(NCCc2cc(C)n(C)n2)[nH]c(=NC2CCC(C(N)=O)CC2)nc2sccc12 N1(C(=O)Cn2ccnn2)CC(NC(C23COCC(C2)OC3)=O)C(C2CC2)C1 Cc1nc2cccc(C(=O)NCC(CNC(=O)C(C)(C)c3cscn3)CO)n2n1 C1(NC(N(C2CN(C(=O)C(C3CCCCC3)F)C2)C)=O)CC(F)(CF)C1 C(c1cccn1C)=CC(=O)NC1CC(NC(C2CC(CC)(CC)C2)=O)C1 N1(C(C2(C(N)=O)CCC2)=O)CCCC(C2CCN(C(N3CSCC3=O)=O)C2)C1 C(=O)(CC(C)(C)O)N(CCC(=O)N(C1CC(=C)C1)C)CC=C CCC(F)(F)CC(=O)NC(CCN(C)C)C(=O)N1CCCCC1CC(N)=O C1(C(N(C)CC2CCN(C(c3cc(CC)on3)=O)CC2)=O)CC2CCCC2C1 C1(N(C(=O)C=C(Cl)Cl)CCOC)CCN(C(=O)C(c2ccc(C)o2)C)CC1 c1(CCC(=O)NCC2CC3(CCN(C(C)=O)CC3)C2)nc(O)c2ccccc2n1 N1(C(c2cn(CC)nc2)=O)CC(CCNC(C2CC(O)C2)=O)OC(C)C1 C=Cc1cncc(C(N2CC(O)CC2C(=O)N(CCC)C2CC2)=O)c1 c1(N(C(Cc2cc(C)on2)=O)Cc2ccccc2)nc2ccccc2[nH]1 N1(C(CN(C2CC2)CC)=O)CCN(C(=O)CSc2ncccn2)C2CCCC12 N1(C(c2c(C)c[nH]c2)=O)CC2CCC(C1)C2C(=O)NCc1cccc(Br)c1 c1(C(N2CCC(CCOC)(NC(C=CSC)=O)C2)=O)c(C2CC2)nc(O)nc1C n1(CC(N2CCC(c3cn(CCCNC(COC)=O)nn3)C2)=O)c(C)ccc1C CCC(C)(C)C(O)C(=O)N1CC(N2CCN(C(c3cnsc3C)=O)CC2)C1 C1(CNC(C(CC)(C)C)=O)CCCCN(C(=O)C2=CCCC2)CC1 c1(CN2CCCC(CC(=O)OCC)C2)cncc(P(C)(C)=O)c1 N1(C(CC2CCN(C)C2)=O)CCOC2(CCN(C(c3cc(O)ccc3O)=O)C2)C1 C(=O)(C(C)C(O)C(C)C)N1CCC(NC(c2ccc(C(=O)OC)c(C)c2)=O)C1 C(N=C(NCc1ccccc1-n1cccc1)N1CC2C(CF)C2C1)S(C)(=O)=O C(=O)(CC(C)(C)CC(=O)NCC(O)CNC(c1ccsc1C)=O)OC Cc1c(C(=O)N(C)CC2CCCCN2C(C2CC(C)(O)C2)=O)cncc1Br N1(C(CCN(CC=C)C(c2coc(C(C)C)n2)=O)=O)CCC(c2ccon2)C1 CCC(C(=O)NCCN(CC(C)O)C(C1(CF)CC1)=O)n1ccc(C2CC2)n1 CC1(NC(C2CCCS(=O)(=O)C2)=O)CCCN(C(=O)C(C2CC2)C2CC2)C1 N1(C(CN(C)C)=O)CCC(NC(C2CC2(F)F)=O)C(c2ccccc2)C1 C1(N(C(CCSCCCC)=O)CC)CCCN(C(c2cc(C(C)C)on2)=O)C1 c1(OC)ccc2c(c1)OC(NC(C1CCC(C)(C)C1)=O)C2 C12(CNC(c3nc(COC)sc3)=O)CC(CO1)N(C(C1CCCC(C)(C)O1)=O)C2 CC1(CCNC(C2(C)COC2)=O)NC(=O)NC1=O N1(C(C(C)(C)CO)=O)CCC2(CCCCC2NC(=O)CSCC(F)(F)F)CC1 c1(COC)ncsc1C(=O)NCCCC1CCCN1C(=O)CCC1CCOC1 N1(C(CNC(c2cccc(C)c2)=O)=O)C2CCC1C(NC(=O)C(C)(C)C(C)C)C2 CS(=O)(=O)c1cccnc1N1CCCC(NC(=O)C=Cc2nccs2)CC1 C(CCCC(=O)NCC1(CO)CN(C(=O)Cc2sccc2C)C1)OCC C1(NC(c2cn(C)nc2)=O)CN(C(=O)C=Cc2cccc(CO)c2)C(C)(C)C1 N1(C(C(c2ccoc2)NC(CCN(C)CC)=O)=O)CCN(Cc2ccco2)CC1 N1(C(c2ccsn2)=O)CCC(C(F)F)(CNC(=O)C(F)CC2CCOCC2)C1 c1(N(C)C)ccc(C(=O)NCC(O)CCNC(c2cc(C(C)(C)C)on2)=O)nn1 C(CCCC(C)C)NC(=O)C(O)Cn1cncn1.C1(OC)C(=O)N2CC1C2 N1(C(c2c(C)[nH]cc2)=O)CC=C(CCNC(=O)CC(C)C(F)F)CC1 c1(OC)c(C)cc(C(=O)NC2CS(=O)(=O)CC2NC(=O)C(C)(C)C2CC2)cc1C c1(CC(=O)NC2(CNC(C3(C)C(C)(C)C3)=O)CCC2)ccc(C2CCC2)cc1 CC(C)CS(=O)(=O)CCC(=O)NC1CCN(C(=O)C(O)CC2CCCCC2)C1C c1(C2C(=O)O2)sc(C)cc1C.C(C)(CC(C)C)N(CCC(=O)OCC)C N1(C(c2nn(CC)c(C)c2)=O)CC2CC(NC(=O)CCc3cnn[nH]3)C2C1 CC1(C)CCN(C(C2CC(NC(c3ccc(F)cn3)=O)C2(C)C)=O)C1 c1(OCC)cccc(C=CC(N2CCCC2c2ccc3cc[nH]c3c2)=O)c1OC c1(OC)cccc(C(c2ccccc2)NC(C2CC(O)CCO2)=O)c1 N1(C(c2cnc(C)[nH]2)C(=O)NCCNCC)CC2CCC(C1)N2CCOC C1(C(=O)NCC(CNC(c2cnc(O)c(F)c2)=O)F)CCCC12CCOCC2 C1(C(N2CC(O)(CCc3cn(Cc4ccco4)nn3)C2)=O)CCS(=O)(=O)N1 C1(C)(CCC(=O)NCCOCCCNC(C(C)c2ccsc2)=O)CC1(F)F c1(C(=O)NCCN(C(=O)C(CC)NC(N)=O)CCC)ccc2nsnc2c1 N1(C(COC(C)=O)=O)CCC2CC2(NC(c2ccc(CO)c(Cl)c2)=O)CC1 N1(C(CC=C)=O)CCCCC(NC(=O)C(c2cccnc2)O)C1 CC(C)C(C(=O)N1CCN(C(=O)CC2CCCC3(CC3)C2)CC1CO)C(C)C N1(C(CC2C(C(C3(C(=O)NC4C5CCC(C5)C4)CC3)C)C2)=O)CCCOCC1C N1(C(CN(CC)CC)=O)CC2C3CCC(C(N(C(=O)C(C)(C)C)CC)C3)C2C1 c1(C(=O)NCC2CC(NC(C3(C#N)CCC3)=O)C2)cc(O)nc2ccc(Cl)cc12 C1(COC)(NC(c2c(C)noc2C)=O)CCCN(C(C2CCOC(C)(C)C2)=O)C1 N1(C(C(C=C=C)C)=O)C2CCC1CN(C(c1cc(C(F)(F)F)cc(N)c1)=O)CC2 C1(NC(CC2(NC(C)=O)CC2)=O)CN(C(c2cncc(C(C)(F)F)c2)=O)CC1C C=C1CC2CCCC(C1)N2C(=O)C(C)(CSC)NC(c1nnc(S)n1C)=O C=CCC(C)(CNC(=O)C(C)N(C)C(C1CCOC1CC)=O)CO C(CC(=O)N(C(C)C(=O)NC(C)(C)COC)CC(C)C)OC C12(NC(=O)CC3CC(NC(c4cccc(CO)c4)=O)C3)CCCC1OCC2 C1(C(=O)NC(c2ccccc2)C(=O)N(CCC(F)(F)F)C)CC2CCC1CC2 C1(C(=O)NCCCN(C(C)C)C(c2cc(Cl)ccc2F)=O)CC1C1CC(F)(F)C1 O=C(C(O)CNC(=O)CNC1=NCCS1)N(c1cccnc1)C1CCCC1 c1(C(N2CC=C(CNC(c3cnc(CC)[nH]3)=O)CC2)=O)ccn2[nH]c(=N)nc2c1 C(=O)(C(C)C(C)NC(=O)OC(C)(C)C)NC(C(=O)NC)Cn1cccn1 C1(NC(c2c(C)cc(CO)cc2)=O)CCCC12CCN(C(C1(O)CCC1)=O)C2 Cc1ncc([N+](=O)[O-])n1CC(N1CC(NC(c2nc(=O)n(C)[nH]2)=O)C(C)C1)=O C1(NC(CCC2C(C)(C)C2)=O)CC2(CCN(C(=O)Cc3ccc4c(c3)CCC4)C2)C1 C(C1=NOC2CC12)(c1nnnn1C1CC1)N(C)C(c1cccc(OCC(N)=O)c1)=O c12nc3ccccc3n1CCS2.CC(CC(N)=O)C1CCCO1 C#Cc1cn(C)nc1C(=O)N(C1(CC(=O)NC2CCC3(CCC3)C2)CC1)C N1(C(CCC2CC(NC(c3cc(OC)no3)=O)C2)=O)CC=CC(O)C1 C(CC(C)C)(C(=O)N1CC(NC(c2sncc2C)=O)CC(F)C1)NC(C)=O c1(OC)cncc(C(=O)N(C2CN(C(c3cc(C)c(C)[nH]3)=O)CCC2C)C)c1C C1(C2(O)CN(C(=O)CSS(C)(=O)=O)C2)(CNC(C2CC3CC(OC)C3C2)=O)CC1 c1(CC)cccc(C(N2CCC(O)(CNC(C3(C)CC(C)(C)C3)=O)C2)=O)n1 C12(CCC(=O)NCCc3nc(C4CC4)no3)CCC(CC1)C2 Cc1ccncc1C(=O)NCCn1cnc(C(=O)NCCc2cnco2)c1 Cc1conc1C(=O)NCCOC(C)(C)CNC(=O)C=Cc1ccsc1 C1(C2(O)CCC(NCc3cc(C)oc(=O)c3)CC2)(C(=O)OC)CC1 c1(C(=O)NC2C(OC)CN(C(=O)CCC3CC3(F)F)C2)ccc(O)c([N+](=O)[O-])c1 C1(NC(Cc2cc(OC)no2)=O)CN(C(c2ccc(C(C)C)cn2)=O)CC2CC12 C1(C(N(C(C)CNC(c2c(F)ccc(C)c2F)=O)CC)=O)CCc2nn[nH]c2C1 c1(C(=O)NC(CCCCNC(C(C2CC2)SC)=O)C)cccn2nccc12 c1(OCC)oc(C)nc1C(=O)NCC1CCCN1C(=O)C(F)=CCCF Cc1c(C(N2CCCN(C(c3cccn3C)=O)CCC2)=O)[nH]c2c(C)cccc12 N1(C(c2c(C(C)C)ncs2)=O)CCC2(CC(NC(C34CC(CC(C)O3)C4)=O)C2)C1 C1(OCC(=O)OCC(CCC=C(C)C)C)CCC(C2CC2)C1 C(=O)(C(C)(O)CC(F)(F)F)N1C(CNC(CCOC(C)C)=O)CC1 N1(C(C(CCC)NC(=O)C(C)c2ccsc2)=O)CC2C(=O)NC(=O)C2C1 N1(C(CC(C)F)=O)CC2CC(C1)N(C(c1ccnc(C(F)(F)F)c1)=O)C2 c1(C(=O)NC2CC(NC(C(CC)OCC)=O)C2)sc2ccc(F)cc2c1C C(=O)(C(F)(F)C(O)CC)NCC1CC(F)(CNC(C(CC=CC)CC)=O)C1 N1(C(CCC#C)=O)CC2CC2(NC(c2c(Cl)n[nH]c2CC)=O)C1 C1(C(=O)N(C)CCOCCCNC(=O)Cc2ncoc2C)(CC)CCC(O)CC1 C(=O)(C(C(C)O)N(C)C)NC1CCN(C(C2C(OC)(OC)CC2)=O)C1 CC(CC(F)(F)F)C(=O)NCc1ccc(CNC(=O)C(=O)Cc2cccs2)cc1 N1(C(C2(CNC(C3C(C(C)C)OCC3)=O)CC(C)(C)C2)=O)CC2COC(=O)C2C1 N1(C(c2c(NC)scn2)=O)CCN(C(=O)C(C)OC2CCCC2)C2CCC12 c1(C(=O)OC)cccn(CC(N2CCC(NC(=O)C(Cl)=CCl)C2)=O)c1=O c1(NC2CN(C(CCCSC)=O)C(C)C2)nccc(S(C)(=O)=O)n1 N1(C(C(CC#CC)NC(=O)Cc2ncccc2F)=O)CC2(CCCCC2)C1 c1(CC)nc(C)oc1C(=O)NCCc1ccc(CNC(C2CCCC2C)=O)cc1 C1(C(=O)NCCCOCC#C)CCN(C(C2CC=CCC2)=O)C1 N1(C(Cc2c(C)n[nH]c2)=O)CC(NC(c2ccc(CO)c(F)c2)=O)CC(C)C1 n1(CC)ccnc1CNC(=O)C(C1CCN(C(C2(CC(C)C)CCC2)=O)C1)C N1(C(Cc2c(C)ncnc2C)=O)CCCC1C1CCCN1C(=O)CCOC1CC1 c1(CSCC(=O)OC(c2ccc(F)cc2)C(=O)OC)ccc(C#N)cc1F N1(c2cc(C)c(NC(=O)NS(C)(=O)=O)cc2)CCCC(C)(C(C)C)CC1 C1(NC(c2c(C)cc(F)cc2)=O)CC2CC(C1)N(C(c1ccnnc1C)=O)C2 c1(C(=O)NC2(C)CCCN(C(=O)CC=C(Cl)Cl)C2)cc(O)nc2ncccc12 C(C)(C(C)CC(C)C)(c1n(CCCOC)nnn1)Nc1ccc(F)cc1SC N1(C(C(c2ccc(C)cc2)C)=O)CCN(C(c2n[nH]c(C)c2F)=O)C(CCO)C1 C(C(O)C(=O)NCCN(C(=O)COCc1nccn1C)CC1CC1)SC CN1N=C(C(=O)NCC(CC(=O)NC2CCCC3(CCC3)C2)C2CC2)CCC1=O C#CC1(C(N2CCC2C(C)O)=O)CN(C(C2CCCCC2)=O)C1 c1(N2C(C(N3CC(C)C(NC(N)=O)CC3)=O)CCC2)cnc(C#N)c(C#N)n1 C1(C(=O)NC2CCN(c3cc(O)ncn3)C2)CC(=O)N(CCOc2ccccc2)C1 C(C1=CCCN(C(=O)CCCC2CC2)C1)NC(=O)Cc1c(F)cccc1Cl C1(NC(C(CC)(C)O)=O)CN(C(=O)CCn2cnc3ccccc23)C2(CCC2)C1 N1(C(C(C#C)(C)C)=O)CCC(CC(N)=O)(NC(c2ncccc2SC)=O)CC1 C1(CNC(c2ncn(C)c2)=O)CC2(CC2)CN1C(=O)CC(=O)NCC1CC1 N1(c2cc(C)c(C#N)cn2)CCC2(CN(C(=O)Cc3ccnn3C)CC(C)O2)C1 Cc1ccc(OC2CCN(C(=O)C(N)Cn3cccn3)CC2)cc1F C1(NC(CCC=CC)=O)CCN(C(=O)CCn2cccnc2=O)C(C)C1 N1(CC(=O)NCCN(CCC)C(c2ccc(COC)[nH]2)=O)CCCC1C C#CCC(O)C(=O)NC(C)CCNC(=O)CC1(CCCC)CC=CC1 C1(C(N2CCC(C)(NC(CC3(C)CC3)=O)CC2)=O)CC2(C1)CC1(CCC1)C2 CC(C)(C)C(O)C(=O)NCCC1(NC(c2cc(C(C)(F)F)on2)=O)CCOCC1 N1(C(=O)OCC)CCC(O)CC1CC(=O)NCC(C)OCCO C(=O)(CCC(=O)NCCCN(C1CCCC1)C(c1ccsn1)=O)NCC C1(NC(c2ccc(SC)o2)=O)CCC2(CC1)CN(C(=O)CC(C)N(C)C)CCO2 c1(C(N2CCC3C(NC(C4N(C=O)CCOC4)=O)C3C2)=O)c(F)cc(Cl)cc1F c1(OC)cc(C(N2CC3CC3(NC(=O)C(C(C)C)N3CCCC3=O)C2)=O)ncn1 C1(N(C(=O)CC2(C)CC2(Cl)Cl)C)CCCCC1NC(c1cn(C)c(O)n1)=O CCC(CC(=O)NC(CC1CC1)C(N1CCN(C(C)(C)C)CC1)=O)CC(C)C C(=O)(N(CCC(=O)OC)OC)c1ncc(OC)nc1.N12CCC(C1)CC2 N1(C(C2(COC)C=CCC2)=O)CC2CCC(C1)C2NC(c1cnc(C(C)C)o1)=O C1(C(=O)NC(C2CCCCC2)(C#C)C)CC2CCC1C(=O)C2 C(CCNC(c1nc(C)c(C)s1)=O)(C(=O)NC(c1cnc[nH]1)C)OC C1(CNC(c2c(CC)scc2)=O)CCCCN1C(=O)CCn1ccnc1C N1(C(COCC(C)C)=O)CCN(C(=O)CC(O)CCc2ccccc2)C(CO)C1 Cc1cccc(NC(=O)CCC2(NC(C3CC(F)C3)=O)CCCC2)c1 N1(CCC(N2CCC(C3N(C(c4cc(C)[nH]n4)=O)CCC3)C2)=O)CCC(C)CC1 Cc1cc(Br)ccc1C(=O)NCC1COCCN(C(=O)CC(C)O)C1 Cc1ccnc(C(N2CCCCC2CNC(C2CC2c2ccc(F)cn2)=O)=O)c1 C(=O)(C(CC(F)F)C1CCC1)OCc1n(C)ncc1Br c1(C(CC)NC(=O)N(CCF)CC)csc(C)c1 c1(C(=O)NC(C)C(CO)NC(C2CN3CCN2CC3)=O)[nH]nc2ncnc(O)c12 c1(CC(=O)N(C)CC2CN(C(c3cscc3F)=O)CCO2)cccc2sccc12 Cc1cnn(C(C)C(=O)NC2(CCNC(=O)CSC3CCOC3=O)CCCC2)c1 c1(NC(C(C)OCCOS(C)(=O)=O)C)ccc(OCC(=O)O)cc1 c1(CCC)ccc(CC(N2CCCC2Cc2cn(CCCCOC)nn2)=O)cc1 C1(N(C(=O)CN(C2CC2)CC)CC)CCCN(C(=O)C(CO)c2ccccc2)C1 C(=O)(C1=CC2(CCOC2)C1)NCc1c(C(N2CCC(C)(C(=O)NC)C2)=O)c[nH]n1 CC(CC(=O)N1CCC2(CC2)CC1C(N1CC(n2ccnc2)C1)=O)C(C)(C)C C=CCC(CNC(=O)C=CC1CCCN1C)C(=O)NCc1nnc(O)o1 C=CC(C)(CCOC)C(=O)N1CCC(CF)(NC(c2cccc(F)c2Cl)=O)C1 N1(C(c2cnc(NC(C)=O)o2)=O)CC(NC(c2ccc(C3CC3)s2)=O)CC(F)C1 Cc1cc(C(N2CCCC(CO)(NC(=O)C=C3CCC3)C2)=O)c2ccccc2n1 CC1CCC(CC(N2CSCC2C(=O)NC(C)(CO)C2CCCC2)=O)CC1 CC(CCCCNC(c1csc(S)n1)=O)NC(C1CCCC1(C)C)=O N1(C(C23CCCCC2C3)=O)CCC=C(C(=O)NC2CC(OC(C)(C)C)C2)C1 c1(OCC)cc(C)ccc1C(=O)N(C)CC1COCCN1c1nc(Cl)c(C#N)s1 C12(NC(=O)C(C3CCC3)C3CCC3)CC1CNC2.c1(C(C)=O)cnc(C2CC2)o1 Cc1nc(CNC(C2C3CCCC23)=O)oc1C(=O)Nc1ccc(N(C)C)nc1 C1(CC(=O)OC)CC2(CCN(CC(=O)N(C)CC3CC3)CC2)CO1 c1(NC(c2nc(C(C)OCC)sc2)=O)ccccc1-c1noc(C(F)(F)F)n1 c1(C(N2CC(SC)C(NC(c3coc(C(C)C)n3)=O)C2)=O)cc2c(ncn2C)s1 CCCC(C(=O)NC1CC1NC(c1ccc(O)nc1)=O)NC(=O)OC(C)(C)C C1(OC)CN(C(=O)CCCCN(C)C)CC1NC(=O)Cc1ccc(Br)s1 CC1(C(=O)NCC(=O)NCC(=O)NCCOC(N)=O)CCC(=O)C1 C(C(C)NC(=O)CCC)(C(C)C)NC(C(C1CCCC1)OCC)=O.C1(=O)CO1.CC C(=O)(C1c2ccccc2C2CC1C2)N1CCN(C(C2CC(C)C2)=O)CC1C(F)F C=CC(C)CC(=O)NC(C12CCC(CC1)C2)CNC(C1CC(=O)N(C)C1)=O N1(NC(=O)COc2c(O)ncc(C)c2)C(=O)NC2(CCCC(C)(C)C2)C1=O N1(C(c2c(C)csc2)=O)CCOCC(C(=O)N(CC(O)CN(C)C)C)C1 C(CS(C)(=O)=O)(C(=O)O)NC(C(=O)NC1C(C)CN(C(=O)OC(C)(C)C)C1)=O c1(N(CCOC)CCNC(C2(C)CCCNC2=O)=O)ncnc2c1nnn2C C(=O)(CC(O)CC(C)(C)C)N1C(C(=O)NC2CC(C)(CC)OCC2)CCCCC1 C1(C(=O)NCC(N)=O)CN(C(=O)Cc2cn3ccccc3n2)CCC1(F)F C(=O)(CCCC(=O)NC1(C(N2CC(=O)NCC2C)=O)CC1(C)C)OC N1(C(C2(CNC(CC3CC(SC)C3)=O)CC3(CC3)C2)=O)CC2(CCC2O)C1 C(CNC(=O)CC1CC(SC)C1)(C(C)(C)C)NC(C1CC(C)(CC)C1)=O N#CC1(O)CC(CN(C(N2CCCC2C2CC(F)(F)C2)=O)Cc2ccco2)C1 C1(C(=O)NC(C(C)SC)C)CC2(CCC2)CN1C(=O)C(C)N(C)C c1(OC)cc(C)c(C(N2CC(C)OC(C)C2C)C(=O)NC2CC(F)(F)C2)c(C)c1 C=CC(C)(C)C(=O)N1CC(OC)C(NC(c2cnc(N3CCOCC3)s2)=O)C1 c1(C(c2ccccc2)OC)nc(C)cc(=NC2CC(c3ccccc3)C3CC23)[nH]1 C1(CN(C(=O)C(=O)N2CC(N(C)C)C2)C)CCCCC1CC(F)(F)F O=S1(=O)CCCC(n2nc(-c3cccnc3)nc2-c2cc(C3CC3)no2)C1 CC1CCN(C(=O)C(F)C2CCCC2)C1C(=O)Nc1cnn(C)c1C(N)=O C(=O)(CC(F)(F)F)N(C1CCCC1)CCCNC(=O)C=Cc1cn[nH]c1 c1(N2C(C)CC(NC(c3cnc(CC)nc3O)=O)C2)nc2ccc(F)cc2o1 C1(C(=O)NCC(CC)Nc2nccc(-c3cnccn3)n2)CCS(=O)(=O)N1 c1(C(=O)NCC2CCCC2NC(c2cnn(C(F)(F)F)c2)=O)ccc(O)nc1 C(CC(C)(c1nnnn1CCCC1CC1)NCC1(n2cc(Br)cn2)CC1)N(C)C C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC(CNC(c1cc(C)oc1C)=O)(C)C N1(C(C2OCCN(C)C2)=O)CC2C3CCC(C2C1)N(C(c1cc(N)ccn1)=O)C3 c1(C(N2CCC3(NC(c4c(C#N)scc4)=O)C(C2)C3)=O)nccn2ccnc12 c1(C(N(CC(=O)NC2CCS(=O)(=O)C2)C)=O)cnn2c1OCC(F)C2 C(=O)(C(F)(F)CF)N1CCC(OC(=O)Nc2ccccc2)C1.O=C1CN1 N1(C(C(CCC)OC)=O)CC(NC(=O)C=Cc2ccsc2)C2(CC2)C1 C1(=CC(=O)NCCC(C)NC(=O)C2=CCCSC2)CCCCCC1(F)F c1(NC(C23CC(NC(c4cccc(F)n4)=O)(C2)C3)=O)nc(Cl)ccc1[N+](=O)[O-].O=CCCl c1(C(=O)NC2CCC(Nc3cc(OCC)ncn3)CC2)n[nH]c2c1CCC2 C(=O)(C1CCCc2ncc(C)n21)N1CC(CC)N(C(=O)COCCF)CC1 C(=O)(C1=CCCC1(C)C)NC1CCN(C(c2c(C)nc(C(C)C)nc2)=O)C12CC2 C#CC1(O)CC(C(=O)NCC(C)CNC(c2cc(C(C)(C)C)oc2C)=O)C1 c1(-c2cncc(OCC)c2)ncc(Nc2ccc(O)c(OC)c2)c(COC)n1 CC(C)CC(CN(C(C)CO)Cc1ccccc1)C(=O)OCc1ccccc1 c1(C(=O)NC(C)CC2CN(C(C3CSCCS3)=O)C2)cc2c(cn1)OCCO2 N1(C(CC2CN(C(C3(CC=C)CC=CC3)=O)CC2C)=O)CCC(O)CC1C C1(C(=O)NC(CCOC)CNC(=O)Cn2nnc(C)n2)(CO)CCCCO1 CC(C)C(F)(CNC(=O)CC1CC(N(C)C)C1)C(=O)NOCC(C)(C)C C(=O)(CCCCC(=O)N1CC(F)CC1C(N1CCC(F)(CO)C1)=O)OC C(=O)(C(C)(C)CCNC(=O)C=C(C)C1CC1)N(CCCOC)CCO C(=O)(CCCC(F)F)NCC(C)CN(C)C(c1ccc[nH]1)=O c1(C(=O)NC(CNC(CC(CC)C)=O)C2CCC2)cc([N+](=O)[O-])c2nsnc2c1 Cc1cn2c(=O)c(C(N3CC(CNC(=O)C(=O)N(C)C)CC3C)=O)cnc2s1 CC(O)(CC(=O)NC1(CNC(c2ccc(CCO)cc2)=O)CCOC1)C(F)(F)F c1(NC(N2CCCC(c3n(C(C)C)c(S)nn3)C2)=O)cc2c(Br)cccc2[nH]1 c1(OC)cc(C(=O)OC)ccc1Oc1ccccc1I.C12(COC1)CNC(=O)N2 C1(CNC(=O)N(C(c2cccc(C(F)(F)F)c2)CO)CCl)CCc2cccc(Br)c2C1 c1(C(=O)NC(C2CN(C(C3(C)CC(F)C3)=O)CCO2)C)cc2n(n1)CCC2 C(=O)(C(CCOCCO)NC(c1ccc(O)nn1)=O)N1CC(C)(N(C)C)C1 c12nc(cc(C)n1)N1CCCC1C2.C1(C(C)=O)CCCN(C(=O)C#CC2CC2)C1 N1(C(c2cn(CCCC3CC3)nn2)C)CCN(CCC2CCCC2)CC1 C(=O)(N1CC(C)(O)CO1)C1CC(NC(C(COC)(C)OC)=O)C1 c1(NC(N2CC(C)(C(F)(F)F)OCC2)=O)ccccc1S(=O)C(F)(F)F c1(C(N2C(CNC(C(C=CCCC)O)=O)CC2)=O)ncc2ccccc2c1O c1(C(=O)NCCCN(C)C(c2cccnc2C2CC2)=O)ccc(O)c(Br)c1 Cc1nn(C)c(Cl)c1C(=O)NCC(CO)NC(c1cnn[nH]1)=O C#CCC(C(=O)NCC1(CN(C)C(C2C(C)C2(F)F)=O)CC1)C1CC1 C12(C(=O)NC(C)CCC(=O)NCC3CCC3(F)F)CC(C)(CCO1)C2 N1(C(c2cc(CC)nn2C)=O)CCN(C(C2CCCC2F)=O)C(CO)C1 N1(CCC(N2CC(C)C(NC(=O)COCC3CCCC3)C2)=O)CCP(C)(=O)CC1 C1(CC(=O)N(CC(C2CC2)OC)C2CC2)C2CN(C(=O)Cn3ccccc3=O)CC12 C(CC(C(=O)N1CC(C(=O)NCC2NC(=O)NC2=O)C(C)C1)OC)OC Cc1ccc(NC(NOC(=O)OC(C)(C)C)=O)s1 Cc1cc(NC(c2cc(CNC(C34CCC(CC3F)C4)=O)no2)=O)cnc1C C1(C(=O)NC2CCC(C(F)C(=O)N(CCCC(C)C)C)C2)(OC)CCSC1 C1(C(=O)NC2CCN(C(CSCCC)=O)CC2C)CNC(=O)CC1(C)C C(=O)(C1CCCc2sccc21)NC(CCNC(c1c(C)nns1)=O)(C)C S(=O)(=O)(c1ccc2c(c1)CC(=O)N2)NCC(=O)NCC1CN(C(C(C)OC)=O)C1 N1(C(C2C(OC)CCCC2)=O)CCN(C(C2CN(C(=O)NC)C2)=O)C(CO)C1 c12cncc(c1)C(=O)N(CC)CCN2C.C1(NC(CC)=O)CCN1C1CC1 N1(S(CC)(=O)=O)CCCCC1C(N1CCCC(CNC(c2ccnn2C)=O)C1)=O Cc1ccc(-c2noc(COC3CC(NC(C4CCCO4)=O)C3)n2)cc1 N1(S(c2cccc(Cn3c(N)nnn3)c2)(=O)=O)CCCC2(CCC(=O)N2)C1 C12C3CCC(C3)N1C(=O)C2.c1(C(=O)NCCCCCN(C)C)cccc(F)c1F C1(C(=O)NC(COC)C(=O)OC)CCN(C(c2conc2C)=O)C12CC2 c1(C(=O)NCC(CNC(C(C)c2ccon2)=O)O)ccc(O)cc1 C=CCC(C(=O)N(CC(C1CCC1)OC)C)NC(c1cccnc1S)=O C(CCCCC(=O)N(CCCO)C)N(C(C1N(CC)CCOC1)=O)C C1(NC(Cn2cc(-c3ccc(C)nc3)nn2)=O)CC(=O)NC1(C)C C(CCCCC(=O)NCCc1ccccn1)N(C(=O)CC1CC1C1CC1)C c1(SCCC(N2C(CNC(C3CC34CC4)=O)CC2)=O)ccccn1 c1(C(=O)NCC(CC=C)NC(=O)C(N2CCOCC2)(C)C)ccc(CO)c(F)c1 c1(NCC2CCCC3CN(C(CCCC)=O)CC32)nc[nH]c2ncc(C(N)=O)c1-2 CC1CC(NC(=O)C(F)(F)c2ccccn2)CN1C(=O)CN1CCC(C)(C)C1 Cc1nc(=N)[nH]c(=NCC(C)CNC(C23CCC(CC2)CC3)=O)[nH]1 C=CCC(F)(F)C(=O)NCC1(CNC(=O)CCSCC(C)C)CC12CCC2 N1(C(c2ccc(CC)cc2)=O)CCC2(NC(=O)CN3CCCCCC3)CC2C1 c1(N2CCC(CC=C)(CNC(=O)C(C)C(C)C)C2)cc(=O)n(C)c(=O)n1C N1(C(C(C)OCC=C)=O)C(CNC(C2CC2OC(C)(C)C)=O)CC2CCCC12 C1(CCC)(NC(C(CC)F)=O)CCCN(C(=O)CCc2c(F)cccc2F)C1 c1(C(C(=O)NCC2CC(NC(c3nc(CC)sc3)=O)C2)O)ccc(Cl)c(Cl)c1 c1(CN(C2CN(C(c3c(OC)ncc(Br)c3)=O)C2)C)ccc2c(c1)CCCO2 N1(CC(=O)N(CCNC(=O)Cc2cccs2)CC)CCC(C)(O)C1 N1(C(C(CC)SC)=O)CC(C(=O)NCCS(C)(=N)=O)CCC1C c1(CNC(=O)CC2CCN(Cc3ccsc3)C2)cc(F)cc([N+](=O)[O-])c1 CC(C)C1=NOC(C)(C(=O)NC2CCCC(NC(=O)Cc3cnoc3)C2)C1 C1(C)(C(=O)NC(CCNC(c2c(OC)ncnc2C)=O)C)Cc2ccccc2N1 C12(C(N(C)Cc3cccnc3O)=O)CCC(NC(=O)CC3CC3(C)C)(CC1)C2 C=C(C)C1OCCC1C(=O)NCCCC(N1CCN(C)CC1C)=O c1(C(=O)NCC2(C)CCCN2C(C2CC23CC3)=O)nc[nH]c2nccc1-2 CC1CC(NC(=O)CSC2CCC2)CN(C(=O)CNC(c2ccccn2)=O)C1 C(CN=C(NC1CC1)N1CCC(CS(C)(=O)=O)C1)c1c([N+](=O)[O-])ccc(OC)c1 C(CN=c1ccn2c(Br)cnc2[nH]1)=CCNC(c1c(F)ccc(C)c1)=O Cn1cc(C=CC(=O)NCCc2ccc(CNC(C3C4COCC34)=O)cc2)cn1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(=O)C(S(C)(=O)=O)C2CC2)CC2(CCC2)C1 CS(=O)(=O)c1ccc(Cl)c(S(=O)(=O)N2CCC(O)(c3ccc(F)nc3)CC2)c1 N1(C(c2n(C)ccn2)=O)CCCN(C(c2cc(C(F)(F)F)ns2)=O)CC1 C1(NC(c2cc(C)ncc2)=O)CCN(C(C2CC2C2CC2C)=O)C12CCC2 C12C(C1(C)C)COC(C)C(=O)N2.c1(C(=O)NC2CCCC2)cnn(C2CCC2)n1 C1(CC#N)CCCN(C(=O)Nc2ccc(OCCCc3ccc(Cl)cc3)cc2)C1 C(CS(N)(=O)=O)N(C)C(C1CC(O)(CNC(C2CCSCC2)=O)C1)=O c1(CCCC)ccc(C(=O)NC2C=CCN(C(=O)Cc3ncoc3C)C2)cc1N c1(OC)cc(C(=O)NC2CCC2NC(=O)CC(C)F)cc(OC)c1O C=C(C)C1CN(C(C23CC(C)(CN2C(c2cc(C#N)oc2C)=O)C3)=O)CCO1 C(=O)(CC(C)CC(F)(F)F)N1CCOCC(NC(C(C)NS(CC)(=O)=O)=O)C1 c1(CC)cc(-c2ccc(C(N3CC(F)CC3C(=O)OC)=O)nn2)ccc1F C1(CC(=O)NC2CC3CN(C(C4(O)CCCC4)=O)CC3C2)CCCC2(CCC2)O1 C1(O)(CC)CCC(NC(=O)C=CCN(C(=O)COC2(C)CCC2)C)CC1 C(=O)(C(C)(C)CCCO)N1CC(CC)N(C(=O)COCCOC)CC1 C(=O)(C1CCc2cc(F)ccc21)N1CCC(F)(CNC(=O)CCC2CC2)CC1 C12(C(=O)NCC3(O)CCCN(C(CCCCC=C)=O)C3)CCC(CO)(CC1)CC2 c1(CC(=O)NCCCOCCNC(C2CSCCS2)=O)noc2cc(F)ccc12 c1(C(C)NC(C(Cc2cc[nH]n2)NC(CC=C=C)=O)=O)ccccc1F C(CC(N)=O)(C(=O)NC1CCN(CC2CC2)C1)NC(C1(C#N)CCCC1)=O CCC(C)CC(=O)NC1CC1NC(c1ccncc1Cl)=O C1(C(=O)NCCCCNC(C=C2CCC(C)(C)CC2)=O)CCC(C2CCCO2)O1 c1(OC)ccccc1NC(c1cn(C2CN(C(=O)COCC(F)F)C2)nn1)=O c1(OC)cc(C)cc(C(=O)NCC(CNC(c2cc(O)nc(O)n2)=O)OC)c1C C1(O)(CCNC(C2CCOC(=O)N2)=O)CCCN(C(=O)CCOC2CCC2)C1 n1(C2CCN(C(C(NOC)=O)=O)CC2)ncc2c1CN(C(=O)CCC(N)=O)C2 CC(C(=O)NC1CC(C(F)F)(NC(C2CC23CC3)=O)C1)S(N)(=O)=O C12(NC(C3C(CC)C3)=O)CCCN(C(=O)CCc3cc(Cl)cs3)CC1C2 C1(C2CC2)(C(=O)NCC2CCC(=C)CC2)CN(C(=O)CC(C)n2cccn2)C1 C1(F)(C(N(C(C(=O)N(CC(CCC)O)C)C)C2CC2)=O)CC=CCC1 C1(CNC(c2ccc(F)s2)=O)CCC2CN(C(=O)CC3CCC=CCC3)CC12 C#Cc1cccc(C(N2CCCC(CNC(=O)CC3CCCO3)C2)=O)c1Cl N1(C(C(CC=CCC)C)=O)CCOCC(C(=O)NCc2cncc(C(N)=O)c2)C1 C(=O)(C(C)(C)NC(C)=O)NC1CC(C(N(CCN(C)C)CC)=O)C1 C(=O)(CCCC#N)N(CCC(=O)N(C)CCc1ccccn1)CCO c1(C(N(C2CN(C(C(=O)NCC)=O)CC23CC3)C)=O)ccn2c(C)cnc2c1 c1(N(C2CN(Cc3c(O)cccc3Cl)C2)C)ncc2[nH]ccc2n1 N1(CC(=O)N(CCSC)CC)CC(=O)Nc2ccccc21 C1(NC(c2cccnc2F)=O)CCC2CN(C(C3CC4C(C3)C4(F)F)=O)CC2C1 CC(C)C(C)(CNC(=O)C(C1CC1)NC(C1CC(=O)C12CCC2)=O)C(C)C c1(C(=O)NCC(C)N(C(=O)C(Cl)=CCl)C)ccnc(N2CCC(C)C2)c1 CCCC(C(O)C(=O)NC1(CCOC)CCC1)NC(c1coc(C(C)C)n1)=O Cc1ccc(-n2cc(C(C)(C)NC(=O)C(c3cncn3C)N(C)C)nn2)c(Br)c1 Cc1ccc(CC(=O)NCC2CN(C(=O)CC3COC(=O)C3)CCO2)c(Cl)c1 N1(C(C(C)(C2CCC2)NC(Cc2ccc(C)o2)=O)=O)CCC(C(C)(C)C)CC1 c1(OC(N(C(C(=O)N(C)C)=O)Cc2ccccc2)=O)cncc(C(N)=O)c1 N1(C(C(CCC)C=O)=O)CCC(NC(=O)CC(CC)CC)CC(C)(C)C1 N1(C(c2c(N(C)C)cccc2)=O)CCC2(CC2C(=O)NC2CCC(F)(F)C2)C1 N1(C(=O)CCCc2cccs2)CC2CCN(C(=O)C3CCc4nccn43)CC2C1 n1(CCC)cc(Cl)c(-c2nc(-c3coc(SC)n3)no2)n1 C1(C(N2CCC(NC(C(CC=C)C)=O)(CC)CC2)=O)CCCCC(F)(F)C1 CCC(O)CC(=O)N(CCCNC(c1cccc(Cl)n1)=O)CC Cc1sc2ccccc2c1C(C(=O)NCCC1CC1)N(CCC(C)C)C C1(C)(C(=O)NC(C)C(C)NC(=O)CC(C)(F)F)CC(C#N)C1 C(c1cnccn1)=CC(=O)NC1CC(CCC(=O)N(CC#CC)CC#C)C1 c1(C(N2C(C(=O)NC(C#N)C(N)=O)CC2)=O)c(F)cc(Br)cc1Cl C1(CCC)CN(C(C2CCCCCC2)=O)CC1NC(=O)Cn1c(C)ccc1C N1(C(CCCCC=C)=O)CCC(C2CC2)(CNC(c2cc(C)nc(C)c2)=O)C1 C1(CNC(c2cc(COC(F)F)on2)=O)CCCCC1NC(c1cnns1)=O c1(CNC(C(F)=C(C)C)=O)ccc(C(=O)NCCN2CC3CC3C2)o1 C1(C(C(=O)NC(C)(C)C)N(C(C(=O)OC)C)C)CC12CCOCC2 c1(C(=O)NCC2(F)CN(C(CC3(C=C)CC3)=O)C2)ncncc1OC c1(OC)c(Br)ccc(F)c1CN1CCOCC1CC(=O)Nc1onc(C)c1Cl c1(C(C(=O)OC(=O)NCC(CNC(C)(C)C)CO)OC)ccccc1 C(C(CC)(CC)NC(=O)CC1CCC(=O)NC1)NC(C(CC)C1CCC(=O)N1)=O c1(C(=O)Nc2ccc(C#C)cc2)cccc(C(=C)C)c1.C1(CCF)C(=O)N1 C(CC(C)(C)C)(C(=O)NCc1cncc(C(N2CCC(C)(C)C2)=O)c1)OC c1(C(=O)NC2CCN(c3c(Br)cnc(C)n3)C2)nc(C(C)C)c2ccccn12 C1(C(=O)NCC2(O)CCN(C(Cn3c(C)ccn3)=O)C2)CN2CCN1CC2C CC(CC(N)=O)C(=O)N(C1CCCN(C(C2(C(c3ccoc3)=O)CCC2)=O)C1)CC C1(C(=O)NCC2OCCN(C(C3C(CC)CCC3)=O)C2)CC2(CCC2)CO1 N(C(=NCc1ccc(N2CCOC(C)C2)nc1)NCC1(C)CC1)C(C=C)C c1(-c2ccc(C(=O)Nc3cnc(OCCOC)nc3)nc2)cc(F)ncc1O N1(C(CSCCCC)=O)CC2CCC2(CC(=O)NOCCCC(F)(F)F)C1 c1(C(=O)NC2C(C)CCN(C(c3nncn3C3CC3)=O)C2)ccn2nnnc2c1 C(=O)(CC(C)(C)CNC(C1CN2CCC1CC2)=O)NCc1ccc(C)o1 C(=O)(C(C)C(F)(F)F)N(C1CCN(C(c2coc(CN(C)C)n2)=O)C1)CC#C C1(C(=O)NC2C(NC(c3ccc(N(C)C)cc3)=O)CCC2)COCC(C)(C)O1 C12(NC(c3cc(C(C)C)[nH]n3)=O)CC1CN(C(c1ncncc1Cl)=O)C2 C(=O)(C(CN(C)C)NC(C1(C2CCCC2)CC1)=O)N(CCC#C)C CN1CCCC(CNC(c2coc(CNC(=O)CCc3cnoc3)c2)=O)C1 CC1CCC(C(=O)NC2CCC(C(N3CCCC3CCC(C)(C)C)=O)C2)O1 N1(S(CC(=O)OCC)(=O)=O)CC(NC(c2c(F)cccc2I)=O)CC(C)C1 C(=O)(C(CC1CCCC1)N(C(CSC)CC(=O)OC(C)(C)C)C)NC(CC)C Cc1ccc(C(C)N(C(=O)CNC(=O)CCCN(C)C)C)c(C)c1 c1(C(=O)NC)cccc(C(=O)NC(C)(C)C(C)NC(C2CN(C3CCOC3)C2)=O)c1 C(=O)(C1=CCOCC1)N1C(CNC(c2c(SC)cccc2)=O)COCC1 N1(C(C23CC(NCc4cc(F)ccc4Cl)(C2)C3)=O)CCC(O)C(F)C1 CC(C)C(C)CC(=O)N1CCC(C(C)C(=O)NCC2=NOCC2)CC1 c1(CC)cccc(CC(=O)NC2CCC2NC(C2CC(C)(C)CO2)=O)c1 C(CNC(=O)CSCC1CCCO1)(CC(F)(F)F)NC(=O)CSC1CC1 Nc1cc(C(=O)NCC2(NC(=O)CC(F)(F)F)CC2)cc(O)c1Cl C1(NC(COCCOCC#C)=O)CCN(C(c2csc(CO)n2)=O)CC12CCC2 c1(C(C)(C)C)ccc(Cl)cc1C(N1CC(C(N)=O)(CNC(=O)Cc2cn[nH]c2)C1)=O C1(C(=O)N(C(C)CC(=O)NC(CN2CCCC2)CO)C)(COC)CCCC1 n1(CC)nc(C(=O)N(CC(C)O)CCNC(=O)C(O)c2cnc[nH]2)c(C)n1 C#Cc1cc(C(N2CC(NC(=O)C(C)(C)CC=C)C3(CC3)C2)=O)cc(Cl)c1 C12(C(=O)NCCc3cocn3)CCC(CC1)N(C(C1(O)CC3CCC1C3)=O)C2 c1(C(=O)OC(C)(C)C)cc(O)n(C(=O)CC[SH2]CC=Cc2ccc(F)cc2)n1 n1(CC)ncc2c(NC(CNC(=O)CS(=O)(=O)C3CC3)C(C)C(C)C)ncnc12 N1(C(C2C(CC)CCO2)=O)CCCC2(C1)CN(C(=O)C(C)(C)n1ccc(C)n1)C2 C(=O)(C1=CCCOC1)N(C1CCN(C(c2c(CCC)nco2)=O)CC1)CCCC Cc1cc(Cl)c(C(=O)NCC(O)CNC(=O)C(C)C2CCCO2)cc1C C1(C(N2CC3CC(NC(C4CSCC(=O)N4)=O)C3C2)=O)(OC)CCS(=O)(=O)C1 Cc1cc(=NC2CCc3nnc(N4CCC(CN5CCCC5)C4)n3C2)[nH]cn1 C(=O)(C1=CCOC1)N(C1CCCCC1)CCNC(c1nc(CCCCC)sc1)=O c1(C(N2CCN(C(c3cnc(SC)s3)=O)C(C)C2C)=O)cnc(C)c([N+](=O)[O-])c1 c1(C(N2CC(CC)N(C(=O)COC(C)C)CC2)=O)cc2c(s1)C(C)(C)CCC2 N#CC12CN(C(=O)Cc3cnn(Cc4ccccc4)c3)CC1CS(=O)(=O)C2 S(=O)(=O)(c1ccccc1CCC#N)NCc1c(C)cc(F)cc1 CC(C)CC(O)C(C)C(=O)N1CCC(NC(c2ccc(CO)s2)=O)C1C(C)(C)C N1(CC2CCCC(C(=O)OC)C2)C2CCC1CC(=O)NC2 C1(NC(c2cccc(OC)c2)=O)CC2CN(C(=O)Cc3nncn3C)CC2C1 CC1(C)CN(N2CCC(c3ncccc3Cl)CC2)CC1CO C(=O)(C1SCCc2sccc21)NCCNC(c1c(C)n[nH]c1)=O C1(CNC(C=C(COC)C)=O)CCN(C(=O)CCC(=O)c2ccccn2)C12CC2 N1(C(C(CCC2CC2)NC(CCCN=[N+]=[N-])=O)=O)CCC2(CCOC2=O)C1 C#CCC(C(=O)NCCC(O)CNC(c1cnccc1C)=O)C1CC1 S(=O)(=O)(c1cccnc1N1CCC(F)(F)C(CO)C1)NC1CC(OC)C(OC)C1 N1(C(c2n(CC)nnc2)=O)C(C(=O)N(c2ccccc2)CCO)CCC1C c1(C(=O)NC2C(CNC(=O)CCc3nc[nH]n3)COC2)cc2ncccc2o1 S(=O)(=O)(c1ccnc(F)c1)Nc1cccc(NCC(=O)OC)c1 C(CCCC(CO)NC(=O)CC(=O)N(C)C)NC(c1cccc(OCCC)c1)=O Cc1cccn(CC(=O)NC2(C)CCN(C(C3CC(C)(F)C3)=O)C2)c1=O C(=O)(C1=CCC(NC(C2(O)CCC2)=O)C1)NCC(CC)N1CCCC1 c1(C(=O)NC)cccc([N+](=O)[O-])c1Cl.C(=O)(C(=O)NCC(C)(C)O)NCCOCC S(=O)(=O)(c1cccc(F)c1)NC(c1ccccc1C(N1CCC(S(N)(=O)=O)C1)=O)=O CCC(C)(CC)C(=O)N1CCC(C)C(CNC(c2csc(-c3nc[nH]n3)n2)=O)C1 CCCCC(=O)NC1CCN(C(C23CSC(C2)C3)=O)C1 Cc1csc2c1CN(C(=O)CC1CC(C)(C)OC1(C)C)CC2 CCCN=C(N(C)CCOc1ccc(Cl)cc1)N(C)CCc1ccn(C)n1 c1(C(N(CCCNC(C2CC(C3CCC3)C2)=O)C)=O)ccc(S(N)(=O)=O)cc1F n1(CC)cc(Br)c(CC(=O)NCC(C)(C)Cn2cc(C(C)(C)C(C)C)nn2)n1 c1(C(=O)NC)cc(=NCC(C)SC)nc(-c2ccncc2)[nH]1 C1(C(C)NC(C23CC(C#N)(C2)C3)=O)CCCN(C(=O)Cn2cnnc2O)C1 C1(NC(CCCOCCOC)=O)CCC(C)(CNC(c2csc(S)n2)=O)C1 C1(CC)CC(O)CCN1C(=O)CCCC(C)NC(=O)CC1OCCO1 CC1(C)CC(NC(c2ncoc2C2CCC2)=O)CN(C(c2ccccc2O)=O)C1 c1(NC(Cc2c(-c3c(CC)scc3)cccc2)=O)c(OC)cccc1O C1(NC(c2ncc(OC)nc2)=O)CCC2CN(C(=O)Cc3n[nH]c(C)n3)CC2C1 N1(C(C(C)SCC)=O)CC(C(=O)NC(c2ncc[nH]2)C)C2(CC2)C1 c1(C(=O)NC2CN(CC(=O)N(C(C)C3CC3)C3CC3)C2)cc2cccnn2n1 c1(C(N(C)CC2CCN(C(c3c(CC)c[nH]c3)=O)C2)=O)cc(F)ccc1C(F)F Cc1csc2ncc(C(N3CC(CNC(c4coc(C(C)C)n4)=O)C3)=O)n12 c1(CCC(N2CCC(c3ccc(F)cc3)CC2)=O)cnc2ccccn12 N1(C(c2cc(C)on2)=O)CC2CC(C1)C2NC(=O)CCNc1ccc(N)cc1 N1(c2nccc(OC)n2)CC=C(CNC(=O)CN2CC(=O)N(C)C2=O)CC1 C(C1=CCN(C(=O)CN2CCC(C)CC2)CC1)NC(C(CCOCC)OC)=O c1(C(N2CCC(NC(C3(SC)CC3)=O)C(CO)CC2)=O)c(Cl)nc2sc(C)cn12 CC1C(CC(=O)NCC2(F)CC(NC(=O)C(C)c3ccsc3)C2)C1(F)F Cc1cc(CC(=O)N(CC(C)NC(c2c(Cl)csc2Cl)=O)C)cc(C)c1 C(=O)(CS(=O)(=O)CCO)N(C1CCN(C(=O)CC2CCC2(C)C)C1)CCC c1(C(=O)NC2CCN(c3ccc(CC)cc3)CC2)ccc(N)c(F)c1F C1(NC(C2(CCC)CCC2)=O)(CNC(C2CCC3CC23)=O)CCCC1 c1(-c2ccc(OC)nc2)ncc(C(=O)NCc2cccnc2)cc1OC c1(OC)cc2c(cc1C(=O)NC1CC1NC(c1ccccc1F)=O)CCC2 C1(C(=O)NC2CCC2)CCCN(C(C2(Br)CC2)=O)C1.N1CCSCC1 C1(C)(CNC(C(F)=CC)=O)CCC(NC(=O)C=Cc2nccs2)CC1 C(CN=C(NCC1CC2CCC1CC2)N1CCC(C(C)(C)C)C1)CS(=O)(=O)N.CS c1(SC)ccc(C(=O)N(CC(C)N(C)C(C2CCN(C)C2=O)=O)C)c(Cl)c1 N1(C(C2CC23CCOCC3)=O)CCC(O)C(F)(F)C1.c12c[nH]nc1CCNC2=O C1(C(=O)NCCC(CC)(C)O)CCC2(CC2)N1C(c1oncc1C)=O C1(O)(Cn2cc(-c3n(C)c(Cl)cn3)nn2)CCCN(C(C2CC2C(=O)O)=O)C1 c1(C(N2CCC(CNC(COCC)=O)C(C)C2)=O)cccc2c1NC(=O)CC2 N1(C(C(C)Cn2ccnc2)=O)CCCC(C)(NC(C2CCCC(C)(C)O2)=O)C1 C1(NC(C(c2cn(C)nc2)=O)=O)CC2CCC1C(NC(=O)C(F)CC1CCC1)C2 c1(C(=O)NCCC2(NC(CN(CCC#C)C)=O)CC2)snnc1C c1(C(C2CN(C(=O)C3=CCCC3)CCO2)n2cc(C(C)O)nn2)cc(F)cc(Cl)c1 C1(C(C)NC(C2C(OCC)C2)=O)CCN(C(C2CCN(C(C)(C)C)CC2)=O)CC1 N1(C(C(CC)OC2CCCC2)=O)CCC(CNC(c2ccc(C#N)o2)=O)C1(C)C N1(C(c2ccn(C(C)C)n2)=O)CCC(C)(C)C1CNC(=O)C(C)c1ccsc1 CN1CCCCCC1C(=O)NCC1(NC(=O)Cc2ccc(Cl)nc2)CCOC1 CCCCC(CC)CC(=O)N1CC(F)CC1CC(N1CCN(C2CC2)C(C)C1)=O N1(C(CC(C)(C)C)=O)CCC2(CCCN2C(C2CCC3CC3C2)=O)C1 c1(C(=O)NC2CCC(NC(c3c(C)onc3Cl)=O)C2)cc2ccccc2oc1=O CC1CCCC=C1C(=O)N1CC2CCC(NC(=O)CSc3ccncc3)(C2)C1 c1(NC(=O)NCCCCCC)cccc2c1NC(=O)CC2 C1(C(=O)NCC2CN(C(c3ccc(C(C)C)o3)=O)CC2O)CC(C2CC2)=NO1 N1(C(c2n(COC)ncc2)=O)CC(NC(=O)C(C)(C)Br)C(SC)C1 C1(NC(C(C)N(C(C)=O)C)=O)CN(C(=O)CCC2(C)CC2)CC1n1ccnn1 C=CCCCCC(=O)N1CC(OC)CC1CNC(c1cc(O)n(C)n1)=O C1(CN(C(=O)CCCC2CC2(C)C)C)CCN(C(=O)C2=CCC2)CC1 c1(C(=O)NC(C(CO)NC(CCSC)=O)C)cnn(C2CCC2)c1C c1(C(=O)NCC2N(C(C3C(C)CC=CC3)=O)CCOC2)ccc2nonc2c1 N1(C(CCC)=O)CCCCC1C(=O)NCC(C)(C)CNC(=O)CSc1cccs1 N1(C(c2cnn(C(C)C)c2N)=O)CCN(C(=O)Cc2ccc(Cl)s2)CC(O)C1 c1(C(N2CC(C)C(NS(=O)(=O)c3cccnc3)C2)=O)cc(O)ccc1[N+](=O)[O-] CC1CN(C(=O)Cn2ncnn2)CC(C(=O)NCC2(CO)CCCCC2)O1 C(C(C)C(F)C(=O)N1CC(C)(C#N)C1)NC(C1(CC#C)CCC1)=O c1(COC)nc(COC(C)(C)C)cc(=NC(C)c2cc(N(C)C)cc(F)c2)[nH]1 C=CCC(C)C(=O)N(C1CCN(C(c2cc(C3(Cl)CC3)n(C)n2)=O)C1)C N1(C(c2cc(C)c(C)nc2C)=O)CCCC(C2CN(C(=O)CSC(F)(F)F)C2)C1 C1(C(=O)NCCC(C)NC(C2CC3(CCOCC3)C2)=O)CCCCC(F)(F)C1 N1(C(C2CC(CN(C)C)C2)=O)CC2(CCN2C(=O)Cc2cc[nH]n2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CCC(C)C)C(=O)NCCCSC(F)F Cc1cn(C(C)C)cc1C(=O)NC(C)CCCNC(c1nncs1)=O c1(NC(C(C)N(C(c2c(CC)cncc2)=O)C2CC2)=O)cnc2ccccc2c1 C12(C(=O)Nc3cc(C)c(Cl)cc3)CCCC1CN(C(=O)CCC1(C)N=N1)C2 Cc1nc(C(=O)NCC(C)(CC(C)C)NC(c2nc(C)oc2C)=O)cc(O)n1 C#CCC(O)C(=O)NCC(=O)N(C1CCN(C(=O)C(c2ccc(F)cc2)(F)F)C1)CC C1(C(=O)NC(c2nc[nH]n2)C)CC2C=CC1N(C(C13C(=O)C4CC1C3C4)=O)C2 S(=O)(=O)(c1cccc2c1CCCC2)C(NNC(=O)Cc1cc(Cl)ccc1Cl)=O C1(C(N2CCCC2c2cc(C)cs2)C(=O)NCCC)CC2C(C1)C2(F)F c1(C(N(C(CC(=O)N2CC(OCCOC)C2)C)C)=O)cc(C)c(CO)o1 C1(C(N2CC(CNC(c3c(C)ncs3)=O)OCC2)=O)COCC(=O)N1C(C)C CC1C(NC(=O)CC2CCC(C)(O)CC2)CCCN1C(=O)Cn1ccnn1 N1(C(c2ccnc(Nc3ccccc3)c2)=O)CCCC(O)(c2nn[nH]n2)C1 Cc1cc(-c2ccc(C(=O)Nc3ncn(C4CC4)n3)nc2)cnc1C#N c1(-n2c(Cc3cccc(C)c3)nc(CSC)n2)cc(Cl)ccc1F C1(F)(CNC(c2ccc(SC(F)F)cc2)=O)CCCN(C(C2COCCO2)=O)C1 C(CCCCCNC(c1ccc(C2CCOC2)s1)=O)NC(C1(CC#C)CCC1)=O CCCS(=O)(=O)c1ccccc1OC(=O)C(N1CCC(COC)(SC)C1)=O CC1(C(=O)NCCC2(NC(c3cccnc3O)=O)CCCC2)CCC2CC2C1 C(CC(N)=O)(C(=O)NC(CC(C)C)C(C)C)NC(C(CC)N(C)C)=O N1(C(c2cc(C3C(C)C3)on2)=O)CC(C2(NC(=O)Cn3cnc(C#N)n3)CC2)C1 c1(CNC(CNC(C(C)OCCC=C)=O)=O)ncc(C(C)C)[nH]1 c1(OC)c(Cl)cc(C(=O)NCC2CN(C(=O)C(C(C)O)N(C)C)C2)c2ncccc12 C1(C(N(CCCN(C(C(C)NC(N)=O)=O)C)C)=O)CC1C1CCCC1 C(=O)(CCC(C)(F)F)NCC1N(C(C2(OC)CCC2)=O)CCC1C N1(C(C2C(CC(C)(C)C)C2)=O)CCCC(CCNC(=O)COCC2CC2)CC1 C1(CNC(C2CCN(C)C2)=O)CN(C(=O)C=C2CCC(C)(C)CC2)CC(C)(C)C1 c1(N2CCC(c3ccc(OC)cc3)(OC)C2)nc2cc(Br)cnc2s1 C1(CCC(=O)NCCN(C(CC=CCC)=O)C2CCCC2)CCN(C)C1 c1(C(=O)OC)cc(CNC(C2CCN2C(=O)C(C2CC2)SC)=O)nn1C c1(OC)cc(C(=O)NCCN(CCOC)C(c2c[nH]c(=N)o2)=O)nc(C)c1 CC(O)C(N)C(=O)NC1CCN(c2ccncc2)C1 c1(C(C)=O)cc(C(=O)NCC(C)(C)CNC(=O)CCOCC(F)F)cnc1C c1(C(=O)OC)cc2c(s1)CCS(=O)(=O)C2.c12cnc(cn1)Cc1nc-2no1 C1(NC(N2CCC(CC(C)(C)C)C2)=O)CC(=O)N(C)C1c1ccccc1 n1(CC)ncc(C(=O)NCCC(C)N(C(=O)CCC2CCCN2C)C)c1C C(CCc1ccccc1)(C(F)(F)F)NC(=O)COC12CCC1CNC2 c1(C(N2CCC(NC(C(CC)C(C)(C)CC)=O)C2)=O)cc(O)nc2cnccc12 c1(NCC(=O)Nc2c[nH]nc2-c2nccs2)ccc(F)c(Cl)c1F n1(CC(=O)NC2(C)CN(C(C3CC3C#N)=O)C2)nc2ccccn2c1=O N1(C(C(CC2CCCC2)OC)=O)CCC(CNC(C2(CC(C)C)CC2)=O)C1(C)C CC1CN(C(c2ccccc2C(F)F)=O)CC1CNC(C1(CN(C)C)COC1)=O N1(C(C2(C)CC(=C)C2)=O)CC2CCCC(NC(c3cncc(OCC)c3)=O)(C2)C1 Cc1cc(C(N2CCCC2(C)C(=O)NC(C)CCO)=O)nc2ccccc12 C(=O)(CCCCCC(C)O)N(CCNc1nc(C(C)C)cc(C)n1)C C1(NC(C(C(C2CC2)OCC)N2CCCC(C(=O)NC)C2)=O)CCC(F)(F)CC1 N1(C(C2(C)CC2(F)F)=O)CC2CC2(NC(c2ccc(C#N)[nH]2)=O)C1 C12(NC(=O)C3CC3)CCCC1N(C(=O)Cc1ccoc1)CC2 CCC(C)C(O)C(=O)N1CCC(F)(CNC(=O)Cc2cc(F)ccc2C(F)(F)F)C1 c1(OC)ccc(F)c(CN2CCCC(NC(C3(O)CC3)=O)C2)c1 Cc1cc(C)c(CC(N2CCCC(O)(CNC(=O)CC(C)(F)F)C2)=O)c(C)c1 Cc1cn2cc(C(N3CCC4CN(C(=O)CCCC(C)C)CC4C3)=O)ccc2n1 Cc1ccc(OCCC(N2CCC(OCc3cccs3)CC2)=O)c(Br)c1 N1(C(C2(SC)CC2)=O)CCC(CNC(=O)CCCSCC(C)C)C(C2CC2)C1 c1(C(=O)NCC2(CN(C)C(c3cccnc3)=O)CC2)[nH]nc2c1CCC2(C)C C#Cc1ccnc(C(=O)NCC(C)(C)OCC(N2CCCC(CC)(CC)C2)=O)c1 C(=O)(C(C)CC(C)(F)F)NCCCC1OCCN(C(C(COC)(F)F)=O)C1 CCC(O)C(F)(F)C(=O)NC1CCCC(NC(=O)C(c2cccn2C)=O)C1 N1(C(c2cccc(SCC)c2)=O)CCN(C(=O)CCC2CCCOC2)CC1CF C1(NC(C(C)S(N)(=O)=O)=O)CN(C(=O)Cc2ccon2)Cc2nccn2C1 CCCCCC(O)CC(=O)NCCC1CC(NC(c2cc(C3CC3)n(C)n2)=O)C1 c1(C(=O)NCCCNC(CCSc2cn(C)nc2)=O)cc(O)nc2ccccc12 CC(C)C(F)(CNC(=O)C(=O)NCC(F)F)C(=O)Nc1ccc(Cl)cc1O N1(c2ccc(S(=O)(=O)NCC3CN(C)C3)c(Cl)c2)CC2CS(=O)(=O)CC2(C#N)C1 C1(CC(=O)NCC2N(C(c3c(C)cccn3)=O)CCCC2)CCCC(C)(C)CC1 C1(C(N(CC(CCC)O)C)=O)CCN(C(=O)C(N)=O)C1(C)C C(C)(C(C(=O)NCCc1ccncc1)NC(c1ccsc1Cl)=O)OC C1(CNC(c2cc(CC)[nH]n2)=O)CCN(C(c2c(C)cnn2C)=O)CC1C Cc1cc(C(=O)NCCCOCCNC(c2ccoc2C)=O)c(C)n1NC(N)=O c1(OC)ccc2c(CC(=O)NC3(c4cccc(O)c4)CCCC3)coc2c1 CC(C)(O)C#CC(=O)NCC1(C(C)(C)C)CCN(C(C2CN3CCN2CC3)=O)C1 C=CCCC(C(=O)N=c1ccn(C2CC2)[nH]1)NC(=O)C(O)C(F)(F)F C#CCCCCC(=O)NC1CCC1NC(=O)CCn1ccnn1 N1(C(c2n(CCC)ccc2)=O)CCC(O)(CNC(=O)CCCN2CCCCC2)C1 C1(C)(C(=O)OCC)CCN(C(=NCCCF)NCC2(C)CC2(Cl)Cl)C1 c1(NC(N2CCC(O)(N3CCCC3=O)C2)=O)cc(F)c(N2CCNCC2)c(F)c1 c1(CC(N2CC(N(C(CN3CC(CC)C3)=O)C)C2)=O)ccc(-n2cccn2)cc1 C(CCCC(=O)NCc1ccc(CNC(=O)CC2CCC3CC23)cc1)NC(C)=O C1(CNC(c2cc(C)n(CCO)n2)=O)CCCN(C(=O)C=CCO)CC1 Cc1ccc(C(N2CC(NC(=O)Cc3ccnn3C)C3CC23)=O)cn1 C#Cc1ccc(NC(=O)C(C)(C)C#CCNC(=O)COC2CCC2)c(C)c1 C(=O)(CC(CC(C)C)NC(C1CCCC(CF)C1)=O)NCC(C#C)(C)C c1(C(=O)NC2CN(C(C3C4CC4C4CC34)=O)C2)c[nH]c2cccc(Br)c12 C1(F)(CNC(c2c(C(C)C)n[nH]c2)=O)CCN(C(c2ncoc2C2CCC2)=O)C1 c1(OCC)cc(Br)c(C)nc1NC(C1CC1NC(=O)Cn1cc(Br)cn1)=O N1(CC(=O)NCCCCCN(C)C(C2(C)CC2(C)C)=O)CCC(C)(C)C1 c1(C(=O)NCCC(N2CC(CNC(COC)=O)C2)=O)cnn(CO)c1C.O(C)C C(=O)(C(F)C(C)(C)O)NCC(C)CC(=O)N(C)CC1OCCC1(C)C c1(N2CCN(C(Cc3cc(C)cc(F)c3)=O)CC2C)ncc2c(C)cn(C)c2n1 N1(C(C2CCC(CC)CC2)=O)C2CCC(C2)C1CNC(C1CC12CCC2)=O N1(C(c2nc(CC)oc2)=O)CC(NC(=O)CCC2CC2(C)C)CC(C)(C)C1 c1(N(CCC(=O)OC)CCNC(C2CCC2)=O)ccnc(-c2ccccc2C)n1 N1(C(C(C)=C2CCCC2)=O)CCCCCCC1C(=O)NC(c1ccoc1)C CCC(C)(CO)C(=O)NCC(CNC(c1csc(N2CCCCC2)n1)=O)OC N1(C(=O)CCc2ccc(F)c(F)c2)CCN(C(=O)CCOC2CC2)CC(O)C1 c1(C(N2C(C(N3CCC(OC)C3)=O)CC3CC32)=O)cn(CC#N)c2ccccc12 Cc1cn2ccnc(C(N3CC(NC(=O)CCCn4cccn4)C4CC34)=O)c2n1 N1(C(CNC(C)=O)=O)CCC(C)C1NC(=O)OC(C)(C)C.c1(O)cnncc1Cl Cc1noc(C(C)C)c1C(N1CCC(C)(NC(=O)C(C)c2ccco2)C1)=O C(=O)(C1=NOC(C)(C)C1)NC(C(C)C)C(C)NC(c1cc(Cl)c(F)cc1Cl)=O CCC(CNC(C1C2CCC1CC2)=O)(CC)NC(=O)CC1CCC(C)O1 c1(C(=O)NC2(CNC(c3cocn3)=O)CCCC2)ccnc(-c2ccccn2)c1 c1(C(=O)NCC2CN(C(c3c(C)csn3)=O)CC(C)C2)cnc2ncccn12 c1(C(=O)NC(C2OCCN(C(C(C)=C3CC3)=O)C2)C)ccc2c(c1)CCN2C C#CCC(O)C(=O)N(C(CNC(c1cc(C(N)=O)co1)=O)C1CC1)C N1(C(c2c(CC)c[nH]c2)=O)CCC(F)C(NC(=O)C(C)C#N)C1 n1(NC(C(C)N(CCOC)CCNC(=O)C=CCN2CCC2)=O)nccn1 CS(=O)(=O)c1cccc(Cl)c1C(=O)NC1CC(O)CN(C(=O)Cc2cnns2)C1 c1(CN2C(C(N3CCC(C(F)(F)F)C3)=O)CCCC2)cc(Br)nc(Br)c1 C1(C)(C(=O)NCC(C)(C(C)C)NC(c2c(OC)nn(C)c2)=O)CCC(=O)NC1 Cc1cccc(Cl)c1C(=O)NC(C)CC(C)NC(C1CCCN1CC(C)C)=O Cc1sc2ccc(F)cc2c1C(=O)NCCCNC(C1CCN1C1CCCC1)=O c1(C(=O)NCCC(C)N(C(=O)Cn2cnnn2)C)cnc2n1CCOC2 C(=O)(C(CO)C(F)(F)F)C(=O)CONC(C1CCCCN1C)=O.CNCC c1(C(C)C)ncc(C(=O)NC2CCCN(C(c3n[nH]cc3F)=O)C2)cn1 c1(C(=O)NCCCCn2cnnc2)ccc2cnnn2c1 N1(C(C(CO)OC)=O)CC2(CCN(C(=O)CCC(C)CN(C)C)C2)C1 C1CCC(=O)NC1C.N1(C(C2CC(=C)C2)=O)CC=CCC1 Cc1nc(CCNC(=O)CC2CCCC2NC(=O)C(O)CN(C)C)cs1 C1(NC(c2cncs2)=O)CN(C(=O)CC2OCCO2)Cc2ccnn2C1 Cc1cc(N2CC=C(CCNC(=O)C(C)Cc3ccco3)CC2)n2ncnc2n1 C(=O)(C(C#N)C(C)C)N(CCOC)CCNC(C1C(Cl)(Cl)C12CC2)=O N1(C(=O)CC2CCC(NC(C3C4C5CCC(C5)C34)=O)CC2)Cc2cccnc2C1 C1(NC(C(CC)SC)=O)CCN(C(=O)C(C2CC2)OCC)CC1CC N1(C(c2ccn(CC)n2)=O)CCC(C(F)(F)F)C(NC(C2CC2C#N)=O)C1 c1(OC)c(F)c(NC(C2(c3cn(C4CCOC4)nn3)CC2)=O)cc(F)c1F c1(C(=O)NC2CCN(CCCNC(C(CC3CC3)OC)=O)C2)ccc(N)c(F)n1 c1(C(=O)NCC(C)N(C(C(C)OCCC#C)=O)C)ccc(C(C)(C)C)nc1 C1(NC(c2cc(OC)c(C(C)=O)cc2)=O)CN(S(=O)(=O)N=S(C)(C)=O)CCN1 c1(C(N(C)Cc2ccccc2)=O)cccc(COC2CN(C(=O)CC#N)C2)c1 C1(CNC(N2CCC(n3cnnn3)C2)=O)CCC(F)(CC2NC(=O)NC2=O)CC1 c1(CC(=O)N(C2CCN(C(CC(C(C)C)O)=O)C2)CCO)ccc2nsnc2c1 C1(C(C)NC(CC(=O)OC)=O)CCCN(C(=O)CS(=O)(=O)N(C)C)C1 C(CC(C)C)(C(=O)NCCN(CC(F)F)C)NC(COCC(=C)C)=O N1(C(c2c(C)n(C)cc2)=O)CCCC(NC(=O)CSc2n[nH]c(O)n2)C1C c1(OC)c(C(N2CCC(C(C)C(=O)N(CCN=[N+]=[N-])C)C2)=O)cnn1C c1(CC(=O)NCC(C2N(C(C(C)OC)=O)CCC2)(C)C)ccc2c(c1)CC2 CN1CCCC1C(=O)NCC(CNC(=O)CC1CC(F)(F)C1)CO C1(NC(c2cc3scnc3[nH]2)=O)CN(CC2CN(S(=O)(=O)C(F)F)C2)CCC1CO C1(C(=O)OC)CC2OCCC2N1C(=O)C=Cc1sccc1C C(=O)(CCCCC(C)(C)C)N1CCN(C(c2c(C)ccnc2)=O)CC1C(C)(C)C CCCCCC(O)C(=O)N(C(c1ccc(O)cc1)(C)C(=O)O)CC Cc1cnc2c(C(=O)NC(C)CCCNC(c3cnc(C#N)s3)=O)cccc2n1 c1(C(=O)NCC(CCNC(c2cc(C)sc2)=O)(C)C)coc2cc(O)ccc12 N1(C(C(CC#C)C2CC2)=O)CC2CCC2(CNC(=O)COC(C)(C)C)C1 C1(N(C(C(F)OC)=O)C)CC2CC1N(C(c1ccoc1C1CC1)=O)C2 C=CCC(C)(C)CC1C(=O)NC2C(C)(C)CCN1C2.c1(C(=O)OC)ccccc1Cl C=CCC(CC=C)C(=O)NC1CCCN(C(C2CC(C)(C)CN2C)=O)C1 Cc1ccc(N(C(C2CCOC(C)C2)C(=O)NCCOC(C)(C)C)C)nc1 C1(C(C)C)CN(C(=O)C2CC2C2CCC(C)(C)CO2)CCN1C(=O)Cn1cccn1 C1(C)(N(C)C)CCN(C(=O)C(C)(C2CCC2)NC(=O)CCc2cccn2C)CC1 C(=O)(C(C)C(O)C(C)CC)N(CCC(=O)NCCCCCCCC)C1CC1 C1(NC(CC2CN(C)C2)=O)CC2(C1)CN(C(=O)C(c1cnn(C)c1)N(C)C)C2 C(N=C1NC2CC2CN2CCN1CC2C)c1ccccc1.C(=O)(NCC)OCC C1(CCCC)CCCN(C(=O)CN(CCC)C(C2CCCC2OC)=O)C1 N#Cc1ccc(NC(C2(F)CCN(C(c3cccnn3)=O)C2)=O)c(Cl)c1 C(C(C(=O)NC1CCCOC1)C(C)(C)C)NC(C(C)CC1CC1)=O C1(C)(C(=O)NCC(CO)NC(C2(C)N(C(CCC)=O)CCC2)=O)CCCCCC1 c1(NC2CCN(C(C(CCC)NC(N)=O)=O)C2)cc2nc(C(C)(C)C)nn2cn1 c1(C(N2CCC(CNC(c3cnc(OC)nc3)=O)C2)=O)cccc2cccnc12 CC1(C(=O)Nc2cccc(NC(C3NC(=O)C4CCC34)=O)c2)CCC(F)(F)C1 C1(CNC(c2c(SC)ccs2)=O)CCN(c2nccc(CC#N)n2)C(C)C1 C1(NC(c2coc3ccccc23)=O)CCC(O)CN(C(=O)CC2CCCO2)C1 CN1CC(NC(C2(F)CN(C(=O)C(O)CC3CCCC3)C2)=O)C2(CC2)C1 c1(N2CCC(NC(C(=O)NCc3nnc(C(C)(C)C)s3)=O)C2)ccc(Br)cc1F C1(C(=O)NCC(C)CNC(=O)CCCNC(N)=O)CC12CCCCC2 CCCCC(CNC(c1cnn(C)c1)=O)NC(c1cccc(CC(F)(F)F)c1)=O C1(C(=O)NCC(C)N2CCC2)CCCC1CNC(C12COCC1C2)=O c1(C(=O)NCC(C)(C2CC2)NC(=O)C=CC2CCOC2)c(Cl)csc1Cl c1(C(=O)NCC2(NC(C3C(=C)C3)=O)CCOC2)ccc(CN(C)C)cc1 C1(C(=O)NCC2CC(O)CN2C(c2cscc2C(F)F)=O)CC12CCCCC2 Cc1c[nH]nc1C1(N)CC1.n1(C)cc(C2CN(C(C3COCC3C)=O)C2)nn1 N1(C(C(=O)NC)=O)CC(C)OC2(CCN(c3ccc([N+](=O)[O-])cc3C#N)CC2)C1 C(c1cnc(O)nc1O)=CC(=O)NC1CC2(C1)CC(NC(=O)Cn1cccn1)C2 C1(NC(c2ncc(OC)nc2)=O)CCCN(Cc2cc(C)ccc2O)CC1 c1(NC(c2ccc(OC)cc2)CO)ncc(C)cc1S(=O)(=O)NC1CCCSC1 Cn1nc(O)cc1C(N1CC(F)CC1CC(=O)NCC1CC1(Cl)Cl)=O c1(OCCOCC)cc(CNC(=O)NC2CCS2(=O)=O)ccn1 CC1OC(C)C(C(=O)NCC2CN(C(=O)CCn3cncn3)CCO2)C1C C1(C(N(C(C(=O)NCC#CC)C2CC2)C)=O)CCN(C)C1=O C1(NC(COC2CCCC(C)C2)=O)CN(C(=O)CCC(F)(F)F)C2(CCC2)C1 CC1CCCC1(C(=O)NCc1nc(=O)o[nH]1)NC(=O)CCc1ccoc1 CC(C)S(=O)(=O)CC(=O)N1CC2CC1C2NC(=O)CC1COCC(C)(C)O1 N1(S(CC)(=O)=O)CCCC1C1C(C(=O)NC(c2nn[nH]n2)=O)C1 c1(CCC)ccc(C(=O)NC(C)CN(C(=O)C(C)OCC2CC2)C)cc1 C1(C(=O)OC)CCCCC1C(N1CCC(CC(C2CC3CCC2C3)=O)C1)=O C(N=c1ccc(Br)c(S(=O)(=O)NC2(C)CC2(C)C)[nH]1)C1(OCC)CCCC1 n1(CC)cc(C(=O)NCC(C)(CNC(=O)C(C)C)OC)c(C2(CC)CCCC2)n1 c1(C(N(N2CCC(c3ncccc3Br)C2)C(C)C)=O)cccc(N(C)C)n1 N1(C(C2(C)CC(NC(C34CCN(CC3)C4)=O)C2)=O)CC2CCC(C1)C2C#N C12(NC(c3cc(CO)[nH]n3)=O)CCCC1N(C(c1cc(=O)cc(Cl)[nH]1)=O)CCC2 C1(NC(C(C=CC)O)=O)CCC(O)CN(C(=O)CCOc2cc(F)ccc2F)C1 C=CC(C)(C)CC(=O)N1CCCC1C1(C(=O)NC(CC(N)=O)C2CC2)CC1 c1(-c2n(C(COC)C)nc(-c3ccccc3C)n2)cnc2c(c1)nc(O)n2C c1(C(C)C)scnc1C(=O)NC1CCCC1CNC(=O)CC(C)N(C)C C(=O)(CS(=O)(=O)CC(=O)NC1CCN(C(C2(C(F)F)CCCO2)=O)CC1)OC Cc1nc(C2CC2)ccc1C(=O)NC1(C)CC(NC(=O)C2=CCSC2)C1 C1(C(N(C(CNC(=O)CSc2nncn2C)CO)C)=O)C(F)(F)C12CC2 C1(CNC(c2[nH]cc(CC)c2)=O)CC(C(=O)Nc2cnc(OC)nc2)=NO1 CCC(CC(F)(F)F)C(=O)NC1CCC1CNC(=O)COCc1nnc(S)n1C c1(NC(C(C2CCN(S(C)(=O)=O)CC2)C)=O)cccc(NC(C2COCCO2)=O)c1 c1(NC(c2nc(C)c(Br)s2)=O)ncc(F)cc1Cl N1(C(COc2cccc(C)c2F)=O)CCN(C(C2CC2F)=O)C(C#N)C1 c1(C2(C(N3C4C(NC(C=C(CC)C)=O)C(CC4)C3)=O)CC2)ccc(Cl)c([N+](=O)[O-])c1 CCC(C)(C)CC(=O)N1CCC(CC(N2CCCC2C(C)(C)COC)=O)C1 Cc1cccc(-n2nnc(-c3nc(C4CC4)nn3Cc3ccccc3Br)c2C)c1 c1(NCC2CC(C#N)C2)nc2c(s1)CC(C(=O)O)CC2 c1(OC)cnc(C(=O)NCC2CC(NC(=O)CC(C)C3CC3)CC2O)nc1 c1(OCCC)ccc(CN2CCC(CC(=O)NC(C(=O)OC)C(C)C)C2)cc1 N1(C(C2CCN(C(C)C)C2)=O)CCCCC1(C)CO Cc1cc(C(=O)NCC(CC(F)(F)F)NC(=O)C(C)C2(O)CCC2)cnc1C C1(CC)CN(C(c2ccc(C(=O)OC)c(F)c2)=O)CCN1C(c1occc1F)=O C(=O)(C1=CC2(CN(C(=O)CC(=O)NC3CC3)C2)OC1)NC1CC(C)OC(C)C1 c1(CCC)cc(C(N2CC(NC(=O)Cc3cc(C)on3)CCC2C)=O)cc(O)n1 c1(-n2c(CC(C)CO)nc(CO)n2)ccc(F)cc1F N1(C(=O)OC(C)(C)C)CC2CC(C(=O)NC3CCN(CC(=O)O)C3(C)C)(C2)C1 N1(C(CC=CCC)=O)CC2CCC1C(NC(=O)C=CC1CCCC1)C2 C=C(Br)CN=c1nc2c(cnn2C(C)C)c(N2CCS(=O)C(C)(C)C2)[nH]1 c1(C(=O)NCC(C)N(C(c2c(CC)nco2)=O)C)cc2occc2s1 C12(CNC(c3n(CC)cc(Cl)c3)=O)CC(CCO1)N(C(=O)C1=CCOC1)C2 c1(C(N(C2CCCN(C(=O)CCCC(N)=O)C2)CC)=O)ccc(N)c(F)c1 c1(C(=O)NC(CCNC(c2nn(CC)c(C)c2)=O)C)cn2cc(Cl)cc(Cl)c2n1 c1(C(=O)NCCC(C)NC(c2ncccc2O)=O)ccc(S(N)(=O)=O)o1 N1(CC(=O)NCCCN(C(=O)CCc2cnn(C)c2)C(C)C)CCC(F)CC1 N1(C(c2n(CC)ncc2)=O)CCC(C(N2CCOC(CC)CC2)=O)C12CC2 c1(C(C2(C)CCCO2)NCCCC)nnnn1CC1CCCO1 C1(CS(=O)(=O)NCC23C(OC)(CCC2)OCC3)C2CC3CC(C2)CC1C3 C12(C(=O)NC3CCN(C(=O)C(c4ccc(F)cc4)O)C3)CCN(C1)S(=O)(=O)C2 C1(NC(=O)CCc2cncnc2)CCN(C(=O)C(c2ccccc2)F)C12CCC2 C=CCC(CC)C(=O)NCC(CC(F)(F)F)NC(c1cnc(N)c(N)c1)=O C=C(Cl)C(C)(C)C(=O)NCC(C)(CC)NC(C1OCCC1C(F)(F)F)=O C(CC(=O)N1CCN(CCF)CC1)(C(C)OC)NC(CC)=O c1(C(N2CC(CC(N3CCC(O)(CC)C3)=O)C2)=O)cc2ncccc2[nH]1 c1(C(N(CCOC)CCNC(C2CCC3C(C2)C3(F)F)=O)=O)ccc(C)c(Cl)c1F C(C(=O)NC1CC(C#N)C1)(C(C)(C)C)NC(c1ccc(C)nn1)=O N1(Cc2c(C)cccc2)CCC2(CC1)COC(C(=O)NC1(C(=O)O)CCOC1)C2 Cc1cc(C(N2CCN(Cc3ccccc3N(C)C)CC23CC3)=O)cc(Br)c1 C1(NC(c2ccc(Br)c(F)c2)c2n(C(C)C)nnn2)C(=O)NCC1(C)C C=CC1(NC(c2csc(C(F)F)c2)c2nnnn2CCCCCC)CCOCC1 N1(CC(=O)N(C)C(C2(C(=O)OCc3ccccc3)CC2)=O)CC2C(C1)C2(C)C c1(C(N2CC(NC(c3cn(CCO)nn3)=O)C2)=O)ccc(CCn2cccn2)nc1 CC(=O)CCCCC(=O)NC1(CNC(=O)CC(C)C(F)F)CCOC1 C1(NC(CC=CC)=O)CC2CC(NC(=O)CCCCNC(N)=O)C1C2 N1(CC(=O)NC(CC=C)CNC(c2ccc(C#N)cc2)=O)C(=O)C(C)C(C)C1=O C12(C(=O)NC3CCC(O)C(F)C3)CCC(n3cc(CC4CCC4)nn3)(CC1)C2 C1(C(N(C2(C#C)CC2)C)=O)CCN(C(=O)C(C)NC=O)CC1(C)C c1(C(c2ccc(F)cc2)NCc2ccc(C(=O)OC)s2)ccnc(Cl)c1 C(=O)(C(F)C(C)C(F)(F)F)NC(CC(C)NC(C(C(C)C)F)=O)C c1(OC)ncc(-c2n[nH]cc2C(=O)NCCOc2cnn(C)c2)cn1 CCC(CC(=O)NCC(CCO)NC(=O)CCSC)C(C)(C)C C(CCNC(=O)NC(C)(C#N)C(C)C)(C(C)C)OC C(c1c(F)cccc1F)=CC(=O)NCC1C(C)CCN1C(=O)COCC1CC1 c1(NC(=O)C(C)CC2CCCC2)ccc(C)nc1.C1(C)(C)CN(CC)C(=O)CO1 CCC(C)C(O)C(=O)NCC(C)N(C(=O)C(F)(F)CCNC(=O)OC(C)(C)C)C c1(NC(C)=O)cc(F)ccc1C(=O)NC(C(C)NC(c1nocc1C)=O)C(C)C Cc1ccc2[nH]cc(Cn3cc(-c4ccccc4)nn3)c2c1 C1(C2CCOCC2)(C(N(C(CNC(c2cnn(C3CC3)c2)=O)C2CC2)C)=O)CC1 C(=O)(C1=C(C)OCCS1)N(CC(=O)NCCC(C)N(CCC)C)C(C)C Cc1ncnc(O)c1C(N1CCN(C(C2(F)CC=CCC2)=O)CC1)=O c1(OC)ccc(C2CC2)c(C(=O)NC(C)CN(C(=O)C(n2ccnc2C)C)C)c1 c1(C(N(C2CN(C(c3cccnc3F)=O)C2)C)=O)c(Cl)ccnc1Br C(CC(O)CNC(c1ccc(Cn2cc(Cl)cn2)o1)=O)NC(CC#N)=O C1(NC(c2n(CCC)ncc2)=O)CCCCC1CNC(=O)C(C)(C)c1ccsc1 n1(CC)nc(C(=O)NCc2csc(C(=O)NCc3conc3C)c2)c(C)n1 Cc1ccc(C(=O)NCCC2CN(C(=O)CCCC3CC3)CCO2)cc1C N1(C(C(CN(C)C)NC(C(CC)n2cncn2)=O)=O)CCCOCC1 C=CC(C)C(C)C(=O)NCCCN(CCCCNC(c1cnc(CC)s1)=O)C1CC1 CC1(C(=O)NCc2ccc(CCNC(c3ccc(=O)oc3)=O)cc2)CC(C#N)C1 C(=O)(C1=CCCOCC1)NC1C(CC(C)(C)C)CN(C(C2CC(O)C2)=O)C1 c1(C(N(CCCCNC(Cc2ccc(C)s2)=O)C)=O)cncnc1C1CC1 C(=O)(CCCCC(C)(C)C)NCCCC(CCCC)NC(=O)C(CC)(CC)CO C1(C(=O)NC(C(C)(C)NC(c2ccc(C)s2)=O)C)CCOCC1(C)C c1(C(=O)NC2CCN(CC(C)(C)O)C2)cccc2cnccc12 C12(C(N3CCCCC(NC(C(C)N(C(C)=O)C)=O)C3)=O)CCC(CF)(CC1)CC2 c1(C(N2CCC(NC(C3(C(=O)OC)C=CCC3)=O)C2)=O)ccnc(O)c1Br C12(NC(CCC(C)OC)=O)CCOC(CNC(C3(C)CCC(O)CC3)=O)(C1)C2 c1(C(=O)NC2(CC)CC2)nc(C2CCCCC2)sc1C Cc1ccc(CC(=O)NCC2CCCN(Cc3ncc(Br)s3)C2)cc1 CCC(C(=O)NCC(O)C(=O)NCc1csnn1)SC CC1CC(C(=O)NCC2CCN2C(=O)COC2CCCC(C)C2)CC(C)(C)C1 C(C)(C)(CC(=O)NCc1cc(C(N2CCC(C)C2)=O)cs1)SC C1(CNC(C2(CC)COC2)=O)N(C(=O)C(C)Oc2cccnc2)CCC1(C)C C(=O)(C(C)(C)C(C)(F)F)NCC1CC(Nc2nc(C)cc(C(=O)NC)n2)C1 n1(CC=C)c(N2CC(C)(C(N)=O)C2)nnc1CCc1ccc(Br)cc1 Cc1nn(C)c(C(F)(F)F)c1C(=O)NCC1CCCN(C(c2cn[nH]c2)=O)CC1 N1(C(C2(C=C)CCN(C(C34CSCC3C4)=O)C2)=O)CCCC2(CCOC2)C1 c1(OC(C)C)cccc(C(=O)N(C2CCCNC2=O)C)n1 C1(N(C)C(C2CC3(CCC3)C2)=O)CC2CC1N(C(C1C=CCCC1)=O)C2 c1(C(N2CCN(C(c3cncc(C)c3C)=O)C(CF)C2)=O)cccc2ccsc12 Cc1ccc(C(=O)NCCCN(C(=O)CC2CCCC(=O)N2)C2CC2)nn1 C1(C(=O)NCC(C)NC(=O)OC)CCN(C(c2cc(O)nc(O)n2)=O)C12CC2 N1(C(C)C(=O)N(C)C)CC=C(CNC(=O)CCc2cc(Cl)cs2)CC1 C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)N1CC(C)C(C)(N(C(=O)C=CCF)CC)C1 C1(CC)C(NC(c2ccoc2)=O)CCCN1C(=O)C=CCF N1(C(c2cn(C)nc2C)C(=O)NC)CCC(N(C)C)C(C)C1 C(=O)(C(F)C(C)CNC(N1CCOCC1=O)=O)N(CC(C)C)CCO C(=O)(CC(O)CC(C)(C)C)N1CCC(C(=O)NC2CC(OC(C)C)C2)C1(C)C C1(NC(C2(CC=C)CN(C(C3CCCC(C)(C)C3)=O)C2)=O)C=CC(C)(C)CC1 N1(C(c2cn(C(C)C)nn2)=O)CC=C(CC(=O)NCC2CCOC2C)CC1 c1(OC)cncc(CCC(=O)NC2CCC(NC(C3CCOC(=O)N3)=O)C2)c1 C1(CNC(C2(C)C(C)(C)C2(C)C)=O)CN(C(c2cnc[nH]c2=N)=O)C2(CCC2)C1 C1(NC(C2CCN(C)C2)=O)CC2CN(C(=O)Nc3cc(Cl)cc(Cl)c3)CC2C1 C1(N(C(c2ccc(CNC(C)=O)s2)=O)C)CCCN(C(C2CCC3(CC3)C2)=O)C1 c1(-c2cc(C)c(O)nc2)nc(C2Cc3ccccc32)nn1C(C)C C1(NC(C2C(C)(Br)C2)=O)CCCCC12CCCN(C(=O)CCn1cncn1)C2 C(C(C(=O)NCC1(C#N)CCC1)C(C)(C)C)NC(C1(OCC)CCOC1)=O N1(C(COC)=O)CC(OC(c2cnn(C)c2)C(=O)NCC(CC)CC)C1 C#CC1CCCCN1C(C1CCCCC1CNC(=O)Cc1ncccc1F)=O c1(C(C(=O)NCc2cn(-c3cccc(Br)c3)nn2)O)cccc(Cl)c1 c12[nH]nc(c1Cl)C(=O)N1CC(C)(C1)NC2=O.c1(CC)nc(-c2nc[nH]n2)sc1C c1(C(=O)NC2C(CNC(COCCOCC)=O)CCC2)cccc(N(C)C)c1 C(=O)(C(C(C)C)NC(c1ccc(OCCC2CCOC2)cc1)=O)N(CC)CC C1(N(C(C(C)SC)=O)CCO)CCN(C(C2(c3ccccc3)CCCC2)=O)CC1 c1(N(C)C)cncc(C(N2CCOC(CNC(C3(CCN=[N+]=[N-])CC3)=O)C2)=O)c1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC2(CCCN(C(C34CCCC(CO3)C4)=O)C2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCOC)CCNC(c1cnc(CC(C)(C)C)o1)=O CCC(CC)CC(F)C(=O)N1CCC(C(=O)NCCCCC2CC2)(CC)C1 c1(CC)cc(C(N2CC3CC3(NC(c3cn(C)cc3C)=O)C2)=O)ncn1 C1(NC(CNC(COc2c(C)occc2=O)=O)=O)CN(C)CCN(C)C1 C1(CS(=O)(=O)NCC(c2ccccc2)C)CCC2(CCOCC2)CO1 n1(C(C)(C)C)ccc(=NC(=O)C(=O)NC2CCC2)[nH]1 Cc1nnsc1C(=O)NCC(C1CC1)N(C)C(c1cn(C(C)C)nn1)=O C(=O)(C(C)(C)CF)NC1CC(N(C)C(c2ncoc2CCC(F)(F)F)=O)C1 N1(C(C23C(CN(C(CC4CCCC(=O)N4)=O)C2)COC3)=O)CCCC2(CCCO2)C1 N1(C(C=CC2(C)COC2)=O)CC=CC(C(=O)NCc2nc[nH]n2)C1 CS(=O)(=O)C1CCCC1C(=O)NCC1CN(C(=O)Cn2ncnn2)CCO1 c1(CCCC)ccc(Cc2cn(C(C)C(=O)N(C(C)C)CC)nn2)cc1 CN=c1cc(C(=O)NC2CCOC2C(=O)NCC(C)(C)C(F)F)cc[nH]1 c1(C(C2CC3CCC2C3)NC(=O)NCCN2CC=CC2)cccc(F)c1 N1(C(C2CC(C)C2)=O)CC2CCC(NC(c3ncc[nH]3)=O)CC2C1 C1(CO)CCC2CN(c3cc(NCC(CO)C(F)(F)F)ncn3)CCC2C1 c1(C(=O)NCC2N(C(CCN(C)CC)=O)CCCC2C)sc2cccnc2c1Cl Cc1ccc(C(F)(F)C(=O)NCc2nccn2C(c2ccccc2)C)c(Br)c1 C12(C)CCCN(CC1)C(C(=O)Nc1ccccc1)c1ccnc(c1)C(=O)C2=O.COOC c1(CCC(N2CCC(N(C)C(C3CCCS3)=O)C2)=O)cc2ccccc2c(=O)o1 c1(C(=O)NC(C)CNC(c2ccc(C(F)F)cn2)=O)cc2cc(Cl)cnc2o1 C1(C2CC2)(CNC(C2(CN(C)C)CC2)=O)CCN(C(=O)C(O)CC(F)(F)F)C1 C(=O)(CC(C=C)CC)N(CC(=O)NCCCCCC#C)C1CC1 CC(C)CC(C(=O)NC1COCC1C(=O)N(C1CC(C(N)=O)C1)C)C(N)=O N1(C(CC2N(C)CCOC2)=O)CC2CCCC2(NC(=O)CCCCC2CC2)C1 C1(NC(CC(C(C)C)O)=O)CC2(CCN(C(C34CCOC3CCOC4)=O)CC2)C1 C(CCCC(C)NC(=O)C(F)CC1CCCCC1)NC(c1c(C)nco1)=O C1(N(C(c2ccon2)=O)CC)CCC(NC(C2CCCCC2F)=O)CC1 Cc1ncc(CN(C(c2snnc2C)C(=O)NCC2CCCO2)C)[nH]1 c1(C(=O)NCC2(F)CCN(C(C3(C=C)CCC3)=O)C2)oc2c(Cl)cccc2c1C CNS(=O)(=O)N1CCC(C(=O)NC(C)CNC(=O)C(C)CN(C)C)CC1 c1(NC(CCC(=O)NCCC2CC(C)OC(C)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NCCN(C(=O)C(c2cncn2C)O)CCOC)ccc2sncc2c1 C(C(C)(CC(C)C)NC(C1CC(SC)C1)=O)NC(C(CC)(C)OC)=O C1(CC=C)CCCCC1NC(C)(C#N)COC(=O)C=Cc1ccccc1 c1(C(=O)NC)cccnc1NC(C1CC(CNC(c2ccn(C3CC3)n2)=O)C1)=O C12(C(=O)NC(c3ccncc3F)C)CCC(CC1NC(=O)CC1CC=CC1)C2 O=C(C1SCCc2sccc21)NCCNC(c1cnc(-c2ccccc2)[nH]1)=O c1(C(C)C)ccc(N(C(C)C=CCCc2ccccc2)C(C)C)cc1 C1(C(=O)NC(C2CCCN2C(c2sccc2C(F)F)=O)(C)C)CN2CCN1CC2 c1(C(=O)NCC(C)(C2CCC2)NC(C2CCCC(O)C2)=O)cncc(C(F)F)c1 C(=O)(C(Cc1cc[nH]n1)NC(C1CCN(C)C1)=O)NCCN(CCC)CC C=CCCC(C(=O)NCCc1ncccc1F)NC(=O)CCC1OCCO1 c1(C(N2C(CC(N3CCC=C(C)C3)=O)CC2)=O)ccn2cncc2c1 C1(NC(CCC(C)(C)F)=O)CC2CCC(C1)N2C(c1cc(F)c(F)c(O)c1F)=O Cc1cncn1C.c1(C2C(=O)NN2CC(C)C)cc(C(C)(C)O)on1.CCC(C)C N1(C(C2(C(C)C)CC2)=O)C2CCCC1CN(C(=O)COc1ccccc1F)C2 Cc1nnc(NC2CCCCC2CNC(C23CC(CO2)C3)=O)c(C#N)c1C N1(C(CSCC(C)=O)=O)CC2COCCC2(NC(c2cnc3ncccn23)=O)C1 C(=O)(CCCC(=O)OC)NC1CC2(C(C(N3C(CC#C)CCCC3)=O)C2)C1 N1(C(COC2(C)CCC2)=O)CC2CC2(CNC(=O)COC2(C)CC(CC(=O)O)C2)C1 C1(C(=O)NCC(C)(O)CNC(=O)C(C2CCCCCC2)O)OCC2CCCCC12 C1(C(C)NC(C2(F)CCC2)=O)CCCN1C(C1CCC(=O)N1)=O c1(C(=O)NC2CCC(CNC(C(CCN(C)C)O)=O)CC2)cccc2cncn12 N1(C(CCCC#C)=O)CC2CCC2(C(=O)NCC(c2ccc(C)cn2)O)C1 N1(C(c2ccc(C)cn2)=O)CCCC2(NC(=O)CCc3ccncn3)CC2C1 CN=c1nc(N(C)CC2CCCS2)[nH]c(=NC(C)c2nc(=N)[nH][nH]2)[nH]1 c1(CC(=O)NCc2ncn(C)c2)cc(F)c(Oc2cccc(F)c2)c(F)c1 N1(c2cc(NC(C)CC(N)=O)nc(COC)n2)CCN2C(=O)C(=O)NCC2C1 c1(C(=O)OCC)csc(CNC(=O)Cn2cc(C(O)CO)nn2)n1 c1(N2C(CNC(Cn3ccc(C)c3)=O)CC2)cncc2ccccc12 C(=O)(C(F)(F)CO)NC(C1(O)CN(C(C2(C(=O)OC)C=CCC2)=O)C1)C N1(C(c2cc(C#N)cs2)C(=O)NCCCSC)CCCCCC1c1cccnc1 Cc1cccc(Cl)c1CC(=O)N(C)CCN(C)C(c1coc(C(C)C)n1)=O CC1C(NC(=O)C(F)(F)c2ccnn2C)CCCN1C(c1nccc(N)c1Cl)=O C1(CNC(C2(C(=O)OC)CC2)=O)CCN(C(c2cc(Cl)ccc2Cl)=O)CC1(F)F c1(CCN(C(C(=O)NC2C(C3C(C)C3)C2)=O)C)cccc([N+](=O)[O-])c1 C1(=CC(=O)NC2CC(C(=O)OC)CC2O)CCCCC1(C)C C1(C(NOCC#C)=O)CCN(C(C2CC2OC(=O)N(C2CC2)CC)=O)C1 c1(C(N(CCN(C)C(c2cc3sccc3[nH]2)=O)C)=O)cc(Cl)ccc1C(F)(F)F CCCC(C(=O)NCCn1cccc1)OOC1CC(N(C(=O)COC(C)=O)C)C1 c1(N(CC(O)CO)C)cn2c(n1)CCN(CCC(N1CCCNC(=O)C1)=O)CC2 c1(C(=O)NCCCC(C)NC(c2c(C)nn(C)c2F)=O)ccc(F)c(C)c1N c1(C(=O)NC(C#C)CC2CCOCC2)nn(C)c2c(Br)cncc12 c1(C(=O)NC2CC(CCNC(C(C)n3ccnn3)=O)C2)cnc2c(c1)CCCO2 c1(CC)onc(C(=O)NC(C)(CNC(C2COCC2C(N)=O)=O)C(C)C)c1C c1(SCc2n(C)nc(COCc3ccccc3)n2)cc(C#N)cc(C#N)c1 C1(CCOC)CN(C(C2CCCN2C(C)=O)=O)CCN1CCC(C)F c1(NC(C2(C)CCN(C(C(=C)F)=O)C2)=O)ccc(C)cc1C O=C(CC(O)Cc1ccccc1)NCC1(F)CC(CNC(=O)COCC(F)F)C1 c1(C(N2CC(C(=O)OC)C2)=O)nc(C)no1.C(C)(C=O)N(C(=O)CC)CCC C(c1cccc(F)c1)=CCC(=O)NC1C2CCN(C(C3COC(=O)N3)=O)C12 c1(C(=O)NC2(C)CN(C(C(CCSC)NC=O)=O)C2)ncc(F)cc1C C(C(CNC(=O)CC1CCCN1C(C1CC1CCOC)=O)C(C)C)OC N1(C(c2n(CC)ncc2)=O)CCCC(C(F)(F)C(F)(F)F)C1.CC(=O)O c1(SCC(=O)NC2CCCCC2NC(c2c(Cl)n[nH]c2C2CC2)=O)ccc(F)cc1 C12(NC(=O)CNC(N3CCCC3)=O)CC(CNC(C3SCCS3)=O)(C1)C2 C1(CNC(C(C)(F)c2ccccc2)=O)(CNC(=O)C(N)=O)CC12CCC2 C1(C(=O)Nc2ccc(SC)cc2Cl)(COC)CCCN(C(=O)CC(C)CF)C1 C1(CC(=O)NCC(CCC)(C)C)CN(C(C2CC(OC3CC3)C2)=O)CCC1C N1(C(c2c(C)ncs2)=O)CCCC2C(CCCN2C(=O)Cc2ccon2)C1 C1(NC(=O)OC(C)(C)C)C(CNC(c2cc(C3CCC3)on2)=O)CCC12CCC2 n1(CC)cc(C(N2CCC(n3cc(CNC4(C(=O)OC)CC4)nn3)C2)=O)c(C)n1 C1(CC(=O)NC(c2ncn(C)n2)C)(OC)CN(C(=O)CC2CCCCO2)C1 N1(C(CCCOC)C(=O)N(C)CC)CC2CCC(NC(=O)OC(C)(C)C)C2C1 Cc1cc(C(=O)N(C2C(OC3CC3)COC2)C)nc(Cl)c1 c1(OC)ccc2sc(C(c3nnnn3C(C)(C)C)Nc3ccccc3)c(C)c2c1 C=CC(C)(CC)C(=O)N1CCN(C(C2CC(N3CCOCC3)C2)=O)C(CF)C1 C1(NC(C2CC(=C)C2)=O)CC2CCC(C1C)N2C(=O)C(c1ccc(N)cc1)(C)C c1(CC)cnc(CC(N2CC(n3cc(CNC(C4(C)CCCO4)=O)nn3)C2)=O)[nH]1 N1(C(C(CC)(C)COC)=O)CC2CC(C)N(C(c3cccc4ccoc34)=O)C2C1 Cc1cnc(C(=O)NCC2COCCN2C(=O)C(C)c2cncs2)cn1 Cc1csc(C(C)C(=O)N(C)CC2CN(C(c3cn(C)nn3)=O)C2)n1 C1(C(=O)NCC(CNC(=O)C=CC2CCC2)O)C2CC3C(C2=O)C13 c1(CC)ccc(C(N2CCC(COC)(NC(=O)CNC(=O)C(C)CC)C2)=O)cc1 N1(C(CC2CCN(C)C2)=O)CCCCC2(CCN(C(=O)CCC3CCCO3)C2)C1 C1(CSC)CCCN(C(=O)C(C2CCNCC2)OC)C1 N1(C(c2nc(C(C)C)oc2)=O)CC(NC(c2cc(CF)on2)=O)CCC1C N1(C(Cc2cn(CC)nn2)=O)CC2CN(C(c3cc(O)nc(O)n3)=O)CCC12 Cn1cc2ncc(C(=O)NCC3CC(NC(c4cnc(=N)[nH]c4)=O)C3)cc2n1 C(=O)(C1=CCN(C(C2COCCO2)=O)CC1)NC(c1ccc(C)s1)C c1(CCC)cc(C(=O)NCCN(C)C(c2cc(C(C)(F)F)on2)=O)sc1C c1(OC)ccc(C(N2CCCCC2CN(C(=O)C2=NOCC2)C)=O)c(F)n1 C1(C(N2CC(NC(c3cc(Br)nc(Br)c3)=O)C(F)C2)=O)CCCCC1(F)F N1(C(CCC(=C)Cl)=O)CCC2(CCCN(C(C3Cc4ccncc4N3)=O)C2)C1 N(C1CCNc2ccc(OC)cc21)C(C(C=C)n1cccn1)=O C#Cc1ccnc(C(=O)NC2CC3CC2N(C(c2cc(C)oc2CC)=O)C3)c1 C(C(C(C)(C)C)NC(c1cc(Br)n[nH]1)=O)NC(CN1C(C)CCC1)=O N1(C(CC(C)(C)N(C(C(CC)N(C)C)=O)C)=O)CC(O)(C2CC2)C1 N1(C(CC2CC(=O)NC2)=O)CCC2(CCCC2NC(c2nocc2Cl)=O)CC1 C1(CC(=O)NCCc2nnc(C)s2)CC(C)(C)CN1C(=O)CC1CCCCO1 c1(OC)ccc(C=CC(N2CC(NC(c3nc(Cl)cs3)=O)CC(F)C2)=O)cc1F C1(C#CC(=O)N2CCCC(N(CCO)C(c3sccc3SC)=O)C2)(CC)COC1 O=S(=O)(c1ccc(NCCF)cc1Br)NC(CC1CCCCC1)CO C1(CNC(Cc2cccc(OCC)c2)=O)CCCN(C(c2ncoc2C)=O)CC1 c1(OC)ccc(C)cc1C(=O)NCC1(F)CCN(C(c2cc(C)nc(O)c2)=O)C1 c1(C(=O)NCCN(C(C2C(c3ccc(C)o3)C2)=O)C(C)C)c(C)ccc(Cl)c1F Cc1cccc(CNC(=O)C(C)N(C(=O)Cc2ccnn2C)C2CC2)c1 N#CC1CCN(C(c2ccccc2C2CCC2)=O)C1 C1(NC(C(C=C)(C)C)=O)CN(C(=O)C(C)(C2CC2)OC)Cc2nccn2C1 c1(SC(C)C(C)NCC2CC2)ccc(Br)c(F)c1F c1(C(N(C)CCn2cc(CC3CCCCO3)nn2)=O)occ2c1CCCC2 C(=O)(CCS(C)=O)NC(CCOC)CNC(C1(C(=O)N(C)C)CC1)=O C(C(C)(C)CNC(=O)C(F)C1CCOC1)N(C(C1C(C)C1)=O)C C(=O)(CCCCCCS(N)(=O)=O)NC1C(C)CN(C(c2ccncn2)=O)CC1C O=C1CCSc2ccc(C(=O)NCC3CCCN(CCC(F)(F)F)C3)cc2N1 C(=O)(CC(C)(CN(C)C)C(F)(F)F)Nc1ccc2cnn(CCOC)c2c1 N1(C(c2cc(CC)ncc2)=O)CCCCCC1C(=O)NCc1ncoc1C1CC1 C(=O)(C1=NOC(CNC(=O)CC23CCC(CC2)CC3)C1)N1C(C)COCC1 C#CCC(C(=O)NC(c1scnc1C)C)NC(n1cnc(NC)n1)=O N1(C(C(C)(C)CF)=O)CC2CCC1C(CNC(c1snc(Cl)c1Cl)=O)C2 c1(SC)sccc1C(=O)NCC1CC1NC(c1ccc(C2CC2)s1)=O C1(NC(C(C(C)O)(F)F)=O)CC2CC(NC(=O)Cc3cnc[nH]3)CC2C1 C1(NC(C(C)NC(C)=O)=O)COC2(C1)CN(C(=O)C=C(C)c1cccs1)C2 N1(C(c2c(C)n(C)nn2)=O)CCn2nc(CNC(=O)C=CCO)cc2C1 N1(C(c2cc(C)n(C)n2)=O)CC2(C1)C(NC(=O)C#CC1CCCC1)CCS2(=O)=O N1(C(CCC)=O)CCC(NC(c2ccnc(F)c2)=O)C1C N1(C(c2c(CC)nn[nH]2)=O)CCOCC(CNC(C2(C)CCCCCC2)=O)C1 c1(C(=O)NC(CNC(C(C)NC(=O)C2CC2)=O)(C)C)cc(C2CC2)ncn1 c1(OC)ccc2c(=NCC(C)SC)[nH]c(=NC(C)Cc3cccn3C)[nH]c2c1 CCCCCCN1CCC(N(CCC)C(C2CC(OC(F)F)C2)=O)C1 c1(C(=O)NCC(C)(CC)NC(c2cn(CC=C)nn2)=O)cc(F)c(C)cc1Cl C(=O)(CCC(F)(F)C(F)(F)F)NC(CNC(C(C)NC(C)=O)=O)(C)CC(C)C c1(C(N2CCC(O)(CNC(C3N(C)CC(O)C3)=O)C2)=O)cc(Cl)cc(F)c1F C1(N(C(CCSCC)=O)C)CN(C(=O)CCOc2cccc(C(N)=O)c2)CC1O c1(C(=O)NC2C(OC)CN(C(=O)COC(F)F)C2)ccc(Cl)c(F)c1N C1(CC#C)(C(=O)NCCNC(=O)Cc2cn[nH]c2)CCN(C(=O)CCN(C)C)C1 CCS(=O)(=O)c1cccc(C(=O)NCCNC(=O)CC2CCOC(C(C)C)C2)c1 C1(CNC(C(C)NC(CC)=O)=O)C(C)CCN1C(C)=O.C12CN(C1)CC(=O)N2 CC(C)(CN=c1nc(N2CC=CC2)c2c([nH]1)CSC2)N1CCc2ccccc21 C(=O)(CCCC(C)(C)C#N)NCCCOCCN(C(c1c(C)cc(C)o1)=O)C Cc1nc(CC(=O)NC2CCCC2CC(N2CC(F)(F)C2)=O)co1 c1(C(N2C3(CNC(C(C)C4CCC4)=O)CCC2CC3)=O)c[nH]c2cc(F)ccc12 c12ncc(cn1)NC(=O)C1CCN1C2=O.c1(C(=O)OC)coc(C(N)=O)c1 CC1CCC=C1C(=O)N1CC(F)CC1CNC(=O)CCc1cn[nH]c1 C1(F)(CNC(CN(C)C2CC2)=O)COCCN(C(C2(O)CCCC(C)(C)C2)=O)C1 c1(OC)cccc(CNC(C23CC2CN(Cc2ccccc2OC)C3)=O)c1F C(c1ccc(C)nc1)=CC(=O)NC(CCNC(c1c(OC)cc(C)s1)=O)(C)C N1(C(Cc2cn(CC)nn2)=O)CC(=O)CC1C(=O)NCC1CC2(CC2)CO1 C(C(=O)NCCC(C(C)C)NC(=O)CCCn1ccnn1)(C(C)(C)C)SC C(C(=O)N(C)CCOCCNC(C1CC(C)(O)C1)=O)(C(C)(C)C)OC c1(C(=O)NCCCCCCNC(CC(=O)N(CCC)C)=O)ccc(F)c(F)c1N c1(C(=O)NC2CCN(C(=O)CO)C23CC3)cc2sc(Br)cc2[nH]1 C(=O)(C1Cc2ccccc21)NC1CC(C)N(C(=O)CCOCCN(C)C)CC1 c1(C(N(CCCNC(C2CC(C)SCC2)=O)C2CC2)=O)oc2ccccc2c1Cl C(=O)(C(C)C(C)O)N1CC(CC)(NC(C2(CC(C)C)CCCC2)=O)C1 c1(C(=O)NC(C(=O)NCCC#C)C2CC2)cccc(C#C)c1C c1(C(=O)NCC(CC)NC(C2CC2CC(C)C)=O)cc(OC)nc(F)c1 C(CC(C(=O)N=c1cc(C2CC2)n(C)[nH]1)NC(=O)Cc1ccoc1C)OC c1(C(=O)NCc2c(CCNC(c3nn(C)c(O)c3)=O)ocn2)cccc(F)c1Cl c1(Cc2nc(CC(CCC)C)n(-c3c(C)noc3C)n2)nc(C)cc(CC)n1 N1(C(C(=O)NC2CCCN(c3ccc(F)cn3)C2)=O)CCC(O)(C2CC2)CC1 C12(NC(CC=C)=O)CCCC1CN(C(=O)COc1c(F)cccc1F)C2 Cc1ccc(C(=O)NC(CC(F)F)C(=O)NC2CC(C(C)C)C2)cc1C Cc1cc(C(=O)NC2(C)CC2Br)c(Br)cn1 C(CC(C)(C)C(=O)Nc1cccc(CO)c1)NC(CCNC(=O)OC)=O C(=O)(C(O)CCCc1ccccc1)NCC(C1CCOCC1)(C)OC C1(CN(C(c2c(C)noc2)=O)Cc2ccccc2)NC(=O)CC1c1ccccc1 c1(C(N2C(CNC(C(CC=C)c3ccccc3)=O)CC2)=O)cc2n(c1)CCOC2 C1(C(N2C(CNC(c3ccc(C(F)(F)F)cn3)=O)CC2)=O)COCCOC1 Cc1c(NC(=O)NCc2cn(C)nc2C(F)(F)F)ccc(C#N)c1F c1(CC(=O)NC2CC(CNC(CC3C(C)C3)=O)C2)cccc(Cl)c1Cl N1(C(c2cc(C)ncn2)=O)C2CCC(C2)C1CC(N1CCC(C)(CN(C)C)C1)=O C1(NC(C2CCCN2C(C2C(C)(C)C2CC2CC2)=O)=O)C2CCCCC12.C1CC1 C(=O)(CCC(=O)C(C)(C)C)N1C(C(=O)NC(CCCC)CC)CC2(CCC2)C1 c1(OC)cc(CC(=O)N(CCNC(=O)C=Cc2cocn2)C2CC2)ccc1C CC1(C)CCCCN1C(=O)CSCCNC(C1CC(=O)C1(C)C)=O c1(N2CC(CCC)OCC2)nc2ccsc2c(=NCC2CCCS2)[nH]1 C12(CNC(C(C)(C)OC)=O)CN(C(c3ccc(C(C)(F)F)cc3)=O)CC1CCO2 C1(NC(C2OCCN(C(C(C=C)NC(C)=O)=O)C2)=O)CC2(CC(OC)C2)C1 Cc1c(Br)cc(C(=O)NC(C)Cn2cc(CC(CO)C3CC3)nn2)c(=O)n1C N1(C(c2nc(Cl)cs2)C(=O)NCCCSC)CCN(C)CC1CC(C)C CCC(CNC(=O)C=CC1CCC1)(CC)NC(=O)C(C1CCCCC1)F C1(CNC(C2CCN(CC)C2)=O)C(C)CCCN1C(c1coc(SC)c1)=O C(=O)(C1=CC2CCC(C1)C2)N1C(CCC(=O)NC2C=CCCCC2)CCCC1 c1(C(N(CCNC(C2C(=C)C2)=O)CCOC)=O)cnc(P(C)(C)=O)cn1 c1(OC)ccc(C(=O)NC(C)C(C(C)C)NC(c2ccc(C(C)C)nc2)=O)cn1 CC1=NN(C)C(=O)C1CC(=O)NC(C)Cn1cc(C2CCC(C)(C)CC2)nn1 c1(C2CCC(=O)N2)cccc(Nc2ccc(C3CCOCC3)cc2)c1 c1(CC(=O)NCCCCC(C)NC(c2nocc2Cl)=O)ccc2[nH]ccc2c1 N1(C(C2(CC)CCCN2C(=O)C=Cc2ccccc2)=O)CC(C)CC(C)(C)C1 C1(C(N2C(C)C(C)N(C(c3cc(F)n(C)n3)=O)CC2)=O)CC2(C1)CC1(CCC1)C2 C(CC(O)C(=O)NOCC(=O)NC1CC(=O)N(C)C1)NC(C)=O N1(C(C2(C)CC2(F)Cl)=O)CCCCC(NC(c2ccoc2)=O)C1 C12(NC(=O)Cn3cccc3)CN(C(=O)Cc3cc(C(F)F)no3)CC1CS(=O)(=O)C2 n1(CCC(=O)N(CC(C)NC(C2C(=C)CC2)=O)C)nc(O)c2ccccc12 C(C(C)C(C)C(=O)NC1C2CN(C(c3cnc4n3CCS4)=O)CC12)OC C12C(CC(=O)N1C)C(=O)OC2=O.c1(OC)ccccc1 C(=O)(CCC(C(C)C)NC(=O)CC1(CSC)CC1)NC(COC)(C)C(N)=O C(c1cocn1)=CC(=O)N(C(C)C(=O)NC1(C2CCCO2)CC1)CC CCCCCC(O)CC(=O)NC(C1CC(NC(C2(CC(C)C)CC2)=O)C1)C N1(C(C(Br)=C(C)C)=O)CC(C)CN(C(C2CCN(CCO)C(=O)C2)=O)CC1C c1(CC(=O)NCC(C(C)(C)C)NC(CCCOCCOC)=O)ccc(Cl)c(C)c1 c1(C(=O)NC(C2CN(C(=O)CC3(O)CCN(C)CC3)C2)C)cc2n(n1)CC(F)C2 CCCCCCC(=O)NC1CN(C(=O)CC23CCCN2CCC3)C(C)(C)C1 C1(CCC(=O)Sc2ccc(Cl)nc2)CCCCN(CC2CC(C)C2)C1 C1(CN(c2nnnn2CCc2ccccc2)CCCOC=C)CCOC1C C1(CNC(CCN(C(C)=O)C)=O)N(C(=O)CSCC2CCCO2)CCC1(C)C C=C(C)CC(C(=O)N1CC(F)(CC)C1)NC(c1ccc(C)c(C)n1)=O N1(C(C(CCC)NC(N)=O)=O)CC2CCC1C(CNC(=O)CCC=C(C)C)C2 C1(C(=O)NC2CCCCN(C(C(C)n3ccnc3)=O)C2)C2CCC(C2)C1(C)C N1(C(c2ccc(C)o2)=O)CCC(C)C1CNC(=O)C=CCN1CCCCC1 C=CCCCCC(=O)NC1CC(NC(=O)C=Cc2ccccc2)C12CCC2 N1(C(COCCNC(c2cc(C)c(O)nn2)=O)=O)CCCC(C)(O)CC1 C1(NC(C23C(NC(C)CCCN(C)C)C4CC2C3C4)=O)CC(C)N(C)CC1C C1(C(=O)NCCNC(c2coc(C(F)F)c2)=O)CC2CCC(C1)O2 CC1COC(C(=O)NC2CC(NC(c3nccn3C)=O)C2)C1 C(CCN(C)C)(C(=O)N(C)OC)N.C(CCCC(=O)CCC=CC)=CC=CC N1(C(C2C(C#C)C2(C)C)=O)CCCC(CNC(=O)C2=C(Cl)CC2)CC1 C1(C(N(CCCNC(c2cncc(OC)c2)=O)C)=O)CCc2nc(=N)[nH]cc2C1 c1(C(N(CCCNC(C2(NC(=O)NC)CC2)=O)C)=O)cccnc1F N1(C(C=CCCC)=O)CCCC(C)C1CNC(c1cc(C#N)oc1C)=O C1(CNC(c2c(SCC)nccn2)=O)CCN(C(=O)CC2(C)CCCCC2)C12CC2 Cc1ccc(C#N)cc1S(=O)(=O)NC1CCC(C(=O)Nc2nncs2)CC1 c1(C(N2C3(CCCC3)CCC2=O)=O)cccc(C)c1C#N.C1(OCC)CCN(C)C1 N1(C(C(C)CC2CCC2)=O)CCC2(CC1)CC2NC(c1cc(Cl)c(Cl)cc1Cl)=O c1(C(N2CCC(CCF)C2)=O)cc2c(Br)c(Cl)ccc2s1 C1(NC(CCCC(C)NC(c2cc(C(F)F)[nH]n2)=O)=O)CC12CCCCCC2 C1(c2nnnn2Cc2nnn(C)n2)(NC(c2c(C)nns2)=O)CCN(C)CC1C C(=O)(CC(C)(C)CC(C)=O)NCC1(NC(C2=CC(C)(CC)C2)=O)CCCCC1C c1(C(c2n(CC=C)nnn2)NCC2(F)CCOC2)cc(Br)c2ccccc2c1 N1(CC(C)OC)CCC(NC(c2cccc(-n3ccc(C)n3)c2)=O)C(O)C1 C(=O)(CC(CCCC)NC(c1nnc(S)n1C)=O)NC(C#C)CC N1(C(c2ccc(C)c(O)n2)=O)CCCN(C(C2CCCOC2)=O)CCC1 CCCCCCC(C)C(=O)NC(CNC(c1cccc(SCC)c1)=O)CC CCC(C)CCCC(=O)NCCN(CCOCCO)C(C1CCCOCC1)=O CCCCC(CC)CCC(=O)NC1CN(C(=O)CN2CC(C)(OC)C2)CC1C c1(C(=O)NC2CC(C(=O)NCC(C3CCC3)OC)OCC2)ccn2cncc2c1 C1(C(N(CCCCC2CC2C)C(C)=O)=O)OC2CCC1CC2.C12CN(C1)C2=O C1(C(C(=O)NCCSCC(=O)NCCc2cccs2)O)CCCCC1 n1(CC)nc(-c2cn(C(C)CC(=O)N3CCC3(C)C)nn2)cc1C CCCC(=O)NNC(=O)NC1CCCC(C)CC1 c1(NC(C2CC(NC(C(C=CC)O)=O)C2)=O)ccnc(CC)c1 N1(CC(N2CC(CC(N3CC(NC(C)=O)C3)=O)C2)=O)CCCC(C(=O)OC)C1 N1(C(C2CC3CCC2C3)C(=O)NC)CCCc2n[nH]cc2C1 C1(NC(C2(CO)CNC(=O)C2)C)CN(C(c2sccc2C#N)=O)CC(C)(C)C1 N1(C(CC(=O)NCC)=O)CCCC(CCNC(C2(CC)CC2(F)F)=O)C1 Cc1n[nH]cc1C(C(=O)NCC1CCCO1)N(C(C)C(C)SC)C c1(C(N2CCC(N(C(C(N3CCCCC3)C)=O)C)CC2)=O)ncnc2ccsc12 C1(C(N2CC(F)(C(=O)NC3CCN(C(N)=O)C3)C2)=O)CCC2(CCC2)O1 C1(C)(C(=O)NCC2C(C)(C)C2)CCCN(C(=O)CC2CCC2)C1 N1(C(c2c(C)occ2)=O)CCC(CCCCCNC(=O)COCC2CC2)CC1 CCCC(C(=O)NCC(C(=O)N(CCN=[N+]=[N-])C)OC)C(C)C C=C(C)CC(C(=O)NC1(CC(=O)NC(c2ccns2)C)CCCC1)OC C(=O)(CCCCCC(C)C)NC1C(OC)CN(C(C2CCCC2O)=O)C1 CCCCC(CC(=O)N1CCOC(CC)C1)NC(C1CC(CCC)C1)=O N1(C(C(C)C)=O)CCC(CCNC(c2ccc(N)c(Cl)c2)=O)CC1C N1(C(C(C)O)=O)CC(NC(c2ccc(N3CCOC3=O)cc2)=O)CC12CCCC2 C=CCC(CNC(=O)CCc1nccn1C)C(=O)N(CCCN1CCCC1)C c1(OC)ccc(I)cc1CN1CCN(C(C2CC2C)=O)C(C)C1 C1(N(C(C(CC)C)=O)CC)CCN(CCC(=O)Nc2ccccn2)CC1 c1(C(=O)NC(CC2CN(C(CC(C)C)=O)C2)C)ccc2[nH]nc(CC(C)C)c2c1 C1(C(=O)NC2C(C)C2(C)C)CC2(CC2)CN1C(c1ccsc1Cl)=O c1(C(=O)NCC2C3CCC(C3)N2C(C2CCC(O)C2)=O)cc2cccc(O)c2[nH]1 C#CCCCC(C)C(=O)NC1(CCC(N2CC(OC)CC2CO)=O)CCCC1 N1(C(C(CC)O)=O)CC(F)(F)CC1CCNC(c1sncc1Br)=O c1(C(N2CC(NC(Cc3c(C)scc3)=O)C2)=O)cc(N(C)C)ccn1 CC1CC(C(=O)NCCN(C)C(C2CC3CCC(C2)N3C2CC2)=O)CCS1(=O)=O C(=O)(C(C)(C)C(O)CC)N(CCC)CCNC(=O)C1CC1.c12nnn(n1)C2 CCCCCC(C(=O)O)n1ccnc1-c1ccccc1-c1sccc1C1CC1.OC Cc1ccc(C(N2CCN(C(=O)CN3CC(C)(C)C3)CC2CF)=O)c(N)n1 C(=O)(C1=CCC2CCC1N2C(c1csc(Cl)n1)=O)N1C(C)(C(=O)NC)CC1 c1(CNC(C2C(NC(c3nc(N(C)C)oc3)=O)CCC2)=O)c(Cl)cccc1Cl CC1(C)OC2(CNC(=O)C=Cc3cccc(Cl)c3)CC1(NC(=O)CS(N)(=O)=O)C2 C(=O)(C(C)C1=CCCC1)NCCCCC(C)NC(c1cccc(NC(C)=O)c1)=O CCCC(C(=O)NCCC(C)NC(c1cc(CN(C)C)on1)=O)c1ccccc1 c1(CC)nc(C)ncc1C(=O)NCCC(C)(C)CNC(c1cn(C)cn1)=O C(C(C(C)(C)C)NC(c1nc(O)c(C)s1)=O)NC(Cn1ncc(C(=O)OC)c1)=O C(=O)(CC1OCc2cc(Cl)ccc21)N1CCC(O)(CC(N2CCCC2)=O)CC1 N1(Cc2c(C)cc(C)[nH]2)CC2CC1CN2C(=O)CNCc1cccc(Cl)c1 c1(C(C(C)NC(C2CC3(CC3)C2)=O)NC(CNS(NC)(=O)=O)=O)ccc(F)cc1 C12(NC(CSCCCC)=O)CC(CNC(C3CCCN(C)C3)=O)(C1)OC2C c1(CN2CC(NC(c3ccccc3OC(F)F)=O)C2)ccc(F)cc1Cl c1(C(N2CC(NC(C(C)NC(=O)CC(F)(F)F)=O)C2)=O)cnc2c(c1)COCC2 Cc1cccc(C(=O)C(N2CC(NC(c3nc(C)c(C)[nH]3)=O)CC2C)=O)c1 c1(C(=O)NC2C(CNC(C3(NC(=O)OC)CCCC3)=O)C2)ccc(Cl)c(F)c1 N1(C(CNS(N)(=O)=O)=O)CCN(C(c2cc3c(s2)CCC3)=O)C2CCCCC12 C=C(F)C1(CC(=O)N(CCN(C)C(c2ncsc2CC)=O)C(C)C)CCC1 c1(CCC)ccccc1C(=O)NC(C)CCNC(=O)CCC1CCOCC1 C1(C2CCN(C(=O)C=Cc3ccn(C)c3)C2)(NC(c2ccc(F)nc2F)=O)CC1 Cc1ccccc1C(=O)NC1CCC(N(C)C(c2n[nH]cc2Cl)=O)C1 C1(NC(C2CC(NC(CS(CC)=O)=O)C2)=O)CCOC(C)(C)C1 c1(NC(=O)CCc2cc(F)ccc2[N+](=O)[O-])ccc2ccccc2n1 C1(N(C(c2cn(CCF)nn2)=O)CC)CCN(C(C2(OC)CCC(C)C2)=O)CC1 C(=O)(C(C)C(O)C(C)C)N1C(C)CCC(C(=O)Nc2c(C)c(CO)ccc2)C1 c1(OC)ccc(CCNC(C2CCCN(CC(N)=O)C2)=O)c(OC)c1 N1(C(c2csc3c2CCCC3)=O)CC(NC(=O)C(F)(F)C(F)F)CC12CCCC2 Cc1cc(C(=O)N(C)CC2CCN(C(=O)COCc3ccncc3)CC2)oc1C c1(C(=O)NC2(C)CCN(CC(=O)NCC(C)C)C2)n[nH]c2c1COC2 c1(OC)cnc(Cl)[nH]c1=NCCC1CCN(C(=O)C(c2ccc(F)cn2)(F)F)C1 N1(CCCl)CCC(C(C(=O)OCc2csc(Br)c2)NC(=O)CC2C=CCC2)CC1 C(=O)(C(=O)C(C)(C)C)N1C(CNc2c(C(C)=O)cccn2)CCC1 c1(C(=O)NC2CN(C(C(C(C)O)NC(N)=O)=O)C2)cc2cccc(F)c2o1 C(CCCCCNC(=O)CC1CC(C)=NO1)NC(c1cc(OCC)n[nH]1)=O C1(C(=O)NC(C)CCCl)C2CN(C(c3cccnc3C(=O)N(C)C)=O)CC12 N1(C(c2cc[nH]c2C2CC2)=O)CCCC(CO)(Nc2ncc(Br)cn2)C1 C(=O)(C1=CCN(C(C2(C3CC3)CCCCC2)=O)CC1)NCC(NOCC)=O C1(C(=O)NCC(CO)NC(C(C)=C(CC)C)=O)CCc2nnnn2C1 C1(C(C(=O)NC(CC)CNC(=O)CCn2ccnn2)C)CCC(=O)N1 c1(OC2CCc3c(cccc3)C2)n[nH]c(=NC2CCCCC2)o1 c1(CC)ccc(C(=O)C(=O)NCc2c[nH]nc2C2CCN(C(C)(C)C)C2)s1 S(=O)(=O)(CCCNC(=O)C=CBr)NC1(C)CN(C(c2cn(CC)nc2)=O)C1 C1(CNC(CCc2onc(C)n2)=O)CN(C(C2CC2C(F)F)=O)CCN1C c1(CC)nnc2n1CCCC2C(=O)N1CCCC(N(C)C(C2OCCO2)=O)CC1 c1(C(=O)NC(C)CCC(=O)NCC2NC(=O)NC2=O)cccc(F)c1F N1(C(COCCCCC)=O)CC2CN(C(=O)Cc3cc(C)ns3)CCC2(CO)C1 N1(C(C(F)=CCC)=O)CC(C)CCC1C(N1CCC(CN(C)C)CC1)=O C1(NC(C(C)SC(F)(F)F)=O)CCCCC1NC(=O)C=Cc1cocn1 CC1CN(C(C2(CF)COC2)=O)CC1NC(C1CCC(n2cccc2)CC1)=O C#CCC(CC(=O)NCCC(C)O)NC(C1CCCC1C(C)C)=O c1(C(N2C(CCNC(COC(C)=O)=O)CCCC2)=O)cc(C)cc(F)c1 c1(C(=O)NCCN(C(c2coc(C(F)(F)F)c2)=O)CC)nn(C)cc1Br C1(C(=O)OC)CCN(C(=O)CCc2ccncc2)C1.C(C(C)NC)OC C1(CCOC)(NC(C2C(=C)C2)=O)CCN(C(=O)CCc2ccc(=N)[nH]c2)CC1 N1(C(CCC=CCC=C)=O)CC(NC(=O)Cc2c(Cl)cnn2C)C(O)C1 C(CCCCC(=O)OC)(C(=O)Nc1cccs1)N(CCOC)CC1CCCCC1 C1(NC(C2C(C)CC(=O)N2)=O)CCC2CN(C(=O)Cn3cnc(=N)[nH]3)CC2C1 n1(CC(N2CC(NC(c3cc(O)no3)=O)(CO)C2)=O)ncccc1=O C(=O)(CCCS(N)(=O)=O)N1CCN(C(=O)NC2C(C)(CC)C2)CC1 C12(NC(=O)COc3cccnc3)CCCC1CN(C(c1cc(F)ccc1F)=O)C2 N1(C(CC(=O)OCC)=O)CC2(CCCC2NC(=O)C(C)N2CC(C)C2)C1 N1(C(c2c(C)cc(F)s2)=O)CCC2(CC1)CC(N)CO2 c1(CC(=O)NCC2COC(CNC(c3cc(CO)on3)=O)C2)ccc(Cl)cc1Cl N1(C(C2CN(CC)C(=O)C2)=O)C2CCC1CN(C(=O)C(F)(F)C(C)O)CC2 C=CC1(C(=O)NCc2ccc(C#N)cc2)CCN(C(C2CC3CC3C2)=O)C1 c1(OC)cc(F)ccc1C(N1CC2CC2(C(=O)Nc2ccc(N(C)C)cc2)C1)=O Cc1c(NC(c2cccc(N3C(=O)CCC3=O)c2)=O)cc(Br)cc1I C(=O)(C1=CCC2(COC2)OC1)N(C)CC1CCCN(C(=O)Cc2csc(S)n2)C1 c1(C(=O)OC)[nH]ccc1C(=O)NC1(C)CC(NC(=O)CCCOc2ccccc2)C1 c1(C(N2CCC(N(C(=O)C=Cc3cccs3)CC3CC3)C2)=O)cnc(O)nc1O c1(C(C(=O)NC2CCOC2)N(c2nc(C)c(C)s2)C)ccc([N+](=O)[O-])cc1Br C1(C(=O)NCC(CNC(C)=O)(C)C)COCCN1C(c1cc(C)on1)=O C(CC(C)CCNC(C1CC2C=CC1C2)=O)NC(c1cc(CC)no1)=O CC(C)(C)C(CCO)CN=C(NCC(F)F)N1CCc2nncn2C1 c1(CNC(c2c(C)csn2)=O)cc(C)c(C(=O)N(C)CC2CC(F)(F)C2)o1 Cc1cccc(CC(=O)NC(C2CN(C(=O)C(O)C3CC3)C2)C)c1Cl Cc1cc(C(=O)NCCCCNC(c2sccc2C(F)F)=O)nn1C(C)(C)C c1(C(=O)OC)c(F)ccc2c1CN(c1nnc(C(=O)OC)n1CC(C)SC)CC2 C(c1cccc(O)c1)=CC(N1C(C(C)NC(=O)CC2CCCC2O)CCCC1)=O C1(NC(=O)CCc2ccsc2)CCCN(C(=O)CCCn2ccnc2)C1 c1(C(=O)NCC(N2CCCC2C2(NC(C3CC3(F)F)=O)CC2)=O)cc(F)cc(F)c1 CC1CN(C(c2ccnnc2S)=O)CCC1NC(=O)CC(=O)NC1CCCC1 N1(C(CC(CC)SC)=O)CC(C(=O)NCc2ccnc(C#N)c2)CC(C)(C)C1 CCC(C)CCNC(=O)COCCNC(c1c[nH]nc1OC)=O CC(c1cccs1)=CC(=O)NCC1(F)CCN(C(=O)CCC2CCOC2)C1 C1(CNC(c2ncccc2Br)=O)CCC2(CN(Cc3ccc(Br)c(F)c3O)C2)O1 C12(NC(=O)Nc3cccc(C4CCC45CCC5)c3)CC3CC(C1)CC(Cl)(C3)C2 N1(C(C(c2scc(C)n2)C)=O)CC2(CCC(CNC(=O)C(C)N(C)C)O2)C1 N1(C(C(C)N(C(C)=O)C)=O)CCC2CN(C(c3ncc(Cl)cn3)=O)CCC12 C(=O)(C(C)(C)CCCNC(=O)C=CC(F)(F)F)N(CC(=O)NC)C c1(C(N2CC(C(C(=O)NC(C)CC(C)C)OC)C2)=O)c[nH]ccc1=O c1(C(N2CCC3(CCC3N3CC(O)C(F)C3)CC2)C)cn(C)c2cc(F)ccc12 CCC(Cc1ccccc1)C(=O)N(C1CC(NC(c2c[nH]nc2C(C)C)=O)C1)C C1(C(N(CCCCNC(C2CSCCS2)=O)C)=O)CCS(=O)CC1 c1(C(=O)NC2CCC(CCC(=O)NCc3nc(=O)o[nH]3)C2)cc2ccccc2o1 CC(=O)C(C)CC(C)C(=O)NCc1ccsc1C(=O)NOCC1CCCO1 C1(CCC=C)(C(=O)NCC#CCNC(c2cc(C3CC3)on2)=O)CCCC1 Cc1nonc1CNC(C1(CCNC(=O)C(O)CC2CCCC2)CCCC1)=O C1(CC(=O)NC(CC)CN(C)C)CCN(Cc2cnc(-c3ccccn3)s2)C1 C(=O)(C(C)(O)CCc1ccccc1)NC(CNC(c1c(C)ncnc1)=O)CC(C)C Cc1ccc(S(=O)(=O)N2CC3CN(Cc4cc(Br)c[nH]4)C3C2)cn1 C1(NC(=O)CCCC2CC2)CN(C(C2(C3CCC3)CC2(F)F)=O)CC2(CC2)C1 C1(CC)CCCN(C(=O)CS(C)(=O)=O)C1C(=O)NCC1(Cl)CCC1 c1(C(N2C(CN(C(C(C)C#N)=O)C)CCC2)=O)cc2ccncc2[nH]1 CCCC(C)(CC)C(=O)NCC1(NC(C2OC3CCC2C3)=O)CCOCC1 C1C(=O)N1CC(C)C.C(CC)(CO)N(C(C=CCCC)=O)C Nc1c(C(=O)NCC2CCCN(C(=O)CCC(F)F)C2)cnn1C1CC1 N1(C(c2cc(=NCC)[nH]cc2)=O)CCC2CCCN(C(=O)Cc3cnns3)C2C1 C1(CC)C(NC(=O)C2=NNC(=O)C2)CCCN1C(=O)CC1CCCCC1O c1(C(N2CCC(NC(C(COC)C)=O)(CF)C2)=O)ccc2[nH]c(=N)sc2c1 C1(NC(CN(CC)CC)C)CCN(C(=O)C(C2CC2)SC)O1 Cn1nc(O)cc1C(=O)NCC1CCCN1C(=O)Cc1ccc(I)cc1 N1(C(CC(C=C)(C)C)=O)CCC(C2CCN(C(c3ccc(CO)nc3)=O)C2)C1 c1(NC)scnc1C(=O)NC(C(=O)N1CCC1)C1CCCO1 c1(CC)nc(C)[nH]c1C(=O)N(CCNC(C1CC1C(N)=O)=O)Cc1ccccc1 N1(C(C2CC(C)(C)C2)=O)CC2C(C(=O)NC34CCC(CC3)C4)C2C1 N1(C(C2CSC2)=O)CCN(C(=O)Cc2csc(S)n2)C(c2cc(F)ccc2F)C1 C1(O)(CNC(C2C(C)CCC2)=O)CCN(C(=O)CN2CC(C)(C)C2)CC1 C#Cc1cccc(C(=O)NC(C)CCCNC(=O)C(C)CC(C)C)c1Cl c1(CC(N2CC(NC(CC(C)(C)OC)=O)C(O)CC2)=O)ccccc1S(C)(=O)=O C1(NC(CCC#CC)=O)CCCC12CN(C(=O)C(c1ccc(F)c(C)c1)(C)C)C2 C(=O)(CC1=CCN(C(c2cc(C)sc2N)=O)CC1)NCc1nccc(C)c1 c1(C(N2CC(C(N)=O)(CNC(c3n(C=C)ncc3)=O)C2)=O)cnn(C)c1C#N c1(C(=O)NCC(C2CCCC2)NC(c2coc(C(F)F)n2)=O)ccc(F)cc1F c1(C(N2CCC(C(C)(C)NC(=O)C(N)=O)C2)=O)ccc(C2=CCOCC2)cc1 C(C)(c1cccc(Cl)c1)=CC(=O)NC1CN(C(COC(C)=O)=O)CC(O)C1 c1(OC)ccc2c(=O)c(C(=O)NC3(CNC(=O)C(F)F)CCC3)cn(O)c2c1 C1(C(=O)NCC2CCC(NC(C(CC)(C)C#N)=O)C2)CN(CP(C)(C)=O)C1 N1(C(C(CCF)NC(C(c2cnn(C)c2)C)=O)=O)CCCC(F)(F)CC1 CCCCC(CNC(C1CCCN1C1CCCC1)=O)NC(c1ccccc1)=O C1(NC(CSCCC)=O)CCCN(C(=O)CC2CCCCO2)C1 c1(CN2CC(NC(c3cccnc3N3CCOCC3)=O)C2)ccc(Br)c(F)c1F C1(C(=O)NC2(CC#C)CCCCC2)CCCCCCN1C(C1CCCOC1)=O C1(C(N(CC(C)OC)C)=O)CCN(C(=O)OC(C)(C)C)CC1C C(=O)(C(Cc1cn[nH]c1)NC(C1(O)CC(O)C1)=O)N(C1CC(O)C1)C C1(NC(C2(O)CC2)=O)CCC2CN(c3cc(O)nc(O)n3)CC2C1 c1(CC(=O)NC(CC)CNC(c2cc(C3CC3)no2)=O)ccc(S(C)=O)cc1 C(C(C)(C)C)N(C(=O)NC)CCOC(C)(C)C CC(C)(F)C(C)(F)C(=O)NC1CCC(CNC(c2ocnc2CC(F)F)=O)CC1 c1(NC(C)CC#N)[nH]c(=NC(C)c2cccnc2C(F)(F)F)nc2c1cnn2C C(CN(C)N1CCC(c2cccc(Cl)c2)C1)N(CCC)CCC c1(CNCCC(C(=O)O)NC(=O)OC(C)(C)C)cccc2occc12 N1(C(CCCSC)=O)C2CCC1CC(N(C)C(C1CCC3(CCCO3)CC1)=O)C2 c1(CN2C(CNC(c3ncc(CC)cn3)=O)CC2)cc(F)ccc1C C1(C(=O)NCC2(OC)CCCC2)(NC(c2cc(C)ns2)=O)CCN(C)C1 C1(N(C(=O)CN=S(C)(C)=O)C)CCC2CN(C(=O)CCC3CCOCC3)CC12 c1(C(N2CCN(CCCNC(c3ccccn3)=O)CC2)=O)[nH]cc2c1CCC2 CCC(C)(C)CCCNC(=O)CCN(C)C(c1cc(O)cc(F)c1)=O C1(NC(C(CSC)c2ccccc2)=O)CCN(C(=O)CCC(C)(C)C)C(C)C1 Cc1nn(C)cc1CCC(=O)NCC1CN(C(c2csc(C)c2C)=O)CC1O C1(COC)(NC(=O)CN2CCC(C)C2)CCN(C(c2ccc(N)cc2F)=O)CC1 Cc1c[nH]cc(C(=O)NC(C2CCCCC2)C(C)NC(c2nnn(C)n2)=O)c1=O c1(C(=O)NCC2CCN(C(c3ccncc3O)=O)C2)cc(F)ncc1Br S(=O)(=O)(c1ccc(F)c(F)c1F)NC(n1ncc2ccc(-c3csc(N)c3)cc12)C C1(C(N(C(CC)CC)CCO)=O)CCCN(C(=O)CCC2CCOC2)C1 c1(C(=O)NC2C3CN(C(=O)Cc4cncnc4O)CC23)cc2ccc(Cl)cn2c1 N1(C(c2ccc(C3CCC3)o2)=O)CCOC(c2cn(Cc3ccc(Cl)s3)nn2)C1 C(C1C(C(N2C3CCC2C(CNC(C2COCCN2C)=O)C3)=O)C1(C)C)=C(C)C C1(NC(Cn2ccc(NC(C(c3cnn(C)c3)OC)=O)n2)=O)CC(=O)N(C)C1=O C1(C(=O)NC2(CCCC)CC2)CC12CCCCC2.C12CCCC(C1)CC(=O)N2 Cc1cc(C)c(NC(C2CC(C3CCC3)C2)=O)cc1Cl N1(C(C(CCC)CC2CCCC2)=O)CC(C)(C(=O)O)C(F)(C(=O)O)C1 CN=c1cc(C(=O)NC2CC(NC(c3cnn(C4C(OC)O4)c3)=O)C2)cc[nH]1 CC1(C)OC(=O)CC1C(N1CCOC(CC(=O)NCC2C3CCCC23)C1)=O CC1C(N(C)Cc2cc(N3CCCC3=O)ccc2F)CCCC1C C1(N(C(CN(CC)Cc2ccc(C)cc2)=O)C)CN(C(C)=O)CCC1O N1(C(=O)Cc2ccc(C(F)(F)F)nc2)CC2(C1)CN(C(c1ccc[nH]1)=O)C2 c1(C(=O)NCCOC2CCN(C(C(C)NC(C)=O)=O)C2)cccc2nc(Cl)cn12 c1(NC(=O)NC2CCC3CC23CO)cccc2c1OCCC2 N1(C(c2nncc(C)c2)=O)CCCCC(NC(C2NC(=O)CC2C)=O)C1 C(=O)(C1=NN(C(C2CCC(N(C)C)CC2)=O)C(=O)CC1)OC N1(C(c2cc(C)cc(F)c2)=O)CCC2(CCCC2NC(=O)C=C2CCCC2)CC1 C12(NC(C#CC(C)(C)O)=O)CCOCC1CN(C(=O)CS(=O)(=O)C(C)(C)C)C2 c1(SC)ccc(-c2nc(C3CC4(COC4)C3)no2)cc1.N1(CC)CCOC1=O c1(C(=O)OC)ccc(OC(F)F)cc1.c12cccc(c1)CCCN(C(C)C)C2=O c1(C(N2C(CC)CN(C(=O)CC3CCC(F)(F)C3)CC2)=O)cc(C)c(F)c(C)c1 C1(O)(CCNC(c2cncc(COC)c2)=O)CCCN(C(=O)CCS(C)=O)C1 c1(C(=O)OC)cc2ccccc2[nH]c1=NC(CNC(=O)C=C(C)Cl)C(C)C(C)C CCC(CC(=O)NC1CCC1NC(=O)C(=O)N(C)C)C(C)C CCS(=O)(=O)CC(=O)N1CC(NC(c2cccc(Cn3ccnn3)c2)=O)C2CC12 C(=O)(C1=CCCCC1)NCc1c(C(N(C(C=C)C2CC2)C)=O)nco1 CC1(C)C(C)(C(=O)NCC2(NC(C3CCCN3C=O)=O)CCCC2)C1(C)C c1(C(C(N2CC(N(C)C(c3cc(C4CC4)nn3C)=O)C2)=O)=O)ccc(Cl)cc1O c1(OC)cncc(C(=O)NCC2CC2CC(=O)NCCN2CCNC2=O)n1 C1(CNC(CN(CC)CC)=O)OCCC1C(=O)NC1(C)CCOC1 C(=O)(C1=CC2CCC(C1)C2)NC(CSCC)C(=O)Nc1cscc1CC C=C1CCC(C(N2C(C(N3CCC(C)(O)C3)=O)CC3CC23)=O)CC1 C(=O)(C1=CC(c2ccccc2)NC(=O)N1)NC(CCCC)CSc1ccccc1 C=Cc1ccc(C(=O)N(CCC(C)NC(c2ccc(COC)[nH]2)=O)C)cc1 CC(CC(=O)N1CC(CNC(c2ncoc2C(C)(C)C)=O)C(O)C1)C(F)(F)F c1(OCC(N2CCCC(CNC(Cc3cnc(C)[nH]3)=O)C2)=O)c(Cl)cccc1Cl C1(CCOC)CN(C(C2OCCCO2)=O)CCN1C(=O)C(C(C)(C)C)OC CC1C(NC(C2CC(O)C2)=O)CC2CCC1N2C(=O)CN1C(C)CCC1C Cc1nc2cccc(C(=O)N(CC(=O)O)CC3CCCO3)n2n1 C1(C(N(C(CN(C)C)C(=O)N(C(CF)CF)C)C)=O)C2(CC2)C12CC2 N1(C(c2cn(CCC=C)nn2)C(=O)NC(C)C(=O)OC)CC(=O)NC(C(C)C)C1 c1(OC)cc(C(=O)N(CC(C)(C)CNC(C2CCCC2C(F)F)=O)C)cc(F)n1 c1(C(=O)NC2CN(C(C3(COC)CCOC3)=O)C2)cc(Cl)cc(C)c1N C1(C)(NC(CC2(N(C(c3cnc(C(C)C)o3)=O)C)CC2)=O)CCC(=O)NC1=O c1(NC2CCN(C(CCN(C)CC)=O)CC2C)cc(=O)n(C(C)C)c(O)n1 O=S(=O)(c1ccc(Br)cc1NCCCF)NCCCN1CCOC(C(F)(F)F)C1 C#Cc1ccc(CCC(=O)N2CC(NC(=O)CC(C)(C)C#N)C2)cc1 c1(C(=O)NCC(CCCC)NC(C2Cc3nccn3C2)=O)ccn2nnnc2c1 Cc1ccc(-c2cccnc2S(C)=O)cc1CO C(=O)(CC1=NNC(=O)C1)N1CC(n2cc(CNC)nn2)C(OC(C)=O)C1 N1(C(N(C)C2CC2)=O)CCCN(C(C2CCC(F)CC2)=O)CC1 c1(C(N(C2CCN(C(=O)C(O)COC)C2)CC)=O)ccc2[nH]c(C)cc(=O)c2c1 C1(C(N(C)CC2CN(C(c3cc(C4CC4)no3)=O)CCO2)=O)CCCC(F)(F)C1 O=C(C#CCNC(=O)C=CC1CC1)NC1CC(F)(F)C1 C(=O)(C(C)(C)CCNC(c1csc(C)c1C)=O)N(CC)CC1CCOCC1 C1(CC#C)CCCCN1C(c1ccc(CNC(c2ccco2)=O)s1)=O N1(C(NNC(=O)C2C(C(C)C)CCO2)=O)CCC12CCN(C)C2 C1(C(=O)NCCN(C(c2nc(C)c(C)s2)=O)CC)CCN(C2CC2)C1=O C#CCCCC(=O)NC(C1CCCN(C(=O)CNc2ccccc2)C1)C N1(C(C2(CC#C)CCC2)=O)CC(CNC(c2c[nH]nc2C(C)(F)F)=O)CCC1C C(=O)(C(C#N)C(C)(C)C)N(CC(C)NC(=O)C1=CC2C=CC1C2)C c1(CN2C(COC)CN(C(c3ccc(SC)s3)=O)CC2)cc(C)c(O)c(C)c1 C1(NC(c2cnsc2)=O)(CO)CCCN(C(=O)CN2CCCC2CO)C1 N1(C(c2n(CC)ncn2)C)CCOCC(C(=O)NCCCCN2CCCC2)C1 C(CCCCCNC(C1CC(=C2CCC2)C1)=O)N(C)C(C1(N(C)C)COC1)=O c1(C(N2CC3(CN(C(CCC=C)=O)C3)OCC2)=O)ccc2c3c(cccc13)CC2 N1(C(N2CCC(C(=O)Nc3ccc(CC)nc3)(CC)C2)=O)Cc2ccccc2C1 S(=O)(=O)(c1ccc2nc(O)[nH]c2c1)N1CCC(F)(CNC(C=CC)=O)CC1 CCC(CC)(CCNC(=O)C(C)OCC(C)C)NC(=O)CC1CCC(=O)N1C C1(C(=O)NCC2(C)CCCN2C(=O)CC2CCC=CCC2)CCc2c[nH]nc2C1 c1(C(CO)NC(=O)CSC2CCOC2)ccc(Cl)cc1 c1(OCC(=O)N(CCC)CCC)c(C)cc(Cl)cc1Cl.C1(=O)CN1 C1(CNC(CCOCCCOC)=O)CCC(NC(C2(F)CC=CC2)=O)C1 c1(OC)ccc(C(C)NC(=O)C(=O)N(CCCn2ccnc2C)C)cn1 CC1CC(NCC2CCN(C(=O)Cc3ccco3)C2)CN1c1ccccc1 C1(O)(CNC(C2(CC(C)C)CCC2)=O)CCN(C(=O)CC2CCCC(=O)N2)C1 N(C1COc2ccccc21)C(C1(c2ccsc2)CC1)=O.C12CC1CNC2=O N1(C(C(CC(C)C)O)=O)Cc2ccc(CNC(=O)C(C)OCC(C)C)cc2C1 Cc1cc(CCC(=O)NC(C)CNC(c2nnsc2C(F)F)=O)no1 CC(C)CC(C(=O)NC(C)(C(N1CCCC(C)(C)C1C)=O)C1CCC1)C(N)=O c1(C(N2C3CN(C(C4(C)COC(=O)OC4)=O)C(C3)C2)=O)nnc2n1CCCCC2 c1(C(=O)NCC(CCNC(C2CCC(OC)C2)=O)(C)C)c(Cl)nn(C)c1Cl Cc1c(NC2CCCC(F)(F)C2)ncnc1N1CCC(OCCF)C1 C1(NC(c2c(C(C)C)n[nH]c2)=O)CC(C(=O)NC2CCCCC2CO)CC1O C1(N(c2nc(-c3cccc(Cl)c3)cs2)C(C)C)CC(C)(C(=O)O)CC1O S(=O)(=O)(c1cc(F)c(Br)cc1F)NC(C1N(CCC#N)CC2C(C)(C)C21)=O C(C(COC)CC(=O)NCCn1cc(C(=O)NC2CN(C)NC2=O)nn1)OC c1(N2CCC(SC)C2)nc(=NCc2sc(C)nc2C)[nH]c2ncn(C)c12 c1(CCc2c(C)[nH]nn2)ccccc1F.N12CCOCC1CSC(C)CCN2 C1(NC(c2nc(C(C)NC(C3CCC(C)O3)=O)oc2)=O)COCCC1O c1(OC)ccc(C(=O)NCC2CCCN(C(=O)Cn3cnccc3=O)C2)cc1 C1(C(=O)NCC(C)N(C)C(c2cccs2)=O)CC2CSCC(C1)C2(F)F C(=O)(CCCNCNC(C(C)C1CCCO1)=O)N(CC(=O)N(C)C)C(N)=O n1(CC)nnc(C(=O)NC(C)(CNC(C2CCCC(O)C2)=O)C(C)C)c1C O=[N+]([O-])c1cc(Nc2ccccc2-c2nc[nH]n2)c2c(c1)OCCO2 C(=O)(C1=C(C)N(C)c2nnnn2C1)NCC(CC=C)NC(C1CCCS1(=O)=O)=O C1(C(c2n(CCCSC)nnn2)NCCC2CC(C)C2)CC2CCC1CC2 c1(CO)cc(CSc2nc(C(O)C3CC3)n[nH]2)ncn1 C(c1ccccc1Br)=CC(=O)N(C1CCCN(C(C(CC)=CC)=O)C1)CCO N1(C(CCCc2onc(CC)n2)=O)CC2CCOC2(CNC(=O)C2=NOCC2)C1 C(CC1CC1)(C(=O)NC1CC(CCC(=O)NC(C)CN2CCCC2=O)C1)OC N1(C(C(=O)NCCC)CC2CCOC2)CC2CCCCCC2C1 c1(NC(C)Cc2c(Cl)cccc2Cl)nc(N2CC3CC3C2)c2cc(Cl)ccc2n1 C1(C)(CN(C(=O)Cc2cn[nH]c2)C)CCCC1NC(=O)CC1C(C)(C)C1(C)C c1(CN2CCCC(NCC(C)Oc3ccccn3)C2)cc(Cl)cnc1Br C1(NC(C2N(C(C)=O)CC(O)C2)=O)CC2CN(C(C3(C(F)(F)F)CCC3)=O)CC12 C(=O)(N=c1ccn(C(C)(C)C)[nH]1)Nc1scc(CNC(CC2CN(C)C2)=O)c1 c1(C(=O)NCC(CC)NC(=O)CC2(OC)CC2)ccc2nccc(C)c2c1 N1(C(COC)=O)CCCCCC(NC(=O)Cc2ccc3nn[nH]c3c2)C1 C=C(Cl)CCC(=O)N(C(CC)C(=O)N(CCF)CCOCCO)C C1(N(C(c2cnc(CC)s2)=O)C)CCCCN(C(C2(CC)CCC2)=O)C1 c1(C(=O)NC2CCC(NC(c3cc(OCC)no3)=O)C2)cc(Cl)c(Cl)n1C C1(C(=O)NC2(COCC)CC2)CC(O)CCN1C(c1[nH]cc(C)c1C)=O C(=O)(C1=CC2(CCOC2)C1)N1CCN(C(c2cccc3c2CCC3)=O)C(CF)C1 C1(C(=O)Nc2ncc(CCO)s2)CN(C(C2CCCO2)=O)CC12CC2 C1(C)(C(=O)NCC(N2CCN(C)CC2)C)CCCN(C2C3CNCC2C3)C1 c1(CC(N2CC(CNC(C(C)CN(C)C)=O)OCC2)=O)ccnc(Cl)c1F N#CC1CN(C(=O)C(Cc2ccco2)NC(=O)CN2CC3CC3C2)CC12CCC2 C12(CNC(C3(COC)CCC3)=O)CC(CO)(CN1C(=O)C1=CC(C)C1)C2 c1(C(N2CCC(C(C)NC(=O)COC(F)F)C2)=O)ncc([N+](=O)[O-])cc1Br c1(C(=O)NCC(C)(CO)NC(C2CCN(C)C2=O)=O)ccc2nonc2c1 Cc1cn2c(C(=O)NCC=CCNC(C3CCC(=O)N3)=O)cnc2s1 C1(NC(c2cnn3ccccc23)=O)CCC2(CCCN(C(=O)COC3CC3)C2)C1 C1(=CC(=O)NCCN(C(C23CCCCC2C3)=O)CC)CCN(C)CC1 C1(CC=C)(NC(=O)CCc2ncc[nH]2)CCCN(C(C2CSCCS2)=O)C1 C1(CC(N2C(CN(C(=O)C(C)(C)Cl)C)CCC2)=O)CC2CCC(C1)C2 C1(CNC(C(C)=CC)=O)CCC(NC(=O)C(COCC(F)(F)F)NC(C)=O)C1 c1(C(C)NC(CC)CNC(=O)OC(C)(C)C)cncnc1 C1(NC(CC2(CSC)CC2)=O)COCCN(C(C23CSCC2C3)=O)C1 c1(C(N(CCC)CCNC(C23CC(CO)(C2)C3)=O)=O)c(F)ccc(Cl)c1[N+](=O)[O-] CCCC(C(=O)OC)C(=O)N1CC(CN(C(=O)CC2CC=CCC2)C)C1 N1(C(c2cc(C)n(C)n2)=O)CC2(NC(=O)CC3CCCN3C)CCC1CC2 N1(C(c2c(CC)ncs2)=O)CCC2(CC2NC(=O)Cc2nc[nH]n2)C1 c1(SCC)ccccc1C(=O)NC1(C)CCOC1.C1(=O)COCCN1.C(CO)O C1(C(=O)NC(C)C(C)n2cccn2)CC2(CC2)CN1C(=O)CC1CCOCC1 N1(C(c2c(C)ccc(F)c2)=O)CCCC2(CCN2S(=O)(=O)CCCCl)C1 CC1CN(C(c2cccc(F)c2)C)CCC1NC(c1cc(Cl)c[nH]1)=O C(=O)(C1CCc2cc(O)cc(=O)n21)N(C(c1ccc(S(=O)(=O)C(C)C)cc1)C)C C1(NC(C(C(C)C)(C)C)=O)C2CCCC1CC(NC(C1CCNC1=O)=O)C2 N1(NC(C(C=C)C)=O)CC2(CNC(=O)N2C)C1.C1(C)(CC)CCc2cn1nn2 c1(OC)ccc(CN2CC3CC2C3C(N2CCCC2C)=O)cc1Cl C1(O)(CNC(CNS(NC)(=O)=O)=O)CCCN(C(=O)CCc2ccc(O)nn2)C1 S(=O)(=O)(c1ccc(NCc2ncnn2C)c(Br)c1)NCC1CC(C)C1 N1(C(CCN(C(CCC)C)C)=O)CCC(O)(CNC(c2oc(C)cc2C)=O)CC1 CC(F)(F)C(F)C(=O)NC1CCOCC1C(N1CC(OCCF)C1)=O N1(C(CCCNC(C(CC)C(F)(F)F)=O)=O)CCC2(CNC(=O)N2)C1 c1(CN2C(C)(COC)CCC2)cc(N2CCN(C(C)=O)CC2)nc(C(F)(F)F)n1 N1(C(c2c(CC)c[nH]n2)=O)CCC(N(C(=O)C(=O)NCC2CC2)CCO)CC1 C1(CNC(C(CC=C)CC)=O)CN(C(=O)COC2CCN(C)CC2)CCC1(F)F c1(-c2cnc(NC(C3CC(CC)(CC)C3)=O)s2)cc(C#N)ccc1F CC1(C)CC(C(=O)NCC2(F)CC2)CN(C(=O)CN2CCC(F)CC2)C1 N1(C(CC(C)(O)C2CC2)=O)CCN(C(c2nc(O)[nH]c(=O)n2)=O)C2(CCC2)C1 Cc1c(N)ccc(C(=O)NCCC(C)NC(C2(C)CC=CCC2)=O)c1Cl C12(CNC(c3cc(OC)c(Cl)s3)=O)CCCC1CCN2C(=O)C1=CCCC1 N1(C(CCC(N2CCCC2)C)=O)CCCC(COCc2ccccc2)C1 C1(C(N(C2CCN(C(c3cscc3OC)=O)C2)CC)=O)COC2CCCCC12 C1(NC(C2CCOC2)=O)CCN(C(=O)Cc2cn3ccsc3n2)CC1O c1(C(=O)NC2C(C)CN(C(=O)CC(C)(C)C)CC2)cc2ccccc2n1CC#N Cn1ncc2c1CCC(C(=O)NCC1CN(C(c3cnnc(O)c3)=O)CC1O)C2 N1(CC)C2CCC1CN(C(=O)CC=CCNC(c1cc(C)cc(O)c1)=O)C2 c1(C(=O)NCC2CCC(NC(CC3(C)CC3F)=O)CC2)onc2c1CCCC2 N1(C(c2nn(CC)nc2Br)=O)CCC2CCC12CNC(=O)CC1=CCCC1 CCCCC(O)C(=O)NCC1(C)CCCN1C(C1CC1C(C)(F)F)=O CCC(C)C(C(=O)N(CCCNC(=O)C=Cc1ccco1)CC)OC c1(OCC#C)ncccc1C(=O)NCCC(O)CNC(=O)Cc1ccsn1 c1(C(c2n(CCCSC)nnn2)NCC2(C)COC2)ccc(C#N)cn1 C(=O)(C(C)(O)CCC)N1CC(CNC(c2c(CCC)n(C)nn2)=O)C1 C(=O)(CCCCCCNC(c1csc(C)n1)=O)NCCC(C(C)C)OC N1(C(C=CC=CCC)=O)CCCC(NC(=O)C=CC2CCOCC2)CC1 CCC(O)C(C)C(=O)NCC1(C)CCCN1C(=O)C(C)n1ccnc1 CCCCC(C(=O)NCCN(C)C(c1cnc(C(C)C)s1)=O)C(C)C C1(NC(=O)C2CC2)CCCC12CN(C(=O)C=CC1CCCO1)C2 c1(NC(CCC=C)=O)cccc(NC(C2(COC)CCCCC2)=O)c1 N1(C(C(C)C2CCCO2)=O)CC(C)N(C(=O)CN(C)Cc2ccccc2)CC1C C(=O)(CCN(OC)C(=O)C(C)CCC(C)(C)C)N1C(CC(=O)OC)CC1 C1(O)(C(=O)NCC(CCNC(C2CCOCC2C)=O)OC)CCCCCC1 C1(NC(Cc2c(C)non2)=O)CC2CC1N(C(=O)CCc1ccc(F)cc1F)C2 c1(CN2C(CNC(c3c(OC)cccn3)=O)COCC2)cc(Br)ccc1OC c1(OC)ccc(Cl)c(C(=O)NCC2(CNC(=O)CCc3ccnn3C)CC2)n1 C=CC1(C(N2CCC(COC)C2)=O)CCN(C(=O)CC2(O)CCCC2)CC1 N1(C(CCc2cccc(OCC)c2)=O)CCN(C(c2[nH]nnc2C)=O)C(C)C1C c1(OC(c2c(Br)cn(CCOC)n2)=O)ccc(C#N)c(Br)c1 N(C1COc2ccc(Br)cc21)C(CCC=C(C)C)C(=O)NC1CC1 c1(OCC)ccc(NC(c2cc(C#N)cs2)c2nnnn2C2CCCC2)c(C)n1 Cc1cc(C(N2CCC(NC(=O)C(C)C(F)F)C2(C)C)=O)ccc1-n1cccn1 Cc1ccc(C(N2CC(NC(c3cccc(O)c3)=O)C2)=O)cc1NS(C)(=O)=O N1(C(CCCc2cc(C)no2)=O)CC(NC(=O)CN(C2CCCC2)C)C2CC12 C1(NC(CCn2c(C)ncc2)=O)C(C)CN(C(=O)C=Cc2cccs2)CC1C C1(c2ccccc2)(NC(C(C=C)O)=O)CCN(C(c2cc(C)co2)=O)C1 C1(NC(c2n[nH]c(C)c2C)=O)CC2CCC1(CNC(=O)Cn1cnccc1=O)C2 C#CC1(C(N2CC(=O)NCC2CC)=O)CCN(C(=O)CC(C=C)CC)CC1 C(=O)(C1CCCc2ncnn21)N1C(CN(C)C(c2csc(C(F)F)n2)=O)CCC1 C(=O)(C1=CCC(C)CC1)NCCC(C(=O)N(C)Cc1c[nH]nc1C)OC CC1(C(F)(F)F)CCCN(C(=NCc2ccc(C#N)s2)NC2CCS(=O)(=O)C2)C1 c1(CN(C(=O)CCC2CC(NC(C3(N(C)C)CCC3)=O)C2)C)ccncc1 N1(C(C(C)CC2CC2)=O)CC2COCCC2(NC(c2cc(C3CC3)cs2)=O)C1 C1(C(=O)NCC(C)NC(C2(Cc3nccnc3N)CCCC2)=O)CCN(C)C(=O)C1 N1(C(C(CC)C#N)=O)CCCC(CO)(NC(c2cc(C)ncn2)=O)C1 C1(CC=C)(C(=O)N(CC(C)C(C)C)C)CCN(C(c2cc(OC)cnn2)=O)C1 N1(C(C2CNC(=O)N2)=O)CC2CCCC(NC(C34CC(CC(F)F)(C3)C4)=O)C2C1 c1(C(=O)NCC2C(C)CN(C(=O)C(C)(C)CO)CC2)cc(S(N)(=O)=O)c(Cl)o1 CC1(C)CCN(C(=O)CCS(N)(=O)=O)CC1NC(C1CCN(C(N)=O)CC1)=O c1(C(N2CCC(NC(=O)C(=Cc3c[nH]cn3)F)C23CC3)=O)cc2ccccn2n1 CC1(C(c2nnnn2CC2CCOCC2)NCc2nncs2)CC2(C1)CC2(F)F N1(C(C2=C(C)OCCC2)=O)CCOC2(CCN(C(C34CCC(CC3)CC4)=O)C2)C1 C1(C(N2CC(F)(CC)C2)=O)CC(C)CCN1C(=O)C(C)CC1CCCC1 N1(C(C(C)c2ccco2)=O)CC2CC(C1)CN(C(=O)COc1cncc(Cl)n1)C2 Cc1ccnc2c(S(=O)(=O)N(C)C)cccc12.C1(N2CCC2)CCC2(CCC2)CN1 C1(NC(c2ccc(C)s2)=O)CN(C(=O)C=C2CCC2)CC1c1ccnn1C c1(OC)cccc(C(N2CCCC(CO)(NC(C3CC3C(F)F)=O)C2)=O)c1O Cc1nc(O)nc(C)c1CC(=O)NCC1(C)CCC(NC(C2CC=CC2)=O)C1 C1(NC(C23CN(C(C(C)NC=O)=O)C(C2)CO3)=O)CCCCCC1(C)C C1(C(N2CC(CNC(c3c(OC)csc3)=O)OCC2)=O)CC(C2CCC2)C1 C12(NC(Cc3c(C)ncc(Cl)c3)=O)CCCC1N(C(C13CCC1CC3)=O)CCC2 c1(C(N(C2CCN(C(=O)CCCC3CCC3)C2)C)=O)cccc(CC#N)c1 C(CN=c1cc[nH]cc1C#N)C1CCN(C(C(C2CCCCC2)OC)=O)CC1 c1(C(=O)NCC(C)(O)CNC(=O)CC2(C#N)CCCCC2)ccc2n[nH]cc2n1 c1(C(C(=O)NC(C(=O)NCC=CCCC)C2CCC2)F)ccccc1 c1(SCC)cncc(C(=O)N(C2CCCN(C(=O)CC3(OC)CCC3)C2)C)n1 C1(O)(C(=O)NC(C)CN(C(=O)Cn2cccn2)C)CN2CCC1CC2 c1(CCC)cc(C(N2CCC(CO)(NC(c3sccc3C)=O)C2)=O)sc1C CCC(C)(C)C(=O)NC(C1CCOC1)CNC(c1ccn(C)c1C1CCC1)=O c1(C(N2CC(F)CC(NC(C=C(C)C)=O)C2)=O)ccc2cccnc2c1 C1(O)(CC(=O)NC(C)C(C)NC(C2CCC(=O)NC2)=O)CCCOC1 n1(CC(=O)NC(C(=O)NC(C(=O)NC)C2CC2)Cn2cncn2)nc(C)oc1=O N1(C(c2ccc(C(C)C)cc2)=O)CCCCCC(NC(C2CC(O)C2)=O)C1 C1(C(N2CC(C(CC)C)C2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)C1C(C)C CCC(C)(COC)C(=O)NC1CC(NC(c2ccc(F)c(CO)c2)=O)C1 O(S(=O)(=O)CCCCCO)C1C(P(C)(C)=O)CCCC1 CCCS(=O)(=O)CC(=O)NC1CC2CC(NC(=O)C(F)CC3CCCCC3)C2C1 c1(-c2cn(CCNC(C(COC)(C)C)=O)nn2)ccc(Cl)cc1F C(=O)(CN=S(C)(C)=O)NCCC(CCNC(C(C)SCCCC)=O)C C1(C2CN(C(=O)CSc3ccc(Cl)cc3)C2)(NC(=O)C(F)CC2CCC2)CC1 C12(CNC(C3(NC(Cn4c(C)ccc4C)=O)CC3(C)C)=O)CCC(CC1)CC2 C1(NC(C2CCCCC2)=O)CN(C(C2CCC(F)(F)CC2)=O)CCC1C(F)(F)F N1(C(c2nc(CC)sc2N)=O)C2CCC(C2)C1CNC(=O)Cc1ncoc1C N1(C(c2ccc(C)cc2)=O)CCC2(CCCC2NC(=O)C=CCO)C1 C1(C(=O)NCc2ccccc2CNC(C2CCOCC2)=O)CCn2nccc2C1 c1(NCC)ccc(C(=O)NC2CC2NC(=O)CCc2ccco2)cc1[N+](=O)[O-] C1(C(=O)NCC2N(C(c3cnc(OC)c(Cl)c3)=O)CC=C2)CC2CC1CC2(F)F N1(C(c2c(C)n[nH]c2)=O)CC(CNC(C2CCC(O)CC2)=O)CC12CCOCC2 c1(C(=O)NCC2(NC(=O)C(Cl)=CCl)CC3CCC2C3)ccn2ccccc12 C1(NC(C=CC(=O)OCCCC)=O)CC2CCC(C1)N2C(c1ccc(SC)o1)=O CN1CCC(C)(C(=O)NC2(C)CN(C(c3ccc(C(C)(C)C#N)cc3)=O)C2)C1=O C1(C)(CCC(=O)NCCN(C(C(C)=C2CCCC2)=O)C(C)C)CCC(=O)N1 n1(CC)nccc1C(C)NC(=O)CCC1(NC(c2cncnc2)=O)CCCC1 C#CCCC(O)C(=O)N1CC(NC(=O)C(C2CC2)SC)C1 N1(C(C2(NC(C)=O)CCC2)=O)CC2CCN(C(=O)C3=NOCC3)CC2C1 N1(C(C(C2CN(C(C3OCCCC3(C)C)=O)C2)OC)=O)CCCC(N=[N+]=[N-])C1 C12(CNC(C(C)C3CCCC3)=O)CCCC1CN(C(=O)Cn1ccnn1)C2 C1(CNC(CN(S(CC)(=O)=O)C)=O)CCN(C(c2cnc(S)n2C)=O)CC1(F)F C(=O)(C1=C(Cl)CCC(C)C1)N1CCC(NC(CCCC=C)=O)C(O)C1 CCC(O)CC(=O)N1CCC(C(=O)NC(C)C(C)(C)CO)(OC)C1 c1(CNC(C(C)n2cccn2)=O)ccc(CNC(c2cc(=N)[nH]n2C)=O)cc1F c1(C(=O)NCCC2OCCN(C(C(CC)C)=O)C2)cc(C)ccc1C(F)(F)F n1(CC(=O)N(CC(=O)NC2CC(CC)C2)CC#C)ccc(C)n1 C(C(C)NC(c1cc(Br)nn1C)=O)(C(C)C)NC(CCNC(=O)OC)=O c1(C(=O)NC(C)CNC(C2(C(C)(C)C)CC2)=O)ccc(C(F)(F)F)cc1Cl N1(CC(=O)N(CCCNC(c2ncncc2N)=O)CCC)C(=O)CCCC1=O N1(C(CN2CCC(C)(C)C2)=O)CCCC2CN(C(=O)CC3CCOC3)CCC12 C1(NC(CCS(C)=O)=O)CCCN(C(=O)COc2ccccc2O)CC1 C(CCCC(CO)NC(C1(OC)CCSC1)=O)NC(c1c(Cl)cn(CC)n1)=O C(=O)(C(C)(C)C1=CCSCC1)NC(CCN(C(C(CCC)C)=O)C)C C1(NC(C2(CC(=O)OC)CC2)=O)CC(NC(C2CCN(C)CC2)=O)C12CCC2 C1(CCC(=O)OC)CCCN1N1CCC(CNC(c2ccccc2)=O)C1 C(C1CN(C(c2[nH]nnc2CC)=O)CC1C(=O)NCc1ccc(OC)o1)=CC CCCCC(C(=O)NC(C(=O)NC1(CO)CCC1)C1CCC1)C(C)C C1(CNC(C(C)Cn2cccn2)=O)CCN(C(c2ccn(C3CC3)n2)=O)CC1 C12(CCOC)CCN(CC1)C2=O.c1(CNC(=O)Cc2cnoc2)cc(Cl)ccn1 C=C=CC(C)C(=O)N(C(CNC(=O)Cc1csc(=N)[nH]1)C1CC1)C c1(C(N2C(CNC(c3ccc(Cl)[nH]3)=O)CC(OC)C2)=O)coc2c(F)cccc12 C1(C(=O)OC)CCCCC1C(=O)NC1CC1CNC(=O)CCC=C(C)C N1(C(c2cc(C)cc(O)n2)=O)CCC2CCCC12CNC(C1(C)COC1)=O n1(CC)ccc(CNC(C2CCOCC2)CCN2CCC2CC(=O)OC)n1 C1(CC(N2CC3CC(Nc4ncnc(Cl)c4CO)C3C2)=O)CCCC(F)(F)C1 CC(C)C(CCC(=O)NCc1nn(C)c(=O)n1C)NC(=O)CC(C)(F)F c1(OCC)ccc(C)cc1C(=O)N(CCCNC(=O)C(c1cccnc1)N(C)C)C c1(COCC)ccccc1S(=O)(=O)NCc1ncnn1C(F)F c1(C(=O)NC2CCN(C(Cn3c(C)nnn3)=O)CC2C)cc2n(c1)CCCC2 C=CCC(C)(C)CC(=O)NC1CN(C(c2ccc(C#N)c(O)c2)=O)CCC1C C1(CNC(c2c(C)ccc(C)n2)=O)CCC2(CCC2)C1NC(c1sccc1C)=O C1(NCC23CC(C(C(=O)NC)N(c4nnnn4C4CC4)C)(C2)C3)CCCS(=O)(=O)C1 C1(C(N(CCCCCNC(C=CSC)=O)C(C)C)=O)CCc2nn[nH]c2C1 Cc1cc(C(N2CC(N3CCCS3(=O)=O)C2)=O)cc(C)c1 CC(C)C(O)CC(=O)NCC1CC(NC(=O)COc2ccon2)C1 N1(C(C(COCC)C)=O)CCOC(C)C1C(=O)NCC(C1CCCCC1)C CC1CCN(C(c2ccc(C(N)=O)s2)=O)CC1NC(=O)CCc1cnoc1 CCC(CC)(C(=O)NCC1CCC(C(=O)NCc2noc(C)n2)C1)OC c1(C(=O)NCCC2CC(NC(C3(C)ON=C(C)C3)=O)C2)sc(Cl)c(Cl)c1C N1(C(C(C=C)C)=O)CCN(C(C2NC(=O)OC2C)=O)C(CCC)C1 C(=O)(CC(O)CC(C)C)NC1C(CNC(CC(=O)NCC#C)=O)CCCC1 CCCS(=O)(=O)C(C)C(=O)NCCCCC(C)NC(=O)CN(C1CC1)CC N1(C(CCSc2nc(C)[nH]n2)=O)CCC2OC(=O)OC2C1 CC1=C(C(=O)NC2CCC23CN(C(=O)C(F)C(C)C)C3)CCCC1 C(=O)(C(C(=O)N(CCC(C)NC(=O)C(N1CCOCC1)C)C)C1CC1)OCC C1(NC(CCCC#C)=O)CN(C(=O)C#CC2CCCCC2)C2(CCOCC2)C1 C=CC(C)CC(=O)NCCC1CCCN(C(=O)C(C2CCC(=O)CC2)F)C1 C1(C(=O)NC2CC(NC(C(C(C)C)NC(C)=O)=O)C2)CCS(=O)(=O)C1(C)C c1(OC)cccc(F)c1CC(N1CC(F)(CNC(=O)CN2CCCC2C)C1)=O C1(C(CN(C)C)NCC2(C)COCCO2)CCN(C(=O)OC(C)(C)C)C1(C)C C1(NC(C2OCC(C)C2)=O)CC2(CCCN(C(=O)CCC3CCCO3)C2)C1 C1(C(N2CCC(OCCNC(C=CCCC)=O)C2)=O)(OC(C)=O)CCSCC1 c1(NC(C)C)ncccc1C(=O)NC1CC(CCNC(C2CCCC(C)C2)=O)C1 C(=O)(C(C)(C)C(C)(F)F)NCc1nc(C(N2CC(C=C)C(O)C2)=O)c(C)o1 C1(O)(CC(=O)N(C2CCN(C(=O)COCP(C)(C)=O)C2)CC)CCOC1 CC(CCCc1ccccc1)C(=O)N(C1CC(NC(c2cc(Cl)cn2C)=O)C1)C n1(CC)cnc(CCNC(C2(n3cc(-c4cnn(C5CC5)c4)nn3)CC2)=O)c1 c1(C(=O)NCC2(C)CCCN2C(=O)CC2CCCO2)c[nH]cc(Cl)c1=O C1(CCNC(CC#N)=O)CCCCN1C(c1cnc(-c2cnccn2)s1)=O Cc1c(Sc2ccccc2C(N2CCC(O)C(CO)C2)=O)cccc1Br CCCC(O)CC(=O)NC1CCCCC1NC(C1(F)CCCCC1)=O C1(C(N2CCN(CC(C)NC(=O)COC3CC3)CC2)=O)CCC(C)NC1=O C1(C(N2CC(C)(NC(c3c(Cl)cc(C)s3)=O)C2)=O)CNC(=O)CC1C c1(C(N2C(C(=O)Nc3ccc(OC)cc3CO)C=CC2)=O)cn2nc(C)sc2n1 N1(C(C2N(C(C3(COC)CC3)=O)C3C(C2)C3)=O)C2COCC1CC(F)C2 c1(NC(C2N(Cc3n(CC)ncc3)CC2)=O)nccnc1Cl c1(C(=O)NCC2CCCN(C(CC(C=C)CC)=O)CC2)cc2cccc(Cl)c2[nH]1 C(=O)(C(C)CCNC(=O)C(C1CCN(C(=O)CCC2OCCO2)CC1)C)OC c1(C(N2CCCC2c2ccccc2Br)C(=O)NCCCC)ccc(C(F)F)cn1 C(=O)(C(C)(C)CC1CC1)NCC(COC)NC(=O)CC(C)C1CCCO1 N1(C(C(=O)NCCCOC)CC2CCCO2)CCN(C2CC2)C(=O)C1.C1(C)CC1 C(=O)(C(C(C)(C)C)N1C(=O)CCC1=O)NC1C(NC(c2scc(COC)c2)=O)C1 c1(C(=O)NCC(C(C)C)NC(c2csc3nccn23)=O)ccn2ncccc12 C=C(Cl)CC(C(=O)NCc1cccc(O)c1F)NC(=O)CSCCC(C)C C1(=CC(N2CC(NC(CCC3CC(OC)C3)=O)C2)=O)CCOCC1 CC(C)(CCCNC(=O)C(O)Cn1cncn1)NC(C1(F)CCCCC1)=O c1(CC)nnc(O)c(C(=O)N(CCC(C(C)C)NC(c2ccon2)=O)C)c1CC c1(NC(c2nccn2C(C)(C)C)C)ccc([N+](=O)[O-])cn1 C1(OC)CCC2(C(=O)NC(C3CCOC3)CNC(=O)Cc3ccoc3C)CC12 c1(C(=O)NCC2N(C(CCC(C)(C)C#N)=O)CC2)cccc2c1CCC2=O C1(c2nc(COC(C)C)nn2-c2cc(F)ccc2C)CCc2ccnn2C1 CC(C)CC(O)C(=O)NCCCN1CCC(NC(=O)Cc2cnnn2C)C1 c1(C(=O)NCC(C)CN(C)C(c2n[nH]cc2Cl)=O)ccc(CO)nc1 C(=O)(C(CC(C)C)C(N)=O)N1CCCC(NC(c2c(F)cc(C)cc2F)=O)CC1 c1(OC(c2ccncc2)C(=O)OC)csc(COOC(F)F)n1 O=C(C#CC1CCCCO1)N1CCC(CNC(C2(O)CCCCC2)=O)C12CC2 c1(C(N2CC(NC(c3cc(C)ns3)=O)C(F)CC2)=O)nc2cccnc2s1 C1(OC)CC(c2nc[nH]n2)N(C(=O)C(CSCc2ccnnc2C)OC)C1 c1(C(N2CCC(NC(CSCCOC)=O)C(F)C2)=O)c(F)ccc(Cl)c1N N1(C(CCNc2ccc(OC)cc2)=O)CCC(NC(=O)C(C)O)C1(C)C C1(NC(CCC(CC)CC)=O)C(C)(C)CN(C(=O)CN(C)CC)CC1(C)C C(C(C)(C)CNC(=O)CC1C=CCC1)N(C(C=C(C)CN1CCCC1)=O)CCO N1(Cc2cn(C(C)C(=O)NCc3ccccc3)nn2)CCC2(CC1)CC2 c1(OC)ccc(C(C2CC2)Nc2ccc(-n3nc(C)cc3C)cc2)cc1Br N1(C(C2C(CNC(c3c(C)noc3N)=O)CCC2)=O)CC2CC(O)CC2C1 c1(NC2(c3n(CC)nnn3)CCC(c3nccn3C)C2)ccc2c(c1)C(=O)NCC2 n1(CC)cc(C2CC2)c(CN(CC(C)(C)CNC(C)=O)C)n1 C1(C(=O)NCCN(C(CCCC#CC)=O)C2CC2)CC12C(=O)Nc1ccccc12 C(CC(CNC(=O)CCC1OCCO1)NC(=O)Cc1nocc1C)OC c1(-c2cn(CC)nn2)cccc(C(=O)NC2CCN(C(=O)OC(C)(C)C)C2)c1 C#CCC(C)(CC)C(=O)NCc1cncc(C(=O)NC(C)C=C)c1 c1(NC(=O)OC)cccc(NC(=O)CC2CC3CC3C2)c1.C12(CCCC1)C(=O)N2 CCCCC(CC)CCC(C)Nc1cccc(C(C)(C)O)c1 CC1CCC(C(=O)NCCCCC(F)(F)F)N(C(=O)CC2CC3C=CC2C3)C1 N1(C(C(C(CC)C)O)=O)CCC2(CCN(C(=O)CNC(c3ccccc3F)=O)C2)C1 C1(C(=O)NCc2cc(C)c(C)o2)CCN(C(C2(C)CC(=O)N(C)C2)=O)C(C)(C)C1 c1(CNC(=O)C=CCO)ncoc1C1CN(C(=O)CCN2CCC2)C1 c1(OCC)ccc(-n2cccn2)cc1S(=O)(=O)Nc1ccccc1C1CCC1 N1(C(CCCN(C(CC(CC)C2CC2)=O)C)=O)CCC(CO)C(C)C1 N1(C(=O)C(=Cc2c[nH]cn2)F)CC(CNC(C2(Cl)CC2(F)F)=O)C(F)(CO)C1 C1(CC(=O)NC2CC(C)OC2=O)C2CCCC2N1C(C1(O)CCSCC1)=O O(N(C)C(=O)C1CC(C(=O)OC)C1)CCCOCC C(=O)(C(C(C)C)OC)NCC(=O)COC1(CCOCCOC)CCCC1.C1CO1 N1(C(CCCN(C)C)=O)CCC(C)(CNC(C2(c3cccs3)CCCCC2)=O)C1 Cc1ccc(O)c(CN(C)C(=O)Nc2ccc(OC3CCN(C)CC3)cc2)c1 C(=O)(C(C#N)C(C)(C)C)N1CCC(C(C)(C)NC(c2c(CC)scc2)=O)C1 CCCCC(C)C(=O)NC(COCC)C(=O)Nc1cscc1C CC1CCCN(C(c2nocc2Cl)=O)C1CCNC(C1(CO)CC(C)(C)C1)=O C1(CC)C(NC(c2cnc(OC)s2)=O)CCN1C(c1ccnnc1)=O C1(NC(C(CC)=CCCC)=O)CN(C(C2CC2COC)=O)CCC1O N1(C(C2N(C(C)=O)CCC2)=O)CC(NC(=O)CCC(N)=O)Cc2ccccc21 CCCC(C)(CCC)C(=O)NCc1nc(CNC(=O)C(C(C)O)N(C)C)cs1 c1(CC(=O)NC(CC)CNC(=O)C(C)(C)c2nncn2C)ccc(F)cn1 S(=O)(=O)(c1cccc2ccccc12)N1CC(NC(c2cc(OC)ncc2)=O)(CO)C1 CCCC(C)CCCC(=O)NC1CCN(C(c2cc(F)cc(Cl)c2N)=O)C1 C1(C(N2CC(C(C)NC(C3(CC)CCC3)=O)OCC2)=O)CCCC(C)(C)CC1 Cc1ccnc(NC2(N3CCSCC3)CC2)n1 C=CC1CN(C(C2CCCC2O)=O)CC1NC(=O)CC1CC=CC1 C1(COCC(=O)NC2CN(C(C34CC(CO)(C3)C4)=O)C2)C2CCCC12 N1(C(C=CCN(C(=O)CCCn2ccnc2)C)=O)CCOC(CN=[N+]=[N-])C1 c1(C(=O)NC2C(NC(CN(C)CC)=O)CCCC2)cccc(O)c1F c1(C(N2CC(C(C)NC(=O)C(C)C3CCCO3)C2)=O)cc2ccccn2n1 N1(CC2CN(C(C)=O)C2)CCC(NC(=NCc2ccnn2C)NCC(F)F)CC1 N1(C(Cc2cc(C)sc2)=O)CC(NC(c2ncsc2C(F)(F)F)=O)C2CC12 C=CCC(CC(=O)Nc1cc(C)sc1C)NC(C1(OC)CC(C)C1)=O C1(NC(CSCC=C)=O)CCN(C(=O)C(C(C)C)NC(=O)OCC)CC1O Cc1ccc(CC(=O)N(C)CC2CCN(C(c3oncc3C)=O)C2)cn1 C(CS(=O)C(F)(F)F)NC(C(N1CCN(CC)CC1)c1ccc(Cl)cc1)=O c1(C(=O)NCC=CCNC(c2n(C)ccc2)=O)cc2c(nc1O)CC(C)(C)CC2 C1(C(N(C(CC(=O)N(C)Cc2onc(CC)n2)(C)C)C)=O)CC(=O)NC(C)C1 N1(C(C(C)C2(O)CCC2)=O)CCCC(C2(NC(=O)CCn3cncn3)CC2)C1 C1(C(=O)NCC(C2CCC2)OCC)(NC(c2[nH]nnc2C2CC2)=O)CCCC1C Cc1ccn2c(C(N3CCSC4(CCC4)C3)=O)cnc2c1.C1CS(=O)(=O)N1 N1(C(C(CC=C)(F)F)=O)CC(NC(=O)COCc2scnc2C)C(S(C)(=O)=O)C1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCC2(CCC2)C(CNC(=O)CCCC(F)F)C1 C1(CC=C)(NC(=O)C=C(C)C)CCN(C(=O)C=CC2CCOCC2)CC1 CC1CN(C(=O)CCn2ccnc2)CC(C)N(C(c2ccc(F)c(O)c2F)=O)C1 N1(C(N)=O)CC(O)CC1C(=O)NC1CC(NC(c2cn(C3CCC3)nn2)=O)C1 c1(CC(=O)NC(CNC(C=C2CCC(C)C2)=O)CCOC)ccc(C(F)F)cc1 C1(C(=O)NCCN(C(=O)C(O)CC(C)C)CCC)CC2C=CC1CC2 c1(NC(N2CC(C3OCCN(C(C(C)C)=O)C3)C2)=O)ccc(N)c(Cl)c1 c1(C(NNC(c2c3n(nn2)C(C)CCC3)=O)=O)cccc2c1OC(C)(C)C2 Cc1cccc(C(N2CCC(C(N3CC[Si](C)(C)CC3)=O)C2)=O)c1N c1(CNC2CC(C(=O)NC(CO)C(F)(F)F)C2)ncc(Cl)cc1F c1(CC)cc(Nc2c(Cc3noc(C)n3)cccc2)cc(O)c1.C(C)(C(=O)O)O C=CCCC(F)(F)C(=O)NC1CC(F)(CNC(c2ccnc(C3CCC3)c2)=O)C1 C1(C(COC)NC(=O)CCCCn2cc(-c3cn[nH]c3)nn2)CCC(F)(F)CC1 C1(NC(CCCOCCC)=O)CCCCN(C(c2cnc(CC)s2)=O)CC1 C=CCC(CC=C)C(=O)NCC1(F)CCN(C(C2OCCC2C)=O)C1 c1(CNC(CCN(C(=O)CC2CC3CCC2C3)CC#C)=O)cnc(O)c(F)c1 C(=O)(CCCCC(C)C)N1C(Cn2cc(C(C)OCC)nn2)CCC1 c1(NC(C(COC)(C)O)=O)ccc(NC(=O)CSc2nncn2C2CC2)c(C)c1 CC(C)(C)CC(=O)NC1CC(NC(=O)C(C)(C)Cc2ccc(O)cc2)C1 N#Cc1cc(C(=O)Nc2cccc(-c3ccc(SC(F)(F)F)cc3)n2)ccc1O C(=O)(C(C)(C)CCCNC(C1CC2CCC2C1)=O)N1C(C)C(C)(C)CC1 C1(CNC(CCN(CC#C)C(C2CCN(OC)CC2)=O)=O)CCCC(C)CC1 C1(C(N2CC(O)(CNC(C(CCC)F)=O)C2)=O)OCCN(C)C1=O C1(CNC(CCC=C)=O)COC(C(F)(F)F)CN1C(=O)CS(=O)(=O)CC N1(CCC(N2C(CNC(C(C3CCCOC3)OCC)=O)CC2)=O)CCN(C)CC1 c1(N(C)C)ccc(N)c(C(N2CCC(O)C(NC(C3CCCS3(=O)=O)=O)C2)=O)c1 Cc1cc(CC(=O)NCCCN(C(=O)C(C)(C)C2CC2)C(C)C)n(C)n1 C1(C(=O)NC2C(CC(=O)N(CC)Cc3ccco3)CCC2)CC2C=CC1O2 c1cc(OC)c(OC)c(OC)c1N.CNS(=O)(=O)NCC(=O)NC.C12CC1NC2=O c1(C(=O)NCC2(C(=O)NC(c3ccc(Cl)nc3)C)CCC2)ccc2occc2c1 C#Cc1cnc(C(=O)NCC2CCC(C(N3CC(C4CCCO4)C3)=O)C2)c(C)c1 CC(C)CC(O)CNCC(c1ccccc1)c1nc[nH]n1 c1(CC)ncc(C(=O)NCC2CCN2C(c2cc(N(C)C)ccn2)=O)cn1 C(C(C)(C)C(=O)N1CC(N(C)C)C1)N(C)C.C1(=O)C(C2CC2)N1C c1(CCC)c(C(=O)OCc2cccc(-c3cn(C)nn3)c2)cnn1C N1(C(CC23C(CN(C(CSCC)=O)C2)CC3)=O)Cc2ccncc2C1 C1(C(N2C(C)CN(Cc3ccccc3)CC2)=O)CN=C2N=CNN2C1 C1(C#N)(C(N2CC(C(=O)NC(c3nnc(C)s3)C)OCC2)=O)CC(F)(F)C1 c1(C(N2CC3C(CNC(c4c(CC)cccc4)=O)C3C2)=O)cccc(Cl)c1N c1(N2CCC(NC(c3cncc(CC)c3)=O)C(F)C2)ncnc2c(Br)cccc12 c1(C(N2CCC(C)(NC(C3CCC(COC)C3)=O)CC2)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(C2C3CCCCC23)C(=O)NCCC2(C)CC2)CCc2c(cnn2CCO)C1 C=C(C)CC(C(=O)NCC1CCCC12CC2)NC(=O)CCc1cnoc1 N1(C(C(C2CN(C(c3cccc(CC)n3)=O)C2)OC)=O)CCCCCCCCC1 c1(COC)nc(N(C)CC2CCCN2C(=O)CCC(C)(F)F)cc(O)n1 C=CCC(CC(C)C)C(=O)N1CCC(CF)(NC(=O)C(CO)NC(=O)C(C)C)C1 c1(C(N(CC(C)NC(=O)Cc2cnc[nH]2)C)=O)cnc(N(C)C)cn1 N1(C(C2(COC)CCC2)=O)CC(NC(c2ccccc2SC(F)F)=O)CC(F)C1 C1(C(C)NC(=O)C=CCN2CCOCC2)CCN(c2cc(C3CC3)ncn2)CC1 C1(C)(CC)C=C(C(=O)NCc2csc(C(=O)N(c3ccccc3)CC)c2)C1 C(C)(CO)(C(=O)N(C(C)CN(C)C)C)NC(CCOCCCOC)=O C1(CCC(C)C)CCC(NC(=O)Cn2cc(C3(C)CCCC3)nn2)CC1 C1(C(=O)NC2CCC(NC(CC(=O)OCC)=O)C2)CC(=O)NC2CCCCC12 c1(OC)nc(C)ncc1C(N1CC(NC(=O)CN2CC(=O)NC2=O)CC1C)=O CCCCCC(CC)C(=O)N(CCCN(C)Cc1ccc(S(C)(=O)=O)o1)C c1(C(N(C2CCCO2)C(C)=O)=O)cccs1.C1C(=O)OCCCS1 CC1CN(C)CCC1N(C(=O)C=CCNC(C1CCCSC1C)=O)C C1(NC(c2c(C)coc2C(C)C)=O)CC2CN(C(c3cccc(N)c3)=O)CC12 C1(NC(C=C(CC)C)=O)CCS(=O)(=O)C12CN(C(c1cc(C)c(Cl)cc1C)=O)C2 C1(F)(C(N2CC(NC(C3C(C(=O)OC)CCO3)=O)C2)=O)CCCN(C)C1 C(c1ccc(F)cc1)=CC(N1CCC(CCNC(N2CCCCC2=O)=O)C1)=O CC1CN2CCN1C(C(N1CC3(CC(NC(C4CCN(C)C(=O)C4)=O)C3)C1)=O)C2 c1(C(N2CCN(C(C3(CC)CC(C)(C)C3)=O)CC2)=O)cnn2c1CN(C)CC2 N1(C(C=C(C)C(F)F)=O)CC(C2CN(C(=O)CC3CC(O)C3(C)C)C2)C1 CC1CCN(C(c2ncnn2C)=O)CC1NC(c1c(Cl)cnn1C)=O Cc1ccc(F)cc1C(=O)NCC1(F)CC(NC(=O)CC2C=NN(C)C2=O)C1 C=C1CCC(C(N2CCOC(CNC(c3ccncc3Br)=O)C2)=O)CC1 CC1CC(C)(C(N2CCC(F)(CNC(c3ccoc3Br)=O)CC2)=O)CCO1 C1(C(=O)Oc2ccc(C)cc2)CCCCN1SCC(=O)NC(C=C)C.CC N1(C(CC2(OC)CC2)=O)CCOC(CNC(=O)CC2(C)OCCO2)C1 S(=O)(=O)(c1ccc(OC)cc1)N1CC(C(N2CC=CC2CO)=O)(C=O)C1.CO Cc1onc(-c2ccccn2)c1C(N1CCC(Oc2ccc(Br)cc2)CC1)=O N1(C(C=C(CC)C)=O)CC2C(CNC(=O)CCc3nnc(C4CC4)o3)C2C1 Cc1sc(Cl)nc1C(=O)NCCCOCCNC(C12CCC(C1)C2)=O O=C(N=c1cnc(Cl)c[nH]1)C1CN(C(c2c(Cl)nc3sccn23)=O)CCN1 CC(C)(C)C1=NOC(C)(C(N2CC3CCC3(CNC(C3CCCC3)=O)C2)=O)C1 C1(NC(CCC2CC3C(CCC)C3C2)=O)CN(C(=O)OC(C)(C)C)CC1OC C1(NC(Cc2ccc(C)s2)=O)CN(C(=O)CCCOC(C)(C)C)CC12CC2 Cn1c(CCOC(=O)CC2(C)CC2(F)F)nc2ccccc12 n1(CCC)nnnc1C(c1ccnn1CC(F)F)NCc1ccc(Cl)s1 c1(C(=O)NC2(CF)CCN(C(=O)CCc3cnco3)C2)ccc2c(c1)COC2 C1(NC(=O)C(O)c2cnc[nH]2)CCC2(CCN(C(C3(C(N)=O)CC3)=O)CC2)C1 CC(C)(CO)CCCNC(C12CC(CN1C(c1cc(CO)ccn1)=O)C2)=O c1(N(C2CCC2)CCNC(c2cnsc2)=O)ncnc2cc(C3CC3)nn12 Cc1c(C(N2C3CN(C(c4n[nH]cc4I)=O)CC23)=O)ccnc1Cl Cc1ccc(CC(=O)N(C)CCn2cc(CN3CCNC3=O)nn2)c(Cl)n1 c1(NC(C=CC(C)(C)NC(CC2CN(C)C2)=O)=O)ccccc1C1CC1 CCC(CC(=O)NC12CCC(CC1)N(C(c1sc(CO)nc1C)=O)C2)C(F)F CC(C)CC(O)CC(=O)N1CCN(C)CC1C(=O)NCCn1cc(C2CC2)cn1 Cc1nc(NC2CCCC2C(N2CCC2(C)C)=O)ncc1Br CC(C)CCCC(N1CCCC1c1cn(C2(C(C)C)CC2)nn1)=O C1(NC(CC(C)CF)=O)CC2CCC(C1)N2C(=O)CCNC(c1cnccn1)=O Cc1cccc(-c2cn(CCOCCNC(=O)CC(C)(O)SCCO)nn2)c1 C1(CNC(C2C(CC)CCC2)=O)CC(F)CN1C(=O)CNC(c1ccoc1)=O N1(C(c2ccnc(OC)n2)=O)CC(OC)CC(NC(=O)C(O)C(C)(C)C)C1 CCC(CC(=O)NC1CCCC(NC(c2cccn3ccnc23)=O)C1)C(F)F C(=O)(C1CCc2ccccc21)NCCCCCC(=O)NCC1N(C)CCC1 C#Cc1ccc(CC(N2CC3CC(C2)C3NC(=O)C=CC2CCOC2)=O)cc1 Cn1nccc1C=CC(N1CCOCC1CCNC(c1cccc(Cl)c1)=O)=O N#CC1(C(=O)NCC2CC(F)CN2c2cc(C(F)F)ncn2)CC2CC2C1 CCCC(F)(F)C(=O)NC(C)C(=O)NCc1cn(C(C)C)nn1 c1(C(N(C2CCN(C(C3CC(=O)N(C)C3)=O)CC2)CC#C)=O)cc(C)c(Cl)cc1C c1(C(C(=O)NC(C)CN(C(=O)CSC(F)F)C)C)c(F)cccc1F C1(C(=O)NC(COC)CO)CC=CC(NC(=O)C=C2CCC(C)CC2)C1 CN1CCCC1(C)C1CCN(C(c2c(OCC3CCCCO3)cccc2F)=O)C1 C1(C(N2CCC(CCC(=O)N(CCC(C)C)CCO)C2)=O)(OC)CC(O)C1 C(c1ccccc1F)=CC(=O)NC1CC(C)(NC(=O)C(Cl)=CCl)C1 C(C)(C)(CC(=O)N1CCOCC1CNC(c1ccn(C2CC2)c1C)=O)OC N1(C(C(C2CCCN(C(c3n(CC)ccc3)=O)C2)C)=O)CCC2C(O)CC12 CN1CCC(C(=O)NC2CC(N(C)C(c3csc(C(C)(C)C)n3)=O)C2)CC1=O c1(OC)ccc(F)c(-n2nc(C(O)CC)nc2C(C(C)C)OC(C)(C)C)c1 c1(N2CCC(NC(c3c(C)nc(O)[nH]3)=O)CC2)nc2cc(Br)ccc2o1 C#CCC(C)(C)C(=O)NCc1ccsc1C(=O)NC1CC(C)(C)OC1=O c1(C(N2CCC(CCNC(C=CC(CC)=CC)=O)C2)=O)ccc[n+]([O-])c1 N1(C(c2c(N)csn2)=O)CC(CNC(=O)CC(F)(F)F)C(O)C1 C1(C(N(C(CNC(c2ccc(C)cc2O)=O)C)C)=O)CC(C2CCCC2)C1 c1(C(=O)NC2(CC=C)CN(C(C3CCS3(=O)=O)=O)C2)cccc(CSCCC)c1 C1(CN(C(=O)CC2(N(C)C(C3CCCC3)=O)CC2)C)CCCC2CC12 c1(CN2CCC(NC(c3sccc3F)=O)C(F)C2)cnc2ccccc2c1 N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CC2CCN(C(C3CCOCC3)=O)CC12 CC(CC(=O)N1CCC(C)(C)C1CC(=O)N(CC1CC1)CC1CC1)C(F)F C1(C#N)(C(N(C(c2ccccc2)CNC(=O)CN2CCCC2)C)=O)CC2CC2C1 C1(C(N2CCCC(CCC=C)C2)=O)CCC(C)(C)N(C(C23CCC(CC2)C3)=O)C1 N1(C(c2c(CC)con2)=O)CCC2(CCC2)C(NC(c2ccc(O)nn2)=O)C1 N1(C(Cc2cn(CC)nn2)=O)CCCC(NC(=O)C(O)c2ccco2)CC1 N1(C(CCc2ccc(C)o2)=O)Cc2n[nH]cc2C1C(=O)N1CC2CCC2(CO)C1 C1(C)(C(=O)NC(C(=O)NC2CCSC2C)C2(C)CC2)CCCCC1 C1(NC(c2cc(C(C)C)on2)=O)CN(C(=O)C=CC2CCC2)CC12CCC2 C(C(C)(C(=O)N1CCCC(CNC(=O)CCN2CCOCC2)C1)OC)OC N1(C(C(=O)Nc2c(C)nsc2)=O)CCc2nn(CCN(C)C)c(=O)cc2C1 C1(C(N(C)CC2(O)CN(C(Cc3c(C)noc3)=O)C2)=O)CCC(C)(C)C1 c1(CC(N2CCC(C)C(NC(=O)C3=CC(C)(C)C3)C2)=O)c[nH]c2cnccc12 c1(C(N2C(C)CN(C(C(C)C)=O)C(C)C2)=O)cccc(N=S2(=O)CCCC2)c1 c1(CC)nccn1C(C)CC(=O)N(CCC(C)NC(C1(C(C)C)CC1)=O)C c1(CC(=O)NCCOCCNC(CC2CC(=C)C2)=O)nc(C)c(C)s1 Cn1nccc1C=CC(N1CCCC1C(N)=O)=O.N12CCC(CC1)SCC2=O C1(CN(CCCNC(C2(n3cccn3)CC2)=O)C(C2CCCC2)=O)CCCOC1 C12(NC(=O)NS(C(C)CF)(=O)=O)CN(C(=O)OC(C)(C)C)CC1(CO)C2 Cc1cc(C(N2CC3C(NC(c4cc(C(F)F)ccn4)=O)C3C2)=O)cc(C)n1 C1(CC(=O)N(CC(C)NC(c2nsc3ccccc23)=O)C)Cc2ccccc2O1 c1(C(C(=O)N(C(CNC(c2c(C)n(C)cn2)=O)C)C)C)ccc(F)c(F)c1 C1(CNC(c2n(C(CC)CC)nc(C)c2)=O)CN(C(C2C(C)C2C)=O)CC1(C)C CCC(C)CC(=O)NC1CC(C)N(C(C2(CF)CC(F)(F)C2)=O)C1 Cc1sc(Cl)nc1C(=O)NCCCOCCCNC(C1(C2CCC2)CC1)=O C1(NC(c2cc(C3CC3)no2)=O)CN(C(c2cc(Cl)no2)=O)C2CC12 N1(CC2CCCC(C)C2)C(=O)CCN(Cc2ccc(-c3cccc(F)c3Cl)o2)C1=O C1(c2ccccc2)(NC(c2ccnnc2)=O)CCN(C(c2c[nH]ccc2=O)=O)C1 c1(C(=O)NC2CC(NC(C(c3ccc(Br)cc3)C)=O)C2)cnc(O)n1C Cc1c(C(=O)NCC(C(F)(F)F)n2cccn2)cc(F)c2[nH]ccc12 c1(OCC)cc(CN2CCOC(CC(=O)NCc3ccsc3)C2)c(Br)cn1.C(C)S C1(C(=O)NCC(CC)(CC)OC)CCC(C)(C)N(C(=O)C(O)C(C)(C)C)C1 c1(N2CCCCC(COC)C2)ccc(S(=O)(=O)NC2CC=CC2)cn1 C(=O)(C(COC)CC(C)C)N1CCCC(O)(CNC(c2c(CC)noc2)=O)C1 N1(C(CSCc2nc(C)[nH]n2)=O)CCSCC1CCNC(=O)CC(F)F CCCCC(CNC(C1CCN(CCC)CC1)=O)NC(=O)COC c1(OC)nscc1C(=O)N(C1CC(NC(=O)COc2ccn(C)n2)C1)C c1(N(c2ncc(Cl)cn2)C)ccc(Br)cc1[N+](=O)[O-] Cc1nc(O)ccc1C(N1CCC(C(C)NC(=O)CCc2cn(C)nn2)C1)=O N1(C(C2CC(CC)C2)=O)CC2CCC2(CC(N2CCOCC23CC3)=O)C1 CC1(C)CC=C(C(=O)NC(c2ccccc2)C(=O)NC2CCC3CC23)CC1 c1(CC)ccccc1C(=O)NC(C)(CNC(C1CCN(C)C1)=O)CC C1(C(=O)NC2CCN(C(CCCCOCC)=O)CC2F)CCN2CCOCC12 Cn1ncc(C(=O)NC2CC(NC(C3CCC3(C)C)=O)C2)c1-n1cccc1 N1(C(c2n(CC)ccn2)=O)CCCC(C)C1CCNC(c1cscn1)=O Cc1ccc(C(=O)NCC(O)CNC(=O)CCc2ccsc2)c(C)c1 c1(OCC(C)C)ncccc1C(=O)NC(C)CCCNC(=O)CC(F)(F)F CCC(CC)C(C)C(=O)NCCCN1CCN(C(=O)C(C#N)=CC2CC2)CC1 c1(N2C(C(N(CCN(C(C3C(CC)C3)=O)C)C)=O)CCC2)ccc(Br)cc1 C(=O)(CCCC(C)(C)C#N)N1CCC(C(N(C2(c3cccc(Cl)c3)CC2)C)=O)C1 C1(C2CC2)(NC(CC=C)=O)CCN(C(=O)CC2CCCC(C)(C)C2)C1 CN1CCOC(SC(C)(C)Cn2c(N(C)CCF)nnc2-c2cc(Br)c[nH]2)C1 N1(C(CC2(C=C)CCC2)=O)CC2CC(C1)N(C(c1ccc3snnc3c1)=O)C2 C1(=O)CCCC2(CC2)N1.C1(C(NOCC(=O)OC)=O)CC=CCC1 C(=O)(C(C(C)(C)C)C1CC1)N1CCC(N(C(c2cc(OCC)n[nH]2)=O)CCO)C1 C(=O)(CC1=CCCC1)NCCOCCC(=O)N(C(C)C)CCc1ccccc1 C1(C)(CNc2c(C)cc(F)cc2)CC(C(C)C)=NO1 N1(C(Cc2ccc(CCC)cc2)=O)CCC2CC2(NC(=O)CCCF)CC1 c1(CN2CCC(C(N(CCn3c(C)ncc3)C)=O)C2)ncccc1Cl C(=O)(C(COC)CC)NCC(C)N(C(C1CC(CC)(CC)C1)=O)C c1(C(N)=O)ccc(S(=O)(=O)NCC2=CCN(C(=O)COCCCF)CC2)cc1 N1(C(C2C(C)OCC2)=O)CCC(CNC(c2cccc(C3(C)CC3)c2)=O)C1(C)C C1(C(=O)NCC(C2CC2)NC(Cc2c(C)nc[nH]2)=O)CCc2ncccc2C1 C1(COC)CN(C(=O)C(C)P(C)(C)=O)CCN1C(=O)Cn1nccc1C c1(C(C)NC2CCC2)cc(OC)ccc1OOc1ccc(NC(=O)OC)cc1 N1(C(Cn2cc(C(C)(C)C)nn2)=O)CCC2C(NC(C3CCCN3N=O)=O)C12 N1(C(C2C(=O)NCC2)=O)CCC2CN(C(C3CC3C3CCC3)=O)CC2CC1 N1(C(Cc2nc(C)[nH]c2)=O)CCC(NC(=O)CC2CC2(Cl)Cl)C12CC2 C1(C(N2CC(C)OC(C)C2)=O)CCCC(C)(C)CC1 C1(C(=O)NCC)COCCN1C=O.C#CC1CC12C(=O)NCCCOCCO2 Cc1ccc(F)cc1C(N1CCC(O)(CNC(c2cnc(Cl)[nH]2)=O)C1)=O n1(CC)nc2c(c1C(=O)NC1(C)CCSCC1)CCCC2 N1(C(Cn2ncc(C)c2)=O)CCC2CCC(NC(c3ccn(C)c3)=O)C12 n1(CC(=O)NC(C2CCCC2)CNC(C=CC(C)C)=O)nc(C)n(C)c1=O Cc1cc(C(=O)NC2CCC(OCC(=O)O)C2)ccc1-c1ccncc1 c1(C(=O)NC2C(NC(CCOCC#C)=O)CC2)ccc(C(F)F)nc1O Cc1cc(C)nc(-c2cccc(NC(=O)CC(C3CC3)C3CC3)c2)n1 Cc1ccccc1-c1nnn(CC(=O)Nc2ccsc2)n1 c1(NC(=O)Nc2nnc(-c3ccccn3)s2)ccc(Cl)c(F)c1 C1(C(=O)NC(CC)CN(C(=O)CCCC(C)(F)F)C)CCc2c(nnn2CC)C1 N1(C(C2(C#N)C(C)(C)C2)=O)CCC2(CC1)CC2NC(c1ccc(C(N)=O)o1)=O C12(C(N3CCC(O)(CNC(=O)C(O)C4CC4)CC3)=O)CCC(C(F)F)(CC1)CC2 CC(C(=O)NC1CC(CNC(C2(C#N)CCOCC2)=O)CC1O)S(N)(=O)=O c1(OC)ccc(C(=O)CC(=O)NCC2CC(O)CN2C(=O)C2=CCC2)cc1F C1(OC)CC(CCNC=O)N(C(=O)C(C)OCCN(C)C)C1.C1(C(=O)N)CCOC1 C(C(C(=O)NCc1nnnn1CC)C(C)C)NC(C1(CC)CC1)=O C1(C)C(=O)N1.C(CC1CC1)(CO)NC(COCCCC)=O N1(C(CCC)C)CC(C(=O)NCCCN(C(=O)COC2(C)CCCC2)C)CC1=O C(=O)(C(C)(F)C(F)(F)F)N1CC(OC)C(NC(c2ccnc3c2CCO3)=O)C1 Cc1cc(C2(C(=O)NC3CC(SCCNC(c4cnnn4C)=O)C3)CC2)no1 CC1CN(C(=O)Cc2ccc(O)c(C(N)=O)c2)CCN1C(=O)C(O)C(C)(C)C C1(CC)CN(C(=O)C=C2CCC(C)CC2)CC1C(=O)N(CCF)CCOC c1(NC(CCC=C)C2CC2)nc(=NCCc2cncn2C)[nH]c2c(C)nn(C)c12 c1(CNC(C(CNC(C(C)OCC=C)=O)C)=O)cnn(C)c1C c1(C(N2CCCC(NC(C=CC)=O)CC2)=O)ccc(S(=O)(=O)NOC)cc1 c1(C(N(C2CCN(C(C3C(CCC)C3)=O)C2)C)=O)ccc(=O)n(CC)n1 c1(C(N2C(CN(C(C(C)=C3CCC3)=O)C)CCC2)=O)cc(Br)nn1C N1(C(C(COC(C)C)NC(=O)CCCC(=O)C2CC2)=O)CCCC(O)(C2CC2)C1 c1(CC(=O)NC(CNC(CCc2n(C)ccn2)=O)C2CC2)cccc2nsnc12 C1(C(=O)NC(CC)C(C)(F)F)CN(C(c2sccc2CO)=O)CC(C)(C)C1 C1(NC(c2c(C)nc(Cc3ccccc3)s2)=O)CC2CCC1N(C(=O)C(C)(C)F)C2 CCC(CC(C)CO)N=c1cc(C)nc(N(C)Cc2nnc(C)n2C)[nH]1 C(=O)(C(C(C)O)N(C)C)NC(C1CN(C(CN(C2CCCCC2)CC)=O)C1)C C1(CNC(=O)NC2CCOCC2SCC2CCCC2)Cc2ccccc2CCO1 C1(CN(S(=O)(=O)CC2CCC2)C)CCCN1C(C1(C(F)F)CCC1)=O N1(C(CC(C)(C)N(C)C)=O)CCC(NC(C2CC(C)(C)OC2(C)C)=O)CC(O)C1 C1(COC)(NC(=O)CN(C)C(C)=O)CCN(C(=O)CC(C2CC2)C2CC2)CC1 C1(C2CCCN(C(=O)CC3OCCO3)C2)(NC(c2c(F)ccnc2F)=O)CC1 CCC(C)(CCC(C)C)C(=O)NCCC1(NC(=O)C(F)C2CC2)CCCC1 C1(C(C)(C)NC(C(c2ccn(C)n2)C)=O)CCN(C(=O)CO)C1 c1(CNC(C2CC(NCc3ccc(C)c(Br)c3)C2)=O)n[nH]c2c1CCCC2 C(CCNC(=O)CSc1ccccn1)(C(=O)NC1CC(C(F)(F)F)C1)OC C1(C(N2CC(CCOC(C)C(=O)NCC3CCCO3)C2)=O)CCCN1C1CC1 CC1CC(C(=O)NC2(CNC(c3cc[nH]n3)=O)CCCC2)CC(C)C1 N#Cc1c(NC(C2(CNC(c3sccc3Cl)=O)CC2)=O)cc(F)cc1F c1(C(=O)NC2C3(CC(NC(C4C(CC)C4(C)C)=O)C3)C2)nccn2nccc12 c1(CCC2C(C)CCN(C(=O)C(N3CCCC3CO)=O)C2)c[nH]c2ccccc12 c1(C(=O)NCCNC(C(CC)Oc2ccccc2F)=O)cc(C)n(C)c(=O)c1 c1(C(=O)NC2C(NC(=O)COc3cncc(Cl)n3)CC2)c(Cl)oc2ccccc12 C1(C(=O)NC(C(=O)OC)C2(C)CC2)CCN(C(c2cc(=O)cc(C)[nH]2)=O)CCO1 N1(C(C(C)OCCl)=O)CCCC2C1CCN2Cc1ccc(F)cc1Cl c1(CC(=O)NCCN(C(=O)CCCc2cnccn2)CCC)ccc(O)cc1 C#CC(C)(C)C(=O)NCC(C)=CC(=O)Nc1ccc(C(C)CC)cc1 N1(C(c2c(N)cn(C)n2)=O)CCC2(CCCN(C(=O)C(F)CC3CCC3)C2)C1 c1(C(=O)NC2CCCC(CNC(CCS(C)=O)=O)C2)cccc2nc[nH]c12 c1(C(=O)NCC2(OC)CCN(C(c3cscc3C)=O)C2)cnccc1C#N N1(c2nnc(C)o2)CCCC(C)(C)C1CNC(=O)CC1CCC(C(F)(F)F)O1 Cc1ccccc1COCC(=O)NCCC1(CNC(=O)CCC(C)C2CC2)CC1 C1(C(N(C2C3CN(C(c4cncn4C)=O)CC23)C)=O)CN2CCN1CC2 Clc1ccc2c(c1)CN(c1nccc(=NCCOCC3CCOC3)[nH]1)CCN2 C(=O)(C(C)(C)CS(N)(=O)=O)N1CCC(NC(c2cc(C)n(C(C)C)n2)=O)C(C)C1 C(=O)(C(COC(C)C)N(C)C)NC(C(=O)NC(C1CCOC1=O)CC)C1CCC1 C(=O)(C1CC(=O)c2ccccc21)NC1C(SC)CN(C(=O)Cn2ncnn2)C1 c1(C(=O)NCCN(C(=O)CC2C(=O)NN=C2C)CC)cncc2ccc(F)cc12 N1(C(C(C(CCC)NC(COCCCC)=O)O)=O)Cc2cccc(C)c2C1 N1(CCC(=O)N(CCN(C(=O)CN2CCCC2=O)C(C)C)C)CCP(C)(=O)CC1 C#Cc1ccc(F)c(C(N2CCC(OCCNC(=O)CC3CCOC3)C2)=O)c1 Cn1cnn(CC(=O)NC2(CNC(c3coc(C(F)F)n3)=O)CCC2)c1=O C1(C(=O)NC2C(C)CN(C(C3CC3(C)Br)=O)C2)CCc2ccccc2O1 C1(NC(c2cccnc2)=O)CC2CC(C1)N(C(c1sncc1Br)=O)C2 CCC(CC(C)C)C(=O)N(C(C)CNC(c1ccnc2cc[nH]c12)=O)CC C(=O)(CCC(C)(C)CCC)N1CC(C=C)C(NC(c2cocn2)=O)C1 C1(CNC(C2(OC)CCOC2)=O)C2CCC(C2)N1C(=O)CCOc1ccccn1 CC(CC(=O)N1CC(NC(=O)COC2CCOC2)CC1C)CC(F)(F)F CS(=O)(=O)c1ccc2c(c1)CN(C(=O)C(=C1CCOCC1)F)C2 C1(C(N(C2CC3CCC(C2)N3)C2C(C)C2)=O)CCc2ccccc2C1 CCC(C)(C#N)C(=O)NCC(C(=O)NC1(CF)CCCC1)N(C)C c1(C(c2n(C)nnn2)NCC(F)CO)cnc(O)c(Br)c1 N1(C(CCN(C(C)C)C)=O)CCS(=O)(=O)C(CCNC(=O)C(=O)NC2CC2)C1 C(CCC(C)C)(C(=O)N1CCC12CCC2)NC(C1ON=C(CC)C1)=O C1(CC(=O)N(CC(COCC(COCCOC)O)O)C)CC(O)C1(C)C N1(C(c2nnn(C(C)C)n2)=O)CCC(C(C)CNC(C2(C(F)(F)F)CC2)=O)CC1 c1(CC(=O)NCC(CNC(CC(C)(C)O)=O)(C)O)cc(Br)ccc1F C1(CC)CCN(C(=O)CC(O)CN(C)C)C(C(=O)NCC=CC(C)(C)C)C1 c1(CC(=O)NCC2(O)CCN(C(C3(C(=O)OCC)CC3)=O)C2)cc(F)ccc1C C(C)(C(N=c1nc(C2CCCC2)[nH]s1)C(C)C)NC(c1c(C)nsc1)=O N1(C(C2CC2F)=O)CCC(n2cccn2)(CNC(C23CSC(C2)C3)=O)CC1 C1(CN(C(C2(CN(C)C)CC2)=O)CC)CCN(C(C2CC(F)C(=O)N2)=O)CC1 N1(C(C2CC23CCC3)C(=O)NCC(F)F)CCN(CC2CCOC2)CC1 Cc1nc2cccc(Cl)c2cc1C(=O)NC1CCCN(C(=O)C(C)(C)C(C)C)C1 c1(C(NOC(C=C)C)=O)ncccc1NC(C1CCNC(=O)C1)=O CCC(C)(C(=O)NCC(C)CNC(=O)CCNC(N)=O)C(N)=O CCC(C)CC(C(=O)NC(C1(N(C)C)CC1)C)NC(=O)C(=O)NCC1CC1 C(=O)(CC(N)CCS(C)(=O)=O)N1CCC(c2ncc(CC)s2)C1 c1(OC)cc(C(=O)NCC(C)N(C(=O)CCN(C)C(C)=O)C)c2ccccc2n1 N1(C(c2n(CC)ccc2)=O)CCC(C(=O)N(C2CCCC2O)C2CC2)C(C)(C)C1 C1(NC(c2c(C(C)NC(=O)CSC(F)F)noc2)=O)CN(C)CCC1O N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)C(=O)NCC2CC2)C(CO)C1 C1(C(N(CC#CC)C)=O)COCCN1C(c1n[nH]cc1C)=O c1(C(=O)OCC)cc(S(=O)(=O)NCCF)c(F)cc1Br Cn1cc(CC(=O)OC2CCCOC2=O)c2ccccc12 c1(C(=O)NCCC(=C)CNC(=O)C(C)CC(N)=O)cc(=O)n(C)cn1 Cc1cn2nc(N3CCn4ncnc4C3)cc2c(N2CCCCC2C)n1 N1(C(C(C)NC(CC)(C)C)=O)CC(NC(c2cccc(C)n2)=O)CC12CCC2 C(=O)(CC(C(F)(F)F)c1ccon1)NCC1N(C(c2cc(C)[nH]n2)=O)CC=C1 c1(C(N2C(C(=O)NC3(C)CN(C(=O)OC)C3)CC2)=O)cc(CO)ccn1 C12(C(=O)Nc3nccc(C(=O)OCC)n3)CC(CO)(C1)OC2C CC(CC(C)(C)C)C(=O)NCC1CCCN(C(c2cc(C(N)=O)ccn2)=O)CC1 c1(SCC(=O)N(C2CCC(NC(=O)CCc3ccco3)C2)C)ccccc1Cl C1(C(=O)NCC2CC[Si](C)(C)C2)(NC(c2nc(OC)oc2)=O)CCC(C)(C)C1 Cc1ccc(CN(C(c2ncc(Br)s2)C(=O)NCC2CC2)C)s1 c1(C(N2CCOCC(NC(c3ccnc(C)n3)=O)C2)=O)nc(C)c(C)[nH]c1=O Cc1sc2ccccc2c1C(N1CC2CC(NC(=O)CC3CCC3(F)F)C1C2)=O c1(C(=O)NCCCCNC(C2C(C(C)C)(CC)C2)=O)ccc(OC)c(F)c1F c1(C(C)C)cc(N2CC(NC(=O)C(C)OCc3ccncc3)CC2C)nc(Cl)n1 N1(C(c2c(C(C)NC(c3ccc(=O)n(C)c3)=O)noc2)=O)CC2CCC(O)CC2C1 c1(OC)ccc(C2(C(=O)N(C3CC(NC(=O)CN4CCNC4=O)C3)C)CC2)cn1 c1(CC)c(C(N2CCOC(CNC(C3(C(N)=O)CC3)=O)C2)=O)oc2ccccc12 c1(C(N2CCC(COC)CC2)C(=O)NCCC)cc(=O)n(C)c(=O)n1C C1(C(=O)NC(CC)CNC(C23CC(CCO2)C3)=O)CCC2(CC1)CC2 C1(CNC(c2n(CCCC(=O)OC)nnn2)c2cnsc2)CCc2cnn(C)c2C1 C(=O)(C1CCCc2ccccc21)NC1(C)CN(C(=O)C2CCCn3ncnc32)C1 c1(C(N2CCN(C(C3C4CNC(=O)C43)=O)CC2)=O)c(F)ccc(I)c1Br C(=O)(C(C)C(C)(C)C)N1C(CC)C(NC(c2cnn(C3CCOCC3)c2)=O)CC1 c1(OC)cc(Br)c(C(c2nnnn2CCC2CC2)NCC2C=CCC2)cc1Cl c1(C(C)C)ccccc1NC(=O)CN(C(=O)Cc1cc[nH]n1)C c1(C(=O)NCC(CNC(C2(C)CCCS2)=O)OC)ccc(C)c2c1CCC2 c1(CC)cc(C(=O)NCC2(F)CC(NC(C3(C(F)F)CCCO3)=O)C2)oc1CC CCC(C)(C(=O)O)NC(=O)C(F)CC1CC(F)(F)C1 C(=O)(CCCSC)N(CCOC)CCNC(=O)COCC(C)(C)C N1(C(CN(CCC)C(C2CC2CC(C)C)=O)=O)CCOCCC1C C1(CCC)CN(C(=O)C(CCSC)OC)CCN1C(=O)CC1(C)CCCC1 c1(C(=O)NCC2C(NC(c3c(C)nc(CC)o3)=O)COC2)cc(OC)cc(C)c1 c1(CC(N2CCC(NC(C(C)SC)=O)C2C2CC2)=O)cc(Cl)cnc1C n1(CC(=O)NCC2N(C(CNS(C)(=O)=O)=O)CC2)ccc(C2CC2)n1 c1(C(=O)NC2(CNC(c3csc(C)c3)=O)CC(OC)C2)sc(C2CC2)nc1C c1(CCNC(C2COCCC2NC(=O)C(F)(F)CO)=O)cccnc1F C1(CNC(C23CC(C)(OCC2)C3)=O)CC2CCC(C1)N2C(=O)CC1CC(F)C1 N1(C(C(=O)NCC2CCOCC2)C2CC2Cl)CCC2OCCCC2C1 c1(CNC2C(C(=O)Nc3cc(OC)nc(C)n3)CCC2)cccc2c1OCCO2 c1(C(=O)NCCCCNC(=O)CCCc2ccncc2)cc2c(s1)COCC2 c1(C(=O)NC2C3CC(NC(C(C=C)OC)=O)CC32)ccc(S(C)=O)cc1 C=CCC(C(=O)NCC1CC(C(=O)NC(C)CS(C)(=O)=O)C1)OC C(CC1CCC1)(C(=O)NC1(CCNC(c2cc(CCO)on2)=O)CC1)OC C1(C(=O)NC(c2cn(CC3C(OCC)COCC3)nn2)C)CC(F)(F)CS1(=O)=O c1(C(N2C(CNC(C=CC)=O)C(COC)CC2)=O)cccc(N=c2cc[nH]cc2)c1 c1(-c2c(C(=O)NC(CC=C)CC)c[nH]n2)ccc(OC)cc1 Cc1ccc2[nH]nc(C(=O)NCC=CCNC(c3sccc3C(N)=O)=O)c2c1 C1(NC(C2(CCC)CC2)=O)Cc2ccccc2C1NC(=O)COCC(F)F N1(C(c2ncn(C(C)C)n2)=O)CC(O)CC1CNC(C1COCCO1)=O c1(C(=O)NC2(CCCNC(C(CC)O)=O)CC2)cn2cc(C)nc2s1 N1(C(c2cnn(CC)n2)=O)CCCCC1CCNC(C1OCCOC1C)=O N1(C(CCC)=O)CC2OCC(NC(c3sc(-n4cccc4)nc3C)=O)C2C1 N1(C(C(C)(CO)OC)=O)CCC2(C1)CN(C(=O)C=CC1CCCCC1)CC(C)O2 N1(CC(COC)O)CC2CCC(NC(c3n[nH]c4c3CCCCC4)=O)CC2C1 C(C)(c1cnn(C)c1)=CC(=O)NCC1(CO)CC(NC(C(C)(C)SC)=O)C1 C(N=c1nc(C(F)(F)F)[nH]s1)C1CCCN(C(c2ccc(C(N)=O)o2)=O)C1 c1(SC)ccc(CCNC(=O)N(C2CCC2)CC2CC2)cc1 c1(NCC2CC(NC(c3cnc(C)nc3O)=O)C2)ncnn2c(Br)ccc12 CCCC(C)C(=O)NCC(c1ccccc1)CNC(=O)CCCNC(C)=O c1(C(=O)NC2C(CNC(CCC(=C)C)=O)COC2)cccc(O)c1Br c1(C(=O)NC2CN(C(COCC(C)C)=O)C2)c(C(F)F)nc2n1CCCC2 c1(CNC2CC3(C(NC(CSc4cccc(C)c4)=O)C3)C2)cccc2c1CCC2 c1(C(=O)OC)ccc(C(=O)NC2CC2CNC(=O)CC2CC(N(C)C)C2)c(O)n1 c1(NC(c2n(C)nnn2)CC2CC2)ccc(S(=O)(=O)CF)cc1 N1(C(=O)Cn2cnc(C(F)(F)F)n2)CCCC2(C1)CN(C(c1ccncn1)=O)C2 CC1(C(=O)NC2CC(CNC(=O)C(c3ccsc3)C3CC3)C2)CC1(Cl)Cl C(N=c1nc(N2CC(C)(C)OC(C)(C)C2)cc(C)[nH]1)c1cnn(CCC)c1C C(=O)(CCCC(CC)NC(=O)C(O)C1CCC1)NCCCOCC=C N1(C(c2cnc(CC)[nH]2)=O)CCN(C(=O)CN(C)CC)C2(CC2)C1 C1(NC(c2c(C)cc(C(F)(F)F)s2)=O)CCC2CCN(C(=O)C=CC3CC3)C1C2 n1(CCC#C)c(N(C)CCSC)nnc1C1CC1C(C)(C)C CCC(C(F)(F)F)NC(=O)C(CCOC)NC(=O)CC1CC2CC2C1 C(=O)(CC(C)(C)C(F)F)N1CCC(C(C)(C)CNC(=O)C(O)C(C)(C)C)CC1 C1(C(=O)NCC2C(NC(CCSCCCC)=O)C2)C(c2ccccc2)C1(C)C.C CCC(C)(CCNC(=O)Cn1cnnc1)NC(C1CCCOC1C)=O N1(C(c2cccc(C3CC3(F)F)c2)=O)CC2(CCN2C(=O)CSc2cccs2)C1 C1(NC(c2cc(C3CC3)no2)=O)CS(=O)(=O)CC1NC(c1cc(Cl)cnn1)=O C1(C(N2CCCC(NC(C(CC)=CCCC)=O)(CO)C2)=O)CC2CCC(C1)N2C CC1CCCCC1(C)n1cc(C2CN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2)nn1 c1(CC)nc(N2CC(CCOC)(NC(C3CCOC3CC)=O)C2)c2ccsc2n1 CC(C)(C)C(=O)Nc1nc(C(=O)NCc2cn(Cc3ccno3)nn2)cs1 C1(CNC(c2ccc(SCC)cc2)=O)CC2CCC(C1)N2C(=O)CCCCSC C(=O)(CC(C(F)(F)F)OC)N1CC(CC=C)(NC(c2cc(CC)[nH]n2)=O)C1 CC(CCCCNC(C1CCSC1)=O)NC(=O)CC1CCN(CCF)CC1 c1(C(=O)NC2CC2NC(c2cnc(C(F)(F)F)o2)=O)cc(Cl)c(F)c(Cl)c1 CCCCCCCCCCC(=O)N1CCC(Cn2cc(C3CCN(C)C3)nn2)C1 c1(C(=O)NC2C3CN(C(C(CCCOC)C)=O)C2CC3)ccc2c(c1)NC(=O)C2 C#CCC(C)(C(=O)NCC(C)C(=O)OC)NC(=O)C(C)NC(=O)OC C1(C(=O)NCCCCC#CC)N(C(=O)COC2CCOCC2)CC12CCCC2 CC(CCN(C)C)C(=O)N(C(C)CNC(=O)COC(F)(F)F)C C12(CC(C)C)CCN(CC1)C2=O.c1(NC(C=CC)=O)cc(OC)cc(Br)c1 c1(C(=O)NC2CCCC(NC(C(C)=C3CCCC3)=O)C2)occ2c1CCOC2 C12(CNC(C(=O)NC(C)C)=O)CC1CN(C(c1cn(C3CCCC3)nn1)=O)C2 C1(C(N(C)CCN(C)C(C2C3(CC3)C23CC3)=O)=O)C2CCC(C2)S1(=O)=O C1(CNC(c2c(CC)n(C)nc2)=O)CC(F)(F)CN1C(c1cc(Cl)on1)=O c1(C(=O)NCC(CNC(C(CC)C#N)=O)OC)coc(S(N)(=O)=O)c1 Cc1ccc(CCCCC(=O)NC2CCC2NC(=O)Cn2nc(C)nc2C)cc1 C#CC1CN(C(=O)NCC(=O)OCCC2(c3cccs3)CC2)CCO1 C1(CNC(c2ccsn2)=O)C=CCN1C(=O)CCCc1cc[nH]n1 O=C(C1=NOC2(CCN(C(=O)Cc3ccc(Cl)s3)C2)C1)Nc1ncc(F)c(Cl)n1 c1(C2(CC(C3CC3)Nc3cccc(CC)c3)CC2)ccc(Cl)cc1Cl Cc1cc(C(N2CCC(NC(C3(F)CCCOC3)=O)C(C)(C)C2)=O)cc(N)c1O c1(C(=O)NCCCN(C2CCCC2)C(Cn2c(C(C)C)nnn2)=O)sccc1Cl N1(C(C2C(C)CCN2C(c2cc(CO)[nH]n2)=O)=O)CC2(C1)CC(C)(O)C2 CC1CN(C)CC(C(=O)N(C(C)CCNC(C2COC(=O)N2)=O)C)O1 C1(CN(C(=O)Cc2csc(S)n2)CC)CCCN1C(=O)C(C1CC1)SC N1(CC(=O)NCC2CCN2C(=O)Cc2nncs2)CCCCCC1 C1(CC(=O)N(CC)CC2CC2)CC(C)(C)CN1C(=O)CSCCC(C)C c1(C(=O)NC(C)(CNC(=O)C(F)(F)C(O)C2CC2)C2CC2)ccc2ncnn2c1 CC1(C)CNC(=O)C1NC(C1CCCCN1C(=O)CCC1CCC1)=O S(=O)(=O)(c1cc([N+](=O)[O-])cc(Br)c1Cl)NCCCc1ccc(OC(C)C)cc1 C1(NC(c2c(C(N(C3(C(N)=O)CC3)C)=O)coc2)=O)CC(C)N(C)CC1C CC(CC(=O)N(C(C)(C(=O)NCc1ccccc1)C1CC1)C)n1cccc1 C1(NC(CC2(C)CCCCC2)=O)CN(C(c2cc(Cl)ccc2F)=O)CC1C#N c1(C(N(CC(C)N(C(C(CC=CC)C)=O)C)C)=O)ccc(N)cc1Br n1(CC)ccc(C(=O)NCC2CC3CCC2N3C(=O)CC2CSCCS2)cc1=O C12(C(N3CCC(CC(C)NC(C(C)OCCCC)=O)CC3)=O)CCC(CC1)CO2 c1(C(=O)NC(CC=C)CNC(C2CCC(F)CC2)=O)cc(O)cc(Br)c1 C(=O)(C(F)(F)C(O)C(C)C)NCC1CN(C(C2(C=C)CCCCC2)=O)CC1C Cc1cc(C(C)N(C)C)c(C)n1C1C(C(F)(F)F)CCN(C(C2(C3CC3)CC2)=O)C1 c1(C(=O)NCC2C(C)(C)N(C(=O)CC3(O)CC3)CC2)n[nH]c2ccc(Br)cc12 C(=O)(CC1=NNC(=O)C1)NCC1CCCN(C(C(c2cc(C)c(F)cc2)=O)=O)C1 c1(NCc2c(Br)ccc(C)c2)ccc(S(=O)(=O)NCCCCF)cc1Br CN(C)S(=O)(=O)N1CC(C(=O)NCCNC(C2CCCC(O)C2)=O)C1 C1(C(=O)NCC2CCN(C(c3nc(CC)[nH]n3)=O)CC2C)CC2(CCCC2)CO1 C1(NC(c2ccc(C(N)=O)o2)=O)CCCC(NC(C2CC(=O)N(O)C2)=O)C1 C1(n2c(-c3ccc(C(C)(F)F)cc3)nc(CC)n2)CCOC(C)(C)C1 C1(NC(CNC(C)=O)=O)CCN(C(=O)C(c2ccccc2F)C)C1C N1(CC)CCCCC1C(=O)NCCNC(=O)C(F)CC1CCCC1 C1(CNC(c2cnc(C)[nH]2)=O)CC(C(F)(F)F)CN1C(=O)CCOCC1CC1 C(=O)(C(F)CCC(C)(C)C)NC(C)C(N1CCC(F)(F)C1)=O C(=O)(C(F)(F)c1nccs1)NCCN(C)C(C1CC(n2ccnn2)C1)=O c1(C(=O)NC(CNC(CNC(C)=O)=O)(C)C2CCC2)cc(C#N)on1 Cc1nc(C(N2CCC(C(C)(C)NC(C3CCCC3C)=O)C2)=O)c2ccccn12 N1(C(C(CN(C)C)(C)C)=O)CC2CC(NC(c3cnn4c3NCCC4)=O)CC2C1 c1(OC)cc(C(=O)NCCNC(C2(C)CC2F)=O)ccc1C(F)F c1(C2(C(=O)NCC(CC#C)O)CC2)ccc(OC)c(C)c1 CC(N=c1cc[nH]c(-c2nccs2)n1)c1ccc(OCC(F)(F)F)nc1 O(P(C)(=O)CCNC(=O)C(=O)OC)CC c1(C(=O)NC2(CC=C)CCCN(C(=O)C(F)C(=O)OC)C2)cc(F)c(F)cc1Cl C=CCC(CC(C)C)C(=O)NCCC1CC(NC(c2ccncc2Br)=O)C1 c1(SCCC(NC2=NCC(C(F)(F)F)N2)=O)c[nH]c2ccc(F)cc12 C12(C(N(CCC(C(C)C)NC(C=CCC)=O)C)=O)CCCN(C1)S(=O)(=O)C2 C1(CNC(C2N(CCC)CCC2)=O)CN(C(c2ncncc2Cl)=O)CC1(F)F CC1(C(=O)NCC23CC2CN(C(C2(CC4CC4)CCC2)=O)C3)CCCNS1(=O)=O Cc1cc(C(N2CCOC(CCNC(c3nsnc3O)=O)C2)=O)c(C)o1 C1(C(=O)NCC2(OC)CCN(C(=O)Cc3cn[nH]c3)C2)CCCCC12CCC2 c1(C(=O)NCCCN(C(c2cc(CO)n(C)n2)=O)CC)cc(Cl)ccc1Cl c1(C(N2C(C(N3CC4CCC3C4)=O)CC(C)C2)=O)cn2cccc(Br)c2n1 N1(C(CCCOC(C)C)=O)CCC(CNC(=O)C=Cc2cnc[nH]2)C1(C)C c1(C(=O)N(C(CC)C(=O)OC)C)cc(N(C)C)cc(C(F)(F)F)c1 N1(C(c2c(CCC)n[nH]c2)=O)CCC2(CC1)COC(CNC(=O)CN(C)CC)C2 C(CCCC(CO)NC(=O)Cc1nc(C)sc1C)NC(c1ncn(CC)c1)=O C1(CCC(=O)NC2CCCC23CC3)CCCCN1C(=O)CCCn1cc(OC)nn1 c1(-c2n(C(CC)C)nc(CSc3ccccc3)n2)cc(C)nc(NC)n1 Cn1ncc2c1CC(C(=O)NC1CCN(C(=O)CCc3cccc(F)c3)C1)CC2 N1(C(C(C)N(C(=O)COCCF)CCC)=O)CCn2ccnc21 C1(N(C(C(=Cc2cn[nH]c2)C)=O)C)CCCCC1CN(S(C)(=O)=O)C Cc1cc(C)cc(S(=O)(=O)N2CCC(CC(=O)NC3CCC(F)(F)C3)C2)c1 Cc1ccc(C2CC2C(=O)NC2CCCN(C(C3C4(CC4)C34CC4)=O)CC2)c(Cl)n1 c1(CCC(=O)N(C2CN(C(=O)C3=NOCC3)C2)C)nc2cccc(F)c2[nH]1 Cc1cc(C(=O)NCCOCCCNC(c2ccnn2CCOCCO)=O)n[nH]1 C1(C(=O)NC2CCN(C(C)=O)C2)CCCCC1CNC(=O)CSCC(C)C C(=O)(C1c2c[nH]nc2CN1C(=O)C=CC1CCOCC1)NC1CN(CC)CC1C c1(N)nc(CC)cc(OC)n1.C1(N(CC)CC)CCC(NC(C2(CCF)CC2)=O)CC1 C12(CCCCC1)C(=O)N2.C1(F)(CN(C)C)CC(NC(c2cc(Br)co2)=O)C1 c1(OC)cc(N(C)C)ccc1CNC1CCN(C(c2cc(O)cc(O)c2)=O)C1 C(=O)(CC1COCc2ccccc21)NCC1CCN(C(CC(=O)OCC)=O)CC1 n1(-c2cnc(C)s2)nc(-c2cccc(OC(C)C)c2)nc1CC1CCC2(CC2)C1 N1(C(C(C2CC2)SC)=O)C2CCC1C(CNC(=O)CC1CC1)C2 N1(c2ccc(S(=O)(=O)NCc3c(C)onc3)cn2)CC(C)OC2(CCCC2)C1 c1(C(=O)NC(C(C)C)CNC(c2coc(O)n2)=O)ccnc2c1CCC2 C(CN=c1[nH]c(=NCCCC(=O)N2CCC2)c2cc(OC)ccc2[nH]1)SCC c1(C(N2CCN(c3ccnc(C)n3)C(C#N)C2)=O)cc(C)cc2[nH]ccc12 c1(OC)cc(C(=O)N(C(c2ccccc2)CNC(=O)CC2C=CCC2)C)n(C)n1 CC(CCC(=O)NCc1cn[nH]c1)NC(=O)C(O)CN1CCCC1 C1(C(C)NC(=O)CNS(C)(=O)=O)CCCN(C(C2CC3CC3C2)=O)C1 c1(OC)cccc2c1OCC(NC(=O)NCCCCc1nc(=N)[nH][nH]1)C2 Cc1ncccc1CC(N1CC(F)CC1CNC(=O)Cc1cccnc1Br)=O c1(CNC(=O)Nc2ccc(C(C)(C)C(=O)O)cc2)ncc([N+](=O)[O-])o1 N1(C(C2C(C(C)C)N(C(c3ncncc3N)=O)CC2)=O)CC(C)C(C)C1C CS(=N)(=O)C1CC(NC(=O)C(O)C2(N)CC2)C1 c1(CC)nnc(N(CCCCN(C(c2ccn(CCn3cncn3)n2)=O)C)C)s1 S(=O)(=O)(c1ccc(N(C)CC)cc1Br)NCCCN(C(n1ccnc1CC)=O)C C1(OC)CN(C(c2cccc(C#N)c2)=O)CCC1NC(=O)CCC1CCC(C)O1 C1(C)(CC(=O)NC(c2cn(C3COCCC3O)nn2)CCC)CCCC1(F)F C1(NC(c2c(CNC(C(C)c3cc[nH]n3)=O)noc2)=O)CC2CCC(C1)O2 CC(CC(N)=O)C(=O)N1CCCC1C(C)(C)C(=O)N(CC(C)(C)C#N)C c1(C(=O)NCCCN(C(COCCCC#C)=O)C)cc2c(nc1O)CCCC2=O C(CCCCC(=O)NC1CCOC1=O)N(C(=O)CC1CC(=O)NC1=O)C N1(C(C(CC=C)C)=O)CCCCC12CC(NC(=O)CCC1CC1(C)C)C2 c1(C(=O)NC2COCCN(C(c3nc(C)sc3)=O)C2)ccc(N)c(C)c1C c1(CC(C)C(N2CC(NC(=O)CSC3CC3)C(CO)C2)=O)ccc(F)cc1F C(=O)(C1CCCc2cncn21)NCC(CNC(c1cc(OC)ncc1)=O)F c1(C(N2CCOCC2)COC)nc2n(n1)CC(C(N1CCCCC1)=O)CC2 c1(OC(C)C(N2CCC(O)(CCNC(c3cnco3)=O)C2)=O)cccc(Cl)c1Cl C1(O)(C(=O)NCC(CCOC)NC(=O)C=C(C)c2ccsc2)CCC(C)(C)CC1 C1(NC(CC(=O)OCC)=O)CC2CCC1CN(C(c1ccc(F)c(OC)c1)=O)C2 C1(c2cncnc2)(C(=O)NC(CC)CN(C(=O)Cn2ncnn2)C)CCCC1 c1(C(N2CC3CCN(C(C4CC(CCC)C4)=O)C3C2)=O)ccc2c(n1)CCOC2 c1(NCC2N(C(C=C(CC)CC)=O)CC2)nc(C)ccc1C#N c1(C(=O)NCC2CN(C(CCCC)=O)C2)ccc(F)c(C(C)(C)C#N)c1 Cn1nnc(C(=O)NC2CCCN(C(=O)C=C3CCOCC3)C2)c1N N1(C(=O)CC2CC2(Cl)Cl)CCN(CCNC(C2(CO)CCC2)=O)CC1 c1(C(=O)NC2C(CC)CN(C(=O)CS(N)(=O)=O)CC2)c(N)cccc1[N+](=O)[O-] c1(OC)cccc(Br)c1CN1CCC(Oc2cnn(-c3ccccc3)c2)CC1 N1(C(C2(NC(N)=O)CC2)=O)CC2(COC(CNC(c3ccc[n+]([O-])c3)=O)C2)C1 Cn1nccc1C=CC(=O)NC(C1CCCCC1)C(=O)NC1CCC2CC12 Cc1nc(C2CCOC2)sc1C(=O)NC(C1CCN(C(=O)C(=O)NC2CC2)C1)C C(c1c(C)coc1C)=CC(=O)NC1(CCO)CN(C(CCC=CCCC)=O)C1 C1(NC(C2CC(N(C)C)C2)=O)CC(O)CN1C(=O)C(c1ccccc1)O N1(C(CC2C(C)C2(F)F)=O)c2ccccc2C(=O)N2CCCC12 N1(C(COCC)=O)CC(C2CCCN(C(c3coc4c(F)cc(F)cc34)=O)C2)C1 c1(C(=O)NCC2CCC(NC(c3c(C)oc(Cl)n3)=O)CC2)cc2ncccc2[nH]1 C(=O)(CC(CN)C(F)F)N1C(c2n(C)ncc2)CCCC1 C1(NC(c2cccs2)=O)CCN(C(=O)C(c2cccc(Cl)c2)(F)F)CCC1CO N1(C(Cc2nc(CC)sc2)=O)CC2CC1CN(C(=O)Cn1cc(CO)nn1)C2 C(=O)(CCC(CC)NC(=O)C(=Cc1ccccc1)C)NCCOCC=C CC(C)C(C)(O)C(=O)NC1CC(C(F)F)(NC(C2CC3CCC(C2)O3)=O)C1 c1(OC)ccc(CN2CCCC(CCNC(=O)CCc3cccn3C)C2)cc1 C(=O)(CS(C)(=O)=O)NCCC(Cc1ccccc1)NC(C1CC(OC)C1)=O CC1CNC(=O)C1NC(=O)C(C)CNC(C1CC1(C)C)=O C(=O)(CCCCCCBr)N1C(N)CC1.c1(COC(=O)NC(C)C)ccccc1 c1(C(=O)NC(CCNC(c2n(C(C)C)ccn2)=O)(C)C)cc(F)c(CO)c(F)c1 N1(C(CCCCCC#C)=O)CCC(N=c2nc(CC3CCCC3)[nH]s2)C(C)C1 C1(NC(C(C2(OC)CCCC2)(F)F)=O)CCCC(CNC(=O)C(F)=CC2CC2)C1 Cn1nnnc1SCC(N1CCC(NC(=O)CC2(n3ccnn3)CC2)C1)=O C=CCC(C)(C)CC(=O)NC1C=CC(CC(=O)Nc2cc(C)cc(C#N)c2)C1 C1(C(C(=O)NC(C2CCCC2)CNC(CN(C(=O)OC)C)=O)F)CCCCC1 C1(C(c2n(CCC(=O)OCC)nnn2)NCC2(CC(C)C)CC2)CCCOCC1 c1(CN2CCC(N(C(c3cccc(C(N(C)C)=O)c3)=O)C)C2)ccc(C#N)cc1 C1(CC(=O)NC(CNC(c2c(COC)scc2)=O)C(C)(C)C)CCCNC(=O)C1 C(=O)(CC(O)C(C)(C)C)NC1(COC)CCCN(C(C2CSCCS2)=O)C1 C1(C(=O)NCc2cc(CC)no2)(CNC(C2CCC2)=O)CCOCC1 c1(OCCC(=O)N(C2(C(=O)NCCCOC)C(C(C)C)C2)C)cccnc1 C1(C(N2CCC(C3CCCN3C(c3ccco3)=O)CC2)=O)CCC(=O)N1C1CC1 c1(C(=O)NCCC2(NC(Cc3nc(CC)sc3)=O)CC2)cc(C)cc(F)c1 c1(SC)cccc(C(=O)NCCCOCCNC(c2cc(Cl)ccn2)=O)c1 C=C(C)C(CC(=O)NC(C(=O)Nc1cnc(C)c(C)c1)C1CC1)OCC C1(N(C(C(CC)NC(C)=O)=O)C)CC2CCC(C1)N2C(C12CS(=O)(=O)C(C1)C2)=O C1(NC(CC(CC)C)=O)COC2CN(C(=O)COCC(F)F)CC12 CC1CCC(NC(c2cc(N)cc(O)n2)=O)CN1C(=O)CCC(N)=O c1(CC(=O)N(CCNC(C(C2CCCCC2)OC)=O)C)ccc2ccccc2c1 C1(C(C)NC(C(c2ccccc2)C)=O)CCCN1C(c1cn(C2CCC2)nn1)=O C(=O)(C1=CC2CC(C1)CC2O)NCC(CC)(C)NC(c1cccc(C)n1)=O N1(c2nccc(SC)n2)C2CCC1C(C)C(NC(=O)COC1CCCCC1)C2 Cc1ccc(C(=O)NC2CCCC2(C)CNC(C2COCCN2C)=O)c(N)c1F c1(C(=O)Nc2nc(-c3cc(Br)cs3)cs2)cc(O)c2occc2c1 Oc1cc2c(nn1)CN(Cc1c[nH]nc1-c1cc(F)cc(F)c1)CC2 c1(OC)ccc(O)cc1CNC1CCCC(C(=O)NCc2cccc(O)c2)C1 C1(C(=O)NC(CCOCC)C)COCC1NC(C1(Cl)CC1(F)F)=O C1(CC(N2CC(CCNC(C3COC(=O)N3)=O)(OC)C2)=O)SC2=NCCN2C1=O CCC(C(=O)NCCOC1CN(C(c2cc(C3(C)CC3)n[nH]2)=O)C1)C(C)(C)CC C1(C(N2CC(C(N)=O)OCC2)=O)CCCN(C(c2cccs2)=O)C1 N#Cc1ccc(C=CC(=O)NC2CC2NC(c2ccc(F)c3[nH]ccc23)=O)cc1 N1(C(C2CCC(=O)N2)=O)CC2CCCC2(C(=O)NCCOC2CCCCC2)C1 c1(C(=O)NCC2(C)N(C(=O)C=CC3CC3)CC(OC)C2)cccc2c1OCCC2 N1(C(C2(F)C(C)OCC2)=O)CCCCC(NC(c2ccncc2Cl)=O)C1 c1(C(N(CC(CNC(c2cc(COC)sc2)=O)C)C)=O)ccc(N)c(Cl)c1 C12(NC(c3c(C)c(Br)ccc3)=O)CCCC1N(C(=O)CCC(C)(F)F)CC2 C(C(O)C(C)(C)C)N(C(CN(C(c1n(CCC)ccc1)=O)CCC)=O)C C1(C(N2CC(C(=O)NCCC=CC=C)(SC)C2)=O)CCC(C)(C)OC1 CC1(C(N2CCCC(C(N)=O)C2)=O)CCN(Cc2ccc(C#N)cn2)CC1 CCC(CC)CCCn1nc(-c2ccncc2)nc1CCCOC1CCCCC1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(C2CC(C)CC(C)C2)=O)CC(C)C1 C(=O)(CCC(CC)OC)N1C(CCC(=O)NC(c2n(CC)ncn2)C)CCCC1 N1(C(c2occ(C)c2)=O)CC2CCCC2(C(=O)NOC2CCOC2)C1 C1(O)(C(N2CC(C(=O)NC(c3ccccc3)C#C)(CC)C2)=O)CCOCC1 c1(OC(C)C)ccccc1C(=O)NC1CC1CNC(C1CCC(O)CC1)=O CC1(C)CCc2nc(CNC(=O)NC3(c4nnnn4C)CCC(CO)C3)sc2C1 N1(C(C(C)CSC(F)(F)F)=O)CCCC(N(C)C(C2COC2)=O)C1 c1(OC)cc(C(=O)NCC2COCC2NC(C2C(C)(C)C2(F)F)=O)c(N)cc1F C(C)(C(C)(C)NC(=O)C=CCN(C)CCO)NC(C(C)O)=O C1(NC(=O)C(=C2CCCCC2)F)CC2CC1CN2C(=O)COCc1nc[nH]n1 Cc1ccc(C(=O)NCC2(C)CCN(C(c3ncoc3C(C)(C)C)=O)C2)c(C)n1 c1(CC)cccc(CC(=O)NCCCOCCOCCNC(=O)CC(C)O)c1 C1(C(=O)NCC(C)CNC(=O)C(c2ccc(O)cc2)=O)CCc2n[nH]cc2C1 C#Cc1ccc(C(N2CC3C(CNC(c4cscc4OC)=O)C3C2)=O)cn1 C=C(CNC(C1CCN(C(c2cc(C#N)[nH]c2C)=O)C1)=O)C1CCOCC1 c1(C(N2C(C)(C(=O)NC3(CC=C)CCOC3)C=CC2)=O)cc(C)nc(C)c1 N1(C(C(C)SC)=O)CC2=C(C1)CN(C(c1ccc(-c3ccc(C)o3)s1)=O)C2 N(C(=NCCN(C1CC1)CC)N(C)CC1CCN(C(=O)OC)C1)C(CC)C c1(Cn2cc(C3(NC(C4(CO)CCC4)=O)CC(F)(F)C3)nn2)ccc(CF)cc1 C1(CN(C(=O)CC2COCCO2)C)CCCCN1C(=O)Cc1cnn(C)c1 C1(C(=O)NCCCCCCNC(c2c(OC)nccc2)=O)OCC2CCCC1C2 CC(C)CC(CO)NC(=O)NC1CCCC(NC(=O)C(C)(C)c2ccccc2)C1 C(CN=c1c(Br)c[nH]cc1[N+](=O)[O-])C1C(C)CCCN1C(c1ccco1)=O c1(C(N2CC=CC(NC(C(C)OCC#C)=O)C2)=O)cc(F)cc2cccnc12 C(=O)(CC(=O)NC1CC(NC(=O)CC(C)n2ccnc2)C1)OCC C1(NC(N2CCC(CN(C)CC)CC2)=O)COc2ccccc2O1 C1(CC)CCN(C(=O)CN2CCC(OC)C2)C(C(N2CCCN(CC)CC2)=O)C1 c1(C(=O)NCCC2CC(C(=O)NCC(C)(C)C(N)=O)C2)ccc2cncn2c1 c1(C(=O)NC2CCCC2NC(C2CCC=CCC2)=O)cnc(O)cc1C(F)(F)F c1(CC(N2CC3CCC3(CNc3cn(CCO)nn3)C2)=O)ccc2nc[nH]c2c1 N1(C(C2CCOCC2)=O)CC2(C1)CC2(F)F N1(C(c2c(C)ncnc2)=O)CC(NCc2ccc(Br)cc2C(=O)O)CC(C)C1 C1(N(C(C=CCCC(C)C)=O)C)CCC(NC(C2CCOC2=O)=O)CC1 C1(C(=O)OCc2c(C)cc(C)s2)CC2CCCCCCC12 C(C(COC)C(=O)N(C(C)CC(=O)NC1(C)CCCC1O)C)OC N1(C(c2cc(CC)[nH]n2)=O)CCC2CC1CN(C(=O)COC(C)CC)C2 C12(C(=O)NC3CC(CNC(C(CC)=CC)=O)C(O)C3)CCC(C)(C1)OC2 C(c1cn(C)nn1)=CC(=O)NCC(CNC(=O)C(CC1CCC1)OC)OC CON1CC(C(=O)NCC2(O)CCN(C(=O)C(c3cccc(C)c3)=O)C2)CC1=O N1(C(CCc2ccc(C)nc2)=O)CC2CCCC2(CNC(=O)C2=CCCC2)C1 CC1CC(=O)NC(C(=O)NCC2CC3C2CCN3C(=O)CCC(C)(C)C)C1 N1(C(C(CCC)N(C)C)=O)C2CCC1C(CNC(c1ccc(C)cc1SC)=O)C2 c1(CC(=O)N(CC(C)C(=O)NC2CCC(=O)NC2)C)ccc(O)cc1 CCCCCCC(=O)NC1(C)CCN(C(=O)Cc2cc(Br)cs2)C1 C(C)(C)(CCCNC(=O)CC1CC(C)N(C(=O)CSC(F)F)C1)OC C1(CN(C(c2ccon2)=O)CC)CCCN1C(=O)CC(c1ccccc1)OC C1(CCNC(c2cnc(CC(C)(C)C)s2)=O)CCN(C(c2cc(F)cs2)=O)CC1 C1(NC(c2cnc(Br)s2)=O)CN(C(c2cccc(F)c2I)=O)CC(F)(F)C1 c1(C(=O)NC2C(OC)CN(C(=O)CCc3nc(C)c(C)[nH]3)C2)cc(O)nc(C)n1 N1(C(CC2CN(C(C3CC(C(C)C)C3)=O)CC23CC3)=O)CC(CO)C2(CCC2)C1 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC(CC=C)CNC(C12CC(CO)(C1)C2)=O c1(CN2CCN(C(c3nncc(OC)c3)=O)CC2)ccc(Br)c(C#N)c1 Cc1ccc(=NCCC(=O)N2CC(CC(C)NC(=O)C(CO)C(C)(C)C)C2)[nH]c1 C1(NC(c2ccncc2N2CCCC2)=O)CCCCCN(C(=O)C2=CCOC2)C1 c1(NC(=O)NC(CCN(C2CCCCCCC2)C)C(N)=O)ccn2c1CCCC2 C(=O)(C1CCc2cccc(F)c21)N1CCN(C(CC(CC)(F)F)=O)C(C(F)F)C1 C1(NC(CC2(COC)CC2)=O)CCCCCN(C(c2[nH]cc3c2CCC3)=O)C1 N#CC1(C(=O)NCCCCNC(c2ccc(-c3cn[nH]c3)cn2)=O)CC2CC2C1 c1(OC)cccc2c(C(=O)NCC3(OC)CN(C(=O)CCOC(C)=O)C3)n[nH]c12 O=S(=O)(c1c(Cl)cc(Br)cc1Cl)N1CCCC1c1nc2ccccc2[nH]1 C(=O)(C1CCc2cccnc21)N1CCCC(C)(NC(C2(COC)CC=CC2)=O)C1 c1(CCC(N2CC3C(NC(c4ccc(Cl)cn4)=O)(C3)C2)=O)nc2ccccc2[nH]1 c1(-c2nc(-c3c(C)cc(C(=O)OC)s3)on2)c(F)ccc(C)c1F c1(OC)cc(CC(N2CCC(C(C)NC(=O)Cc3cn[nH]c3)C2)=O)ccc1Cl C(c1cccc(Cl)c1Cl)=CC(=O)NCc1nc(-c2cccc(OC)c2)oc1 C(C(C)(C(=O)NCC1CCCC(CO)C1)NC(C1CCC(F)(F)C1)=O)SC C1(CNC(C(C)C2CCCC2)=O)CN(C(c2cc(N)cc(O)c2)=O)CCCO1 Cn1nc(-c2cn(CCCCC(=O)NCCCOCC3CC3)nn2)cc1N c1(C(N2CC(C)CC(NC(C(C)OCC=C)=O)C2)=O)ccc2sc(C)nc2c1 CS(=O)(=O)c1ccc(C(N2CCCC(CCNC(C3CC(=O)N3)=O)C2)=O)o1 n1(CC(N2C(CN(C(CC3C(C)C3(F)F)=O)C3CC3)CCC2)=O)cccnc1=O c1(C(N(CC(CNC(Cn2c(C)ccn2)=O)O)C)=O)ccc(C2CC2)cc1 N1(C(c2c(C)con2)=O)CC2CC1CN(C(=O)Cc1c(F)cc(F)cc1F)C2 C(=O)(C(C)C(=O)NC1CC(NC(=O)CSC)C1)OC c1(C(=O)NC2C(C)CC2)n[nH]c2c1CN(C(C1(C#N)CCCCC1)=O)C2 C(=O)(C(C)CCC(C)(C)C)N1C(C(=O)Nc2c(OC)ccc(Cl)c2)CC(O)C1 CCC(C)(CCNC(=O)CCc1cncn1C)NC(c1cc(C)n(C(C)C)n1)=O S(=O)(=O)(c1ccc(F)cc1F)N1C(C)(C(=O)NC2CCCOC2)CC1 c1(COC)ccc(C(N2CC(CNC(C3CCC(N(C)C)C3)=O)(OC)C2)=O)s1 c1(C(N2CC(SC)C(NC(=O)C(C)(C)C(C)C)C2)=O)ccc(C#N)cc1C c1(SCC(=O)NC2CC2CNC(c2cncc(O)c2Cl)=O)nc2ccccc2s1 c1(CC(C(=O)NC2CC(CC(=O)OCC)C2)O)cccc(C(F)(F)F)c1 C1(C)(C(=O)OC)CCN(C(C2(F)CN(C(C3CCCCS3)=O)C2)=O)C1 C1(C(=O)NC(CNC(C2CCC(C)S2)=O)(C)C)COCCOC1 Nc1c(C(=O)NCC2(O)CCCN(C(C3CCCC(=O)N3)=O)C2)ccc(Cl)c1O S(=O)(=O)(c1ccc2oc(=O)c3ccc(Br)cc3c2c1)N(CC(C)O)C(C)(C)C c1(N(CC(N2CCCCC2c2ccccc2F)=O)C)ccnc(C#N)n1.C(C#N)N c1(CC(=O)NC2CC(N(C(C(C3CC3)OC)=O)C)C2)ncc(Cl)n1C c1(C(=O)NC(CC)CN(C(=O)C(O)CC(F)(F)F)C)ccc(O)c2ncccc12 C(C(CC1CCCC1)C(=O)NC1CC(C)OC1=O)NC(c1nc(CC)sc1)=O N1(C(C(C)=C(CC)C)=O)CCCC1CN(C(c1n[nH]cc1CC)=O)CC c1(C(=O)Nc2cc(C)c(NC(C3CC3C3CC3)=O)cc2)nncc2ccccc12 C1(NC(CC2(C=C)CCC2)=O)CC(NC(=O)CCNC(C)=O)C12CCC2 C(=O)(CCC(CF)CF)NC1CN(C(Cn2c(C)ncc2)=O)CC(C)C1 c1(C(=O)NCc2onc(CC)n2)ccc(CNC(c2cc(OC)n[nH]2)=O)nc1 c1(C(=O)NC(C)CNC(=O)C(C)(C)Cc2cnn[nH]2)ccc(O)nc1Cl CCC(C#N)C(=O)NC(C1CCN(C(C23CCC2CC3)=O)CC1)C N1(C(CC(C=C)(C)C)=O)CCC(NC(=O)C=CC=CC)C(CO)CC1 C(=O)(C(F)(F)CC(C)C)N(C(C)CNC(=O)C(C)Sc1ccc(F)cc1)CC C1(C(=O)NCC(C)(C)CNC(C2(C#N)CCOCC2)=O)CCc2nccn2CC1 c1(C(N2CC(F)(CNC(c3c(CC)cco3)=O)C2)=O)cc2c(C)c(F)ccc2[nH]1 Cc1nn2cccnc2c1C(=O)Nc1cccc(CNC(=O)CCC(C)(C)O)c1 C(=O)(C(F)CC(C)(C)NC(=O)C(CO)C(F)(F)F)N(C)CC1(O)CCCC1 N1(C(C(CC#C)C2CC2)=O)CCC(NC(c2ncsc2C)=O)CC(C)(C)C1 CCC(C)(O)C(=O)NC1CCOC1C(N1CC(C#N)C1)=O Cc1ccc(N2CC(NC(=O)CC3COCCN3C(c3cscn3)=O)CC2=O)cc1 C1(NC(CSSC)=O)CN(C(=O)COCC2CCCCO2)CC1C(F)(F)F N1(C(CC(CCC)O)=O)CCC(C2CC2)(NC(c2coc(C3CCC3)n2)=O)C1 S(=O)(=O)(c1cccc(F)c1)NC1C(O)CCN(Cc2cccc(OC)c2O)C1 N1(C(=O)Cn2nnc(C3CC3)n2)CCOC2(CCN(C(c3nncs3)=O)CC2)C1 C(=O)(CCC(=O)NN(C)C)N1C(C(=O)NCC2CC(=C)C2)C=CCC1 C#CC1CCCCN1C(=O)C(c1ccoc1)NC(=O)CN(C)C C1(NC(=O)N(C2CC(c3ccon3)C2)CCN2CCCC2)CCOC1 CCC(C)CCCC(=O)N1CCN(C(=O)C(C)Cc2ccccc2)C(C)C1 N#CC1CN(C(c2cc(F)ccc2Cl)C(=O)NCCCOCC2CC2)C2(CC2)C1 CCCC(C(=O)NC1CCC(NC(C2(CC(C)C)CC2)=O)CC1)C(C)C N1(C(c2cc(OC)n[nH]2)=O)CC2C3CCC(C2C1)N(C(C1CCCC(O)C1)=O)C3 C(C(F)(C(=O)N1CCC(C)C1CO)C(C)C)NC(c1c(OC)nn(C)c1)=O N1(C(C2(CC=C)CC2)=O)CC(n2cc(-c3cncc(Cl)c3)nn2)CC1C c1(NC)ccc(C(=O)NCC2(NC(c3cccs3)=O)CCOC2)nc1 C1(NC(c2scc(C)c2)=O)CC2(C1)CC(NC(c1cc(C)c(C(F)F)cn1)=O)C2 C1(NC(C2CCCN(C(CCC)=O)C2)=O)CC(C)CN(C(=O)C2=CCCCC2)C1 CC1CC(NC(=O)CC2C=CCC2)CN(C(=O)COc2ccc(O)cc2)C1 C(=O)(C1=C(Cl)CCC1)NCC1(C)CCN(C(c2ccc(CC(C)C)nc2)=O)C1 C1(CN(CC(=O)N(C)CC2(C3CC3)CC2)C)CCCN1C(C1CCCC1)=O C1(C(=O)NC)CCN(C(=O)CCN(CCCO)C(c2cccc(CO)c2)=O)C1C C1(OC(CCC)C(=O)N2CCC(NC(=O)C3=C(C)OCC3)C2)CC(=O)NC(=O)C1 c1(C(=O)NC(CC(=O)NC(CC=C)(C)C)C2CC2)ccc2c[nH]nc2c1 N1(C(CC(C)(C)O)=O)CC(O)CCC1C(=O)NCC1CC2(CC2)C(=O)O1 C1(C(=O)NC2(CSC)CCC2)CN(C(=O)CNc2ccc(Cl)cc2)CCO1 C1(CNC(C2CCN(C(C3(C)CCC4CC4C3)=O)C2)=O)CCn2ncnc2C1 N1(CCC#C)CCN(C(C2C(NC(=O)CCC3CCCO3)C2(C)C)=O)CC1 C1(C(C)NC(=O)CC2CC=CCC2)CCN(C(=O)C(C)C2CCCO2)CC1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CN(C(Cc2cn(C(C)C)nc2)=O)C1 C1(COC)C=CCCN1C(=O)CC1C(NC(c2cc(OC)cs2)=O)CC1O C(=O)(C(C)CC(C)CC)NC1(CCNC(c2cnc(CCCC)[nH]2)=O)CCCC1 c1(C(CNC(=O)COCC2CC2)CNC(c2coc(Cl)c2)=O)ccccc1 c1(C(=O)NCCNC(c2csc(Cl)c2)=O)cccc(C2COC2)c1 c1(CC)ccc(-c2nc(C(C)SC)nn2CC2CCCO2)cn1 CCC(C#N)(CC)C(=O)NCC(C)C(N1CCC(SC)CC1)=O Cc1oc(C)c(C(=O)NCC2C=CCN2C(=O)CN2CCC2C)c1Br C1(CNC(C2CCCCC23CC3)=O)CC2(C1)CN(C(=O)CCCN1CCCC1)C2 Cc1nc(-c2cc(CNC3CC(C(N)=O)(N(C)C)C3)cs2)cs1 Cc1nc2cccc(C(=O)NC3(CNC(C4CCS(=O)(=O)C4)=O)CC3)n2n1 c1(C(N2C(CO)CC(NC(c3ccc(CC)o3)=O)C2)=O)cnc2n1C(C)CCC2 C#Cc1cnc(C(N2CCN(C(c3cc(C)co3)=O)C(CC)C2)=O)c(C)c1 n1(CC(=O)NCC(C)(C)NC(C2C(C(=O)OCC)CCO2)=O)nc(C)c(Cl)c1C C(=O)(C1=COCCC1)NC(C)CCCCNC(=O)C(O)c1ccsc1 C(=O)(CC(O)CC(C)(C)C)NC1(C(=O)NCCOCCC)CCC1 C(=O)(C1=CCS(=O)(=O)C1)N1CCC(CN(C(=O)Cc2ccncc2Cl)C)C1 CC1CC(CNC(=O)C(c2ccccn2)O)CN(C(=O)CN2CC3CC3C2)C1 C(CCC(C(=O)N(CC1CC1)OC)NC(=O)CCC1CC1CC)OC Cc1ccc([N+](=O)[O-])c(C(N2CC(N(C)C(c3ccc(N)c(Cl)n3)=O)C2)=O)c1 C1(CN(C(CCCNC(C)=O)=O)C)CC(F)CN1C(C1COC(=O)O1)=O N1(C(C(C)C)=O)CC2(CCOCC2)CC1CNC(c1ccn2ncccc12)=O CC1C(NC(=O)CCc2ccc(Cl)s2)CCN1C(=O)CC1(CO)CC1 N#Cc1ccc(C(=O)NC2CCCCC2NC(=O)CSCCC(F)(F)F)cc1F N1(C(CCC(C)OCC)=O)C2CC1CN(C(C1CCC(C3CC3)O1)=O)C2 c1(C(N2CCC(O)(CCNC(C(C)(C)C)=O)CC2)=O)coc2c(F)cc(Cl)cc12 C1(N(C)C(c2cccnc2O)=O)CN(C(=O)C(F)C2CCOC2)CC12CC2 c1(C(=O)OC(C)(C)C)cc(=O)c2ccccc2[nH]1.C12C=CC(CC1)CC(=O)N2 c1(CN2CCCC(N)(CO)C2)ncn2ccccc12 CC(C)C(C(=O)NC(C)(C)C(C)NC(=O)CN(C1CCC1)C)Sc1ccccc1 C1(CNC(CNC(=O)OC)=O)CC2COCC2N1C(C1CC2(C1)CC2F)=O Cc1noc(CCC(N2CC(F)(CNC(=O)Cc3nnc(O)s3)C2)=O)n1 Cc1c(CCNC(CCCC#N)c2nnnn2CC2CCOC2)cnn1C C12(CNC(CCCN(CCC)CCC)=O)CN(C(C3C(C)C3(F)F)=O)CC1CCO2 N1(C(c2ncccc2F)=O)CC2C(C1)C2(F)F Cc1cccc(C(=O)NC2CC=C(C(=O)N(C34CC(C3)C4)C)C2)c1N C1(N(C)C(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC2(C(F)F)CC2)CC1 c1(NC(C2CN(S(CCC)(=O)=O)CC2O)=O)cnc2c(F)c(F)ccc2c1 C(=O)(C(C)C(F)(F)F)NC(COCC)C(=O)NCCc1ccnn1C C(CCF)(C(=O)NC1(C)CCOCC1)NC(c1cc(OCC)n[nH]1)=O c1(OC)cc(OC)c(C(=O)NCC(O)CNC(=O)C=CS(C)=O)cc1N Cc1cc2c[nH]nc2c(C(N2CC(NC(C3CCCOCC3)=O)C2)=O)c1N c1(C(=O)NC2C(CNC(c3ccc(C(N)=O)cc3)=O)CC2)cncc2ccsc12 C1(C)(C(N2CCC(NC(C(COC)C)=O)C(O)C2)=O)CCC(C)(C)CC1 N1(C(c2n(CC)cc(Cl)c2)=O)CC(CNC(c2cnc(C)s2)=O)CC(C)C1 c1(CN2CC(NC(c3ccc(Br)cn3)=O)C(O)C2)cc(Cl)ncc1Br C(=O)(N=c1cc(C(F)(F)F)[nH][nH]1)C1N(C(C(C)(C)OC)=O)C2C(C1)C2 C1(NC(CSC)=O)CC2CN(C(=O)Cc3cccc(OC(C)C)c3)CC2C1 C1(C(N2C(CN(C(=O)C=CCO)CC)CCC2)=O)C(F)(F)C12CCC2 n1(CC)ccc2c(NC(=O)CNC(=O)CCn3ccnc3C(C)C)cccc12 Cc1cc(C(=O)NCCC2(NC(C3CC34CCC4)=O)CCC2)ns1 C1(C(=O)NC2CCC(NC(CCCc3ncc(C)o3)=O)CC2)CCC(C)(C)CC1 N1(C(c2c(C)c(Cl)ccc2)=O)CCC2(CC1)CN(C(C1CCCO1)=O)CC2CO C1(OC)(CNC(c2cc(C)ncc2C)=O)CCN(C(c2c(C)csc2Cl)=O)CC1 C1(CC=C)CC2CC(O1)CC(=O)O2.C12(C(=O)NC)CCCC1C2(F)F C(=O)(C(C)(C)C(=O)NCCC1COCCN1C(C12CCC(C)(C1)OC2)=O)N(C)C N1(C(C2OCCN(CC)C2)=O)CCOCC(C(=O)N(C2CC(F)(F)C2)C)C1 C(C)(C)(CC(=O)N(C1CCOCC1)CC)N(C(C1C(CC)CCO1)=O)C O=CN1CCCC1C(=O)NC1CC2(C1)CC2C(=O)NCC1(O)CSC1 c1(OC)cc(C(F)(F)F)ccc1CC(C(=O)O)NC(=O)C(c1cccc(C)c1)C Cc1ccc(C(=O)NCC(C)(C)NC(=O)CC2CCCCC2C)c2c1NCCC2 Cc1cc(Cl)c(C(N2CCCC(CCNC(=O)C=Cc3cn(C)cn3)C2)=O)cn1 CCC(CC)(CO)C(=O)N1CCN(C(c2cc(C(N)=O)c[nH]2)=O)C2(CC2)C1 N12CCn3nc(cc3C1)C(=O)NCC2=O.N1(C(C(=O)O)=O)CCC(CO)C(O)C1 CC(C)CS(=O)(=O)CCC(=O)NCCOCCNC(c1ccnc2c1CCO2)=O N1(C(C2C(C3C(C)C3)C2)=O)CC2CC(NC(c3cc(C(C)(C)C)no3)=O)CC1C2 c1(C(=O)NC23CCN(C(c4n(C)ncc4)=O)C2CCC3)cnc2[nH]c(O)nc2c1 C(CC(=O)N1CC(NC(c2ccn(C)c2)=O)C(C)(C)C1)(C(N)=O)NC(C)=O c1(CC)csc(CC(=O)NC2CCN(C(=O)Cc3ccccc3)C2)n1 C1(C(N(C)CC2CCN(C(c3c(C)cn(C)c3)=O)CC2)=O)COCC(C)(C)O1 N1(C(Cc2cc(C)no2)=O)CCCC1(C)C(=O)NCC1CCCC1N(C)C c1(C(N(CC(CC)NC(=O)Cc2nocc2C)C)=O)conc1C C=CCCC(C)(C)C(=O)N1CCC(C(F)C(=O)NCc2ccnc(CO)c2)C1 N1(C(C(C)(C(C)C)OC)=O)CCC2(CCCCC2NC(=O)Cn2cccn2)CC1 Cc1cccn2cc(CC(N3CCN(C(C4CCCN4C(C)C)=O)CC3)=O)cc12 n1(CC(=O)NC2(COC)CN(C(c3cc(CC)[nH]n3)=O)C2)cc([N+](=O)[O-])cn1 C1(CSCC(=O)N(CC(C)NC(c2ccc(C(C)(C)C)[nH]2)=O)C)CCCCO1 CS(=O)(=O)c1cncc(-c2cnccc2C(=O)NCC=CC2CC2)c1 C(C1CCCO1)=CC(=O)NCCCOCCNC(C1CC1C(F)F)=O C1(NC(c2cc3n(n2)CCO3)=O)CC1C1CCN(C(C2(O)CCC2)=O)CC1 c1(C(=O)OC)ccccc1C(=O)NC1CCN(C(=O)CSC(C)C)CC1 C(=O)(C(C)(C)C(C)(C)O)N1C(CNC(c2c(CC)oc(C)c2)=O)CCCC1 c1(C(=O)NCC(C)NC(c2cc(CF)on2)=O)nccn2ccnc12 c1(OC)nc(C)c(C(=O)NC2CCC(C(=O)Nc3nc(C)c(C)s3)C2)s1 Cc1cccc2[nH]cc(CC(=O)NC3CC(F)CN(C(C4CC4C#N)=O)C3)c12 N1(C(C2(C=C)CC2)=O)CC(NC(=O)Cc2ncn(C)c2C)C(C)C1 c1(C(=O)NCC(CN(C)C(c2nnn(C(C)(C)C)n2)=O)O)ccc2nnnn2c1 CCC(CC(=O)N(C1CN(C(C2CNC(=O)CC2C(F)(F)F)=O)C1)C)C(C)C Cc1cc(F)cc(NC(C2(F)CCN(Cc3cnn(C4CC4)c3)C2)=O)c1Br C(=O)(C(CCC(N)=O)N(C)C)NCCOCCNC(c1cnn(CCC)c1Cl)=O C=C(Cl)CC(C(=O)N(CCCCO)C)NC(=O)CCN(C1CCC1)C N1(C(CC(=O)NCC)=O)CCC=CC1C(=O)N(CCC(C)C)CCO c1(OC)ccc(CO)cc1C(=O)N(C)CC1(NC(C2CC3C=CC2CC3)=O)CC1 C1(NC(c2cc(O)n(C)n2)C)CCCCC1NC(c1ccccn1)=O c1(CCC(N2CC(C)N(C(=O)C(CO)NC(N)=O)CC2)=O)nc2ccccc2o1 C=C1CON(C(=O)C(CCF)NC(=O)C#CC2(C)CCCO2)C1 N1(C(C=CSC)=O)CCN(C(C23CCC(C)(C2)OC3)=O)CC1C1CCC1 C1(C)(CNC(C2CCC(C(N(CC(=O)OC)CCOC)=O)O2)=O)CCCCO1 c1(C2CCC(C(N(C3CCCCN3)CC)=O)C2)cccc(F)c1 c1(C(=O)NC2CN(C(C3CC4(CSC4)C3)=O)CC2C(F)F)cc(=O)cc(Cl)[nH]1 c1(C(N2C(C3(NC(C(CC)(C)COC)=O)CC3)CCC2)=O)ccc2c(c1)CCN2 CN1CC(C(=O)NCC2CCN(C(=O)COC3COC3)C2(C)C)CCC1=O S(=O)(=O)(c1ccc(NCC(CC2CC2)CO)c(Br)c1)N1CCOC(C)CC1C C(CCCCCC(=O)NCc1cnns1)NC(C1OCCC(C)(C)C1)=O N1(C(Cn2nc(C)oc2=O)=O)C2CCCC1CC(NC(=O)C1=NNC(=O)CC1)C2 CC1CCC(C)N1C(c1cc(NC(c2cccnc2I)=O)cn1C)=O Cc1ncc(C(=O)NC(C(=O)NC(c2nnc(C)o2)C)C2CCCC2)c(C)n1 N1(C(C2(CNC(C3CC34CCOC4)=O)CC(=C)C2)=O)CCC2(C1)CN(C)C2 CC1CCC(C)(C)N1C(=O)CCC1CCN(C(=O)Cc2ccon2)C1 Cc1sc2ccccc2c1CNC(=O)Nc1ccc(=O)n2c1CCC2 Cc1cc(C)c(C(N2CC(NC(=O)C(=O)NCC3CC3)CC(O)C2)=O)c(N)c1 c1(C(=O)NC(CC)(CNC(=O)CC2(O)CCCOC2)CC)ccc(S(N)(=O)=O)o1 N1(C(C(CC#C)C)=O)CCCC(NC(c2cncc(Cl)c2)=O)CC1 c1(C(c2nnnn2C)NC(c2ccc(C)o2)C)cc(CO)ccc1[N+](=O)[O-] C12(NC(CNC(C)=O)=O)CC(CNC(=O)CCS(=O)(=O)NC3CC3)(C1)OC2(C)C N1(C(c2c(Cl)cn(CCC)n2)=O)CC2CC(NC(=O)Cc3csc(C)n3)C1C2 c1(OC)c(Br)ccc(F)c1C(C(=O)NC1CCCC1)N(C)Cc1ccc(Cl)cc1 Cc1cc(C(=O)NCc2nc(CNC(=O)CCC3CC(F)(F)C3)cs2)no1 N1(C(C(CC)CC(C)C)=O)CC2(C1)CN(C(=O)C=Cc1cccnc1C)CCO2 Cc1cccc(CC(=O)NCCN(C(=O)C(c2nc(C)cs2)C)CC(C)O)c1 Cc1c(CC(=O)NC(CNC(=O)CC(C)c2ccncc2)C(C)(C)C)ncn1C C1(COC)CC(CNC(c2csc(Cl)n2)=O)N(C(=O)C2=CCOC2)C1 c1(OC)cc(C(=O)NCC2CN(C(c3snnc3C)=O)CCO2)cc(Cl)c1 Cc1ccc(NC(C2CC(O)CN2C(=O)C(Cl)(Cl)Cl)=O)cc1N1CCOCC1 C(C(C)CC(F)(F)F)NC(CC1N(C(c2c(COC)cco2)=O)CCOC1)=O CCC(C)(C#N)C(=O)N(C)CC1(O)CN(C(c2ccc(CC(C)C)s2)=O)C1 N1(C(CCOCCOC)=O)CC2CC(NC(=O)CSC3CCCCO3)C2C1 C12(NC(C3CC=CCO3)=O)CCCN(C(c3coc(Br)c3)=O)CC1C2 C1(C(N2CC(N(CC(C)C)C)C2)=O)CC2(CC2)CN1C(=O)CCCNC(N)=O c1(CN(C(c2cnc(C(C)OCC)s2)=O)C)ccc(CO)cc1.C(=O)(CC(C)(C)O)N c1(C2C(F)(C(=O)NC3C(NC(c4cnco4)=O)C3)C2)ccccc1 C(CC(C)C)(C(=O)N1CC(N(C(=O)CC=Cc2ccc(F)cc2)C)C1)NC(C)=O C1(NC(C2(OC(C)C)CCC2)=O)CC(C)CN(C(=O)C(C)(C)O)C1 C1(NC(c2cnc(C(F)(F)F)nc2)c2onc(C(F)(F)F)n2)CC2CCCC2O1 C(=O)(C(C(=O)N1CCOC(CNC(=O)Cc2cccc(C)c2)C1)OC)OC N1(C(=O)NC(CC)CC)CCCC2(COc3ccccc32)C1 C1(CCCC)CCCC1(c1nnnn1CC(=O)OC)NCCOCC(C)(C)CCC Cc1cc(O)ncc1C(=O)NC1CN(C(C2CC2C)=O)CCC1F C1(N=[N+]=[N-])(C(N2CCC(SCC(=O)NCC(C)C)CC2)=O)CCNCC1 C#CCC(CC(F)F)C(=O)N1CCC(C2CC2)C1C(N1CC2CC(CO)C(C2)C1)=O C(CCCCC(=O)NC(CCOCCO)C(=O)NC1CC(CCO)C1)=CCCC c1(C(N2CCC(F)(CNC(CC(C)F)=O)C2)=O)cc(Cl)cc(Cl)c1 C1(C(=O)NC2CCN(C)CC2C)(CC)CCCN(C(c2c[nH]nc2Cl)=O)C1 c1(C(=O)NCC2C(C)CN(C(=O)CN3CCC(C)(O)C3)C2)ccc(C#N)c(O)c1 N1(C(c2cc(C)cc(Cl)c2)=O)CC2OCC(NC(=O)CS(=O)(=O)CC)C2C1 C(=O)(C#CC1(C)CCCO1)NC(C1CN(C(=O)C(C(C)(C)C)n2ccnn2)C1)C N1(C(C2N(C(CCc3onc(C)n3)=O)CCN(C)C2)=O)CC(C)(C2CCC2)C1 N1(CC(N2c3ccc(C(=O)OC)cc3CCC2)=O)C(=O)NC2(CCCCC2C)C1=O C(COC)(C(=O)NOC(C)(C)C(=O)OC)NC(CCCCOC)=O C(CC(C)C)(C(N)=O)N(C(C1CC(N(C(CCc2cc(C)on2)=O)C)C1)=O)C Cc1c(C(=O)NCCN(C(=O)CC(C)CF)C)oc2c1ccc1ccccc21 c1(C(=O)NCCC2CN(C(c3c(C)nc(O)[nH]3)=O)C2)ccc([N+](=O)[O-])s1 N1(C(C2CC(=C)C2)=O)CCCC1C(C)NC(=O)C(C1CCOCC1)F c1(C(=O)NCCN(C(C(CSC)C)=O)CCOCCO)nc(C(F)(F)F)oc1C c1(C(N2CCC(NC(Cc3c(C)nc[nH]3)=O)C2)=O)nc(Br)ccc1F N1(CC)CCOC(C(=O)NCC2CCCN(C(C3CC(n4cncn4)C3)=O)C2)C1 Cc1ncc([N+](=O)[O-])cc1C(=O)N(C(C)CNC(=O)CC1CCOCC1)C C(=O)(CCC=C(C)C)N1CC(CCCCNC(C=CC=CC)=O)C1 N1(c2ccc(C)cc2)CCN(CC(N2CCC(C(N)=O)CC2)=O)CC1C n1(CC)ncc(Cl)c1C(=O)NC1CCC(C)(CNC(=O)CCC2OCCO2)C1 c1(C(=O)NC2CC(CCNC(C(C3CCCCCC3)C)=O)C2)ccc(N)cc1F Cc1nn2cc(C(=O)NCCCCCN(C)C(c3ccc(C(N)=O)[nH]3)=O)nc2s1 CN1CC(C(N2CC(CNC(c3ccoc3C(F)(F)F)=O)C2)=O)OCCC1=O C1(NC(c2n(C(C)C)ccc2)=O)CCCN(C(C2CC23CC(C)(C)C3)=O)CC1 c1(C(=O)NC2(C)CCN(C(c3ccc(C(C)=O)o3)=O)C2)cncc2cccnc12 C1(N(C(C(CCOC)NC(=O)CC(=O)NC2CC2)=O)C)CC(C)(C)CCO1 Cc1nc(O)nc(C)c1CC(=O)NC1CC(NC(c2cc(CC(C)C)on2)=O)C1 c1(CC(N2CC(OC)(CNC(=O)C=CC3CC3)C2)=O)ccc(C)cc1Cl N1(C(CC2(C=C)CN(C(c3nscc3C)=O)C2)=O)CC2NC(=O)OC2C1 CN1CCC(C)(CNC(c2conc2CNC(=O)CC2CCCC2)=O)CC1 N12CCCOC(C1)CCC(C)(C)C2.c1(N(C)CCO)cnn(C)c1 C1(C(C)C)CN(C(=O)C(CCC2CC2)NC(C2CC(F)C(=O)N2)=O)CCO1 C(=O)(CC(C)(C(F)F)N(C)C)NCC1CCN(C(c2cnc(OC)c(C)n2)=O)C1 C1(F)(CNC(C(COC)OC)=O)CCN(C(=O)CCCCc2cnn[nH]2)CC1 c1(C(N(CCOC)CCNC(c2ncc(Cl)nc2Cl)=O)=O)cc(F)cc(N)c1N CC1=C(C)CC(C)(C(=O)NCCCN(C)C(c2cc(Br)sn2)=O)CC1 c1(CNC(C(N2C(c3onc(C)n3)CSCC2)=O)=O)cc(Br)cc(F)c1F CC(O)C(C)(C)NC(=O)C(C1CCN(C(=O)C(F)C2CCCC2)C1)F C(=O)(C(C)(C)OC(C)=O)OCC.C12C(C1(F)F)CN(CC(=C)CC)C(=O)C2 N1(C(CC2CC(CC)C2(C)C)=O)CC2CCC(C1)N2C(=O)C(C)(C)N1CCCC1 C1(NC(c2ccc3oncc3c2)=O)CC2CCCCCC2C1 CC(C)CC(Cn1cc(C(C)CC2CCCC2)nn1)NC(c1conc1CO)=O C1(CNC(CC(CC)C2CCC2)=O)CC12CCN(C(C1CN(C(N)=O)C1)=O)CC2 C1(C(=O)NCCCC(=O)OCC)CC12CCN(C(c1cn(C3CC3)nn1)=O)CC2 C12(NC(c3cnn4c3CCC4)=O)CCCC1CN(C(c1cc(Cl)ns1)=O)C2 c1(C(=O)NCCC2CN(C(C3CCC(O)C3)=O)C2)cc(Cl)c2c(c1)OCCO2 C1(NC(C(C)(F)C(C)(C)F)c2n(CCCCCC)nnn2)CC2(CCCCC2)C1 c1(NC(C2(F)CN(C(C)=O)C2)=O)ccc(C)cn1.C12OCCC1C(=O)NC2 c1(C(=O)NCC(c2ccccc2)CNC(CCSC)=O)cccc2c1CCO2 N1(C(CCNC(=O)OC)=O)CCC2CCN(C(c3ccc(C(N)=O)o3)=O)C2C1 N1(C(c2cnn(CC)c2C)=O)CCOCC12CCCCC2 C(CCNC(c1cscc1C(F)(F)F)=O)(C(C)C)NC(CC=CC=C)=O Cc1cc(C(=O)NC(CNC(C2CCCC2(C)C)=O)CO)nn1CCO N1(C(CC=CC=C)=O)CCN(C(=O)Cc2c[nH]nc2O)C(CCC)C1 c1(C(N2CCC(NC(C3CCCC4CC34)=O)C2)=O)ccc(Br)c(Cl)c1 C(N=c1ncc([N+](=O)[O-])c[nH]1)C1(CC=C)CCN(C(=O)CN(C)C2CC2)C1 c1(C(=O)NCC2(CNC(=O)Cn3cnccc3=O)CCCC2)cc(Cl)ncc1Cl c1(C(=O)NC(CNC(CCC(=C)Cl)=O)CCOC)ccc(C)cc1SC Cc1noc(C(C)C)c1NC(N1CCCC1Cn1cc(C(=O)O)nn1)=O n1(CC(N2CCC(N(C(=O)COC3COC3)C)C2)=O)nc2c(n1)CCCC2 c1(CN2CCN(CC(N3CC(O)CC3CO)=O)CC2)cc(Cl)cnc1Br C(=O)(C1=CC2CCCC12)NC1CC(CNC(COc2cc(C)c(Cl)cc2)=O)C1 C#CCC(C)C(=O)N1CCCC1C(C)NC(c1cnn(C(C)C)c1Br)=O C(=O)(C(O)CCNC(=O)NC12CCC(CC1)C2)NC(C)=O CC(C)(C)C(O)C(=O)N1CC=CC(NC(=O)CCn2cccc2)C1 CCCC(C)(C)CC(=O)NC1CC2(C1)CC2C(=O)N(C)Cc1cn(C)nn1 n1(CC)ccc(C(=O)NC(Cc2ccco2)C(=O)NCC(C)(O)CN(C)C)c1C C1(C(N(CC(C)CNC(c2ccc(N(C)C)cn2)=O)C)=O)CCc2nc[nH]c2C1 c1(C(N(C2CCN(C(=O)C(C)(C)F)C2)C)=O)ccc(C2CC2)cc1F C1(C(=O)NCCCCNC(C2CCCC(C(F)(F)F)O2)=O)(CC)CNC(=O)C1 N1(C(C2C(CC)CCC2)=O)CCCC(NC(c2ccc(O)c(C)c2)=O)CC1 C=CC(C)(O)C(=O)N1CC(C(C)NC(c2cnn(C(F)F)c2)=O)C1 CC1CC(C)(C)CCC1NC(=O)CCC1(C)CN(C(c2cc(Cl)no2)=O)C1 C(CCC(C)C)(C(=O)NCC12CCC(C1)C(=O)N2)NC(CCC(=C)Cl)=O c1(C(C(=O)N(CC(C)CNC(c2cn(C)c(O)n2)=O)C)(F)F)cccc(F)c1F N1(C(c2ncccc2F)C(=O)NCC2CC2)CCN(c2ccc(Cl)cc2)CC1 N1(C(CNC(c2cccc(OCCNC)c2)=O)=O)CCN(C)C(=O)C1 CC1CCCn2cc(-c3ccc(NCC4CC(C(F)(F)F)CO4)cc3)nc21 N1(C(CC(C(=C)C)OCC)=O)CC2CCC(C(=O)NOCC3CCC3)(C2)C1 N#Cc1ccccc1-c1cn(C2CCCN(S(=O)(=O)C3CC3)C2)nn1 C12(CNC(CCC)=O)CCC1CCN2C(c1csc(Br)c1C)=O CCCC(C)(CC)C(=O)NC1COCC1CNC(=O)C(Cl)=CCl C(C)(C)(CC(F)C(=O)NCc1n[nH]c2c1CCC2)NC(CCNC(=O)NC)=O C1(O)(C(C(=O)NCC(CNC(C2C(C)(CC)C2)=O)C)(F)F)CCOCC1 C1(N(C(=O)CC2CCOC2)C)CCCN(C(C2(C)CC2(Cl)Cl)=O)CC1 C(=O)(C1CCc2cc(F)ccc21)NCCN(C)C(C1CCCCC(=O)N1)=O CC(=O)CCN=C(NCC1(CO)CCCOC1)NC(c1cncnc1)C CC1CCCC1(C(=O)NCCN1CCCCC1=O)NC(=O)CCC(C)N(C)C C(=O)(C(O)C(C)CC)NCCC1(NC(COCC#C)=O)CCCC1.C1(C)CC1 C(C(CNC(C12CSCC1C2)=O)C(F)(F)F)NC(CCCC)=O C1(NC(C2(CC=C)CCC2)=O)CCC(C)N(C(c2sc(C)cc2C)=O)C1 N1(C(C2CCCN(C(C3(C#C)CCCC3)=O)CC2)=O)CCC(C)C2(CCC2)C1 C1(NC(=O)C(Cc2cc[nH]n2)NC(C2CCSC2)=O)CC(C2CC2)C1 C(CN=C(NCCC1CCOCC1)NCC1CCOC1)c1c(C)cn(C)n1 C1(C#N)(CC(=O)NC2(C)CC(NC(c3cc(C4CC4)no3)=O)C2)CCOCC1 c1(C(N(CCCNC(=O)C(F)CC2CCC2)C2CC2)=O)nccn2nccc12 C1(NC(COCC#C)=O)CCC(N(C(=O)Cn2nnc(C3CC3)n2)C)C1 CC1=C(C(=O)N2CCN(C(=O)C=CC(C)C)CC(C)(C)C2)CCC(C)(C)C1 c1(CC)cn2c(C(=O)NC(C)C(C(C)C)NC(=O)CCNC(N)=O)cccc2n1 C1(C(N2CC(C3(NC(Cc4n(C)ccc4)=O)CC3)C2)=O)CCC2(CCOC2)O1 CC1(C)CCN(C(=O)CCC2CCOC2)CC1C(=O)NC1(CO)CCCCC1 Cc1cc2occ(C(N3CC(O)(CNC(c4cncc(F)n4)=O)C3)=O)c2cc1C C(C)(CC(C)(C)CO)NC(CC(C)(C)n1cc(COCC(=O)OC)nn1)=O c1(C(=O)NCC2CCN(C(COCC#C)=O)C2)cc(O)ccc1Br C1(C(=O)NCCCOCC)CCCC12CCN(C(c1cscn1)=O)C2 C=CCCC(C(=O)NCC(c1ccco1)OC)NC(=O)CCn1cnnn1 Cc1[nH]c(C(C)C)c(C)c1C(=O)OC.c12c(cccc1O)CC1(CC1)CNC2 CC1CN(C(=O)CCN2CCCC2=O)CC1NCc1ccc(C#N)s1 C=CCCC(CC(C)C)C(=O)N1CCN(C(=O)CC2CCN(C)CC2)CC1CO N1(C(c2n(CC)c(O)nc2)=O)CCN(C(c2ccc(N)cc2F)=O)C2CC12 c1(OCC(=O)NCC2CC2NC(=O)Cc2cc[nH]n2)ccccc1 C(=O)(CCC(C)(C)C(=O)NC(C)CC(C)NC(=O)CN1CC2CCC1C2)OC N1(C(C2(CC)CCCC2)=O)CCC(CO)(CNC(C2CC2C(F)(F)F)=O)C1 c1(C(=O)NC2CN(C(CCC)=O)CC2c2ccccc2)nc(C)c(C)nc1C c1(C(=O)NC2CC(CNC(c3occ(C)c3C)=O)C2)nc(C(C)C)ncc1Br c1(C(=O)NC2CCN(C(c3onc(C)n3)=O)C2)ccc(P(C)(C)=O)cc1 CC(=O)CCN=C(NCC(CO)C1CC1)N1CCc2cccc(Cl)c2C1 c1(CC)nn(C)c(Cl)c1C(=O)NCCC1CCCN(C(C2(C)CC(C#N)C2)=O)C1 c1(N(CC=O)CC)ccnc(Cl)c1.N1CC(SC)C1 CC(C(CO)NC(=O)C(C)C1CCC1)NC(=O)Cn1cnc(-c2ccccc2)c1 CC1(C)CN(C2CCCN(C(=O)Nc3c[n+]([O-])n[nH]3)C2)C(=O)O1 CC(C)C(CC(=O)NCC1CCC2(C1)OCCO2)C(=O)OC(C)(C)C C1(N(C(c2nc(N(C)C)oc2)=O)C)CCCN(C(c2cn(C(C)(C)C)cn2)=O)C1 Cc1nc2n(n1)CCN(C(=O)C(C(C)C)NC(=O)C1=C(Cl)CCOC1)C2 C(=O)(C(C)C(O)CC)NCc1onc(-c2ccc(CC)cc2)n1.N1(C)CCOC1=O c1(C(=O)NCCN2CC2=O)cc(C)nc(O)n1.c1(N(C(C)=O)C)ccccc1 N1(C(c2c(C)cc(Br)cc2)=O)CCCC2(NC(C3CCCC3)=O)CCCC12 N1(C(c2csc(C(F)F)n2)C(=O)NCCC2CC2)CCN(c2cncnc2)CC1 C12(C(N(C)CC3N(C(C(C(C)C)(C)O)=O)CCC3)=O)C3CC(CC13)C2(F)F C#CCCCC(=O)N1CCC(CCOC)(NC(=O)C(CO)OC)C1 C1(C(=O)NCc2cccc(NC(=O)CCC(C)SC)c2)(CC)CC(C)(C)C1 C(C(CNC(=O)CC1CC(C)=NO1)CO)NC(C1(SCC)CC1)=O C12(NC(CCSC)=O)CCN(C(=O)CS(=O)(=O)N(C)C)CC1C2 O=C(C1CCCn2cnnc21)NCCCCCNC(C1OCC2CCCCC12)=O c1(OC)cncc(CCC(=O)NC2CCC(CC(=O)NC3(C)CC3)CC2)c1 C(C1=CCN(C(=O)Cc2cscn2)CC1)NC(c1cc(C2CC2)cc(F)c1)=O N1(C(C=CSC)=O)CCN(C(C23COC(CS(C)(=O)=O)(C2)C3)=O)C(C)C1 c1(C(=O)NCCS(C)(=O)=O)n[nH]c2c1CN(C(c1cc[nH]n1)=O)C2 CC1(C(=O)NCCc2ocnc2CNC(C2(O)CCSC2)=O)CCCO1 Cc1cccc2cc(C(N3CCCCC3C(C)NC(=O)COCCO)=O)[nH]c12 C(CC)(CC(=O)N1CC=CC1COC)N(C(C1C(=C)C1)=O)C N1(C(Cn2ccc(C)c2)=O)CCC(CNC(=O)Cc2cc(C)nn2C)C(O)C1 CCC(CCCC(=O)N1CCC(CC(C)C)CC1)NC(C1CCCC(=O)C1)=O CC1CCC(C)(C(=O)NCCCCNC(=O)CCc2cnccn2)C1 c1(C(N(C(CCSC)C)C)=O)csc(CNC(=O)OC(C)(C)C)n1 C(CC)(c1ccccc1)=CC(=O)NC1(CNC(C(CC#C)C2CC2)=O)CCCC1 c1(C(=O)NC2CCCC(NC(CCNC(C)=O)=O)CC2)cc2sc(Cl)cc2[nH]1 c1(NCC(C(CC)C)O)ccc(S(=O)(=O)NCc2c(C)cc(C)cc2C)cc1Br c1(NC(CCSCC(C(F)(F)F)OC)=O)cc(Cl)ccc1C c1(OCC(=O)NCC2CCCCN2C(=O)C(F)(F)C2CC2)ccc(F)cc1 N1(C(CC(C)(C)C)=O)CCN(Cc2cocn2)CC1C#N C1(CNC(C(C=C=C)C)=O)CCCC2(CN(C(=O)C#CC(C)(C)O)C2)O1 N1(c2nc(N(C)CC3CCCO3)nc3c2scc3)CCN2C(CNS2(=O)=O)C1 C1(OC)CC(CNC(C2(C(C)(F)F)CC2)=O)N(C(=O)C(C)CSC(F)(F)F)C1 C1(C(=O)NCC2CC(O)CN2C(=O)Cc2ccsc2Cl)CCC=CCCC1 c1(C(C(=O)N(C2CN(C(C3CC=CC3)=O)C2)C)O)cccc(Cl)c1 c1(CC2(C)CC2)nc(-c2cc[nH]n2)n(-c2ccc(F)nc2)n1 CC1CCC(CNC(C2(N(C)C)CC2)=O)CN1C(=O)CCCn1c(O)nnc1O c1(C(N2C(CNC(CCC#C)=O)CC(C)(C)C2)=O)cc(C)cc(Cl)c1N CCC(CC)C(C)NC(=O)CC1COCCN1C(C1CN(C)C(=O)N1)=O c1(C=O)cnc(O)c(C)c1.C(C(C(=O)N)N1CCC1(C)CCO)SCC N1(C(C2(COC)COC2)=O)CCCCC1C(=O)Nc1cccc(C)n1 N1(C(CCCC=C)=O)C(C)CN(C(=O)CC2(O)CCCCC2)CC1C S(=O)(=O)(c1ccccc1F)N1CCN(CCCNC(c2cnc(Cl)cn2)=O)CC1 N1(CC(=O)NC2C3CC2N(C(C2CC2CF)=O)C3)C(=O)NC2(CCCCC2)C1=O CC(C)CC(C(=O)NCC1CCN(C(c2cc(O)cc(Br)c2)=O)C1)C(N)=O Cc1oc(C#N)cc1C(=O)NCCOC1CCN(C(=O)CC(C)CF)CC1 c1(CN(C(C(=O)NCC(CC)O)=O)C(C)C2CC2)ccc(N2CCCC2=O)cc1 CC#CCCCC(=O)N1CCC(n2cc(CNC(=O)C(F)C(C)C)nn2)C1 c1(CC)cc(C(=O)OC)c(C)cc1Br.c1(-c2c[nH]nn2)cc(-c2ccsc2)c(Cl)s1 C1(C(N2CCN(C(C3OCC(C)(C)C3)=O)CC2)=O)CC2CCC(C1)O2 C(CCc1ccccc1)(C(=O)NCSC1CCOC1)N(C)CC1OCCC1CN c1(NC)cc(C(N2CCC2CNC(C2CC(C)=NO2)=O)=O)cc(C2CC2)c1 CC1Oc2ccccc2C1NC(=O)C(c1ccc(C(C)(C)C)cc1)(C)C C1(NC(c2c(C)oc(C(C)C)c2)=O)CN(C(=O)CSc2cnn(C)c2)C(C)(C)C1 N1(C(c2nnn(CC)c2C)=O)CCC(CNC(c2cnc[nH]2)=O)C(C)C1 c1(CC(C)NC(=O)C(C)C(C)c2ccc(F)cc2)cnc2ccc(F)cc2c1 C1(C(=O)NCCNC(c2ccco2)=O)CCc2ncnn2C1.C123CC1CN(C2)C3=O N1(C(CCCn2c(C)ncc2)=O)CC2CN(S(=O)(=O)C(Cl)(Cl)Cl)C2C1 C(=O)(C(CC1CC1)NC(=O)Cn1nccc1C)NCC1(SCC)CC1 N1(C(c2ccc(C)c(I)c2)=O)CCC(C)N(C(c2cc(CO)cc(Br)c2)=O)CC1 c1(OC(C)C(=O)N(C)CC2CCN(C(=O)C(C)(F)F)C2)ccc2c(c1)CCCC2 C(CC1CC1)(CC(=O)N1CCCC(C(C)C)C1)NC(COCCC=C)=O C1(C#N)(C(N(C(C)CCNC(c2c[nH]nc2C(C)(C)C)=O)C)=O)CCCOC1 C1(OCC(C)C)CC(N(C=O)C(c2cccc(C(C)C)c2)C)C1(C)C N1(C(c2c(C)nn[nH]2)=O)CC(C)CN(C(=O)CC2C=CCCC2)C(C)C1 C12(NC(C(C)OCCCC)=O)CC(CO)(C1)OC21CN(C(=O)CC(CC)SC)C1 c1(C(=O)NC23C(CN(C(C4C(C=C)C4)=O)C2)C3)nnc(O)c2c1CCCC2 C1(C(N2CC(NC(c3ccc(-c4cn[nH]c4)cc3)=O)C2)=O)CN2CCCC1CC2 Cc1cc(C)c(C=CC(=O)NC2CCC(NC(=O)CC3CN(C)C3)C2)cc1C N1(C(C2(F)CCN(C(c3ccccc3F)=O)C2)=O)CC2(CCNC2=O)C1 CC1(C)CCC(C(=O)NCC(C)(C2CC2)NC(=O)Cc2ccncc2Cl)C1 N1(C(c2cnc(C(C)C)o2)=O)CC(F)CC1CNC(c1cc(C2CC2)ns1)=O C(=O)(C(C)(C)C(F)F)NC(C)C(C)NC(c1cccc(SC(F)(F)F)c1)=O C1(C(=O)NCC2CCCN2C(=O)CCOCC(F)(F)F)C=CC=CC=C1 C(=O)(N1OC2CCC1CC2)C1C(NC(c2c(C)scn2)=O)CCCC1 c1(C(=O)NC(CC=C)CNC(c2ccc(C)cc2N)=O)nnn2c1C(=O)NCC2 CC#CC1CCN(C(=O)C(C)(C2CCC2)NC(c2cnc(C)nc2)=O)C1 Cc1ncc(Cl)c(C(=O)NCC2CCN(C(c3cc4[nH]ccc4s3)=O)CC2C)n1 C1(CNC(Cc2n(C)ccn2)=O)CN(C(C2CCS(=O)(=O)CC2)=O)C2CCN1C2 C1(C(N(C2CN(C(C(C)(C)N(C)C)=O)CC2(C)C)C)=O)CCc2ccccc2O1 C1(NC(c2c(C)n[nH]c2)=O)CCN(C(c2cc(C(C)(F)F)n[nH]2)=O)C(C2CC2)C1 C1CCC(C)NC(=O)COC2(CC2)C(=O)N1.c1(COC(C)=O)n[nH]c(O)n1 C1(C)(C(N2CCCCC(C(NOCCOCCOC)=O)C2)=O)CC(=O)N(C)C1 Cc1[nH][nH]c(=N)c1C(=O)N(CCCCN(C(=O)CCCOc1ccccc1)C)C c12noc(=O)n1CC2.C1(CC)CCCCN1C(=O)C(C)(C)c1cc[nH]n1 C(=O)(CCCCC(=O)NC1CC(C)(CNC(C2CCNC2=O)=O)C1)OC CC1OCCCC1C(N1CC(CC(C)(C)CNC(c2sccc2Cl)=O)C1)=O C(CCC(=O)NC(C1CCCC1)CNC(C1(CSC)C=CCC1)=O)OCCOC Cc1ccc(C)c(C(=O)NCC(C2CC2)NC(=O)C(C(C)O)NC(C2CC2C)=O)c1 c1(OC2CCN(C(c3c(C)cccn3)=O)C2)ncnc2sc3ccccc3c12 N1(C(=O)CC(F)(F)C(F)F)CCN(C(c2ccc(Cl)nn2)=O)C2CCCCC12 O=C1CCOC(C(N2CCOC(CCNC(=O)COc3ccon3)C2)=O)C1 c1(C(N(C2CCCCC2C)CCC)=O)cc(OC)nc(OC)c1 C(=O)(C1C(C)S1)N(CC(O)CC1CC1)C.C(C)(C)(C)OC(=O)OC(C)(C)C Cc1cc(N)c(C(N2CCC(O)(CN(C)C(C3OCCC3C)=O)C2)=O)c(F)c1 N1(CC(N2C(n3cc(C4(C)CCCC4)nn3)COCC2)=O)CCC(=O)NC1=O CC1CN(C(C2(C(F)F)CCC2)=O)CC1NC(=O)Cn1ccc(C(F)(F)F)n1 c1(OC)cccc(CC(=O)N(CCCNC(=O)C(O)C(C)OC)C)c1 c1(C(N)=O)ccc(CNC(c2coc(CNC(=O)COC3CCCC3)n2)=O)cn1 c1(C(N(C2CCN(C(c3ccnc(Cl)c3F)=O)C2)C)=O)ccc(Cl)c(Cl)c1Cl N1(c2cc(CC)ncn2)CCCC(C2(NC(C3CCC(=O)N(CC)C3)=O)CC2)C1 C1(CNC(c2c(CC)c[nH]n2)=O)CC2CC1CN2C(c1ccc(N)cn1)=O c1(OC)cccnc1C(=O)NCCC1CCC(NC(=O)Cc2cnsc2)C1 C1(C(=O)NC(c2nccc(C(F)(F)F)n2)C)CNc2ccnn2C1 c1cc2n[nH]cc2c(-c2ccc(C3CCCN3)cc2)n1 n1(CC=C)nnnc1C(c1nnc(C2CC2)s1)NC(C)Cn1cnnc1 CC(C)(C)C(C(=O)NCCC1CCCO1)NC(C1COCC1(C)C)=O c1(C(=O)NC(CNC(Cc2cc(C)sc2)=O)CC(F)(F)F)ccc2nc[nH]c2c1 CC(C)CCC(=O)C(=O)NC12CC(C(N3CCC(O)C(C)C3)=O)(C1)C2 O=S(=O)(c1ccc(N2CCCC(CCCO)C2)c(Br)c1)N1CCN(CCO)CC1 c1(C(=O)NCC(CC)NC(=O)C(O)C2CC2)ccc(O)c(C(C)=O)c1 C(CCC(=O)NCc1ncccn1)N(C(C=CC=CC)=O)C C1(CNC(c2ccc(CO)o2)=O)CN(c2nccc(Br)n2)CCO1 CC1(C)CCCC1CCNC(=O)C(C)(C1CC1)NC(c1cc(O)cs1)=O CC(CN(C)C)CC(=O)N(C1CCN(C(C2(n3ccnc3)CCCC2)=O)CC1)C C(C(N=[N+]=[N-])C(=O)N1CCCC1(CNC(=O)C(C)(C)C1CCC1)COC)OCC N=c1cc(C(N2CCCC2c2c(F)cccc2Cl)=O)c(F)c[nH]1 C12(C(=O)NCCC(CC)(C)C)CCC(CC1)N(C(c1cc(C)c(C)[nH]1)=O)C2 C(=O)(CC(C)C(=O)N1CCC(N=[N+]=[N-])C1)OC.c1(C2C(=O)N2)c(C)cccc1Br CC(C)C(CNC(=O)C(c1ccc(Cl)s1)C)NC(=O)CCCOC1CCOCC1 CCC(C)C(C(=O)N1CCOC(C(=O)NC2COCC2N=[N+]=[N-])C1)N(C)C c1(CC)nncn1NC(=O)C(Cn1cncn1)NC(C1CCN(C)C1=O)=O CCCCC(CC(=O)NCC(C)C(F)(F)F)NC(=O)C(C)N=[N+]=[N-] c1(C(=O)NCC2N(C(C3OCCN(C)C3)=O)CC2)coc(S(N)(=O)=O)c1 c1(C(N2C(C)CC(NC(C(C)=C3CCC3)=O)C2)=O)cc2c(Br)cccn2n1 c1(C(=O)NC2C(NC(C(CC)C#N)=O)CCC2)cc(Cl)ccc1O N1(C(CC(=O)NCC)=O)CC(NC(C2CCCCC2(F)F)=O)C(S(C)(=O)=O)C1 CCC(C)(Cl)CNC(=O)COCCNC(=O)CCC1CCOC1 C1(C(=O)NC2(C(F)(F)F)CC3CCC2C3)CCC12CCOCC2 C1(NC(C(C)(C)OCC)=O)CCN(C(c2ccccc2C2CC2)=O)CC(C)(C)C1 C(CN=c1[nH]c(N2CCC(OCC3CCCO3)CC2)nc2c1CCC2)NCC c1(C(=O)NC2C=CCN(C(CSCC(=O)OC)=O)C2)ccc(F)c(F)c1F N1(C(C(C2CC2)SC)=O)CCC(=CCNC(C2CCCC23CC3)=O)CC1 c1(CN2CCCC(CNC(c3cc(F)c(Br)cc3Cl)=O)C2)ccc2cc[nH]c2c1 C1(CC(=O)NCC(C2CC2)NC(=O)C=CCn2cncn2)CC(O)C12CCC2 C1(NC(c2c(C)n(CCO)nc2)=O)CCCCN(C(C2OCC3CCCC23)=O)C1 c1(C(N(CCN(C(CN(C(C)=O)C)=O)C)C)=O)csc(C(C)(F)F)n1 N1(C(C)=O)CCC(C(=O)N(C2CC(NC(=O)CC(C)(C)C)C2)CC2(F)CC2)CC1 N1(C(CC(CCCC)O)=O)C2CCCC1CC(NC(=O)CCc1ncco1)C2 C#CC1(C(=O)NCCC2CN(C(=O)C(C(=O)OC)OC)CCO2)CCCC1 CC1CC(=O)NCC1C(=O)NCC1=CCN(C(C2CCCC(F)C2)=O)CC1 C1(N(C)C(c2coc(C(N)=O)c2)=O)C2CN(C(=O)C(C)(C)C)CC12 c1(C(C)C(=O)NCC(C(C)(C)C)NC(c2ccoc2)=O)ccc(Br)c(Cl)c1 C(=O)(C(O)CC[S+](C)C)NCCC1CCCN(C(C(C)Cc2cnc[nH]2)=O)C1 C1(C(=O)NCc2conc2C)(CC)CCN(C(c2cn(CCO)nn2)=O)CC1 CC1(C)Cc2[nH]nc(C(N3CC4CC3C4NC(=O)C3=CCCCC3)=O)c2C1 N1(C(C2C(C)CCC2)=O)CC2(CCC(NC(=O)CC3CCOCC3)CC2)C1 C#Cc1cnn(C)c1C(=O)NCCc1ccc(CNC(C2CCSC2)=O)cc1 C=CCC(CNC(=O)CSC(F)(F)F)NC(=O)CC(=C)Br C1(OCCNC(=O)OC(C)(C)C)CCCCN1CC(F)F C(c1ccc(F)c(OC)c1)=CC(N1C(CNC(C(C)=CC)=O)CC(O)C1)=O N1(C(C(CCC)F)=O)CC(NC(=O)Cc2ccc(O)cc2Cl)CC12CCCC2 C1(NC(C(c2ccccc2C(F)(F)F)C)=O)C2CC1N(C(c1cn[nH]c1)=O)C2 c1(C(=O)Nc2ncc(C(C)(C)C)o2)ccc2c(c1)C(=O)CCC2 C1(CC)C(=O)NCCCN1C(C1(NC(=O)CCc2cnoc2)CC(F)(F)C1)=O C1(C(N(CC(C)CNC(=O)COC(F)F)C)=O)C2CNC(=O)C12 C1(N(C(=O)CC2CCCN2C(=O)CC2(NCC)CCC2)CC)CCN(C)C(=O)C1 N1(C(CS(CC)(=O)=O)=O)CC2(CCCC2)C1C(=O)NC1CC2CCC1O2 c1(C(C)NC(CN(C(=O)C(C2CC2)OC)CCOC)=O)ncc(C)o1 c1(CNC(C2CCN(Cc3cc4n(n3)CCC4)CC2O)=O)cc(Br)ccc1O N1(C(CC(COC)C)=O)CC(C2CN(C(=O)CCc3cccn3C)C2)C1 N1(C(CSCCC=C(C)C)=O)CCCCC1C1CCCN(C(=O)CO)C1 c1(CC(N2C(C)C(NC(=O)CCN3CCC3)CC2)=O)cc(F)ccc1F C1(C(N2C(CNC(C=C(C)C(C)C)=O)CC(O)C2)=O)CC12CCCCC2 C(=O)(C(CC(C)C)c1ccc(Cl)cc1)NC(CNC(c1c(C)scn1)=O)(C)CO c1(OCC(=O)N(C2CCN(C(c3n[nH]cc3C3CCC3)=O)C2)C)ccccc1 C1(CN(C)C(C2CCC=CCC2)=O)CCCCN(C(C2CC2(C)C)=O)C1 CCC(C(=O)NC(CC)CCCC(=O)NC1C2CCCCCC12)C(C)(C)CC C(CN=C(NCC1(C)CCCCC1)NC1CCCS(=O)(=O)C1)OC c1(CC)ccnc(C(=O)NC(C2CCCN2C(=O)Cc2sc(C)nc2C)C)c1 C1(CCNC(c2c(C)scn2)=O)CN(C(C2CC3(C2)OCCO3)=O)CCCO1 C(=O)(CCCN=c1[nH]c2ccccc2s1)NC(CNC(C(CN(CC)CC)F)=O)C c1(C(=O)OC)nc(C(=O)NCCN(C(=O)C(O)CC2CC2)C)cs1 c1(C(=O)NC(C2C(C)CCC2)C2CN(C3CC3)C2)cccn(C2CCSC2)c1=O c1(CC)c(NC2CCC(CNC(=O)C=Cc3cn(C)cn3)C2)ncnc1Cl c1(C(N(C2CCCN(C(C3(C#C)CC3)=O)CC2)C)=O)nc(C)[nH]c2nccc1-2 c1(C(=O)NCCNC(Cc2c(C)nc(Cl)cc2)=O)cc2cccc(Br)c2o1 c1(CC(=O)NC2C(C)(NC(C(CC=C)CC)=O)CCC2)cccc([N+](=O)[O-])c1 c1(COC)ncc(C(=O)N(CCCN(C)C(C2CCCC(C)C2)=O)C)c(O)n1 C12(NC(Cc3cccc(OC)c3)=O)CCN(C(=O)C=C3CCN(C)C3)CCC1C2 NS(=O)(=O)C1CCc2ccccc2C1NC(c1cc(Br)ccn1)=O N#Cc1cncc(C(=O)NNC(C(C(=O)O)C2=CCCS2)=O)c1 C(=O)(C1CCCc2nc[nH]c21)NCC(C)CNC(=O)C=C(Cl)Cl C1(C(=O)Nc2ccccc2Cl)CN(C(=O)COc2ccccc2)CC1O c1(CNC(=O)NC2C(OC(C)(C)C)CCCCC2)cc(O)c2sccc2c1 C(CC(=O)N1CC=C(CO)CC1)(C(C)(C)C)NC(c1scc(OC)c1)=O Cc1nc(NC(C2CSC2)C)cc(=NCc2ccc(OCC(C)C)nc2)[nH]1 CN=c1[nH]c(C(N2CCC(NC(=O)C(c3cncn3C)N(C)C)C2)=O)cs1 Cc1ccnnc1C(=O)NC1CCCC(CN(C(=O)CC(C)(F)F)C)C1 c1(NC(c2cccc(OC)c2C)=O)ncc2ccc(C3=CCCCO3)cc2n1 C1(CNC(CC2(NC(c3ccc(CC)nc3)=O)CCC2)=O)CCOC(C)(C)C1 C1(C(=O)NC(C)CNC(=O)C(c2ccccc2)C)COC2(CO)CC1C2 n1(CCC)nc(C)c(NC(C2CC(C)N(C(=O)COCC3CCCC3)C2)=O)c1C C1(CCNC(C2(CC#C)CC2)=O)CCCCN1C(=O)CCn1cc(Cl)cn1 CC1CC(C(N2CCOC(C)(CNC(c3cc(Cl)no3)=O)C2)=O)CCN1C N1(C(c2nc(CCOCC)oc2)=O)CCN(C(=O)Cc2cnnn2C)CCC1C c1(C(=O)NCC2CC(c3ccccc3)CO2)cc(Cl)cc2c1OCC2 c1(C(N2CCC(NC(C(C=C)(F)F)=O)CC2)=O)cc(C)c(C)c(F)c1 C=CCC(F)(F)C(=O)NCC1CC(NC(=O)C(CCF)NC(=O)OC(C)(C)C)C1 N1(C(=O)NCC2CCC3(CCCC3)O2)CCN2CCNCC2C1 O=C(C#CC1CCCO1)N1CCCC(CNC(c2cnc(CC3CC3)s2)=O)C1 c1(C(N2C3C(NC(C=C(CC)C)=O)CC(C3)C2)=O)ccc(Cl)c(C#N)c1 c1(OC)ccc(C)cc1S(=O)(=O)N1CC(OCCN=[N+]=[N-])CCC1C C(=O)(C(C#N)C(C)(C)C)NC(CC#C)CC(=O)N(C)CC1CC(O)C1 C1(CN2CC(CNC(C3(CC)CC3)=O)C2)CCOC(C)C1 N1(C(CC(C)(C)C)=O)CCCC(C)(CNC(C2CC23CC(OC(C)(C)C)C3)=O)C1 C(CC(C(=O)NCC(O)CNC(C1CCCCC1OC)=O)OC)OC N1(C(c2cc(C)c(C)o2)=O)CC2CC(NC(c3cnc4[nH]cncc3-4)=O)CC2C1 Cc1cc(N)cnc1C(N1CCC(C(O)CNC(=O)C(C(C)O)N(C)C)CC1)=O c1(CC(N2CC(N(C(c3c(Cl)ncc(C)c3)=O)C)C2)=O)ccc(S(C)=O)cc1 C1(NC(CC2(OC)CCC2)=O)Cc2ccccc2C1NC(=O)C(C)C1CCCO1 N1(C(C2CC(NC(C3C(C)(C)C3(F)F)=O)C2)=O)CCCC(O)CC1 C12CCCN(CC1)C(=O)C1(CCCC1)Oc1ccc(cc1)C(=O)N2CC.N(C)OC S(=O)(=O)(c1cnc(NCC2(C)CS(=O)(=O)C2)cc1C)NC(CC=C)CO CC1NC(=O)CCC1CNC(C1CC2(CC2)CN1C(c1cncn1C)=O)=O c1(C(N(c2c(C)ccs2)C)=O)ccc(CC2CCNCC2)cc1 C=CC(C(=O)NCC1CC1C(N1CCC(CC2CCC2)C1)=O)OC S(=O)(=O)(c1cccc(C(N2CCCC2CNC(=O)CC2CCOC2)=O)c1)NC c1(C(=O)OC)ccc(N2CCOCC2CN(C)C(c2ccsc2C)=O)nc1 N1(C(C2(C#C)CC(=O)C2)=O)CCC(C)C(CC(=O)NCCN2CCOCC2=O)C1 c1(C(N2CCC(C(=O)NCC(C)CCO)C2)=O)cccc(CC#N)c1 c1(C(C(N2CCC(CNC(c3c(CC)cncc3)=O)C2)=O)O)cccc(C)c1F Cn1c(C(=O)NC(CNC(=O)COC2CCOC2)C2CC2)ccc1[N+](=O)[O-] c1(C(C)(C)C(=O)NCCCNC(c2ccn(CC(F)F)n2)=O)c(F)cccc1F c1(OC)cnc[nH]c1=NCCNC(c1cccc(C)c1C)=O C1(CO)(Cn2cc(-c3cccc(C(=O)O)n3)nn2)CC=CCC1 CCC(C)C(O)C(=O)N(C(C)CNC(=O)CCc1ccc(Cl)c(F)c1)C Cc1sc2cncn2c1C(=O)NC1(CC(=O)O)CCSC1 c1(C(=O)NC2C(NC(C(CCCC)(C)F)=O)C2)ccc2sc3ccccc3c2c1 C1(C(N(CC(C)NC(c2c(CC)c[nH]c2)=O)C)=O)CCC(CC)CC1 c1(NC(=O)CC2CCN(Cc3ccc4ncoc4c3)C2)cc(Cl)cc(Cl)c1Cl C1(C(N2CC3CC(Nc4ccnc(CO)n4)CC2C3)=O)CCCC2(CCC2)C1 C(=O)(C1=CC(C)(C)C1)NCC=CCNC(C1(OC)CCC(C)C1)=O c1(C(=O)NC2C(NC(C(C)OCCOCC)=O)C2)ccccc1F N1(C(C2CC(C)(C)C2)=O)CCC2(CC2C(=O)Nc2ccnc(-c3ccccc3)n2)C1 N1(C(C(C)(C)NC(=O)OC(C)(C)C)=O)CC=C(CNC(c2ccno2)=O)CC1 N1(C(CCCC)=O)CC2CCCC1C2CNC(c1ccc(-n2cnnn2)cc1)=O CC(C)CCCCC(=O)NC(C)(C(N)=O)c1cccnc1 C(CCCCNC(C1CCC(=O)N1)=O)N(C(CCOC(C)C)=O)C C1(NC(CCc2cc(C)on2)=O)CC2(C1)CC2NC(c1nc(C(C)C)oc1C)=O CCCN=c1[nH]c(N2CCN(C)CC2)nc2ccc(Cl)cc12 c1(CC(N2CCN(C(C(C)S(C)(=O)=O)=O)CC2)=O)ccc2c(c1)NC(=O)C2 C(=O)(C(C)(C)CC(F)F)N1CC(C(N(CC(CC)(C)OC)C)=O)C(C(C)C)C1 C1(CNC(c2cnc(NC(C)=O)o2)=O)CCC2(CCC2)C1NC(=O)CC(C)(F)F c1(C(N(CCCCNC(C2(C(F)(F)F)CCC2)=O)C)=O)cc2cccc(F)c2s1 c1(C(N2CCCC(N(C(CCCOC)=O)C)CC2)=O)ccc(P(C)(C)=O)s1 C(C)(C)(CCCNC(C12CCC1CC2)=O)NC(C1CCC(OC)C1)=O C1(C(=O)NC(C(=O)OCC)SC)(OC)CCN(C(=O)C2=CCCC2)C1 c1(NC(CCC2N(C(C(CC)(C)O)=O)CCC2)=O)nc(F)c(Br)cc1Br N1(C(c2cc(C)[nH]c2C)=O)CC(NC(c2cc(C(C)C)n(C)n2)=O)CC1(C)C CC1(CN(C(=O)CCC2CCCO2)CC2CC2)CC1(F)F Cc1cccc2c1OC(C(=O)NCCCCCCNC(C1(C)CNC(=O)C1)=O)C2 N1(C(c2c(C)sc(O)n2)=O)CCC(F)C(NC(c2cc3occc3s2)=O)C1 Cc1ccc(F)cc1C(N1CCCCC1CCNC(C1CC2CC2CC1C)=O)=O N1(C(CCCC(C)C)=O)CCN(C(c2cnc3n2CCCC3)=O)CC(C)(F)C1 N1(C(CSCc2nc(C)sc2)=O)CCN(C(=O)OCc2ccccc2)CC1C Cc1cc(C(=O)NC2(CNC(=O)CCCC3CCOCC3)CCC2)no1 CC1COC(C(=O)NC2(C)CC(NC(=O)CSc3nnnn3C)C2)C1 C(CC(=O)NC(C)C)(OCC)OCC.C(=O)(C(=O)NCC)NCC1CC1 c1(CNC(CN(C)C(N)=O)=O)nnc2n1CCN(C(=O)CN=c1cc[nH]cc1)C2 C1(NC(C(c2nc(C)sc2)=O)=O)CCC(NC(C23CCC(C2)C3)=O)CC1 C1(NC(=O)C(c2ccc(F)cc2)F)CCC12CN(C(=O)CC1COCCOC1)C2 N1(C(C(C)N2CCCC2)=O)CCC(NC(C2C=CCCC2)=O)C12CCC2 c1(C(N(C)CC2CCCC(NC(=O)Cn3cncn3)C2)=O)c[nH]nc1S(N)(=O)=O c1(CCNC(C2COCCN(CC3CC4CCC3N4)C2)=O)nc2c(o1)CCSC2 C=C(C)CC(C(=O)NCCC(CNC(=O)C=C1CCC(C)(C)CC1)OC)NC(C)=O C#Cc1ccc(NC(=O)NCC(c2ccc(OC(F)(F)F)cc2)(F)F)c(C)c1 CC(CNC(C1CCC(NC(C2CC2(F)Cl)=O)C1)=O)C(C)(F)F CC(C)(F)C(=O)NCCOC1CCN(C(=O)CN2CC(F)(F)C2)C1 Cc1cc(C(=O)OC(c2nc(C(=O)N(C)C)co2)C)ccc1Br C1(NCC=C(C)C)CC2CCC1CC2NC(=O)CC1COC(=O)C1 N1(C(CCC)=O)CCCCC1C(N1CCC(N(C)C(c2coc(CO)c2)=O)C1)=O C1(NC(CC2(CC)CCC2)=O)CC2CC(C1)N(C(=O)Cc1ccc(F)cc1)C2 N1(C(C2C(CNC(C3=CCN(C)C3)=O)CCC2)=O)CC23CCC2(COC3)C1 N1(C(C2N(CC)CC2)=O)CCN(C(C2CCCCCC2)=O)C(c2nccn2C)C1 c1(NC(=O)NCC2(C(=O)NC)CCCC2)ncccc1O C(CN=C(NC1CC1)N1CCC(n2cccn2)C1)c1cc(F)c(Cl)cc1 C1(NC(C=Cc2cnc(C)s2)=O)CCC12CN(C(=O)C(C)NC(N)=O)C2 c1(C(=O)NCC(C(C)C)(C)NC(=O)CC2=CCN(C)CC2)cc2scc(Cl)c2[nH]1 c1(NC(C(C)(N(C(=O)Cn2ccnc2)C)C2CC2)=O)cccc2c1OCC2 C1(N(C)C)CN(C(C(=O)NCc2ccc(F)cc2)C2CCOC2)CC1C1CC1 C1(CC(=O)N(CCOC)CCOC)CC(C)(C)CN1C(=O)CCN1CCCCC1 c1(CNC2C3CN(c4nccc(C)n4)CC32)c(O)cccc1O CN1CC(C)(C(N2CC(N(C)C(C3C4C5CCC(C5)C34)=O)C2)=O)CCC1=O C1(NC(c2cccc(COC)c2)=O)CCN(C(=O)C=C(C)C(F)F)C(C2CC2)C1 N1(C(C2(CCC=C)CC2)=O)Cc2ccccc2C(NC(c2cn(CC)nn2)=O)C1 CC(C)CC(C(=O)N=S(C)(=O)c1nccn1C)NC(c1ccco1)=O C#CCCC(O)C(=O)NCC(CNC(c1cc2occc2s1)=O)C(F)(F)F N1(C(c2cnc(N(C)C)s2)=O)CCC(C)(C)C1C(=O)NC1CCC(F)(F)C1 N1(CCC)CCCN(N2CCC(C(=O)N(C)OC)CC2)CC1 Cc1[nH]c2ccc(F)cc2c1CCC(=O)NCCS(C)=O C1(NC(C2CN(C(CCOC(C)C)=O)C(C)(C)C2)=O)CC(C)N(C)CC1C C1(C)(CNC(CCOCC(C)C)=O)CCCN(C(C2(Br)CCC2)=O)C1 C1(C(N2CCN(C(C(CCC)O)=O)CC2C(C)C)=O)CCCC(F)(F)CC1 c1(C(=O)NCC2(C(F)F)CCN(C(C(C)(C)OC)=O)C2)c(F)ccc2[nH]ccc12 N1(C(C=C(CCC)CCC)=O)CCCOC(CNC(c2ccn(CC)c2C)=O)C1 N1(C(CC(CNC(C2CCC(CO)CC2)=O)OC)=O)CC(O)CC(O)C1 C(=O)(CC(F)(F)C(F)F)NCC(C(C)(C)C)NC(=O)CC1CCCS(=O)(=O)C1 C(=O)(N=c1ccn(CCc2ccccc2)[nH]1)C1CCCC(C(C)=O)CC1 N(S(=O)(=O)N1CCN(CC(C)O)CC1)C(C(=O)NCCCCCC)c1cn[nH]c1 N1(C(C2C(CC)CCO2)=O)CC(NC(=O)C2=COCC2)C(SC)C1 C1(N2C(C(N(C)C)=O)CCC2)CCN(C(C2(CC(=O)O)CCOC2)=O)CC1 C1(NC(C(C(C)C)NC(C(CO)OC)=O)=O)CCCCC12CC2 Cc1cc(C(=O)N(C)CCNC(=O)CC2CCS(=O)(=O)C2)c(N)c(Cl)n1 N1(C(C2C(C(C)C)OCC2)=O)CC=C(C(=O)NOCC2CCOCC2)C1 c1(NS(CC)(=O)=O)ccc(-c2nc(C)c(NCc3ccc(F)cc3)s2)cc1 Cc1c(C)n(CC(F)(F)F)c2ncnc(NC(C3CCCSC3)=O)c12 c1(-n2cc(C(=O)NC(CNC(CSCCC)=O)CO)nn2)cccc(C)c1 C1(OC)C=CCN(C(C2CCCC2CNC(c2n[nH]c(C)c2C)=O)=O)C1 Cc1cc(NC(C2CSCN2C(C2C3CC(=O)CC23)=O)=O)ncc1F c1(N2C3CN(C(CC(C)n4ccnc4)=O)C(CC3)C2)ncc2cccnc2n1 c1(NC(=O)C=Cc2cnccn2)nc2c(s1)CC(NC(C1CCSCC1)=O)CC2 C(=O)(C#Cc1cccc(F)c1)OC.N1(C(=O)OC(C)(C)C)CC2CC1CO2 CC1(C)CCC(C(=O)NCc2cc[nH]n2)CN1C(C1CCCN1C=O)=O Cc1ncncc1C(=O)NCC1CN(C(=O)CC(C)CF)CCO1 CC(CCC(=O)N=c1ccn(CC2CC2)[nH]1)NC(c1cccc2ccoc12)=O CC(C(=O)N1CCC(F)(CNC(C2CCCC3(CC3)C2)=O)CC1)S(C)(=O)=O C(c1c(Cl)cccc1Cl)=C(C)C(=O)NCC(F)CNC(=O)CCP(C)(C)=O C1(C(=O)NC(c2cccnc2)C(=O)NC(COC)CO)OCCC1C(C)C Cc1ccc(-c2cn(Cc3ccc(C(N4CCCC4CSC4CC4)=O)o3)nn2)cc1 C(C(C)(C)CC(=O)N1CCN(C)CC1C(=O)NCc1cccnn1)OC C(=O)(CC1=CCCC1)NCCC(=C)CNC(=O)CC1CCCC(C2CC2)O1 c1(C(=O)NC(CNC(c2c(C)occ2)=O)C(C)C)cnc2c(C)cccc2c1 N1(C(=O)NC(c2cn(C)nc2)CO)CC(Cn2cccn2)Cc2ccccc21 C(=O)(C(CC(C)CC)NC(c1cc(C)nnc1O)=O)NC(CC#C)(C)C c1(C(=O)NC2C(C)N(C(C3CC34CCC4)=O)CC2)cccc2oncc12 C(=O)(C=CS(F)(F)(F)(F)F)NCCCC1CCN(C(C2(CC#C)CCC2)=O)CC1 C1(NC(c2c(CC)noc2)=O)CCCC(CNC(=O)COC2(C)CCCC2)C1 c1(OC)ccc2nc(N3CC(C)OCC(C)(C)C3)[nH]c(=NCCC(C)(C)C)c2c1 Cc1cncc(CC(=O)NCCCN(C)C(C2(N(C)C)CCCOC2)=O)c1 N(C(=NCCCF)NCc1cnc(-c2c(Cl)cccc2Cl)s1)C(C)COC(F)F C1(CCCNC(C(C)c2ccco2)=O)CCCN1C(c1nocc1Cl)=O c1(C(=O)OCC)c(OC)ccc(S(=O)(=O)NCc2nc(SC)ns2)c1C N1(C(c2c(C3CC3)ccc(OC)c2)=O)CCC2(CCC(NC(=O)C(F)F)CC2)C1 CC1CC(C(=O)NC(C)CN2CCN(C(=O)CCc3cc[nH]n3)CC2)CCO1 Cc1ccc(NC(C2CCN(c3ncc(Br)c(C)n3)CC2O)=O)cc1CN(C)C C12(C(=O)NC3CCN(C(C4CCC(C)O4)=O)CC3)CC=CC(C1)OC2 N1(C(CN(C)CCO)=O)CCC(NC(c2coc(C(F)F)n2)=O)C(F)(F)CC1 c1(CN(C(C(=O)NC(c2c(OC)nccc2)C)=O)C2CC2)ccc(F)c(C)c1 c1(NC(CCNC(C)=O)=O)cccc(NC(C2CC(C(F)(F)F)(OC)C2)=O)c1 c1(C(N2CCC(O)(CNC(CCCCSC)=O)C2)=O)cc(Cl)cc2c1NCCC2 CCC(CC)C(=O)N1CCCCC1C1CCCN(c2ncnc(=N)[nH]2)C1 c1(NC(=O)CC2COCCN2Cc2cc(F)ccc2I)cc(C(=O)O)c(F)cn1 c1(SCc2onc(-c3n(C)nc(C4CCCC4)c3)n2)c(I)ccnc1F C1(F)(C(N(C2CCCC(C)C2)C)=O)CCCN(C(c2cnn(C)c2Cl)=O)C1 c1(N(C(=O)NC2CCN(C(C)=O)CC2)C)ccc2c(c1)S(=O)(=O)N=C2Cl C1(CN(C(C2(C(=O)NC)CCC2)=O)C)CCCCN1C(C1CCCS1(=O)=O)=O C1(OC)C(C(=O)Nc2cccc(C(=O)Nc3ccccc3)c2)C2CCCC12 C1(C(N2CCC(C(C)NC(c3ccc(C(C)O)cc3)=O)C2)=O)CC(C)(C)CN1C c1(C(=O)NC2CN(Cc3c(C)cc(Br)cn3)CC2C(=O)O)cc2ccccn2n1 N1(C(C(C)(C)SC)=O)CCN(C(c2ccc(NC(N)=O)cc2)=O)C(CO)C1 C(=O)(CCCC=O)NC(C(=O)N(CC)CC)CC1CCC1.C(C)(C)(C)OC(=O)CO Cc1csc(C(C)NC(C2CC(CO)CN2)=O)n1 c1(C(N2C3CC(NC(C(C)n4ccnc4)=O)C3CC2)=O)noc2c1CCCCC2 C1(O)(C(=O)NC(CC(C)C)CNC(=O)CC2CCC23CCC3)CCC(C)(C)CC1 O=S1(=O)CC2CC1CN2C(=NCCCCl)NCCc1cccc(F)c1 C1(C(=O)NCC(CNC(c2c(CCC)occ2)=O)O)CCCC(O)C1 N1(C(=O)C=CCN2CCC2)CC2CCC(C(=O)NN3CC=CC3)(C2)C1 c1(N(C(c2sc(C)c(O)n2)C(=O)NCC2CCCOCC2)C)ccc2c(c1)CCC2 CC(C)CC(C(=O)NCC(=O)N(C)O)NC(c1cc(Cl)c[nH]1)=O c1(C(=O)NC(C(C)NC(C2(C)CS(=O)(=O)C2)=O)CO)ccc2c(c1)CC(C)(C)O2 N1(C(C2C(C(=O)OCC)C2)=O)CCN(C2CCN(C(c3csc(C)c3)=O)C2)CC1 c1(C2C(=O)N2)nc2cc([N+](=O)[O-])ccc2o1.C(CN(C)C)SC C(=O)(C(C)(C)C(O)C(C)C)NC1CCC(CC(=O)NCC(CC(=O)OC)O)CC1 c1(C(=O)NCC2(CNC(CN(CC)CC)=O)CCC2)cc(F)cc2ccccc12 C(=O)(C(C)(C)CCCNC(=O)NC1CC(O)C12CCC2)N(C)C C1(NC(C(C)CF)=O)CCC2CN(C(c3cc(O)ccc3Cl)=O)CC2C1.C1(C)CC1 CCCCCCC(CC)C(=O)N1CCCCC(NC(c2ccc(C(F)F)s2)=O)C1 N1(C(c2ccc(NC)cc2)=O)CCC2(NC(=O)C(C)c3cncs3)CCCC12 N1(C(C(C2CC2)OC)=O)CC(CN(C)C(c2cc(F)sc2Cl)=O)C2(CC2)C1 CCC(CO)CCNC(=O)C(F)C1CC(NC(=O)C(C)OC(C)=O)C1 C1(CNC(C(=O)N(C)C)=O)OCC2CCN(C(c3cc4ccccn4c3)=O)CC12 CC1CC(NC(C2(c3ccncc3)CC2)=O)CCN1C(C12CC(C)(C1)C2)=O C(CCN=C(NCC)NC1CC(C)N2C1C=C(C(C)C)OC2CC)n1c(C)cc(C)n1 C(=O)(C(CNC(=O)CCOCC)(CC)CC)NC(CC#C)C(=O)OC C1(C(=O)NC(CNC(Cn2c(C)ncc2)=O)(C)C2CCC2)CCCCN(C)C1=O C1(NC(CC2(C=C)CCC2)=O)COCCN(C(=O)C(CC)=CC)C1 O=C(CC(F)(F)F)N(CCC(=O)O)CC1CCCCN1Cc1ccccc1 N1(C(C(=O)NC2C(CC)C(O)C2)=O)CCCCC(CCC(=O)NC)C1 C(C(=O)NCc1ccco1)(C(C)(C1CC1)OC)N(CC#CCOC)C c1(C(N(CCNC(CCN2CCC(C)CC2)=O)C(C)C)=O)ccc(Cl)nc1O N1(C(C(CCC)F)=O)CCC(C)CC1C(=O)NC1CCCCC1OCC CC1CCCCC1(C)C(=O)NC1CCOCC1C(=O)Nc1cccc(C(F)F)c1 C1(OC)CN(C)C(C)(C(N2CCC(N(C)C(c3cccc(N)c3C)=O)CC2)=O)C1 N#Cc1ccc(O)c(C(=O)NC2CCC(NC(c3cncc(Br)c3)=O)C2)c1 C(C)(C)(CC(=O)Nc1ccc(C(C)(C)C)cc1)OC N1(C(CN(C)CC)=O)C2CCCC1CN(C(c1cnc3nccn3c1)=O)CC2 c1(C(N(C(CNC(CC(C(C)C)OCC)=O)C)C)=O)ccc2c(c1N)CCCC2 N1(C(=O)NC(C)CC#N)CC2CC1C(c1ccccn1)(C(F)(F)F)C2 CN1CCN(C(c2nccn2C)=O)C(C(=O)NC2CN(C)C(C)(C)C2)C1 c1(CC(N2C(Cc3c(C)ccc(C)c3)COCC2)=O)cccc2c1OCO2 C1(CNC(C(COC)(C)C)=O)CCN(C(=O)C(C)c2cccs2)CC1C c1(C(N2CC3C(CNC(CNC(C)=O)=O)(C3)C2)=O)cc2ccccc2o1 c1(OC)nn(C)cc1C(=O)NCCCC(=O)N1CCC1C(C)C CC1CCC(C(N2CCCCC2CCNC(=O)CN2CCCOC2=O)=O)CC1 C12(C(N3CCC(CNC(c4ccn(C5CC5)n4)=O)C3)=O)C3CCC(CC13)C2(F)F C12COCCN1C2=O.C1(C(=O)OCC)CC(F)CN1C(=O)Cc1cc(Br)cs1 C1(C(N2C(C(N(CC)CC3CCCO3)=O)CC=CC2)=O)CCC(O)CN1C C#CCCC(O)C(=O)NCC1CC(NC(=O)C(C)=C2CCC2)C1 CC(C)CC(O)C(=O)N(C1CCCCCC1)CCNC(C1CCS1(=O)=O)=O C(CC(C)CC(C)(C)C)OC(C(c1c(OC)cccc1)(C)C)=O c1(CO)ccc(F)cc1.c1(C2C3(CC3)C(C)N2)nnnn1C1CC1 CCCCC(O)CC(=O)NC1CC(NC(=O)C(F)Oc2ccc(Cl)c(F)c2)C1 N1(C(c2ccc(C)nn2)=O)CC2(CCC2)CC1C(=O)NC(C)CC(N)=O C1(NC(COc2cc(C)on2)=O)CC2CC(C1)N(C(=O)CC1CC3(CCC3)C1)C2 N1(C(C2N(C(C)=O)CCC2)=O)CC=C(CCNC(=O)CCCn2ccnn2)CC1 CCCCC(C(=O)N1CCC(C)(C(=O)OCC)C1)NC(c1ccc(C)cc1O)=O N1(C(=O)CCCCN2CCCC2)CCN(C(=O)CCc2ccon2)C(CO)C1 C1(C(N2CCCC(C(C)O)C2)=O)CCC(C)(C)N(C(C2CCCN2C=O)=O)C1 C1(OC)CCN(C(=O)NC2(CNC(C)=O)CCOCC2)C(c2ccccc2)C1 CCC(N=c1[nH]c(=NCCC(O)C2CC2)c2[nH]ccc2[nH]1)C(C)C Cc1cc(C)c(C(=O)N(C)CCN2CCN(C(=O)C(C3CC3)N(C)C)CC2)[nH]1 CC1CCCCCCN1C(=O)C=CC1CCCN1C(=O)CS(C)(=O)=O C1(CNC(c2ccc(CO)o2)=O)CC(O)CN1C(=O)Cc1sccc1Cl C1(C(N2C(CCC=C)CCC2)=O)CN(C(c2cc(C(C)=O)on2)=O)CCC1(C)C c1(C(=O)NC(c2nc(C)on2)C)cc(CNC(=O)C(C)c2ccsc2)ccn1 N1(C(=O)C=C2CC2)CCN(C(=O)CCc2cncs2)C(C(F)F)C1 N1(C(C2C3CCC2(c2cccs2)C3)=O)CCN(C(=O)Cn2cccc2)C(CO)C1 c1(OCC)nc2ccc(C(=O)N(C3CN(C(C4CC4Cl)=O)C3)C)cc2[nH]1 C(=O)(C1=CCCN(C(=O)Cn2ncccc2=O)C1)Nc1c(C)nn(C)c1 c1(OC)ccc(C(=O)NC2CCCC(NC(=O)CNS(=O)(=O)C3CC3)C2)cc1O c1(CC(=O)NC2CCN(C(c3cnn[nH]3)=O)CC2)csc2c(F)cccc12 c1(C(=O)Nc2cccc(Cl)c2CO)c(F)ccc(Br)c1Cl C(=O)(C1=NNC(C(F)(F)F)C1)NCC1OCCN(C(c2ccc(N)cn2)=O)C1 c1(NC(C2CN(Cc3ncccc3F)CCN2)=O)cnc2cc(Br)ccc2c1 Cc1ncnc(C(N2C(C(=O)N(C)Cc3ccco3)CC2C)=O)c1C C1(C(=O)NCC(C)N(C(c2cc(CC)no2)=O)C)CCCCNC1=O CC1(C)CCC=C(C(=O)NC(CNC(C2CC(F)C2)=O)CO)C1 N1(C(c2c(C(C)C)[nH]cc2)=O)C2CCC1C(F)C(NC(=O)COC1CCCC1)C2 C1(NC(C(C)SC(C)C)=O)CCCCC1NC(c1ccc(-c2nc[nH]n2)cc1)=O C1(OC)CCN(C(C2(C)CCN(C(c3ccc(O)cc3)=O)C2)=O)CC1 c1(C(=O)NC2C(CO)CCN(C(CN(C)CCO)=O)C2)cc2cc(Cl)ccc2o1 CC(C(=O)N(C1CC2CCC(C1)N2C(c1cc2sccc2[nH]1)=O)C)C1=CCCC1 C=CCC(C)C(=O)NC(CNC(=O)Cc1ccc(CC)cc1)CC(C)C c1(-n2cc(CN(C(=O)Cc3ccccc3)C(C)C)nn2)ccc(C(C)(C)C)cc1 C(c1ccc(C)c(C)c1)=CC(=O)NCC(CC=C)NC(c1nn(CC)nc1C)=O N1(C(c2c(C(C)C)ccs2)=O)CC2(C)CC1C2NC(=O)C=CC(F)(F)F Cc1cn2ccc(C(=O)NC3CCCC3CNC(=O)CCOC(C)C)cc2n1 CCCCC(CC)CC(=O)NC12COCC1CN(C(c1csnc1OC)=O)C2 CN1CCCCC1C(=O)NC(C)(CNC(=O)C=CC1CCOC1)C1CC1 C(C(CC(C)C)C(=O)N1CC(F)(F)CCC1C)NC(c1cn(CC)nn1)=O N1(C(C(CC2CC2)OC)=O)CC(NC(c2c[nH]c3ncccc23)=O)C2(CCC2)C1 c1(OCC)cc(CC(=O)NC2(CNC(=O)CCc3ccsc3)CC2)ccc1C CCC(CNC(=O)C(C)NC(=O)C(C)(C)C)(CC)NC(C1(C)CC=CCO1)=O N1(C(C(C)CC(=O)c2cccc(Br)c2)=O)CCCC2(C)COCC12 c1(CNC(C2CCN(C(C(C)=C(CC)C)=O)C2)=O)oc(C)nc1C c1(C(COC(=O)C(F)(F)F)=O)cccc(Cl)c1N.CC1C(=O)N1 c1(NCC2N(C(=O)COc3ccncc3)CCCC2)ccc([N+](=O)[O-])cc1 c1(OC)ccc(C(C)NCC(CNC(=O)NC(C)(C)C)CC2CC2)cc1 C1(C(=O)NC2CC=CC2)(CNC(c2ccnn2CCF)=O)CCCO1 C12(C(=O)NC3C4CN(C(C(C)NC(C)=O)=O)CC43)CC3CC(C(=O)N1)C2C3 N1(C(C2N(C(CC)=O)CSC2)=O)CC(NC(c2ccc(C3CC3)s2)=O)C2(CC2)C1 C1(c2nc(COCCCOC)on2)CCN(C2CC(c3ccccc3)C2)CC1 c1(C(=O)NC(CNC(C=CCCC)=O)C(C)(C)C)c(CC)nc2sc(C)cn12 C1(CNC(CC(C)OC)=O)CN(C(c2ccnc(F)c2N)=O)CC(C)(C)O1 C(c1cc2ccccc2n1C)=CC(N1C(C)C(NC(=O)Cc2cnc[nH]2)CC1)=O C(=O)(C(O)C(C)(C)C)NCCCN(CCCCNC(c1cnnc(O)c1)=O)C C1(C(N2CCC(COC(C)=O)C2)=O)CC1C1CN(C(=O)Cc2nocc2C)C1 c1(C(=O)NCC2CC(F)(CNC(CC(C)SC)=O)C2)ccc2ccncc2n1 CC(CC(=O)NC1CC(O)(Cn2cc(CC3CCCCC3)nn2)C1)C(C)(C)C n1(CC)ncc(Cl)c1C(N1CCOC(CNC(C2(C)COC(=O)C2)=O)C1)=O c1(C(N2CC(N(C(=O)Cn3cnc(C#N)n3)C)C2)=O)nc(O)nc(O)c1N C1(n2cc(C3N(C)CCC3)nn2)(C(=O)NCC(F)(Br)Br)CCCCC1 c1(C(=O)NC(CN(C(c2cnc(O)c(F)c2)=O)CC)C)c(F)c(C)cc(N)c1F Cc1cccc(C=CC(=O)NCC2CC2CNC(c2nccnc2C(N)=O)=O)c1 c1(C(=O)NCCCCN(C(C2C=CC(C(=O)OC)C2)=O)C)cc(C)c(Br)o1 Cc1ccc(C(N2CC(CNC(c3cnncc3C)=O)CC2C)=O)c(Br)c1 C(C1(O)CCc2cc(F)ccc21)NC(C(=O)N(CCC(C)(C)C)C)=O C(=O)(CC(CCCC)NC(=O)Cn1cccc1)N(CC(CCCC)CC)C N1(C(C(C)(C)C2CC2)=O)CCCC2(C1)CN(C(=O)CC1CCOC1)CCO2 CC1(C)CCN(C(C23CCC(CC2)C3)=O)CC1NC(c1cccc2ccsc12)=O C1(C2CCCN(C(=O)Cn3ccnn3)C2)(NC(C(C)Cc2ccccc2)=O)CC1 c1(C(=O)NC(CC)CN(C(=O)CC2CCC(=O)N2CC)C)ncnc2sccc12 CC1CC(C(N2CCC(Br)C2)=O)N(C(=O)COCCSc2ccccc2)C1 c1(C(=O)NCC(C)N(C(=O)C(C)C2(O)CCC2)C)ccn(CC(F)F)c(=O)c1 C(CCCCCN(C(=O)Cc1csc(N(C)CC)n1)C)NC(CN(CC)CC)=O N1(C(c2n(CCOC)ncc2)=O)CC2CC(C1)CN(C(=O)C(O)CC(C)C)C2 C1(CC(=O)NC2C(C)=NNC2=O)CC(C)(C)CN1C(c1cnn(C(C)C)c1)=O c1(CC(C)NCc2cccc(OC(C(=O)OC)C)c2)cc2ccccc2s1 CN1C(=O)CCC1(C)CNC(c1nnnn1CC1CC1)(C)CC1CC=CCC1 c1(COC)nc(N2CCN(C(C3(C)CC4CCC3C4)=O)CC2)cc(O)n1 N1(C(CNC(c2cccnc2)=O)=O)CC(NC(C2C(F)(F)C23CC3)=O)C(C(F)F)C1 c1(OC)cccc(C(=O)NCCC(O)CNC(=O)CCC(=O)N2CCCC2)c1 N1(C(=O)OC(C)(C)C)CCCC1(C(F)(F)F)CNc1cnc(F)cn1 C1(CC)(CC)CN(c2nnnn2CC2OC(=O)CC2(C)C)CCS1=O.N(C)C C1(NC(c2cc(OC)n[nH]2)=O)CN(C(C23CC(C)C2C3)=O)CC2(CCC2)C1 C(CCCOC)(C(=O)NCc1cccc(Cl)n1)NC(C(C)OCC#C)=O C1(C2(O)CCC2)(C(=O)NCCCCC(=O)NCC(=O)NCC(F)F)CC1 N1(N(C(F)(F)C(F)(F)F)C2(c3onc(N(C(C)=O)CC)n3)CC2)CCCC1COC C1(NC(CC2(OC)CC2)=O)CC2CCC1CC2NC(C1CCCC(F)C1)=O c1(C(N2CCCC(CNC(C(CC#C)C)=O)C2)=O)n[nH]c2ccc(F)cc12 CC(O)C(C(=O)N1CCCCC1C1CC1)NC(N)=O.C12CC(C1)N2 Cc1cc(C)nc(-c2cn(CCCC(=O)N(C)CC3CCOC3C)nn2)n1 C1(CNC(c2c(C)cno2)=O)CC(C)N(C(=O)COc2ccc(C(C)C)cc2)C1 c1(C(=O)NC2C(NC(CCOCC)=O)C2)cccc(NC(C2CCOCC2)=O)n1 C(C(N=c1nc(C2CCCC2)[nH]s1)C1CCC1)NC(=O)Cc1ccc(Cl)cc1 C1(C(=O)NC(CNC(CCCNC(=O)OC)=O)C)CCCCC(=O)N1 N1(C(C(CCC)CNC(C2CC(C(C)C)C2)=O)=O)CCCC2(CCC2)C1 C(C1=NOC2CN(C(C3(F)CCCC3)=O)CC12)NC(c1cccc(CO)c1)=O c1(C(N(CCNC(c2c(C)cncc2)=O)C)=O)coc2c(F)cc(Cl)cc12 N1(C(CCCOCC=C)=O)CC(OC)CC1C(=O)NC(CN(C)C)CCO c1(C(N2CC(CNC(C=C3CCN(C)C3)=O)C2)=O)ccc2cc(Cl)ccc2n1 c1(C(N2CC(O)(CNC(c3cc(SCC)ncc3)=O)C2)=O)[nH]cc2c1CCCC2 C1(C(=O)NCCC2(C)CCOCC2)CCCCCN1C(C1CCS1(=O)=O)=O N1(C(c2cc(COC)no2)=O)CC(CNC(c2c[nH]nc2OC)=O)C(O)C1 C1(C)(CN(C=O)Cc2c(C)c(Cl)c(Cl)cc2)CCOC2(CCC2)C1 c1(C(N(C(CN(C(CC(C)OC)=O)C)C)C)=O)[nH]cc(C(C)=O)c1C C1(NC(C(CC)OCC)=O)CC(F)CN(C(=O)C(C)(C)n2ccc(C)n2)C1 Cc1cc(C(=O)NCCCN(CC(=O)N(C)C2CC2)Cc2ccccc2)sc1C c1(C(=O)OC(c2cc(C)sc2C)C)ccc(Br)cc1F N1(C(c2ccc(NC)cc2Cl)=O)CC2(CCCN(C(C3CCCC(F)C3)=O)C2)C1 C#Cc1cccc(C(=O)NC2CCC(C(=O)Nc3cnc(C)c(C)n3)C2)c1 Nc1cc2[nH]cnc2cc1C(N1CCOC(CCNC(c2ccns2)=O)C1)=O C(CC(=O)N1CCC1CNC(c1ccc(CN=[N+]=[N-])cc1)=O)(C(N)=O)NC(C)=O C(=O)(C(C)(C)C(F)(F)F)N1CCC(CN(C(=O)CS(=O)(=O)NC2CC2)C)C1 C(=O)(C#CC1CCOC1)NCC1C(C)CN(C(=O)C2=NOC(C(C)(C)C)C2)C1 CCC(C)(CO)C(=O)N1CCCC1Cc1cn(CCN2CCCC2C(=O)O)nn1 C1(C(=O)NCCOCCNC(c2c(C(N)=O)cccc2)=O)CCC12CCCO2 C1(=CCNC(C2(c3n(C)ncc3)CC2)=O)CCN(C(=O)C=Cc2cc[nH]n2)CC1 N1(C(=O)CSCc2ncc[nH]2)CCN(C2COCC2NC(=O)CCCF)CC1 c1(CCC(=O)NCCCN(C(c2ncsc2C)=O)CC)ccc(F)nc1 c1(NC(C2CCCN(C(C3(C(=O)OC)CC3)=O)C2)=O)ccc(F)c(F)c1Cl c1(-c2nnc(N3C(c4cc(C)no4)CCC3)s2)ccc(C#N)cc1 N1(C(Cc2c(C)nn(C)c2C)=O)CCCC2CN(C(C3(C)CCCCO3)=O)CC12 N1(CC(=O)NCC(CCOC)O)CCN(C(=O)C(C)O)CC1 c1(C(N(CCC(=O)NCC2CC23CC3(F)F)CC)=O)nccc2[nH]ccc12 c1(C(=O)NCC(CN(C(C(CN(C)C)O)=O)C)O)sc(F)cc1Cl N1(C(C=CCC)=O)CCN(CC(C)(C)NC(=O)Cc2cc(COC)on2)CC1 CC(C)CC(CO)NC(c1cc(CNC(C2CC(C)(C)CO2)=O)ccn1)=O N1(C(C(C2CCCN2C(=O)CC2CC2C2CC2)C)=O)CCN(C2CC2)CC1 N1(C(Cc2nc(C(C)OC)sc2)=O)CCN(C(c2cc(C(C)C)on2)=O)CC1C C(=O)(C(C)N=[N+]=[N-])NC1CCN(C)C1.CC1C(=O)NCCN1C1CC1 CCCCCCCCNC(C1CCN(C(=O)CCP(C)(C)=O)C1CC)=O c1(C(=O)Nc2cnn(CCO)c2)cccc(-c2cccnc2N2CCOCC2)c1 N1(C(c2c(C)cn(C)c2)=O)CC=C(C(=O)NCC2(C)NC(=O)NC2=O)C1 C1(C(=O)NCC(C)(O)CNC(=O)CCc2cc[nH]n2)CSC2(C)CCC(=O)N12 C(C(CC(C)C)NC(=O)CC1CN(C)C1)NC(COC(CC)(C)C)=O N1(C(c2cc(C#C)c(C)cc2)=O)CCCC12CCN(C(=O)CC(O)C(C)C)C2 c1(C(=O)NC(C2CCCN2C(=O)Cc2cn[nH]c2)C)ccccc1C#N c1(C(N(C2CCN(C(=O)C(O)CCS(C)=O)CC2)C)=O)nnn2c1CSCC2 c1(C(N(C2CC(C(=O)NCCN(CCOC)C)C2)C)=O)cncnc1C N1(C(c2c(CC)cno2)=O)CC2CCN(C(=O)Cn3cc(S(N)(=O)=O)cn3)C2C1 c1(OC)ccnc(C(=O)NCC2(O)CC(NC(c3ncnc(O)c3F)=O)C2)c1F N1(C(CCCC)=O)CCN(C(=O)C(c2cccnc2)O)CC1c1cccc(F)c1 CCS(=O)c1ccccc1C(=O)NCC(C)CNC(=O)Cc1nnc(S)n1C C1(NC(c2c(C)n[nH]c2C)=O)CCN(C(C23CCC2C3)=O)C12CC2 N1(C(CCOCCOC)=O)CC(C)(NC(=O)CC2CCOC2)C1 c1(C(N(CCN(C(=O)CCC2CCC2)C(C)C)C)=O)cc2cccc(Br)n2c1 C1(C(N2CCCC2CCNC(C2(F)CC2)=O)=O)CC2CCC1CC21OCCO1 c1(CC2C(C(=O)OCC(C3(C)CC3(F)F)=O)CCC2)ccc(F)cc1 N1(C(c2cc(C)c(Br)cc2)=O)CC(NC(=O)C=Cc2cc[nH]n2)CC2(CC2)C1 c1(C(N2CC(C)C(CNC(=O)CSC(C)(C)C)C2)=O)cc2c(ncn2C)s1 c1(CN2CCC3CN(C(C(C)(C)F)=O)CC3C2)nccc2cc(Cl)ccc12 C1(C(N(C(C)C(=O)OC)CCC)=O)CC2CCC(C1)N2C(c1cnc(C)c(C)c1)=O N1(c2ccc(S(=O)(=O)N3CCC(F)(F)CC3)nc2)CCc2cc(F)cc(Cl)c2C1 C1(NC(C(N2CCC(O)CC2)C)=O)CN(C(C2C3CC4C(C3)C24)=O)CC1O C1(CNC(C(C)C2CC2)=O)CCCCN1C(C1CCC(CN2CCCC2)O1)=O CC1CC2(CC2)CN1Cc1cc(C(F)(F)F)ccc1-c1sccc1C#N C#CCCC(O)C(=O)NCC=CCNC(c1nc(C)ccc1Br)=O C1(NC(c2cnc(C)n2C)=O)COC2(C1)CN(C(C1CCCN1C1CC1)=O)C2 CC1(CNC(c2csc(C(F)F)c2)=O)CC(NC(C2(C3CC3)CC2)=O)C1 C1(O)(C(C(=O)NC(CNC(c2cscc2F)=O)CO)(F)F)CCCCC1 n1(CC)nnc(CNC(=O)CN(C(C2CCCC2OC)=O)CC)n1 C(N=c1[nH]c(=NCC2(C3CC3)CC2)c2ccccc2[nH]1)c1nc(N(C)C)sc1 c1(C(=O)NCCN(CCC)C(c2cscc2Cl)=O)ccc(NCC)cc1 O=C1OCc2cc(NC(=O)CC3(NC(c4ccc(O)nc4Cl)=O)CCC3)ccc21 C(=O)(C(CC)(CC)CO)NC(CCOCC)C(=O)NCc1cncc(C#N)c1 C1(C(N2C(C(C)C)CC2)=O)(C(C)C)CCCN1C(=O)Cn1cccc1 C(CCCCC(=O)NC1CCC1N(C)C)N(C(c1nncc(NC)c1)=O)C Cc1cc(Cl)cc(C(=O)NC(CNC(C2CC(C(C)C)=NO2)=O)C(C)(C)C)c1N C1(C(N2CC(C)(NC(=O)Cc3cccc(C#N)n3)C2)=O)CCn2ncnc2C1 c1(N(CCCNC(C(Cc2c(C)n[nH]c2C)C)=O)C(C)C)ncnc2onc(C)c12 Cc1ncnc(C)c1OCC(=O)NCCC(C)NC(C1NC(=O)OC1(C)C)=O N1(C(C(C)=C(CC)C)=O)CCC(CNC(c2ccc(C(C)O)cc2)=O)(COC)C1 c1(CC)nc(C)c(C(C)N(C(c2cncn2C)C(=O)NCC(C)C)C)s1 c1(OC)ncnc(C)c1C(=O)Nc1cncc(N(C(=O)OC(C)(C)C)C2CC2)c1 c1(C(=O)NC2(CNC(C3C(C)OC(C)C3)=O)CC2)cc(N)cc2c1OCCO2 N1(CCC)CCC(NC(=O)NC(C)CN(c2ccccc2)C)CC1 C1(O)(CCNC(CN(C(COC)=O)C)=O)CCN(C(=O)Cc2cn(C)nc2C)C1 c1(C(=O)NC(CNC(C2N(CCCC)CCCC2)=O)C)c(Cl)nc2ccccn12 N1(C(C2(OC)CCCOC2)=O)CC2CCC(C1)N2C(c1scnc1C(F)F)=O c1(C(N(CCNC(=O)C(CCO)N(C)C)CC)=O)ccnc2[nH]cnc12 c1(C(=O)NC2CN(C(c3c(C)nccn3)=O)C(C)C2)cncc2nc[nH]c12 c1(NC(Cn2ncc(CC)c2)=O)ccc(NC(c2nc(Cl)sc2C)=O)c(C)c1 C(=O)(CCC(=O)NCCC(C(C)C)NC(N)=O)N(CCC)CCC.C(=O)(CC(C)F)N c1(NC(N2C(c3cn(CCCOC)nc3)CCC2)=O)sc(C)cc1C C1(CNC(C2CCN(C)CC2)=O)(NC(c2cnn[nH]2)=O)CCC(F)(F)CC1 C(=O)(C1=CS(=O)CCC1)N1CC(NC(C(C(C)C)SC)=O)(CO)C1.c1(N)ccccc1 N1(CC(C)C)CCC(C(N2CCOCC2CNC(C2CC3C=CC2O3)=O)=O)CC1 C(N=c1nnc(O)c(C)[nH]1)C1CCN(c2cccc(OC)c2)C1 c1(CC(=O)NC(CNC(c2ccn3cnnc3c2)=O)CO)ccc2c(c1)CCC2 N1(C(C2C(C(=O)OC)C2)=O)CCC(C2CC2NC(C2(CC(F)F)CCC2)=O)CC1 C(=O)(C1=CCCOCC1)N1CCC(CNC(C(c2cncn2C)OC)=O)(OC)C1 C1(NC(C(C2CC2)OCC)=O)CC1C1CCCN(C(=O)C2=CCCCC2)C1 c1(OCC)nc(C)cc(C)c1CN(C(=O)C(C(C)(C)C)n1c(C)cccc1=O)C C1(NC(=NCCCC)NCCc2cccc(OC)n2)CCC2(CCOCC2)CC1 c1(NC(C(CC)Br)=O)ccc(C2CCCN(Cc3n[nH]cc3Cl)C2)cc1 C(CC(C)(C)NC(=O)CCC1CCC(NC(=O)CCc2cnn[nH]2)C1)N(C)C O=C1CCC(C(F)C(=O)NCC2CC2NC(C2(N3CCOC3=O)CC2)=O)CC1 C1(C(=O)NC2(CCC(=O)N(CCOCC)CC)CCC2)OCCOC1C N1(C(C(C)OCC)=O)CCC(CCNC(=O)CN2CCC(OC)CC2)(OC)CC1 n1(CC(=O)NCC(CNC(c2ncoc2-c2ccco2)=O)OC)cnnc1O c1(NC(C2CN(C(c3c(OC)csc3)=O)C2)=O)cc(C)c(Br)cc1F c1(C(N2CC(OCCOCC)C2)=O)nc2ccccc2nc1C C1(C(COC(c2ncncc2Cl)=O)=O)CSc2ccccc2O1 c1(OCC(=O)NC(CNC(C(C)OC)=O)CO)ccccc1Cc1ccccc1 c1(OCC)ccc(CN2CCCC(O)(CNC(C)=O)C2)cc1[N+](=O)[O-] c1(CC(=O)NC2C(CNC(COCc3scc(CC)n3)=O)CC2)ccc(C)cc1 C1(C)(CC(N2C(C)(CCC)CC2)=O)CCN(C(=O)CN2CCOC2=O)C1 n1(CC(=O)NC(CCCNC(C(C)NC(CC)=O)=O)C)cnc2c1CCCC2 C(C)(CNC(=O)C(C)=C(C)C)(CNC(=O)CCC1(C)CC1(F)F)OC C1(C(N(CC(=O)NCCc2cnccn2)C2CCC2)=O)CC2(CC2)C1 N1(Cc2c(C)nn(C)c2)CCCC(NC(c2ccc(Cl)c(Cl)c2)=O)CC1 c1(C(N2CC(CNC(C3(CS(C)(=O)=O)CCC3)=O)C2)=O)cnc(O)s1 c1(NC(C23C(CN(C(c4cc5sccc5s4)=O)C2)C3)=O)nc(Cl)ccc1[N+](=O)[O-] C1(O)(CCNC(C2(C)COC2)=O)CCN(C(=O)C(C)(C)C2CCOCC2)C1 c1(C(=O)NC(C(=O)OCC)CC2CC2)ccc(I)c(N)c1 C1(CC(C)C)(C(=O)NC2CCCN2CCOC(C)(C)C)CCOCC1 Cc1cccc2cc(C(=O)NCCC(C)NC(C3(C(C)C)CCCO3)=O)oc12 CC1CCCN(C(=O)C=CC(=O)N(C)C)C1CCNC(=O)COC1CCCOC1 c1(C(N2CCC(C)(NC(Cc3c(C)noc3)=O)C2)=O)ccc2nonc2c1 CCS(=O)(=O)CC(=O)N1CCC1C(N1CCOC(C)CC1)=O N1(C(C2CC(C)CN(C(=O)C(C3CC3)C3CC3)C2)=O)C2CCC1CC(F)C2 C=Cc1ccc(C(=O)N(C2CCC(NC(=O)CN3CCCCC3)CC2)C)cc1 CC1(CO)CN(C(C23CC(NCc4cccnc4F)(C2)C3)=O)CCC1O N1(C(C2N(C(C)=O)CSC2)=O)CCC(NC(=O)CC(F)(F)F)C(F)(F)CC1 C(=O)(C1c2ccccc2C2CC1C2)N1CC(NC(=O)C=Cc2ccco2)C2C1C2 N1(C(CN(C(COC)=O)C)=O)CCCCCC1CNC(=O)C(O)C(C)C C1(NC(c2cccc3nonc23)=O)CN(C(c2cc[nH]c2)=O)CC1C1CC1 C1(F)(C(=O)NCCC(C)NC(=O)CC2CCOC2C)C(C)(C)C1(C)C N1(C(c2c(C)nco2)=O)CCC2CCCC12CNC(c1cc(C)n(C)c1)=O N1(C(CCOCC)=O)CC(NC(=O)C(C)(C)CN2CCN(C)CC2)C(C)C1 N1(C(C(C)OCC2CC2)=O)CC2CC2(CNC(=O)C(c2ccc(Cl)s2)=O)C1 c1(OCC=C)ccc(Cl)c(C(=O)NCC23CC2CN(C(=O)C=CCO)C3)n1 c1(NC(=O)N(C2CN(C(c3ccoc3)=O)C2)C2CC2)ccccc1C(F)(F)F C1(C(=O)NCCC2(OC)CCC2)CC2CC2N1C(=O)CCc1ccsc1 CCC(C)C(C)C(=O)NCC1(C(=O)NC23CC(C)(C2)C3)CCCO1 C1(NC(C2(C#C)CCC2)=O)CCC(C)(CNC(C23CC(F)(C2)C3)=O)C1 C1(C2CCN(C(c3cccc4sccc34)=O)C2)(NC(CC=CC=C)=O)CC1 C(=O)(CC(C)(C)CC(=O)NCCN(C(=O)Cn1ccc(Br)n1)C)OCC C=CCC(C)C(=O)NC1CC(C(C)NC(C2CCCC2(C)C)=O)C1 C1(c2ccccc2)(CN)CCC(O)CC1.C1(CNC)CCCN(C)C1c1ccnn1C C(=O)(C1=C(C#N)CCC1)NC(CC)CNC(=O)C(C)CNC(C1CCCC1)=O c1(C(=O)NCCN(C(C)C)CC)cnn(C)c1O CN1C(=O)C(=O)N(CC(=O)NC2CCN(C(C3CCCOC3)=O)C23CC3)C1=O CCC(C)(C(=O)NC1CCN(C(=O)Cc2cccc(OC)c2)C1C)C(N)=O C=CCC(C(=O)NCCc1n[nH]c(C)n1)NC(=O)C(O)C(C)C CCCC(O)CC(=O)NCCC(C)N(C(=O)CCCNC(c1ccccc1)=O)C c1(C(N2CCCC2c2cn(-c3cccnc3F)nn2)=O)cc(F)cc(Br)c1Cl C1(NC(C(C=CCCC)O)=O)CCCN(C(=O)CSc2nncs2)CCC1 C(=O)(C(CCOC)OC)N(CCOC)C.O(NC=O)CC.C12CC1NC2=O C1(CN(C(=O)C(O)CC2CCCC2)C)CCCN1C(c1csc(Br)c1)=O C1(CNC(CN(C)CC)=O)CCN(C(c2c(NC(=O)OC)c[nH]c2C)=O)CC1O N1(C(C(C(C)C)(C)C)=O)CC(C)OC2(CCN(C(c3n[nH]c4c3CCC4)=O)C2)C1 CON(CCC(=O)NCC1(C)CC(C)=NO1)C(=O)CC(C)F c1(OC(C(N2CCCC(c3nc(C)c(C)s3)C2)=O)(C)C)cc(F)cc(F)c1 C12(N(C)C)CC3CC(C1C3)CN2.C(CCCS(C)(=O)=O)NC1CN(CC)C(=O)C1 C1(OCC)CN(C(=O)C=CCN(C)C)CC1NC(c1[nH]ccc1C1CC1)=O C1(C2CN(C(=O)C(C)O)C2)(NC(C(C)CC2CCC2)=O)CC1 C1(CN(C(c2c(OC)scc2)C(=O)NC2CC2)C)CCCC1(C)C C(=O)(CCC(C)(C)C#N)NCCC1CN(C(C2(CC(C)C)CCC2)=O)C1 N1(C(C(C)=CC)=O)CCCC(C2CN(C(=O)CCn3cc(Br)c(C)n3)C2)C1 Cc1cc(C(=O)NCCN(C(=O)C2=CCCC2C)C2CC2)c2[nH]cnc2c1 C1(OC)CCCC(NCc2ccc(-n3cccn3)cc2Cl)CC1 c1(C(=O)NCCCCC(C)NC(c2cc(Cl)nnc2O)=O)ccc(F)c(F)c1F C1(OC)C(C)(C)C(OC(=O)CCn2ccc(C(F)(F)F)n2)C1(C)C.C(C[Si](C)(C)C)O N1(C(C=C(C)C2CC2)=O)CC(C)(C)C(NC(=O)C(C(C)C)C(C)C)C(C)(C)C1 N1(C(C(C)SC)=O)CCN(C(=O)Cn2ncc(Br)c2C)C(CF)C1 CC1CN(C)CC1C(=O)NCC1(F)CC(NC(c2cc(O)nn2C)=O)C1 CC(=O)CC(C)(C)CC(=O)N1CC2CC(C1)N(C(c1nc3ccccn3n1)=O)C2 N1(C(CC(CCC)(C)O)=O)CCC(Nc2nc3cccc(Br)c3o2)C2(CCC2)C1 C(=O)(C#CC1(C)CCCO1)N1CC(CCOC)N(C(=O)C=CC(C)(C)C)CC1 Cc1c(C(=O)NC2CCC(NC(c3csnc3Cl)=O)CC2)nnn1C N1(C(CC2CC(C(C)(C)C)C2)=O)CCC(O)C(NC(C2(C)C=CCC2)=O)C1 c1(C(CCC)=O)cc(C(F)(F)F)ccc1F.C12C(C1C(=O)OCC)C(=O)OC2=O c1(C(=O)NC2(CCNC(C(CC)(CC)OC)=O)CC2)cc(OC)c(OC)cc1F CN1CC(C)(C(=O)NCC2(CNC(c3csnn3)=O)CC23CCC3)CC1=O c1(C(=O)NCCN(C(CCN(CCC)C)=O)C)cc(CN(C)C)on1 c1(C(N2CC3(C(NC(c4c(CC)con4)=O)CC3)C2)=O)cc(Cl)c(F)cc1O C(C(=O)N1CC(C)(C(F)C(=O)NC2CC(=O)N(CC)C2)C1)(C(C)C)OCC C(CC(C(=O)N1CCC1C(=O)OC)NC(=O)CC(C)(C)C)OC N1(C(C2C(=C)CC2)=O)C2CC1CN(C(c1cc(OC)cc(F)c1)=O)C2 C12(NC(=O)CN3C(=O)CNC3=O)CCN(C(c3ccncc3Br)=O)CCC1C2 CC(C)CCN=C(NCCn1cccn1)N1CCCC(CCC(C)C)C1 Cc1nc(CN2CC(C=CC3CCCO3)C2)sc1C(=O)O N1(C(C2C(C(C)NC(c3ccc[nH]3)=O)C2)=O)CC2CC3CC2C1C3 c1(OC)c(C(=O)NCC2(C)CCN(C(=O)Cn3cc(Cl)cn3)C2)csc1C C1(C)(C(=O)NC(c2cncc(F)c2)C)CCCN1C(c1cc[nH]c(=N)n1)=O c1(C(=O)NCCCC2(NC(=O)CNC3C(C)OCCC3)CC2)cccc([N+](=O)[O-])c1 c1(C(=O)NCC23CC2CN(C(C2CC2C2CC2)=O)C3)cccc(F)c1C(F)(F)F O=C(CCCCC(F)(F)F)NCC1CCN1C(c1cccn1C1CCCC1)=O C1(C(=O)NC2(C=C)CCC2)CCN(C(=O)C(C(C)(C)C)OC)O1 c1(CNC(=O)NCC(c2cccc(OC)c2)O)cccc2c1OCCCO2 Cc1ccc(CNC(=O)C(c2ccccc2)N2CCCC2)c(O)n1 c1(CNC(C(C2CC2)OCC)=O)cc(C(=O)NC2CCCC2)co1 c1(C(N2CC3C(CNC(c4ccncc4Br)=O)(C3)C2)=O)cc(F)cc(F)c1Br c1(OC)cccc(C(=O)NCC(C2CCCC2)NC(=O)C=CC2CCOC2)c1N CC(CN(C)C)CC(=O)N(C1CN(C(=O)CC(Cl)Cl)CC1O)C N1(C(=O)COc2cccc(CO)c2)CCOCC(CNC(C2CCC(O)C2)=O)C1 c1(C(=O)OC)cc(NC(c2ccc(CO)cn2)c2nnnn2C(C)C)ccc1C N1(C(CCC#N)=O)CC(F)CC1C(c1ccccn1)NC(=O)CCCCC1CCSS1 Cc1ccc(C(=O)CCC(=O)N2CC3C(CNC(=O)CCC(C)C)C3C2)cc1 Cc1nn(C)c(C)c1C(C)C(N1CCCC1CN(C(=O)Cc1cnnn1C)C)=O c1(C(=O)NC(C(=O)N(CCC)CCC)C2CCOC2)cccc(F)c1 C1(OC)CC2(C(=O)N(CCC(C)NC(c3cccn3C(C)C)=O)C)CC12 c1(CC=C)ccccc1C(=O)NCC12CC(CNC(=O)CCC(C)OC)(CO1)C2 C1(C#N)(C(=O)NCC(C2CC2)NC(C(=Cc2cnc[nH]2)C)=O)CC2CC2C1 N(C)(S(=O)(=O)N(C)C)CC(=O)N(C)CC1CN(C(C(C2CC(F)(F)C2)OC)=O)C1 C1(C(CC(C)(C)C)NC(C23COC(CF)(C2)C3)C)CCS(=O)(=O)CC1 c1(C(=O)NCC2CC(NC(c3c[nH]c(=N)o3)=O)C2)cccc(Cl)c1Br Cc1ccc(C(C)(C)C(=O)NC2CC(CNC(C3CCCS3)=O)CC2O)cc1 C(=O)(C(C)CC(C)C)N1CCC(C(C)NC(CCN(CCCCC)C)=O)CC1 Cc1ccc(CNC(=O)C(=O)NCc2ccc(O)cc2F)c(F)c1F C1(CC)(NC(c2cccc(N)n2)=O)CCCN(C(=O)C(CC)c2ccccc2)C1 C(=O)(CCS(C)(=O)=O)N1CC2C(CNC(C(c3cccc(C)c3)F)=O)C2C1 CC(C)C(CNC(c1cccn1Cc1ccccn1)=O)NC(=O)CC(C)F c1(C(N2CCN(C(CC(C=C)C)=O)C(C(C)C)C2)=O)c[nH]c2cc(Cl)ccc12 C1(NC(C)=O)CN(C(c2ccnc(OCc3ccccc3F)c2)=O)CC12CCC2 C1(C(=O)OC)CCCN1NC(=O)CNC(C1CCSCC1)=O C(N=C(NC1CC1)N1CCOC(C2CC2)C1)c1ccc(SC)cc1 c1(NC(CC2C(CNC(CN(CCC)C)=O)C2)=O)cncc(CC)c1 C1(C(N(C(C)C)Cc2cccc(Br)c2)=O)CCCN(C(=O)C(=O)N(C)C)CC1 N1(C(CC2(CNC(c3ccnnc3)=O)CC2)=O)CC2CCC(CO)(C2)C1 c1(C(N(CCN(C(CCN(CCC)C)=O)CC)CC)=O)cccc(C)c1 C#Cc1c[nH]nc1C(=O)N(C1CCCN(C(C2CCSC2)=O)C1)C C1(NC(CC(C)n2cccn2)=O)CCC2(CC1)CCN(C(C1CC(C)(F)C1)=O)C2 Nc1c(-c2noc(C3CCCN3c3nccs3)n2)cnn1CCO N1(C(c2ccc(C#C)o2)=O)CCC(NC(C2C3CN(C)CC23)=O)C2(CCC2)C1 N1(C(c2cccc(-c3ccc(O)nn3)c2)=O)CC2CCC(C(=O)O)(C2)C1 N#CC1CCCCC1NC(C1C2CC1N(C(=O)CCCNC(N)=O)C2)=O C1(O)(N(C(=O)C(=O)NCC(F)(F)F)C)CCN(C(=O)CC(F)(F)F)C1 N1(C(CCC=CC(C)C)=O)CC2CC(NC(=O)Cc3cc(C4CC4)on3)C2C1 N1(C(CC2CC(C)C2)=O)CCN(C(c2ccnn2C)=O)C(CF)C1 c1(C(CC)NC(N2CCCC2CCCc2ccccc2)=O)cc(Cl)cc(Br)c1 Cc1ccc(N2CCCCC2)c(S(=O)(=O)N2CCC(C)(CN3CCCC3C)C2)c1 c1(NC(=O)NCCC(CCNC(C2CN(C(C)=O)C2)=O)C)ccccc1S(C)=O Cc1ccc2c(c1)CCC2C(=O)NCCC1CC1C1CC1 C1(CCNC(Cn2c(C)nnn2)=O)CC(F)(F)CN1C(c1cccc(F)c1O)=O N1(CC(N2CCCC(C(C)=O)C2)=O)CCCNC(=O)C1C c1(C(N2CC(C(C)NC(C=CSC)=O)OCC2)=O)cc(F)c(C)cc1Cl c1(CC(=O)N(C(C)CNC(c2cncnc2)=O)C)ccc2c(c1)CC2 C1(NC(=O)Cc2cnccc2Cl)COCCN(C(=O)CC2CCCCC2(F)F)C1 N1(C(c2n(CC#C)ccc2)=O)CC2(CC(CNC(C3CCCCC34CC4)=O)C2)C1 c1(NC(C2CCN(C(=O)CCc3cncnc3)CC2O)=O)nc(Cl)cnc1Br C1(O)(CNC(CCCCNC(N)=O)=O)CCCN(C(c2cc(O)nc(Cl)c2)=O)C1 c1(CN2C(C(N(CC#C)Cc3ccccc3)=O)CC(F)C2)ccc(Br)c(F)c1 C12(NC(c3ccn(CC)c(=O)c3)=O)CCCC1N(C(=O)CNC(N)=O)CCC2 CCC(CC(=O)NCCCC(=O)Nc1ccc(O)cc1)C(C)C c1(C(N(CCNC(C(=O)N(C)C)=O)C)=O)ccc(O)c2ncccc12 Cn1cnc2c(NCc3nc[nH]n3)nc(N3CC(C)(C)OC4(CCC4)C3)nc12 C1(C(=O)NC(C2CC2Cl)=O)OCCNCC1N(C1CC1)CC S(=O)(=O)(c1c[nH]ccc1=NC1CCN(CC)C1)NC(c1ccc(OC)cc1F)C c1(C(=O)NC2C3CN(C(C4CC5CC4C5)=O)CC23)ccc(F)c(Cl)c1 CC(CCC(=O)N(C)Cc1ccnn1C)NC(=O)COC(C)(C)C C(=O)(CC(C)(C)C(C)(F)F)N1CCCC(C)(NC(c2ccc(=NCC)[nH]c2)=O)C1 C1(C(=O)NCC2(C(N)=O)CN(C(CCC(=O)OC)=O)C2)CCN(S(N)(=O)=O)CC1 Cc1nc(C)n(O)c1C(=O)NCCC1CCCN1C(c1cccc(C2CC2)c1)=O C1(NC(CC=CC=C)=O)CCN(C(=O)C=Cc2cccc(F)c2)CC1CC N1(C(c2c[nH]c(=NC)o2)=O)CC(C(=O)NC2(C)CC3(CC3)C2)CC12CCC2 C(=O)(CC(O)CC(C)(C)C)N1CC(C)(CC(=O)OC)C1.C1(C(C)C)CN1 CC(C)C(O)C(=O)NCCC1CN(C(C2(C)CC2(Cl)Cl)=O)C1 c1(C(=O)NC2C(CC(=O)NCCOC3CCCC3)C(O)C2)cnnc(O)c1 c1(CCNC(C2N(S(CCC)(=O)=O)CCC2)=O)ccc(C(C)=O)cc1[N+](=O)[O-] Cc1cc(=O)c(C(=O)NC2CCC(N(C)C(C3(F)CC3)=O)CC2)c[nH]1 C(=O)(C(C)C1=CCCC1)NCC(C)CNC(=O)CN1CCC(O)CC1 CC1CN(C(=O)CC23CCC2CN(C(=O)C(c2ccccc2)F)C3)C(C)CO1 C1(c2n(-c3ccn(CC(F)F)n3)nc(C3CC34CC4)n2)Cc2ccc(F)cc2O1 N1(C(C2C3N(C(COCC(=C)C)=O)C(CC3)C2)=O)CC2(C1)CC(C)(F)C2 Cc1cn2ccnc(C(=O)NC(C)CCCNC(c3nc(Br)c[nH]3)=O)c2n1 c1(SCC(=O)NCCOCCNC(c2c(CC)nn[nH]2)=O)nc2ccccc2s1 Cc1sc(Br)nc1CC(=O)NC1CCCCC1NC(=O)Cn1ncnn1 N1(C(C(C)n2ccnc2)=O)CCCC1C=CC(=O)NCCSCCO N1(C(c2ccc(OCC)nn2)C(=O)NC)CCC(N(C)OC)CC1 C1(C(N2CCCC(NC(c3c(CC)cno3)=O)C2C)=O)CCc2cn(C)nc2C1 C1(NC(C2CC(=C)C2)=O)CC2CC(NC(c3c(Cl)ccc(F)c3N)=O)CC2C1 C=CC1CCCCN1C(C1(CNC(c2ccco2)=O)CCCCC1)=O C1(C(=O)NC2(C(=O)Nc3cccc(C4CC4)c3)C(C)(C)C2)CCCC(=O)C1 C1(C(=O)NCC(CC)NC(=O)CNC(=O)COC)CCCC(F)C1 Cn1nc(C(=O)NC2CCCC2CNC(=O)C=CC(F)F)cc1Cl c12nnnn1NC(=O)CC2.C1(C(=O)OC)(Cc2cccs2)COC1 c1(C(=O)NC2CC(NC(c3c(CC)cco3)=O)C2)ccc2ncccc2n1 N1(C(CCC(C)N(C)C)=O)CCN(C(c2ccc(C(F)F)o2)=O)C(C)C1 C(=O)(C(F)C(=O)N(C(C)C(=O)NCCCn1cc(C)cn1)C)OCC CCCC(O)CC(=O)N1CCN(C(C2(C(=O)NC3CC3)CCC2)=O)CC1C Cc1sc(Br)nc1NC(c1ccc(Cl)cn1)c1nnnn1CC1CCOC1 N1(C(CC2C(C)C2)=O)CCC2(NC(=O)CNC(C3CCOCC3)=O)CCCCC12 c1(C(N(CC(CNC(CC2CCC(C)CO2)=O)C)C)=O)ccc(N)cc1Br CC1CN(C(=O)CC2CCOC2C)CC1(C)C(=O)NCCC1CC(F)C1 c1(C(=O)NC(c2cn(CC3CCCC3)nn2)CCC)cccc2c1C(=O)NC2=O CC(C)(CCCC(=O)N1CCCC(N=[N+]=[N-])C1)NC(=O)C1=COCC1 C1(C)(C(=O)NC(C2CN(C(c3ccc(CN(C)C)s3)=O)CCO2)C)CCC(F)(F)C1 c1(C(=O)NC2CCCN(C(C3C(OCC)C3)=O)C2C)cccc(S(=O)(=O)CC)c1 C(CC(C(=O)N(C)CC1CN(C)CCO1)NC(c1ccc(O)cn1)=O)OCC C(CC(=O)NC1CCCC(NC(c2c(Br)n[nH]c2C)=O)C1)(C(N)=O)NC(C)=O c1(-c2n(CC(C)Sc3ncccc3-c3ccc(F)cc3)ccn2)ccccc1C#N C(=O)(CCCCCCC(=O)OC)N1C(C)CCC(NC(C(C=C)O)=O)C1 CCCC(C)(O)C(=O)NCC1CCCC1C(=O)NC1CNC(=O)C1 C(=O)(C(C)(C)CS(C)(=O)=O)NCC1(NC(C=Cc2nnn(C)n2)=O)CCC1 c1(C(N(CC(C)NC(C(C)CC(F)(F)F)=O)C)=O)coc2c1NC(=O)CCC2 c1(C(=O)NC(C2CC(F)CN2C(C2CC(=O)C2(C)C)=O)C)cc(C(F)F)n(C)n1 S(=O)(=O)(c1c[nH]c(C(N2CCC(CCNC(C3COC(C)C3)=O)CC2)=O)c1)NC C12(NC(C(C)(C)C)=O)CC1CN(C(=O)C(C)(C)Oc1ccccc1)C2 c1(C(N2CCCC(O)(CN(C(CCCCC#C)=O)C)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C1(C2CCN(C(c3cc(C4CC4)nc(Cl)c3)=O)CC2)(NC(=O)CCC2CC2)CC1 C(=O)(C1=C(C)OCCC1)NCC1N(C(C(CC)CC)=O)CC(C)CC1 c1(C(N(C2CCCN(C(c3c(C)nn[nH]3)=O)C2)C)=O)c(Cl)cncc1Br CCC(F)(F)CC(=O)N(C1CN(C(C2(c3ccccc3)CC2)=O)CC1F)C N1(C(C(c2ccc(C)cc2)N(C)C(=O)OC(C)(C)C)=O)CC(=O)NC(=O)C1 Cc1ccc(OCC(=O)NCC2CC(NC(c3cc(Br)[nH]n3)=O)C2)cc1 c1(CC)cc(NC(=O)C(c2cccs2)NC(C2CCC3(CC3)C2)=O)ccc1C C12(NC(c3ccc(N(C)C)cn3)=O)CC(C1)N(C(=O)COCC1CCCOC1)C2 C1(CNC(C(COCC)n2cc(Cn3cccc3)nn2)=O)CC(C(C)(C)C)=NO1 C(=O)(C1=C(F)CN(C(=O)CC(C)c2ccco2)CC1)N(CC(C)C)CCOC N1(C(CCC2CCN(C(=O)OCC)C2)=O)CC(=O)N(CC2(C)CSCCO2)C1=O N1(C(c2n(C)c(S)nc2)=O)CCC12CN(C(=O)CSc1cn[nH]c1)C2 Cc1cc(NC(c2cc(Br)sc2C)=O)ccc1NC(C1CCCO1)=O C12CC=C(C(=O)N1C)C2.C(CCC(=O)NC)N(C)C c1(C(=O)OCC)ccc(C(N2CCC(NC(=O)CC3CCC(O)C3)C2)=O)cc1F N1(C(C=Cc2cn(C)nn2)=O)CCN(C(C2(CC(F)F)CC2)=O)C2(CCC2)C1 c1(N(CC(C)O)C)cc(C(=O)NCC=CCNC(=O)C(O)C2CCCC2)ccn1 c1(C(N2C(CN=c3nn[nH]n3C)CC(C)(C)C2)=O)cc(F)cc2cccnc12 Cc1cc2c[nH]nc2cc1C(=O)NC1(CNC(c2c(F)ccc(Cl)c2F)=O)CC1 c1(C(=O)NCC(CNC(C(C(=C)C)(C)C)=O)F)cc2ccc(C(C)(C)C)cc2[nH]1 C1(C(=O)OCC(c2ccc(N(C)C)cc2)=O)CN2CC(CCC2=O)O1 Cc1ncc(C(=O)NC(C)(C)CCNC(C2(C)CCCCC2C)=O)cc1Cl N=c1[nH][nH]cc1C(=O)NC1(CCC(=O)NCCc2nccs2)CCC1 N1(C(C=CC(C)C)=O)CCCC1C(C)C(=O)NC(C)CC(=O)NCc1ccccc1 c1(C(=O)NCC2OCCN(C(C=CCN(C)C)=O)C2)cc(O)cc(=O)o1 c1(C(=O)NCCC2N(c3nnc(CC)s3)CCC2)[nH]c2ccc(C)cc2c1C c1(C(=O)NC2(CO)CC2)ccc(F)c(N2CCC2)c1 C(=O)(C1=CCS(=O)(=O)C1)N1CCC(N(C(=O)CC2CC3CC3C2)C)C1 N1(CC(CN(C)CCO)O)CCC(N2CCCC2=O)CC1 c1(CN(C)C(=O)NC(c2ccc(F)cc2F)CF)n[nH]c2ccccc12 Cc1cnn(C)c1C(=O)NCC1(N(C(c2[nH]cnc2C#N)=O)C2CC2)CCCCC1 C(C(C)C(F)C(=O)NOC1CC1)NC(C(C)N(C(C)=O)C)=O c1(OC)cc(C(N2CC(N(C)C(C3CCCC3C)=O)C(O)C2)=O)cnc1OC Cc1ccc(-c2nc(C3CSC3)n(CC3OCCCC3(C)C)n2)cc1F c1(CC(=O)NC2C(NC(c3cnc(C)[nH]3)=O)CCOC2)cccc(C)c1Br N1(C(C(CC2CN(C(C3CC(=C)C3)=O)C2)F)=O)CCCC(C)(C)C1C N1(C(C(C#C)(C)C)=O)CC2CC(NC(c3ccc4c(c3)CC4)=O)C(C2)C1 Cc1sc2ncc(C(=O)NCCN(C(C3CCC4C3C4(F)F)=O)CC3CC3)n2c1C C1(N(C(C(C=CC)O)=O)CC)CCCN(C(=O)C(c2ccccc2SCC)O)C1 C1(CC)CCN(C(c2ccc(C3CC3)o2)=O)C1CNC(=O)Cc1nonc1C c1(NC(CSCC)=O)[nH]c2cc(-c3cccc(C(=O)NCCO)c3)ccc2c1C CCC(CN=c1[nH]c(=NC(C)c2ncc3ccccn23)c2[nH]ccc2[nH]1)N(C)C C(=O)(C1=CCCCC1)N(CCC(N1C(C)CCCC1)=O)CCCO C1(NC(=O)C(N2CCCC2c2cccs2)=O)CCCC2(CC2)C1 C1(NC(=O)NC(C2CS(=O)(=O)C2)C(=O)O)C2Cc3ccc(Br)cc3C12 CC1CCCCN1CC(N1CC(O)CC1C(=O)N(C)Cc1cnccn1)=O C1(C#N)(C(N2CC(OCCC(=O)NCC(C(=O)OC)(C)O)C2)=O)CC12CCC2 C(C1(O)CCCc2ccccc21)NC(C1(CCc2ccccc2)CC1)=O C1(CNC(Cc2cc(C)on2)=O)C2CN(C(C3CC3Cc3ccccc3C)=O)CC12 c1(C(=O)NCC2CN(C(CCCC=C)=O)CC2O)cc2c(C)cccc2o1 C(=O)(CS(N)(=O)=O)NCC1N(C(CN(C)C(c2ccccc2)=O)=O)CC=C1 N1(C(CC(C=C)CC)=O)CCC2CN(C(c3ccc(C(F)(F)F)nc3)=O)CCC12 C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1CCCN(C(C(CCC)(C)O)=O)C1 C(=O)(C(C)CC(F)(F)F)Nc1c(C)cc(C2(O)CCOCC2)cn1 c1(C(=O)NCC2CCCC(NC(=O)CCSC(F)(F)F)C2)ccc2snnc2c1 c1(NC(c2cc(COC)no2)c2nnnn2CCCSC)ccc[n+]([O-])c1 C(CCCCC(=O)N1CC(O)CC1(C)C(=O)NCCC(=O)OC)OCCC CCC(CO)C(=O)NCCCOC1CCN(C(c2ccc(OC)cc2)=O)CC1 c1(C(=O)NC2CN(C(c3n[nH]c(C4CC4)c3Cl)=O)C2)cc2c(cc1O)OCO2 C12CN(CCO1)C2=O.C=CC1(CNC(C2(C(c3ccccc3)=O)CC2)=O)CCC1 c1(N2C(C)CC(NC(C(Br)=C(C)C)=O)C2)nc(C)nc(O)c1C C1(C(C)C)CN(C(C2(Cc3cccnc3)CC2)=O)CCN1C(=O)CN=S(C)(C)=O c1(CC(N)C(=O)NC2CC3CCN(C2)C3)ccc2c[nH]nc2c1 C#CC1(O)CCN(C(C2C3CC4C(C3NC(=O)Cc3cc[nH]c3)C24)=O)CC1 Cn1ncc2cc(C(N3CCC4(CC(NC(C5(O)CC(C)(C)C5)=O)C4)C3)=O)sc12 CCC(C)C(O)CC(=O)NC1CCCC(C(=O)Nc2ccc(CCO)cc2)CC1 c1(C(N2CCC3(C(C(=O)Nc4cncnc4O)C3)C2)=O)c(Cl)ccc([N+](=O)[O-])c1Cl CCC(CC(=O)N(CCC(N1CC2(CCC2)CC1CO)=O)CC)CC(C)C C=CCC(C(=O)NCCOCCCNC(c1cn[nH]c1)=O)c1ccccc1 c1(C(=O)OC)ccc(C(=O)NC2CCCC2NC(C2(C3(C)CC3)CC2)=O)c(C)c1 C1(C(N2C3CC(NC(CC(=O)NCC)=O)CC2CC3)=O)CN(S(=O)(=O)N(C)C)C1 N1(C(C=C(C)Cl)=O)CCCC1CCNC(=O)C(c1ccccc1)C C1(N(C(CCC=C=C)=O)C)CN(C(c2cc(CO)oc2C)=O)CC12CC2 c1(NC(CN(C)CC)=O)c[nH]nc1C(=O)NOC(C)(C)C(=O)OC N=c1nc(N2CCCC(F)(F)CC2)[nH]c(=NCCN2CCCC2)[nH]1 N1(C(C=CC2(C)COC2)=O)CC(F)CC1CNC(C1(CF)CCOCC1)=O c1(OC)ccc(CO)cc1-c1cccc(-c2nn[nH]n2)c1.C12CC1C(=O)N2 N1(C(CSc2n(C)ccn2)=O)CC2(CCN2C(C2CC23CC3)=O)C1 Cc1c(C(F)(F)F)cc(C(=O)NCC(CO)NC(C2CC2(Cl)Cl)=O)cc1N N1(C(C2COCCN(C(c3nncc(OC)c3)=O)C2)=O)CCC(C2(C)CC2)C1 C1(C(=O)NC2(COC)CN(C(C3(C4CC4)CC3)=O)C2)Cc2ccccc2S1 Cc1ccnc(NC(c2cc3n(n2)CCCC3)=O)c1C#N c1(C(C(=O)NC(CN(C(c2cccs2)=O)CC)C)C2CCCC2)cnn(C)c1 Cc1cc(C(=O)NC2CCC(F)(CNC(=O)C(C)(C)C#N)C2)c(F)cc1F S(=O)(=O)(c1cc(C)cnc1NCc1csc(=NC)[nH]1)NCC(CC)CCO c1(NC(C2CCCC(NC(Cn3c(C)ncc3)=O)C2)=O)ccc(O)c(F)c1 CCC(C(=O)NC(C)(C)C(C)NC(=O)CNC(=O)NC1CCOCC1)C(C)C O=C(CC1CC(=O)Nc2ccccc21)NC12CC1CN(C(c1sccc1F)=O)C2 C1(C)(NC(c2n(CC=C)ccc2)=O)CCN(C(=O)CCOC(C)=O)CC1 Cc1ncnc(C)c1NC(C1CCN(C(=O)C2(C)CCCN2C)O1)=O N1(C(C(CCCC)(F)F)=O)C2CC=C(C(=O)NOC3CCC(O)C3O)C1CC2 c1(C(N2C(C)CC(NC(C34CCN(CC3)C4)=O)C2)=O)ccc2c(c1)OCO2 Cc1ccc2c(c1)SC(C(N1CCCC(NC(=O)C3=C(Cl)CCC3)CC1)=O)C2 C1CC(O)C(=O)N1.c1(C(N2CCC(CCSC)C2)=O)ccc(-c2cc[nH]n2)cc1 C1(C(C)NC(c2cnn(C3CC3)c2)=O)CCCCN1C(c1cc(CO)on1)=O N1(C(c2c(CNC(c3n(C)ncn3)=O)n[nH]c2)=O)CCN2CC(O)CC2C1 c1(CN(C(=O)C(C)(C)c2csc(C(=O)OC(C)(C)C)n2)CC)c(F)cncc1Cl Cc1nc2ccc(C(=O)NCC(C)(O)CNC(C3CCOC3C)=O)cc2o1 c1(C(N2CC(C)C(NC(c3ncc4n3CCCC4)=O)C2)=O)ccnc2cc[nH]c12 c1(C(=O)NC2(C)CCN(C(CCNC(C)=O)=O)C2)cnn2ccsc12 Cc1ccc(C(C)(C)C(=O)NC2CCC2CNC(=O)C=Cc2sccc2C)cc1 c1(C(N(C2CCCN(C(C(CC)n3cncn3)=O)C2)C)=O)nnc(O)cc1O CCC(CC)C(=O)N1CCC(C(=O)NC2(c3noc(C)n3)CC2)(C(C)C)C1 C1(NC(C2(CC=C)COC2)=O)CCOC(CNC(=O)CC2(O)CCC2)C1 c1(CC)nn(C)cc1C(=O)NC1CC(F)(CNC(c2cccc(OC)c2)=O)C1 c1(CC)[nH]nc(C(=O)NCCC2CN(C(=O)CC(C)SC)CCCO2)c1[N+](=O)[O-] c1(CC)c(C(=O)NCCCCCNC(=O)C(C)O)cnn1C(CC)CC CC(C(=O)NC(C1CCN(C(=O)C=Cc2ccc(O)cc2)C1)C)C(C)(F)F N(C1COCc2ccccc21)C(C1N(Cc2c(C)scn2)CC(F)C1)=O C1(C(N(CCCC(=O)NC(C(=O)OC)CO)C)=O)CN(C)C(=O)N1 c1(CC(N2C(C)CCC(NC(c3cnc(C)[nH]3)=O)C2)=O)cccc2ncccc12 N1(C(C(CC)CC)=O)CCC(C2CCN(C(C3(N(C)C)CC3)=O)C2)CC1 c1(OC)ccc(C)nc1C(=O)Nc1cccc(CNC(C2(O)CC2(C)C)=O)c1 C#Cc1cnc(=NCCCCC(C)NC(c2ncoc2C2CCC2)=O)[nH]c1 C(=O)(C(O)CCS(C)=O)NC12CC(NC(C=CC(=O)N(C)C)=O)(C1)C2 C1(C)(CCNC(C2(CC(C)C)CC2)=O)CCN(C(C2CCCCO2)=O)C1 C(=O)(CCCCC(N)=O)N1CCC2(NC(CCC(=O)NCCC)=O)C(C1)C2 Cc1cn(C)cc1C(=O)NC(c1ccnn1C)C(=O)N(CC(C)O)C C(=O)(CC(O)CCSC)NC1C(NC(c2c(CCC)nsc2N)=O)CCC1 c1(C(=O)NC2CCCCC2CNC(C2(C(F)F)CCC2)=O)ccc2c(c1)CCO2 C=C(Cl)CCC(=O)N(CC(C)NC(=O)CCCOc1ccc(C)cc1)C N1(C(CC(C=C)C)=O)CCCC2(C1)CN(C(=O)C(C1CC1)OCC)C2 C1(CC)CN(C(=O)C(=O)Nc2cc(F)ccc2OCC(F)(F)F)CC(C)(C)C1 c1(CC)nc(=N)[nH]cc1C(=O)NC1CC12CC(NC(=O)Cn1cccn1)C2 c1(OCC)ccc(NC(N2CCCCC2Cc2cc3ccccc3[nH]2)=O)cc1C#N c1(C(=O)NC2CC(CCNC(C3C(C)CN(C)C3)=O)C2)ccnc2ncccc12 C1(C2CCN(C(c3cn(C(C)C)cn3)=O)C2)(NC(CC(C(C)C)OCC)=O)CC1 N12CCC1CN(C)CC2=O.c1(CC(=O)NCc2ccco2)cnsc1 CCC(CC(=O)N1CCCC1(C(=O)Nc1ccc2nccn2c1)CC)CC(C)C N1(C(COCC(=O)NC)=O)CCC(C(=O)NC2CCN(C)C2C)(CF)C1 C12(C(=O)NCCNC(c3cnc(OC)c(Cl)c3)=O)CCCCC1CCC2 C(=O)(CCCC(CC)NC(=O)Cc1c(C)n[nH]c1C)NC1(C=C)CCCCC1 C1(CNC(CCC(=C)C)=O)CN(C(c2sc(C(C)(C)C)nc2C)=O)CCC1(C)C C1(NC(CC2CC(CC)C2)=O)CCCN(C(=O)CC2CC3CC3C2)CC1 Cc1ccc(C(C)C(N2CCCC2CC(=O)NCCCO)=O)cc1 c1(C(=O)NC(CC#C)C(=O)NC(c2ncc(C)[nH]2)CC)cnc(O)cc1C c1(C(=O)NC(C(C)NC(C=CCCC=C(C)C)=O)C)cc(C(F)(F)F)cc(Cl)c1 CC1CCCN(C(C2CCC3CCC23)=O)C1.C1(CCN(C)C)N=N1 C(=O)(C(C)(CO)NC(c1ns[nH]c1=O)=O)N(C1CC1C1CC1)C N1(C(C(CCSC)O)=O)C2CCCC1CN(C(=O)CC=Cc1ccccc1)C2 C1(N(C)C(c2ccc(-c3ccc(CO)o3)[nH]2)=O)CS(=O)(=O)CC1O CC1CCCCC1(C)C(N1CCC(CF)(NC(c2cc(C(N)=O)[nH]n2)=O)C1)=O C1(N(C(CNC=O)=O)C)CCC(NC(C2CC(OCc3ccccc3)C2)=O)C1 c1(CC(=O)NCC23C(CN(C(C(C)OCC4CC4)=O)C2)C3)c[nH]c2ccccc12 N1(C(=O)COCC2CCC2)C2CCCC1CC(NC(C1(C(F)F)C=CCC1)=O)C2 N1(C(C2(C(C)C)COC2)=O)CCC(CNC(=O)CCSC(F)(F)F)C1 c1(C(=O)NCC2CC(CNC(C3(O)CCCC3)=O)C2)cc2cccnc2s1 c1(OCC#C)ccc(CN2CC(F)(C(=O)Nc3cc(C)c(Cl)cn3)C2)cc1OC C1(NC(=O)CN2CCCCC2=O)C2CCC1N(C(=O)CC1CCCCC1O)C2 C(=O)(C1CCOc2ccc(F)cc21)NCCC(C)(C)NC(=O)C1=CCCC1(C)C c1(CCN=C(NC2C(C=C)C2)NCCc2cn(C)cn2)c(C)[nH]c2ccccc12 Cc1c(Br)noc1C(N1CCCCC1Cn1cc(C2CC(F)(F)C2)nn1)=O Cc1c(F)ccc(C(=O)NC(C)CNC(=O)CCS(N)(=O)=O)c1N N1(C(CCSc2n(C)nnn2)=O)CCN(C(C2CCCCC23CC3)=O)CC(O)C1 N1(C(C(N2CC(C)C2)C)=O)CC(C(N2CCC(NC(N)=O)C2)=O)C2(CCC2)C1 C1(CC)CCN(C(=O)Cc2cn[nH]c2)C1C(=O)NCCC(=O)NCC1CC1 C(=O)(CS(=O)(=O)C1CC1)NCC1C2CN(C(c3cc(C)c(O)cc3)=O)CC21 Cn1ncc(CC(C(=O)O)NC(=O)CC2CC(C(=O)O)C2)c1O c1(C(=O)NC2C(CNC(Cc3cc(C)on3)=O)CC2)ccc2c(c1)OCC2 CCC(C)(C)CCCC(=O)N1CC=CC1Cn1cc(C(c2ccccc2)O)nn1 C1(C(N(CCC)CCNC(c2ccnn2CCC)=O)=O)CCC(=O)N1CCC c1(CCC(=O)Nc2nc3cccc(C(=O)OC)c3[nH]2)c(Cl)cccc1[N+](=O)[O-] Cc1cncc(C=CC(=O)NC2CC3CCC2N3C(c2nc(Cl)sc2C)=O)c1 c1(NC(C2N(C(C(C)SC)=O)CC(OC)C2)=O)ccc(C)cc1N(CCO)CC C1(C2CC2)(C(=O)NCc2cc(C)n(C)n2)CN(C(C2CCCC2F)=O)C1 CCC(C)(C(=O)N1CCC(O)(CNC(=O)C(C)Cc2ccnn2C)CC1)C(N)=O C(C(C)(C)CN=[N+]=[N-])NC(c1ccc(CNC(C(C)c2ccco2)=O)o1)=O Cn1[nH]c(=NC(=O)C2CC3(C2)CC2(CCC2)C3C(=O)O)n(-c2ccccc2)c1=O C(=O)(C1=CS(=O)CCC1)NCC(CNC(c1cc(F)ccc1N)=O)OC N1(C(C(CCC=C)(C)C)=O)CCC2(CC1)CN(C(c1cc(Cl)cc(Cl)c1F)=O)C2 C1(CC(=O)NCCCCCNC(c2c(CCC)occ2)=O)CCC(=O)N1C C1(C(N2CC(CCC)N(C(=O)CNC=O)CC2)=O)Cc2ccncc2N1 N1(C(C(CC(C)C)F)=O)CCc2sccc2C1CNC(=O)Cc1ccnn1C S(=O)(=O)(c1ccc2[nH]c(=NCCOCC(C)C)ccc2c1)N(CC=C)CC1CC1 Cn1ncc(NCc2cnc(-c3ccccc3)[nH]2)c1C(F)F C1(C(=O)NC(c2ncc(C)cn2)C)CC(F)CCN1C(=O)Cn1ncccc1=O C(CCSC)(C(=O)N1CC(NC(=O)Cn2nccn2)C(O)C1)OC CCCC(C(=O)NCCC(C)NC(c1cn(C2CC2)nc1C)=O)OCC CS(=O)(=O)CC(c1ccccc1)NC(c1ncn(Cc2ccccc2)n1)=O CC1CN(C(C2CCC(F)(F)CC2)=O)CCC1N(C(=O)CN=S(C)(C)=O)C C1(CC)CN(CC)CCN1C(=O)CC1(CNC(c2c(C)nn(C)c2N)=O)CC1 CC(C(=O)N1CC(O)(C(C)(C)CNC(C23CSCC2C3)=O)C1)C(C)S(C)(=O)=O c1(C(=O)NC(C(C)NC(=O)CCCC(=O)N(C)C)CO)cnc2[nH]cnc2c1 c1(OCCC(N2CCC(F)(CNC(C(C)SCC)=O)C2)=O)ccc(Cl)c(C)c1 c1(OC)nc(NC2CC3CCCC(C2)N3Cc2cocn2)nc2ccccc12 CC(C)(F)C(C)(F)CNC(C1(CO)CN(C(=O)C2=CCCCO2)C1)=O C1(C(=O)NC(c2ccno2)C)CC12CN(c1ncc(Br)cn1)C2 C(=O)(CCCCCCCC(=O)OC)NCC(N(C(CSCC)=O)C)C1CC1 Cc1cnc2c(C(N3CCCC3CNC(=O)Cc3ccns3)=O)cccc2n1 Cc1ccc2oc(=NC3CN(C(=O)C(O)C4CC4)CC(C)(C)C3)[nH]c2c1 C12(C(=O)NC3C(CNC(C4SCCS4)=O)CC3)CCC(CO)(CC1)C2 C1(NC(C2CC23CCOC3)=O)CN(C(c2cc(Cl)nc(Cl)c2)=O)C2CCCCC12 C1(CC)CN(C(=O)CCc2cn[nH]c2)CCC1NC(=O)CCc1cnn(C)c1C C12(CNC(c3cccc(C)c3)=O)CC(C1)C(NC(=O)C(c1cncn1C)O)CO2 c1(CNC(=O)NC(C(=O)OC)CCc2ccncc2)cn2cc(Cl)cc(C)c2n1 c1(CC(N2C(C3CCN(C(C(=O)NC)=O)C3)CCC2)=O)ccc(C)c(OC)c1 c1(C(CC(=O)N2CC(N(C)C3CC3)C2)OC)ccccc1F N1(CC)CCOC(C(N2CCC(C(C)(C)CNC(=O)CC(C)F)CC2)=O)C1 C1(C)(NC(C=NOC)=O)CCCCC1C(N1CC2CCC(C1)O2)=O c1(C(=O)NCCN2CCN(C(C(C3CCC(=O)N3)C)=O)CC2)ccc(Cl)cc1O N1(C(CCCC)=O)CC(C(=O)O)C2(C1)CN(C(=O)CC(C1CC1)C1CC1)C2 c1(C(=O)NCCC=CC)cc(C(=O)OC)cs1 c1(OC)cc(C2(C(N3CC(NC(C4(Cl)CC4)=O)C(F)C3)=O)CC2)ccc1Cl N1(C(C(CC)CC)=O)CCC(NC(c2ccnc(Br)c2N)=O)CC1C c1(OC)ccc2c(C(N3CCC(C)(NC(c4cc(C)co4)=O)C3)=O)n[nH]c2c1 N1(C(c2[nH]c(=NC)sc2)=O)CCCC(NC(c2c(C)cc(C)oc2=O)=O)CCC1 CCC(CC(=O)NC1C2CN(C(C3(C)CNC(=O)N3)=O)CC12)C1CC1 C(c1ccc(C2CC2)cc1)=CC(=O)NC1C2CC1N(C(C1(F)CCOC1C)=O)C2 C(=O)(CC(C)C(C)(C)C)N(CC(=O)N(C)CCF)CCOC c1(CCC)cc(C(=O)NC(C2CCN(C(=O)CC3(OC)CCCC3)C2)C)ccn1 c1(C2(NC(CN(C(CC3(OC)CCC3)=O)C3CC3)=O)CC2)nncn1C C1(C(N2CCCC(CCC#C)C2)=O)CCN(C(=O)C(C)=C(C)C)CC1(C)C C1(C)(NC(CC(C=C)C)=O)CCCN(C(=O)COCC)C1 N1(C(C)=O)CCC(C(=O)NCCC2CC3CCC2C3)CC1 N1(C(COCC#C)=O)CCN(C(C)CNC(C2CC(C)N(C)C2)=O)CC1 C(c1ccc(Cl)cc1Cl)=CC(=O)NCC(C)N(C)C(C1CCOC(=O)CC1)=O C1(C(=O)NCC2(CCF)CC2)CCN(C(=O)C2CC2)O1 N1(c2ncc(C)cn2)CCC2CCN(C(=O)CC3CC4CCC3O4)CC2C1 CC1CCN(C(=O)CCc2cn(C)cn2)C(CNC(=O)CC(Cl)Cl)C1 c1(C(=O)NCC(C)(O)CNC(=O)Cc2cocn2)ccc(C2(O)COC2)cc1 c1(N2CC(NC(=O)C(C)(C)O)CC(C)(C)C2)ccc([N+](=O)[O-])c(C(N)=O)c1 C(=O)(CC(C)(C)O)NC1C(CNC(c2scc(C(C)=O)c2)=O)C1 C=CCC(CC(=O)N(C1COCC1OC)C)NC(=O)CC1CCCSC1 CC1CN(C(=O)Cc2sccc2Cl)CC(C)C1NC(=O)CCc1cncs1 C(=O)(C1=CCCCCC1)N1CCC(CNC(C(CN(C)C)c2ccccc2)=O)C1 N1(C(CNC(C)=O)=O)CCCCCC(NC(=O)C(F)(F)CN(C)C)C1 C(=O)(C1=CCCN(C(=O)CC(=O)NCCC2CCC(C(F)(F)F)CC2)C1)OC Cc1ccc(S(=O)(=O)Nc2ccsc2C)cc1C(=O)N(C)CC1CC1C c1(C(=O)NCC(CNC(c2ccc(OC)s2)=O)O)sc(C)cc1Cl c1(NC(C)=O)cc(Cl)ccc1C(=O)NCCC1CN(C(C2(C)CC2)=O)CCO1 c1(CC(N2CCC(OCCNC(C(CC(C)C)O)=O)C2)=O)ccc2ocnc2c1 CC(C)(F)CCC(=O)NC(CNC(=O)CCNC(=O)OC(C)(C)C)C1CC1 C1(NC(C=CC2(C)COC2)=O)CC=C(C(=O)NC2CC(O)C2)C1 CC(C)(C)CC(C)(C)C(=O)NCCOCCNC(C1N2CCC1(C)C2)=O Cn1cncc1C(O)C(=O)NCCC1(NC(c2ccco2)=O)CCC1 C1(C(C)C)CCN(C(=O)C(c2ccoc2)NC(C2C3CC4C(C3)C24)=O)CC1 N1(C(C(C(C)NC(c2nc(CCC)oc2)=O)C)=O)CC2CCC(C1)C(=O)N2 N1(C(C(c2cnn(C)c2)NC(c2c(OC)cncc2)=O)=O)CCN(C)C2CC12 C1(C(=O)NCC(C)NC(CN(CCOC)C)=O)CC(OC(C)=O)C1 C=C(C)CC(C(=O)NC1CC12CC(NC(=O)C(COC)N(C)C)C2)OC Cc1cc(C#N)cnc1C(N1CCC(C)C(N(C)C(C2CCCN2C)=O)C1)=O c1(NC(C2C(NC(c3cc(O)cc(F)c3)=O)CCCC2)=O)cncc(F)c1I N1(C(C(N(C(CC(CC)C2CC2)=O)C)C2CC2)=O)CCC(CO)C(O)C1 CCC(C)C(C(=O)Nc1cnccc1C)N(C)C(c1cc(COC)on1)=O C(=O)(CCCC(C)(F)F)N(CCCNC(=O)CCc1cncnc1)CC c1(C(N2C(CCNC(c3n(CC)ccc3)=O)CCCC2)=O)c[nH]c2cccnc12 C1(NC(C2C(C)=C2)=O)CC2CCC(C1C)N2C(=O)C(F)(F)c1ccccc1 N1(c2ccc(C(N3CCC(c4c(C)ccnc4)C3)=O)cc2)CC(C)(C)OC1=O c1(C(N2CC3C(NC(CCOCC#C)=O)(CC3)C2)=O)c[nH]c2ccncc12 N1(CCNC(C(CCC)C)=O)CCN(C(c2cnc(Cl)cc2N)=O)CC1 C1(CNC(CN(CCOC)C)=O)CN(C(=O)C(C)c2ccsc2)C2CCCC2O1 C12CCCN(C1)C(=O)C(C)N(CC)C2.C(C(=O)N)=CC=CC.C1CC1 c1(C(N2C(CNC(C3C(c4onc(C)n4)C3(C)C)=O)CC2)=O)ccnc(C)n1 c1(CC)ccc(F)c(C(=O)N(CC(O)CNC(C2(COC)CCCO2)=O)C)c1 C1(CC(=O)OC)CN(C(c2ccn(COC)n2)=O)C(C)(C)CO1 n1(C(C)C)cc([N+](=O)[O-])c(=NC2CC(NC(=O)CCCc3ccsc3)C2)[nH]1 CC(C)C(CNC(=O)Cc1ccc(Br)s1)NC(=O)CNC=O C=CCCCCCN=c1cc[nH]cc1S(=O)(=O)N1CCCC(O)C12CCC2 N1(C(COCCC)=O)CC(CNC(C2CCN(CCS(N)(=O)=O)CC2)=O)C(C)C1 c1(NC(C2CC(O)CN2C(=O)C=Cc2cccs2)=O)ccc(Cl)nc1Cl c1(NCC(=O)NCCCN(C(=O)CC2CSCCO2)CC)ccc(C)cc1 N(C1CCc2c1cnn2CC)C(c1ccc(Br)cc1)C(=O)NC(C(CC)CC)=O c12nocc1C(=O)NC2C.N1(C(C)=O)CCC1C(C)C.C1(=O)CN1 C=CCC(C(=O)N1CC=CC1(C(=O)N(C)CCc1nccs1)COC)C(C)C CCC(CC(=O)N1CCCC1CNC(C1(Br)CC12CCC2)=O)OC c1(C(C#C)N(CCC2CC(NC(=O)OC(C)(C)C)C2)CCC)ccco1 Cc1cc(C)c(C(=O)NCC2CCCC(NC(c3c(C)coc3C)=O)C2)c(=O)o1 C(=O)(Nn1cnnc1)c1c(C)nn(-c2ccc(Cl)cc2)c1 n1(CC(=O)NC(C2CN(C(C3CC(=C)C3)=O)C2)C)cc(C(F)(F)F)cc1C C1(NC(c2cn(CCC)nn2)=O)CCOC(C(=O)NC2(C)CC(C(N)=O)C2)C1 c1(-c2cn(CCC(=O)N(C(c3ccc(C)cc3)C)C)nn2)cccc(F)c1C#N C1(C(=O)NCC(C)(C)OCCNC(C2(N(C)C)CC2)=O)CCCN1N=O Cc1oc(C(=O)NCCn2cc(CNC(=O)Cc3cccs3)nn2)cc1CO C#CC1(C(=O)NCC2CC2NC(C2CC2c2nncn2C)=O)CCCCC1 N1(C(C2(NC(C)=O)CCC2)=O)CC(NC(C2(C)CC(C)(C)C2)=O)C(C)C1 C=CCC(C)C(=O)NC1CC1NC(c1cccc(OCC=C(C)C)c1)=O c1(C(N2C(CN(C(CNC(C)=O)=O)C)CCCC2)=O)cccc2cnnn12 c12ccc(cn1)c(=O)[nH]2.N1(CCNC(C(C)NC(CC)=O)=O)CC(C)(O)C1 C(=O)(CP(C)(C)=O)N1CCCC(CCC(=O)NCC2(CC)CCCC2)C1 C1(CNS(C)(=O)=O)CN(C(=O)C(N2CC3CCCCC23)=O)CCCO1 C1(C(=O)NC2CC(N(C)C(c3cocn3)=O)C2)CC(c2ccc(Cl)cc2Cl)=NO1 c1(C(=O)NCC2(NC(C3C(C#C)C3)=O)CCCCC2)ccc2nccnc2c1 CC1CCCC1(C(=O)N(C)CCc1cnn(C)c1)NC(=O)CN(C)C c1(C(N2CC(CC(C)NC(=O)C(C)n3ccnc3)C2)=O)ccc(CO)nc1 C(=O)(C(C)CCCC(C)=O)NCC1C(NC(CCC(CC)OC)=O)CCC1 N#Cc1ccc2nc(NC(C3C=CCN3Cc3cc(Cl)ccc3Br)=O)[nH]c2c1 c1(C(N(C2CCC(C)CC2)C(C2CC(C)(C)C2)=O)=O)noc2cc(Cl)ccc12.CC=CCl C1(NC(c2c(C)n[nH]c2)=O)CC(CNC(=O)C=Cc2ccco2)C(O)C1 N1(C(C2CC(C)(CC)C2)=O)CCCCC(C(=O)NC(c2cccnc2)CC)C1 n1(CCCN2C(CC(=O)OCC)CCC2)c(=O)oc2ccccc12 c1(C(N2CCC3(C(=O)Nc4ccc(I)cc4F)CC3C2)=O)cc(C2CC2)ncc1Br CN1CCN(C2CCN(C(=O)NC3CCN(C4CCCC4)C3)CC2)C1=O c1(C(=O)NCC(C)CN(C(=O)CCCOc2cccnc2)C)cc(Cl)nc(Cl)c1 CC1(C(=O)NCC(C2CC2)NC(=O)CCCC(F)F)CCC(=O)NC1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCC(NC(=O)C(=O)N=S(C)(C)=O)C(CO)CC1 N1(C(C2C(C)(C)C2(F)F)=O)CCN(C(c2ccoc2Br)=O)C(CC2CC2)C1 c1(NC(CCOC)C(F)F)cc(N2CCC(NC(=O)OC(C)(C)C)C2)nc(C)n1 N1(C(c2c(CC)n[nH]c2)=O)CCCCC1CNC(=O)CCCN1C(=O)CCC1=O Cc1nc([N+](=O)[O-])cn1CCC(=O)NCC1(F)CCN(C(C)C(=O)N(C)C)CC1 c1(C(=O)OC)ccc(O)c(C2CN2)c1.C(C(C)CC(=O)OC)C(=O)OC(C)(C)C C(=O)(N1OC2CCC1CC2)C1CC(C)CN(C(=O)CCCC(C)(C)C)C1 C#CCC(C)(C)C(=O)N(C1CCN(C(=O)C=Cc2cn(C)cn2)CC1)CC(C)C N1(C(c2cc(COC)[nH]n2)=O)CCC(CNC(=O)CC2(CO)CC2)C(C)C1 N1(C(c2ccc(OC)c(-c3ccccc3F)c2)=O)CC(=O)N(C)C2CC12 c1(O)ccccc1F.CC(CCC(=O)NC1CCCCC1)NS(=O)(=O)C(F)(F)F Cc1cc(N)c(C(=O)NCC2CCC2NC(C2CCCC2(C)C)=O)cc1F C(=O)(CCCC(C)CC)N(C1CCCN(C(c2cc(C)c(CO)cn2)=O)C1)CC Cc1cccc(C(F)C(=O)NC(CNC(c2scnc2C)=O)CO)c1 C1(CCNC(C2(CC=C)CCOC2)=O)CSCCN1C(c1cccc(CO)c1)=O O=C1CN(C(=O)COc2cccnc2)C(C(=O)NC(C2CCOC2)CO)CN1 CCC(C)C(C)C(=O)NCC(C1CCCN1C(C1CC(=O)C1(C)C)=O)(C)C C(=O)(C(C)(C)CC(C)(C)C)NCC(CC=C)NC(=O)C#CC(C)(C)C c1(C(OC)OC)ccc(NC(c2cccc(C(F)(F)Cl)c2)=O)cc1 N1(CCNC(C2CCOC2C(=O)NC2(CC3CC3)CCC2)=O)CCCOCC1 Nc1ccc(Cl)cc1C(=O)NCC1(O)CCN(C(C2CCNC2=O)=O)C1 c1(C(=O)NCCN(CCC)C(C2(CO)CCCC2)=O)cc(C)cc(Br)c1 C#CCC(CC(=O)NCc1ccc(CC)cc1)NC(C1(CC)CCOC1)=O C(=O)(C(F)CCC(C)C)N1CC(CNC(c2c(C)cc(C#N)s2)=O)C(C)C1 Cc1cc(CC(=O)NCCNC(=O)CC2CCN(CC(F)(F)F)CC2)cc(F)c1 C1(C2CCN(C(=O)Cn3nnc(=O)[nH]3)CC2)(NC(C(=O)NCC)=O)CC1 CC12CCCC(C(=O)NC3CC(CNC(c4ccc(Br)cn4)=O)C3)(CO1)C2 c1(C(N(C)CC2N(C(C(F)OC)=O)CCCC2)=O)cnc2c(c1)NCC(=O)N2 N1(C(=O)CCn2cncn2)CC2CC1CN2Cc1ccn(-c2ccccc2)n1 Cc1nsc(C(=O)NC(C)CCC(=O)O)c1N CN(S(=O)(=O)N1CC(O)C(O)C1)Cc1cccc(C(F)(F)F)c1 C(=O)(C(C)CCCC(C)=O)NCC1CCN(C(CN2CC(=C(C)C(F)F)C2)=O)C1 C1(CC(=O)NCCCCNC(Cc2scc(C)c2)=O)OC(C)(C)OC1=O C(=O)(CC(C)(C)COC)N1CC(NC(COc2c(CC)cccc2)=O)C(OC)C1 C1(CNC(CS(=O)(=O)NCC)=O)CC2CC1CN2C(=O)C(F)n1ccnc1 c1(C(=O)NCC(CC)NC(=O)CCn2nc(C)nc2C)ccc(O)c(F)c1 C1(C(N2CCCC(NC(C3(C)CS(=O)(=O)C3)=O)C2)=O)CCC2CC2CC1 c1(C(=O)NCCC(C)NC(=O)CC2(O)CCCC2)cc(Br)c2[nH]nnc2c1 C1(N(C)C(c2cnc[nH]2)=O)C=CCN(C(=O)CC(=O)OC(C)(C)C)C1 c1(SCC)ccc(-c2nc(C(c3ccccc3F)C)nn2CCCSCC)cc1 CN1CCCC(C(=O)NC2CN(C(=O)CCCn3ccnc3)C2)C1 C(=O)(C(CC)C(C)(C)CC)N1CC(CC)(NC(=O)C(C(C)(C)C)n2ccnn2)C1 C1(CC)CN(C(=O)Cc2cccnc2Cl)CCC1NC(=O)Cc1nc(C)cs1 c1(NC(C2CCC(CNC(C(OCC)OCC)=O)CC2)=O)cnc(O)c(F)c1 c1(C2C(C(=O)NC(c3nc(C(C)(C)O)no3)C)C2)cccc(Br)c1 C12(CC(=O)NCC=CCNC(C(C)OCC=C)=O)CC3CC(CC(C3)C1)C2 N1(C(c2c(CC)nc(C)o2)=O)CC(NC(c2cnc(C)s2)=O)CC2(CC2)C1 c1(C(N(C)Cc2cn(CC3CCOC3)nn2)=O)n[nH]c2c1CSCC2 Cc1cnc(Br)cc1NC(C1CN(c2nc(C(C)C)ns2)CCO1)=O c1(C(=O)NC2CCN(C(CCC3C(C)(C)C3)=O)C23CC3)c[nH]c2cc(F)ccc12 C1(C(=O)NCCNC2C(C)C(C)CN2C(=O)OC(C)(C)C)CCc2cnnn2C1 C(C(C(=O)NCC(C1CCC1)NC(=O)CCc1n[nH]c(=N)s1)OC)OC c1(CC(=O)NCC(CNC(C2CN(C(C)C)C2)=O)OC)cn(C)cn1 N1(C(C(COCC)C)=O)C2CCC1CN(C(=O)C(C)(C)C(F)F)C2 CC1OCCOC1C(=O)NCC(C)(C)CN(C(=O)CCc1ccccc1F)C c1(C(=O)NCCCCCCNC(c2ccc(O)c(F)c2)=O)c(F)cncc1Cl C(C(=O)N(C)OC)NC(C1C(NC(COCC(C)C)=O)CCC1)=O N1(C(c2c(CC)cc[nH]2)=O)CCOC(C(=O)NC2COC(C(F)F)C2)CC1 C(N=c1cc[nH]c(C#N)n1)C1(C(C)C)CCN(C(=O)C(C)Oc2cccnc2)C1 n1(CC(=O)NC2CC(CCNC(c3cn(C)nc3)=O)C2)cccc(N)c1=O c1(OCCC)ccc(C=CC(=O)NC2CN(C(C3(C)CC(F)C3)=O)CC2C)cc1 c1(C(=O)NCC2CC(C)N(C(C3CC3(F)F)=O)CC2)snc2ccccc12 C(CC(=O)NC(CSC)CO)N(C(=O)COCCCN(C)C)CC#C c1(CN2CC(C)N(C(=O)CS(=O)(=O)NC(C)(C)C)CC2)cccc([N+](=O)[O-])c1N C(CCCCC(=O)N1CCC(C)(CNC(=O)CCN2CCC2)C1)NC(C)=O C#CC1(O)CCN(C(=NCc2ccc(Cl)cc2C(=O)OC)NC2CC2)C1 Cc1cc2cc(C(=O)NC(C)CCCNS(C)(=O)=O)[nH]c2cc1Cl Cc1c(F)ccc2c(=O)c(C(=O)NC3CCCC34CN(C(=O)CCF)C4)c[nH]c12 Cc1cccc2c(C(N3CCC(C)C3CNC(c3cccc(Cl)c3F)=O)=O)n[nH]c12 Cc1nc(C)c(C(=O)NC2CCOC(CNC(=O)Cc3cccnc3)C2)o1 c1(CC)c(C(=O)N(C)CCNC(=O)CSC(C)C)cnn1-c1ccccc1CC C1(NC(C(COC)(C)C)=O)CCCN(C(c2cccc(OC(F)F)c2)=O)CC1F C12(CNC(C(C)c3cccs3)=O)CCCC1N(C(=O)C(C)NC1CCCC1)CC2 N1(C(C2(OCC)CCCC2)=O)CCCC2(NC(=O)CC3(C)CC3(F)F)CC2C1 n1(CCC)ncc(C(=O)NC2CCC(NC(c3c(Cl)nsc3Cl)=O)C2)c1C C#CCCC(O)C(=O)N1CC(NC(=O)C(C)=C(C)CC)C(C)C1 c1(OCC)cccc(SCC(=O)NCC(CO)NC(=O)CC(C)c2ccco2)c1 Cc1ccc(C(=O)NC(C)CCc2ccnn2C)c(-n2ccnc2)c1 C1(N(CCc2cn(CC(CC)O)nn2)C)Cc2ccccc2OC1C(F)(F)F CC1(C)COCC1CNC(=O)C(=O)NCc1nnc(Cc2ccc(Cl)cc2)o1 c1(N2C(CNC(C(CCCOC)C)=O)CCC2)ccn2nccc2n1 c1(C(N2CC(CNC(C(C)n3cccn3)=O)OCC2)=O)nccc(C#N)c1F N(C1c2ccccc2CC1NC(=O)CCCCCO)C(C1CN(C)C(=O)N1)=O C1(NC(CCOC)=O)CCCCC12CCN(C(=O)CC(=O)OC(C)(C)C)CC2 C(=O)(C1=CS(=O)CCC1)NC1CC2CC(NC(c3ccc(CN(C)C)o3)=O)CC21 c1(CC)nc(C)ccc1NC(=O)NCc1ccc(C)c(OC(F)F)c1 c1(-c2nc(C3CCC(F)(F)C3)nn2C2CCOC2)cnc2cnccn12 C1(CC(N2CC(NC(c3cnnn3C3CC3)=O)C2)=O)CCC=CCC1 N1(C(Cn2nc(C)c(Cl)c2)=O)CC(C)CCC1CNC(=O)CC1CN(C)C1 N1(c2ccnc(NC(CC(CC)C)=O)n2)CCc2[nH]nc(C(F)(F)F)c2C1 C1(O)(CN(C(C(C2CCCC2)OC)=O)C)CCN(C(=O)C=C2CCN(C)C2)C1 c1(C(=O)NC(C(=O)N(C)CC2CC(=C)C2)c2ccoc2)ccc(C)nc1O C1(C)(C(=O)NCC2C(NC(C(C(C)C)O)=O)CCC2)CCN(C)CC1 Cc1c(Cl)c(C(=O)NCC23CC2CN(C(C2CCCCC2O)=O)C3)nn1C c1(C(=O)NC(C(=O)N(CC(CN(C)C)O)C)C2CC2)cccn2ccnc12 C1(CNC(=O)Nc2cccc(C(C)C)n2)CCC2(CCCCCC2)O1 Cc1ccc(C(=O)NC23CC(NC(=O)C(c4cc(F)cc(F)c4)C)(C2)C3)c(O)n1 N1(C(CNC(CCC)=O)=O)CCSCC1CCNC(C1CS(=O)(=O)C1)=O C=CC(C)(CCOC)C(=O)NC(C)CC(C)NC(c1ncnn1C)=O CC1C(C(=O)NCCCN(C(=O)CCC(N)=O)C2CC2)=Cc2ccccc21 C1(CNC(c2n(CC)ccn2)=O)CN(C(C2CCCC2O)=O)CCC1(C)C C1(NC(C2C(NC(c3ccnc(Cl)n3)=O)CCCC2)=O)CC2CCCC(C1)C2 CC(CN(C)C(C1CC(CF)C1)=O)C(=O)NCc1nc(=O)o[nH]1 C(=O)(C#CC1CCCCO1)N1CC(C)(NCc2coc(-c3ccc(F)cc3)n2)C1 C1(CC)CCN(C(C2CC(O)C(F)C2)=O)C1C(=O)N(C)Cc1ncco1 c1(OC)ccc([N+](=O)[O-])cc1NC(=O)CC1C(=O)Nc2ccccc21 C1(NC(c2c(C)cns2)=O)CC2CN(C(c3cc(O)cc(N)c3Cl)=O)CC2C1 N1(C(=O)COCCCF)CCC(C2OCCC2NC(=O)CSC2CC2)CC1 c1(C(=O)NCC(=C)CCNC(=O)C(C)C(O)C(C)C)cc2c(Cl)cc(Cl)cc2[nH]1 Cn1ncc2cc(-c3ccc4c(C(=O)NCCF)n[nH]c4c3)ccc12 c1(Sc2ccnc(-c3nc(C)sc3)n2)cc(C)cnc1C#N c1(OC)cccc2c(C(=O)N(C(C)CCNC(=O)CSC)C)csc12 C1(CNC(c2cc(CNC(C3C(COC)CC3)=O)on2)=O)CSCCO1 N1(C(C2N(C)CCC2)=O)CCC2(CCCN2C(c2ccc(C(C)(F)F)nc2)=O)C1 N1(C(Cc2nc(CC)sc2)=O)CC(NC(=O)C#CC2(C)CC2)C(S(C)(=O)=O)C1 CCC(C)(CO)CN=c1[nH]c(=N)[nH]c(=NCc2nc3cc(OC)ccc3n2C)[nH]1 Cc1c(C(=O)NCC(O)CNC(C2C3(CC3)C23CC3)=O)ccc(Br)c1F C1(C(=O)NCCn2c(C)nc(C)n2)CN(C(c2nnc(S)n2C)=O)CC1C1CC1 C(=O)(C1=CCCCCC1)N1CC(C)C(CNC(=O)Cn2cnc3ccccc23)C1 C1(O)(CNC(c2nc(C(C)OC)sc2)=O)CCCN(C(C2(CC(F)F)CC2)=O)C1 C12(CNC(C)=O)CCC(CNC(=O)C(C)(C)c3cnsc3)(CC1)OC2 CC1=C(C(=O)NCCC2CCCN(C(=O)CCc3ncc[nH]3)C2)SCCO1 Cc1sc(C(N2CCC(NC(=O)C(C)n3ccnc3)CC2)=O)nc1Br c1(C(N2CCOCC2COC)C(=O)NCCC(=O)OCC)cc(Cl)c(OC)cc1Cl c1(C(N2CCC(CNC(CC3(CC)CCC3)=O)C2)=O)cc(F)ccc1OC CCCCC(CC)C(=O)NCCCOCCNC(=O)C(C)c1ccco1 c1(C(N2C(CNC(CC(CCSC)O)=O)C=CC2)=O)cc2cc(F)ccc2s1 N1(C(C2ON=C(C)C2)=O)CC=CC(NC(=O)CCC(=O)N(C)CCN(C)C)C1 N1(C(C(c2ccc(F)cc2)(C)O)=O)CCCCC(NC(=O)C=C2CCOCC2)C1 N1(C(C(CC)C(C)O)=O)CC(CO)C2(C1)CN(C(=O)C(C)=C1CCCC1)C2 C1(SC)CN(C(c2coc(C(F)F)c2)=O)CC1NC(=O)CC1CSCCO1 c1(-c2nc(CCOC)nn2CCF)cc2ccc(OC)nc2[nH]1 C1(C(N2CCC(NC(C=CC=CC)=O)C2C)=O)CCC(C)C(C)C1 C1(CNC(CC(=O)N(CCCOC)C2CC2)=O)CC1C1CCCC1 C(=O)(C(C)(C)C(C)C)NCC1CC(NC(Cc2c(C)nsc2)=O)C1 C1(NC2CCN(C(C(=O)OCC)=O)C2CCl)CCOC12CCOCC2.C(C)(C)C N1(C(C(CC)N(C)CC)=O)CC(NC(C2CN(C(N)=O)C2)=O)CC(F)C1 C1(C(=O)NCC2C(NC(Cc3cc(CC)no3)=O)COC2)OCCN(C)C1=O c1(C(=O)NC(C2CCCCN2C(=O)C(=O)NCC(F)F)C)ccc([N+](=O)[O-])n1C C1(C(N(C(C#C)C)C)=O)CN(C(C2CCC(CO)CC2)=O)CC(C)O1 C1(CNC(C2(CC)CCNC2=O)=O)CCN(C(c2c(C)noc2C)=O)C(C)C1 C(C(=O)N1CC=C(C)CC1)(C(C)(C)C)NC(C(CC)=CCCC)=O N1(C(CC2(CC)CC2)=O)CCN(CC(C)NC(C2CCC(C(C)C)CC2)=O)CC1 N1(C(c2n(C)nc(CNC(C3CCC(=O)C3)=O)c2)=O)CCCC12CCOCC2 c1(SC)ccc(C(=O)NC2CN(C(c3cncc(C(C)C)c3)=O)C2)cc1 C1(C(=O)NCC(C(=O)NC)O)CC2CCC(C1)N2C(=O)COC(C)C c1(CC)onc(C(N2CC(C(=O)NCCC(C)C(=O)OC)(COC)C2)=O)c1C c1(SCCC(=O)NC2CC(F)(CNC(CC3CC(C)C3)=O)C2)ccc(F)cc1 c1(C(=O)NC(C2(O)CCN(C(CC(CC)C3CC3)=O)C2)C)cc(OC)nc(Cl)c1 C1(NC(c2ncccc2C2CC2)=O)CCCCCC1NC(C1CC(CF)C1)=O C1(O)(C(N(C2CCCN(C(=O)Cn3cc(C4CC4)cn3)C2)C)=O)CCCCCC1 N1(C(CN(C2CC2)CC)=O)CCC(C)(NC(=O)C(c2ccccc2)C)CC1 C1(C(N2CC(OC(CC)=O)C2)=O)C2CC3C(C2NC(=O)C(C)CC2CCCC2)C13 N1(C(=O)NCC2(CC)CC2)CCN(c2cc(C)ccc2OC)C(=O)C1 C(=O)(C1=CC(C)(C)C1)N1CC(CCNC(c2c(C)cc(CO)o2)=O)C(C)C1 c1(OC)cccc2nc(NC(c3n[nH]c(C)n3)=O)sc12 C#CC1(C(N2C3CCC2CC(CO)C3)=O)CCN(C(=O)C(F)C(F)(F)F)CC1 N1(C(c2cc(C)cc(C(F)F)c2)=O)CCC(C2CC2C(=O)O)CC1 N1(C(C)C)CCCC1CC(=O)NC1(C)CC(NC(=O)C=Cc2ccco2)C1 c1(CC)ccc(F)c(C(=O)NC2CCN(C(=O)C=CCOC)C(C)C2)c1F Fc1cc(CSc2cc(C3CC3)cc(Cl)c2)c2ncccc2c1 N1(C(CCC=C(C)C)=O)CCC2(CC1)CN(C(c1scnc1C(C)C)=O)CCO2 C=CCCC(=O)NCc1ccc(C(=O)NCC(F)Cl)s1 C1(C#CC(=O)NC2CC(F)(CNC(=O)CCCC(C)=O)C2)(CC)COC1 c1(NC(CCCC2(C)NC(=O)NC2=O)=O)ccc2[nH]c(C(F)F)cc2c1 N1(C(c2ccn(CC)c2C)=O)CC(N(C)C(C2CCC(=O)NC2)=O)C(C)(C)C1 c1(OCC(=O)NC(C(C)NC(Cc2c(C)noc2Cl)=O)C)nc(O)nc(O)n1 N1(CC(=O)N(CCCNC(C2(C3CC3)CCCO2)=O)C)CCC(=O)NC1=O c1(C(=O)NCC2CCN(C(c3c(C(C)C)c[nH]n3)=O)C2)ccc(S(C)(=O)=O)o1 C(=O)(C1=C(C)OCC1)N(CCC(=O)NCC1CC12CC2)CC=C CCCC(C(=O)NC(C1CC2(CCC2)C1)C)NC(=O)CN1CC2CC2C1 c1(C(N2C(C)C(O)CCC2)=O)c2c(nn1C)CCN(C(=O)Cn1cccn1)C2 c1(C(N(C2CCN(C(=O)COCC(=O)NC)CC2)CC)=O)ccc(N)cc1OC C1(NC(c2c(CC)occ2)=O)CC2CN(C(=O)CC3(N4CCCC4)CC3)CC2C1 C1(C(N2CCCC(CN(C(C3(CC(C)=O)CCC3)=O)C)C2)=O)C2CCC(F)(F)C12 C1(C(C)NC(c2c(CC)cco2)=O)CCCN(C(C2(C#N)CC2)=O)C1 c1(N2C(C(=O)Nc3ncnc4c3CCC4)CCC2)ccn2ncc(Br)c2n1 C1(NC(CC(C)C(F)F)=O)CN(C(c2cc(C#N)cs2)=O)CC(C)(C)C1 C12(C(=O)NC3(CCNC(CCn4ccc(C)n4)=O)CC3)CCCC1CC(=O)C2 CCC(C(=O)NCC(C)NC(=O)Cn1cnc(Br)c1)Sc1ccccc1 C(=O)(C(C)(O)C(C)C)NC1CC(CNC(C(COC)Cc2ccc(Cl)cc2)=O)C1 CC(C)(C)CC(C)(C)C(=O)NC1C2CCC1CN(C(=O)C(O)C(F)(F)F)C2 C(=O)(C1=CS(=O)CCC1)NC1(CO)CN(C(CC(n2c(C)cc(C)n2)C)=O)C1 N1(C(C(C2CCCC2)OC)=O)CCCC(CO)(CNC(c2ccc(O)nc2)=O)C1 c1(C(=O)NC2CN(C(C(C(C)C)C(C)C)=O)CC2O)cc2c(F)c(F)ccc2s1 C(=O)(C1CCCc2sc(=N)[nH]c21)NC1CCCN(C(C(C)(C)c2cccs2)=O)C1 c1(OCC)ccccc1NC(C1CC1NC(=O)C(CC)OCC)=O N1(C(CCC(C)=O)=O)CC2CC(C(=O)NCCCC3CC3)CC2C1 C(=O)(CCCn1cncn1)NC(C(=O)NC(COC)COC)C1(O)CCC1 n1(CC)ncc(Cl)c1C(=O)NC1CCCC1NC(c1nc(Cl)oc1C)=O c1(CNC(C)COc2ccccc2)cnc(Cl)cc1Br c1(C(=O)NCCNC(=O)C(=O)Nc2ccccc2CO)cc(Cl)ccc1F C1(C(N(CCNC(C2CCS(=O)(=O)C2)=O)CC)=O)Cc2ccccc2N1C(C)=O Cc1c(C=CC(=O)NCC2(F)CN(C(=O)Cc3ncc(Cl)s3)C2)cnn1C C#CCC(Cc1ccccc1)NC(=O)CCSCC(=O)Nc1ccccc1 C1(C(N2CC3C(NC(CC4C(=O)NC(=O)N4)=O)C3C2)=O)C2C=CC(C2)C1CO C(CN=c1[nH]c2c(c(=NCC3(CSc4ccncc4)CC3)[nH]1)CSC2)OC(F)F c1(OC)nc(C(=O)NCC2CC2NC(C2(C)CC2(C)C)=O)sc1C C(=O)(C1CCc2cccc(Cl)c21)N1CCC(CCNC(=O)OCC)CC1.C(=O)C(=O)N CCC(C(=O)N(C1CCN(C(c2cc[nH]c2C2CCC2)=O)C1)C)C(C)C N1(C(c2c(C)nns2)=O)CCC2(C(=O)N(C)C)CCCC12.C1(CO)C(=O)N1 C(=O)(CS(=O)(=O)C(C)C)N1C2CC(CNC(c3c(OC)cccc3)=O)C1CC2 C1(NC(CC=C=C)=O)C(C)CN(C(=O)COC(F)F)CC1C c1(NC(C2CCCN2Cc2ncc3ccccn23)=O)ccc(Br)c2ccccc12 Cc1nn(CC(N2CCCC2C2CCN(CC3CCCCN3C)C2)=O)c(=O)n1C C1(O)(CNCC(CCC)NC(C)=O)CCN(Cc2ccccc2)C1 C1(CNC(c2cc(OCC)no2)=O)CN(C(=O)C#CC2CCCO2)CCC1(C)C N1(C(C(CC)NC(C)=O)=O)CCN(CC(N2CCCC2C(=O)NC)=O)CC1 c1(C(=O)NC2CC(CS(C)(=O)=O)C2)cccc(S(=O)(=O)CF)c1 CC(C)(C)C1=NOC(C(=O)NC2CC(C)(NC(=O)CCNC(=O)CO)C2)C1 CN1CCN(C(C2Cc3nnsc3S2)=O)C(CNC(=O)Cc2ccnn2C)C1 C(=O)(C1OCCc2ccccc21)NCCCC(C)(C)NC(=O)C=CC1CCOC1 n1(CC)nc(C)cc1C(=O)NCCC1CCN(C(C23CCCC2C3)=O)CC1 c1(SC)ccccc1C(C)NC(=O)NC1(CO)CC(C(=O)O)(CO)C1 C1(CC(=O)NC2COCC2NC(=O)C2=CCC2)CCC(c2ccccc2)CC1 CC(CC(=O)N1Cc2ccncc2C1)C(C)(C)NC(=O)C(F)C(C)(F)F C(C(C)C(=O)OC(c1cnn(-c2ccccc2)c1)C)OCC.c1(CN)ccccc1 c1(NC(C2C(C(N(C(c3cncc(F)c3)C)C3CC3)=O)C2)=O)cc(Cl)n(C)n1 C=C1CCN(C(=O)CC(C)N(C)C)C(C(N2CC(CO)C3(CC3)C2)=O)C1 c1(C(=O)NC2(C3CCN(C(Cn4ccc(C)n4)=O)CC3)CC2)occ2c1CCC2 N1(C(C2(C#N)CCCC2)=O)CCOC(C(NC[Si](C)(C)C)=O)CC1 C(=O)(CS(=O)(=O)c1ccccc1C)N1CCC(CNC(C2CC(C)(CC)C2)=O)C1 n1(CC(=O)N(CC(CNC(C(CC)(C)O)=O)O)C)ncc2ccccc12 CC(C)C(C(=O)NCCN(C)C(C1COCCN1C)=O)NC(c1ccccc1)=O C(=O)(C(CNC(=O)COCCC(C)C)C(C)C)NC(C)COC.C(CS)OC N1(C(C(CCC)C(C)C)=O)CC2CCCN(C(c3ccn(CCF)n3)=O)C2C1 c1(C(=O)NC2CCN(C(c3c(N)nccn3)=O)CC2CO)nc[nH]c2ncnc1-2 C1(NC(Cn2cc(C(C)O)nn2)=O)CCC(NC(=O)CC2CCCO2)CC1 N1(CCC(=O)NC(C2CCCN(C(C(CC)CC)=O)C2)C)CCSC(C)(C)C1 Cc1ccc(CNC(=O)CN2CC(C)CCC2OC(=O)C2CC2)c(C)c1 C12(C(=O)NC(CC)(CC)C(C)C)CCCC1CN(C(=O)CCc1cccn1C)C2 C(C(CC1CC1)C(=O)N(C1CCSCC1)C)NC(C=CC(C)C)=O Cc1cc(C(=O)NCCOCC(N2CCCC2(C)C2CC2)=O)[nH]c1C c1(CCC)c(C(N2CC(CN(C(=O)C(F)(F)CN3CCCC3)C)C2)=O)cnn1C Cc1cnsc1C(c1nnnn1C1CCC1)NCCCNC(N)=O c1(C(N(CCNC(C2=CC(C)CC2)=O)C2CC2)=O)cc2c(F)c(F)c(F)cc2[nH]1 CC(CC(C)(C)C)C(=O)NC1CC(CNC(c2cccn2CCC)=O)C1 c1(C(C)NC(c2ccc(S(=O)(=O)NC)o2)=O)cc2cc(F)ccc2o1 c1(C(=O)NCCC(C)(C)NC(C2C(=C)C2)=O)nnn(-c2ccccc2)c1C CC1(N=c2[nH]nc(C(F)F)o2)CCC(COC2CCCC2)CC1 C1(C)(CNC(C2CN(CC)C(=O)C2)=O)CCCN(C(C2CCC(C)CC2)=O)C1 N1(C(C2C(C(=O)OC)CCC2)=O)CC2CC1CN2C(=O)CCCn1cccc1 c1(CNC(C=C(CC)CC)=O)cccc(C(=O)NC2CC2(C)C(C)C)n1 C1(CC(=O)N(CC(=O)NCc2cscc2C2CC2)C)CCCCCC1 N1(C(CC(C)SC)=O)CC2(CCN(Cc3cn4ccccc4n3)CC2)CC1C C1(c2n(CCCCCC)nnn2)(NC(c2cc(Br)no2)C)CCN(C(C)C)C1 N1(C(c2cnc(C)c(N)c2)=O)CCOC2(CCCN(C(=O)C(O)CC(C)C)C2)C1 c1(OC)ncc(F)c(NC(=O)C(C2CCN(Cc3ccc(F)cc3Br)CC2)C)n1 N1(C(CC2ON=C(C)C2)=O)CCCCC(C(=O)NC2CCCC2C(N)=O)C1 Cc1cnc(F)c(C(=O)NC2(C3CCCCN3C(C3CC(C)(C)C3)=O)CC2)c1 c1(C(N2CCC(C)(NC(CCOCCOC)=O)CC2)=O)c(F)ccc(F)c1OC CCCC(O)CC(=O)N(C)CC1COCCN1C(c1ccccc1CC#N)=O c1(N2CCCN(C(C)C)CC2)nc(=NCCSC(F)(F)F)[nH]c2c1CCCC2 c1(C(c2n(C)ncc2)O)c(Cl)cc(C#N)cc1Cl.N12C(CC3CC13)CNC2=O c1(C(=O)NC2(CN(C(C3C(C(=O)OC)C3)=O)C)CC2)cccn(O)c1=O CC1=CC(c2ccccc2)=Cc2nc1[nH]c(-c1cccc(Cl)c1)csc2 C(C(CC(C)C)C(=O)NC(C)Cn1cc(C)cn1)NC(C(CCC)C#N)=O c1(Sc2nc(N3CCCC(OC)C3)c(Br)cn2)ccc(C#N)cc1F c1(CC)ccc(C(N2CCC(O)(C(C)NC(=O)CCc3nncn3C)C2)=O)nc1 C1(CNC(c2c(CC)occ2)=O)CC(C)(C)CN1C(=O)Cc1cc(O)nnc1O C1(NC(c2c(OC)cccn2)=O)CN(C(=O)C(C2CC2)OC)CC12CC2 N1(C(C(CC)F)=O)CCC2(NC(C3C(c4ccccc4)C3(C)C)=O)CCCC12 C1(NC(C2N(C(C)=O)CCCC2)=O)CC12CCN(C(=O)CC(C)C(C)C)CC2 c1(-c2nc(Cc3ccc(OC)nc3)nn2C(C)C)cc2ccc(C)cc2nc1Cl c1(C(=O)OC)ncccc1NC(N1CCCC(Cn2cc(C(C)(C)O)nn2)C1)=O CC1CN(C(=O)CC2CCN(Cc3cc[nH]c3)CC2)CC(C)O1 Cc1ccc(F)c(OCC(=O)N(C(CNC(C2CC3CC3C2)=O)C2CC2)C)c1 c1(C(=O)NCCN(C(C2COCC2C(F)(F)F)=O)CC)ncoc1C1CCCO1 C1(CC(=O)NC2C(NC(CCN(CC)CC)=O)CCOC2)CCCC(C)(C)O1 N1(C(c2ccc(CCC)s2)=O)CCC2CCN(C(c3nccc(C)n3)=O)CC2C1 c1(C(N)=O)cc(Br)ccc1NC(C1CC(F)CN(C(c2ccnc(F)c2F)=O)C1)=O c1(SCC(=O)NCC2N(C(C3(C4(C)OCCO4)CC3)=O)CC2)c(F)cccc1F S(=O)(=O)(CC(C)(C)CCC(=O)O)CN1CC2(CN(C3CCN(C(=O)OC)C3)C2)C1 C1(NC(C(c2cccnc2)NC(C(C)C)=O)=O)CC2CC1C(O)C2O c1(NC(c2ccc(F)cc2)C#C)nc2c(F)cccc2o1 c1(C(C(=O)NC2CN(C(C3CC3CF)=O)CC2O)O)ccc(Cl)cc1Br C(C(CNC(=O)CCNC(=O)NC)OC)NC(CSCCCC)=O c1(C(N(C2CCN(C(C3(C)CCCC3)=O)C2)CCC)=O)cc(F)c[nH]1 c1(NCC(COC)C)nc(C)cc(=NCC(C)(CO)c2ccccc2)[nH]1 CC1=NS(=O)(=O)NC=C1C(=O)NC(CNC(=O)CS(=O)(=O)CCOC)C1CC1 c1(OC)cnc(C(N2CCC(C)C2CNC(c2c[nH]nc2F)=O)=O)c(F)c1 C(=O)(CC1=NN(C)C(=O)C1)NC1CCCCCN(C(C=C2CCC(C)CC2)=O)C1 c1(C(=O)NCC2(F)CC(CNC(CC3(C=C)CC3)=O)C2)nc(C2CC2)oc1C c1(CC(=O)N(C2CCN(C(=O)C(C)SCC)C2)CC#C)csc2nccn12 c1(C(CN(C=O)CC)C)ccc(OC(F)F)cc1.C12(CO)CN(C1)C(=O)N2 C1(C)(NC(c2nc(COC)sc2)=O)CCN(C(=O)C2=CSCS2)C1 c1(C(=O)NCC(CNC(C2(C)CCC2)=O)OC)cn(Cc2ccccc2)nn1 N1(C(C(C)(N(C(CSCC)=O)C)C2CC2)=O)CCn2c(cnc2C)C1 C1(NC(c2ccc(SC)o2)=O)C=CCC(C(=O)NCC2(c3ccon3)CC2)C1 N1(C(CC(C)(C)OC)=O)C2CCCC1CC(NC(=O)Cc1csc(Cl)c1)C2 N1(C(CC)C)CCN(C(=O)C(CNC(=O)C(C)(C)NC(C)=O)CC2CC2)CC1 C1(NC(c2cc(C(C)(C)C)sc2)=O)CCCC(NC(C2COCCO2)=O)C1 C1(NC(C(C2CCC2)NC(c2ccc(C(N)=O)[nH]2)=O)=O)CC(F)(F)C1 C1(OC)CC(C(=O)NC2CCOCC2F)N(C(=O)C(C)CO)C1 CC(CNC(C1CC1c1cccc(Cl)c1Cl)=O)CS(N)(=O)=O CC(=O)CCCC(=O)NCC(C(C)C)NC(c1ccccc1C#N)=O C1(NC(c2cn(CCOC)nn2)=O)CN(C(c2cocn2)=O)CC1n1ccnn1 c1(OC)ccc2cc(C(=O)NCC3(NC(C4CC45CCOC5)=O)CC3)nnc2c1 N(C)(C1CCCc2cccnc21)C(=O)NC(C)C(C)Oc1ccccc1 CC1OC(C)C(C(=O)NCC(c2ccc(CO)cc2)O)C1C C1(C)(C(=O)NCCCN(C(CCc2onc(CCC)n2)=O)C2CC2)CC(O)CN1C c1(C(C)C)nccnc1NC(C1CN(CCC2CC2C)C1)=O c1(NC(c2ccc(OC)c(OC(C)C)c2)=O)cc(O)c2ccsc2c1 c1(C(=O)NCCNC(CC(c2ccc(C)cc2)(C)C)=O)c(C)ccc2nonc12 c1(C(c2nn[nH]n2)N(C(CC2CCCC2)C(N)=O)C)ccccc1F c1(C(N2CCC(=CCNC(C(C)N3CCC3)=O)CC2)=O)cnc2c(c1)CCOC2 N1(C(C(CN(C)C)OC)=O)CC(Oc2cccc(Br)c2)C(O)C1 CC(C(C)(C)O)N(C)C(C1CCN(C(=O)C=CC2CCOC2)C1)=O c1(OCCOC(c2c(C(C)C)cnn2C)=O)ccc(Br)cc1Br c1(C(N2C(CC)CN(Cc3ccc(F)cc3Cl)CC2)=O)cc2cccc(C)n2n1 C(=O)(CCCCC(N)=O)NC(C(=O)NC(C1CCOC1)C#C)(C)CSC C1(C(N(C2C(C)C2)C)=O)C2CC2CN1C(=O)CC1CCSC1 c1(NC(c2cccc(-c3ncco3)c2)=O)cccc(Cl)c1C(F)F N1(C(c2c(C)c(F)ccc2)=O)CCC2CN(C(=O)C(C)C(F)(F)C(F)F)CCC12 CC1(C)CCN(C(C2CCC(=O)NC2)=O)C(C(=O)NC2(CO)CC(F)(F)C2)C1 c1(C(=O)NCC2C(C)CCN(C(=O)Cc3cccn3C)C2)cccc2c1OCO2 C(CCCC(C)(C)C(=O)NNC(=O)CSCCF)N(C)C.C1CCCC(=O)O1 c1(OC)ccc(F)c(C(=O)NCCC2COCCN2C(C2CCCS2(=O)=O)=O)n1 C1(C(=O)NCc2n(CC)cnc2)CC(F)(F)CN1C(=O)C(=O)NOC CCC(CCCC(=O)NCC(O)CC(C)C)NC(C1C2CCC(F)C12)=O C(=O)(C1CCCn2nccc21)N1CC(C)CC(NC(c2cnc(C)s2)=O)C1 c1(C(=O)NC2C3(CCN(C(c4c(C)n(C)nc4)=O)C3)C2)cccn2ccnc12 c1(C(=O)NC2CCC(n3c(C)nc(C)n3)CC2)cc(N)c(C)cc1Br c1(CN(C(C(CCSC)NCC2CCCO2)=O)C2CC2)c(C)cccc1Br.C1CC1 C1(NC(=O)CCCC2CCOCC2)CN(C(C2CC=CCC2)=O)CC2(CCC2)C1 c1(C(=O)NC(CNC(C(CC)C#N)=O)(CC)CC)cc2cc(C)cc(C)c2[nH]1 C1(C(N(CC(C)(C)CNC(c2[nH]ccc2C)=O)CC)=O)CCCC(C)CC1 C(=O)(C(CCC(C)C)NC(C)=O)NCC(=C)CCNC(=O)C=CBr C(C(N)=O)(C(C)(C)C)ONC(c1c(C)n(-c2ccccc2Cl)nn1)=O C1(CNC(C(=O)NC(C)C)=O)CN(C(=O)C(N)CCC(N)=O)CCC12CCOC2 C=CCC(C(=O)N1CCC(C)(CCNC(=O)C=Cc2ccccc2)C1)NC(C)=O c1(CN2CCN(C(c3ccc(C)c(O)c3)=O)C3C2C3)cnc2ncccn12 C1(SC)COCC1NC(=O)C(C1CCN(C(=O)C=CC(F)F)C1)F NC(=O)CCC(C(=O)NCC1(c2cn(CC3CCC(=O)O3)nn2)CC1)n1ccnn1 C1(NC(C(CSC)(C)C)=O)CCN(C(c2nn(C)c(N)c2C)=O)CC1C c1(C(=O)NCC2CC(NC(C(=O)NC3CC3)=O)C2)cc(-c2cnccn2)[nH]n1 N1(C(C2C(CC)OCC2)=O)CC=C(C(C)(C)C(=O)NC(C2CC(F)(F)C2)C)C1 C1(C(N2C(C)C(NC(=O)Cc3ccncc3Cl)CC2)=O)CN(S(N)(=O)=O)C1 C1(O)(CNC(C2CCCS2)=O)CCCN(C(=O)C(O)COCc2ccccc2)C1 c1(C(CC)O)cn(CC)nn1.C12CCCN1C2.c12ccnn1C(C)C(=O)NC2=O N1(C(C23CC(OC(C)=O)(C2)C3)=O)CCN(C(C2CCc3n[nH]cc3C2)=O)CC(O)C1 Cc1cc(F)c(CC(=O)NCC2CN(C(C3CCSC3)=O)CC(C)(C)C2)cc1F c1(C(=O)NC(C(C)C)CNC(=O)CCCCCNC(N)=O)cccc2nn(C)cc12 N1(C(Cc2ccc(C)cc2)=O)CCOC2(CCN(C(=O)C(O)C(C)(C)C)C2)C1 N1(Cc2c(CC)cccc2)CCC2CN(C(C3CCNC(=O)C3)=O)CCC12 CCC(CC)C(F)C(=O)N(C1CCN(C(=O)Cn2cc(C(C)O)nn2)C1)C c1(C(N(C(C)CCNC(=O)COCc2ccccc2)C)=O)ccnc2[nH]ncc12 C(=O)(N(CCC(=O)NC1CCCC(CC)C1)OC)c1ncc(CC)cn1 C(C(=O)C1CCOc2ccccc21)OC(CCn1nc(C)c(Cl)c1)=O C#Cc1ccc(CNC(=O)C(=O)NC(C2OCCC2(C)C)C)cn1 CCCN(OC)C(=O)CN(CCc1cc(C2CCC2)cc(OC)c1)C(C)C C(=O)(C1CNC(=O)c2ccnn21)NCCNC(CCC1C(C)(C)C1)=O C=CC(C)(C)C(=O)NC(CCN(C(=O)C(C)Oc1cccnc1)C)c1cccs1 C1(C)(c2onc(C)n2)CCN(N2CCCC(c3nccc(CC4CC4)n3)C2)C1 C1(CC(N2CC(CC#C)OCC2)=O)CN(C(=O)CCC(C)=O)C(C)(C)C1 c1(C(=O)NCC(CNC(C(CC(=C)C)C)=O)F)cc(F)c(F)cc1F C1(NC(C2C(CC)N(C(=O)CC(C)CC(C)C)CC2)=O)CC2COCC(C1)C2 c1(OC)ncc(CN2CCC(C(C)C(=O)Nc3cnccc3OC)CC2)cc1Cl C1(N(C(C2N(C)CCC2)=O)C)CC2CCC(C1)N2C(=O)CNC(=O)CN(C)C CCC(CC)C(F)C(=O)N1CC(F)(C(N2CC(CC)OC(C)C2)=O)C1 c1(C(C)C)cccc(C(N2CCC(NC(=O)CCc3cncs3)C(F)C2)=O)c1N C1(C(=O)NC(C23CC(CO2)C3)C)COC2(C1)CN(C(=O)CCCC1CC1C)C2 Cc1nc(C)c(CC(=O)NCC2(C)CC(C(=O)NCC(CO)N(C)C)C2)s1 Cc1c(C(N2CC(SC(F)F)C2)=O)cnn1C1CCOCC1 C1(O)(C(=O)OCC)CCN(C(C2C(C)(C)C2(C)C)C(=O)NCCOC)C1 C1(CNC(c2cn(CCC)nc2)c2nnnn2C(C)C)CCC2(CC2)C1 C=CC1OCCCC1C(=O)NC(C)(CNC(c1ccnnc1O)=O)CO C(=O)(C1CCc2cc(Br)ccc21)NC(C(C)(C)NC(C=CC(C)C)=O)C c1(NC(c2ccc(C(C)C)cc2)c2n(C(CC)C)nnn2)c(SC)cccc1C c1(C(N2CC(C)OCCC2)=O)cc(S(=O)(=O)N2CCSCC2)c[nH]1 C(=O)(C(C)(C(F)F)c1ccccc1)N1CCC(NC(Cc2c(C)non2)=O)CC1 C1(CNC(C2(COCC)CC2C=O)=O)CN(C(=O)C2=COCCO2)CCC1C CC(C)C(O)C(F)(F)C(=O)NC1CCC(NC(=O)C(F)C(F)(F)F)CC1 C1(C2CCN(C(=O)CC3(C=C)CCCCC3)CC2)(NC(C2(CC#C)CC2)=O)CC1 c1(C(N2CC3CN(C(Cc4cc(C)on4)=O)C3C2)=O)cc(Br)cc([N+](=O)[O-])c1Cl C1(C(=O)NC(COCC)C(=O)N(C)CCOCCN(C)C)CC1C1(C)COC1 C1(NC(=O)CC2CCCCC2)CCN(C(C2CC3(CC3)CO2)=O)CC12CCC2 C1(C)(COC)CC(NC(c2ncc(C(F)F)s2)=O)CN1C(=O)Cn1nnnc1C CC1CCCC(O)(C(=O)NC2(CNC(=O)CCF)CCCC2)CC1 c1(N(C)C)ccc(C(=O)NCCC2(NC(C3CCC(=O)O3)=O)CCC2)nc1 C(CCCCC(=O)NC(C)(C)C(N)=O)N(C)C(c1cc(O)nc(O)n1)=O c1(C(CNC(c2c(C)ncs2)=O)NC(=O)C(O)CC2CC2)ccc(F)cc1F CCC(C(=O)NCC(C)NC(=O)C(C)(C1(C)CC1)OC)n1cncn1 C1(C(N2CCC(C)C2CNC(C2CCCN2C=O)=O)=O)CCc2nnc(O)n2C1 c1(OC)ccc(F)c(N)c1C(=O)NC1CCCCN(C(=O)C#CC2CCCO2)C1 Clc1cc(Br)c(C(c2nnnn2CCCC2CC2)NCC2CC23CCC3)s1 c1(C(C)=O)ccc(NC(=O)C(C)NC(Cc2ccccc2Cl)C(=O)O)cc1Cl c1(CC(N2CC(CC(=O)NCC(C(=O)OCC)O)(OC)C2)=O)ccnc(O)c1 C(C(C)C(=O)NCCOC1CN(C(=O)CCCc2nccs2)C1)SC c1(C(N2C(CNC(CCCC(C)=O)=O)CN(C)CC2)=O)cn(C)c(=O)nc1O N1(C(C(CCC)C)=O)CCc2c(-c3ccc(F)c(F)c3)cccc2C1 N1(C(C2CC(C#C)(O)C2)=O)CCC2(CC1)CC(C)N(C(c1coc(CC)n1)=O)C2 c1(N2CCC(CC=C)(N(C(=O)CCN(C)C(C)=O)C3CC3)C2)ncnc2scc(Br)c12 Cc1cc(NC(=O)C(=O)NCCC2CCCN2C(=O)N(C)C)c(C)o1 c1(C(C)CC(=O)NCC(CO)NC(C2SCCS2)=O)c[nH]c2ccccc12 c1(NC(CC2CC3(CN(C(CCOC)=O)C3)C2)=O)cc(F)c(O)c(F)c1 C(C1=CCN(C(=O)C=Cc2ncco2)CC1)NC(=O)CSc1ccccn1 N1(c2onc(-c3cnn(C)c3C(F)(F)F)n2)CC2CCCC(C1)C(=O)N2 C1(C)(C(=O)NC2C3CC(NC(C4C(C)(O)CCC4)=O)CC32)CCCCNC1=O c1(CC)c(C(=O)NCC2C=CCN2C(=O)CN2CC(C)C2)cnc2ncnn12 O=S(=O)(c1ccc(N2CCC(CCO)C2)cc1Br)NCCN1CCCCC1 c1(C(=O)NCCN(C(C2CCC(C)=C(C)C2)=O)CC)c(N)c(C(F)(F)F)nn1C n1(CC)cc(C(N2CC(NC(c3occc3C)=O)CC2C)=O)c(C(C)(C)C)n1 N1(C(C(CC2CC2)NC(C2CC3(CCO2)CC3)=O)=O)CC2(CCC1CO)CC2 Cc1cc(=O)ccn1CC(N1CCN(C(c2cnc(S)n2C)=O)C(CCO)C1)=O c1(C(=O)NCCC(C)N(C(=O)C(CC(F)F)C2CCC2)C)ccc2cncn2c1 N1(C(c2c(C)ocn2)=O)CC(CC(=O)NC2CCCC2(F)F)CC1(C)C CCC1=C(C(=O)N2CCCC2C2(O)CN(C(C3CC(C(C)C)=NO3)=O)C2)CCCO1 c1(C(N2CC3C(NC(CP(C)(C)=O)=O)(CCC3)C2)=O)ccc2c(c1)CCC2=O Cc1cc(C(=O)NCC2CC(NC(=O)COCCN(C)C)C2)ccc1Cl CCCCC(C)(F)C(=O)NC(CNC(=O)C(C)Sc1ccc(F)cc1)C(C)C N1(C(C(COC)(C)OC)=O)CC2(CC(NC(c3cc(Cl)ccc3N)=O)C2)C1 N1(CCC)C(=O)CCC1C(=O)NCCOCCN(C(=O)C(CC)SC)C Cc1cc(F)ccc1S(=O)(=O)N1CCC12CCN(C(=O)CCC1CCC1)CC2 C=C(Cl)CC(C(=O)NCC(C)(O)CCCC)NC(=O)Cc1cnns1 c1(C(=O)NC(CCCCNC(C(CC(C)C)F)=O)C)cc(S(N)(=O)=O)co1 C1(CNC(c2c(CC)onc2)=O)CCC2(CCC2)C1NC(=O)CCn1ccnn1 c1(C(=O)OCC)cnc(NC(=O)C(=O)NCC(C)C(C)O)c2cncn12 c1(OC)cc(O)ncc1C(N1CC2CC2(CNC(C2CC3(CC3)CO2)=O)C1)=O C1(CNC(C2OCCN(C(c3c(C)cc[nH]3)=O)C2)=O)CCOC(C)(C)C1 c1(OCC(=O)NC(CN(C(=O)COC2(C)CCCC2)CC)C)ccc(F)cc1F C(=O)(CCCC(=O)NC1(CNC(=O)C(C)(O)C2CC2)CCOC1)OCC C12(C(N3CC(F)(C(=O)OC)C3)=O)CC(CO1)N(C(=O)CSc1nc[nH]n1)C2 C1(CNc2ncnc(N3CCC4(CCCO4)C3)c2)CC2OC(C)(C)OC2C1 C(=O)(C1SCCc2sccc21)N(C)CC1CCCN(C(=O)C(N)=O)C1 C=CC1CN(C(C2CC3C=CC2CC3)=O)CC1NC(=O)COCCCCC c1(CC(=O)NCC(C2CCN(C(=O)Cn3cccc3)CC2)O)ccc(F)nc1 C(=O)(C(CCNCCC(C)(C)CSC)NC=O)OCC C1(C)(C(=O)NC(C)CN(C(=O)C(F)=C2CCCC2)C)CCCCO1 C(=O)(C(C1=CCSC1(C)C)N1CC(=O)NCC12CCC2)NCC=C c1(C(CC)(C)NC(c2ccc(CC(C)C)cc2)=O)ccc(Br)c(F)c1 C1(O)(C(C2CCCC2)NC(=O)NCCCC#C)CCCCC1 N1(C(c2cn(CC(N)=O)nn2)=O)CC(C2CN(C(=O)CC3(O)CCC3)C2)C1 N12CC3(CCC(O3)C1=O)C2.N1(CC(C)N(C(=O)C(F)(F)F)CCCl)C(=O)CCC1=O c1(C(N2CCC(CNC(=O)CC(O)c3ccccc3)C2)=O)c(O)cccc1Br N12CCC(CC1)NC(C)C=CC2=O.C(=O)(CCN(C)C)NCCO C(C(C)(C)CC(=O)N(C(c1ncccn1)C)CC1CC1)OC.C12(CCC1)C(=O)N2 c1(CC(=O)NC2CCN(Cc3nc(CC)on3)C(C)C2)c[nH]c2c(C)cccc12 C1(C(=O)NCC(c2nccs2)C)CC2CCCC2N1C(=O)C1=COCCC1 CCC(O)C(=O)NC1CCCC1NC(=O)CCc1nnc(C(F)F)o1 c1(C(N(C2CC(C)OC2=O)C2CC3(CC3)C2)=O)ccc(Cl)c(Cl)c1 C1(C)(C(=O)NC(C)C(CO)NC(=O)CCC2CCOCC2)CCCCO1 c1(C(=O)NCCC(=C)CNC(=O)C2=CC3C=CC(C2)C3)ccnc2ccccc12 c1(CC)cc(C(=O)NC(C)(CNC(=O)CCOC)C2CC2)ccc1F Cc1nc(O)ccc1C(=O)N(CC(C)N(C)C(c1cn(C)nc1Cl)=O)C C1(NC(C2C3(CC(NC(CCSC)=O)C3)C2)=O)CN(C)CCC1O c1(C(=O)NC(C2CCN(C(C(CC)=CC)=O)C2)C)nccc2ccncc12 C1(OCC)(OC)CC2(CCN(C(CC3COC(C)(C)O3)C(=O)Nc3cccs3)C2)C1 C12(COC)CC(CNC(=O)CCOC)(CN1C(=O)CCN1C(=O)CCC1=O)C2 C1(CC(=O)N(C2CCN(C(=O)C(C)N(C)C)C2)CCC)CCCOCC1 CC1CN2CCN1C(C(=O)NC1CCC(CNC(=O)C(C)(C)CO)C1)C2 C12(CNC(c3c(C)sc(Cl)n3)=O)CCCCC1CN(C(=O)C(F)(F)C(C)O)C2 C12(C(=O)NCCN(C(c3cn(C4CCOC4)nn3)=O)CC)CCC(CC1)C2(C)C c1(NC(C2(F)CCN(C(C3CCC(=O)N3)=O)C2)=O)c(F)cc(Br)cc1Cl N1(C(CN2CCC(OC)C2)=O)C2CCC(C2)C1C(=O)NC(c1ncn(C)n1)C C1(F)(C(N2CCC(CC=C)(NC(=O)Cc3nnc(C)n3C)C2)=O)CCS(=O)(=O)C1 CCC(CC)CCCN(C(=O)CN(C(=O)C(CSC)OC)C)C N1(C(c2c(CNC(CCCOCC)=O)occ2)=O)CCC(C)C1C c1(N2CC(CCNC=O)(OC)C2)ncc2c(n1)COC2.c1(CN)cccc[n+]1[O-] C(CCC1CC1)(C(=O)N(C)Cc1cccc(C)c1)NC(C=CC(CC)C)=O Cc1nnc2n1CCCC2C(=O)NCC(F)CNC(c1cccs1)=O CC(C)C(C(=O)NC1CN(C(=O)Cc2cncc(C(F)(F)F)c2)CC1C)NC=O C1(C(=O)NC2CCCN(C(CC3C(CC)C3)=O)C2)CCCCCN1C C1(S(C)(=O)=O)(C(=O)NC(CN(C)C(C2CC2CF)=O)Cc2ccccc2)CCC1 Cc1[nH]nc2cc(C(=O)N(C)CCN(C)C(C3(Cl)CC3)=O)ccc12 c1(CC(=O)NCC2CC(CNC(C3C(C(=O)OC)C=C3)=O)C2)cccc([N+](=O)[O-])c1 c1(C(N2CCC(C)(NC(c3cc(CC)c(F)cc3)=O)C2)=O)ccn2c1CSCC2 C(C1CCCCC1)=CC(=O)N(C1C2CN(C(C3(C(F)F)CCOCC3)=O)CC12)C N1(C(c2c(=N)[nH]cnc2)=O)CC2(C1)C(NC(c1ccsn1)=O)CCS2(=O)=O N12CCN1C(CC(F)F)C2.N1CCOCC1.C(CC=O)SCC(N)=O N1(C(CCCOC)=O)CCC(CNC(=O)C2=COCCC2)C12CCC2 N1(C(C2SCCCS2)=O)CCC(OCCNC(C2(C(O)C(F)(F)F)CC2)=O)CC1 c1(NC(C2C(C)CCN2C(C2CCC3CC23)=O)=O)ccc2ncnn2c1 N1(C(=O)OCC)CCC(c2ncc(C(=O)NC(C)CO)s2)CC1 C(C(C)(O)CCOC)NC(=O)CS(=O)(=O)NC.C=CC1C(=O)O1 CCCC(C)(C)C(=O)N(CC(=O)N(C)Cc1cn(C)nn1)C C(c1ccccc1Br)=CC(N1CCN(CCNC(C(C)(C)OC)=O)CC1)=O c1(OC)ccc(CC(=O)N(C)CC2CN(C(C3CC(NS(C)(=O)=O)C3)=O)C2)cc1 C(CC(C)C)(C(=O)NC1CC(C(CO)NC(=O)CC2CNC(=O)O2)C1)NC(C)=O C1(C(N(CC(=O)NC(c2ccns2)C)C(C)C)=O)CC2CCC1O2 c1(OC)cc2c(O)cccc2cc1C(=O)NNc1cccc(C(F)C(F)(F)F)n1 CCCCCCC(=O)N1CCC(C)(C(=O)NCCC2CCCCC2O)CC1 Cc1ccc(=O)n(CC(=O)NC2CCC(CNC(=O)CCCC(N)=O)C2)c1 c1(OC)c(C(N2CCCC(O)(CNC(=O)Cc3cncnc3)C2)=O)ccc(F)c1F C(=O)(C1=COCCC1)N1C(C(=O)NC(C)(C)CN2CCCCCC2)CSCC1 c1(CC)ncc(Cl)c(C(N2CC3CCC3(NC(=O)C(C)C(C)C)C2)=O)n1 C1(CNC(C=CC)=O)CC(O)(CNC(=O)C(c2cnn(C)c2)SC)C1 N1(C(C2CN(CC)C(=O)C2)=O)CCCC2(CNC(c3cscc3F)=O)CCCC12 c1(OC)ccc2c(=NC(C)N3CC=CCC3)[nH]c(N3CCC(C)C3)nc2c1 Cc1nccc(C(=O)NC2CCC(NC(=O)C(C)(C)n3cnnn3)C2)n1 C(=O)(C(C)(C)CCNC(=O)CC1CCSC1)NC(c1c(C)nccn1)C Cc1cc(C(=O)NCCCCC(CO)NC(C2CC(C)(C)CN2C)=O)cc(O)n1 C1(C(=O)OC)CN(C(=O)C=CC(C)NC(=O)CC2OCCC2C)CC(=O)N1 C(=O)(C(C)(C)CC(F)F)NC1C(CC)CN(C(=O)C=Cc2cnn(C)c2)C1 C#Cc1ccc(CCC(=O)N(C2CCN(C(=O)C(CC)C(C)C)C2)CCC)cc1 c1(C(=O)NC2C(F)CCN(C(c3n(C)c(S)nc3)=O)C2)cnc2c(n1)CCCC2 N1(C(C(COC)N(C)C)=O)CC(O)CC1(C)C(=O)NCC1CC[Si](C)(C)C1 c1(OC)nc(C(=O)NCC=CCNC(=O)COc2ccc(F)cc2C)cc(O)n1 O=C(CCCc1nccs1)NCC1(c2ccccc2)CCCO1 c1(C(N2C(C(N(CC(F)F)C)=O)CC2)=O)cn(C)cn1 C1(OC)CC2CCCCN2C1NC(=O)NCC(F)CO c1(-n2cc(CN(C(=O)C(F)n3ccnc3)C)nn2)ccc(F)cc1Br C1(NC(CCOCCC)=O)CCOCC1NC(=O)Cc1cnsc1 N1(C(C(=O)NC(c2ncc(C(=O)OCC)s2)C)=O)CCCCC1CCO C1(C(=O)NC(C(C)(C)NC(c2c(C)c[nH]n2)=O)C)CCCN(Cc2ccncc2)C1 C1(CC=C)(NC(=O)C(C)CC=CCC)CCCN(C(=O)CN2C(=O)CCC2=O)C1 c1(NC(C2(CC=C)CCCC2)c2nnnn2CC)cnc(OC)c(C2CC2)c1 C(=O)(C(F)C(C)CC(C)(C)C)NC(CC)CN(C)C(C1Cc2ccccc2O1)=O C1(C(=O)NCC2(C#C)CCC2)(NC(=O)C(CN(C)C)CC)CCCCC1 N1(C(c2ccc(Cl)[nH]2)=O)CC2=C(C1)CN(C(c1cnc(C(F)F)cn1)=O)C2 C(CC(=O)NCC1CCC(=O)NC1C)(C(F)(F)F)NC(C(NOC)=O)=O N1(C(C(CC)F)=O)CC2CC1CCC2NC(c1ncn(-c2ccccc2)n1)=O C(=O)(CC1=CCOCC1)N(C(C)C(=O)NCC1(C)CCCC1O)CC c1(N2CCC(N(C(=O)C(=O)Nc3ccc(C)cc3)C(C)=O)C2)cc(C)ncc1CO c1(C(=O)NCC2(F)CC(NC(CN3CCC(C)(O)C3)=O)C2)ccc2c(c1)NCC2 C(=O)(C(O)CCNC(=O)C(O)C1CCC1)NC(c1ncc[nH]1)C C1(CCn2ncc(C)c2)CCN(C(=O)C(=O)NC2CCC(C)N2)CC1 N1(C(c2ccc(CC)o2)=O)CCOC2CN(C(C3CCOC4(CCC4)C3)=O)CC12 c1(-n2ncc(C(N(C3CC(NC(CCN(C)CC)=O)C3)C)=O)c2)ccccc1F C1(NC(c2cnsc2)=O)CCC2(CC1)CN(C(=O)CN1C(=O)CCC1=O)CCO2 N1(C(C(C)=C(CC)C)=O)C2CC1CN(C(c1ccccc1Cl)=O)C2 n1(CC)nc(SCc2ccccc2)nc1-c1ccc(F)s1 C1(C(N(CC(C)NC(c2c[nH]nc2C(F)F)=O)CC)=O)C(C)(C)C1(C)C N1(C(c2c(SCC)n[nH]c2)=O)CCC(C(=O)N(C(C)C(=O)OC)C)CC1(C)C C1(C(=O)N)CCn2ncnc2C1.C12(CCC1)C(=O)N(C1CC1)CCCS2.CCO Cn1c(C(=O)NC(CO)CCCCNC(c2cc(O)cs2)=O)cc2sccc12 N1(c2ncc(CC)s2)CC(c2ccc(Br)cc2)CCC1=O C1(C(=O)Nc2cccc(CF)c2)Cc2ccccc2C(=O)O1 CCCC(C(=O)N1CC(NC(=O)CCc2ccnc(Cl)c2)C(O)C1)OCC1CC1 c1(NC(C2OCCN(Cc3c(OC)cccn3)C2)=O)c(C#N)cnc2ccnn12 CN1CC(O)CC1C(=O)NC1CCC(C)(CNC(=O)Cc2cn[nH]c2)C1 c1(C(N2CC3(CN(C(c4ccc(CC)cc4)=O)C3)C2)=O)cc(C)ccc1[N+](=O)[O-] C1(NC(C(C)(C)NCC2CC3C=CC2C3)=O)C2CC3CC1CC(O)(C3)C2 Fc1cc(F)c2[nH]c(=NCc3ccc(Cl)cc3)[nH]c(=NCC(Cl)=CCl)c2c1 C(=O)(CCCC(C)(C)C)N1C(CNC(C2(C)C(C(=O)OC)CC2)=O)CCCC1 CC1=C(C(=O)N2CCC(C)(CC(=O)NCCC(CC)CO)C2)COCC1 C(=O)(C1=CCCS1)N1CCC(C(C)(C)NC(=O)CSCC2CCOCC2)C1 N1(C(c2cc(OC)ncc2F)=O)CCC2(NC(=O)CCC3CC3(Cl)Cl)CCCC12 CC(C(=O)NCCC1(C(=O)NC2CC(C(F)F)C2)CCCC1)S(C)(=O)=O c1(OC)ccc(Br)c(C(N2CC3CCC2CN3Cc2cnc(C)cn2)=O)c1F C1(CC=C)(NC(C2(CC)CC2)=O)CCCN(C(=O)C(C)Cc2ccc(F)cc2)C1 C(=O)(CCC(F)(F)C(F)F)N1CCC(NC(c2cc(OC)no2)=O)C(CO)C1 c1(NC(C2N(C(C3CC=C(C)CC3)=O)CCOC2)=O)ccc(CN(C)C)cc1C c1(OCC)ccc(C(=O)NC(C2CN(C(=O)C(C(C)C)NC=O)C2)C)cc1 C(C(C)NC(C1(C(=O)CN(C=O)C2CC2)CC1)=O)OC.C(C(C)C)CN(C)C C1(NC(c2ccc(C)[nH]2)=O)CCN(C(C2(C)CC2(F)Cl)=O)CC1F N1(C(C2(C(C)(C)C)CCC2)=O)CC2C(CNC(C3(C)CCCCC3)=O)C2C1 C=CCCCC(C)(C)C(=O)NC(CCC)CC(N1CCCC2(CCCC2)C1)=O CCCCCCC(C)C(=O)N1CCCC(CC(=O)NCC(C)(C)CSC)C1 CON1CCC(CC(=O)N(CC(C)N(C)C(C2C(F)(F)C23CCC3)=O)C)CC1 CC(C)CCCCCC(=O)NC1(C(N2CC(c3nc(=O)o[nH]3)C2)=O)CCOCC1 C(C1CN(C(=O)C=C2CCC2)Cc2ccccc21)NC(C1(COC)CC1)=O C#CCCCCCCC(=O)N1CCN(CCNc2ccc([N+](=O)[O-])c(Br)c2)CC1 C(C)(C(=O)NC1CCC1CNC(=O)Cc1cnoc1)(C1CC1)NC(C)=O c1(NC(C(C2CCCC2)NC(CCCC#C)=O)=O)ccc2ncnn2c1 C1(NC(c2c(C(C)(C)C)ocn2)=O)COC2(C1)CN(CC1CCCOCC1)C2 C(=O)(CC(C)C1CC1)NCC(C)N(C)C(c1csc(-c2ccsc2)n1)=O c1(C(N(C2CC3N(C(C(CC)(C)O)=O)C(CC3)C2)C)=O)ccc2c(C)[nH]nc2c1 CC1(NC(C2CCCC2(F)F)=O)CCN(C(c2ccc(-c3cccs3)[nH]2)=O)CC1 c1(C(=O)OC)cc(NC(=O)C(=O)Nc2cc(F)c(O)c(F)c2)cc(F)c1F CCC(C)(CNC(C1(F)CCN(C(C2(SC)CCC2)=O)C1)=O)CO N1(C(C(CC(F)F)NC(C2CC(CCC)C2)=O)=O)CCOC2COCC2C1 Cc1cc[nH]c1C(N1CCC(n2cc(Cl)cn2)C1)=O C1(O)(CNC(CC(=C)Br)=O)CCCN(C(c2ccc(C)n(C)c2=O)=O)CC1 N1(C(c2c(N)c3c(cn2)cccc3)=O)CCN2CCN(C(=O)CC3CC3)CC2C1 c1(C(N(C(CNC(COCCCC)=O)C)C)=O)cnn(CCN(C)C(C)C)c1C CC1=C(C)CC(C(=O)NC2CC3(C2)CC(NC(c2cc(Cl)cnn2)=O)C3)CC1 C1(CCNC(C2CC(CCC)C2)=O)CCN(C(=O)CCOC(C)C)C1 C#CCC(CC(F)F)NC(=O)CN(C(=O)C(C1CCOCC1)O)CC(C)C c1(OC)ccc(NCCN(C)C(=O)NC(c2ccsc2C)(C)C)cn1 N1(c2snc(CC)n2)CCC2CCN(C(C3CC(C(C)C)C3)=O)CC2C1 N1(C(C2N(CCC)CCC2)=O)CC2CCC(NC(c3ccc(=O)oc3)=O)(C2)C1 N1(C(CCOC(C)C)=O)CC(NC(C2CCNC2=O)=O)C(C(F)(F)F)C1 C1(CCNC(C(COC)O)=O)CCCCN1C(c1csc(C(N)=O)n1)=O C1(NC(CSSC)=O)CN(C(c2cnn3cccc(Cl)c23)=O)C2(CCOCC2)C1 Cc1c(C(=O)NCC2CN(C(C3(N=[N+]=[N-])CC3)=O)C2)cc(C2CCCC2)n1C C1(C(=O)NCC(C2CCN(C(c3ccc(Cl)o3)=O)CC2)(C)C)CCCOCC1 C(C(N)=O)(C(N)=O)NC(c1c(CNC(CC)=O)ocn1)=O C(CC(C(=O)NC1C2CCC1CC2)NC(=O)CC1CSC1)=CC N1(C(c2c(COC)cco2)=O)CCCC(C)C1CNC(=O)C(C)C(F)(F)F C1(NC(C=CCN(CC)CC)=O)CN(C(c2cnnn2C)=O)C2(CCOC2)C1 C#CC1(C(N2CCC(CO)C(O)C2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1 CCCCS(=O)(=O)CC(=O)NC1CCCN(C(=O)CC2CC2(C)C)C1 C12(CNC(c3nc(C(C)C)sc3)=O)CC1CN(C(C1(C)CC(C#N)C1)=O)C2 c1(OC)ccc(C(N2CCC(CN(C)C(C3CC(S(N)(=O)=O)C3)=O)C2)=O)cc1O c1(CC)n[nH]cc1C(=O)NC1(CNC(c2coc(CN3CCCC3)c2)=O)CCC1 c1(C(N2CC(C(C)NC(C3CC(C(F)(F)F)C3)=O)OCC2)=O)ccc(F)cc1Cl c1(OC)nccc(C(=O)N(CC(C)(C)CNC(C2CCCC(C)C2)=O)C)n1 N1(C(C)C)CCCN(C(C2CCCCN(C(=O)C(c3ccccc3)C)C2)=O)CC1 c1(C(=O)NCCCN(C(=O)Cc2cnccn2)C)cnc(P(C)(C)=O)cn1 C1(C(N2CC(C3(CNC(CCC(CC)C)=O)CC3)(O)C2)=O)CC2(CCCCC2)C1 C(C(C)(C)CS(C)(=O)=O)NC(C(=O)NC(CC(C)C)C(N)=O)=O C1(C(N2C(CN(C(=O)CCC(C)(C)C)CC)CCC2)=O)C(O)C(=O)N(C)C1C C1(C2CCN(C(C3CCC3)=O)CC2)(NC(C(C)Cc2ccc(F)c(Cl)c2)=O)CC1 CCS(=O)(=O)C=CC(=O)N1CCOC(CN(C(=O)C(F)C2CCC2)C)C1 N1(C(c2ncc(C(C)C)nc2)C(=O)NCC2COC2)CC(C)CC(C)C1 C1(NC(C(c2cccc(F)c2)(C)C)=O)COC2(C1)CN(C(c1cc(O)cs1)=O)C2 N1(C(CCC2C(C)=NOC2=O)=O)CCCC(NC(C2(n3cnnn3)CC2)=O)C1C C1(C(=O)NC2C(CNC(CSCCCC)=O)C2)CCc2cnnn2C1 N1(C(c2cnc(Cl)cn2)=O)CCN(Cc2c(Cl)cc(Br)cc2Cl)CC12CC2 C(C(O)CC(=O)NCC(C1CCN(C(c2cc(CO)ccn2)=O)CC1)F)N(C)C C1(NC(COC(C)=O)=O)CCCCCC1C(=O)NC(C)(C)CCF C(=O)(C(C(C)C)N(C(c1cnn(C2CC2)c1)=O)C1CC1)N(C1CCN(CC)C1)C N1(C(C2(CC)CCCCC2)=O)CC2CN(C(=O)C3=COCCC3)CCC2(CO)C1 C1(COC)CN(C(C2CC(c3cccc(F)c3)C2)=O)CCN1C(=O)C1=CCOC1 C#CC(CC(C)(C)C)NC(=O)CC1(CNC(=O)C(O)Cn2cncn2)CC1 C1(C(=O)NCCCC(=O)NCCC(C)(O)C2CC2)CCCC(=O)CC1 S(=O)(=O)(c1ccc(NCC(C)C)c(F)c1)NCc1c(C)nc(C)s1.C12CN(C1)C2 Cc1cccc(C(CNC(C2CC(=O)N(C)C2)=O)NC(c2csc(O)n2)=O)c1 CCCCCC(O)C(=O)NC1CCN(C(C2(C(N3CCCC3)=O)CC2)=O)C1 c1(C(=O)NC(CCCNC(C(C)OCCC=C)=O)(C)C)nc(Cl)ccc1OC N1(C(CNCCC)=O)CCc2ccsc2C1C CC1CCCC(C)N1NC(=O)C1CCO1.C1(OC(C)(C)C)CCCN1C(=O)O CC1NC(=O)CCC1NC(C12CC(CO1)N(C(=O)CCS(N)(=O)=O)C2)=O C1(n2cc(C3CCN(C(=O)CC45CCCC4C5)C3)nn2)CCC(F)(F)CC1 C1(O)(C(C)NC(C=COCC)=O)CCN(C(c2c(C(F)(F)F)coc2C)=O)C1 CCN=c1[nH]cc(C(N2CC=CC2CNC(C2CCN(CC)C2)=O)=O)s1 c1(C(N)=O)ccc(CNC(c2n[nH]cc2NC(=O)COc2ccsn2)=O)cc1 C(CC(C)(C)C(=O)NCCOC1CCN(C(=O)CCCCO)C1)OC c1(N2CCOCC(NC(CC(CC)(C)C)=O)C2)nc2c(cc1C#N)CCC2(C)C N1(C(C2C(C)=C2)=O)CCC2(CCCCN(C(=O)C(N3CCC(O)CC3)C)C2)C1 C1(CC=C)(NC(c2ccns2)=O)CCCN(C(=O)C(C)COC)C1 N1(C(CCCC(C)=O)=O)CCCC2(CCCN2C(c2csc3ccccc23)=O)C1 CCC(C)CCCC(=O)NC(C)C(N1CCNC(=O)C1C)=O c1(Cc2ncc(N)nc2)ccc2cccc(-c3ccccc3)c2n1 N1(C(COCCOCCOC)=O)CCC(C(C)COC)C1.C12CC(C1)NC(=O)C2 c1(CC)ccccc1OCC(=O)NC12CC1CN(C(=O)CN1CCCCC1=O)C2 c1(C(=O)NC(C2CC2C(N2CC(F)CC(F)C2)=O)C)cnccc1C#N C(=O)(N(CCC(=O)NC1CC2(CCC2)C1O)OC)C1C(C(=C)C)OCC1 C1(NC(c2c(CC)nn[nH]2)=O)CC2CCC1CN2C(c1ccc(Cl)s1)=O N1(C(CCCc2cc(C)sc2C)=O)CCCCC(CNC(=O)C2=NNC(=O)C2)C1 C#Cc1cc(N(CCN2CCOC(C)(COC)C2)C2CC2)cc(N)c1 c1(CC2(C(=O)OC)CC2)cccc2ccccc12.C1C(=O)N1CCOC C(=O)(C1=CCCOC1)N(C(C(=O)NCCC=CCCC)CC)C c1(C(C(N2CCN(CCCNC(C=CCOC)=O)CC2)=O)C)c(F)cccc1F C1(C(=O)NC2C(NC(C(CCC)C)=O)CCC2)CC2CCC(C1)C2=O c1(C(=O)NC2CC(CNC(C3(OCC)CCC3)=O)C2)ccc2c(C)noc2n1 CC(O)(CC(=O)N1CC(N2CCN(C(C3CN(CC(C)C)C3)=O)CC2)C1)C1CC1 C(=O)(C(CNC(=O)C(O)CN1CCCC1)NC(c1cc(Br)no1)=O)OC N1(C(C(C)SCC)=O)CCC2(CC2)CC1C(=O)NCC(=O)N(CC(C)C)C1CC1 CC1CCCC(C)N1C(=O)C(=O)NCCCOCCNC(=O)Cc1c[nH]nc1O c1(C(=O)NCCC(C)NC(Cc2ccc(C)c(O)c2)=O)cc2ccc(O)nc2s1 C1(CC#C)(C(=O)NC(C2CCN(C(=O)CCN(C)CCO)CC2)C)CCCCC1 N1(C(c2c(NC)nccc2)=O)CC(CO)C2(C1)CN(C(C1CC(C(F)F)C1)=O)C2 C1(CCC)(NC(C2CCCOC2)=O)CCN(C(C2CCCOCC2)=O)CC1 c1(NC(C(=O)NCCN(CCC)C2CC2)=O)cc2c(cn1)C(=O)CCC2 C1(NC(Cc2c(C)ncs2)=O)CCN(C(C2(CO)CC2(F)F)=O)CC1O c1(CC(=O)NC(CC=C)CNC(=O)CC2CCSC2)c(Br)cnn1C c1(C(=O)NCC2CCCC(NC(C3CC(O)(CC#C)C3)=O)C2)ccc(O)cc1F C(C(C)CC(=O)N(CC(=O)N(C)Cc1nnnn1C)C)OC C1(CNC(C(C=C)O)=O)CCCCN(C(c2c[nH]c(=NC)o2)=O)CC1 C1(NC(C=CC2(C)COC2)=O)CCOCC1C(N1CC(NC(=O)N(C)C)C1)=O C1(N(CC(=C)C)C)CCCN(C(=O)COC(C)C)C1.c1(C2C(=O)N2)ccccn1 N1(C(COCCCC)=O)CCN(C(=O)C(=Cc2ccco2)C)CC1CCOC N1(C(CC(CC)C2CC2)=O)CCN(C(=O)CCN2CCN(C)CC2)CC1SC C1(C(=O)NCCC(CNC(c2[nH]ccc2C2CC2)=O)O)CC2(CCCC2)CO1 C1(CC=C)(NC(C2CCCN(C)C2)=O)CCCN(C(=O)CC2CCC(C)C2)C1 c1(C(=O)NC2(CO)CN(C(CC(C(C)C)O)=O)C2)cn2c(Br)cccc2n1 C1(C(C(=O)NCC2(C(=O)OC)CC2)C)CCCCN1C(C)=O.C1CC1NC=O Cc1ccc(C(C)CC(=O)N2CCC(CNC(c3nocc3Cl)=O)C2)cc1 N1(C(CSC(C)(C)C)=O)CC2CCCC(CNC(=O)C3Cc4ccccc43)C2C1 C1(C(N)=O)CCN(C(C2CC2CNC(=O)CCCF)=O)C1 c1(NC(n2cc(-c3ccnc(Cl)c3)nn2)=O)c[nH]c2c(CC3(CO)CC3)cccc12 CCS(=O)(=O)C=CC(=O)N1CCCC1C1N(C(c2ccc(C(C)C)c(O)c2)=O)C1 CCCC(C)CS(=O)(=O)N(CC(C1CCCCC1)(C)O)C c1(CN2C(C)(C(=O)Nc3cc(C(F)F)cnc3Br)CCC2)cc(F)c(Cl)cc1O C12(NC(CCCc3c(C)ccs3)=O)CCOC(CNC(c3cnco3)=O)(C1)C2 C=Cn1nncc1S(=O)(=O)Oc1ccc(C(=O)OC(C)CC)cc1 C(=O)(CCC(CC)NC(c1cc(COC)on1)=O)N1CC(C)(OCC)C1 N1(C(C(CC)(C)C#N)=O)C2CCC1CC(CNC(=O)CN1CCCCS1(=O)=O)C2 c1(C(C)C)cccc(CC(=O)NCC2CCN2C(C2(F)CC2(Cl)Cl)=O)c1 C(=O)(CC(F)(F)Br)NC(CC)COC.C(=O)(COCC(F)F)NCCNC C(=O)(C(O)CCN(C)C)N1CCC(CNC(c2cnc(NC)s2)=O)C1 c1(C(=O)NCC(C)CNC(=O)CC2C=CCCC2)nccc(Cl)c1O CC1CN(C(=O)CC2CC(=O)NC2=O)CCN(C(c2c[nH]nc2F)=O)C1 c1(C(C)=O)cc(NCC(C)NC(c2ncoc2C(F)(F)F)=O)ccc1[N+](=O)[O-] C(N=c1cc[nH]c(C#N)n1)C1CCCN(C(C(=O)N(C)C)=O)C1 C(=O)(N1CC(O)CO1)c1c(CNC(C2(CSC)CCC2)=O)cnn1C N1(C(CCCCC)=O)CCC2C1CCCN2C(=O)COC(=O)NS(C)(=O)=O C1(CC)(NC(C2CC(C)C2)=O)CCCN(C(c2oc(Br)nc2C)=O)C1 C(N=c1[nH]c(N2CCOC(C3CC3)C2)nc2c1COC2)C1C(C)(C)NC(=O)O1 c1(CC(C)C(=O)NCC2CCCC2NC(=O)CN2CCCCC2)ccccc1F c1(C(N(CCOCCCN(C(C2(C(=O)NC)CC2)=O)C)C)=O)sccc1Cl N1(C(C(C(C)C)Sc2ccccc2)=O)CCCC(O)(C(N)=O)C1 CCC(CO)(C(=O)NC1C=CCC(C(=O)NCC(F)C2CCC2)C1)OC N1(C(C(c2cn(CC)nc2)(F)F)=O)CCN(C(C2CC23CCC3)=O)C2(CCC2)C1 C1(NC(Cc2c(C)cc(C)s2)=O)CCN(C(C2CCC(C)(C)CO2)=O)C12CCC2 CC(C)CCCCCC(=O)NCC(C(=O)NCC1(O)CC(C)(C)C1)N(C)C CC1(C)CC(CNC(C2CCCO2)=O)N(C(c2cc[nH]c2C2CC2)=O)C1 N1(C(c2cc(=NC)[nH]cc2)=O)CCC(C)(C)CC1C(=O)NCCC[Si](C)(C)C C(CC(O)CC(=O)N(CCCCNC(C1CCSC1)=O)C)SC c1(C(=O)NCCC(C)(C)NC(C2COC(=O)N2)=O)ccc(O)cc1Cl C(=O)(CS(=O)c1cc(Br)ccc1OC(=O)CSC)N(C(=O)CC(C)CF)CC C1(C(N(CC(C(=O)NCc2nnc(C)s2)C)C)=O)CC2COCC2C1 CC(C)(CCCNC(C1CC2CCC2C1)=O)C(=O)N1CC(N2CCCC2)C1 c1(C(c2nnnn2-c2cccc(Cl)c2)CC)ccc(F)cc1Br.C(COCC)(CO)N Cc1cccc(SCC(=O)NC(C)(C)CN(C)C(c2cnn(C3CC3)c2)=O)c1 N1(C(CC(=C)Br)=O)CCC(C(C)C)CC1CNC(c1coc(C)c1)=O c1(C(=O)NC2CC(CNC(c3ccc(C)nc3O)=O)C2)nn2cccnc2c1Cl c1(SC)cc(C(N2CCCC2CN(C(=O)Cc2ccco2)C)=O)c(Cl)cc1Cl N1(C(C(c2ccn(C)c2)C)=O)CCC(F)(C(=O)NOC2CCOC2)C1 c1(SCC)ccccc1C(N1CCOC(CCNC(C2(F)CC2)=O)C1)=O C(=O)(C1=NN2CC(C)CN=C2N1)NCC(C1CC1)NC(C1CCC(CC)CC1)=O c1(CC(c2ccccc2)NC(C2(F)C3CCCC23)=O)ccccc1Cl C1(NC(c2c(OC)ccs2)=O)CC2CC(C1)N(C(c1c(F)cc(O)cc1F)=O)C2 C(C#Cc1ccccc1)N(C1CCOCC1)CC1CCCO1.O=S1(=O)CCN1 N1(C(C=CCC)=O)CCN(C(c2sncc2C)=O)C(C)C1C C(=O)(CCCS(N)(=O)=O)N1CC(NC(C2C(C(C)C)C2)=O)C(c2ccccc2)C1 C(=O)(C(C#N)C(C)(C)C)NC(C(=O)NCC(C)Cn1cccn1)C1(C)CC1 N1(C(CC2(NC(C)=O)CCCC2)=O)CC2(CCN2C(=O)CC(C)n2ccnc2)C1 C1(C(=O)NC2C(C)(C)CN(C(c3cnc[nH]3)=O)CC2)CCc2nccn2CC1 N1(C(CSCCC(C)C)=O)CCC(C2CC2)C1C(N1CCC12CCCCC2)=O C(CC(C(C)C)NC(C1CCCC(NC(=O)C(N)=O)C1)=O)OC c1(-c2cn(C3CCCC(C(F)F)CC3)nn2)ccc2ncccc2c1 C1(CNC(Cn2c(=N)nc[nH]2)=O)CCC2CN(C(c3ccc(N)c(F)c3)=O)CC12 O=C1NCC2CN(Cc3ccc(Cn4cccn4)cc3)CCC2N1 c1(C(N2C(C)CCN(C(C3CS(=O)(=O)C3)=O)CC2)=O)cc(F)cc2cc[nH]c12 CC1(NC(c2ccsc2-c2ccccc2)=O)CCN(C(C23CCC(C2)C3)=O)C1 CCC(C)(C)C(=O)N(CC(C)N(C(=O)CCc1cocn1)C)C N1(C(C(C)(C)OCCCCC)=O)CCCCC2(CCN(C(=O)C=CCOC)C2)C1 c1(NC(C)=O)cnc(N2CCCC2C(N2CCC(C3CCCN3)CC2)=O)c(C)c1 CCCCC(CC)CC(=O)NCC1(NC(c2nn(C)c(N)c2C)=O)CCOC1 Cn1cc(C(=O)O)cc1CNCC1(c2ccc(F)cc2)CCC1 N1(C(c2c(C)c(O)ccc2)=O)CCC2(CC1)CN(C(=O)C(O)C(F)(F)F)C2 c1(C(=O)NC2CCC(C)N(C(=O)CCC3CCCC3)C2)ccc(P(C)(C)=O)s1 C1(NC(COCCC)=O)CCC2(CC1)CCN(C(C1CN3CCC1CC3)=O)CC2 Cc1cnc(C(=O)NC2CCCCC2CNC(c2c(CO)noc2C)=O)c(F)c1 C12(C(N(CC(C)NC(=O)COCC(=O)Nc3cccs3)CC)=O)COCC1C2 C(=O)(C(N)CCC(=O)C(C)Oc1ccccc1C(F)(F)F)OCC CN1N=C(CC(=O)N2CCC3(CCCN3c3nc(C4CC4)ns3)C2)CC1=O c1(OCC(c2cn(CC)nc2)O)cnc2[nH]cc(C)c2c1 C1(CNC(Cc2cn(C)nc2)=O)CCCC(Cn2cc(C3COCC3O)nn2)C1 N1(C(CC(C)C2CCCCC2)=O)CC2(NC(c3cc(Br)c[nH]3)=O)CC1C2 c1(C(N(CC(CNC(C(C)OCCCC)=O)C)C)=O)c(Cl)csc1Cl N1(C(C(C=CC)O)=O)CC2CCCC(C1)N2C(=O)C(C1CC(F)(F)C1)O C1(C(=O)NCC(C2CCCC2)NC(c2ccn3ccsc23)=O)CC2(C1)CC(O)C2 CCC(CC(=O)NCCN(C(c1ccnc(OC)n1)=O)CC1CC1)C1CC1 c1(C(N(CC(C)NC(c2cc(C(N)=O)ccn2)=O)CC)=O)cn2ccccc2n1 c1(C(N2CC(CC(N3C(C(N)=O)C(O)CC3)=O)C2)=O)ccc(Cl)c(C#N)c1 CC1C(NC(c2cnc(-c3ccoc3)s2)=O)CCN1C(C1CC12CCCC2)=O C(=O)(C1=C(CC)OCCC1)N(CCC(=O)NC1CCN(CC)C1)CC#C CCC(C)CC(=O)NCCN(C(=O)C(c1ccccc1OC)(C)C)CCOC C1(CC(=O)NC(c2ncc(C)o2)C)CC(F)CN1C(=O)CSCC(F)F C(C1=CCN(C(C2CCN2CC)=O)CC1)NC(C1CC(CC)C1)=O C12(C(N(CCNC(c3cnc4[nH]cncc3-4)=O)CC)=O)C3C4C1C1C2C3C41C#N C1(CNC(C(C)(C)OCC)=O)CC2CN(C(c3cccnc3O)=O)CC12 c1(C(N2CCC(NC(C3C(=C)C3)=O)C2C)=O)cc(OC)ccc1[N+](=O)[O-] N1(C(C2C3(CN(Cc4c(C)n[nH]c4C)C3)C2)=O)CC(C)N(C)CC1C C1(NC(C(C)OCOC)=O)CC2(C1)CN(C(C1CCCN(C)C1)=O)C2 N1(C(C(C)=C(C)C)=O)CCCC1C1CCCCN1C(c1cnc2ccsc2c1)=O C=CCCCCCCC(=O)N(CCCNC(C1CCCN(C(C)=O)C1)=O)C1CC1 N1(C(C2CCN2C2CCCC2)=O)CC(F)(F)CC1c1nc(-c2cccc(F)c2)no1 CCCC(O)CC(=O)N1CCC(CNC(=O)CN2C(=O)CN(C)C2=O)C1 O=C(CCCCn1cc(C2CCCN(CC3(CC4CC4)CCCO3)C2)nn1)OC N1(C(c2c(CC)n(CC)nc2)=O)CCOC2(CCN(c3ncc(I)cn3)C2)C1 C(C1CCCC1)=C(C)C(N1CCC(CC(=O)NC(C)(C)C(C)O)C1)=O C1(C(=O)NC(CNC(c2c(SC)cc(C)cc2)=O)(C)C)CCCC2CCCN12 N1(CC(N2CCC(C(=O)NCc3nc(C)[nH]n3)C2)=O)CCOCC1=O c1(C(N(C(C(=O)N(C)C(c2ccn(CCF)n2)=O)(C)C2CC2)C)=O)nncn1C c1(SC)nccc(=NC(=O)c2cncc(NC(=O)COC3CCCC3)c2)[nH]1 S(=O)(=O)(c1ccncc1)N1CC(F)CC(C(=O)Nc2cc(C)cc(Br)c2)C1 c1(C(=O)NCC2N(C(c3ccc(C)nn3)=O)CC(F)C2)csc2ccncc12 c1(OC)c(Cl)cc(O)c(Cl)c1C(N1CCN(C(C2CCC(O)C2)=O)C(CO)C1)=O C1(CC#C)CCN(C(C(=O)NCC(=C)C)C2CC2(Br)Br)C1 CCC(C(=O)NCCN(C)C(C1CC1C(=O)OC)=O)SC C1(NC(CCCC)=O)C2CC1N(C(=O)Cc1cc(C(F)(F)F)co1)C2 C1(O)(C(=O)NCc2onc(COC)n2)CCN(C(=O)C(C)(C)C(C)C2CC2)CC1 c1(C(=O)NC2CCC(NC(C=CS(C)=O)=O)C2)ccc2c(c1)CCCC(=O)N2 C1(C(=O)Oc2c(C)nnc(Cl)c2)CCOC2(CCOC2)C1 N1(C(CC(=C=C)C)=O)CC(C(N2CC(OC(F)F)C2)=O)C2(CC2)C1 Cc1cc(C(=O)NCCn2cc(CNC(c3cnsn3)=O)nn2)ccc1O CC1SCCCC1C(=O)NC1COCCC1C(=O)N(CC(C)(C)C#N)C C12(NC(c3c(C)onc3C3CC3)=O)CCOCC1CN(C(=O)C(C)(C)C#N)C2 c1(N2CCN(C(C)CO)CC2)nc2c(c(=NCC3CC=CC3)[nH]1)COC2 Cc1nc2c(o1)CCCC2CC(=O)NC1(CNC(=O)C#CC(C)(C)C)CC1 C1(C(N(CC(CC)C)C)=O)(CNC(C2CC(=O)C2)=O)CC12CCC2 CCCC(O)CC(=O)N1CCCCC1CCN(C)C(c1ncoc1CC)=O O=C(N1CC(O)CCO1)C1CC2CC1CN(C(C1(F)CC=CCC1)=O)C2 C1(NC(=O)CN2CCCNS2(=O)=O)CCCC12CN(C(c1ccnnc1O)=O)C2 N1(C(C2C(CC)C2)=O)CC2CCN(C(c3cnc(OC(C)C)cn3)=O)C2C1 c1(N(CC(=C)C)C)nc2cccnc2c(=NCC(C)C(Cl)(Cl)Cl)[nH]1 CC(CC(=O)NCC1CCCC1NC(=O)C=Cc1cnn(C)c1)C(F)F c1(OC)nn(C)cc1Oc1cc(NC(c2ncccc2F)=O)ncn1 N1(C(c2occ(C)c2)=O)CC(C)(C(=O)NC2CC(=O)N(C)C2)CC1(C)C C(=O)(C#CC1CCCCO1)NC(C)CNC(c1ccc(N)cn1)=O C1(CNC(c2c(SC)cccc2)=O)CC12CCN(C(=O)Cn1nnc(C)n1)CC2 CN1C(=O)NCC12CN(C(=O)C(O)CNC(=O)C=CC1CC1)C2 Cc1ccc(F)c(NC(C2(CNC(c3cnn(CCF)c3)=O)CCCC2)=O)c1 C(=O)(C(CC1CNC1)NC(c1cn(C2CCC2O)nn1)=O)OC N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCC(NC(=O)C=CC(=O)NC3CC3)CC2C1 c1(C(=O)NC2CCCN(C(=O)C=CCO)CC2)cc2ccccc2oc1=O C1(CNC(c2c(CC)ncs2)=O)N(C(=O)CC2CCOC2(C)C)CCCC1(C)C C1(CC(=O)N(C2CCCN(C(c3cc(C(N)=O)cs3)=O)C2)C)CCCN(C)C1 C1(CC=C)(C(=O)N(CCC(=O)NC)C2CC2)CCN(C(=O)C(O)CSC)C1 C1(CNC(c2c(CC)[nH]c(=N)s2)=O)CN(C(c2cocc2C(N)=O)=O)CC12CC2 C(C(C)(C)CC(=O)N1CCC(C)(C)C1CNC(=O)C=CBr)OC Cc1cc(Br)ncc1C(c1nnnn1-c1ccccc1)NCC1CCCC1(C)C [N-]=[N+]=NCCCCCCCS(=O)(=O)NCC1CN(c2nncs2)C1 C(CCNC(C1(F)CCCCC1)=O)(C(=O)NCCC1CCCO1)OC c1(OCC)ccc(C(N2CC3CN(Cc4ccsc4)C3C2)=O)cc1OC C#CCC(O)C(=O)NCC1CN(c2nnnn2C)C1.C12(F)CN(C1)C(=O)C2 c1(OC)cccc(S(=O)(=O)N2CCC(C(C)Nc3ncc(F)cn3)CC2)c1 c1(C(=O)NCCN(C(C2CCCC2O)=O)CC)nc(-c2ccco2)sc1C N1(C(c2c(C)occ2)=O)CCCC1C=CC(=O)NCCF c1(CC(N2C(CN(C(CC(C=C)C)=O)C)CCCC2)=O)c(C)nc(CC)nc1C c1(C(=O)NC(C(C)NC(=O)Cn2ccc(C(F)F)n2)C)c(F)ccc(C#N)c1F C1(C)(C(=O)NCCN(C(C2CC(N3CCCC3)C2)=O)CC)CC=CCC1 N1(C(c2cc(C)c(C)o2)=O)CC2C3CCC(C2C1)N(C(=O)CN1CC1CCCC)C3 C1(COC)(CNC(=O)Cc2ccc(C(N)=O)cc2)CCCN1C(=O)C1=CCCC1 c1(C(N2CC(O)(C3CCCN3C(c3cnn[nH]3)=O)C2)=O)ncsc1Br C1(C(C)NC(c2n(CC)cnn2)=O)CN(C(=O)Cc2ccnc(F)c2)CCO1 c1(C(N(CC(CNC(CCC(=O)NCCC)=O)C)C)=O)ccc(OC)c(F)c1O N1(C(C(C)(C)C2CCC2)=O)CCN(C(C2CCCC2O)=O)C(c2cn[nH]c2)C1 c1(C(=O)NCC2(C(C)NC(=O)CCc3cncnc3)CC2)nc(C)n2ccccc12 C(CNC(c1csc(Br)n1)c1nnnn1CCCF)(C(F)(F)F)OC C12(C(N(CCCO)CCC)=O)CC(CCO1)N(C(=O)CCNC(C)=O)C2 C(=O)(CC(O)C(C)CC)NCC(CC(=O)N(CC)Cc1ccoc1)O C1(C#N)(CC(N2CC3C(C(=O)NCC4C(C)C4)(C3)C2)=O)C2CC3CC(C2)CC1C3 C1(NC(C(C)N(C)C)=O)(CNC(C2CCC3CC23)=O)CCC(C)(C)CC1 C=C1C(NC(c2nn(C)c(Cl)c2CN2CCNC(=O)C2)=O)CC2CC1C2(C)C C1(CNC(CNC(CN(C)C)=O)=O)CCCCN1C(c1csnc1Cl)=O N1(C(CCc2n(C)cnn2)=O)CCC2CN(C(c3ccsc3Br)=O)C2C1 N1(C(C(C2CC2)OCC)=O)C2CCC1C(NC(c1ccc(=O)n(CCO)c1)=O)C2 C1(N(C)C)CCCC(C(=O)NCC2CCCN2C(c2ccc(CCF)cc2)=O)C1 C(=O)(C(C)C(C)(F)F)NCC1(C(C)(C)C)CCN(C(C(N2CCOCC2)C)=O)C1 CC1=C(C)CC(C(=O)NC2(CNC(C3CCN3C)=O)CCCCC2)CC1 c1(N(CCCC(=O)NC2CCC2)C)ccc(F)cc1Cl N1(C(C(C)n2ccnc2)=O)CCC2(CCOC2)C(CNC(C2C3COCC23)=O)C1 C(=O)(C1=CCCN(C(=O)C(C)OCCC(C)C)C1)NC(CC(=O)NC)C1CC1 C1(C(=O)NC2C(CC=C)CCC2)CN(C(C2CCCNC2=O)=O)CCC1(C)C c1(C(N(C(C)CNC(C2CC(O)C2)=O)C)=O)csc2ccc(F)cc12 C1(NC(C2CCC(=O)NC2)=O)(CNC(C2C3CC4C(C3)C24)=O)CC2CCC1CC2 CC1CCC(F)(F)CN1C(=O)C(CC1CCCC1)NC(=O)CCP(C)(C)=O C(=O)(CC(C)(C)CC(F)(F)F)NC(C(C)(C)NC(CCCC#C)=O)C C1(C(N2CCC(O)(C(C)C)C2)=O)COC2(C1)CN(C(=O)C1=CCOCC1)C2 C1(NCC(N2CC(NC(C3C(=C)C3)=O)(CO)C2)=O)CCN(C2CC2)CC1 C1(SC)CCN(C(=O)C=C2CCN(Cc3cc(-c4ccccc4)n[nH]3)C2)C1 C1(CCNC(C=CC=CC)=O)(C(=O)NC(c2ccco2)COC)CCC1 S(=O)(=O)(c1c[nH]ccc1=NCCn1ccnn1)NCCC(C)O C(CCCCCNC(=O)C(c1nc(C)cs1)C)NC(c1cnc(OCC)s1)=O c1(C(=O)NC2C(SC)CN(C(=O)CCc3cc(C)nn3C)C2)cc(O)nc(O)n1 c1(CC(=O)NC2(CN(C(CC=C)=O)C)CC2)ccc(Br)cc1OC c1(N2CCN(C(=O)NC)CC2)ncnc2c(Br)csc12 c1(C(N2C3C(C(C)=O)C(C3)C2)=O)nn(C)c(NCc2cc(Cl)ccc2OC)c1Cl N1(C(c2c(OC)nc(C)cc2)=O)CC2CCC1CC2NC(c1coc(C)c1)=O CC1CC(NC(=O)CSCC(c2ccccc2)=O)CN1C(C1CC2(CC2)C1)=O c1(CC)oc(C(=O)NCC2CC(C(=O)NC(CC3CC3)COC)C2)cc1C c1(C(N(C(CNC(c2c(C)cc(C)cc2C)=O)C)C)=O)cc2nc[nH]c2cc1N S(=O)(=O)(c1ccc(N2CCC(c3ccc(C)cc3)C2)c(Cl)c1)N(CC=C)C C1(OC)(NC(=O)N(C)Cc2ccc(Oc3cccc(Cl)c3)cc2)CCCC(C)C1 C1(NC(c2ccc(C)c(C)n2)=O)CCC2CN(c3cc4nncn4cn3)CC2C1 n1(CC)cnc2nc(=NCCSC3CCCCC3)[nH]c(NCCCS(C)=O)c12 CCCCC(=O)NC(C)(C)CN(C(=O)Cc1cnn(C(C)C)c1)C N1(Cc2ncc(C)o2)CCC(O)C(N(C(=O)CCCNc2ccccc2)C)C1 Cc1ccc2[nH]c(C)c(CNC(=O)NCCC(F)(F)C(F)F)c2c1 c1(CCC(NNC(=O)N2C(CC(=O)NC)CCCC2)=O)ccnc2ccccc12 N1(C(CCc2n(C)ncc2)=O)CC2(C)CN(C(=O)CC3(O)CCC3)CC2(C)C1 C1(CNC(c2c(CC)onc2)=O)CN(C(=O)CC2CCS(=O)(=O)C2)CCC1(F)F C(=O)(CCC(F)(F)C(F)F)N1CC(CNC(c2ccc(C)c(C)c2O)=O)C(C)C1 c1(NC(CCC2CC(NC(C3CCN(C)C3=O)=O)C2)=O)cccc(C#N)c1 CCC(CC)C(C)C(=O)N(CCCN(C)C)CCNC(=O)CC1CCS(=O)(=O)C1 N1(C(C(C)CNC(=O)CN2CCC(C)C2)=O)CCCC12CCOC2=O C#Cc1cccc(CNC(=O)COCCNC(C2CC3CCCC3C2)=O)c1 N1(C(=O)CCc2cc(F)ccc2Br)CCC(N2CCC(CO)C2)C2(CC2)C1 c1(OCCC)ccc(CC(=O)OC2CCN(C)C(C)C2)cc1C c1(C(=O)NC2C(CC)CCC2)n[nH]c2c1CN(C(C(=O)NC)c1ccsn1)CC2 N1(C(c2c[nH]c(=N)s2)=O)CC2OCC(NC(c3ccc(O)nc3)=O)C2C1 C1(C(=O)NCC(CNC(C2N(C(CCC)=O)CCC2)=O)O)(CC)CCCCC1 C1(CC(=O)NC(C)CC2CN(C(C3(OC)CC3)=O)C2)(OC)CCC1 O=C1COCC2(C(N3CCC4(CCCC4CC(=O)O)CC3)=O)CCCCN12 Cc1cncc([N+](=O)[O-])c1N1CCC(C(C)NC(c2nc(C)c(C)nc2O)=O)C1 C1(OC)CN(C(=O)CN2CCCCCC2)CC1NC(C1ON=C(C)C1C)=O c1(C(=O)NC2CC(N(C(C(C(C)C)NC(C)=O)=O)C)C2)cc(C(F)F)cc(Cl)c1 Cc1c[nH]c(C(=O)NCCNC(=O)C(C(C)C)NC(C2CCCCC2)=O)cc1=O N1(C(c2ccc(C#C)cc2F)=O)CC2CCCC(NC(=O)CC3(OC)CC3)(C2)C1 CC1CN(C(C2(NC(=O)C(N)=O)CCC2)=O)CC(CNC(N)=O)O1 c1(C(N2CCC(N(C(C(C)OCC#C)=O)CCO)C2)=O)c(F)ccc(Cl)c1F C(N=c1[nH]cnc2c1COC2)C1N(C(C2C(C)CC(=O)N2)=O)CCC1 C=CC(C)(C)CC(=O)NC1(C)CCN(C(C2(CC=C)COC2)=O)C1 C(=O)(CC(c1ccccc1)NC(N)=O)NCC(CC)NC(c1ccc(CO)o1)=O c1(OC)cc(C)[nH]c(=NCC(C2CC2)N(C)C(C2COc3ccccc3O2)=O)n1 c1(-c2cnc(NC3C=CCN(C(COC(C)(C)C)=O)C3)s2)c(F)cc(F)cc1F C#CCC(CC(=O)NCC(C1CCCCC1)OC)NC(c1cc(F)cnc1O)=O C1(C(=O)NC)CC(C)CN(C(C2CCCCC2NC(c2[nH]cc(C)c2C)=O)=O)C1 c1(C(=O)NCCc2ccc(OCCC=C)cc2)cnn2cccnc12 c1(CCN(C)CC2(N)CC2C(F)(F)F)ccc(F)cc1F C1(OC)CN(C(=O)Cc2nncn2C)CC1NC(C1(NC2CC2)CCC1)=O Cc1nnc(O)c(C(=O)NCC2CCCN2C(C2CCCC3C2C3(F)F)=O)c1C c1(C(=O)NCCC2CCCN(C(c3coc(Br)c3)=O)C2)cc2cnccc2[nH]1 O=C(N=c1ccc(C2CC2)n[nH]1)c1csc(N2CCNCC2)n1 C=CC(C)(O)CC(=O)NCC(CC(=O)Nc1cnn(C)c1)C1CCC1 N1(C(C(C)C(C)(F)F)=O)CC(C)(C)CCC1CNC(c1ccc(C(F)(F)F)[nH]1)=O c1(OC)ccccc1C(=O)NCC(C)(O)CNC(c1ccnn1C1CC1(F)F)=O N1(C(c2c(N)nc(Cl)cc2)=O)CCC(C2CCCN(C(c3csc(S)n3)=O)C2)C1 C1(NC(C2CC(SC)C2)=O)CCC(F)(CNC(C2(C(F)F)CCCC2)=O)C1 C(C(=O)N(CC(F)(F)Cl)C)(C(C)(C)C)NC(C(C)CO)=O Cc1nn(CC(N2CC(CNC(=O)Cc3cnc(C4CC4)[nH]3)C2)=O)cc1Br N1(C(C2C(C)(C)CCC2)C=O)CC(O)C(C)(C)C1.N1(CC(F)F)CCCC1 Cc1cccnc1CCC(N1CCOC(CN(C(=O)C=Cc2cc[nH]n2)C)C1)=O c1(OC)ccc(CC(N2CCC(OCCNC(C3(C)CS(=O)(=O)C3)=O)C2)=O)cc1 C1(CN(C(C(C=C)O)=O)C)CCN(C(C2(OC)CCC2)=O)CC1 CCC(C)C(c1ccccc1)NC(=O)CC1CN(Cc2ccc(Cl)o2)C1 C1(C(=O)NCCC2(O)CCC2)CCC2CCC1N2C(c1cc2ccccc2o1)=O N1(C(C(CC)n2ccnc2)=O)CCC(CO)(CNC(=O)C(CC)N(C)C)C1 N1(C(C2C(C)(C)OC(=O)C2)=O)CCN(C(C2CC(OC3CC3)C2)=O)CC(C)(F)C1 Cc1cc(C(N2CC3CC3(CNC(=O)Cc3nncn3C)C2)=O)nc(C)n1 Cc1nc(Br)oc1C(=O)NCC1CN(C(=O)C(c2ccccc2)C)CC1C N1(C(C2CC(C)(NC(C3CC4CCC4C3)=O)C2)=O)CC(C)(C)C2CCCC12 O=C(C1=Cc2ccccc2C1O)N1CC(NC(C23CC(C2)S(=O)(=O)C3)=O)C1 N1(C(C=Cc2c(C)coc2C)=O)CC(C2CCCCN(C(C3CCCS3)=O)C2)C1 Cc1nc(CNC(C)(CCCO)c2nnnn2CC2CC2)sc1CC1CCOC1 Cc1c[nH]c2ncc(C(N3CC(NC(C4CC4CCN(C)C)=O)C3)=O)cc12 N1(C(COCC(C)C)=O)CCC(NC(c2ccn3ncccc23)=O)C(F)(F)CC1 N1(C(C2(COC)CC2)=O)CCC2CCN(C(=O)C(C(C)(C)C)c3cc[nH]n3)CC12 N1(C(c2c(C)cncc2C)=O)C2CCC1CN(C(=O)Cc1ccc(F)cn1)C2 C(=O)(N=c1ccn(C2CC2)[nH]1)NC1(CN(CC(CC)OC)C)CCCC1 C(=O)(C(CNC(=O)C=CC1CC1)CC1CC1)N(CCCO)CC#C c1(C(N2CC(c3nn[nH]n3)(C(=O)NCC)C2)=O)cc(C2CC2)cc(F)c1 N1(C(CC=C)=O)CC2CN(C(=O)NCc3cc(SC(C)(C)C)nn3C)C2C1 c1(C(=O)NCCc2ncc(C)s2)cnc(S)n1-c1ccccc1 C1(C(C)(C)C)(CNC(=O)CC(O)C2CCCC2)CCN(C(=O)C2=CCCO2)C1 Cc1cc(Br)cc(C(N2CC(CNC(=O)C(C)(C)CO)C3CC23)=O)c1N C(=O)(CCC(C)(C)C#N)NC1(CNC(C=Cc2c(C)cccc2)=O)CCCCC1C C1(OC)CN(C(C2CC(=O)CC(=O)C2)=O)CCC1NC(=O)COC1CC1 CCC(C)C(C(=O)N1CCOC(C(C)C)CC1)N(C)C.N12CCC(OC)C1C2 C1(CS(CC)(=O)=O)CCC2(CC1)CC(O)C2.C(C)(CC(C)C=O)NCC(=O)NC N1(C(c2cn(C)c(=O)cc2)=O)CCC(C2(NC(=O)Cc3cncnc3)CC2)C1 C1(C)(COC)CN(N2C(CC=O)CC(O)C2)CCO1.C1(CC=O)CCCCC1 c1(CNC(c2c(COC)noc2)c2nnnn2C2CCCCC2)ccc(Cl)cc1 c1(SC)ccc(C)c(OC(=O)CC#N)c1.C1(C)(C)C(=O)O1.C1CCN1CCO c1(N2CCN(C(C=CC=CC)=O)CC2)ccc([N+](=O)[O-])c(OCC)c1 c1(SC)cc(C)c(C(N2CCC(NC(=O)C(C)(CO)NC(C)=O)C2C)=O)s1 c1(C(N2CC(n3cc(C4(C(=O)OCC)CCCO4)nn3)C2)=O)cccc(C#N)c1 C(CCCS(=O)(=O)CCO)NC1C(OC)CCCC1 c1(OC)c(F)cc(C(N2CC(O)CC2C(=O)Nc2nnc(C(C)C)o2)=O)cc1F C(CC(C(C)(C)C)CC1(C=O)CC1)N(C)C1CC1.C1(COCC(=O)N)CCCO1 CN1CCOCC1CC(=O)NC1(CNC(=O)CCCC#N)CC1 C1(NC(c2cc(C)n(C(C)C)c2)=O)COC2(C1)CN(C(C1C3CN(C)CC13)=O)C2 c1(CC)cc(OC)ccc1C(=O)NCCCN(C)C(c1csc(C(N)=O)n1)=O N1(C(CC)=O)CCC(CNC(C2(C)CCN(C)CC2)=O)C12CC2 Cc1nc(C(=O)NCCNC2CN(C(=O)CN3CCCC3C)C2)c(Cl)cc1C#N CCCC(O)C(=O)N(C1CN(C(c2ccc(S)cc2)=O)CC1O)C CC1CC(CNC(c2ccc(-n3ccnc3)nc2)=O)CN(C(C2(CO)CC2)=O)C1 c1(C2(NCC)CC2)cccc(F)c1F.C1(N(C(C(=O)NCC)=O)C)CC(C=O)C1 C1(C(=O)NCC(C)N(C(c2c(CC)noc2)=O)C)CCCC(=O)C1 N1(C(CNC(C2C(CC#C)CCC2)=O)=O)CCCN(CCO)CC1 c1(OC)c(C(=O)NC2C3CC2N(C(C2CNC(=O)N2)=O)C3C)ccnc1F C1(C)(CNC(c2n(CC)nc(C(C)C)c2)=O)CN(C(=O)CSCCF)CCO1 N1(C(c2ccc(C(N)=O)nc2)=O)CCC2CCCC12CNC(=O)CCCF N1(C(C(n2c(C)ncc2)C)=O)CC(C(N2CCC3(CC2)CC3)=O)CC(C)C1 c1(N(C(CNC(C(C)CO)=O)C)C)ccn2ccnc2n1 C1(NC(=O)C2=CCSC2)CC(F)(F)CC1NC(c1csc(Br)n1)=O N1(C(c2c(C)ncnc2C)=O)CCCC2CN(C(C3(F)CCOC3)=O)CC12 c1(C(=O)OC)cnc(C2CC2)nc1.C1(C2C(=O)O2)CCCCO1 N1(C(c2nc(OCC)sn2)=O)CC(NC(=O)C(CCSC)OCSC)CC2(CC2)C1 N1(C(C23CC(CSC)(OC2)C3)=O)CCCC(N(C(=O)Cc2csc(C)c2)C)CC1 Cc1cnn(C)c1NC(=O)CN1CCN(CCN)CC1 C(=O)(C(C)(CO)NC(=O)C(C)O)NCc1cc(C(=O)OC)n[nH]1 C(CC(=O)N1CCNC(=O)C1)(C(F)F)NC(C(CC)COC)=O c1(N(C)Cc2cc(NC(C)=O)ncc2)nc2cc[nH]c2c(=NCCC(F)F)[nH]1 C#CC1(NC(C2CC(NC(=O)C3=CCCC3)CCO2)=O)CC2CCCC12 N1(C(C(C(C)C)F)=O)CCC2CC1CN(C(=O)Cc1cccc3ncccc13)C2 C1(NC(C2(C(C)C)CCN(C(C(C(C)C)OCC)=O)C2)=O)CCCCC1C#N C1(OCC)CN(C(C2CCN(c3nc(=N)[nH][nH]3)C2)=O)CC1NC(c1cnns1)=O CCC(C)C(O)C(C)C(=O)NCC1(C(N2CC3CC2CN3C(C)C)=O)CCCC1 N=c1nc(C(N2CC(=O)NC(c3ccccc3)C2)=O)cc(N)[nH]1 c1(C(=O)NC(C(C)C)C(C)NC(C2(C)C(C)(C)C2(C)C)=O)cccc2occc12 C1(C)(NC)CC1(F)F.CCC1CNC(=O)N1C c1(OCC(C)C)ccc(C(=O)NC(CNC(C2CCOC(C)C2)=O)C(C)C)cc1 c1(C(N2CC(C)C(NC(=O)CCNC(C3CCC3)=O)C2)=O)ccc([N+](=O)[O-])cc1 N1(C(c2nc(C)sc2C)=O)CCC2CN(C(=O)CCC3CCCOC3)CCC12 CC(C)C(C(=O)N1CCOC(CCNC(C2C=CCC2)=O)C1)C(C)C c1(C(N2CCC(NC(C(C)C3CN(C(C4CC4)=O)C3)=O)C2)=O)ccccc1C#N C12(CNC(C3C(=O)NCC3)=O)CCCC1CN(C(=O)Cc1c(F)cccc1F)C2 CN1CC2CCC1C(NC(C1(NC(C3CC(C)(O)C3)=O)CC1(C)C)=O)C2 N1(C(C2CCC(=O)NC2)=O)CCC2(CCC2CNC(c2csc(Cl)n2)=O)CC1 Cc1nc(C(N2CCCC2C2(C(=O)NC3CCCSCC3)CC2)=O)c(C)o1 c1(N2CC(C(=O)OC)C2)ccc2c(n1)CN(C(C1CCNC1)=O)CC2 c1(OC)ccc(C(N2CC(C3CNCCN3)C2)=O)c(C)c1C C(C(N=[N+]=[N-])C(=O)N1CC2CC1(C(=O)NCc1nccs1)C2)OCC c1(C(N(CC(C)C)C(=O)NC(C2CCOC2)C)C)cccc(Cl)c1 N1(C(C(C(=O)OCC)(C)C)=O)CC2(NC(C3CCCS(=O)(=O)C3)=O)CCC1CC2 c1(NC(N2CCN(CC(=O)Nc3c(C)cc(C)s3)CC2)=O)cccc(C#N)n1 n1(CCNC(=O)C(F)=CC2CC2)ccc(C(=O)NC(c2cccnc2)CO)c1 c1(C(N2CCC(N)CC2)=O)n[nH]c2cc(CN3CCC(N(C)C)C3)ccc12 c1(C(N2CCC(F)(CNC(c3c(C)ocn3)=O)C2)=O)ncnc(O)c1Br c1(C(N2CC(NC(=O)CC3CNC(=O)C3)C(C(F)F)C2)=O)ncc2ccccn12 c1(C(N2CCC(N(C(=O)CCc3nccs3)CCC)C2)=O)cc2cn[nH]c2cn1 Cc1ncc(Br)cc1C(=O)NC1CN(C(=O)C(C)(C)N(C)C)CC1F c1(C(N2CCC(NC(c3c(C)onc3CO)=O)C2)=O)c[nH]cc(Br)c1=N C1(C(=O)NCC2CC(CNC(CCC(C)OCC)=O)C2)CC2CC(=O)C1O2 C1(CC)CCCCCCN1C(C1CCC(CNC(c2coc(C)c2)=O)CC1)=O c1(C(N(C)CC2C(NC(CC(CN(C)C)O)=O)CCC2)=O)cc(F)cc(Cl)c1N N1(CC#N)CCOCC(C(=O)NC2CC3OCCCC23)C1 Cc1cc(C(=O)NCC2(CNC(=O)CN3CCC(C)(C)C3)CCC2)c(N)c(C)c1 c1(C(=O)OCC2(C#N)CCOCC2)cccc2c1COC2 c1(C(=O)NCC(C)(C2CC2)NC(C(CN(C)C)N(C)C)=O)cccc(CC#N)c1 C1(NC(Cc2c(C)occ2)=O)CCN(C(=O)CCC2CCCCN2C)CC1O CCCC(C)C(C)NC(=O)C(C)(C)CN(C)C(c1ccsc1Cl)=O c1(C(=O)OC)cncc(NC(c2ccccc2Oc2cnccc2C)=O)n1 n1(CC(=O)OCC)[nH]cnc1=NC(=O)C1CC1C1CC1c1ccccc1 C1(CN(C(C2C(C)CCC2)=O)C)CC(F)CN1C(=O)CSC1CCS(=O)(=O)C1 C#Cc1ccc(C(=O)NC2(C(=O)N(CCO)CCOC)CC3CCC2C3)nc1 C1(C(C)CC2(NC(=O)CC=CC(C)(C)C)CC2)CCN(C(C2(OC)CCOC2)=O)CC1 N1(C(C(Cc2ccc(N)cc2)N(C)C)=O)CCC2(C)C(C1)C2(Cl)Cl N1(C(c2c(C)cc(Br)o2)=O)CCC2(C1)CN(C(=O)C(C)(C)CF)C2 c1(OC)cnc(C(N2CCN(C(=O)C=C(C)Cl)C(C)C2)=O)c(F)c1 c1(C(N(CCC(C)NC(C2CCC(C)CC2)=O)C)=O)ccc2cc[nH]c2c1F C1(CNC(C(CCC)N(C)C)=O)CN(C(=O)C(O)CCn2cncn2)CCCO1 N1(C(CN2C(C)CC3(CC3)C2)=O)C2CCC1CC(C(N1CCC(O)C(F)CC1)=O)C2 c1(C(N2CC(CCNC(C=CS(C)=O)=O)OCC2)=O)nccc2cc[nH]c12 C(C(=O)N(C)CCOCCCN(C)C(c1ccsc1)=O)(C(C)(C)C)NC(C)=O C1(C#N)(C(=O)NCC2OCCN(C(c3c(CCC)nsc3N)=O)C2)CCCOC1 c1(C(=O)OC)cc(C2CCCN(C(=O)CCc3csc(=N)[nH]3)C2)cc(F)c1 C(=O)(C(=O)N=c1ccn(C2CCCC2)[nH]1)NCCC(Cl)=C(C)C C=CC1CCN1C(=O)CC(C)N(C(=O)CSCC(N)=O)C CC1C(=O)N1C=O.COCON(CCC(=O)O)C Cc1cccc(C(=O)NC2CC(NCc3ccc(OC(F)F)nc3)C2)n1 c1(N2CC(C(N(C)NC(Cc3cccc(CC)c3)=O)=O)C2)nc(OC)c2ccccc2n1 C1(CCNC(=O)CCNC(C2CCC2)=O)CCCN(C(=O)Cc2cc[nH]n2)C1 N1(C(C(C)OCC#C)=O)CCC12CCN(C(c1ccn(C)c1CC)=O)CC2 CCC(C(=O)NC(C)(C)CCNC(=O)Cc1ccsc1Br)N(C)C N1(C(Cc2ccc(C)c(C)c2)=O)CC(NC(C2(C)CC2(F)F)=O)CC12CCC2 C=CCC(C(=O)NCC1(C(=O)NCCC2(C)CC2)CCCO1)NC(C)=O N(C(=NCCC(C)=O)NCC1(C(F)(F)F)CC1)CC1(OCC)CCOC1 C12(NC(C(C=C)C)=O)CCCC1(F)CN(C(=O)CC1CCCCC1)C2 Cc1cc(C(=O)NC(C)CCNC(c2cnns2)=O)c2c(c1)CCO2 c1(C(=O)N(C2CC2)Cc2cccnc2)cccc(Br)c1O.C12(CCC1)C(=O)N2 N1(C(c2cc(OC)nn2C)=O)CCCCC(CNC(c2cncc(CO)c2)=O)C1 CC1OC2(C(=O)NC3CCC(CNC(c4cccc(=O)n4C)=O)CC3)CCC1C2 C(=O)(C1CCCc2nccc(N)c21)NC(C)CNC(C1CC(O)C1)=O n1(CC)cccc(COC(C2CC2C(=O)OC)=O)c1=O C1(N(C(c2cnn(CC)c2C)=O)C)CN(C(=O)CCC2CCC(=O)N2)CC12CC2 Cc1csc(C=CC(=O)NC2CC(NC(c3ccc(Br)cc3)=O)C2)n1 c1(CC(=O)NCC(N(C(C(C)SC)=O)C)C2CC2)ccc(-n2cccc2)cc1 c1(C(N2CCN(C(CCCOC)=O)CC2C)=O)cc2occc2n1C c1(CC(=O)NCC#CC(=O)NC2(C(=O)NCC)CC2)cccnc1C N1(C(CN)=O)CC(C2CCN(C(=O)CC(Cl)Cl)CC2)C1 N1(C(c2ccc(-n3cc(Cl)cn3)c(Cl)c2)=O)CCN2CCc3ccccc3C2C1 C1(NC(C2N(C(c3c(CC=C)cccc3)=O)C(C)C2)=O)CCCN2CCCC12 C(=O)(C(C(C)(C)C)SCCCN)OCc1nc(-c2ccc(OC)cc2)on1 C(=O)(C1=CC2(CCOC2)C1)N1CC(C(C(=O)NCc2ccccc2C#N)OC)C1 C(=O)(CC(CNC(=O)Cc1cn(C)cn1)OC)N(CC(CC)C)C c1(C(C(=O)NCC2CC2)N(C(C(CC)C)C)C2CC2)ccccc1C c1(C(C)=O)nc(C(N2CC(O)(CCNC(=O)C(F)n3ccnc3)C2)=O)cs1 C=C=CCCC(=O)NCCCOCCOCCNC(c1ccnn1CC(F)F)=O C1(NC(c2c(CC)nco2)=O)CC(OC)CN(C(=O)C(F)OC)C1 c1(C(c2n(CCCF)nnn2)NCc2conc2C2CC2)cc(Cl)ccc1F c1(OC)cc(C(=O)NC2COCC2NC(=O)CC(C)n2ccnc2)cc(C)c1 c1(C(N2C(CC)CN(C(C3(O)CC3)=O)CC2)=O)cc2ccccc2nc1C C1(NC(C=CCOC)=O)CCCC(NC(c2cc(O)ccc2OC(F)F)=O)CC1 c1(C(C(=O)NC(CN(C(=O)CC(C)C2CC2)CC)C)(C)C)ccccc1C C1(C2(O)CN(C(C)=O)C2)(CNC(C)(C)C)CC1.N12CCN(CC1)NC(=O)C2CC N1(C(C2C(c3n(C)ccn3)C2)=O)CCCCC(NC(C2C=CCCC2)=O)C1 c1(C(CC(=O)OC2CCN(CC(F)F)C2)(F)F)nnc2n1CCC2 S(=O)(=O)(CCC(=O)N1CC(F)(F)CC1CNC(=O)CCC1CCC(C)O1)NC C(CCCCC(=O)N1CCC(n2ccnc2)C1)NC(C1N(CC)CC1)=O c1(C(=O)NCC2CCC(NC(C3(F)C(C)OCC3)=O)C2)ccc2nn[nH]c2c1 Cc1ccn(C)c1C(=O)N(CC(C)N(C(=O)C(C)Cc1ccccc1)C)C N1(CCCNC(CC2C(C(C)NC(c3cnn[nH]3)=O)C2)=O)CCCCC1C c1(N2CC(C)C(NC(=O)Cc3cncnc3)CC2)ncc(Br)cc1[N+](=O)[O-] C#CCCCCCCC(=O)NC1CC(O)CN(C(c2cc(C#N)c[nH]2)=O)C1 N(C1CCCc2cn(C3CCCC3)nc21)C(C(C)Cc1cnc[nH]1)=O N1(C(C(C)N2CCC2)=O)CC(NC(=O)CCc2ccsc2)CC12CCC2 CC1(C)CN(C(C2CNC(=O)O2)=O)CC(CNC(c2ccc(F)c(Cl)c2)=O)O1 c1(C(=O)NCCC(C)NC(C(C)(C)OC)=O)ccc2c(c1)C(C)(C)CO2 c1(C(N2CC(O)(CNC(C=C(C)c3ccccc3)=O)C2)=O)cc2cccnn2c1 C=CC(C)(O)CC(=O)NCC1CCC(NC(C)=O)C1 C12(CNC(C3(CN(C)C)CCCO3)=O)CC1CNC2=O.N12CC(C1)C(C)C2=O c1(CC(=O)NC(CNC(C(C)OC)=O)CCOC)cccc2cn[nH]c12 c1(CNC(C(=O)OC)Cc2ccccc2OC(F)F)nc2ccc(O)cc2s1 c1(N2C(C)CC(NC(C(C3CCC3)OC)=O)C2)cc2nnc(C)n2cn1 c1(C(=O)NC2CN(C(C(COCC)C)=O)C2)cc2cncn2c(O)n1 C1(C(N2CCC(COC)(NC(c3nccnc3N)=O)C2)=O)CC(S(C)(=O)=O)C1 c1(CCC)sc(C(N2CC(CNC(C3(C)CC3F)=O)C2)=O)cc1CC C1(CCN(C(C(=O)NCCCOC)CC2CCC2)C)CCCC(C)C1 CCC(CCC(=O)NC(Cc1ccc(Cl)cc1Cl)CC(C)C)OC C1(O)(CC)CCCN(C(C2C=CCCN2C(c2sccc2C#N)=O)=O)C1 O=C(CCCC(F)(F)CO)NC(CNC(c1cccnc1O)=O)CO N1(C(C2CCC(CN(C)C)O2)=O)CC2CCC2(CNC(c2ccc(F)cn2)=O)C1 CC(C)(Cl)C(=O)NCC12CC(NC(=O)Cc3cn(C4CC4)cn3)(C1)C2 C1(NC(C2C(NC(C(CO)N(C)C)=O)C=CCC2)=O)CN2CCCC1C2 C1(CNC(C2N(C)C(=O)NC2)=O)(NC(c2cccc(Cl)c2)=O)CC2CCC1CC2 C1(NC(C2(CC)CC(F)(F)C2)=O)CCC(F)(F)CC1.C12CC(O)(C1)CNC2=O N1(C(C=C)=O)CC2(CCC2)CC1CNC(c1csc2nnsc12)=O c1(NC(=O)NC(C2CCCCO2)C2CC2)ccc2cccnc2c1 N1(C(C(C)CC2CC2)=O)CC(C)CCC1C(=O)N(c1cccn(C)c1=O)C C1(C(=O)NC(C(C)NC(=O)CCNC(=O)CO)CO)CCN(C2CC2)C1=O C1(C(=O)NCCC(C)NC(=O)C(C2(O)CCOCC2)(F)F)CC2(CC2)CN1C CS(=O)(=O)C1CCN(C(=O)NCC2C3CCC4C(C3)C24CO)CC1 CC1CN(C(c2nnc(S)n2C)=O)CCC1NC(c1coc2c1COC2)=O C1(C(C(=O)NC(CC)C)N(C2CCCC2)C)CCN(C(CC)C(=O)O)C1 c1(C(N2CC(O)CC(NC(=O)CCc3cnccn3)C2)=O)cncc2c1CCC2 C1(CNC(=O)C=CC2CCCC2)CC2(CCC2)CN1C(=O)Cc1cccc(F)c1 C1(NCC(CN(C(C)C)C(C)C)O)CCCC(C(F)F)CC1 O=CN1CCCC1C(=O)NCC1COCC1NC(=O)CCc1ccccn1 N1(c2nc(C)c(C(=O)O)s2)CCN(CC(=O)Nc2cccc(Br)n2)C(=O)C1 c1(NC(c2ccc(Br)cc2Cl)COC)nc(Cl)cc2ccc(F)cc12 N1(C(CCC=C)=O)CCCCC1c1n[nH]cc1C(=O)Nc1ccsc1C N1(C(c2cc(C)n(C)n2)=O)CCC(C(=O)NCC(O)C(C)O)C12CC2 C1(CC)(NC(C2CCCC2C2CC2)=O)CCCN(C(=O)C2=COCCC2)C1 CC(O)C(C)(C)CN=c1cccc(S(=O)(=O)NCC(C)(N(C)C)C2CC2)[nH]1 c1(-n2cc(C(=O)NC(C(C)NC(=O)C(N)=O)CO)nn2)cccc(C(F)(F)F)c1 c1(C(=O)NC2CC(CNC(COCC#C)=O)C2)cc(S(=O)(=O)NCC)ccc1Cl c1(C(N2CC(C(=O)Nc3cccc(C(=O)NC)n3)C2)=O)cc(OC)c(O)c(I)c1 N12CCC(S1(=O)=O)C(=O)OC1CC2C1.c1(C(=O)OCC)cc(OC)ccn1 c1(-c2cn(CC)nn2)cc(C)nn1C.CCC(=O)C1(C(C)NC=O)CC1 CC(CCOc1ccccc1)C(=O)Oc1ccccc1CN1CCC(O)C1 CC(CC1CC1)C(=O)NC1CCC1CNC(c1cnc(O)o1)=O N1(C(C(CC)NC(N)=O)=O)CCCCC(NC(=O)COC)C1 c1(C(=O)NC2(C(=O)NC(C(=O)NC)CC(C)C)CCCC2)c[nH]c2cnccc12 C1(NC(Cc2c(CC)con2)=O)CN(C(=O)C(CCSC)OC)CC1C n1(CC(=O)NCCN(C(C(C2CC2)OC)=O)C2CC2)nc(C)cc1C(F)F Cc1ccc(C(=O)NC(CC2CC2)C(=O)NC2CC(=O)NC2=O)n1C Cn1cc(S(C)(=O)=O)c(C2CCCC2)n1.C1(C)(c2ncno2)Cc2ccccc2C1 N1(C(c2c(C)ccs2)=O)CCOCCC1C(=O)NCC1(O)CCC(C)C1 c1(C2C(C(=O)NCC(CC)NC(c3ncoc3C)=O)C2(C)C)cccc(Br)c1 C1(=O)C(C)C(C)NC(=O)C2CN1C2.C1(n2cccn2)(N)CCC1.C(=O)(NC)N Cc1ccc(C(=O)N(CC(O)CNC(C2CC(C3CC3)=NO2)=O)C)c2c1CCC2 c1(OCC)cc(OC)c(C(=O)Nc2[nH]ccc2C(=O)NCCOC(C)(C)C)cn1 C=C(C)CCCC(=O)NC1CCC(N(C(=O)Cc2cccc(OC)c2F)C)C1 C=Cc1ccc(-c2c[nH]nc2C(=O)Nc2cc(C)cnc2O)cc1 CC(C)C(O)(C(=O)N1CCC2(CCCN2C(=O)C=CC(=O)N(C)C)C1)C(F)(F)F c1(C(=O)NC(C)Cn2cc(C3(N(C)C)COC3)nn2)nncc2ccccc12 CCCC(C(=O)NCC12CC1CN(C(=O)COCC=Cc1ccccc1)C2)C(C)C C(CCCOC)(C(=O)NC12CC(CO1)C2)NC(C1C(=C)C1C(=O)OC)=O c1(C(=O)NC2C(NC(=O)CCCCc3cccc(O)c3)C2)cc(F)ccc1F c1(N2C(C(N(C)Cc3n(C)sc3)=O)CC(F)(F)C2)ncc2c(Br)cccc2n1 C1(C(=O)NCCCC(=C)Cl)CC(NC(=O)CCC=CCC=C)CCO1 c12cccc(c1)C(=O)N2.CC(C)(O)C(=O)N(CCC#N)CCC#N C(CN=c1[nH]c(=NCCN2CCCC(C)C2)[nH]c2cc[nH]c12)NC(CC)(C)C C(=O)(CCCC(=O)N1CC(C)CCC1C(=O)NCc1ccc(F)cc1F)OCC N1(C(=O)COCC2CCCC2)CCN(C(c2cccc(F)c2O)=O)C2(CC2)C1 N1(C(CC(=O)NCC)=O)CC2(CC(CNC(c3cncc(C)c3)=O)C2)C1 C12(NC(=O)CC3(C(F)(F)F)CC3)CCCC1N(C(c1ccnc(Cl)c1F)=O)CC2 c1(NC(CC)=O)ccc(O)c(C(N2CCN(C(=O)C=C(Cl)Cl)C3CC23)=O)c1 C1(C(=O)NCCN(C(C(C)(CO)NC(C)=O)=O)C2CC2)CCCCCN1C C1(CCNC(C2(CCC)CC2)=O)CCCN(C(c2cc(OC)ncc2F)=O)CC1 Cc1ccc2c(n1)C(NC(c1nnnn1C(C)C)CC1CCS(=O)(=O)C1)C2 N1(C(CC(CC)C)=O)CCC2CCN(C(=O)C(O)Cc3cnc[nH]3)CC2C1 C1(OC)CN(C(C2CC(F)CN2C)=O)C(C)(CNC(=O)C2=CCCC2)C1 S(=O)(=O)(c1cccc2cccnc12)N1CCC(NC(=O)CC2COCCO2)C1 C1(CNC(c2cc(C)[nH]n2)=O)COCC2(CCN(C(=O)CN3CCSCC3)C2)O1 C1(CC)CN(C(c2ccc(C(=O)CF)cc2)=O)CC1NC(=O)C(C)CSC C(=O)(C1=CC(C)(C)C1)N1CC(CCNC(c2ccc(C(C)C)cc2)=O)C(C)C1 C(c1cccc(N)c1)=CC(N1CCC(N(C(c2c(CC)cno2)=O)CC)C1)=O Cc1cncc(CCC(=O)NC2CC(NC(C3CC3C#N)=O)C2)c1 c1(NC)snc(C)c1C(=O)NC(C)CC(C)NC(c1cn(CC2CC2)nn1)=O Cc1ccc(F)cc1C(=O)NC1CCCC1CNC(C1CCC(N=[N+]=[N-])C1)=O c1(C(C(N2CCCC(C(=O)NC3C(OC)CCC3)C2)=O)(F)F)cnc(O)nc1O N1(C(C(CC=CC)C)=O)CC(C(N2CCCC2CNC(N)=O)=O)C(F)(F)C1 C=Cc1ccc(C(=O)NCC2CCC(NC(=O)C(C)C3CCOC3)CC2)cc1 Cc1ccc2oc(=NC(C)C3CN(C(=O)CCC4CC4(Cl)Cl)CCO3)[nH]c2c1 c1(C(N2CC=CC2CNC(C2CN(C3CCC3)C2)=O)=O)ncc(Br)cc1F c1(C(=O)NCCN(C(=O)C(C)SC(F)(F)F)CCOC)cc(N)cc(O)c1C C1(=O)C(CC(C)C)n2nnnc2C(C2(OC)COC2)N1.c1(OC)ccc(Cl)cc1 N1(C(CCCn2c(C)cc(C)n2)=O)CCN(C(=O)CSCCC#N)C(C)CC1C C1(NC(=O)COC2CN(C(C3CN4CCC3C4)=O)C2)CCC2CC1CO2 C1CCC(=O)N1CCOCCO.n1(CC(=O)NCC(=O)NC2CC2)ncnn1 C(=O)(CCCCCC(=O)OCC)NCC(CNC(CS(CC)(=O)=O)=O)(C)C c1(C(=O)NCCCNC(=O)Cn2cccn2)cc(CO)on1 C(=O)(C(C)(F)C(C)(C)F)NC1C(NC(c2ccnc(OC(C)C)c2F)=O)C1 C12(C(=O)NC3C(NC(C(C)(C)C)=O)CCCC3)CC(CO)(CCO1)C2 CC(C)CC(CNC(C1CC2(C1)CC2F)=O)NC(C1(Oc2ccccc2)CC1)=O N(C(=NCCCF)NC1CCc2sc(Cl)cc21)CC(c1c(C)cccc1)(C)C N1(C(C2(CC(C)=O)CCCC2)=O)CCC(CCNC(c2csc(C)c2)=O)CC1C c1(-c2c(CNC(c3ccc(N4CCCCCC4)nc3)=O)c[nH]n2)cccc(Cl)c1 CCS(=O)CC(=O)N1CCC(C)(NC(=O)C=CI)C1 N1(C(c2nc(C(c3ccccc3)NC(N)=O)no2)=O)CCC(COC)C1(C)C C(=O)(C1=CCCCN(OC(C23CC(C(C)C)(CO2)C3)=O)CC1)OC c1(CC(=O)NCC(C)N(C(=O)Cc2ccc(CO)cc2)C)cccc(Br)c1 CC1CCN(CC(=O)NC(Cc2cc[nH]n2)C(=O)NCCn2ncnn2)CC1 C=C(C)CC(C(=O)N(CC(C)CNC(c1ccoc1C)=O)C)NC(C)=O C1(NC(C2(OC)CCCC2)=O)CCN(C(C2CCCN2C(N)=O)=O)C1C1CC1 C1(CC)C(C(=O)NCC(F)(F)C(=O)OC)CCN1C(=O)Cn1c(O)nnc1O c1(C(=O)NC2(C)CC(NC(C3C4CCC3(c3cscn3)C4)=O)C2)cc(Cl)ccn1 C1(C(=O)NCc2cn(CC)nc2)CC2(CCN(C(c3nc(C)c(Br)s3)=O)CC2)C1 N(C(=NCCc1ccc(Cl)cc1Cl)NCCc1ccc(F)c(Br)c1)C1CC(C)C1CO c1(NC2CC3CN(C(C4(F)CCCC4)=O)CC32)ncc2c(n1)COC2 c1(C(=O)NCC2N(C(C3=C(C)OCC3)=O)CCC2)c[nH]c2ccncc2c1=O Cc1ccc(C(N2CCN(Cc3c(C)noc3C)C3CC23)=O)c(I)c1 c1(C(N2C(CC(=O)NCCCC)CCCC2)=O)cc(OC)ccc1C.C1(=O)CO1 C1(CNC(C(C)(C)OC(C)C)=O)N(C(=O)C(C)O)CCC1(C)C C12(C(N(CCNC(c3coc(Cl)c3)=O)CC)=O)CCCC1CC(F)(F)CC2 C1(C(N2C(CCNC(C3C(CC)C3)=O)CSCC2)=O)C2CC3C(C2=O)C13 C1(CC#C)(C(=O)NCCC2CCN(C(C3CCNC(=O)C3)=O)CC2)CCCCO1 c1(C(CC)N(C(C2CC(=C)CN2C(=O)OCC)=O)C)cc(F)ccc1F CC1(C)CC(NC(=O)C(c2ccco2)NC(C2CC2C2CC2)=O)C1 C1(NC(C(CC=CC)NC(c2csnn2)=O)=O)CC(C)CC(C)(C)C1 C1(CN(C(c2ccc(CSC)o2)=O)C)CN(C(C2(C(F)(F)F)CC2)=O)CC12CC2 N1(C(c2nn(CC)nc2C)=O)CC2=C(C1)CN(C(=O)CC1CCC(C)CC1)C2 c1(C(=O)NC2(CNC(c3c(OC)c(F)ncc3)=O)CC2)cc(F)c(F)cc1F C12(C(=O)NC3CCN(CCC)C3)CC1CCN2C(=O)Cc1nonc1C C1(C(N(CCOCCCN(C(CC(=O)N(C)C)=O)C)C)=O)CCCC2CCCN12 Cc1ccc(CC(N2CC3(CC3)CC2CNC(c2cn[nH]c2)=O)=O)cc1F C12(C(=O)Cc3ncc(OC)cn3)C(N)C3CC1C2C3.C(=O)(C(CC(C)C)OC)N c1(N2CCN(C(CNC(c3c(CC)[nH]nc3Cl)=O)=O)CC2)ccn2nccc2n1 N1(C(CN2C(C)CC2)=O)CC2(C1)CN(C(c1ccc(=O)n(C)n1)=O)C2 N1(C(c2ccnn2CC2CCC2)C(=O)NC2(C)CC2)CCOC2CCC12 CN1CCC(C)(C(=O)NC(CNC(c2cncc(-n3ccnc3)n2)=O)C2CC2)C1 N1(C(C)C)CCOC(CNC(=O)C(N2CCC(c3ccccc3CO)C2)=O)C1 N1(C(C2(c3ccc(C)cc3)CCCCC2)=O)CCCC(NC(C2COC2)=O)C1C c1(OC)ccc(CCCCC(=O)N2CC(NC(=O)COC(F)F)C(C)C2)cc1 C1(CC(N2C(CN(C(c3cc(OC)cnn3)=O)CC)CCC2)=O)COC(C)(C)CO1 N1(C(CCC(=O)NCC)=O)CCCN(C(=O)C(C)(C)NC(c2ccco2)=O)CC1 Cc1cc(F)cc(C(N2CC3CC2CN(C(=O)CCC2CC2(C)C)C3)=O)c1N C1(OCC)CN(C(=O)Cn2ncnn2)CC1CNC(c1cc(Br)co1)=O N1(CC)C(=O)CCC1CC(=O)NCC1CCC1NC(=O)CCSc1nccn1C C1(O)(CCNC(C(C)(CO)OC)=O)CCN(C(c2ccc(N(C)C)cc2)=O)CC1 C(CO)(C(=O)NCCCC1(O)CC1)NC(C1C(C)(CC)C1)=O c1(C(N2CCN(C(c3c(Cl)cnc(CC)n3)=O)CC2)=O)noc2cc(Cl)ccc12 C1(CC(=O)Nc2cnsc2)(NC(=O)CC2CCC2)CCC1 C1(NC(c2cc(C(=O)OC)sc2)=O)CC(NC(=O)C(C)C(C)F)CC1O CC1CCN(c2nc(=N)nc(N3CCOC(CSC4CC4)C3)[nH]2)CCS1(=O)=O c1(N2C(C)(CNC(=O)C3=CCC3)CC(F)(F)C2)ncnc2ccc([N+](=O)[O-])cc12 O=C(CCC(=O)N1CCCCC1)N1CCCC1NCc1ccccc1I C(=O)(C1SCCc2sccc21)N(CCNC(c1ccnc2ncccc12)=O)CC CC#CC1CN(C(C2CN(C(C3(COC)CC=CC3)=O)CCO2)=O)C1 C1(NC(C(CN(C)C)O)=O)CC2(CCCCN2C(c2cnc([N+](=O)[O-])n2C)=O)C1 c1(CC)c(N2CCN(C(=O)C(C)N(S(=O)(=O)CC)CC)C(C)C2)nc(C)nc1Cl C(=O)(C1CN(C)C(=O)c2ccccc21)N1C(CN(C(CC(CC)CC)=O)CC)CC1 CC1CCCN(C(=O)C(=O)NCCC2CCN(CCCS(=O)(=O)N(C)C)C2)C1 C1(C(N2CC(C)(CC)C2)=O)CC(NC(=O)C(c2ccn(C)c2)C)CCO1 CCCCC(CCCC)C(=O)N1CC2CCN(c3ccnc(C4CCC4)n3)C2C1 C12(NC(CC(CC)(F)F)=O)CCCC1CN(C(=O)C(CSC)c1ccccc1)C2 Cc1noc(C)c1CN(C(=O)C(C1CCN(C(c2cnc(=N)[nH]c2)=O)C1)F)C C(=O)(CCC(=O)N1CC2CC2(NC(c2csc(C(C)(C)C)c2)=O)C1)OCC c1(CCC)sc(C(N2CCC(CF)(NC(=O)Cc3cccnc3)C2)=O)cc1CC C(=O)(CC(C)CNC(C1CCN(C(=O)CC(C)C2CCCO2)C1)=O)NC C(=O)(CC(C)CNC(=O)CCCC1CC1C)NCC1(COC)CN(C)C1 c1(C(=O)NCCN(C(=O)CCc2ccn(C)n2)CC)cc(F)cc(S(N)(=O)=O)c1 C#Cc1ccc(C(=O)NC2(C)CCN(C(C34CC(c5ccccc5)(C3)C4)=O)C2)cc1 N#CC1(C(N2CCC(NC(C3CC=CC3)=O)C2)=O)CCCCCC1 CC1(C)CCCC(C)(NC(C2CCN2C(=O)CC2CCCC23CC3)=O)C1 c12nn(C)c3c1CN(CC3)C(=O)CCCNC2.CC(C)C(=O)NCCNC(N)=O c1(C(N2C3CC(NC(CC4CCN(C)C4)=O)C3CC2)=O)cccc(C#CCO)c1 N1(Cc2cc(C)ns2)CCC2C(CCCN2C(C2CCCN2CC(F)(F)F)=O)C1 CCC(C)C(=O)C(=O)N1CCC(CC)C1CNC(=O)C(C)(F)F CC(N=c1[nH]c(=NCC2(OCCO)CCOC2)[nH]c2cc[nH]c12)c1c[nH]ccc1=O C(=O)(CCCCCCNC(=O)C(C)(O)C1CC1)N(C)CC1CCN(C)C1 c1(CC)ncccc1C(=O)NCCSc1ccccc1F.c1(C=O)[nH]cc(C)c1C CCCC(C(=O)NC(CNC(C1CC(=O)N(c2ccc(F)cc2)C1)=O)CO)OC C1(C(N2CC(CNC(C3CCCS(=O)(=O)C3)=O)C2)=O)CC(C2CC2)=NO1 c1(C(N2CC(CC(C)NC(C(=O)NC(C)C)=O)C2)=O)cc(Br)sc1Cl N1(C(CS(CC)(=O)=O)=O)CCC12CCCN(C(c1cnc3ccccn13)=O)C2 C(C(=O)NCC(F)C1CCC1)(C(C)(C)C)NC(C(CC)N(C)C)=O Cc1cc(N)n2ncc(C(N3CC(F)(CNC(=O)C(C)P(C)(C)=O)C3)=O)c2n1 c1(OCC=C)ccc(C(=O)NC2C=CCN(C(C3CC4CCC4C3)=O)C2)cc1 N#CC1CN(C(=O)CCC(N)=O)CC1NC(=O)C1=COCCC1 Cc1ccc(C)c(C(=O)Nc2cc(C)n(-c3ccc(Br)cc3)n2)c1O C1(NC(C2CCN(CC)C2)=O)CCCCC1CC(=O)NOCCOC C(=O)(N=c1[nH]c(Cl)c(C#N)s1)c1c(C)nn(CC(=O)N(C)C)c1C C(=O)(CCC(=O)c1ccccc1N)N(C)CC1(NC(C(C)SC)=O)CC1 OCCCC(C(=O)O)NCc1ccc(-c2ccncc2)cc1 C1(CNC(CN(C(C(C)C2(O)CCC2)=O)C2CC2)=O)CC2OC1C1CC21 C1(NC(c2c(CC)scn2)=O)CN(C(=O)CC2CCCCC2)C(C)(CC)C1 N1(C(CCOCC#C)=O)CC2CCC1CN2C(C1CC1(F)C(=O)OCC)=O CCCS(=O)(=O)c1ccc(C(=O)NC2C3CN(C(C4CC=CCC4)=O)CC23)cc1 c1(C(N(CC(C)N(C(C2C(OCC)C2)=O)C)C)=O)ccnc(N(C)C)c1 CCC(C)C(CC(=O)NCC1CCOC1)NC(=O)C(CC)(CC)OC CC1OC(C)CC1CC(N1CC(CN(C)C(C2CC2C)=O)C1)=O c1(C(N2CCCC(O)(CNC(C(C)O)=O)C2)=O)cn(C)c2c(Cl)cccc12 Cc1cc(C(F)F)nn1CC(N1CC(CNC(=O)Cc2csc(S)n2)CC1C)=O C1(CCN(C(=O)CC(C)(C)F)C)CCCCN1C(=O)C=Cc1cc[nH]n1 N1(C(C(F)=CCC)=O)CC(OC)CC(NC(=O)CCn2nc(C)c(C)c2C)C1 c1(C(N2CCN(C(C3(CC#C)CCC3)=O)CC2CC)=O)cccc2oc(=N)[nH]c12 C(=O)(C1CCCc2n[nH]cc21)NC1CC(O)CCN(C(C2CN(C)C2)=O)C1 CCC(CC(=O)N1CC(C(C)(C)O)(CNC(c2cccc(O)n2)=O)C1)SC n1(C(CC)CC)nc(C2CC=CCC2)nc1-c1cnoc1C CC1CCN(C(=O)C=Cc2cncc(O)c2)CCN1C(C1CC1F)=O C1(C(N(C(CC)=O)C(C)C)=O)CCCN1NC(=O)c1ccc(C)nc1 c1(C(=O)NCC(C)N(C)C(c2ccc3nn[nH]c3c2)=O)ccnc2c1ccn2C c1(OC)cccc2sc(C(=O)NCC3CCN3C(C3CCC(F)(F)CC3)=O)cc12 c1(C(N(CCOC)CCNC(c2ccncn2)=O)=O)nc(C)c(N(C)C)s1 N1(CC2CCN(C(c3cc(C)ns3)C(=O)NCC(C)C)C2)CC(C)OC(C)C1 c1(OC)cc(CNC2(c3nnnn3C)CCCC2)c(C)cc1C CCC(CCCC(=O)NCC(=O)NCC(F)F)NC(C1(COC)CC=CC1)=O CC1CN(C(C2COCCN2C)=O)CC1NC(c1cc(CO)on1)=O c1(C(=O)NC2CC(NC(C3CC4CC4C3)=O)C2)cc2cc(Br)cn2cn1 C=C(C(=O)NC1CN(C(c2ccc(C)cc2OC)=O)CCC1F)C(F)(F)F C1(CC(=O)N(C(C)COC)CC)C2CCCC2N1C(=O)C=Cc1cc[nH]c1 C1(CNC(c2c(C)nccn2)=O)Cc2ccccc2CN1C(C1(N(C)C)CC1)=O CC(C)CCCC(C)C(=O)NC(c1nc(C(=O)NC(C)Cc2nn[nH]n2)co1)C C1(C(=O)NCCNCCCNC(c2c(SC)cccn2)=O)CC(C)(C)CN1C n1(C2(C(=O)NC(CNC(C(C)NC(C)=O)=O)CO)CC2)ncc(Br)n1 C1(C)(C(N2CC(c3c(CNC(CC=C)=O)nco3)C2)=O)CCCCCC1 Cn1nc(C(=O)NCCC2CCN(C(=O)C=Cc3ccccc3)C2)cc1Cl c1(C(=O)NCC(C(=O)NC2COC(C(C)C)C2)OC)ccc(O)cn1 c1(CN(C(C)C2CC2)CC23CC(F)(CO2)C3)nnc2n1CCC2 c1(C(=O)NCCC(C)NC(c2cc(C#N)ccn2)=O)cccc2c1NC(=O)CO2 C(=O)(C1=CC2(CN(C(C3(C)CCCC3O)=O)C2)OC1)NCCOCC#C C1(C(c2csnn2)NCc2nnnn2C(C)(C)C)(OC)CCCC1 c1(NC(=O)NC(C#C)CC(C)(C)C)oc2ccc(Br)cc2c1C C1(NC(C2C(=C)C2)=O)CN(C(c2ccccc2COC(C)(C)C)=O)CC1(C)C C1(C(N(C)CC2(NC(c3cnc4n3CCS4)=O)CC2)=O)CN(CP(C)(C)=O)C1 c1(N2CCC(N(C(=O)Cc3cncnc3)C)CC2)nc(C(F)(F)F)ccc1C#N N1(C(C2C(C)=CCS2)=O)CCOC(C)C1C(=O)NCCCC1CC(C)C1 C1(CC(=O)NCC(C)CNC(C2CS(=O)(=O)C2)=O)CC2C=CC1CC2 N1(C(Cn2ncc(C)c2)=O)CCCCC1Cn1cc(C(N2CCCC2)C)nn1 C1(CCNC(c2n(CCCC)nnn2)c2ocnc2CC)CCC2(CCC2)O1 c1(C(=O)NCCCC2OCCN(C(C(CC=CC)C)=O)C2)cc([N+](=O)[O-])oc1C c1(NC(C2(CCOC)CCNCC2)=O)ccc2c(ccn2C(C)=O)c1 N1(C(CCC#N)=O)CC2CC1CCC2NC(=O)CCc1ncc[nH]1 c1(OC)cc(=NC(=O)N2CCCC(O)(CCCCn3ccnn3)C2)[nH]n1C N1(C(CSCCCC)=O)CCn2nc(C)c(CNC(=O)CCC3CCOC3)c2C1 c1(C(=O)NC2(CF)CCN(C(C(COC)(C)O)=O)C2)ccc(OC)cc1OC c1(C(=O)NC)csc(C(c2nnnn2C2CC2)NC(C)CC(=O)OC(C)(C)C)n1 N1(C(C(C)OCCCC)=O)CC(N2CCCC(CC(N)=O)C2)C(F)C1 N1(C(c2cc(CC)no2)=O)CCC(C(=O)NCC2C(=O)NN=C2C)C(O)C1 C(C)(C(CC(=O)NCCn1ccc(=O)cc1)NC(C1(C2CC2)CC1)=O)OC C1(CC)CN(C(c2cnn(CC)c2)=O)CCN1C(=O)Cc1cccc(F)c1OC c1(C(N2CCN(C(C(CC)COC)=O)C(C)C2C)=O)ccc2nc(CO)[nH]c2c1 N1(C(C2(CNC(C(C)SC(C)C)=O)CC(C)(C)C2)=O)C2CCC1CC1(C2)N=N1 C1(O)(CC(=O)N(C(CNC(=O)Cc2csc(=N)[nH]2)C2CC2)C)CCOCC1 Cc1nc(Cl)ccc1CC(=O)N(C1CN(C(=O)C(C)c2ccsc2)C1)C C(CC1CCCO1)(C(=O)NN(C)CC1(O)CC(Cc2ncc(C)[nH]2)C1)OCC N1(C(CS(N)(=O)=O)=O)CCC(NC(C2CN3CCN2CC3)=O)C(C(N)=O)C1 C(=O)(C(C)(C)CC1CCC1)N1CCC(N(C(C(N2CCCCC2)C)=O)C)C1 c1(C(=O)NC(CCN(C)C(c2ccns2)=O)c2cccs2)nc(=O)n(C)[nH]1 C(=O)(C(O)CCNC(C1CC(O)CN1C(C1CC=CC1)=O)=O)OC c1(CNC(CC2(NC(C=C(C)c3ccco3)=O)CC2)=O)ccn(C)c(=O)c1 c1(N(C)C)nc(C(=O)NC2(C)CCN(C(C3(Cl)CC3)=O)C2)[nH]c(=N)n1 c1(CC)cccc2[nH]c(C(=O)NCCCCCNC(=O)COC(C)C)cc12 C1(C)(C(=O)NCC2(F)CCN(C(C3CCC(=C)CC3)=O)C2)CCCNC1=O N1(C(C(CC)C(C)C)=O)CC2=C(C1)CN(C(c1ccc(Cl)cc1)=O)C2 C1(NC(C2C(CC(C)C)C2)=O)CC(C)(NC(=O)CC(C)n2cccn2)C1 c1(N2C(CNC(c3ccc(C)s3)=O)COCC2)ncc2cccc(O)c2n1 c1(C(=O)NC2C3CN(C(C4(COC)CCCC4)=O)CC32)ccc(=O)n(CCF)n1 c1(C(=O)NC2C(NC(c3ccc(CSCCC)o3)=O)CCC2)cc(N)ccc1Cl N1(CCNC(C=CC)=O)CCCN(C(c2cn(C)nc2-c2ccccc2)=O)CC1 C1(C(C(=O)NC(C)CCNC(c2cc(Cl)n(C)n2)=O)C)CCC(C)(C)CC1 CC(C)(C)CC(C(=O)NC1CC2C=CCC(C1)C2)NC(c1c[nH]c(=O)cn1)=O C1(CNC(=O)COC2COC2)CCN(C(=O)CCc2cncc(F)c2)CC1 N1(C(c2c(CC)c[nH]n2)=O)CCCC(CN(C(=O)CC(C)(C)F)C2CC2)C1 c1(C(=O)NCC(C)(CC(C)C)NC(Cc2c(C)occ2)=O)nc(O)nc(O)c1F C(=O)(C(CC(C)C)ONC(C12CCN(CC1)CC2)=O)NC(c1ccnc(O)c1)C C12(CC(=O)N(CC(CC)NC(c3c(Cl)c(C)nn3C)=O)C)CCCN1CCC2 c1(CNC(CC(C2CC2)NC(c2ccc(=N)[nH]c2)=O)=O)cc(O)cc(F)c1 C1(CN(C)C(c2cscc2C(F)F)=O)COCCN1C(=O)C=CC(C)(C)C N#CC1(C(N2CCCCC2CNC(c2ccnnc2S)=O)=O)CC2CC2C1 C1(C(N2CCC(CCNC(c3cc(CO)[nH]n3)=O)C2)=O)Cc2ccccc2CO1 c1(N2CC(C(N)=O)(CNC(C(C)OCc3ccccc3)=O)C2)ncnc(=N)[nH]1 N1(C(C2OCCC(C)(C)C2)=O)CCC2(C=C(C(=O)NC3CCN(CCF)C3)C2)C1 C1(COC)CCC(C(=O)NCCCN(C(=O)CN2CC=CC2)C)C1 c1(C(=O)NC2CC(C)(NC(c3c(C(C)C)ccs3)=O)C2)cncc(C2CC2)c1 c1(OC)cc(NCC2C3CN(C(C4COC(C)C4)=O)CC23)ccc1[N+](=O)[O-] c1(C(N2CCCN(CCNC(C(C(C)O)C)=O)CC2)=O)cnc2n(c1=O)CCS2 N1(C(C2CCC(CNC(C3CC=CCC3)=O)O2)=O)CC(C2CC2(F)F)C1 Cc1cc(F)ccc1CC(=O)Nc1cc(C(F)(F)F)ccc1N1CCCCC1 c1(CCC(=O)N(CCN(C(CCNC(=O)NC)=O)C)C)ccc(F)cc1F C1(C(=O)Nc2c(CC)nn(C)c2)COC2(C1)CN(C(=O)CC1C=CCC1)C2 Cc1cc(C(=O)NCC2N(C(CC3C(CC)C3)=O)CC2O)ns1 C1(NC(C2CCC(CNC(C3(CSC)CC3)=O)C2)=O)Cc2cncn2C(=O)N1 Cc1cccn2ncc(C(=O)NC3CC(F)CN(C(=O)C(C)c4ccco4)C3)c12 C(=O)(C1COCc2ccccc21)NCC(CNC(c1cnn(CC)c1C)=O)(C)C C(C)(CC(=O)OC)SC.N1(C)CCOCC1.c1(C2C(=O)N2C2CC2)cn(C)nn1 c1(C(N2CCCC(NC(C3C(C(C)C)C3)=O)C2)=O)cc(N)c(Cl)cn1 N1(C(CC(COC)(C)O)=O)CC2(C1)SCCC2NC(=O)CN1C(=O)CNC1=O C12(C(=O)NC(c3cccc(C)c3)C(=O)Nc3c(OC)nsc3)CCC(CC1)CO2 C12(C(=O)OC)COCC1CN(C(=O)C(=O)NC1CCCC1C1CC1)C2 C1(NC(CCN(C)CCO)=O)CCCN(C(c2ccc(F)nc2F)=O)CC1 C(C(CC(C)C)C(=O)NC(CC(=O)NCC1(C2CC2)CCCO1)C(F)(F)F)OC c1(NC(N2C(c3n(C)ncc3)CCC2)=O)cc(C#N)cnn1 C1(NC(C=CC(C)NC(c2nc(C)n(C)c2)=O)=O)CCCCCC1C C1(C(=O)NCC2CC(NC(c3c(C)nc(C)[nH]3)=O)C2)CC1C1(C)COC1 C1(C(=O)NCC=CCNC(C2CCCN(CC)C2)=O)CCc2nncn2CC1 Cc1ccccc1NNC(=O)C=CCN(C)C CC(CN1CCCC1)CN=c1cc[nH]cc1Cl C(CN=c1[nH]c(=N)[nH]c(=NCC(c2ccco2)C2CCCC2)[nH]1)N(C(C)C)C N1(C(C(C2CN(C(C3(OC)CCCC3)=O)C2)O)=O)CC(C)CCCC1C C(=O)(C1=NOC(c2ccccc2)C1)NCC1C(NC(CC2C(OCC)CC2)=O)C1 C12(C(N(C(C)(C)CNC(=O)COc3cccc(O)c3)C)=O)CC1CCC2(F)F C1(C(C)C)CN(C(c2cnc(O)o2)=O)CC1C(=O)NC(C)CCO C1(NC(C(C)CO)=O)CC2(CCCCN2C(=O)CNS(N)(=O)=O)C1 c1(C(=O)NC2CCC(CCNC(c3ccc(CC)o3)=O)C2)ncc(C)cn1 c1(CC(CN(C)C(C2(C)CSC2)=O)NC(C=C(CSC)C)=O)ccccc1 c1(CN(CC(=O)NCCC(C)N(C)C(C2CC=CCO2)=O)C)ccccc1 C1(CNC(CC2CC(CC)C2)=O)(OC)CN(C(c2coc(C)n2)=O)C1 N1(C(CCC(C)O)=O)CCC(CNC(=O)COC2CCCCC2C)C1(C)C c1ccccc1.C12CC(C1)COC2=O.C12(CC1)C1C(C1)NC2=O.CCOC C1(CN(C(=O)CC2CNC(=O)O2)C)CN(C(C2C=CCS2)=O)CCO1 N1(C(CCC(C)(C)OC)=O)CC(C(=O)NC(C)Cc2ccncc2)CCC1(C)C c1(C(N(C(CNC(C2(CO)CC(F)(F)C2)=O)C2CC2)C)=O)cccc2sccc12 CCCCCC(=O)NCC(=O)N(CCNC(=O)C(O)CN1CCCC1)CC c1(C(=O)NCCCNC(c2ccc(F)c(F)c2F)=O)ccc2nc[nH]c2n1 C1(CNC(C2(C=C)CCC2)=O)CN(C(c2ncc(OC)nc2OC)=O)CC1(F)F C1(CCC)(NC(=O)Cn2nc(C)cc2C)CCCN(C(c2cc(=O)n(C)o2)=O)C1 c1(OC)ccc(C)c(C(=O)NC2CN(C(=O)C(C)(C)C(=O)N(C)C)CC23CC3)c1 S(=O)(=O)(c1cccc(F)c1)NC1C(C(=O)NCC2CCCC(C)C2)C1 c1(C(=O)NC2(C)CCN(C(CCn3ncc(C)c3)=O)CC2)ccn2ccnc2c1 CCCC(CC(C)C)C(=O)NCCN(C(=O)CC(C)(C)C(F)(F)F)C1CC1 N1(C(C=C(CC)C)=O)CC2(CCC(CNC(=O)C(c3ncccc3F)(F)F)O2)C1 c1(C(=O)NCC2(F)CC(CNC(COCCC)=O)C2)ccncc1OC(C)C c1(C(=O)NCC2N(C(C=Cc3scc(C)n3)=O)CCC2)cccc(C)c1O C1(N(CCN)C)CCCN(S(=O)(=O)C(F)F)C1 N1(C(c2c(CC)con2)=O)CCCCC(NC(=O)C(C)NS(C)(=O)=O)C1 c1(CC)c(NC(=O)C(=O)NC(c2ccnc(Cl)c2)C2CC2)cnn1C Cc1[nH]nc(C(N2CC3CC2C3CNC(C2CCCC2)=O)=O)c1Cl c1(CN(C(C2CCN(c3ccccn3)CC2O)=O)CC2CC2)c(F)cccc1F c1(OC)cc(C)c(C(N2CCC(CN(C)C(C3(C#N)CCCO3)=O)C2)=O)c(C)c1 c1(C(N2C(C(=O)NC(COCC)C(C)C)CC(F)C2)=O)cnc(C)c(C#N)c1 N1(C(C(COC)O)=O)CC2CC3CC2C1C3NC(c1cc(C(F)(F)F)ccn1)=O c1(C(N2CC(C)(CC(=O)Nc3ccc(F)c(CO)c3)C2)=O)cc(F)c(O)c(F)c1 C12(C(N3CCC(CN(c4nccc(OCC)n4)C)C3)=O)CC3CC(C(=O)N1)C2C3 N1(C(COCC(=C)C)=O)CC(OC)C(NC(=O)CSc2nccn2C)C1 O=C(C#CC1CCCC1)N1CC2(CC3CN(N4CCC5CCCC45)C3)CC1CO2 N1(C(c2c(OC)nsc2)=O)CCCN(C(c2coc(SC)c2)=O)C(C(C)C)C1 N1(C(CCC=C)=O)CCC(C(N2CCCC(C=C)C2)=O)C12CC2 Cc1cc(Cl)ccc1C(=O)NC(C)(CNC(c1cc(F)n(C)n1)=O)CO c1(CC)cccc(C(=O)N(C)CCN(C)C(c2cc(C(F)(F)F)on2)=O)c1O c1(NC(C(CC)C)=O)cnc(Cl)cc1C(=O)Nc1ccccc1C(C)(C)O N1(CCC)CCC=C(c2c[nH]nc2C(=O)Nc2ccc(-c3cscc3C)nc2)C1 N1(C(CC(C)(F)F)=O)CC2(C1)CN(C(c1ccc(F)cc1C(F)(F)F)=O)CCO2 c1(C(N2CCCC2CC2CN(C(c3cc(C(=O)OC)sc3)=O)C2)=O)nc(O)sc1C C1(CC#C)(NC(C2CC(C(F)C(=O)NCCC=CCOC)C2)=O)CCOC1 C1(CCNC(C(N(C(C(C2CC2)SC)=O)C)C2CC2)=O)CCCCCC1 C12(C(=O)NC(CCC(=C)C)C)CCC(CC1NC(C13CC(CO)(C1)C3)=O)C2 CC1=C(C)CC(C(=O)NCCC2COCCN2C(=O)CN2CCCCC2)CC1 C1(c2n(C)ncc2)CCCC(N=c2ccc3c([nH]2)CCCC3=O)C1 C12(NC(C3C(CNC(C(C)c4ccsc4)=O)CC3)=O)CCCN(CCC1)C2 c1(NC(C(=O)NC(CN(C(c2ccc(I)cc2)=O)CC)C)=O)ccc(NC)cc1 c1(OC)cc(C(=O)NC2CC(CN(C)C(c3ccn(CC4CC4)n3)=O)C2)[nH]n1 c1(CNC(C2CCCN2C(=O)COC2CCOC2)=O)cc(F)cc(F)c1 C(=O)(CCC(=O)NCCN(C(=O)COC1CCOCC1)C(C)C)NCCCOC C1(N(C(=O)C(C)(C)NC(=O)Cc2cncs2)C)COC(C)(C)C1 c1(C(=O)Nc2n[nH]c(Cn3c(O)nnc3O)n2)ccc([N+](=O)[O-])nc1 N1(C(CN(CC)CC)=O)CCC(F)(F)C(CNC(c2cc3cnccc3o2)=O)C1 C1(C)(NC(C(C=C)OC)=O)CCCCC1C(=O)N(CC(=O)OCC)CC C(=O)(C(=O)N=S(C)(C)=O)NC1CN(C(c2ccc(C(C)(C)C)o2)=O)CC(O)C1 CCC(CC(=O)NC1CCC1NC(=O)C(C)(C)CC1CCC1)C1CC1 c1(CN(C)C)cc(O)ccc1F.C12CCCCC1NC(=O)c1c[nH]c(c1)C(=O)N2 N1(C(C(C)C(F)F)=O)CCC(NC(=O)C=Cc2ccncn2)C12CCC2 N1(C(C2(C#N)C(C)(C)C2)=O)CCC(C2(NC(=O)C(F)C(C)(C)O)CCC2)CC1 c1(C(=O)NCC2OCCN(C(C3(COC)CCCCC3)=O)C2)nccc(Cl)c1C c1(C(=O)NCCS(CC)=O)cnc(CNC(C2(C)CCCCC2)=O)nc1 CCCCS(=O)(=O)CC(=O)NC1CN(C(C2CN3CCN2CC3)=O)CC1C C=CCCCC(C(=O)NC1CCC1)N1CCCC(c2ccncn2)C1 c1(C(N2CCC(OC)(CNC(=O)C(C)OCC(C)C)C2)=O)c(C)cccc1O c1(OCC)cc(C(=O)NCCC2CCN(C(C3CC3CF)=O)C2)cc(Cl)c1O C1(CNC(C2CCC(=C)CC2)=O)CN(C(c2ccsc2OC)=O)CC1(F)F C1(NC(c2scc(C)c2)=O)COC2(CCN(C(=O)CCc3ccccc3Cl)C2)C1 C(CS(C)(=O)=O)N(C)C(C1CNC2CC12)=O C1(NC(c2ccc(Cl)nn2)=O)COC2(C1)CN(C(C1C(F)(F)C13CCC3)=O)C2 C1(C(C(=O)NCC(=C)CC)C)CCCN(C(c2cnn(CC)c2C)=O)C1 C(N=c1ccc(C#N)c[nH]1)C1CN(C(Cc2ccc(CC)s2)=O)C(C)C1 c1(C(=O)NC(CN(C(c2c(C(C)C)ncs2)=O)C)C)cccc(O)n1 C1(NC(Cc2nc(C)sc2)=O)(CNC(=O)C(c2cnn(C)c2)C)CCCCCC1 N1(C(c2onc(OC)c2Br)=O)CCC(NC(=O)Cc2csnn2)C(F)C1 c1(C(=O)NC2COCCN(C(C3C(C4C(C)C4)C3)=O)C2)ccc2nncn2c1 c1(CC(=O)NC(CNC(c2c(C)c(N)cnc2)=O)C)cnc2n1CCCC2C N(C1CCCOc2ccc(C)cc21)(C(CS(CCC)(=O)=O)=O)C1CC1 C(=O)(CCCC(N)=O)NC(C(C)NC(c1cc(C(C)C)[nH]c1C(C)C)=O)CO CC1CN(C(c2ccc3c(n2)CCOC3)=O)CC(C)N(C(C2CC=CCO2)=O)C1 C(CC(C)C(=O)N1CCCC1CNC(c1cc[nH]c1C(C)C)=O)OC N1(C(c2c(C(=O)OCC)cnn2C)=O)CC2CC(NC(=O)C(C)(C)SC3CC3)C1C2 Cc1cc(C)c(CN2CCC(N(C)C(c3cc(Cl)nnc3O)=O)C2)cc1C N1(CC(=O)N(C(C2CCCOC2)=O)CC)CCC(Cc2ccccc2O)CC1 C1(C(=O)NCCOCCOCCNC(C=NOC)=O)CCC(=O)N2CCCC12 C1(O)(C(C)NC(C(CCC)O)=O)CCN(C(c2cnn(C)c2)=O)CC1 N1(C(C)C)CC(C(=O)NC(C)CCNC(c2cn(C)nc2C(C)(F)F)=O)CC1=O Cc1csnc1C(=O)N(C1CCCC1)CCNC(=O)CC1CC1 CC#CC1CCN(C(=O)C(C(C)C)NC(c2cscc2OC)=O)CC1 C1(C2CCC2)C(=O)S1.C1(CN)CCC1.C(C)(C)(CNCC(=O)OC)OC(C)C CCCCC(O)CC(=O)NCC1CN(C(C2CN(C)C(=O)N2)=O)CCCO1 c1(C(N2CC(C(N3CCOC4(CC4)C3)=O)C(F)C2)=O)nccc2cc[nH]c12 c1(C(C)C)cc(=NCC2CCCCN2C(=O)CNC(c2ccccc2)=O)[nH]cn1 c1(NC(CN2C(NCC(C(C)C)c3ccnn3C)CC2)=O)ccnc(Cl)n1 C=CC(C)(C)C(=O)N1CCC(CCC(=O)NCC2COC(=O)N2)CC1 C1(C)(NC(C(C)Cc2ccncc2)=O)CCC(NC(=O)OC(C)(C)C)C1 c1(COC(=O)CC2(c3ccco3)CC2)csc(C2CC2)n1 c1(CC2(C(=O)NC3(CNC(c4c(C)[nH]cc4)=O)CC3)CC2)ccccc1F C1(C(C(=O)N(C(c2ccc(Cl)cc2)COC)C)N)Cc2ccccc2C1 N1(C(N2C(CSCC)CCCC2)=O)CCN(c2ccccc2CSCC)C(C)C1=O c1(C(N2C(COC)CN(C(c3ccsc3)=O)CC2)=O)cn2cc(C)sc2n1 CN1CCN(C(=O)CCCCCCn2cc(C3(O)CC3)nn2)CC12CCCCC2 C12(CNC(c3n[nH]cc3Br)=O)CCC(C1)N(C(=O)CCC1CCCC1)C2 c1(NC(C(C)(C#N)c2ccccc2)=O)cc(Br)ccc1F N1(C(C(CCCC)O)=O)CCN(C(C2CCC(=O)O2)=O)CC(C)(C)C1 C1(NC(C(CC)=CCCC)=O)CCSC12CN(C(C1CCCN1S(C)(=O)=O)=O)C2 C#Cc1cccc(OCC(N2CCN(C(=O)CCCCN(C)C)C(CC)C2)=O)c1 CC(CCCNC(C1(F)CCOC1)=O)NC(=O)CSCCN(C)C N1(CCC(=O)NCCN(C(=O)C(O)(C2CC2)C2CC2)CC(C)O)CCNC(=O)C1 C12(NC(C(CC(C)C)O)=O)CCCC1N(C(c1cnc(-c3cccs3)[nH]1)=O)CC2 c1(C(N(C)CC2OCCN(C(C(C#C)(C)C)=O)C2)=O)ccc(OCC)c(Cl)c1 c1(C(=O)NCC23CC(NC(C4(SC)CC4)=O)(C2)C3)cccc(N2CCCCC2)c1 c1(C(=O)NCC2(F)CN(C(C3CC34CCOC4)=O)C2)nnn2c1C(=O)NCC2 c1(C(=O)NC2C(NC(c3cnc(CC)nc3C)=O)CC2)ccc2nn(C)cc2c1 c1(CC(=O)NC23CC(C2)N(C(=O)C(O)C2(O)CCC2)C3)ccc(O)c(O)c1 C1(CNC(Cn2c(C)ncc2)=O)CN(C(=O)C(C)C(C)(C)C)CC1(F)F Cc1ccc(C(=O)NCC2(O)CN(C(=O)C=CCOC3CCOCC3)C2)c(N)c1Cl C(=O)(C(CCC1CC1)NC(c1cc(C(F)F)[nH]n1)=O)NCCc1cc(C)on1 C1(CNC(C2C(OCC)CC2)=O)CC2(CC(OCC3CC3)C2)C1 CCC(CCC(=O)NC1CCC(C)N(C(=O)CC2(OC)CCCCC2)C1)OC c1(CC(=O)NCCNC(CCCN(C(C)=O)C)=O)ccc(N2CCOC2=O)cc1 C(=O)(CC(C)(C)S)N1CCC(C(=O)NC2(CC(=O)O)C(C)C2)C1.C(C)(C)(C)NC=O N1(C(CCC#C)=O)CCN(C(c2conc2COC)=O)CC1CCO c1(NC(C2CC(NCc3c(CO)nn(C)c3O)C2)=O)c([N+](=O)[O-])ccc(Cl)c1Cl c1(SC)ccc(Cl)c(C(=O)NC2CN(C(c3cccc(C)c3O)=O)CC2O)c1 C(=O)(C#CC1CCCOC1)N1CCCN(C(C2CC2(F)F)=O)CC1CO c1(C(=O)NCC2C(NC(c3c(C)ncs3)=O)CC2)ncccc1N(C)C c1(CC)cc(C)ccc1C(=O)N(C(C)CCNC(=O)C=CC(=O)NC1CC1)C N(C(=NCCCCl)NC1CCCCC1C)Cc1c(C)cccc1OC(C)(C)C c1(CC(C(=O)NC2CC(C(C)(C)C)C2)NC(COC)=O)ccccc1Br c1(C(=O)NC2(CF)CCN(C(C=CC)=O)C2)cc(OC)c(C)c([N+](=O)[O-])c1 C1(NC(c2ccsn2)=O)CCN(C(C2(F)CCCC2)=O)CC1F C(=O)(C1CCc2cccc(O)c21)N1CC(C2CC2)C1.c1(CC)ccc2cc1NC2=O C=C(Cl)CCC(=O)N1CCC=CC1C(=O)NOCCC(C)O C1(CCNC(C2(COC)COC2)=O)CCN(C(c2cncn2C2CC2)=O)CC1 c1(CNc2ccc(C(N3CCC(O)(C(F)F)C3)=O)nc2)cc(F)cnc1Cl C1(CNC(c2nccc(CC)c2)=O)CCN(C(c2sc(C)cc2C)=O)C12CCC2 c1(CNC2C(C(=O)NCc3cnccn3)CCC2)ccc2cc[nH]c2n1 c1(CC(=O)NC2COCC2NC(C2CNC(=O)N2)=O)ccc(-n2cccc2)cc1 N1(C(C2CC(C)NC(=O)C2)=O)CCN(C(=O)Cc2c(F)cccc2F)CC(O)C1 c1(C(=O)NC2CCC(C(=O)Nc3c(C)ccnc3Cl)OC2)ccc(I)c(F)c1F Cc1c[nH]c(CC(N)=O)c1C(=O)NCC12CC(NC(c3ccncn3)=O)(C1)C2 N1(C(c2nn(C(C)C)nc2Br)C(=O)NCc2ccco2)CC(C)S(=O)(=O)C(C)C1 CCC(CC(=O)NCCC(C)NC(=O)COC)C1CCC1 N1(C(C=CCC)=O)CCOCC1CN(C)C(c1ccc(N2CCOCC2)nc1)=O N1(C(C2CCN(C)C2)=O)CCC(C2(NC(C3OCCOC3(C)C)=O)CCC2)CC1 c1(OC)ccc(S(=O)(=O)NCc2ccco2)cc1C=C1CCC(C(=O)O)CC1 C(CC(=O)N1CC2CCN(C)C2C1)(C(F)(F)F)NC(C(C(CC)C)=O)=O C12(NC(COCCCOC)=O)CCC1CN(C(c1cc(N)nc(Br)c1)=O)C2 c1(C(=O)NC(CC)CNC(=O)COC(C)C)sc(O)nc1C N1(C(C(C)SC(C)C)=O)CC2CC1CCN2C(c1cccnc1)=O C12(CC(N3C(C(=O)OC)C=CC3)=O)CCC1CN(C(=O)C1=C(C)CC1)C2 N1(C(Cc2nc(CC)sc2)=O)CCN(C(C2CS(=O)(=O)CCO2)=O)C(CC)C1 c1(C(N2CC(NC(c3nc(C)sc3)=O)C(F)(F)CC2)=O)cc(O)cc([N+](=O)[O-])c1 N1(C(CC(C=C)(C)C)=O)CCC2(C1)CN(C(C1CCCCS1)=O)CCO2 c1(C(N2CC3CCCC(C2)N3C(c2cnns2)=O)=O)c(F)cccc1[N+](=O)[O-] c1(C(=O)NCCCN(C(C2C(OCC)C2)=O)C(C)C)cn(C2CCOC2)nn1 Cc1ccccc1CCNC(C)(CCCO)c1nnnn1C1CCOC1 Cc1cc(C(=O)NCCCN2CCC(NC(c3cc(F)n(C)n3)=O)C2)cn1C Cc1c(C(=O)NCC2CC2NC(C2(Cl)CC23CCC3)=O)cncc1Br CC1C(NC(c2c[nH]c(=O)cn2)=O)CCN1C(=O)CC1CSCCS1 c1(N2C(CNC(C34CCC(CC3)C4)=O)CC3(CCC3)C2)ccc([N+](=O)[O-])cc1 C1(C(N2CCC(O)(CC)C2)=O)CCC(C)CN1C(=O)CCC1(C)CC1 CC1(C)C=C(C(=O)NC(C2CCCCC2)CNC(c2cc(Br)c[nH]2)=O)C1 N1(C(c2csc(C)n2)C(=O)NCCOC)CCCC(CC(C)C)(CO)C1 c1(CC)ccc(O)c(NC(=O)C=CCNC(C2CCCC2C(C)C)=O)c1 C1(C(=O)NCCN(C(=O)CCC2CCCCN2C)C(C)C)CC2CCC(C1)C2 Cc1cnccc1C=CC(N1CC(O)(CCNC(=O)C(n2cc(C)cn2)C)C1)=O Fc1ccc2c(CNCc3ccc(C4CCC4)cc3)n[nH]c2c1 CC(C)C(C(=O)NCC(C1CCCCN1C(c1cnc(O)n1C)=O)(C)C)N(C)C c1(OC)cc(C(=O)NCC(C2CC2)N(C)C(C2CCN(C(N)=O)CC2)=O)n(C)n1 CCCCC(C(=O)NCC(F)CNC(C1(CCOC)CCCC1)=O)NC(N)=O CCC(CCCO)NC(=O)CC1CN(C(=O)CCc2nncn2C)CCO1 C1(C(=O)NC(C2CCCN2C(=O)CC2(O)CC2)(C)C)CCC(F)(F)CC1 Nc1cccc(C(=O)NCC2(NC(=O)CCCc3ncco3)CCCCC2)c1 C(=O)(C(CCF)NC(=O)C(C)CN(C)C(c1nscc1C)=O)OC CCCCC(O)C(=O)NCCOC1CN(C(c2cncnc2C)=O)C1 N1(C(C2CC3(CSC3)C2)=O)CCN(C(c2cnncc2O)=O)C(CC(F)F)C1 c1(CCC)n[nH]c(=NCC2CCCC2NC(=O)CCOCCN(C)C)s1 Cc1cccc(C(=O)N(C2CCN(C(=O)C(Cc3cccc(Cl)c3)=NO)C2)C)n1 C1(NC(C=CCC)=O)CN(CC2CC(CC(=O)OC)C2)CCC1C C1(CC)(NC(=O)C(CC2CCCC2)NC(=O)Cc2cnccc2C)CCOCC1 c1(OC)ccccc1C(=O)NCC1CN(Cc2csc(Br)c2)C1 N1(C(c2scc(C)n2)C(=O)NCC2CC2)CCCC(c2cc[nH]n2)C1 c1(C(C)(C)C)ccc(C(=O)NCC(O)CCNC(=O)CC2CCOC2)cn1 N1(C(c2c(OC)cncc2)=O)CCN(C(c2cccc(C)c2O)=O)C(C)C1C c1(C(=O)NCC2(CNC(C3(COC)CCCCC3)=O)CC2)cc2cccnn2n1 N1(C(Cn2c(C)cnc2)=O)CC2=C(C1)CN(C(c1ccsc1C(F)F)=O)C2 C(CCC(C(=O)NC1(c2nc[nH]n2)CC1)NC(C1CCC(O)CN1C)=O)OC c1(OC)ccccc1C(C)Nc1cc(NC(C2(S(C)(=O)=O)CC2)=O)on1 c1(C(=O)NCC(CC)NC(=O)C(c2cccc(C)c2)(C)C)cc2n(c1)CCC2 Cc1cc(CC(=O)NC2CCN(C(c3cnn(C)n3)=O)C2)nn1C N1(C(=O)C(O)Cc2ccccn2)CCC2(CC1)OCCCO2 N1(C(c2ccc(CF)cc2)=O)CCC(CN(C(C23CC(F)(C2)C3)=O)C2CC2)CC1 N1(C(c2c(CC)scn2)=O)CC(NC(c2ocnc2CC)=O)CC1(C)COC CCCCCC(C)(CC)C(=O)NCC(CCOC)NC(=O)CN1CC(=O)NC1=O c1(C(N2CC3COCC3C2)=O)cc2c(-c3cccc4cc[nH]c34)cccc2[nH]1 C1(C(N(C2CCCC2)CCNC(c2c(C)[nH][nH]c2=N)=O)=O)CCCCC1(C)C c1(NC(c2ccc(-c3cccc(C(=O)NC)c3)cn2)=O)c(F)c(F)cc(F)c1F c1(NC(c2c(Br)cn(CC)n2)c2nnnn2CCCF)c(F)cc(Cl)cc1Br c1(C(N2CC(CC(CNC(CCSC)=O)(C)C)C2)=O)c(Cl)cncc1Cl c1(OCCN2CCC(CC(=O)NC(CC)C3CC3)C2)ccc(C)nc1CO N1(C(C=CC(C)(C)C)=O)CCCC2(CC(NC(=O)Cc3ccc4nsnc4c3)C2)C1 c1(NCCCN(CC)CC)ncc(S(=O)(=O)N2CCOC(C3CC3)C2)cc1Cl CCCC(C(=O)N1CCC(OCC(=O)NCC2(F)CCCCC2)C1)OCC CC1(C)CCC(CC(=O)NC2CN(C(c3ccc(C#N)o3)=O)CC2(C)C)CC1 C1(CC(=O)N(CCCCN(C(CC2CC(=C)C2)=O)C)C)CCCCO1 N1(C(CCC=C)=O)Cc2n[nH]cc2C1C(=O)NCC=Cc1ccccc1 c1(CN2C(c3ccc(C(=O)O)cc3)CCCC2)coc2cc(F)cc(F)c12 N1(C(c2c(C)ccnc2)=O)CCN(Cc2ccc(Cl)cc2Cl)CC1C C(CC(F)(F)F)SCC(=O)NCCN(C(=O)CC1CCOC1)Cc1ccccc1 Cc1cc(N2CCC(c3ccccc3)CC2C)nc(N2CCC(C)(C)C2)n1 C(=O)(C1Cc2ccccc21)NC(C1CCCC1)CNC(C(C(C)C)(C)O)=O C=CCC(F)(F)C(=O)N1CCC2(NC(c3cc(OC)n[nH]3)=O)CC2C1 N1(C(c2c(OC)c[nH]n2)=O)CCC2(CC1)CN(C(=O)CCC1NC(=O)NC1=O)C2 N1(C(C2CC(=C)C2)=O)CC(NC(C2(CC(C)C)CC2)=O)CC(F)C1 N1(C(C(=O)N(C)C)=O)CC2CN(C(c3coc(CN)n3)=O)CC12 N1(C(c2ccccc2OCCF)=O)CCN(C(=O)C(F)C2CC2)C(C2CC2)C1 c1(OC)ncc(C(=O)NCC(c2ccccc2F)NC(c2cscn2)=O)c(C)n1 c1(C(N2CC(C)CC(C)(C)C2)=O)c(F)ccc2n[nH]cc12 Cc1cc(C(=O)NCC(O)C(=O)NCC2CCOCC2(C)C)cnc1O c1(CC)cccc(C(=O)NCCCN(CCCNC(=O)CC2(C)CCOC2)C)n1 O=C(C1=CS(=O)CCC1)NC1CN(C(c2ncn(-c3ccccc3)n2)=O)CC1O C1(C)(C(=O)NC(CCCNC(CC2(C=C)CCC2)=O)C)CNC(=O)C1 C1(N=[N+]=[N-])(C(N2C(C#C)CCCC2)=O)CCN(C(c2ccc(CC)nc2)=O)C1 C12(C(=O)NC(C3(O)CCN(C(c4ncn(C(C)C)c4)=O)C3)C)CCCC(C1)OC2 C(C)(C)(CC(F)C(=O)NC(CO)C1(C)CC1)NC(C(C)n1ccnn1)=O C(=O)(C1=CCCCC1C)N1CCC(NC(c2nc(C)nc(O)c2)=O)(CO)C1 n1(CC)ccc(CNC(C2(CNC(c3cncn3C)C3CC3)CC2)=O)n1 C(=O)(CC(C)(C)C)NCC(CN(C(Cc1nc(CC)sc1)=O)C)C Cc1[nH]nc2c1CCC(C(N1CC3COCC(C1)C3NC(=O)CCC(C)C)=O)C2 CCC(CCC(=O)NC(COC)CCO)NC(=O)C(CC)N(CC)CC N1(C(C(C2CC2)OCC)=O)CC(=O)CC1C(=O)NC(CO)C(N)=O N1(C(Cc2cccc(C#C)c2)=O)CCC2(CC1)CC(Nc1nccc(C)n1)CO2 N1(C(C2CC(CC)(CC)C2)=O)CC2CCCC2(NC(=O)Cc2csc(Cl)n2)C1 C#CC1(O)CCN(C(=NCC2C(C)(C)C2(F)F)NCC(=C)C)C1 c1(N(CC(=O)NC(CN)CC(C)C)S(C)(=O)=O)ccc(Cl)c2occc12.CCO C(=O)(C1=CCCCC1)NCC(C)N(C(C1CC(O)(CC#C)C1)=O)C C1(C(=O)NC2CCN(C(CCSC)=O)C2C(C)(C)C)CC2(C1)CC1(CC1)C2 C1(C(=O)NCCC(C)NC(C(C)NC(C2CCCCC2)=O)=O)CC12CCCCC2 C#CC1(CNC(C2(F)CCN(C(C3OCCC3C(C)C)=O)C2)=O)CCCC1 c1(C(=O)NC2C(NC(C3(OCC)CCCC3)=O)COC2)cnn2c(Cl)cccc12 C(CC(C)(C)C#N)NC.n1(CCCNC=O)cc(C2CC2)nn1 C(=O)(C1=CCCCC1)NCC1C(NC(Cn2c(C)nc(C)n2)=O)CCC1 C1(NC(c2ccc(OC)cc2Cl)CO)CCCCC12CCCC2 C(=O)(CC(C)C(C)C(C)C)N1CC2CC(Nc3cc(SC)nc(SC)n3)C2C1 c1(CC)cc(C(=O)OCc2nc(NC(C)C(=O)OC)cc(O)n2)cc(C)c1 c1(NC2CCN(C(C3(C4CCCO4)CC3)=O)C2)ccc([N+](=O)[O-])c2cccnc12 c1(C(N2CCCC(NC(CCC(CC)C)=O)C2)=O)c(OC)cc(OC)cc1N N#Cc1ccc2[nH]cc(CN3CC(Nc4ccncn4)CC(F)C3)c2c1 c1(OC)ccc2c(N3CCC(O)(CC(=O)OCC(=O)N(C)C)CC3)ncnc2c1 O=C(CCCC1CC1)NC1CCN(C(=O)C(c2ccoc2)=O)C1 c1(C(N2CC(N(C)C(C3CCCCN3C)=O)C2)=O)cc2c(s1)CCSC2 N1(C(Cn2ncc(C)c2)=O)CC2CCC(C(N3CC4C(C(N)=O)C4C3)=O)(C2)C1 C1(CNC(c2c(OCC)nccc2)=O)CCCCCN1C(=O)Cc1csnc1C Cc1cc(C)c(C(N2CC3(C2)CN(C(c2cc(C(F)(F)F)no2)=O)C3)=O)cc1N c1(-c2c(F)ccc(OC)c2F)ncn2c1CN(C(=O)C1=COCCC1)CC2 C1(C(=O)NCC2CC(C)(C)OCC2)CCN(C(=O)CCCC2CCC2)C(C)(C)C1 C1(CC(=O)NC(C)CC(=O)NCc2ccn(CCF)n2)COCC(C)O1 c1(NC(=O)NCC2C(=C)C2)cnc2ccc(F)cc2c1 c1(C(N2CCC(NC(C(C)CO)=O)CC2)=O)ccc(Br)c2cn[nH]c12 c1(CN2CCC(NC(C(CCSC)NC(C)=O)=O)C(F)C2)cc(F)c(Cl)cc1C CCC1=NOC(CC(N2CCC(CCNC(c3nc[nH]c3C(C)(C)C)=O)C2)=O)C1 C(c1nc(C)c(C)[nH]1)=CC(=O)NCCN(C(=O)Cc1ccnc(Cl)c1F)CC C1(NC(=O)Cc2ccsn2)CCCN(C(=O)CCc2cccc(Cl)c2)CC1F C(=O)(C(C)C(O)CC)NCCC(C)N(C(c1cnn(CC)c1Br)=O)C Cc1sc2ncc(C(=O)N(CCC(C)NC(C3(C)CCCO3)=O)C)n2c1C N1(C(C(N2CCOC2=O)C)C2CC2)C2CCC1CN(C(=O)CC(C)P(C)(C)=O)C2 c1(C(=O)NC2CC(C)N(C(=O)Cc3ccon3)C2)cccc2c1CCC2 Cc1cc(=NC(=O)C(=O)NCC2CN(C(C3CCCC3C)=O)C3(CCC3)C2)[nH]o1 Cc1c(C(N2CC(n3cc(-c4ccc(F)cn4)nn3)C2)=O)[nH]ccc1=O c1(CC(C)C)ccc(C=CC(N2CCN(C)CC2CNC(c2cnc[nH]2)=O)=O)cc1 C12CCCN(C1)C(=O)CSCC2.C1C(=O)N1C1CC1.C=CCSC(C)C CC(C)CC(O)C(=O)N1CC(C(N2CCC(OCCF)C2)=O)CC(C)C1 c1(OC)ccnc(C(=O)NCC(C2(O)CN(C(C3(C4CC4)CC3)=O)C2)(C)C)c1C C(=O)(CCC(=C)C)NCCOCC#C.C12CCOCC1C(=O)NCC(=O)N2 O(NC(=O)C(C)(C1CCC1)NC(=O)C=C1CCOCC1)CCN(C)C C1(C(=O)NCCN(CCC)C(c2cc3scnc3[nH]2)=O)CCCC1S(C)(=O)=O C1(NC(C(COC)OC)=O)CCCCN(C(=O)CC2CCCS(=O)(=O)C2)C1 c1(C(=O)NCC(C)(CO)NC(c2cc(C)ns2)=O)cc(S(C)(=O)=O)c(C)o1 C(=O)(C1=CC2CCC1C2)NC1CN(C(c2c(C)[nH]c(C#N)c2)=O)CC12CC2 c1(C(=O)NC(C2CCC2)C)ccnc(CN(C(C2CC2F)=O)C2CC2)c1 N1(C(c2c(C)n(C(C)C)nn2)=O)CCCN(C(=O)COCC(C)(C)C)CC1 N(C1CCc2cc(F)ccc21)c1nnc(CC(C)C)n1Cc1cccs1 c1(C(N(CC(C)N(C(C(CC#C)C2CC2)=O)C)C)=O)nccc(Cl)c1C C1(CNC(c2c(Br)ccc(C)c2)=O)CC2(CCN(C(C3CCO3)=O)CC2)C1 C1(N(C(C2CC(C(=O)Nc3cccc(F)c3)C2)=O)CCF)CCCN(C(C)=O)C1 c1(C(=O)NC(C)CN(C)C(c2csnn2)=O)ccc(C(F)(F)F)cc1C(F)F C1(NC(C(CC)=CCCC)=O)CCN(C(=O)C(C)c2ccco2)C1C C(CC(=O)NCC(C)C(C)C)(CC(C)C)NC(c1ccc(C)c(C)c1)=O N1(C(C2CCC(C)S2)=O)CCCC2(C1)CN(C(c1cncc(F)c1)=O)C2 N1(C(c2c(CC)cncc2)=O)CC(C)C(NC(=O)C=Cc2cnc(C)s2)C(C)C1 CC(CCCNC(c1cn(Cc2ncccn2)nn1)=O)NC(c1csc(Cl)c1)=O C12(C(=O)OC)CCCC1(C(=O)NC1CC(CNC(c3coc(COC)n3)=O)C1)C2 C1(C)(CC(=O)NC(CN(CC)CC)C)CCN(C(=O)C=CC2CC2)C1 c1(CC(=O)NC2CCC(F)(CNC(Cc3cn(C)nc3)=O)C2)ccc(F)c(F)c1 CCC(C)CCCC(=O)N1CCCC1C(N1CC(OC(=N)O)C1)=O c1(C(N2C(CN(C(CCC)=O)C)CCCC2)=O)cc(C(=O)OC)ccc1C C1(C(N2CCC(NC(=O)Cn3cnnn3)(CO)CC2)=O)CS(=O)(=O)CC12CC2 C1(C)(C(NOCC2(COC)CC=CC2)=O)CCCCC1 c1(CNC(C2OCC(C)(C)C2)=O)ccc(Br)cc1O.C12(C)CC(C1)NC2=O c1(CNC(CCC2CC(OC)CN2C(=O)OC(C)(C)C)=O)c(Cl)cccc1Br Cc1cc(Cl)c(C(N2CCC(C)(CNC(=O)Cn3ccsc3=N)C2)=O)s1 c1(C(N(C2CN(C(C(CC(C)C)O)=O)CC23CC3)C)=O)cnc(O)c2ccsc12 c1(-c2scc(-c3cc(-c4n(CCCCC=C)ccn4)n[nH]3)c2)ccc(OC)cc1 O=C(COc1ccc(-c2nn[nH]n2)cc1)NNC(=O)NC1C=CCCC1 c1(CC)ccc(C(=O)N(CC(C)CNC(=O)C(O)Cc2cccs2)C)cc1CC c1(CC)ccc(SC)cc1CN1CCCC(CO)C1CO N12CCC(C#N)(C1)NC(=O)C13N(CCC1C3)C2=O.CC(C)(C)O.C(=O)(C1CC1)N c1(C(=O)NCC2CCN(c3snc(CCC)n3)C2)ccnc2[nH]nnc12 C1(Cn2cc(CSC)nn2)CCN(C(c2cc(Cc3ccccc3)[nH]n2)=O)CC1 Cc1cc(C(N2CCCC(C(=O)NCCN(CCO)CCO)C2)=O)cc(C)c1Br CN(NC(=O)C(C)(C)CCCn1cc(CC2CC2)nn1)CC(F)(F)F.C1C(=O)N1 c1(NC(C2CC(F)CN2Cc2c(F)cccc2Br)=O)ncnc2cc[nH]c12 C(=O)(CC1=CCN(C)CC1)NCC1(O)CCCN(C(c2c(NC)snc2C)=O)C1 c1(NC(N2CCC(CN(c3cn(CC)cn3)C)C2)=O)ccc(OC)c(F)c1 c1(C(=O)NC(C)C(C)NC(c2onc3ccccc23)=O)cc2nc[nH]c2cc1N C1(CNC(CC=C(C)C)=O)CN(C(=O)CCOCC2CCCC2)CCC12CCC2 N1(C(C(C)n2cccc2)=O)CC(NC(=O)CCc2cnc[nH]2)CC2(CC2)C1 C1(NC(C=CC(CC)C)=O)C(CC(=O)N(CC(C)OC)C)C1(C)C O(NC(=O)CC1C(NC(=O)CNc2ncccn2)CC1O)CC Cc1ccc(NC(N2CCN(C(=O)C(Cl)(Cl)Cl)C3CC23)=O)c(Br)c1 CC1(C(N2CC3CC3(CNC(c3ccnnc3O)=O)C2)=O)CCNC1=O c1(CC(C)C)noc(CN(CC(O)CN(C)C(c2coc(Br)c2)=O)C)n1 c1(NC(c2n(CCC)nnn2)(C)CCI)cccc(F)c1C N1(C(C(Br)=C(C)C)=O)CC=C(CCNC(=O)C(C)C(C)O)CC1 c1(CC(CN2CCC(COCC)(CO)CC2)=O)ncc(C)c(OC)c1C N1(C(COC(CC)C)=O)CC2CC(NC(C3CN4CCN3CC4)=O)C2C1 c1(OC)c(NC(=O)CNC(Cc2ccco2)CO)cc(C)cc1C c1(C(N2CCN(CC(=O)NCC(CC)OC)CC2)=O)cccc([N+](=O)[O-])c1OC C(C)(C(C(=O)N(C1CCCC1O)C)NC(=O)CCCN(C)C(C)C)OC N1(CC(=O)Nc2cc(C)no2)CCC(NC(C2CCC(F)C2)=O)CC1 CCCCC(CC(=O)N1CC(n2cnnc2)C1)NC(C1C2CCC(F)C12)=O CCCCCC(=O)NCC(=O)NCCC1CCCCN1C(=O)C=C1CCOCC1 C12(COC)CC(C(=O)NC3CN(C(=O)CCc4ccc(C)o4)C3)(CO1)C2 C1(C(=O)NCCCOCC=C)CC(C)CN(C(C23CC(CO)(C2)C3)=O)C1 C(C(CC1CC1)C(=O)Nc1ccc(OCF)cc1)NC(CCn1cnc(=N)[nH]1)=O N1(C(CSCCCC)=O)CCN(C(c2cccc(C(=O)OC)c2)=O)C(C)CC1C C#CCC(C)(C(=O)NC(CC)CCO)NC(=O)C(O)C=CC C1(CC(=O)NCC(CC)NC(c2ccncc2)=O)COC(C)(C)C1 CCC(CC(=O)NC(C(=O)NCCCC(C)(C)C)C1CC1)C(C)(C)C N1(C(C2(N(C)C)CC2)=O)CC(C2CCCN(C(C3CCC4(C3)CC4(F)F)=O)C2)C1 C(C(CC(C)C)C(=O)NCC(CO)NC(=O)C(C)(C)C(N)=O)OC Cc1cc(C(=O)NCC2COCCN2C(c2cc(C(C)C)sn2)=O)sc1Cl N1(C(C2CCC(N(C)C)CC2)=O)CC2CC1CC2C(N1CC(O)C1)=O CCCCC(CCCC)NC(C1(C)CC(O)CN1C(=O)Cn1nccn1)=O N1(C(C(C(C)C)C)=O)CC2(CC(NC(c3cccc(O)c3Cl)=O)CO2)C1 C1(n2cc(C(=O)Nc3ccc(OC4CCCCC4)cc3)nn2)CCCS(=O)(=O)C1 N1(C(C2C(OC)CCC2)=O)CCN(CCCCCNC(=O)CCCC#N)CC1 C1(CN(CCC(=O)O)Cc2ccc(OCC)c(Br)c2)CCc2ccccc2O1 Cc1ccc(NC2CC(=O)N(c3ccc(OC(C)C)cc3)C2)cc1I C1(NC(c2cc(CO)on2)=O)CC2(C(=O)NCC34CCCC3OCC4)COC1C2 C(=O)(CC(C)(C)C(=O)OC)NC1(CN(C(C(C)=C(CC)C)=O)C)CC1 N(S(=O)(=O)N1CC(O)C1)CC(=O)NC(Cc1cc(OC)c(O)cc1)C C1(CNC(C2(C(=O)NC)CC2)=O)CCN1C(=O)CCc1cnc[nH]1 N1(C(C2(C)N(C(c3cncc(C)n3)=O)CC=C2)=O)CCC(O)C(C)(C)C1 Cc1cc(Cl)c(C(=O)NC(Cc2cn(-c3ccc(Cl)cn3)nn2)CC(=O)O)s1 n1(CCC)cccc1C(=O)NCC1(CC(=O)NCC(c2cn(C)cn2)O)CC1 c1(C(C(=O)OCCOC)N(C(C(=O)OC)C(C)OC)C)ccc(F)cc1Br C1(C)(C(=O)NCC(C2CCN(C(C(CC)OC)=O)CC2)(C)C)CCC(=O)NC1 C1(C(N2CCN(CCOCC)CC2)=O)CC(=O)N(C)C1c1cnn(C)c1 c1(CN(C(C)C)Cc2ccc(C(C)(C)C)cc2)ccccc1[N+](=O)[O-] n1(CC(=O)N(CC(N2CCC(CC=CC)C2)=O)CC#C)ncccc1=O Cc1nn(C)c(C)c1C(C)C(=O)NC1CCCC1NC(c1n[nH]cc1F)=O C1(NC(=O)C=Cc2cscn2)CCN(C(=O)Cc2cn[nH]c2)CC1CO N1(C(c2c(C)c[nH]n2)=O)CC(C)CN(C(C2CCN(CC3CC3)CC2)=O)CC1C C(=O)(C#CC(C)(C)CNC(C1CC2(CCC2)C1)=O)N(CC(O)C1CC1)C C(CC(C)(C)C(=O)N=c1ccn(CCF)[nH]1)NC(C1CCCC(C)CC1)=O C1(C(=O)NC(CCCC)C(=O)NC)CC(F)CN(CC2CC3C=CC2C3)C1O C(C(C(F)(F)F)NC(=O)C(n1cc(-c2ccc(C(F)(F)F)cn2)nn1)C)OCC c1(CN2C(CCC(N3CCCC(C(=O)OC)C3)=O)CCC2)cc(Br)ccc1Cl N1(C(c2ccc(OC)o2)=O)CC2CCC(N(C(=O)Cc3cccc(F)c3)C)C2C1 c1nc(C(C)C)cc(C)n1.C(C)(C)(C(=O)NC)SC.C12CC(C1)NCC2 N1(C(C(C)(F)F)=O)CC2CCC1C1CN(C(=O)CN=c3ccc(C#N)c[nH]3)CC21 N1(C(CC)=O)CCOC2(CCC(N(C3CC3)C(=O)C3CC3)CC2)C1 C=CCC(CNC(C1(OCC)CCCOC1)=O)C(=O)NC1COC(C(C)C)C1 C(=O)(CC1COCc2ccccc21)NCC(C)NC(c1cc(Cl)c(F)cc1O)=O Nc1nonc1C(=O)NC1CCC(CCNC(=O)CNC(c2ccco2)=O)C1 C(C(CC1CC1)C(=O)NCCCOC1CC1)NC(CC1(C)CCOC1)=O C(=O)(C1CCc2ccccc21)N1CCCC(O)(CNC(C(C)(C)O)=O)C1 c1(C(N(C2CC3(N)CC2C3)C)=O)cccc(N=[N+]=[N-])c1 Cc1ccc(C(F)(F)F)cc1CNC(C1(C)CCN1Cc1cc(Cl)cc(I)c1)=O c1(C(N2CCC(C)C2)C(=O)NCCOCC)cc(C(C)(F)F)ccn1 N1(C(C(CCSC)OC)=O)CCCC(O)(CNC(=O)CCSCC(N)=O)C1 N1(C(C2N(C(c3ccc(N)c(F)n3)=O)CC(O)CC2)=O)CCN2C(=O)OCC2C1 Cc1nc2cc(Cl)ccc2cc1C(=O)NCCC(C)NC(C1(C)CC2CC2C1)=O C(CC(C)C(=O)NCC1CCCN1C(=O)CN1C(=O)CCC1=O)=CCC Cc1cccc2c1OC(C(N1CCC3CN(C(c4nc(Cl)cs4)=O)CC3C1)=O)C2 N1(C(C(C)OCC2CCCO2)=O)CC(O)CC1CNC(c1ncc(F)cn1)=O c1(C(=O)NC(C(C(C)C)C)CNC(c2cnc[nH]2)=O)cc(S(C)(=O)=O)ccc1O Fc1ccc(-c2nc(C(=O)CC(F)(F)c3ccccc3)cs2)c(F)c1 C=CCCCCC(=O)NC1(CO)CCCN(C(c2onc(C)c2C)=O)C1 CCCC(C)CC(=O)N1CC(C2(NC(c3ccc(=NC)[nH]c3)=O)CC2)C1 c1(OC)ccc(C=CC(=O)NC2CCN(C(C3(F)CCS(=O)(=O)C3)=O)C2)cc1O N1(C(CC(CC)O)=O)CCCC(C)(NC(c2cc(OC)ccn2)=O)C1 O=C1CC(CC(=O)N2CCOC(CC3(CNC(C4CCCC4)=O)CC3)C2)=NN1 C12(C(N3CC4N(C(c5nnn(C)c5N)=O)C(CC4)C3)=O)CCCN1S(=O)(=O)CC2 C1(NC(C2CC2(Cl)Cl)=O)COCCN(C(C2CC3(CCC3)CO2)=O)C1 C(=O)(CC1=CCCCC1)N1C2CC(CNC(c3c(COC)cc[nH]3)=O)C1CC2 N1(CC(=O)NC)CCN(CCCN(C(c2cc(C)cs2)=O)C(C)C)CC1 C#CCC(O)C(=O)N(C(C)CCNC(c1ccc(-n2[nH]c(O)nc2=O)cc1)=O)C C1(CNC(C2CCN(CC)C2)=O)CN(C(c2ccnc(S)c2)=O)CC12CC2 C1(C2(N)CCC2)(C(=O)NCC(CC#N)(F)F)CC1 CC1CCCN(C(=O)C(C2CCN(C(c3ccc(-c4ccco4)o3)=O)C2)C)C1 CCCC(C(=O)NCC(C)N(C)C(C12CCC(C#N)(CC1)CC2)=O)S(N)(=O)=O N1(C(C(=O)N(CCCOC)CCCOC)=O)CC(OC)C(F)C1 C1(C(N2CC(NC(c3cccc(C)c3C)=O)C(C)CC2)=O)CCCC2CCCN12 C#CC(CC)(CC)NC(C1CC1CNC(=O)CC1CCC(C)CO1)=O C1(O)(CC=C)CCN(C(=O)CCNC(c2ccncc2NC)=O)CC1 CC1(C)CN(C(C2CCC(=O)N2)=O)CCC1C(=O)NC1CCCCC1 CCC(CC)(CC(=O)OC)C(=O)NCCCCCCNC(=O)CN1CCNC1=O c1(C(=O)NC2(CC=C)CCN(C(=O)COCC)C2)cnn2c(Cl)cccc12 c1(N(CCCN(C)C(C2OCC2(C)C)=O)C)ncnc2cnccc12 N1(C(C(C)N(C(=O)CCN2CCCC2=O)C)=O)CCC(O)CC1C N1(C(C(CNC(c2nc(C)oc2C)=O)O)=O)CCC(C2(C)CC2)CC1 c1(C(c2n(CC=C)nnn2)NCC2C(C)(C)C2(C)C)c(Br)c(C(F)(F)F)nn1C Fc1cc(-c2csc(-c3ccc(F)cc3)n2)c2c(c1)CCC2 n1(CCC(=O)NC2C(NC(C(C)SCCCC)=O)CC2)nc(C)cc1C N1(CC)OCC(NC(=O)CNC(=O)CNC(=O)CC2CCSCC2)C1=O c1(C(=O)NCC(C)N(C(C2CC(O)(CC#C)C2)=O)C)ccc(O)c(C)c1C CN=c1[nH]c(=NCC2CNC(=O)C2(F)F)[nH]c(=NC(C)c2ccc(Cl)nc2)[nH]1 C1(CNC(C(C)O)=O)CCCN(C(=O)C(O)CCn2cncn2)CC1 c1(C(C)C)cc(C(N2CC(NC(C3CCC3F)=O)C2)=O)nn1-c1ccccn1 CCC(CC)CCC(=O)NCC1CN(C(c2ccc(O)c(CO)c2)=O)CC1C c1(C(=O)NCC(CNC(c2cc(C)c(N)cn2)=O)CO)cn2cc(Cl)cnc2n1 C1(NC(C(CC)N(CC)CC)=O)CC(N=c2nc(SC)[nH]s2)C12CCC2 N1(C(C2(CN(C)C)CC2)=O)C2CCC1CN(C(=O)CC1CCCC1O)C2 C1(C(N2CC(C(C(=O)N3CCC3)NCC3CSCCO3)C2)=O)(CO)CCCCO1 C(=O)(CCCC(=O)N(C)C)N1C(CNC(c2c(C)n(C)nc2)=O)C=CC1 Cc1cc(C(=O)N(C)CC2CC(F)CN2C(=O)CC2CCC(=O)N2C)cnc1O C1(C(=O)NC(COC)(C)CO)CCC2(CC2)N1C(=O)CCc1csnn1 CN1CCCC(CC(N2CC(O)CC2C(=O)NCC2CC[Si](C)(C)C2)=O)C1 N1(C(C2(C#C)CC2)=O)CC2CCC1CN(C(c1c(F)cc(OC)c(F)c1F)=O)C2 C(CCc1ccccc1)(C(C)N=c1ncnc(C)[nH]1)NC(c1n(CC)nnc1)=O C1(CNC(C(C2CCC2)OCC)=O)(NC(=O)CN(C)C(=O)C2CC2)CCOC1 C1(N(C)C(C2COCCO2)=O)CCCCN(C(c2ccnc(S)c2)=O)C1 c1(NC2C(C)CN2C(=O)OC(C)(C)C)cc(Br)cc2c1OCCC2=O Cc1cc(Nc2nc(C(=O)Nc3csc(C(F)(F)F)n3)cs2)ncn1 c1(OC)nc(C(C)C)ccc1CN(CCC(C)O)CCO C1(NC(C=CCCC)=O)(CSC)CCN(C(c2ccc(SC)nc2)=O)C1 C1(NC(C(C)(C)OCC)=O)CCCCC1NC(=O)CSc1ccccc1C C(=O)(C(C)C(C)NC(=O)C=C(C)C(C)C)NCCOCC#N Cc1cccc(C(F)C(N2CCC(NC(c3sccc3Br)=O)C2)=O)c1 C1(C)(CNC(CCC#CC)=O)COCCN(C(c2sc(OC)nc2Cl)=O)C1 c1(CNC(CN(C)CC)=O)ccc(C(=O)Nc2cnccc2C)cc1 C(CCC(=O)NC(C)CN(C(=O)C(C1CCCCC1)C)C)SC C1(NC(C(C)CC2CC2)=O)COCCC1NC(=O)CCc1cc[nH]n1 c1(C(N2CC(NC(c3c(C)c(O)ccc3)=O)C3(C2)CC3)=O)nccc2occc12 C12(NC(C(C)C#N)=O)CCCC1CN(C(c1ccc(OCC(F)F)cc1)=O)C2 c1(C(N2CCC(O)(CNC(C(CCC#C)O)=O)C2)=O)ncnc2ccsc12 CCC(CC)CC(=O)N1CCC(C(N2CC(N3CCC3)C2)=O)C1CC c1(C(=O)NCCOC2CN(C(=O)C(F)(F)C(F)(F)F)C2)cncc2ccccc12 C1(NC(=O)COCCCF)CCN(C(=O)Cc2ccco2)C1c1ccccc1 Cc1cc(C(N2C3CCC2CN(C(=O)C(O)CC(C)C)C3)=O)cc(=O)n1C CC1CC(NC(C2CCCN2C)=O)CN(C(c2cn(C3COC3)nn2)=O)C1 C1(NC(c2cc(OCC)no2)=O)CCCOC12CCN(C(=O)CCF)CC2 C(=O)(C(F)C(=O)NCC(C1CCCCC1)NC(c1cncc(F)n1)=O)OCC c1(C(C)=O)c(NCCC2CC(NC(=O)CS(N)(=O)=O)C2)nc(C)nc1Cl CC1CN(C(c2c(F)cc(C#N)cc2F)=O)CC(C)N1Cc1ccccc1 c1(C(N(C2CCN(C(=O)Cc3cscn3)C2)CCC)=O)ccnc(C)n1 c1(-c2nc(CN(CCC)C(=O)NC(C)Cc3nc[nH]n3)on2)ccc(C)cc1 C1(NC(c2ccc(C)n2C)=O)CN(C(=O)C(F)(F)c2ccnn2C)CC12CC2 C1(C(=O)NC(c2cccnc2)C(=O)NC(CCC)CO)CC2(CCC2O)C1 Cc1cnc(C(=O)NC(C2(O)CN(C(=O)CCCC3CCCCC3)C2)C)cn1 CCN=c1[nH]c(C)c(C(N2CC(CNC(=O)C(F)(F)CC3CC3)C2)=O)s1 C1(CNC(C(CC)OC2CCCC2)=O)COCCN1C(=O)CN1CCOCC1=O C1(CNC(C2CN(C(=O)NC)C2)=O)CCCN(C(c2cccc(O)n2)=O)CC1 CCC(C)C(C)C(=O)NCCC1CCN(C(=O)Cc2cncn2C)CC1 c1(C(N2C(C)CCC(NC(CN(CC)CC)=O)C2)=O)cc(=NS(C)(=O)=O)cc[nH]1 c1(C(=O)NC2(C3CN(C(C(COC)(C)C)=O)C3)CC2)ccn2cnnc2c1 C=CCCC(CC(C)C)C(=O)N1CCCC(C)(NC(=O)Cc2cnco2)C1 c1(C(=O)NC2CC(C)(NC(C(C=C)O)=O)C2)cc2ccc(F)cc2nc1C Cc1cc(Br)ccc1-c1noc(C(OC(C)(C)C)SCC2CCC2C(N)=O)n1 C1(NC(Cc2c(C)n(C)cn2)=O)CCC2(CC1)CN(C(C1C=CCC1)=O)CCO2 CC1(NC(C2CCO2)=O)CC(C(=O)NC2CC(C(C)(C)C)C2)C1 c1(C(=O)NC2CC3(C(NC(=O)COC4CC=CC4)C3)C2)cccc2[nH]cc(Cl)c12 C1(CC)CCCN(CC(=O)NC(C)CCCNC(c2cncnc2)=O)C1 C1(C(=O)NC(c2ccccc2)C(=O)NCc2ccco2)CC(Cl)(Cl)C1 CC1(C)COC(CCC(=O)NCC2(NC(=O)CCCc3ccc(F)cc3)CC2)C1 N1(C(C2(C)CCCN2)=O)CCC2C1CCN2C(c1ccc(NS(C)(=O)=O)cc1)=O C=Cc1ccc(CNC(C2N(C(=O)CC34CCCC3C4)CCC2(C)C)=O)cc1 c12ccc(nc1)NCCC2.CC(C(=O)NC)NC(N)=O.c1(C=O)nc[nH]n1 C1(CC(=O)NCCC(C)N(C(=O)CCC2CCCO2)C)C=CCCC1 c1(C(N2CCC(S(=O)(=O)NC)C2)C(=O)NCCOC)cc(O)nc2ccccc12 c1(C(=O)NC(C)CNC(=O)CN(C)C(=O)OC(C)(C)C)ccnc2[nH]c(O)nc12 C1(CC(N2CCC(C(=O)OC)C2)=O)OCC2CCN(C(=O)COC(=O)NCC)CC12 C1(C(C)(C)C)C(=O)NCCN1C(=O)C(C)(C)C1CCN(C(=O)CC2C=CCCC2)C1 Cc1cc(OC(c2ccc(OCc3cccnc3)cc2)=O)ccc1Cl c1(NCc2scc(CN(C)C)n2)ncc(S(=O)(=O)N2CCCC3CC23)cc1Cl N1(C(c2ccc(C)cc2C)=O)CC2(CCCC2)C1C(=O)NCC(O)C(F)F C(CCC(N)=O)(C(=O)O)NC(c1ccc(C2CC2)cc1)=O C1(CC(=O)NCc2cc(COC)no2)CCCCN1C(=O)CSc1cn[nH]c1 C12(CNC(c3cc(C)c(C)nn3)=O)CC(CCO1)N(C(=O)CC1(CO)CC1)C2 C1(C(=O)NC2CC3(C(C(=O)NC4CN(CC)C4)C3)C2)C2CCCCCC12 c1(N(CCCN2C(=O)OCC2)C2CC2)ccc2c(c1)CCC2 O=C(C#CC1CCOC1)NCC1(O)CC(NC(C2Cc3nccn3C2)=O)C1 CON1CCC(C(=O)NC(C)CCNC(C23CCCCC2C3)=O)CC1 C(=O)(C(S(C)(=O)=O)C1CC1)NCC(C)(C1CC1)NC(C(CC)(C)C)=O c1(N2CC(n3cc(-c4c(C)cn(C)n4)nn3)C2)ccc(Br)c(Cl)c1F c1(C(NNC(=O)N(c2ccc3nnsc3c2)CC2CC2)=O)cccc2[nH]ccc12 N#Cc1ccc(COC(c2cccn2CCc2ccccc2)=O)c(F)c1 c1(C(=O)OC(c2nnc(C3CCC3)o2)C)ccc(Cl)c2cccnc12 N1(C(C2CC(=O)N2)=O)CC2CCN(C(c3cc(Br)cnc3Br)=O)C2C1 CN1CC(OC(F)F)N(S(=O)(=O)Oc2cccc(Br)c2F)CC1=O N1(C(C2(CC)COC2)=O)CCCN(CCCCNC(=O)CCC2CCOC2)CC1 c1(C(N2CC(O)(CNC(C3(OCC)CCSCC3)=O)C2)=O)cc(N)cc(O)c1C c1(C(=O)OC)cc([N+](=O)[O-])ccc1NCC(F)C(F)(F)F N(C(=NCc1ccc(OC)c(OC)c1)N(C)Cc1ccc(Br)c(F)c1)C(CC)C C1(n2cc(C(CCC)=O)nn2)CN(C(c2ncoc2C(F)(F)F)=O)CC1C C=CC1CN(C(=O)CC2CN(C(=O)C(C)(C)OCC)CC2C)CC1O c1(C(=O)NCC(C)CNC(=O)C(N2CCCCC2)C2CC2)cccc(C(F)F)c1 C1(NC(COCCCC#C)=O)CC2CCC1CN2C(=O)C(c1ccc(C)o1)C N1(C(C(CC)F)=O)CC2CN(C(c3ccnc(N4CCCCC4)n3)=O)CC2C1 c1(C(=O)NC2(CCNC(C3CCN4CCCC4C3)=O)CC2)cccc2cc[nH]c12 N1(C(c2c(NC)cccc2)=O)CC=C(C(=O)N2Cc3ccncc3C2)CC1 C1(O)(CCNC(C2(C=C)CC2)=O)CCN(C(=O)CC2CC(=O)NC2=O)C1 N1(C(c2c(CC)cccc2)=O)CCOCC(CNC(=O)C(C)(C)CCF)C1 c1(C(N)=O)ccnc(C(=O)NCCC2CCCN2C(=O)Cc2cnc[nH]2)c1 C=CCC(CC(F)F)C(=O)NC1(CO)CN(C(=O)C(O)CCCC)C1 c1(OCCNC(C2C(OC)C2)=O)cccc(OCc2ccc(C)cc2)c1 C(=O)(CC(C)(C)C(F)F)N1CCC(NC(Cc2c(C)nc(C)s2)=O)C1C C(=O)(C(CN=[N+]=[N-])OC)N1CC(COC)(NC(c2cc(OC)n[nH]2)=O)C1 c1(C(N2CCCSCC2)=O)ccc(-c2cc[nH]c2)c2c1OCO2 C1(NC(c2cc(C)sc2C)=O)CC(F)CN(C(C2CC2c2ccncc2F)=O)C1 c1(CC(=O)NC(CNC(c2ccc(SCC)nc2)=O)(C)CO)cccc(C)c1F c1(OC)cc(CNC(C2CC(F)CN(C(=O)CN(C3CCC3)C)C2)=O)ccc1C c1(C(N2CC(NC(CN(C)CC)=O)C2)=O)ccc(C)nc1OC c1(C(=O)NCCCC(O)C(=O)N2CC3(C=CCO3)C2)cnn2ccc(Cl)c(F)c12 CCCCCCCC(O)CC(=O)N1CCN(Cc2cnc(Cl)c(Cl)c2)CC12CC2 Cc1cc(C(=O)NC(C)CCN(C)C(c2ccc(F)cc2)=O)c(Br)c(C)c1 Cc1nn(CC(N2CCOC(c3ncc[nH]3)C2)=O)cc1Br C12(C(=O)NC34C(CN(C(C5(CCOC)CC5)=O)C3)C4)CCC(F)(CC1)CC2 C1(NC(CCSCC)=O)CCN(C(=O)CCCc2cccnc2)CC1F C1(C(=O)NCC(C23CCC(CC2)C3)NC(C(CC)OC)=O)CC(=O)CCO1 C1(C)(C(N2CC(NC(c3c(OC)scc3)=O)C(C)C2)=O)CCC(C(C)(C)C)CC1 c1(NC(C(n2cc(C(N(C)C)C3CC3)nn2)(C)C)=O)ccc2c(c1)OCO2 CC(C)C(N=[N+]=[N-])C(=O)N1CCC1C(=O)NCC1(C)CCC(=O)N1 N1(C(C=CC=CC)=O)CC(NC(C2C(C)C2C)=O)C(c2cncn2C)C1 C1(NC(CNC2(C)CN(C(c3cc(OC)ns3)=O)C2)=O)CN(CP(C)(C)=O)C1 N1(C(C2(CC=C)CN(C(=O)CC(C)C=C)C2)=O)CC2C(CO)C2C1 c1(CN(C)C(C2CC(C(F)(F)F)C2)=O)ccnc(C(F)(F)F)n1.C12CCN1C2 C1(C#N)(C(=O)NCCC2(O)CN(C(Cc3nc(C)oc3)=O)C2)CCCC1 N(C1=COCCC1)C(C1C2CN(C(=O)CN3C(=O)C=CC3=O)CC12)=O C1(C(N(C(CC)CC)CC(C)C)=O)CCCN(C(c2csc(C)c2C)=O)CC1 N1(C(C=CCC)=O)CCC2(CCCC2NC(c2cc(C(C)C)on2)=O)C1 c1(OCC(=O)NC2(CC)CCN(C(=O)C(C)c3cc[nH]n3)C2)ccc(F)c(F)c1 C1(NC(c2nc(C)oc2C)=O)CC2CCC1(NC(=O)CC1(C)OCCO1)C2 N1(C(c2cc(CC)oc2C)=O)CCC(NC(=O)CCCc2sccc2C)C(C)C1 C12(CNC(c3ccccc3F)=O)CC1CN(C(=O)C(c1ccccc1F)O)C2 CC1=CCC(C)(NC(C2CN(C(C3C4CC5C(C4=O)C35)=O)C2)=O)CC1 C1(C(=O)NCCN(C(=O)C(C)(C)Cc2ccc(Cl)cc2)C)CCC(C(N)=O)CC1 N1(C(c2c(C)onc2CO)=O)CC2(CCCCN2C(=O)CSS(C)(=O)=O)C1 O=CN1CCN(C(C2(F)CN(C(=O)Cc3c(Cl)cccc3Cl)C2)=O)CC1 CCC(O)CCNC(C1(CNC(=O)C(C2CCOCC2)C)CCC1)=O N1(C(C2(OC)CCOCC2)=O)CC(NC(=O)CC2(CS(C)(=O)=O)CC2)CCC(O)C1 C1(C(=O)NCC(CNC(c2ncn(CC)n2)=O)F)CCC2C(C1)C2(F)F c1(NC(=O)NC2(CC(=O)Nc3ccc(Cl)nc3Cl)CCCC2)ccc(Br)c(F)c1 N1(c2scc(C)n2)CCCC(C(=O)NCCSC23COCC(C2)C3)CC1 C(=O)(C1=NNC(=O)C1)NCC#CC(=O)NC1(CC(=O)OC)CCC1 C1(C(=O)NCC(CC)(C)C)CCN(C(c2cncn(C)c2=O)=O)CC1O c1(NC(CC2C(CNC(CC=C=C)=O)C2(F)F)=O)ccc(C)cc1CC c1(C(N2C(C)CN(C(=O)CC3CCC(C)C3)CC2)=O)ccc2ocnc2c1 C1(NC(=NC)NCc2c(OC)ccc(F)c2O)CCN(CC(F)(F)F)C2(CC2)C1 c1(C(N(CC(C)C)C)=O)cnc(CNC(c2ccn(CCF)n2)=O)nc1 C(=O)(C(CCOC)NC(c1c[nH]c(=O)cn1)=O)NCC#C N1(C(CSc2ccc(OC)cc2)C(=O)NCC(C)C)CCC(S(=O)(=O)C(C)C)C1 C1(NC(C(C=C)C)=O)CC2(C(=O)NCCC#CCO)COC1C2 C1(CCOC)(NC(=O)CCC2CCCCC2)CCN(C(=O)CC2C=CCC2)C1 c1(C(=O)NC2C3(CN(C(C(CSC)O)=O)C3)CCC2)cc2c(F)ccc(F)c2[nH]1 C(=O)(CC(C)C(=O)N1CC(CNC(c2cc(F)ccc2C)=O)C1)OC N1(c2ccnc(NCC(COCC)(C)CO)n2)CCOC2(CCCC2)C1 C1(CC(=O)N(C)Cc2ccc(CNC(=O)CC(C)(C)O)cc2)CCCC(C)(C)C1 Cc1noc2cc(C(=O)NC(C3CCCN3C(c3cnc(O)s3)=O)(C)C)ccc12 C(C(O)C(=O)N(CCCCCNC(=O)CCC1CC1(C)C)C)SC N1(C(CC(CC)O)=O)CC(NC(=O)Cn2ncn(C)c2=O)C(C)(C)C1 N1(C(C(c2ccoc2)NC(C2C(OC)CC2)=O)=O)CCCC(C2(C)CC2)C1 N1(C(C(C)NC(c2ccoc2)=O)=O)CCC2C(C1)CN2C(=O)CCC1CCOC1 CC(C)C(F)(F)CC(=O)N(C)CCC1CCN(C(c2cnc3n2CCS3)=O)CC1 C=CCCCCCCC(=O)OC.C1CCCN(C(=O)C(C)ONC(=O)OC(C)(C)C)C1 C12(C(=O)NC3(C)CC(NC(=O)C(C4CCOCC4)F)C3)CC3CC1C2C3 N1(C(CCC(CC)C)=O)CCn2ncc(C3(NC(=O)C(=O)N(C)C)CCC3)c2C1 c1(-n2cc(C(=O)OC)nn2)ccc(C(N2CCCCC2C)=O)cc1.C12CCN(C1)C2 N1(CCNC(C2C(c3onc(CC(C)C)n3)C2)=O)CCN(Cc2cccs2)CC1 C1(CNC(CCC(C)OC)=O)CN(C(c2cc(F)ccc2Cl)=O)CCC12CCC2 N1(C(C#CCNC(c2c(CC)oc(C)c2)=O)=O)CCSCC(C)C1 N1(C(C2N(C(=O)OC(C)(C)C)CSC2)=O)CC2CN(c3nccc(Br)n3)CC12 C1(NC(=O)CC2CCC3CC23)CC2(CCCCN2C(c2ccc(=O)n(O)c2)=O)C1 C(=O)(C(CCF)NC(=O)C=Cc1cc[nH]n1)N1CC(CC(=O)OC)C1 CCC(C)C(O)CC(=O)NCCCC(C)(C)NC(c1cn2ncccc2n1)=O c1(C(=O)NCC2CCC(NC(CCOC)=O)C2)cc(N(C)C)cc(C#N)c1 n1(CCC(=O)NC(c2occc2Br)C)cc(CCSC(F)F)nn1 c1(C(=O)NCC(C(=O)OC)C2CCCCC2)c(-n2cnnn2)sc(C)c1C Cc1cc(S(N)(=O)=O)cc(C(=O)NC(C)C(C)NC(=O)CN2CCCCC2)c1C CCC(C)CCCCC(=O)NC1CCN(C(c2cc(Br)n(C)c2)=O)C1 c1(OC)nn(C)cc1C(=O)NCC1CC(F)CN1C(c1nc(=N)cc[nH]1)=O CC(C)CC(C(=O)N1CC2(CCC2)CC1C(=O)N(C)CC1CC1)C(N)=O C1(NC(CC(C(C)C)OCC)=O)CN(C(c2ccc(C#N)o2)=O)CC12CCCC2 C1(c2cn(C(C(=O)OC)(C)C)nn2)CCCN(C(C2C3CN(C)CC23)=O)C1 Cc1ccc(=N)[nH]c1C(N1CCC(C)(CNC(C2CC23CC(O)C3)=O)C1)=O CCC(CC(=O)NCC12CC(CO1)N(C(=O)C1=NOCC1)C2)C(F)F N1(C(C2(SC)CC2)=O)CC2(CNC(=O)CCc3nnc(C)n3C)CC1CO2 c1(NC23C(CN(C(C(C)OCCCC)=O)C2)CCC3)[nH]c(=O)n(C)c(=O)c1C#N C1(C(N(CCC(C)O)C)=O)CCC=CC1NC(=O)CC1CCCC(=O)C1 C(=O)(CC(C)(C)C(=O)N1CC(CC(C)NC(=O)C=CBr)C1)OC c1(OC)ccc2[nH]c(C)c(C(=O)NC(C)CN(C(=O)COCCN(C)C)C)c2c1 C1(NC(c2cc(C(C)C)c(Br)cc2)=O)CC12CCN(C(C1CCCOC1)=O)CC2 CC1=NOC(C)(C(=O)NCCCN(C(c2ccc(OC(F)F)nc2)=O)C2CC2)C1 C(CC(=O)Nc1cccc(C#N)c1)(C(C)(C)C)NC(CCCOCCC)=O CC(CC(=O)N1CCC(CNC(C2(C(C)(C)C)CCC2)=O)C12CC2)C(C)(C)C c1(CN=C(NCC(COC)(C)C)NCC(C)(C)C)cccc(C#N)c1F c1(C(=O)NCC2(CN(C(C=CC(C)(C)SC)=O)C)CC2)cn2cccnc2n1 CCCC(C(O)C(=O)N1CC(C(=O)NCC)C1)NC(=O)Cc1csc(C)c1 C(=O)(C(C#N)C(C)(C)C)NCC1(CNC(C(C(C)C)n2ccnc2)=O)CC1 C1(NC(C2(CC#C)CCCC2)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1O C1(CNC(=O)Cc2ccccc2F)CN(C(c2csnn2)=O)CCC12CCOC2 c12nnc(n1CC(=O)OC(C)(C)C)n2Cc1cc[nH]n1.c1(COC)cccnc1C N1(C(C(Cn2ccc(C)n2)C)=O)CC(C)CN(C(=O)C(C)CC2CCC2)CC1C c1(C(C)NC(=O)NCC2CCSC2)c(F)cccc1Cl c1(OC)cc(F)c(F)cc1NCc1cc(O)cc(Br)c1 C(c1cccc(C(F)(F)F)c1)=CC(=O)NC1CN(C(CCC#C)=O)C2C1C2 C1(C(=O)NCC2(O)CCN(C(Cn3c(C)nnn3)=O)CC2)CCc2nnnn2C1 c1(C(C)=O)csc(C(=O)N(C)Cc2cn(CC3CCOC3)nn2)c1 C(=O)(C1=COCCC1)NC1CN(C(C2(CC#C)CCCO2)=O)CC1CCC C1(NC(C(N(C(CCC(=C)Cl)=O)C)C2CC2)=O)CCOC(C)(CC)C1 N(C1CCCc2ccoc21)c1nccc(N(C)CC23CC(CO2)C3)n1 CC1CCc2[nH]nc(C(=O)NC3CCN(C(C4CS(=O)(=O)C4)=O)CC3C)c2C1 c1(C(N(C)CC2N(C(Cc3nnc(C)o3)=O)CCCC2)=O)cc(C)c(F)cc1N c1(CNC2CCC(C)(C)CC2C(N2CCNC(=O)C2)=O)ccc2ccccc2c1 c1(N2CCCC(O)CC2)nc(N2CCOCC3(CCC3)C2)c2ccsc2n1 Cc1c(C(N2CCC(F)(C(=O)N(CC(C3CCCC3)O)C)C2)=O)cccc1F c1(C(N(CCN(C(=O)C=CC(F)(F)F)C(C)C)C)=O)cnc(N(C)C)cn1 C(=O)(C1=C(Cl)CCC1)NC(c1ccc(C)cc1)CNC(=O)C(C)O c1(C(=O)NCC2(C)CCN(C(Cc3nnc(C)o3)=O)C2)ccc(F)cc1Br c1(C(c2nnnn2C(C)C)NC(C=C)COC)c2c(nn1C)CCCC2 C1(CNC(CCC#C)=O)CCC2(CCN(C(=O)C(F)C(F)(F)F)CC2)CO1 c1(C(N2CC(NC(CCCN(C(C)=O)C)=O)C(C)C2)=O)cc2occc2s1 C12(NCCNC(CN3CC(=O)NC3=O)=O)CC3CC1(C1OCCO1)CC3C2 c1(C(=O)NCCCN(C(C2CCCC2C2CC2)=O)CC)cc(OC)cnc1F c1(-c2onc(CCc3ccc(F)c(Cn4ccnc4)c3)n2)nc2c(s1)CCNC2 c1(C(N2CCNCC2)=O)ccc(S(C)(=O)=O)cc1.Cc1sc(O)nc1 CC(CNC(=O)CC1(C)CCC1)C(F)C(=O)Nc1cncc(C2CC2)c1 N1(C(CC(COC)C)=O)CCC(C)(CNC(=O)CC2CCN(C(C)=O)CC2)CC1 c1(OC)ccc(C(=O)NC2CC3(CNC(=O)O3)C2)c2ccoc12 C1(OC)CCCC(CC(=O)N(CCCCNC(c2ccc(C(F)F)s2)=O)C)C1 C1(NC(C(N2CCN(C)CC2)C)=O)CCCC(NC(c2cc(C#N)on2)=O)C1 c1(C(=O)NC2(CNC(CC3CCC(C)C3)=O)CCCCC2)cc2sccc2n1C c1(C(=O)NCCCCCN(C)C(C2CSCC(=O)N2)=O)ccc(Cl)c(O)c1 C12(CNC(CC(C=C)C)=O)CC(CCO1)N(C(C1CC(C3CC3)C1)=O)C2 Cn1ccc(C(=O)NC2CCCC2NC(c2ncoc2-c2ccco2)=O)n1 c1(C(C)(C)C(=O)NCC2CC2NC(=O)CC2CC=CCC2)ccccc1Cl c1(C(N2C3(CNC(C(C)(C)OCC)=O)CC(C2)C3)=O)cc(C)nc(Cl)c1N N1(C(C(C)OCCC=C)=O)CC(C(=O)NCC2CCC3(CC3)CO2)C2(CC2)C1 C(C(C)CC(=O)NCC1(C(=O)NC2CC(=O)N(C3CC3)C2)CCC1)OC C1(C2CCCN(C(=O)C=C3CCC3)C2)(NC(Cc2ncc(C)s2)=O)CC1 C1(NC(C(C)NC(=O)NC)=O)CC2CN(C(c3cccc(F)c3Cl)=O)CC12 N1(C(c2cc(OCC)no2)=O)CC2(CCC2)CC1CNC(=O)C1=C(C)OCCS1 C1(OC(CSCCC=C)=O)CCCC(=O)N(C)C1 Cc1ccc(CC(N2CC3CC2C3CNC(c2cncc(C3CC3)c2)=O)=O)cc1 c1(CNC(c2c(C)cns2)=O)ccc(CN(C)C(C2CCN2C)=O)cc1 c1(C(N2CC(NC(c3c(COC)cco3)=O)C(F)C2)=O)cc2ncccc2[nH]1 CC1CN(C(C2(C)CCCCC2(F)F)=O)CC(C)N(C(=O)C(=O)CC(C)(C)C)C1 C1(C(N2CC(CCC=C)(C(N3CCC(CC)C3)=O)C2)=O)CC2CCCC2C1 CC(C)(CC(F)C(=O)N1CC(=O)NC(=O)C1)NC(=O)CS(C)(=O)=O C1(CC(N2CC3(CCN(C(C4C(C)C4)=O)C3)C2)=O)CCC2(CC1)OCCO2 C1(CN(C)CCN2CCC(CSc3ccccc3)CC2)CC(N)CCOC1 c1(C(=O)NC(C2CN(C(c3cnc(O)c(F)c3)=O)CCO2)C)cc2cscc2s1 C=CCC(C(=O)NCC1(CNC(C2CC(O)CN2C)=O)CCC1)c1ccccc1 C1(c2nnnn2CCC2CC2)(NC2(CC)CCC2)CCOC(P(C)(C)=O)C1 O=C(NOC1COC1(F)F)C(c1cccc(C2(OC(F)F)CC2)c1)C(F)(F)F CC1Oc2c(C(=O)NC3CCCN(C(=O)C4=CCCS4)C3C)cccc2NC1=O Cc1cc(Cl)cc(C(=O)NCC(O)CN(C(=O)CC2CCCC2)C)c1O C12(CNC(C3CCN(C)C3)=O)CC(NC(C3CCCS3(=O)=O)=O)(C1)C(C)(C)O2 C1(CC(=O)NCCC(C)NC(c2ccc(C(C)(C)C)cn2)=O)OCCOC1(C)C N1(C(C2C(=O)OCC2)=O)CCCC(N(C(=O)CCn2cnnn2)CC2CC2)C1 N12CC3OCCCC3(C1)C2=O.N1(C(C)C(=O)NC)CCN(c2ncccn2)CC1 c1(C(=O)OCC)ocnc1-c1cn(CC(=O)N(C(C)CO)C)nn1 N1(C(C)C)CCCC1C(=O)NC1COCC1C(N1CC(c2nncs2)C1)=O Cc1ccc2nsnc2c1C(N1CCCN(C(c2cc(C(N)=O)cs2)=O)CC1)=O Cc1ccccc1CC(=O)NCCCCC(=O)N(CC(C)(C)C)CCO FCCN=C(NCCN1CCOCC1)N1CCN(CCC2CC(C3CC3)C2)CC1 C1(C(=O)NCCC(C)N(C(C(C)CO)=O)C)CC(N=[N+]=[N-])C1 CCCC(C(=O)NC1(C)CC(NC(=O)CN2CCCC2CO)C1)N(C)C Clc1ccc(C2=CCN(c3ccc(Br)cn3)CC2)cc1 Cc1cc(F)ccc1CNC(C1CCCC(NC(=O)CSc2ccccn2)C1)=O c1(CC(N2C(C3(NC(C4N(CC)CC4)=O)CC3)CCC2)=O)cnn(C)c1C C1(NC2(C(N(C(C)C)C)=O)CC2)CCN(C(=O)COCC2CCC2)C1 C1(C(C(=O)NC(C2CCCC2)C#C)C)CCN(C(=O)Cc2cncn2C)C1 CN1CC=C(CC(=O)N(C2(C(=O)NC3(C4CCCO4)CC3)CC2)C)CC1 c1(CC)ccc(C(=O)NCC2(C)CCC(NC(=O)CSCCN(C)C)C2)nc1 c1(OC)ccc(CN2CCC(O)C(C(=O)Nc3cccnc3I)C2)c(Cl)c1 c1(C(CC(=O)OC)O)nc2ccccc2[nH]1.C12CC(C(=O)O)CN1C2 C1(CNC(CCOC)=O)COCCN1C(C1CC2CC2C1)=O C=CCCCC(C)(C)C(=O)N1CCC(C(C)C(N2CCOC3COCC23)=O)C1 CC(C)(O)C(F)(F)C(=O)N1CC2CC(NC(c3csc(Cl)c3Cl)=O)CC2C1 C1(CC(=O)N(CC(C)N(C(C2CN(C(=O)NCC)C2)=O)C)C)CCCS1(=O)=O c1(OC)ccc(CN(C)C(C2CCCN(C(=O)CO)CC2)=O)cc1OC(C)C C1(O)(CNC(CCCC#C)=O)CCCN(C(c2ccc(OC)nc2F)=O)C1 N1(CC23N(Cc4n(CC(C)C)ncc4)C(CC2)CC3)CCc2ncsc2C1 C1(C(=O)NC(CNC(=O)Cc2cnns2)C2CCC2)(COC)CC=CCC1 Cc1ccncc1C(=O)NC(c1nocc1C(=O)NC1(C(C)(F)F)CCC1)C C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC(CN(C(CSC(C)C)=O)C)(C)C C1(NC(C2(C)CC(=C)C2)=O)CC2CCC(C1C)N2C(c1csc(=NC2CC2)[nH]1)=O CCC(C(=O)N1CCC(CN(C)C(C2CC(n3cnnc3)C2)=O)C1)N(C)CC C=C(Cl)CC(C(=O)NC1CC(OCC)C1)NC(c1nccs1)=O C(=O)(CCCC(C)(C)C#N)NC1CCN(C(c2ccc(OCC)nc2)=O)CC1C N1(C(C2CN(C)C(=O)N2)=O)CC2(C)CN(C(C3CCC(C)CC3)=O)CC2(C)C1 Cc1ccc(Cl)c(O)c1C(N1CCC(C(C)NC(c2cc(Cl)cs2)=O)CC1)=O C1(C(=O)NCCC(CC)C)CCN(C(=O)CCCSC)C12CCC2 Cc1c(NC(C2CCCCN2C(c2ccc(F)cn2)=O)=O)ccc(Br)c1F N1(C(C2CCC(CN(C)C)O2)=O)CCOC(CNC(c2nccn2C(C)C)=O)C1 N1(C(c2ncccc2C(F)(F)F)C)CCC2(C1)CN(Cc1cccc(Cl)c1F)C2 CC1CN(C(=O)C(c2ccccc2)O)CCC1CNC(c1csc(C(N)=O)n1)=O C1(CNC(COCCCOC)=O)CN(C(=O)C(C)(C)c2cccnc2)CC1C CC1(CNC(=O)C(O)CC2CCOCC2)CC(O)(CO)C1 Cc1cccc2c1ccn2CC(N1CCN(C(=O)C(C)O)C(CF)C1)=O C1(F)(CNC(C2(NC(N)=O)CC2)=O)CC2CCC(C1)N2C(c1ccnn1CCF)=O c1(CC(=O)NC2CN(Cc3cncc(F)c3)CC2O)ccc(Br)cc1Br N1(C(c2cc(CCC)[nH]n2)=O)CC2C(C1)C(=O)N2.C(CSC(C)C)OC CCCCC(C(=O)NCc1c(C)cccc1C)NC(=O)C(CC1CC1)OC N1(CCNC(CCN(C(c2ccc(CC)o2)=O)CC2CC2)=O)CCCC(O)C1 C(CCC(N)=O)(C(=O)N(CCO)CC1COCC1O)NC(=O)OC(C)(C)C C(=O)(C1=CC2CCC(C1)C2)NC1C(CC)CN(C(=O)CCc2nc(O)n[nH]2)CC1 O=C1CN(CCNC(C2CC23CCC3)=O)CCN1.c12ccc(nc1)Cn1cc-2nn1 Cn1ccnc1CCC(N1CC(CO)(NC(C2OCCC2c2cccs2)=O)C1)=O C=C=CCN=c1nc2ncn(CC)c2c(NCC(=O)NCC2CC2)[nH]1 NC(=O)CCCC(=O)NC1CCN(C(C23CCN(CC2)C3)=O)C1 N1(C(c2oc(CC)c(C)c2)=O)CC(CNC(c2ccc(C)cn2)=O)C2(CCC2)C1 c1(C(CNC(=NC)NCc2cc(-c3ccc(F)cc3)n[nH]2)(C)C)ccc(F)cc1 N1(C(C=CC(=O)N(C)C)=O)CCC(F)(CNC(C2CCCN(C(N)=O)C2)=O)C1 c1(C(=O)O)[nH]nc(NCc2cn(C3CCCCC3)nn2)c1-c1ccccc1 C(=O)(C#CC1CCOCC1)N(C1CCN(C(c2c(C)cc(O)nn2)=O)C1)CCO c1(C(=O)NCCC(C)NC(C2CC2c2cccs2)=O)cc(O)nc(C2CC2)n1 C1(C2CCN(C(=O)CC3=CCCC3)C2)(NC(CC2(CC(N)=O)CC2)=O)CC1 C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCC2(N(C(CC(CC)C)=O)CCC2)C1 C(=O)(C(CNC(=O)CNC(=O)CC)CC(C)C)N1CCCN(CC=C)CC1 C(=O)(C(CNC(=O)Cc1n[nH]c(C)n1)CC(C)C)N(CCC)CCC c1(C(N2C(CCN(C(C(CC#C)OC)=O)C)CCCC2)=O)ncn2c1CCC2 CCCCCC(O)CC(=O)N1CC2(CC2)CC1CC(=O)NCc1ncc(C)s1 Cc1cc(NC(C2(NC(c3cn(C)cn3)=O)CCOCC2)=O)cc(Cl)c1 C1(c2onc(CC(C)C)n2)CCCCN1C(C(=O)NCC1CC1)C1CC1C(C)C C(=O)(C1CCc2nnc(C)n21)NCCC(C)N(C(c1cc(CCC)on1)=O)C C1(NC(c2c(CC)c[nH]c2)=O)CCN(C(C2CCNC2=O)=O)C(C)C1 N1(C(c2c(CC)onc2C)=O)CC2CC1CC2CNC(c1ccns1)=O Cc1cccc(N)c1C(N1CC(C)(NC(=O)CC2CCC2C2CC2)C1)=O C1(n2cc(-c3n(C)ncc3)nn2)C2CN(C(=O)C(=O)NC3(C)CC=CCC3)CC12 c1(OCC(=O)NCCCNC(CC=CCCCCC)=O)ccc(C(N)=O)cc1 c1(C(=O)NCC(CN(C(=O)CC23CCCC2C3)CC)(C)C)cccc(F)c1F Cc1cccc(C(=O)NC(CNC(c2cccc(-n3cccn3)n2)=O)CO)c1 C(CCC(C)C(=O)NCC(C1CCCN1c1nnc(C)s1)(C)C)OC CCC(C)CCCC(=O)NC(CNC(c1ccnn1C1CCC1)=O)CO c1(C(=O)NCC(C)NC(C2CC(N(C)C)C2)=O)cnc(Cl)c(N)c1 C1(NC(C(C)N(C)C)=O)CC12CCN(C(c1c(F)cc(O)cc1F)=O)CC2 Cc1ccn2ncc(C(=O)N(C3CCCC(NC(c4cnc(O)s4)=O)C3)C)c2n1 CC(C)C(CCN(C)C(C1CC(Cl)(Cl)C1)=O)NC(C1(N(C)C)CC1)=O c1(COC)cccc(C(N2CCC(C)(NC(C3CCCCO3)=O)C2)=O)c1 c1(C(N2CCC(NC(C3C=CCC3)=O)C(O)C2)=O)cc2ccccc2oc1=O CC#CCC(C(=O)N(C)Cc1ccncn1)NC(=O)COCC1CCCO1 N1(C(c2c(C)onc2)=O)CCC2(CCCC(CNC(=O)C(F)C3CCC3)O2)CC1 C1(C(=O)OC)CC(C(=O)NN2CCC(SC)C2)CC(C(=O)OC)C1 C1(NC(C2C(C(=O)OC)CCC2)=O)CCN(C(=O)CC(C)(C)O)C1C N1(C(CCC(=O)Nc2nnc(C)s2)=O)CC2(C1)OC1(C)CC2(c2nn[nH]n2)C1 CN1CCCC(CC(=O)NCC2CCCN(C(=O)CC3(C)N=N3)C2)C1 Cn1nccc1C1(NC(C2CCOC2CNC(c2ccco2)=O)=O)CC1 CCCCCC(O)C(=O)NCC1(OC)CN(C(C2CC3(CCC3)CO2)=O)C1 C1(CNC(C(C)C2CCCC2)=O)CCCCC1NC(=O)CC1CCSC1 C12(C(=O)OCc3c(C)c(Cl)ccn3)C3C4C1C1C2C3C41C c1(C(=O)NCC(CCOC)NC(C2CCCN2C=O)=O)sc(OC)nc1Cl C=CCC(C)(C)C(=O)NCC1CCN(C(=O)C=CCC)CC1C N1(C(Cc2n(C)ccn2)=O)CC2CS(=O)(=O)CC2(NC(=O)CN=S(C)(C)=O)C1 C1(CNC2(NC(=O)Nc3ccc(O)cc3)CC(CO)C2)CCS(=O)(=O)N1 C(=O)(CC(O)(CCC)CCC)N1C2CC(CC(NC(C(C=C)(C)C)=O)C2)C1 C12(CNC(CCCN=[N+]=[N-])=O)CCCC(CN1C(=O)CCNS(C)(=O)=O)C2 CC1(OCC(=O)NCc2ccc(Cl)s2)CN(C(=O)Cc2cncs2)C1 c1(N2CCC(OCC(C)(C)C)C2)nccc2sccc12 C1(NC(c2ccnc(OC)n2)=O)CCCCC12CCN(C(c1ccsn1)=O)C2 c1(C(=O)NC)ccc(CNCC2CCCCN2C(c2ccnc(S)c2)=O)cc1 CCCC(C)(O)CC(=O)N1CCCC1CCNC(c1cc2ccncc2o1)=O c1(C(N2C(C3CCN(C(C(N)=O)=O)CC3)CCC2)=O)ccc(O)c(F)c1 N1(C(CNC(CSC(C)C)=O)=O)CC(N(C)C2CC2)CC1C C1(NC(c2ccncc2Cl)=O)CCC2(CC1)CC2NC(c1ccc(=O)oc1)=O C1(C(=O)NCC2C3CN(c4nc(C5CC5)nc(=N)[nH]4)CC32)CCc2nnnn2C1 C1(CC(=O)NC(c2cn(C)nc2)C(=O)NCCCCCN=[N+]=[N-])NC(=O)NC1=O c1(C(=O)NC2CC(F)(CNC(C(CC)(C)C(F)F)=O)C2)ccc2nnc(O)n2c1 CCC(CC(=O)NC1COCCC1NC(=O)Cc1cncc(O)c1)CC(F)(F)F Cc1ccc(-c2nc(CC(N3CC(C(C)NC(C4CC4Cl)=O)C3)=O)cs2)cc1 CC(CCC(=O)NCC1CCCC1NC(=O)CNC(N)=O)c1ccccc1 C1(C(=O)NCC(C(C)O)C)(CNC(C2CCN(C)C2)=O)CCCCC1 c1(OC)ccc(C2C(=O)N2)cc1.c1(OCC(CC2CC2)CO)ccc(OC)nc1 C(=O)(CC(O)CCCCC)N1C(C#C)CN(C(=O)C(O)CCSC)CC1 Cc1cnn2ccc(C(=O)NCC(C)(CO)NC(=O)CCNC(N)=O)nc12 N1(C(c2n[nH]cc2Cl)=O)CC=CC(C(N2CCN(C3CCC3)CC2)=O)C1 C1(C(=O)NC2CC(OC)C2(C)C)CC(F)(F)CN1C(=O)CCN(C)CCO S(=O)(=O)(c1ccc(C)c2ncccc12)Nc1ccc(CC)c(C(=O)OC)c1 C1(CNC(C2CC(C)C2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)C2(CCOCC2)C1 C=CCC(CNC(C1(CC)CCC1)=O)C(=O)NCCc1c[nH]nc1O Cc1ccc(C(=O)NCC2(NC(c3cc(C)[nH]n3)=O)COC2)c(O)c1 N1(C(C(CCOC)OC)=O)CCCC(F)(CNC(c2cc(O)ncn2)=O)C1 C#CCCCCCC(=O)NCC1CCN(C(c2n[nH]c(C)n2)=O)CCC1(F)F c1(C(N(CC(C)NC(=O)Cc2cncs2)CC)=O)ccnc(OC(F)F)c1 N1(C(C(C)SC(C)C)=O)CCCCC(CNC(=O)CN2CCCC2C)C1 c1(C(N(C2CC(N)C2)C)=O)ccnc(-c2cccc(Cl)c2)n1 CCCCC(CN1CCCC(C#N)C1)CC N1(C(C(C)CO)=O)CC(C(=O)NC2CC(CO)(CO)C2)C2(CCC2)C1 C1(C(=O)NCC2(CNC(CC(=O)OC)=O)CC23CCC3)CN(C)CCN1C c1(C(=O)NC2CC(CNC(C3C(C)(C)CO3)=O)C2)ccc(CC2CC2)cc1 CCC(C)CC(C(=O)Nc1cc(CO)ccc1O)NC(c1coc(C(N)=O)c1)=O C1(N(C(Cc2cc(C)ns2)=O)C)CN(C(c2ccn(C)c2)=O)CCC1CO C1(OC)CC(NC(=O)C(F)C(C)C)CN(C(=O)C(C)(C)COC2CCCC2)C1 Cc1cc(C)c(C(=O)NCC2C=CC(NC(=O)Cc3c(C)noc3C)C2)c(O)n1 C1(NC(C(CC)C2CCOCC2)=O)CN(C(c2c(C)nsc2C)=O)CC1OC C#CC1CCC(NC(C2CCN(C(=O)C=Cc3ccccc3)CC2)=O)C1 c1(SCCC)ccc(C(=O)NC2CN(C(C3CCC3)=O)CC2O)cc1 c1(N2CCS(=O)(=O)CC2)cccc(S(=O)(=O)NC2CCSC2)n1 C1(C(C)NC(CC2(C=C)CC2)=O)CCN(C(c2cc(COC)nn2C)=O)CC1 Cc1nn(C)c(C(=O)N(C)CCCCCNC(=O)CCC(=O)OC(C)(C)C)c1Cl c1(CC)cc(NC(CNC(c2cnn(C)c2Cl)=O)C(C)C(C)C)nc(C)n1 c1(C(N(C2CCCN(C(c3nnn(C)c3C)=O)C2)CC)=O)cc(Br)c(C)o1 C1(C(=O)OC)CN(C(C(=O)Nc2cc(C(=O)OC)cs2)c2ccon2)CCCO1 c1(SC)cnn(C)c1C(=O)N(C)CCN(C)C(c1csc(C(C)=O)n1)=O N1(C(c2c(SC)nccc2)=O)C2CC1CN(Cc1cnccc1Cl)C2 C1(c2nc(CCCN(CC)CC)nn2-c2ccc(Br)nc2)CCC2CCCCN12 CCC(C)CC(=O)C(=O)N1CCC(C(=O)N(CCCF)CC)C1 Cc1nn(CC(N2CCCCC2CN(C(=O)Cc2cc[nH]c2)C)=O)c(=O)n1C N1(C(C(CCC)NC(N)=O)=O)CCC(NC(c2[nH]c(C)nc2CC)=O)C(O)C1 c1(CC(CC)C)nc(-c2cccc(Br)n2)nn1-c1cccc(OC)c1 c1(C(=O)NCc2nc3ccccc3[nH]2)cccc2ccc(Br)cc12 CCCC(CCC)C(=O)N1CC2C=CC1C(C(N1CC3CC1(CO)C3)=O)C2 N1(C(C)=O)CCC2(C(=O)N(CCC(C)C)CC(OC=CC=O)=O)CC2C1 C(CCC(=O)NCC1(c2ccccc2)CCCC1)C1C(C)C1.[nH]1cc(C2CC2)nn1 N1(C(C(C(C)C)SC)=O)CC2CCN(C(c3cccc4nc[nH]c34)=O)CC2C1 N1(C(Cc2c(C)nc[nH]2)=O)CCC2C(CCN2Cc2cnccn2)C1 C1(NC(C(C)NC(CC)=O)=O)CCN(C(=O)CC(O)c2ccccc2)C12CC2 c1(C(=O)OC)ccc(NC(N2CCOC(CC(C)(C)C)C2)=O)c2c1CCCC2 C(c1ccc(C(F)F)o1)=CC(N1CCC(CN(C(c2c(C)cns2)=O)C)C1)=O C#Cc1ccc(C(=O)NCC2CCN(C(=O)OC(C)(C)C)CC2C)cc1 Cc1c(F)ccc(C(=O)NC2(CO)CCCN(C(=O)CC3CCC(=O)N3)C2)c1N c1(C(=O)NCC2N(Cc3c(C)ccs3)CCC2)cnc(C)nc1C C(C)(C(C(=O)N1CCCC1C(C)(C)NC(C1CC=CCC1)=O)N(C)C)OC CC(c1ccsc1)=CC(=O)NCC1COCC1NC(C1CCCCO1)=O Cc1nc2cc(C(=O)NC(CNC(=O)C(CO)NC(N)=O)CC(C)C)ccc2o1 c1(SC)nc(N(C(CNC(C2CC23CCCC3)=O)C2CC2)C)cc(Cl)n1 C1(CC)(NC(C2CCCCN2S(C)(=O)=O)=O)CCCN(C(=O)COCCCF)C1 Cc1c(CC(N2CCOC(CCCNC(c3cncs3)=O)C2)=O)cnn1C CC1(C)C2CCC1(C(N1CCC(C(=O)NC(C(O)CO)C3CC3)(CO)C1)=O)C2 N1(C(C2CC(=O)N(c3cccc(Cl)c3)C2)=O)CCC(c2nn[nH]n2)C(F)(F)CC1 N1(C(C2C(=C)CC2)=O)CCOC(C)(CNC(=O)CC2CC3CCC2CC3)C1 C=CCC(F)(F)C(=O)N1CC(CC=C)(NC(C2(Cc3cccnc3)CC2)=O)C1 CCC(CC(=O)N1CCC(C(=O)NCCOCCOC)C12CC2)C(F)F C(=O)(CC(C(F)(F)F)NC(c1cnc(C(C)C)o1)=O)NC1CCN(CC)CC1 N1(C(c2c(C)nns2)=O)CC(CO)C2(C1)CN(C(=O)CCOC1CCOCC1)C2 Cc1cc(C(=O)NC2CN(C(=O)CCc3ccc(S(N)(=O)=O)o3)C2)cc(=O)n1C C1(NC(CC2CC(OC)C2)=O)CN(C(c2cncc(C3CC3)c2)=O)C(C)(C)C1 N1(C(CC2(OC)CC2)=O)CCC(C(=O)NCCCC2C=NNC2=O)CC1C C(C(C)(O)C(=O)NCC(c1ccc(F)cc1)NC(=O)CS(N)(=O)=O)OC N1(C(C(CC=C)C)=O)CC(F)(F)CC1CNC(c1n[nH]c(CO)n1)C Cc1nn2ccccc2c1C(=O)NC(C1CCCC1)CNC(=O)Cc1cnsc1 C(=O)(C(C(C)(C)C)NC(=O)C(C)CCN(C)C)NCCC(=O)NC C1(C(C(C)C)C#N)CCN(Cc2ccc(-c3csc(C(N)=O)c3)s2)CC1 Cc1cncc(OCC(=O)OCC2CCCC(N(C)C(C3(C)CCCS3)=O)C2)n1 C1(CCNC(C2CC(O)(CC#C)C2)=O)CSCCN1C(c1cscc1C#N)=O CC(N=c1nc(C(C)(C)C)s[nH]1)C(C)c1ccc(F)cc1 C1(O)(C(CNC(=O)CC2CCOC2)NC(C2C(OC)CCC2)=O)CCCCC1 c1(CC(=O)NCC2(CNC(C(CC(=O)OC)(C)C)=O)CC2)ccc2nccn2n1 N1(CCCNc2cccc(OC(CC)C)n2)CC(C)OC(C)C1 c1(OC)cc(C)c(CN2CC(C(N3CCC(CC(N)=O)CC3)=O)C2)cn1 C1(CC=C)(NC(C2CC2C2CCCO2)=O)CCN(C(=O)C#CC2(C)CC2)CC1 c1(CNC(c2c(CC)ncs2)=O)ccccc1CN(C)C(C1(F)C2CCCC12)=O C(=O)(C(C)(C)NC(C1CCOC1C1CC1)=O)NC(C(=O)OC)C1CC1 c1(C(N2CC(O)(CNC(C(=O)OCC)=O)C2)=O)cc(COC(C)(C)C)nn1C c1(CC(=O)NC(C2CC=CCC2)C(=O)NC(c2ncccn2)C)c[nH]ccc1=O C1(CN(C)C(c2c(Cl)csc2Cl)=O)CCCN(C(c2cc(C#N)no2)=O)C1 CC1(C)CCC=C1C(=O)NC1CCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)C1 c1(C(N(C2CCCC(NC(=O)C3=COCCC3)C2)C)=O)cc(O)cc(O)n1 C=Cn1nccc1C(=O)NCCCCC1CCCN(C(=O)CN(S(C)(=O)=O)C)C1 C1(CN(C)C(C2CCC(F)(F)C2)=O)C2CN(C(c3cccc(CO)n3)=O)CC12 C1(NC(c2cc(C)cc(Cl)n2)=O)CCN(C(c2c(C)ncn2C)=O)CC12CCC2 c1(CC)nn(C)c(C(=O)OCC2CCN(c3ccncn3)C2)c1Cl CC1CCN(C(C2CC3(CC3)C2)=O)CCN1C(=O)CCCCCc1cccs1 N1(C(c2c(N)c(O)nc(O)n2)=O)CC2CCN(C(=O)CCCF)CC2C1 c1(CC)cc(C(=O)NC2CC(C)(NC(C3CCCCC3F)=O)C2)c(C)nn1 C#CC1CN(C(=O)C(C(C)O)NC(=O)CSCCOC)CCO1 Cn1ccc2c(C(N3CCCC(NC(=O)C4=COCC4)CC3)=O)cccc12 C1(C#N)(OC)CC(C(=O)NC2C=CC(C(=O)NC(CO)CC(C)C)C2)C1 C(=O)(C1CCc2ccc(C)cc21)N1C2(CCN(C(C(C3CC3)OCC)=O)C2)CCC1 C1(N(C(CCC=C)=O)CCF)CCCN(C(c2nc(Cl)c(Cl)s2)=O)C1 c1(-c2nc(CC(C(N)=O)Cc3ccc(F)cc3)on2)c(O)ccc(F)c1Br N1(C(COc2cc(C)on2)=O)CC2C3CCC(C2C1)N(CCC1CCCO1)C3 c1(NCC(CC)CCO)[nH]c(=NCc2cccc(Br)c2C)nc2c1ncn2C Cc1cccc(NC(C)C(=O)Nc2ccsc2C(=O)NCC(F)F)c1 C1(OC)CCC(N=c2nc3c(cnn3C)c(NC3CCN(C(C)(C)C)CC3)[nH]2)C1 C1(C(=O)Nc2cccc(I)n2)CC2CCCCC2N1Cc1cccc2[nH]ncc12 Cc1cc(NC(c2coc(Br)n2)c2nnnn2CC2CCCO2)ccc1O C1(C(=O)NC(C2(O)CN(C(c3c[nH]c(=O)s3)=O)C2)C)CC2CCC1O2 C1(C(N2C(CNC(c3c[nH]nc3C3CCCO3)=O)CC2)=O)CCc2c[nH]nc2C1 C1(CNC(c2n(CCCSC)nnn2)c2cnsc2)(OC)COCC1(C)C Nc1cc(C(=O)NCC2CCCC(NC(=O)COC3CCCC3)C2)cnc1N C1(c2ccccc2)(NC(c2cc(F)cs2)=O)CCN(C(c2ccnnc2)=O)C1 C=C=CCCC(=O)NCC1(C(=O)NCC=CCCOC)CC1 Cc1cc[nH]c1C(=O)NCC1CCCN1C(C1CCC(=O)N1)=O c1(C(=O)NCC(C)NC(C2(C(=O)C3CC3)CC2)=O)ccncn1 c1(NC(C)=O)ccc(F)c(C(=O)NCCC(C)N(C)C(c2ccsn2)=O)c1 CN1C(=O)CC(NC(C2CC2CNC(=O)C(=O)C(C)(C)C)=O)C1=O C1(NC(CN(CC)CC)=O)CCCCC1NC(c1oc(C(F)F)cc1C)=O CCCCCC(C(C)(C)C)NC(N1CCCC(CC#N)(CO)C1)=O Cc1ccc2nc(C)cc(C(N3CCC(NC(=O)C(C)CN(C)C)C3)=O)c2c1 N1(C(CC2(C(=O)NC(c3c(C)ccc(Br)c3)=O)CCC2)=O)C2CCC1CN(C)C2 C(CC(=O)N1CCC1C)N(C(=O)C(N1CCCC1)C)CCC N1(C(C2C(C(=O)OC)C2)=O)CCC2(CC1)CCN(C(=O)CCc1ccoc1)CC2 c1(C(=O)Nc2cc(OCC)nc(OC)c2)c(C)cc(C)nc1OCC(F)F n1(CC)nnc(C(=O)NC(C)C=CC(N2CCC(C3CCO3)CC2)=O)c1C C(C(C)C)(C(O)C(=O)NC(COC)C(=O)NC(c1ccc(F)cn1)C)OC CC(CO)N(C(=O)CC1(CN(C)C(C2CC2Cl)=O)CC1)C N1(C(c2cnc(CC)[nH]2)=O)CCC(NC(c2cc(C3CC3)nn2C)=O)C(C)C1 c1(C(N2CCn3c(C)cnc3C2)=O)ccc2nc(C)c(C)nc2c1 N1(CC(C2CCOC2)OCC)C(=O)CN(CCc2ccccc2)C1=O C(N=c1ccnc(NCC2CCCCS2(=O)=O)[nH]1)C1(C=C)CCOCC1 N#CC1(C(N2CC3(C2)CN(C(c2ncc(Cl)cc2Cl)=O)C3)=O)CCCOC1 C1(NC(c2cc(OCC)ncc2)=O)CCC2CN(c3ccc(C#N)cn3)CC2C1 c1(C(=O)NC(c2ccc3c(c2)CN(C(=O)CC#N)C3)C)ccnc2c1ccn2C C(=O)(C(F)C(=O)NOC(CO)C(C)C)OCCN(C1CCCCCC1)CC CCC(C)C(C)C(=O)N(CC(CO)(CO)NC(=O)C=C1CCN(C)CC1)C N1(C(c2nc(CCC)oc2)=O)CCC(CNC(=O)C(C2CCC(=O)N2C)C)CC1 c1(C(=O)NCC2(C=C)CCOCC2)n[nH]c2c1CN(C(=O)C(C)(C)OCC)C2 c1(OCCCC(=O)NCCCC(C)NC(COC)=O)ccccc1[N+](=O)[O-] c1(CC)nc[nH]c1C(=O)N(CCCNC(c1cncn1CC)=O)C C12(C(=O)NCCSCCC=C)CCC(CC1NC(=O)C(CC)NC(=O)NC)C2 C(CC(C)(C)C(=O)N1CCCC(NC(N)=O)C1)SC.C12CCCCN1C2=O N1(C(Cc2cc(C)on2)=O)CC(NC(=O)C(Cl)=CCl)C2CC12 C1(NC(C(C)(N(C(CCCCN(C)C)=O)C)C2CC2)=O)CCC(C#N)CC1 c1(C(=O)NCC(CC)(C)NC(c2snnc2C)=O)cccc(N(C)C)c1 C=C=CCCC(=O)N(CCC(C)NC(c1c[nH]c(C(N)=O)c1)=O)C c1(C(N2CCC(C)(CCNC(C3COCCO3)=O)CC2)=O)ccc(S(N)(=O)=O)o1 O=C1CCN(CC(=O)NC2CCC(NC(=O)C(c3ccc(F)cc3)O)C2)C(=O)N1 c1(OC)ncc(C(=O)NCCCCCn2cc(C(O)CC(C)C)nn2)cn1 C1(NC(c2n(C)ncc2)=O)CCN(C(=O)CC2CCOC2=O)C12CCC2 N1(C(C2C(c3ccc(C)nc3)C2)=O)CCC2(CC1)CN(C(=O)CC(O)C(C)C)C2 c1(C(N2C(CNC(CC3(C)CCC3)=O)CC3CC32)=O)ccc(O)c2c1CCCC2 c1(CC(N2C(C(C)(C)NC(C3C(COC)C3)=O)CCC2)=O)c(O)nc(=N)[nH]c1C N1(C(C(C)SCC)=O)CC2CCC(C1)C(NC(c1cc(C(C)C)[nH]n1)=O)C2 C(=O)(C(C)CC(C)C(C)=O)NC(C(=O)N(CC(COCC)O)C)c1ccoc1 Cc1cc(C(=O)NC2(C)CC(NC(=O)CCCCCN(C)C)C2)cc(C#N)c1 c1(NC(C(C)NC(Cc2cc(OC)c(C)cc2)=O)C)cc2nncn2cn1 C(=O)(C1=CS(=O)(=O)CCC1)NC(c1ccc(C)cc1)CNC(=O)Cn1nccn1 C(C(=O)N=c1ccn(CCO)[nH]1)(C(C)(C)O)NC(c1c(C)nc(O)s1)=O C1(C(N2CC(CC)(CC)C2)=O)N(C(=O)Cc2nonc2C)CC12CCCC2 c1(C(=O)NCCN(C(=O)CC(C)C2CC2)CC)ccc2c(C)cc(Cl)nc2c1 C1(C(=O)NCCCOC=C)CCCCC1CNC(=O)Cn1cnnn1 C(=O)(C1CC(C)Cc2c[nH]nc21)NC1CC(NC(C2(CC#C)CC2)=O)C1 N1(CC(=O)NCCC2CC(NC(C34COCC3C4)=O)C2)CCCOC1=O c1(-c2cccc(OC)c2F)ccc2c(c1)CCN(C(=O)CCCCBr)C2 C1(C(=O)NC(c2nc(CC)[nH]n2)C)CCCN1S(=O)(=O)N(C)C c1(OC)nccc(C(=O)NCCCN(C(=O)C(C)C(F)(F)F)CCO)c1F Cc1csc(C(c2nnnn2CCN(C)C)NC(Cc2cccnc2)C(=O)O)n1 C1(C(=O)OC)CCN(C(C2COC3(CN)CC2C3)=O)C2(CCC2)C1 Cc1ccc(=O)n(CC(N2CCCC(NC(=O)C(S(C)(=O)=O)C3CC3)CC2)=O)n1 C1(C(C2CCCC2)SCC(C)O)CCOC1 Cc1oc(C)c(C(=O)NC(CNC(=O)C(C)(C)OC(C)C)C(C)C(C)C)c1C c1(OCC(=O)NCC2N(Cc3ccn(CCOC)n3)CCC2)ccc(Cl)cc1 c1(N2CCC(C)(C(C)C)CC2)nc(NC(C)Cc2ccnn2C)c2ncsc2n1 CC(C)C(C#N)C(=O)N1CC(CCO)(NC(=O)C(Cc2ccccc2)C(C)C)C1 c1(CC)c(C(=O)NC(C)CCNC(=O)CCc2ccc(Cl)cc2)csc1C N1(C(c2cnc(COC)[nH]c2=N)=O)CCN(C(=O)C(O)CC(C)C)CC12CC2 C1(CCN(C(CC(C)C)=O)C)CCCCN1C(=O)C(COC(C)(C)C)N(C)C N1(C(c2cc(C(C)C)[nH]n2)=O)CCCN(C(C2CC3CCCCCC23)=O)C(C)C1 c1(OC)cccc(CN2CCC(NC(c3c(Cl)cccc3Br)=O)C(F)C2)c1Cl c1(OC)cccc(C(=O)NC(C2CCCN2C(=O)CC(C)NC(N)=O)C)n1 N1(C(C(CNC(C(C)CC2CCC2)=O)CC2CC2)=O)CCOCC2(CCC2)C1 c1(NC(COC)(C)COC)nc(C)ccc1Br c1(OC(C(=O)N(C(CC)C)CCCC(F)(F)C(F)F)C)ccccc1Cl C(=O)(CC(F)(F)F)NC(C1CN(C(c2ccnc(S)c2)=O)C1)C c1(CC)nc(OC)c2ccccc2n1.N1(C)CCCC1c1cc(C)no1 N1(C(C(C)C#N)=O)CCC2(CCCCN(C(c3cnc4n3CCS4)=O)C2)C1 Cc1sc2ncc(C(=O)NCC3C4CN(C(=O)C(C)CN(C)C)CC34)n2c1C c1(C(=O)NCC(C)NC(C2C3COCC23)=O)[nH]ccc1CC1CCC1 C(=O)(C(O)C(F)(F)F)N(CC(C)C(=O)N1CCC1(C)CCO)C N1(C(C(C)N(CC(F)(F)F)C)=O)CC2(CCN(C(C3NC(=O)C4CCC34)=O)C2)C1 N1(C(c2c(OC)scc2)=O)CCCN(CCNC(C2CC(C)C2C)=O)CC1 c1(C(=O)NC2CN(C(C(CC=C)C)=O)CC2C)c([N+](=O)[O-])c(C)nn1C N1(C(c2cc(CC)ncc2)=O)CCN(C(=O)C(C)P(C)(C)=O)CC1CC(C)(C)C n1(CC(N2CCC(C)(CNC(CCC=C)=O)C2)=O)c(C)c(C)sc1=O C1(C)(C(=O)NCCCOC=C)CCCN(C(=O)Cc2ccccc2C#N)C1 N1(C(c2c(NCc3cccc(C(=O)O)c3)ccs2)=O)CCc2ccccc2CC1 C(=O)(CC1=CCN(C)CC1)N(CCNC(C1OCCCO1)=O)CC c1(N2CCC3(CC(O)C3)C2)nc(=NCCN2CCc3ccccc32)[nH]c2c1CCC2 Cn1nc(C(=O)NCC(C2CCOC2)NC(c2cnnn2C)=O)c2c1CCSC2 Cc1cc(C(=O)NCCCOCCNC(c2ccnnc2C)=O)ncc1F CC1CC2(CCN(C(=O)Cc3cnns3)CC2)CN1C(=O)C(O)C1CC1 C1(CNC(=O)C=CC2CCOC2)CC2COCC2N1C(c1ccc(O)nc1Cl)=O c1(C(=O)NCC(CNC(CSc2cccc(C)c2)=O)F)ccc2nc(Cl)nn2c1 C1(NC(CC2CCC(NC(COCCSC)=O)C2)=O)CC2CSCC2C1 N1(C(C=C2CCC(C)C2)=O)CCCCC1CNC(C1CC(O)C1)=O C(=O)(C(C)CN(C(=O)C(C)N(C)C(c1cocc1C)=O)C1CC1)OC Cc1nc(O)nc(O)c1CC(=O)NCCCC1(N(C(=O)CC2(C)CCCC2)C)CC1 C12(NC(CC(C=C)(C)C)=O)CC(C)(C1)OC21CCN(c2ccncn2)CC1 c1(C(N2CCCC(C(C)NC(=O)CN3CCCC3=O)C2)=O)cc2c(s1)CCC2 C1(CCC)(NC(c2oc(Br)cc2C)=O)CCN(C(=O)CCC(C)C)CC1 N1(CCC(=O)NCCCN(C)C(C2(F)CC=CC2)=O)CCCCCC1 N1(C(COC2(C#C)COC2)=O)CC2(C1)CN(C(=O)C(CC)SC)CCO2 C(=O)(CCCCC(N)=O)N(CCCNC(Cn1nc(C)n(CC)c1=O)=O)C1CC1 Cc1cc(CN2CCCC(C(N3CCCC34CC4)=O)CC2)ccc1F C(CCNC(C1(C)COC1)=O)(C(=O)N1CC2CC2(CO)C1)OC N1(C(C(COC)N(C)C)=O)CCCC(CO)(NC(c2ccc(F)cc2F)=O)C1 c1(C(=O)NC2CC(NC(C(C)OC3COCCC3)=O)C2)cc(C#N)ccc1O CN1CCC(CC(N2CCCC(C(C)(C)C(=O)NCC(C)(O)C3CC3)C2)=O)CC1 c1(NC(c2n(C)nnn2)(C)Cc2cc(F)cc(Br)c2)cc(C(F)(F)F)c(Br)cn1 Cc1cc(NC(=O)CC2C3CCC(C3)N2C(=O)CCCN2CCCC2)cc(O)c1 C1(CC(=O)NC2(C)CCN(C(=O)CSCCC#N)CC2)CCC2(CCC2)CO1 c1(CC(N2C(C)(CNC(CC(=O)OC)=O)CCC2)=O)cccc2nsnc12 C1(NC(C2(COC)COC2)=O)CCCN(C(c2cc(C(C)C)oc2C)=O)C1C CC1CC(C)N(C(c2cnco2)=O)CCN1C(c1cc2nccc(Cl)c2s1)=O C(N=C(NC1CC1)N1CCC(CC2CCCC2)C1)c1cn(CC)nn1 C(=O)(C(CO)C1CC1)N(CCNC(C(C)C)=O)C C1(NC(c2[nH]cc(C)c2)=O)CC2C1CCN2C(=O)Cn1nc(C)n(C)c1=O c1(C(=O)NC2CCN(C(c3cnc(C(=O)OCC)s3)=O)C2)c(Cl)nn(C)c1Cl CC1CC(=O)NCC1C(N1CCN(C(=O)C(c2ccccc2)C)CC1C)=O CCCC(CC)CCC(=O)NCC1CC(NC(=O)C2=CCCC2)CCO1 C1(C(N2C(CNC(C3(CC=C)CC=CC3)=O)CC2)=O)CCC(C)(C)CC1 N1(C(Cc2c(C)n[nH]c2C)=O)CC2CCCC2(CNC(C2CC2F)=O)C1 C1(C(N(C)Cc2nc(C)sc2)=O)CCN(C(=O)C23CC(C#N)(C2)C3)O1 n1(CC(=O)NC(C(C)C)C(C)NC(=O)C(Cl)=CCl)cc(F)ccc1=O C(C(CC(F)(F)F)NC(=O)C(C(C)(C)C)C1CCC1)NC(CC=C)=O c1(C(N2CC(=C(CNC(c3ncccc3F)=O)F)C2)=O)ccc(=O)n(C2CC2)c1 C1(CN(C(CC(C)c2ccco2)=O)C)COCCN1C(=O)Cc1cncs1 CCC(C)(CNC(=O)CCCCCSC)C(=O)NC1CN(C(C)C)C1 C1(C(=O)NCC2N(C)CCC2)CC(O)CN1C(=O)CC1CC2(CC2)C1 c1(NC2CCC(CNC(=O)OCC)C2)cc(OC)cc(OC)c1Cl c1(NC(C(=O)NC(C(=O)NCC(C)C)C)=O)cccc2c1CNC2=O C1(C(C)C)CCC(C(=O)NCC2CCCCN2C(c2sccc2C(F)F)=O)CC1 CCC(C)C(=O)NC(C)CC1CN(C(=O)C=C2CCC(C)C2)C1 CCC(C)CCCC(=O)N1C2CCC1C(C(=O)NCc1nc(C)c(C)[nH]1)C2 c1(CCC(=O)NCCN(C(c2cnc(C)o2)=O)C2CC2)ccc2[nH]ccc2c1 c1(C(C)(C)NC(C)C)cn(CCCCCNC(=O)Cc2ncoc2C)nn1 C1(NC(C(F)=CC)=O)(COC)CCN(C(=O)Cn2cnnc2O)CC1 C12(C(=O)NCC3C(NC(C4N(C(C)=O)CCCC4)=O)CCC3)CC(C)(C1)OC2(C)C Cc1cccc2ccc(C(=O)N(CC(C)NC(=O)C(Cl)=CCl)C)nc12 c1(C(N2CCCC(CN(C(CNC(C=CC)=O)=O)C)C2)=O)cc(C)[nH]c(=NC)n1 c1(-c2nc(CN(CC#C)C)on2)ccccc1F.C(F)(F)F c1(C(=O)NCCCN(C(=O)CSCC2CCCC2)C)ccc(N)c(F)c1 N1(C(C(=O)OC)=O)CC2CC2(CNC(=O)CC(C)SC)C1 C=Cc1cnn(C)c1C(N1CCCC(CNC(=O)C(C)(CO)OC)C1)=O c1(C(=O)NCC2CCC(NC(c3cc4n(n3)CCC4)=O)C2)ccc2cnnn2c1 C1(C(N2CCC(C)(CNC(c3cnc(N)cn3)=O)C2)=O)CC(S(C)(=O)=O)C1 c1(N2CCN(C(CCc3cccc(C)c3)=O)CC23CC3)ncnn2ccc(Br)c12 CC(C)(C)C(C#N)C(=O)NC1C=CC(C(=O)NCCC2CCC2)C1 C=CCCC(CC(C)C)C(=O)N1CCN(C(=O)C(C)(C)C(C)C)CC1CF C12(CNC(=O)CC3CC=CC3)COCCN1C(=O)CN(C(=O)C=Cc1cn[nH]c1)C2 N1(C(c2n(CC)c(O)nc2)=O)CCC2(CC2C(=O)NC(C)(C)CC2CCC2)C1 C(=O)(C1=CCCN(C(C(=O)NC2CC(F)(F)C2)C(C)CC)C1)OC NC(=O)CC(C(=O)NCC1CCCC1F)NC(=O)C1=CCSC1 N1(C(c2c(COC)c(C)on2)CC)CCCCC1C(N)=O.C123CC(C1)(C2)NC3=O Cc1ccc(I)c(C(=O)NCC2CCN(Cc3ncsc3C)C2)c1 C(CC(=O)NNC(=S)NCc1ccc(F)cc1)NC(CCOCC)C(=O)O C1(CNC(C(C)c2ccco2)=O)C(C2CC2)CCN1C(c1cncn1C)=O CCCCC(CC)C(=O)N1CC(F)(C(=O)NCC2CSCCO2)C1 C12(NC(Cn3ncc(C)c3)=O)CCCC(CN(C(=O)CCc3ncc[nH]3)C1)C2 c1(C(=O)NC(CC)CNC(=O)CC2(CN(C)C)CCC2)ccc(N)c(F)c1 CC(CCCCNC(=O)CC1(O)CCC1)NC(c1cnn(C)c1C(C)(F)F)=O C(=O)(CC(O)CC(C)C)N1C(COC)(CNC(=O)C(C)(C)C2CCC2)CCC1 CCCCCCC(=O)N1CCC(C(=O)NC2CN(CC(F)F)C2)(OC)C1 c1(C(=O)NC)ccc(NC)cn1.C1(O)(C(C(=O)C2(COCC)CC2)=O)CCCCC1 Cc1nc(=N)[nH]c(C)c1C(=O)NCC1(CNC(C23CCCN(CC2)C3)=O)CCC1 N1(C(c2cccc(CC=C)c2)=O)CCN(C(=O)CC(C)COC)CC(C)C1 C1(NC(=O)CC2Cc3ccccc3O2)CN(C(C2(Cl)CC2)=O)CCC12CCC2 Cc1ncc(NC(c2nnnn2C2(C)CC2)C2CCC2)cc1C(N)=O C#Cc1ccc(CC(=O)NC(CNC(=O)Cc2ccco2)C(C)C(C)C)cc1 c1(C(=O)NCCC(C)CCNC(C2(C)CCC2)=O)nnc(O)nc1O CC(C)C(F)(F)CC(=O)NCC1(F)CN(C(c2cc(C#N)cs2)=O)C1 N1(C(c2c(CCC)nco2)=O)C2CCC(C(=O)Nc3ccc(SC)cc3)C1CC2 O(N1C(=O)c2ccccc2C1=O)CC(=O)N(C)Cc1ccc(CO)cc1 C1(CNC(C(C)(F)F)=O)CCC2(CCN(C(C3CCSC3)=O)CC2)CO1 N1(C(c2cc(C)c(C)s2)=O)CC(NC(c2ccn(C(C)C)n2)=O)CC(F)C1 C1(CC)C(C(=O)NCc2cc(OC)n(C)n2)CCCN1C(C1COCCO1)=O C=C(C)C(O)CC(=O)N1CCN(C(c2ccc(CC(C)C)cc2)=O)C(C2CC2)C1 CON(CCC(=O)NC(C)CC(C)(C)OC)C(=O)C1C2CCC(F)(F)C12 c1(C(=O)NC2C(NC(CCn3c(C)ccc3C)=O)CC2)cc2ccc(F)cc2o1 Cc1c(C(N2CCCC2CNC(=O)COc2ccc(F)cc2)=O)cncc1Cl c1(C(=O)NC(CC)(C)CNC(=O)C(C(C)O)N(C)C)ccc(=NC)[nH]c1 c1(NC(C(=O)NCC(CNC(C2N(CCC)CCC2)=O)(C)C)=O)ccc(Cl)cc1 c1(OCC(=O)NC(CNC(c2cc(C3CC3)ncn2)=O)CO)cccc(Br)c1 CCCCC(O)C(=O)N1CCCC1C1(C(=O)NCCC(C)(C)O)CC1 N1(C(C2CCC(=O)C2)=O)CCC(C2CC(NC(C3CCCCC(=O)N3)=O)C2)CC1 c1(CC(=O)NC(C(C)NC(C2(n3ccnc3)CCCC2)=O)CO)ccc(O)nc1 C(CCCC(=O)NCCC1(O)CCN(C(C2(Br)C(C)C2C)=O)C1)OCC c1(-c2cccc(COCCOC(=N)O)c2)nc2c(s1)CCCC2 c1(C(N2CCCC(O)(CNC(CCSCC)=O)C2)=O)cnc2c(c1)COCC2 N1(C(C2(O)CC(C)(C)C2)=O)C2CCC1CN(C(C1CC1c1ccc(F)cn1)=O)C2 CCC(C)(CO)C(=O)N1CCN(C(c2ccc(C)c(Cl)c2)=O)C(C(C)C)C1 N1(C(=O)CCCc2nccs2)Cc2ccccc2C(c2cccs2)C1 c1(C(C(=O)NCC(C)(C)CNC(=O)CNC2CCC2)(F)F)cc(F)cc(C#N)c1 Cc1cnc(-c2cn(CCC3CN(C(=O)C(c4ccc(Cl)cc4)C)C3)nn2)nc1 CN1CCN(C(=O)CCc2cncnc2)C(CNC(c2cscc2C(N)=O)=O)C1 c1(CC(=O)NC2CCN(C(C(COCC)C)=O)C2CC)ccc(C)cc1Cl c1(OC)n[nH]cc1C(=O)NC(CO)C(C)NC(C1CC1c1ccoc1C)=O CC(C)C(C(=O)NCC1CCCCC1NC(c1ccc(Cl)nn1)=O)n1cccc1 c1(OC)cc(C(=O)NC2CN(C(C34CC(O)C3C4)=O)CC2OC)cnc1OC C1(C(C(=O)NC2CC2)NC2CCCN(c3cn(C)nc3)C2)CCS(=O)(=O)C1(C)C C1(NC(CC(CC)NC(=O)CC2C(=O)NN=C2C)=O)CCN(CC)C(C)C1 C1(CC(N2CCCC(N(C(c3cc(OCC)n[nH]3)=O)C)C2)=O)COC(C)(C)CO1 CN(CCc1ccccn1)N1CC2CCCC(C1)N2c1ccccc1F C(=O)(C(C)(C)CC(=O)N(C)C)NC(CN(C)C)C(N1CC(C2(C)CC2)C1)=O C=CCCCCCCCNC(c1ccc(O)c(Br)c1)=O C1(CNC(C(CCO)N(C)C)=O)CCCCN(C(=O)C(N)=O)C1 CCCCC(C(=O)NCC1CC(NC(C2CSCN2C(C)=O)=O)C1)C(C)C C(=O)(C1Cc2ccccc21)NCC(C)(C)CNC(c1c(F)cccc1Cl)=O C(=O)(C1=CC2(CCN(C(=O)C(=O)C(C)C)C2)C1)NC1(c2c(C)nn[nH]2)CC1 c1(C(=O)NCC(C)(CC(C)C)NC(C=NOC)=O)cc(S(N)(=O)=O)cn1C c1(OC)cc(F)c(C(=O)NCC2CCN2C(c2cccn3ccnc23)=O)c(F)c1 N1(C(C(C2CC2)SC)=O)CCOCC(CNC(=O)COCCF)C1 C1(CNC(CCOCCC)=O)CCC(N(C)C(C2(F)CCOC2C)=O)CC1 C1(OCC(=O)NCC2CC2NC(=O)CN2CC3CC3C2)CCCCCC1 c1(CC(C)C)ccc(C(C)C(=O)N(CC(=O)NCc2ccccn2)C)cc1 Cc1ccc(C(=O)NC2(CCNC(c3ccc(C(F)(F)F)o3)=O)CCC2)c(C)n1 C(=O)(CC(C)C(F)F)NCCC(=C)CNC(=O)COc1cccc(C(C)(C)C)c1 CCC(CC)(CC)C(=O)NC1CN(C(=O)CSc2ccc(F)cc2)C2CC12 N1(C(C2C=CCN(C(c3n(C(C)C)ccc3)=O)C2)=O)CCOC(C)C1C C(=O)(C(C)(CO)NCc1cnccc1C1OCCO1)OCC C(N=c1[nH]c(=NCCN2CCCC2C)[nH]c2c1COC2)c1nccc(CC)c1 c1(CN(CC(c2ccc(C(C)C)cc2)O)C=O)c(Br)cccc1[N+](=O)[O-] c1(OC)cc(OC)cc(CNC2(c3nnnn3CCC3CC3)CSCC2C)c1 N1(C(Cn2nnc(C)n2)=O)CCOCC(NC(c2cccc(N)c2F)=O)C1 c1(C(=O)NC2(CC(=O)NC(CC3CC3)C3CC3)CC2)cnccn1 C1(C(=O)NCCN(CCC)C(c2cccn2C)=O)CCCC1S(C)(=O)=O CCS(=O)(=O)C=CC(=O)N1CC2(CCN(C(c3cc(Cl)ccc3C)=O)C2)C1 c1(C(=O)NCc2nc(CNC(c3n(C)c(O)nc3)=O)sc2)cncc([N+](=O)[O-])c1 Cc1ccc(F)c(S(=O)(=O)NCCNC(=O)NC23CC(C)(CCO2)C3)c1 c1(NC(C2CCC(N)(C(F)(F)F)CC2)=O)ccc(S(=O)(=O)N(C)CC)cc1 CC(C(=O)NC(Cn1cccn1)C(=O)Nc1cccc(Cl)c1O)C(F)(F)F C(=O)(C1=CC2CCCCCC12)NC(CNC(c1c(C)c(F)c(F)cc1)=O)(C)C C12(C)CCCCC1C(=O)O2.C=C1CCC(C(=O)NCC)CC1 C1(C(=O)NC(c2cccnc2)C(=O)NCCC2(C)CCCC2)CC1C1CCC1 c1(C(=O)NC(C2CN(C(=O)CSCCN(C)C)CCO2)C)c(F)cc(F)c(F)c1F Cc1cc(C(N2CCOCC2C(=O)NCC2C(C)C2C)=O)c(N)s1 C1(C(=O)NC2(CC#C)CC2)CCN(C(=O)CNc2ccccn2)C1C(C)C C1(NC(c2c(C)csc2)=O)CCC2CCN(C(=O)Cc3ccccc3)C12 Cc1cc(CC(=O)N(CCNC(=O)CCF)CCOCCO)cs1 c1(C(=O)NCC2CCC(NC(CCCOCC)=O)CC2)cccc(Cl)c1Cl c1(C(=O)NCCN(C(c2nnn(C)n2)=O)C2CC2)cc(Cl)ccn1 N1(C(c2cc(C)c(C)[nH]2)=O)CC(C)C(C)(C(=O)NCCCc2cccs2)C1 N1(C(C2(C)C(C)(C)C2)=O)C(C(=O)NC2C3CCCC23)C2CC(O)C1C2 CC1CCC(Cl)=C(C(=O)NCC(C)(O)CNC(=O)Cc2ccncc2Cl)C1 C(=O)(C1=NOC2(CCC2)C1)NC1(CCOC)CCN(C(c2ccsc2C#N)=O)C1 CN1C(=O)CCCc2occ(C(N3CCC3CNCc3ccnc(O)c3)=O)c21 c1(CC)nc(C)ncc1C(=O)NC(C)CC(C)NC(c1ccc(OC)nc1Cl)=O c1(C(=O)NCCC(CNC(CC2ON=C(C)C2)=O)O)cccc2c1CC(C)(C)C2 CC(CC(C)(F)F)C(=O)N1CC2CC(O)C1C2NC(c1ccn(CCN(C)C)n1)=O Cc1ccc(O)c(C(N2CCC(NC(c3cn(C)cn3)=O)C(C)C2)=O)n1 C1(NC(CN(C2CCSC2)C)=O)CCN(C(C2CN3CCC2CC3)=O)CC1O Cc1ccc(C(=O)NC2CCCC2NC(=O)C(n2cc(Br)cn2)C)s1 c1(CC(C)C)ccccc1C(N1CC(N(C)C(C2CC(F)C2)=O)C(O)C1)=O N1(C(COCC)=O)CC2CC1CCC2NC(C1CC2(C1)CC2F)=O C1(C(=O)NC(CN(C)C(C2CC2c2cnn(C)c2)=O)(C)C)CCC(C#N)CC1 C1(C)(NC(c2c(CC)noc2)=O)CCCN(C(=O)C(C)(F)CC2CCCC2)C1 N1(C(C2CCC(SCC)O2)=O)CCC(CC(NCP(C)(C)=O)=O)C1(C)C C1(C(=O)NCCC)CCC(n2cc(CCC(C)O)nn2)C1 C(=O)(C#CC1(CC)COC1)N1CC2C(C(=O)NC3(CCC)CC3)(C2)C1 C1(F)(C(=O)NC(C2CCN(C(CS(C)(=O)=O)=O)CC2)CO)CCC(F)(F)CC1 N1(C(C#CC2(C)CC2)=O)CCN2C(=O)C(NC(c3cnccn3)=O)CC2C1 C12(CCNC(c3cc(C)on3)=O)CCC1CN(C(=O)C=C(C1CC1)C1CC1)C2 c1(C(N(C2CCCC(NC(=O)C(C)(C)c3cccs3)C2)C)=O)cnc(=N)[nH]c1 CN1C(=O)CCCC1C(=O)NCC1CCN(C(c2cncc(F)c2)=O)C1 C(=O)(C(C)(O)C(C)C)NC1CC(CCC(=O)Nc2ccc(OCC)cc2)C1 N1(C(C)=O)CCC(C(=O)OS(=O)(=O)c2ccc(F)cc2)C2CCCC12 S(=O)(=O)(c1cc(Br)c(Br)cc1F)N(CCN(C(C)C)C)C C1(C(N(CCNC(C(C)n2ccnc2)=O)CCOCCO)=O)CC12CCC2 C(=O)(CC(O)(CC)c1ccccc1)NCC(CC)NC(=O)CCCCCF C1(OC)CCCC(C(N2CCC(C)(NC(c3n[nH]c(C)c3O)=O)C2)=O)C1 N1(C(CSCCC)=O)CCC(NC(C2CC3(CC3)CO2)=O)CC1c1ccccc1 C1(C)(C(N(CCCO)CCC)=O)CCCN(C(c2ccc(F)s2)=O)C1 c1(N(C(C(CC)C)=O)C(=O)CN2CC3CC2CO3)ccc(Cl)cc1 C=CC1(CC(=O)N(C2CCCC(NC(=O)CC3CCC3)C2)C)CCCCC1 Cc1sc(C)c(S(=O)(=O)N2CC3(CO)CCCC3(F)C2)c1Br C1(C(N(CCN(C(C)C)C(C2CC(CCO)C2)=O)C)=O)CCC(C)C1 c1cc2ncc(N3CC4CCN(c5ncncc5I)C4C3)cc2[nH]1 c1(OC)ccc(C(=O)NCC2CN(C(C3(C#N)CC3)=O)CC2O)c(F)c1F C(=O)(C(C(C)C)N1CCCC1=O)NC(C1N(C(c2cc(C)on2)=O)CCC1)C C1(C(N2CCC(NC(C=COCC(COCC)O)=O)C2)=O)CCCCC1OCC C(=O)(CC(C)c1nn[nH]n1)N(C(C)CN(C(=O)C(C)N(C)C)C1CC1)C C(CN=[N+]=[N-])(C(=O)N(C)Cc1ncn(C)n1)NC(c1c[nH]c(=NC)s1)=O C1(N2CCN(c3c(C#N)nccn3)CC2)CCOC12CCOC2 c1(CNC(=O)CC2CCN(C(c3ncc(Cl)cn3)=O)C2)cc(F)cc(Br)c1 C(CCN(C(=O)CC1CCCC(=O)N1)C)(C(C)(C)C)NC(c1c(C)onc1)=O C1(C(N(C(CCCC(=O)OC)=O)CC(C)N(C)C)=O)CCn2ncnc2C1 C1(NC(C2CN(CC)C2)=O)CCN(C(=O)CCP(C)(C)=O)CC1(C)C C#CCC(C)(C)C(=O)NC1CC(C)CN(C(=O)CCCc2ccc(F)cc2)C1 c1(C(N)=O)ccc(C(=O)Nc2ccc(N(C)C3CC3)cc2)cc1.N12CCOC(C1)C2 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N1CCC(C)C(CNC(=O)CO)C1 Cc1cc(C)n2nc(C(=O)NC(C)C(C)(C)NC(c3c[nH]c(=O)cn3)=O)nc2n1 C1(N(C(=O)CC2CCC(C3CC3)O2)CCC)CCN(C(C2(F)CCC2)=O)CC1 C1(N(C(CC=CCNC(C2N(CC)CCCC2)=O)=O)C)CCCCC1(C)C CCCC(C(=O)OC(C)(C)C)NC(c1ccc(F)cc1)C(=O)OC CCCC(F)C(=O)NCCC1(NC(C2CCCN(CCC)C2)=O)CCC1 c1(C(=O)NC2CN(C(CN(CCCCCC)C)=O)CC2O)cc(F)ccc1O n1(C(C)C)ccc(CC(N2CCC2CNC(C2CCOC2C2CC2)=O)=O)n1 C(c1ccccc1[N+](=O)[O-])=CC(=O)NCCOCCCNC(C1CCC(O)C1)=O C(C1(O)CCc2ccccc21)CCONC(=O)OC(C)(C)C c1(CCNC(CCN(C(CC)=O)CC2CC2)=O)ncnn1C.N12CC(C1)C2=O c1(C(N(CC(CN(C(CCCC(C)=O)=O)C)O)C)=O)cc2c(F)ccc(F)c2[nH]1 C(=O)(C(CC)C(C)(F)F)N1C(CN(C(c2cn(C)nc2SC)=O)CC)CCCC1 NC(=O)CCC(=O)N1CC(OCCNC(=O)Cc2cn[nH]c2)C1 C(=O)(NNC(=O)NCCNc1cccc(OCC(F)F)c1)SCC(N)=O CC1(C)CCC(CC(=O)NC23CCN(C(c4sccc4C(F)F)=O)CC2C3)CC1 C1(NC(CCCCCOC)=O)(CO)CCCN(C(=O)C(O)CSC)C1 c1(C(N(C)CC2(O)CCN(C(C(C)SC(C)C)=O)C2)=O)ccc2c(c1)CCO2 c1(COC)cc(O)nc(NCCCc2cc(C(=O)O)ccc2C)n1 CC1(CN=c2ccnc[nH]2)CCCN(C(=O)CCc2ccccc2)C1 S(=O)(=O)(c1cc(F)c(OC)c(Br)c1)N1CCN(c2ccc(OC)c(Cl)c2)CC1 c1(OC)ccnc(CC2CCCCC2C(N2CC(O)CC2C(=O)O)=O)c1OC N1(C(CC(CC)OC)=O)CCC2(CC1)CN(C(c1cnc(Cl)[nH]1)=O)C2C(C)C Cc1cccc(C)c1C(=O)Nc1cc(-c2c(C)noc2C)cnc1Cl C1(NC(c2c(CCC)n(CC)nn2)=O)CCN(C(=O)C=CCOC)CC1F c1(-c2nc(-c3nccc(OC)c3)nn2C2CCOCC2)ncc(C#N)cc1C S(=O)(=O)(c1csc(C(=O)NCC2CCCN2C(C2CC(C3CC3)=NO2)=O)c1)NC Cc1cc(C(F)F)n(CC(=O)NCC2COC(CNC(=O)C(F)(F)C3CC3)C2)n1 c1(C(=O)NC(CCNC(C(C)NC(COC)=O)=O)C)ccc(Br)c(N)c1 C1(C)(NC(C2(CNC(C3CC(OC)C3)=O)CCC2)=O)CC1(C)C CC(CCCNC(=O)Cn1nnc(C2CC2)n1)NC(C1CC(n2ccnc2)C1)=O CC1(CNC(C2(C3CCCN3C(=O)C(F)(F)CO)CC2)=O)CC2CC2C1 n1(CC(=O)NC2(C(N3CCOC(CCF)C3)=O)CC2)cccnc1=O C(=O)(CC1=NNC(=O)C1)N1CCN(C(CC(CC)C2CCCC2)=O)CC1 CCC(C)C(O)C(C)C(=O)N1CC(F)(F)CC1C(N1CCC(F)(F)C1)=O C12(C(N(C(CCCC)C)C)=O)CCC(NC(c3cccc(C)c3)=O)(CC1)C2 C1(CNC(CCC(=O)NCCC)=O)CC(C)(C)CN1C(=O)Cc1ccc(Cl)nc1 N1(C(c2sncc2C)=O)CCC2CN(C(=O)C(C3CCCCC3)C3CC3)CC2C1 c1(SC)cccc(C(=O)NCC(C)CNC(C23CC(C)(CCO2)C3)=O)c1Cl c1(C(N2C(CNC(C=C(C)C3CC3)=O)CC2)=O)ccc(=O)n(CC(C)O)c1 N1(C(CCCC)=O)CCN(CC(=O)NCC(=O)NC(C)(C)C)CC1 c1(C(C)C)ccoc1C(=O)NC(C)CC(C)NC(C1CC(C(=O)OC)C1)=O c1(C(=O)NCC(CO)NC(CCc2ccc(C)s2)=O)ccc2sccc2c1 C=CCS(=O)(=O)CCNC(C1CC(C)(C)C12CC2)=O C(=O)(C(C(C)O)NC(C1CCOC1C)=O)OC C1(CC(=O)Nc2ccc(CNC(COC(CC)C)=O)nc2)COCC(C)(C)O1 CC1(C)CCC(C(=O)NCC2CCC2)(NC(C2C3CCC(F)(F)C23)=O)C1 N(C1CCCn2c(C)nnc21)CC(c1cc(C)n(-c2cccnc2)c1C)=O N1(C(CCCCCN(C(=O)C(Cl)Cl)C)=O)CCC2CCCC2CC1 c1(OC)ccc2c(c1)OCC(C(=O)N1CCC1CNC(=O)CC1(O)CCC1)=C2 c1(OC)ccc2c(=NC(C)c3cc[nH]n3)[nH]c(=NCC(C)(C)C(F)(F)F)[nH]c2c1 N1(C(C2CC(CC)C2)=O)CCC2(NC(C3CCC(C(=O)OC)CC3)=O)CC2C1 N1(C(C(CC)CC2CCCC2)=O)CC2(CCC(NC(=O)CCC(C)OC)CC2)C1 c1(CC)cc(=NC(=O)C2CCC(C)N2C(c2cc(C)nc(C)c2)=O)[nH]n1C C(c1ccc(F)c(Cl)c1)=CC(=O)NCC1CN(C(c2c(C)nn(CC)c2C)=O)C1 C1(O)(C(N(CCOCCCNC(C(CC)NC(N)=O)=O)C)=O)CC(F)(F)C1 CCC(CNC(C1CC2(CCO1)CC2)=O)(CC)C(=O)N1CCC1C1CCCCC1 C1(C)(CNC(COCC)=O)CC(F)(F)CN1C(c1cc(C)cc(Br)c1O)=O C1(CNC(C23CC2CNC3)=O)CC(O)(Cn2cccn2)C1 Cc1nc(CC(=O)NC2CCCN(Cc3cn(-c4ccn(C)n4)nn3)C2)c(C)s1 CC1CC(N=c2[nH]c(N3CCC(OCCC(C)C)CC3)nc3c2CCCC3)CS1 Cn1ncc2c1CN(C(C1CC3CC3N1C(c1cc(C#N)c[nH]1)=O)=O)C2 c1(C(=O)OCC)cccc(C#CCNC(CCO)C(C)(C)C)c1 C12(CC(=O)NCC(C)(O)CNC(c3ccc(F)s3)=O)CCC(CC1)C2 c1(N(C)C)ncc(C(=O)NC2CN(C(=O)CCNS(C)(=O)=O)CC2CO)cc1Cl CC(CC(=O)N1CCCC(CC(=O)N(C2CCCC2)CCO)C1)CC(C)(C)C CC1(C)CC(=O)NC1CNC(C1(C)CN(C(C2CC3(CC3)CO2)=O)C1)=O C(CCNC(C1COC1)=O)(C(C)C)NC(C(C)(C)N(C)C)=O C=CC(C)(C)CC(=O)NCC(C)CN(C)C(c1ccc(OCCOC)cc1)=O Cc1cc(C(=O)NC(C2CCCCC2)CNC(=O)C(C)OC2COC2)cs1 C(=O)(N=c1[nH][nH]c2c1CN(Cc1cc(C)ccc1OC)C2)c1c(C#C)cccc1 CN=c1nc(N2CCOC(C)(C(F)F)C2)[nH]c(=NCC2(OC(C)C)CCOC2)[nH]1 C1(CNC(=O)CCC2CC2)CCC2(CCC2)C1NC(=O)CCNC(C1CCC1)=O CC1CC2CN(C(=O)CCc3ccc(C#N)cc3Br)CC2N1C(C1CC1F)=O Cc1cccc(C)c1NC(=O)C(Cc1cc[nH]n1)NC(=O)CN1CC2CC2C1 CCC(CCOC)C(=O)N1CCC(O)(C(C)NC(=O)CCCCC2CC2)CC1 Cn1c(C(N2CC(CNC(=O)C(O)c3ccsc3)CC2(C)C)=O)cccc1=O C1(C(F)(F)F)(C(=O)NCC(C)N(C(=O)CCC2CC2(C)C)C)CCO1 CCCCCCC(C)C(=O)NC(C)CNC(=O)Cc1cc(F)c(N)cc1F N1(C(COCCC#C)=O)CC(CO)CC1C(=O)NCC1(c2cccc(Cl)n2)CC1 C1(CNC(CCc2cn(C)nc2)=O)(CO)CC12CCN(C(c1cncs1)=O)CC2 N1(C(c2c(SC)cccc2)=O)CC(NC(=O)CC2(C)CCCO2)C2(CCC2)C1 n1(CC)ccnc1C(=O)NCCc1cc(C(F)F)n[nH]1 N1(C(CCCC#C)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)CC(C)(F)C1 C(CCCCC(=O)NC)OCC.N12CCN(CC1)CC(=O)N1CC(C1)C2=O O=S(=O)(c1cccs1)NCC1CCN(CC2(c3cccc(Cl)c3)CC2)C1 C=Cc1cc(C(=O)NC(CNC(=O)CCc2nc(CC)no2)CC)cc(F)c1 C1(CC(N2C(CN(C)C(C3CCCC4CC34)=O)COCC2)=O)CCCC(F)(F)C1 C1(NC(CC)=O)CCN(C(C2CC2c2cc(Cl)ccc2C(F)(F)F)=O)C1(C)C C#CCC(C(=O)N1CC(F)(F)C1C1CC1)NC(=O)CCC1CCCOC1 O=C(C=CSc1ccccc1)NC1(CNC(c2ccns2)=O)CC1 C1(C(=O)NOCC2(C)N=N2)(CC=C)CCN(C(=O)C(C2CCCCC2)F)C1 CCC(C(=O)NCC1CCN1C(c1sccc1SC)=O)Oc1ccccc1 C(C(O)C(=O)NC1CC(O)C1CC(=O)NCC(C)(C)CO)=CC C1(CNC(NCC(C=C)(C)C)=NCC2CCCN2CC)COC2(CCCCC2)O1 Cc1cc(C)c(C(c2nnnn2C2(C)CC2)NCCn2cc(Cl)cn2)c(C)c1Br N1(C(c2c(C)noc2)=O)CCCC(C)C1CNC(c1coc(O)n1)=O c1(C(N2C(C)C(NC(C34CCC3C4)=O)CCC2)=O)ccc([N+](=O)[O-])c2cccnc12 Cc1cc(C(=O)N(CCCNC(=O)C2=NOC(C(C)(C)C)C2)C)ncc1F C1(NC(C2N(CC)C(=O)CC2)=O)CC(O)CN(C(=O)C(N2CCN(C)CC2)C)C1 c1(C(N2CCC(CN(C(C(CCOC)C)=O)C)C2)=O)cc2c(C)cccn2n1 C(=O)(CC(F)(F)C(F)F)N1CCC(CNC(C2C(C(C)(C)C)C2)=O)C1 CC#CCC(CO)N=c1cc2c(n[nH]1)-c1ccccc1CCC2 C1(C(N)=O)COCCN(C(C2CCC=CC2NC(C2CC23CCCC3)=O)=O)C1 C(=O)(C(CC(C)C)NC(=O)Nc1c(C)cnn1C)NCC(=O)N(CC)CC C1(C(N2C3C(NC(C4CC(OC)C4)=O)C(C3)C2)=O)CC1C1CCCC1 c1(C(=O)NCC2(C(C)NC(=O)CSCC(N)=O)CC2)cnc2n1CCS2 C1(C(=O)NC(C#C)(C)C)CCN(C(=O)CN(CC)CC)C1(C)C C1(Cn2cc(C3(OC)CCCC3)nn2)CCN(C(=O)CC2NC(=O)NC2=O)CC1 C#CCCCCC(=O)NC1(CNC(C23CC2COC3(C)C)=O)CCCCC1 Cn1cc(Cl)cc1C(=O)NC1(C)CC(NC(C2(CC3CC3)CCCO2)=O)C1 c1(C(=O)NC2(CC=C)CN(C(c3c(C#C)c[nH]n3)=O)C2)ccn(CC)c(=O)c1 c1(C(=O)NC2CN(C(CCSC)=O)C(C)C2)ccc(C)c(C#N)c1 c1(CC(=O)NC2CN(C(CCSCC)=O)CC2F)ccc(S(=O)(=O)NC)s1 c1(C(=O)NC(CNC(C2CC3CC(=O)C2C3)=O)C2CC2)cc(F)cc(F)c1 c1(CC(=O)NCC(C)(C2CCC2)NC(C(CCC)O)=O)cccc(Cl)c1Cl O=C(NNC(=O)C1CC(C(=O)O)C1)C1(N2CCCS2(=O)=O)CC1 C1(CNC(CN(C)C(c2cccn2C)=O)=O)CCC1(F)F N(C1CCc2c(F)cccc21)CCNC(C1CC1C1CC1)=O Cc1c(N)ccc(C(N2CCCC(NC(C3CCc4n[nH]cc4C3)=O)C2)=O)c1C CCCC(CC(C)C)C(=O)N1CCC(NC(c2csc3cncn23)=O)C(C)(C)C1 Cc1ccc2c(c1)C(=O)N(CC(=O)NC(C1CCCO1)Cc1cccs1)C2=O C1(C(C)NC(=O)CSCc2ccccc2)CCN(C(c2ccon2)=O)C1 N1(C(c2c(C)nc(C)n2O)=O)CC2CCCC2(CNC(C2CCS(=O)(=O)C2)=O)C1 N1(C(c2ccc(C)c(O)c2)=O)CCC2CCCC12C(=O)N(CC(C)O)C CCCCC(C(=O)N(CCC)CC)NC(c1cc(O)cc(Cl)c1)=O CCC(C(=O)N(CC(O)CN(C)CCOCCOC)C)c1ccco1 Cc1cc(C)n(C(C)C(=O)NC2CC2NC(=O)CCc2ccc(CO)cc2)n1 N1(C(C2CC(C)OCC2)=O)C2CCC1CC(NC(C1CCc3nncn3C1)=O)C2 c1(C(C(=O)NCC2(NC(C(C3CCCOC3)OC)=O)CCC2)O)ccc(F)cc1 c1(C(CNC(C(CCC)O)=O)NC(c2cn[nH]c2)=O)ccc(F)cc1F c1(C(N2CCC(C(=O)OC)(C(C)C)C2)C(=O)NC(CC)C)c(C)cnn1CC c1(C(N2C(CC(=O)NCC3(OC)CCCOC3)CC2)=O)cc[nH]c2nccc1-2 c1(CNC2(C(=O)Nc3ccc(CC)c(Cl)c3)CCC2)ccc(F)c2ccccc12 c1(NC2CN(C(c3c(C)ncn3C)=O)CC2C)ncc([N+](=O)[O-])cc1F N1(C(CCC=CC)=O)CC(NC(=O)Cc2cc(Cl)ccc2O)CC12CCC2 CC1CC(NC(=O)C=Cc2ccncc2)CCN1C(=O)CC1(CS(C)(=O)=O)CC1 c1(C(=O)NC2C(NC(CS(CCOC)(=O)=O)=O)CCC2)ccc2sc(C)nc2c1 N1(C(C2CC2F)=O)CC2CCCN(C(c3ncsc3Br)=O)C2C1 C(=O)(CC(CC)C(C)(C)C)NC(N1CCC(Nc2nc(F)ccc2Cl)CC1)=O c1(NC(CCNCc2c(OC)ccnc2Cl)=O)cc2c(nc1O)CCC2 CC12CN(C(c3cc(Cl)cs3)=O)CC1(C)CN(C(C1(Br)CC1)=O)C2 CC(C)(O)C(C(=O)N1CCC12CCCC2)NC(=O)C(CO)NC(N)=O N#Cc1ccc(CN2CC(C(=O)NCCc3cc[nH]n3)CC(F)C2)c([N+](=O)[O-])c1 CC(CC(F)F)C(=O)N1CCN(C(=O)C(C)OCCN(C)C)CC1C C(=O)(C(C)(C)C(F)(F)F)NC1CC=C(C(=O)NC(C(C)(C)C)C2CC2)C1 CCC(CN(C)C)CC(=O)N1CCN(C(=O)CC2CCNC(=O)C2)CC1 c1(C(=O)NC2CC(CO)N(C(C3CC3F)=O)C2)cc(C2CC2)nc(O)c1 c1(C(N2CC(NC(c3cn[nH]c3)=O)CC(C)C2)=O)cc(C(F)(F)F)cc(Cl)c1F c1(OCC)cnc(N2CCNCC2C(N2CCCC2c2cccc(Br)c2)=O)nc1 N1(C(CCCOCC)=O)CC(C(=O)NC(C)CC2CCCCC2)CC1(C)C C(C(C)(O)CC(=O)NC1CCC1NC(=O)C=CCN(C)Cc1ccccc1)OC c1(C(N2CC(CNC(CC3C=NN(C)C3=O)=O)C2)=O)c[nH]c2nc(F)ccc12 c1(C(N2CC(C=C)C(NC(=O)C(C3(O)CCCC3)F)C2)=O)nccn2ccnc12 Cc1csc(CCC(=O)NCCCCNC(C2(CO)CCCO2)=O)n1 CC1CCCN(C(C2(C(N)=O)CC2)=O)C1CNC(=O)CC=CC(C)(C)C c1(C(=O)NC(C2CCN(C(CC3(CSC)CC3)=O)C2)C)cc2sccc2n1C C1(C(=O)NCC2C(CNC(C3CC4CCC3O4)=O)C2)CC2(C1)CC21CC1 N1(C(C(CC)N(C)C)=O)CCC2CN(C(=O)Cn3cc(C#N)cn3)CC12 c1(C(=O)NC2(CCC(N3CCC(O)CC3)=O)CCC2)c[nH]c2ccccc12 Cc1cc(CNC(=O)C(C)Cc2ccncc2)oc1C(=O)N(C1CC(CO)C1)C c1(CC)noc(C)c1C(=O)NCC1CCC(C(=O)NC2CN(C)NC2=O)CC1 c1(COC)c(C(=O)NC(C)CCCC(=O)O)sc2ccccc12 c1(C(N2CC(N(C)C(C3CCC(=O)N3C)=O)C(O)CC2)=O)[nH]nc2cnccc12 Cc1cc(C(N2CCOCC2CN(C)C(c2csc(C(N)=O)n2)=O)=O)cc(C)n1 c1(N2CC=C(C)C2)ccncc1S(=O)(=O)N1CCN(c2cc(F)cc(Br)c2)CC1 C12(NC(=O)CO)CCC(CNC(c3ccc(Cl)c(Cl)c3)=O)(CC1)OC2 C(=O)(C1=CCCCC1)NCC1N(C(C(C)SC(F)(F)F)=O)CC1 c1(CC(=O)OC)cccc(CC(=O)N(C)CCNC(=O)Cc2cnn(C)c2)c1 CCCCC(CC(=O)NC1CN(C)CC1(C)C)NC(=O)CNC(N)=O N1(C(C2C(C(=O)OC)C2)=O)CCCC(C(N2CC(n3ccnn3)C2)=O)C1C C(=O)(CCCC1CCCC1)N(C1CCC(NC(=O)CCc2ccncc2)C1)C Cc1[nH]nc(C(=O)NC2CC(CNC(C3(C#N)CC3(C)C)=O)C2)c1[N+](=O)[O-] C(C(O)C(=O)N1CCCC1CNC(=O)C(F)=CCCF)=CCCC N1(C(c2c(C)onc2)C(=O)NC2CC2)CCC2(CCOCC2)C(C(C)C)C1 C1(OCC)CCCCC1N=c1[nH]c(=NCc2ccc(Br)cc2F)[nH]c2c1CSC2 c1(C(N(C2CCCC(N(C(c3ccc(C)o3)=O)C)C2)C)=O)cc(Cl)cnc1C Cc1nc(C(N2CCC(OCC(=O)N(C)CCc3cccs3)C2)=O)cs1 CN1CCC(C)(C(=O)NC2CC(CNC(c3ccc(CO)o3)=O)C2)C1=O c1(C(C(=O)NC(Cc2nnc(C)o2)=O)O)cccc2c1OCC2.C1CC1 C1(NC(C(CC=C)NC(C)=O)=O)(CNC(C2CCC3CC23)=O)CCCCC1 N1(Cc2n(CC)ncn2)CCC2(CCN(C(=O)Cc3cn4c(n3)CCCC4)C2)C1 C1(C(=O)NC(CN(C(=O)C=Cc2ccc(OC)cn2)CC)C)CCCCNC1=O C(C(C)(CC(C)C)NC(C1CC2CCC(C1)O2)=O)NC(C1(CC)COC1)=O c1(N(CCC)C(C2CC2)C2CC2)nc(-c2ccccc2)ncc1F C1(C2CC2)(CNC(CCc2cn(C)nn2)=O)CCN(C(=O)C2=CCCSC2)C1 S(=O)(=O)(c1ccc(N2CCC3(CC2)CC3)c(C#N)c1)N(CC(COC)C)C1CC1 c1(SC)cccc(F)c1C(=O)NCC(C)NC(C1(O)CCC(C(F)(F)F)CC1)=O C1(C)(CNC(C2(C(F)F)CC(=C)C2)=O)CCCN(C(c2cnc(N)s2)=O)C1 N1(C(CCCNC(=O)OCC)=O)CCC(C)(CCNC(C2(C)CCCC2)=O)C1 N(C(=NCCN1CCOC(C)C1)NC(C1CCOC1)C)Cc1scc(C)n1 N1(C(C2(C)C(C)(C)C2)=O)CC2CC1C2NC(=O)CCCn1ccccc1=O CCCC(C#N)C(=O)N(C(C)CNC(=O)CSc1ccccc1OC)C C=CCC(CC=C)C(=O)NCCOCCN(c1cc(OC)cc(F)c1)C C(C(C)(C(=O)NCC1CCCC1(C)CO)NC(=O)COc1cnn(C)c1)SC C1(NC(C#CC(C)C)=O)CC(C)CN(C(c2cnn(C(C)C)c2F)=O)C1 C1(C2CCC2)(C(=O)NC2CC3(C(NC(C4CCN(OC)CC4)=O)C3)C2)CC1(F)F c1(NC(C)=O)cnccc1C(=O)NCCCC(C)(C)NC(=O)CSC1CCCO1 C1(F)(CNC(COCCOCC#C)=O)CCC(CNC(C2CCS2(=O)=O)=O)C1 Nc1c(C(=O)NC23CC(CNC(=O)Cc4nc[nH]n4)(C2)C3)cc(Cl)cc1Cl N1(C(=O)OC)CCCCC1C(N1CCN(CC)CC1)=O.C12CN(CCO1)C2=O N1(C(c2c(C)ccs2)=O)CC(C2(NC(=O)CCCN3CCCCC3)CC2)C1 Cc1nc(C(C)C)oc1C(=O)NC1CCCCC1NC(c1ccncc1F)=O C1(COC)(CNC(=O)C=C(C)C)CCCN1C(C1CCCO1)=O N1(C(CCC=CC)=O)CCCC2C1CCN2C(=O)C(c1ccncc1C)C c1(C(N(C2CCN(C(c3nc(OC)c(C)s3)=O)C2)CC)=O)c(C)noc1C1CC1 CCC(C)(F)C(=O)NCC(C)(CC)NC(c1cnc(=N)[nH]c1)=O Cc1cc(Cl)cc(NC(C2CC3CC3N2Cc2ccn(CCF)n2)=O)c1I Cc1cc(F)cc(C(=O)NCC2CCN(C(=O)C(N3CCSCC3)C)CC2)c1C C#CCC(C)(CC)C(=O)NCC12CC(CN1C(=O)Cn1cc(C(=O)OC)cn1)C2 C1(C(=O)NCc2noc(C)n2)(NC(C(C)OCC=C)=O)CC(O)C1 Cn1c(C(=O)NC2C3CC2N(C(=O)CN2CCCC2)C3)cc2cc(Cl)ccc12 C(=O)(CC1=CCCCC1)NC1(C)CN(C(c2ccc(C(F)F)c(F)c2)=O)C1 N1(C(C(CSC)C)=O)CCC(CNC(c2cnc(Cl)cc2N)=O)C(O)C1 CC12CC(NC(=O)NCC3(CO)CC34CCC4)C(CO1)C2 c1(C(=O)NC2(C)CCN(C(=O)CC3CC3(Cl)Cl)C2)cc2ccncc2s1 N1(Cc2ccccc2)CCCC1CC(=O)NC1C(OC(C)C)COC1 c1(CNC(C(=O)NC(c2cccnc2)C)=O)cccc(N2CCCCC2)c1 C(=O)(CC(CCCC)NC(C1(CCC)CC1)=O)N(CC#C)CCF C(CN=c1[nH]c(=NCc2cc(C)cc(Br)c2)[nH]c2c1SCC2)OCC=C c1(OC(C)CNC(=O)CCOCC(=O)Nc2ccccc2)ccc(Cl)cc1 C1(CNC(=O)CCc2ccoc2)CCN(C(=O)Cc2cccc(F)c2O)CC1O c1(C(=O)NC(CCOC)CNC(c2ccn(C)n2)=O)ccc(C(=O)OC)cc1F N(C(=NCC(=C)C)N1CCCCCCCCC1)CC1C(C=C)OCC1 c1(CN(C)C)cc(C(=O)NCCOC2CCN(C(=O)CCCC3CC3)C2)ccn1 c1(C(=O)NCC2N(C(Cc3c(OC)ccnc3)=O)CC2)cc2c[nH]nc2s1 N1(C(c2ccon2)=O)CC2(CCN(C(c3cc4c[nH]cnc-4n3)=O)CC2)C1 C(=O)(CC(F)(F)C(F)(F)F)NC1CCCN(C(C(c2ccccc2F)C)=O)C1 C1(CNC(COCC(=C)C)=O)CC(F)CN1C(=O)CC1CC(C)C1 CCCCCS(=O)(=O)CC(=O)NC1(C)CCN(Cc2nnc(C3CC3)o2)CC1 Cc1ccc2c(=NC3CCC4CCCC4C3)[nH]c(=NCC3(CSC)CC3)[nH]c2c1 c1(CC)c(C(N2CC(C)(NC(c3ccnn3CC)=O)C2)=O)cnc2ncnn12 c1(-c2c(C)c(F)c(F)cc2)ccc2nc(C(=O)Nc3cccnc3CO)sc2c1 N1(C(CNC(C)=O)=O)CCC(NC(=O)C=C2CCC(C)C2)CC(O)C1 C1(CNC(C(N2C(C(=O)OC)CC2)C)=O)CC2C=CC1O2 C(=O)(CC(=O)NC1CC1CNC(c1cn(CCC(C)C)nn1)=O)OCC c1(OCCC(=O)N(C)CC2N(C(C(C)=C(C)C)=O)CCCC2)ccc(F)cc1Cl c1(OC)ccc2c(c1)CCCC(NC(C1CC(CN)C1)=O)C2 C(=O)(C1SCCc2sccc21)NCC1N(C(c2c(CCC)n(C)nn2)=O)CC1 CC1(C)CC(C(=O)N(C2CCCC2)CCNC(C2(C#N)CC2C(F)(F)F)=O)=NO1 C1(CC(=O)NCC(CC)NC(C23CCCN2CCC3)=O)CC(C)(C)C(=O)N1 N1(C(C=CC)=O)CC2(C1)OC1(CO)CC2(NC(=O)Cc2csc(Cl)c2)C1 Cc1c(CC(=O)N(C(C)CCNC(=O)CC2CC2(C)C)C)oc2ccccc12 CCC(CC)(C(=O)N1CC2CC(C(=O)NOCc3nc[nH]n3)CC2C1)C(C)C C=CCN=C(NCc1ccc(C#N)cc1)NCc1cn(C(C)C)c(=O)nc1O c1(C(=O)NC(C(C)NC(c2ccc(C)cc2O)=O)C)ccn2c(C)cnc2c1 CN1C(=O)CCCC1C(N1CC(CC(=O)NCC(CO)C2CC2)C2(CC2)C1)=O O=C(C(O)CC1CC1)NCCCC1CCCN1C(=O)Cc1cnco1 N1(C(C23CC(OC)C2C3)=O)CCC(C(=O)OC)(NC(=O)CCC(C)(C)F)CC1 N1(c2n(CCOC)c(-c3ccc(C)c(C)n3)nn2)CCOC2COCC12 N1(C(CCC#C)=O)CC(NC(=O)Cc2csc(SCCN(C)C)n2)CC(O)C1 Cc1cc(C(N2CCC(C(C)NC(=O)CCCc3cncs3)C2)=O)nc(O)c1 Cn1nc([N+](=O)[O-])cc1C(N1CCCC1C(C)(C)NC(C1CC2C=CC1O2)=O)=O C1(CNC(C=COCC)=O)(CNC(C2(c3cccs3)CC2)=O)CC12CCC2 c1(N2CCN(C3CC(CC(=O)OCC)OCC3)CC2)ccccc1S(C)(=O)=O N1(C(CC2C(C)C2)=O)CCN(C(C2CN3CCN2C(C)C3)=O)C2(CCC2)C1 C1(OC)CC2(C1)CC(N=c1ccnc(NCC(CO)C(F)(F)F)[nH]1)C2 C(O)CC(C)N=c1nc(-c2ccccc2)[nH]c(=NCC(C)(C)CS(N)(=O)=O)[nH]1 c1(C(NNC(=O)C2N(C(C)C)CCC2)=O)cn(C)c2c(cnn2C)c1=O c1(CC(=O)NCC(CNC(C(=O)NCC)=O)(C)O)ccc(F)cc1C c1(C(=O)NC2CC(NC(CC3CCC(C)O3)=O)C(O)C2)n[nH]c2c1CCC2 N1(C(C(CCN(C)C)NC(C(C)CC2CCCC2)=O)=O)CCCC2C(O)CC12 c1(C(=O)NCC2CCCN2CCN2CCNC2=O)ccnc(-c2ccccc2)n1 c1(C(N(C(CNC(C2N(CC#C)CCC2)=O)C)C)=O)ncnc2sccc12 N1(C(C2(C)CN(C(C(n3c(C)ncc3)C)=O)C2)=O)CCC2(C=CCO2)CC1 c1(NC(c2cccc(C3CC3)c2)c2n(CC(=C)C)nnn2)ccc(Br)cc1Cl c1(C(N2CC(CNC(C(C)n3ccnn3)=O)OCCC2)=O)cc(C#N)ccc1F C1S(=O)(=O)N2CC(N=C3NC4=C(C(=NCC1CSC)N3)COC4)CC2 CC#CCC(C(=O)NCC1NC(=O)NC1=O)NC(=O)Cc1ccc(C#N)cc1 C12CCCCN1C2.C1(C(=O)NCCS(=O)(=O)N(C)C)C(F)(F)C12CC2 c1(C(=O)NC(C2CCCCN2C(=O)CCOCC2CC2)C)cncc2sccc12 N1(C(=O)CC2CC=CC2)CCC2CCCN(C(=O)CNC(C3CCOCC3)=O)C2C1 C#CCC(C)(C(=O)N1CCOC(CF)C1)NC(=O)C(n1nccc1C)C Cc1nn(C)c(C)c1CC(N1CC(CCNC(=O)C=Cc2cnn(C)c2C)C1)=O c1(C(C(=O)NC2CC2)N(C(C)CC(N)=O)CC#N)c(F)cccc1Br CN1CCN(C(=O)C=Cc2cnn(C)c2)C(C(=O)NCc2cn(C)cn2)C1 N1(C(C(C)OCCOC)=O)CC2(CC(NC(c3cc(C(N)=O)no3)=O)C2)C1 C1(C(=O)NC2(CC(=O)NCc3cn(C)nc3)CCC2)CN2CCC1C2 c1(C(=O)NCCC(C(C)C)N(C)C)nc(Cl)cn2ccnc12 Cc1csc(Cl)c1C(N1CC(NC(=O)C(C(C)C)c2ccn(C)n2)C(O)C1)=O C(=O)(C(C)(O)C(F)(F)F)N(C(C)C)CCNC(C1CCN(C2CC2)C1=O)=O N1(C(C(C(C)O)C)=O)C2CCC1CC(NC(C1CC3C(C1)C3(F)F)=O)C2 N1(C(=O)NCc2c(C(=O)OCC)cco2)CC=CCC12CCCC2 c1(C(N2CCOC(C3CC(F)(F)C3)C2)C(=O)NCCCOC)ccc(C#N)s1 C(=O)(CCCCC(=O)N1CCC(CNC(=O)CC2(C)CCCO2)C1(C)C)OC c1(C(=O)NCC2C(NC(c3occ(C)c3)=O)CCC2)sc(F)cc1Br C1(CNC(C(C2CCOCC2)C)=O)CC2CCC1N2C(=O)C=Cc1ccoc1 c1(C(=O)OC(C)C(N2CCC(C(N)=O)C(C)(C)C2)=O)ccc(F)c(F)c1F C=CCCCC(C)(C)CNC(c1cn(CCNC(C2(CC(C)=O)CC2)=O)nn1)=O C(CN=c1[nH]c2c(c(=NC3CCOC(C)C3)[nH]1)COC2)OC(C)C C1(C(N(CC2=CCCOC2)C)=O)CN(C(C2(C)SCCCS2)=O)CC1(C)C N1(C(=O)Cc2ccon2)CC2CC(C1)N(C(=O)C(F)CC1CC1)C2 CC1CN(C(c2ccoc2C2CC2)=O)CC1CNC(=O)COCC(F)(F)F c1(OC)oc(C)nc1C(=O)NCC1CCC(NC(c2cc(CCCO)on2)=O)C1 C1(CNC(C(C(CC)O)C)=O)CN(C(c2[nH]nnc2C)=O)CCC12CCOCC2 Cc1cc(C#N)cnc1C(N1CC(NC(C2CCCC(=O)N2)=O)CC1C)=O C1(OCC)CCN(N2CCC(N3CCCS3(=O)=O)C2C)C1C C(=O)(C1=COCCO1)N1CCN(c2c(NC(CCOC)=O)cccn2)CC1 C1(Cc2cn(C(N(CCOC)CC)=O)nc2)Cc2ccccc2C1O S(=O)(=O)(c1ccccc1)NCCC(=O)NCC(c1ccc(F)cc1)C(C)C Cc1ccc(C(=O)C(=O)NCC2CC(NC(C3CC3c3cccc(F)c3)=O)C2)cc1 N1(C(C(C)N(C(C(C)OCCOC)=O)C)=O)CCCC(C)(C)C1C Cc1cc(F)c(CN2CC3CC3(C(=O)NCCOc3ccccc3)C2)cc1Br C12(CNC(CC(=O)NCC#C)=O)CCCC1N(C(c1ncccc1Cl)=O)CCC2 N1(Cc2ccc(-c3cn(C)nc3)cn2)CC2(CC2C#N)C1 c1(C(=O)NC2C(NC(C3(C#C)CCC3)=O)CC2)ccc(F)c(OC(F)(F)F)c1 CC1CCC(C)(C=CC(=O)NCC2(O)CN(C(=O)Cc3cccnc3N)C2)C1(C)C C(C(C)(C)CC(=O)NC1CC(C(=O)NCC2C=CCCC2)C12CCC2)OC C(=O)(C(C(C)(C)C)OC)NCCC1(O)CCN(C(c2c(OCC)nccc2)=O)C1 N1(C(C2C(OC)CC2)=O)CCN(C)CC1CNC(=O)COc1c(F)cccc1F c1(C(=O)NCCN(C(CC2COCC(C)O2)=O)CC2CC2)ccc(Cl)c(F)c1F c1(NC(C(CC)(C)CNC(=O)CC2CNC(=O)O2)=O)ccc2nc[nH]c2c1 C12(C(N3C(C)CC(NC(=O)CCOCCN(C)C)C3)=O)CCC(C(F)(F)F)(CC1)C2 c1(C(N(C(C)CNC(c2cncc(CO)c2)=O)C)=O)cnn2cccnc12 c1(C(=O)OCC)cccnc1NC1CCN(C(=O)Cn2ccc(C)n2)C1CC c1(CC)nc(C)[nH]c1C(=O)NCCC1CCN(C(c2cc(C3CC3)no2)=O)C1 C(C)(N=c1[nH]c(=N)[nH]c(=NCCc2ccc(Cl)cc2C)[nH]1)c1ncc(C)cn1 CN1CCN(C(=O)C(F)C2CCC2)C(C(=O)Nc2ccc(OC(F)F)nc2)C1 c1(C(C)C)ccc(C(=O)N(C)CC2CCCN(C(=O)COCC3CC3)C2)cc1F C(=O)(C(C(=O)NCC=CCC(=O)N(C1CCC2CC12)C)OC)OC C(=O)(CCC(C)(C)NC(=O)C(F)CC1CCOC1)NC1C(C=C)COC1 N1(C(C(CC)=CC)=O)CCC(CCNC(=O)CCC2CCCC2)C(F)(F)CC1 N1(C(C(C)(F)c2ccccc2)=O)CCC2(C1)CN(C(c1ccnc(O)c1F)=O)C2 CCCS(=O)(=O)C(C)C(=O)N(CC(C)NC(=O)Cc1cccnc1F)C Cn1ncc(C(=O)NC(CNC(=O)COc2ccc(C(F)(F)F)cc2)CO)c1Cl C(c1cccc(Br)c1)=CC(=O)NC1COCCN(C(=O)C(=O)NC2CC2)C1 CC1CCCCC1C(N1CCCC1CC(N1CSCCSC1)=O)=O C1(O)(C(C)NC(c2cc(C(N)=O)no2)=O)CCN(C(c2csc(CO)n2)=O)C1 C1(C(=O)NCCN(C(C23CC(O)C2C3)=O)CC2CC2)C2CCC1(c1cscn1)C2 c1(C(N(CCCNC(c2cc(=O)cc(Cl)[nH]2)=O)C)=O)ccc2c(=O)ccoc2c1 CC1CCN(C(C2CCCCC(=O)C2)=O)CCN1C(c1cnccn1)=O c1(N(C(C(CC(C)C)O)=O)C(c2ccc(F)cc2)C)ncnc2cccnc12 N1(C(c2c(C)nco2)=O)CC(NC(c2ccc(COc3ccccc3)o2)=O)C(F)C1 CC1(C(=O)NCC2CC(O)CN2C(=O)CCOCC2CCC2)C=CCCC1 c1(C(=O)OCC)c[nH]c(=NCC2(C)CCCN(C(c3sccc3SC)=O)C2)cn1 N1(C(C(CC(=O)OC)C)=O)CCC2CN(C(c3cn(CC(N)=O)nn3)=O)C2C1 CC(=O)CCCC(=O)N1CCCC1CN(C)C(C1CCCCNC1=O)=O c1(CC)ncc(C(N2CC(C(=O)NC(CO)C(N)=O)(SC)C2)=O)s1 C1(C(=O)NC2CCC2NC(C2(O)CCCC2)=O)Cc2nccn2C1 c1(C(N2C(CN(C)C(c3scnc3Cl)=O)COCC2)=O)ccc(F)c(CO)c1 C1(NC(Cc2cc(C)on2)=O)CN(CC(N2CCCCC2)=O)CCC1C C1(N=[N+]=[N-])(C(=O)NCC(C)CC(C)O)CCN(C(C2CN3CCN2CC3)=O)C1 c1(C(=O)NC2C(CNC(CCc3nnc(C)o3)=O)C2)ccc2occc2c1 N1(C(C(CC)n2ccnc2)=O)CCC(C(C)CNC(=O)Cc2ccoc2)CC1 N1(CC(N2C(CCNC(=O)C=CC3CCCC3)CCCC2)=O)CCS(=O)(=O)CC1 C1(C(N2CCC(C(=O)Nc3ccc(Cl)cc3)(CF)C2)=O)COc2ccccc2O1 N1(C(C=C(C)Cl)=O)CCC2CN(C(=O)C(CO)c3ccccc3)CC2C1 N1(CCC(=O)Nc2cc(OC)cc(OC)c2)CC2CC(F)CC2C1 Brc1ccc2occc2c1N1CCC(C2CCCC2)C1 N1(C(=O)CC2CCC=CCC2)CCN(C(=O)CCCC(F)(F)F)C2CCCCC12 C1(CNC(c2cc[nH]c2)=O)(CO)CCCN(C(C23CCCCC2C3)=O)C1 N1(C(c2c(C)coc2)=O)CCC(C2CC(NC(C3CCC=CCCC3)=O)C2)CC1 n1(CCC(N2CC(NC(CC=CCC)=O)C(C)C2)=O)cc(C#N)c(O)nc1=O c1(NC(C(C)NC2CCCC3(CC2)CC3)=O)ccc(S(N)(=O)=O)cc1 C1(NC(C2C(C(N)=O)C2)=O)COC2(C1)CN(C(c1c[nH]c(=S)cn1)=O)C2 N1(C(c2c(C)nco2)=O)CC(NC(c2ccn(-c3ccncc3)n2)=O)CC1C NS(=O)(=O)c1ccc(CN(C2CCC(F)(F)C2)C(=O)Nc2cc(F)cc(F)c2)s1 Cn1ccn2ncc(CNC(C3CC4(CC4)CN3C(=O)OC(C)(C)C)=O)c12 C12(NCC(c3ccc(OC(C)C)cc3)O)CNCC1CCO2 c1(C(=O)NCC2N(C(C=C3CCC(C)C3)=O)CC2)cnn2c1CCCC2 C1(C(N2CCN(C(c3cc(SC)c(C)o3)=O)CC2)=O)CCC=CCCC1 c1(C(N2C(CCOC)CN(C(=O)CC3CC3(C)C)CC2)=O)cc(S(C)(=O)=O)co1 c1(C(=O)NCC(C)(C2CC2)NC(c2c(OC)nn(C)c2)=O)c(Cl)ccc(C)c1N N1(C(C2CC(=C)C2)=O)CCCC2(NC(=O)CC3CCC34CCC4)CCCC12 Cc1cc(=O)ccn1CC(N1CCC(F)C(NC(=O)C(C)c2ccsc2)C1)=O C(=O)(C#CC1CCCC1)NCC(C(N1CCCC(C)(C)C1)=O)C1(O)CCC1 C(=O)(C(CCC(N)=O)NC(C1(CF)CC1)=O)NC(CCN(C)C)C(C)(C)C N1(C(CSc2ccc(C)cc2)=O)C(C(N2CCCC2CF)=O)C2CC(O)C1C2 c1(NC(C2CCCN2C(=O)Cn2cncn2)=O)ccc(O)c(CO)c1 N1(C(C=C(CC)CC)=O)CCCCC1CNC(C1(CCS(N)(=O)=O)CCC1)=O.CN1CC1 c1(C(=O)NCC2(C)CCC(NC(c3sccc3F)=O)C2)ccc2nc[nH]c2c1 C1(OC)CN(C(c2cc(Cl)cc3c2OCC3)=O)CC2(CCC2)C1 c1(CC)ccoc1C(=O)NCCNC1COC(C)C1 C1(NC(c2c(OC)cc(Cl)cc2)=O)CC2CN(C(=O)CC3CC3C)CC2C1 c1(C(N2CCC(NC(CCC3CC(OC)C3)=O)C2C)=O)cc([N+](=O)[O-])n[nH]1 c1(C(N2CC(NC(C(C)NS(C)(=O)=O)=O)C(F)CC2)=O)ccc2ccn(C)c2c1 c1(OC)ccc(CCC(=O)NC(C)(C)CNC(c2sc(=N)[nH]c2C)=O)cc1 N1(C(c2cnc(OC)s2)=O)CC(C2(NC(=O)Cc3ccncc3Cl)CC2)C1 C1(NC(c2n(CCC)nnn2)C2CCSCC2)CCc2cnc(C)n2C1 Nc1ccc(C(=O)NC2(CCCNC(C3Cc4nccn4C3)=O)CC2)cc1F N1(C(c2c(COC)scc2)=O)CC2CCC2(CCNC(c2ccnc(O)c2)=O)C1 C1(C(=O)NC(CC(C)C)CNC(c2cc(Cl)sc2Cl)=O)CCc2nc(O)[nH]c2C1 C1(CNCc2n(CCCC)nnn2)CNC(=O)C(C)(C)C1 C1(C(N2CC(NC(C(C)=C3CCC3)=O)C2)=O)CC(c2cccnc2)=NO1 C1(C)(CNC(c2c(OC)nn(C)c2)=O)CCCN(C(C2CC(F)C(=O)N2C)=O)C1 Cc1nc(NC(=O)OC(C)(C)C)co1.C12COCC1n1cc(nn1)-c1csc2n1 C(=O)(C1=CCCCCC1)N1CC(CNC(c2cc(CC)nnc2C)=O)OCCC1 C1(CC(=O)NCCCN(C(C)C)C(c2ccnn2CC2CCC2)=O)CNC(=O)O1 Cc1c(F)ccc(C(=O)NC2CCCCC2NC(c2ccc[nH]2)=O)c1C#N C(C)(C)(C(=O)NC1CC(NC(C2CCC(C(=O)OCC)C2)=O)C1)SC.C(C)(C)C C(=O)(C(CC(C)C)NC(c1ncncc1OC)=O)NCC(CCOC)O c1(C(=O)NCC(C)N(C(=O)CC2CSCCS2)C)nc(=N)[nH]c2ccccc12 C1(C(C)(O)CNC(c2ccncc2)=O)CCN(C(c2coc(C3CC3)n2)=O)CC1 C1(C(=O)NC(C)CN2CCC(O)CC2)(NC(c2ccco2)=O)CCCCC1 C1(C(=O)NC2CN(C(C3N(CC)CC3)=O)C(C)CC2)C2CCC3(COC(=O)C13)O2 C(=O)(C(C)(C#N)CC)NCC1CCN(C(c2c(OCC=C)cccn2)=O)C1 C(C)(CC1CCC1)(CN=c1cc(NCc2sc(C)cc2Br)nc(C)[nH]1)OC C(=O)(C(C(C1CC1)OC)N(CCCOC(C)CC)C)NCC Cc1cccnc1C(=O)NC1C=CCN(C(C2CN(C(N)=O)C2)=O)C1 N1(C(c2c(C)ncs2)=O)CCN(Cc2ccc(CBr)cc2)CC1C#N N1(C(c2c(CC)nccc2)=O)CC(C(=O)NCc2ccc(C)nn2)CC(C)(C)C1 c1(NC(c2cc(C)ncc2C)=O)cc(C)n(C)c(=O)c1 C1(Cn2cc(C(N3CCOCC3)C)nn2)CN2CCCC2CO1 c1(CC(=O)NCC2CC(NC(C(CC)N(C)C)=O)C2)cc2ccccc2nc1O c1(C(=O)NCC2N(C(=O)C=Cc3cn[nH]c3)CCN(C)C2)nccn2nccc12 C1(C(=O)NC2CCC(NC(C3(C)CCC3)=O)C2)Cc2ccccc2C1(C)C C(CCCCO)N(C(C)C)C(c1ccn(CCNC(=O)C=C2CCOCC2)c1)=O C1(O)(CCNC(=O)Cn2cccn2)CN(C(=O)C(C2CCCCC2)O)C1 C1(CC(=O)NCC(C)(C)NC(=O)CC(c2cccc(F)c2)O)CCC12CCC2 C1(NC(CC=CCC)=O)C2CCC1N(C(C1(OCC)CCCC1)=O)C2 n1(CC)c(C(=O)NC2(C)CC(NC(C3CCC(C)C3)=O)C2)cnc1O N1(C(c2c(OC)noc2C)=O)CCC2(C1)CN(C(C1CCC3(CC3)C1)=O)CCO2 c1(NC(c2cc(CC)n(C)n2)c2nnnn2CC)ccc(C(N)=O)c(C)c1 c1(C(c2nnnn2CCOCC)NCC(=C)CC)cccc(F)n1 c1(C(=O)NC2CCCCN(C(CC3C(CC)C3)=O)C2)c(C)cc(C)nc1O CON1CCC(C(=O)NCCCCCNC(C2(S(C)(=O)=O)CC2)=O)CC1 C1(CC(=O)NC(C(=O)NCC(=O)NCC(C)C)CC2CCCC2)CCCCO1 C12(C(N3C(COC)CCC3)=O)CC(C)(CN1C(=O)C(C1CCCCC1)C)C2 C1(COC)(NC(=O)CSCC(C)C)CCN(C(=O)COc2ccon2)CC1 C#CCC(C)(C)C(=O)N1CCN(CCNC(=O)CC(CC)c2ccccc2)CC1 N1(C(C(CC)C#N)=O)CCC(O)(CCNC(=O)C(COC)OC)CC1 C1(NC(C2C(C)=C2)=O)CN(C(c2cnn(CC(F)F)c2C)=O)CC2(CCC2)C1 C1(CNC(c2cn(CCC)nc2)=O)CC(F)(F)CN1C(=O)C(F)CC(C)C c1(CC)[nH]nc(Cl)c1C(N1CCCC1CCNC(C1CC1c1cccnc1)=O)=O N1(C(c2cc(C)sc2)=O)CCC(C(C)C(=O)N(C)Cc2nccn2C)CC1 c1(C(C)(C)C)nnc(CNC(=O)NCc2n[nH]c(=N)s2)s1 C(=O)(C1=C(F)CN(C(=O)CC2COC(=O)C2)CC1)NC1(C)CSC1 C(CCC1CC1)(C(=O)NCC(O)C1(Cl)CC1)NC(CCCOCCC)=O N1(C(c2cn(CCC)nc2)=O)CCC(NC(=O)C(N2CCCC(C)C2)=O)C(C)C1 C1(C(=O)NC2CC(CNC(C(C)P(C)(C)=O)=O)C2)CCN(S(N)(=O)=O)CC1 c1(C(c2nnnn2CCCC2CC2)NC2C(OC)CN=C2)cccc([N+](=O)[O-])c1C CN1CCOC(C(N2CCCC(O)(CNC(c3nn[nH]c3Cl)=O)C2)=O)C1=O C(=O)(C1=CCCCC1)NC(C(=O)NCC(C1CCC1)OCC)(C)CO CC#CCCCC(C)(c1nnnn1CCCC1CC1)NC(COC)CC(=O)OC C1(C(=O)NCC2C(C(N(C)CCn3cccn3)=O)C2)CC2CCC2C1 C1(C(=O)NOCCOC(C)C)(CC=C)CCN(C(=O)CC(C)COC)C1.OC CCC(C(=O)N(C1(C(=O)NC2CC(C(=O)OC)C2)CCC1)C1CC1)C(C)(C)CC CC1(C)OCCOC1C(N1CC(F)CC1CNC(C1CCSCC1)=O)=O C(=O)(CC(F)(F)F)N1CC(CC=C)(C(=O)NCCCc2nc[nH]n2)C1 c1(CNC(C(C)OCCOC)=O)ccc(C(N2CC(N(C)C)C2)=O)cc1 c1(C(=O)NC(CC(C)NC(c2cccc(NCC#C)c2)=O)C)ccc(O)cc1F c1(NC(C2(NC(c3c(C)cccc3)=O)CC2)=O)ccc(Br)nc1Br C12(C(=O)NC(CC(C)NC(c3cc[nH]c3)=O)C)CC3CC(C1)CC(O)(C3)C2 N1(C(C=CC(C)C)=O)CC(N(C(=O)C=CC=C(Cl)Cl)C2CC2)Cc2ccccc21 Cc1cc(Cl)c(C(=O)N(CC(O)CNC(=O)C=CC2CCOC2)C)cc1[N+](=O)[O-] Cc1cc(=O)n(C)nc1C(N1CCC(C2(NC(c3cccc[n+]3[O-])=O)CC2)C1)=O CC(=O)CCCC(=O)NCC1CCN1C(c1cccc(SCC#N)c1)=O C#Cc1ccc(CCC(=O)NC2CCCCC2NC(C2CCCN2CC)=O)cc1 C12(CNC(C(C)OC)=O)COCCN1CCN(C(c1cc(C)cc(F)c1N)=O)C2 c1(C(N2C(C=O)CC2)=O)csc(S(N)(=O)=O)c1.c1(NCC)scnc1C(=O)OC c1(C(C)NC(c2cnc[nH]2)=O)ccc2c(c1)CN(C(C1C(C)(C)C1(C)C)=O)C2 c1(-c2cn(C3C(C)(C)CCC3)nn2)ccc(Cl)c(I)c1 N1(C(C(C=C)c2ccccc2)=O)CCCC(C2CN(C(=O)C(C#N)CC)C2)C1 C1(C(=O)NCC(COCC)O)(NC(C)=O)CCNC1=O C=C(C)CC(C(=O)N1CC(O)(C(F)(F)F)C1)NC(=O)C(C)c1cccs1 N1(C(C(C(C)O)C)=O)CCCC(C2CN(C(=O)CC3CC4CCC3C4)C2)C1 C1(C)(NC(CCCc2nc(C)sc2)=O)CCN(C(C2CC2c2cccnc2)=O)C1 C1(C(=O)NCCC2(O)CCC2)CCCN(C(C2COCOC2)=O)CC1 CC(C(CO)NC(c1cnc(-c2ccccc2)s1)=O)NC(C1CC(C)(C)O1)=O c1(COCC(=O)N(C)Cc2ccc(C(=O)O)o2)cn(CC2CC2(F)F)nn1 N1(C(CCCC=C)=O)CCN(C(=O)CCc2nccn2CC)C2CCCC12 C(C(C(C)C)NC(=O)CNc1ccncc1)(c1ccccc1)NC(C=CC)=O C1(NC(C=C(C)C(F)F)=O)CCOC12CCN(C(c1ccc(CO)cn1)=O)CC2 c1(C(N(C(c2ccccc2)(C)C)C)=O)ccc(CNC(c2ccco2)=O)cc1 C1(C(=O)NC2CC(C)N(C(C3(C)CC(F)(F)C3)=O)CC2)CCc2nnnn2CC1 C1(C(=O)NC2CCN(C(C=CCCC(C)C)=O)C2)C2CC3C(C2)C13 c1(OC)ccc(NC(=O)C(c2cnn[nH]2)N(C2(CCO)CC2)C)cc1 Cc1cc(C(N2CCOC(C(F)F)CC2)=O)cc(C)c1.C(=O)(C(C)C)N CC1CN(C(=O)CCCCN(C)C)CC(C(N2CCCC2C(O)CO)=O)O1 C(=O)(C(C)(C)C(C)(F)F)N1C(CN(C(=O)C(C#N)C(C)(C)C)C)CCC1 N1(C(C(c2ccccc2F)OC)=O)CCC(CO)(NC(c2cnoc2C)=O)CC1 C1(C(=O)NC2C(OC)C(O)C2)(CC)CCCN(C(c2n[nH]cc2Cl)=O)C1 N1(C(C(=O)NC(c2ccc(C(C)C)cc2)C)=O)CCc2ncccc2C1C c1(CNC(C(CC)C)=O)ccc(CNC(C2C3CC(=O)CC23)=O)cc1 c1(C(N2CC(O)(CNC(c3nc(CCC)sc3)=O)C2)=O)cc(C2CC2)nc(O)c1 C(CC1CCC1)(C(=O)NCC1=CCCC1)NC(=O)Cn1cnnn1 C(=O)(C(C)(C)CCCF)N1CCCC(CC=C)(NC(=O)C(C)OC)C1 c1(C(=O)NCC(CC(=O)OCC)O)cc2c(ccn2C)[nH]1 c1(OCC(CN2CCC(c3onc(CCC(C)C)n3)C2)O)ccc(Cl)cc1Cl C1(NC(Cc2c(C)ocn2)=O)CCC(F)(CNC(=O)C(C)(O)C2CCOCC2)C1 C1(C(=O)NC(C)CCF)CC2CN(C(c3ccc(F)cc3)=O)CC2C1 C1(O)(C(C)C)CCCN(CCC2(CN)CNC2)C1 c1(NC(C(C(C)C)SC)=O)cccc2c(-c3cn(C)nc3C(F)(F)F)cccc12 N1(C(CN(C(C)=O)C)=O)CCOCC1CCNC(c1cc(O)n(C)n1)=O C#CCS(=O)(=O)CCNC(=O)C(=O)Nc1cccc(N(C)C(C)=O)c1 N1(C(CC=CCC)=O)CCN(C(C2(F)CCOC2)=O)CC1c1ccc(F)c(F)c1 C1(C(C(=O)NCCCSC)N(C)C(c2ccccc2Br)C)CC2CCC1O2 N1(C(c2cccc(N(C)C)n2)=O)CCc2[nH]nc(C(=O)NCC=C(Cl)Cl)c2C1 CC(C)(C)C(=O)NCCC(=O)NCCCOCCNC(=O)C=C1CC1 C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1(C)CCCN(C(=O)CC2CC=CCC2)C1 Cc1ncc(C=CC(=O)N(CCCNC(C23CC(C)C2C3)=O)C(C)C)s1 CC(C)C(C(=O)N1CC2CC1(C(N1CC(c3nncs3)C1)=O)C2)N(C)C Cc1ncc(Cl)cc1CC(=O)NC1CN(C(c2cnc3sccn23)=O)CC12CC2 CCCC(CO)NC(=O)C(C1CCN(C(=O)C=Cc2ccc[nH]2)C1)C c1(N(CC)CC2(CO)CCCC2)ccncc1S(=O)(=O)N(C)CC.C(CC#N)N c1(C(N2CCC(NC(C=CSC)=O)(CO)C2)=O)cc(S(C)(=O)=O)oc1C Cc1cn(-c2ccccc2F)nc1C(=O)NC(C)C(C)S(C)=O N1(C(C(C=C)(C)O)=O)CC2(COC(CNC(c3cnc(C)nc3C)=O)C2)C1 Cc1cccc(CC(=O)NCC23CCC(CN2C(C2CC2(Cl)Cl)=O)C3)c1F c1(OC)cc(C(=O)NC2CC(CNC(=O)Cn3nnnc3C)C2)ccc1OC C1(C(=O)NC2C(CNC(CCc3nc(C)sc3)=O)C2)CC1C1CCC1 N1(CCNC(C2C(C)(C(F)F)C2)=O)CCC(CNC(=O)CC2CC2C2CC2)CC1 N1(C(C=CCC(C)(C)NC(C2CCC(=O)C2)=O)=O)CCN2C(=O)NCC2C1 CC1(C)CC(CNC2CCC3(CCC3)CO2)C(C)(C)O1 C(=O)(CC(C)(C)C)N(CC(C)(C)CNC(c1cc(C)co1)=O)CC c12c(cccc1F)NC2=O.c1(C(N(CCNC)CCOC)=O)ccc(CO)cn1 CC(F)(CNC(c1cc(Cl)n[nH]1)=O)CNC(C1CC1C(N)=O)=O CC(CO)C(=O)NC1(C2CCCN2C(c2cnc(-c3cnn(C)c3)s2)=O)CC1 c1(C(=O)NCCc2ccsc2)cc(O)nc2c1CN(C(c1cscn1)=O)CC2 N1(C(CCC2N(C(C=C(C)C(C)C)=O)CCCC2)=O)CC2CC(C1)N(C)C2 c1(C(=O)NCC(C(C)C)NC(C2CCCC2C(F)F)=O)ccncc1Cl c1(SC)ccc(CNCc2ccn(CC(F)(F)F)n2)o1.C12CCC(C1)C(=O)N2C CC1(C)CN(C(c2cc(C(C)(C)C)on2)=O)C(CNC(=O)CC2CC=CC2)CO1 c1(C(N2CC(C(=O)NCC(=O)NC(COC)CO)C2)=O)coc(COC)n1 C12(NC(=O)Cc3ccnc(F)c3)CCCC1N(C(c1coc(Cl)n1)=O)CCC2 c1(C(N2CCC(NC(C3CC3C(F)(F)F)=O)C2)=O)[nH]c2ccccc2c1Br c1(OC)ccc(CS(N2CCCC2C(N2CCCC(O)C2)=O)(=O)=O)cc1 C(=O)(C(CCN(C)C)NC(c1coc(C(F)F)c1)=O)NCC1(CO)CC(C)C1 N1(C(C=CCC)=O)C(C(=O)NC2COCCC2OC)CCC12CC2 C(=O)(CC1=CCOCC1)NCCC1N(C(c2c(C#N)scc2)=O)CCSC1 CC1CN(C(C2C(C)C2C)=O)CCCN1C(=O)CCCSc1ccc(Cl)cc1 CCC(CN(C(C(CNC)O)=O)CCN1CCCC(C)CC1)CC(F)F C1(C)(CNC(C(n2cc(CCCCO)nn2)C)=O)COc2ccccc2O1 C1(C(=O)NC(CC2CC2)CC2CC2)C2CNCC1C2 Cc1ccc(O)c(CC(=O)NCC2CCN(C(=O)CCF)CC2)c1 C1(NC(C2CC(F)(F)C2)=O)CC2(CCN(C(C3COCC4(CCC4)O3)=O)CC2)C1 N1(C(C2(OC)CCCCC2)=O)CC2CCC(C1)N2C(=O)CCc1cc[nH]n1 C1(C(N2CC(O)(CNC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)(CC)CCC(O)CC1 Cc1cc(C(=O)NCC2CC2C(=O)NCC(C)(C)C(=O)N(C)C)ccn1 C1(CNC(CC(C)OC)=O)CCCCN(C(c2c(Br)n[nH]c2C)=O)C1 C1(C(c2nnnn2C2CCOC2)NCCCSCC)C2(CCC2)C12CCC2 C1(NC(=O)NC)CCN(C(c2ccc(CNC(=O)CC(=O)NC)nc2)=O)C1C c1(CC(=O)NCC(CNC(c2cc(C)sn2)=O)O)ccccc1CC(N)=O N1(C(CCC(C(=O)OC)(C)C)=O)CC2CCCC1CN(C(=O)C1=NOCC1)C2 C(=O)(CCCCC(C)=O)N1CCC(C(=O)N(C)CC2CCOC2)(OC)C1 N1(C(c2sc(C)c(Br)c2)=O)CC2(C1)CN(C(=O)C1=CCCS1)CCO2 C1(C(=O)NCCN(C(=O)C(O)C(C)C)CCC)CCC2(CC1)NC(=O)NC2=O C1(CC=C)(CNC(CC2N(C(COCCC=C)=O)CC2)=O)CC=CC1 c1(C(=O)NC2C(C)(C)CCN(C(=O)Cc3ccsc3)C2)csc2cc(Cl)cnc12 C1(C(NOCC=C)=O)C(C)OCCN1C(=O)C(C)SCC C12(CNC(C)=O)CC3CC(CC(C3)C1NC(=O)Cn1cc(C(=O)OC)nn1)C2 c1(C(=O)NCCC(CC)(CC)NC(=O)C(F)=C(C)C2CC2)cccn2c(O)nnc12 c1(C(N2C(CCCNC(C3CCC(C4CC4)CC3)=O)CCC2)=O)cccc(F)n1 N1(C(CC(C)CF)=O)CC2CCCC2(CNC(c2ncn(C)n2)=O)C1 c1(CNC(COC)=O)n[nH]c2c1CN(C(=O)Cc1ccc(C)cc1Cl)CC2 C1(C(=O)NC2CCNC2=O)(NC(c2coc(CO)c2)=O)CCCCC1 CC(C)CC(CNC(C1(CNC(c2ncccc2F)=O)CC2(CC2)C1)=O)CO C1(NC(C2(COC)CC2)=O)CS(=O)(=O)C12CCN(C(=O)C(C(=O)OC)OC)CC2 c1(C(=O)NC(C2CCN(C(=O)CC(O)C3CC3)CC2)C)cc2ccccc2n1C N1(C(c2cncc(OC(C)C)c2)=O)CCCC(CNC(=O)CC(=O)N(C)C)CC1 C1(C(C)NC(Cc2nc(C)[nH]n2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC1 N1(C(C(C)=CC2CC2)=O)C2CCC1CN(C(=O)CC(C)(C)C(=O)OC(C)(C)C)C2 C1(C(C)(C)C)(CNC(C(CC)F)=O)CCN(C(C2(COC)CCC2)=O)C1 N1(C(C(COCC)C)=O)CC(NC(=O)Cc2cnc(C)s2)CC12CCCCCC2 C1(C(N(C(C)C)CC2CCC2)=O)CCC(CNC(c2cnn(CCO)c2)=O)C1 CC1(C(N2CCN(C(c3cc(C(N)=O)[nH]n3)=O)CC2)=O)CCC12CCC2 c1(OC)ccc(C)nc1C(N1CCCC1CCNC(=O)CCc1nncn1C)=O n1(C(C)(C)C)ccc(=NC(=O)C(C2CCCO2)NC(c2ccccc2F)=O)[nH]1 C(=O)(CCC1C(=O)Nc2ccccc21)NCC(CNC(C(C)=C1CC1)=O)O C(=O)(CCC(F)(F)CCO)N1CCC(C(F)(F)F)(OC)CC1 Cc1coc(C(C)(C)C)c1C(=O)NC1CC1CNC(=O)CC1CCCC(=O)N1 C(=O)(C1=NNC(=O)CC1)N1CCC(CCNC(C2=C(C)CCC2)=O)CC1C c1(C(=O)NCCCNC(C2C(c3cn(CC)nc3)OCC2)=O)c(Br)c(C)nn1C c1(CC(=O)NCC2CCC(NC(C3(C)COC(=O)N3)=O)C2)ccc2sccc2c1 c1(Nc2ccc(CNC(=O)NCCSCC=C)cc2)cc(C)cc(Cl)c1 c1(C(=O)NC(CNC(C(CCC)NC(N)=O)=O)C)cc(C)cc(Br)c1O n1(CCC)nc(C)cc1C(N1CC2CC1C2NC(c1ccnc(N(C)C)c1)=O)=O Cn1nc(C2CC2)cc1C(C1CCNC1)NS(=O)(=O)CC1CCC(C(F)(F)F)O1 N1(C(C=Cc2scc(C)n2)=O)CCC(C2(NC(c3cn(C)c(=O)cn3)=O)CC2)C1 C1(NC(C=CSC)=O)COC2(CCN(C(C3(C4CCCCC4)CC3)=O)C2)C1 C1(CCNC(C2OCC2(C)C)=O)(OC)CN(C(=O)Cc2csc(C(C)=O)n2)C1 N1(C(C2(C)CCC(=O)NC2)=O)CC23CCCC2(C1)CN(C(=O)Cn1cccc1)C3 N1(C(=O)OC(C)(C)C)CC12CC(C)(C(=O)N(CC(O)C(N)=O)CC1CC1)C2 Cc1cn2nc(C(=O)NCC3CC3NC(c3cc(N)ccn3)=O)cc(C)c2n1 c1(NCc2cc(OC)nn2C)[nH]c(=NC(CCO)C(F)F)nc2c1ncn2C c1(C(N2C(CNC(c3c(C)ncc(C)c3)=O)CCC2)=O)ccc2c(C)noc2c1 O(NC(=O)C(CCOC)N(C)C(c1cncc(OC)c1)=O)CC1CC(=C)C1 c1(-c2nc(C(C)C)sn2)nc(-c2nc[nH]n2)nn1CC1(C)CCCC1 C1(CNC(CN(C2CC2)CC)=O)CC(O)CN1C(=O)CC(C)(C1CCC1)N(C)C C1(C2CCCCC2)(C(=O)NC2CS(=O)(=O)CC2NC(=O)COC2CCC2)CC1 CCCCC(CC(=O)N(CC1=CCCOC1)C)NC(=O)C(C)c1cccs1 C(=O)(C(C)CS(C)(=O)=O)NC(C)Cn1cc(CNC(=O)CN(C)C2CC2)nn1 c1(C(=O)NCC(O)CNC(c2cnc(-c3ccco3)s2)=O)cccc(C(F)F)c1 c1(C(=O)NC(C(C)NC(C2C3CC4C(C3)C24)=O)C)ccc2ccnn2c1 CC(C)C(C(=O)NC(C)CF)NC(=O)CN1CCCNC1=O C1(NC(C23CC(COC)(OC2)C3)=O)CN(C(=O)C(F)(F)C2CC2)CCC1C C1(CC(=O)N(CCNC(C2N(C(C)=O)CCC2)=O)C(C)C)CCC(=O)N1C Cc1ccnnc1C(=O)NCc1ccc(C(N2CCCC2)=O)nc1 C=CCCCC(C(=O)N(CC(F)(F)CO)C)NC(=O)C(F)CC1CCOC1 N1(C(CNC(CC(C)C)=O)=O)CC2C(CC(=O)NC(C)Cc3nccn3C)C2C1 c1(C(=O)NCCC2CN(C(C(C)C3(CO)CC3)=O)C2)cnccc1C1OCCO1 c1(OC)cnc(F)c(C(N2CC(NC(C3CC34CCOC4)=O)CC2C)=O)c1 c1(OCCC(=O)NCCNC(=O)C(C)(C)c2ccsc2)ccc(F)cc1.CC1CO1 C1(C2CCC2)(C(N2CC(CNC(C=CC)=O)C(C)C2)=O)CC1(F)F c1(CC(=O)N(C2CCC(NC(C=COCC)=O)CC2)C)cc(F)ccc1O C1(C(=O)NC2CN(C(=O)OC)C2)CN(Cc2cc(F)cc(C#N)c2)CCC1(F)F c1(C(=O)NCCC(CC)(C)NC(C2C3CCCCCC23)=O)cc([N+](=O)[O-])sn1 N1(C(C2N(S(CCC)(=O)=O)CCCC2)=O)CC2CCC(C1)N2C(=O)C(O)C(F)F C1(CNC(CNS(N)(=O)=O)=O)CCCC2(CN(C(C3CCCCC3(F)F)=O)C2)O1 C1(C(CNC(c2cc(CCC)on2)=O)C)CCN(C(c2cnccc2C)=O)CC1 C(=O)(C1=CC2(CN(C(=O)C(C(C)O)N(C)C)C2)OC1)N1CCC(CC)(OC)CC1 Cc1oc(C)c(C(=O)N(CC(C)CNC(C2CC3CCC2CC3)=O)C)c1Br c1(C(N2CC(NC(c3ccc(OC)s3)=O)C3C2C3)=O)ccc([N+](=O)[O-])c(C)c1 c1(-c2cscc2)ccc2ncsc2c1.Cc1cnc(-n2ccnc2-c2ccncc2)s1 N1(C(CC=C(C)C)=O)CC2CCC(C1)N(C(=O)C=Cc1ccc3c(c1)OCO3)C2 CN1N=CC(CC(=O)NCC2CC2CNC(c2cccc(CC#N)c2)=O)C1=O N1(CC(=O)NCC(C)NC(c2c(SC)snn2)=O)CCCCCCC1=O C1(CNC(CN(C(C2CCOC2)=O)CC)=O)CCCC1(C)OC C1(C(=O)NCC2N(C(c3c(C)snn3)=O)CCC2)CC12CC(F)(F)C2 Cc1cc(C)c(C(=O)NC2CC(NC(=O)C(=O)NC(C)C)C2)cn1 CCC(C)C(CC(=O)NCc1ccc(Cl)nc1)NC(c1cccc(CC#N)c1)=O c1(C(=O)OC(C)(C)C)ccc(NCC2C=CCN2Cc2cc(Br)co2)cc1O Cc1cc(N)cnc1C(N1CCOC(C2CN(C(=O)CCP(C)(C)=O)C2)C1)=O c1(C2(C(=O)NCCCNC(c3occc3C3CC3)=O)CC2)cc(F)ccc1F C1(NC(C(C2CC2)OC)=O)(COC)CCN(C(c2cn(C3CCC3)nc2C)=O)CC1 c1(C(=O)NCC(C)(O)CNC(=O)C=CC=C(Cl)Cl)[nH]ncc1C#N C1(NC(CCC(C)C)=O)COC2CN(C(=O)CC(c3ccc(F)cc3)C)CC12 c1(OC)ccc(C(=O)NCC(F)CNC(=O)C(C)Cn2ccnc2)cc1C(C)C c1(C(=O)NCC2CC(C)N(C(=O)CCCN=[N+]=[N-])C2)cnc2c(c1)NCC2 C#CCCCCC(=O)NCCN(C(=O)Cc1ccns1)CCOCCO c1(C(C(=O)NC(C2(O)CCN(c3nnc(CC)s3)C2)C)O)ccc(F)cc1C C1(CNC(C(C)(C)C2CCCCC2)=O)CCCCN1C(=O)Cc1ccc(O)cc1 c1(C(N2CCC(NC(C(C(C)O)N(C)C)=O)C2)=O)c[nH]c2ccc(F)cc2c1=O c1(C(=O)NCC(CC(=O)NC2(CC=C)CCCCC2)C)cc(C#N)oc1C C(C(=O)NOCC(C)(C)O)(C1(O)CCC1)NC(C(N1CC(C)C1)C)=O Cc1cc(C#N)c(O)nc1C(=O)N(C1CN(C(=O)CC2CC(O)C2(C)C)C1)C c1(C(N2C(C(N(CC(F)(F)F)C)=O)COCC2)=O)ccc2n[nH]cc2c1 c1(C(N(CCCNC(c2cn(C)nn2)=O)CC)=O)cccc(OCC(F)(F)F)c1 C(=O)(C(C#N)C(C)C)N1CC(n2cc(SCc3cc(OC)no3)nn2)C(O)C1 CCCCC(O)C(C)C(=O)NCCOC(C)(C)CNC(C12CCC(C1)OC2)=O c1(OC)c(C(=O)NC2CC2c2cccs2)cnn1-c1ccccc1 C1(NC(C2CCC(CC)O2)=O)CCCCN(C(=O)Cc2nc[nH]n2)C1 c1(C(=O)OC)ccn2c1CN(C(c1ncccc1Br)C(=O)NC1CCCC1)CC2 C1(CN(C(C2C=CCCC2)=O)CC)CCN(C(C2C(C)C2C)=O)CC1 c1(C(=O)NCC(=C2CN(C(=O)Cc3ccccc3)C2)F)cc2occc2s1 CN1CC(C(N2CCC2CNC(=O)CCCc2cccs2)=O)NC1=O C1(C(=O)NCCc2c[nH]nc2O)(CC)CCCN1C(=O)CC1CC(OC)C1 c1(CCC(N2CCC(COCC#C)C2)=O)cccc(C)c1Br C=CCC(CC(=O)N1CCOCC1CC(N)=O)NC(=O)CC(C1CC1)C1CC1 C1(N(C(c2c(C)scc2)=O)C)CCN(C(C2(C)C=CCCC2)=O)CC1 c1(C(N2CCC(N(C(=O)Cc3cn(C4CC4)cn3)C)C2)=O)cncnc1C1CC1 N1(C(CC(=O)OC(C)(C)C)=O)CCCC(NC(C2CC2(F)F)=O)C(F)C1 c1(C(=O)NCC(CCCC)NC(=O)CCCNC(N)=O)cccc2nc[nH]c12 N1(C(CCSC)=O)CC2(C1)SCCC2NC(c1nnc(S)n1C)=O c1(C(=O)NC(CNC(c2ccc(CCC=C)cc2)=O)(C)C)cc(Cl)cnc1O c1(C(=O)NC(CCC)CNC(=O)CCCn2ccnc2)cncc(N)c1 C1(=CCNC(CN(C)C)=O)CCN(C(=O)CCC2CC2(C)C)CC1 c1(-n2c(CSc3ccccc3)nc(C(C)OCC)n2)ccc(Br)c(F)c1 C1(C(=O)NCc2ncc(C)nc2)CN(C(=O)C(C)(C)F)CC1(F)F c1(C(N(C2CCN(C(CCOCC)=O)C2)C)=O)ccc(C)c(C)c1Cl CC1(C)COCCC1C(=O)NC1(C)CC(C(=O)NC2(C(C)(C)O)CN(CC)C2)C1 C1(C2CC2)(NC(c2cc(Cl)ccc2C(F)(F)F)=O)CCOC1 c1(C(N2CC(C(=O)NCc3cn(C(C)C)nc3)OCC2)=O)cc(Cl)cc(Cl)c1O C1(NC(CS(N)(=O)=O)=O)CCN(C(c2cc(F)c(N)cc2F)=O)CCC1CO CCCCCC(O)C(C)C(=O)N1CC(O)(CNC(C2CCSC2)=O)C1 N1(C(CCc2c(C)nn(C)c2C)=O)CCCN(C(=O)C(C)C2CCC2)CCC1 c1(C(=O)NC2CC(C)(NC(C3(CC)CCC3)=O)C2)cccc(F)c1Br c1(C(CNC(=O)C=CBr)NC(C(CSC)OC)=O)ccccc1F C=CCCCC(C(=O)N1CC2(CCC2(C)C)C1)NC(C1CCC1C(=O)OC)=O c1(OC(C)C(=O)NCc2ccc(CNC(=O)C=CC3CC3)cc2)ccc(F)nc1 Cn1ccc2ccnc(C(=O)NC3CC(F)(CNC(C4CCCS4)=O)C3)c12 Cc1nc(C(C)NC(=O)C(C2CCC2)NC(C2CC2(F)Cl)=O)n[nH]1 Cn1c(SCCC(=O)NCCCOCCNC(=O)C(N)=O)nc2ccccc12 Cc1occc(=O)c1OCC(=O)NC1CCC(NC(c2ccnnc2)=O)CC1 c1(C(C(=O)N(CC(C)NC(C2OCCCO2)=O)C)O)cc(F)cc(F)c1 C=CCC(Cc1ccccc1)C(=O)NC1CC(C)(NC(C2CC2C=C)=O)C1 c1(C(=O)NC(c2cc(C)cc(F)c2)C(=O)O)ccccc1S(=O)(=O)C(F)F CCC(C)CCCCC(=O)NC(CC1CC1)CC(=O)NCC1(O)CCC1 N1(C(CCCCN(C)C(c2cn[nH]c2)=O)=O)CCC2(CCCCO2)C1 CC1=NN(C)C(=O)C1CC(N1CCC(c2cccc(N3CCCS3(=O)=O)c2)C1)=O C1(CNC(C2CC(C)N2C(=O)C(C)(C)C2CCCC2)=O)CC2CCC1O2 C(c1cccc(F)c1F)=CC(=O)NC1CC(C)(NC(c2cnc(CC)s2)=O)C1 C(=O)(C1=CCCOCC1)N1CCCC(C(=O)NC2CC(C(N)=O)C2)(CC)C1 C(=O)(C(C)(C(C)C)NC(C)=O)N(CCNC(C1CC1C#N)=O)CC C(=O)(C1=NOC(C(C)(C)C)C1)NCCC(C(C)C)NC(C(C=C)OC)=O c1(CNC(C(c2cnn(C)c2)C)=O)c(Br)ccc2ccccc12 C1(C(CC)O)CCC(NC(=O)NC2C3CN(C(C)(C)C)CC23)CC1 N1(CC(=O)NCCc2cn(CCCC)nn2)CCC(F)(F)C1 C(=O)(CS(=O)(=O)C1CCCC1)N(CC(C)NC(C1(F)CCCOC1)=O)C N1(C(C)=O)CCOC(C(N2CC(CO)(NC(=O)C(C)CN(C)C)C2)=O)C1 c1(C(=O)NC2C(C=C)CN(C(=O)CCNS(=O)(=O)CC)C2)cc2ccccn2c1 c1(CN(C(C(=O)NC2CC3CC(OC)C3C2)=O)C)cn2cc(Cl)ccc2n1 C1(CNC(C2C(NC(CCSCC)=O)COC2)=O)OC(=O)NC1(C)C CC1C(NC(C23COC(CCO2)C3)=O)CC2CCC1N2C(=O)CCCC(=O)C1CC1 c1(CC(=O)NCC2CC(O)CN2C(c2cccnc2)=O)cc(Cl)cc(Cl)c1 Cc1cc(NC(=O)C(=O)NC2CC3CC(C(N)=O)CC23)cc2cccnc12 Cc1nn(C)c(C)c1CC(=O)NC1CC(O)CN(C(c2cc(=O)cc(Cl)[nH]2)=O)C1 N1(CCOC)CCCC(NC(C2(CN)CCCOC2)=O)C1 N1(C(c2cc(C)oc2)=O)CCC(F)(CNC(C2(CO)COC2)=O)CC1 c1(C(=O)NC2C3CN(C(C4CCN(C(C)=O)C4)=O)CC2C3)ccc(C)c(C)c1O N1(C(CCn2ccc(C)n2)=O)CC2CC(O)C1C2NC(c1cnc(O)o1)=O c1(-c2scc(CC(=O)NC3(C)CC(CN=[N+]=[N-])C3)n2)ccc(F)cc1 N(C1CCCc2c1cnn2C)C(C(n1cc(-c2ccccc2Cl)nn1)C)=O c1(C(N2C(C)C(NC(=O)C(C)(C)N(C)C)CC2)=O)ccc(N)c(N)c1 Cc1cc([N+](=O)[O-])c(F)c(C(=O)NCCC(O)(C(F)(F)F)c2ncco2)c1F c1(C(=O)NC(CCN(C(C(CCOC)C)=O)C)C(C)C)[nH]nc2c1CCC2(C)C CC1(C)C=C(C(=O)NCC(O)CC(=O)NCc2cccnc2O)C1 O=C(N=c1cc(C2CC2)[nH][nH]1)C1CCCCN1Cc1ccc(Cl)o1 c1(N2C(CNC(C(CCC)(C)O)=O)CCC2)nc2c(C)c(C)ccc2s1 c1(SCC)cccnc1C(=O)NCC1(C)CCN(C(=O)C(C(C)C)SCC)C1 N1(C(CNC(C)=O)=O)CCCCC(NC(c2cc(F)cc(Cl)c2)=O)C1 C=CCC(C)(CC)C(=O)NCCCN(C(=O)Cc1ccc(OC)c(Cl)c1)CCO c1(C(=O)NCC(CN(C(=O)C(F)(F)CO)C)O)ncc(Cl)cc1F N1(C(CC(C)O)=O)CCC2C(C(=O)NCCc3ncc[nH]3)C2C1 c1(C(=O)NC2CC(NC(CS(CC)=O)=O)C2)cc(O)nc(OC)n1 C(CC(C)C)(C(=O)NCc1cnc(C)s1)NC(CC=C)=O C1(C(N2CC3C(NC(Cn4c(C)nc(C)n4)=O)(C3)C2)=O)OCC2CCCC1C2 CC1(C(=O)NC23CC2COC3(C)C)CCN(C(C2CC(=C3CCC3)C2)=O)CC1 N1(C(C(C)OCCC=C)=O)CC2(CCC2)CC1CNC(=O)Cn1ncnn1 N1(C(C(C#C)(C)C)=O)CC2(NC(C3CCOC3c3nccn3C)=O)CCC1C2 C(=O)(C1=CCc2ccccc21)NCCC(=C)CNC(C1CC2CCC1C2)=O C(C)(C)(CCC(=O)N(C)Cc1ncc(C)o1)NC(c1cc(CC)oc1C)=O c1(C(N(CCC(C)NC(CC(=O)NCC)=O)C)=O)ccc2ccn(C)c2c1 C(CC(=O)N1CCOC(CCNC(C2CCCN2C)=O)C1)(C(F)(F)F)OC C(CC(=O)N(C)Cc1nncs1)(C(F)(F)F)NC(CC=C)=O c1(OC)cccc2scc(C(=O)NC3(C)CN(C(=O)CN(C4CCCC4)C)C3)c12 CC1CN(C(c2coc(-c3ccccn3)n2)=O)CC1NC(=O)CC1CC(C)(C)C1 Cc1cc(N)c(C(N2CCCC(CNC(C34CC3CCC4(F)F)=O)C2)=O)c(F)c1 c1(NC(c2nc(O)n[nH]2)C)[nH]c(=NCC2CCOC(C)C2)nc2c1cnn2C N1(C(CN(CCC)C)=O)CCN(CC(C)NC(c2cnc(CC(C)C)[nH]2)=O)CC1 c1(NC(CNC(C(COC)C)=O)C(C)(C)C)ccc(C(F)(F)F)cc1[N+](=O)[O-] C(N=c1[nH]nc(CC(C)C)s1)C1CN(C(C=CCC)=O)C(C)C1 c1(C(=O)NCC(C)N(C(C23C(CN(C(CC)=O)C2)C3)=O)C)cc(CC)cnc1O C(C(=O)NC12CC1CN(C(c1csc(C)n1)=O)C2)(C(F)(F)F)OC(C)=O c1(N2CC(C)(NC(CC(c3c(C)n[nH]c3C)C)=O)C2)nccc(S(C)(=O)=O)n1 C(N=c1cc[nH]c(=NCCc2cncc(C)c2)[nH]1)C1(OCC)CCS(=O)(=O)CC1 N1(C(c2c(CC)nns2)=O)CCOC(CCNC(=O)CCSC(F)(F)F)C1 N1(C(CS(C)(=O)=O)=O)CCC(O)(CNC(c2ccnc(CO)c2)=O)CC1 C1(C2CCCN(C(=O)Cn3nnc(C)n3)C2)(NC(CC2CC(OCC)C2)=O)CC1 CC1(CNC(c2ccc(-c3nc(=O)n(C)[nH]3)cc2)=O)CCS(=O)(=O)CC1 N1(C(CC(CCC)C)=O)CC2CCCC2(CNC(c2ccc(C3CC3)nc2)=O)C1 c1(C(=O)NC(C)CCNC(C2(C)CC3(CC3)C2)=O)ccc(N)c2ccccc12 C(CCCCCCCO)=CC(=O)NCCCCCNC(c1cn2c(n1)SCC2)=O Cc1cccc(SCC(=O)NC2CCCC2NC(C2CC(C#N)C2)=O)c1 c1(CC(=O)NCC2C3CN(C(C(CC)(C)O)=O)CC32)ccc2ncnn2c1 C1(C(=O)NC(CC)CC(=O)NC2CCCC2N(C)C)CCN(C)C(=O)C1 N1(C(C2(C)COC2)=O)CC2(NC(=O)C3=CCCCO3)CCC1C2 c1(C(=O)Nc2c(OC)ccc(C#N)c2)c[nH]ccc1=Nc1ccccc1 c1(C(N(CCCN(C(C(C)n2cccn2)=O)C)C)=O)cc2cc(F)ccc2cn1 N1(C(C(C)OCCOCC)=O)C(C(N2CCC(N(C)CC)C2)=O)CCC12CC2 N1(C(C2CCCN2C2CC2)=O)CCC(F)(F)C(CNC(C23CCC(C2)C3)=O)C1 C(CCCOC)(C(=O)Nc1cccc(CC)c1)NC(CCCC=C)=O c1(C(=O)NC(C=C)C)coc2cc(N)c(C3=CC(C)(C)CC(C)(C)C3)cc12 CCC(CNC(=O)CC1CCC2CC12)(CC)NC(=O)CN(C)S(N)(=O)=O CC1(C)CCc2onc(C(N3C4CCC3CN(C(=O)C(C)(C)CF)CC4)=O)c2C1 C(c1cnc(O)nc1O)=CC(N1CC2(CCN2C(=O)Cc2cccs2)C1)=O c1(C(C(N2CC(CC)C(NC(=O)C=CCF)C2)=O)C)c(C)cccc1C c1(C(N2CC(NC(CCc3n(C)cnc3)=O)C3(C2)CC3)=O)cnc2n1CCOC2 N1(C(C2C(C=C)CC2)=O)CC(CNC(c2cccnc2OCC)=O)CC(C)(C)C1 c1(C(N2CCC(NC(c3c(C)nc(C)s3)=O)C(C)C2)=O)cc(F)cc2c1CCC2 CC(C)CC(CC(C)C)C(=O)N1CCCC2(NC(C3CCNC3=O)=O)CCCC12 N1(C(=O)OC(C)(C)C)CCCOCC1SCCNC(=O)CC(F)(F)F C1(C(=O)NC(C)CCNC(=O)C(C(C)C)N(C)C)CNC(=O)CC12CCOC2 CCCCC(C(=O)NC1CC12CCN(C(=O)COCC(C)(C)C)C2)C(C)C CC1CCOCC1C(=O)NCC(CO)NC(c1ccsc1)=O c1(CC)cncc(C(=O)NCC2(NC(c3cc(C)c(CC)s3)=O)CCOC2)c1 c1(CNC(C2C(CC)OCC2)=O)cccc(CN(C(=O)CC2(C)CC2(F)Cl)C)c1 c1(CNC(=O)CC2CN(Cc3cc(I)ccc3O)CCO2)ccc2cc[nH]c2c1 N(C1CCCc2ccccc21)C(CS(Cc1c(Cl)c(OC)cc(OC)c1)(=O)=O)=O C(C)(C(C)(C)C(=O)NC1CCC(O)C1)NC(CC=CCCCCC)=O C1(NC(c2cocn2)=O)CN(C(c2ccc(O)c(Cl)n2)=O)CC1C1CC1 N1(C(c2ccc(I)s2)C(=O)NCCCC2(C)CC2)CCN(CC(C)(F)F)CC1 N1(C(Cc2c(OC)cccc2Cl)=O)CC2(CCCN(C(=O)C(C)OC)C2)C1 C(N=c1ccnc(C)[nH]1)C1CCCCN(C(CNS(CC)(=O)=O)=O)C1 c1(OC)cc(C)c(C(=O)NCCC(C)N(C(=O)C(C)NC(C)=O)C)cc1OC C1(CNC(CCc2ccc(C)o2)=O)CN(C(c2ccn(CCF)n2)=O)CC1(C)C C1(NC(CSCCOC)=O)CCN(C(c2cnc(O)n2C)=O)C(C2CC2)C1 C1(N(C)C)CCCCC1N=c1nc(N(CCC(N)=O)C)c2c([nH]1)CCOC2 c1(NC(=O)CC(=O)N(CC2CCN(CC)CC2)CC)cc(SC)cc(Cl)c1 N1(C(c2n(CC)cnn2)=O)CC2(CNC(C3(C#N)CCCCC3)=O)CCC1CC2 C(=O)(C1=CC(C)(CC)C1)N1C(CNC(c2n(C=C)ncc2)=O)CC1 CC1CCc2[nH]c(=NCc3ncc[nH]3)[nH]c(=NCCP(C)(C)=O)c2C1 Cc1cccc(Cl)c1CN1CCCC(c2cc[nH]c(=N)n2)C1 C1(C(N2CC(NC(C3(CC(C)=O)CCC3)=O)C2)=O)CCN(c2ccccc2)C1 C1(COC)(NC(=O)CC(C)(C)O)CCN(C(c2ccnc(C(F)(F)F)n2)=O)CC1 CC1(C(=O)Nc2cncc(Br)n2)CC12CCN(C(c1ccc(O)c(O)c1)=O)CC2 c1(CC(=O)NC(C(C(C)C)NC(=O)CC2(O)CC2)C)c[nH]c2cnc(Cl)cc12 C1(C2CCN(C(C3(N(C)C)CC3)=O)C2)(NC(Cc2c(C)nc[nH]2)=O)CC1 CCCCC(=O)C(=O)N1CCCC1CNc1cccc(C(=O)NC(C)=O)c1 C1(C(N2CC(N(C)C(c3ccc(N)c(O)c3)=O)C3(C2)CC3)=O)Cc2ccccc2S1 c1(C(C(=O)OC(COCC)C)C)ccc(C(C)(C)C)cc1 CC(CCN(C)C)C(=O)N1CC2C(NC(c3cc(C(C)(C)C)c[nH]3)=O)C2C1 N#Cc1cnc(C(N2CC3CC3(C(N)=O)C2)=O)c(Cl)c1 N1(C(c2c(C)nn[nH]2)=O)CCN(C(=O)CNc2ccc(C(F)(F)F)cn2)C2CC12 C=CCCCCCCCC(=O)NC(C)(CNC(c1cccn1C)=O)C1CCC1 C(C(=O)N1CCC(NC(c2cc(Br)c(C)o2)=O)C1C)(C(F)(F)F)OC(C)=O C12(C)CCN(C1)C(=O)CCO2.Cn1cc(CCC(=O)NC2CCCCC2)nn1 C1(C(N2CC(CC#C)C2)=O)CC(NC(c2nocc2C)=O)CCO1 N1(C(C2CC(C)OCC2)=O)CC(NC(=O)C(N2CCCCCC2)C)CC1(C)C C1(C(=O)NCC2CCN(C(C(CC)C#N)=O)CC2)CCc2nnc(O)n2C1 C=CCC(CNC(C1CCS(=O)(=O)C1)=O)C(=O)NOCC(C)C c1(CNC(=NC)NCC(C)(C)CCCO)cccc(S(N)(=O)=O)c1 N1(C(C2(NC(c3cnc(S)nc3)=O)CC(CO)C2)=O)CC(F)(F)C1C1CC1 CC1OCCN(C(=O)NCC(=O)NC(C)(C)C)C1CN1CCCC1 c1(C(N2CCN(C(C(CC=C)(C)C)=O)CC2C2CCC2)=O)cnc2nccn2c1 C1(CN(C)C)CCC(C(=O)NC(CNC(c2ccn(C3CCC3)n2)=O)C2CC2)O1 Cc1ccc(C(N2CCCCC2CCNC(C23CCC(C2)C3)=O)=O)cc1O C(=O)(C(F)(F)C(C)(C)O)N1C(CC(=O)NCCCCC=C)CCCC1 C#Cc1ccc(C(=O)N(CC(C)NC(C2C(C)C2C)=O)C)cc1C N1(C(=O)C(F)CC2CC2)CCC2CN(C(C3(F)CC3)=O)CC2C1 c1(C(N2CCC(C(N(C3CCN(C)C3)CCC)=O)C2)=O)cccnc1Br C(=O)(CC(=O)N(C1CCCC1)CCN(C(=O)CN1CCCC1C)C)NCC CC1COCC(CC(=O)NCc2nc(C(=O)N(CC3CCCO3)CC3CC3)co2)O1 Cc1cc(C(N2CC(CNC(C3(C)CCOC3)=O)C(C)C2)=O)sc1C N1(C(=O)COCc2nc[nH]n2)CC(NC(=O)Cc2cccc(Cl)c2Cl)CC(O)C1 C(=O)(C1=CCCC1C)NC(CN(C(C1(c2cccnc2Cl)CC1)=O)CC)C N(C)(C[Si](C)(C)C)C(c1c(C(=O)NCCN(C(CC)C)CC)cco1)=O C(C(C)CC(=O)NCC1(CCCNC(=O)COC(C)C)CCCC1)OC c1(CC)nc(C)c(C(=O)NC2CCCC2C(=O)N(C(CO)C2(C)CC2)CC)o1 Cc1ccncc1CCNC(=O)C(C1(C)CC1)NC(C1CC1(F)Cl)=O C(=O)(CCS(N)(=O)=O)NCc1nnn(C)c1C(N1CC(CN=[N+]=[N-])C1)=O CCC(C)C(=O)NCC(N1CC=CC1CNC(=O)CC1CC(NC(C)=O)C1)=O C(=O)(C1Cc2ccc(F)cc21)NCC(=C)CCNC(=O)CCc1ccc(O)cc1 C(=O)(C#CC1CCCCO1)N(CC(C)O)CCNC(=O)CCC1CCOCC1 N1(C(C)CC2CCOCC2)CCC(O)C(C(=O)NCCOC2CC2)C1 c1(C(N(CC(CNC(c2c(CC)cno2)=O)O)C)=O)nccc2ccn(C)c12 S(=O)(=O)(c1cnc(NC(c2ccc3c(c2)CCO3)C)cc1C)NCCCCCC N1(C(c2c(COC)noc2)C(=O)NCc2ccc(F)cn2)CC(CO)OCC1C CCCC(C(=O)N1CC(C)(C)C1C1CCN(C(=O)C=C(C)C(C)(C)C)CC1)OC Cc1cc(C(=O)NCC2(CNC(C3CCS(=O)(=O)N3)=O)CCC2)ccc1C(F)F N1(C(c2c(C)onc2)=O)CCN(C(=O)C(=O)N(C)C)C(CCO)C1 N1(C(C(C)NC=O)=O)CCC(CNC(=O)CN2CCNC(=O)C2)C12CCC2 N(C(=NCCCCCCO)NCC1CC2CC1C2)CCN1CC(C)OC(C)C1 C(CCCCCNC(=O)COCC1CCCO1)NC(=O)CCc1cc(Cl)cs1 C1(CNC(c2nc(COC)oc2)=O)CN(C2C(C(=O)OC)CCC2)CC1C(C)C C1(C(=O)NCC(CC)NC(=O)Cn2nnnc2C(C)C)Cc2cc(Cl)ccc2O1 c1(C(N2C(C)(C)CC(CNC(=O)C(C)(O)C(F)(F)F)C2)=O)ncccc1S(C)(=O)=O N1(C(c2ccn(C(C)C)n2)=O)CCOC(CN(C(=O)C(C)CCN(C)C)C)C1 c1(OC)cc(I)c(C(N2CC(C(=O)Nc3c(Cl)ccnc3Br)C2)=O)cc1OC N1(C(C=CCOCCOC)=O)CC(CNC(=O)C=CCCC(C)C)CC1C CC(C)C(F)C(=O)NCc1ncc(C(=O)N(C)CCC2CCCC2)cn1 C=CCC(C)(C)C(=O)NC1CC2CC1N(C(=O)CCc1ccc(C(N)=O)nc1)C2 C12(C(=O)NCCN(C(Cc3n(C)ccc3)=O)CCOCCO)CCN(CC1)CC2 n1(CCCOC(C(=O)OC)C)cc(C2CC(NC(=O)OCC(C)C)C2)cn1 c1(N(CC(CC)O)CC2CC2)nc2ccccc2c2ccccc12 N1(C(CC2CCCN(C(C3CN(C)C3)=O)CC2)=O)CCCC(C2CCC2)C1 C(=O)(C1CCCc2scnc21)N1C(CNC(c2n[nH]c3ccnc(Cl)c23)=O)CC1 c1(C(=O)NC(CC)CNC(c2ccn(C(C)C)n2)=O)nc(C)ncc1Cl N1(C(CC(CC)CN(C)C)=O)CC(NC(=O)CCOC2CC2)C2CCCC12 CCCCC(C(=O)NC1CN(C(=O)COCC2CCCC2)C2(CCC2)C1)C(C)C CCCS(=O)(=O)C(C)C(=O)NCC1CCCN1C(c1ccc2nn[nH]c2c1O)=O c1(C(N2CCC(C(C)NC(C=Cc3ncc(C)[nH]3)=O)C2)=O)ccc(C)c(CO)c1 CC1=C(C(=O)N(CCCNC(c2cnn(C)c2F)=O)C2CC2)SCCO1 c1(OC)ccc(C(=O)NC2CCC(CNC(C34CCC(C)(C3)OC4)=O)C2)cc1Cl CC1(C)CC2(CN(C(=O)CONC(C3CCCC4(CC4)C3)=O)C2)C1 c1(C(N2C(C)CC(CNC(=O)Cc3sccc3Cl)C2)=O)ccc2ncnn2n1 c1(CC)ccc(C(N2CC(NC(=O)CC3(OC)CCOCC3)CC2C)=O)cc1N C(C)(C)(C(=O)NCC1(CO)CCC1)C1(C)CC1.C1(C(C=O)F)CCOCC1 C1(C(=O)NC2(CC(=O)NC3C(SC)COC3)CC2)CC(C)CCO1 O=C(C1=CS(=O)CCC1)NC1CN(C(=O)COc2ccsc2)CC1CC1CC1 Cc1cc(C(=O)NC(CC2CC2)C(N2CCCC(C#N)C2)=O)nc(C)c1 C=CC1CN(C(C2CCCC3(CC3)C2)=O)CC1NC(C1(CC2CC2)CC1)=O CCC(C)CCCC(=O)N1CCOCC1CC(=O)NCC12CCC(CC1)O2 CC1CN(C(C2C3CN(C(=O)CC4CCSC4)CC23)=O)CC(C(N)=O)O1 C1(O)(CNC(C(C)OCCC#C)=O)CCN(C(c2cc(CCC)n(C)n2)=O)CC1 C(=O)(C(F)C1=CCCCC1)N1CCC(C2N(C(c3cnc(Cl)cn3)=O)CCC2)C1 CC(C)CC(C(=O)NCC)C(N)=O.c1(Cc2ccc(C)o2)c2c(nn1C)CCSC2 N1(C(Cn2ncc(C)c2)=O)CC(CNC(c2cn(C)nn2)=O)C2CC12 C1(C2CCCCC2)(C(=O)NC(C2CCN(C(C3CC4(CSC4)C3)=O)C2)C)CC1 c1(C(N(CC(C)CNC(=O)C(C)N(C)C(C)=O)CC)=O)ccoc1C(=O)OC C1(C2CC2)(NC(C(N)=O)=O)CCN(C(c2cnnc(-c3ccccc3)c2)=O)C1 c1(C(=O)NC(C(C(C)C)NC(c2cnsc2)=O)C)ccc2c(c1)S(=O)(=O)NC2 N1(C(C2(CCOC)CCC2)=O)CCCC2(NC(=O)C(C)OC3COC3)CCCC12 c1(CC(=O)NC2CCC(N(C(=O)CCOC3CC3)C)CC2)ccc(F)cc1Cl c1(C(N2C(CNC(CCCN(C(C)=O)C)=O)C=CC2)=O)ccnc(SC(F)F)c1 CCCCCCCCCCC(=O)N1CCC(N(C(=O)C(=O)C(C)(C)C)C)C(C)C1 C1(C(N(CC(CO)(CO)NC(C2CSCCS2)=O)C)=O)C2CCCCCC12 c1(Nc2cc(C(F)F)nc(C)n2)cccc(C#N)c1N CC1CCC(NC(c2cnc(=N)[nH]c2)=O)CN1C(=O)Cc1cccc(F)c1 N1(C(c2c(N)nccn2)=O)CC=C(CCNC(c2csc(Cl)c2Cl)=O)CC1 C(=O)(CC(C)(C)C)NC(C)C(=O)N(C(C)CNC(c1cc[nH]c(=N)n1)=O)C C(=O)(C(C)C(C)(C)C)N1CC(CNC(c2cc(CCC)c(C)s2)=O)C(C)C1 C1(C(N(C)CC2(CO)CCC2)=O)CC(NC(c2ccc(O)cc2F)=O)C12CCC2 c1(C(C(C)NC(=O)Cn2cnnn2)NC(C2C(CCC)C2)=O)ccccc1 CS(C)(=O)=NCC(=O)NCCN(C(C1CC1c1ccncc1F)=O)C1CC1 C1(c2n(CCCOC)nnn2)(Nc2ccc(Br)cc2C#N)CC2(CCOCC2)C1 CC(C)C(CNC(=O)CC1CC12CC2)NC(c1cc(-c2ccoc2)[nH]n1)=O Cc1cn(C(C)C)cc1C(=O)NCC(O)CCNC(=O)CCc1ccn(C)c1 c1(CN(C(C2COC3(CCC3)C2)C(=O)NC)C)cc(Cl)c(C)cc1Br N1(C(c2c(C)nns2)=O)Cc2[nH][nH]c(=NC(=O)c3ccc(O)cc3)c2C1 C1(C(N(C)CC2CCN(C(=O)Cc3cccnc3)C2)=O)CCC2(CCCC2)CC1 c1(C(=O)NCC(C2CCC2)NC(=O)COC2CC=CC2)cc2c(Cl)nccc2o1 Cc1ncc(C(N2CC(C)(C)CC2CNC(=O)C=C2CCCCC2)=O)cc1N C1(C(N(CC(CC)NC(C2CN(C(C)=O)C2)=O)C)=O)OCCOC1(C)C Cc1ccn(CC(=O)NC(C)(C)CNC(c2cc(-c3ccccc3)cs2)=O)n1 C1(C(=O)NC2CC(CCNC(c3c(C)nccc3Cl)=O)C2)CC2CCCC(C1)C2 C1(C(N2C(CC)CCC2)=O)(NC(=O)Cn2nccn2)CCCC1C c1(C(=O)NCCC(C)NC(C2CCOCC2)=O)ccn2ccsc12 Cn1ccn2cc(C(N3CCC(C)(CNC(C4C5CCCC45)=O)C3)=O)nc2c1=O CCCCC(CCC)C(=O)N(c1ncc(C#N)cc1C)CC C(=O)(C1=CCCCC1C)N1CC(CC=C)(C(=O)NCC2CC(CO)CO2)C1 Cc1oc(C2CC2)nc1C(=O)NCC1CCCN(C(c2cn(C3CC3)cn2)=O)C1 c1(CC(=O)N(CC(CNC(C2(CC)CNC(=O)C2)=O)O)C)c(Cl)c(CC)nn1C N1(C(C(C)NC(c2ccco2)=O)=O)CCN(C(C2CCC3(CC3)C2)=O)C(CO)C1 C12(NC(CCCCC)=O)CCCC1(F)CN(C(=O)C(C(C)(C)C)OC)C2 C1(CCNC(CCC(=C)C)=O)CN(C(=O)C2=CS(=O)CCC2)CCS1(=O)=O C(CCC(O)C(=O)NC1CC2CC2C1)NC(CN1CC(C)(OC)C1)=O CCCCC(C(=O)NC1CCN(C(C2CCC2)=O)CC1F)C(C)C Cc1cccc(C(N2CCC(O)(C(=O)NOC(C)C)C2)=O)c1N CC1CN(C(C2CC3(C2)CC(O)C3)=O)CCCN1C(=O)CCc1cncc(F)c1 N1(C(CC2(C(=O)OCC)CCC2)=O)CCOC2C(C(F)(F)F)C12 Cc1cnc(Cl)[nH]c1=NCC1CCC2(CCC2)C1NC(c1ccc(Cl)c(Cl)c1)=O C(CC(C(C)C)NC(c1ccc(C)nn1)=O)N(C(C(CC)N(C)C)=O)C c1(C(=O)NCC2C(NC(C(c3c(C)ccc(F)c3)=O)=O)C2)ccc2nsnc2c1 N1(C(C(C)OCCCC)=O)CCN(C(=O)Cc2ccc(Cl)cn2)CC1C1CCC1 n1(C(C)C)cc(C(=O)NCC(n2cc(CC(C)(O)CC)nn2)C)c(Br)n1 N12CCCC(CC1)C2=O.C(CC(COC)NC(=O)CSCCC(C)C)OCC C(C)(CC(F)(F)C(F)(F)CC)(c1n(CC=C)nnn1)NCc1ccc(Br)c(C)c1 c1(C(CC(C(C)C)(C)NC(C2CC2C)=O)=O)cc(S(=O)(=O)N2CCCC2)c[nH]1 N1(C(CC(CC)C)=O)CCC2(C1)CN(C(c1csc3c1CCCC3)=O)CC(C)O2 n1(CCOC)nc(C(=O)Oc2ccc(F)cc2)nc1-c1ccc(C(C)(F)F)cc1 O=C(C(C1=NOC2CC12)N1CCN(Cc2ccoc2)CC1)NC1COC1 c1(OC)nc(N(C2C3CNCC23)C(c2ccc(Cl)cc2F)=O)ncc1F N1(C(c2cc(CC)[nH]n2)=O)CC(NC(c2ccc(NC(=O)OC)cc2)=O)CC1C CC1CC(C)N(C(=O)CCCCCc2ccccc2)CCN1C(c1cncs1)=O c1(N(C(C(=O)OCC)c2cccs2)C)cncc(F)c1C.C12CCCN(C1)C2=O c1(C(=O)OC)cc(C(=O)NC2CN(C(c3nnsc3C)=O)CC2C)ccc1F C1(CNC(c2c(CC)non2)=O)CN(C(C2(O)CCOCC2)=O)CC2(CCC2)O1 c1(NCCCOC)cc(Br)ccc1S(=O)(=O)N1CC2CC1CS2=O N1CC2(C1)CN(C(=O)CNC(C1CC(=O)C1)=O)C2.c1(OC(F)(F)F)ccc(CCC)[nH]1 Cc1cnc(NCc2ncccc2C)c(S(=O)(=O)NCC2CCC(O)C2)c1 c1(CC)ncc2c(n1)CCC(C(=O)NCCCNC(C1CN(CC(C)C)C1)=O)C2 c1(C(=O)NC(C2(OC)CCC2)C)c[nH]nc1CNC(c1cc[nH]n1)=O Cn1nc([N+](=O)[O-])cc1C(=O)NC1CCC(CNC(C2(C#N)CCCCC2)=O)C1 c1(CN2CCC(N(C(=O)C(c3c(F)cccc3F)(F)F)C)C2)cc(O)nc(=N)[nH]1 C(C(C)CC(=O)N(C)Cc1cncnc1)NC(C(C1CCC1)OCC)=O CC1CCN(C(c2cncc(C(N)=O)c2)=O)CC1NC(C1OCCCO1)=O C1(CN(C(c2ccc(OC)o2)=O)C)CN(C(=O)CCC(C)(C)F)CC12CC2 c1(C(N2CCC(N(CC(C)O)C)CC2)C(=O)NCCSC)csc(C#N)c1 N1(C(c2n(CCC)ncc2)=O)CCC(NC(=O)Cc2nocc2C)C1C c1(NC(c2nnnn2CC2CCCO2)(CC)C)ccc(OC)cc1CC C1(C(=O)NCc2cc(CC3CC3)on2)(OC)CC(CC(=O)CCc2cnn[nH]2)C1 N#Cc1ccc(C(N2CCC=CC2C(=O)NOCC2CCOC2)=O)cc1 N(C(=S)NNC(=O)C(C)(C)c1ccc(C(N)=O)cc1)C(C)C N1(CCC)CC(OCC(=O)NC(c2cc(Cl)c(Cl)s2)=O)CCC1=O CC(C)(Cc1ccccc1)CC(=O)NCC(O)CNC(C1CCSC(=O)C1)=O c1(C(N(C2CCCN(C(=O)CS(N)(=O)=O)C2)CC)=O)ccc(=NC(=O)OC)[nH]n1 c1(C(N(C(CCNC(C#CC(C)C)=O)C)C)=O)cc2cc(N)ccc2[nH]1 c1(C(=O)NCC(CCCC)NC(C2CC2F)=O)cc(F)c(F)cc1NC(N)=O c1(C(=O)NCC2CCC(NC(CCCCC)=O)CC2)ncc2c(F)cccn12 N1(C(CC(CC)SC)=O)CCN(C(c2cc(C)cc(Cl)c2)=O)CC1C(C)C N1(C(C(C(C)O)(F)F)=O)CCCC2(CCCN2C(=O)CC23COC(C)(C2)C3)C1 C1(C)(CNC(=O)NC2(CC)CCCC2)CCCN1C c12nc(C)c(o1)C(=O)NC2.C1(C)(CN(C(CCC)=O)C(C)(C)C)CCCC1 C1(NC(C2C(C(N)=O)C2)=O)C=CCN(C(c2ccnc(C3CC3)n2)=O)C1 c1(C(=O)NCCNC(CC(C(C)C)O)=O)cc(Cl)c(O)c(Cl)c1 Cc1ccncc1C(c1ccc(Br)cc1)NCc1nnnn1C1CCOC1 C(=O)(C(Cc1ccccc1)NC1(C(=O)OC)CC(C)C1)NCC(C#C)C N1(C(C2C(C#C)C2)=O)CC(NC(=O)Cc2ccc(C(F)(F)F)nc2)C(O)C1 c1(C(=O)NCC2CCCN(Cc3cc(F)cc(Cl)c3)C2)cn2cc(Cl)ccc2n1 c1(C(C(=O)NCCC2C(C)(C)OCC2)F)ccc(Br)cc1Cl C(=O)(C1=CC2(CN(C(C3CC(=O)C34CCC4)=O)C2)OC1)NC1CN(CCC)C1 C1(N(C(=O)COCC2CC2)C)CCN(C(=O)C)C1.C=C1CC1C(=O)OC(C)(C)C N1(C(c2c(CC)nc[nH]2)=O)CCC(NC(c2nc(Cl)sc2C)=O)CC1C c1(C(=O)NC2CC(C(=O)OCC)C2)cnc(N)cn1.C1(=O)CCNC(=O)CN1 N1(C(c2cscc2C(F)(F)F)=O)CC2CCC1CN2C(=O)CC1CCC1 C1(C(C)NC(c2nnc(C)s2)=O)CCCCN1C(c1cnn(C(C)C)c1)=O c1(C(N2C(CCCC)CN(C(=O)C(C)O)CC2)=O)cn2ncnc2nc1C Cc1nc(N2CCN(C(C(=O)NC(C)C)c3cnsc3)CC2)sc1C C1(CC2CC2)CCCC1NC(c1nc(C(C)NC(C(C)OCC(C)C)=O)on1)C c1(OC)ccc(C(CNC(C2(C(F)(F)F)CC=CC2)=O)NC(=O)C=C(C)Cl)cc1 C1(CCC)(NC(c2cc(C)nc(C)c2)=O)CCN(C(=O)C=C2CCC2)CC1 C(=O)(CC(C)P(C)(C)=O)NCC(CC)NC(=O)Cc1csc(NC(=O)C(C)C)n1 C1(C2(O)CCN(C(=O)CSC(C)C)CC2)(NC(c2cnc(CCC)s2)=O)CC1 C1(C(C)C)(C(=O)NCCS(C)(=N)=O)CCN(C(C2CCC(=O)NC2)=O)C1 c1(NCCCCNC(C2CC(C)OC(C)C2)=O)cc2nncn2cn1 Cc1cnn2ccc(C(=O)NC(C)(C)C(C)NC(=O)C=CCN3CCCC3)nc12 CCC(F)(F)CC(=O)NCc1ccc(CCNC(C2CC2(Cl)Cl)=O)cc1 N1(C(C2C(OC)CCC2)=O)CC(CNC(=O)CCSC(F)(F)F)C(C)(C)C1 C(C(COC)CC(=O)C12C(C1(F)F)C(=O)N(C(C)C)CCNCCC2)OC Cc1nc(O)nc(C)c1CC(N1CC(CNC(=O)C(C)CC(F)F)C(C)(C)C1)=O C(CNC(c1c(Br)noc1C1CC1)=O)(C(C)(C)C)NC(C1C(CC)C1)=O CC1=C(C)C(NC(N2CCCN(CC(C)(C)O)CC2)=O)CCC1 C(=O)(N=c1[nH]n(CC(=O)OC)cc1I)NCCC(=O)Nc1c(SCC)cccc1 CC(CC(=O)NC1CC2CCC1(C(N1CCCCCCC1)=O)C2)C(C)(C)C Cc1ccnc(CN2CCN(CC(=O)Nc3cccc(C(C)O)c3)CC2)c1 C1(NC(c2cn(C)nn2)=O)COCCC1C(=O)NC(C1CCC1)C1CCC1 c1(C(N(CCNC(CC(c2ccc(C)cc2)C)=O)C)=O)cncc(F)c1C N1(C(CCSCC)=O)CCC(CO)C(NC(=O)CCc2ncccc2C)C1 C(CCCC(=O)NC1CCC(CC(=O)NCC(c2ccnn2C)O)CC1)SC c1(C(N2C(C(=O)NCc3nn[nH]n3)CCOCC2)=O)cccc2cncn12 C(=O)(CC(C)C(C)(C)NC(c1ccc(CO)cn1)=O)NCc1n(CC)c(C)nc1 N1(C(c2cc(C(=O)NC(C3(CC)CC3)C)n(C)n2)=O)CCC(=C(F)F)CC1 C1(C(=O)NCC2(NC(c3c(C)cccn3)=O)CCCCC2)NC(=O)OC1(C)C C#CC(C(C)(C)C)NC(c1ccc(CNC(=O)C(C2CCOCC2)F)nc1)=O C(=O)(C1=NOC2(CCC2)C1)N(C)CC1CN(C(=O)C(F)C2CCCC2)CCO1 C12(CNC(CCOC)=O)CC(C1)C(NC(=O)CN1CCS(=O)CC1)CO2 C#CCCCC(C)C(=O)NCCC(=O)NC1CC1.C12CN(C1)C(=O)CNC2=O C1(CNC(Cc2c(C)nc[nH]2)=O)CCCCN(C(C2(c3ccccc3)CCC2)=O)C1 C1(C(=O)NCC(C)(CO)NC(CCOCC(=O)OC)=O)CCC2(CCC2)C1 c1(C(=O)NC2CCC(N(C(COC)=O)C)C2)c(C(F)(F)F)ncn1O c1(C(N2CCC(CNC(CC(CC)OC)=O)C2)=O)cc(C(C)C)ccc1F N1(C(=O)Nc2c(-c3ccccn3)ccc(C)c2)CCC(O)C(C2CC2)(CO)C1 Cc1cccc(CNC(=O)C(O)C2CN(C(=O)C3=CCN(C)C3)C2)c1O CC(=O)C(C)CC(C)C(=O)N(CCC(=O)Nc1ccc(C)cc1C)C CC(C)CC(F)(F)C(=O)NC1CC12CC(CNC(C1CSCN1C(=O)OC)=O)C2 N1(C(COCCC)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1=CCCCC1 CCC(C(=O)NCC1(C(N2CC(O)C(F)C2)=O)CCCCC1)C(F)(F)F c1(C(N2C(C(=O)NCCN(C(=O)C=CBr)C)CCC2)=O)ccc2[nH]c(=N)oc2c1 CN1Cc2cc(CNC(=O)NCC3OC4CCC3C4)ccc2C1=O C1(C(N2CC(C)(C)CC(NC(CC3(OC)CC3)=O)C2)=O)CC2(CCCC2)CO1 c1(C(C(CN(c2ccccc2Cl)CCOC)=O)C)ccc(-c2ccccc2)cc1 c1(C(=O)NCC(C2CCC2)Nc2ccnc(C3CC3)n2)cc2occc2s1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)N1CCCCC(CNC(CC(C)O)=O)C1 CC(CC(F)F)C(=O)N(C1CCCCC1N(C(=O)CC1(C)CCC1)C)C c1(NC2CC3CN(C(CC(CC)(C)C)=O)CC32)ccc2c(n1)CC(C)(C)CC2=O C1(CC)CN(C(=O)C(C)OC(C)(C)C)CCC1NC(=O)CC1CCC(C)CC1 C1(CC)CCC(C(=O)NCC(C2CCCCC2)NC(=O)CC(C)c2ccco2)O1 C(C(=O)N1CCCO1)NC(=O)CC(CC1CC1)NC(C1CC2(CCO1)CC2)=O Cc1nc(N2CCC(CNC(C3(C)CC(O)CN3C)=O)CC2)cc(C(F)(F)F)n1 C1(C(N2CC3C(CN(C(C4(COC(C)C)CC4)=O)C)C3C2)=O)CNC(=O)CC1C C1(CCC)(NC(=O)CCN(C(=O)CCC2CCC2)C(C)C)CCNC1=O N1(C(=O)CC(C2CC2)NC(C2(C3CC3)CC2)=O)CC2(CCC2O)C1 N1(C(c2c(OCCC)cccn2)=O)CCC2C1CCCN2c1ncc(F)cn1 N1(C(c2cnn(C)c2Cl)=O)CCCN(C(C2C3COCC23)=O)CC1CO N1(C(C(C)OCCOC)=O)CC(CC(=O)NCCCCSC2CCCC2)(OC)C1 C(=O)(C(C)C(F)(F)F)NC(CCOCC)C(=O)NC1CCN(COC)C1=O C1(CC(=O)NC2C(CNC(C#CC(C)C)=O)CCCC2)CCCS(=O)(=O)C1 C(CCC(N)=O)(C(=O)N1CCCC1N(c1cccc(Br)c1)C(=O)C1CC1)N(C)C N1(C(C(C2(O)CN(C(Cn3nnc(C)n3)=O)C2)F)=O)CCN(C)CC1C c1(OC)cccc2c1CN(C(c1ccc(Cl)cc1-c1ccccc1)=O)CC2 C1(C(=O)NCCN(CC(C)O)C(c2nn[nH]c2Cl)=O)CC(C)CC(=O)N1 CCCC(C(=O)NC1(C(=O)NCCSCCOC)CCCCC1C)C(C)C N1(C(C2(C)CC2(F)F)=O)CC2(CCC(N3CCC4COCC4C3)CC2)C1 c1(C(N2CCCC(O)(c3ccccc3F)C2)C(=O)NCC)noc2c1COCC2 c1(CCC(C)NC(=O)NC(CCOCC)CO)ccc(Cl)cc1 N1(C(CC2N(CC)CCC2)=O)CCN(C(c2ncccc2CO)=O)CC1C1CC1 c1(C(=O)OC)ccc(O)cc1CN1CCC(O)(CCN(C)C)CC1 C1(O)(C(C)NC(Cc2ccc(CC)cc2)=O)CCN(C(=O)C(CC)OC)CC1 CCCC(C#N)C(=O)N1CCCC(CCNC(=O)CCc2ccc(F)cc2Cl)C1 N1(C(CSCCCC)=O)CC=CC1CNC(=O)C(n1cc(Br)cn1)C C1(C)(C(N(CCCN(C(c2cc(OC)n[nH]2)=O)C)C)=O)CCC(=O)N1 n1(CCC)ccc(C(=O)NC(C2CCCCC2)CNC(=O)C(CC)N(C)C)n1 N1(C(CC=C)=O)CSCC1C(=O)NC(C)CN(C(c1cc(C(F)F)no1)=O)CC N12Cc3ccccc3C1CNC1=CNC=CC1=NC2=O.CC(C)(C)OC(N)=O C1(CNC(C(CC)(C)N(C)C)=O)(COC)CCN(C(=O)CC(C)(C)C)CC1 N1(C(CNC(C(CC)CC)=O)=O)CCN(C(C2CC(=O)N(C)C2)=O)C2CCC12 N1(C(=O)OCCN(C2CC2)CC)CCCC(CCO)CC1 Brc1cc2c([nH]1)CCN(c1nc(N3CC=CC3)c3c(n1)CSC3)C2 Cc1ccc2oc(C(=O)NCC3(C)CCN(C(C4C5CCN4CC5)=O)C3)cc2c1 C(CCN=C(NCc1cscc1C)NC1CCS(=O)(=O)C1)=CC c1(C(=O)NCCC2CN(C(CCSCC)=O)C2)ccc(OC)cc1Br CC(Cc1cc(F)c(F)c(F)c1)N=c1ccn2ncc(S(=O)(=O)NC3CC3)c2[nH]1 c1(N(CC(CO)NC=O)C)cc(Br)c(C(=O)OC)o1.c1(OC)nc(CO)cs1 C1(NC(CC2N(C)C(=O)CC2)=O)CC2CC1N(C(c1occc1Br)=O)C2 C1(C(C)(C)C)CCN(c2nnc(-c3cncc(O)c3)n2C)CC1 c1(C(=O)NCC2(C)CCN(C(C(C=C)OC)=O)C2)cc2c(nn1)CCC2 CCC(C)C(=O)NCC1CCN(C(=O)C(C)OCCC(C)C)C1 N1(C(c2nc(CCC)sc2)=O)CCOCC1CNC(=O)C(C1CCC1)OCC C(C(C(C)C(C)C)NC(c1cnnc(C2CC2)c1)=O)NC(Cc1cc(C)on1)=O N1(C(C(CC)Cc2ccccc2C)=O)CCC2CCC(NC(=O)COC(C)=O)C12 N1(C(C2N(C)CCC2)=O)CC2(C1)CN(C(C1CC(F)(CO)C1)=O)C2 c1(OCC)ncccc1C(=O)NCC1CCC1NC(=O)CCC(=O)NCC(F)F C1(O)(C(C)NC(c2ccccn2)=O)CCN(C(=O)Cc2csc3nccn23)CC1 C1(NC(c2c(CC)n(CC)nn2)=O)C(C)CCN(C(=O)C(C)c2ccsc2)C1C c1(N2CCCC(NC(C(C(C)(C)C)O)=O)(CO)C2)c(F)cccc1[N+](=O)[O-] N1(C(CCc2n(C)ncc2)=O)CCC(O)C(NC(c2cc(O)nn2C)=O)C1 N1(C(c2cnc(C3CCC3)s2)=O)CC2CC1CN2C(c1coc(C2CC2)n1)=O N1(C(CC2CCN(C)CC2)=O)CC2CC1CCC2NC(C1CCCC1O)=O C1(C(=O)NCc2n(CCC)ccn2)CC(N=[N+]=[N-])CN1C(=O)CCNC(=O)OC c1(C(=O)OCC)n[nH]c(=NC2CC(NC(c3ccc(C)c(F)c3)=O)C2)s1 C1(NC(C(C2N(C(=O)OC(C)(C)C)CCC2)O)=O)(CO)Cc2ccc(Cl)cc2C1 c1(OC(C(=O)NCCCC(C)NC(CC=C=C)=O)C)ccc(C)cc1Br N1(C(C(C(C)(C)C)O)=O)CC2CCN(C(=O)C3=COCCO3)CC(C2)C1 N1(C(C=CC(C)NC(=O)COC2CCOCC2)=O)CC(F)CC(F)C1 c1(C(CC)N(C)C)cc(OC)cc(OC)c1Cl.N1CCC(S(=O)(=O)N2CCCCC2)C1 C(CCCCCC(=O)NCC1CN(C(=O)CCc2c(C)n[nH]c2C)CC1C)SC c1(C(N2CCCCC(N(C)C(C3CC(F)(F)CS3)=O)C2)=O)ccc2[nH]ccc2n1 N1(C(C(CC)COC)=O)C2CCC1CC(O)(CNC(c1cn(C(F)F)cn1)=O)C2 C1(C(=O)N)C=CCCN1C(=O)C(O)CN1CCCC1.c1(C2(C)CC2)ccc(F)cc1 C1(C(N(C)C)=O)CCN(C(c2cncs2)=O)CC1O C1(C(N(OCC)CC)=O)C(CC)CCCN1C(=O)CC(C)CC C(=O)(CC(C(F)F)NC(=O)CCC1CC1C)NCCOCCC#C N1(C(C2CCC(C)(CC)O2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1CCO N1(C(Cc2cc(C)n(C)n2)=O)CCCC2C1CCCN2C(=O)CSC(C)C N1(C(C(OCC)OC)=O)CC2(C(=O)NC(C)CCOC)CC1CO2 C1(C)(CNC(c2ccc(C)o2)=O)CCC(NC(=O)Cc2csc(NC=O)n2)C1 C12(C(N3CC(C(C)NC(=O)CC4(C)CC4)OCC3)=O)CCOC1CCOC2 C(=O)(C(C(=O)NCC(CC(=O)NCC(CC(C)C)OC)OC)OC)OC c1(C(=O)NC(C)CN(C(=O)CC2OCCC2(C)C)C)cnc2[nH]cncc1-2 C1(C(N(CCOCCN(C(c2cc(CC)[nH]n2)=O)C)C)=O)CCCC2(CC2)C1 N1(C(CN(C(C)=O)C)=O)CC2CCCC(C1)N2C(=O)C(N1CCCC1CO)=O Cc1nnccc1C(=O)NC(CNC(C1(CF)CCC1)=O)C(C)C C(C(=O)N1CCN(CCCNC(C2CCCSC2)=O)CC1)(C(C)C)NC(C)=O c1(NC)cccc(C(=O)NCC23CC2CN(C(C2CCCN2C)=O)C3)n1 c1(C(=O)NCC2N(C(COC)=O)CCC2(C)C)ccc(S(N)(=O)=O)nc1 C1(C(N2CC3C(NC(c4c(O)cc(O)cc4O)=O)C3C2)=O)CCCCC(F)(F)C1 c1(C(N2CC(NC(c3cc(C(C)C)[nH]n3)=O)C(O)C2)=O)ncnc2c1CCCC2 N1(C(CC2C(=O)NC(=O)N2)=O)CCN(C(=O)Cc2cc(C(F)F)no2)C2(CCC2)C1 Cc1cccc(CN2CCCC2(C)C(N2CCC(=O)CC2)=O)n1 c1(C(=O)OC)ccc(=NCC2(C)CCN(C(C3CSCCS3)=O)CC2)[nH]c1OC c1(C(=O)NC2CCC(NC(CCS(C)=O)=O)C2)cc(F)ccc1C(F)F C=CC(C)(O)CC(=O)NC1CN(C(c2ccc(C)c(N)c2)=O)CC1C c1(C(=O)NC(C)Cc2cn(Cc3cccnc3)nn2)ccc2cnn(C(F)F)c2c1 C1(NC(c2cc(C(C)C)sn2)=O)CN(C(c2ccnc(OC(F)F)c2)=O)CC1F C1(C(=O)NC2C(C(C)(C)C)N(C(=O)CCS(N)(=O)=O)CC2)CC2CCC(C1)O2 C(C(C(C)C(C)C)NC(=O)CC1(C)CC1)NC(CCc1ccc(C)cc1)=O C(=O)(CC(C)CCCCCC)N1C(CCNC(C=CCCC)=O)CC(OC)C1 C1(NC(C2C(=C)CC2)=O)CC1C1CCN(C(c2cccc(CO)c2C)=O)CC1 C(=O)(C1=NNC(=O)C1)N1CCCC(C(C)NC(CCc2ccc(C)cc2)=O)C1 C1(O)(C(=O)NC2CCC(CCNC(C(=O)NCC)=O)C2)CCC(C)(C)CC1 Cc1nc2[nH]n(C)c(=O)c2c(C)c1CCNC(=O)C(N)CC1CC1 C1(CC(=O)N(CCCNC(c2c(C)nc(C3CC3)[nH]2)=O)C)CN2CCN1CC2 Cc1coc(C2CC2)c1C(=O)NCC1CC(F)CN1C(=O)CC1CCCO1 N=S1(=O)CCN(C(=O)C(C2CCC2)NC(=O)Cc2ccon2)CC1 N1(C(c2c(CC)nn[nH]2)=O)CCC2CCC(C1)N2C(C1CCCN(C(C)C)C1)=O c1(C(=O)NC(c2ccccc2)C(=O)NC(c2ccccc2)C#C)cscc1Cl c1(C(N2CC(CCO)(NC(c3ccc(CC)cn3)=O)C2)=O)ccc2cncn2c1 C(=O)(C(C(=O)OC)OC)NCC(CNC(CCSCCCC)=O)(C)O c1(N2CCCC(NCC(=O)OC)C2C)ncnc2c1ncn2CCC(C)(C)CO c1(N2CCC(CC=C)(NC(C3CC4(C3)CC4F)=O)C2)cnc2ccccc2n1 Cc1nc(N2CC(NC(=O)CCc3cn[nH]c3)CC3(CC3)C2)c(Cl)cc1C#N C1(C(=O)NCC2C(CNC(CC3(C#N)CC3)=O)C2)CCc2nnc(O)n2C1 C(=O)(C(F)S(=O)(=O)c1ccccc1Br)N1CC(C)(C)OC(C)(C(F)(F)F)C1 C1(NC(C(CC=C)CC=C)=O)CC1C1CCCN(C(c2occc2C)=O)C1 S(=O)(=O)(c1cnc(N2CCC(CC#N)C2)cc1C)NCC1C(CCCC)CCC1 C1(C2(O)CN(C(c3ccccc3SCCCC)=O)C2)(CNC(C2C(=C)C2)=O)CC1 C1(CNC(c2cc3c(s2)CCC3=O)=O)CCN(C(=O)CC2CCCC2)C12CCC2 C(=O)(C#CC1CCCC1)N1CCC(CCNC(CSc2n(C)c(S)nn2)=O)CC1 Cc1cccc(C(N2CC(C(=O)Nc3ccnn3C(C)(C)C)C(F)C2)=O)n1 c1(C(N2CC(NC(c3n(C)cnc3)=O)CC3(C2)CC3)=O)cccn2[nH]c(=N)nc12 Cc1ccc(C#N)cc1C(=O)NCCC1(O)CN(C(=O)CCCCCF)C1 C1(NC(CC(C)SC)=O)CCN(C(c2ccc(C(F)(F)F)c(N)c2)=O)C12CC2 C1(CC=C)(NC(c2cccc(CCCCC)c2)=O)CCN(C(=O)C(O)CC)C1 C1(C(=O)NCC(C(C)C)NC(C2(C(C)(C)C)CCCC2)=O)CC(=O)N(C)C(=O)N1 c1(CNC(C2CC(C)(NC(c3ccc(OC)cc3)=O)C2)=O)ccnc(C#N)c1 C1(C(=O)NC(CC=C)CO)CC2(CC2)CN1C(c1cc(CC)ccc1O)=O CC1=CCC(C)(C(N2CC3CC(C2)C3NC(C2CCCC3CC23)=O)=O)CC1 C1(CNC(c2cscc2F)=O)CC2(CC2)CN1C(=O)Cn1cccn1 C1(CCCNC(C2(CSC)CCC2)=O)CN(C(=O)CCC2CC2(C)C)CCO1 C1(NC(CC2N(C(COC3(C#C)COC3)=O)CC2)=O)CC2CC1CC2(C)O N12CCC(CC1)C(=O)OC(C)C2.N1(C(C2CCC2)=O)CCN(C)CC1 N1(C(CSCCC(C)C)=O)CCN(C(=O)CCc2cn[nH]c2)C(CC(=O)N(C)C)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)N1CC(CNC(C(CCSC)NC=O)=O)C1 C#Cc1cncc(C(=O)NC2(C)CN(C(c3sc(C(C)OC)nc3C)=O)C2)c1 Cc1nn(C)c(=O)c(C(N2CCC(C)(NC(c3cnc(C(C)O)s3)=O)C2)=O)c1C C1(C(N2C(C(N3CC(CC(C)(C)C)C3)=O)CSCC2)=O)CCC=CCCC1 CC1CCCC(C(=O)NC23CC(C2)N(C(c2csc(C#N)c2)=O)C3)CC1 N1(C(CNC(CCC)=O)=O)CCN(CC(=O)NOC2C3CCC2CC3)CC1 c1(C(N(CCC)CCNC(=O)CC2CCCCC2C)=O)cnc2n1CCC2 C12(C(=O)NCC3OCCN(Cc4cccc(C)c4)C3)CCC(C)(C(=O)O1)C2(C)C CC1(C(N2CC(NC(c3ccc(-c4ccco4)s3)=O)C2)=O)CCCCNC1=O c1(NC(C2OCC(C)(C)NC2)=O)cnc2ccc(F)cc2c1 N1(C(c2c(OC)ccnc2)=O)CC(CNC(c2coc(N(C)C)n2)=O)CC(C)C1 CCC(C)(CC)C(=O)N1CCCCC1Cn1cc(CCCC(C)O)nn1 C1(CN(C(C2(COC)CCOC2)=O)C)CCCCN1C(c1csc(C(F)F)n1)=O c1(OC)cccc(Cl)c1C(N1CCCCC1C(=O)Nc1cc(O)nc(O)n1)=O N1(C(CCC(=O)OCC)=O)CCN(C(C23CC(C)(C2)OC3C)=O)C2(CCC2)C1 C1(CCC)(NC(=O)Cc2ccoc2C)CCCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 C(CC(C(=O)NCCCC1CCCN1C(=O)CC1(OC)CCC1)OC)OC C1(NC(c2cc(CC)c(C)s2)=O)CN(C(=O)C(C)CC(C)(C)C)CCC12CCC2 C1(CCNC(C2C(C(C)(C)C)C2)=O)CN(C(=O)Cc2ccc(F)nc2)CCCO1 CC1CCN(C(=O)CCCn2c(O)nnc2O)C(CNC(=O)CCC(C)(F)F)C1 c1(SCC(=O)NCC2(OC)CN(C(C3(Cl)CC3)=O)C2)ccc([N+](=O)[O-])cc1 C(=O)(C(C)CC(F)(F)F)NC1CC(CCNC(c2cc(CC)ncn2)=O)C1 c1(C(N2CC(C(=O)NC(CCCC)CO)OCC2)=O)ccc(F)nc1C c1(NCC2CC(C)(C)OC2)ncccc1S(=O)(=O)N1CCC(c2ccc(Cl)s2)C1 c1(NC(C(=O)NC2C(SCC)CCCC2)=O)ccc2[nH]ccc2c1 C1(CC)CC(C)CN(C(=O)C=C(C)CNC(C2(OC)CCC2)=O)C1 c1(N2CCC(C(C)NC(=O)CCCC3CCC3)C2)ncc(S(C)(=O)=O)cc1Cl c1(COC)cc(C(N2CC3(C2)CN(C(C2CCCC(O)C2)=O)C3)=O)ccc1OC N1(C(C(CCOC)C)=O)CCC(CNC(c2ccsc2C)=O)C(O)C1 C1(C(N(C2CCC(=C(C)C)CC2)c2cnsn2)=O)CCC2CCC1N2C1CCC1 N1(C(c2ccc(C#C)cc2)=O)CC2CCN(C(C3CC3F)=O)C2C1 C=CCCCC(C(=O)NCc1noc(C(C)C)n1)NC(=O)CCC(C)(C)N(C)C c1(C(=O)NC(CC)(CNC(=O)Cc2c[nH]nc2O)CC)cc2ccncc2[nH]1 C1(C2CC2)(NC(c2c(C)nco2)=O)CCN(C(C2(C)CCCS2(=O)=O)=O)C1 N1(C(CC=CC=C)=O)CCN(C2CCN(C(=O)CC3(CC)CC3)C2)CC1 N1(C(C2C(C(=O)OCC)C2)=O)CCCC(CO)(NC(c2occ3c2CCC3)=O)C1 N1(CC(N2CCC(F)(CNC(C3ON=C(CC)C3)=O)C2)=O)C(=O)CC(C)(C)C1=O n1(CC(=O)NC(C2CC(NC(C(C)=C3CC3)=O)C2)C)cnnc1O C(=O)(C1=NN(CCO)C(=O)CC1)C(=O)C1=CCCOC1.C1(N)CC2(C1)CC(C)C2 c1(OC)cc(C(N2CC(C(C)NC(=O)Cc3ccc(Cl)nc3C)C2)=O)cc(C)n1 C(C1c2ccsc2CCN1C(=O)COc1cccnc1)NC(C(C=C=C)C)=O c1(C(N(C2CCC(NC(c3cc(C)[nH]n3)=O)C2)C)=O)sc2ccc(F)cc2c1C C1(NC(c2nc(C)sc2)=O)CCN(C(=O)CC2CCCC(C)(C)C2)CC1F N1(C(=O)NC(C2CCCOC2)CC)C2CCC1c1ccccc12 N1(CC)CCN(C(=O)CC23CCC2CNC3)c2ccccc21 C1(CNC(c2nc(C)[nH]n2)=O)CCC2(CN(C(=O)CC3CCCS3(=O)=O)C2)O1 C(=O)(CC(C)C(C)C)NC1(CC(=O)NCCC2(OC)CCC2)CC1 CCC(C)CC(C)C(=O)NC(CC)(CC)CCNC(=O)C(F)=C(C)C1CC1 c1(C(=O)NCC(=O)NCCCC2CCCN2C(=O)Cn2ncnn2)ccccn1 c1(C(=O)NC(C2N(C(c3cnc(C(C)C)[nH]3)=O)CCC2)C)nn(C)cc1[N+](=O)[O-] C12(C(=O)NCC(C(C)C)(C)C)COCC(c3ccc(Br)cc3)(C1)C2 CC1CCCC1(C)C(N1CCCC1CNC(c1cc(=O)n(C)o1)=O)=O C1(CC(C)CC(N2C3CCC2CC(n2ccnn2)C3)=O)CCC2(CCC2)CO1 c1(C(=O)NC(C)(CNC(=O)C=Cc2ccco2)CO)ccc(C#N)cn1 C1(NC(CC2CC(=C)C2)=O)CCC(F)(CNC(=O)C(CC)=CC)C1 CC1(NC(=O)Cc2cccs2)CCC(N)CC1.C(=O)(CCCN1CCCC1)N C1(c2nnnn2CC2CCOC2)(NCc2cc(C)[nH]n2)CCCOC1 c1(C(=O)NC(CN(C(=O)CC(C)CC(C)C)CC)C)cc2c(s1)CCC2=O Cc1nc(C(=O)N(C)CC=CC(=O)NOCCO)cs1 c1(OCC)ccc(C(=O)NCC2CCN(C(=O)C=CC(=O)NC)C2)cc1C#N C1(C(=O)NCc2ccnc(C)c2)(NC(CCCNC(C)=O)=O)CCCC1C N1(C(C2C(NC(c3cc(C)sc3C)=O)CCC2)=O)CC2CC(C)C2C1 c1(C(=O)NC(CC(=O)N(C2C(C)COCC2)C)CC2CC2)ccc2ccoc2c1 c1(C(N2CCC(N(C(CC(=C=C)C)=O)CC)C2)=O)ccc(C(=O)OC)c(C)c1 C1(NC(C2C(C=C)CC2)=O)CCC(NC(c2ccc(C3CCC3)nc2)=O)CC1 C1(CNC(CCc2cnc(C)s2)=O)CN(C(c2n[nH]c(C)c2C)=O)CCCO1 C(C(C)(CC(C)C)NC(c1cc(OC)ncn1)=O)NC(C(CC=C)OC)=O C1(C(=O)Nc2cccc(C(C)=O)c2)CC(C)(C)CCN1C(c1cccnc1C)=O C1(=O)C(C(N(OC)C)=O)(CCC)NC(=O)NCCC1 Cc1ccc(Br)c(CNCC2CCCN2C(c2sc(Cl)nc2C)=O)c1 CC1CN(C(c2cncc3c2CCC3)=O)CC(C)N(C(=O)Cc2nccn2C)C1 c1(C2c3[nH]nc(OCC)c3CCC2N)ccc2c(c1)CS(=O)(=O)C2 N1(C(c2cc(C)oc2C)=O)CC2(CC2)CC1C(=O)NC12CC1COC2(C)C c1(C(=O)NCC2N(C(C3C(CC)CCO3)=O)CCC2)cccc2nc(CO)[nH]c12 C12(C(=O)NC3CCN(CCC)C3)COCC1CN(C(=O)Cc1nocc1C)C2 N1(C(=O)Cc2cn[nH]c2)CC2CC(C1)N(C(c1cccc(F)c1F)=O)C2 c1(OC)c(C(N2CCC(F)C(NC(=O)Cc3cncs3)C2)=O)c(C)nn1C c1(C(=O)NCCC(C)N(c2ccnc(CO)n2)C)cccc(-c2nnco2)c1 c1(OC)ccc(C(N)CC(=O)N2CCCC2C(=O)NC(C)(C)C)cc1 C(=O)(C(F)C(F)(F)F)NCC1CN(C(c2c(COC)cccc2)=O)C(C)CC1 N1(C(=O)Cc2cc(Br)cs2)CC2CCN(S(=O)(=O)C(Cl)(Cl)Cl)CC2C1 C1(NC(CS(=O)(=O)NC)=O)CCCN(C(c2cn3ccsc3n2)=O)C1C Cc1cc(C(F)(F)F)cc(C)c1S(=O)(=O)Nc1cc(F)ccc1O C1(C(N2CCC(N(CCC)C(c3scnc3CC)=O)C2)=O)CCN(C)S1(=O)=O S(=O)(=O)(c1ccc([N+](=O)[O-])cc1)C(COC(=O)CC1CCCC2(CCNC2)O1)=O C(C1SCCc2ccccc21)C(N1CCCC(c2ccccc2)(C(=O)OC)C1)=O C(C(CC(C)C)C(=O)NCC1CCCCS1)NC(C1CCN(CC)C1)=O c1(C(=O)NCC(CN(C(Cc2c(C)n(C)nc2)=O)C)O)ccc(Cl)nc1O c1(C(N2CCCCC(NC(Cc3c(C)noc3)=O)C2)=O)cc2n(n1)C(C)CCC2 c1(COC(C(C2C(COC)C2)CCCCl)=O)sccc1S(N)(=O)=O C(C1c2ccsc2CCN1C(=O)C(O)CC1CC1)NC(c1ccon1)=O c1(C(=O)NC2CN(C(Cc3c(C)n[nH]c3)=O)CC(O)C2)[nH]c2ccccc2c1Cl c1(C(=O)NC(C)CNC(C2CC2c2nc[nH]n2)=O)ccc(-n2ccnc2)nc1 Cc1c(C(=O)NCC(C2CCCC2)NC(=O)C(F)F)cnn1CCN(C)C CC(CNC(c1snc(Cl)c1Cl)=O)CN=c1[nH]c2cc(F)cc(F)c2o1 C(CC(C)C(=O)NCC(O)CC(=O)N(CCS(C)(=O)=O)C)OC c1(NC(N2CC3CN(C(C4C(C)OCC4)=O)CC3C2)=O)ccc2ccccc2c1 Cc1cnc(Cl)c(S(=O)(=O)Nc2nc(C(=O)N=c3cc(CCO)[nH][nH]3)cs2)c1 c1(C(N2CC(NC(C3C(C)C3)=O)C(N(C)C)C2)=O)c(-n2cccn2)nc(O)nc1C Cc1cccn2cc(C(N3CCCN(C(=O)Cc4csc(=N)[nH]4)C(C)C3)=O)cc12 C1(NC(CCN(C(CCCCSC)=O)CC2CC2)=O)CCC(=O)NC1C C(CNC(C1CCCOC1)=O)(CCC)NC(C1(C#C)CC1)=O C1(C)(C(F)(F)F)CCC(NCCCCOC2CC2)C1 C1(CC(=O)NC2CC(NC(c3c(CC)noc3)=O)C2)CN2CCN1CC2 N1(CC)CC2(CCN(C(C3(C)CC3(F)Cl)=O)CC2)CNC1=O C1(COC)CC(CNC(=O)CCC2CCCN2C)N(C(c2ccc(C#N)o2)=O)C1 C1(CC)CN(C(=O)C(C)c2ccco2)CCC1NC(c1ncc(Cl)cc1F)=O c1(C(=O)NCC2N(C(CC=CC)=O)CC(F)C2)cc2c(nc1O)C(C)(C)CCC2 C(=O)(CCC(CC)NC(c1cncc(O)c1)=O)NC1(COC)CC=CC1 c1(CNC(C=CCN(C(C(CN(C)C)O)=O)C)=O)cccc(CO)c1 c1(C(=O)NC2(CF)CCN(C(c3c(C)ccn3C)=O)C2)n[nH]c2c1CC(C)CC2 Cc1cc(C(N2CCC(CO)(CNC(C3(O)CCOC3)=O)CC2)=O)cc(C)n1 C1(CNC(C(CCN(C)C)O)=O)CN(C(c2ccc(C3CC3)s2)=O)CC(C)(C)C1 Cc1sc(C(N2CCC(C)(NC(=O)C(O)CCc3ccccc3)C2)=O)nc1O CCC(C)(O)C(=O)NOCC(=O)NCc1ccc(C)cc1 C(=O)(C(O)CC(C)(C)C)NC1C(C(N(C(C)C)CCF)=O)CCOC1 CC1CCN(C(C2(F)CCC2)=O)CC1CN(C)C.C12(CC1)N(C)C2=O C1(CC)CN(C(C2(C)C(C)(C)C2(C)C)=O)CCC1CNC(C1(C)CC=CCC1)=O C(=O)(C(C)(O)C(F)(F)F)NCCC(C)CCNC(c1ccc([N+](=O)[O-])o1)=O N1(C(c2ncc(C)cc2F)=O)CC(NC(=O)CC(O)C(C)C)CC(F)(F)C1 N1(C(c2c(C)nc(O)s2)=O)CCC2(CC(C(N3CCC(CO)C(C)C3)=O)C2)C1 c1(C(N2CCCCC(CNC(CC(C=C)CC)=O)C2)=O)cc(N)c(Br)c(F)c1 C1(NC(C2CCC(C(N)=O)C2)=O)CCCCCCC1O.CC12CCCN(C1)C2=O C=CCC(C(=O)NC1CN(C(c2ncncc2Br)=O)CC1O)C(C)C c1(CC(=O)NC2CN(C(c3n(C=C)ncc3)=O)C(C)C2)nc(F)c(F)cc1F CC1CC(C)N(C(=O)CN(C2CC(C#N)C2)C(c2c[nH][nH]c2=N)=O)C1 C(C(C)(O)CC(=O)NCCCCNC(=O)C=C(C)CN1CCOCC1)OC c1(C(=O)OCC)cnn2c1OCC(NC(=O)NC1(Br)CC13CCC3)C2 C1(C2CC2)(CNC(Cc2c(C)ccc(C)c2)=O)CCN(C(C2CCC2)=O)C1 c1(C(N2CCCC2C2CC2)C(=O)NCCOC)cc(F)cc(Cl)c1 N1(C(CN2CCC(C)CC2)=O)CC2CC1CN(C(c1cc(CC3CC3)on1)=O)C2 N1(C(C(CN(C)C)N(C)C)=O)CCC(C(=O)NCC(N)=O)C12CCC2 S(=O)(=O)(c1cccnc1NCc1ccc2nsnc2c1)NC(C1CCOC1)CC c1(C(N2C3C(NC(COCC=C)=O)C(C3)C2)=O)coc2c1C(=O)NCC(C)(C)C2 c1(OC)ccc(-n2nc(CCC(F)(F)F)nc2CCCc2ccnc(Cl)c2)cn1 c1(N2CCC(OCc3ccc(OCC)cc3)CC2)ncnc2c1oc1ccccc21 c1(COC)ccccc1C(=O)NC(CNC(=O)Cc1csc(C)n1)C1CCC1 C(=O)(C1CCC(=O)c2ccccc21)N1C(CCNC(C2CCS2(=O)=O)=O)CCC1 c1(OC)ccc(NC(C)=O)cc1NC(C1CC1C(N1CC2CCC(C1)O2)=O)=O C(=O)(C1Cc2c(Cl)cccc21)N1CCN(C(c2ncc(CC)nc2)=O)C(C)C1 C1(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)CN(C(c2ccoc2)=O)CCC12CCOC2 C(=O)(C1CS(=O)(=O)c2ccccc21)NC1(CC=C)CN(C(=O)C(S)C2CC2)C1 N1(C(C2C(C)CCO2)=O)CCC(C2CC2)C1C(=O)NCC1(n2ccnn2)CC1 c1(C(N2CCCC(NC(c3ccc([N+](=O)[O-])cc3)=O)C2)=O)nc(O)nc(O)c1F c1(N2C(C)CN(C(c3cnn(C)c3C(F)F)=O)CC2)cc(Cl)nc(S(C)(=O)=O)n1 N#CC1(c2ccccn2)CCN(Cc2ccccc2-c2cn[nH]c2)CC1 C(C(C)(C)C(=O)N1CC(NC(c2cccc(CS(C)=O)c2)=O)C(C)C1)NC(C)=O C(=O)(C(CC(C)C)CC(C)C)NCCC(C)N(C(C1CC2(ON=C(C)C2)C1)=O)C c1(CS(C)=O)ccccc1C(=O)NC1CN(C(C2(C)CCC(=O)C2)=O)CC1F N1(C(c2c(CC)n(C)cc2)=O)CCC(NC(c2cc(C)sn2)=O)C(O)C1 N1(C(CCC(=O)NCCCOC)=O)CC2CC(C1)CN(C(C1CCN(C)C1)=O)C2 N1(C(c2cc(OC)ncc2)=O)CCC(C2CCN(C(=O)C=NOC)CC2)C1 CC1CCCN(C(=O)Cn2ccc([N+](=O)[O-])n2)C1CNC(=O)Cc1nc(=N)[nH][nH]1 N1(C(C#CC(C)C)=O)Cc2ccnn2CC(NC(=O)CC(C)c2ccncc2)C1 CCC(C#N)C(=O)N1CC(NC(c2ccc(-c3ncc[nH]3)nc2)=O)C(O)C1 c1(CN(CC(C)NC(C2CC2C(C)(F)F)=O)C)ccc(F)c(Cl)c1 CCCCC(O)C(=O)NCC1CCCCN1C(=O)C(c1c(C)noc1C)C c1(C(=O)NCC2(C)N(C(CCCC#CC)=O)CCC2)[nH]cc2c(=O)n(C)ccc12 N1(C(C(C)NC(N)=O)=O)CC(O)(CCNC(c2cc(C3(C)COC3)no2)=O)C1 C#Cc1cccc(C(=O)NCC(CC=C)NC(c2cc3ncccc3o2)=O)c1Cl c1(CC(=O)NC2C(CNC(CN(S(C)(=O)=O)C)=O)CCC2)cc2ccccc2s1 C(=O)(C1COc2ccccc21)N1CCC2C(NC(C(C)OCC#C)=O)C2C1 N1(C(Cc2c(CC)con2)=O)CCC(OCCNC(C2OCC2(C)C)=O)CC1 CCC(O)C(O)C(=O)NCCOc1cccc(C)c1C c1(COC(C(C(C)C)OC)=O)c(C(F)(F)F)cccc1F C1(NC(CCCCSC)=O)CC2(C1)CN(C(=O)C(C)Sc1nnnn1C1CC1)C2 Cc1nn(C)c(C)c1C(C)C(=O)NCC(O)CCNC(=O)CSC(C)(C)C c1(CN2CC(C(N3CCC(OCC)CC3)=O)OCC2)cc(C)nc(COC)n1 c1(C(N2CC(COC)N(C(C3(CO)CC3)=O)CC2)=O)cc(Br)c(F)cc1F c1(C(N2CC(NC(COCCCC)=O)C(C)C2)=O)cc(O)nc2[nH]c(=N)ccc12 N1(C(C2(OC)CCC2)C(=O)NC2CCOC2)CCN(C(C2CC(C)(C)C2)=O)CC1 CCC(C)C(=O)NCC(=O)NCCC(=O)NCC1CCSC1 C(CNC(=O)C(C1(O)CCCCC1)CC)(C(C)(C)C)NC(C(C=C)O)=O C1(CC)CCC(c2nnnn2CCCSC)(NCC2CCCCCO2)CC1 C(=O)(CCC(CF)CF)NC1CCCC(C(N2CCC(C)(CO)C2)=O)CC1 CN1CCOC(C(=O)NCc2ccnc(C(=O)NCC(C)(C)N(C)C)c2)C1 CCC(C(=O)N(CCNC(=O)Cc1ccccc1)NC(C)=O)C(C)C.CN c1(C(=O)NCC(CN(C)C(c2cn(C)c(=O)n2C)=O)O)c[nH]c(=O)c2ccnn12 CCC(C(=O)NC1COCC1C(=O)NCC1CCCC12CC2)C(C)C c1(CC(C)NC(C(N2CCC(CC)C2)=O)=O)ccc(Cl)c(C(F)(F)F)c1 N1(C(C2CCC(CC)CC2)=O)CCCC(N=c2cnc(F)c[nH]2)CC1 CCCCC(C)(F)C(=O)NC1CCN(C(c2cc(C#N)no2)=O)CC1 c1(C(N2C(CC(=O)NC(CC)C(N)=O)CC2)=O)cnc(-c2ccccn2)nc1O CC1CC(C(=O)NCC2(C3CCC3)CC2)CN(C(c2cncc(Cl)c2)=O)C1 N1(C(C2(C)CC(=O)C2)=O)CC2(CC(C(=O)NCc3ccc(O)nn3)CO2)C1 C1(CC(NOCC(C)(C)C)=O)CCCN(C(C2CCCSC2)=O)C1 C1(CNC(=O)CCSC(F)(F)F)CC2CC2N1C(=O)Cc1ccccc1F c1(NS(C)(=O)=O)cccc(CNn2cc(-c3cnn(C4CC4(F)F)c3)nn2)c1 CC1CCC(C(=O)NCCCN(C(=O)C(F)=C2CCC2)CCO)S1 N1(C(Cn2c(C)nnn2)=O)CCC(CC(=O)NC2C=CCCC2)C1(C)C N1(C(C(Cc2ccco2)NC(CCNC(=O)CO)=O)=O)CCNC(=O)C1 C1(C(N(CCN(C(CC(COC)(C)C)=O)C)C(C)C)=O)CCC2CCCCN12 C1(NC(C(C)NC(C)=O)=O)CCOCC1NC(c1cnon1)=O c1(C(=O)NCC2CCCN(C(c3cccc(C)c3N)=O)C2)cnc2[nH]ccc2n1 C(=O)(C(COC)N(C)C)NCCCN(C(c1cnc(C)[nH]1)=O)CC c1(NCc2cc(OCC)c(OC)c(C(=O)O)c2)ccc2c(c1)CC(C)O2 c1(NC(=O)NCc2ccsc2)ncc(C(=O)NCC(CO)C2CC2)s1 CC1(C)COC(C(=O)NCC2C=CCN2C(C2CC(=O)CCO2)=O)CO1 c1(OC)ccc2c(c1)C1=NC(=NC(C)C(c3ccco3)N1)N2.C(CN(C)C)SC C(=O)(C(F)C(C)(F)F)N(CC(C)N(C(C(N1CCOC1=O)C)=O)C)C CC(CC1CCC1)C(=O)N1CCCC1CCNC(C1CN(C(=O)N(C)C)C1)=O c1(C(=O)NC2(COC)CN(C(C3(C)CC3(F)F)=O)C2)[nH]c2ccc(F)cc2c1C c1(CC(=O)NC2CCC(NC(CC(C)C)=O)C2)cccc(C(F)(F)F)c1 C1(NCC(N2C(C(C)CC(=O)O)CCC2)=O)CCS(=O)(=O)C1 c1(CC(=O)NC2CC(c3c(C(=O)OC)cccc3)C2)c(C)ncnc1C C1(CN2CC(c3ccc(C)s3)OCC2)CCC2(CCC2)CO1 c1(C(=O)NCCN(C(c2cnccc2C)=O)CC)cnc(O)cc1C(F)(F)F C(=O)(C(O)C(C)(C)C)NCC(c1ccccc1)NC(c1cc(COC)on1)=O C(=O)(CC1=CCCC1)N1C(C(C)NC(c2ccc(C(F)F)cn2)=O)CCC1 c1(C(=O)NC2(CF)CCN(C(=O)CC3CSCCS3)C2)cnc(F)c(Cl)c1 C(=O)(CN=c1cc(Nc2ccccn2)nc[nH]1)N(CC(CO)C(C)C)CC=C C(=O)(CCCCC(=O)Nc1c[nH]nc1C(=O)N(C)CCc1ccncc1)OC C1(C(=O)NC(CN(C(CNC(CC)=O)=O)C)(CO)CO)CN2CCCN1CC2 C(=O)(CCCC(F)(F)F)N(C1CCCN(C(c2c(C)ccc(N(C)C)c2)=O)C1)C C1C(C)CC(=O)N1CCN(C)C.C1(C(C=O)NCC)COCC1C(F)(F)F Cn1ncc(NC(=O)CC2(C)CCN2C(=O)CP(C)(C)=O)c1Cl CC1(CNC(C23CC(CO2)C3)=O)CCN(CCc2cccc(F)c2)CC1 C(=O)(C(CC(C)C)C(C)C)NC1C2(CCC(NC(c3c(C)ccnn3)=O)CC2)C1 O=C(C(O)C(F)(F)c1ccccc1)Nc1ncc(Cl)cn1 C1(CNC(CCS(N)(=O)=O)=O)(CO)CC12CCN(C(=O)Cc1cnoc1)CC2 c1(C(=O)NC(C2CCCN2C(C2CCC(=O)N2C)=O)C)ccc(F)nc1 c1(CC(C(=O)NCC(CN(C(C(C)OCC=C)=O)CC)(C)C)C)ccccc1C S(=O)(=O)(c1ccc(NCC2CN(C(C)C)C2)cc1Br)N1C(CC)C(C)CC1 CCS(=O)(=O)c1ccc(F)c(C(=O)N(CC(C)NC(=O)C(O)CC(F)(F)F)C)c1 c1(C(=O)Nc2cccc(CNC(C(COC)C)=O)c2)cncc(C)c1C C(CCCCCSc1ccc(Cl)cc1)N(C(=O)C(F)F)C(=O)CC12COC(C1)C2 C1(CC(=O)NCC2(COC)CN(C(c3cc(CO)[nH]n3)=O)C2)CCCCN1C c1(OC)ccc(NC(N(CC2=CCOCO2)c2ccccc2)=S)c(C)c1 Cc1ccc(C(=O)N(CC(=O)NCc2ccn(C)n2)CC2CC2)o1 C(=O)(C1CCc2c[nH]nc21)N1CC2C(CNC(C34CCC(O)(CC3)CC4)=O)C2C1 Cc1cnn(C)c1C(=O)NC1CCCN(C(C2(C#N)CCCO2)=O)C1 N1(C(c2cc(OC)no2)=O)CCC2CN(C(=O)C(C)Cc3ccco3)CC12 N1(C(C(CCC)C)=O)CCN(C(=O)CN2CCC(F)(F)C2)CC1c1ncc[nH]1 CC12CCC(C(=O)NC3C4CC5C3C5C4C(=O)NC3CNC(=O)OC3)(CO1)C2 c1(C(=O)OCCNCCSC)ccc(C)c(CO)c1 C1(C(N2CCCC2CN(C)C(c2csc3nnsc23)=O)=O)(OC)CCCCCC1 CCCC(C(=O)NCC1OCCC1C(=O)NCC#CC(F)(F)F)NC(N)=O C(CCC(N)=O)(C(=O)NCc1cncnc1I)n1cc(-c2c(C)nccn2)nn1 C#CC1CN(C(C2CCC(C)(CC)O2)=O)CCN1C(=O)CCc1cnc[nH]1 N1(C(C(C=C)(C)C)=O)CC(C2CCCN(C(=O)CC3COCC(C)(C)O3)C2)C1 C#CCCC(C(=O)N(CC(=O)NC)C)NC(C1SCC=C1C)=O C1(CC)C(NC(c2cc(C(F)F)ccn2)=O)CCN1C(C1CCOC1=O)=O CCS(=O)(=O)C=CC(=O)NC1CCCCC1CNC(c1cccc2sncc12)=O c1(C(=O)NCC(C2(O)CN(C(=O)Cn3cccn3)C2)(C)C)ccc(N)c(N)n1 n1(CC)cc(C(N2CC(CCCCNC(c3cccs3)=O)C2)=O)c2ccccc12 c1(C(N(C2CCCN(C(C3(CCCC)CCCC3)=O)C2)C)=O)occ2c1CCC2 CC(C(=O)NC(C(=O)NC1CNC(=O)C1(C)C)C(C)(C)O)C(C)(C)C C(=O)(C1=CC2(CCOC2)C1)N(CCN(C(CC(COC)(C)C)=O)C(C)C)C C1(Nc2cc(C)sn2)C2CC(O)C1N(C(c1cccc(C(=O)OC)n1)=O)C2 C1(NC(C2CC3(CCOC3)C2)=O)CN(C(C2CC3CC3C2)=O)Cc2nccn2C1 N1(C(c2ncc(C)o2)C(=O)NCC)CCC2C(O)CCCC2C1 C1(NC(Cc2c(OC)nccc2)=O)CCN(Cc2cc3occc3s2)CC1C C(C#C)(CSC)OCCNC(CNC(CNC(=O)OCC)=O)=O c1(OC)ccc2c(C(=O)NCC3CCN(C(C4CC(O)C4)=O)CC3C)c[nH]c2c1 n1(CC)ncc(Cl)c1CC(=O)NCC1CC1NC(=O)C(C)C#N C1(C(=O)NCCN(C(C2CC3CCC2CC3(F)F)=O)CC)CCC2(CCC2)CO1 C(=O)(C1=CC(C)CC1)NC1(C)CCN(C(c2cccc(C)n2)=O)C1 C1(C(=O)NC(C)(C)C)CCC(CCC(O)COC2CCOCC2)CC1 c1(CS(=O)(=O)NC(C)CCCOc2ccccc2)ccc(C)cc1 N1(C(CC(C)n2cccn2)=O)CCCN(c2ccc(C#N)cc2)CC1 C(=O)(CC(C(F)F)NC(C1(C#N)CC2CC2C1)=O)NC(C(=O)OC)(C)C C(=O)(C(C(F)(F)N)C1CCCC1)C(=O)OC(C)(C)C.CC1CC(=O)N1.C(C)(C)C N1(C(c2c(C)cn(C)c2)=O)CC(C)CN(C(C2CC(C)(C)CCO2)=O)C(C)C1 c1(OCC(=O)NCC2(COC)CN(C(=O)CCC3CCCC3)C2)ccccc1Cl Cc1noc2ncnc(N(C)CCOCCNC(=O)C3=COCCC3)c12 C(CCC(=O)N1CCCC1C1CCN(C(=O)CCN2CCC2)C1)OC(C)=O C1(O)(CCNC(C(C)(C)C2CC2)=O)CCCN(C(=O)Cc2cccnc2)C1 C=CCC(CNC(C1CC(=C)C1)=O)NC(=O)CC1(n2cncn2)CC1 C(=O)(C1CCOc2ccccc21)N1C(CNC(=O)CCc2cccc(O)n2)CC1 Cc1nc(CC(N2CC(NC(=O)CCc3cccn3C)C(C)C2)=O)[nH]c1C C(C(C)C)(C(O)C(=O)N1CC(O)(CNC(c2cc(OC(F)F)n(C)n2)=O)C1)OC Cc1cc(=O)n(CC(=O)N(C)CCNC(=O)C(CCO)N(C)C)c2ccccc12 N1(C(Cn2c(C)cc(C)n2)=O)CCC(NC(c2cc(CO)oc2C)=O)C(F)C1 N1(C(C(=C)C(F)(F)F)=O)CCC(C)(C)CC1C(=O)NCCNS(C)(=O)=O C1(NC(CCCn2nc(C)c(Br)c2)=O)CCC2(CCC2)C1CN c1(CN(C)C)ncc(C(=O)NC2CC(NC(=O)COC3CCC3)C2)[nH]1 CCC(CC1CCCCC1)C(=O)N(CCN(C)C(C1(OC)CCCC1)=O)C(C)C N(C(=NCCC(C(C)C)N(C)C)NCC1CCN(c2ccccc2)C1)CCOC CCCC(C(=O)NC1CC(NC(=O)CCn2cc(C)cn2)CC1O)NC(N)=O c1(C(C)NC(=O)C(N2CCC(SCC(N)=O)CC2)=O)cccc(Cl)c1 C1(CNC(c2c(C(C)C)onc2)=O)CC2CC(C1)N(C(c1ccc(=N)[nH]n1)=O)C2 C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1C(NC(C2(O)CCCC(C)(C)CC2)=O)CC1 Cc1ncc(C(N2CC(O)(CCNC(c3nncn3C3CC3)=O)C2)=O)c(C)n1 Cc1ccccc1C(C)CC(=O)N(C)C.C12(CC1(F)Cl)C(=O)OC2 N1(C(CC(C=C)C)=O)CC(C)(C)OC2(C1)CN(C(=O)CC1CSCCS1)C2 c1(CNC(C(N2CC3CCC3C2)c2cc(OC)ns2)=O)ccc(F)cc1 C(=O)(CS(=O)(=O)C(C)(C)C)N(C(CNC(CC1C(C)CCO1)=O)C1CC1)C N1(C(C(C2CN(C(C3N(CCC)CCC3)=O)C2)O)=O)CCC(O)C1CC C1(CN(C(COCCOC)=O)C)CCN(C(c2cnn(CCN(C)C)c2)=O)C1 c1(CC(=O)NC(C(=O)NCCSCC)C2(O)CCC2)ncn(C)c1C C1(OC)(CNC(=O)C(c2cccc(Br)c2)(F)F)CCSCC1 N1(C(C(CC)C#N)=O)CC2=C(C1)CN(C(c1cnn(CC3CCCC3)c1)=O)C2 c1(N2C(=O)CC(C(N(CCCNC(=O)Cn3ccnn3)C)=O)C2)cc(F)ccc1F c1(C(=O)NCCOCCN(C(COCC(=C)C)=O)C)cc(Cl)n[nH]1 C1(C(=O)NCc2cccnc2)CCCN(C(c2c[nH]c(=S)cn2)=O)C1 c1(C(=O)NCCn2cc(CC(C)(C)O)nn2)ccc([N+](=O)[O-])cc1 C1(NC(CCC=CCC=C)=O)CCN(C(C2CC(=O)N(CCC=C)C2)=O)C1C N1(C(CN(C2CC2)CC)=O)CCC2CN(C(c3coc(S(=O)(=O)NC)c3)=O)C2C1 C1(C(N(CCCc2ccco2)C)=O)CC2CC2N1C(c1ns[nH]c1=O)=O C1(O)(COC)CCCC1NC(C1CCCN(C(c2ccc(C)cc2)=O)C1)=O N1(C(Cn2ncc(C#N)c2)=O)CCC2CCCC12CNC(c1cc(Cl)c[nH]1)=O C(N=c1[nH]c2c(c(=NC3CN(C)CC3C)[nH]1)CCC2)C1(CC)CCCCC1 C1(CNC(C2CCC(N(C)C)C2)=O)(NC(=O)CC2(C)CC2)CCC(C)(C)CC1 C1(C(=O)NC2(CN(C(CCCn3c(C)ncc3)=O)C)CC2)CC(C)N(C)C1 N1(C(C2(CC#C)CC2)=O)CC(NC(C2CC23CCSCC3)=O)CC(F)(F)C1 c1(CC(=O)NCCCNC(C2(Cc3ccncc3)CC2)=O)c[nH]c2nccc(Cl)c12 CC1(C)CN(C(=O)C(=O)N2CCC2c2cccc(F)c2)C(CNC2CC2)CO1 CN1CC(C(=O)NC(CC2CC2)CC(=O)NCCc2ccco2)CCC1=O C(=O)(C#CC1CCC1)NCC1C(NC(CCc2c(C)n(C)nc2)=O)CCCC1 C(N=c1nc(C)c(Br)c[nH]1)C1(C)CCN(C(=O)Cn2cccn2)CC1 c1(CNC(C2(CN(C)C)CC2)=O)ccc(CNC(C2CCCN2C=O)=O)cc1 CCC(C)C(C)CCNC(C12COC(C)(C1)C2)=O C(=O)(N1CC2COCC2O1)C1C2N(C(C(C(C)C)C)=O)CC(C=C2)C1 c1(CC)ccc2cc(C(=O)NC3CC(C)(NC(C4CC4Cl)=O)C3)[nH]c2c1 c1(CN2CCC(CC(=O)N(CCOC)Cc3ccc(Br)s3)C2)c(Cl)c(C)nn1C c1(-c2cc(C)nc(C)c2)ccc(S(=O)(=O)NCC2CCC(=O)NC2)cc1C C1(C(N2CC(C)(NC(=O)C(F)CC3CC3)C2)=O)CCCC(C#N)C1 C1(NC(c2cnn(C(C)C)c2Cl)=O)CC2CC(NC(C3(CO)CCC3)=O)CC12 CC1COCCC1NC(C12CC1CCN2C(c1cnco1)=O)=O CN1N=C(C(=O)NC2CCOCC2C(N2CCC(C(C)(C)C)C2)=O)CCC1=O C(=O)(C1=CCC(C)CC1)NCC(C1CCC1)NC(c1ccn(CCOC)n1)=O c1(OCCC)cc(OC)ccc1C(=O)NC(C)CN(C(=O)C(C)C1CCC1)C Cc1cc(N(C(c2cc3sccc3s2)C(=O)NCc2nnn(C)n2)C)cc(C)c1 O=C(C1=CCS(=O)(=O)C1)N1CC(CNC(C2CC(O)C2)=O)C2CC12 C1(C(N(CCCCSC)C2CC2)=O)CC12CN(C(=O)OC(C)(C)C)C2 Cc1nc(NCc2ccc(OC(F)F)cc2)cc(=NC(C)CC(C)N(C)C)[nH]1 C(CC(C(C)C)NC(=O)CCC1CCC(=O)C1)NC(C=C(COC)C)=O C1(C(F)F)(OC)CCN(C(c2cc(Cl)ccc2C)C(=O)NC2(C)CC2)CC1 Cc1ccc2[nH]cc(CC(N3CCCC3C(C)(C)NC(C3CC3F)=O)=O)c2c1 c1(OCC=C)ccc(C(=O)NC(C)(C)C(C)NC(=O)CCCCN(C)C)cc1 c1(C(=O)NC(CC=C)CNC(C2CCC3(CC3)C2)=O)ccc(Cl)c(C)c1Cl N1(C(c2cnn(CC)c2C)=O)CCC(CO)C(NC(c2ccc3c(c2)CC3)=O)C1 N1(C(C2(c3ccccc3)C(C)C2)=O)CCC(NC(=O)CC2(C(=O)OC)CCC2)C1 CC(C(C)(C)NC(=O)Cn1nnc(-c2ccco2)n1)NC(C1CCOC1=O)=O C1(C)(C(=O)NCc2cc(C)ncc2)CCCN(CC(c2ccccc2)C2CC2)C1 N1(C(C(n2ccc(C)n2)C)=O)CCC(C)N(C(=O)C(=O)Nc2ccccc2)CC1 CC(CC(F)F)C(=O)NC1CCCC1(C)CNC(=O)C(C1CCCCC1)N(C)C C(=O)(CS(=O)(=O)C1CCCC1)N(C(C)CCNC(=O)CCc1ccon1)C c1(CNC(=O)NC2CCN(c3ccccc3)C2)c(F)cc(F)cc1F c1(C(=O)NCc2nc(C)oc2)cc(C)sc1Br O=C1CC(NC(=NCC2CC2)NCC(=C2CCCC2)F)CCN1 c1(OC)cc(NC(=O)C(=O)NCC2COCCN2C2CC2)c(C(C)=O)cc1OC C1(C(=O)NC2CCC(NC(c3n(C(C)C)ccn3)=O)C2)CCc2nc(O)[nH]c2C1 c1(C(=O)NC2C(c3cn(C)[nH]c3=N)C2)oc(=O)c2ccccc2c1-c1ccccc1 c1(C(N2CCCC(C(CNC(c3cc(C)sc3)=O)(C)O)C2)=O)cc([N+](=O)[O-])c[nH]1 c1(CC(C)C)ncc(C(=O)NCC(C)NC(c2cncn2C(F)(F)F)=O)[nH]1 CCCC(C(=O)NCCCN(C(=O)C(CC)CC)CC(C)C)OC c1(C(=O)NCC2C(NC(CCCCC)=O)CCC2)cc(C)nc2c(C)c(C)nn12 N1(C(Cc2ncn(C)c2)=O)CCC2(CCCN(C(C3CC3F)=O)C2)C1 C1(C(NNC(=O)NCCCCN2CCCCC2)=O)CCC2C(C1)C2(F)F C#CC1CC(NC(C2C=CC(NC(C3(N(C)C)CCC3)=O)C2)=O)C1 CCCC(C(=O)NC1(N(C)C)CCCC1)NC(=O)CSCC(N)=O c1(-c2occ(C(=O)NC(CC=C)CNC(=O)C(C)NC(C)=O)n2)ccccc1F N1(C(C(CC=C)N(C)C)=O)CCCC2(CCN(C(=O)CCc3cncs3)C2)C1 N1(C(CCS(C)=O)=O)CC2(C1)CN(C(c1ncc([N+](=O)[O-])cc1F)=O)CCO2 C(=O)(C1=C(C)OCCS1)NC1(CC(=O)NC(c2ncc[nH]2)CC)CC1 N1(C(CN(C)C(=O)C2CC2)=O)CCCC1(C)C(=O)Nc1ccc[n+]([O-])c1 C1(CNC(C2C(C)(C)CC2)=O)C(C2CC2)CCN1C(C1CC2(CCC2)C1)=O C(C)(CCCN=c1[nH]cc([N+](=O)[O-])cc1CO)NC(c1c(C)ccc(F)c1)=O Cc1ccsc1C=CC(=O)NC(c1ccccc1)C(N1CCCCC1CF)=O Cc1cc(C(=O)NCCCOCCNC(=O)CC(C)F)ncc1N C1(C(=O)OC)CCC1C(=O)NCCC(C)SC Cc1nc(N)c(CC(N2CCC(C)C(NC(c3cc(C)n(C)c3)=O)C2)=O)c(O)n1 Cc1cc(O)ncc1NC(=O)CC1CC(C)(C)CN1C(=O)CCCN=[N+]=[N-] c1(CNC(=O)N(CCN2C(=O)CNC2=O)C2CC2)cccc(Br)c1O C1(NC(CS(N)(=O)=O)=O)CN(C(=O)Cn2cnnc2O)CCC1O N1(C(Cc2cc(OC)cc(F)c2)C)CCC2(CCS(=N)(=O)CC2)C1 C=CC(C)(C)CC(=O)N1CC2CCC1(CNC(=O)COC1CCCC1)C2 C1(NC(CS(CC)=O)=O)CCC2(CC1)CN(C(=O)C#CC1(C)COC1)C2 C1(NC(COC2CN(C(c3c(C)cc(F)s3)=O)C2)=O)CN2CCC1(C)CC2 c1(C(=O)OC)cc(OC)c(OC)cc1C(=O)NC1CC(O)(C(F)(F)F)C1 c1(CC)sc(C(=O)NCC(C)(CO)NC(=O)C(O)C(F)F)cc1C C1(CC=C)(N(c2ccc(N)cc2)C(C2CC2(C)Br)=O)CCN(C(=O)CC)C1 CC1(C)CN(C(=O)CCN2CCCC2)CC1NC(=O)Cc1ccon1 c1(OC(C)C(=O)NC2CC(NC(=O)CC3COC(C)(C)C3)C2)cccc(F)c1 C1(CNC(c2ccc(-c3ccco3)[nH]2)=O)COCCN(C(=O)CC2CCCO2)C1 N1(C(c2c(C)c[nH]n2)=O)CCC2(COCC(CNC(=O)C(F)=C3CCCC3)O2)C1 N1(CCNC(CC2C(C)CCC2)=O)CCN(C(c2cn(C)[nH]c2=N)=O)CC1 C=CCCCCC(=O)NC(C1CCCN1C(c1cnc(O)c(F)c1)=O)C N1(C(C2(F)CCN(C(c3c(OC)ccc(Cl)c3)=O)C2)=O)CCc2cccnc2C1 c1(NC(C2N(C(c3nc(COC)oc3)=O)CC(O)C2)=O)cccn2ncnc12 CC(CC(=O)N1CCCC1C(=O)NCCC12CC(CO1)C2)C1CC1 c1(CC(=O)NCC2C(CNC(=O)CC3CCOCC3)CCC2)c(F)cccc1F C1(CNC(c2c[nH]c(=NC)o2)=O)C(C)CCCN1C(c1cccnc1O)=O c1(NC(=O)NCc2c(OCC)nccc2C)cc(C)c(F)cc1Cl O(NC(=O)C(C)(C)CCNC(=O)CC(C)n1cccc1)CC(C(C)C)O C=C1CC2(C1)CC(C(=O)NCC1(O)CCN(C(C3(C(F)(F)CC)CC3)=O)C1)C2 C1(F)(C(=O)NC2CCC(NC(c3n[nH]c(C)c3C)=O)C2)CCN(C)CC1 Cc1cc(C=CC(N2CC3CN(C(=O)C(O)C(F)(F)F)CC3C2)=O)ccc1F c1(N(c2ccccc2)C(C)=O)nnc(-c2ccco2)n1CC(C(C)C)N(C)C c1(C(N2CCC(C)OC(C)C2)=O)coc2c1N(C)C(=O)CCC2 NS(=O)(=O)c1ccc(C(=O)NCCC2CCCN(C(C3(CF)CCC3)=O)C2)cc1 C1(CC(=O)NC2C(CNC(C(C)(C)N3CCOCC3)=O)C2)CCCC(O)C1 CC(CC(N)=O)C(=O)NCCCC1(CNC(C2CC2CN(C)C)=O)CCCC1 N1(C(C(COC)(C)C)=O)CC2(NC(c3ccc[n+]([O-])c3)=O)CCCC2(F)C1 c1(C(=O)NC(CNC(CCNC(c2cccc(C)c2)=O)=O)C)cc2n(n1)CCC2 O=C(N=NCC(=O)NCC(C1CC1)NC(=O)C1CC1)N=c1cc[nH]cc1 N1(C(C(N2CCCC(CSC)C2)=O)=O)CCC2(CCCOC2)C1 C(=O)(C(C#N)C(C)(C)C)N(CCCNC(c1cc(C(F)(F)F)ccn1)=O)C(C)C C1(NC(C(n2ccc(C)n2)C)=O)C=CCN(C(c2cccnc2N)=O)C1 Cc1ccccc1C(N1CC(NC(=O)Cc2ccccc2C(F)(F)F)C(O)C1)=O C(=O)(CC(O)CC(C)C)NC1CC(OCC(N2CC(CC)OC(C)C2)=O)C1 C(CCCCCCCO)=CC(=O)NC1C=CC(CNC(CC(C(C)C)O)=O)C1 c1(C(N(C(CC)C(=O)N2CCCC2CC)C)=O)ccnc(C)n1 C1(NC(C(COC)(F)F)=O)CC2CC1N(C(=O)COCc1ccnn1C)C2 C1(C)(NC(CC(C)SC)=O)CCN(C(=O)CC(C)(C)NC2CCCC2)C1 C(C)(CO)(C(C)(C)O)NC(CNC(CC)=O)=O C1(C(CC(N2CCCC(c3nc(C)c(C)[nH]3)C2)=O)N)CCC(F)(F)CC1 c1(C(C(=O)N(CCN(C(C)C)C(C2CCCS2(=O)=O)=O)C)C)cccc(Cl)c1 N1(C(c2nnn(C)n2)=O)CCCC2(C1)CN(C(=O)CCCC1CCCO1)C2 C(=O)(CC(O)CC(C)C)NCC1C(C(N2CC(CC)C2)=O)CC1 C1(CNC(c2ccc(CCC)[nH]2)=O)CC2CCC(C1)N2C(C1(O)CCOC1)=O n1(CCC(=O)NC(C2CN(C(=O)C3=COCCO3)C2)C)ncc2ccccc12 C(=O)(C(F)(F)CN(C)C)NC(C)Cn1cc(CCN(C)C)nn1 N1(C(c2cc(C)c(C)[nH]2)=O)CCN(C(=O)Cc2cccn2C)CC1C(F)F C(=O)(C#CC1CCCCC1)NC(C(C(C)C)C)CNC(C12CCC(CC1)CC2)=O C(=O)(CCCC(CC)NC(C)=O)N(CCN(C(=O)C=C1CCCC1)CCC)CC c1(OC)ccc(OC)c(C(=O)NC(C2CN(C(c3cccn(C)c3=O)=O)C2)C)c1 c1(N2CC(NCc3ccccc3)OCCC2)ncnc2cc[nH]c12 N1(C(c2cc(C)c(C3CC3)cc2)=O)CC2CC(NC(=O)C=CC3CC3)CC2C1 c1(C(=O)NC(CNC(c2cc(C)nc(C)c2)=O)(C)CO)cnc2sc(C)c(C)n12 Cc1ccc(C)c(CN(C)C(C2CCCC2NC(C2C=CCCC2)=O)=O)c1 CC1=C(C(=O)NCCCCN(C(=O)CCc2ccc(O)nc2)C)CCS1(=O)=O C1(C(=O)NC2CC(C)C2)CCCC1NC(c1nc(Cl)cs1)=O C1(CCNC(C(F)=C(C)C)=O)CCN(C(=O)CCCCCF)CC1(F)F CC1CC(C(N2CCOC(CN(C(=O)CN(C)C(=O)C3CC3)C)C2)=O)CCN1C c1(OC)ncccc1S(=O)(=O)Nc1nc(-c2cnoc2)cs1 N1(C(COCCOC)=O)CCC2CN(C(c3ccnc(OC)c3)=O)C2C1 N1(C(c2cc(OC)c(C)cc2)=O)CC(NC(=O)C(N)=O)C2(CCOCC2)C1 c1(OCC)ccc2c(c1)CC(C(=O)NCc1coc3c(F)cc(F)cc13)CO2 c1(C(=O)NC2(C)CCN(C(=O)CSCc3ncc[nH]3)C2)cccn2nncc12 CC(C)(C)CCC(=O)NCC(F)CNC(C1CCCOC1)=O c1(C2CC(c3ccc(CC)cc3)C2)nc(CO)c2c(n1)CCCC2 c1(C(=O)NCC2(O)CN(C(CCc3ccc(C)cc3)=O)C2)cc(C)c(C#N)cn1 c1(C(N2C(C(C)NC(C(C)=CC)=O)CCC2)=O)ccc(C)cc1OC Cc1nc2ccccn2c1C(=O)NC12CC(NC(C34CCC(C)(C3)OC4)=O)(C1)C2 c1(CC)[nH]c(=N)sc1C(=O)NCC1(C)CC(NC(=O)Cc2ccco2)C1 c1(Sc2ccc(OC)cn2)ccc(C(N2CCCC2(C)CO)=O)c(C)n1 CCC(CC(=O)NC(C)CCNC(=O)CCc1nc(C(C)C)no1)SC c1(C(=O)NC(c2ccccc2)C)ccc(S(=O)(=O)NCC2(O)CCOCC2)cc1 C1(C(N2C(C3CCN(C(C4(C=C)CCC4)=O)C3)CCC2)=O)Cc2cccc(F)c2O1 C1(NC(c2ccc(O)cc2)=O)CC2CC1CN(C(c1cn(C3CC3)cn1)=O)C2 c1(C(=O)NC(CCNC(C)=O)Cc2ccccc2)sccc1S(=O)(=O)C(F)F C1(COC)(NC(c2c(C)nn(C)c2C)=O)CCN(C(=O)C(C2CC2)N(C)C)CC1 N1(C(C(C)Oc2cccnc2)=O)CCC2C(C1)CN2C(=O)CCc1nccs1 N1(C(CCC(=C)Cl)=O)CCC(CNC(C2CC2c2cnn(C)c2)=O)C1(C)C c1(C(=O)NC2CC(SCCNC(C3N(C)CCC3)=O)C2)ccc(NS(C)(=O)=O)nc1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC(NC(C2(C#N)CCC2)=O)C(C)C1 C1(CC)CCN(C(=O)C(C)OC)C1C(=O)NOCc1sc(C)nc1C C1(CCC(=O)OC)CCCN(C(c2ccccc2C(C)C)C(=O)NCC(C)C)C1 C(c1ncccc1C)=CC(=O)N(CCC)CCNC(C1CC1(C)Br)=O N1(c2nc(C)nc(C)c2F)CC2(CN(C(=O)CC3CCCS3(=O)=O)CC2CO)C1 c1(C(C(=O)NCC(C(C)C)NC(=O)C(F)F)OC)ccccc1Br N1(C(C(C=C)CC)=O)CCCC(C(=O)NC(c2ccccc2F)C)CC1 CC(C#N)C(=O)NC1CCOC1C(N1CCC(C(F)F)C1)=O CC(CNC(C1(CO)CCC1)=O)CC(=O)NCC=C1CCSCC1 CC1CCCN(C(c2cc(Cl)nc(Cl)c2)=O)C1CNC(=O)CC1CS(=O)(=O)C1 Cc1cc(CSCC(=O)NCc2cc(-c3ccco3)no2)cc(C)c1OC(F)F CC1(C)CN(C(=O)COCC=Cc2ccccc2)CC1C(=O)O c1(CNC(=O)NCCNC(CC(CC)C)=O)ccc(Cl)cc1C(=O)OCC Cc1sc(N)c(C(=O)NC2(CCO)CCCSC2)c1C CC(CC1CCC1)C(=O)NC1CC(C)(NC(c2ccco2)=O)C1 CN1CC(NC(=O)CCC(C)(C)NC(=O)CCC(=O)NC2CC2)C2(CC2)C1 c1(NC(C2C(NC(Cc3cccc(C)c3)=O)C2)=O)cnc(Br)c(Cl)n1 C(=O)(C(CC#CC)NC(c1cccc(OC)n1)=O)N1CCC(C#C)C1 C(CN=c1cc(C)[nH]cc1C(=O)OC)C1N(C(c2ccc(CC)s2)=O)CCCC1 N1(C(CC(=O)N(C)C)=O)CCN(C(C2(C)COCC2(F)F)=O)CC1CO Cc1ncc(C#N)cc1NC(C1(C(C)NC(=O)C(C)N(C)C)CC1)=O c1(-n2ccc(C(=O)NCC(N(C(CC=C)=O)C)C3CC3)n2)ccc(F)cc1 c1(-c2cn(CC(C)NC(C3CCCC(=O)N3C)=O)nn2)cc(Cl)c(N)c(Cl)c1 CC1(C)C(CC(=O)NC2(c3cn(C(C)(C)C(=O)O)nn3)CCCOC2)CC1O C1(O)(CN(C)C(c2cc(C(F)F)cs2)=O)CCN(C(C2(N(C)C)CC2)=O)C1 C1(OC)CC(CNC(=O)CNC(C)=O)(NC(C2CCSC2)=O)C1 C(=O)(C(C)(C(C)C)OC)N1CC(F)(CNC(c2c(CC)c(C)sc2)=O)C1 S(=O)(=O)(C1CCOCC1)N1CCC(O)(C(=O)NCCCN2CCCCC2=O)CC1 c1(C2CN(OC(C(C)=CC)=O)C2)c(C)cccc1Cl C1(NC(=O)Cc2cc[nH]n2)CCC2(C1)CN(C(c1c(C)nc(N(C)C)s1)=O)C2 C1(OC)CCC12CC(C(N1CC(NC(c3nc(Cl)sc3C)=O)C1)=O)C2 O(NS(=O)(=O)c1ccc(F)cc1)CC1CC(c2ccc(C)cc2C)(C(=O)O)C1 c1(OCC(=O)NC2C(NC(c3c(C)snc3)=O)CCC2)ccc(F)cc1Cl C(=O)(C(C)(C)C(C)O)N1CC(CCC)C(C(=O)NC2CN(C3CC3)C2)C1 CC(c1ccccc1F)=CC(N1CCC2(NC(=O)Cc3cc[nH]c3)CC2C1)=O CCN=c1[nH]c(C(=O)NC2CCN(C(=O)C(C)(COC)OC)CC2CO)cs1 CC(C)(CN=c1[nH]c(=NCC2CC=CCC2)c2ncccc2[nH]1)S(C)(=O)=O N1(C(CCc2c(C)n[nH]c2C)=O)CCCN(C(c2csc(O)n2)=O)C(C(C)C)C1 C1(C(N2CCC(NC(C34CCC(CC3)C4)=O)C(F)C2)=O)CN2CCCC2CO1 C(=O)(CC1=CCN(C(C2C3CCCCC23)=O)CC1)NCc1n(C)cnn1 c1(NC(c2cc(-c3ccoc3)on2)=O)nc(-c2ccccc2)cs1 N1(C(CCOCCOCC)=O)C2CCC1C(CNC(=O)C(C)c1cccs1)C2 N1(CCC)C(=S)NC(c2cn3cc(F)ccc3n2)C(C(=O)OC)=C1C1CC1 Cc1nonc1C(=O)NCc1nc(C(=O)N(C)Cc2cnco2)co1 C(C)(CNC(=O)C=CCCC(C)C)(C(C)C)NC(C(Cc1c(C)nc[nH]1)O)=O O=S(=O)(CCN=c1[nH]c(=NCC2CCCSCC2)[nH]c2c1COC2)C(F)F C1(C(=O)O)CCCN(Cn2ccc(-c3cccc(F)c3)n2)C1 CC1CN(C(C2(C(C)(F)F)CC2)=O)CCC1CNC(c1ccncc1O)=O C1(C(N2CCC(O)(CNC(CSC(C)C)=O)C2)=O)CCc2nnnn2CC1 C1(CNC(C2C3CCCOC23)=O)CCC2(CCC2)CN1C(=O)CC1(CO)CCC1 C1(OCCN(CCOCc2ccc(C(=O)O)cc2)C)(CO)CCC(CC)CC1.CC N1(C(C2CCN(CC)C2)=O)CCC(O)(CN(C)C(c2csc(C)c2N)=O)CC1 N1(C(C(C)n2ccnc2)=O)CCC2(CCC2)C(CNC(c2cnn(C)n2)=O)C1 c1(CCNC(C2CCCCC2)CCC)nc(N(C)C)cc(N2CCOC(C)C2)n1 N12CC3(CC1CO3)NC1CC3C(C3C1)C2=O.C(=O)(C(C)(C)C(=O)OC)OCC C#CC1(N(CCCCCC)C(=O)CNC(=O)C(C)(C)Cl)CCCC1 c1(CN2CC3N(C(C4C(C)CCC4)=O)C3C2)cccc(Br)c1F C1(C(CNC(c2cc(C(N)=O)[nH]c2)=O)F)CCN(C(C2(CF)CC2(F)F)=O)CC1 N1(C(C(=O)NCCCCNC(C=C(C)C2CC2)=O)C)C(=O)CCC1=O c1(N(CCCNC(CCc2onc(CC)n2)=O)C2CC2)cc(O)nc(O)n1 C1(CNC(C=COCC)=O)CN(C(=O)C(C)Cc2ccco2)CCCO1 C1(CCNC(C(CN(C(C2C(CCC)C2)=O)C)C)=O)CCCC12CC2 N1(C(c2cnc(CC(C)(C)C)o2)=O)CCCC(NC(=O)C(C)(O)C2CCC2)CC1 c1(C(=O)NC2(C)CC(NC(=O)CCF)C2)ccc(-c2cccs2)cn1 Cc1cnc(CNC(C2CCCCCC2NC(=O)CCCOC(C)C)=O)c(C)c1 CC1CCC=C1C(=O)NCCC1CCN(C(C2CCCCN2C(C)C)=O)CC1 Cc1cc(C(N2CC3CCCCCCC23)=O)cc([N+](=O)[O-])c1 N1(C(C)=O)CCN(CC(=O)N(C(C)(C)C)C2(c3ccno3)CC2)CC1 C1(C(=O)NCC2C(NC(c3ccc[nH]3)=O)CC2)CC(=O)N(c2cccnc2)C1 C1(NC(C2(OCC)CC2)=O)Cc2ccccc2C1NC(C1CC(C(C)C)=NO1)=O n1(CC)cc(S(=O)(=O)NC2(c3ccccc3OC)CC2)c([N+](=O)[O-])n1 N1(C(c2c(F)ccc(C)c2)=O)CCC(C)(C)CC1C(=O)NC(C1CCC1)C c1(C(N2CC(NC(CC(C)(F)F)=O)C(C)(C)C2)=O)cc(F)cc2ccccc12 Cc1ccc(Cl)c(CNCC23CCCC2C3)c1 c1(NC(=O)C(=O)Nc2ccc(Br)nc2)cccc(C(F)(F)CF)c1 N1(C(c2c(OCC)cccn2)=O)CC(NC(C2COC2)=O)CC2(CCOCC2)C1 CCCCC(F)C(=O)NCC1(OC)CN(C(=O)CN(CC)CC)C1 Cc1[nH]c(C#N)cc1C(N1CC(C)(C)CC1CNC(C1CC(N(C)C)C1)=O)=O c1(NC(C23CC(NC(C4C5CCC(F)C45)=O)(C2)C3)=O)ncc(F)cc1F c1(N(CCCN(C(C(C)C2CCOC2)=O)C)C)nc(N(C)C)nc2c1CCC2 c1(C(=O)NCC(CNC(c2ccnc(C)c2Br)=O)C)cccc2c1CCN2 N1(CCNC(C=CCN(C)C(c2ccnc(O)c2)=O)=O)C(=O)CCC1=O C1(C(N2CC(NC(=O)CCC3CCC3)C2)=O)CCCCC1n1cc(Br)cn1 c1(C(=O)NCCOCCN(C(=O)C2=CCC2)C)cc(N)c2ncccc2c1 C12(C(N(C)CC3CN(C(C4(C)CC4(F)F)=O)CCO3)=O)CCCC1C2(F)F n1(CC(=O)NC2C(NC(Cc3cccc(C)c3)=O)COC2)ncc2cccnc12 C1(NC(C2C(C)(C)C2C(=O)NC2CCC2CO)=O)CCCSCC1 Cc1ncc(NC(=O)C(C)NC(=O)C(C)CSc2ccccc2)cc1C#N c1(CNC(C(C)C)=O)cc(C(=O)NCc2nc(=O)o[nH]2)n[nH]1 C1(C(N2CCCC(N(C(c3scnc3C)=O)CC)CC2)=O)CCc2nnnn2C1 N1(C(CC2ON=C(C)C2)=O)CCC=CC1C(=O)NCC(c1ccsc1)C C1(C(=O)NC2CCCC2C(=O)NCC(=O)N(C)C2CC2)(CC)CCCC1O C1(O)(CCNC(C2CC(C)OC2)=O)CCN(C(C2(C)CCNC2=O)=O)CC1 Cc1[nH]ccc1NC(=O)CCOC1CN(C(=O)CN2CCSCC2)C1.C1CO1 N1(C(C2(C(CC)=O)CC2)=O)CC(NC(=O)Cc2cccc(OC)n2)C2CCCCC12 N1(C(C(C)OCCCC)=O)CC(C2(NC(=O)CCCCNC(N)=O)CC2)C1 c1(C(=O)NCC2(CNC(C3(CSC)CCC3)=O)CC2)cc2cccnn2n1 C1(N(C(CCOCCOC)=O)C)CN(CC)C(C)(C)C1.C12C3CN(CC13)C(=O)C2 N1(C(C(n2c(C)ccn2)C)=O)CCCCC(NC(=O)CN2CCN(C)CC2)CC1 C1(C(=O)NC(C(=O)NCC)C)(CC)CCCN1C(c1ccncc1)=O N1(C(C)=O)CCCC1(C)C(N1CC(NC(=O)C=Cc2ccsc2Br)C1)=O N1(C(c2cccc(C)c2Cl)=O)CCC(C2CC(NC(=O)Cc3csc(Cl)c3)C2)C1 c1(OC)ccc(S(=O)(=O)CC(C)C(=O)OCC2COCCN2C(C)=O)cc1 c1(NC(CC2CCN(C(c3cnc(C(C)N)s3)=O)C2)=O)cccc(F)c1 CC(C)CCC(F)C(=O)N1CCCC1C(C)(C)C(N1CCC(C=O)CC1)=O.N(C)C C1(NC(c2nc(OCC)oc2)=O)CC2CC1N(C(=O)C(c1nc(C)cs1)C)C2 c1(C(N2C(c3c(C)n[nH]c3C)CCC2)=O)ncc2conc2n1 C1(N(CC(=O)OCC)CCOC)CCCC(C)C1.C(C(F)F)SCC N1(C(C2CC(SC)C2)=O)CC(C)(C)OCC1CNC(=O)Cc1n[nH]c(C)n1 CC(C)(C)C(CC(=O)NC1(CCF)CC(O)C1)NC(C1CC2(CCC2)C1)=O c1(CN2CC(CC)N(C(c3ccsc3C)=O)CC2)cc(Cl)c(O)c(Cl)c1 C(CCCCC(=O)NC1CS(=O)(=O)CC1NC(C1CC(=C2CC2)C1)=O)OCC c1(N2CCC(CSC)C2)nc(C)cc(=NC(C)c2nncn2C)[nH]1 c1(CCC(=O)NC2(C)CN(C(=O)CN3CCCC3)C2)cc(Br)ccc1F c1(CC)nc2ccccc2cc1C(=O)NC1CCC(NC(=O)Cc2csnn2)C1 c1(OC)ccc(CN2CCC(N(C)C(c3cc(F)ccc3C)=O)C2)c(OC)n1 C1(CC=C)(NC(c2csc([N+](=O)[O-])c2)=O)CCN(CCCC2CCOC2)CC1 C1(CC)C(NC(C2(F)CCCCC2)=O)CCCN1C(c1cscc1SC)=O c1(C(N2CC(CC(=O)NCCC(C)(C)C)OCC2)=O)cccc2c1CCCC2 C(=O)(CC(C(C)(C)C)NC(=O)C1=C(Cl)CCC1)N(C)Cc1cnco1 C1(CNC(C(C)O)=O)(CO)CCN(C(C2CCCSC2)=O)CC1 c1(CC)noc(C(=O)NC2CCOCC2NC(=O)COCc2ccncc2)c1C C1(C(=O)NC2(CC=C)CN(C(=O)CC(O)CN(C)C)C2)CC(=O)N(CC2CC2)C1 C1(NC(C2C(COC)CN(C(=O)CCCn3cccn3)C2)=O)CC2CCC1CC2 c1(Cc2nc(C(N(CC)CC)C)on2)ccccc1[N+](=O)[O-] C(=O)(C(C)CC=C(C)C)NC1(CCNC(CCCSC)=O)CC1 C1(C(=O)NCCCN(C(c2c(CC)noc2)=O)C(C)C)CCCCC1O c1(C(=O)NC2CCCCN(C(CCOC)=O)C2)cc(OC)cc2ccccc12 c1(C(N2CC(SCCOC)C2)=O)[nH]nc2cc(Cl)c(Cl)cc12 C12(C(=O)NC3CCC(NC(C4CCCS4)=O)CC3)CCCN(CCC1)C2 c1(C(N(CC(CNC(C2(CC)CCCCC2)=O)C)C)=O)nn(C)c2c1CCCC2 C(N=c1cc(C)nc(N(C)CC2(C)CCCO2)[nH]1)c1c(C)nc(CCC)o1 CC1CN(C(C2(CCNC(C3CC3C(F)(F)F)=O)CC2)=O)CCS1=O c1(C(N(C(CC(=O)N(C(C#C)C2CCC2)C)C)C)=O)ccc(C)n1C Clc1ccc2[nH]cc(CNCC3CCC34CCC4)c2c1 C(C)(C(C)(C)C(C)(C)O)NC(C)OCC(COC)(C)O C(=O)(CCS(=O)(=O)N1CCC(C(=O)NCc2ccc(C)c(OC)c2)C(O)C1)OC N1(C(C=CSC)=O)CCCC2(CNC(=O)CC(C)n3ccnc3)CCCC12 C1(C(CNC(C(C)(C)O)=O)(C)C)CCCCN1C(c1ccnc(OCCO)c1)=O C1(C(C)NC(CC(C)C2CC2)=O)CCN(C(c2ccncc2C(F)(F)F)=O)CC1 C(=O)(C1CCCc2nnn(C)c21)NC(C)CNC(=O)C(C)n1ccnc1 C(=O)(CCN(OC)C(=O)CC1CCCC1(F)F)NC(C=C)C1CC1 C(=O)(CCCCCC(C)O)N1CCC(NC(CCOCCC)=O)(COC)C1 C(=O)(CCC(C(C)C)NC(C1CC2CCC(C1)O2)=O)NCCCCC(=O)OC C1(NC(C2C(O)CCN2C(C2CC3(CSC3)C2)=O)=O)(CO)CCCCCC1 c1(-c2cc(C(N(CCC(C)NC(c3nocc3Cl)=O)C)=O)[nH]c2)ccc(Cl)cc1 C1(OC)(CNC(C2CC2c2ccncc2)=O)CCN(C(=O)CCC=CBr)C1 C1(CC)COC(C)(C)CN1C(C1CN(C(=O)COC2CC2)CCO1)=O N1(C(C(C)OCc2ccccc2Cl)=O)CCN(C(c2n[nH]cc2Cl)=O)C2CCC12 CN=c1[nH]cc(C(=O)NCC(C)(C)CN(C(=O)C=Cc2ncc(C)[nH]2)C)s1 C1(NC(c2c(C)coc2)=O)CCN(c2nc(C3CCCCC3)ns2)CC1O N1(CC(=O)NCC2CN(C3CC3)C2)CCC(O)C2CCCCC12 c1(CNC(c2cccnc2)CC)ccc(N2CC(F)(F)C2)nc1 CC1(O)CCN(Cc2cnn3c2CCC3)CC1F.C12CCCC1NC2=O CCCC(C(=O)NCC(C1CC1)NC(c1cc[nH]c1C1CCC1)=O)OC Cc1cc(C)c(C(=O)NC2(C)CCN(C(C3(C#N)CCOC3)=O)C2)o1 N1(C(C(C2CCOCC2)C)=O)CC(O)CC1C(=O)NCCP(C)(C)=O N1(C(C2(CC#C)CCC2)=O)CCC(C)(CNC(=O)CCn2cccn2)C1 C1(C(=O)NCCC#CCC)CCN(C(=O)c2ccc(F)cc2C)O1 Cc1nc(N2CCC(C)C2CNC(c2n[nH]c(C)c2Cl)=O)c(F)c(C)n1 N1(C(c2c(CC)nns2)=O)CCC(O)C(NC(=O)CC2CCCOC2)C1 c1(C(=O)NC2(CNC(CCSCC)=O)CCC2)ccc2c(c1)CCC2=O C1(C2CN(C(c3cc(O)cc(Cl)c3)=O)C2)(NC(CNC(CCCCC)=O)=O)CC1 c1(OC)cc(C(=O)NC(C)CCN(C)C(C2CC(CCO)C2)=O)ccc1OC c1(C(=O)NCCCN(C(=O)COc2ccn(C)n2)C(C)C)n[nH]cc1[N+](=O)[O-] O=[N+]([O-])c1ccc2c(c1CNCc1csc3cccc(F)c13)CCN2 Cc1nc(O)nc(O)c1CC(=O)NCC(O)CNC(c1ccc(S(N)(=O)=O)o1)=O c1(C(N2CC(CN(C(=O)CSc3ccccn3)C)OCC2)=O)cc(N)cc(Cl)c1 C1(NC(C(C)(C)OC(C)=O)=O)C=CCN(C(=O)C(c2ccnn2C)O)C1 N1(C(Cc2c(C)nc(O)nc2C)=O)CCC2CC1CN(C(=O)CC(O)C(C)C)C2 C(=O)(C(C)(C)CC#C)NC1CCCC(NC(C(C)NC(CC)=O)=O)C1 N1(C(c2cnc(CCC)o2)=O)CCN(C(=O)C(C)O)C(c2ccc(F)cc2)C1 N1(C(C2CC3(CC(OC)C3)C2)=O)CCC2(CC(NC(c3ncccn3)=O)C2)C1 N1(C(c2c(C(C)C)n[nH]c2)c2nnnn2CCCF)CCC2(C1)CC2(F)F C(=O)(C(C)(C)CCOC)NCCCN(C(CCCCOC)=O)C C(=O)(CC(C)(C)C(=O)N1CCC(F)(CNC(c2cc(F)c(F)cc2F)=O)C1)OC CC1=C(C(=O)NCCC2(CNC(=O)CCn3ccc(C)n3)CC2)CCCC1 O=C1CCC(C(=O)NCC#CCNC(=O)CSC2CCCCO2)C1 C1(C(N(C2CCN(C(C(CC)C(C)C)=O)C2)CC)=O)CCc2c(ncn2C)C1 C#CCC(CC(=O)NCc1cc(C)c(C)o1)NC(C1(OC)CCSC1)=O CC(C(=O)NC(C(=O)NCc1ncco1)C1(C)CC1)=CC(C)(C)C Cc1ccc(NC(=O)CCN(C(=O)Cn2cnnn2)C2CC2)cc1Cl N1(C(c2ccnc(OC)c2F)=O)CC2CN(C(C3(C)CC=CC3)=O)CC2(C)C1 C1(C(=O)NCCCSCC)CC(C)N1C(=O)Cc1cnc(C)s1 N1(C(CCN(C(C(n2ccc(C)n2)C)=O)C)=O)CC(C)C(C)C1C C(=O)(C(C)CC(C)(C)C)N1C(CNC(c2cnc(NC(C)=O)o2)=O)CC(F)(F)C1 c1(C(CCNc2n(CC)c(CC)cn2)=O)cc(F)ccc1F c1(C(=O)NC(C(C(=O)OC)O)C)cc(C(F)(F)F)cc2nc(C3CC3)[nH]c12 C1(NC(C(CCC)O)=O)CC2CC(NC(=O)CCSc3ccc(C)cc3)C1C2 N1(C(CC=CC=C)=O)CC2CC2(CNC(=O)CN2CCCC2=O)C1 c1(C(N2CC(NC(c3c(C)ncnc3)=O)(CO)C2)=O)ccnc2[nH]cnc12 Cn1ccc(C(C(=O)NC2COC2)N(C2CC2)Cc2ccccc2)c1 Cc1cc(C(=O)NCC2CN(C(=O)Cc3csnc3C)C2)c(C)s1 c1(C(=O)OC)csc(C(=O)NCC(C)CNC(=O)C(c2cncn2C)O)c1 CC1(C)COC(CC(=O)NCC2CC(NC(=O)C(C)(C)C3CCCC3)C(O)C2)C1 C1(O)(C(N(CC#C)C)=O)CCN(C(c2cccnc2)=O)CC1 C#CCCCCCC(=O)NC1CCCCCN(C(c2cscc2C(F)(F)F)=O)C1 CCC(C(=O)NC1(c2cn(CCC=C(C)C)nn2)CC(F)(F)C1)C(C)C c1(CNCC2C(c3n(CC)nnn3)CC=CC2)cnc2n1CCC2.C1(S)CC(C)(C)CO1 C(C)(CCCCN=c1nc(C)c(C(=O)OC)c[nH]1)NC(C(C=C)(C)C)=O c1(CC)ccc(OC)cc1C(=O)NCC1CN(C(=O)Cc2ncc(C)cc2F)C1 c1(C(=O)NCC(CNC(Cn2nc(C)c(Cl)c2)=O)O)cc(C)n(C(C)C)c1C Cc1cc(C#N)cc(C(N2CCCC(CO)(NC(=O)C=Cc3ncc[nH]3)C2)=O)n1 c1(CC(=O)NC(CC)CNC(=O)CN2CCSC(C)(C)C2)csc2nc(C)cn12 c1(N2CCN(CCOC(C)C)CC2)nc(=NC2CSC(C)C2)[nH]c2c1CCC2 Cc1cc2nc(C(=O)NCCC(C)NC(=O)CCc3cncn3C)cn2cc1C C1(CC=C)(N(C(=O)C(C)=C2CCC2)CCC(=O)C(C)(C)CF)CCCCC1 c1(CCC(=O)NC(C(=O)NCC(C)(C)F)Cn2cccn2)c[nH]c2cnccc12 c1(OC)cc(NC(N2CCN(C(=O)C(=O)N(C)C)CC2)=O)c(F)cc1C#N C1(F)(CNC(C(C2CCN(C(=O)Cc3ccc[nH]3)C2)C)=O)CCCCCC1 c1(NC(c2ccc(COC)c(Br)c2)=O)sc2c(c1C(=O)O)CCC2 c1(OCC)ccnc(N(C(C)CCNC(=O)C(C)=CC2CC2)C)n1 C(=O)(NNc1ccc(S(=O)(=O)C(F)(F)F)cc1)C1CCC(NS(C)(=O)=O)C1 CN1CCC(CC(N2CC(F)CC2C(N2CC(C)(C(F)(F)F)C2)=O)=O)C1=O C1(O)(C(C)NC(c2cc(Cl)n[nH]2)=O)CCN(C(=O)CN2C(C)CCC2C)CC1 C(=O)(C(C)(O)C(F)(F)F)NCCC(C)NC(c1cccc2occc12)=O CC1(C(=O)NCC(O)C(=O)NC2(CO)CCOC2)CC(=O)C1 c1(C(=O)NCC(CC)NC(=O)C(C)(C)CO)cc(Cl)c(F)cc1Br c1(C(N2CCC(C(C)(C)NC(C(C)=C3CC3)=O)C2)=O)ccc(Cl)cc1 C(=O)(CCCCC(=O)NC(CCF)C(=O)N1CC(OC)C(F)C1)OC Cc1cc(C)c(C(=O)NCC2CCN(C(=O)C(c3cccc(Cl)c3)O)C2)o1 C1(OC)CC(c2nncn2C)N(C(c2cn(C3(N)CC3)nn2)=O)C1 C12CN(CCO1)C2=O.c1(N(CC(C2CCCC2)=O)C)ccnc(S)n1 C(CCC(C)CC(=O)N1CCC(CC(=O)Nc2cccnc2Cl)CC1)=C(C)C N1(C(c2c(C)snc2)=O)CC2CC(NC(C34CCCC3CCC4)=O)CC2C1 CCC(C)C(C(=O)N1CCCCC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C1)NC(C)=O Cc1ccc(C(=O)NC2CCC2NC(c2cnn(CCO)c2N)=O)cn1 c1(CNC(CN(C(C(c2ccccc2)C)=O)C2CC2)=O)ccc(=O)n(C)c1 C(c1cccc(Cl)c1)=CC(=O)NCC1(F)CCCN(C(C2(CO)COC2)=O)C1 C(=O)(CCC(F)(F)C(F)F)NC1CC2(CC(CNC(CC(C)SC)=O)C2)C1 Cc1ccc2c(CC(=O)NC3CCCCC3N(C)C(C3CC3C)=O)coc2c1 c1(C(=O)NC(CCOC)CNC(=O)C(C)NC(C)=O)cnn2cccnc12 c1(C(=O)NCC2C(NC(=O)Cn3cccc3)CCCC2)cnc2ccccn12 N1(C(C(CC)OCC)=O)CC2CCN(C(c3ccc[nH]3)=O)C2C1C C(CC(C)(C)C(=O)N1CC(CC)OCC1C)NC(CCCOCC)=O c1(C(=O)NC2C(NC(C(CC)=CC)=O)CCCC2)nnc(O)c(Br)c1O C(=O)(CC(F)F)NCCC1CC(NC(C2CC(n3cnnc3)C2)=O)C1 C=CCCC(C(=O)N1CCN(C(=O)NC)CC1)NC(C1CC(C)(C)CN1C)=O C(=O)(CCC(=O)NC)N(CC(C)(C)CNC(C1CCSC(C)C1)=O)CC C1(CNC(C(CCC)CC)=O)CC2(CCN(C(c3c(Cl)cnn3C)=O)CC2)CO1 c1(C(N2CCC(N(C(c3ccc(Cl)o3)=O)CC)C2)=O)cncc(P(C)(C)=O)c1 C1(CNC(C2CC(CCC)C2)=O)CN(C(c2cc(N)c(F)cn2)=O)CC(C)(C)C1 CS(C)(=O)=Nc1ccc(C(=O)NC2CCCCN(C(C3CC3(F)F)=O)C2)nc1 C1(C(=O)Nc2ccc(C(=O)NC3CC3)cc2)CC1C1CCCCC1 c1(N(C(=O)CCN(C(=O)C=CC(C)(C)C)CCO)CC)ncoc1C Cn1ncc(Cl)c1C(N1CC(NC(C2CC2F)=O)CC1CO)=O C1(C(=O)NCCC(C)F)CCC(C)(C)N(C(=O)C=CC(C)(C)C)C1 Cc1ccc(CC(=O)NCCN2CCN(C(c3cc(O)no3)=O)CC2)cc1F C1(C(C)(C)NC(C(C2CC2)OCC)=O)CCCN1C(=O)CC1CC1 C1(NC(C(CCC)C)=O)CN(C(c2[nH]cnc2C#N)=O)CCC12CCC2 Nc1ccc(F)c(C(N2CC(NC(C3CS(=O)(=O)C3)=O)CC3(CC3)C2)=O)c1F C1(Nc2cc(OCC)ncn2)CN(C(=O)Cc2ccc(Cl)c(F)c2)C(C)(C)C1 C1(O)(C(C)NC(CSC(C)C)=O)CCCN(c2nccc(-n3ccnc3)n2)C1 N1(C(C(CC2CN(C(C3CC(O)(CC#C)C3)=O)C2)F)=O)CCNC(=O)C1(C)C C1(C(N(C)CC2N(C(C(C(C)C)=O)=O)CCCC2)=O)CC1C1(C)COC1 Cc1cc(F)ncc1NC(c1cc(-c2cncc(C(F)F)c2)[nH]n1)=O Cc1cc(CC(N2CC3(C2)CN(C(=O)CC2CC(=O)C2)C3)=O)ccc1CO N1(C(c2ccnc(C)n2)=O)CC2CC(CNC(c3cnsc3)=O)CC1C2 C1(CCNC(CC=CC)=O)CCCCN1C(=O)CCSCCC c1(C(N2C(CNC(C3(OC)CCCCC3)=O)CCC2)=O)cc(C(C)C)cc(F)c1 C1(C)(C(=O)NCC(CC=C)NC(c2cc(C(C)(F)F)on2)=O)CC(C2CC2)=NO1 CON1CC(C(=O)NC(C(=O)N2CCS(=O)CC2C)C(C)(C)C)CC1=O CCC(C)(C)CN=C(NCc1ccco1)N(C)CC(C)(CC)OC C1(N(CCC)C(c2nsc(OC)n2)=O)CCN(C(=O)CC2CCC2OCC)CC1 c1(C(N2C(CN(C(=O)CC(C)F)CC)CCCC2)=O)nc2ccccc2nc1C c1(C(C)=O)c(O)cccc1F.C1(CN2CCC3C2CC(=O)OC3)CCS(=O)(=O)CC1 C#Cc1cccc(C(=O)NC2CC(C)CN(C(c3ncn(C)n3)=O)C2)c1F C1(C(=O)OC)(OC)CCSC1.C1(=O)CSCCN1CCOC.C1(=O)CN1 CC(C)(C(=O)NCC1(CNC(c2cc(Cl)no2)=O)CCC1)C1CCCCC1 c1(CN(C2CCCCC2)Cc2ccc(F)cc2)cc(F)ccc1Br c1(C(C(=O)NCC(CO)NC(C(=O)NCC)=O)(C)C)ccc([N+](=O)[O-])cc1 c1(OCC(C)N(C(c2ccc(CC)o2)=O)CCOC)c(C)cc(C)cc1C n1(CC)nnc2c1CCC(C(=O)NC1CC13CC(NC(c1cc(Cl)no1)=O)C3)C2 C=C(C)C1CCC(C)(O)C(NC(=O)NCCN2CCC(NC(C)=O)CC2=O)C1 n1(CCC(=O)OCC)nnnc1C(C(C)(C)N1CCOCC1)NCCSC(C)C O=C(CCCCC(F)(F)F)NCCCC1CCCO1 C1(C(N(CCCC)CCCO)=O)C2CC3C(C2N(C(C2OC4CCC2C4)=O)CC)C13 N1(CC(c2ccc(OC)cc2)NCC(=O)NCC#N)C(=O)c2ccccc2C1=O c1(OCC(N2C(CC)CC2)=O)ccc(F)nc1OC.c12ccc(cc1)CN2C C12(NC(c3c(C)con3)=O)CCCC1N(C(=O)CCOCC(C)(C)C)CC2 Cc1nn(C)c(C)c1OCC(=O)NC(C)C(C)NC(c1cc(C2CCC2)[nH]n1)=O O(NC(=O)C(C)(CSC)NC(=O)Cc1cnoc1)CC(=C)C c1(CC(=O)NC2CN(C(c3c(N)cccn3)=O)CC2F)ccc2nn[nH]c2c1 N1(C(C(C)OC)=O)CC(N=[N+]=[N-])CC1C(=O)N(C1CC(C)(C)C1)C Cc1cc2c(C(N3CC4CC4(CNC(C4CCC(=O)C4)=O)C3)=O)ccc(C)c2[nH]1 C(=O)(CCCCC#N)N1C(C(C)(C)NC(C2N(CC(C)C)CCC2)=O)CCC1 N1(CC(=O)N(C(C)C)C(C)=O)CCN(C)C(CNC(=O)CCC2CC3CCC2C3)C1 N1(C(c2n(CC(C)C)ncc2)=O)CC2CC1CN(C(c1nnc(C(C)C)s1)=O)C2 c1(C(N(C)CC)=O)cccc(NC(C2CSC(C(F)(F)F)C2)=O)c1 C1(CN(CCCN(C(c2cn(C(C)C)nc2)=O)C)C)CC(C)(C)CO1 Cc1nc(F)ccc1C(=O)NCCOC1CN(C(=O)CC2CCC(=O)N2C)C1 C1(NC(c2nc(OCC)oc2)=O)CCN(C(=O)C(CC)N(C)C)C1C C1(CSC)CC(OC(C)(C)C)CN1C(C1CCOC(C2(C(=O)OC(C)=O)CC2)C1)=O N1(C(C(C(C)C)(C)c2nn[nH]n2)=O)CCC2(C=CCO2)C1 Cc1cccc(C(N2CCN(C)C(C(=O)Nc3conc3C)C2)=O)c1C C(c1ccc(NC(=O)Cc2ccc(C(N)=O)nc2)nc1)=CC(=O)OCC C#CC1(OCC(N2CCC(C(C)NC(=O)Cc3cnc(C)s3)C2)=O)COC1 C1(C(=O)NCC(n2cc(-c3ccn(C)n3)nn2)C)CNC(=O)O1 c1(CNC(C(Cc2ccoc2)NC(Cc2cn(CC)nc2)=O)=O)cccc(C)n1 CN1C(=O)CN(C(c2nc(Br)sc2C2CCOC2)=O)c2ccccc21 C1(NC(C(CCC)NC(N)=O)=O)C2CCCC1CC(NC(c1c(C)nsc1N)=O)C2 N1(C(C(=O)OCCNC(Cc2ccc(OCC)cc2)=O)C)CCC(CC)CC1C N1(C(C2CC(C(C)(C)C)C2)=O)CC(NC(C2(F)CC=CC2)=O)CC2(CCC2)C1 Cc1oc(S(C)(=O)=O)cc1C(=O)NCCC1(O)CN(C(=O)CC=C(Cl)Cl)C1 c1(CC(N2C(Cc3cn(CCCN(C)C)nn3)COCC2)=O)cc(Cl)ccc1O n1(C(C)C)ccnc1CNC(=O)C(C1CCCCC1)NC(=O)CCOC(C)C N1(CC)CCC2CSCC2C1.N12CCOCC1C2.c12cnc(cn1)c(=O)[nH]2 C(C(CNC(=O)CC(C)c1ccco1)CO)NC(C1(COCC)CC1)=O c1(CNC(CCCNC(C)=O)=O)n[nH]c2c1CN(C(C1CC1(C)C)=O)CC2 N1(NC(C(C)(CC)Nc2n(CCCOC)nnn2)=O)CCCC(C(F)(F)F)C1=O N1(C(CC)=O)CCC2C(C1)NC(=O)CN2C(c1cc([N+](=O)[O-])oc1C)=O N1(C(C(C)SCC(c2cnn(C)c2)O)=O)CCN(C(=O)C2CC2)CC1 C(C1CCCCCC1)=CC(=O)N(C1CCCCN(C(c2c[nH]nc2Br)=O)C1)C N1(C(CN(C(C)=O)C2CC2)=O)CCOCC1CCNC(SS(C)(=O)=O)=O c1(SCC)nccnc1C(=O)Nc1cccc(CNC(=O)C(CC)OC)c1 C1(C(N(C2CCC(CNC(C3CC(C)OC3)=O)CC2)C)=O)CCC2(C1)CC2(F)F n1(CC)ccc(C(N2CCOCC2CNC(c2cnc(COC)s2)=O)=O)cc1=O c1(CC(=O)N(C2CCN(C(=O)CCc3ccccn3)C2)C)sccc1Br CC(C)(O)C#CC(=O)NCCCOCCCNC(=O)C(C1CCCO1)C1CC1 N1(C(C=CCC)=O)CCCC(N(CCF)C(c2csc(-c3ccccc3)n2)=O)C1 O=C1CC2CNC1=CC=C(Br)C=C2OCC1CCC(C(F)(F)F)C1 c1(C(N(C2CN(C(c3ccn(CCF)n3)=O)C2)C)=O)c[nH]c(-c2ccncc2)n1 CC1(CCO)CCN(CCSc2cccc(Cl)c2)CC1 C1(NC(CC2C(C)OCC2)=O)CC2(CCN(C(=O)CCSC(F)(F)F)CC2)C1 N1(C(C(=Cc2ccccc2)CC)=O)CC=C(CCNC(C2CC2F)=O)CC1 c1(CC(=O)NCC(CC)NC(c2cccc(OC)c2)=O)cn2cccc(C)c2n1 C(=O)(CCC(F)(F)F)NCCCCCCNC(Cn1ncc(CC)c1)=O N1(CC(=O)NC(CN(C(=O)CCC2CCOC2)C)(C)C)CCCC1CO C(C(C)(O)CC(=O)NCCC1CCN(C(=O)C(C2CCCCCCC2)O)C1)OC c1(OC)ccc(C(N2CC=CC2CNC(=O)CC2CC2(Cl)Cl)=O)cc1O C12(CCNC(CC)=O)CCC(C1)N(C(=O)CN1CCCC1CO)C2 CC1(C(=O)NCCCCCNC(=O)CCc2cn[nH]c2)CCC(=O)NC1 C1(NC(C2C(CC)C2)=O)COC2(C1)CN(C(=O)C(C)(C)C(C)(C)O)C2 c1(C(=O)Nc2scc(C(=O)NC)n2)c(-c2ccccc2)noc1C.C1(=O)CCN1 C1(NC(Cc2nc(C)sc2)=O)CCCC(N(C)C(c2cc(Br)co2)=O)C1 CC(CNC(C1(NC(N)=O)CC1)=O)C(F)C(=O)N=c1ccn(CCO)[nH]1 c1(C(N2CC(NC(C3(N(C)C)CCC3)=O)C3C2C3)=O)cc2n(n1)CCC2 C1(CNC(C(C)NC(N)=O)=O)C2CCC(C2)N1C(=O)CN1CCN(C)C(=O)C1 C1(C(=O)NCc2ccc(CN(C)C(C3(O)CC3)=O)cc2)CCn2ncnc2C1 c1(C(N(CCNC(CC2CC(=C)C2)=O)C)=O)cc(OC)cc(F)c1 CCCCCCC(C)C(=O)NCC(O)C(=O)NCc1ncc[nH]1 C(CNC(=O)C(c1cncnc1)C)(C(=O)NOCCCOC)OC C=C1CCC(NC(=O)CC2CC2CNC(=O)CN2CCCNC2=O)CC1 c1(C(=O)NC2CCC(C)N(C(=O)CN3CCSCC3)C2)ccnc2ncnn12 c1(C(c2n(CCOC)nnn2)NCC2(C)C=CCCC2)ccc(C)n(C)c1=O CCC(CO)CN=c1[nH]c2c(c(=NCCN3CCS(=O)CC3)[nH]1)COC2 C=CCN=c1[nH]cc(C(=O)Nc2nc(CC(=O)OC(C)(C)C)cs2)s1 CCC(CC(=O)NCC1(CC(=O)NCC2CC2(F)F)CC1)CC(C)C c1(C(=O)NC2C(NC(C(C(CC)C)NC(C)=O)=O)COC2)ccc(F)c(C)c1C#N O=C(CC1CCC(NC(c2coc(C3CC3)n2)=O)C1)NOCC1CC1 c1(-c2cccc(C(CO)NC(c3cc(C)cc(F)c3)=O)c2)ccc2nccn2c1 Cc1cc(C(F)F)oc1C(N1CCC(NC(=O)CCCCc2cnn[nH]2)C1C)=O N1(C(C23CC(CC)(C2)C3)=O)CCCC(CNC(=O)Cc2cccc(OC)n2)CC1 N1(C(c2cnc(CC)nc2)=O)CCC(C(=O)NCC(C2CCCCC2)C)C12CC2 c1(C(N2C(C)CC(NC(C3OCCC3(C)C)=O)CC2)=O)cc2cnccc2o1 C1(CC)CN(C(C2CCCNS2(=O)=O)=O)CCN1C(=O)COC(F)(F)F c1(OC(C)C)nc(C(=O)N(CCCNC(=O)C(F)(F)C2CC2)C)cc(O)n1 c1(OC)nccc(C(=O)N(CCC(F)(F)F)CCC2CCCNC2)n1 c1(C(=O)NC(CC)(C)CNC(=O)C(C)C2(O)CC2)cc(F)ccc1Cl C(CC1=CCN(C(=O)C(O)C2CCC2)CC1)NC(C(C=C)(C)CC)=O C12(C(N3CCC(F)(CNC(C45CC(C)C4C5)=O)C3)=O)CCC(CC1)CC2 N1(C(c2cn(CC)nc2C)=O)CCCCCC1CNC(c1n[nH]cc1F)=O CCCC(C(=O)NC(C)CCSC)NC(c1[nH]nnc1C1CC1)=O N1(CC)CC(CNC(C2CCN2C(=O)CCCc2cccc(Cl)c2)=O)OC1=O c1(C(=O)Nc2ccc(NC(C3(CC)CCCO3)=O)cc2C)cnn2c1CCCC2 CC(C(C)(C)C)=CC(=O)NCC1CCN(C(=O)C(F)(F)C2CC2)C1 C1(c2nc(CC(C)OC)nn2-c2ccc(C(C)C)cc2)CCC(=O)N(C2CC2)C1 N1(C(CC2CCN(C(C3N(CC)CC3)=O)C2)=O)CCCC(C)(C#N)C1 CCC(CC(=O)N1CCCC1C(C)NC(=O)C=CC(F)(F)F)c1ccccc1 C1(C(=O)NCCCC(C)(C)NC(C2CCCN2N=O)=O)(CC)CCOCC1 N1(C(Cc2cc(C)sc2)=O)CCC(O)C(NC(=O)C=C2CN3CCC2CC3)C1 N1(C(c2cc(CCC)[nH]n2)=O)CCCCC1C(=O)NCCCC1(O)CC1 CC(C)CC(C(=O)N1CCC(C(=O)N(C)Cc2ncnn2C)(C(C)C)C1)C(C)C N1(C(=O)NC(C(CC)O)C)CCC2(C1)CC2(F)F CC(C(F)C(=O)NCCN(C(=O)Cc1ccc(Cl)cc1F)C)C(F)(F)F C(=O)(C(C)(C)C(O)CC)NC1C(CC)CCN(C(=O)OC(C)(C)C)C1.C1CCO1 N1(C(c2c(OC)ccnc2F)=O)CC(CNC(C2CCC2(F)F)=O)OC(C)(C)C1 C1(CC)CN(C(=O)CN2CC(C)(OC)C2)CCN1C(C1CN(C(C)=O)CCO1)=O c1(C(=O)NCCC2(NC(CC3C(C)=NNC3=O)=O)CCC2)cncc([N+](=O)[O-])c1 c1(C(=O)NCC(CO)NC(CCc2cnn(C)n2)=O)ccc(N)cc1F C(=O)(C1=COCCC1)NC1CC(C(=O)Nc2c(C(C)=O)csc2)C1 C(=O)(C#CC1CCCC1)NCC(N1CCN(C(C2(C)CNC(=O)C2)=O)CC1)=O N1(C(Cc2n(C)ncc2)=O)CCC(NC(=O)C2=CSCCO2)CC1C1CC1 CC(C(CO)NC(=O)CCc1ccco1)NC(C1CCCC1c1nc[nH]n1)=O c1(C(C)=O)ccc(C(=O)NC(C2CCCCN2C(c2cc(CF)on2)=O)C)nc1 c1(CC(=O)NC2CC3COCC3N2)cc(F)cc2c1OCOC2 CC1CCN(C(=O)CC2CC2)C1CNC(c1cnccc1Br)=O C(CN=c1[nH]c(=NCC2CC(C)CO2)c2ncccc2[nH]1)c1cc(C)c(Br)cc1 c1(CC(=O)NCCN(C2CC2)Cc2n(C(C)C)ncc2)ccc(Cl)c(Cl)c1 C(C)(C(=O)NC1(CC(C)C)CCC1)NC(C)=O.c1(CC=CC(=O)NC)ccsc1 c1(NCC(C(C)(C)C)NC(C(CCC)OC)=O)cc(=O)n(C)c(O)n1 N1(C(c2cccc(CC)n2)=O)CC(C(=O)NCC(C)(C)C)CCC1(C)C N1(C(CSCC=C)=O)CC(NC(=O)Cn2ncnn2)C2(CCS(=O)(=O)CC2)C1 CNS(=O)(=O)NCC(=O)NCC(C1CCCC1)NC(=O)CCNC(N)=O C(=O)(CC(CC)CCC)NC1(CC=C)CCN(C(c2cc(Cl)cc(Cl)c2)=O)C1 c1(C(=O)NCCN(C(CC(CC)SC)=O)C(C)C)ccc2ncc(Br)n2c1 c1(C(=O)NCC(CO)NC(c2n(CC)ncc2)=O)cc(C)n(C(C)(C)C)n1 N1(C(c2n(C)c(O)nc2)=O)CCC2(CNC(C3(S(N)(=O)=O)CC3)=O)CCCCC12 c1(NC)ccc(NC(=O)C(CSC)OC)cc1.N12CCOC(C1)CCC(=O)NO2 C1(C(=O)NC(CC)(CNc2cc(=O)n(C)c(O)n2)CC)CCOC2(CCC2)C1 c1(NCC(=O)NCC(c2ccccc2)N(C)C(c2cnsn2)=O)cncc(N)c1 N1(C(C2CC(OCC)C2)C(=O)NC(C)CC)CCOC(CN=[N+]=[N-])C1 c1(CC)nnc(C)cc1C(=O)NCC(C(C)C(C)C)NC(c1cc(C)c(C)[nH]1)=O c1(CNC(=O)NCC2(c3ccc(Cl)cc3)CC2)noc2c(F)cccc12 N1(CC)CCC2(CC1)CCN(c1ccccc1SC)C2.c12ncc(s1)[nH]c2=O CCN=c1[nH]c(C(=O)NC2CN(C(=O)CNC(=O)C(C)(C)C)CC2C)cs1 CC1(C)CCC(C(N2CC3(NC(=O)CC4(O)CCOC4)CC2C3)=O)C1 C(=O)(C(O)C(C)C)NCCN(C(=O)C(CC)n1cncn1)CCC c1(-c2c(SC)scn2)ccc2c(c1)CN(C(C1CC(O)CN1)=O)CC2 Cc1cccnc1-c1cn(CC(F)CCN2CCN(C(=O)C3=CCC3)CC2)nn1 c1(OC)ncc(C=CC(=O)NCC(C)NC(c2ccc(=O)n(O)c2)=O)cn1 C1(F)(C(=O)NC(c2cc(C)cc(C)c2)CC(=O)OC)CC2(CCC2)C1 C(CC(C)(C)C)(c1n(CCCSC)nnn1)NCC1CC1(Br)Br C12(NC(C3C(N=[N+]=[N-])COC3)=O)CCC(CC1n1cc(C(C)(C)OC(=N)O)nn1)C2 Cc1ncc2n1CC(C(=O)NC(C)CNC(=O)CCC1CCCOC1)CC2 C(=O)(CC1=CCN(C)CC1)NC1CCC2(CNC(CCC(=O)NCCC)=O)C1C2 C1(C(=O)NCCCN(C(=O)C(C)(C)C2CCC2)C)CC1C1CCOCC1 C1(CNC(C(c2ccccc2)SC)=O)CC(NC(C23CC(C)(C2)C3)=O)C12CCC2 CC(C(=O)NCC(C1CCCCC1)NC(=O)C(C)(C)CN1CCN(C)CC1)C(F)F CC1CCCCCN1C(C1CCN(C(C2CCNC2=O)=O)C(C)C1)=O C1(N(C(CN2CC(C)(CC)C2)=O)C)CCCCC1C C1(N(C(=O)C(O)CSC)CCOC)CCN(C(C2(OC)CCSCC2)=O)CC1 c1(N2C3CC(CF)CC2CC3)nnc(C2CCCn3cnnc32)n1C1CCC1 C1(N(C(=O)COC2CC(F)(F)C2)C)CN(C(C2CCC3(CC3)C2)=O)CC1O N1(C(C(N=S(C)(C)=O)=O)=O)CC(NC(c2ccc(=N)[nH]n2)=O)CC12CCCOC2 C1(NC(CSc2n(C)ccn2)=O)CN(C(c2cnco2)=O)C2(CCCCCC2)C1 c1(N(CCC)CCN2CCCC2)ccc(COC)o1 C=CC(CC)CC(=O)N1CCCOC(CNC(c2csc(C(N)=O)n2)=O)C1 c1(C(=O)NCC2(OC)CN(C(c3nnn(C(C)C)c3C)=O)C2)cccc(C#N)c1 c1(OC)ccc(C(N2CC3CC2C3NC(c2sccc2SC)=O)=O)cc1C(F)F c1(CCC(N2C(CCC)CN(C(C3SCCS3)=O)CC2)=O)cnc2ccccn12 C1(C(F)(F)C(=O)NCC2C=CC(NC(C3CCC3(F)F)=O)C2)(OC)CCCC1 C(N=c1nc2scnc2c(NCC(=O)N(C)C)[nH]1)N1CC(c2cccc(C)c2N)C1 C1(C(=O)NCCC(C)N(C(c2nn(CC)c(C)c2)=O)C)CC12CCCCCC2 CCC(O)CC(=O)N1CCSCC1C(=O)NC1(CCCCO)CC1 C(c1cccc(F)c1)=CC(=O)NCC12CC(NC(C3CCNC(=O)C3)=O)(CO1)C2 C1(C(N2CC(NC(c3ccc(C)cc3O)=O)C(C)C2)=O)CCCC1P(C)(C)=O c1(C(N2C(C)(CNC(CC=C)=O)CCC2)=O)cc2c(C(C)C)nn(C)c2s1 N1(C(C(N(C(CCC=CCC=C)=O)C)C2CC2)=O)CCCCN(C)CC1 c12nocc1CNC1CN(C1)C2=O.C1(N(C(=O)CC(O)C2CC2)C)CCCCC1 c1(-c2c(Cc3ccc(F)cc3)scc2)ccc2oc(Cl)cc2c1 N1(C(C2CC(C)(C)C2)=O)C(CNC(=O)CCn2ccccc2=O)CC2COCC12 CC1=NOC(C(=O)NC2CC(CNC(=O)Cc3coc(C(F)F)n3)C2)C1 C1(CNC(C2(C(=O)OCC)CCO2)=O)CC(C)CCN1C(=O)CCCCC1CC1 C1(C(N(C(C)CNC(C2CC3CC2CC3O)=O)C)=O)CC2(CCCCC2)C1 c1(-c2cc(C(C)Nc3cccc4c3OCO4)c(Cl)nc2)ccc2ccn(C)c2c1 C(=O)(C#CC(=O)N1CC(NC(=O)C(C)(O)C2CC2)C(O)C1)N(C)C N1(C(c2cnc(Br)n2C)C(=O)NC(C(=O)OC)C)CC2CC1CS2(=O)=O c1(C(=O)NCC(C)(CO)NC(CC(C=C)C)=O)ccc([N+](=O)[O-])cc1 Cc1cc(C)c(C(=O)N(C2CN(C(=O)CC3CCOC3C)C2)C)c(C)c1 c1(C(N(CCNC(=O)COCP(C)(C)=O)CC)=O)cc(C)c(C)[nH]1 Cc1c(NC(C2CN(C(=O)COC3CCCCC3)CCC2O)=O)cccc1F C1(CNC(CCc2nnc(C(C)C)o2)=O)CCN(C(C2CC2(F)F)=O)C12CCC2 N1(C(C=CC(C)(C)SC)=O)CCCCC1C(C)NC(c1cc(Cl)cn1C)=O C(C)(c1cccc(Cl)c1)=CC(=O)N(C)CC1N(C(CCCCCC)=O)CCOC1 N1(C(C(=O)N(C)Cc2cnc(-c3ccccc3)s2)=O)CC2CC3CC(C2)CC1C3 CC#CC1CN(C(C2COCCC2NC(C2CCC3(CC3)C2)=O)=O)C1 C(c1ccccc1)=C(CC)C(=O)NC1COCC1NC(=O)CN(C1CCSC1)C C1(NC(c2cnc(Cl)c(Cl)c2)=O)CCN(Cc2ncccc2C(F)(F)F)CC1F C1(C(N2C(CC(=O)NC(c3ccn(C)n3)CC)CCC2)=O)CC(C(C)C)=NO1 N1(C(c2c(C)ncn2C)=O)C(C)C2CC1C2NC(c1ccc(=O)oc1)=O C1(CN(C)CC2(C)CC=CCC2)CCCN(C(C2(C3CCC3)CC2)=O)C1 N1(C(CCCNC(=O)CC2CCC=CCC2)=O)CCC(O)CC12CC2 CC12CCCN1C2=O.c1(C(=O)NCC2(N3CCCC3)CCC2)ncsc1C1CC1 C1(C)(CC(=O)NCC(C)N(C)C(c2cc(-c3ccc(Cl)s3)[nH]n2)=O)CCCC1 C1(NC(=O)COCC(F)F)C2CC1N(C(c1ccc(Cn3cc(Cl)cn3)o1)=O)C2 C1(C(N2CC(NC(C(CCCC)C)=O)C2)=O)(OC)CCCC(C)(C)C1 C1(CC(=O)OCC)CCCCN1C(N1CC(NCC)C1(C)C)=O c1(C(=O)NCC=C2CCN(C(=O)CC3(O)CCOC3)CC2)nc2c(s1)COCC2 c1(C(N(C2CCCCC2)CCNC(C2CC23CC3)=O)=O)ncc2[nH]ncc2n1 c1(OC)cc(C(=O)NC(C)C(C)NC(c2c(C)nsc2Br)=O)n(C)n1 N1(C(C(C2CCN(C(C(C(C)C)NC(C)=O)=O)C2)(C)C)=O)CCSC2(CCC2)C1 C1(O)(CNC(=O)C=Cc2nc[nH]n2)CCN(C(=O)CCCC2CC2)C1 C1(CNC(c2nc(CC)oc2)=O)CN(C(=O)CCCn2nc(C)nc2C)CC1C c1(OC)c(C(=O)NC2CCN(C(c3cnn(C(C)C)n3)=O)CC2O)occc1=O C12(CNC(C(CC)C)=O)CCC(NC(c3ccnc4c3CCO4)=O)(CC1)CO2 N1(C(C(c2ccnn2C)NC(C2CN(C)C(=O)C2)=O)=O)CCC2C(O)CC12 c1(C(N2CC(NC(=O)CCCc3cccnc3)C3C2C3)=O)cc(O)cc(F)c1F c1(C(N2CC(F)(CNC(c3c(C)onc3)=O)C2)=O)cc(-c2cccs2)ncn1 CC(C)CC(O)C(=O)NCC(CC1CC1)C(=O)NCC1C(C)C1C c1(OC(C)C)ccc(CC(=O)NC2CN(C(c3cccc(N)c3)=O)C2)cc1 n1(CC)cc(C)c(C(C(=O)NCC2CCOC2)N(C(C)COC)C)n1 c1(C(=O)NC2C(CNC(=O)CC3CCCO3)C2)cc([N+](=O)[O-])n[nH]1 c1(NC(C(C(C)C)CNC(c2cccc(O)c2F)=O)=O)cc(C#N)ccc1O c1(CC)nc(C)sc1C(=O)NCC1CN(C(=O)CC2CNC(=O)O2)C1 C1(CC(c2cccc(C)c2C)NC(CCC)C2CCCC2)CCC(F)(F)CC1 N1(C(c2n(CC)ncc2Cl)=O)CC2CCC(C1)N2C(C1CCCN1C(=O)NC)=O N1(C(CCSCCC)=O)CC(C(C)(C)O)(CNC(C2CC2Cl)=O)C1 Cc1ccn(CC(=O)NC2CCN(C(=O)COC3CC(F)(F)C3)C23CC3)c(=O)c1 c1(-c2n(-c3ccn(CC)n3)nc(CCC(C)C)n2)cccc2cnnn12 Fc1ccc2scc(CNC(=NCC(F)F)NCc3ncccc3F)c2c1 c1(NC(c2[nH]cc(C(N)=O)c2)=O)ccc2nc(S)oc2c1 c1(CN2CC3(C(C(=O)Nc4c(C)ccc(Br)c4)C3)C2)nc2ccccc2[nH]1 C1(C)(CN(C)C)CN(c2nnc(CSC(F)F)s2)C1.CCCCCN(CC(=O)OCC)C c1(C(N2C(C(C)NC(CSCCOC)=O)CCC2)=O)cnc2ccc(F)cn12 C1(c2nnnn2CCCNC(C2CSC2)=O)(OC(C)C)CCCOC1 C1(N(C(=O)CCSc2nncn2C)C)CN(C(c2cc(CF)on2)=O)CC1O c1(C(N2C(CC(=O)NCCCCCN=[N+]=[N-])CC2)=O)cccc2ccoc12 CCCC(C)CCN=c1[nH]c(N2CCC3(CC2)CN(C)C3)nc2c1CC(C)CC2 c1(COC)ccc(C(c2nnnn2C2CCCC2)NCC2(C#N)CC2)o1 CC(C)(C#N)CCCC(=O)N1CCC2(CC2)CC1C(N1CCC(CCO)CC1)=O c1(N2CCC(CCC)(CO)C2)cc(N(C)C)nc(NCC2CCC(C3CC3)C2)n1 N1(C(C2CCN(CCC(C)(C)O)CC2O)=O)CCC2(CC1)OCC(C)(C)CO2 c1(OC)cc(C(N2CC(CNC(=O)Cc3nccn3C)C3(CC3)C2)=O)cnc1O C(=O)(N=c1cc(Cl)c(C#N)c[nH]1)C1CC2(C(CNC(=O)OC(C)(C)C)C2)C1 CC1CCC(O)CN1C(=O)CC1(CNC(C2CC(C)(C)C2)=O)CC1 C(C(O)CC(=O)NCCN1CCCCC1=O)NC(CCc1cn(C)nn1)=O C1(C(=O)NCC(CCC)NC(C2CCN(C(C)C)CC2)=O)CCS(=O)(=O)N1 C1(=CC(=O)N(C)CC2(NC(C(c3c(C)cccc3)C)=O)CC2)CCC(C)(C)CC1 N(C(=NCC#Cc1cnn(C)c1)NCC1CCC1)CCCc1c(C)cccn1 N1(C(CNC(=O)OC)=O)CC2CN(C(=O)C(c3ccc(F)cc3)N(C)C)CC2C1 C(=O)(C1OCCc2c(O)cccc21)NCC1CC(NC(c2cc(C)nn2C)=O)C1 N(C(=NCCC=CBr)NCC1CCS(=O)(=O)N1C)CC(=C)C C1(CNC(c2cc(CC)oc2C)=O)CCCCCN1C(=O)C=C1CCCC1 c1(OC)ccnc(-c2cn(C(C)C(=O)NCC(c3cnc[nH]3)C)nn2)c1 Cc1nc(C(=O)NCC(O)CCNC(=O)COc2ccccc2O)c(=O)[nH]c1C n1(CC(=O)NCC(N(C(=O)C=C2CC2)C)C2CC2)cncn1 CC1CCOCC1C(=O)NC1CCCC1C(=O)NCC1CCCN(C)C1 C(=O)(CCCN(C)N=O)N(CCC)CCNC(=O)Cc1cnn(CC)c1 c1(C(=O)O)sccc1S(=O)(=O)N1CCCC(C(=O)NCc2cc(Br)ncc2Br)C1 c1(C(N2CC3CC(C2)N(C(C2CCC4(CC4)CO2)=O)C3)=O)cnc2ccoc2c1 C1(NC(Cc2cn(C(C)C)nc2)=O)COCCC1NC(C1CCC(O)CC1)=O C(=O)(CCC(F)(F)Cn1cc(CC(C)O)nn1)NC(C(C)C)C(=O)NCCO N1(C(C2CC(OC)C2)=O)CCn2c(CNC(C3(Cl)CC34CCC4)=O)nnc2C1 C(N=c1[nH]c(=NCCN2CC=CC2)[nH]c2cc[nH]c12)c1c(C)c(F)c(F)cc1 c1(C(=O)NCC(CN(C(c2nc(C)nn2C)=O)CC)(C)C)cc(C)c(O)c(N)c1 c1(C(=O)NCCN(C(=O)CCCS(N)(=O)=O)C)cc([N+](=O)[O-])cn1C c1(CCC(=O)N(CC(C)(C)NC(C2C(C#C)C2)=O)C)ccc(Br)cn1 N1(C(C2C(COC)C2)=O)CC2(CC(NC(c3cn(C)nc3C3CCCC3)=O)C2)C1 N1(C(C(C)=Cn2ccnn2)=O)CCCC2(CCN(C(c3occc3F)=O)C2)C1 C1(C(N2CC3(CN(C(C(C)CF)=O)C3)OCC2)=O)CCc2cc(F)ccc2O1 c1(C(C)=O)ccc(O)c(C(N2CC3CC2C3C(N2CC(C)OC(C)C2)=O)=O)c1 c1(OC)cc(C(=O)NC2CCCN(C(c3ccc(N)cn3)=O)C2)sc1Br C(C(F)(F)CCC(=O)NCCC(C)(C)C)n1cc(C(C)NC(C)=O)nn1 C=CCN=c1[nH]cc(C(N2CCC(F)C(NC(C3CC(OC)C3)=O)C2)=O)s1 C1(CNC(C(C)O)=O)CCC2(CCN(C(=O)CC3COC(=O)C3)CC2)CO1 N1(C(c2c(C)cn(C)c2)=O)CCCC(C)C1CCNc1nccnc1F C(=O)(CCC(N)=O)NC1(C(=O)NCC(C)C2CC2)CSC1 C(CCCCC(=O)N(C1CCCCC1)C)N(C(C(C)=C(C)C)=O)C N1(C(C2C(CC)N(C(=O)CCC=CC(C)C)CC2)=O)CCC(C)(OC(C)=O)CC1 N1(C(C2C3CN(C(c4ccc(Br)c(Cl)c4)=O)CC32)=O)CCCC(F)(F)C1 C(=O)(C(C)CCCC(C)C)N1CCC(COC)(NC(=O)Cc2ncoc2C)CC1 C1(C(=O)NC(C)(CO)C2CCCC2)CCN(C(=O)C=Cc2cocn2)CC1O Cc1ccc(Cl)c2[nH]c(C(=O)NCC3C4CCC(C4)N3C(=O)CN(C)C)cc12 c1(C(N2CCSCC2CCNC(C23CC(CN2C2CC2)C3)=O)=O)ccnnc1Cl c1(C(=O)OC)cc2c(NC(C)(C)CNC(=O)CC3CCCCC3C)ncnc2[nH]1 C(C(O)CN=c1ccc2ncc[nH]c-2n1)NC(C1(C)CC2CCC1C2)=O C1(NC(C(N2CCC(C)CC2)=O)=O)CN(C(C2CCN2S(C)(=O)=O)=O)CC1(C)C C1(O)(C(N2CC(c3ocnc3CNC(c3cc(Cl)cs3)=O)C2)=O)CC2CCC1C2 C1(NC(c2cnn(C(CC)C)c2C)=O)CC2(C1)CN(C(c1occc1CC)=O)C2 N1(C(CC(CC)C)=O)CC=C(C(=O)N(CCN(CCN(C)C)CC)C(C)C)C1 c1(C(=O)NC(C2OCCN(C(CCSCC)=O)C2)C)cc([N+](=O)[O-])ccc1SC C1(OC)CC2(C1)CC2NC(=O)CCC1(NC(=O)COCC2CC2)CCC1 CCC(C)(C)CC(=O)N1CCC(CNC(c2cnc3n2CCS3)=O)(OC)C1 c1(CC(=O)NC(C(C)(C)C)CNC(C2CCCO2)=O)noc2cc(F)ccc12 Cc1cn2c(n1)CC(C(N1CCN(C3COC(C)(C)OC3)CC1)=O)C2 C1(CC(=O)NCC2CCCN(C(c3cncnc3)=O)C2)Cn2ccnc2NC1=O C1(C(=O)OC)CC(CN)CN(C(=O)COc2cc(C(C)(F)F)ccc2Cl)C1 C(CC(C(=O)NC1CCCC12CC2)NC(=O)Cc1ccc[nH]1)SC c1(C(C)OC(c2csc([N+](=O)[O-])c2)=O)cccc([N+](=O)[O-])c1 c1(CC)c(C(=O)N(CC(C)NC(C2(c3ccno3)CC2)=O)C)sc2ccccc12 C=CC(C)(C)CC(=O)N1CC2(CNC(=O)C(C3CCCCCCC3)O)CC1CO2 c1(C(=O)OC)ccc(NC(c2ccccc2)C2CC(=C3CC3)C2)cc1 C(=O)(CCC(CC)NC(C1(C)CCOC1)=O)NC1(C#C)CC1 C1(CC(=O)N(C(C)CCNC(C2CC2C(C)C)=O)C)(NC(C)=O)CCCCC1 C1(NC(c2cc(COC)cn2C)=O)COC2CN(C(=O)COCC3CC3)CC12 C1(NC(CCOCC#C)=O)CN(C(=O)CC2CC(O)C2(C)C)CC(C)(C)C1 C(=O)(CCN=C(NCc1ccc(Br)c(C)c1F)NCC(C)COC)NC C(=O)(C(C)C(F)F)NCCCC1(CNC(N(C)CC2(OC)CCC2)=O)CC1 Cc1ncc2n1CCC(C(N1CC3CN(C(=O)C(C)SC(F)(F)F)CC3C1)=O)C2 C1(OC)CC(C(=O)N(C)Cc2ccncc2F)N(C(=O)Cc2cnns2)C1 CN1CCCC(C(C)(C)C(=O)NC2CC(n3cc(CC(O)C4CC4)nn3)C2)C1 c1(C(N2CCC(N(C(=O)CCC(=O)C3CC3)CC)CC2)=O)cc2n(n1)CCC2 c1(C(N)=O)cnc(NC(N2CCCCC2C2CCNC2=O)=O)c(Cl)c1 c1(C(N(CC(C)N(C(=O)C(F)=C2CCC2)C)C)=O)ccnc(OCC(F)F)c1 Cc1nc(Cl)ccc1NC(N1CC(C2NC(=O)NC2=O)C1)=O C1(NC(c2c(CC)occ2)=O)CCCCC1NC(=O)C(C)(C)n1cnnn1 N1(C(C=CC)=O)CCCC(CN(C(=O)COC2CCC(C(N)=O)CC2)CC)C1 CC1CC(NC(=O)CC23CC(CO2)C3)CN1C(=O)Cn1cc(CN(C)C)nn1 c1(CSC)cccnc1C(=O)NCC=CCNC(=O)C(F)C1CCC1 CC1CCN(C(=O)Cn2cc(CNC(c3cn(C)cc3Cl)=O)nn2)CC(C)O1 C(c1c(Cl)cccc1Cl)=CC(N1CCC(CC(C)NCN2CC(N(C)C)C2)CC1)=O C=CCC(C)(C)CC(=O)NCC1CCC(C)N(C(c2ccc(Cl)c(C)c2O)=O)C1 c1(C(=O)NC(C2CCCN2C(=O)CC2CCCOCC2)C)nc2c(s1)CN(C)CC2 Cn1c(=O)nc(O)c2nc(C(=O)NCC3CC(C(F)(F)F)CN3)[nH]c12 c1(C(=O)OC)ccc2nc(N3C(=O)NC(CCF)C3=O)ccc2c1 C(C(F)(C(=O)NCc1ccn(CC)n1)C(C)C)NC(C(C)OCC#C)=O c1(C(N(C(CCNC(CC(C)=C(C)C)=O)C)C)=O)cccc2c1CCC2 N#CC12CCC(NC(C3CCCCN3C(=O)CC3NC(=O)NC3=O)=O)(CC1)CC2 C1(CC(=O)OC)CN(C(c2csc([N+](=O)[O-])c2)C(=O)NC2CC2)C(C)(C)C1 C1(NC(c2nccc(OC)c2O)=O)CC2(CCN(C(C3CCCC34CC4)=O)C2)C1 CC(CO)C(=O)NC1CC(CNC(=O)CCNc2ncccn2)C1 CC1(C(=O)NCC2CC23CC3)CCCN1C(C1CCC1C(N)=O)=O O=C(CN1C(=O)Cc2ccccc21)NC1CC2C1CCN2C(=O)CC1(CO)CC1 c1(OC)ccc2c(=NC(=O)c3nnn(C4CCS(=O)(=O)C4)c3C)[nH]oc2c1 CC(CC(C)(C)C)C(=O)N(CC(C)C(C)(C)C)C.C1=CNC1=O c1(C(C(=O)NCC(N(C(C(c2ccc(C)o2)C)=O)C)C2CC2)C)ccccc1C N1(C(C2CN(CC(C)C)C2)=O)CC(O)CC1CNC(=O)Cc1csc(S)n1 c1(C(=O)NCCCC(C)NC(Cc2cccc(C#C)c2)=O)cc(S(C)(=O)=O)co1 c1(C2(CCNC(=O)C(=O)NCC3CC3OCc3ccccc3)CC2)cccnc1 C1(COC)CN(C(c2cnc3n2CCC3)=O)CCN1C(C1CC(F)C(=O)N1)=O N1(C(C(C)N(C(=O)CC2CCCO2)CCC)=O)CCCC(C#N)C1 C1(C#CC(=O)C(=O)CN(C)CC)(CC)COC1.C(C(C(C)(C)C)Nc1ncccn1)N C1(NC(C(C)(C)C)=O)CN(C(=O)CCN(c2cnccn2)C)Cc2nccn2C1 C(CC(C)CCNC(c1ccc(-n2cccn2)cc1)=O)NC(COCCC#C)=O c1(OCC=C)ccc(C(=O)NCC2CCN2CC2CC(C)CO2)cc1 c1(CC)cccc(C)c1C(C(C1C2COCC12)C(=O)NCSc1ccccc1)C C1(C(=O)NCCN(C(C)C)C)CCCCN1C(c1cccnc1)=O N1(C(c2[nH]c(=N)sc2)=O)CC2CC1CCC2NC(C1CC1c1ccccc1)=O N1(C(c2n(C=C)ncc2)=O)CC(=O)NCC1C(=O)NCC1CCCO1 c1(CC(=O)NC2COCC2NC(C2(CF)CC2)=O)cnc(C(F)(F)F)s1 N1(C(CC=C)=O)CC(CNC(c2cccc(N(C)C)n2)=O)CCC1C C1(C(C)C)CN(C(=O)C(C)(C)C2CCCO2)CCN1C(c1cccc(O)c1Cl)=O c1(CNC(c2cc(Br)n(C)n2)c2n(CCCC)nnn2)cccc(C(N)=O)c1 Cc1nc2ncccc2cc1C(=O)NC(C1CCN(C(=O)C=CC2CC2)CC1)C C(c1ccccc1)=CC(=O)NCC1CN(C(=O)Cc2cccc(F)c2)C2CC12 C=CC1(C(=O)Nc2cc(C)cc(Cl)c2)CCN(C(c2nccnc2N)=O)C1 c1(OC)ccc2[nH]c(=NCC=CC3CC3)[nH]c(=NCC3CC(CO)CO3)c2c1 Cc1ccn(CC(N2CC(NC(=O)CC3CCC(C)(C)C3)C2)=O)c(=O)c1 c1(OC)ncc(C(=O)N(CCCCNC(C2CCC2C(N)=O)=O)C)s1 c1(CNC(c2ccc(-n3c(C)nnc3)cc2)=O)cccc2cn[nH]c12 O=C(CCC(=O)NC1CCCC1CNC(=O)CC1CC12CC2)Nc1nccs1 C1(OC)CC(NC(c2cnc(Cl)n2C)=O)CN(C(=O)C(=O)NCC(F)F)C1 c1(C(=O)NC(C2CCN(C(Cc3cn(C)nn3)=O)CC2)(C)C)cc(O)cc(O)c1 CC(CC(=O)NCc1ccsc1)C(C)(C)NC(=O)COCC(F)F c1(C(N2C3CC(CNC(c4c(C)c[nH]c4)=O)C2CC3)=O)coc2cc(C)ccc12 c1(C(=O)NCc2c(C(=O)NCC3(CO)CC(C)C3)[nH]cc2)ccc(F)cn1 C1(C(N2CCCC(C(C)NC(c3ccc(OC)cc3)=O)C2)=O)CN(C)CCN1C C1(CNC(COCCCOC)=O)CN(C(C2(CC(C)C)CC2)=O)C(C)CCO1 N1(C(c2c(C)ccn2C)=O)C2CCC1C(CNC(=O)Cc1ccc(O)nc1)C2 N1(C(C23CCC(OC)C2C3)=O)CCCC(CO)(NC(=O)CNC=O)C1 C(c1cccc(F)c1Cl)=CC(N1CCC(C)(NC(=O)C(F)(F)F)CC1)=O c1(C(=O)NCCc2cc(C)ns2)coc2c1CN(C(=O)C(C)n1cncn1)C2 C1(C)(C(=O)NCC2(O)CCCN(C(c3c(CC)scn3)=O)C2)CCC(F)(F)CC1 CCC(CNC(=O)C(F)CC1CCOC1)(CC)C(=O)NCC1(C)CC2CCC1C2 c1(C(C)(C)OC)ccc(C(=O)NC2CC(C)(NC(=O)Cc3ccon3)C2)cc1 c1(C(=O)NCC2(OC)CCC(C)C2)c(C)nn(C)c1-n1cc(C)cn1 CC(C)CCCCCC(=O)NCC1CCCCN(C(=O)C(=O)N=S(C)(C)=O)C1 N(C(=NCCn1cccn1)NCCSC1CCC(F)(F)C1)CC(C)(C)C C(CCC(C(=O)Nc1ccccc1)NC(=O)OC1CC2CC1CC2O)OC C1(NC(c2ncn(C(C)C)n2)=O)CCN(C(=O)Cc2cccc(C(F)F)c2)CC1O Cc1cc(C(=O)NOCC(=O)NC23CCCC2C3Br)c(C)o1 N1(C(c2cn(CC)nn2)=O)CC2(CO)CC1(C(N1CC=CC1(C)CO)=O)C2 CC1c2ccccc2OC1CNCCCOc1ccccc1 C(=O)(CC(F)(F)C(C)C)N1C(CCNC(C(n2ncc(C)c2)C)=O)CC(F)(F)C1 N1(C(CCCOCC)=O)CCC2CCCC12C(=O)Nc1c(C)nc(O)nc1O Cc1cc(CC2OCCOC2C)cc(C)c1.C1C(C)CC2(N=N2)CNC(=O)N1 C1(C(=O)NCCN(CC(F)F)C)CC2CC2N1C(=O)Cc1ccccn1 c1(C(=O)NC(C2(O)CN(C(c3cnccn3)=O)C2)C)cc2c(nc1O)CCOC2 CCCC(O)CC(=O)N(C)Cc1cc(OC)cc(OC)c1 N1(C(CC(CCC)C)=O)CC2CCCC2(C(=O)Nc2ccc(COC)cc2)C1 CCCCC(C)CCC(=O)N1CCC2C1CCN2C(=O)C(c1ccccc1)=O c1(CC(C(=O)NCC2CN(C(C(C=CCCC)O)=O)C2)C)ccccc1C C1(NC(CC=CC)=O)C2CCN(C(c3cnc(OC)s3)=O)C12 N1(Cc2ccc(C#C)cc2)CC2CN(C(c3n[nH]c(C)c3C)=O)CC2C1 CC(C)(C)C(=O)C(=O)NC1CCCC(NC(c2cc(Cl)ccc2C2CC2)=O)CC1 N#CC1(C(=O)NCC(CNC(=O)CCc2cc(Cl)no2)CO)CC2CCC1CC2 c1(C(=O)NC2C(CNC(CC(C)CF)=O)C2)cc(N=S(C)(C)=O)ccn1 C(=O)(C(CO)C(F)(F)F)NCCCN(C(C(CCC)C#N)=O)C N(C(=NCc1c(N(C)C)noc1C)NC(c1ccccc1)C)C(CC)C c1(CNC(CN2CC(CC)C2)=O)ccnc(N2CCCC2)n1.C12(COC1)C(=O)N2 Cc1cccc(F)c1C(=O)NCC1CN(C)CCN1c1cc(C2CC2)ncn1 c1(N(C)CC2OCCN(C)C2)nc(N2CCC3(CCC3)CC2)nc2c1CCC2 CC#CCC(C(=O)NC(CSCCOC)C1(C)CC1)NC(=O)OC(C)(C)C C1(c2ccccc2)(CNC(Cn2c(C(C)C)nnn2)=O)CCN(C)CC1 c1(C(=O)NC2C(CNC(CN(C)CC)=O)CCC2)cc(F)cc2cnccc12 c1(NC(c2ccc(O)nc2)=O)ccc(C#N)c(C(F)(F)F)c1.CC12CN(C1)C2=O N1(C(C(C)=O)=O)CCC2(CCCC2NC(c2ccnc(F)c2)=O)CC1 c1(C(N2CC(CN(C(CC(=C)Br)=O)C)OCC2)=O)cnc2c(c1)CCCC2 C1(CC(=O)NC(C)(C)CNC(c2csc(SCC#N)n2)=O)CCCOCC1 C(=O)(C1CCc2c[nH]nc21)N1CC(C(C(=O)NC2(C)CCCC(C)(C)C2)OC)C1 c1(C(N2CCC(NC(CN3C(C)CCC3)=O)C(O)C2)=O)cc2cc(F)ccc2o1 c1(C(=O)NCC2(CNC(c3cn(CC(=O)OC)nn3)=O)COC2)cc(Cl)c(Cl)s1 C1(CC(=O)N(C)CC2(O)CN(C(=O)C(F)(F)C(F)F)C2)Cc2ccccc2O1 n1(CC)cnc2nc(N3Cc4cccnc4C3)nc(NCC(CN(C)C)OC)c12 C(=O)(CC(=O)OC(c1ccccc1)C(=O)OC)OCC.C1CN(C)C(=O)N1 c1(NC(C23CCN(C(C(C)=C(CC)C)=O)CC2C3)=O)cc(C(C)=O)ccc1C#N C1(C)(C(=O)NCC2C(C)CN(C(=O)CN3CCC3)C2)COC(=O)OC1 N1(C(N(CCSc2ccccc2)Cc2scc(C)n2)=O)CCCC2(CCCCO2)C1 Cc1nnn(NC(=O)C2CCCCN(C(=O)CCCCCF)C2)c1C c1(C(N2CCN(C(c3cc(C)sn3)=O)C(CF)C2)=O)ccc(O)c2c1CCCC2 N1(C(CCOCCOC)=O)CCC(N=c2nc(C3CCCCC3)[nH]s2)C(C)C1 c1(CCC(=O)NCC(CN(C(=O)CCC2CCCC2)C)O)ncc(C(C)(C)C)o1 Cc1ccc(C(C)C)cc1C(=O)NCC1CN(C(=O)Cc2ccoc2)C(C)(C)C1 c1(C(=O)NC(CCNC(CC(=O)OC)=O)C)cc(OC)nc2ccccc12 C1(C(=O)NCC(CSC)OC)CC=CCN1C(c1nc(=N)cc[nH]1)=O c1(C(C)=O)cc(=NCC2CC(NC(c3c[nH]cc(Cl)c3=O)=O)C2)[nH]cc1[N+](=O)[O-] C1(C(N2C(CNC(CN3CC(C)(OC)C3)=O)CC2)=O)C2CN(C)CC12 c1(CC(=O)NCCC2CCN(C(C(N3C(CC)CCC3)=O)C)C2)ccccc1F C#Cc1cccc(NC(=O)CC2(OC)CN(C(=O)CC3NC(=O)NC3=O)C2)c1 N1(C(c2c(C)csc2)=O)CCC(NC(=O)CC(C)(C)O)C(C(N)=O)C1 C1(OC)CCC2(C(=O)NC(C3CCN(C(C4CNC(=O)N4)=O)CC3)CO)CC12 C1(CN(C(C2C(C(=O)OC)C2)=O)C)C2CN(C(=O)CCc3ccc(C)s3)CC12 c1(NC(CCCSC(C)(C)C)=O)cc(Cl)c(Cl)c(Cl)c1.C12CC(CO1)C(=O)NC2 c1(CC)ccc(S(=O)(=O)NCC(F)N)s1 C1(C(N(C2CC(C(N(CC(=C)C)CC(=C)C)=O)C2)C)=O)CC2CCC2C1 c1(C(=O)NC(CCC(=O)N(CCOCCOC)C)C)ncc(F)cc1N C1(C)(C(=O)NC2CCN(C(CN(S(CC)(=O)=O)C)=O)CC2)CC(OC)CN1C CC1CCN(CCO)CCN1C(c1ccc(Br)cc1I)=O Cc1cc(C(N2CC(CNC(=O)Cn3nnnc3C3CC3)C3CC23)=O)c(C)s1 N1(C(CCCOCC)=O)CCCC2(CCN(C(C3CC34CCCC4)=O)C2)C1 C1(Cc2n(-c3ccn(C(C)C)n3)nc(-c3ccnn3C)n2)CCCS(=O)(=O)C1 Cc1nc(C(=O)NC(CCN(C)C(c2ccc(C(C)F)cc2)=O)C(C)C)c(C)s1 C1(NC(C2(CC=C)CN(C(=O)CCCOC(C)(C)C)C2)=O)CCN(C)CC1C C1(C(N2CC(F)(CNC(c3onc(C)n3)=O)C2)=O)CCCSC1C CC1CCC(CC(=O)NC2CCC(CNC(C3(O)CCCCCC3)=O)C2)CC1C C(=O)(C(C)CC(C)(C)C)N1CC(COC)N(C(=O)Cc2cncn2C)CC1 N1(C(C(C2CCCCC2)OCC)=O)CCC(n2cc(CCC#N)nn2)C1 CC1(C)CCCCC1C(=O)NC1(CC(=O)NC(Cc2ccco2)CO)CC1 N1(C(CCOC(C)C)=O)CC2(C1)CN(C(c1sc3cccnc3c1Cl)=O)CCO2 N1(C(c2c(OC)cccn2)=O)CCCN(C(=O)CN=S(C)(C)=O)CC1C(C)C C1(NC(=O)CC2CC23CC3)CN(C(c2cnc(Cl)[nH]2)=O)CCC12CCOCC2 C1(CC)CN(C(=O)Cc2ccc(OCCCC#N)cc2)CCN1C(=O)CC1CC1 c1(C(N2CCCC(CNC(C3CCCCS3)=O)C2)=O)cc(O)nc(C2CC2)n1 C12(NC(C(n3cc(Br)cn3)C)=O)CC1CN(C(=O)COCC1CCCC1)C2 C#CCC(C)(CC)C(=O)N1CC(NC(=O)CSS(C)(=O)=O)C(c2nccn2C)C1 c1(CC(C(=O)N(CC)CC)NC(C2(F)CCNC2)=O)ccc(O)cc1 C(=O)(C1=C2CCCN=C2NN1)N(CC(C)NC(c1ccnc(Cl)c1Cl)=O)C C=C(C)CC(=O)NCCCCNC(C1SCCS1)=O CC1CN(C(=O)CCN2CCCC2=O)CC1NC(=O)C(C)Cc1ccccc1 C1(NC(C(COCC)C)=O)CC2(CCC(NC(c3cc(CC)no3)=O)CC2)C1 C12(C(N(C3CN(C(CCN4C(C)CCCC4C)=O)C3)C)=O)CCCCC1OCC2 c1(N(C2CN(C(c3c(O)ncc(SCC)c3)=O)C2)C)nc2ccc(O)cc2s1 c1(C(N2CCCC(NC(CN(C3CCC3)C(C)=O)=O)C2)=O)cc2ccsc2s1 C12(NC(C(C)SC)=O)CCCC1N(Cc1c(F)cccc1F)CC2 c1(C(=O)NCC(C)N(C(CC(C)O)=O)C)cccc(O)c1 N1(C(C2C(=C)CC2)=O)CCCC(N(C)C(c2cc(COC)[nH]n2)=O)CC1 C1(CCSCCN(CC)CC)CN(C(=O)OC(C)(C)C)CCN1C c1(C(=O)NCC(C)(CO)NC(CC(C)c2ccco2)=O)cnncc1O C(=O)(C(C)(C)C(C)(C)O)NCCN(CC(C)O)C(c1n(CC)ncc1)=O Cc1cc(C)c(C(=O)NCCC2(NC(C3C=CCCC3)=O)CC2)cn1 C(CC(C(=O)OC(C)=O)OCC)NC(=O)Oc1ccccc1.C12CCC(C1)OC2 C(C)(C)(CNC(=O)CN(C)C1CC1)OCCCNC(CNC(CC)=O)=O Cc1cccc(C(=O)NC2CCN(C(=O)Cc3ccsn3)CC2)c1F C(C1OCc2ccccc21)NC1CCCC(C(C)C)N1 C1(C(=O)NC(CC(=O)OCC)C)C(C)OCCN1C(=O)C(C(C)OC)OC c1(CN2CC(C(=O)NC3CC(=C)C3)OCC2)ccc(C(=O)O)cc1Br C(=O)(C(C)(C)CC(C)C)NCC(=CC(=O)Nc1c(CC)onc1C)C C(c1ccc(C)cc1)=CCC(=O)N.C(C(=O)C(CN)=O)N(CC)CC.C12(CC1)CC2 C1(CN(C(CCC=C=C)=O)C)CCCN(C(=O)CC2(O)CCCN(C)C2)CC1 c1(N2CC3N(C(c4c(C)c(Cl)ccc4)=O)C3C2)ncnc2sc(C(C)C)cc12 C1(C=O)CCC(=O)N(C)C1.n1(CC(=O)NCCCN(CC)CC)cc(C)cn1 C(C)(C)(C(=O)NC(CNC(c1cnoc1-c1cccs1)=O)C(C)C)SC c1(C(=O)NCCCN(C(CCC=CC)=O)CCO)cc2cc(F)cc(F)c2[nH]1 C1(C(=O)NC(C#C)C)CC(C)(C)CCN1C(c1ccncc1O)=O C1(NS(CCc2c(C)ncs2)(=O)=O)CCCC(C)C1 C(=O)(C1CC(O)c2ccccc21)NCCNC(c1onc(OC)c1C(F)(F)F)=O Cc1oc(Cl)nc1C(N1CC(O)(C(F)C(N2CC(O)C(O)C2)=O)C1)=O Cc1cc(C)c(C(=O)NCC2(F)CC(CNC(c3c[nH]c(=N)o3)=O)C2)s1 Cc1cnc(C(=O)NCCC2(C(=O)NCC3(O)CC(C)(C)C3)CCC2)cc1C C1(C(=O)OC)CCC(C)(C(=O)N(N2CCC(N=[N+]=[N-])C2)C)C1(C)C C(=O)(CCC(C)(C)F)N1CC(CC(CNC(CC(C)CN(C)C)=O)(C)C)C1 C1(NC(C2CC2F)=O)CC2CC1CN(C(c1cccnc1I)=O)C2 C(=O)(C#CC1CCCO1)N(C)CC1CCN(C(CC=C)=O)C1 C1(C(=O)NCC2(CCOC)CC2)CC2CN(C(c3nccn3C)=O)CC2C1 N1(C(c2c(OC)cc(C)cc2)=O)CCC(C2(NC(C3Cc4cscc4C3)=O)CC2)C1 Cn1nccc1C(C1CC1)NC(=O)C(O)CC1CCOCC1.n12cc(nn1)CC2 C1(CC)CN(C(=O)COC2CCN(C)C2=O)CCN1C(C1CC2(C1)CC(C)C2)=O c1(C(N2CCN(C(c3c(C)nco3)=O)CC2C(C)C)=O)ccc2c(c1)OCCO2 c1(-c2cccc(COC)c2)cnn2c(C=CC(N3CC4COCC4C3)=O)c[nH]c12 C(=O)(C(CCC)C(=O)NC(CC(=O)NCCCC(C=C)(C)C)C(F)F)NCC N1(C(CCC(C)c2ccccc2)=O)CC2(CCC2NC(c2ccnn2CCF)=O)C1 n1(CC(=O)NC2CC(NC(CN=S(C)(C)=O)=O)C2)ccc2nc(O)nc(O)c12 C12(NC(CCCC#C)=O)CC(C)(C1)OC21CCN(C(=O)C(C)C(=O)OC)CC1 c1(C(=O)NC(CN(C(c2ccc(C)nc2)=O)CC)C)c(C)nn(C2CC2)c1Cl c1(CNC(=O)CC2(O)CCCOC2)ccc2c(c1)CCC2NC(=O)C1=CCC1 C1(CC(=O)N(CCC(N)=O)C)CC(C)(C)CN1C(=O)C1=CCCC1 C1(N(C(c2ccc(CCC)[nH]2)=O)C)CC2CCC(C1)N2C(c1coc(C)c1)=O N1(C(Cc2nc(COC)sc2)=O)CCC2(CC1)CN(C(=O)C=C(C)Cl)CC(C)O2 C1(NC(=O)CCC(F)F)CCCC(NC(=O)COc2ccc(F)c(F)c2)CC1 C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)CCCCNC(N)=O)C2CCCC12 c1(C(=O)NC2CC(C(=O)OCC)OCC2)[nH]c2c(c1C)CCCC2 CCCCC(C(=O)OCC(=O)NC(c1ccc(OCC(C)C)cc1)C)N(C)C c1(N(C2CC(CO)C2)C)nc(=N)[nH]c(=NCCCc2cccc(Br)c2)[nH]1 C(CC(O)C(=O)NCC(C)CN(C(=O)CSC(F)F)C)SC C(=O)(C(O)CCCNC(C1CC12CCCCC2)=O)N1C(C(=O)OC)CCC1 C12(CNC(c3c(C)nn[nH]3)=O)CN(C(c3cc(CO)[nH]n3)=O)CC1CS(=O)(=O)C2 n1(-c2c(C(=O)O)ccc(F)c2)nnc2ccccc12.C1(C(=O)O)CS(=O)(=O)N1 C1(C)(C(=O)NC2(CC=C)COC2)CC2(C1)CC2(F)F N1(C(c2c(CNC(CCC(CC)C)=O)cco2)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(OC)cccc(NC(C(c2cnn[nH]2)N(C2CCC2)C)=O)c1 N1(C(c2nc(CC)[nH]n2)=O)CCC(=CCNC(=O)C(CSC)c2ccccc2)CC1 C1(CCC(F)(F)F)(COC(=O)CC2CCC(C(F)(F)F)O2)CCCCC1 C1(C(N2CC3C(NCc4c(OCC)cccc4)(C3)C2)=O)CCc2nc[nH]c2C1 c1(N2CCN(C(C=CC=CCC)=O)CC2)cc(=O)n2cc(Cl)ccc2n1 N1(C(c2nc(C)sc2)=O)CC(CNC(=O)C(C)N(C)C(C)C)C(F)(F)C1 c1(OC)cc(F)cc2[nH]c(CNc3cnn(-c4ccccc4F)c3)cc12 C12(COC(c3c(N)ncc(Br)n3)=O)CCCC(=O)N1CCC2.C12CCN(CC1)C2=O N1(C(c2c(C)cc(F)s2)=O)CCCN(C(=O)CCc2cnc(O)[nH]2)CC1 N1(C(c2cc(OC)n[nH]2)=O)CCC(C2CC2)C1CNC(=O)C(O)C(C)(C)C N1(C(c2cc3ccccn3c2)=O)CCN(Cc2ccco2)C2(CCOCC2)C1 C=CC1(CC(=O)N(C)Cc2ccccc2F)CN(C(=O)Cc2ncccc2C)C1 N1(C(C(C)C2CCC2)=O)CC(=O)NCC1C(=O)Nc1cccc(F)c1 C1(COC)(NC(=O)CN(C)C(c2ccoc2)=O)CN(C(=O)C(C)CO)C1 c1(C(N2CCC(O)(CNC(COCCCOC)=O)C2)=O)cnn2c(=N)[nH]cnc12 C1(CC)CN(Cc2ccc(Br)cc2C(F)(F)F)CCN1C(=O)Cc1ccccc1 C(C(CC(C)C)NC(C1CN(C(C)C)CCO1)=O)NC(CCc1ccc(C)o1)=O O=C(CC(C(F)F)NC(c1cccc(F)c1O)=O)NCCC(O)C1CCCC1 c1(CC)ccc(C)cc1C(=O)NCC1CCN(C(C2CC3CC3C2)=O)C1 C=C1Cn2c(C(=O)NC(CCN(C(=O)C(C)(C)SC)C)C(C)(C)C)nnc2S1 C1(NC(CC2CCC(=O)NC2)=O)(CNC(c2ccc(Cl)cn2)=O)CCCCCC1 c1(C(=O)NC2CC2NC(C2CC(F)(CO)C2)=O)cnc(Cl)s1 C1(NC(c2ncn(C)n2)=O)C2CCN(C(c3cncc(N)n3)=O)C12 N1(C(c2cn(C)nc2O)=O)C2CCC1C(F)C(NC(=O)CC1CCCO1)C2 Cc1cccc(Br)c1OCCNC(c1cc(C#N)c(Br)s1)=O C(C)(O)(CC(C)C)NC(CC1C(C(=O)OCC)C1)=O.C1C(=O)NCCO1 CC1(C(=O)N(C2CCNCC2)CCO)CCOC1 O=C(C1=CCS(=O)(=O)C1)NCC1(CNC(C2CC23CCOC3)=O)CCC1 C(CC(C)(C)CC(=O)NC(C)(C)CC=CC(=O)NC1CC(C)(O)C1)OC N1(C(C2C(C)=C2)=O)CC2CCCN(C(C3CCC(=O)N(C4CC4)C3)=O)C2C1 C1(CNC(C(c2cn(C)nc2)O)=O)CN(C(=O)Cc2cocn2)CCO1 c1(COC(C2C(c3ccc(C)cc3)CCCC2)=O)ccc(N)c(F)n1 c1(C(=O)OC)ccc2c(CNCc3ccc(N(C)C)nc3)c[nH]c2c1 CCC(C)(C)CCCC(=O)N1CCC(CC(=O)N(C(C)CC)CCO)CC1 n1(CCNCc2c(N(C)C)cccc2)cnc2cc(Br)ccc12 c1(C(N2CCC(NC(c3n(C)nc(C)c3F)=O)C2)=O)ccc(C#N)cc1Br c1(C2C(C)(C)NC(=O)CC(=O)N2C)ccc(F)cc1.C(C)(C)(C)NC(=O)OC1CC1 c1(C(=O)NC2C(OC)CN(C(=O)Cc3ccn(C)c3)C2)ccc2c(c1)CC(C)O2 C(C#Cc1ccccc1)N(C(C(=O)NC)CC1CC1(Cl)Cl)C Cc1nccc(C(=O)NCCCNC(C2(C3CCCO3)CC2)=O)c1C c1(C(=O)OC)ccc(S(=O)(=O)Nc2ccccc2OCCF)c(C)c1 C1(C(=O)Nc2ncc(-c3ccc(C(=O)NCC=C)cc3)s2)CCCCC1(F)F N1(C(c2nc(C(C)C)sc2)=O)CC(NC(=O)CC2CCOC2=O)CCC1C C1(CC)CN(C(=O)CCOCCOC)C(CNC(=O)CCCOC)CO1 c1(NC2CC(C(N3C(C=C)CC3)=O)N(C(=O)OC(C)(C)C)C2)cc(C)cc(O)n1 c1(C(=O)NCCC(C)CCNC(C2(C)CCCS2)=O)ccc2c(c1)OCC(=O)N2 Cc1csc(CC(=O)N(CCCC(=O)NCCC2CCC(C)O2)C)c1 c1(C(=O)NCC2C(NC(C(C(C)(C)O)F)=O)CC2)cc(N)c(F)cc1F C12(NC(=O)C=CC3CCC3)CCCC1CN(C(c1c[nH]nc1-c1cccs1)=O)C2 CCCC(C(=O)NCc1csc(C(=O)NC(C)(COC)C(N)=O)c1)OC CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)COCC(F)F)C2CCCCC12 c1(C(N2CCCC(C(=O)NCCc3ccc(C)cc3)C2)=O)ccc2[nH]ccc2c1 c1(CCC)cc(C(=O)NC2CC(OCCN)C2(C)C)c(C)o1 N(C1CCCc2ccc(C(C)(C)C)cc21)C(C(=O)N(CC)Cc1ncccn1)=O c1(C(N(C(CC(F)F)C(=O)NC2C=CCC2)C)=O)ccc(=O)n(C)c1 Cc1cc(O)ccc1C(=O)N(CC(C)CNC(C1(F)CCS(=O)(=O)C1)=O)C n1(CC)cc(S(=O)(=O)NCC2(n3cccn3)CC2)nn1 CC1(C(=O)NCC2CC2CNC(c2cc(-c3ccoc3)on2)=O)CCCCC1 C(CCCCNC(=O)C(C)C1(NC(=O)CSC(F)(F)F)CC1)N(C)CC N1(C(C(C)(C)NC(=O)NCC=C)=O)CCCN(C(=O)C(C)(C=C)CC)CCC1 CCC(C)C(O)C(=O)N1CCC2C(NC(=O)CC(CN(C)C)CC)C2C1 N1(C(CCCCN(C)C)=O)CCN(C(C2CCC(N=[N+]=[N-])CC2)=O)CC12CCC2 C1(NC(CS(C)(=O)=O)=O)C(CNC(C2(C(F)(F)F)CCCC2)=O)CCC12CCC2 C1(CCC)CN(C(C2CCC2C)=O)CC1C(=O)NC1CCCC1F N1(C(c2c(C)scn2)=O)C2CCC1C(NC(c1ccc(OCCF)cc1)=O)C2 C#Cc1cccc(C(=O)NC(C)(CNC(=O)CCC(C)CC)CO)c1 CCC(C)C(CC(=O)NCC1CCCCO1)NC(=O)Cc1ccn(C)n1 c1(CNC(C=C(C)Cl)=O)ccc(C(C)NC(c2cc(C)no2)=O)cc1 C(CC(C(=O)NCCCCN(C)C)NC(=O)CSc1ncc[nH]1)SCC N1(C(CC2(OCC)CCC2)=O)CCOCC(NC(=O)C(C)OCCN(C)C)C1 N1(C(C(C(=O)OC)OC)=O)CC2(CCC2)CC1CNC(=O)C=Cc1ccc(C)s1 C1(C(=O)NCCOc2c(OC)cccc2)CCC2(CC2)N1C(c1ccncc1Cl)=O C(=O)(CCCCC(N)=O)NC(C(=O)NCC(C)CC1CCC1)CCN1CCCC1 C1(C(=O)NCCC2CC(F)C2)(CNC(=O)CCCn2ccnc2)CCCCC1 S(=O)(=O)(c1c[nH]ccc1=NC(C)CCC(C)(C)C)Nc1cccc(C(C)C)c1 c1(C(N(CCN(C(=O)CC2CCCC2(F)F)C)C)=O)cnc2c(F)cccc2c1 c1(C(=O)NC(C(C)NC(=O)CSc2nncn2C)C)cccc2ncnc(O)c12 Cc1nc(CC(=O)NCCCc2ccncc2F)c(Cl)s1 c1(-c2c(F)ccc(C(=O)Nc3cc(OC(C)C)n[nH]3)n2)ccc2oc(C)nc2c1 C(C(C)CC(=O)N1CC(c2ccccc2)(NC(=O)CC2CC2(Cl)Cl)C1)OC c1(C(C)O)ccc(C(N2CCCC2CN(C(=O)C(c2ccccc2)F)C)=O)cc1 c1(C(=O)NC2CCC(N(C(Cc3cc(C)sc3)=O)C)C2)ccc(C2CC2)cn1 C1(CC(=O)NCCSCCOC)CCCC1NC(c1nccn1C(C)C)=O C1(C(=O)NCC(CCOC)NC(c2cc(OC)n[nH]2)=O)Cc2cc(C)ccc2S1 O=S(=O)(c1nc(N2CCCC2)ccc1Br)NCC(c1ccccn1)NCCCCF CC1=C(C(=O)N(C)CC2CCCN2C(C2(CN(C)C)CC2)=O)Cn2nnnc2N1C C1(C(=O)NCC(CO)NC(C(C=C)(C)C)=O)CCn2cc(CC)nc2C1 CCCC(C)CCCC(=O)NCCOCCCN(C(=O)CCC1CCC1)C C1(C(=O)NCC(CNC(Cc2nc(C)oc2)=O)F)CCCS(=O)(=O)C1 C1(NC(c2c(OC)c(Cl)ccc2)=O)CC2CC(C1)N(C(=O)C(C)(C)C#N)C2 Cc1cc(NC(=O)C(=O)NC(c2cccc(Cl)c2)Cn2cccn2)ccc1N n1(C(C)C)cc(OCC(=O)NC2CCC2CNC(=O)C=CC2CC2)cn1 CC(C)CC(O)C(=O)NC(CC(=O)NCC1CC=CCC1)C(F)F c1(OC)ccc(C(N2CC3CN(Cc4ccccc4Cl)C3C2)=O)cc1OC C1(C(N2CC(OCCNC(CC3CC(=O)NCC3)=O)C2)=O)CCC([N+](=O)[O-])CC1 C1(NC(C=Cc2ccc(C)o2)=O)CC1C1CCN(C(=O)C(O)CC2CC2)CC1 CCC(C(=O)NC(C1(O)CN(C(=O)C=CC(F)(F)F)C1)C)OC1CCCCC1 CN=c1[nH]cc(C(N2CCC(C(C)C(=O)NC3CCC(C)(C)C3)CC2)=O)o1 C(C(C)C(=O)N1CCC1C(=O)NCCCc1nncs1)OC C1(CNC(C(CCCC)O)=O)CCCC2(CN(C(=O)C(C)(C)O)C2)O1 C1(CC)CN(C(=O)CNC(N)=O)CCN1C(c1ccnc(-n2cccc2)c1)=O c1(C(N2CCC3(CCC3)C(CO)C2)C(=O)NC2CC2)cc2c(cn1)OCCO2 C12(NC(=O)CC34CCCC3C4)CCCC1N(C(c1ccc(Cl)cc1F)=O)CC2 C1(CNC(C=NOC)=O)CN(C(C2CC(n3ccnn3)C2)=O)CC(C(F)(F)F)O1 N1(C(C(C)CN(C)C)=O)CC(C2(NC(=O)C=CC3(C)CCOCC3)CC2)C1 N1(CC)CCCN(C(=O)Nc2ccc(F)c(N(C)C)c2)CC1=O.c1(C)ccccc1 N1(C(c2ccc(OC)nc2)=O)CCCN(C(C2(C)CC(C)OC(C)C2)=O)CCC1 O=C(NOC1CC2CCC1C2)C1=CC(O)C(NC(C2CCSCC2)=O)C1 c1(C(C(=O)NCCCCN(C(C(n2cc(Cl)cn2)C)=O)C)(C)F)ccc(F)cc1 C1(C2C(CN(C(=O)C)C)C2)CC12CCC2.C1(CC(=O)NCC2(C)CC2)CC(C)=NO1 N1(C(Cn2ncc(C#C)c2)=O)CCCCC(NC(=O)C(C=C)CC)C1 Cc1ccc(CC(=O)NC2CN(C(=O)CCc3ccccc3O)CC2F)cc1Cl N1(C(C(=O)N(CCCN2CCCC2=O)CC=C)=O)CCN(C2CC2)CC1C N(C1CCCOc2cc(Cl)ccc21)C(=O)NCC1(c2ccon2)COC1 C1(NC(=O)C=Cc2cc[nH]n2)CC2CN(C(c3n[nH]c4c3CCSC4)=O)CC2C1 C1(C(N2CCN(C(C(COC)N(C)C)=O)CC23CC3)=O)CNC(=O)CC12CCC2 C1(CC(=O)Nc2cc(OC(C)C)ncn2)CCOC(C)(C)C1.c12ncccc1O2 C(c1ccc(O)c(O)c1)=CC(=O)NCC(C)(C1CC1)NC(=O)CSC(F)F Cc1sc(Cl)c(C(=O)N(C)Cc2cn(CC(c3cccc(Cl)c3)(F)F)nn2)c1C N1(C(C(CC#C)O)=O)CCC(O)C(N(C(=O)CCCc2ccc(F)c(F)c2)C)C1 N1(CC(N2CCC(c3n(C(C)C)cnn3)C2)=O)CCC(=O)NC1=O c1(C(N2C(C(=O)NC3C(CCC)C3)CN(C)CC2)=O)ccc(C#N)c(C)c1 C(=O)(CCCNC(N)=O)NC1(C(=O)NC2(CC(C)C)CC2)CC1 CC(C)(C)CC(C)(C)C(=O)NC1(CC(=O)NCC(CO)C2CC2)CCC1 Cc1nn(C)cc1C(=O)NC(CNC(c1cncc(-c2ccoc2)c1)=O)C(C)C C1(NC(c2c(OC)oc(C)n2)=O)CCN(C(=O)CC(=O)NC2CC2)CC1C(C)C c1(N2CC(C(N)=O)OCC2)cccc(S(=O)(=O)NC(Cc2ccsc2)CO)n1 C(=O)(C1CCCc2ccccc21)NCC(CC=C)NC(=O)CSCc1cscn1 C(N=C(NCc1cccc(C(F)(F)F)c1)N1CCC1)c1ccc(C)cn1 C12(CNC(C=C(CCC)C)=O)CCC1CCN2C(=O)Cc1ccnnc1O N1(C(C2N(CCC)CCC2)=O)CCC2C(CCN2C(c2ncc(F)cc2N)=O)C1 C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NCC(C1(O)CCN(C(=O)CC2CC2)C1)C N1(C(C(CN(C)C)O)=O)CC2CC1CN2C(C1(Sc2ccccc2)CCC1)=O c1(NCCC(C(C)C)N(C)C(c2cccc[n+]2[O-])=O)ncc([N+](=O)[O-])cc1Cl C(=O)(C1CCCn2cncc21)N1CC2CCN(C(c3cccc(C)c3)=O)C2CC1 CCCCCC(O)C(=O)NCC1(CNC(c2cc(OC)ncn2)=O)CCCC1 C1(C(C)NC(c2c(C)cccc2)c2ccccc2)CC2CCC1CC2 Cc1c(NC(C2CC(=O)N(CC(C)C)C2)=O)cccc1C(C)C Cc1ccc(F)c(C(=O)NC2CCN(C(c3ccc(N)cc3C)=O)C(C)C2)c1 CC(C)C(F)(F)CC(=O)NC1CCC(N(C)C(c2cc3n(n2)CCO3)=O)C1 c1(C(=O)NC2CCCC(CNC(C3CCCCC3)=O)C2)cnc(O)c([N+](=O)[O-])c1 C12(C(=O)OC(c3ccc4c(c3)CC(=O)N4)C)CC3CC(CC(C3)C1)C2 N1(C(CC2N(CC)CCOC2)=O)C2CCC1(CNC(=O)C(C)(Cl)Cl)CC2 C(C(C)(C)CC(=O)N(CCCn1ccnc1)C)NC(C(C(C)C)=O)=O CC1(CNC(=O)C(F)(F)CC2CCCO2)CC(F)(F)CN1C(=O)CC1COC(=O)N1 CCC(O)C(=O)NCCC(O)CNC(=O)C(F)(F)c1ccncc1 CC(F)(F)C(C)(C)C(=O)N1CCCCC1Cc1cn(Cc2ccccc2F)nn1 CC(C)C(O)C(=O)NCCn1cnc(C(=O)NCc2cscn2)c1 c1(C(=O)OC)cc(OC)c(S(=O)(=O)N(C)Cc2cc(OC)ns2)s1 N1(C(Cc2c(C)nn(C)c2C)=O)CC2CCC(C1)N2C(=O)N(C)C1CC1 N1(C(c2cc(CNC(C(C)C(F)F)=O)[nH]n2)=O)CC(O)CC12CCC2 N1(C(c2ccc(CSC)o2)=O)CC2(CCN2C(=O)CC(=O)N(C)C)C1 C1(N(C(C2ON=C(C)C2)=O)C)CCCN(C(=O)CC#N)C1 C1(NC(CCN(C)CC)=O)CCCCC1NC(c1nccnc1C)=O Cc1ncn(C)c(=O)c1C(N1CCN(C)C(CNC(c2cnncc2O)=O)C1)=O N1(C(c2ccn(C)c2)C(=O)NC)CCCC(C(=O)Nc2ccccc2)C1 C(=O)(C1=C(Cl)CCC(C)C1)N1CCC(NC(C2CC(CCC)OCC2)=O)CC1 c1(C(=O)NC2CCN(C(C(F)=CC)=O)CC2CC)sc2ccccc2c1C(=O)OC c1(C(N2C(C)CCC2)=O)cccc(C#N)c1.c12ccccc1NC(=O)C2 Cc1nccc(C(=O)NCC(N2CCC(O)(C(N)=O)C2)=O)n1 c1(NC(C(CC2CCCC2)NC(C(CC)C)=O)=O)ccc(C)cc1C c1(CC(N2C(CNC(CC(C)N(C)C)=O)C=CC2)=O)cccc2cnccc12 c1(-n2ncc(CN(C)C(c3nccn3Cc3ccccc3O)=O)c2)cccc(F)c1 N1(C(C(CCOC)NC(=O)C2=C(C)CCC2)=O)CCN2C(=O)NCC2C1 C1(C(C(=O)NCCCCC(=O)NC)(C)C)CCCCN(C(C2CCOC2)=O)C1 c1(OC)cc(C(=O)NC(CO)C(C)NC(=O)CN(C2CCSC2)C)cc(C)n1 C(C(O)CC(=O)CC(=O)NC1COC(C)(C)C1)NC(CC)=O C1(C(=O)NC(COC(C)C)C)CCCN1NC(=O)C1COCC1C(N)=O c1(SC)nc(O)nc(C)c1C(N1C2CCC1CN(C(C1(F)CC1C)=O)C2)=O C(=O)(C1Cc2c(Cl)cccc21)NCC(C)(C)NC(C1CC1C1CC1)=O N1(C(C2C(=O)NCC2)=O)CCCC(C2CCN(C(c3coc(Br)c3)=O)CC2)C1 c1(C(=O)NC2CN(C(c3c(C)nc(C)s3)=O)CC23CC3)cc2cccc(Cl)c2s1 C1(CNC(C(c2ccccc2)C)=O)CC(F)(F)CN1C(C1CC2(CCO1)CC2)=O Cc1nc(N(C)C)sc1NC(C1(CC(C)C)CCCC1)=O.C123CC(C1)(C2)NC3=O N1(C(C(CO)OCC)=O)CC(OC)C(NC(c2cccc(OC(F)F)n2)=O)C1 CCCC(CCCO)C(=O)NCC(C)(C1CC1)NC(=O)CCn1cncn1 O=C(C1=CCCCC1)NC1CN(C(=O)CCC2CCCC2)CC1F C1(C(N(CCOC)CCNC(c2ccc(C3CC3)[nH]2)=O)C)CCCCC1OC N1(C(C(C(C)NC(c2scc(OC)c2)=O)C(C)C)=O)CCN2CC(C)CC2C1 c1(NC(C2CCN(C(C3C(C(=O)OCC)C3)=O)CC2)=O)ccc(C(N)=O)c(Cl)c1 C1(OC)(CNC(=O)C2=CCCSC2)CCN(C(c2cc(C)cs2)=O)CC1 C1(C(F)(F)F)(C(=O)OCC2CC2C2CC2)CC2CCC1C2 CN1CC(C(=O)NC2CC(NC(c3cnn(C)c3C(F)F)=O)CC2O)CC1=O C1(NC(C(C)(C)SC)=O)CCC2CC1CN2C(=O)CCC(=O)N(C)C C(=O)(CCCCCCNC(C1CC(O)CN1C)=O)Nc1c(C)ncnc1 N1(c2cc(OC)ncn2)CC=C(CNC(C2CCCC2c2ccccc2)=O)CC1 c1(C(=O)NCC=CCNC(C(=O)N(C)C)=O)c(C2CC2)nc2sccn12 C(=O)(C(C(C)C1CC1)N1CCCC1CC1CC1)NC(C)C CCCCC(F)(F)C(=O)NCCCN(C)C(c1cc(F)cc(F)c1OC)=O c1(C(N2CC(NC(c3nc(CC)sc3)=O)C(C)C2)=O)cc(O)nc2c1CCCN2 N1(C(C(CC)(F)F)=O)CC23CCCC2(C1)CN(C(c1cccc(N)c1C)=O)C3 C1(CC(N2C(C=C)CCC2)=O)CCN(C(C2C=CCCC2)=O)C1(C)C C1(CC)CN(C(C)C)CCO1.C(CC(=O)NC1C(=O)NC12CCC2)SCC N1(C(C2C(C(C)(C)C)OCC2)=O)CCC2(CC1)CN(C(c1cscn1)=O)CCO2 C1(c2ncc(C(=O)OC)s2)CCN(c2nnnn2Cc2cc(C3CC3)no2)CC1 C1(CC=C)(C(=O)NC2(C)CC2(C)C)CN(C(=O)CCc2ncccn2)C1 CCCCC(CC)CC(=O)NCc1cc(C)c(C(=O)N(CC(C)OC)C)o1 C1(CCC)CCC(CNc2ncc(CN(C(=O)CNCC)C)nc2)CC1 n1(CC)ncc2c1CC(C(=O)NC1CN(C(=O)C(=O)NC3CC3)CC1(C)C)CC2 N1(C(CNC(C(CC)C)=O)=O)CCN(C(c2sc(C)nc2C)=O)CC1CC(F)F C#Cc1cc(F)c(C(=O)N(C)CCN(C)C(c2ccc(=NCC)[nH]c2)=O)cc1F C1(CCOC)(NC(=O)CSCCC#N)CCN(C(=O)Cc2cscn2)CC1 CCCC(C)CCCC(=O)N(C1CC2CCC(C1)N2C(c1cn(C)[nH]c1=N)=O)C N1(C(C(CCSC)OC)=O)CCC2C(C1)CN2C(=O)CN1CCCCC1 c1(NC)ccccc1C(N1CC(N(C(=O)CCC2CCCO2)C)C(O)C1)=O CN1CC(C)(NC(c2ccc(Cl)c(Cl)c2)C#N)CCC1=O N1(C(C(=O)N(C(C)CNC(=O)CC2CC3CC3C2)CC)=O)CCCC(C)C1 c1(C(=O)NC(CCNC(Cc2cccc(C(=O)OC)n2)=O)C)cncn(C)c1=O c1(C(N2C(C(=O)OC)CC(OC)C2)=O)nc(C)[nH]c2nccc1-2 CC1(CNC(C2(CC(F)(F)F)CC2)=O)CCC(NC(c2ccc(F)cc2)=O)C1 CC(CCC1CC1)NC(=O)CCN(C(=O)CCn1cncn1)CCCO C(CC1CCCCC1)(C(=O)N(CCNC(=O)C(C1CC1)OC)C1CC1)OC C1(C(c2ncccn2)C(=O)NCCCC)CN(C(=O)OC(C)(C)C)CCC1C N1(C(CSCC#C)=O)CCC(C2CCCN(C(=O)C(c3cnn(C)c3)C)C2)C1 c1(N(C(C2CN(C)C(=O)N2)=O)CC)ccc(Cl)cn1.C12(c3ccccc3)CN(C1)C2 c1(C(N2CC(C)C(CNC(c3coc(Cl)c3)=O)C2)=O)c(F)ccc(Cl)c1N c1(CC(N2CCN(C(C(CC=C)(C)C)=O)CC2C)=O)csc2sc(C)cc12 N1(C(C(C)CC2CCCC2)=O)CCCC(C2CCN(C(=O)CS(N)(=O)=O)C2)C1 CN1CCN(C(C2CC3CC3N2C(=O)Cn2nc(Cl)ccc2=O)=O)C(CO)C1 C(=O)(C(C)(C)C(F)(F)F)N(CCCCN(C(=O)CCC1CC1(F)F)C)C Cc1nc(NCC2CN(C(c3cc(Cl)no3)=O)CCC2C)c(Cl)cc1[N+](=O)[O-] C(c1cccc(Cl)c1)=CC(=O)NC1CCC(N(C(=O)CCN2CCCCC2)C)C1 C1(C(=O)NCCCOCCCNC(CC2C(C)CCO2)=O)CCC(N=[N+]=[N-])CC1 CCS(=O)CCNC(=O)C(C)CNC(=O)C(N1CCOC1=O)C C=CC(C)(C)CCN=c1[nH]c(=NC2CCC(C)(SC)CC2)c2cc(OC)ccc2[nH]1 c1(N2CCC(NC(=O)NC3CS(=O)(=O)C3)CC2)ccc2nncn2n1 C1(NC(c2ccc(C(C)=O)s2)=O)CCCC(NC(c2ccn(C)n2)=O)CC1 NC1CCCC1NC(=O)C(=O)NC1CCN(Cc2ccccn2)C1 N1(C(C2CC(OC)CN2C(=O)CN2CCC(C)C2)=O)CCCOC(C)C1 N1(C(C(CCC)CNC(=O)C(C)CO)=O)CCCC(C)(C#N)C1 c1(C(N2CCC(CNC(c3cc(C)ns3)=O)C2)=O)cc2c(C)cccn2n1 C1(NC(C(C)OCCC#C)=O)CN(C(=O)Cc2ccc(C)nc2Cl)CC1N=[N+]=[N-] C1(C(N2CC(NC(CCc3c(C)nccc3)=O)(CO)C2)=O)Cc2nnc(C)n2C1 CC(C(=O)N(CCCN(C)C(c1noc2c1CCCCC2)=O)C)C(C)S(C)(=O)=O c1(C(=O)NC2CN(C(C3CCC4CC34)=O)CC23CCC3)cnn2cccc2c1 c1(C(=O)NCC2C(C(=O)NC(C(C)C)CN(C)C)C2)c(O)cccc1F c1(C(N2CC(OCCNC(CC3N(C)C(=O)CC3)=O)C2)=O)cc(O)nc(O)n1 N1(CC(=O)N(CCCNC(CC(C=C)C)=O)CC)C(=O)NC(CC)(CC)C1=O c1(CC(N2CCN(C(c3ccc(C#C)cc3)=O)C3C2C3)=O)ccc2c(c1)CCC2 C1(C(=O)NC(C2CCN(C(c3nccn3C)=O)C2)C)CCCCC1(F)F N1(C(CCN(C(=O)CNC(=O)OCCF)C)=O)CCCC(OC2CCCC2)C1 C(c1ccccc1S(=O)(=O)c1ccncc1)N(C1CS(=O)(=O)CC1O)C Cc1ccc(CC(=O)NC(C)CCNC(=O)C(c2cncnc2)C)c(F)c1 C1(N2C(NC(=O)NCC=C3CCSC3)CC2)CCOCC1 c1(C(=O)NCCC(C)(C)NC(c2scnc2C2CC2)=O)ccc(CO)nc1 C(=O)(C(CC(C)C)C(N)=O)N1C(CS(=O)(=O)N(CC)CC)CCC1 CCS(=O)c1ccccc1C(N1CCCC(CNC(=O)CCNC(C)=O)CC1)=O C(C(CC1CC1)C(=O)NCCN1CC(CF)C1)NC(C1(C)CC(=C)C1)=O CC1CCN(C(c2ccc(C#N)o2)=O)CC1CNC(=O)C(C)(C)CF C1(C)(NC(c2n(CCC(=O)OCC)nnn2)c2ccn(C)n2)CCCOC1 C1(CNC(CN2CC(C)C2)=O)CCC12CCN(C(C1(F)CCOC1)=O)CC2 C(C(=O)N(CC(=O)NCC1CCCO1)C1CC1)(C(C)C)OCC N1(C(CC2CN(C)C2)=O)CCC(C)(C)C1CNC(C1CCC(=O)N1C)=O C(=O)(C1Cc2c(Cl)cccc21)NC(C)CCNC(c1csc(CO)n1)=O Cc1cccc(CS(CC2(NC(C3COC(C)C3)=O)CCC2)(=O)=O)c1 c1(CNC(C2(C(F)(F)F)CCC2)=O)cnn2c1CN(c1nccc(CO)n1)CC2 N1(C(C2CCC(=O)C2)=O)CCN(C(=O)Cc2ccsc2Cl)C(c2ncc[nH]2)C1 C1(C2CC2)(CNC(c2csc3nccn23)=O)CCN(C(=O)C=Cc2cncs2)C1 N1(C(c2c(CCC)nco2)=O)CCOCC1CN(C)C(C1CCCOC1C)=O C(c1ccc(C)c(Cl)c1)=CC(N1CC2C(CNC(C(C)SC)=O)(C2)C1)=O C1(OCC(=O)NCCC2CCN(c3ccc(CC)cc3)C2)Cc2ccccc2C1 N1(C(c2cc(C)ncn2)=O)CC(NC(=O)CCc2ncc(C)[nH]2)CC(O)C1 N1(C(CCN(CC(C(C)C)C)C)=O)CC(NC(=O)CN(C2CCC2)C)CC1CO N(C(=NCc1ccc(OC(F)F)cc1)NCc1ccsn1)C(C1CCCCO1)C c1(C(=O)NCCNC(c2c(OC)ccc(C(N)=O)c2)=O)cccc2oc(C)nc12 c1(C(=O)NC2C(CNC(C(C(CC)C)NC(C)=O)=O)C2)ccc2c(c1)CCCN2 N1(C(c2c(C)n(C)cn2)=O)CCN(C(=O)Cc2nnc(O)s2)C(CO)C1 c1(C(=O)NCC2N(C(c3nc(COC)oc3)=O)CCCC2)ccc(S(C)=O)cc1 c1(C(N2CC(CNC(C3CCC(C)C3)=O)OCC2)=O)cc(O)nc(C2CC2)n1 c1(-n2cc(C(N(CCNC(Cc3c(C)con3)=O)C)=O)nn2)ccc(Br)c(F)c1 C(=O)(CCCNC(c1ccoc1)=O)NCC(CNC(C1C(C)CC1C)=O)OC CN1CCC(CC(=O)NC2CCC(CNC(c3nc(=O)n(C)[nH]3)=O)CC2)C1=O C1(CN(C(=O)CCC2CCCN2C)CC)CCN(C(C2C=C(C)CS2)=O)CC1 c1(CC)ccccc1SCCNC(Cc1ccc(C)cc1)C(F)F N1(C(C(C(C)C)OC)=O)CC2(CCCC2)C1C(=O)NCC(=O)N1CCCO1 c1(C(=O)NC2(CNC(C(COC)(C)C)=O)CCCCCC2)cccc(F)c1C#N N1(C(C(c2ccc(C)o2)C)=O)CC2(C)CC1(C(=O)NC1CCOC(C)C1)C2 c1(CCC)nc(C)c(C(=O)NCCN(C(=O)C(c2cccc(OC)c2)OC)CC)o1 c1(C(=O)NCC2(F)CC(NC(c3c(C)onc3)=O)C2)cc2c([nH]1)CCC(C)C2 c1(C(=O)OC)n[nH]c(C2c3n(nnn3)CCCN2)n1.C1(C(C)(C)OC)CC2CC2C1 C(c1cc(C)ccc1OC)=CC(N1CC(O)CC(NC(C2C(C=C)C2)=O)C1)=O C(=O)(C(C)(F)C(C)(C)F)NCC(CNC(c1ccc(C)nc1N)=O)C c1(C(=O)NC2C(C=C)CN(C(=O)C(C)NC(=O)CC)C2)cn(C)c2ncccc12 CCC(F)(F)CC(=O)N(C1CCCCN(C(=O)Cc2ccc(F)cc2)C1)C N1(C(c2n[nH]c(CC)c2C)=O)CCC2(C=C(C(=O)N3CCC=CC3CC)C2)C1 c1(CNC(C23C(CN(C(CCSC)=O)C2)C3)=O)c(C(=O)O)[nH]c2ccccc12 C(=O)(C(CN(C)C)C(C)C)NC1C(N(CC=C)C(C2CCCCC2O)=O)OCC1 CCC(CC(=O)NC1(CO)CCCN(C(c2ccc(C#N)o2)=O)C1)CC(F)(F)F Cc1cc(C)n(CC(=O)NCC2CCN(C(C3(C)CCC3C(=O)OC)=O)CC2)n1 Cc1cc2cc(C(N3CCN(C(C4(C(N)=O)CC4)=O)CC3)=O)[nH]c2cc1Cl N1(C(C2C(C)=C2)=O)CCCC2(CCN(C(=O)C(F)(F)c3nccs3)CC2)C1 C=Cc1cncc(C(N2CC(NC(C3C(C)C3C)=O)C(CO)C2)=O)c1 c1(CC)ncc(C(=O)NC(CN(C)C(c2cscc2C2CC2)=O)CC)[nH]1 C(CC)(CCCC(=O)NOCc1ccc(F)cc1)NC(C1C(=C)C1C(=O)OC)=O c1(C(=O)NC2(CCC(N3CCC(OCC#C)C3)=O)CCCC2)nc(C)sc1C C1(NC(CC(C)(C)C(=O)O)=O)C(F)(F)C12CCC2.n12cc(nn1)COCCC2 C1(C(=O)NCC(COC)O)CCOCCN1C(C1CCC(=O)O1)=O CN1CCN(C(c2ccn3ccsc23)=O)C(CNC(=O)COCCF)C1 C1(C#CC(=O)NC2CCC(C)N(C(=O)C=CCNC(C)=O)C2)(CC)CC1 C#Cc1ccc(C(=O)NCCN2CCN(C(=O)C(C3CCOC3)OC)CC2)nc1 CC1CCCCCN1C(c1cccc(-c2cn(CCOC3CCOC3)nn2)c1)=O C1(CCC)CCCN(C(c2cc(CNC(c3cncs3)=O)on2)=O)CC1 N1(C(C2C(CN(C)C)C2)=O)CCC(NC(=O)Nc2scnc2C(F)F)C1 c1(C(=O)NCC(C2CCN(C(C(CC)(C)C#N)=O)CC2)C)cnc2ccnn2c1 C1(C(C)C)CN(C(=O)CCC2CCC(C)O2)CC(=O)N1 c1(NC(C(C)NC(C2CC(=C)C2)=O)(C)C)cnc(C#N)cn1 C(C1CN(C(c2[nH]cc(C)c2C)=O)CC1C(N1CC(C)CC1CC)=O)=CC c1(OC)cncc(C=CC(N2CCC(NC(=O)C(O)CC(N)=O)C2(C)C)=O)c1 N1(C(C2C(C(=O)OC)CC2)=O)CC(CN(C(=O)CC2CC2)C)C2(CC2)C1 C(=O)(CC(c1ccccc1)c1ccccc1)NCC#CCNC(C1C(=C)CC1)=O CCCCC(CC)CC(=O)N1CCC2CCCC12C(=O)NCCC(O)C(F)F c1(C(=O)NCC(CC(C)C)NC(c2c(CC)scn2)=O)cc(Cl)cc(F)c1N C(C)(C(=O)NC1CCC1NC(C1CCN1C)=O)NC(CC)=O C1(NC(CC2CCC(N)C2)=O)CC2(CCC2O)C1 Cn1cc(-c2nc(C(=O)NC3CC(NC(=O)CC45CC(C4)C5)C3)co2)cn1 N1(C(C(CCCC#C)C)=O)CC(C2CCCN(C(C3(CSC)CC3)=O)C2)C1 C1(N(C(=O)CC2COCCO2)C)CN(C(c2ncccc2N)=O)CC12CC2 C#Cc1ccc(NC(=O)C(=O)NCc2noc(-c3cccc(F)c3)n2)c(Cl)c1Br CC1(C(=O)NCCOC2CCN(C(c3ccnn3C(F)F)=O)CC2)COCCO1 N1(C(C(CC)n2ccnc2)=O)CCC(C(=O)NCc2nccnc2C)CC1(C)C c1(CSC)cccc(C)c1NC(=O)C(N1CC2CC(NC(=O)OC(C)(C)C)C1C2)=O CC1CN(C(c2ccco2)=O)CC1NC(C1(Cc2ccccc2Cl)CC1)=O C=C1CC2(C1)CC(C(=O)NC1CCCN(C(=O)Cn3nc(O)ccc3=O)CC1)C2 N1(C(c2c(C(F)(F)F)nn(C)c2Cl)=O)CCCC2(CCN2C(c2ccno2)=O)C1 C1(CCC#C)CCCN1C(C1CCCC1CNC(=O)C(F)C1CCOC1)=O c1(OCCC)cccc(CN(C2CC2)C(c2ccc(C3CC3)cc2)C)c1 O=C1Cc2cc(C(=O)NC3(CNC(c4cc5n(n4)CCCC5)=O)CC3)ccc2N1 C1(NC(CCOC(C)C)=O)CCC(N(C)C(c2nnn(C)c2C(F)F)=O)CC1 CCC(CC(=O)NCC1CCN1C(=O)CCCn1ccnc1)C1CC1 N1(C(C(=O)NCC)=O)CCN(CCN(C)C(c2occc2C2CC2)=O)CC1 c1(OC)cccc(NC(=O)C(N2CCC(C(F)F)(OC)C2)c2ccsc2Cl)c1 N1(C(c2ccc(C(=O)OC)o2)=O)CCN(C(=O)C=CBr)C(C)CC1C c1(C(=O)NCC2C(C(=O)NCC3(O)CN(C)C3)CCCC2)cnc2cc[nH]c2c1 C(=O)(CC(c1ccccc1)n1cnnn1)NCC(C)NC(=O)C(C)OC(C)(C)C C1(CNC(CCCC)=O)C2CCCC1N(C(=O)COC1CN(C(C)=O)C1)C2 c1(-n2cc(C3CCC(F)(F)CC3)nn2)nc2ncccn2n1.FC(F)S c1(NC(=O)Cc2ccc(NC(c3ccccc3)=O)cc2)ncnc2scc(Br)c12 C(=O)(CCC(=O)N1CCCC1(C(=O)N(C)CC1CCSC1)CC)NCC C(=O)(CCCC(C)(C)NC(c1cc(C2CC2)on1)=O)N(C(CC)C1CC1)C c1(C(N(C)CC2OCCO2)=O)cn2c(n1)CN(C(c1ccc3nc[nH]c3n1)=O)CC2 c1(C(=O)NCC(C)N(C(c2cnc(CCC)s2)=O)C2CC2)cn(C(C)C)nc1C c1(OC)ccc(Br)cc1C(N1CCC(CN(C(=O)C(F)C(F)(F)F)C)C1)=O C(=O)(CCC(=O)NN(C)C)NC1CC(NC(C=CC(C)(C)SC)=O)C1(C)C CC1(CNC(C2(CNC(c3nsnc3O)=O)CC3(CC3)C2)=O)CC(F)(F)C1 C1(CCNC(C2CC2c2ccccn2)=O)(OC)CN(C(=O)C=Cc2cncs2)C1 C1(C)(CC(=O)NCC(C)(C)NC(C2(N(C)C)CCCCC2)=O)CC1(Cl)Cl Cn1ncc2c(O)cc(C(N3CCN(C(=O)CC(C)(C)F)CC3C3CC3)=O)cc12 C1(CC(N2CCC(CNC(CC(COC)C)=O)CC2)=O)CCC2(CC1)COC2 C1(C(N2CC(O)(CNC(C(CC)n3ccnc3)=O)C2)=O)CN(S(=O)(=O)N(C)C)C1 N1(C(CCC2CCN(C)CC2)=O)CC(NC(C2CC(C)(C)CO2)=O)CCC(O)C1 C1(NS(CCCCC)(=O)=O)CC=C(c2ccc(F)cc2)CC1 c1(CC(N2C(C)CCC(NC(C3OCCCO3)=O)C2)=O)noc2cc(F)ccc12 N1(C(CC(C)(C)C)=O)CC2(C1)CN(C(c1cccc(-n3cnnn3)c1)C1CC1)C2 c1(OCCC(=O)NCC(CNC(=O)C=Cc2cc[nH]n2)F)ccc(F)cc1 C1(C(=O)NC(C#CC)(C)C)CCC(C)(C)N(C(c2cnc(Cl)n2C)=O)C1 C(=O)(CC(O)CCSC)N1C(CCNC(C2N(CCC)CCC2)=O)CCC1 c1(C(=O)NCCOCCCNC(CC2CN(C)C2)=O)cc(S(N)(=O)=O)n(C)c1 C1(NC(C2OCC(C)(C)C2)=O)CCC2CCN(C(C3CCCCCC3)=O)C1C2 c1(C(N2CC(O)(C(CNC(CCC)=O)(C)C)C2)=O)cc2c([nH]1)CCC(C)(C)C2 N1(C(c2c(C)nc(O)cc2)=O)CCC(C2CC2)C1CNC(=O)C1=CC2CCCC12 N1(c2c(S(=O)(=O)NCc3ncc(CC)o3)cccn2)CC2(C)CN(C)CC2(C)C1 CCCC(CCCNC(=O)CCC1CCOC1)NC(=O)C(C)(C)C1CCCC1 c1(C(CC=C(C)C)NC(=O)C(F)CC2CCC2)c(C)cccc1Br.C1CN1 C1(CC(=O)NCCOCC(F)F)CCCN(C(C2C=CCS2)=O)C1 C12(CNC(c3nnc4ccccn34)=O)CN(C(C3CC=CCC3)=O)CC1CCO2 CC1CCC(C(=O)NC(c2ccno2)C)N1C(c1c(Br)cnn1C)=O C(=O)(CCS(C)=O)N(CC(C)(C)CNC(=O)Cc1csc(C2CCCC2)n1)C CC1CCCCC1CC(=O)N(CCCCN(C(=O)C=Cc1ccc(Cl)s1)C)C C1(CCNC(c2ccc(C)nn2)=O)CN(C(c2c(C)csc2C)=O)CC(C)O1 N1(C(Cn2cc(C(C)=O)nn2)=O)CCC(C)C1CNC(c1cc(C)sc1C)=O N1(C(c2c(-c3cn(C)nc3)cccc2)=O)C2CCC1CC1(C2)N=N1 c1(C(=O)NC(CN2CCN(C(CCC(C)OC)=O)CC2)C)cncc2sccc12 c1(OCC)ccc(-c2nnc(CN3CCCC(CNS(C)(=O)=O)C3)o2)cc1 Cc1noc(C)c1CC(C)C(=O)NCC1CC(F)CN1C(C1CCCC(O)C1)=O c1(C(C)=O)[nH]c2ccccc2c1C(=O)NCC(C(C)(C)C)NC(C1CC1F)=O N1(C(C(=O)NC2CC2)=O)CCCCC(C2CN(C(C3CCO3)=O)C2)C1 C12(C(N3CC(C)OCC3)=O)CCN(C(=O)C=CC3CCCC3)CC1C2 c1(C(=O)NCCCN(C)C(c2cc(C(F)F)no2)=O)ncc(Br)cc1F c1(C(N2CCC(N(C)C(c3ccc(Br)nc3Br)=O)C2)=O)ccc2ncccc2c1 C1(NC(C(CCOC)NC(=O)C(C2CCOCC2)O)=O)CC2COCC(C1)C2 C=C1CC(C(F)(F)F)(C(=O)NCCN(C)C(c2cscc2CC)=O)C1 C1(C)(CC(=O)N(CCN(C(C2C(C=C)C2)=O)C)C)CCCCC1 C1(C(=O)NC(c2ccccc2)CNC(C(CSC)C)=O)(C(F)F)CCCCC1 N1(C(c2c(CC)ncs2)=O)CC2(CCCCN(C(=O)C(C)(C)CNC(C)=O)C2)C1 c1(N2C(C(CNC(C(C(C)C)N(C)C)=O)(C)C)CCC2)nccc(C#N)n1 N1(C(c2cnc(SC)s2)=O)CCC2(CC1)CC(NC(=O)CCCC1CC1C)C2 C(=O)(CCCC(C)(C)CC)N1C(CCC)CN(C(c2conc2C2CC2)=O)CC1 N1(C(c2c(C)ccs2)=O)CCC2(CCC(CNC(=O)C(O)C(F)(F)F)OC2)CC1 CCCCC(CC)C(=O)N1CC(NC(=O)C(C)(C)C(=O)NC)CC(C)(C)C1 C1(NC(CC(C)(C)NC(C2CCCC(OC)C2)=O)=O)CN(C)CC1(F)F N1(C(CNS(CCCC)(=O)=O)=O)CCCC2C1CCN2C(c1ccc[n+]([O-])c1)=O C1(NC(=O)CC2COCCN2C(C2COCCO2)=O)CCC2(CC1)N=N2 C1(C(N(C(CC)CO)C)=O)CN(C(=O)C=Cc2cn(C)cn2)C(C)(C)C1 C(N=c1nc(N2CCC(CCN(C)C)C2)c2[nH]ccc2[nH]1)C1CCCN(CC)C1 CCC(C)CC(C)N(C(=O)CCC(C)NC(=O)C(C)CCN(C)C)C C1(CC=C)(NC(c2cc(CSC)on2)=O)CCCN(C(=O)C=C2CCSCC2)C1 N1(C(C2CCCN(CC(C)C)C2)=O)CC2CC(NC(C3CC(O)C3)=O)C(C2)C1 Nc1c(C(N2CCOC(CNC(=O)CCSC(F)(F)F)C2)=O)sc2nccnc12 N1(C(C(c2ccco2)NC(C=Cc2n(C)ncc2)=O)=O)CCC(O)C(C)(C)C1 N1(C(c2c(C)cc[nH]2)=O)CC(NC(=O)CCN2CCC(C)CC2)CC1C c1(N(C)C)nc2ccsc2c(=NCCN(C(c2cnccn2)=O)C2CC2)[nH]1 N1(C(C2(OCC)CCOCC2)=O)CCOCC(NC(c2nnc(S)n2C)=O)C1 N1(C(C(C)(C)C)=O)CC(NC(c2ncccc2C(F)(F)F)=O)CC(C(F)(F)F)C1 c1(OC)cc(C(=O)NCCN(C(=O)C(C)CC2CCCO2)C)sc1Br C(=O)(C1=COCCC1)NCc1ccc(C(N(C(C)CO)CC2CCC2)=O)cn1 N1(C(CCC(C)=O)=O)CCC12CCN(C(c1cc([N+](=O)[O-])ccc1C)=O)CC2 c1(COC)nnc(C(=O)NCCC2CCN(C(=O)C(C)OC3CCCCC3)C2)s1 C1(CC)CN(C(=O)Cc2ccc(C)cc2Br)CCN1C(=O)CSC1CCCCO1 c1(C(N2CCC(N(C(c3ccc(C(C)=O)[nH]3)=O)C)C2)=O)cc(O)nc(O)n1 c1(OC(C)C(=O)N(C2CN(C(=O)C(C)(C)C3CC3)CC2F)C)ccc(F)c(F)c1 N1(C(c2c(CC)nc(=N)[nH]c2)=O)CCCN(C(=O)CC2C=CCCC2)C(C)C1 C1(N(C)C)(C(N2CCC(CNC(=O)Cn3nnc(C(C)(C)C)n3)C2)=O)CCCC1 N1(C(C(CCC)O)=O)CCC2(CCC(NC(=O)CCC3CCC3)C2)C1 CC(CC(C)NC(=O)Cn1nnc(=N)[nH]1)NC(=O)C(c1ccccc1)C1CC1 C1(C(=O)Nc2c(COC)nsc2)C(C)CCN1C(=O)CN1CCCC1 C1(C2CN(C(CSCC#C)=O)C2)CN(C(=O)COCC(=C)C)CCO1 N1(C(C(N2CCOC2=O)C)=O)CCCC(C(N2CCCC2C(=O)NC2CC2)=O)C1 c1(C(C)NC(CN(C2CC(C#N)C2)C(C(C)=C2CCC2)=O)=O)nncn1C Cn1ccc(C(=O)N(CCCCCCNC(C2CCOC(=O)N2)=O)C)cc1=O C(CCN=c1[nH]c(=NCc2ccsc2)[nH]c2c1SCC2)c1ncn(C)n1 C12(C(=O)NCC(C)(C)NC(=O)CCCS(C)(=O)=O)CC3CC(CC(C3)C1)C2 c1(C(=O)NCC(C)N(C(CC=C(C)C)=O)C)ccnc(N2CCCCC2)n1 C1(C(=O)NCC(C)CN(C(=O)C#CC2CC2)C)(COC)CCCCO1 C(=O)(C1Cc2ccccc21)NC(C)(C)CCNC(=O)Cc1cnc[nH]1 CC1CC(COC(C2(NC(=O)OCC3CCCCC3C)CCCCC2)=O)C(C)O1 Cc1ccc(C)c(S(=O)(=O)N2CC3C(C2)N3C(c2cc[nH]c3ncc(I)c2-3)=O)c1 c1(C(=O)NCC2CCN(C(c3ccc(C(C)=O)cc3)=O)C2)ccnc2[nH]ncc12 Cc1cc(C(N2CC(CNC(c3nn(CCO)nc3C)=O)CC(C)C2)=O)cc(F)c1 N1(C(C(C)Oc2c(OC)cccc2)=O)CC2=C(C1)CN(C(c1cscc1C)=O)C2 C(=O)(C1=CC2CCCCCCC12)NC1CC(CNC(C(=O)NCC(F)(F)F)=O)C1 N1(C(c2c(C)n(C)nc2)C(=O)NCC2CCCO2)CCC2CCCC12 c1(NCCCCCN(C(C)C)C)ncccc1S(=O)(=O)NCC1OCCC1(C)C N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC2CCCC12C(=O)NC1CC(=O)NC(=O)C1 Cc1n[nH]c(C)c1C(=O)NC1CCN(Cc2cn(C3CCC3F)nn2)CC1 C=CCCCC(=O)NC(C1CCOC1)CNC(c1cc(C(F)F)ncn1)=O C1(N(C)C)(C(N)=O)CN(C(C2CCC(NC(=O)CC3CC3C(=O)O)C2)=O)C1.C1CC1 C1(C(N2CCC(CN(C)C(C3CCCC3(C)C)=O)C2)=O)CSCC(=O)N1 C1(CNC(C(C#C)(C)C)=O)CCC2CN(C(C3(C(=O)N(C)C)CC3)=O)CC12 CCC(CO)(C(=O)NC1C=CC(C(=O)NCc2ccccc2OC)C1)OC c1(CC(=O)NCCNC(c2[nH]n(C)c(=O)n2)=O)ccn2cncc2c1 N1(C(C2=C(C)CCC2)=O)CC2OCCN(C(c3cc(F)cc(F)c3N)=O)C2C1 CC(C)CC(C(=O)NC(C)(C)C)N(C(=O)CC(c1cc(F)cc(F)c1)N(C)C)C C(=O)(C(C)(C)C(C)NC(=O)CCC1CCOC1)N(CCCC(O)CO)C C1(NC(c2ccc[nH]2)=O)CCN(C(=O)Cc2cnns2)C12CCC2 Cc1ccc(F)c(C(=O)NC(CN=[N+]=[N-])C(=O)NCC2(N(C)C)CC2)n1 C=CCCCCCC(=O)NCC1CCC1NC(c1cc(C)cc(O)c1)=O C1(C(N(CCNC(C)=O)C)=O)CCCN(C(c2cn(C)nc2C)=O)C1 C1(NC(COC)=O)CN(C(C2CC3C=CC2O3)=O)C2CCCCC12 c1(C(=O)NCCCCCN(C(C(CC=C)C)=O)C)ccc2c(c1)NC(=O)CCC2 C1(CNC(C=CC(CC)=CC)=O)C(C2CC2)CCN1C(c1nccn1CC)=O N1(C(C=C(C)C)=O)CCOC2(CCN(C(=O)CNC(=O)C3CC3)CC2)C1 c1(C(N2CCCCC(N(C)C(c3ncncc3Cl)=O)C2)=O)coc2c1CCCC2 N1(C(C(=O)NC(C)C)=O)CCN(C(=O)CCc2ccoc2)CCC1C N1(C(C(CCC)C)=O)C(C(N2CCC(CC(C)C)C2)=O)C2(CC2)C1Cl C#CC1CCC(C(=O)N(C)CCNC(=O)Cc2cnsc2)CC1 CC(C)S(=O)(=O)CC(=O)NC1CCCC1NC(=O)CCn1ncc2ccccc12 C(=O)(C1CCCc2sccc21)N1C2CCCN(C(c3[nH]cc(C#N)c3)=O)C2CC1 c1(C(=O)NC(c2cccnc2)C(=O)N(CCC(C)C)CCO)cc2cnccc2[nH]1 C1(C)(CNC(c2cc(SC)oc2)=O)CCCN1C(=O)Cn1cccn1 CN1CCCC(CCC(=O)N(C2C3CN(C(C4(F)CCC4)=O)CC23)C)C1 C=C(C)CCCC(=O)NC1CCC12CN(C(c1ccc(Cl)cc1Br)=O)C2 C#CCCCCCCCNC(=O)C1=CCCN(C(C2(C#N)CCOC2)=O)C1 N1(C(CNC(C)=O)=O)CC2(CCC2)CC1CNC(=O)Cc1ccc(F)cc1 C1(CNC(c2c(C)scn2)=O)CN(C(=O)CCC(C)C#N)C(C)(C)C1 CC1(NC(=O)CSc2ccc(F)cc2)CCN(C(C2(C)COCC2(F)F)=O)CC1 N1(C(CC(C(C)C)OCC)=O)CCN(C(c2cc(OC)cs2)=O)CC(CO)C1 N1(CC(N2C(C(N)=O)CC2)=O)CCN(C(=O)CC(O)C2CCCC2)CC1 C1(NC(CSCc2cccc(C)c2)=O)CC12CCN(C(C13COCC1C3)=O)C2 c1(C(=O)NCC23CCC(CC2)OC3)ccc2c(c1)CC(C(F)F)O2 CCC(CC(C)C)C(=O)N1CCC(C(=O)NCC23CCCN2CCC3)O1 C1(NC(C2CC(OC)C2)=O)CC2CC1N(C(c1ccc(-c3csnn3)cc1)=O)C2 c1(NC(C=Cc2n(C)ncc2)=O)ccccc1N=[N+]=[N-].C12C3CC1N(C3)C2=O C1(C(=O)NCC(C)NC(C=C(CCC)C)=O)CC(CC)(CC)C1 O=C1CC(C(N2CC3(C2)CN(C(c2csc(S)n2)=O)C3)=O)Oc2ccc(Cl)cc21 c1(OC)nc(C(=O)NC2CCCN(C(=O)CC3(C)CC3)C2)sc1C C(C(C)CC(=O)N(CCCNC(=O)CCC(=O)OC(C)(C)C)CCO)OC N1(C(CS(CC)=O)=O)CCCC(C)(C(=O)NCC(=O)OCC2CC2)C1 C1(C(N2C(C(=O)NCCc3ncccn3)CC(OC)C2)=O)CCC(O)CN1C N1(C(C)=O)CC2CC1CN2N1CCCC1C=O.c1(C)c(C)coc1C C(CC(CC)C(=O)NC1CC2(C1)CC2NC(=O)CC1(CS(C)(=O)=O)CC1)=CC Cc1c(C(=O)NC2CCN(C(=O)CCC3CCCN3C)CC2)ccc2c1CCC2 c1(C(C2CCOC2)CNC(c2n[nH]cc2Br)=O)ccccc1.C1C=CCN1 C1(OCC#C)CN(C(=O)C=C(C)CNC(=O)COC2CC2(C)C)C1 N#Cc1cccc(NC(=O)CNCCc2ccccc2Br)c1 Cc1cc(C(=O)NCC(c2ccc(F)cc2)NC(=O)CC(C)(F)F)cn1C N1(CC)CCC(N(C(=O)C(C)(C)NC(=O)COCc2nc[nH]n2)C)C1 c1(C(N2C(C)CN(C(COCCOCC)=O)CC2C)=O)cncc(S(C)(=O)=O)c1 C1(C(N(C(c2cscn2)CO)C)=O)C2CN(C(=O)CCC(=O)N(C)C)CC12 C1(COC)(CNC(=O)C(C)c2ccco2)CCN(C(C2CC(C)CCO2)=O)C1 C1(C(N(CCC(=O)OC)CC)=O)CC(C)CCN1C(c1nnn(C)c1C)=O N1(C(c2ccc(C)n(C)c2=O)=O)C2COCC1CC(NC(C1CCCOC1)=O)C2 c1(NC(C(=O)N(CCOCCOC)C)=O)cc(C(F)(F)F)cc(N)c1 c1(CN2CC(C(=O)Nc3ccc(SC)cc3)OCC2)c(Cl)cnc(Cl)c1Cl C(=O)(CC1CNc2ccccc21)NC1(C)CN(C(=O)Cn2cc(C3CC3)nn2)C1 c1(C(C(=O)N(CCNC(C2(OC)CCCC2)=O)C)=O)ccc2c(c1)CCCC2 C1(c2c(SC)csc2)NC(=O)N(CCF)C2=C1C(=O)NC2(C)C C(=O)(CS(=O)(=O)CC(C)C)NCCC1(O)CCCN(C(c2[nH]cc(CC)c2)=O)C1 C1(C)(C(N(CCCCCC)C)=O)CCCN1C(=O)C(F)C1CCC1 C1(NC(c2cncc(C)c2Cl)=O)C2CC3CN(C(=O)C(C)O)C1C3C2 N1(C(CCCCCCSC)=O)CC(NC(=O)CN(C)C(C)C)CC12CCCCC2 C(C(C)(C)C(=O)NC)NC(C1(C2N(C(c3c(COC)cco3)=O)CCC2)CC1)=O c1(COC(CCN(CC(C)C)C(=O)OC(C)(C)C)=O)ccc(CCN(C)C)cc1 N1(C(c2ccncc2-c2ccc(-c3nn[nH]n3)cc2)=O)CCN2CCNC(=O)C2C1 c1(C(N)=O)cn(CCC2CC2)nn1.N1(C(c2ccsn2)=O)CC2(C1)CN2 C1(NC(C2CN(C(CCC)C)C(=O)C2)=O)CCCCCC1NC(=O)Cc1ccoc1 C1(CNC(=O)CN(C(=O)C(C2(O)CCCC2)F)C2CC2)CC2(CC2)C(=O)O1 C#Cc1ccc(C(=O)NCC2CN(C(C3CC4COCC4C3)=O)CCO2)cc1C C(=O)(C1=C(Cl)CCOC1)N(CCCCC(=O)N(C)CC1CCN(C)C1)C c1(C(=O)NCC(CC)NC(=O)Cc2cc(C)ccc2C)c2c(c[nH]c1=N)CCC2 CC1(C)CCOC(C(=O)NC2(C)CC(C(=O)NCC3CCC=CCC3)C2)C1 C1(S(C)(=O)=O)(C(N(CCN(C(=O)C=C(Cl)Cl)C)C)=O)CCOCC1 c1(OC)ccc(Br)c(C(N2CCCC2CNC(c2cccn(CO)c2=O)=O)=O)c1 c1c(C)nc2ncnn2c1C.C(C(N=[N+]=[N-])C(=O)NOCCC(F)(F)F)OC(C)=O N1(CC)CCCCC1C(N1CCC(C(C)NC(=O)CCc2cc(C)on2)C1)=O c1(C(=O)NCCCN(C(=O)Cc2cocn2)Cc2ccccc2)ccncc1O N1(C(c2c(CC)ncs2)=O)CC2(COC)CC1(CNC(=O)C(C(C)C)SC)C2 c1(C(=O)NCC(n2cccn2)C)ccc(Cl)cc1CN(C)C N1(C(C(CC)NC(N)=O)=O)CCC(F)(CNC(C2Cc3nccn3C2)=O)CC1 c1(-c2nnc(COC(Cc3cnc(C)[nH]3)=O)o2)cccc(NC(N)=O)c1 CCC(=O)CCC(=O)N1CCC(O)C1C(=O)Nc1cnc(Cl)c(C)c1 C(=O)(C1=NOCC1)NCc1c(C(=O)NC(CCC)C2CCC2)c[nH]n1 CC1(C)CCOC1C(=O)NCC1(C)CCN(C(C2(NC(N)=O)CCCCC2)=O)C1 C1(C(=O)NC(CCNC(CCCNC(C)=O)=O)C)CCCCN1CC(F)F C1(C)(NC(N(CCN(CC(F)(F)F)C)CC)=O)CCCCO1 C(=O)(C(CCCC)NC(=O)C(CC)CCNC(=O)OCC)NCCC(=C)CSC S(=O)(=O)(c1cnccc1N1CC23CCCC2(COC3)C1)NCc1c(C)coc1C C1(O)(CNC(CC(CC)OC)=O)CCCN(C(=O)CSC)C1 N1(C(c2c(CSCC)cccc2)=O)CCCC(C)(NC(=O)C(C)n2cccn2)C1 c1(C(N2CCCC(O)(CCNC(CC(CC)C)=O)C2)=O)cc2ccnc(Cl)c2s1 c1(C(=O)NC2(CNC(C(C)(C)c3ccccc3)=O)CC2)ccc2c(c1)CC(=O)N2 N1(C(COCC(C)C)=O)CCN(C(C2CN3CCC2CC3)=O)CC(C)(C)C1 c1(NC2CCN(C(=O)NC(COC)C)CC2)nccc(N2CCCC2)n1 c1(C(N2CCC(NC(c3ccco3)=O)C(F)C2)=O)cc2cc(Cl)cnc2[nH]1 c1(C(=O)NCCC2(NC(C3CCC(CC)C3)=O)CCC2)nccc2ncncc12 C1(C(=O)NCCCCNC(CC(C)F)=O)CCC2(CCOCC2)O1 c1(CN2CC(C(N(CCN(C)C(C3CCC(=O)N3)=O)C)=O)C2)ccccc1 n1(CC)c(NC(=O)N(C)CCc2cccs2)nc2c1CCOC2 c1(CC)nccnc1CNC(=O)CONC(c1cnc(N)cn1)=O C1(NC(=O)C(Cl)=CCl)CCCC12CCN(C(c1cnc3ccncc3c1)=O)CC2 N1(C(C(CC=C)(C)CC)=O)CC2(NC(=O)CCSCC)CCCC2(F)C1 c1(C(N2CCCc3sccc3C2)=O)c(C(F)(F)F)nc2n1CCCC2 C(=O)(C(CCSC)OC)NC(CC)CNC(c1occc1C)=O c1(C(N2C(CNC(CSCC(C)=O)=O)C(C)CCC2)=O)ccc2ccnn2c1 c1(NC(N2CCCCCC2)=O)ccc2c(=O)n(-c3ccc(F)cc3)c(S)nc2c1 Cc1oc(CO)cc1C(=O)NC1(CN(C)C(C2CC(N3CC(O)C3)C2)=O)CC1 C1(C(=O)NCCC(C)(C)N(C)C)(CC)CCCN1C(=O)CN1CC2CC2C1 N1(C(Cc2cccc(SC)c2)=O)CC(NC(C2(F)CC2)=O)CC12CCC2 C1(C(=O)CN2CCCC(n3nncc3C(F)(F)F)C2)CCC2(CCOCC2)CO1 C(=O)(C(C(C)C)N(C)C)N1C(C2(NC(c3c(C)[nH]cc3)=O)CC2)CCC1 Cc1cc(Br)ccc1C(C)NC(=O)CCSCc1ccccn1 CC1CN(C(=O)CCc2nccn2C)C(C)CN1C(=O)CSCc1ncc[nH]1 CC(C)C(C(=O)N1CC(F)CC1CNC(=O)CC1COC2CC1C2)n1cccc1 C1(CC(=O)NC2CC(NC(c3nc(C)sc3)=O)C2)COC2CC1C2 C(C)(C)(CC(=O)N1CC=CC(C(=O)NC(C)Cc2nn[nH]n2)C1)OC O(NC(=O)C(C)C(F)(F)F)C(CC(C)C)C(=O)NC(C)(CO)C(C)(C)O CCC(CCC(=O)NCc1ncc(C)o1)NC(C1CCN(CC)C1)=O CN1CCN(C(c2cnn(-c3ccccc3)n2)=O)CC1CNC(c1cc[nH]n1)=O C1(C)(C(=O)NCC2C(CNC(CNS(NC)(=O)=O)=O)C2)CC2(CC2)C1 c1(C(=O)NC(CCOC)CNC(=O)C(C)CC2CCCC2)cccc(C)c1Cl c1(NC(=O)NC(c2ccc(C)cc2)CC(=O)O)cnc(-c2nn[nH]n2)cc1O c1(CC(=O)NCC2CCCN2C(C2SCCCS2)=O)ccncc1Cl C1(C(=O)NC2CCC(NC(C(C=C)(C)O)=O)CC2)CCC2(CC1)NC(=O)NC2=O C1(C(=O)NC2C(SC)CN(C(C3CCC(N(C)C)C3)=O)C2)CCc2c[nH]nc2C1 c1(C(=O)NC(C2(CNC(CC(C)SC)=O)CC2)C)occ2c1CCC2 C(=O)(C1=CCCSC1)NC(CCNC(c1c(C)nc(COC)s1)=O)(C)C C(CCC1CCC1)(C(=O)NC(c1ccccn1)CO)NC(Cc1n(C)nnc1)=O C(=O)(CC(C)C(=O)N1CCN(CC(=O)NC(C)(C)CCCF)CC1)OC CCCC(C(=O)NC(C)C=CC(=O)NCc1coc(C)c1)N(C)C c1(NC(C)=O)cccc(C(c2nnnn2C(C)C)NCC(C)OC(F)F)c1 CC(C)(C)C(=O)NCCCC(=O)NCC(C1CC1)NC(c1cc[nH]c1C1CC1)=O c1(C(=O)NC(CC)CN(C(=O)C(O)C2CC2)CC)cccc2nc(O)ccc12 c1(N(CC(COC)(F)F)C)nc(=NC(C)c2nnc(C)s2)[nH]c2c(C)nn(C)c12 C(=O)(C(F)C(F)(F)C(F)(F)F)NC(CCCNC(c1c(C)nc(C2CC2)o1)=O)C C(=O)(CCC(=O)NC1C2CC(NC(=O)CC3C=CCC3)CC12)NCCC c12nnc(o1)CC1(C)CN(C1)C(C)C2.C1(C)(NCCC)CC1 c1(C(=O)NC(C(C)NC(c2cn(C)cn2)=O)C)cc2ccccc2c(O)n1 C1(CNC(C(C)OCC)=O)C(C2CC2)CCN1C(c1cc(C)n(C)c1)=O c1(C(=O)NCCC(C)NC(=O)CCc2csc(-c3ccco3)n2)cn(C)nc1Cl c1(COC)nc(NCCSC(F)F)cc(=NC(C)c2nc(CO)n[nH]2)[nH]1 c1(C(C(=O)NCC(N(C(C2CC(CC)(CC)C2)=O)C)C2CC2)C)ccccc1F N1(C(C2CCCSC2)=O)CCN(C(C2CCc3nnnn3C2)=O)C2(CC2)C1 C1(C(=O)OC)CC2CNCC(C1)C2NC1CCCC(C(=O)OC)C1 C#CCC(C)(C)C(=O)N(C)CC1(CNC(=O)CC2CCCC(C(F)(F)F)C2)CC1 C(=O)(C(C(C)O)N(C)C)NC(CNC(CC1CC(CC)C1)=O)CO Cc1c(F)ccc(C(N2CC(CNC(=O)CCCn3cncn3)C(C)C2)=O)c1N C1(CCCNC(c2cnccn2)=O)CN(C(c2cncc(O)c2)=O)CCO1 c1(CCC)ccc(-c2nccn2CCC(O)CNC(=O)OC(C)(C)C)cc1 C(N=c1cc(Cl)nc(C(C)OC)[nH]1)n1cc(C(=O)OC)nn1 C1(N(C(=O)CC2(O)CCC2)C)CN(C(c2[nH]ccc2C2CC2)=O)CC1(C)C N1(C(C=C(COC)C)=O)CCC(C(C)CNC(=O)COC2CCC2)CC1 C=CC1OCCCC1C(=O)N(CC(C)(C)NC(=O)C1=NOCC1)C c1(C(C)C)nc2[nH]ccc2c(=NCCCn2cnnc2C)[nH]1 c1(OC)ccc(C(C)C)cc1ON(C(=O)COCC(F)F)C(C)C S(=O)(=O)(c1ccc(C(=O)NC2(CNC(=O)CCOCC(C)C)CC2)o1)NC C1(C(=O)NS(c2cc(OC)ncc2)(=O)=O)CCC2(CCN(CCO)CC2)O1 C1(CN2CC(C(=O)OC)N(C)CC2)OC(=O)CC12CCNCC2 N1(C(CCCC)=O)CC2(CCN(C(c3cccnc3O)=O)CC2)C1C(C)C CCC(CCC(=O)Nc1cccc(Cl)c1O)NC(=O)Cc1coc(C)n1 N1(C(CC2CC(C)(C)C2)=O)CCOC(CC(N2CCCC(C(C)(C)C)C2)=O)C1 c1(OC)cccc(CC(=O)NCCCCC2CN(C(C3CSCN3C)=O)C2)n1 Cc1nccnc1C(=O)NC1C=CCN(C(=O)C=CCn2cncn2)C1 C1(C(=O)Nc2cncc(F)c2)(COC)C=CCN1C(C1C=CCCC1)=O c1(CNC(C23CC(NC(c4nc(CC)sc4)=O)(C2)C3)=O)ccc(C(=O)O)cn1 c1(N2CCC(CNC(N(c3ccccc3C(N)=O)C)=O)CC2)cnnc(O)c1Cl c1(OC)ncnc(C)c1C(=O)N(CCCCN(C(=O)CN1CCS(=O)CC1)C)C c1(CC)nc(=N)[nH]cc1C(=O)NCC1CC1NC(c1ccncc1C(F)F)=O O=C(C1CCCc2ncccc21)N1CC2(C1)CN(C(c1cnc(Cl)s1)=O)C2 N1(C(CCOC)=O)CC(C(C)(C)C)CC(CNC(=O)C(c2cnn(C)c2)O)C1 c1(NC(C2(C(C)C)CCN(C(C)=O)C2)=O)cn(C2CCc3c(Br)cccc32)nn1 N1(C(C2(CCOC)CC2)=O)CC(N(C(=O)CC(C)C2CC2)C)C2(CC2)C1 C1(C(N(CCCC(=O)NC(c2c(C)ccnc2)C)C)=O)CCCC(C#N)C1 C(C(C)(C)C(C)(F)F)NC(CC1(N(C(Cc2c(C)cccc2)=O)C)CC1)=O c1(OC)c(C(=O)NC(CNC(=O)C(C)c2ccco2)CC(C)C)csc1Cl c1(C(C(=O)N(CCNC(c2c(CC)ocn2)=O)C2CC2)O)ccc([N+](=O)[O-])cc1 C1(N(C(Cc2c(C)con2)=O)C)CCC(NC(=O)Cn2cc(Cl)cn2)CC1 c1(CCC(=O)NC(C2N(C(C=CC)=O)CCCC2)C)ccc2c(c1)OCCCO2 c1(OC)cc(OCCc2ncccc2SC)ccc1[N+](=O)[O-] C(=O)(C(C)(C)C(N)=O)NCC1(OC)CCN(C(CC(COC)C)=O)C1 c1(C(=O)NC2CN(C(Cc3nc(C)sc3)=O)CC(O)C2)cc2c(nn1)CCCC2 c1(C(N2CC(NC(=O)COC3CCCC3)CC(C)C2)=O)c(S(N)(=O)=O)ncn1C N1(C(COC2(C)CCC2)=O)CCC(NC(=O)C(C)(C)C2CC2)CC1C1CC1 c1(C(=O)OC)ccc(O)c(C(=O)NCCCN(C(=O)C(F)C2CCC2)CCO)c1 c1(C(=O)NC2CN(C(CCC#C)=O)C(CC)(CC)C2)ccc2c(=O)ccoc2c1 C#CC(C(C)(C)C)NC(=O)C=CC(C)NC(C1CC(=O)CCO1)=O C1(NC(c2ccc([N+](=O)[O-])cn2)=O)CC2CC(C1)CN(C(c1nocc1Cl)=O)C2 C1(NC(CCOCCC)=O)CCCC1(C)CNC(=O)C(C)(CC)OCC N1(C(=O)NC2(C(N3CC(F)(F)C3)=O)CCSC2)CCC1 N1(C(Cc2c(OC(C)C)cccc2)=O)CCCCCC1CNC(c1cnsn1)=O N1(C(CCCC)=O)CCCCC(NC(C2CC(CCC)C2)=O)C1 C1(C2CC2)(C(=O)NCCCCCCNC(=O)C(F)n2cccn2)CC=CC1 N1(C(CCSC)=O)CC(NC(=O)CCC2CNC(=O)N2)CC12CCCCCC2 c1(CC(N)C(=O)N(CCO)CC2CCOC2)ccc(O)c(Br)c1 c1(C2(C(N3C(CCCNC(C(C)N(C)C)=O)CCC3)=O)CC2)cncc(Br)c1 C1(CCC(=O)NCC2(CNC(c3n(CC)ccn3)=O)CCC2)CCCC(O)C1 C1(C)(CC)C=C(C(=O)NC2(C(C3(NCC=CC(=O)NC)CC3)=O)CC2)C1 C1(NC(c2c(OC)ccnc2)=O)(CNC(C2CCOC2C)=O)CC2CCC1CC2 N1(C(C23OCC(N)C(C2)C3)=O)CC2CC(C1)CS(=O)(=O)C2 C12(CNC(c3nc(CC)oc3)=O)CN(C(C3CCOC3C)=O)CC1CCO2 N(C(=NCCc1ccccn1)NCC1(CO)CCC12CCC2)C(CC)C c1(C(N(CCCNC(C(C)Oc2cccc(C)c2)=O)C)=O)cc(C)ncc1C C=CCC(C)C(=O)N1CCC(NC(=O)C(C)(C)Cc2ccccc2Br)C1 C1(CC(=O)N(CC(C)OC)C)CC(C)(C)CN1C(c1ncccc1C)=O C1(C(=O)N(CCN(C(=O)C(C#N)CC)CCC)CC)CCCN(C(N)=O)C1 C(c1ccco1)=CC(=O)NCC1CCN1C(=O)CC1COC(=O)N1 O=S(=O)(CCn1nccn1)COCc1ccccc1 c1(C(=O)NCC2(NC(C(CC)NC(C)=O)=O)CCC2)nccc(OC)c1C c1(CC(=O)NC(C2CCN(C(CCC=C=C)=O)C2)C)c(C)cc(C)nc1O Cc1ccc(Cl)c(F)c1C(N1CCCCC(NC(=O)CCC2CCCCO2)C1)=O Cc1ccc(CN2CCN(CCOC(F)(F)F)CC2)cc1NC1CC1(C)C c1(C(=O)OC)c(OC)cc(NC(C2C3CN(C(C4(C5CC5)CC4)=O)CC23)=O)cc1O C1(NC(c2cccnc2Cl)=O)CCCN(C(C2(C(F)(F)F)CCC2)=O)C1 N(C1CCCn2nccc21)C(C1=CCCN(C(C(COC)(C)OC)=O)C1)=O C1(CNC(CC(C)OC)=O)CN(C)CCN1C(=O)CCCc1cnccn1 CC1CCc2nc(C(N3CCC(CN(C(=O)CC(C)(C)F)C)CC3)=O)cn2C1 C(=O)(CC(F)(F)CC(=O)OC)NC1CC(CNC(C(CC)(C)CC)=O)C1 N(C1CCc2c1ccc(OC)c2F)CC(=O)NC(CCC)(C)C c1(CC)ccc(C(=O)N(CCCNC(=O)CCCC2CC2C)C)[nH]1 N1(C(C(CC)SC)=O)CC2CC(O)C1C2NC(c1cc(C)c(Cl)cc1OC)=O c1(NCC(N(OCC=CC)C)=O)cc(C(F)(F)F)n(NC2=NCCCS2)n1 c1(C(=O)NCC2N(C(C(C(C)C)NC(C)=O)=O)CC2)nnc(O)c(Br)c1O C(=O)(C1CCCc2c[nH]nc21)NC(CN(C(c1c(F)cc(CC)cc1F)=O)C)C c1(SC)c(C(=O)NCC(C2CCCC2)NC(=O)CC2CC(F)C2)cccc1F C(=O)(C1=CCCC1C)NCCC(Cc1ccccc1)NC(C1CN(C(C)=O)C1)=O C(N=c1[nH]c(=NCC(C2CC2)OCC)[nH]c2ccsc12)C1(OC)CCN(C)C1 CS(=O)C1CN(C(=O)CCCn2cc(-c3nc(C4CC4)cs3)nn2)C1.C1C(=O)N1 c1(C(=O)NCCC(CCNC(C(CC(C)C)O)=O)C)cc(S(N)(=O)=O)co1 C1(c2n(CC)nnn2)(NCCCSC)CC(C)(C)OC(C)(C)C1 C(C(=O)NCC1CN(C(C2(O)CCC2)=O)CC1C(F)(F)F)(C(C)C)NC(C)=O Cc1cc(S(N)(=O)=O)cc(Br)c1C(=O)NCC1(Cc2cccc(F)c2)CC1 N1(C(C(COCC)(C)C)=O)CCC(NC(=O)Cc2nn(C)cc2Cl)C(C)C1 C1(NC(C2(CC=C)CCCC2)=O)CN(C(C2(CCC)CCC2)=O)CCC1F C1(NC(CCc2c(OC)cccc2)=O)CCOC2(CCN(C(=O)C(C)C)CC2)C1 NC(=O)CCCC(=O)N1CCC(F)C(NC(=O)C=Cc2cccc(CO)c2)C1 CCCCC(O)C(=O)N1CC(=C(F)CNC(c2cccn2C(C)C)=O)C1 C1(NC(CCC(C)OC)=O)CCCC2CN(C(c3cnn(C(C)C)n3)=O)CC12 CC(=Cn1ccnn1)C(=O)NC(CNC(=O)CSc1cnn(C)c1)C(C)C N1(C(c2c(CC)occ2)=O)CCCC(NC(c2[nH]ccc2COC)=O)C(F)C1 C1(NC(C(C)Sc2c[nH]c(=N)s2)=O)CC(F)CN1C(=O)CC1CCCN1C C(=O)(N=c1cc(C(C)(C)C)o[nH]1)C1N(C(C2N(C)CC(O)C2)=O)CCC1 N1(C(CC(C(C)C)O)=O)CCCC2(CC(NC(=O)CCC3(C)CC3)C2)C1 c1(C(=O)NCCC2(NC(C=CC(C)C)=O)CC2)cc(O)nc2ncccc12 CC1CC(CO)(NC(C2CCC2CNC(=O)CCn2cccn2)=O)C1 C1(NC(CC(C)C(F)F)=O)CCC2(CC1)CN(C(c1cc(Br)c(O)cc1F)=O)C2 CC(CC(N)=O)N=c1nc(NCCC2CCCCC23CC3)c2c(F)cccc2[nH]1 C=CCCCCCC(=O)NC1CC(C)CN(C(c2ncc(C)cc2C)=O)C1 N1(C(C23N(C(c4c(OC)n[nH]c4)=O)CCC2C3)=O)CCC(F)(C#N)C1 C(N=c1cc[nH]c(=NCCc2cc(C)cc(C)c2)[nH]1)c1cn(CC)nn1 Cc1coc(C(=O)NC(C)C(C)NC(=O)CCCc2ccc(C)s2)c1 C=CCC(C)(C)C(=O)NCC(=C)CCNC(c1ncoc1CCC(F)(F)F)=O C1(C(=O)NC(CC)CN(C)C)(CC)CCCN1C(c1ccc(C2CC2)o1)=O C12(C(=O)NCCn3c(CC)ncc3)COC(C1)C(NC(C1(C)CCCCO1)=O)C2 c1(C(=O)NC(C(C)C)CNC(C2CC3C(C2)C3(F)F)=O)ccc2[nH]c(=N)oc2c1 c1(C(=O)NCC(C)(CC(C)C)NC(Cc2c(C)ccs2)=O)ccc2cccnn12 C(=O)(CC(O)CC(C)(C)C)NCC=CCNC(c1c(C)c(O)ccc1)=O C1(C(N2C(C(N3CCC(OCCF)C3)=O)CCCC2)=O)CC2CC1CC2O C(=O)(C1CCc2nccn21)NC(C1CCCN1C(c1cccc(OCF)c1)=O)C N1(C(C(c2c(C)nn(C)c2C)C)=O)CCC2(CC1)CC2NC(c1n[nH]cc1F)=O c1(C(=O)NC2CCC(NC(C(Br)=C(C)C)=O)CC2)nc2nc(C)ccn2n1 C(=O)(C(C(C)(C)C)C1CCCC1)N(CCCNC(C1CC(C#N)(OC)C1)=O)C CCC(CC)(C(=O)NCC(F)CNC(c1cc(C)cc(C)n1)=O)c1ccccc1 Cc1cc(F)ncc1C(N1CCC(CN(C)C(c2ccccc2Cl)=O)C1)=O C(=O)(C(O)CCSC)NCC1(NC(c2ccc(COC)[nH]2)=O)CCCC1 C1(NCC)CCCC(N=c2cc(C)[nH]c(=NCC3(C)CCCC(C)(C)C3)[nH]2)C1 C12(CNC(CN(C3CC3)CC)=O)CC(CC)(CN1C(=O)CCc1scnc1C)C2 C(CCC(C)C(=O)N1CSCC1C(=O)NCc1cncc(OC)n1)OC N1(C(C2(C#N)CC(=O)C2)=O)CC2(CCC(CNC(c3c[nH]cc(Cl)c3=O)=O)O2)C1 CC1(C)Cc2nc(Cl)ccc2C(NCC2CCC3COCCC3C2)C1 CC1CCC(NC(c2ccc(CNC(c3ccco3)=O)nc2)=O)CC1 C1(O)(C(C)NC(=O)C=Cc2cc[nH]n2)CCN(C(C2C3COCC23)=O)CC1 N1(c2cc(C)[nH]c(=NCC3COC(C)(C)CO3)n2)CCCCC2(CCOCC2)C1 C1(CNC(CCCc2c(C)ccs2)=O)CCCCCN1C(C1CCCOC1C)=O C1(CNC(CCCN(C)C)=O)(NC(=O)C(F)n2ccnc2)CCC(F)(F)CC1 N1(C(CSC(C)C)=O)CC(N(C)C(C2CC3(CC3)CN2C)=O)C(C)(C)C1 CC1CN(C(=O)C(=Cc2cccn2C)F)CCCN1C(=O)C=CCO C1(C)(COC)CC(NC(=O)CC2(CO)CC2)CN1C(c1cnoc1C)=O C1(COC)CN(C(=O)CN(C)S(N)(=O)=O)CCN1C(C1CCCNS1(=O)=O)=O c1(N(C)CC2CCOC2)nc(=NCCC2CC(=O)N(C)C2)[nH]c2c1SCC2 CCCCCC(O)CC(=O)NC(C)C=CC(N1CC2(CC(F)C2)C1)=O c1(CC)cc(NC(=O)C(Cn2cccn2)NC(c2cc(C)on2)=O)cc(C)c1 C(=O)(C(O)CC(C)(C)C)N1C2(C(=O)NCc3ccc(C)c(C)c3)CC2CC1 n1(C(CC)C)nccc1C(=O)N(C1CN(C(=O)COC(C)CC)C1)C c1(C(=O)NC2CCCCN(C(CCN(CCC)C)=O)C2)cc2cccnc2cn1 CC1CCC(C)N1CC(=O)NCCC(C)(C)NC(=O)C=Cc1ccc(C(N)=O)o1 c1(CC)ccc(NC(=O)C(=O)NC(CN2CCCC2)CC(C)C)cc1 C12(NC(CC3C(C)(C)OCC3)=O)CCC(NC(=O)C(O)C(F)(F)F)(CC1)C2 c1(OC)ccc2ncnc(N3CC(NC(c4nc[nH]n4)=O)C(F)(F)C3)c2c1 N1(C(CN(CCC)C)=O)CCCC(C2CCN(C(C3(CO)CC3)=O)C2)C1 CC1CN(C(C2CC3CCCC23)=O)CCN1C(=O)CNC(c1ccccc1F)=O c1(CCC(=O)NCCCN(C(=O)C(C)n2cccc2)CC)cccc(C)c1 C1(C(N(CC#N)Cc2ccccc2)=O)CCCN(c2ccc(F)cn2)CC1 C12(C(N)=O)CC(NC(=O)Nc3ccc([N+](=O)[O-])cc3)(C1)C1(CCC1)O2 C1(CC(=O)NCC2CCC2C(=O)NCC2CN(OC)C2)(COC(C)(C)C)CCC1 c1(C(=O)NCC2C(CNC(c3cc(C)nnc3)=O)C2)cc(C)c(O)c([N+](=O)[O-])c1 c1(C(=O)NC(CN(C(C(C(CC)CC)C)=O)CC)C)cc(OC)c2c(c1)OCO2 N1(C(C2CCCC(=O)N2)=O)CCC2CC2(NC(c2ccc3sccc3c2)=O)CC1 N1(CC=O)c2ccccc2CCC1C.C(C(C)=CC(=O)OC)SC c1(C(=O)NC2CN(C(C(C)Cc3ccccc3)=O)C2)ccc2c(c1)CCCC2=O c1(C(=O)NC23CN(C(CC4CC(OCC)C4)=O)C(C2)C3)ccnc(Cl)c1OC N1(C(Cc2ncc(CC)[nH]2)=O)CCC2CCCN(C(=O)CCCC3CCC3)C2C1 Cc1nc(C(=O)NC2(C(=O)Nc3ccccc3C)CCCCC2)cc(O)n1 c1(C(=O)NCCCCCN(C(c2cc(C(C)C)[nH]n2)=O)C)ccc(F)cc1Cl Cc1cc(NC(C2CC(F)CN(c3ncncc3F)C2)=O)cc([N+](=O)[O-])c1C C(=O)(C1=CCCC1C)N1C(C)(C(N2CC(C#C)(F)C2)=O)CCC1 N1(C(CCN(CC=C)C(c2cn(C)cc2C)=O)=O)CC2(CCCC2)C1 c1(C(=O)NCC2CC(C)CN(C(C3CCC3(F)F)=O)C2)ccn2ccnc2c1 c1(C(=O)NCC2CCCC(NC(C=C(C)C3CC3)=O)C2)cccc2nc(O)oc12 Cc1nccc(C(=O)NCC2(NC(=O)C3=CCCS3)CCOC2)c1C c1(OC)ccccc1C(C)N(C(=O)CNC1CCCS1)C CC1(CNC(c2ncccc2F)=O)CCN(C(=O)CCc2nc(C3CC3)no2)C1 N1(C(C(C)=CC2CC2)=O)CCC(NC(=O)CSc2ccccc2O)C(C)C1 c1(N2CC(CCC)C(CC)C2)ncc(C)cc1S(=O)(=O)CC.C1CN1CC.CC c1(CCC(N2CCC(N(C(C3CC(=C)C3)=O)CCC)C2)=O)cccnc1Cl CON1CCC(CC(N2CCCC2CNC(c2cnc(C(C)=O)s2)=O)=O)CC1 c1(-c2n(CCCC)nc(CC(C)CC)n2)ccc(C2=CCCC2)cc1 C(=O)(C1=NOCC1)NC(COC)C(=O)NCC1(C)CC1 C1(C(=O)NC2CC(CNC(COCCN(C)C)=O)C2)C(C#N)C1(C)C Cc1cccc(C2(C(=O)NC3CCCC3NC(c3scc(C)c3C)=O)CC2)c1 C#Cc1cc(F)c(C(N2CC3(NC(c4ccc[nH]4)=O)CCC2C3)=O)cc1F C(=O)(CS(=O)(=O)CCO)N1CCOCC(NC(c2c(C(C)C)ccc(F)c2)=O)C1 CCC(CC(=O)NCCCOCCCNC(C1(C)CC(=O)N(C)C1)=O)CC(C)C c1(CC(C(=O)OCC)NCc2nc(-c3cccn3C)sc2C)cccc(O)c1F c1(CC(=O)Nc2c(C)cnc(C)n2)ccc(F)cc1[N+](=O)[O-] c1(CC)ccc(NC(C2CC2C(=O)NCCCN(CC)CC)=O)cc1F C1(NC(Cc2c(C)nccc2)=O)CC(C)CN(C(=O)Cc2cncn2C)C1 CCCC(CC(C)C)C(=O)NCC1CC(NC(c2ccc(O)cc2C)=O)C1 Cn1nc(C(=O)NCC2(O)CCCCC2)c2cc(C3=COCCC3)ccc12 N1(C2C(CO)CCCC2)CC2CC(O)C(O)CC2C1 Cc1cn2c(C(=O)NC3CCSC34CN(C(C3CCC(C)(C)C3)=O)C4)cnc2s1 c1(CCNC(c2n(CC=C)nnn2)c2cn(C)cn2)cc(F)ccc1Br c1(OC)cc(Cl)cc(CN2CC3CN(C(c4cc(C)n(C)c4C)=O)CC3C2)c1O C#Cc1ccc(F)c(C(=O)NCC(C)NC(C2CCN(CCO)C(=O)C2)=O)c1 CCC(C(=O)NCC1(F)CCN(C(=O)C(c2ccn(C)c2)C)C1)C(C)(C)CC C(C(C)C(C)C(=O)N1CCC(NC(C2CC(N3CCCC3)C2)=O)C1(C)C)OC C(=O)(C(C)(C)C1=CCSCC1)N(CCCN(C(CCCCN(C(C)=O)C)=O)C)C c1(NC(CN2CC(NC(CC3C(C)OCC3)=O)C2)=O)ccc(OCC(F)(F)F)cc1 c1(SC)cc(C)c(C(=O)NCCCC(C)NC(=O)CCOc2ccccc2Cl)o1 C(=O)(C1CCCc2nn(C)cc21)N1C(C(C)NC(c2cc(Cl)no2)=O)CCC1 CC(C)CC(C)C(=O)NC1CN(C(c2ccc(F)s2)=O)C1 c1(C(=O)NCC(=O)NC(C(C)NC(C2C=CCCC2)=O)CO)cccc(C(N)=O)c1 c1(CC)noc(CCC(=O)N(CCN(C(C2CC2Cl)=O)CC)CC)n1 CC1CCCC1C(=O)NC1(C)CC(NC(=O)C=CC=C(Cl)Cl)C1 Cc1cc(=NC2CCC(NC(=O)C(C)C(C)(F)F)CC2)[nH]cc1C#N C(=O)(C(CO)C(F)(F)F)NC(C)CNC(c1cc(-c2ccccc2)n(C)n1)=O C1(CC(=O)NCC2CC(N(C(=O)C(O)c3ccco3)C)C2)CCC(=O)CC1 N(C(=NCC(C)C(F)F)NCc1cc(C)on1)C(COc1c(OC)cccc1)C c1(C(=O)NCC(COC)NC(c2ccn(CC)n2)=O)c(Cl)ccc(C)c1O CCC(Cc1ccccc1)CC(=O)NC(C)CCNC(=O)CCC(=O)N(C)C N1(C(C2(CSC)CC2)=O)CCC(C)N(C(=O)COCC2CCOC2)CC1 C1(C(N2CCCC(CN(C(=O)C(O)C(C)C)CC)C2)=O)CCC(O)CN1C c1(C(N2CCC(NC(c3ccc(CO)nc3)=O)C(O)C2)=O)cc2cc[nH]c2cn1 CC1CN(C(c2ccccc2F)=O)CC(C)C1NC(c1c(F)cnn1C(C)C)=O C1(NC(C(SC)SC)=O)C2CCC1CN(C(C1CC3(CC3)C1)=O)C2 C1(C(=O)OC)CCC(C)N(C(C2(NC(C3CC4(CCC4)C3)=O)CCC2)=O)C1 c1(CC)cnn2c(NCC(c3ccc(Br)c(F)c3)C)cc(Cl)nc12 Cc1nn(CC(=O)OCc2nc(=O)o[nH]2)c(=O)c2ccccc12 c1(C(N2CC(N(C(c3c(C)coc3)=O)C)C2)=O)c(C)nc(C)nc1C C(=O)(CCCC(=O)NCC(C)NC(C1CCCN1C1CC1)=O)NCC C12(CNC(C3(CC#C)CC3)=O)CC1CN(C(C1CCCN(C(=O)N(C)C)C1)=O)C2 N1(C(c2c(C(C)(C)C)ocn2)=O)CCCC(CC(=O)NCCc2ncc[nH]2)C1 Cc1cc2occ(C(C(=O)NC3CCCC3)N(C)CC3CC3C)c2cc1C CC1CC(C)N(C(c2ncc(C(F)F)s2)=O)CCN1C(=O)Cc1cccnc1F Cc1cn(C)nc1C(=O)N(C)CC1(O)CN(C(c2c(C)nsc2NC2CC2)=O)C1 N1(C(C2CCC(C)(CC)O2)=O)CCOC2CN(C(=O)CC3(O)CCOCC3)CC12 Cc1nnc(N2CCC(C)(NC(c3coc(CC4CC4)n3)=O)C2)c(C#N)c1C N1(C(=O)CC2CCS(=O)(=O)C2)CC(C2CN(C(=O)CCCF)C2)C1 c1(-c2cc(CC)cc(Cl)c2)nc(OC)nc2c1CC(C)CC2 N1(C(C(OC)OC)=O)CCC1(C)CC(N1CCC(c2nc[nH]n2)C1)=O CCC(C)CCC(=O)NC1(COC)CN(C(c2cc(C(C)(C)C)on2)=O)C1 N1(C(CC(C)(C)N(C(c2c(CC)n[nH]c2)=O)C)=O)CCCC(C)(C#N)C1 c1(OC(c2ccsc2)CNC(C(=O)N(C)C2CC2)=O)ccc(F)cc1 C1(NC(=O)Nc2cccc(Cl)c2O)CN(C(N2CC=CC2)=O)CCC1CO c1(C(N(C2CCN(C(=O)CCC(C)(C)C)C2)C)=O)cnn2c(=N)[nH]cnc12 Cc1cc(NC(=O)C(=O)N2CC(c3cc(C)n(C)n3)C2)cc(Cl)n1 O=C(CN=c1ccc(F)c(Br)[nH]1)NCCn1c(=O)oc2ccccc12 C12(NC(c3cnn4cccc(Br)c34)=O)CCCC1(F)CN(C(=O)CO)C2 C1(CCn2cc(C3C(C)C3)nn2)CN(C(=O)C(F)C2CCOC2)CCO1 N1(C(c2cc(C)c(O)nc2)=O)CC2CC(CNC(C3CC(=C4CC4)C3)=O)CC1C2 c1(NC(C(N2C(CC(C)C)CC2)=O)=O)cnn(CC(F)(F)F)c1C c1(CCC(=O)NC(CC)CNC(C2CC3CC3C2)=O)ccc2c(c1)CCO2 c1(OC)ccc(C(=O)NCc2cccc(CNC(=O)C=CSC)c2)c(N)c1 CC1(C(N2CCC(NC(C3CCCO3)=O)C(O)C2)=O)CCC(=O)CC1 c1(CNC(C2OCCN(C(C(C)=CC(C)(C)C)=O)C2)=O)nc(C)cc(C)n1 n1(CC(=O)NCC2(NC(CCCCOCC)=O)CC2)cnc2ccc(C)cc12.OCC c1(C(=O)NCC2(C)CCN(C(C(C)C#N)=O)C2)cc(O)nc2ccccc12 C(=O)(C1=CC2CC=CCC12)N(CCNC(c1cnc(CC)[nH]1)=O)CCOC N1(C(C(C)Sc2ccccn2)=O)CCC2(CC1)CC2NC(=O)C(C)(CO)CO c1(OC)ccc2c(C)c(C(N3CCC(C(C)NC(=O)C=C(C)C)C3)=O)[nH]c2c1 c1(CCC(=O)NC2CN(C(C3(CC)CCCCC3)=O)C2)cc(Br)ccc1F CC1=CCC(C)(C(=O)NCC2CN(C)CCN2c2ccnc(C3CC3)n2)CC1 c1(C(=O)NC2C(C)CCN(C(c3c(C)nc(=N)[nH]c3)=O)C2)cn2ccncc2n1 C1(C(=O)NCC2(NC(CCCC)=O)CCCCCC2)CC2(CCCC2)CO1 CCC1=C(C(=O)NCCN2CCN(C(=O)CCc3nccn3C)CC2)SCCO1 C1(NC(c2ncccc2F)=O)CC2CC(NC(C3CN(C4CCC4)C3)=O)C2C1 c1(C2C(CC(N3CC(NC(C(c4ccccc4)OCC)=O)C3)=O)C2)ccccc1 C1(NC(CS(CC)(=O)=O)=O)CCCC2CN(C(=O)CC3(C#N)CC3)CC12 c1(C(=O)NCCC2N(C(CC(C)C3CC3)=O)CCOC2)ccc2c(c1)CCCO2 c1(C(=O)NC2C(NC(CN(CCOC)C)=O)C2)csc([N+](=O)[O-])c1 C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CN(C(=O)CC2CCC2)CC12CCOCC2 C#CC1(C(=O)N(CC(C)NC(=O)C(C)Oc2ccc(Cl)cc2)C)CCOCC1 C1(C(=O)NCC2CCC(=O)NC2)CC2(CCN(S(=O)(=O)c3ccc(Br)s3)CC2)C1 CCC(CC)C(F)C(=O)N(C1CC(C(=O)NCCCCCCCO)C1)C N1(C(c2cc(CC(C)C)on2)=O)CCC2(NC(c3c[nH]cc3Br)=O)CC2C1 O=[N+]([O-])c1cc(Cl)c(Cl)cc1CN(CCc1cccc(Cl)c1)Cc1ccccc1 Cn1cc(CNCC(c2ncon2)C)cc1C#N N1(CNC(=O)CC2CC2CC2(C(=O)NCC)CC2)CC2C(C(=O)OC)C2C1 N1(C(C(C)NC(=O)NC)=O)CCC2CCC(C1)N2c1nc2ccc(N)cc2s1 C1(CCCNC(C=CCOC)=O)CCCCN1C(C1CC2(CSC2)C1)=O C(=O)(C(CSc1ccccc1)C(C)C)NCCCOCCN(C(C(C)SC)=O)C c1(NC(C)C(N2CCC(C(O)CO)CC2)=O)cccnc1O N1(C(C2C=C(C)CS2)=O)CCC(C2(NC(=O)CC3(C)CCOC3)CC2)CC1 Cc1cc(NC(C2CCCCO2)=O)ccc1NC(c1nn[nH]c1Cl)=O N1(C(CSC)=O)CCC(C(=O)Nc2cc(COC)nc(C(C)C)n2)(N(C)C)CC1 c1(C(C(N2CC(CC(C)NC(=O)CC3CCCOCC3)C2)=O)O)cccc(Cl)c1 C1(C2CCN(C(C3CN4CCCN3CC4)=O)C2)(NC(CC(C)CN(C)C)=O)CC1 C(=O)(C(C)(C)CNC(C1CC1C#N)=O)NCC1(N(C)C)CCC1 N1(C(C(C(C)C)C#N)=O)C(C(=O)NCC2(C)CSC2)C2CC(O)C1C2 Cc1cnc(C(=O)NCC2CCN2C(=O)CCOc2cc(F)cc(F)c2)c(F)c1 C1(C)(CCC(=O)N(C)Cc2nncn2C)CN(C(=O)CCC2CCC(=O)C2)C1 c1(CCC)n[nH]c(=NC2CCCC3CN(C(=O)C(=O)CC(C)C)CC23)s1 C1(NC(c2c(OC)ccs2)=O)CN(C(=O)C(C)=C(C)C)CC1N=[N+]=[N-] C1(CNC(=O)CCCc2ccsc2)CC2(CCC2)CN1C(=O)C1=CCOC1 C(c1cccnc1)=C(C(=O)NC(C(C(C)NC(CCCOCCOC)=O)C)=O)C#N C(=O)(CC1=CCN(C)CC1)N(CC(CNC(C(CC)CC1CCCC1)=O)O)C c1(NC(c2csnn2)=O)cccc2c(C3(C(=O)O)CC3)cccc12 c1(OC)ccc2occ(C(=O)NC3CCC4CC3CN4C(=O)CCC(N)=O)c2c1 N1(C(CSCC#C)=O)CC(NC(=O)C(C(C)C)N2CCCC2=O)C(CC)C1 c1(C(=O)NC(CNC(C(CC)O)=O)C)ccc(O)cc1-c1ccc(F)cc1 N1(C(C)=O)CCc2c(N(C)C)cccc21.C12CCOC1C(=O)N2.C12CN(C1)C2=O CCCC(C)(CC)C(=O)NCC1(NC(C2CC(C)CCO2)=O)CCOC1 N1(C(C(C)NC(N)=O)=O)CC2CCC(CNC(=O)C(C)(F)C(C)(C)F)C2C1 c1(C(=O)NC(c2ccccc2)C(=O)N(C)C)nc(=O)n(C)[nH]1 c1(C(=O)OC)c[nH]c2cc(NC(c3csc4c3CCCC4)=O)ccc12 c1(C(N2CCC(CCNC(C(CC)NC(N)=O)=O)C2)=O)ccc(SC)cc1OC N1(C(CCc2c(N)cccc2)=O)CCN(C(=O)Cc2cnns2)CC1C1CC1 C(=O)(CCCC(F)(F)CO)N1C(CNC(CN(C2CCSC2)C)=O)CCCCC1 N#CC1(C(N2CCOCC(NC(=O)Cc3cn[nH]c3)C2)=O)CCCOC1 CCCCCC(O)CC(=O)N1CC2(CCN2C(=O)CSc2cn[nH]c2)C1 Cc1cccc2c1N(C(=O)NC1CCCN(Cc3ccccc3)C1=O)CCC2C C(=O)(C1=CCC(C)CC1)NCCc1c(C(=O)NC(C2CCOCC2)C#C)c[nH]n1 C12(NC(C(C)NC(C)=O)=O)CCCC1N(C(c1c(Cl)ccc(F)c1F)=O)CC2 N1(C(=O)CC2(O)CCCCC2)CCC(C(F)(F)F)C(NC(=O)C(Cl)=CCl)C1 c1(C(C(=O)NCC2(F)CC(NC(CCC#C)=O)C2)C)ccc(F)c(Cl)c1 c1(OC)cc(C(=O)NCCN(C)C(C2CC3(C2)CC2(CC2)C3)=O)c(N)cc1F c1(C(N(C2CCN(C(C(C(C=C)C)C)=O)CC2)CCC)=O)cnc2ccsc2c1 c1(C(N(CCC)CCNC(C2SCCC2C)=O)=O)sc2ccccc2c1CSC C1(CCC)CCCC1OC(C1CC1(C)C(C)C)=O N1(C(c2cn(C)c(=O)cc2)=O)CC2(CCCC2)C1C(N1CC(O)CC1CO)=O CCC(N=c1[nH]c2c(c(=NCCCn3ccnc3)[nH]1)COCC2)c1ccccc1 Cc1cc(CC(=O)N(C(c2ccccc2)CNC(c2cocc2C)=O)C)on1 C(=O)(C(CCCC(C)C)N1CCC(C)(CS(C)(=O)=O)CC1)NCC C1(C(N2CC3C(CNC(=O)C(F)OC(F)(F)F)C3C2)=O)C2Cc3ccccc3C12 CC1CC(=O)NC(C(=O)NC(c2ccccc2)CNC(=O)CCCN(C)C)C1 C(CC)(C(=O)N(C)CC1CCCN1C(=O)C(C)OCc1ccccc1)=CCCC CCCCC(O)C(=O)N1CC(O)CC1C(N1CCCC1c1ccc(OC)cc1)=O C(CC(=O)NOCCO)C1CCN(C(C2N(CC)CC2)=O)C1 C1(OC)CN(C(=O)CN2CCCNS2(=O)=O)C(C)(CNC(=O)COC(F)F)C1 C1(NC(CCC=CC(C)C)=O)COC2(CCN(C(C3(C#N)CC3(C)C)=O)CC2)C1 C(=O)(C1=CCN(C(=O)CCc2nc(O)n[nH]2)CC1)NC(c1ccncn1)C c1(C(N2CCCC(C(=O)NCC3C(C)CCC3)CC2)=O)ccc2cc[nH]c2n1 C=C=C(C)CC(=O)NCC1CCCC(CNC(=O)Cc2cc(C)oc2C)C1 C=CCC(C)(CC)C(=O)NCC1CCC(C(=O)NCC2(C(N)=O)CC2)O1 N1(C(CCC)=O)CCC2(CC1)CN(C(C1(CO)CC(C)(C)C1)=O)C2 N(C(=NCCCCSC)NCc1ccnc(N2CCN(C)CC2)c1)C(C=C)C c1(C(=O)NC2CC(NC(C(COC)C)=O)C(O)C2)cnc(N(C)C)c(F)c1Cl C1(O)(c2cn(Cc3ccc(OC)cc3)nn2)CCN(C(N2CCCC2=O)=O)CC1 CC(CN=c1[nH]c2ccccc2cc1C#N)N(C(=O)CC1CCCC1C)C N1(C(CNC(=O)OCC=C)=O)CCC(CCOC)(NC(C2CC(O)C2)=O)C1 N1(C(C(n2cc(C)nc2)(C)C)=O)CCCC2CN(c3ncncc3Cl)CCC12 C1(C(=O)NCCCC(C)(C)C)CN(C(=O)C=CC(=O)NC2CC2)CC1(F)F Cc1ncnc(C)c1C(=O)NCCN(C(=O)C(O)CCn1cncn1)C c1(OC2(C(=O)NC(CC)CN(C)C(c3occc3C)=O)CC2)ccc(F)cc1 C12(CS(=O)(=O)N3CC(c4ccon4)C3)CCCCC1OCC2 c1(C(=O)NCC(C)N(C)C(C2CCC2C)=O)nc[nH]n1 CC1=C(C(=O)NC(C2(CNC(=O)CC3CC(C)(C)CO3)CC2)C)C(C)(C)CCC1 c1(-c2cc(C(=O)NCCCN(C(=O)CCS(C)=O)CC)n[nH]2)ccc(Cl)cc1 C1(CC(=O)N(C2CCC2)CCNC(COCCCC)=O)CC(CC)=NO1 c1(-c2c(C(C)O)cccn2)ccc2c(c1)CCCC2 c1(C(=O)NC23CC(NC(C(C(C)O)C)=O)(C2)C3)ccnc2ncccc12 CC(C)C(C)CC(=O)N1CCCC(N(C)C(c2ccnc(C#N)c2)=O)CC1 N1(C(CCC2C(C)C2)=O)CCC2(CCN(C(=O)Cc3cccnc3)C2)C1 C1(C(=O)NC2C(CNC(CCCN(C)C)=O)CC2)CCC(F)(F)CC1 Cc1cc(Cl)nc(N)c1C(N1CCC(CNC(=O)Cc2cccc(CO)c2)C1)=O c1(C(N2C(C)CCC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)nnn2c1C(=O)NCC2 N1(C(CC=CCC)=O)C(CNC(=O)CN2C(=O)CNC2=O)CC2COCC12 C1(NC(=O)CC2CC3CCC2C3)CCN(C(C2CSC2)=O)CC1F CCCS(=O)(=O)NC(C)C(=O)NCC(C1CCCCC1)NC(=O)COC(C)CC CCCCCCC(F)C(=O)N1CCC(O)(CNC(C2CCCOC2C)=O)CC1 C1(CNC(c2cc(OC)no2)=O)(OC)CCN(C(C2CCNC2=O)=O)C1 c1(CCC(N2CC(CNC(C3(C)CC4CC4C3)=O)C2)=O)cc2ccccc2o1 CCC(CC(F)F)C(=O)N1CC(O)(C(C)NC(=O)CC2CC3(CCC3)CO2)C1 c1(C(CO)NCC(=O)NC2CCCC23CC3)ccccc1Cl C(=O)(C1c2c[nH]nc2CN1C(=O)CCCNC(N)=O)NC(C)CS(C)(=O)=O c1(C(N2CCC(NC(c3cncc(OC)c3)=O)CC2C)=O)cc(O)cc(N)c1Cl C1(NC(C2CC(OC)(OC)C2)=O)CC2CC1CN(C(=O)C=C1CCC(C)CC1)C2 C1(C(N2CCC(C(=O)Nc3ccn(C)n3)CC2)=O)(CC)CCNC1=O c1(NCC(C(CC)C)O)ccc(S(=O)(=O)NCc2nnn(C)c2C)cc1Br N1(C(C(=C(C)C2CC2)F)=O)CCCC(CO)(NC(=O)CC2CCCCN2C)C1 C1(NC(CSCC#C)=O)CN(C(=O)CCc2ncc(F)cn2)CCC1C C(=O)(CCC(C)(C)C(=O)N1CCN(C(c2cccnc2C(F)(F)F)=O)CC1)OC C1(CC#C)(C(N2CCCC(N(C)C)C2)=O)CCN(C(=O)CC(C)F)C1 Cc1cc(F)cc2[nH]c(C(N3C(C)CC(CC(F)(F)F)C3C)=O)cc12 c1(NCC2CCN(C(C(C)(C)O)=O)C2)cc2c(cn1)C(=O)CCC2 C12(CNC(c3c(CC)cc(F)cc3)=O)CCC(NC(=O)CSC)(CC1)CO2 c1(OCC)ccc(C)nc1C(=O)NCCC(C)N(C(=O)C=Cc1cnc[nH]1)C C1(=O)C(NN(C)C)C1=O.C(C)(CNC(=O)C=CCSC)SC N(C1CCOc2ccccc21)C(c1nccc(-c2cccnc2)n1)C C(C(C)(C)CC(=O)N1CCCC(CNC(=O)Cn2cc(Cl)cn2)C1)N(C)C CC1CN(C(c2cnc(Cl)cn2)=O)CCN1C(c1cccnc1Cl)=O C(C(C)(C)CNC(=O)CCNC(c1ccccc1)=O)N(C(=O)CC1C=CCC1)CC C1(NC(CC(=C)C)=O)CCSC12CN(C(=O)C(F)=CC1CC1)C2 CC(C)CCC(O)C(=O)NC(C(=O)NC1CC1(C)C)C1CC1 c1(CC)cc(Cl)ccc1C(=O)NCC(C)(C)NC(C1OCCC1CC)=O C=CC(C)CC(=O)NCC=CC(=O)N(CCO)CCOC CCCCC(C)(F)C(=O)NCCC1CC(NC(c2ccc(C(N)=O)s2)=O)C1 Cc1ncc(C(N2CC(F)(CNC(=O)CC(F)(F)Cl)C2)=O)n1C C1(C(=O)NCc2ccc(CNC(CCCC(N)=O)=O)cc2)CCn2cnnc2C1 C1(NC(CCCC(=O)NC)=O)CC2CCC(C1)N2C(c1cn2c(n1)CCC2)=O Cc1ccc(C(=O)NCC(C2CC2)NC(c2cnc(C3CC3)nc2C)=O)cc1N Nc1cc(C(=O)NCC(CO)NC(=O)C(O)C2CCCC2)ccc1Cl C1(C2(O)CN(C(c3ccoc3Cl)=O)C2)(CNC(C23CCC(CO)(CC2)C3)=O)CC1 CC1CC2CN(C(c3cnccn3)=O)CC2N1C(c1cccc(Cl)c1)=O c1(C(=O)NC(C2CC=CCC2)C(=O)N(CC(COCC)O)C)cn(C)nc1C C1(CC=C)(NC(=O)CC2CCNC2=O)CCN(C(=O)C(=O)C(C)(C)C)CC1 N1(C(CS(C)(=O)=O)=O)CCC2(CC1)CC(N1CCC3(CCOC3)C1)C2 c1(SCC(C(=O)OC)NC(=O)CC2(c3nn[nH]n3)CC2(C)C)cc(F)cc(Br)c1 c1(C(=O)NCC2N(C(CCCC=C)=O)CC(O)C2)cc2c(C(F)F)nn(C)c2s1 c1(CC(=O)NC(CC(C(C)C)N)C)cccc2cccnc12 N1(C(C(CCC)O)=O)CCC2(CCN(C(c3c[nH]c(-c4cccs4)n3)=O)C2)C1 C1(NC(=O)CC2CCCC(=O)N2)C2CCC1CN(C(c1cn3ccccc3n1)=O)C2 C1(NC(C2CC(C)OC2)=O)CC2CCC(C1)N2Cc1cn(C)nn1 C(=O)(C1=C(Cl)CCCC1)NCCCN(C(c1nnc(O)cc1C)=O)CC c1(C(c2n(CCCOC)nnn2)NCC2CC(C)(C)C2)cccc(F)c1Br c1(COC)cc(C(=O)NC(CNC(C2CC2F)=O)C2CCC2)n(C)n1 c1(C(=O)NCCC(C)NC(C2CC2CF)=O)cc(Br)n2ccccc12 Cc1ccccc1C(N1CC(NC(c2cnc[nH]2)=O)C(F)C1)=O C=CCC(C)(C(=O)NCC1CC2(CC2)CN1C(=O)CCN1CCOCC1)N(C)C C1(C(=O)NC2CCC(NC(c3c(CC)nn[nH]3)=O)C2)CC(C2CCC2)C1 N1(C(COC)=O)CCn2nc(CNC(c3cc(C(=O)OC)cn3C)=O)cc2C1 Cc1cc(O)c(Cl)cc1C(=O)NCCN(C(C1CC2(C1)CC2F)=O)C(C)C C1(C)(C(N(C(C)CCNC(C2CCCCN2C)=O)C)=O)CCCC(F)(F)C1 c1(C(=O)NCCCC(C)NC(CC(C)c2ccncc2)=O)ccnc(F)c1F N1(C(C2(COC)CC(=O)C2)=O)CCCC(CC(=O)NCc2cnn(C)c2)C1 Cc1cccc(Cl)c1C(=O)NCC1CCCN1CC(n1cccn1)C c1(C(=O)NC(CC)CNC(C2C=CCC2)=O)cccc(C(=O)C2CC2)c1 N1(C(c2c(CC)noc2)=O)CC(O)CC1CNC(C1CC2(CCC2)C1)=O c1(CNC(CNC(CC)Cc2ccccc2)=O)cc(F)c(Br)cc1O C1(C(N2CCCC(CCC#C)C2)=O)CCC(O)CN1C(c1ccn(CCC)n1)=O O=C1CCC2(CN1)CN(C(=O)CC1CC(O)CN1C(=O)CCn1ccnc1)C2 C123CCC(CC1)(CO2)NC3=O.N1(C(C)C)CCOC(C(N2CC(N(C)C)C2)=O)C1 c1(OC)cc(C#N)ccc1CN1CCOC(C(=O)Nc2cc(Cl)cc(C)c2Cl)C1 C1(C(N(CC(C)N(C)C(c2ccc(Cl)c(F)c2F)=O)C)=O)CC1C1CCCCC1 C12(C(N3CC(N(C(=O)CCc4cnccn4)C)C(O)C3)=O)CCCN1CCC2 C(CC)(C(=O)NC(C1(O)CN(C(=O)Cn2cc[n+](C)c2)C1)C)OCC c1(OC)cc(C(F)(F)F)ccc1C(=O)NC(C)(CNC(=O)CC(C)O)CO c1(C(=O)NC)ccc(C=CC(N2CC3CC2CN3C(=O)C2=C(Cl)CCC2)=O)cc1 C1(CNC(C(C)N(C(C)=O)C)=O)CC2(CO1)CN(C(C1(F)CCCCC1)=O)C2 C(C(CC1CC1)C(=O)NCCCC1CCOC1=O)NC(C1C(CC(C)C)C1)=O c1(C(=O)OC(c2ccc(OC)c(Cl)c2)CC(=O)OC)ccc(C(=O)OC)c(C)c1 C(N=c1nc2c(ncn2C)c(NC2(C(=O)Nc3ncccn3)CC2)[nH]1)CC(C)C N1(C(CC(CC)C2CCC2)=O)CCCC(CNC(=O)C(c2cncnc2)C)CC1 n1(COCC)nc(C)c(CC(=O)NCC(C(C)(C)C)NC(=O)CCOC(=N)O)c1C C(CNC(c1cc(C)ccc1C)=O)(C(C)C(C)C)NC(C1(SC)CC1)=O Cc1ccc2c(n1)CN(C(c1ccnc(Cl)c1)C(=O)Nc1ccc(F)cc1)C2 C1(NC(c2nc(OC)oc2)=O)CCC(C)N(C(c2cc(C3CCC3)nn2C)=O)C1 Cn1nc(C(N2CC3CC(NC(c4cccc(Cl)n4)=O)C3C2)=O)c2c1CCOC2 CCC(C)(C)C(O)C(=O)NC1CN(C(=O)Cc2c(C)noc2C)CC1OC C(=O)(C1=CCCCC1)Nc1cccc(NC(C2C(C)(C)COC2)=O)c1 Cc1cc(CNCC(CO)NC(c2ccc(C(N)=O)nc2)=O)ccc1[N+](=O)[O-] C12CC3CC1CN3C(=O)CN2C(=O)CCCSC.C(C)(C)(C)OC(=O)NCC(=O)O N1(c2nc(C)[nH]n2)CCCC(NC(=O)NC(c2ccncc2O)C)C1=O C=CCC(C(=O)NCC(CC=C)NC(c1cc(CC)ccc1Cl)=O)C(C)C C1(C(N(c2ncc(C)cn2)CC2CCNCC2)=O)CCc2nc[nH]c2C1 N1(C(C(C(C)C)C)=O)CCC2(CCCCN(C(c3ccnc(CO)c3)=O)C2)C1 N1(C(c2cnc(C)o2)=O)CCN(C(C2(C)C=CCC2)=O)CC1C(F)F c1(C(N2CCC(O)(CNC(C3(C)CC3(F)Cl)=O)CC2)=O)ccnc2[nH]cnc12 N1(C(=O)CCc2cccs2)CCCC2(CCCN(C(c3ccc(Br)s3)=O)C2)C1 CN1C(=O)CSC1=CC(=O)NC1CCN(C(c2cnc(S(C)(=O)=O)s2)=O)CC1O C12(Nc3cc(C(C)=O)ncn3)CCCC1N(C(C1CN(CP(C)(C)=O)C1)=O)CC2 c1(C(=O)OC)c(C)[nH]c(C(=O)NCC2(NC(c3n[nH]c(C)c3C)=O)CCC2)c1C C(=O)(C(C)CCCC(C)C)NCC1CCN(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)C1 c1(C(N2C(CNC(C(C(CC)C)O)=O)CCCCC2)=O)cc2ccncc2s1 N1(C(C(C)(CSC)NC(COC(CC)C)=O)=O)CCC(C)=C(F)C1 C(CC(F)(F)Cn1cc(-c2cnccc2Cl)nn1)NC(=O)COC(F)(F)F N1(C(c2cc(-c3c(CNC)cc(F)cc3)[nH]n2)=O)CC2CCN(C)CC2C1 N1(C(C=CC)=O)CCC(NC(c2cnn(CCC(F)(F)F)c2)=O)CC1C1CC(OC)CC1 O=C(C(F)CC1CCOC1)NCC1(F)CN(C(C23CCC(C2)C3)=O)C1 c1(C(=O)OC(c2ccccc2)C(=O)N(CCC)C(C)C)ccn2ncccc12 CCCCC(CNC(=O)CC(F)(F)F)NC(C1(CC2CC2)CCC1)=O c1(CC)n[nH]c(=NCC(C)(CC)C(N)=O)s1 C1(CCOC)CCN(C(=O)C(C2CC2)NC(=O)CCCC2CC2)C1 C1(C(=O)NCc2ccccc2CNC(=O)C(C)SC)(COC)CCCCC1 c1(C(N2C(C(N(CCC=C)CC)=O)CSCC2)=O)ccc(Cl)c(F)c1F c1(C(N)=O)csc(NC(=O)CN2CCOC2=O)n1 c1(C(=O)NC2CN(C(C(CC(C)C)O)=O)CC3C2C3)ccc2c(n1)OCCO2 N1(C(c2cc(C)on2)=O)CCC2CC12.c1(C(=O)NC(C)(C)C)cccc(CCO)c1 CC(C)(Cl)CC(=O)N1CC(NC(c2cccnc2N)=O)C(c2ccccc2)C1 C1(CC)CN(C(=O)Cn2ccccc2=O)CC1NC(C1(C)CC(C)(C)C1)=O c1(OCC)ccc(C(=O)OC)cc1Cl.c1(C(N(C(=O)NCCO)C)C)ccccc1Br C(=O)(C(O)C1=CCCCC1)N(CCN(C(C(C)n1ccnn1)=O)C)C c1(C(C)C)ccc(C(=O)NC(Cn2cncn2)C(=O)N2CC(CF)C2)o1 C(=O)(C1=C(C)OCCS1)NC1CN(C(c2cc(COC)oc2C)=O)CC1C(F)F N1(C(COC(CC)CC)=O)CC=CC(NC(c2ccn(C(C)C)n2)=O)C1 C1(c2scc(C(=O)O)n2)(C2(NC(=O)C(Cc3ccsc3)CO)CC2)CCCCCC1 c1(C(C)C)ccc(F)cc1C(=O)NCC1C=CCN1C(=O)C=CBr N1(C(c2cc(OC)n[nH]2)=O)CCC(CNC(c2cc(O)cs2)=O)CC1 c1(CC(N2C(CC)C(NC(c3ccccc3Cl)=O)CC2)=O)cc2ccccc2o1 N1(C(c2c(C)onc2)=O)CCCCCC(NC(c2ccnnc2O)=O)C1 c1(C(N2CC(SC)C(NC(=O)C(C)(C)CO)C2)=O)cc([N+](=O)[O-])oc1C C#CCC(C)(C(=O)NC(C)C(C)(C)CC)NC(C1CC2(CCO1)CC2)=O c1(C(N2CC3C(CCNC(C(C)=C(CC)C)=O)(CC3)C2)=O)cnc2ccccn12 c1(C(=O)NC(C(CO)NC(c2c(C)n(CCO)nc2)=O)C)ncc(Cl)cc1F C1(C)(C(N2CCOCC(CNC(CCOC)=O)C2)=O)CCCCC1(F)F c1(CC(=O)NCCOCCN(C)CC2CC(C)OC2)cc(F)ccc1Br Cc1nc(C)c(C(=O)NC2(CNC(C3CC(=O)N(C(C)C4CC4)C3)=O)CC2)o1 C#CC(C)(C)C(=O)N1CC(O)(CNC(C2CCN(C(=O)CC)C2)=O)C1 C1(CC)CN(C(C2(Cl)CC2)=O)CCC1NC(c1c(C)coc1C(C)C)=O Fc1cc(Br)cc(F)c1C1(NCC=CC=Cc2ccccc2)CC1 CN1CCCC(C(=O)NCCC(C)(C)CNC(=O)CCF)C1=O c1(C(=O)NCCC(C)NC(c2cccc(OC)c2)=O)occ2c1CCC2 c1(C(N2CCC3C(NC(=O)CCC(F)(F)F)C3C2)=O)cc2ccccn2n1 c1(C(N(CC(C)NC(c2cc(CSCC)on2)=O)CC)=O)ccc(C)nn1 c1(C(=O)NC(COCC)C(=O)NCCc2noc(C)n2)cccc2c[nH]nc12 C1(NC(N(CCCC2CCCOC2)CC)=O)CCN(c2ccccc2F)C1=O O=C(C(CCCC1CC1)N1CCCC1c1ccccc1Br)NC1CC1 C(CCCC(CO)NC(=O)CN1CC2CC2C1)NC(C1C(C(C)C)C1)=O c1(-c2cccc(F)c2)cncc2cc(Cl)ccc12 CCC(O)C(C)(C)C(=O)N1CC(NC(=O)Cn2ncc(O)nc2=O)C1 C1(CC(=O)NCC2CC23CC3(F)F)C2CCCC2N1C(=O)CC1CCC(O)C1 c1(N2CC(C)C(NC(C3CC4CCCCN4C3)=O)C2)ncnc2ccc(Cl)cc12 C1(OC)CC2(CCC(CN(C(C(=O)NC3NC(=O)NC3=O)=O)C)CC2)C1 CC1(C)C2CC(NS(=O)(=O)CC34CCC(C3)C(=O)N4)CC12 c1(N(C)Cc2scc(C)n2)ccc(Cl)c(S(=O)(=O)N2Cc3cccnc3C2)c1 c1(CN2CCC(C(N3C(C(N)=O)CCC3)=O)C2)cc(Cl)c(Cl)cc1O N1(C(C(CCOC)NC(c2[nH]ccc(=O)c2C)=O)=O)C2CCC1CC1(CC1)C2 C1(C(F)(F)F)(SC)CCCN(C(=NCC2(CF)CC2(F)F)NC(C)C)C1 c1(C(=O)NCC=CCNC(C2(SC)CC(O)C2)=O)cc(Cl)c(Cl)cc1C CC1CN(C(=O)CC2CCC2)CC(CCNC(c2csc(C(F)(F)F)n2)=O)O1 O(C1CCc2ccc(Cl)nc21)C(=O)NC1CC(n2c(C(=O)OC)ccn2)C1 N1(C(c2cc(OC)ns2)=O)CC2(NC(c3ccc(CO)nc3)=O)CCCC2(F)C1 C1(COC)C=CCCN1C(C1CC(O)CN1C(C1CCC(C)(C)C1)=O)=O N1(C(c2n(CC=C)ccn2)=O)CCCCC(NC(C2(CS(N)(=O)=O)COC2)=O)C1 N1(C(C(C)NC(CC)=O)=O)CC(N(C)C(c2cc(C(C)(F)F)n[nH]2)=O)C2(CC2)C1 c1(C(N2CCC(C(=O)NC(CC)C(=O)N3CCOCC3)CC2)=O)ccc(C)cc1 c1(-n2c(C3CCCCN3)nc(COCC)n2)ccc(CC)c(C)c1 c1(C2C(=O)NC3CCC(C3)N2)c(F)cccc1F.C(C(=O)N(C)C)=CC=CCC c1(OCC(N2CC(CCNC(c3ccccc3)=O)C2)=O)cc(Cl)ccc1Cl S(=O)(=O)(c1ccc(Br)cc1NCC1(S(C)(=O)=O)CC1)NCC(=C)c1ccccc1 C1(OC)CN(C(c2cn(C)cn2)=O)CCC1NC(c1coc(SC)c1)=O CCC(C(=O)N1CCCC1C(=O)N(CCCF)CCN(C)C)NC(N)=O Cc1csc2c(C(=O)N(C(C)CNC(=O)Cc3n[nH]c(=N)s3)C)cccc12 C1(N(C(c2cccc(C)c2)CO)C(c2cc(C)oc2C)=O)CCNCCC1C C12(C(N(C)Cc3ccccc3O)=O)COCC1CN(C(C1CCC(F)(F)C1)=O)C2 C1(CC=C)(NC(=O)Cc2csc(C)n2)CCN(C(=O)CC2COCC2O)C1 C1(C(N(C2CCC(NC(CC(C)F)=O)CC2)C)=O)CC2C=CCC(C1)C2 C(=O)(C(C)CCC(C)(C)C)NCCC1=CCN(C(CCc2cnc(C)o2)=O)CC1 CCS(=O)CC(=O)N1CC(F)CC1CC(=O)NCCCF c1(C(N2CC(O)CC2CNC(C2CC(F)(CO)C2)=O)=O)c(F)cccc1F c1(OC)ccoc1C(=O)N(CCC(=O)NCCc1cnc(C)[nH]1)C1CC1 N1(C(CN(CCOC)C)=O)CCN(C(c2coc(C(F)F)n2)=O)CC(CO)C1 C1(C(=O)NC(CCCC)CO)CCC(C)(C)N(C(=O)C(O)C(C)C)C1 Cc1cccn2c(=O)c(C(=O)NNC(=O)NCC3CCNC3)cnc12 c1(OC)c(C(=O)NCCCCC(C)NC(=O)CC2CCC(C)C2)nc(O)nc1O C1(NC(c2cc(OC)no2)=O)CC(F)CN(C(C2(CO)CCCO2)=O)C1 C12(C(=O)NCCOC(=O)C3CC3)CCOC1CS(=O)(=O)C2.C1Cc2nccnc2C1 N1(C(C(C)NC=O)=O)CCC(CNC(C2CN(C(C)C)C2)=O)C1 S(=O)(=O)(c1ccc(Oc2ccccc2Br)cc1)NC(C1(C)C=CCN1)=O Cc1nn(CC#N)nc1CNC(=O)NC1CC(C(=O)OC(C)(C)C)C1 c1(C(=O)NCC23C(CN(C(C(CC)(F)F)=O)C2)C3)cn2c(n1)C(=O)N(C)CC2 O=C(C1=CCN(C(C2(CO)CCC2)=O)C1)NCC1CC(CO)CO1 C1(NC(C2CCC3CCC23)=O)CCN(C(=O)CSC2CCOCC2)C12CCC2 C1(NC(C2CC(=O)NCC2)=O)CCN(C(c2cc(C(F)F)ccc2F)=O)CC1O c1(C(N2C(CC)CC(C)C2)=O)ccc2c(n1)CN(C(=O)CN1CCCC1)CC2 C1(CNC(C(C)NC(C)=O)=O)CCN(C(=O)Cc2ccon2)C(C)C1 N(C(=NCC(C)C#N)NC(C)CCN1CCOCC1)CC(=O)NC(COCC)C N1(C(C(CCC)OC)=O)CCC2CN(C(c3cnn(CC4CCCC4)c3)=O)C2C1 Cc1c(C(=O)NC2CC2NC(=O)CCc2nccs2)cnc2c(Cl)cccc12 C=C1CCC1(C(=O)OC)C(=O)N(CCC)CCNC(=O)Cc1cccs1 N1(C(C2C(C)(C(C)C)C2)=O)CCC(C)(C(=O)N(C2CCC2)CCO)CC1 C(=O)(C(F)C(C)CNC(C1C2CCC(F)C12)=O)NC1CCCC(OC)C1 N1(C(C(=O)NCC)=O)CC(CNC(=O)C(CC)OCC)CC12CCOCC2 N1(C(c2cn(CCC)nc2)=O)CCCC(C2(NC(=O)CSC)CC2)C1 C1(C(N2CCC(CN(C(C(C)C(C)(F)F)=O)C)CC2)=O)Cc2ccccc2C1 C=CC1CN(C(C2C=CCS2)=O)CC1NC(=O)CC1C=CS(=O)(=O)C1 c1(C(=O)NCC2(C)CCCN2C(=O)C2=CS(=O)CCC2)nccc2c1NCCC2 C1(C(=O)OC)CC(n2cc(CSC)nn2)CN1C(c1ccc(Br)nc1)=O C(=O)(C(O)CC(F)F)NC(C(C)C)CCN(C)C(C1CCCCN1C)=O N1(CC(=O)NCCN(C(=O)C(c2ccc(F)c(F)c2)O)C)CCP(C)(=O)CC1 c1(C(=O)Nc2cnc(C(F)(F)F)cn2)ccc(I)c(I)c1 C1(CN(C(C2CC(=C)C2)=O)CC)CCN(C(c2cn(CCC(C)C)nn2)=O)C1 Cc1nc(CCC(=O)NC2CC(CNC(C3(CC(C)C)CC3)=O)C2)oc1C N1(C(CN2CC(C)(OC)C2)=O)CC(CNC(C2(F)CC=CCC2)=O)C(C)C1 c1(C(=O)NCC2(NC(CCCCC(N)=O)=O)CC2)ccc2nnn(O)c2c1 C1(OC)CN(C(=O)CCCn2cc(C)cn2)CC1NC(=O)C(N1CCSCC1)C c1(OC)nc(C(=O)NCCC(C)NC(=O)C=CC2CCCN2C)sc1C C(C(=O)N1CCC1CC(=O)NC(C)(C)CO)(C(C)C)NC(C)=O CC(C)C(=O)NC(C(=O)NC1(c2nn[nH]n2)CC1)C1CCCO1 C#CC12CCC(C(=O)N(CCNC(=O)C(CC=C)C(C)C)C(C)C)(CC1)CC2 c1(OC)ccc(OC)c(C(N2CCC(NC(=O)C(=O)NCCSC)C2)=O)c1 Cc1cc(C(N2CC(c3ccccc3)(NC(C3CC3c3sccc3C)=O)C2)=O)n[nH]1 CC1(C)CCCN(C(=O)C(F)C2CCCC2)C1CNC(=O)CCC1CC(F)(F)C1 c1(C(=O)NCC(CC)(C)NC(c2ccco2)=O)cc(OC)c(OC)cc1F CCC(C#N)(CC)C(=O)NC1CCN(C(=O)Cc2nc(C3CC3)nn2C)CC1C C1(OC2(C#C)COC2)CCCN(CCCOc2n[nH]c(C(=O)OC)c2Cl)C1 c1(N(C(=O)CN2CCOCC2CC2CCNC2)C2CC2)ncc2ccsc2n1 CCC(C)C(O)CC(=O)NC(Cc1ccco1)C(=O)NCc1nc(CO)n[nH]1 N1(C(c2c(CC)nc[nH]2)=O)CCCCC1C1CCN(C(C2(P(C)(C)=O)CC2)=O)C1 C(C(O)C(=O)NC1(CCCCNC(c2cnc(C3CCOCC3)s2)=O)CC1)SC N1(C(Cc2ccc(C(C)C)cc2)=O)CCCC(C)(C(N2CCCC(C)C2)=O)C1 c1(C(C)NC(=O)COc2cnn(C)c2)cnc(Cl)nc1C1CCC1 c1(N2CCC(C)(CC)C2)ncc(S(=O)(=O)NCC(C2CCCCC2)F)cc1Cl C1(C2C(C)C2)CCCN(C(CCc2ccsc2)C(=O)NC2CCCCC2)C1 CCCCC(C)NC(C1(NC(=O)CC2(O)CCCC2)CC(F)C1)=O C1(CCNC(c2cncn2C2CC2)=O)COCCN1C(c1cnc(C2CC2)s1)=O N1(C(C=C(C)C(F)F)=O)CCC(C)(C)C(CNC(=O)CC2CCOCC2)C1 c1(C(N2CC(CCCCNC(Cc3cc(C)nn3C)=O)C2)=O)ccc(C)c(Br)c1 C#CCCN=C(NCC1(COC)CCCC1)N1CCC(S(C)=O)(C(=O)OC)CC1 N1(C(CNC(c2cscn2)=O)=O)CC2CC1C2NC(C1CC1c1ccsc1)=O C(=O)(CCCC(C)(C)C)NC1C(C)(CNC(C2(COCC)CC2)=O)CCC1 N1(C(c2ccnc(C)n2)=O)CCC2CCC(C1)N2C(C12CC(C)(C1)OC2(C)C)=O c1(CNC(C(CC)C)CO)cc(F)c(C)cc1Br n1(CC(=O)NCC(C)CNC(C2COC(=O)C2)=O)ccc(=O)c([N+](=O)[O-])c1 c1(C(c2ccccc2OC(F)(F)F)O)ccncc1Cl.c12ccccc1N2 C1(CNC(C(c2ccccc2)C)=O)C(C)CCN1C(=O)CC(=O)OC(C)(C)C N1(C(N2CCCC2C2CC2)=O)CC2C(CC(=O)Nc3cncc(Br)c3)C2C1 N1(C(C2N(C(C(C)Cc3cnc[nH]3)=O)CSC2)=O)CC(N2CCCC2)C(O)C1 c1(OC)ccc(C(=O)NC(C)C(C)NC(=O)C(=O)N(C)C)cc1Cl c1(OCC)ccc(S(=O)(=O)NCCCC(=O)N(C)C)cc1C(=O)OC Cc1cc(C(=O)NCCC(O)CNC(=O)C(c2ccccc2)F)ccc1[N+](=O)[O-] CC(C(=O)NCc1cc(C(=O)N(CC(F)F)C(C2CC2)C2CC2)cs1)C(F)(F)F C1(CC(=O)N(C(C)CCNC(=O)Cc2ccco2)C)CCS(=O)(=O)CC1 c1(C(N2CCCC(NC(=O)C(F)(F)CC3CCCO3)C2)=O)coc2c1COC2 Cc1ccc(C(=O)NCC2COCC2NC(=O)C(C)(C)C(C)C)cc1C Clc1ccc(C2(c3ccncc3)CC2c2nc(C3CC4CC4C3)no2)cc1 c1(CC(C)C)cccc(C(N2CCCC(C(=O)NCC3CC3(C)C)C2)=O)c1 c1(C(=O)NCC2CC(CNC(=O)CC3CCCCC3O)C2)cc(F)cc(F)c1O CC(C)CC(CNC(=O)CCC(C)(C)C)C(=O)N1CC(C)(C)CCC1CO C(=O)(C#CC1CCCCC1)NC(C(=O)N(C)CC1(OC)CCC1)CCN(C)C C1(NC(C2(OC)CC2)=O)CCN(Cc2sc(Cc3ccccc3)nc2C)CC1 N1(C(c2n(CCC)ccc2)=O)CCC2(CCN(C(C3(C)CCCC3(F)F)=O)C2)C1 Cc1ccn2c(COC(c3cccc(OC(F)(F)F)c3)=O)cnc2c1 c1(C(=O)NCCNC(C2CCCN(C(C(CC)F)=O)C2)=O)cc(O)ccc1C C(=O)(C1=NN(C)C(=O)CC1)N1CC(CNC(CCOCCCOC)=O)C(O)C1 C=CC1(CC(N2CCOC(CCO)C2)=O)CN(C(=O)C(=Cc2ccco2)C)C1 C(=O)(CP(C)(C)=O)NCCCC(C)NC(=O)Cn1nnn(-c2cccs2)c1=O Cc1cc(CC(C)NC(=O)OC(C)(C)C)cc(C)c1.C1CCN1S(C)(=O)=O c1(OC)cc(C#N)ccc1CN1CCCC(C(N2CCCC(O)C2C)=O)CC1 c1(NC(=O)OC(C)(C)C)cnc(F)cc1NCC(=O)NC(c1ccc(Br)cc1)C CC1(CC(=O)NC(CO)CCC2CC2)CCN(C(=O)CCc2cnn[nH]2)C1 C12(CNC(c3cccc(CSC)c3)=O)CCC1CCN2C(c1c(C)cnn1C)=O N1(C(C(C#N)CC2CC2)=O)CCC(NC(c2cc3scnc3[nH]2)=O)C12CC2 CC(C)C(C#N)C(=O)NC1(CC(N2CCCC(CC(N)=O)C2)=O)CCCCC1 C(=O)(NNc1cccc(F)c1Cl)C1CN(C(=O)OC(C)(C)C)C(C)(C)CC1 c1(C(N2C(C(C)NC(CC=C)=O)CCC2)=O)nc(CC)n2ccccc12 CC1=NN(C)C(=O)C1CC(=O)N(C)CC1COCCN1C(=O)CSc1cn[nH]c1 N1(C(c2cc(C#C)c(C)cc2)=O)CCC(N=c2[nH]ccn3nnnc23)C(C)C1 CC1(O)CCC(C(=O)NCC(O)CNC(c2cc(N)cc(N)c2)=O)CC1 Cc1ccc(NC(C2(NC(=O)CN=[N+]=[N-])CC(F)(F)C2)=O)cc1C C(=O)(CC(F)(F)C1CCNCC1)N1CC(NC(c2c(C)cco2)=O)C1 c1(N(C)CC2CCN(C(C(CCC)N(C)C)=O)C2)nc(Cl)nc2cnn(C)c12 C1(C(=O)NCC2(C(N(C3CCCC3)C)=O)CC=CC2)CCOC1(C)C C1(C(=O)OC)C(CNC(=O)C(C)(C)NC(=O)CCOC(C)C)C1(F)F C1(C(=O)OC)CC(OC)CN(C(C2(OC)CC(C)C2)=O)C1.C(C)(C)S N1(C(Cc2c(C)con2)=O)CC(O)CCC1C(N1CC(CC(C)C)C1)=O C(=O)(C(F)C(=O)NCC(C)N(C(=O)C(c1c(C)noc1C)C)C)OCC C1(CC(=O)NC(CC)C(=O)Nc2nc[nH]n2)CCCCN1C(N1CCCC1)=O C=C=CCCC(=O)N(CC(C)(C)CNC(c1nocc1Br)=O)C N1(C(c2cc(OC)n[nH]2)=O)CCC(CF)(NC(c2ccn(CC(C)C)n2)=O)C1 C1(NC(C(C)CF)=O)C2CC3CN(C(=O)Cn4ncn(C)c4=O)C1C3C2 c1(CNC(CC2CNCC(C)O2)=O)nnc2n1CCNC2 CC1CN(C)CC(C(=O)NC23CC(CNC(=O)COCC4CCCOC4)(C2)C3)O1 C=CCCCCCCCC(=O)NC(C)CNC(=O)CC=Cc1ccc(C)cc1 C1(C(=O)OC)CC(NCC(F)(F)CCNC(=O)OC(C)(C)C)C1(C)C CC(C)CC(C(=O)NC1CC(F)CN(C(c2cccc(F)c2C2CC2)=O)C1)N(C)C c1(C(=O)NC(C(c2ccccc2)NC(c2c(C)csc2)=O)C)ccnc(CO)c1 O=S(=O)(c1cc(CO)co1)NC1CC(=O)N(COCC2CC2)C1 C(CN=c1nc(N2CCOC(C)C2)c2ccc(C(F)(F)F)cc2[nH]1)N(C(C)=O)C C1(NC(=O)C=C2CCOCC2)CC(F)CN(C(=O)CCc2nnc(C(F)F)o2)C1 N1(C(=O)NCC(=O)Nc2ncccn2)CCc2onc(C(N3CC(O)C3)=O)c2C1 C1(NC(C(C)c2cccs2)=O)CC2CC1N(C(C1(N3CCOCC3)CC1)=O)C2 c1(Cc2nc(C(N3CCC(C4CC4)C3)C(=O)NC(C)C)sc2)ccc(F)cc1F N1(C(CSC)=O)CCC2(CC1)CC(NC(=O)CCc1cc(C)sc1C)CO2 c1(C(=O)NC(Cc2ccc(CNC(C(CC)C)=O)cc2)C)cc2sccc2n1C CC1(CNC(C2CCC(NC(c3cn[nH]c3)=O)C2)=O)CCCCO1 CC(CN=c1[nH]c(C#N)c(Cl)s1)NC(C1(C2CCCO2)CC1)=O c1(OC)ccc(C)c(C(N2CCC(C)(C(N3CCC(n4ccnc4)C3)=O)C2)=O)c1 N1(C(C2(C=C)CCC2)=O)C2CCCC1CC(NC(=O)C(C)(C)C(C)C)C2 C1(n2cc(C3(NC(C(C)O)=O)CC3)nn2)C=CCC(NC(=O)C=CCO)C1 C12(CC=CCN(C(CN(CC(C)(C)C)C)=O)CCO)CC(CO)(C1)C2 CC(CC(=O)N(CCCOCCNC(c1cccnn1)=O)C)C(F)(F)F C=C(C)C(C)(O)C(=O)NCC(C)(C)Cn1cc(C(C2CCCC2)C)nn1 CCCC(CNC(=O)C(C)(C)CCSC)C(=O)NOCc1ccncc1 Cc1cn(C)nc1C(=O)NC(CNC(c1cnc(Cl)n1C)=O)C(C)(C)C N1(C(CC(C=C)c2ccccc2)=O)CCCN(Cc2nc(F)ccc2Cl)CC1CO c1(OC)ncc(C(N2CCC(C)C2CNC(=O)CNC(=O)C(F)(F)F)=O)nc1C N1(C(c2ccc(CCC)cc2)=O)CC(NC(=O)CO)CC(F)C1 C(N=c1[nH]c(=NCc2nc(Cl)ccc2Cl)[nH]c2c(F)cccc12)C1N(CC)CC1 CC1(CC(=O)NCC2(NC(c3ncoc3C3CC3)=O)CCCC2)CCCCC1 C(=O)(C(F)C(C)C(F)(F)F)N(C1CN(C(c2ccc(NC(C)=O)c(Cl)c2)=O)C1)C N1(C(c2ccc(C)n2C)=O)CCCN(C(c2cc3ccccc3o2)=O)C(CO)C1 N1(CC(N2CCC(NC(C(COCC)c3ccccc3)=O)C2)=O)CCCNC1=O CC(C)(C)CC(O)C(=O)N1CCN(CCNC(=O)CCC2NC(=O)NC2=O)CC1 C(N=c1[nH]cc(C(=O)NCc2ccccc2)s1)c1cc(OCC)n[nH]1 C(C(C)(C)C#CC(=O)NC(c1ccccn1)CO)NC(c1n(CCC)ncc1)=O Cc1cc(C(=O)NC(C2(O)CN(C(=O)Cc3ccc(O)c(C)c3)C2)C)cc(Cl)c1 N1(CC(=O)N(CCCCCCNC(c2ccco2)=O)C)CCCCCC1=O c1(C(=O)NCCC(CNC(=O)Cn2cnnc2O)OC)cnn(C)c(=O)c1 c1(C(=O)NCC(O)CNC(C2CCCC2O)=O)c(O)cc(F)cc1F C1(C(N(CCN2CCCC2)Cc2cn(C(C)C(=O)O)nn2)=O)CC2CCC1C2 c1(C(=O)NC(C)C(C)NC(=O)CCN(C)C)ccnc(CO)c1 N1(C(C2C(C)C2)=O)CCC(F)CC1NCC(=O)NC(C1(O)CCC1)C C1(CCNC(C2C(=C)C2)=O)CCCN(c2ccc(Cc3ccccc3)nn2)CC1 c1(NC(=O)CN2CCN(Cc3sc(Cl)nc3Cl)CC2)ccc(Br)c2ccncc12 C1(CC)CN(C(=O)CC23COC(C)(C2)C3)CCC1NC(c1cc(C)n(C)n1)=O c1(C(=O)NC2CCC(CNC(C3CCC(CC)O3)=O)C2)cc(Cl)ncc1F c1(C(N2CCN(C)CC2CNC(c2cc(C#N)c[nH]2)=O)=O)n[nH]c2ccccc12 C1(CNC(CCC(C)SC)=O)CCN(C(c2c(Cl)cncc2Cl)=O)CC1C C(=O)(C(CO)N(C)C)NCCC(C)NC(=O)CCCc1ccsc1 c1(C(C(F)(F)F)NC(C2CCCOC2)C)cc(OCC(F)(F)F)ccc1O N1(C(CN2C(C)CCC2C)=O)C2CCC1CN(C(=O)Cc1cccc(Cl)c1)C2 C1(CNC(c2nc(C)c(C)[nH]2)=O)C(C)CCCN1C(=O)CCNC(=O)C=CCl c1(C(N(CCOCCNC(CC(=O)NCC)=O)C)=O)c[nH]c2cccnc12 c1(CC)c[nH]c(C(N2CCCC2CN(C(=O)CSC(F)(F)F)C2CC2)=O)n1 C1(CC(=O)N(CCNC(=O)CCc2cnc(O)[nH]2)CC)CCS(=O)(=O)C1 c1(C(=O)NCC(CC(C)C)NC(c2c(C)cccc2)=O)nc(C)c(N)cc1C N1(C(C2C(C)CC2C)=O)CCC2(C1)CN(C(c1ccc3nc[nH]c3n1)=O)C2 CCCCCC(C(=O)NCCN1CCCC1=O)N1CCC(C)S(=O)CC1 C1(N(C(C(C)=C2CC2)=O)C)CN(Cc2ccn(C3CCCC3)n2)CC1F Cc1cc(CO)oc1C(=O)NCC1CCN(C(C2CCC(C)(CC)O2)=O)CC1 CONC(=O)C(=O)NCc1cccc(C(=O)N(C2CCCC2)C2CC2)n1 c1(C(=O)NCC(C2CC2)NC(C2(C)CCSCC2)=O)ccc(F)c(C#N)c1 c1(C(=O)NCC(CNC(c2nc(C)c(C)s2)=O)F)noc2c1CC(C)CC2 c1(C(=O)NCC2C(C)(C)C(NC(=O)Cc3cccs3)C2)c(F)ccc2c1OCC2 CCC(C)(O)C(=O)NCCNC(c1ccc(NS(N)(=O)=O)cc1)=O N1(C(CNS(C)(=O)=O)=O)CC2CN(C(C3CCCC(=O)N3)=O)CCC12 N1(C(CC(=C)Br)=O)CC2CCC(C1)N2C(=O)C(C#N)C1CC1 c1(C(N(CC(C)NC(CS(CC)=O)=O)C)=O)cnc(Cl)c(F)c1N C1(CCC(=O)NCc2cc(C)ns2)CCCN(C(C2(CCN(C)C)CC2)=O)C1 C1(C(=O)NCC(C)NC(C2(N(C)C)CC2)=O)CC1(C(C)C)CO c1(CC)nn(C)c(N2CCC(CNC(c3cc(C)sc3C)=O)C2)c1[N+](=O)[O-] c1(C(=O)NC(C(C)NC(CCC(=O)NC)=O)C)cnc2ccncc2c1 c1(CC)ccc(C(=O)NC2(CNC(C3CC(O)CN3C)=O)CCCC2)nc1 C(C)(C)(CCCNC(=O)C(n1cc(C2CCCN(C)C2)nn1)C)N(CC)CC C1(CC=C)(NC(=O)CCC(F)F)CCCN(C(=O)Cc2ccc(F)c(Cl)c2)C1 S(=O)(=O)(c1cnc(NC2CCC(CC(C)C)C2)cc1C)NCc1ccc(C)cn1 C1(C(C)C)(C(=O)NCC2CCN2C(=O)C(F)C2CCOC2)CCOC1 N1(C(C(=O)NCC)=O)C2CCC1CN(C(c1cc(=O)n(C)o1)=O)C2 CC1CN(C(c2cc(N)c(Cl)cn2)=O)CCN1C(c1cnc(C(F)F)s1)=O N1(C(C(CCC)OC)=O)CCC2C(C(=O)N(C)CCC3CCCC3)C2C1 N1(C(C(C(C)C)OCC(C)C)=O)CCN(C(C2CCC(N=[N+]=[N-])C2)=O)CCC1C CC(CCNC(=O)C(O)CNC(=O)C(N1CCOCC1)C)CCO c1(C(=O)NC2C(C)CN(C(=O)C(C)N3CCC3)CC2)ccc(F)c(C#N)c1 C1(C)(CNC(c2cc(C)on2)=O)CCC(NC(=O)Cc2nccn2C)C1 c1(C(=O)NC(C2CCN(C(C(CC)COC)=O)CC2)C)cc2n[nH]cc2cc1C C1(C(N(CC(C)CNC(=O)CC2CC2)C)=O)CSC(c2ccccc2)=N1 Cc1ccc2c(C(=O)NC3CCCN(C(C45CC(O)C4C5)=O)C3)csc2c1 C1(CC(=O)OC)CCC2(CC1)CCN(C(=O)NC1CCCCC1N1CCCC1)C2 N1(C(CCSCCCC)=O)CC2(CCC2NC(=O)CSc2nnc(C)s2)C1 c1(C(N2CC(NC(CC(C)c3cccnc3)=O)C2)=O)ccc[n+]([O-])c1 C1(NC)CN(C(=O)C(N2CCCCC2C(=O)NS(=O)(=O)C2CC2)=O)C(C)(C)C1 C1(NC(CCCC)=O)CN(C(C2CCN(C(=O)C3CC3)CC2)=O)CCC1C c1(C(N(C)CCn2cc(CC(C)(C)C)nn2)=O)ccc2[nH]nc(Br)c2n1 Cc1cccc(OCC(=O)NCCNC(c2cccc(Cn3ccnn3)c2)=O)c1 Cn1nc(C2CC2)cc1C(=O)NCC1CCN(C(=O)CN2C(=O)CNC2=O)CC1 C1(C(=O)NC2C(NC(c3c(C)cc(CC)o3)=O)CC2)SC2C=CC1CC2 C1(NC(c2n(CC#C)cnn2)=O)CC(O)CN(C(C2(C)CCCCC2)=O)C1 Cc1cc(Cl)ccc1C(=O)NC(C1(O)CN(C(=O)C(O)C(F)(F)F)C1)C CC(C)CCC(C)N(C)C(C1OCCC1CNC(C1(F)CCOC1)=O)=O N1(C(CC(CC)SC)=O)CCCC(CNC(C2CCCCN2CC)=O)CC1 c1(C(=O)NC(C2CCCN(C(CCCC(C)=O)=O)C2)C)cnc2[nH]c(O)nc2c1 N1(C(c2c(C(C)C)ocn2)=O)CCC(C2CC2NC(C2C(C)C2C)=O)CC1 N1(C(CCCC(CC)C)=O)CCOC2(C1)CN(C(C1CCC(=O)NC1)=O)C2 c1(C(N2CC3C(NC(C4CCC(=O)N4)=O)(C3)C2)=O)cc(F)cc2cnccc12 N1(C(C(CC)C#N)=O)CC2(CCC(CNC(c3nc(C4CC4)oc3C)=O)O2)C1 CC(C(=O)NC1CC(CNC(=O)C=CC(=O)N(C)C)CC1O)C(F)(F)F c1(CCC(=O)N2CCC2c2ccc(F)cc2)ccc(-c2cccnn2)cc1 C1(C(=O)NC(C2CC(NC(C=C(CCC)C)=O)C2)C)COCC1(C)C Cc1nn(CC(=O)NCCNC(C2(c3ccc(O)cc3)CC2)=O)cc1Br N1(C(C(n2ccc(C)n2)(C)C)=O)CCCC(O)(CNC(c2ncccc2F)=O)C1 C(=O)(C1=Cc2ccccc2OC1)NC1CCN(C(C(CCCC)CCCC)=O)C1 c1(C(N(CC(=O)OC2CC(CC)C2)CC2CC2)=O)ocnc1C1CC1 N1(C(Cc2cc(C)sc2)=O)CC2COCC2(C(N2CC(c3ccncc3)C2)=O)C1 c1(C(=O)NC2(CF)CCN(C(C(C)OCCCC)=O)C2)c[nH]c2cccc(F)c12 N1(C(C2C(NC(Cc3c(C)n[nH]c3)=O)C2(C)C)=O)CC2OCCN(C)C2C1 N1(Cc2cc(C)[nH]n2)CCC(NC(c2ccc(F)c(C)c2)=O)C(F)C1 C1(COCC)(NC(=O)Cn2cncc2C)CN(C(=O)CCc2nc(C)no2)C1 c1(C(=O)NCC=CC)cnc(CNC(c2snnc2C)=O)nc1 c1(C(=O)NCC(CCC)NC(=O)CN2CC3CC3C2)ccc(F)c(C)c1F c1(C(=O)Nc2cccc(NC(C(CSC)(C)C)=O)c2)cc(O)ccc1C C(=O)(CCC(=O)NN(C)C)N1C(C(NOCC(=C)Cl)=O)C(CC)CCC1 c1(C(N2C(C)(C)C(CNC(C3CCCC3O)=O)CC2)=O)cc(C#N)c(N)cc1O N1(C(C(CC=C)CC)=O)CC23CCCCC2(C1)CN(C(=O)C(C)C1CCCC1)C3 Cc1nnc(O)c(C(N2CCC(CO)(NC(=O)CC3CC3(C)C)CC2)=O)c1C c1(N2CCC(C(N3CCC(C(F)(F)F)CC3)=O)C2)ncc(Br)c(O)n1 C1(C(N2CC(C(=O)NCCc3cccnc3C)(CC)C2)=O)C2CCC(C2)C1C N1(C(C2(COC)CCCC2)=O)CCC(C)C(CNC(=O)Cc2ccc(Cl)cc2)C1 c1(NC(C2(CNC(CCSC)=O)CCC2)=O)cccc(Br)c1Br c1(CNC(CC(C)C2CC2)=O)cc(C(=O)NCc2ccsc2Cl)ccn1 S(=O)(=O)(c1ccc(NC)cc1Cl)NCc1c(CC)cc(Cl)cc1 c1(CC)nnnn1C(C1(NC(C2(CF)CC2)C)CC1)NCCO.C(C)(C)(C)OCC c1(C(=O)Nc2ccc(C(F)(F)F)nc2)cc2[nH]ccc2cc1C1=CCSCC1 CC1(C)CC(C(=O)NC2CC3(C2)CC(C#N)C3)CN(C(c2cc(C#N)cs2)=O)C1 C#CC(CNC(=O)CN(C(=O)C(C)COC)C1CCC1)C(C)C C1(F)(CNC(Cc2ccc(OCC=C)cc2)=O)CCN(C(=O)C(O)CF)CC1 C1(NC(c2c(OC)cc(Cl)cc2)=O)CN(C(c2n[nH]c(=N)[nH]2)=O)C2CCCCC12 c1(OC)cc(C(N2CC(CNC(C3CCC3C)=O)C2)=O)c(C)cc1O N1(CC(=O)NC2C3CN(C(COCC)=O)CC32)C(=O)c2ccc(Br)cc2C1=O N1(C(C2(C(N(C)C)=O)CCCSC2)=O)CCC2(CC1)SCCS2 c1(C(C(=O)NCC(C)NC(=O)Cc2ccco2)O)ccc(OC(F)(F)F)cc1 c1(OC(C)C)ccc(C(N2CC(CNC(=O)CCC(=O)N(C)C)C(O)C2)=O)nc1 c1(CNC2CCC(CN)C2)ccc(Br)cc1[N+](=O)[O-] C1(C(=O)NCC2=CCN(C(C3C(OCC)CC3)=O)CC2)CCn2nnnc2C1 C(C)(CCCCO)NC(CONC(C1CC(OC)(OC)C1)=O)=O c1(CC(=O)OC)ccccc1CC1CCN(C(=O)CCSc2nccn2C)C1 N1(C(c2c(C)n[nH]c2)=O)CCOCC(CNC(=O)CCc2cccc(Cl)c2)C1 C(=O)(CC(C)C(F)F)NCCNC(c1occ(C)c1C)=O N1(CC(=O)N(CC(C)NC(c2c(C)n[nH]c2)=O)C)C(=O)NC(C)(C2CC2)C1=O CC(C)(C)CC(=O)NCC1CCCCC1CNC(C1CCC=CO1)=O c1(C(CN)=O)ccc2occc2c1.N1(C(c2ccc(C)o2)=O)CC2CC(C(=O)O)C1C2 c1(C(=O)NCC2(OC)CCN(C(=O)C=CC(F)(F)F)C2)c[nH]cc(C)c1=O c12ccccc1C(=O)N2.c1(C2C(C(=O)OCC)CC2)nnc(C(C)OC(C)C)s1 c1(OCC(C)C)ccc(C(=O)NC(C)CN(C(=O)Cn2ccnc2)C2CC2)cc1 C1(C(=O)NC(C2CCCN(C(C3C(OC)CCCC3)=O)C2)C)CN2CCC1CC2 N1(C(C(C=C)CC)=O)CCCCC2(CCN(C(=O)C(CO)OC)C2)C1 C1(NC(Cc2cccc(OCC)c2)=O)CN(Cc2cn[nH]c2)CC1C#N Cc1csc(C(=O)OCc2ncc(-c3ccc(Br)cc3)o2)c1C N1(C(c2c(C)ncs2)=O)CCC(C(N2CC3C(C2)C3(C)C)=O)C(O)C1 Cc1cc(C(N2CCCC2(C)CNC(C2(C)CC=CCO2)=O)=O)ncc1N C1(C(=O)NCC(COCC)(C)C)CCCCCCN1C(=O)C1=CCCOC1 OC1CCN(CCC2CCC3(CC2)OCCO3)C12CCSC2 C1(C(=O)OC)CN(C(=O)NCc2cccc(OC3CC3)c2)C1(C)C C(=O)(C1=NOC(C)(C)C1)NCCC1CN(C(C(C)n2ccnn2)=O)C1 N1(c2n(Cc3ccc(C4C(C(=O)OC)CCO4)s3)nnn2)CC(=O)NC(=O)C1C c1(C(N(C(CC(C)C)C(=O)NCCc2cnccn2)C)=O)ccc2c[nH]nc2c1 C1(C(N(CC(C)O)CCNC(c2cncc(C)n2)=O)=O)CCCN2CCCCC12 C1(C(=O)NC2(C)CCCOC2)C2CCC(C2)C1NC(=O)CCCC1CCC1 c1(C2C(N(C(=O)NC(c3ncccn3)C)C(C)C3CC3)C2)ccccc1 Cn1cnc2c1CCCC2C(=O)N1CCC(C)(NC(c2cnc(C(F)F)s2)=O)C1 C(=O)(C1CCCc2nn(C)cc21)NCC1N(C)CCN(C(c2csnc2Cl)=O)C1 C#CC1(C(N2C(CO)CC2CO)=O)CN(C(=O)CC2COCC(C)O2)C1 C1(C)(CC)CC(NC(=O)C(F)C(C)CNC(C2(CO)CCOCC2)=O)CCO1 C(CN=C(NCC(c1cc(Cl)cc(Cl)c1)O)NC1CCC1)N1C(=O)CCCCC1 c1(C(=O)NC2CN(C(C3CCC(C)CC3)=O)C(C)C2)cc(N)c(F)c(F)c1F c1(C(C)(C)C)ccc(C(N2CCC(O)(NC(=O)COC(F)(F)F)C2)=O)cc1 C(=O)(CC(CC(C)C)NC(=O)C(O)CN(C)C)NC(C1CCCC1)CC C12(OC)CCCC(CC(NC(c3ccc(S(C)(=O)=O)o3)=O)C1)C2 c1(OC)nc(C)ncc1C(=O)NC1CC(CO)N(C(C2CCC(=O)N2C)=O)C1 Cn1cc2c(CN3CCCC(C(=O)Nc4c[nH]c5ncccc45)C3)cccc2n1 C(CC(=O)N1CC(F)(CO)C1)(C(F)(F)F)NC(CC(CC)(C)C)=O C(C(CC(C)C)C(=O)N1C(C(N2CCOCC(C(C)C)C2)=O)CCC12CC2)OC c1(C(N2CC(C)C(=O)CC2)=O)c[nH]c2ccc(-c3cccc(C#N)c3F)cc12 Cc1cnc(C(N2CCC2CNC(=O)C=CC2CCCCCC2)=O)c(F)c1 N1(C(C2(COC)COC2)=O)CCCC2(CCCNC2)C1 C12(C(=O)NC3CCC(N(C(c4cn(CC)nc4)=O)C)C3)CCC(CC1)OC2 N1(C(c2c(CC)nc[nH]2)=O)CCC(NC(C2CC(CCO)C2)=O)C(CO)C1 Cc1cc(=NCC(C)(C(C)C)NC(=O)COC2CCCCC2C)[nH]c(Cl)n1 c1(C(=O)NC(CNC(CCc2cnc(C)s2)=O)C2CC2)cc2cc[nH]c(=O)c2s1 CC1CCN(C(C2OCCC2CNC(=O)C(C)(C)C(N)=O)=O)CCS1 C=CCCC(C(=O)OC)NC(=O)CCC1(C)CN(C(=O)CCc2ccnnc2)C1 N1(C(C(CCC)C)=O)CC2CCN(C(c3cc(F)c(C(F)(F)F)cc3F)=O)C2C1 C(N=c1nc2sccc2c(N2CCC(O)C(F)C2)[nH]1)c1c(OC)cccc1.C1(C)CC1 c1(C(N2C(CNC(c3scc(C(C)=O)c3)=O)CCC2)=O)cn(C)nc1C(C)C C1(CC=C)(C(=O)NCCN2CC3CC3C2)CCN(C(=O)C(F)CC2CCOC2)C1 C(=O)(C#CCCCC#N)Nc1n(C)ccc1.c12ccc(cc1)C(=O)N1CCC(C1)C2 c1(OC)ccc(C2CC2)c(C(N2CC3CC3(NC(c3csc(O)n3)=O)C2)=O)c1 c1(N2CCCC(C(=O)Nc3cccc(F)c3I)C2)ncnc2c(F)cccc12 C(CC(=O)NC1CCOCC1(C)C)(C(C)OC)NC(COCCCC)=O CCCCC(O)C(=O)NC(CO)CCCCNC(C1(Br)CC1)=O c1(C(=O)NC23CN(C(C4(COC)CCCO4)=O)C(CC2)C3)cnc(O)n(C)c1=O C(C)(C)(CCC(=O)N(C)CC1CCCN1C(c1nc(Cl)sc1Cl)=O)OC C(=O)(CCC(F)(F)F)N1CCC(CNC(C(CC)Cc2ccccc2)=O)CC1 CCC(C)(F)C(=O)NCCC1CCCCN1C(=O)C1=COCC1 C1(NC(C2C(C)C2)=O)CN(C(=O)CCn2ccccc2=O)CCC1C(F)(F)F n1(CC(=O)NC2C(NC(c3cnc(C(C)C)s3)=O)CC2)cc2ccccc2n1 c1(-c2nc(C(C)NCCNC(C)=O)on2)cccc(F)c1 N1(CC(N2CCOC2=O)(C)C)CC(=O)N(CCCN2CCCC2)C1=O C1(NC(C2(CC)CCN(C(=O)CC3OCCC3(C)C)C2)=O)CCCCC1N=[N+]=[N-] c1(C(=O)NCC2(CNC(CCCOCC=C)=O)CC2)cc2n(n1)CCCC2 N1(C(C(F)OC)=O)CCC(C2(NC(c3ccc(CN(C)C)cc3)=O)CC2)C1 c1(OC)cc(C)c(C(=O)NCC2(OC)CN(C(=O)C(C)(C)C(N)=O)C2)cn1 N1(C(C2C(C(=O)OCC)C2)=O)CCN(C(=O)Cc2n[nH]c(=NC)s2)CC(C)(C)C1 Cc1ccc(C#N)cc1C(=O)N(C)CCN(C(=O)CN1C(=O)CC(C)(C)C1=O)C C(CCCCCC(=O)N1Cc2ccccc2CO1)NC(C(C)C#N)=O C1(NC(C=C2CCN(C)C2)=O)CCCCN(C(=O)CC2CCCCC2O)C1 N1(C(C2CCCOC2)C(=O)NC2CC(C(=O)OC)C2)CCCC(CO)CC1 C1(NC(C(CC(=O)O)C2CC2)=O)CCc2cncn2C1 N1(C(CS(=O)(=O)N(C)C)=O)CCC(CNC(=O)CN2CCSCC2)C(C)(C)C1 N1(CC(=O)NC(C)CCNC(=O)CCC2NC(=O)NC2=O)Cc2ccccc2C1 N#CCCCCC(=O)NCC12CC1CN(C(=O)C(F)=C1CCC1)C2 c1(C(N2CCCC(NC(CCSCCC)=O)C2)=O)cnc2[nH]cc(C)c2c1 N1(C(C2(CCOC)CCC2)=O)C(C(=O)NCCC2CCOC2)CC1C c1(C(=O)NCCC2CCCN(C(c3c[nH]nc3C(F)F)=O)C2)c[nH]nc1[N+](=O)[O-] c1(OC)ccnc(COCC(N2CCOCC2CNC(C2OCC2(C)C)=O)=O)c1 N1(C(C2C(COC)C2)=O)CC2C(NC(=O)CCCc3csc(C)n3)C2C1 N1(C(C(CC)(C)OC)=O)CCN(C(c2cnn3ccsc23)=O)CC2(CC2)C1 N1(c2snc(-c3cccc(C)c3)n2)CCC(C)(NC(c2sccc2F)=O)CC1 C(c1ncc(C)[nH]1)=CC(N1CC(O)(CCNC(c2c(CCC)nco2)=O)C1)=O C1(CC)(NC(c2cccc(NC)c2)=O)CCN(C(c2cc(Cl)cnc2Cl)=O)CC1 N1(C(C(c2ccc(Cl)cc2)(C)C(C)(C)C(=O)NS(C)(=O)=O)=O)CCC(O)C(F)(F)C1 C1(C(C)NC(c2cc(-c3ccco3)[nH]n2)=O)CN(C(c2c[nH]c(=N)o2)=O)CCO1 N1(C(CC(=O)NC)=O)CCC2(NC(c3[nH]nc(OC)c3Cl)=O)CCCC12 CC1CN(C(C2CC(C)(C)CO2)=O)CCN1C(c1cnc(C(C)(F)F)s1)=O c1(C(=O)NCC(C)(C2CC2)NC(C(CC)C2CCOCC2)=O)cncn(C)c1=O N1(C(C(COC)(C)C)=O)CC2CCC(C1)C2CNC(=O)C(C)CSC(F)(F)F C1(NC(CC(=O)NCC)=O)CCCC1(C)CNC(C1CCCN1C(C)C)=O c1(C(N2CC(NC(C3CC3C3CC3)=O)C(O)C2)=O)c(F)ccc2nc[nH]c12 c1(C(=O)NC2(CF)CCN(C(C=CC(C)(C)C)=O)C2)cncc2ccsc12 C1(NC(CC(CCC)N(CC)CC)=O)CCN(C(=O)C(C)C(F)(F)F)CC12CC2 c1(C(N2C(CNC(CCCOC)=O)CC2)=O)cc(Br)c(Cl)cn1 N1(C(C2(SC)CCC2)=O)CCC(F)(F)C(CNC(=O)CC2CCC(F)(F)CC2)C1 CC(C)CCCC(C)C(=O)N(CCC(=O)NC1CN2CCCC1C2)CCO C(=O)(C(C(C)C)OCC)NCC1(C(=O)NC(CSCC)CO)CC1 c1(OC)cc(C(N2CCN(C(C3CCC(C#N)CC3)=O)C(CO)C2)=O)ccc1C CC1(C)CN(C(=O)C2=CCCOC2)CCN(C(c2c[nH]c3cc(F)ccc23)=O)C1 c1(C(N(C2CN(C(C(CC)C(=O)OC)=O)CC2(C)C)C)=O)sc2nccn2c1C c1(C(=O)NC(CC)CNC(c2cncn2C2CC2)=O)oc2cc(Cl)ccc2c1C CC(C)CC(CC(C)C)C(=O)N1CC=CC(NC(c2ccsc2C(F)(F)F)=O)C1 CCCCC(C(=O)NC1CCN(C(c2coc(C(N)=O)c2)=O)C1C(C)C)N(C)C Cc1cc(CC(=O)N(C2CN(C(=O)CC3CCOC3=O)CC2(C)C)C)ccc1F c1(SC)ccccc1C(=O)NCC1(O)CCN(C(=O)C(C)C(C)C)C1 c1(NC(C)=O)ccc(CCNC(c2cnccc2C)c2nnnn2C)cc1 c1(C(=O)O)cccc(C(CO)Nc2cccc(C3CCCC3)n2)c1 C1(C(=O)OCC)CCC2C(=O)N(CCc3cccnc3)C(=O)N2C1 N1(C(C=CC(C)C)=O)CC2CCC(C1CO)N2C(c1ccn(CCO)c(=O)c1)=O C(N=c1cc[nH]c(-c2ccc3nonc3c2)c1)C1C(C)CCCC1 c1(C(=O)NC2(C)CC(NC(c3cc(CF)on3)=O)C2)ncc2ccccn12 C(CC(C(C)C)OC)NC(CN(C1CCN(C(COCCC)=O)C1)C)=O C(C(C)C(F)C(=O)NCCc1ccc(O)nc1)NC(Cc1c(C)cnn1C)=O C1(C(=O)NCCCOCCNC(C2CC(C)(F)C2)=O)CC2(C1)CC2(F)F c1(CC)cc(C(=O)NCC2(NC(=O)C(C)c3ncco3)CCC2)cc(F)c1 C1(CC(=O)NC2(CC)COC2)CCN(C(=O)CC(C)(C)CN(C)C)C1(C)C c1(C(N2CCC(NC(CN(C3CCSC3)C)=O)C(F)C2)=O)ccnc2[nH]nnc12 C(=O)(C(F)C(C)CNC(=O)CC1CC=CC1)Nc1cnc(OCC)nc1 c1(CNC(C(C)Cc2cnco2)=O)ccc(CNC(C2CCOC2)=O)cc1 N1(C(C=CSC)=O)CC2(CCCC2NC(c2cccc(C(C)(C)C)n2)=O)C1 C(=O)(C1=NN(CCO)C(=O)CC1)N1CC(NC(C(CCS(C)=O)O)=O)C1 N1(C(C=CCC2(NC(C(CCC)C)=O)CCC2)=O)CCc2ccccc2C1 C(c1ccccc1)(C(F)(F)F)=CC(=O)N(CCCNC(C1CC1(C)C)=O)C C#CC1CCN(C(C)=O)CC1.C1(C(C)(C)C)C(=O)NC(CCC)c2cn1nn2 C1(NC(CC2(C)CN(C(=O)OC(C)(C)C)C2)=O)C2CN(CC3CCOCC3)CC12 Cc1cc(Cl)cc(C)c1C(=O)NC1CC2CC(NC(=O)C(C)CC(F)(F)F)CC12 Cc1cc(CNC(=O)C(C)CN(C)C(C2CS(=O)(=O)C2)=O)nn1C c1(C(=O)NC(CN(C(C(C)NC(CC)=O)=O)C)C)cc(OC)cc2c1CCC2 Cc1ccc2cc(C(N3CCN(C(=O)CCC(N)=O)C(C)C3)=O)[nH]c2c1 N1(C(n2cc(-c3cn(C)nc3)nn2)=O)CCN2CCCCC2C1.C12C(C1(F)F)C2 c1(CN2CC(CNC(c3cc(S(N)(=O)=O)oc3)=O)C2)cc(=O)n2ccsc2n1 CC(C)CC(O)C(C)C(=O)NC(CSC1CC1)C(=O)NC(CCO)C1CCCC1 N1(Cc2onc(CCC)n2)CCC(NC(=O)CC2CCCCO2)C(O)C1 C1(CC)CC(C)CN(C(c2ccc(CNC(c3ccc(C)cc3C)=O)o2)=O)C1 C1(CNC(CCCC#C)=O)CCN(C(c2cc(Cl)c(C)c(Cl)c2)=O)CC1(F)F C1(NC(CN(S(CC)(=O)=O)C)=O)CC12CCC(NC(c1c[nH]cc1C)=O)CC2 c1(C(C(=O)NCC(CC)NC(C2CCCN2C=O)=O)(F)F)ccc(F)cn1 Cc1cccnc1C(=O)NC1CC(NC(=O)CCCc2cccc(Cl)n2)C1 c1(C(=O)NCC(CC)(C)NC(c2ccc(Cl)cn2)=O)ccc(Cl)c2cccnc12 c12ccc3nc(sc3c1)N2.C1(C(=O)Nc2c(C(=O)OC)n[nH]c2)CC=C(C)CC1 Cc1ccc(F)cc1CC(=O)NC1CCN(CC2CCOC(C)C2)CC1 C(CN=C1NCC2(CC(F)(F)C2)CN1)SC.C1(NC(C)=O)(CO)CCCCC1 C(C)(CC(=O)NCC(C)(C1CC1)NC(=O)CC1CCC1(C)C)SC N1(C(c2n(CC(C)C)ncc2)=O)CCC(C2CCN(C(=O)C=CCO)CC2)C1 N1(C(CN(C(=O)C(F)(F)F)CC)=O)CCC(CNC(c2cnc(COC)o2)=O)C1 N1(C(c2cc(OC)no2)=O)C2CCC1C(NC(=O)CN(c1ccccc1)C)C2 C=C(C)C(O)CC(=O)N1CCN2CC1c1cc(c(C)[nH]1)C2=O.CS(C)(=O)=O C1(CNC(CCCC=C)=O)(OC)CCCN(C(C2CN(C(N)=O)C2)=O)C1 C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(NC(C=C(C)Cl)=O)C12CC2 CCCCCCC(C)NC(=O)C=CC(C)(C)NC(C1CC2(CCC2=O)C1)=O c1(C(=O)NCCC(C)NC(C2CN(CCC)C(=O)C2)=O)c(N)ccc(Cl)c1F c1(NC(CC)CNC(C2(F)CCC(C)CC2)=O)nc(C(C)C)ccc1C#N C(=O)(CC(=O)OC)N(CC(=O)NCC1CN(CCC)C1)C(C)C N1(C(CC2(OC)CN(C(=O)C(C)(C)SC)C2)=O)CCC(N=[N+]=[N-])CC1 C(=O)(C(CCF)NC(C1(NC(c2ccc(C#N)o2)=O)CCSC1)=O)OC N1(C(=O)OC)CCN(CC2(NC(=O)C(C)OCC3CC3)CC2(C)C)CC1 Cc1cnccc1C(=O)N(CC(C)(C)NC(=O)CC1(O)CCOC1)C C#Cc1cc(F)c(C(=O)NCC2(F)CN(C(=O)C(CN(C)C)C(C)C)C2)c(F)c1 c1(NC(c2ncc(F)cc2F)C)nc2c(c(=NCC(C)C3CCC3)[nH]1)COCC2 c1(C(N(C(CCc2ccccc2)C(F)F)C)=O)c(F)cc([N+](=O)[O-])cc1Br C1(CC)CCN(C(c2csc(C)c2)=O)C1CNC(=O)CCCOC(C)=O c12cccc(c1)CC1CCN1C2=O.n1(CC2CCC2)cc(C(C)(C)C)nn1 c1(C(N2CCC(NC(c3c(OC)c(C)sc3)=O)C(C)C2)=O)nn(C)cc1[N+](=O)[O-] C(C(C)(C(=O)NOC(c1ccccc1)C)NC(c1[nH]nnc1C)=O)SC c1(SC)ccc(C(=O)NCC(O)CN(C)C(c2coc(CN(C)C)c2)=O)cc1 Cc1[nH]c2cc(Br)ccc2c1C(=O)NC1CC(NC(=O)C2=NOC(C)C2)C1 N1(C(COCCOCC#C)=O)CCC(C)C(N(C)C(c2ccsc2SC)=O)C1 N1(C(C(N2CCOC2=O)C)=O)CCC(C(=O)NC2CCC3(CC3)C2)C12CC2 C(N=c1[nH]cnc(NCc2ccc(C(F)(F)F)cc2)c1C)c1c(Cl)ccc(C)c1 c1(C(=O)OC)ccc(F)cc1C(C)OC(=O)NC1(CO)CC(F)(F)C1 N1(C(C)=O)CC(O)CC1C(=O)NC(c1cccc(Cl)c1)CNC(C1(C)CC1)=O C(c1ccc2c(c1)COCC2)=CC(=O)NC(CC)CN(C)C(c1cnc(S)[nH]1)=O n1(CC)ncc(C(=O)NCC2CN(C(C3(c4ccc(F)cn4)CC3)=O)C2)c1Cl Cc1cncc(C(=O)NC2CN(C(C3C4CCCC34)=O)CC2C)c1Cl c1(OC)ccc(C(=O)NC2CC2CNC(C2(O)CCOC2)=O)cc1C1CC1 C1(NC(=O)Cc2sccc2Cl)CN(C(C23CC(F)(C2)C3)=O)CC2(CC2)C1 C1(C(N(C(C(=O)N(CCN=[N+]=[N-])C)(C)C2CC2)C)=O)CCC(C2CC2)C1 n1(CCCC(=O)OC)c2nnc1CN2.C1(N(CCC(C)C)C)CCN(C)C1 c1(CCC(=O)NCC2CCCN2C(C2(CF)CC2)=O)cccnc1Cl c1(NCCOC2CCN(c3nc(OC)nc(OC)n3)C2)ccc2nnsc2c1 c1(NC(C)C#N)ccc(S(=O)(=O)NC(c2cn(C)c3cc(Cl)ccc23)C)c(Cl)c1 C1(C(N2CCCC(NCC=C)C2)C(=O)NC(C)(C)CC)CCOC(C)(C)C1 C(CC(=O)N=c1cc(-c2ccsc2)o[nH]1)N(CC)CC c1(C(=O)NC2CCCC(NC(C3CCC(N(C)C)C3)=O)C2)cnc2n1CCCC2 C12(C(=O)NCc3ccc(CC)o3)CC(CCO1)N(C(C1CCOC1C(C)C)=O)C2 C1(N2CC2=O)CCOCC1C(C)C.CC(C)CCNCC1CCCC1 N1(CC)CCC2(C1)OCc1ccccc12.c1(N(CC(O)CO)C)ccc(C=O)cc1 c1(C(N(CC(CNC(CNC(CCC)=O)=O)C)C)=O)ccnc(F)c1N CN(CC(=O)Nc1cnc2ccccc2n1)N1CC(C)(F)C(C)C1 CC1C(C(=O)NCC2(F)CCN(C(=O)CN(c3ccccc3)C)C2)=NOC1C C1(C(=O)NCC(CNC(C(CCCC)C)=O)(C)C)CC(=O)c2cc(Cl)ccc2O1 C(c1cc(C)c(C)cc1C)=NC(CCN(CC(O)C(=O)OC(C)(C)C)C(C)=O)=O c1(CC(N2CC(CC(C)NC(C(CCC)OC)=O)C2)=O)ccc(C)c(Cl)c1 c1(C(=O)NCC2N(C)CCN(C(c3c(CC)[nH]cc3)=O)C2)ccc(F)c(F)c1C C1(C(=O)N(C(CNC(c2ccc(CN=[N+]=[N-])o2)=O)C2CC2)C)(COC)CCCO1 C(=O)(C1=CCCSC1)N(CC(C)NC(c1cnc(OC(C)C)cn1)=O)CC CC1CCC(F)(C(N2CC=CC(NC(=O)CSc3nnc(S)s3)C2)=O)CC1 N1(C(c2ccc(NC(C)=O)o2)=O)CCOC2CN(C(C3CCC(=O)NC3)=O)CC12 N#Cc1ccccc1OCC(=O)NCC(CO)NC(C1COCC1C(F)F)=O c1(C(=O)NC2(C)CCN(C(Cn3c(C)ccc3C)=O)C2)ncc2n1CCCC2 C(=O)(C(C)CC(F)F)N1CCC(OCCCNC(CC2ON=C(C)C2)=O)CC1 C(=O)(C(CC)(CC)OC)NCc1cncc(C(N(c2c(CC)cccc2)C)=O)c1 N1(C(CC=C)=O)CCC2(C1)CN(C(C1(c3ccno3)CC1)=O)CCO2 c1(CC)n[nH]c(CNC(c2ccc(-c3ccc(F)cc3)o2)C)c1Br n1(CCCC)nnnc1C(c1nnn(C)n1)NC(C)C(=O)OC(C)C C#Cc1cn(C)nc1C(=O)NC1CN(C(c2nc(O)sc2C)=O)C1 Cn1c(O)nc(N2CCC(C#N)(CN3CCCC3)CC2)cc1=O C1(NC(C2(SC)CCC2)=O)CCCCCC1NC(=O)CC1(C)CCCO1 N1(C(C(C(C)(C)C)=O)=O)CCOCC(C)(CNC(C2CCCCCC(=O)C2)=O)C1 c1(N(C2CCN(C(c3cn[nH]c3)=O)C2)C)nc(Cl)nc2c1S(=O)(=O)CC2 CCC(O)C(C)(C)C(=O)N1CC2(CC(CNC(=O)CCOCC3CC3)C2)C1 C=CC1(O)CCN(C(C2(NC(=O)C=CC3CCOC3)CC(O)C2)=O)C1 C#CCCCCC(=O)NCC1CCC(NC(=O)C(C)CSc2ccc(F)cc2)C1 N1(C(COCC=C)=O)CC=CCC1C(=O)NC1CCN(C)C1 c12ccc(cc1)C(CC)CN2.N1(CC)CC(=O)N(c2cncc(Cl)c2)C1 CCC(CC(=O)OC(c1cccnn1)C(=O)OC)OC(C)=O N1(C(C(C=C=C)C)=O)CC(C)(C)OCC1CNC(c1cc(C)n(C)c(=O)c1)=O Cc1cc(C(=O)NC2CN(C(=O)Cn3ncnn3)CCC2CO)c2c(c1)CCC2 C(=O)(C1=C(C)OCCC1)N1C(C2CCN(Cc3ccnc(COC)c3)C2)CCC1 c1(C(=O)NC(CCNC(CCCNC(C)=O)=O)C)ccc2c(c1)OCC(=O)N2 c1(OCC)ccc(C)cc1C(=O)NC1(C)CCN(C(=O)C(C)(Cl)Cl)CC1 C12(C(=O)NCc3c(CNC(=O)CC(F)(F)F)cccc3)CCCN1CCC2 c1(C(=O)NCC(CC)NC(c2c(CC)scc2)=O)ccc(F)c2occc12 C1(C(N(CCOC)CCNC(=O)CCCc2nncn2C)=O)CCCC(O)C1 CC(C)C(F)(CNC(c1cnn2c1OCC2)=O)C(=O)NC1(C2CCC2)CC1 CCCCC(=O)C(=O)N1CCCC(NC(=O)Cc2ccc(OC)nc2)CC1 C1(C(=O)NCC(N(C(CCCC)=O)C)C2CC2)COCCOC1 C1(O)(CNC(=O)COCC(F)(F)F)CCN(C(=O)CNC(=O)C(F)(F)F)CC1 CCCCC(C(=O)N(C)CCNC(c1c(I)n[nH]c1C)=O)C(C)C C1(C(=O)NCCOCCN(C(=O)CSc2cnccn2)C)CCCCO1 C=C1CCC(C(=O)NCCC2CCCN(C(C3CC(F)CN3C)=O)C2)CC1 c1(C(=O)NC(CC)CC(=O)NCC2COCC(C)O2)ncc(F)cc1F CCCC(CC)C(=O)N1CC(OC)CC1CNC(=O)Cc1sccc1C N1(N2CC(NC(c3ccc(CC)cc3)=O)C2)CC2(C1)CN(C(=O)C(F)C(C)C)C2 C1(c2n(C3(C)CC3)nnn2)CC2CCCC(C1)N2C(c1sccc1Cl)=O N1(C(c2scc(OC)c2)=O)CCC(C)C(N(C)C(c2ncoc2CC(C)C)=O)C1 c1(C(C)=O)ccc(OCC(F)(F)F)c(CC(=O)NC(C2(CSC)CC(F)(F)C2)C)c1 N1(OCc2c(C)cccc2)CCCC(CCO)CC1 c1(N2CCCC(CNC(CC(CC)C)=O)CC2)ccn2ncc(I)c2n1 c1(CCC(=O)NCC(C)(C)NC(C2C(C#C)C2)=O)cc(Br)cc2c1OCC2 C=CC1(C(=O)NC(C)CCC(C)C)CCN(C(c2ccsc2Cl)=O)C1 c1(CC(=O)NC(CCNC(c2c(C)nc(SC)s2)=O)C)cc(C)ccc1F n1(CC(=O)NCCC2(NC(c3cc(C)nc(C)c3)=O)CC2)c(C)cc(C)nc1=O C1(C(N2CCC(O)(CCNC(c3c(C)onc3)=O)C2)=O)CC2CCC(C1)O2 N1(C(C(C2CCN(C(c3cc(OC)nn3C)=O)C2)F)=O)CC(N(C)C)CC1(C)C c1(CCC(N2CCCC2CCNC2CCCSC2)=O)nc(=N)[nH]cc1C(=O)OC c1(NCCNC(=O)N(C)C)ncc(S(=O)(=O)NCCC(C)CC2CCCO2)cc1Cl c1(OC)ccc(C(O)C(N2CCC(F)(C(=O)NCCC#N)C2)=O)cc1 CC1(CNC(C2CC2C(N)=O)=O)CCCN1C(=O)CCc1cccnc1 c1(C(N2CCC(C)(NC(C34CCC(C3)C4)=O)C2)=O)ccnc2ccccc12 c1(C(N(C2CCN(C(=O)Cn3cc(CO)nn3)C2)CC)=O)cnc2cc[nH]c2c1 c1(-c2cc(CC(=O)Nc3ccnc(Br)c3F)ncc2)cc(F)cc(F)c1O c1(CN(C(=O)Cn2nc(C3CC3)cc2C(=O)O)CCC)ccccc1CC N1(C(C2N(C(C)C)CCC2)=O)CCN(CCN(C)C(C2(C)CCCC2C)=O)CC1 N1(C(C2(C(CC)=O)CC2)=O)CCCC(C2CCCN(C(=O)C(O)CCSC)C2)C1 C12(NC(c3cc4cccnc4[nH]3)=O)CCCC1CN(C(c1cc(Cl)no1)=O)C2 N1(CC=CCC(=O)O)CCC2(CC1)CC(C(=O)Cc1cccc(N(C)C)c1)CO2 C1(CNC(C2CN3CCCC3CO2)=O)CN(C(c2cnc(S)[nH]2)=O)C2(CCC2)C1 c1(C(=O)NCC(CNC(c2nc(Cl)oc2C)=O)OC)cnn(CCN(C)C)c1C CC1(CNC(=O)CC2CC3CCC2C3)CCCN1C(=O)CC1CCCOC1 S(=O)(=O)(c1ccc(C)c(C)c1)N1CCC(N(c2c(Br)ccc(OC)n2)C)C1 Cc1nc(N(C)C)sc1C(=O)Nc1cccc(NC(=O)CSCc2cccs2)c1 c1(NC(C2C(C(N3CC(C)C(O)CC3)=O)C2)=O)nc2nccc(Br)c2o1 C1(C)(C(=O)NCC(CNC(CN(CCC)C)=O)CO)CCCCN1C(C)=O N1(C(Cn2ncn(C)c2=O)=O)CC(CNC(=O)C=Cc2ccn(C)c2)C(F)(F)C1 C(C(C)(C)C(=O)NC(C)CN1CCN(C(=O)Cc2cn(C)nn2)CC1)OC N1(C(C(C)C)=O)CCC2CN(C(c3cccc(CO)c3)=O)CC12 N12CCC(C1(C)C)CC(=O)N1CC3(N2CC3)C1.C1(C(C)C=O)CCOCC1 c12ccc(cc1)NC2C.C1(C(C)N)CCN(CCCN)CC1 c1(C(C(=O)NCCC(C)NC(C2COC(C)(C)C2)=O)(F)F)ccccc1F C1(NC(c2c(C#C)cnn2C)=O)COC2(CCN(C(=O)CCN(CC)CC)C2)C1 C12(NC(N3CCC(O)(C(C)C)C3)=O)CCC(C1)OC2C c1(C(=O)NCC(CNC(C(COC)C)=O)(C)O)nc(OC(C)C)ccc1Cl c1(CC=C)ccccc1C(=O)N(CC(=O)Nc1cc(Br)cs1)C C1(CC#C)CN(C(=O)C(C)N(C(=O)C2=C(C)CC2)C2CC2)CCO1 C1(N)(NC(=O)CC2CCN(Cc3c(C)c[nH]n3)C2)CCC(C)(C)C1 C1(CN(CC(=O)N(C(C)CNC(c2ccncc2)=O)CC)C)CCC(F)(F)CC1 N1(C(C2(C=C)CCN(C(=O)CCN(C)C)C2)=O)CCC2(CCOC2)C1 c1(C(N2CCCN(C(C3(C=C)CC3)=O)CC2C)=O)cc(F)cc2ccoc12 c1(NCC(C)NC(c2c(OCC)nc(C(F)(F)F)cc2)=O)ncccc1[N+](=O)[O-] C(=O)(C1=CCC(F)(F)CC1)NCC1N(C(c2cc(CC)c(C)s2)=O)CC(F)(F)C1 c1(NC(N(C2CC(C)(C)C2)C)=O)ccn2ccnc2n1.N12CC3CC1CC3C2=O c1(CCNC(=O)NCCCC(O)CO)cc(F)c(F)cc1I c1(C(=O)OC)nc(NCC2CCCCN2C(c2cnc(C)s2)=O)sc1C C1(NC(CNC(CC)=O)=O)CC12CC(NC(c1ccc(C)s1)=O)C2 N1(C(CC=C(C)C)=O)CCCC2(CCC(NC(=O)C(C)(C)C3CCC3)C2)C1 C1(NC(=O)Cc2nc[nH]n2)CC(NC(C2CC(=C3CCC3)C2)=O)CC1O C1(CNC(c2cccc(CSC)c2)=O)CN(C(=O)CCOC2CCC2)CCC1C c1(C(=O)NCC2(C)N(C(C3C(C=C)C3)=O)CCC2)cc2n(c1)CCS(=O)(=O)C2 c1(C(=O)NC2C(CNC(C(c3cccc(C)c3)C)=O)C2)cccc2nccn12 c1(CC(C)NC(C2C(CO)C3CCCC23)=O)cc2ccccc2s1 N1(C(CCC(CC)=O)=O)CC2CCC(N(C)C(c3ccc(CC)[nH]3)=O)C2C1 C1(C(=O)NCCNC(C(CCCC)F)=O)CCOC2(CCC2)C1 c1(OC)cc(Br)cc(F)c1CN1CCCC(C)(C(=O)NC2CC(C)C2)C1 CC#CC1CCN(C(c2ccnnc2N2CCCCC2)=O)CC1 C#CCC(CC#C)C(=O)N1CC(CNC(=O)CC(CC)C2CCC2)C2(CC2)C1 C1(C(=O)NCC(C)(C)CCNC(C2CCC(=O)N2)=O)OCCCC1(C)C N1(C(Cc2c(C)nc(S)s2)=O)CCC(NC(=O)C(C)P(C)(C)=O)C(F)C1 C1(SC)CCCN(C(=O)C(CN2CCCC2)c2ccccc2)CC1.N12CCC1C2 C1(NC(c2cc(F)c[nH]2)=O)COCCN(C(C2CCOC2)=O)C1 C1(C2CCN(C(=O)C=CI)CC2)(NC(CCCC#C)=O)CC1 Cc1cc(C(N2CCCC23CCN(C(=O)C(C)CC(F)F)C3)=O)cc(C)c1C#N CC12CC(CC(=O)Nc3ccccc3C3CCNCC3)(CO1)C2 N1(C(C(C)N=[N+]=[N-])=O)Cc2occ(C(N3CCC(N(C)C)C3)=O)c2C1 N1(C(CN)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccc(Br)s1 C1(C(N(CCCCNC(C(CCCC)F)=O)C)=O)CCc2nncn2C1 C(=O)(CCCCCS(N)(=O)=O)NCC(CNC(C1(C)CCN(C)CC1)=O)CO c1(C(N(C2CC(NC(CSCCOC)=O)C2)CC)=O)ccnn1CC(F)(F)F c1(C(=O)NC2CCN(C3CCN(C(C4CC(=C)C4)=O)CC3)C2)ccc(F)c(F)c1 c1(C(=O)NCC2(F)CC(CNC(c3c(C)snn3)=O)C2)nccn2nccc12 C1(NC(c2c(C)cn(C)n2)=O)CCC12CN(C(=O)Cc1cc(Br)cs1)C2 C1(NC(CC=C)=O)Cc2ccccc2N(C(=O)CCCc2cc(C)no2)C1 CC(CCC(C)(C)C)C(=O)Nc1cc(-c2cccc(F)c2C(F)(F)F)ccn1 c1(C(=O)NCCC2CCN(C(c3ccc(C)n3C)=O)C2)cc(Cl)ccc1Cl C1(C(=O)NCC(Cn2cc(C3(C)CCOC3)nn2)OC)CC1C1CCCC1 c1(C(N2CCC3(CC2)CC3)C(=O)NC(C(=O)OC)C)cccc(C)c1Br C=CCCC(C)(C)C(=O)NCC(C)(C)CNC(=O)C(c1ccc(Cl)cc1F)O Cc1cc(Oc2cccc(NC(c3cnn4ccsc34)=O)c2)cc(C)c1C C1(CC(N2CCOC(CN(C(=O)CCCCC3CC3)C)C2)=O)(OC)CCCCC1 c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC(C)CN(C)C(C1(F)CC1)=O C=CCC(CC(C)C)C(=O)N1CC(F)(F)CC1CNC(c1ccsc1Br)=O N1(C(C(C)(C)C2CC2)=O)CC(NC(=O)Cn2nc3c(n2)CCCC3)C2(CCC2)C1 c1(CN2CCC(COCCC)C2)cc2ccc(Br)cc2nc1Cl CCC(C)C(O)C(C)C(=O)NCC(C)(C)C(=O)NCC1CCN1CC Cc1ccc(C(C)(F)F)cc1C(=O)NC1CCC(NC(c2cn[nH]c2)=O)CC1 c1(C(N2C(C(=O)Nc3ccc(-c4n(CC)cnc4)cc3)CC2)=O)nc(F)ccc1F OC1CCN(Cc2ccccc2)CC1NC1CCN(C2CC2)CC1 CC(C)(C(=O)N1CCC(NC(=O)CC(=O)NCC2CC2)C1)c1cnc[nH]1 C1(NC(=O)CCCCc2cnn[nH]2)CCCCCN(C(=O)CC2CCCC2)C1 C(=O)(N=c1ccn(CCCO)[nH]1)C1(CNC(C(CCC)C#N)=O)CC1 c1(OCCNC(=O)CNC(C2CCOCC2)=O)ccc(Cl)nc1 c1(C(N2CC(N(C(=O)C(F)CC3CCC3)C)C2)=O)c(F)ccc(F)c1O C(=O)(C(=O)N=S(C)(C)=O)NCCC1N(C(c2c(OC)cc(F)cc2)=O)CCOC1 C=CC(C)(O)CC(=O)N1CCCCC1CCNC(c1cc(O)n(CC)n1)=O c1(C(=O)NCC(=O)NC(C)C(C)NC(c2cn(C)nc2Cl)=O)c(F)cccc1Cl C#CC(C)(C)C(=O)N1CCN(C(C)CNC(=O)CC2CC3CCC2C3)CC1 c1(C(=O)NCC(C(C)C)NC(c2ccc(C#C)nc2)=O)c[nH]c2nccc(Cl)c12 Cc1nccnc1C(=O)NCc1nc(C(=O)N(C(C)C)CC2CCC2)co1 c1(SC)cccc(F)c1C(=O)NCC1CCCN(C(C2(C#N)CCCO2)=O)CC1 c1(OC)ccc(F)c(C(=O)NCCCCCNC(=O)CC2CCC(=O)NC2)c1N N1(C(CNC(=O)OC(C)(C)C)=O)CCC2CN(C(=O)CN3CSCCSC3)CC12 c1(C(=O)NCC(CC(C)C)NC(=O)C(C)(C)CC(F)F)ccc2nc(O)oc2c1 c1(C(=O)OC)c(NC(C2CCN2C(c2ncc(Br)cc2C)=O)=O)sc2c1CCC2 C(C(C(=O)NNC(=O)CNC(c1c(F)cccc1Cl)=O)n1cc(C(C)O)nn1)OC C1(O)(CNC(C(C)(CO)OC)=O)CCCN(C(c2coc(C#N)c2)=O)C1 C1(N(C(CCN(CCC)C)=O)CCNC(=O)CCNC(N)=O)CCCCC1 c1(C(=O)NCC(C)CN(C(=O)C(c2cscn2)N(C)C)C)ccc([N+](=O)[O-])s1 C(CCCCNC(=O)C(C)(C)c1nncn1C)N(C(CNC(CCOC)=O)=O)C N1(C(C2CCN(C)C2=O)=O)CC(NC(C2CC(F)(F)C2)=O)CC(F)C1 C(=O)(C(C)C(C)C(C)(C)C)N1CCC(N(C(=O)CCCS(C)(=O)=O)CCC)CC1 c1(NC(C2C3CN(Cc4cnc(C(F)(F)F)nc4)CC23)=O)ncnc2sccc12 C(=O)(CCCC(=O)NCC(C)(O)CNC(c1cc(F)ccc1CC)=O)NCC c1(C(=O)Nc2cc(CSCC)c(Cl)cc2)sc2ccccc2c1CC CCCC(C(=O)N(CC(C)(C)CNC(=O)CN(c1nnc(C)n1C)C)C)C(C)C CCCS(=O)(=O)CC(=O)NC(C)(CNC(=O)Cc1ccc(Cl)nc1C)C1CCC1 N(S(=O)(=O)N1CCOCC1CC(=O)OC(c1cccs1)=O)C1CC(OC)C1 CCC(N=c1ccnc(N2CCN(CCOC)CC2)[nH]1)c1ccc(F)cc1F c1(CC(N2CC(C)C(NC(C3(C)CC3C)=O)C2)=O)cc2ccccc2o1 C1(NC2(c3n(C)nnn3)CN(C(C3CC4(CC4)C(=O)O3)=O)C2)COCC(C)(C)O1 C=CCN=C(NCC1CCOCC1C)NC1CC(C(N)=O)C1 N1(C(c2c(C)ccc(OC)n2)=O)CC2(COC(CNC(=O)C=CCF)C2)C1 CC(Cc1cnc[nH]1)C(=O)NCC(O)CCNC(=O)CCc1cncn1C c1(OCC(N2CC(CCNC(CCNC(C)=O)=O)C(C)C2)=O)cccc(C#N)c1 N1(C(c2cncc(C(C)C)c2)C(=O)N(CC)C2CC2)CCN(C)CC1CCO C1(C(=O)N(CC2C(C(N(C3(C)CC3)C)=O)CCO2)C2CC2)C(C#N)C1(C)C c1(C(=O)NCC2(C)CCC(NC(C3(CC)CCC3)=O)C2)cc(F)cnc1O C1(O)(CNC(c2ccc(F)cc2)=O)CCN(C(c2ccccc2CO)=O)CC1 c1(OC)c(C)nc[nH]c1=NCC1(F)CCN(C(C2(OC)CC2)=O)CC1 N1(C(c2cn(C(C)(C)C)nc2)=O)CCC2CCCC12CNC(c1cnn[nH]1)=O CC1C(C)N(C(c2ccncc2F)=O)CCN1C(=O)Cc1csc(S)n1 C1(C(=O)NCCc2nnc(C)n2C)CN(C(C2CC3(CCC3=O)C2)=O)CC1(C)C N1(C(C(CCCC)C)=O)CC2CCCCC2(CNC(c2ncoc2C2CC2)=O)C1 C1(CNC(C(c2ccccc2)NC(CC)=O)=O)CC2CN(C(=O)C(F)(F)CC)CC12 Cc1nc(C(C)C)ccc1C(=O)NC1COCC1CNC(c1cnc(S)n1C)=O c1(CC)ccc(OC)c(C(N2CC(O)CCC2C)C(=O)NC(C)(C)C)c1 N1(C(C(C)Sc2nncn2C)=O)CCC(NC(=O)CC2CC=CCC2)C12CCC2 N1(C(c2nccc(C)c2)=O)C2CCC1CC(NC(c1cccc3nonc13)=O)C2 C(C(CC1CCCC1)C(=O)NOC1CCC1)NC(C(CC=C)NC(C)=O)=O N1(C(CN(CCOC)C)=O)CCN(C(c2ncccc2N)=O)CC12CC2 CC1CC(NC(c2cc(C3CCCN3C)[nH]n2)=O)CN1C(=O)C(C)n1cccc1 C1(OC)(CF)CCN(C(C2(C(C)N)CCCN2C(=O)OC(C)(C)C)=O)C1 Cn1cc(C(N2CC(NC(=O)CCc3cn[nH]c3)C(O)C2)=O)ncc1=O C12(C(N(C)Cc3ccccc3F)=O)CCN(C(=O)CCCCC#N)CCC1C2 C1(C(N2CCCC(NC(C(C)(C)C3CC3)=O)C2)=O)CC(=O)c2ccccc2C1 N1(C(CCCc2ccc(C)s2)=O)CCCCC(NC(=O)COCC2CC2)CC1 N1(C(CC2CC(=C)C2)=O)CC2CN(C(=O)CC3COCC(C)(C)O3)CC2C1 c1(CN2CCOC(C)(C(=O)NCc3c(C)n[nH]c3)C2)nnc2ccccn12 c1(C(N2CCCC(CCNC(C(CC)=CC)=O)CC2)=O)cc2nc(=O)ccn2[nH]1 CC(CO)(C(=O)N1CC(C(N)=O)C1)NC(c1coc(C(F)F)c1)=O C(=O)(C1=CCC2CCC1N2C(=O)C(CC(C)(C)C)OC)NCC(COC)(O)CO C1(CC=C)(NC(C(C)OCCC=C)=O)CCN(C(=O)C2=CSCS2)CC1 C1(NC(CN(CCC)C)=O)CC(C2CCN(C(C3(C#N)CC=CC3)=O)C2)C1 C1(NC(=O)C=Cc2nccs2)C2CC1N(C(c1cc(C(F)F)ccn1)=O)C2 Cc1cc2c(=NC(=O)NCCCC(C)C)[nH]cc(Br)c2c(=O)n1CC C12(C(=O)NCCn3cc(C(=O)NC(CN(C)C)CO)nn3)CCCC1CCC2 C1(N(C)C(c2cnn(C3CC3)c2Cl)=O)CN(C(C2CCCS2(=O)=O)=O)CC1(C)C C(=O)(C(C)(O)C(C)(C)C)N1CC2CC(NC(c3cc(C)on3)=O)C2C1 C1(NC(COCC)=O)CN(C(c2ccc(-c3ccco3)nc2C)=O)CCC1F c1(NCC(=O)NC(c2ccc(C)cc2)CCCC)ncnc2cnn(C)c12 C(=O)(CC(C)(C)CNC(C1COCC1C(N)=O)=O)N(CCCC)C1CC1 C1(C2(C)CC2)(C(C(N2CCC(N(N3CC(CC(C)(C)C)C3)C)C2)=O)=O)CC1 n1(CCC)ncc(C(=O)NC2CC(C)(NC(=O)CN3CCCC3C)C2)c1C CCC(CN(C)C)CC(=O)NCCOCCN(C(=O)CCc1cnn(C)n1)C c1(C(=O)NC(CC(C)NC(c2cc(C(F)F)ccn2)=O)C)nnn(C)c1N c1(CC)[nH]nc(Cl)c1C(=O)N(CCCNC(C1CCC(=O)N1C)=O)CC N1(C(CSC)=O)CCC(C)CC1CNC(=O)C(C(C)O)NS(C)(=O)=O O(C=CC(=O)NCC(C1CCOC1)NC(C1(C#N)CC1)=O)CC N1(C(C2C(C=CC)CN(C(=O)CC3(OC)CCC3)C2)=O)CCc2nncn2CC1 c1(OC)ccc(C(N2CC(C(=O)NCCCCCCO)C2)=O)c(OC)n1 Cc1cc(F)ccc1C(=O)NCC1(O)CCN(C(=O)CC2(O)CCCCC2)C1 C(=O)(C(CN=[N+]=[N-])NC(=O)C(c1ccccc1)F)N(C)CC1CCN(C)CC1 c1(NC(=O)OCC)cnc(C(=O)NC2CN(C(=O)C(C)Cc3cnc[nH]3)C2)cn1 N1(C(C(COC)C)=O)CC2CN(C(c3ccnc(-n4cccc4)c3)=O)CC12 c1(C2(C)N(C(C(=O)NC(C)Cc3cn[nH]c3)=O)CCC2)ccc(F)cc1F CC1(C)CCN(C(=O)C(c2ccccc2)O)CC1NC(c1ccccc1)=O CC(C)C(F)C(=O)NCCC(O)CNC(c1cccc(-n2ccnc2)c1)=O CC(c1cnn(C)c1)=CC(=O)NCC1(C)CC(NC(C2(C)CC3CC3C2)=O)C1 c1(C(C(=O)NCCN(C(C=CC(CC)=CC)=O)C2CC2)C)cccc(Cl)c1 O=C(C(Cn1cccn1)NC(=O)C(O)C1CCC1)NC1CCCC1F c1(CC)cc(C(=O)NC2CCN(C(=O)C=CC3CCC3)C23CC3)ccc1OC c1(NCC(N2CC(CCNC(C(C)C)=O)C2)=O)cccnc1Cl S(=O)(=O)(CC(=O)NCC1(C)CCCN1C(=O)CCN(CCC(C)(C)C)C)NC N#CC1(C(N2CCC(CF)(NC(C34CC(F)(C3)C4)=O)C2)=O)CC2C=CC1C2 C123CCCC1N(CC2)CCC1CC1CNC3=O.c12sccc1C2.CO.CO C1(CNC2CC(CC)SC2)CCN(C(=O)OC(C)(C)C)CC1 c1(C(=O)NCC(CC)(CC)NC(=O)CC2(C3CC3)CC2)nccn2nc(C)cc12 C1(NC(=O)C(O)C(F)F)CC2CCCC(C1)N2C(c1c(Cl)cnn1C1CCCC1)=O C=CCCC(C(=O)NCCN(C)OC)NC(c1cnns1)=O C1(C(=O)NCC2CCCCN2C(=O)Cc2n[nH]cc2Br)CC12CCSCC2 C(N=c1[nH]c(=NCc2ccc(C(F)F)o2)[nH]c2ccccc12)C1C(C)C1 C(=O)(C1=CN=C2N=CNN2C1)N(CC(C)NC(=O)CC1CCCC(C)(C)O1)C CC(CO)C(C)N=c1[nH]c(=NCCC2(C)CC2)[nH]c2c1COC2 N1(C(CCCC#C)=O)CCC(CO)C(NC(c2ncn3c2CCC3)=O)C1 c1(CCC(=O)N(C2CN(Cc3cnn(C)c3)C2)C)ccccc1Br O=C(C1=CC2(CCOC2)C1)N1CC2CCC(C1)N2C(C12COC(F)(F)C1C2)=O N1(C(COC(C)C)=O)C(CC(=O)NC(CC2CCCC2)CO)C2CCCC12 c1(C(=O)OC)cc(S(=O)(=O)NCc2nn(C)c(Cl)c2I)sc1C N1(C(C(C)=C2CC2)=O)CC2CC2(CNC(c2cc(-c3ccco3)no2)=O)C1 N1(COC)CC(C(=O)NCC2(O)CCN(C3CC3)C2)CC1=O.C12(CC1)C(=O)N2 C1(NCC2N(c3nc(C)cc(C)n3)CC3(CC3)C2)CCc2n[nH]cc2C1 C1(C(C(=O)NC2CC(CNC(=O)C(O)C3CCC3)C2)OC)CCC(F)(F)CC1 C(=O)(C1=CC2CCCCC12)NC1CC(C)N(C(=O)CSc2n[nH]c(=N)s2)CC1 CC(C)(CO)C(=O)N1CC(C)(CCC(=O)NCC2CC=CCC2)C1 c1(C(=O)NCCCCCNC(C2(CC#C)CCCCC2)=O)c(OC)cccc1Cl C1(NC(C(COC(C)C)C)=O)CC2CC(NC(c3c[nH]c(C(N)=O)c3)=O)CC12 C(CCC(C)C(=O)N1CCC2C(C(=O)NC3CCC3C(=O)OC)C2C1)OC C1(N(C(c2nccc(CC)c2)=O)C)CCCCN(C(C2CCN(C)C2C)=O)C1 C1(C(CNC(C(COC)C)=O)(C)O)CCN(C(c2cnc(N(C)C)s2)=O)CC1 c1(OC)cccc(C)c1C(N1CCC(O)(CCNC(C2CCC2(C)C)=O)C1)=O C(=O)(C1OC(=O)c2ccccc21)N1CC(O)(CNC(=O)C=CC2CCCCC2)C1 N1(Cc2ccnc(C)c2)CCCC1C1CCCN1C(c1cc(CSC)[nH]n1)=O Cn1nc(C(=O)NCC2(CNC(=O)C3=CCCOCC3)CC2)c2c1CCSC2 C1(NC(CNC(=O)OC)=O)CCN(C(=O)CCC2CC(C)C2)C12CCCC2 N1(C(c2c(OCC)ncnc2C)=O)CC2CCCCC2(CN)C1 CC1CN(C(C2CCCN2C)=O)CCC1NC(C1(C(=O)NC2CC2)CCC1)=O C1(NC(C(C(C)C)OC)=O)COCCN(C(=O)Cc2cc(C(C)C)no2)C1 CC(CC(F)(F)F)C(=O)NCC1CC(NC(=O)CCC(F)F)C1 C(=O)(CCCC(=O)NCCC1CCCN1C(=O)CCc1cnn[nH]1)N(CC)CC C1(NC(CCC=C=C)=O)COC2C(NC(c3sccc3OC)=O)COC12 c1(CC)c(C(N2CC(CCNC(=O)CC3CCOC3(C)C)C2)=O)nnn1C C1(C(=O)NC(C)(CNC(=O)C=CCF)C2CC2)CC2(C1)CC2F N1(C(=O)NCc2cn(CC)nc2C(C)(C)C)Cc2ccccc2N2CCCC2C1 CC(CS(C)(=O)=O)C(=O)NC(c1ccccc1F)CNC(=O)C(F)=C1CCC1 CC12CC(CC(=O)NCCNC(C3CCC3c3ccc(O)cc3)=O)(CO1)C2 c1(C(=O)NC2C(CNC(Cc3cnc(C)s3)=O)CC2)cc(N)ccc1[N+](=O)[O-] c1(CNC2C(C(=O)Nc3cnc(CC)nc3)C2)ccc(Br)c(C)n1 CC1CC(NC(=O)CCc2cnc(O)[nH]2)CN(C(C2CCC(=O)N(C)C2)=O)C1 n1(CCCC)nccc1C(=O)NCCOCCN(C(=O)CCCN(CCC)CC)C c1(C(N2CCC(CC(=O)NCc3cnccn3)C2)=O)coc2c(F)cc(F)cc12 N(C(=NCc1cnnn1C)NC1C(C)(C)C1(C)C)C(CC)C C(=O)(CS(=O)(=O)C(C)C)N1C(C)CC(CNC(C(CC)c2ccccc2)=O)C1 C(=O)(C(COCCCN(C(CN(CC)CC)=O)C)N(C)C)N.C(C)(C)(C)ON c1(CC(=O)NCC2CCC(NC(=O)CCc3nc(Cl)no3)C2)cc([N+](=O)[O-])n[nH]1 c1(C(N(C2CCN(C(CSC)=O)CC2C)C)=O)cccn2ccnc12 C(=O)(C(C)(C)OC)N(CCN(CC(CC)O)C)C CN1CC2(CC2)CC1C(=O)NC(CCC1CCC1)C(=O)N1CCC(F)(F)C1 C1(C(=O)NCCCCCCC)CN(C(c2cc(CC)on2)=O)C2(CCC2)C1 c1(C(=O)NCC(C)(C)CNC(C2C(F)(F)C23CC3)=O)[nH]c2ccccc2c1C#N N1(C(C(C)C2CCCC2)=O)CCCC(N(C(c2ccc(CO)o2)=O)C2CC2)C1 c1(C(N2CCC(NC(C(C)C3CC3)=O)(CF)C2)=O)ccn(C)c(=O)c1 Cc1cccc(C(=O)NCCC2(CNC(c3ccco3)=O)CC2)c1C(F)(F)F N1(C(C2(F)CCCC2)=O)CC(O)CC1C.CC1C(=O)NCC2N1CC2 c1(C(=O)NCCNC(C2(C)C(C(=O)OCC)C2)=O)ccccc1S(=O)C(F)(F)F C1(C(=O)NC(c2cccnc2)COC)CC(C)C1(C)C c1(C(=O)NC(CC=C)CNC(=O)CCOCC(F)(F)F)cn(C)nc1OC C1(NC(C2(F)CCC2)=O)CCC2CN(C(C3(F)CCOCC3)=O)CCC2C1 C1(NC(C2(OC)CCC2)=O)CCN(C(c2csnn2)=O)CC1O CCC(O)C(C)C(=O)NCCOCCN(C(=O)C(C1CC1)SC)C N1(C(c2scc(C#N)n2)C(=O)NCc2cccs2)CCCCCC1CCO c1(C(=O)NCC2C(NC(C(C)OCC)=O)C2)c(O)nc(C)c([N+](=O)[O-])c1C C1(CNC(C(C(=C)Cl)(C)C)=O)CC2(CCC2)CN1C(c1sccc1C1CC1)=O Cn1cnc(C(=O)NC(C(=O)NCC2CC23CCC3)C2CCC2)c1 N1(C(=O)Cc2cnc(C3CC3)[nH]2)CCCCC(CNC(C2(Br)CC2)=O)C1 c1(NCc2nccc(C)c2)ccc(C(=O)NC2CC(=O)NC(=O)N2)cc1C c1(CCNC(N2CCC(Nc3ccc(C)cc3)C2)=O)cccc(S(C)(=O)=O)c1 N1(C(C(CC)OC)=O)CC(NC(c2cc(COC)[nH]n2)=O)C(n2cccn2)C1 C1(C(=O)NCC2CN(C(c3c[nH]cc(C)c3=O)=O)C2)COc2ccc(F)cc2C1 CC1(C)CCC1C(=O)NCCCCCC(=O)CCc1ccc(-c2ccccn2)o1 CC12CCN(C(C3CSC3)=O)C1CN(C(=O)C=CC1CCC1)C2 c1(CC(NNC(=O)C2N(C)CCC2)=O)c(Br)ccc(Cl)c1F c1(CNc2cc(CCC)nn2C)c(F)ccc(F)c1F c1(NC(=O)NC(C(N2CCN(C3(C#N)COC3)CC2)C)=O)ccc(F)cc1Cl c1(CC(=O)NCC2C(C)(C)CCN2C(c2cc(Cl)no2)=O)ccc2c[nH]nc2c1 CN1CCN(C(c2cnsn2)=O)CC1CNC(c1coc(Cl)n1)=O C1(C)(CC)CN(C(=O)CCOCC2CC2)CCO1 C(=O)(C1=CCCCC1)NC1CC(CC(=O)N(C2CCC2)C)C1(C)C C(=O)(C(CCC)C(C)C)NC1(CCC(=O)NC(CCCC)COC)CCCC1 C12(NC(c3c(C)onc3)=O)CCC(C1)N(C(=O)CC(O)CN(C)C)C2 CCCC(C)(CCC)C(=O)NC1C(CNC(=O)CC2CC(=O)NC(=O)C2)C1(F)F C1(C(=O)NC2CC(CCNC(=O)CSc3cccnc3)C2)C2CNC(=O)C12 c1(C(N2CCCC(CN(C)C(C3(F)CC3)=O)C2)=O)cc(C(F)(F)F)cc(O)c1 c1(OC)ccc(O)c(C(=O)N(C2CCN(C(=O)C(C)C)CC2)CCO)c1 c1cc(C(F)(F)F)ccc1F.c1(NC(C(=O)N(C(C)C)NC)=O)nc(C2CC2)no1 N1(C(C(=O)NCCCC)C2CC(CC)C2)Cc2c[nH]nc2C1 n1(CC)cc(CCN(C2CC(O)C2)CC2(CC)C(C(=O)OC)C2)c(C)n1 C=CCC(C)(C)CC(=O)NC1CC(O)(CNC(=O)CC2COCCO2)C1 C(c1ccc(Br)s1)=CC(=O)NCC1C(NC(C(=O)N(C)C)=O)CC1 n1(CC(=O)NC(COCC)C(=O)NC(c2cncn2C)CO)ncn(C)c1=O CCCCC(O)C(=O)N1CC(C(=O)NC(C)C(F)F)(CC)C1 c1(C(=O)NCCN2CCN(C(COC(CC)C)=O)CC2)ccc(C)nc1C(C)C c1(N2CC(CNC(C(C(CC)C)C)=O)OCCC2)c(C)c(C)nc2ncnn12 c1(C(=O)NCC2CCC(NC(c3c(OC)csc3)=O)CC2)cccc(C)c1F C(C(=O)N1CCCO1)NC(C(CN(C)C(C1C2CC3C(C2=O)C13)=O)(C)C)=O c1(C(=O)NC2C(CC)CN(C(=O)C(F)(F)CC3CC3)CC2)ccc2c(c1)CCCS2 c1(C(=O)NCC(CNC(C(c2ccc(C)nc2)=O)=O)C)c(Cl)nn(C)c1Cl c1(OC)cc(Br)ccc1CNC1CC(NS(=O)(=O)C(F)(F)F)C1 N1(C(c2n(C)cnc2)=O)CCN(C(=O)CCNC(C2CCCCC2)=O)CC1CF Cc1cc(NC2(c3nnnn3C3CCC3)CC(C)N(C)C2)cc2n[nH]cc12 N1(C(=O)OC(C)(C)C)CCC(CNCC23CC(C(=O)O)C(C2)C3)CC1 c1(C(=O)NC2C(CNC(C(C)Sc3ccccn3)=O)CC2)cc(O)n(C)n1 Cc1c(-c2cn(-c3c[nH]nc3C)nn2)cccc1Br c1(CC(=O)NC2C(NC(C(C)OCCCC)=O)CCC2)cccnc1Cl c1(C(=O)NCC2(NC(C(CC)F)=O)CCC2)ccc(Cl)c2c1OCCO2 C1(CN(C(COCCC)=O)CC)CCCN(C(=O)C2CC2)C1 c1(C(c2n(C(CC)C)nnn2)NCc2cncn2C(C)C)c(Cl)nc(Cl)n1C N1(C(CC(C)C(C)(C)NC(C2CC3CCC3C2)=O)=O)CC2(C)COCC2(C)C1 c1(C(N2CC(CO)C(C)C2)=O)cccc(-n2cc(CNC(C3(F)CC3)=O)nn2)c1 C(=O)(C(C)S(C)(=O)=O)N1CC(C(C)NC(c2noc(C)c2Br)=O)C1 C(CN=C(NC1CCOCC1)NC1CC1c1ccc(F)cc1)c1ccc(OC)cc1 N(C(=NCc1ccoc1)N1CCC(F)(CN2CCCC2)C1)Cc1n(C)ncc1 Cn1cc(CNC(=O)C(C2CCN(C(=O)CSC3CC3)C2)F)nn1 c1(Nc2scc(C)c2)nc(N(C)CC2CCOCC2C)c2ncn(C(C)C)c2n1 N1(C(c2c(OCC)ccc(C)n2)=O)CCC2(CC1)COC(CNC(=O)C(C)C)C2 C1(CNC(C=CSC)=O)COCCN1C(C1(c2ccc(Cl)nc2)CC1)=O c1(CC)c(C(=O)NC(c2ccccc2)C(C)NC(=O)C(F)=C(C)C)cnn1C c1(NC(c2ccncc2O)=O)sc2c(c1C(N1CCCCC(F)(F)C1)=O)CCC2 c1(C(=O)OCc2cc(OC(F)F)ccc2F)cc(O)ccc1[N+](=O)[O-] Cc1cc(C(F)(F)F)nc(N2CCCC2CCNC(c2c[nH]cc(C)c2=O)=O)n1 Nc1c(C(=O)NCCCOCCNC(C2(CO)CC2)=O)cnc2ncnn12 c1(C(CONC(=O)Nc2ccnc(C(F)(F)F)c2)=O)ccc(F)cc1F CN1CCC(C(=O)N(C2CCC2=O)CC(N2CCCC2)=O)C1 c12cc(C)ccc1CNC2=O.C1(NC(CSCC)=O)CCCCC1n1cccn1 N(C(=NCC(=O)NC1CCC1)NCC(C(F)(F)F)N1CCOCC1)C1C(C)C1 Cc1cccc2c1CCN(C(C1COC3(C1)CN(C(=O)CNC(=O)C1CC1)C3)=O)C2 Cc1csc(=O)n1CCCC(=O)NC(CNC(c1cccc(Cl)c1)=O)CO c1(OC)ccc(Cc2cc(C)n(C)c2)c(C(F)(F)F)c1.C12C3CN(CC13)C2=O c1(C(=O)NC2CN(C(=O)C3=CC(O)CCC3)C2)cc(Cl)c2ccncc2n1 CC1CCN(CC(=O)NC2CC(C(C)NC(c3cc(C(F)F)cs3)=O)C2)C1 C(=O)(C1=CC2C=CC(C1)C2)N1C(CCN(C)C(c2ncccc2F)=O)CCCC1 CC(C)(C)CC(O)CNC(c1ncoc1CNC(c1sccc1C#N)=O)=O c1(C(=O)NC(C(C)C)CNC(C2COCC2(C)C)=O)c(Cl)cncc1Cl Cc1cc(C)c(CC(=O)NC(CNC(=O)C=CC2CCOC2)C2CC2)s1 C(C1c2ccccc2CN1C(C1CCCC1O)=O)NC(CSCCC)=O CC1CCC(CNC(=O)C(C)(O)C2CC2)CN1C(=O)CN1CCCCC1C Cc1oncc1C(=O)NC1CCC1NC(=O)C(C)(C)Oc1ccccc1 C#CC1(C(=O)NOC2CCCC2)CCN(C(C23CCC(C2)C3(C)C)=O)CC1 c1(-c2nc(COC)nn2-c2ccc(Cl)c(F)c2)cncc2nc(O)[nH]c12 N1(C(C(C)CCO)=O)C2CCC1C(C)C(NC(c1cc3c(o1)CCCC3)=O)C2 C#CC1(C(=O)NCC(CSC)OC)CCN(C(C2CCC(C)O2)=O)C1 C#Cc1ccc(F)c(C(=O)NC2CCN(C(=O)CN3CCCS3(=O)=O)CC2O)c1 Cc1c(C(=O)NCC(CC(C)C)NC(C23COCC(C2)C3)=O)cncc1N c1(OC)ccc(CO)cc1C(=O)NC1CC(NC(C)C2CC2)C1 CCC(CC(=O)N1CC2(CC(NC(=O)CNc3cnn(C)c3)CO2)C1)C(C)(C)C C1(CC)CCCC1N=c1[nH]c2c(c(=NC3CCCN(C)CC3)[nH]1)COC2 c1(CC)ccc(C(N2CCC(O)(C(C)CNC(=O)C3=CCCC3)C2)=O)cc1F c1(C(=O)NC2C(NC(C3(NC(C)=O)CCC3)=O)COC2)nccn2nc(C)cc12 N(C1COc2cc(Br)ccc21)C(=O)NCCCCOc1ccccn1 C(=O)(C1=CCc2ccccc21)NC(C)CN1CCN(C(C2(F)CC2C)=O)CC1 C1(CC(=O)NCC2C(C)(C)CCN(C(=O)C3CC3)C2)Cc2ccccc2NC1=O CC(C)C(F)(CNC(=O)CCc1cn[nH]c1)C(=O)NCC1(F)CCOC1 c1(N(CCN(C)C(c2c(F)ccc(F)c2Cl)=O)C)cc(=O)n2ccccc2n1 C=CC(CCC)CC(=O)NCCC(C)N(C(=O)C1=CCCCC1)C Cc1[nH][nH]c(=NC(=O)C2CC2C(=O)Nc2ccc3c(c2)CC(=O)N3)c1Cl CN1CCN(C(C2NCC23CC3)=O)CCN(C)CC1 C(=O)(CC(C)(C)C(F)F)N1CC2C(N(C(=O)Cc3cc(C(F)(F)F)c(O)nn3)C)C2C1 N1(C(c2cnc(C(C)C)o2)=O)CCOCC1CCNC(=O)CCc1cc[nH]n1 C(C1CCCN1C(c1ccc(CN(C)C)o1)=O)=CC(=O)NC1C(C)COC1 C(C)(C(F)(F)C(F)(F)F)N1CC(C(=O)OC)C(F)(F)C1 c1(C2(C(N(CCN(C(=O)Cc3nc(=N)[nH][nH]3)C)C)=O)CC2)ccc(O)cc1 CC1CCC(C(=O)NCC(F)(F)Cn2cc(CCNS(C)(=O)=O)nn2)CC1 N1(C(c2cc(C)c(C)[nH]2)=O)CCC2(CCC2)C(NC(C2CCC2)=O)C1 Cc1ccc(C)c(C(=O)NC2(CC(N3CCN(CCC(C)(C)C)CC3)=O)CCC2)c1 C1(F)(CNC(c2ccn(CC(F)(F)F)n2)=O)CCN(C(C2(CO)CC2(F)F)=O)C1 Cc1c(C(=O)N(CCCNC(C2CCC3(C2)CC3(F)F)=O)C)nn2ccccc12 C(=O)(C(C)(C)COC)NC1(CC)CCC1.C12CCC(C1)C(=O)N2.C(C(F)F)O CC12CCC(C(=O)NCC3(NC(C4CC4CF)=O)CCCC3)(CC1)CO2 C(C(=O)NC(C(C)NC(=O)C(=O)NCCC(N)=O)C(C)C)(C(C)C)SC N1(Cc2ccc(CCC)s2)CCC(O)(C(=O)NC(c2cncnc2)C)C1 c1(C(N2CCC(C(C)CNC(=O)CC3CC3(C)C)CC2)=O)nccc(Cl)c1O C(=O)(C1Cc2ccccc21)N1CCC(O)(CNC(c2n[nH]c3c2CCC3)=O)CC1 C1(CNC(C(C=CC)O)=O)COC(C)(C)CN1C(=O)CN(C1CCS(=O)(=O)C1)C c1(C(=O)NC(CNC(Cc2c(C)ocn2)=O)(C)C)oc(CO)nc1C N1(C(C(CC(C)C)N(C)C)=O)CCC2(CC1)C(NC(=O)CCNC(N)=O)CS2(=O)=O C1(COC)CN(c2nnc(C(C)C)n2CCC#N)CC(C)O1 CC1CN(C(C2(F)C(C)(C)C2(C)C)=O)CCC1C(N1CCC1C(N)=O)=O CN1CCN(C(=O)Cn2cc(Br)c(Br)n2)CC1c1cn(C2CCCCO2)nn1 N1(C(CCNC(=O)OCC)=O)CCCCC1CN(C)C(C1CCC1C(C)(C)C)=O N1(C(C2CC(C)(NC(c3snc(C)c3N)=O)C2)=O)CC(C)(C)C2COCC12 c1(C(C)(C)C(=O)NCC2(NC(=O)COCCCF)CCOC2)ccc(F)c(F)c1 c1(NC(=O)CCOCC(F)F)cccc(NC(c2c(C(F)(F)F)coc2C)=O)c1 N1(C(CCCCCCC)=O)CC2(CCOCC2)CC1CNC(=O)C(F)CC C(=O)(C1Cc2ccccc21)N1CCC(NC(c2csc(Br)n2)=O)C12CC2 c1(C(=O)NCC(=O)NC(c2nc(CC)on2)C)c(COC)cnn1C C1(C(N2CCC(OC)C2C)=O)CC(N=[N+]=[N-])CN1C(c1ccnc(C)c1C)=O C1(NC(C2ON=C(CC)C2)=O)CN(C(=O)C2=CCCCCC2)C2CCCC12 c1(C(N2C(CNC(C3CC(C)(F)C3)=O)CC3(CC3)C2)=O)ccc2c(c1)NCC2 c1(C(N2CCN(C(C3=NNC(=O)C3)=O)CC2CF)=O)cc2n(c1)CCCNC2=O Cc1cc(C(N2CC3CCC2CN(C(=O)C(C)(C)F)C3)=O)ccc1[N+](=O)[O-] C12(NC(c3n(C)cnc3)=O)CCC1CN(C(=O)CSc1n[nH]c(=N)s1)C2 n1(-c2cc(C(=O)NC(CNC(COC(CC)C)=O)C3CC3)on2)c(C)ccc1C c1(C(C)=O)ccc(C(=O)NCCC(O)CNC(=O)CCCF)c(F)c1 c1(C(C(N2CCC(N(C(=O)CCCN(C)C)CC)CC2)=O)(C)O)ccc(F)cc1 Cc1nc2cc(C(N3C4CCC3CC(NC(=O)CC(C)C(F)(F)F)C4)=O)[nH]c2s1 C#CC1(NC(=O)CC(C)(C)N(C(=O)C(C#N)CC)C)CC2CCCC12 N1(C(CCN(C(C(C=C)CC)=O)CCO)=O)CC2CC1CN2C c1(NC(=O)NCC(C(=O)OC)(C)C)cc(NCC2(N(C)C)CC2)ccc1[N+](=O)[O-] N1(C(C(CCC)NC(N)=O)=O)CCN(C(c2nncn2CC)=O)CC12CCC2 Cc1cc(C)c(CC(=O)NCCCN2CCN(C(=O)CN(C3CCC3)C)CC2)s1 C(CCCCCCN(C)C)N(CC(=O)NCC(c1ccccc1)(C)C)CCC c1(C(N2CCC(CC=C)(NC(=O)CN(C)CCO)C2)=O)ccnc(F)c1N c1(CC(=O)N(C)CCNC(C2CCC(=O)N2C)=O)cc(Cl)cc(Cl)c1.C1(C)CC1 N1(Cc2ccn(CC)n2)CCN(C(c2ccccc2C2CC2)=O)CC1 C1(C(=O)NCCCN(C(c2cn(CC(F)F)cn2)=O)CC)CCCCC1F c1(NC)cnccc1C(=O)N(C)CCN(C(c1csnc1Br)=O)C(C)C N1(C(c2ccc(C)o2)=O)CCC(C(=O)Nc2nccc(C(F)F)c2F)C(O)C1 c1(N2CCC(CNC(CC)COC(F)(F)F)C2)cccc(OC(F)(F)F)c1 C1(CNC(C(C)OC)=O)CC(O)CN1C(c1c[nH]c(=N)s1)=O N1(C(c2c(C)nc(CC)o2)=O)CC(NC(=O)CN(C)C2CC2)C(C2CC2)C1 C1(NC(=O)OCCC=C)CCN(C(=O)C(C)CCOCC)CC1 c1(N2CCCCC(CC)C2)nc(=N)[nH]c(=NC(C)Cc2cccn2C)[nH]1 c1(C(=O)NCC2CC(O)(CNC(C(C=C)C)=O)C2)ccnc(C)c1C c1(Sc2ncnc3scc(C)c32)nc(O)c2ccccc2n1 c1(C(=O)NCCCCN(C(CCC(=C)Cl)=O)C)cc2c(s1)CCCCCC2 C(=O)(C(CNC(=O)C(C)CC1CCCC1)CC(C)C)N1C(C#C)CCCC1 N(C(=NCCC1(OC)CCC1)NC(C)C)CC(c1ccc(F)cc1)OC N1(C(CN2CCC(C)CC2)=O)CCN(C(C2CCC3CCC2O3)=O)C(CCO)C1 C(=O)(C(O)CC(N)=O)NCC(=O)NC(C)C(N1CCC(NC(=O)CC(F)(F)F)C1)=O c1(OC)cccc(Br)c1-n1cc(CN2CC3CC(C(=O)O)C2C3)nn1.C1(C)C(=O)N1 C1(CN(C(=O)CCc2cnc[nH]2)C)CCCC(NC(=O)C=C2CC2)C1 c1(OC)cccc(F)c1C(=O)NC1CCCC(N(C)C(C2CC(SC)C2)=O)C1 C(CN=C(NCc1cccc(C)c1Oc1ccc(Cl)cc1)NC1CC1)OC Cc1cnc2n1CCC(C(=O)NC1(CN(C(=O)Cn3cccnc3=O)C)CC1)C2 C1(C#N)(C(=O)NC(C)CNC(=O)C(C)Oc2cc(Cl)cc(Cl)c2)CC12CCCC2 CS(=O)c1cccc(C(N2CC=CC(NC(=O)C(F)(F)c3csc(Cl)c3)C2)=O)c1 C=CCCCCCC(=O)NCCN(C1CCCCC1)C(C1CC2C=CC1O2)=O c1(CNC(C2(C)CCCC2)c2nnnn2CCCOCC2CC2)ccc(Cl)cn1 S(=O)(=O)(c1cccc(=NCCc2ncc(C)o2)[nH]1)N(C)CC c1(C(N2CCN(c3c(C(C)C)c(F)ccc3)CC2)=O)[nH]nc2c(=O)n(C)cnc12 c1(C(C)C)ncc(C(N2CC(N(C(=O)C(C)CC3CCC3)C)C2)=O)o1 Cc1csc2cc(C(=O)NCCC3CCCN(C(=O)CC(C)C)CC3)[nH]c12 C1(N(C(=O)Cc2csnn2)C)CN(C(C2CCC(=O)O2)=O)CC1O N1(C(c2c(C)cn(C)c2)=O)CCC2(CC1)CC2C(=O)NCc1c(O)cccc1F c1(OC)ccnc(C(c2nnnn2C(C)C)NCCC2CCCO2)n1 C1(C(F)F)(NC(CC(C)SC)=O)CCN(C(=O)CCCCN2CCOCC2)C1 C1(NC(c2c(OCC)cccn2)=O)CN(C(=O)C(F)CC2CCC2)C2CCCC12 C1(CN2C(C(CC)C)CCC2)COC2(CCC2)CN1 c1(OC)ccc(CC(=O)NCC2CCCCN2C(c2ncoc2C2CC2)=O)cc1 CCC(C)CC(C(=O)NCCN1CCCOCC1)NC(=O)COc1ccccc1 C(=O)(C#CC1(C(F)(F)F)CC1)N1C(C)CC(CNC(c2cccnc2Cl)=O)C1 N1(c2nc(NC3C(C)C3C)nc3c2ccs3)CCOC2(CCC(C)(C)C2)C1 c1(CN(C(c2cn(C)c(-c3ccccc3)cc2=O)=O)CC)ccccc1[N+](=O)[O-] c1(C(=O)NC(CC)CNC(=O)C(C(C)C)n2cnnc2)ccc2[nH]nc(N)c2c1 c1(C(N(C2CCN(C(C3CC3C)=O)CC2)CC#C)=O)cc(C2CC2)nn1C C1(CNC(C=CCOC)=O)C2CCCC1N(C(=O)C1=CCCCO1)C2 n1(CC)ccc2cc(CNC3(CO)CCNC3)ccc12 N1(C(C2CC2C(=O)NCC#C)=O)CC(C)(NC(=O)CCC2CCC2)C1 c1(C(C)C)cc(CNC(=O)C(C)(C2CC2)N(C(=O)CCCC2CC2C)C)no1 CC1CN(C(C2(N(C)C)CC2)=O)CCC1N(C(=O)CSc1cccc(Cl)c1)C C1(CC=C)(C(=O)NC2COC(=O)C2)CN(C(C2CC3CC3C2)=O)C1 O(C=CC(=O)NCC(C1CC1)N(C(=O)Cc1ccsc1)C)CC C1(CC)CN(C(=O)COc2c(Cl)cccc2Cl)CCN1C(c1cc(Br)cs1)=O C#CCCN=C(NCC1(C)CCN(C)CC1)N1CCCC(COC(F)F)C1 C12(NC(c3ccnc(O)c3)=O)CCCC1N(C(=O)CC1COC(=O)C1)CC2 C1(C(N(C)Cc2c(C)nn(C)c2)=O)CC(NC(c2ccsc2C)=O)C12CCC2 C(=O)(CC1COc2cc(O)ccc21)N(CCCN(C(C(C(CC)O)C)=O)C)C C1(CCC)(NC(=O)CC(C)N(C)C)CCCN(C(=O)C(=Cc2cnc[nH]2)C)C1 CC1CC(C)CN(S(=O)(=O)N(C)C2CCCC(C(=O)O)C2)C1 C1(NC(CNC(CC)=O)=O)CCOC(C2CCN(C(c3ccc(C)[nH]3)=O)CC2)C1 N1(C(c2onc(C)c2C)=O)CC(NC(=O)COCCCC(C)C)C2(CCC2)C1 c1(C(C)C)ccc(C(=O)NC(CNC(=O)Cc2ccc(O)cc2)C(C)C)cc1F Cc1oc(C#N)cc1C(N1CCCC1(C)C(=O)NC1(C2CCCC2)CC1)=O C1(CNC(c2onc(CC)c2C)=O)C(C)CCCN1C(c1cnc(C(C)C)[nH]1)=O c1(C(N2C(C)CC(NC(=O)CCc3ccn(C)c3)C2)=O)cc2cnc(Cl)cc2s1 C1(C)(C(N(OC)Cc2ccccc2)=O)CN(C(c2oncc2C)=O)C(C)(C)C1 C1(CNC(Cc2cn(CC)nn2)=O)CC(C)(C)CN1C(=O)COC(F)F CN1CCC2CN(C(=O)CN(C(c3ccc([N+](=O)[O-])o3)=O)CC3CC3)CCC12 C1(CNC(C(c2ccc(F)c(F)c2)C)=O)CN(C(C2COCCO2)=O)C(C)(C)C1 C1(C(=O)NCC2(C)CN(C(=O)CC3=CCCCC3)CCO2)CCn2nncc2C1 C1(N(CCC)C(C2CC2c2cccc(O)c2)=O)CCN(C(=O)C(C)(C)C)CC1 S(=O)(=O)(c1cc(Br)sc1Br)NCc1c(C)ccc(N(C)C)c1 CCC(COC)C(=O)NCC(C)(C)CN(C)C(C1(C2CCCO2)CC1)=O c1(C(=O)NC(C(C)c2ccsc2)=O)cc(C(F)F)ccc1Cl.C12CCCN1C2 c1(C(N2CC(CC(C)NC(C3CC(=O)NC3(C)C)=O)C2)=O)cc(F)c(F)c(F)c1 N1(C(C2CSC2)=O)CCC(C2CCCN(C(=O)CNc3ccccc3Cl)C2)C1 O=S(=O)(c1ccc(Cl)cc1F)NC12CC(NCc3ncc(Br)cc3Br)(C1)C2 n1(C(C)(C)C)ncc(C(=O)NCC#CCNC(C2C3CCC(=O)C23)=O)c1Cl C(=O)(CCCCCC(C)C)NC(c1cccc(C)c1)CNC(CC1C(CC)C1)=O c1(CC(=O)OC)ccc(=NC(C)c2ccc(C(F)F)cc2)[nH]c1N1CCOCC1 CC1CC(NC(=O)CCC2CC2)CN1C(C1(C2CCCO2)CCC1)=O N1(CC#CC)CCCC(C2CCN(C(c3ccc(C(=O)N(C)C)cc3)=O)CC2)C1 Cc1cc(=NC2CC(Cc3ccccc3)C2)[nH]c(=NCCc2ccc(F)cc2)[nH]1 C1(NC(c2cc(C3CC3)cc(C3CC3)c2)=O)CC2CN(c3ncns3)CC2C1 c1(CC(=O)NC2C=CC(CNC(c3c(C)cn(C)n3)=O)C2)cccc2sccc12 C(=O)(C1=NN(C(C)C)C(=O)CC1)NCCC(C(C)C)NC(CC1CC(CC)C1)=O N1(C(C2(Br)C(C)(C)C2)=O)CCCC2(CCN(C(c3ncncc3Cl)=O)C2)C1 N1(C(c2ccc(C(C)C)cc2)=O)CCCCCC1C(F)F CCC(C)C(O)C(C)C(=O)NCCC1CCCCN1C(c1nnsc1N)=O C(=O)(C1c2c[nH]nc2CN1C(C1CC(OC(C)=O)C1)=O)N1CC(CC)OCC1C C(CCN(C)C)(C(=O)NCC1(O)CC1)NC(C(C)SC)=O C1(NC(c2ccc(CC)c(Cl)c2)=O)CC2CCC(C1)N2C(c1n[nH]cc1OC)=O C1(NC(C2CCC(C)CC2)=O)CCN(C(=O)CC2CC(F)(F)C2(F)F)C12CCC2 N1(C(=O)CCn2cncn2)CC2CC1CCN2C(c1ccc(C(O)CF)cc1)=O C1(C(=O)NCC(C)NC(=O)Cc2ccno2)(OC)CCC(C)CC1 C12(C(=O)NCCOC3CN(C(CC4C(C)CCC4)=O)C3)CC(C)(C1)OC2C C1(NC(C2C(C)(C)COCC2)=O)CCC2(CC1)CCN(C(=O)C(F)F)CC2 c1(OC)c(F)cc(NC(C2(C)CCCN(Cc3ccc(Br)cc3Cl)C2)=O)cc1F C1(C(=O)NC(COCC2CN(C(=O)OCC)C2)=O)(CC)OC2CCC1CC2 C12(C(=O)NCC3(O)CN(C(CCc4c(C)noc4Cl)=O)C3)CC(CO)(C1)OC2C c1(CC)snc(C)c1C(=O)NCC1CC(CNC(C2(CC(=O)NC)CC2)=O)CO1 C#CCC(C)(C)C(=O)N(C1CC(NC(=O)C(C)Cc2ccco2)C1)C C1(N(C(=O)COc2cccc(F)n2)C)CCCN(C(=O)C=C(C)C(C)(C)C)C1 Nc1cc(F)c(Cl)cc1C(=O)NCC1CC(NC(C2CC23CCCC3)=O)C1 C(=O)(C(C)(C)CC(F)(F)F)NCC(C(C)C)NC(=O)CC12CCC(=O)N1CCC2 C1(C(N2CC(NC(CC(C)C(F)F)=O)(CN(C)C)C2)=O)CC2(C1)NC(=O)NC2=O Cc1nc(C)c(C(N2CCC2CNC(c2cnc(C(F)F)cn2)=O)=O)nc1C C(=O)(C1=CS(=O)CCC1)NC(CN(C(c1n(CC)nc(C)c1)=O)CC)CC CC1(CS(=O)(=O)NCC(C2CC2)C2CC2)CCCC(F)(F)C1 N1(C(CCn2c(C)csc2=O)=O)CC2(C1)CN(C(=O)CC1CCOC(C)(C)C1)C2 N1(C(c2c[nH]cc2C2CC2)=O)CCN(C(C2CCS2(=O)=O)=O)C2(CCC2)C1 CC1CCC(NC(c2ccnc(F)c2Cl)=O)CN1C(c1cc(Cl)nnc1Cl)=O C1(C(N2CC(OC)C(F)C2)=O)CCCN(C(=O)C(F)C(C)(F)F)CC1 C1(NC(CCCC#C)=O)CC2(C1)CN(C(c1cnc(C(C)(C)C)nc1)=O)C2 C(C(C)(O)C(=O)NC1CCCC1CN(C)C(c1cn(C2CC2)cn1)=O)OC NS(=O)(=O)N1CC(C(N2CCOC(CCNC(C3OCCCO3)=O)C2)=O)C1 O=C1CCC(C(=O)NC2CC(CCC(=O)NCc3ccncc3)C2)O1 C(=O)(C(C(C)(C)C)NC(c1n[nH]cc1Cl)=O)NCC(C)Cn1cccn1 C1(C(=O)NC2(CNC(C(C)(C)F)=O)CCOCC2)CC2CCCCCC12 c1(CC)cc(F)ccc1C(=O)NC1CCC(C)(CNC(=O)C=CCCC(C)C)C1 c1(NC(c2nnnn2CC2CCOCC2)(C2CCCO2)C)cccc(F)c1 C1(OCC(N2CCC(O)(CNC(C(F)OC)=O)C2)=O)CCC(F)(F)CC1 Cc1cc(C)n2ccc(C(=O)NCC3C(C)CCN3C(=O)CC(C)(C)O)c2n1 c1(OC)ccc(C(N2CCC(NC(C3(C)CCCN3C)=O)C(F)C2)=O)nc1OC Cc1nc2ccc(C(N3CC(NC(=O)COCC4CC4)C(C4CC4)C3)=O)cc2s1 CCC(C)CC(C(=O)NC1COCCOC1)NC(=O)C#CC(C)(C)O N(C(=NCCC(O)c1ccc(C)o1)N1CCN(Cc2ccnn2C)CC1)C(CC)C CC#CCCCC(=O)N1CC=CC1(C(N1CCC(C)=C(C)C1)=O)COC C1(OC(CC)C(=O)c2ccccc2)(CCOOC2(C)CC2)CCCCC1.C(C)(=O)NC c1(C(N2CC(CNC(c3cnn(C)n3)=O)OCC2)=O)ccc2cc[nH]c2c1F c1(N(C(=O)CC2CCC(=O)N2)CCNC(CC2(OC)CC2)=O)ccc(Cl)nn1 N1(C(C2CCCN(CC)C2)=O)C(C(=O)NCc2ccc[nH]2)C2CC(O)C1C2 Cc1cccc(SCC(=O)NC2(C)CCOC2)c1.C(C)(C)(C(F)(F)F)NC(=O)COC c1(C(=O)NC2CCCN(c3nc(O)cc(C)n3)C2)c(F)ccc2ccoc12 Nc1c(C(=O)NCC2CCN(C(C3CCC3(F)F)=O)C2)cccc1C(F)(F)F C1(OC)CC2CC(C(=O)OCc3ccc(C(C)C)c(C)c3)CC2C1 C12CCCN(C1)C2=O.C(C)(C)(C(=O)NCC(C1CCC1)OC)NC(=O)NCC=C CCCC(C)CC(=O)NCC1CCCC(CNC(c2csc([N+](=O)[O-])c2)=O)C1 c1(C(=O)Nc2cn(Cc3ccc(OC)cc3)nc2)ccc(C)c(Br)c1OC c1(CC(N2CC(C)(NC(=O)CC(O)c3ccccc3)C2)=O)cc2ccccc2s1 C1(NC(c2cc(C)cc(C)c2)=O)CCN(C(=O)Cc2sc(S)nc2C)CC1(C)C c1(C(N2CCCCC(CNC(CC3CC(=C)C3)=O)C2)=O)nccc2ccccc12 c1(NC)cccc(C(=O)NC(C(=O)NCC2(C)CC3CC3C2)C(C)OC)n1 C(C(C(=O)N(C1CC1(C)C)C)NC(=O)CCc1nncn1C)OC(C)C c1(CC)cc(C(=O)N(CCO)Cc2ccccc2OC)c(C)o1 C(CNC(c1ncc(C(F)(F)F)s1)=O)(CC(C)C)NC(C(CC)n1cccn1)=O c1(C(N2CCC(O)(CNC(C3(OC)CCSCC3)=O)C2)=O)cc(N)c(C)cc1C C1(NC(c2ccc(CC)[nH]2)=O)CCCC(NC(C2(CCO)CC2)=O)CC1 C1(O)(C(=O)NCC2N(C(CSCc3n[nH]c(=N)s3)=O)CC2)CN2CCC1CC2 CN1N=CC(CC(=O)NCC2CC(NC(C3CCC(C)CC3)=O)C2)C1=O N1(c2ccc(S(=O)(=O)NCC3(CC#N)CC3)cn2)CCc2ccncc2C1 Cc1ncc(Br)cc1C(=O)NCC1CN(C(c2ccc[nH]2)=O)CCC1C N1(C(C(CC)(C)C)=O)CCC2(CC1)CN(C(C1COC3(CCC3)CO1)=O)C2 Cc1cnc(C=CC(=O)NCC2CC(C)N(C(c3cccc(C(F)F)n3)=O)C2)[nH]1 c1(C(N2CC(N(C(c3cc(C(C)=O)on3)=O)C)C2)=O)cc2c(C)nn(C)c2s1 c1(C(N(CCCn2cc(CC3(CO)CCC3)nn2)C)=O)c(F)cc(Cl)cc1F Cc1ncc(C(N2CC(O)(C(F)C(N3CC(O)(C(C)C)C3)=O)C2)=O)n1C C=CC(C)C(=O)N1CCCC1CCCNC(=O)CC1CCOC1=O c1(C(N(C2CCCN(C(C=COCC)=O)C2)CCO)=O)ccc(C(F)F)cc1Cl C1(SCC)CCC(NC(=O)NCC(Cc2ccccc2)NC(=O)OC(C)(C)C)O1.C C1(NC(C(C)SCCCC)=O)CN(C(=O)Cc2c[nH]c(=N)nc2O)C2CCCC12 C1(C(=O)NCc2scc(C(=O)NCc3cnccc3Cl)n2)CC2(CCC2)C1 N1(C(C(C(C)C)SCC)=O)CCC(NC(c2[nH]c(O)nc2C)=O)C(CO)C1 C1(NC(C2N(OCC)CC2)=O)CC(F)(CNC(=O)CC=C(C)C)C1 C1(C(=O)OC)N(C(c2cc(C)c(=O)n(C)c2)=O)CCOC1(C)C CN1C(=O)COCC1CNC(C1CC(N(C)C(c2cc(Cl)no2)=O)C1)=O N1(C(CC(CCC)C)=O)CCC(C)C(NC(=O)CC2CC3CCC2O3)C1C C1(C(=O)NC2CC(CC)(CC)C2)C2CCN(C(=O)C=CCO)CC12 C1(CC)CC(C)CN(C(C2CCCCCC2NC(=O)Cc2cnns2)=O)C1 Cn1cc(CN2CCN(CC3CCCO3)CC2)c(C(F)(F)C(F)(F)F)n1 c1(OC)ccc(C(=O)NC2CN(C(=O)CCC(N)=O)CC2n2ccnn2)cc1O c1(C(=O)NCC(C)(C(C)C)NC(CC(=C)C)=O)ccc(O)c(F)c1F Cc1nc2cc(C(N3CCC(CNC(=O)C4=NNC(=O)C4)C3)=O)cc(Br)c2[nH]1 C#CC(CCC)NC(=O)NC1C(OC(C)(C)C)CC1OC c1(C(C(N2CCN(C(COC)=O)CC2COC)=O)(F)F)nc2ccccc2s1 c1(CN(CCCC(F)(F)F)c2cc(-c3ncccn3)ncn2)cc(F)cc(Br)c1 N1(Cc2cccc(OCC)c2)CCC(NC2CCCC(CCC(=O)O)C2)CC1C CC1(C)C(CC(=O)NCC(C2CC2)C2CC2)CCN1C(=O)CSCC(F)F N1(C(C2(CCC=C)CC2)=O)CCC(O)(CCNC(=O)CCC(C)(C)C)C1 c1(CN(CCC(Cc2ccccc2)COC)CC)cccc(CNC(C)C)c1 C1(CN(C(=O)C=C2CCOCC2)C)C2CN(C(=O)CC(C)(C)O)CC12 CC(CCCC(=O)NCCC1CC(O)C1)NC(C1CC(=C2CC2)C1)=O C1(CC)CCC(C(=O)NCCN(C(C2CCCCC2O)=O)C(C)C)CC1 C#CCC(C)(C(=O)NCCN1C(=O)CNC1=O)NC(=O)C(CC(C)C)OC C(=O)(CCCCCn1cc(-c2cc(F)ccc2OC)nn1)OCCSCC c1(C(N2C(CNC(c3ncn(CC)c3)=O)CC(F)C2)=O)ccc(C(C)C)nc1C C1(NC(c2c(C)cc[nH]2)=O)CC2CC(NC(=O)C(c3cccnc3)O)CC12 CCCC(C)(CC)C(=O)N(CCCOCCNC(c1ccoc1C(C)C)=O)C N1(C(CC(C=C)CC)=O)CCC(NC(=O)CCc2nccn2C)C(F)(F)CC1 c1(CC)nn(C)cc1C(N1CC(CNC(=O)CC(C)(C)O)CC1C)=O C1(C2(NC(C3CC34CC4)=O)CC2)CCCCN1C(c1ccns1)=O C#CCCCC(C(=O)N(C1COC1)Cc1ccco1)N1CCOCC1(C)C C1(C(N2CCC(C#C)C2)=O)CCN(C(=O)CCNC(=O)OC)CCO1 C1(NC(CC2C(NC(c3cnc(C)s3)=O)CCCC2)=O)CCC(C2CC2)C1 C1(C(=O)NC23CC(F)(C2)C3)C2CCCC2CN1C(C1CCCCC1)=O C1(O)(CC2CN(C(=O)OC(C)(C)C)C2)CCC(NC23CC2CN(C)C3)CC1 C1(C(=O)NCC#CC)CN(C(=O)CC2CCOC2=O)CC1OC N1(C(C(=O)NCC(=C)C)c2ccns2)CCC(C(=O)OCC)C1 N1(C(CCOCC#C)=O)CC(OC)CC(NC(c2cc(C)nc(C)c2)=O)C1 N1(C(C2C(C(=O)OC)CC2)=O)CCOCC1CCNC(c1cncn1C)=O CC1(C)COCC(C(=O)NCC2(NC(=O)CC34COC(C)(C3)C4)CC2)O1 N1(C(C2=NOC(C)C2)=O)CC(NC(=O)COC(F)(F)F)C2(CCS(=O)(=O)CC2)C1 c1(OC)cnc(C(=O)NCCCN(C(=O)CCN2CCCC2=O)C)nc1 c1(SC)nn(C)cc1C(=O)NCCCC(C)(C)NC(=O)COc1ccsn1 C1(N2C(=O)CC2)CCCOCC1.c1(CN(C2CCC2CF)CC)ccc(F)cc1 C(C(CC(F)(F)F)NC(C1CC(CF)C1)=O)NC(=O)Cc1ccc(Cl)s1 Cc1cccnc1CC(N1CCC(N(C(=O)C(C)Sc2ccc(Cl)cc2)C)C1)=O C(=O)(C1=NNC(=O)C1)NC1CC(O)(CNC(c2cnc(CCC)s2)=O)C1 C1(C)(NC(c2ccc(OC)s2)=O)CCC(NC(=O)CC2(C(F)(F)F)CC2)CC1 C=CC1(CC(N2CCCCC2CCNC(C2OCCO2)=O)=O)CCOCC1 C12(NC(CC(C)SC)=O)CC3CCC(C1C2)N3C(=O)CSCc1cccnc1 c1(C(N2CCOCC(NC(C(CC=CC)C)=O)C2)=O)cc2n(n1)CCCNC2=O CCC(CC)C(=O)N1CCC(Cc2cn(Cn3nc(C)cc3C)nn2)C1 C1(C(N2C3CC(NC(C4N(C(C)C)C(=O)CC4)=O)(C3)C2)=O)CCc2nccn2C1 N1(C(C=CC(CC)C)=O)CCC2(CC1)CCN(C(C1OCC3CCCCC13)=O)C2 N1(C(C2CC(NC(=O)CC3CC(C4CC4)C3)C2)=O)CCN2CC(O)CC2C1 C(=O)(N=c1ccn(-c2nccc(C)n2)[nH]1)C1C(Oc2c(OC)cc(C)cc2)C1 C1(C(=O)NC2COCCO2)CC2CC(C1)N(C(=O)COC1CCOCC1)C2 C1(C(N2C(C(C)NC(=O)CC(C)(C)C)CCC2)=O)COc2ccc(F)cc2C1 N1(C(CCOCCC)=O)CCN(C(C2CC2CC(C)C)=O)C(CF)C1 CCC(C)(C(=O)N1CCC(NC(=O)C(C)Sc2ccc(C)cc2)C1)C(F)F CC(C)C(C#N)C(=O)N1CC=CC1C(N1CCC2(CC1)N=N2)=O C1(CCC)(NC(=O)CNC(c2ncccn2)=O)CCN(C(c2cncs2)=O)CC1 N1(C(CCCOC)=O)CC(NC(=O)C(N2CCCCCC2)C)CCC1C CCC(C(=O)N1CC(C(=O)NCC(C)=CCO)C(F)C1)C(C)(C)CC C1(C(=O)NC(c2ccc(CNC(=O)C3=CSCS3)cc2)C)CC2(CCCO2)C1 Cc1cc(C)n2ncc(C(=O)NCCCc3cn(Cc4ccccn4)nn3)c2n1 N1(C(C2(CC(C)C)COC2)=O)CC2(CC(NC(=O)C=Cc3cccnc3)CO2)C1 [N-]=[N+]=Nc1ccccc1C(N1CC2CCC(NC(C3CNC(=O)N3)=O)CC2C1)=O N1(C(Cn2ncn(C)c2=O)=O)CC2CN(C(=O)Cc3ccco3)CC2(C)C1 C1(C(=O)NCC2(F)CC(CNC(=O)OC(C)(C)C)C2)CCC(C)CN1C(=O)C1CC1 N1(C(C2(OC)CCC2)=O)CCN(C(=O)C(C2(O)CCCCC2)O)CC1 c1(CC(=O)NCC)ccc(C)c(OC(F)F)c1.C1(C)C(C)(C)N(CC)CC(=O)N1 C1(C(=O)NCCC=C(C)C)CNC(=O)CN1C(=O)C=CC1CC1 c1(SC)nn(C)cc1C(=O)NC(C)(CNC(=O)COc1ccn(C)n1)CO N#CC1(C(N2CC(CNC(C3COCCOC3)=O)C(O)C2)=O)CCSCC1 C1(NC(C(n2ccc(C)n2)C)=O)CC(F)CN(C(c2ccc(C(C)(C)C)o2)=O)C1 c1(NC(C2(F)CCN(C(C(C=C)O)=O)C2)=O)cccc2c1OCO2 N1(C(=O)NC(C)C(C2CCCCC2)C)Cc2cc(Cl)nc(Cl)c2C1 c1(C(=O)NCC(C(=O)OC)Cc2ccoc2)ccc(OC(F)(F)F)c(F)c1 c1(CC)cccc(C(=O)N(C2CN(C(c3cc(CC(C)C)c[nH]3)=O)CC2O)C)n1 N1(C(c2ncc(OC)nc2)=O)CCN(C(c2ccc(F)c(O)c2F)=O)C2(CC2)C1 C(C(=O)N1CCCc2ccnn21)OC1CN(C(c2c(C)cc(C#N)cc2)=O)C1 N1(C(C2(c3cc(C)no3)CC2)=O)CCC(NC(=O)CC(O)C(C)C)C(O)C1 N1(C(COCC)=O)CC(C)(C)C1C1CCN(C(C2(C)CS(=O)(=O)C2)=O)CC1 C1(CNC(c2c(C)c[nH]n2)=O)CC(C)N(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 c1(C(N2CC(N(C)C(c3sncc3Br)=O)C2)=O)coc(C(N)=O)c1 C1(CC(N2CCCC(Nc3ccccc3)C2)=O)CC2(CCN(CCF)CC2)CO1 c1(OC)ccc(C(=O)C(=O)NCC2CCCCC2NC(=O)C(C2CC2)SC)cc1 C1(CNC(CSCCCC)=O)CN(C(c2nc(Cl)cs2)=O)C2CCN1C2 N1(C(CCn2ccc(C)n2)=O)CCC(C)(C)CC1C(=O)N(CC(F)Cl)C C1(CCNC(C(C=C)O)=O)CCCCN1C(=O)CNc1cnn(C)c1 C1(C(=O)NCC2(C(N3CC=CCC3)=O)CC2)CC2C=CC1CC2 c1(CNC(CCCCC)(C)c2nnnn2C2COC2)cc2c(Cl)n[nH]c2cc1F c1(C(=O)NCCCC(C)NC(c2cnn(C)n2)=O)cn(C)c(=O)cn1 C1(C)(CC)CCC(C(=O)NC2CCOC2C(=O)NC2CC3C=CC2O3)O1 c1(OC)cc(=NC(=O)CNC(C2CCC(=O)C(C)C2)=O)[nH]n1C C1(C(N(CCCC(CC)CC)C)=O)C2CCCC2CN1C(c1cnc(C)n1C)=O C(c1cncs1)=CC(=O)NC(C(=O)N(CCCN(C)C)CCC)C1(C)CC1 C1(NC(CC2(C=C)CN(C(c3cc(C)c[nH]3)=O)C2)=O)(CO)CC2CCC1C2 O=S(=O)(c1nc(N2CCC(C(F)F)C2)ccc1Br)NCC1(CO)CCCC1 S(=O)(=O)(c1cccc(=NCCCCCC(C)C)[nH]1)NCCOc1cc(C)nn1C c1(C(=O)NC2CC(CNC(C(CC#C)O)=O)C2)ccc2ncc(Br)cc2c1 c1(C(N2CCC(NC(CS(CCC)(=O)=O)=O)C2)=O)csc2ncnc(O)c12 C1(C(CC)NC(=O)C=CCNC(=O)CSC(F)F)CCOC1 C1(C(N2CC(CCC)C2)=O)CCCCC1(C)NC(c1cc(Cl)n(C)n1)=O Cc1cc(NC(=O)CCN(C(C2(C)CCCC2C)=O)C2CC2)cc(CO)c1 C12(CNC(=O)NCc3cccc(C(N)=O)c3Cl)CCCN1CCC2 c1(CC(N2CCC(CCNC(C3CC(OC(F)F)C3)=O)CC2)=O)cccnc1O CCC(C)(C)C(O)C(=O)N(CCC(=O)N1CC(C2CC2)(OC)C1)OC C1(C(=O)OCC2CCCC2NC2CC2)CC2CC(F)(F)CC(C1)C2(F)F C1(NC(c2cn(CC)nc2)=O)CC1C1CCCN(C(c2cocc2C)=O)C1 CC1CN(C(=O)C(C)O)CCCN1C(=O)CNC(c1cc2c(s1)CCOC2)=O N1(C(C(CC)=CCCC)=O)CCC2CCN(C(c3conc3C)=O)CC12 CC1CN(C(C23CCC(CC2)OC3)=O)CCN1C(C1CC1C(C)(F)F)=O C1(CCNC(c2n(C(C)C)ccn2)=O)CCN(C(=O)C(C)(C)C#N)CCC1(F)F C1(CNC(=O)CSC(F)(F)F)CCC(NC(c2cn(-c3ccccc3)cn2)=O)C1 CCCC(CNC(C1CC1(Cl)Cl)=O)C(=O)NCCOCCO C1(C(=O)NC(CN(C(c2csc(C(C)C)n2)=O)CC)C)CCCCCS1(=O)=O N1(C(c2ccc(CNC(c3c(C)ccn3C)=O)s2)=O)CCSCCC1C C(=O)(CCN(OC)C(=O)C1(C(=O)OC)CC(O)C1)N1CCC(C#C)C1 c1(N(C)CC2CCC(C)(C)CC2)nc(NCc2cc[nH]n2)c2ncsc2n1 N1(C(COC(C)C)=O)CC(NC(=O)CN2CCCCCC2)C(c2ccccc2)C1 C1(NC(c2ccc[nH]2)=O)CCCCC1CNC(C1(C(F)F)CCC1)=O C(C(CC1CC1)C(=O)NC(CN(C)C)CO)NC(C1C(COC)CC1)=O c1(CC)ncc(C(=O)NCC(C2CC2)NC(=O)CCC#N)[nH]1 c1(C(=O)NCCc2c(C)n(C)nc2)cc(F)c(Cl)c(F)c1 C(C(C)(C)C(=O)NC1CCC(C(=O)NCCN2CCC(CO)C2)C1)N(C)C C1(CNC(=O)CC2CCSCC2)CCN(C(=O)CCCF)CC1C1CC1 CCCCCCC(F)C(=O)NC1CC(CNC(C2CC2CF)=O)C1 C(C)(CCC(F)(F)F)NC(c1c(CNC(CCC#C)=O)cco1)=O C(=O)(C1c2ccccc2CN1S(=O)(=O)C1CCOCC1)NC(C)CN(C)C O=C1CCC(CC(=O)NC2CCOC2C(=O)NC(c2ncccn2)C2CC2)N1 n1(CC(=O)N(C)Cc2ccc(-c3nn[nH]n3)cc2Cl)ccc(=O)n(C)c1=O N1(C(c2c(C)c(F)cnc2)=O)CC(C2CN(C(c3c(F)ccc(F)c3Cl)=O)C2)C1 C(CCCN(C(=O)C=CCC1(NC(C2CC2C2CCCO2)=O)CCC1)C)N(C)C C#CC1(NC(=O)CC2CCN(C(=O)CC(=O)OCC)C2(C)C)CC2CCCC12 C=CCCC(CC(C)C)C(=O)N1CCC(CC)(NC(c2cc(CO)on2)=O)CC1 c1(CC(C)C)nc(C(=O)N(C2CN(C(=O)Cc3nncs3)C2)C)cs1 C(=O)(C(C)(C)C(=O)NC1CCC1CNC(=O)CCCc1ccc(C)c(C)c1)OC N(C(=NCCNC(C1(CSc2cccnc2)CC1)=O)NCC(F)(F)Cl)CC N1(C(CNS(CC)(=O)=O)=O)CC2(CC2)CC1CNC(C1CC(OC(F)(F)F)C1)=O N1(C(C2(C)CC2F)=O)CCC2(CC1)CN(C(c1ccc(Br)c(F)c1)=O)C2 C(=O)(C(F)C(C)C)N(CC(c1ccc(C)cc1)(NCC)SC)C.c12ccc(s1)C2 C(=O)(CC(C)(C(F)F)N(C)C)N1CC(C)C(NC(c2cnnn2C2CC2)=O)C1 N1(C(C=CCC)=O)CCn2nc(CNC(=O)C(CC3CCCCC3)CC)cc2C1 C1(C)(C(N(CC(C)N(C(=O)CCCSc2ccccc2)C)C)=O)CC(=O)N(C)C1 c1(-n2c(Cc3n(CC)nnc3)nc(C(C)OC)n2)ccc(F)c(Br)c1.C(C)C N1(C(c2ccncc2Cl)=O)CC(CO)C2(C1)CN(C(C13CCC(O)C1CC3)=O)C2 c1(CC(=O)NC2(C3CCN(C(=O)CC4=CCCC4)C3)CC2)n[nH]c2ccccc12 Cn1ccc(SCCNC(=O)Nc2scnc2Cl)c1 N1(C(C2(NC(c3c(C)noc3)=O)CCCC2C)=O)C2CCC1CN(C)C2 N1(C(C(C2CCC2)OC)=O)CC2=C(C1)CN(C(C1CCC1C(C)(C)C)=O)C2 c1(OC)ccc(F)c(C(=O)NCC2CN(C(=O)CCS(C)=O)C2)c1N Cc1nc2c([nH]1)C(C(=O)NC1CN(C(=O)C(F)=CCCF)CC1C)CCC2 c1(CC(=O)NCCC(C)CCNC(=O)Cn2ncccc2=O)cc(F)c(F)cc1F c1(C(N2CCC(OC(C)C)CC2)C(=O)NC(CC)C)ccc(C)nn1 N1(C(CC=CCC)=O)CCCC(C)(NC(C2CCN2C2CCCC2)=O)C1 CN1CCOC(C(=O)NC2(CNC(C3(C(F)(F)F)CCCC3)=O)CC2)C1 c1(CC)ncc(C(=O)NC2(C(=O)NC(C)Cc3ccco3)CC(CO)C2)o1 N1(C(C2C=CCN(C(C3(OCC)CCOC3)=O)C2)=O)CCCC(F)CC1 C1(C(=O)NCC2CC(NC(=O)CCN3CCCC3=O)C2)CCC=CCCC1 C(=O)(C(CC(F)F)NC(=O)C(C)N=[N+]=[N-])NC1CC(C)(C(=O)OC)C1 C1(C(C)C)Oc2ccc(C(N3CCCN(C(=O)C(F)F)CCC3)=O)cc2NC1=O CC(C)(C(=O)NCCn1cc(C(=O)NC2CC23CCC3)cn1)C1CCOC1 C1(C(=O)NCCC(=O)NCCCC)CCCN(C(c2c[nH]c(=S)cn2)=O)C1 C(=O)(CS(=O)(=O)CC(C)C)NCC#CCNC(C(c1ccc(OC)cc1C)C)=O c1(C(C(=O)N(CCC(=O)NCC=C=C)CC)(F)F)ccc(F)cc1 C1(C(=O)NCCN(C)C(C2CN3CCCC2C3)=O)CCC(C)(C)OC1 N1(C(CCNS(CC)(=O)=O)=O)CCCCC(NC(=O)CCC(C)(C)N(C)C)C1 C1(NC(=O)CCCN=[N+]=[N-])CC12CCC(NC(c1c(CC)nccn1)=O)CC2 C1(CC)CN(C(=O)CCc2ccon2)CCN1C(=O)C(N1CCN(C)CC1)C c1(CCC)nc(-c2cn(C(C)(C)C)nc2Br)n(CCC)n1 C1(C(N2CCC(CN(C)C)C2)=O)CCN(C(c2ccc(F)s2)=O)C1(C)C C1(CNC(c2sccc2C2CC2)=O)CC2(CC(NC(C3C4COCC34)=O)C2)C1 CCCCCCCNC(=O)CC1CCCN(C(C2(C(C)(F)F)CC2)=O)C1 C1(NC(CSCCC(C)C)=O)CCC(NC(=O)Cc2n[nH]c(=N)s2)C1 C(=O)(C1=CCCC1)N1CC(Cn2cc(CNC(c3ccc(CC)o3)=O)nn2)C1 C(C)(C)(CC(C)(C)C)NC(CCC(C)NC(c1ccc(O)cc1F)=O)=O c1(C(CC)C(=O)NCC23CC(C(C)(F)F)(C2)C3)c(C)noc1C C(=O)(C(CCCCC)CCCCC)NCC1N(C(C(C)=CC)=O)CCOC1 c1(C(=O)NCC2OCCCN(C(C(C)=CC)=O)C2)cc(O)nc2[nH]c(=N)ccc12 Cc1n[nH]c(C)c1C(N1CCCC(CNC(=O)C=Cc2cc(C(N)=O)co2)C1)=O N1(C(c2cc(C)ns2)=O)CCC=C(C(=O)N2CCC(C(=O)N(C)C)C2)C1 N1(C(C(CC=C)OC)=O)CCCC2(CCCN2C(=O)CC2(OC(C)=O)CCC2)C1 C12(CC(=O)NC3CC3NC(=O)CSc3nnc(S)s3)CCC(CC1)OC2 c1(C(=O)NCCC2N(C(C3C(C)OCCO3)=O)CCC2)cccc2ncnn12 c1(C(=O)NCCN(C(C2CC(C)C2(C)C)=O)CC)cccc(CO)n1 C(CN=c1cc(C)nc(SC(F)F)[nH]1)C1CCCN(c2nc(O)cc(C)n2)C1 CCC(C)CC(C)C(=O)N1CCOCC1c1cn(-c2cccc(C)c2C)nn1 N1(C(COC(C)C)=O)CC(CNC(c2cc(Cl)no2)=O)C(F)(F)C1 CCC1=C(C(=O)N2CCC(NC(=O)Cc3nonc3C)C23CCC3)CCCO1 c1(C(=O)NC2CCC(C)(CNC(C3CC(C#C)(O)C3)=O)C2)cc2sc(C)cc2s1 CC12CCC(C(=O)NC3CCCC3CNC(C3CCC4(CC4)C3)=O)(CO1)C2 CC(C)(C)C(C#N)C(=O)NC1(C(N2CCC(F)C(F)C2)=O)CCC1 N1(CCCn2cc(C(CC)N(C)C)nn2)CCCCC1C N1(CC(N2CC(O)(CNC(C(c3scc(C)n3)C)=O)C2)=O)CCN(C(C)C)CC1 CC1(CO)CN(Cc2sccc2Cl)CC1C(=O)O c1(OC)cn(C)c(C(=O)Nc2nc(C(N)=O)c(Br)nc2Br)cc1=O CON=CC(=O)N(C1CCN(C(C2CC2C(=O)NCCO)=O)C1)CCO C1(C(=O)NCC(C)CN(C)C(c2cc(Br)no2)=O)CCC(=O)N1 C(C(=O)N=c1ccn(CCC)[nH]1)(C1CC1)NC(CC(C=C)CCC)=O C(=O)(N1CCS(=O)(=O)CCO1)C1(C(=O)OCCOCCOC)CCC1 C1(CC=O)COCCN1C(c1ccc(C2CC2)cc1)=O.c1(CCO)nc[nH]n1 Cc1cc(COCC(=O)N(CC(=O)NC2COCC2OC(C)C)C)on1 Cc1cc(C(=O)NC(C)CC(C)NC(C2CCCCO2)=O)nnc1C C(CCC(C)CC(=O)N(CC(C)(C)NC(=O)CCC1CCCOC1)C)=C(C)C CCC(CC(=O)N1CCC(C(=O)NCCC2CCCCC2)CC1)SC c1(C(=O)OC)ccc2c(c1)CCN(N1CCC(C(F)(F)CO)C1)CC2 CCCC(CNC(=O)COCCCOC)C(=O)NC(c1ccnn1C)CO [N-]=[N+]=NCCCC(=O)N1CCOCCC1C(N1CCC(OCC(N)=O)C1)=O C(=O)(C1=CC2(CCOCC2)C1)N1CC(CC(C)(C)C)N(C(C2CCCO2)=O)CC1 C(N=c1[nH]c2c(F)cccc2o1)C1OCCCN(C(C(C2CCC2)OCC)=O)C1 c1(C2C(NC(=O)NC(c3ccc(F)cn3)C)C2)ccccc1F C(=O)(C#CC1CCOC1)N(CCN(C(=O)CC1COC(C)(C)CO1)C)C c1(C(=O)NCC2CCC(NC(c3cnc(CC)[nH]3)=O)CC2)occ2c1CCOC2 c1(C(=O)OCCCC2CCOC2)ccc(F)cc1OC(F)F C1(C(=O)NC2C3C=CC(C3)C2CO)C2Cc3cc(Cl)ccc3C12 C1(CNC(C(C)N(C(C(C)OCCN(C)C)=O)C)=O)CCCC2(CC2)C1 C1(C(N2CCCC(N(C)C)C2)=O)CCN(C(=O)CCc2cnccn2)C(C)(C)C1 N1(C(CCc2cnc(C)o2)=O)CCCC(O)(CNC(=O)CC(C)(C)C(F)F)CC1 C1(C(=O)NCCOC(C)=O)CC2(CCO1)CC2.C12C=CCN(C1)C2=O C1(C(=O)NC2(C)CCCN(C(C3CC4CCC(C3)S4)=O)C2)Cc2cccnc2C1 C(CCNC(=O)Cc1conc1C)(C(C)C)NC(Cc1cn(CC)nc1)=O c1(CC(=O)NC2C(CNC(C=CCC)=O)CC2)c(OC)cc(Br)cc1OC CCCC(C)(O)CNC(=O)C(C1CN(C(=O)CC2CC(=O)NC2=O)C1)OC C1(NC(c2[nH]c(C)c(-c3ccccc3)c2)=O)CCC12CCN(C(=O)C(C)C)CC2 c1(C(N(C)CC2(CNC(C(C)C(C)(F)F)=O)CC2)=O)cc2cccnn2n1 C(c1c(Cl)cccc1Cl)=CC(N1CCC(O)(CNC(C2(C)CCOC2)=O)CC1)=O C(=O)(CC(O)CNC(C1CN(C(=O)COC(C)=O)CCO1)=O)OC C1(NC(C(CNC(=O)OC(C)(C)C)O)=O)CC(F)(F)CC1CNC(=O)CC(C)F c1(C(N2C3C(NC(C4CC(=O)NC4)=O)(CCC3)CC2)=O)cc2ccccc2cn1 N1(C(C2(C)CC=CC2)=O)C2CCC1CC(C(=O)NCCC(C)(O)C1CC1)C2 c1(N2CCC3(C(C(=O)NCC(=O)NC4CC4)C3)CC2)ncc2cccc(Br)c2n1 N1(C(Cn2c(C)cc(C)n2)=O)CC2CC(CN3Cc4cncnc4C3)CC2C1 Cc1oc(Br)cc1C(=O)NCCNC(=O)C(C)NC(=O)CC1CCCCC1 c1(C(N2CCC(NC(C3CC3c3ccccc3)=O)C2)=O)ccc2nc(O)sc2c1 Cc1cccc(C)c1C(O)C(=O)NCCCC(C)NC(C1CCCCNC1=O)=O CC(C)(CO)C(CO)NC(C1(NC(=O)C2=CCC2)CC(O)C1)=O c1(OCC)nc(C)ccc1C(=O)NC1CCCCC1NC(c1nc(C)oc1C)=O C1(NC(c2c(C)nn[nH]2)=O)CCC(C)(CNC(=O)CC2CC=CC2)C1 c1(NC(N2CCCC(C(=O)Nc3c(C)nsc3)CC2)=O)cnc2ccc(F)cn12 c1(CC(C(=O)NC2N(C(C=CCOC)=O)CCSC2)(C)C)ccc(C)c(C)c1 CC1=NN(C)C(=O)C1CC(N1CC(O)(CNC(C2(CCO)CC2)=O)C1)=O C1(NC(C(CC)OCC)=O)CN(C(=O)CCc2ccnn2C)CCC1F c1(C(c2ccc(N3CCN(S(C)(=O)=O)CCC3)nc2)C)cc(Br)c2cn[nH]c2c1 C1(CNC(Cc2cc(CC)no2)=O)CN(C(=O)CC2=CCCCC2)CCC1(F)F C(CCN(C)C(C1CC1c1ccncc1)=O)(C(C)C)NC(CCCC)=O CC1(C)C(NC(C2(C)CCC(=O)N2)=O)CCN1C(c1ccnc(C(F)(F)F)n1)=O n1(CCNC(N2CCCC(C(OC)OC)CC2)=O)ccc2cc(F)ccc12 C1(CN(C(c2ccc(CO)s2)C(=O)NCCCF)C)CCCCN1CCl.S(C)(=O)(=O)N c1(C(C)N(C(=O)CC(c2ccccn2)NC(=O)C(F)(F)F)C)cn(CCF)nn1 C1(C(=O)NCCC2CCCOC2)CC(O)CCN1C(c1ccc([N+](=O)[O-])o1)=O c1(OC)cc(C(=O)NCC2CC(NC(=O)C(C)(C)F)C2)cc2c1OCO2 C(CNC(=O)CC1C=NN(C)C1=O)(CCCC)NC(CC1(OC)CCC1)=O C(=O)(C(CCOC(C)(C)C)OC(=O)C(c1ccccc1O)C)OC C=CC(C)(O)CC(=O)NCC(C)(C)CNC(C1(C)C=CCCC1)=O c1(C(N(C2CN(C(C(C(CC)C)C)=O)C2)C)=O)cccc2c(C)[nH]nc12 C1(OC)C(OC)CN2C1CC2=O.c1(NC(=O)C(F)(F)F)c(C)coc1C Cc1cccc(C)c1C(O)C(=O)NC(C)(CNC(c1ccc(C#N)[nH]1)=O)C1CC1 CON1CC(C(N2CCCCC2CC(=O)N(C)Cc2cccnc2)=O)CC1=O CCC(CO)(C(=O)NC1CC2CC(NC(c3coc(C4CCC4)n3)=O)CC12)OC C1(c2n(C)ccn2)N(C(c2cc(-c3cccc(F)c3)no2)=O)CC1(C)C N1(C(C=CC)=O)CCN(C(=O)C(O)C(C)C)C(c2cnn(C)c2)C1 c1(C(=O)NC(CC(N2CC(CCC)OCC2)=O)CC2CC2)cccc(=O)n1C C(=O)(CCCCN=[N+]=[N-])N1C(CC(=O)N(CC(=O)N(CC)CC)C)C2CCCC21 c1(C(N(CC(CNC(C(=O)N(C)C)=O)O)C)=O)nc2c(s1)COCC2 C1(NC(c2c(CC)con2)=O)COCCN(C(=O)C(C)OCC2CCCCO2)C1 CC1CN(C(=NCc2ccccc2-c2ccco2)NCC(F)F)CC(C)(C)C1F c1(C(N2CC(C(CN3CCCCCC3=O)OC)C2)=O)cccc(Cl)c1C c1(C(N2CC(C(C)(C)O)(CO)C2)=O)nn(CC(F)(F)F)cc1C#N N1(C(C2N(C(CC(CC)O)=O)CC(O)C2)=O)CC(=O)NC(=O)CC1 N1(c2n(CCC(=O)NC(C)C)c(Cc3cscn3)nn2)CCC2C(CCN2C)C1 c1(NC2CCC(NC(COc3ccc(C)cc3)=O)C2)ccc(C#N)cc1O C=CCCCC(C(=O)N(C(C)C(C)(C)O)C)NC(C1CC1C(F)F)=O C(=O)(C1=CCC(F)(F)CC1)NC1C(CC)CN(C(c2cscc2Cl)=O)CC1 C(C(C)(O)CC(=O)NC(C)(C)CN(C)C(C1CN(CC(C)C)C1)=O)OC c1(C(=O)NC(CNC(C2C(C)CCC2)=O)(C)C)ccc(N(C)C)nn1 C(CCC(C)C(C(=O)NCC(C)C)N1CCN(c2cncc(F)c2)CC1)=C(C)C N1(C(C=CC(C)(C)SC)=O)CC2CC2(CNC(=O)CCC2CCOC2)C1 C1(C(=O)NCC2CC(=O)NC2)C2CCC(C2)C1NC(C12CCCN1CCC2)=O CN1CCCC(CC(N2CCSCC2C(=O)Nc2ccccc2O)=O)C1 C1(C(=O)Nc2ccno2)CN(C(=O)CCC2CCC2)CCN1 c1(C(C(C)NCC2CCN(C(=O)OC(C)(C)C)C2)O)ccc(Br)cc1 c1(C(=O)NCCC(C)(C)NC(C2C(CC)CCO2)=O)ccn2nccc2n1 C1(NC(CCC2COC(C)(C)O2)=O)CC12CCC(NC(=O)CCC(F)(F)F)CC2 c1(NC(N2CC(OC)C2)=O)ccc(-c2coc(O)n2)cc1 CC(F)(F)CCC(C(=O)O)NC(c1cc2ccncc2[nH]1)=O c1(C(CNC(=O)NCC23C(CN(C(C)=O)C2)C3)C)ccc(F)c(F)c1 N1(C(c2cnc(CC)s2)=O)CCC(O)(CN(C)C(C2CCCC2C(C)C)=O)C1 c1(OC)ccccc1NC(N1CCOC(C(N2CC(C)C(F)C2)=O)C1)=O Cc1cn2c(n1)CCC(C(=O)N(CC(O)CN(C(=O)C(C)S(C)(=O)=O)C)C)C2 N1(C(C2C(=C)CC2)=O)CCC2CCC(C1)N2C(c1c(Cl)ccc2[nH]ccc12)=O C(=O)(C(CC(F)F)N(C)C(c1ccc(C)n1C)=O)NC(c1scc(C)n1)C C(CCS(C)=O)N(C(C)CNC(C1CCSC1)=O)C CS(=O)CC(O)CNC(c1ccc(NCC(F)(F)F)cc1)=O S(=O)(=O)(c1nn(C)cc1Cl)NC(c1cc(N2CCCC(N(C)C)C2)ncc1)=O CCC(CC(=O)N1CC2CCN(C(=O)CCc3cnc(O)[nH]3)C2C1)C(F)F N1(C(C2ON=C(C)C2)=O)CCC2(CC1)CCN(C(=O)CS(=O)(=O)N(C)C)C2 C1(CNC(C(C(C)OC)NC(C=CCOC)=O)=O)COCC(=O)N1C C1(NC(C2C(CC)C2)=O)CN(C(c2ccc(OC)c(OC)c2)=O)CCC1(C)C N1(C(c2cc(CCC)on2)=O)CCC(C(=O)NCCC(C)C(F)F)C1C C=C(C)CC(C(=O)NCC=CCC(=O)NCC1CC(=O)NC(C)C1)OC C1(C(=O)NC2(CN(C(C3C(=C)C3)=O)C)CC2)C(F)(F)C12CCC2 c1(OCC(=O)N(CC(C)O)CCNC(C2CC(=C(F)F)C2)=O)cccc(F)c1F C#CCCCC(=O)NC1CCN(c2cc(C)oc(=O)c2)C1 N1(C(CNC(=O)OC(C)(C)C)=O)CC2(C1)CN(C(C1CCCCC1)c1cscn1)C2 Cc1cc(C(=O)NC2CN(C(C3CCOC(c4ccccc4)O3)=O)C2)cc(Br)c1 CC1CN(C(c2ncccc2Cl)=O)CC(C)C1NC(=O)Cn1cncn1 c1(SC)cccnc1C(=O)NCC1CC(C)N(C(=O)CCCSC(C)(C)C)C1 C1(C(=O)OC)(Cc2cn(C(C)C(=O)Nc3ocnc3C)nn2)CC=CCC1 C1(C(=O)NC(C2CCCC2)CNC(C(CC)F)=O)CCN(c2ncccn2)CC1 C(c1c(F)cccc1F)=CC(=O)NC(CNC(C(C(=O)OCC)F)=O)C(C)(C)C C1(C(C)(C)NC(C2C(C)=C2)=O)CCN(C(c2ccccc2SCCO)=O)CC1 C(=O)(C(O)C(C)c1ccccc1)N(CCCN(C(c1c(C)nc[nH]1)=O)C)C c1(CC)occ(C)c1C(=O)NCc1ncccc1C(=O)Nc1ccc(SC)cc1 c1(N(C)Cc2nccc(OC)n2)ccc(S(=O)(=O)N2CC(C)C(C)C2C)c(Br)c1 CC1NC(=O)OC12CN(C(C1(F)CCN(C(C3(CO)CCCCO3)=O)CC1)=O)C2 C1(CC(=O)NC(Cn2cc(CS(CC(C)C)(=O)=O)nn2)C)COc2ccccc2O1 N1(C(C2CC(C#N)C2)=O)CCCCCC1C(=O)N(CCCO)CCO N1(C(c2n(C)ncc2)=O)CCC2(NC(c3nn4cccnc4c3Cl)=O)CCCCC12 N1(C(CC2CCC(=O)C2)=O)CCC(C2CN(C(C3CS(=O)(=O)CCO3)=O)C2)CC1 N1(C(c2c(C(=O)OC)[nH]cc2)=O)CCOC(C)(CNC(C2CC2C(C)(C)C)=O)C1 Cc1cc(C(N2CC(C(=O)NCc3ncc(C)o3)C(F)(F)C2)=O)c(C)cn1 c1(N2CCC(NC(C(C(C)O)C)=O)C(CO)C2)ccc([N+](=O)[O-])c(C(N)=O)c1 C1(C(N2CC(CCCNC(c3ccncc3)=O)OCC2)=O)CC2C=CCC(C1)C2 c1(C(c2nnnn2CC2CC2)NCC2C(CCC)C2)c(C)cccc1F C1(C2CCCCC2)(NC(=NCC=C)NC2CCS(=O)(=O)C2)CC1 CC1=NNC(=O)C1C(=O)N(CC(=O)N(C)Cc1ccncc1)C1CC1 c1(OC)ccc(N)c(C(=O)NCCNC(c2cnn(C(C)C(C)C)c2C)=O)c1 C1(CN(C2CCN(C(C3CCCN3C(C)C)=O)C2)CC)CCCCN1CC C(CC(=C)C)(C(=O)NC(=O)CC(C)C)OC(CC=C)=O N1(C(CN(C(C)=O)C)=O)CCC(C)(C)C1C(=O)NCC(CO)C(C)C c1(CC(=O)NC2(C(=O)NCC(c3ccccc3)F)CC(CO)C2)cccnc1O C1(CNC(c2cccc(NC)n2)=O)CCC(C)CN1C(=O)C=CC=C(Cl)Cl S(=O)(=O)(c1ccc2[nH]c(=NC(C)CCC(C)C)sc2c1)N(CC=C)CC1CC1 C(c1ccc(Br)c(Cl)c1)=CC(N1CCC(c2nc[nH]n2)C1)=O c1(C(N2CC(CO)CC2C)C(=O)NCC=C)n[nH]c(C)c1Cl c1(C(=O)NCC2C3CN(C(C4(C(C)C)CCCC4)=O)CC32)cnc2ccccc2n1 C1(CC(=O)N(C2CCN(C(=O)C=CC3CCOC3)C2)C)CCCNC1=O Cc1nc2n(n1)CCN(C(=O)CN(C)C(c1sc(C)cc1C)=O)C2 C=Cn1nncc1C(=O)N(C)CC1(O)CN(C(C2COCCO2)=O)C1 c1(C(N2CCN(C(CCCC=C)=O)C(C)C2C)=O)ccc(S(N)(=O)=O)nc1 c1(C(N(C)Cc2cn(C(c3ccccc3)C)nn2)=O)ccc(C(F)F)cc1Cl C(C(C)(C(=O)N(C1CCOC1)C)NC(=O)CC1CCC(C)(C)O1)SC C(=O)(C(F)(F)CCn1cccn1)NC1CC(C)N(C(c2cnc(O)s2)=O)C1 C1(COC)COCCN1C(C1CC(F)CN1C(=O)Cc1ccc(Cl)cn1)=O c1(N2CC(=O)NCC2)nc(=NCc2cncc(F)c2)[nH]c2c1CCCC2 c1(C(N(C2CCN(C(C(C(CC)O)(F)F)=O)C2)C)=O)ccc(O)c2ccccc12 C(=O)(C(O)C(C(C)C)OC)N1CCC(C(=O)NC2(CCC)CCOC2)CC1 O=C1Cc2cc(C(N3CCC4(NC(=O)CC(F)(F)F)CC4C3)=O)ccc2CN1 C1(C(N2C(CN(C(C=CC(C)(C)SC)=O)C)CCC2)=O)CCC(=O)N1C(C)C C(C(C)(C)CC1CC1)NC(C(C)N(C(=O)CSC1CC1)C)=O C(=O)(CC1=CCCC1)NC1(C)CCN(C(CCC(=C)Br)=O)CC1 C(N=c1[nH]c(=NCC2CCCN2C(C)=O)c2ccccc2[nH]1)c1n(CC)ccc1 C(=O)(C1CCCc2nccn21)NCCCCCNC(C1(c2c(C)occ2)CC1)=O S(=O)(=O)(c1cnn(C)c1)NC(C(N1CC2C(NC(C3(OCC)CC3)=O)(C2)C1)=O)C C(=O)(CS(=O)CC(F)(F)F)N1CCC(SCc2nccc(=N)[nH]2)CC1 Cc1nc2c(C(=O)NCCC(C)NC(C3CNC(=O)C(C)(C)C3)=O)cccc2o1 C1(NC(C(COC(C)C)NC(c2ccccc2)=O)=O)CCN(C)C1(C)C c1(CCC(N2CC(N(C)C(c3c[nH][nH]c3=N)=O)C2)=O)ccc([N+](=O)[O-])cc1 c1(CC)ccc(CCC(=O)N(CC(C)CNC(=O)C(C)OCC(C)C)C)cc1 c1(C(=O)NC)ccc(OCC=C2CCCCC2)c(NC(=O)NC2CC2)c1 Cc1ccc2c(ccn2-c2cccc(F)c2)c1 CN1CCC(C)(C(=O)NC2CCCC(NC(c3nnn(C)c3N)=O)C2)C1=O C1(C(F)F)(OC)CC(C(=O)NC23CC(NC(c4cnn(CCC#N)c4)=O)(C2)C3)C1 C12(C(N3CC(O)(CNC(C4CC4F)=O)C3)=O)CCC(CC1)O2 c1(N(C(N2C(C(=O)O)CCC2)=O)CCSc2ccccn2)cccc(C(=O)O)c1 S(=O)(=O)(c1ccc(N2CCOC(C)CC2)c(Cl)c1)NC(CC)COCC1CC1 C1(=O)CCCC(=O)N(C2CC2)C2CN1C2.C1(C2(C(=O)NC(C)C)CC2)CCCO1 CCCC(CCC)C(=O)N1CCC(NC(c2cnn(Cc3ccccc3)c2)=O)C1 c1(C(=O)NCC2C(CNC(c3ccoc3Cl)=O)C2)csc2ncnc(O)c12 c1(C(=O)NCC2CN(C(CCCOCCC)=O)CC2O)coc2c(C)cccc12 c1(OC)cc(C(=O)N(C2CC(C(=O)NCCCc3cc(O)n[nH]3)C2)C)ncn1 C1(CCCC)CCC(C(N2CCC(NC(=O)C=CSC)C2)=O)CC1 N1(C(COCCCCCC)=O)CC2CC(C1)CN(C(c1nocc1C)=O)C2 C(CCCCC(=O)NC(C)C(c1ccccc1)NC(=O)C=CBr)SC C1(NC(Cc2cc(CC)nn2C)=O)CC2CC(C1)N(C(c1cccnc1N)=O)C2 c1(OC)ccnc(F)c1C(=O)NCC(O)CNC(=O)C(C)N(C)C(C)=O C1(NC(c2cc(CC)nn2C)=O)CCN(C(C2CC(C#N)C2)=O)CC1(C)C C1(CNC(C(C)SC)=O)C=CCN1C(c1cc(-c2cnn(C)c2)[nH]n1)=O C1(NC(Cc2c(C)ccnc2)=O)CCC(O)CN(C(C2(C)CC2(F)F)=O)C1 CC1CC(C(N2CCOC(c3nccn3C)C2)C(=O)NCCC2CC2)CC(C)C1 c1(C(=O)OCC)c[nH]ccc1=NC1(CC)CCCCN(C(c2cnsn2)=O)C1 N1(C(c2c(OC)cncn2)=O)CCC2(C=C(C(=O)NCC(C)CC(F)(F)F)C2)C1 C(CC(=O)NC1CC2(CC2)C1)(C(F)F)NC(C(C)C1CC1)=O C1(CNC(C(C)NC(=O)Cc2ccc(F)c(F)c2)=O)CCn2ccnc2C1 C(=O)(C1=Cc2cc(F)ccc2OC1)N(C(CNC(C1(C)CC1)=O)C1CC1)C C(=O)(CC(C)(C)C#N)N(CC(=O)NCC(C)(C)OCCO)CCOC C1(C(=O)NC2CC(NC(C3CC(SC)C3)=O)C2)CCc2ncnn2CC1 C(C(C1CCCCC1)NC(c1cc(SC)c(C)o1)=O)(C(C)C)NC(COCC)=O c1(CCC)cc(C(=O)NCCC2(NC(C3(C(=O)OC)CC3C)=O)CC2)c(C)o1 N1(C(C(C)SC(C)C)=O)CC2CCC1C(NC(c1cn(C)nc1C(F)F)=O)C2 CC1CC(NC(=O)CCOCCN(C)C)CCN1C(=O)C(C)(C)c1cncnc1 N1(C(CCCC=C)=O)C(CNC(=O)COc2ccc(C#N)cc2)CC2COCC12 CCC(F)(F)CC(=O)NCC1CCCN(C(c2ccc(N3CCC3)nc2)=O)C1 c1(C(N2CCC(CNC(CC=C=C)=O)(OC)CC2)=O)ccc2c(Cl)nccc2c1 CC(C)C(=O)C(=O)NN1CCCC1C(=O)NCC1CCCSC1 c1(CC(N2CCCC(NC(C3CCSC3)=O)C2)=O)cc(F)cc(F)c1 c1(C(=O)NC(C(c2ccccc2)NC(c2c(C)onc2)=O)C)cc(=O)n(C)cn1 C(=O)(C(O)CC(F)(F)F)N1C(C(C)C)C(NC(=O)CCc2ccccc2Cl)CC1 C1(NC(CC2ON=C(C)C2)=O)CC2(C1)CN(C(c1cc(C)c(F)cn1)=O)C2 c1(NC(C2CCN2C(=O)CCC2CCCC2)=O)cccc(F)c1F C1(C(=O)NC(CC2CC2)C(N2CC3CC3C3CC23)=O)CC2C(C1)C2(F)F C(C(C)C(=O)NOCCC)N(C(c1c(CCC)[nH]cc1)=O)C C(=O)(CC(CC)CC(C)C)NC1(CC(=O)N(c2cn(C)nn2)CC#C)CCC1 c1(CNC(c2ccnc(CNC(C3CCCC(O)C3)=O)c2)=O)cc(O)cc(F)c1 c1(C(N2CCC(N(C(=O)CC3CC34CC4)CC#C)C2)=O)nnn(CCOC)c1C N1(C(CCC(=C)Cl)=O)CCC(C)C(NC(=O)C#CC2CC2)C1 C(=O)(C(O)C1=CCCCC1)N1CCC(CCCNC(c2c(C)ocn2)=O)CC1 CS(=O)(=O)c1cc(N2CC3CC(NC(C4(n5cnnn5)CC4)=O)CC2C3)ncn1 C1(CCC#C)CCCN(C(C2CCN(C(C3CC(SC)C3)=O)C2C)=O)C1 C1(C(=O)NC(C2CN(C(CCNC(COC)=O)=O)C2)C)CCC(C)O1 N1(C(CN(C)CC)=O)CCCCC1C(=O)NCC(F)CN(C)C CCCCCCCC(F)C(=O)NCCN(C(=O)C(C)OCC)Cc1cccnc1 O=C1CC(CC(=O)NCC2CC(NC(=O)CCn3cccnc3=O)C2)CC(=O)N1 c1(C(N2CC(CC34CC(C3)C4)C2)=O)ccc(Oc2ccc(Cl)cc2)cc1 c1(C(C)NS(C)(=O)=O)ccc(C(=O)N(CCCc2ccco2)C)cc1 c1(OC)c(Cl)cccc1S(=O)(=O)NC(c1ccc(F)c(C(F)F)c1)=O C(=O)(CC(F)(F)C(F)F)N(C(C)C)CCNC(=O)COc1nn(C)cc1Br C1(C)(CNC(c2n(CCC)ccc2)=O)CN(C(c2cn(C)nc2OC)=O)CCO1 Cc1[nH]c2ccccc2c1CC(=O)N(C1CN(C(C2(O)COC2)=O)CC1F)C C1(CNC(CCc2ccn(C)n2)=O)CN(C(C2(C)CNC(=O)C2)=O)CCC1(F)F N1(C(C2(C)CC(F)C2)=O)CCc2ccccc2C1CNC(C1(O)CCCC1)=O N1(CC)CCOCC1NC(=O)C(c1ccnn1C)NC(=O)COC1CCCCC1 Cc1cccc(SCC(=O)NCC(CO)NC(c2ccccc2C2CC2(F)F)=O)c1 N1(C(CNS(N)(=O)=O)=O)CCC(C2CC2)C1CNC(c1n[nH]cc1Cl)=O CN1C(=O)CSC1=CC(=O)NCC1CC(NC(=O)CSCc2cccs2)C1 C1(NC(c2ccoc2C2CC2)=O)CN(C(C2CCC3(CCC3)O2)=O)CC12CC2 C1(CNC(c2cnns2)=O)CCCC(NC(=O)C(c2ccc(F)cc2)=O)C1 C1(NC(c2n(C)nc(C3CC3)c2)=O)CC2CCC1CN2C(c1sccc1F)=O Cc1ccc(O)c(S(=O)(=O)Nc2ccc(OC3CCOC3)nc2)c1 C1(C(=O)OC)CCCN(C(c2nocc2C)C(=O)NCCCC2CC2)C1 N1(C(c2n[nH]c(=N)s2)=O)CC=CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 C1(C(=O)NCCC2N(C(C=CCOC)=O)CCOC2)CC2CC1CC2O O=C1COc2ccc(C(=O)NC3(CO)CN(C(C4(CO)CCCC4)=O)C3)cc2N1 Cc1cc(N2CCCC(CNC(C3(C)CCCC3C)=O)C2)n2nc(C)cc2n1 C(=O)(CC(C)CC(C)(C)C)N1CCCC(N(C(c2c(C)ncs2)=O)CCF)C1 c1(NC(=O)CC2CCCO2)cccc(-n2cnnn2)c1.C12CCN(C1)C2=O C1(CCNC(COc2c(C)cc(C)cc2C)=O)COc2ccccc2O1 N1(C(C2C(CC)C2)=O)CC2CCCC1C2CNC(c1ccc(C)cc1)=O N1(C(C(C)OCC(C)C)=O)CC2(CCCC2NC(=O)C=Cc2cnn(C)c2)C1 c1(C(N2C(CNC(C(C(=O)OC)C)=O)CCCC2)=O)ccc2sccc2c1 C(C)(CC(N)C(=O)NCC1(c2cccc(F)n2)CCC1)OC c1(C(N2CC(F)CC(NC(C(CC#C)C3CC3)=O)C2)=O)cc(C)c(F)cc1F c1(OC)ccc2sc(C(=O)NC3(CNC(c4cc(CO)[nH]n4)=O)CC3)c(C)c2c1 N1(C(C(CSC)C)=O)CCC(NC(C2CCCS2)=O)C2(CCC2)C1 c1(C(N(C)CCNC(C2CCCCN(C)C2=O)=O)=O)ccc2c(c1)NC(=O)C2(C)C n1(CC(=O)NC2(CC=C)CCN(C(=O)C=CC=CCOC)C2)ccc(O)nc1=O C(=O)(C1=NOC(C)C1)NCC(C)(C)NC(c1c(CC)n(C)nn1)=O CCCCCC(O)CC(=O)NCCCC(CCC)NC(=O)CC(C)(C)C c1(CNC(NC(CC)CO)=NCCSc2ccccc2)ccc(Br)c(C)c1F C1(NC(CC(C)SC)=O)CCC2CN(c3cc(Cl)c(O)nn3)CCC2C1 CC#CCCC(=O)NC(CO)C(C)NC(C1(CC)CCCCC1)=O c1(-c2n(CCCC)nc(CC(C)CC)n2)c(F)ccc2c1OCC2 Cc1cccc(CC(N2CC(NC(c3sc(F)cc3C)=O)C(C(F)(F)F)C2)=O)c1 Cn1nc2c(c1N)CN(C(C1COCC3(CCC3)O1)=O)C2 c1(OC(C)C)ncccc1C(=O)NC(C1CN(C(=O)C(O)C2CCC2)CCO1)C Cc1cc(C)c(C(=O)NCc2cc(C)c(C(=O)N(CC(C)C(C)C)C)o2)o1 c1(OC)n[nH]cc1C(=O)NC(CN(C)C)C(=O)NCCCn1ccnc1 c1(CC(=O)OC)cscc1NC(N1CCC1c1ccccc1)=O.C1CCC(C)N1 Cc1ccc(F)c(C(=O)NC2(C)CCCN(C(=O)C(C)c3ccon3)C2)n1 c1(OCCNC(C(=O)NC(C#C)CCC)=O)cccc(Cl)c1Cl c1(C(=O)NCC(C)(O)CNC(=O)CCC2CC(C)(C)CO2)cnc2c(c1)NCC2 c1(C(N(C(C)C(=O)NCC2(n3ccnn3)CC2)CC)=O)cc(C)[nH]c1C CN(C(=NCc1ccnc(F)c1)NCc1ccnn1C)CC1(F)CCOC1 N1(C(C2C(CCC)C2)=O)CCN(C(c2ncccc2O)=O)CC1CC(F)F N1(C(CCCc2nc(C)sc2)=O)CCC2(CCCC2NC(=O)Cn2ccnn2)C1 C(C(C)(CC(C)C)NC(C1CC1C(F)(F)F)=O)NC(c1c(C)n(CCO)nc1)=O C(CC(C(=O)NCC1CC12CCOC2)NC(C1C(C)(C)C1(C)C)=O)SC N1(C(Cc2scc(C)c2)=O)CCSCC1C(=O)NC(C)CC(C)(C)C c1(CONC(=O)NCc2c(C)cn(C)c2)ccc2ccccc2c1.OCC N1(C(COCC(=C)C)=O)CC(C)(CNC(C2(OC)CCOC2)=O)CC1(C)C N1(C(c2c(C)nsc2)=O)CCC(NC(c2cc(=O)n(C)s2)=O)C(CO)CC1 CCCCC(O)C(C)C(=O)NCC1(F)CCCN(C(c2cnc(C)cn2)=O)C1 Cc1c(N)ccc(C(=O)NC2CC(CNC(C3CC4CC3CC4(F)F)=O)C2)c1C N(C1CCc2cc(F)ccc21)C(c1cccc(I)c1)c1n(C(C)C)nnn1 O=C1CSc2ccccc2C(NCCNC(c2ccc(N3CCOC3)cc2)=O)C1 CCCC(CNC(C1CN(C(C)C)CCO1)=O)C(=O)NCC(=O)OC N1(C(c2c(C)cccc2)=O)CC(CNC(c2cccc(C)c2C)=O)C(C)CC1C CC1CC(N=c2[nH]c(=NCCC3(C)CCC3)[nH]c3ccc(Cl)cc23)CCS1(=O)=O Cc1cnc(C(=O)NC(C)CN(C)C)cc1C.C12(CCOCC1)C(=O)N2C Cc1cccnc1C=CC(=O)NCC(C(C)(C)C)NC(=O)C=CS(C)=O c1(C(N2CCC(C(C)NC(COCCC#C)=O)C2)=O)cc(Cl)cc2c1OCC2 CN(C)S(=O)(=O)NCC(N1CC(CCNC(C2(CO)CC2(F)F)=O)C1)=O c1(C(N2C(C)(C)CC(C(=O)NC3CCC=CCC3)C2)=O)ccnc2cc[nH]c12 C1(C(N(CC)CC2CCCN2CC(F)(F)F)=O)CCCN(CP(C)(C)=O)C1 c1(C(N2CCCC(N(C(C3(C)CC(C)=NO3)=O)CC)C2)=O)cc(C)c(CO)cn1 C12(C(N3CCC(C)(C)C3CNC(C3CNC(=O)C3)=O)=O)CC(C)(C1)OC21CCC1 C(=O)(C(CC)(CC)CO)N1CC(O)(CN(C(C2CCN(CCCC)C2)=O)C)C1 c1(N2C3CN(Cc4ccc(OC)c(C(C)C)c4)C(C3)C2)ncnc2c1cnn2C C1(NC(CCN(CCC)C)=O)COC2CN(C(C3CCCC(COC)C3)=O)CC12 c1(CNC(CC(C)C2CCCO2)=O)ccc(CCNC(c2coc(Cl)n2)=O)cc1 C1(CC(=O)NC2CCC3(CC2)N=N3)CC2(CC2)CN1C(=O)Cc1ccc(O)nc1 c1(C(N(C(C)C(=O)NC(C)(C)CF)CC)=O)cc[nH]c2nccc1-2 C=CC1OCCC1C(N1CC(OC)C(NC(c2cnn(C)c2SC)=O)C1)=O CCC(C)(CCO)NC(=O)C(C)CNC(=O)Cn1cccn1 CCC(CN(C)C)C(=O)NCC(N1CCN(C(C2CCC(C)CC2)=O)CC1)=O N1(C(c2c(C)con2)=O)CCCOC(CNC(c2ccncc2F)=O)C1 C(=O)(C1=C(C(C)(OC)OC)N(C)C(=O)NC1c1cnc(Cl)c(N)c1)OCC N1(C(C=C2CCN(C)C2)=O)CCC(C)(C)C(CNC(C2(F)CC2)=O)C1 C1(CNC(CCOC2CN(C(C3C(C#N)CC3)=O)C2)=O)CC(C(N)=O)=NO1 C1(CC(=O)NCC2CC(C)(C)C2)CN(C(=O)CC2OCCCO2)CC12CC2 c1(OC)cc(N)c([N+](=O)[O-])cc1CC1(c2cc(F)ccc2F)CC1.SC C=CCC(CNC(=O)C(C)n1cnnn1)C(=O)N(CCCCN(C)C)C C#CCCCCCC(=O)NC(C)(CNC(C1CC2OC1C1CC21)=O)CO Cc1cnc(F)cc1NC(=O)NCC1(Oc2ccccc2)CCCC1 c1(CCC(=O)NC23CC2CN(C(=O)CSc2ccccc2)C3)cc(Br)ccc1F C1(NC(C(C2CCOC2)NC(C=CC(C)(C)C)=O)=O)CN2CCC1(C)CC2 C(CC(C)C(=O)NC1CC1NC(c1cc(C)c(C)[nH]1)=O)=CC CCCC(C)(C)CC(=O)NC(C(N1CC(C)(C(F)(F)F)C1)=O)C1CC1 C1(NC(C2CCCCC2)=O)CN(C(C2CC3CCC(C2)C3)=O)Cc2ccnn2C1 c1(C(C)C)cc(CN2CCc3nn(C)cc3C2)c2ccccc2c1 C(CCC(C)(C)C(=O)Nc1cnn(C)c1Cl)OC C1(CNC(C2C(C(=O)OC)C2)=O)CCN(C(c2cccc(SC)c2)=O)C12CCC2 c1(N(C)Cc2nc[nH]n2)nc(N(C)CC2CCCCO2)nc2c1CSC2 C1(CN(C)C(c2cncn2C2CC2)=O)CCCN(C(=O)Cc2csc(S)n2)C1 CCC(CC)C(=O)NCCCN(C(C1(C)CC1(F)F)=O)Cc1ccccc1 C=CCC(CC)C(=O)NC(C1CC(NC(c2ccnn2CCOC)=O)C1)C C#CCC(C)C(=O)NCCC(CNC(=O)CCOc1ccc(O)cc1)OC c1(C(=O)NCC(CNC(CCCCC)=O)(C)O)nc(C)ccc1C CC1CC(NC(=O)Cc2cccc(O)c2F)CCN1C(c1cnc(Cl)s1)=O C(=O)(C1=Cc2ccccc2C1O)N1C(CCNC(c2c(C)occ2)=O)CCC1 CC1(C(=O)NCC2CN(C(c3ccccc3OCCF)=O)CC2O)CCSCC1 CCC1=NOC(C(=O)NC(C)(CSC)C(=O)N(C(C)CN(C)C(C)=O)C)C1 C1(CC)C(NC(=O)Cc2c(C)cnn2C)CCN1C(=O)Cc1ccc(O)nc1 c1(OC)ccc(C(=O)NCCCCc2cn(-c3ccnc(Cl)c3)nn2)nc1 C12CCCCCC1N2.c1(OCCNC(=O)OC(C)(C)C)ccc(Cl)c(Cl)c1 c1(OC)ccc(C(C)(C)C(=O)NCC(O)CNC(=O)C(n2ccc(C)n2)C)cc1 n1(CCC)nnnc1C(CC1C2CC12)Nc1cncnc1 c1(N2CC(N(C(=O)CCSc3nccn3C)C)C2)nc(Cl)nc2c1cnn2C C1(NC(CCN(CCCCC)C)=O)COCC1n1cc(C(C)(C)CC)nn1 CCCCC(CC)CC(=O)NC1CN(C(=O)CCC(=O)N2CCOCC2)C1 C1(SCC(=O)NC2CC(NC(C(c3cncn3C)N(C)C)=O)C2)CCC(=O)NC1 CC1OCCCC1C(=O)NCC(=O)NCC(=O)NCCN=[N+]=[N-] c1(CNC(C2C3COCC23)=O)ccc(C=CC(=O)NC(CN(C)C)CO)o1 C=C(C)CN=C(NCC(=O)NC(C)C)N1CCCC(NC(C2CCCO2)=O)C1 C1(NC(C(C)OCC)=O)CC2CC1N(C(C1(Br)CC1)=O)C2 CCC(C)(COC)C(=O)NCC1CN(C(=O)C=CC(C)C)CC1(F)F c1(C(N2CC(N(C(c3c(COC)nn(C)c3)=O)C)C2)=O)ccc(C)nc1O CC1(C(=O)NC2CCC(CNC(C3CC=CCC3)=O)CC2)COC(=O)N1 C(=O)(CN=c1ccc(Cl)n[nH]1)N(C)CCNC(=O)C(O)CCS(C)=O c1(C(N2CCCC(CN(C(CCC)=O)C)C2)=O)ccc2oc(O)nc2c1 C(C1COCc2ccccc21)NC(=NCCc1cc(OC)ncc1)NC(C)C C(=O)(C1Cc2c(Cl)cccc21)N1CCCC(N(C(CCCC#C)=O)C)C1 Cc1nc(C)c(CNC(=O)CC(C2CC2)NC(=O)CCOCC(C)C)s1 c1(C(N(CC(CNC(CC(C)CN(C)C)=O)O)C)=O)cnc(O)c2ccccc12 CCC(O)C(F)(F)C(=O)N1CC(O)(CNC(=O)Cc2csc(-c3ccsc3)n2)C1 C1(CC(=O)N(C(C2(NC3CCSC3)CCOCC2)=O)C2CC2)CCS(=O)(=O)C1 N1(C(Cc2c(C)occ2)=O)CCCC(C(C)NC(C2CC=CC2)=O)C1 C1(C(C)NC(=O)CCCc2cccs2)CCCN(C(=O)C(C)(C)CC2CC2)C1 c1(OCCCC(N2CCC(N(C(=O)C(C)C)CC)CC2)=O)ccc(C)cc1 C1(CSc2n(CCCC)c(-c3ccccc3C)nn2)CCC(F)(F)CC1 c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)CC(C)C2)cc(C)c(C)cc1C C1(NC(C2C3CN(C(C4CC5CCC5C4)=O)CC23)=O)CC2CC3C(C2)C13 c1(CCC(=O)NCCN(C(C2CCN(S(C)(=O)=O)C2)=O)CC)cc(C)cc(C)c1 Cc1ccc2oc(C(N3CC4(CCCCN4C(=O)C4=NOCC4)C3)=O)cc2c1 c1(SC(C)C(=O)NC2(CCNC(N)=O)CCOC2)nnnn1C1CC1 C1(NC(CC(COC)C)=O)CC2CCC(C1)N2C(c1ccnc(C(F)(F)F)n1)=O C=C(C)CC(C(=O)N1CCN(C(C2(c3ccc(C)nc3)CC2)=O)C(C)C1)OC C1(CCC)CN(C(c2cc(C3(C)CC3)on2)=O)CCN1C(c1cnn(CC)c1)=O C=CC(C(=O)N(CCC(C)NC(=O)Cc1scnc1C)C)OC c1(C(=O)NCCC(CC)C)nc(C)c(Br)c(C)n1 c1(NC(=O)OCCOCC#C)c(Cl)cc(Cl)cc1Cl C1(CCC(N2CC(CCNC(CC3(CS(C)(=O)=O)CC3)=O)C2)=O)OCCC1(C)C N1(C(C2(C)C(C)CN(C(C(C=CC)O)=O)C2)=O)CCc2c(cnn2C)C1 C(=O)(C(C)CC1CCCCC1)N1CC(C(C)NC2(C(N)=O)CC2)C1.CC1C(=O)N1 C=CC(CCC)CC(=O)NC1CCCC1CNC(=O)CCC(C)(C)C#N c1(CC(=O)NCC2(NC(C3CCC(C)C3)=O)CCCC2)noc2ccc(F)cc12 C(CCC(=O)NCc1ccc(C(=O)NC2(C)CC2(C)C)s1)OC(C)(C)C c1(CCC(=O)NCC=CCNC(CC2CCC(C)(C)O2)=O)nnc(S)nc1O N1(S(C)(=O)=O)CCCC(CC(=O)NCC2CN(C(c3cncc(O)c3)=O)C2)C1 C=CC(C)(O)CC(=O)N1CC(CNC(=O)C(c2cccc(OC)c2)O)CC1C c1(C(N2C(C(C)NC(c3c(C)[nH]nc3Cl)=O)CCC2)=O)nccc2ncccc12 C=C(C)CC(C(=O)NCC(C)(C)C#N)NC(C1OCCCC1(C)C)=O CC(c1cnn(C)c1)=CC(=O)NC1CCC(CNC(=O)CCC(C)(C)F)C1 C(=O)(C1=CC(C)(C)C1)N1C(CNC(CCOc2c(CC)cccc2)=O)C=CC1 CCS(=O)(=O)CC(=O)NCC(C)(C)CN(C(=O)CCN1CCC1)C N1(C(c2ccc(C)c(O)c2)=O)CCC2(C1)CN(C(c1ccc(C(N)=O)cc1)=O)C2 c1(C(N2C(CNC(=O)Cn3nnc(=O)[nH]3)CCC2)=O)cnc2c(c1)NCC2 N1(C(CC=CCC)=O)CC(CC(N2CCCC(O)CC2)=O)C2(CC2)C1 c1(C(=O)NCCN(CCOC)C(c2ncoc2C(C)=O)=O)cnc(C)s1 C(N=c1ccn(CCSC)[nH]1)(c1c(F)cccc1F)c1n(CC=C)nnn1 C1(CNC(C=CC(CC)C)=O)C(O)C(O)CN1C(c1cc(=O)c(OC)c[nH]1)=O c1(SC)ccc(-c2cnc(C(=O)Nc3ccc(Cl)cc3)nc2)cc1F c1(C(=O)NCC(C)NC(C2(C#N)CC2(C)C)=O)ccc(-c2ccc(F)cc2)n1C c1(N(C(=O)CC2CCC3CC23)CCn2cncn2)ccc(NC2CCC2)nc1 CC(C)C(CNC(=O)Cc1cn[nH]c1)Cc1cccc(C(=O)O)c1 c1(OC)noc(C2CC2)c1C(=O)NC(C)C(C)NC(=O)CCc1ccccc1O C(=O)(C1Cc2ccccc21)NC1C2OCC(NC(=O)C=Cc3cnc[nH]3)C2OC1 N1(C(CC(=O)NC(C2CN(C(=O)CC3CCCC3)C2)C)C)CCCC1=O N1(C(CSCCCC)=O)CCN(C(c2cccnc2C)=O)C(C)C1C C1(NC(C23C(C(=O)OC)(CCC2)C3)=O)CN(C(c2cocc2C)=O)C(C)(C)C1 C1(C(N(C)CCOCCO)=O)CN(C(=O)CC2CCCC(=O)N2)CC1F C1(O)(CN(C(C(C)C2CCC2)=O)C)CCN(C(c2ccc(C(F)F)o2)=O)C1 N1(C(CNS(NC)(=O)=O)=O)CC(CNC(=O)CCc2nc[nH]n2)C2(CCC2)C1 C1(NC(CCSC)=O)CN(C(=O)CCCSc2ccccc2)CC1n1ccnn1 C(Cc1ccco1)(C(=O)NCc1ccoc1)NC(C(C)c1ccco1)=O c1(C(=O)NCCCC(CCC)NC(=O)Cc2ccc(C)o2)n[nH]c2c1CCCC2 C1(C(N(CCCNC(c2c(C)csc2)=O)CCO)=O)CCC(=O)N1C(C)=O CCC(CC(=O)N(C(C)C(=O)Nc1cc(C)c(F)cc1O)C)CC(C)C c1(N(C)C)ccncc1CNC(=O)CC1CC=CCC1.C12CCCN1C2=O C1(NC(c2cc(OC)ncc2)=O)CC(NCc2cccs2)C12CCC2 Cc1sc2ncnc(CN(CC(C)C)CCO)c2c1C c1(CN(CC(c2ccccc2)=O)CCN(C)C)cccc(F)c1 N1(C(c2ccnc(OC)c2)C(=O)NC(CC)C)CCCc2c(Cl)cccc21 C(=O)(C1CNC(=O)c2ccnn21)N1CCC(NC(Cc2c(C)occ2)=O)C1 c1(NC(C(C2(C)CC2)NC(c2cc(C)no2)=O)=O)cc(Cl)ccc1O C1(C(N2CCC(C=C)C2)=O)CC12CCN(C(C1CCC(CC)CC1)=O)C2 c1(C(=O)NC2C(NC(C3(OC)CCOC3)=O)C2)cn(C)c(=O)cn1 N1(C(CCC=CC)=O)CCCC(C(C)NC(C2(n3cc(Br)cn3)CC2)=O)C1 c1(C(=O)NC(C)CN(C(=O)CC2CCCO2)C)ccccc1C(C)(C)C C(N=c1[nH]c2c(c(=NCC3CC34CC4)[nH]1)SCC2)C1(C(F)(F)F)CC1 CC1CC(NC(=O)CC(c2cccs2)n2cccc2)CCN1C(=O)Cc1cnns1 CC1=C(C(=O)N(C)CC2C3CN(C(C4CCNC4=O)=O)CC23)CCO1 N1(C(C2CCN(C)C2)=O)CC2CCC2(CNC(c2ccccc2C(F)F)=O)C1 C(=O)(C(C)C(C)CCC)NC1(CC=C)CN(C(c2cnn3ccsc23)=O)C1 C1(c2c(C)n(C)nc2)C(C(=O)NC2CNC(C)C2)CC(=O)N1C c1(CC)c(C(=O)NC2CCC(CCC(N3CCOCC3C(C)C)=O)C2)ccn1C CC1(C)C=C(C(=O)NCC2(O)CC(CNC(C3CC4CC3CO4)=O)C2)C1 CC1(C)CC(CNC(=O)CC2CCCC(=O)N2)N(C(=O)CC2CCC(O)C2)C1 C(=O)(CN=c1[nH]c2ccccc2s1)NCCCNC(C(C)OCC#C)=O c1(CC(=O)NC(CC(C)NC(CCOCC)=O)C)cccc(CC)c1 c1(SC)ccc(C(=O)N(C2CN(C(N)=O)C2)C)cc1.C12COC(C1)CNC2 C1(C(CO)NC(C(C)OCC2CC2)=O)CCN(C(=O)CS(C)(=O)=O)CC1 c1(C(=O)NCCOCCNC(CC2ON=C(CC)C2)=O)cc2c(Cl)ccnc2s1 c1(CC(=O)N(C2CN(C(C3CCSC3)=O)C2)C)cc(F)cc(F)c1 c1(OC)nc(C)c(CC(=O)NC2CCC(CNC(=O)CCN3CCOC3=O)C2)s1 c1(OC)cc(C)c(NC(=O)C(C2CC2)N(C(=O)CC(C)SC)C)cn1 N1(C(C2CC(C#C)(O)C2)=O)CC=C(CCNC(c2cnn3ncccc23)=O)CC1 Cc1nnc(O)c(C(=O)NC2CCCC2CNC(=O)CCCCO)c1C C(CC(C(=O)N1CCC(CF)C1)NC(c1ncncc1OC)=O)=CC C#Cc1cnc(C(=O)NCC(=O)NCCCCCCCC)c(C)c1 CC1CN(C(C2CCCCC2)=O)CC2(CCN(C(c3sc(F)cc3Cl)=O)CC2)O1 C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)CC2CSC2)CC12CCOCC2 C1(CNC(C(P(C)(C)=O)O)=O)CN(C(c2ccc(CCF)cc2)=O)CCC1(F)F C(C)(C)(C(=O)NCCCNC(c1ccco1)=O)NC(=O)OC N1(C(Cc2cc(C)on2)=O)CCC2(CC1)CC2C(N1CCC2(CCC2)C1)=O N1(C(c2ccc(C(=O)OC)s2)=O)CC(C)CN(C(=O)CCc2cnn[nH]2)CC1C C1(NC(Cc2cc(C)[nH]n2)=O)CCN(C(C2CCC(C)C2)=O)CC1 C(=O)(C(C#N)C(C)C)NC1CCCC(C(=O)NCc2cc(CC)on2)C1 CCCC(C(=O)N1CC(C(C)NC(=O)CCOc2ccccc2C#N)C1)C(C)C C#CCCCOC(=O)C(C)N(C(=O)C(C)NC(N)=O)C C(=O)(CCCCCCCNC1(C(F)(F)F)CC=CC1)OC c1(C(N2CC3CC2CN3c2ccc(F)c(C3(CO)CC3)c2)=O)cc2ccccc2o1 n1(CC)nnc(C)c1C(=O)NCC(C)(C(C)C)NC(=O)C(C)OC1CCCCC1 C1(NC(C=C(C)C2CC2)=O)CN(C(c2c[nH]nc2F)=O)CC12CC2 c1(N2CCC(C)(NC(Cc3c(C)cco3)=O)CC2)nccn2nnnc12 CC1CC(NC2CCCC2C(=O)NCCSCCO)CO1 c1(OC)ccncc1C(=O)NC1CCCC1CNC(C1CC(n2cnnc2)C1)=O C12(C(N3CCC(CN(C(=O)COC4CC4)C)C3)=O)COCC1C2(F)F C1(CC)C(NC(C2(C(C)(F)F)CCC2)=O)CCN1C(C1CC(O)CN1C(C)=O)=O N1(C(C2CCN(C(C)C)CC2)=O)CCC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C(F)C1 C1(CNC(C(C2CCC2)OCC)=O)CC2(CCN(C(C3(C)CSC3)=O)CC2)CO1 CCC(C(=O)NC(C)(C)CCCNC(=O)C(C)Cc1cnn(C)c1)C(C)(C)CC C1(C(CNC(c2ccc(CCC)[nH]2)=O)O)CCN(C(=O)C(F)CC2CCC2)CC1 C1(NC(C(N(C(C(C)NC2CCOCC2)=O)C)C2CC2)=O)CCC2CCCC1O2 C1(CNC(c2c(CC)noc2)=O)CC2(CCN(C(=O)Cc3ccno3)CC2)CO1 c1(C(=O)NC2(C)CN(C(CC(C)c3ccccc3)=O)C2)cc(N(C)C)ccn1 C#CC12CCC(C(=O)NC(CNC(=O)C(C)Cc3ccco3)CC)(CC1)CC2 n1(CC(=O)N(C)CC2CCN(C(CCCOC)=O)C2)ncc2ccccc2c1=O C1(C(=O)N)(CO)CC=CCC1.c1(C(=O)O)cncn1CCCOC1CC1 C=CC1CCN(C(C(=O)Nc2ccc(OC)cc2)C23CC(C2)C3)CC1 N1(C(CCCN(CCC)CCC)=O)CC(NC(=O)C(F)C(C)C)CC1CO Cc1cnc(N2CCOCC2)nc1NCC(F)C1CC1 CC1CC(C(N2CCOC(CNC(c3ccncc3)=O)C2)=O)CN1C c1(C(N2CCCC(CCNC(C(C)NC(N)=O)=O)C2)=O)c(Cl)ccc2c1OCO2 N1(C(CNS(N)(=O)=O)=O)CC2CCC1C(CNC(c1ccc(Cl)c(Cl)c1O)=O)C2 c1(NC2(CNC(C=C(C)C)=O)CCCC2)nc(C)nc2scc(C)c12 C1(CC=C)(N(S(=O)(=O)C(F)(F)F)C(c2nnnn2-c2ccccc2)=O)CCSCC1 N1(C(c2cc(OC)n[nH]2)=O)CCC(NC(=O)C(=O)Nc2ccccc2)CC1C C(=O)(CCCS(=O)c1ccc(Br)cc1)N(c1ccc(Br)cc1C(N)=O)C c1(C(=O)NCC2C3(CN(C(CC(C)C)=O)C3)CC2)nn(C)cc1[N+](=O)[O-] N1(C(c2ccc(CC)s2)=O)C2CCC1CC(C(N1CCC1COC)=O)C2 C1(NC(C(C2CC=CCC2)NC(CC2CC(=C)C2)=O)=O)CC2(C1)CC(C#N)C2 C1(C(=O)NCCCN(C(C2CC(F)(F)C2)=O)C2CC2)C2CC3CC(C2)CC1C3 N1(C(C(C)C)=O)CCOCCC1C(=O)NC(c1ccns1)C CCCC(C(=O)N1CCN(C(C2CCC(=O)N(C(C)C)C2)=O)CC1C)C(C)C c1(C(=O)NC2CC(CNC(C3CC3(F)F)=O)C(O)C2)cc(F)ccc1Cl Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)C(C)C(F)F)c(N)c(F)c1 CC(C(=O)NC1CN(C(c2csc(-c3ncc[nH]3)n2)=O)CCC1F)C(C)(C)C C(CC(C)C(=O)NC1C2CN(C(c3ccccc3C)=O)CC12)=CC N(C(=NCC1CCCC(=O)N1)NC1CCCC1)C(C)C Cn1nncc1CCNC(=O)C(C1CCN(C(=O)CC2CC(N(C)C)C2)C1)F c1(CNC(CC=C)=O)cc(C(=O)N(C2CCC(C)C2)C)n(C)n1 c1(N2CC(CCNC(c3ccncn3)=O)(OC)C2)ccnc2nc(C)nn12 C1(OCC)(CC)CCCN(C(=O)C(C(=O)NC)c2ccccc2)C1 C(=O)(C(CCN(C)C)NC(=O)CCc1nccs1)NCCCC1CC(C)C1 CCC(F)(F)C(=O)NCc1nc(C(=O)N(C2CC3(CCC3)C2)C)co1 c1(C(N2CCC(CNC(=O)C(F)CC3CCCC3)C2)=O)coc2c(Cl)cccc12 c1(C(N(CCCCC(=O)N(c2cn(CC)nc2)C)C)=O)cc(C#N)oc1C N1(C(COCCC=C)=O)CCC(C)C(NC(C2CC2(c2ccccc2)C)=O)C1 CCC(CC(=O)Nc1nc(C2CCCCN(C(=O)CS(N)(=O)=O)C2)n[nH]1)C(F)F CC1=C(C(=O)NC2CN(C(c3oc(C)nc3C)=O)CC2C)CCCO1 C1(C(=O)NC(CNC(CCN2C(C)CCCC2)=O)C)CC(F)(F)CCC1(C)C N1(C(C2C(C=C)C2)=O)CCCCCC1C(=O)NCC(=O)NC1CCC1 C1(C(=O)NCC(N2CCN(C(c3n(C)c(S)nc3)=O)CC2)=O)CC2C(C1)C2(F)F C1(NC(c2ccc(CCF)cc2)=O)CC2CC(NC(C3(F)CC3)=O)CC12 c1(OC)ccccc1C(C)(C)C(=O)NCCC1(NC(=O)C2=CCSC2)CC1 N1(C(CC=CCC)=O)CCOC2(CCCN(C(c3nc(C)oc3OCC)=O)C2)C1 c1(CN(C(=O)C(F)C2CC2)CCNC(C2(CCCC)CCC2)=O)ccc(Cl)nc1 N1(C(C(C)OCOC)=O)CC(CNC(=O)Cc2coc(C)n2)C2(CCC2)C1 C(=O)(C(C)N(C)C(C1(C2C=CCC2)CC1)=O)NCC(C)C1CC1 C12(CNC(C#CC(C)C)=O)COCCN1CCN(C(c1nncs1)=O)C2 N1(C(c2ccc(C)cc2N)=O)CCC2(CC1)CN(C(=O)C(C)CCO)C2 CCCCC(C(=O)NC(CSC)CC)NC(=O)Cn1nc(C)nc1C C1(NC(CC2(C)CC2)=O)CCOCC1C(=O)NC1(C)CC(N(C)C)C1 c1(NC(C2(F)CN(Cc3c(C)scn3)C2)=O)ccc(O)c(Cl)c1 CC(CCC(F)(F)F)NC(=NCC1(OC(F)F)CCCSC1)NCC(C)(C)C C1(NC(C(Cn2ccc(C)n2)C)=O)CN(C(c2ncsc2C(C)C)=O)CC1(C)C c1(CNC(C(C)N2CCC2CNC(=O)CS(C)(=O)=O)=O)ncnc2[nH]cnc12 C1(C(=O)NC2CCC(NC(C3CN(C(N)=O)C3)=O)C2)CC(=O)NC(=O)N1 N1(C(C2N(C(=O)C=CCCC(C)C)CCC(=C)C2)=O)CCOC2(CCCC2)C1 C1(CC)(NC(=O)C(C)N2CCC2)CN(C(c2cc(CN)on2)=O)C1 C1(NC(c2ccn(C(C)C)c(=O)c2)=O)CN(C(=O)CC2CCCC2)CC2(CC2)C1 c1(SCC(CC)N(CCCN(C)C)C(C)C)cccc(COC)c1 C1(CC=C)(NC(=O)C(O)CCCC)CCN(C(C2CSCCS2)=O)CC1 N1(C(C(P(C)(C)=O)O)=O)CCCC2(C1)CN(C(=O)CC(C(F)F)n1cccn1)C2 N1(C(c2c(C)ccs2)=O)CCN(C(C2CCCC2C)=O)C2CCCC12 c1(OC)cccc(C(C)=CC(N2CCC(NC(C3CCC(C#N)C3)=O)CC2)=O)c1 C1(NC(CS(C)(=O)=O)=O)CCCCCN(C(c2cccc(S(=O)(=O)F)c2)=O)C1 C1(NC(C(CC)N(C)C)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)CC1F c1(C(=O)NCC2CN(C(C3C(CCOC)C3)=O)C2)cc(S(C)(=O)=O)oc1C C1(OCC)CCCN(C(c2cc(COC(C)(C)C)on2)C(=O)NC)C1 N1(C(CCC=C)=O)CCC(C(=O)NCC(O)C(C)C)C12CC2 C12(NC(C)=O)CCC1CN(C(c1ccsc1OC(F)F)=O)C2 N1(C(CCC(C)NC(=O)C=C2CCOCC2)=O)CC2NC(=O)OC2C1 C1(CC(=O)NCC2(CNC(c3c(C)n(C)cn3)=O)CCC2)COCC(C)(C)O1 N1(C(C(C(C)O)(C)C)=O)CCC(O)(C2(NC(=O)C3=C(Cl)CCCC3)CC2)CC1 N1(C(=O)C(=CC2CCCCC2)F)CCC2(CCN(C(=O)CO)C2)C1 c1(C(N2CCN(C(C3(F)CC=CC3)=O)CC2)=O)nc2ccccc2s1 c1(C(N2CCCC(C(C)NC(CNC(CC)=O)=O)C2)=O)cc(C)c(=O)n(C)c1 C12(NC(CCOCC)=O)CCCC(NC(c3cc(Cl)cnc3O)=O)(C1)C2 c12cccc3[nH]c(cc13)-c1noc(n1)C2(C)C.c1(COC)ccnc(F)c1 N1(C(C(C)O)=O)CCC2(C1)c1ncn(C)c1CCN2C(=O)CCCC(=O)C1CC1 N1(C(Cc2ncc(C)o2)=O)CC(CCNC(=O)COC2CC2)OC(C)C1 C(=O)(C(O)CC(F)(F)F)NC1CCC(NC(c2nc(CC)oc2)=O)C1 N1(C(C(C(C)C)F)=O)CCC2(CCC2)C(NC(c2ccsn2)=O)C1 C1(NC(c2c(NS(C)(=O)=O)csc2)=O)CN(c2cccc(Br)c2)C(=O)O1 c1(C(N(CC)CC2CCCN2C(C2CCC(=O)N2)=O)=O)cccc2sncc12 C(C(C)(F)CNC(C1(COC)CCCC1)=O)NC(C=CCOC)=O C(=O)(C(O)P(C)(C)=O)N(CC(C)(C)CNC(=O)COc1cn[nH]c1)CC c1(C(=O)OC)cc(SC(C2(OC(F)F)CCCCC2)C)ccc1OC c1(CNC(c2cc(COC)[nH]n2)=O)ncccc1C(=O)NCc1cc(C)no1 CC1C(NC(=O)COCC2CCCOC2)CCCN1C(C1CN(C(N)=O)C1)=O N1(C(C(C)OC2COC2)=O)CC(F)(F)CC1(C)CNC(=O)C(C)n1ccnc1 C1(CNC(=O)OCCCCC)CCCC2(CCC2)O1 CC(CNC(c1cnccn1)=O)CC(=O)N(C)Cc1nc(=O)o[nH]1 c1(CN(CCCCCC)C(C)C(C)NC(=O)OC(C)(C)C)ccnc(C(F)F)c1 Cc1ccc(F)c(C(=O)NC2CC(C)(NC(c3n[nH]c(C)c3C)=O)C2)n1 Cc1c(Br)ccc(O)c1C(N1CCC(CCNC(c2cccn2C)=O)C1)=O C1(CNC(c2c(C)cc[nH]2)=O)CCCN(C(c2ccc(C3CC3(F)F)cc2)=O)C1 N1(C(=O)NC2C=CC(NCc3cccc(-c4ccccn4)n3)C2)CCC(F)CC1 C1(C)(C(=O)Nc2c(COC)cccn2)CCCN(C(=O)CSc2nc[nH]n2)C1 c1(CC(=O)NCC(N(C(=O)CC2CC=CC2)C)C2CC2)ccc(C(F)(F)F)cn1 C1(NC(C2N(S(C)(=O)=O)CC2)=O)CCC(CNC(=O)CCc2ccccc2Cl)CC1 C1(C(=O)OC)(C(=O)OC2CCOCC2)CCNCC1 c1(CC(=O)NCC(C(C)(C)C)NC(CC(C)F)=O)ccc(Br)c(Cl)c1 Cc1ccc(Cl)c(N)c1C(=O)N(C(C)CNC(=O)CC1CC1(C)C)C C1(N(C(c2c(CNC(C3C(C)CC=CC3)=O)occ2)=O)C)CCCCC1(C)C C(=O)(C(C(C)OC)NC(c1ccc(C#N)[nH]1)=O)NCC(COCC)O c1(C(N(c2ncc3ccccc3n2)C(C(C(C)C)O)C)=O)cc(Br)cc([N+](=O)[O-])c1 Cc1oc(C)c(C(=O)NCCC2CCN(C(c3ccn(C(F)F)n3)=O)C2)c1C CC1CN(S(=O)(=O)N2CCN(C(c3cccnc3[N+](=O)[O-])=O)CC2)CC(C)O1 c1(-c2cc(C(=O)NCC(C)N(C(=O)CC3OCCO3)CC)[nH]n2)ccc(F)cc1 c1(C(N(C2CCN(C(=O)C=Cc3cn(C)cn3)C2)C)=O)ccc(N)cc1F C1(C)(CCC)CCCN(C(C2COCCN(CCn3cccn3)C2)=O)C1 Cc1ccnc(C(=O)NC2CCC(CCC(=O)N(C3CCCC3C#N)C)C2)c1N C12(CNC(c3c(CC)n(C)nc3)=O)CCC(CC1)N(C(=O)Cn1cnnc1)C2 C=Cc1cncc(C(=O)N(C)CC2CN(C(c3ccn(C4CC4)n3)=O)CCO2)c1 CCC(CC(=O)N1CCOC(CCCNC(c2cccn2C)=O)C1)C(F)F C(=O)(C1=CC2(CCN(C(c3cncc(-c4nn[nH]n4)c3)=O)C2)C1)OCC c1(C(=O)NC(Cn2cccn2)C(=O)NCCc2cscn2)ccnnc1O C1(c2n(CC=C)nnn2)(NCCCCC(=O)OC)CCCC(C#N)C1 S(=O)(=O)(c1cccnc1Cl)N1CC2(CCN(C(C3CCC(F)(F)CC3)=O)C2)C1 C(=O)(C(F)C1=CCCCC1)N1CCC(C)(CNC(=O)CC2(CO)CCCC2)C1 c1(C(=O)NC(CC#C)CC(=O)N2CC(O)C(F)C2)ccc(C)c(C#C)c1 C1(NC(C(C)(C)OC(C)C)=O)CCCN(C(C2(C#N)CC2)=O)CC1 N1(C(C23CC(C)(OCC2)C3)=O)CC(NC(=O)Cc2cncnc2)CC12CCOC2 c1(C(=O)NCC(C)NC(c2nccc(CC)c2)=O)cccc2c1CNC2=O c1(CCC)cc(C(=O)N(CC(O)CNC(c2c(C)n[nH]c2C)=O)C)sc1C c1(CN2CCC(C(=O)Nc3nnc(-c4cccc(Cl)c4)s3)C2)ccc(Br)c(Cl)n1 c1(N2CCN(C(C(C)(CF)c3ccccc3)=O)CC2)cccc(O)c1Br C1(C(N2C(CC(=O)NCC(n3ccnn3)C)CC(F)C2)=O)CC12CCOCC2 c1(C(N(CC(CC)NC(=O)C(C)=C(C)C)C)=O)cn(C)cc(Br)c1=O CCC(C#N)C(=O)NCC1(F)CC(NC(c2ccc(O)nc2)=O)C1 C12(C(=O)NC3CN(C(C=CC(c4cn(C)nc4)=O)=O)CC3F)CCCN(CC1)C2 c1(C(N2CC(NC(C3C(C(=O)OC)C3)=O)C(C)C2)=O)cnn2cccc(Br)c12 N1(C(COC(C)=O)=O)CC(CNC(c2cc(Cc3ccnn3C)[nH]n2)=O)CC1C N1(C(C2(CC(=O)NCC(=O)N(C)C)CC2)=O)CC(C(C2(CSC)CC2)=O)C1 C1(C(N)=O)(CNC(C(C2CC2)OC)=O)CN(C(c2cc(C3CC3)n[nH]2)=O)C1 c1(NC(c2n(CC=C)nnn2)CC2CCOCC2)ccc(C2CC2)c(C)c1 c1(C(C)NC(=O)C(=O)NC2CCCCC2(F)F)cccc([N+](=O)[O-])c1 c1(CN2C(C)(C(=O)NC(c3ccccc3Cl)CO)CCC2)ccc(F)cc1O N1(C(C2C(C(C)(C)C)C2)=O)CCCCC(C2CN(c3nc4ccccc4o3)C2)C1 C1(CC(=O)NC2CC(NC(C3CC(OC)C(OC)C3)=O)C2)CCCCC12CC2 c1(C(N2CCCC(C)(NC(C(CC=C)C)=O)C2)=O)nc2sc(C)cn2c1C CCCCC(CC)C(=O)N1CCC(C2(NC(=O)Cc3sc(O)nc3O)CC2)C1 N1(C(c2c(C)oc(C)c2C)=O)CCC2(CC1)COC(CNC(=O)C1CC1)C2 c1(C(=O)NCC(C2CCCC2)NC(C(C)NC(C)=O)=O)cnc2ccccc2c1 C(N=c1[nH]c(C)c(C(N2CCC(OC)C(F)(F)C2)=O)s1)c1cnc(SCC)s1 C1(CNC(c2c(SC)ccs2)=O)CN(C(=O)CCC(F)F)CCC1(F)F C(N=C(NCC1CCCO1)N1CCCC(CF)C1)c1cccc(OC)c1O N1(C(Cn2ncc(C(=O)OC)c2)=O)CC2CC2(CNC(c2ccc(SC)s2)=O)C1 N1(C(C(C)N(C(C(CCC)C)=O)CCC)=O)CCC(C)(C(=O)OC)CC1 N1(CCC(=O)NCC2C(NC(CCc3nnc(C)o3)=O)CCC2)CCC(O)CC1 C1(CC)CN(C(c2c[nH]c(C#N)c2)=O)CCN1C(C1CCC(F)(F)CO1)=O N1(C(C2(NC(CCC(C)=O)=O)CCSC2)=O)CC2CCC(C1)C2C#N C1(C(=O)NCC(C)N(C(c2nnn(CC)c2C)=O)C)CCc2nnc(O)cc2C1 c1(C(=O)NCC2CN(C(=O)CN3CCOC3=O)CC2O)cc2cc(Cl)ccc2s1 N1(C(=O)CC2OCCO2)CCCC2(C1)CN(C(=O)Cn1cnnc1)CCO2 c1(OC)coc(C(=O)NC2CCCCC2CNC(C2(C)C=CCC2)=O)cc1=O N1(C(C2(SC)CC2)=O)CC(C(=O)NCC2CCCC(C)(C)C2)C2(CCC2)C1 O=C(NNc1ccc(Br)c(F)c1)NCCNS(=O)(=O)C1CC1.C12(CC1)CC2 C1(CCCNC(C2CC2(F)F)=O)CCCCN1C(c1cc(Cl)c(Br)s1)=O c1(N2CCCCC(C)C2)nc(N2CCC(OCCO)CC2)nc2ncn(C)c12 C(=O)(CCCCCn1cc(C2CC2)nn1)N(CC1CCCN(C(C)(C)C)C1)CCOC C1(C(N2CCC(OCCNC(c3cc(CC)sc3)=O)C2)=O)CN(CC)C(=O)N1 C#Cc1cccc(C(N2CCN(C3CCN(C(=O)C(C)CO)CC3)CC2)=O)c1Cl Cc1cncc(C(=O)N(CCNC(c2coc(Cl)n2)=O)C2CC2)n1 c1(C(=O)N(C(C)(CO)C2CCC2)CCO)ccc2occ(CCC(=O)OC)c2c1 N1(CCCCOC)CCC(CNC(c2ccn(CC(C)C)n2)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2CCCCS2)=O)cncc(Br)c1 C1(CNC(c2c(C)cccc2)=O)CC2(CC(NC(c3cc(Cl)cn3C)=O)C2)C1 N1(C(COc2cccc(C(=O)OC(C)(C)C)c2)=O)CC(CO)CC12CCC2 c1(CN(C(C2CCCOC2)C(=O)NCC)C)cc(OC)cc(CC)c1 c1(OC)cc(OC)c(C(=O)NCC2(NC(=O)C3=CCCS3)CC2)cc1OC c1(C(N2C(C(=O)NCCCCCOC)CC(F)C2)=O)ccc(OC)c(F)c1 Nc1nc(Cl)ccc1C(=O)NCCCCCNC(=O)C(F)(F)CF C#CCC(CO)NC(=O)C(CO)NC(=O)CCc1cncnc1 C1(CC(=O)NCCN(C(C(C)c2cc[nH]n2)=O)C)CC(F)(F)C1 C1(CNC(=O)OC(C)(C)C)CC(F)(COCC2CC(C(=O)NC3CC3)C2)C1 c1(OC(C)C)cccc(C(=O)NC2COC(C(F)F)C2)n1 C1(NC(CN(CC)CC)=O)C=CCN(C(=O)CC2(CC)CCC2)C1 N1(c2snc(C(=O)OC)n2)CCC(CNC(=O)CSc2ccccn2)CC1 C(CCCCC(=O)N1CC(OCCNC(c2cc(C3CC3)ccc2Cl)=O)C1)OC c1(NCC(=O)N(CC(C)C(N2CCC(O)C(C)C2)=O)C)ccc(C#N)cc1 CN=c1[nH]c(CNC(=O)NCC2CN(c3nnc(O)s3)C2)cs1 C1(C)(CC)CC(NC(=O)Cc2ccccc2)CN1C(=O)CCc1cccnc1C N1(C(C2CC(OC)C2)=O)CCN(C(c2oc(SC)cc2C)=O)C2CCC12 C1(OC(C)(C)C)COCCN1C(=O)OCc1cccnc1Br c1(C(N2C(CNC(C(C)Cc3ccncc3)=O)CCC2)=O)cc2ccncc2s1 CCS(=O)(=O)CC(=O)NCC1CC1NC(c1cncc(NS(C)(=O)=O)c1)=O C1(C(=O)NCCN(CCCCCCN(C(CCCOC)=O)C)C)OC2CCC1CC2 C(=O)(CP(C)(C)=O)N1CC(C)(CCC(N2C(C)CC2CO)=O)C1 C12(NC(c3cc(F)c(Cl)cc3F)=O)CCCC1N(C(=O)C1=CCC1)CC2 C1(C(N2CCN(C)CC2CNC(=O)CCCC2(C)N=N2)=O)CCOC2(CCC2)C1 Cc1cc(S(=O)(=O)N2CCCCCCC2C(=O)N(C)C)ccc1-c1ccno1 C1(NC(COC2(C)CCC2)=O)CCC(C(=O)NCC2(C)CCCCO2)CC1 C1(C(=O)Nc2c(CCN(C)C)noc2)CN(C(=O)OC(C)(C)C)CC1F c1(C(N2CC(O)(CCNC(c3cc(C(CC)C)no3)=O)C2)=O)ccc(Cl)cc1F N1(C(C(C(CNC(CCCOC(C)C)=O)C)F)=O)CCc2n[nH]cc2C1 c1(C(N(CC(C)NC(=O)COC2(C)CCCC2)C(C)C)=O)cc(O)n(C)n1 C#CCCN=C(NCC1(C)CCOC1)N1CCN(c2ccccn2)CC1 CC1(CNC(c2ccccc2CC#N)=O)CCN(C(C2CC3CCCC23)=O)C1 C1(CC=C)(C(=O)NC2(C)CCCC2)CCCN1C(=O)CC1CCCNC1=O c1(C(=O)NCC2(C(N3C(COC)CC3)=O)CC2)ccc(-c2ccncc2)nc1 N1(C(c2cnn(CC(F)F)c2)=O)CCCC2CN(c3ncc(F)cn3)CCC12 C1(CC=C)(C(=O)NC(c2ccsc2)C)CCCN1C(=O)C(C=C)OC C1(C(=O)NC2CC(C(C)C)OC2)(CC(c2cncn2C)=O)CCN(C)C1 C(C(=O)NC1(CN2CCCCCC2)CC1)(C(C)C)n1ccc(C)c1 c1(OC)ccc(F)c(CC(=O)NC2CN(C(=O)Cn3cc(C)cn3)C(C)(C)C2)c1 N1(C(=O)Nc2c(C)cc(C#N)cc2)CC2CCCC(C(N3CC(O)C3)=O)C2C1 CCC(C)C(C(=O)N1CCC(C(=O)OC)C1)NC(c1ccc(C)nn1)=O N1(C(=O)NC(C)C(C)n2ccnc2)CCC(N2CCC(C#N)C2)CC1 C(=O)(CC(C)CC(=O)N1CC(O)CC1CNC(C12CC(C)(CCO1)C2)=O)OC C1(NC(C(C)N(c2ccccc2F)C(=O)COC)=O)CCOC(c2ccccc2)O1 N1(C(c2c(OC)cc(Br)cc2)=O)CCC(C)N(C(=O)CC2(C#N)CC2)CC1 N1(C(c2cn(C)nc2Br)=O)CCC2(CC1)CC2(C#N)CO c1(CNC(C(C)S(N)(=O)=O)=O)cccc2c1CN(C(c1cc(C3CC3)cs1)=O)C2 c1(C(N2CCC(CNC(=O)C(F)Cc3ccccc3)C2)=O)ccc(O)cc1O N1(C(c2n(COC)ncc2)=O)CCCC(O)(CNC(c2csc(COC)n2)=O)C1 N1(C(C(C)=C(C)C)=O)CCC2CCN(C(=O)C(n3cc(Cl)cn3)C)CC12 c1(C(N2CCCC3(CNC(c4ccnnc4)=O)C2C3)=O)cc(F)c(F)cc1F N1(C(c2cc(COC)[nH]n2)=O)C(C)CN(C(=O)C(C)(C)C(F)(F)F)CC1C CN1CC(NC(C2C3CN(C(=O)OC(C)(C)C)CC23)=O)Cc2ccccc21 C1(NC(Cc2cc(C)no2)=O)CS(=O)(=O)CC1NC(C1CCC(O)CC1)=O C1(C(=O)NCC(CC=C)NC(C2CCC2C#N)=O)CC(C)CC(C)C1 c1(OCC)cc(NCCC2CCC(NC(=O)CCc3cc(C)no3)C2)nc(C)n1 CCC(C)C(CC(=O)N(C)CC1(C#N)CC1)NC(=O)C(C(C)C)C(C)C N1(C(c2nc(-c3ccc(CC)cc3)oc2C)=O)CCN(CC(C)O)C(C)C1 Cc1nnccc1C(=O)N(CCNC(=O)CCc1ncc(F)cn1)C1CC1 C(=O)(C(F)C(F)(F)F)NC12CC(NC(=O)CCC(=O)c3ccccc3)(C1)C2 Cc1cc(C(=O)OCC(=O)Nc2cnc(C)nc2)n2nccc2n1 c1(NC(CN(C)CCOc2ccccc2Cl)=O)cccc(F)c1 N1(C(c2c(C)noc2N)=O)CCCC(CO)(NC(=O)C(O)P(C)(C)=O)C1 c1(NCC(c2ccccc2)CNC=O)ccc(-c2ccccc2)cn1 C1(C(=O)NC(CCCNC(c2cn(CC)nn2)=O)C)CCC(C#N)CC1 C1(CNC(c2oc(CC)c(C)c2)=O)CCC2CN(C(C3(C)CCNC3=O)=O)CC12 N1(Cc2c(OC)nsc2)CCC(NC(=O)CC(=O)Nc2cccc(C)c2)CC1C C12(CNC(c3c(NC)cncc3)=O)CCC(NC(=O)COCC(C)C)(CC1)CO2 C1(CNC(CSCCC)=O)CCCC2(CN(C(=O)CC(C)CC)C2)O1 CC(CC#N)C(=O)N1CCC(NC(=O)CCCOC2CCOCC2)C1 C1(C)(CNC(C2(OC)CCCCC2)=O)CN(C(=O)C(O)CCC(C)C)C(C)(C)C1 CC(C)CC(F)C(=O)NC1CC(CCNC(c2n[nH]c(C3CC3)n2)=O)C1 N1(C(CC(=O)OCC)=O)C(C)CC2CN(C(c3cc(C)c(C)nn3)=O)CC12 Cc1ccnn1CC(N1CC(C)(C(=O)Nc2cnn(C(C)(C)CO)c2)C1)=O c1(C(=O)NC23CC(C(=O)NC(c4cccc(Cl)c4)C)(C2)C3)ncc(Br)cc1Br C12(CCN(C(c3c(C)noc3)=O)CCO)CCC(C1)N(C(=O)CNC(=O)C1CC1)C2 C1(NC(c2c(Cl)cccc2Cl)=O)CCCCN(C(C2(O)CCOC2)=O)CC1 Cc1cc(C(=O)N(c2ncc(Br)cn2)C2CCNCC2)nn1-c1ccccc1 C(=O)(C(C)CCCCCC)NCC=C.C(=O)(CCC1CC1(C)C)N(CC=O)CC#C N1(C(=O)C=Cc2ccsc2)CCC2C(CCCN2C(=O)CN2CC3C=CC2C3)C1 C=CCC(CC(=O)NCC1CCCCN1C)NC(=O)C(C)(C)OC(C)=O C=CCC(C(=O)NC1CC(NC(c2ccc(OC(F)F)c(Cl)c2)=O)C1)C(C)(C)C CCC1=C(C(=O)NCC2(C)CCCN2C(c2cc(N)cc(F)c2)=O)CCCO1 CCC(CC(=O)NC(C)(C)CCCF)NC(=O)Cc1coc(C)n1 N(C1CN(C(C2CC(C)(C)C2)=O)Cc2ccccc21)C(c1c(C)n(C)cc1)=O C=CCCC(CO)NC(C1CC1CNC(=O)C(C(C)C)OC)=O C12(C(C)NC3CCN(c4snc(C)n4)CC3O)CC3CC(CC(C3)C1)C2 C1(C(N(C)CC2CCCN2C(=O)CCN(C2CCCCC2)C)=O)COCCC1(F)F N1(C(Cc2ccc(C)s2)=O)CCN(C(=O)CCCCC#N)C(C2CCCC2)C1 C=C1CC2(C1)CC(C(=O)NC(CNC(=O)C(C)(C)c1nncn1C)C(C)C)C2 O=C(O)C(C(O)c1ccc(F)cc1)NCc1ccnc(Cl)c1 N1(C(C2NC(=O)CC(C)C2)=O)CC2CCN(C(=O)CCP(C)(C)=O)C2C1 C(C(C(=O)NC(CC)(CC)C(C)C)C(C)(C)C)NC(C(CC=C)OC)=O CCC(CN(C)C)C(=O)N1CC(C(N2CCOC(CN=[N+]=[N-])C2)=O)C(F)C1 Cc1nncc(C(=O)NC(c2ccccc2)C(N2CCCCCCC2)=O)c1C C(=O)(C1=CS(=O)(=O)CCC1)N1CC(CNC(C(C)(C)Cc2ccc(O)cc2)=O)C1 C(CCc1ccccc1)(C(C)O)N1CCC(N(CC)Cc2nc(CSC)cs2)C1 c1(C(C2CCOC2)C)cn(CCN(C(c2coc(Cl)c2)=O)C2CC2)nn1 C1(C(C)C)CC(O)CN1C(=O)CC(C)(C)N(C)C(C1OCCC1C)=O c1(C(N2CCC(O)CC2)C(=O)NCCCSC)cncc(C)c1 C1(C2CCC2)(C(=O)NCC#CCNC(=O)CCCc2ccsc2)CC1 Cc1cccc(F)c1CC(N1C2CCC1C(NC(=O)C(c1ccnn1C)O)C2)=O C1(NC(C23OCCC(C)(C2)C3)=O)CCC2CN(C(c3cnc(Cl)[nH]3)=O)CCC2C1 c1(CC)ncncc1C(=O)NC(C(=O)NCC1(COC)CC=CC1)c1cccs1 CC(C)C(CCC(=O)NC(CC1CCCC1)CO)NC(C1CC2(CC2)C1)=O C1(C(=O)NCC(CNC(c2c(C)noc2N)=O)O)COc2ccc(Cl)cc2C1 C12(NC(c3ccc4nc[nH]c4n3)=O)COCCC1CN(C(=O)C1=CCOC1)C2 CCC1=C(C(=O)NC2CC(F)CN(C(=O)C=C(C)C3CC3)C2)SCCO1 CC#CCC(C(=O)N1CCOC(C)(C2CC2)C1)NC(c1csc(Cl)c1)=O CCC(C)C(O)C(=O)NCCCC1CCCCN1C(c1cc(C)n(CC)n1)=O C1(CNC(C2(CCSCC)CCC2)=O)CC(F)(F)CN1C(=O)CC1CCCO1 c1(C(=O)NC2(CCNC(c3c(SCC)cccn3)=O)CC2)cccn2nnnc12 Cc1cccc2oc(=NCC(O)CNC(C3Cc4cncn4C(=O)N3)=O)[nH]c12 C1(NC(C2C(C)C2)=O)CC(NC(c2nscc2Br)=O)C(O)C1 c1(C(C)C)[nH]nc(C(=O)NC(CO)C(C)NC(=O)C2=NOCC2)c1Br c1(C(=O)NC2CCCN(C(c3cccc(OC)c3)=O)C2)cc(C)c(O)c(C)c1 C(=O)(C1=Cc2cccc(Br)c2OC1)NCCC(C)NC(C(CCCC)CC)=O c1(NC(CCSC)C)ccc(S(=O)(=O)NCCC2CCCCCC2)c(Cl)c1 C(N=c1cc(NCCc2cn(C)nn2)nc(C(F)(F)F)[nH]1)C1CCC(C)N1C C12(C(=O)NCC#CCNC(=O)C(c3ccc(Cl)cc3F)O)CC1CCC2(F)F N1(C(CC(CNC(C(C)(C)NC(=O)OC)=O)O)=O)CCC2(CC1)CC2C#N C1(N(c2scc(C)c2Cl)C(=O)CSC(C)(C)C)CCN(CC)CC1 C1(C(N(C)Cc2snc(C)n2)=O)CC2C=CC1N(C(=O)CC1(N(C)C)CC1)C2 C1(CC(C)(C)C)NC(=O)CCN(CCC2CCCCO2)C1=O c1(CNC(C2(CCC)CC2(F)F)c2nnnn2CC)cnc(Cl)cc1Cl N(C1CCCn2nc(CCNC(C)C(=O)OC)nc21)C(CC(CCC(=C)C)C)CO c1(SCC(=O)NCC2(NC(c3ccc(F)cc3)=O)CCC2)ccccc1F CCCC(C)C(=O)NC(C)(C)CCNC(c1scc(C)c1Cl)=O C#CC1CCN(C(=O)Cn2cc(CNC(c3ccsn3)=O)nn2)CC1 c1(NCCN(C)C(c2ccoc2Br)=O)ncnn2c(Br)ccc12 c1(C(=O)NCC2CCCC(NC(c3cc(C)c(C)o3)=O)C2)cc(Cl)c(F)cc1N C(=O)(CC(COC)COC)NCC(C(C)(C)C)NC(C(C1CCCC1)OCC)=O CC1=C(C(=O)NC(C)C(C)C(=O)NC23CCC(CC2)CC3)SCCO1 c1(C(=O)NC(CNC(CC(=O)NCC#C)=O)C(C)C)ccnc(CO)c1 C1(CC(N2C(CC(C)(C)C)CCC2)=O)CC2(CC2)CO1.c12ccn(n1)C1CC1C2 Cc1nc(C2CC2)ncc1C(N1CC(C(C)NC(c2ccc(CO)o2)=O)C1)=O C1(C(N2CCC(C(=O)NC(c3ccc(F)cc3)C)(OC)C2)=O)CN(C)CCN1C C(=O)(C(F)CCC(C)(C)C)N1CC(C(C)NC(C2C=CCN2C2CC2)=O)C1 C1(CC(=O)NCC2CCN(C3CCCCC3)C2)CC12CCOC2 CCC(CCc1ccccc1)C(=O)N1CCC(CNC(C2CC(=C3CC3)C2)=O)C1 CC1CC=CCC1NC(=O)CC1C=CC(NC(=O)CCC2CC2(F)F)C1 c1(-n2ncc(C(=O)NC(CN(C(CCOCC#C)=O)C)C)n2)ccc(Cl)cc1 C(=O)(C(O)CCCC)N1CC(C#C)(C(=O)N)C1.c1(C(C)C)ccncc1 C1(OC)CN2CCCC2(C(N2CCC(n3nc4ccccc4n3)CC2)=O)C1 CN1CCOCC1CC(=O)NCCN(C)C(C1CCCC1c1cn(C)nn1)=O c1(CC)cncc(C(=O)NCC(C2CCOC2)NC(=O)CCCOC)c1 c1(C(N(CC(C)NC(=O)CC2CC=CC2)CC)=O)cnn2ccn(C)c12 C(CC(=O)N1CCC(C)C(O)C1)(C(F)(F)F)NC(c1ncc(CC)cn1)=O c1(C(=O)OC)nccnc1NC(=O)CC1(N)CCOCC1 c1(C(=O)OC)ccc2c(C(F)(F)F)cc(=O)oc2c1.c12cc(cs1)CC(=O)O2 N1(C(C2CCC(C(CC)(C)C)CC2)=O)CCC2C(C1)NC(=O)CCN2C c1(NCC(=C)F)cc(=NCc2nc(SC)n[nH]2)[nH]cn1 C(CC(=O)NCC1CC12CC2)(C(F)F)NC(CCN(CCC)C)=O c1(Nc2c3nc(N(C)C)oc3ccc2)ncnc2c1nnn2C1CC1 Cc1cc(C#N)c(F)cc1NC(c1cc2ccc(-c3ccsc3)nc2[nH]1)=O N1(C(c2nccc(CC)c2)=O)CCC2C(CCN2c2nc(C)ncc2F)C1 c1(C(=O)NCCCN(C(=O)C=C2CCCCC2(C)C)C)[nH]nc2c1COC2(C)C C1(C(=O)NCCc2n(CC)cnn2)CC=CCC1NC(=O)CSC(F)F c1(CC)oc2ccccc2c1CC(N1CCC(CNC(=O)CC(C)(C)O)C1)=O N1(CC2CC(SC)C2)C(=O)CCN(CCc2cccc(F)c2C)C1=O C1(CNC(CCCCOCCC=C)=O)CC2CN(C(=O)C(C)(C)C(C)C)CC12 C(CCC(C)C(=O)NCCC1CN(C(c2cncc(C)n2)=O)CCO1)OC C(=O)(C1=CC2CCC=CCCC12)NC1CC(OCC)C12CCOCC2 Cc1ccc2c(-c3cn(CC4OC(CO)C5OC(C)(C)OC45)nn3)cccc2n1 N1(C(CC2C(CC)C2(F)F)=O)CCCC(CCNC(=O)C(C)CCOC)C1 C1(NC(CC(COC)C)=O)CC2CN(C(=O)Cc3ccon3)CC2C1 c1(OC)ccc(OCC(=O)NC2C3CC2N(C(=O)CCN2CCOC2=O)C3)cc1 c1(C(=O)NCC(CO)NC(c2c(CC)ccs2)=O)cc2c(F)cccc2s1 C(=O)(C1=NNC(=O)CC1)N(C(CNC(Cc1cc(C)cc(F)c1)=O)C1CC1)C CC1CN(C(c2csc3nccn23)=O)CC(C)C1NC(=O)CCOC1CCCC1 CC(=O)C(C)CCN1CC(c2noc(C(F)F)n2)C1 C1(C(N2CC(OCC)C2)=O)CN(C(=O)CSc2cn[nH]c2)C(C)(C)C1 C1(CNC(C2CC2c2ccc(F)cc2)=O)(CO)CCCN(C(=O)C2=CCCC2)C1 N1(CC(=O)NC2(C(N3CC(C(N)=O)C3)=O)CC(F)C2)CCCNC1=O c1(C(N(C)CC2CCCC(NC(CCC(=O)NCC)=O)C2)=O)ccc(Cl)c(C)c1 C1(C(N2C(CN(C(C3(OC)CCCOC3)=O)C)COCC2)=O)CCCCCCC1 n1(CC(=O)N(C(C)CNC(C2CC(CF)C2)=O)C)cccc(C(F)(F)F)c1=O c1(CNCCCCn2cc(-c3cn(C)nc3)nn2)nnc(-c2cccs2)n1C CCCC(C(=O)NC1CC(C(N2CC(F)C2)=O)C1)OCC N1(C(C(C)OCOC)=O)CCC2(C1)CN(C(c1nccc(OC)c1F)=O)CCO2 c1(CC(N2CC(N(C)C(C3CC(c4ccccc4)CO3)=O)C2)=O)ccc(Cl)cn1 C1(NC(C2CCC(OC)C2)=O)CCN(CCNC(c2cc(C(C)=O)[nH]n2)=O)CC1 c1(OC)ccc2c(c1)C(N)(C(=O)c1cnccc1SC)CC2 c1(C(N(CC(C)O)CCNC(CC(CC)(F)F)=O)=O)ccc([N+](=O)[O-])cn1 CCCC(C)CC(=O)N(CCNC(c1cn(C)nc1Oc1cccnc1)=O)CC C(CS(=O)(=O)CC(=O)NCC(CC1CC1)C(=O)NCC(N)=O)OC c1(CC)nc2ccc(Br)cn2c1C(N1CCC(C(C)(C)O)C1)=O C1(C(=O)NCC(O)O)(SCCNC(c2ccc(C3CC3)cn2)=O)CCCCO1 C1(C(=O)NC(CC)(CNC(=O)CCN2CCCC2)CC)CCC2C(CC1)C2(F)F c1(C(N2CCC(CNC(c3c(C(C)C)scn3)=O)C2)=O)cc(Cl)cnn1 N1(C(C(n2cc(Cl)cn2)C)=O)CCCC2CN(C(=O)C(F)=CC3CC3)CCC12 c1(CN2CCN(CCNC(c3cccc(C)c3I)=O)CC2)ccc([N+](=O)[O-])cn1 C(=O)(C1=CC2CCCC12)N1C(CNC(c2c(C#N)cncn2)=O)CCC1 c1(C(N(C(C(=O)NCc2cc(C)no2)(C)C2CC2)C)=O)ccc(O)cn1 c1(C(=O)NC2(C)CCN(C(C3CC4CC3C3CC43)=O)C2)ncnc2ccsc12 c1(C(C(=O)NCC)N(C)Cc2cccc(F)c2)cc(C(F)(F)F)nn1C c1(C(=O)NC2(CC=C)CCN(C(C3(C)CC3(F)Cl)=O)C2)nc[nH]c2ncnc1-2 C(C(=O)N1CC(NC(C2CC(F)C2)=O)C(F)C1)(c1ccccc1)=C(C)C C1(OC)CC(CC(=O)NC2CC(C)(Nc3ncncc3C)C2)C1(C)C C1(C(=O)NCCC2CCN(C(CCC#C)=O)C2)CCCN(CC)C1 C1(N(C(c2cc(SC)n(C)n2)=O)C)CC2CCC(C1)N2C(=O)CC(C)N(C)C CC(C)C(C(=O)OC(C)(C)C)C(=O)NCC1(C)CCCN1C(=O)Cn1ncnn1 CC(CC(=O)N1CCN(CC(=O)NCC2CN(C)C(C)(C)C2)CC1)C(C)(C)C N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CC(NC(C2CC(O)C2)=O)C(N=[N+]=[N-])C1 N1(C(c2cc(CCC)[nH]n2)=O)CC2CCC(C1)N2C(C1(c2cc[nH]n2)CCC1)=O C(CCCC(CC1COCCO1)C(=O)Nc1cccc(Br)c1)OC(C)C c1(OC)ncc(C(=O)NC2CCC(NC(=O)C(F)=CCCF)CC2)cc1C C(=O)(C(C(C)(C)C)OC)NC(CC(=O)NCC(CSC)OC)C C1(C(N(C)CC2CCCN(C(=O)COCCF)C2)=O)CCCCC(C)(C)C1 C1(C(C)C)CN(C(=O)CNC(N)=O)CCN1C(=O)CSc1nccs1 c1(C(=O)NC2CC3(CN(C(C4C(SC)CCC4)=O)C3)C2)ccc(C)c(C)c1N N1(C(c2c(F)cc(C)c(F)c2)=O)CC2CS(=O)(=O)CC2(NC(=O)OC(C)(C)C)C1 S(=O)(=O)(c1cccc(Br)c1F)NC1CN(C(CCNC(C)=O)=O)CC1F Cc1onc(CO)c1C(=O)NC(CNC(=O)CCc1ccc(Cl)cc1)C1CC1 c1(C(=O)NCC(CNC(C=COCC)=O)F)sc(C(F)(F)F)nc1C1CC1 CC1(C)CCCC(C(N2CCN(CCNC(C3CCCOCC3)=O)CC2)=O)C1 c1(C(N2CC(N(C(C)=O)C)C(F)C2)=O)cc2c(Br)cccc2cn1 c1(-c2cc(F)cnc2)cc(F)cc(C)c1NC(c1ocnc1C)=O.C(=O)OCC CCCCCC(O)C(=O)N(C1CN(C(C2(c3cccc(F)c3)CC2)=O)CC1O)C C1(NC(C(Br)=C(C)C)=O)COCCC1CNC(C1(C#N)CC1)=O C(=O)(C(CC(F)F)NC(=O)CCn1ccnc1)N(CC(C)CO)C C1(NC(C(C)SCC)=O)C(CN=c2[nH]nc(C3CC3)s2)CCC12CCC2 C1(C(=O)NC)CCN(C(=O)C(CO)NC(c2c[nH]c(C)c2)=O)C1C c1(OC)cccc(C(=O)NCC2(NC(=O)CCCC(=O)C3CC3)CCC2)c1C C1(NC(C(=O)N(C(C)C)C2CC2)=O)C2CCNCCC12.c12ccc(cc1)oc2=O C1(C(N2CCC(NC(C(CC)(C)CC)=O)C2C)=O)CCn2ccnc2C1 c1(C(C)(N)C(N2CCC(O)(c3cccnc3)CC2)=O)ccc(F)cc1Br C(=O)(CCCCC(C)=O)NCC(CC(=O)NC(CC)C(C)CN(C)C)O N1(C(c2ncn(CC)c2)=O)CCN(C(=O)CCN2CCC2)C2CCCCC12 C1(n2cccn2)(C(=O)NC(C(CCC)C)C)CCN(C(c2cccnc2O)=O)CC1 C1(CCC)CN(C(c2c(C)noc2CC)=O)CC1NC(=O)Cn1cccn1 N1(C(C(C)OCC2CC2)=O)CCC(CCNC(C2(CF)CC2)=O)CC1C C1(C)(CCC)CC(C(C)(C)C)=NO1.C(N=c1cnc(C(=O)NO)c[nH]1)c1c(C)cccc1N c1(C(=O)NCCCN(C(C(=Cc2ccccc2)C)=O)C)ccc(F)c(F)c1 c1(CC)cc(NC(C2CC3(C2)CN(S(=O)(=O)c2cn[nH]c2)C3)=O)ccc1Br N1(C(C(F)=CCC)=O)CC(C2CCCN(C(C3(C4(O)CCOC4)CC3)=O)C2)C1 c1(CC(N2CCN(C3CCCC3C(=O)O)CC2)=O)c(Cl)cccc1Cl c1(C(N2C(COCC)CCCC2)=O)cccnc1N1CCCCC1 C(=O)(C1=CC2CCCCC12)N1CC(N(C(=O)C(C)(C(C)C)OC)CC)C1 CC(C)(C(=O)NCC1CN(C(c2ccc(-c3ccccc3)cc2)=O)C1)C(F)(F)F C(=O)(CC(C(C)C)C(C)C)N1CCN(C(c2cc(COC)sc2)=O)CC1C1CC1 CS(=O)(=O)CCCN1CCC(NC2CCOCC2)CC1 c1(C(N(CCNC(c2sc(F)cc2C)=O)CC)=O)ncnc2c1CCCC2 c1(C(=O)NCC2C(NC(Cn3ncc(C(=O)OC)c3)=O)C2)ncnc(C)c1OC C(CCC(C)C(=O)N1CCN(C(=O)Cc2ccsc2Cl)C(CS(C)(=O)=O)C1)OC c1(C2(C(=O)NC3(O)CC3)CC2)cc(CC(=O)N)no1.C1(C(=O)OCCC)CCC1.C C(C1(O)CCc2ccccc21)N(C=O)Cc1nc(Br)n2c1CNCC2 n1(CC)c(O)nc2ccc(C(=O)NCC(C)N(C)C(c3cn(C)c(C)n3)=O)cc12 c1(NCC(C(=O)NC)(C)C)ncnc(NC2CCCC(CNN(C)C)C2)c1C C1(CNC(=O)C2=CCOCC2)CC12CCN(C(C1CCC(F)CC1)=O)CC2 C1(C#N)(C(N2CCC(N(C(C3CN(CCC)C(=O)C3)=O)C)CC2)=O)CCCCC1 n1(CC)nnc(C(N2CCC2CNC(=O)CCc2n[nH]c(=N)s2)=O)c1C CC1(C)CC(CC(N2CCC(CNC(=O)COCC3CCCCCC3)C2)=O)CO1 OC1CCC2(CC1)CC2CNc1ccc2c(c1)CCC2 c1(CC(C(=O)OC)NCc2ncc[nH]2)cc(F)ccc1Cl C1(NC(C(=O)Nc2ccc3oc(O)nc3c2)=O)COC2(CCCCC2)C1 CS(=O)(=O)c1cccnc1NCC1CC2CCC1N(C(C1CC3CC3C1)=O)C2 N1(C(C2(CCC)CCC2)=O)CC2CC2(NC(=O)C=Cc2ccncc2)C1 C1(C(=O)OC2C(OCCS(=O)(=O)NC)CCC2)CC(C)OC(C)C1 c1(OCC)ccccc1C(N1CC(C(N)=O)(CNC(c2nccnc2N)=O)C1)=O c1(CCNC(=O)CC2CN3CCN2CC3)nc2ccc(Br)cc2[nH]1 N1(C(C(F)=CCC)=O)CCCC(CNC(=O)C(c2cnn(C)c2)OC)C1 CC(C)C(C(C)C)C(C(=O)NCCNC(=O)C1CC1)N1CCC(O)C1 c1(CC)nc(C)c(N(C(N2CCCC2CCCO)=O)Cc2ccccc2O)o1 c1(C(=O)NCC(C)(C)NC(c2ccnn2C2CCOCC2)=O)cn(C2CC2)cn1 C1(NC(c2nc(CNC(c3n(C)nnc3)=O)oc2)=O)CCCC2(C1)N=N2 C1(CNC(c2cccnc2CO)=O)COCCN1C(=O)Cc1ccns1 n1(CC(=C)C)nc(CCC2CCCN2C)nc1-c1csc(C(F)F)n1 CC(C)C(CNC(=O)CCC(C)(C)F)C(=O)NCC1CCC=CO1 c1(C2(C(N3CCC(N4CCC(N)CC4)C3)=O)CC2)ccc(F)nc1Br CCS(=O)CC(=O)NCC1(C(C)(C)C)CCN(C(c2cc(C(F)F)ncn2)=O)C1 C1(NC(c2ccc(O)nn2)=O)CC2(C1)CC(CNC(c1cc(Cl)ncc1Cl)=O)C2 C1(c2nnnn2CC)(NC2(CCCC)CC2)CCC(CC(C)C)C1 N1(Cc2c(C)ccc(C)c2)CC2CN(C(c3cc(C4(C)CC4)on3)=O)CC2C1 N1(C(C(C)(C)C2CCCCC2)=O)CCCCC(NC(C2C3CCC(=O)C23)=O)C1 C1(C(F)F)(CNC(C(C)N(C)C)=O)CCN(C(=O)CSc2cccc(Cl)c2)C1 N1(CC(=O)NCC(CC=C)NC(c2nccnc2C)=O)CCCNS1(=O)=O C1(C(C(C)=C)=O)C=CCN(C(=O)C(C)=C2CCCC2)C1.c1(C(CO)N)ncc[nH]1 C1(C2CC2)(C(=O)NC2C(C)(C)C(O)C2)CN(C(=O)C(F)C2CCCC2)C1 C=C1CC(C(=O)NCCCC)(CNC(=O)C(c2cnn(C)c2)C)C1 CCCC(CCCNC(c1cn(CCO)nc1C)=O)NC(=O)Cn1ccc(=N)[nH]1 C12(C(N3CC(CC(=O)OCC)C3)=O)CCCN(CC1CO)C2 Cc1cnc(F)c(C(=O)NC2CCC2NC(=O)CN2CC3CC3C2)c1 N1(C(CN2CCC(C)C2)=O)CC2CCC(CNC(C3CCOCC3)=O)C2C1 c1(CC)c(C(=O)NC2CCCC2NC(=O)CN(C)C(N)=O)cnn1C c1(C(=O)NCC2CN(C(c3c(C)ocn3)=O)CC2C)c(O)cc(Cl)cc1F N1(C(COCCC)=O)CC2CCCC(CNC(=O)C(O)C(C)(C)CC)C2C1 Cc1c(C=CC(=O)NC2CCCC(NC(C3CC(=O)NC(=O)N3)=O)C2)cnn1C c1(OC)cc(C)c(Cl)cc1C(=O)NC1CCN(C(=O)Cn2cnnc2O)C(C)C1 N1(C(c2ccn(COC)n2)=O)CCCC(C(=O)NC2CCCOC2)CC1 N1(C(c2cncc(NC)c2)=O)CCOCC(NC(=O)C(C)C(F)F)C1 Cc1cccnc1CC(=O)NCC1(C)CCC(NC(=O)CC2CCCCC2)C1 Cc1cc(Cl)nc(Cl)c1C(N1CC2(CCCN2C(c2cc(O)ccc2F)=O)C1)=O C(CCCC(=O)N1CCC(CC(=O)NCC(F)Br)CC1)OC c1(NC(C2N(C(C(C(CC)C)NC(C)=O)=O)C(C)CC2)=O)cc(C)c(F)cc1O Cn1nc(C(=O)NCC2(NC(=O)C=CI)CCCC2)cc1F N1(C(C(C2CC2)OC)=O)CCC2C(C1)CN2C(=O)CNc1ccccc1C(N)=O CCC(CC(C)C)C(=O)N1CC(Cn2cc(C3(C)COC3)nn2)C1 C1(N(C(C(C)OCCOC)=O)C)CN(C(c2ccc(SC)cc2Cl)=O)CC12CC2 c1(COC)nn[nH]c1C(=O)NC(C)CN(C(=O)C(c1ccccc1)N(C)C)CC c1(OC)cc(CN2CCCC(C)(C(=O)N(C)CCN3CCCC3)C2)cc(C)c1 CC(C)C(O)CC(=O)N1C2CCC(C2)C1C(=O)NCCC1CC2C=CC1C2 C1(C(N2CC(OC)C(F)C2)=O)CCC(C)(C)N(C(=O)CCc2nncs2)C1 C(=O)(C1=CCS(=O)(=O)C1)NCC(C)(CO)NC(c1cc(CC)n(CCO)n1)=O N1(C(c2sc(CC)c(C)c2)=O)CCCC2(C1)CN(C(=O)C(COC)N(C)C)C2 N1(C(c2cnc(C3CC3)[nH]2)=O)CCOC2(CCN(C(C3(C4CC4)CC3)=O)C2)C1 C1(NC(CC(C)N(C(C(C)c2ccco2)=O)C)=O)CC2CC3C(C2)C13 C(CC(=O)NOC(CO)C(C)C)N(C(=O)CCc1cn[nH]c1)CC#C Cc1noc(C)c1CNC(=O)C(C)(C)C1CCCN1C(=O)Cc1cc[nH]c1 C(=O)(C(C(C)(C)C)SC)NCC1C(C)CCN1C(c1cc(CO)on1)=O n1(CC(=O)NCC2CN(C(c3c(C)cns3)=O)CC2C)c(C)nc2ccccc12 CC1CN(C(=O)C2=C(Cl)CC2)CCC1NC(c1ccc(C#N)n1C)=O C(C(F)(F)F)(C(C)(C)NC(=O)NC1CCC(C(=O)NC)C1)OCC Cc1c(C(N2CC(O)(CNC(c3cnn(C)c3Cl)=O)C2)=O)nn2c1OCCC2 N1(C(c2cn(C(CC)C)nc2)C(=O)NC2(C(=O)OC)CC2)CCCOCC1 N1(C(C(C)N(CC)CC)=O)CCN(C(c2cnc(CO)nc2C)=O)CC1C C1(C)(CNC(C=C(C)Cl)=O)CCCN(C(c2csc(-c3ccc(F)cc3)n2)=O)C1 n1(C(C)C)ccc2c(C(=O)NC3CC(NC(=O)C(C)(F)C(=O)NC)C3)cccc12 C12(C(=O)NC(CNC(c3c(C)ncn3C)=O)C(C)C)CCC(=O)N1CCS2 C=CCC(C)(O)C(=O)NCCC1CCN(NC(c2cc(OC)no2)=O)CC1 N1(C(=O)Nc2ccc(-c3ncc(C(F)(F)F)cn3)s2)CCc2c(O)cccc2C1 N1(C2CCN(C(C(C)c3ccsc3)=O)C2)CCN(C(=O)C(C)C(C)O)CC1=O C1(C(=O)NC2CC(NC(c3cc(CC4CC4)ccc3Cl)=O)C2)CC2OC1C1CC21 Cc1c(C(N2CCC3(CC3C(=O)NCc3ncccn3)C2)=O)oc2ccccc12 CC1(C)C(C(=O)NCC(C2CCC2)NC(C2C3CC4C(C3=O)C24)=O)CCS1(=O)=O CCCC(CC(C)C)C(=O)N1CCC(C)(NC(C2COC(=O)O2)=O)CC1 Cc1c[nH]c(C(=O)N(C2CC3CC2CN3)Cc2ccc(F)cc2)c1C c1(COC)sccc1C(=O)N(C1CCN(C(=O)CC(C)n2cccc2)C1)CCO C1(NC(C2C(CN(C)C)C2)=O)CN(C(c2coc(C#N)c2)=O)CC1n1cccn1 Cn1nc(Br)cc1C(=O)NCC(O)CCNC(C1CC=CCC1)=O N1(C(CC(CC)SC2CC2)=O)CCCN(C(c2ccc(CSC)cc2)=O)CC1CO C1(NC(COCC#C)=O)CC2CC(C1)CN(C(=O)C1=CCCCO1)C2 c1(C(=O)NC2CCCN(C(C=CSC)=O)C2)coc2c1COC2 c1(CC(N2C(CN(C(C(C)SC(F)(F)F)=O)C3CC3)CC2)=O)nnn(C(C)(C)C)n1 CCCC(CC)CCC(=O)N(C)CCNC(=O)C1=CC(C)(CC)C1 CCCC(CCCNC(C1CCC(F)(F)CC1)=O)NC(=O)C=Cc1cocn1 c1(C(N2CCN(C(c3n(C)ccn3)=O)C3C2C3)=O)ccc(=O)n2c1CCCC2 c1(C(N(C2CC2)CC2N(C(C(C)OCC)=O)CCC2)=O)cccc(N(C)C)n1 c1(CC(=O)N(C2CC(NC(c3c(C)noc3)=O)C2)C)cn2ccccc2n1 N1(C(C(COC)NS(C)(=O)=O)=O)CCC(CNC(=O)CC2CCC(=O)NC2)CC1 N1(C(=O)CC2CCN(C(c3sc(I)cc3Br)=O)C2)CCC(c2nc[nH]n2)CC1 Cc1ccc(C(=O)NCC2CCC(F)(CNC(C3CCSCC3)=O)CC2)cc1C CC1(C)CC2CN(C(C3(C)CCCN3C(c3ccccc3F)=O)=O)CC12 C(=O)(CCCCCF)NC(C(=O)NC(c1c(C)nccn1)C)Cn1ccnn1 CC1CN(C(c2cnn3c2OCC3)=O)CC(C(=O)NCCOC(F)F)O1 C1(C(N(CC(N2CCC2C(=O)NC2CCC2)=O)C)=O)CC2COCC2C1 c1(C(=O)NC(C(C)NC(CCCc2nc(C)sc2)=O)(C)C)cn(C)[nH]c1=N C1(CN(C(=O)C=CC(=O)NC2CC2)C)CCCN1C(=O)C(O)c1ccco1 C(=O)(CCCCCC(C)(C)C)N(CCCCNC(c1cc(O)nn1C)=O)C N1(C(C(F)OC)=O)CCCN(C(c2n[nH]cc2CCC(F)(F)F)=O)CCC1 C(c1cccc(F)c1Cl)=CC(N1C2(CN(C(CN(C3CCSC3)C)=O)C2)CC1)=O N1(C(c2ccc(OC)cn2)=O)CCC(CO)C(NC(c2[nH]cnc2C)=O)C1 c1(C(C)=O)cc(C(N2CCC(NC(c3cnn[nH]3)=O)CC2)=O)c(C)o1 C1(CC)C(NC(=O)C(CO)N(C)C)CCN1C(c1nnn(C(C)C)c1C)=O S(=O)(=O)(c1ccc(NC2CCC(=O)N2)c(Cl)c1)N1CC(N(C)C)C(C)(C)C1 c1(C(=O)NCCC2CC(NC(c3cc(C(N)=O)[nH]c3)=O)C2)ncccc1C(F)F C1(NC(CCc2nc(C)c(C)o2)=O)CC(F)(F)CC1NC(c1cncnc1)=O S(=O)(=O)(c1cccnc1CNCCc1nnnn1C)NC.C1(C)CC(C)(C)CO1 CC(C)(C(=O)N1CCC(CNC(=O)COCC2CCCO2)C1)n1cnnn1 C1(C(N(C2CCCCC2)CCNC(=O)C=Cc2ccccn2)=O)CC2C(C1)C2(F)F C(=O)(C(C)(C)C#N)NC(CC)CNC(c1ccc(-c2cccs2)s1)=O N1(C(C=CC(C)C)=O)CC(CNC(C2CCCC2C2CC2)=O)OC2(CCC2)C1 C1(C(N(C)Cc2onc(CC)n2)=O)COCCN(C(=O)C(O)CCSC)C1 C=CCC(CC=C)C(=O)N1CCC(C(=O)N(C)Cc2ccncc2)C(C)(C)C1 C1(CNC(c2ccco2)=O)CN(C(C2CC3C=CCC(C2)C3)=O)CC2(CCC2)O1 C1(C(N2C(C)CCCC2C)=O)COC2(CCN(C(=O)C(C)n3cncn3)CC2)C1 C1(C(=O)OC(C)(C)C)CN(C(c2cnc[nH]c2=N)=O)CC12COC2 C1(C(=O)NC(c2c(C)nn(C)c2)C)CC2(CC(NC(=O)C(F)(F)C(C)O)C2)C1 N1(C(c2nc(CC(C)C)sc2)=O)CCCN(C(C2CC3C=CC2C3)=O)C(C)C1 c1(C(N(C(C)CN(C)C(C2(C(F)F)CC2)=O)C)=O)ccnc(O)c1 C=CCCC(C)(C)C(=O)N1CCC(C2CC2)(CNC(c2cc(C)n(C)n2)=O)C1 CCCC(O)C(=O)N(C1CCN(C(=O)CC2CC(=O)N2)CC1)Cc1ccsc1 c1(C(N2CC(CN(C)C(C3C4CCCCC34)=O)OCC2)=O)ccc(F)c(O)c1 CC(N=c1[nH]c(=NCCC2CCOC(C)(C)C2)c2c(F)cccc2[nH]1)c1cncs1 CCC(C(=O)N1CCN(C(=O)Cc2ccc(OC)cc2OC)CC1)C(C)O Cc1cccc(CC(N2CCCC2C2(O)CN(C(=O)C=CC=C(Cl)Cl)C2)=O)c1 c1(NC2(CNC(c3c(CC)nns3)=O)COC2)ncc(Br)cc1C#N C1(NC(c2cccc(OCC)c2)C2CCC2)CCc2nc(C(F)(F)F)ncc2C1 c1(-c2cncc(NCc3c(CC)nn(C)c3)n2)cccc(OCC)c1F Cc1cc(F)c(C(N2CC(NC3CCCN3C(=O)C3CC3)C(O)C2)=O)cc1F C1(C(N2CCCN(C(CNS(CC)(=O)=O)=O)CC2)=O)CCC2CCCCN12 CN1CC=C(CC(=O)NC2CC3CCC2(NC(=O)C#CC(C)(C)C)C3)CC1 c1(OC)cccc(C=CC(=O)NC(C)C(C)NC(C2CC(C(F)F)C2)=O)c1 n1(CC(=O)N(CC(O)CN(C)C(c2cnn(C)n2)=O)C)nc2n(c1=O)CCCC2 c1(C(=O)NCCC2N(C(=O)OC(C)(C)C)CC(F)(F)C2)ccnc2c1CCC2 c1(NC(=O)C(C)N)ccccc1NC(COC)=O C1(NC(CN(CCOC)C)=O)CN(C(=O)CC2CC(O)C23CCC3)CC12CC2 CC(C)C(C)(F)CNC(=O)C(C)C(C)NC(c1sccc1F)=O C1(NC(C2CCC(CC)O2)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC12CCC2 CCCCCC(C)CC(=O)N(CCCNC(c1scc2c1OCCO2)=O)C c1(COC(=O)CCc2ccccc2[N+](=O)[O-])ccc2ccccc2n1 C12(NC(CCCOCC)=O)CCCC1N(C(=O)CC1(C3CC3)CC1)CCC2 Cc1c(C(=O)NC2CCN(C(=O)CC(C)c3cccnc3)C2)[nH]c2c1CCCC2 c1(C(N2CC(SC)C(NC(C3Cc4ccccc4C3)=O)C2)=O)cccc(C#N)c1C c1(CC)cc(C(N2CC(CNC(c3cnc(S)[nH]3)=O)CC2C)=O)sc1C c1(C(=O)NCCC2C(C(=O)NCC3(OCC)CCOCC3)C2)cc(C)nc(C)c1 N1(C(C2(OCC)CCCC2)=O)CC2CC(C1)N(C(=O)C(C)C(C)(C)C)C2 CC1(C)CN(C(c2cnnc(Cl)c2)=O)CC1NC(=O)C(c1cc(F)ccc1F)=O c1(OC)ccc(CN=C(NC2CC2)NCC(c2c(C)noc2C)O)cc1Br C1(C(=O)NC2C(CC)N(C(=O)C(CO)NC(N)=O)CC2)CCCCCN1C N1(C(C(C)OCCC(C)C)=O)CCCCCC1CNC(=O)CCCN(C)C(C)=O Cc1cc(F)ccc1C1CC1C(=O)N(C1CCCC1)C(C)(C)C C(=O)(C(CC)C(C)(C)CC)N1C(C(=O)NCC(CC#C)(C)CO)CC1 C(C(=O)N(CC(C)NC(=O)C=CCOc1ccccc1)C)(C(C)C)SC Cc1nc(C(=O)NC(C(=O)N2CC(O)C(O)C2)C(C)C)c(C)o1 c1(CN)cn(CC2CCN2C(=O)Cc2cc(Br)cs2)nn1 C1(NC(C(Cc2ccsc2)NC=O)=O)C=CCN(C(c2ccccn2)=O)C1 C1(NC(COC2(C)CN(C(C(CC)C#N)=O)C2)=O)CC2CC1CC21CC1 N1(C(c2c(CC)cnn2C)=O)CC(NC(=O)CC2CC(OC)C2)CC2(CCC2)C1 C(=O)(CCCCC(=O)OC(C)(C)C)N1CCC(NC(C(CC)COC)=O)C(O)C1 O=C1CC(NC(N2CCN(c3cnccn3)CC2)=O)CN1C1CCCCC1 C1(N(C(CC(=O)NCC)=O)CCO)CCN(C(C2COCCC2C(F)F)=O)CC1 CC1CN(C(c2cc(Cl)sc2Cl)=O)CCN1C(=O)CCCCF c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)C(C)O)cc2c(nc1O)CCCCC2 c1(C(N2C(CNC(=O)CCCc3cccnc3)CCC2)=O)cccc(F)c1 c1(SCC#N)ccccc1C(=O)NCCCOCCNC(C1CC(C2CC2)C1)=O N1(C(COCCC)=O)CC2CC(NC(C3(CC)CCCC3)=O)C2C1 c1(NC(NOCC=C)=O)ccc(OC)c(Cl)c1.c12cn(nn1)CCCC2=O CC(C)CC(O)C(C)C(=O)N1CC2(CC2)CC1CC(=O)NCC1(F)CCC1 N1(C(C(CCC)C(=O)OC)=O)CC2OCCN(C(c3sccc3CO)=O)C2C1 c1(SC)nc(Cl)c(NC(=O)CN(C)C(c2cncc(Br)c2)=O)c(Cl)n1 c1(N(CCCCn2c(C)ncc2)C)cc(F)c(Br)cc1C N1(C(C(=Cc2cccs2)C)=O)CCC(NC(C2(CN(C)C)CC2)=O)C12CCCC2 c1(OC)ccc(C(=O)NCCc2ccc3[nH]c(C)cc3c2)c2[nH]ncc12 c1(OC)cc(C(=O)NCCC(O)CNC(C2CCNC(=O)C2)=O)c(C)cc1O N1(C(C(C(CC)C)O)=O)CC2CCC1C(NC(c1ccc(C3CC3)cc1)=O)C2 c1(C(=O)NC(C)C(C)C(=O)NCCc2ccon2)cc(C#N)ccc1N N1(C(c2n[nH]c(C)c2O)=O)CCC(CNC(=O)CC2CSCCO2)C(O)C1 N1(C(C2(CCCC)CC2)=O)CCC(NC(C2(CN(C)C)CC2)=O)C(C)C1 c1(C(=O)NC2CCN(C(CC(COC)C)=O)C2C)cnc2c(C)c(Cl)ccc2c1 C1(C(=O)NC(C)Cn2cnnc2)CCCCC1(C)NC(=O)CN1C(=O)CNC1=O N1(C(C(C)OCC=C)=O)CCc2c(C(N3C4COCC3C4)=O)n[nH]c2C1 C12(CNC(C=C(COC)C)=O)CC(NC(C3CN(C)C(=O)N3)=O)(C1)C(C)(C)O2 c1(C(=O)NCCCNC(C(C(CC)C)c2ccccc2)=O)cc(C#N)ccc1F c1(OC)cc(CN2CC(F)CC2C(N2CC(F)C(F)C2)=O)cc(C(F)(F)F)c1 c1(N2CCC(OC)(CO)C2)nc2cccc(F)c2c(=NCC(N(C)C)C2CC2)[nH]1 C1(CC)CCC(C)CC1NC(=O)CC1CCN(CC2(C)CCCCC2)C1 c1(C(=O)NCCCN(C)C(C23CC(O)C2C3)=O)c(Cl)ccc(Cl)c1O C1(C(N(CC(C)N(C)C(C2CCC=CCC2)=O)C)=O)CCc2n[nH]cc2C1 N1(C(C2CCC3(CCC3)CC2)=O)CCCC2(CCN(C(C34COCC3C4)=O)C2)C1 C1(C(=O)NCCC(=O)N(C)C)CCN(C(=O)CC#N)C1 O=S1(=O)c2cc3c(cc2Cl)NC(=NCCN1)S3.C1(CCN2CC=CC2)CCOC1 N1(C(c2cn(C)nn2)=O)CCC(C)(CNC(C2C3(CC3)C23CC3)=O)CC1 C(=O)(C1=CCCOCC1)NC(COC)C(=O)NCc1nc(C)no1 C1(O)(CC(=O)NCCC(C)N(C(c2nc(C)oc2C)=O)C)COC(C)(C)C1 c1(C(C)C)ncsc1C(=O)NC(CNC(=O)CC1CCC2CC12)C1CC1 C1(c2nnc(CC)o2)CC(F)(F)CN1C(=O)C(N1CC(C2=NOCC2)C1)=O c1(CN2C(C(=O)NC(CC)C(=O)O)C=CC2)cccc(Cl)c1Br c1(C(C)NC(N(C)CCOC(C)(C)C)=O)ccccc1 N1(CCNC(C2C(C)CCS2)=O)CCN(C(=O)CCc2cccc(O)n2)CC1 C(=O)(C(C)(C)C(=O)NC1CCCCC1CNC(=O)Cc1csc(Cl)n1)NC c1(C(=O)NC(C)CNC(=O)CCn2ncn(C)c2=O)cc(F)cc2c1NCCC2 Cc1sc(CCN)nc1NC(c1ccc(CNC=O)cc1)C CC1(C)CN(C(c2n[nH]c(=N)[nH]2)=O)CC1NC(c1ocnc1C(F)F)=O c1(C(=O)NCC#CCNC(C(C)(C)C2CCCC2)=O)cn2ncccc2n1 Cc1ccc(Br)cc1N(C(c1cccnc1)C(=O)NCc1ccccc1)C C1(C(=O)OCC)CCC(C(=O)OC)CC1.C1(COC)CN(Cc2ccoc2)C1 N1(C(C(C(=O)OCC)F)=O)CCC(CC)(NC(=O)Cc2ccccc2Cl)CC1 C(C(=O)NC1CC2(C1)CN(C(c1ccc(N(C)C)nc1)=O)C2)(C(C)(C)C)SC c1(N2CC(C)(NC(C3C(OC)CCC3)=O)C2)ncc(O)cn1 c1(-n2cc(C3(N(C)C)CCCOC3)nn2)cccc(C(N(C)CP(C)(C)=O)=O)c1 C1(N(C(C(=O)NC(C)CC)c2csnn2)CC=C)CCC(F)(F)CC1 C(=O)(C(C)(C)CCCF)NC1CCCC(C(N2CCC(OC)CC2)=O)CC1 c1(C(=O)NC2(C)CCN(C(C3CCN(C4CC4)C3=O)=O)C2)cc2scnc2[nH]1 c1(N2C3CC(CN(C(C4C(C)CC5CC5C4)=O)C3)C2)ncnc2cccc(Br)c12 C1(CC(F)F)(C(=O)NCC(CC)NC(=O)CC(C)F)CCOCC1 n1(CC)cc2ccc(C(=O)NC3CN(C(=O)C(F)(F)COC)CCC3C)cc2n1 n1(CCC)cc(Cl)c(C(=O)NC2CCCC(NC(=O)CC3CCC(=O)N3C)C2)n1 C1(NC(C(c2ccccc2)OC)=O)CCCC(NC(c2ccncc2)=O)C1 c1(C(=O)NC2C3CN(C(=O)COCc4ccncc4)CC23)ccn2ccsc12 CC#CCCC(=O)NC(c1cccnc1)C(=O)NCc1n[nH]cc1CO.C(C)(=O)O c1(C(N2CCOCC(CNC(c3cc(OC)ns3)=O)C2)=O)ccc(F)c(F)c1O N1(C(Cc2c(C(C)C)con2)=O)CCC2CN(C(C3(F)CCOC3)=O)CC2CC1 Cc1ncn(C)c(=O)c1NC(O)=NCCCCl.N12CCCN(C(CO)C1)C2=O Cc1c(CN2CCN(c3ccccc3)CC2)cccc1O.c12ccc(o1)CN2C N1(C(C2(C(C)(F)F)CC2)=O)CCC(N(CCO)C(C2CCCSC2)=O)C1 c1(OCC(=O)NCC(C)NC(=O)C(F)(F)C(O)C2CC2)c(F)cccc1F c1(C(N2CCC(NC(C(C)Oc3ccccn3)=O)C(F)C2)=O)cc(F)c(Cl)nc1Cl C1(C(=O)NC(CSCC)C(=O)NCCC2(O)CCC2)(CC)CCCO1 c1(OCCCn2cc(C(CSC)C)nn2)ccc(F)cc1.C1C(O)CN1 n1(CC)nnnc1C(c1nncn1C(C)C)NCCC1CCCCO1 C(=O)(N=c1ccn(CCO)cc1C)N1CCCC(C)(c2cn(CCC=C)nn2)C1 n1(CC)ncc(Br)c1C(N1CC2CC1C2NC(C12CCCC1C2)=O)=O CCC(O)C(F)(F)C(=O)N1CC(NC(c2cc(F)ccc2Cl)=O)CC(C)C1 N1(C(C2CC(CC(C)(C)C)C2)=O)CCCC1C1(NC(C2CCCO2)=O)CC1 C(=O)(C(=O)CCC(C)(C)C)NCC(CNC(CCc1n(C)ncn1)=O)O C1(CC(=O)N(CC(C)CNC(C2(CO)CCCCC2)=O)C)CCn2cncc2C1 c1(C(N(C)CC2CCN(C(C3ON=C(C)C3C)=O)CC2)=O)c(F)cc(Cl)cc1F C1(C(=O)NC(c2ccncc2)C)(CO)CCN(C(c2cnsc2)=O)C1 Cc1cccc(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)n2ccnc2)c1 C1(C(N2C(C(=O)OCC)CC2)=O)CN(C(=O)CN2CCCCC2)CC1C CON=CC(=O)N(C(C)CCNC(=O)C(=Cc1cscn1)F)C c1(C(=O)NCC2C(Cn3cc(C(CC)O)nn3)C2(F)F)ccc2c(c1)CC(C)O2 Cc1cc2[nH]c(C(=O)NC3CC3CNC(c3cccc(N)c3Br)=O)cc2o1 C1(CNC(CN(CC)CC)=O)CCC(NC(=O)C(C)n2cncn2)C1 c1(CC)ccc(C(=O)NCCN(C(=O)C#CC(C)C)CC)c(C)n1 c1(C(N(C)CC2CN(C(CCOC)=O)C2)=O)nn[nH]c1C(C)=O N1(C(CC(CCCC)NC(=O)C=CC(C)(C)SCC)=O)CCN2C(=O)NCC2C1 C(=O)(CCCCC(N)=O)NCC1CN(C(C2(C)N(C)CCC2)=O)CC1(F)F C(=O)(CC(C(F)F)n1cccn1)NC(C)C(CO)NC(=O)CS(C)(=O)=O Nc1cnc(CNCCN2CCCOCC2)cn1 C1(C(N2CC(CC)(CC)C2)=O)N(C(=O)Cc2cc(C)no2)CCCC1(C)C C1(C)(C(=O)NC2CC(NC(C(C=C)c3ccccc3)=O)C2)CCC2CC2C1 CCCCCC(O)C(C)C(=O)N(C)CCC1CCN(C(=O)Cc2cnoc2)CC1 C12(NC(c3ccc(C(N)=O)cn3)=O)CCCC1N(C(c1coc(Br)n1)=O)CCC2 C1(CNC(CC2C(NC(C3(COC)CC=CC3)=O)CCC2)=O)CC2(CCCO2)C1 C=CCCCCCC(=O)NC(CNC(=O)C(c1ccccc1)NC(=O)CC)CC CC(C)(C)C(C(=O)NC1CCCN(c2cc(F)ncn2)C1)c1ccccc1 c1(C(N2C(CCC)CN(C(C)=O)CC2)=O)coc2cc(NC)ccc12 c1(N2C(COC)(CO)CCC2)ccc(S(=O)(=O)NC(C2CC2C2CC2C)=O)cn1 N1(C(c2c(C(C)C)noc2)=O)CC2CCN(C(c3ccccn3)=O)C2C1 C1(OC)CN(C(=O)CN2CCC2C)CC1NC(=O)Cc1cnn(C(F)F)c1 c1(C(N2C(C(N3CCC(OCC)C3)=O)(C(C)C)CCC2)=O)cc[nH]c(=NC)c1 C1(CNC(c2[nH]cc(C)c2)=O)CN(C(c2n[nH]c3c2COC3)=O)C2CCCCC12 C=CC(CC)CC(=O)NC1CC(C)(C(=O)NC(c2nccc(C)n2)C)C1 Cc1nc(N)c(CC(=O)NC(C(C)NC(c2n[nH]cc2C)=O)C(C)C)c(O)n1 C(C)(C(O)C(C)C)N(C(CC1(N(C(Cc2cc(C)sc2)=O)C)CC1)=O)C1CC1 C(CC(C)(C)CC(=O)NCC1CN(C(C2(C)CSC2)=O)CCO1)OC c1(C(=O)NC(C)C(C)NC(c2ncc[nH]c2=O)=O)ccc(F)cc1C(F)F N1(C(C2(COC)CCCO2)=O)CCC12CN(C(c1cccc(C3CC3)c1)=O)C2 c1(CC)ccc(C)c(C(=O)NCC2CC(NC(=O)CNC=O)C2(C)C)c1 C(=O)(C(CC=CCl)c1ccccc1)NC1C(NC(c2cnc(C(C)C)[nH]2)=O)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1C(NC(CN2CCP(C)(=O)CC2)=O)C1 c1(C(=O)NCCC(C)N(C(C=C(C)C(F)F)=O)C)ccc2c(c1)C(=O)N(C)C2=O N1(C(C2(OC)CCC2)=O)CCC(C2CC(NC(=O)CSCCN(C)C)C2)C1 c1(CNC(C(C(C)c2ccccc2)N)=O)cc(Cl)cc2c1OCOC2 N1(C(=O)OC(C)(C)C)CCC2(CC2C(=O)OCc2cc(Cl)ccn2)C1 C(CCCCC(=O)N1CCN(C(=O)C2CC2)CC1)N(C1CCCN1C)C c1(C(=O)NCCC(C)NC(C2CCN(C)C2=O)=O)cc2c(s1)CCS(=O)(=O)C2 O=C(C1=CC2CCC(C1)C2)NC(C1CCCCC1)C(=O)NCC(O)CC1CCC1 C12C(=O)NCCN1N2C.c1ccsc1C(=O)O.CC C(=O)(CCCCCCCC1CC1)OC1(C(=O)OC)CC(OC)C1 C(c1cc[nH]c1)=CC(=O)NCCC(C)N(C(=O)Cc1cncnc1)C N1(C(Cc2c(C)con2)=O)CCCCC2(CCN(C(=O)CSCC(F)(F)F)C2)C1 c1(C(=O)Nc2cc(OC)ncc2-c2ccc(OC)cc2F)cc(Br)cc(Br)c1F c1(NC(C(=O)NCC(C2CCOC2)OC)=O)ccnc(C(=O)NC(C)C)c1 S(=O)(=O)(c1ccc(Br)cc1N1CCC(CC2CC2)C1)NCC=Cc1n(CC)ccn1 N1(C(C(C)CC(N)=O)=O)CCC(CNC(=O)C(C)CF)C12CCC2 C1(CCOC)(NC(=O)Cc2nncn2C)CCN(C(C2CCCN2C)=O)C1 c1(CCCSCC)nc(-c2ccnn2C2CCCCC2)n(C2CSC2)n1 CCC(C)C(C(=O)NCCC1CC(NC(c2cccc(F)c2OC)=O)C1)OC Cc1nn(C)cc1C(=O)NCC(C)(O)CNC(=O)C(F)CC1CCCCC1 N1(C(CCCC#CC)=O)CC2CCC(CNC(c3cccc(F)c3)=O)C2C1 Cc1c(C(=O)NC(CCN(C)C(c2ccc([N+](=O)[O-])[nH]2)=O)C(C)C)nn(C)c1N Cc1ccc(COC(c2cc3scnc3[nH]2)=O)cc1C#N CC(F)(F)CCC(=O)NCC(F)CNC(C1CCCN(CC(F)F)C1)=O CC(CO)C(=O)NCC1CCN1C(C1(N2CCCC2)CCC1)=O Cc1c(NC(=O)C(CC2C=CCC2)NC(=O)OC(C)(C)C)oc2ccccc12 C1(CNC(C2CC23CC(O)C3)=O)CCCN(C(C2(C3CC3)CCC2)=O)C1 N1(C(CC(C)C)=O)CCCC(C(C)NC(c2cc(-c3ccccc3)ncn2)=O)C1 C1(F)(C(=O)NC(C)CCCNC(C2(CS(C)(=O)=O)CCC2)=O)CCCCC1 c1(OC)cccc2c(C(=O)NCC(CO)NC(c3cccc(F)c3N)=O)n[nH]c12 c1(C(N2CCCC(CCNC(C3C=CCC3)=O)C2)=O)cc(Cl)ccc1Cl c1(OC)cccc(Cl)c1C(=O)NC(C)CNC(=O)CC(C)c1cccnc1 c1(C(=O)NC(CNC(CC(CC)OC)=O)(C)C(C)C)cc2cc(F)ccc2[nH]1 C1(NC(C=C(CNC(c2c(C(C)C)ocn2)=O)C)=O)CCC2CC2CC1 c1(CCC(=O)N(CCCCNC(=O)C2=C(Cl)CC2)C)nnc(O)nc1O N1(C(CCNC(=O)NC)=O)CCC(C(C(C)C)NC(=O)C(C)C2CCOC2)CC1 c1(NC(c2c(C)nccn2)C)ccncc1S(=O)(=O)NCC1(Cl)CC1(F)F c1(C(N2CC(n3cc(C(C45CCC4C5)C(C)N(C)C)nn3)C2)=O)cnc(S)n1C C(CCCCC(=O)N1CCN(C(c2ccc(Br)o2)=O)CC1CCO)OC C1(NC(CCN(C)CC)=O)CN(C(C2CCCN2C2CC2)=O)CCC1(C)C N1(C(C2=NNC(=O)C2)=O)CCc2ccc(CNC(c3scnc3Cl)=O)cc2CC1 CCC(O)C(C)C(=O)N1CC(C)(C)CC1CNC(C1(C(C)C)CCC(C)CC1)=O CCCCC(C(=O)N1CC2CC2(NC(c2ccc(C)c(OC)c2F)=O)C1)C(C)C C(=O)(C1=CCN(C(c2ccc(F)cn2)=O)CC1)N(CCC(C)(C)O)C S(=O)(=O)(c1ccc(N2CCC(CC(C)(C)C)C2)cc1Cl)NCC(C)(CO)OC C(=O)(C(CC(C)C)ONC(c1cnn(CCO)c1)=O)NC(C=C)CO c1(NC(=O)NC(CC=C)CC2COC(C)(C)C2)c(OCC)cccc1Cl CCCCC(C)CCC(=O)NCC1(C)CCN(C(=O)CSCCN(CC)CC)C1 CCC(F)(F)CC(=O)NCCC(C)NC(=O)CN(c1ccc(Cl)cc1)C c1(OC)cc(C(=O)NCC(C)(C)CNC(C2CC3(CCC3O)C2)=O)cnc1C N1(C(c2c(CC)cncc2)=O)CCC2CN(C(=O)Cc3sc(O)nc3O)C2C1 C(CC(C)(C)CC(=O)N1CCCCC1C(C)NC(C1CC=CC(O)C1)=O)OC c1(C(=O)NCC(CC)C)cc(CNC(C2CCC2OC)=O)nn1C N1(CCN(C(=O)C(C)(O)C2CCC2)C)CCN(C(c2ccsn2)=O)CC1 N#CC1(CC(=O)NCCCNC(=O)CC2CCC3(CCC3)O2)CCOCC1 N1(C(C(C)NC(c2nccc(C)c2)=O)=O)CCCOC(C)C1 C1(CN(C(=O)CN(C)C(C)=O)CC)CCCN1C(=O)CCCc1ccccn1 C1(CC(N2C(CNC(CCOCC#C)=O)CCCC2)=O)COCC(C)(C)O1 N1(C(CC(C)n2ccnc2)=O)CCC2(C1)CN(C(c1ccc(Cl)o1)=O)CC(C)O2 Nc1cnccc1C(=O)NC1CCCCC1NC(c1coc(C(F)(F)F)n1)=O N1(C(C(CC(C)C)C)=O)CC2CC(O)C1C2NC(c1cc(Br)n(C)n1)=O C1(O)(CN(C(=O)C(c2ccc(F)cc2)F)CC)CCN(C(=O)C(O)C(F)F)CC1 C1(C(=O)NC(CNC(CNC(c2ccc(C)s2)=O)=O)C2CC2)CCC=CCCC1 N1(C(c2c(CNC(COCCOC)=O)occ2)=O)CC2CC(C1)N(C)C2 C12(n3c(N4CCC(C(=O)NC(C)CN(C)C)CC4)nnn3)CCC(C1)OC2C C12(C(=O)NCC(C)C(=O)NCC3(C)CCOCC3)CCC(C1)C2(C)C c1(COC)cccnc1C(=O)NCC1CC(NC(C2CN(CC(F)(F)F)C2)=O)C1 C=CCC(CC(F)F)NC(=O)C(c1ccnn1C)NC(c1ncoc1C)=O N1(C(c2ccc(NC(CCC(C)C)=O)nc2)=O)CCCCC(F)(F)C1 C(C)(CCC(=O)NC(C)C(CO)NC(c1coc(C(C)C)n1)=O)OCC C#CCC(C)(CC)C(=O)NCC(C1CCC1)NC(c1sc(C2CC2)nc1C)=O C(=O)(CC(C(F)(F)F)NC(=O)C(C)(C)C(C)(F)F)N1C2C(OC)CC(C2)C1 CC1CN(C(C2CC(O)C2)=O)CCCN1CC=Cc1ccc(C(F)(F)F)o1 c1(C(C(=O)Nc2ccccc2C)N(C2(C#C)CC2)C)cccc(C(F)(F)F)c1F c1(C(N(C2C(N(C(=O)CC3CC4(CC4)C3)C)CCCC2)C)=O)ccc2c(c1)CC2 N1(C(C)CC(N2CC3CCC(C2)O3)=O)CCCCc2ccccc21 C1(CNC(COC(CC)C)=O)CN(C(=O)C(F)(F)CCn2cccn2)CC12CC2 C1(NC(=O)CC2COC(=O)C2)CCC(O)CN(C(=O)CN2CCCC2)C1 c1(C(N(CC(C)NC(=O)C=CCN2CCOCC2)CC)=O)c(C)cc(OC)cc1C C1(NC(c2ccc(OCC)c(C)c2)=O)CC2(CCN(C(=O)CO)C2)C1 Cc1nn(C)cc1C(=O)NCC1CC(C(=O)NCCC(C)N(C)C)CO1 c1(C(=O)NC(CCCNC(CC2(C=C)CCC2)=O)C)cnc(O)n(C)c1=O CCC(C#N)(CC)C(=O)N1CC(CCNC(c2c(F)ccc(F)c2Cl)=O)C(C)C1 Cc1cc(F)ncc1C(=O)Cc1ccc(Br)c(Cl)c1 C1(CC=C)(NC(c2cnn[nH]2)=O)CC2CCC(C1)N2C(C1CC2(CCCC2)CO1)=O CCC(C)C(O)CC(=O)N1CCC(C)(C)CC1C(=O)NCCc1cc(C)no1 C(=O)(C(O)CCS(C)=O)N1CC(CNC(c2ccc(CNC(C)=O)s2)=O)C1 c1(C(N2CCC(NC(C(CC)=CC)=O)C2C(C)(C)C)=O)ccc2c(n1)CCOC2 C1(C(=O)NC(CCCC(C)C)C)CCc2nc(-c3ccc4oncc4c3)sc2C1 c1(C(=O)NC2CCN(C(C3CC(=C)C3)=O)C2)ccc(OCC(F)(F)F)nc1OC N1(C(C=CC(CC)=CC)=O)C2CCCC1CN(C(C1CC(OC(F)(F)F)C1)=O)C2 CC(CCC(=O)NCC(C1CC1)Nc1cc(C(F)(F)F)ncn1)N(C)C Cn1ccc(=NCc2cccc(C(=O)Nc3ccc(Cl)cn3)c2)[nH]1 c1(C(N2CC=CC(NC(C=C(CC)C)=O)C2)=O)cccc2c1CC(C)(C)C2 CC(C)C(O)(C(=O)N1CC=CC(NC(=O)Cn2ncn(C)c2=O)C1)C(F)(F)F c1(C(=O)NCC2CC3(CC(CN)C3)C2)cc2n(n1)CCNC2=O O=S(=O)(c1ccc2[nH]c(=NCC(Cl)=CCl)ccc2c1)NC1CC(C(F)F)C1 N1(C(c2c(C)c(F)ccc2N)=O)CCC2CN(C(=O)CC3CCOC3)CC2CC1 C(=O)(C(C1=CCSC1)N1CC(CSC)OC(C)(C)C1)NC C(=O)(CC(C)C(C)(C)NC(=O)CC1CCC2CC12)NC1(CC(C)C)CC1 N1(c2nccc(OC)n2)CCC(c2nnn(-c3ccc(Br)cc3SCC)n2)C12CC2 C(=O)(CC(C)CC(C)C)N1C(C(=O)Nc2cccc(C)c2)CSCC1 C(=O)(CCCC(F)(F)CO)NC(COC)CNC(c1c[nH]nc1-c1cccs1)=O C(=O)(C(F)C(F)(F)F)N1CCN(C2CN(C(=O)CSc3ccccc3OC)C2)CC1 N1(CCC(N2CC(OC)(CNC(=O)CCc3cn[nH]c3)C2)=O)CCC(O)CC1 c1(CC(=O)C)nc2ccccc2o1.N1(C(=O)CC2CC2F)CCC(F)(F)C1 C(=O)(C1CCCc2scnc21)N1CC(C)(NC(C=Cc2cncc(OC)c2)=O)C1 C#CC1(C(N2CC(Cc3ccc(Cl)cc3)C2)=O)CN(CC2CC2)C1 C1(C(=O)NC2C(NC(C3CC(OC)C3)=O)CCCC2)Cc2ccc(F)cc2O1 CC1CN2CCN1C(C(N1CCCCC(CNC(=O)C(C)(Cl)Cl)C1)=O)C2 n1(CC(=O)NC(CNC(C2CC2C(C)C)=O)(C)C)nccc1COCCOC C1(C(N(C(CNC(CCC=CC)=O)C2CC2)C)=O)CN(C)CC(C)O1 N1(C(c2onc(C)c2C)=O)CCC(C)(CNC(=O)C(C)C2CCC2)CC1 C1(C(N2CC(O)(CN(C(=O)C=Cc3nccs3)C)C2)=O)CCC2(CCOCC2)C1 N1(C(=O)CC(F)(F)Cl)C2CC1CN(C(=O)C(F)(F)CC1CCCO1)C2 c1(C(N(CC=CC(N2CCC(CC=C)C2)=O)C)=O)ccc(=O)n(C)c1 CCCCC(O)C(=O)N1CC2CC2(CNC(=O)C(C)NC(C2CCCC2)=O)C1 c1(C(c2n(CC)nnn2)NC(c2nnc(C)s2)C)ccnc(C(F)(F)F)c1 CCC(C(=O)NC1(C)CN(C(C2CNC(=O)N2)=O)C1)SC CCCC(C(=O)NC1CCCN(C(=O)Cn2cc(C3CC3)nn2)CCC1)C(C)C C(CC1C(=O)NCCCC(=O)N1)=CC.N1(C(C)=O)CC(SCC)C1 C1(NC(CCCOCCOCC)=O)CC2CC1CN2C(=O)Cn1nc(C)cc1C N1(C(C=CC=CC)=O)CC(C)CN(C(=O)CCc2ccccc2Br)C(C)C1 n1(CC(=O)NC2CCNC2=O)ccc(=NCc2n[nH]c3ccc(Br)cc23)nc1O c1(C(=O)NCCN(C(=O)CC2CCCC2C)CCC)ccncc1N(C)C C1(C(N2CCC(N(CCC)C(c3cccc(OC)n3)=O)C2)=O)C2CCC(F)(F)C12 C1(NC(c2c(C)n(CC3CC3)cc2)=O)(CO)CCCN(Cc2ccccc2)C1 c1(CC)nc(C(=O)NCc2c[nH]nc2C(N2CCOCC2CO)=O)c(C)o1 c1(C(N2CCC(NC(Cc3nnc(C)o3)=O)C(F)C2)=O)c(Cl)cc(Cl)nc1N C1(CC(=O)N(CC2CCN(C(=O)COC3CC3)CC2)CC)(OC)CCOCC1 c1(CC)ccc(C(=O)N(CCCN(C)C(c2cn(C3CC3)cn2)=O)C)cn1 N1(C(CSCCN(CC)CC)=O)CC2=C(C1)CN(C(c1cc(C)sn1)=O)C2 c1(C(=O)OC)ccc(COC(c2cc(-c3cn(C)nc3C)no2)=O)cn1 C#CC1(C(N2CC(N(C)C)CC(C)C2)=O)CCN(C(=O)CCSCC)C1 CC1CN(C(=O)NC(c2ncc[nH]2)CO)CCN1c1ccncc1 c1(CC)sccc1C(N1CC(CCNC(=O)CC2CCOC2)(OC)C1)=O N1(C(CCn2cc(CCOC(=N)O)nn2)=O)CCC(O)(c2ccc(F)cc2)CC1 CCCC(CCC)=CC(=O)NC(C1CCN(C(c2cncc(N)c2)=O)CC1)(C)C N1(C(C2N(C(CCc3ncn(C)c3)=O)C3(CC2)CC3)=O)CCC2(CC1)CC2C#N N1(C(C(C)N(C)C(C2CCC(F)CC2)=O)=O)CCCCC2(CCC2)C1 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1CCCN(C(C(C)=CC2CC2)=O)CC1F C12(CNC(Cc3c(C)ccs3)=O)CC1CN(C(=O)CC1CC3C=CC1C3)C2 c1(CC(=O)NCC2(O)CCN(C(CCCOC)=O)CC2)ccc(F)cc1[N+](=O)[O-] C(N=c1[nH]c(=NCCC(C(C)C)OC)c2ccc(C)cc2[nH]1)C1CCN(CC)C1 c1(C(=O)NC2(CCCNC(COCC=C)=O)CC2)ccc2nsnc2c1 C(=O)(C(C)N(C(=O)C=CC(=O)NC1CC1)CCC)NC(C#C)C Cc1cc(Br)cc(C(=O)NC2(CNC(C3CCCCC3C)=O)CCCC2)c1N C12(CC(=O)NC3CN(C(c4ccc(=N)[nH]c4)=O)CC3F)CCCN1CCC2 Cc1nc(-c2nn[nH]n2)ccc1C(=O)NCC(N1CCOC(C(C)C)C1)=O C(C)(CC(=O)NC1C=CCN(C(=O)CC(F)F)C1)(C(F)(F)F)N(C)C C1(CNC(c2occc2Br)=O)CN(C(c2ccc(Cl)nn2)=O)CCCO1 c1(C(N(CC(CC)NC(=O)CNC(=O)OC)C)=O)ccc2c(c1)C(C)(C)CO2 CC1COc2ccc(C(=O)NCC3(NC(=O)CC4CCCN(C)C4)CCC3)cc21 c1(C(=O)NCCN(C(c2cc(Br)ccc2O)=O)CC)nnc(O)c2ccccc12 C(=O)(C(C)C(F)(F)C(F)F)N1C(CC)CN(C(c2nc[nH]c2C(C)(C)C)=O)CC1 C(CC(F)(F)C(F)(F)Br)n1cc(-c2cn(C)nc2C(F)F)nn1 C(c1cccc(Cl)c1)=CC(=O)NCC12CC1CN(C(=O)C(F)=C1CCC1)C2 c1(C(N(CCOCCNC(c2cc(C)no2)=O)C)=O)cccc2oncc12 N1(C(C2CCC(CNC(c3nn(C)c(=O)cc3)=O)C2)=O)CCCC(F)(F)CC1 N1(C(c2c(C)nc(CCC)o2)=O)CC(NC(C2CN(C)CCN2C)=O)CC(C)C1 C(=O)(C1=CC2C=CC(C1)C2)NCC1(NC(CCCCCCC)=O)CCCCC1C c1(C(=O)NC(C)C(C)(C)NC(C2CCCC(O)C2)=O)sc(N2CCCC2)nc1Cl C=C1CCN(C(=O)COCCC(C)C)C(C(N2CC3(CC3CC)C2)=O)C1 c1(C(=O)NCc2cc(C(N(CCC(C)C)C)=O)n[nH]2)cccc2cc[nH]c12 S(=O)(=O)(c1ccccc1F)N1C(CC)CN(c2ncnc(C(F)(F)F)c2Br)CC1 c1(C(C(=O)NC(CC)(C)C)N(C)CC2CCC(C)O2)cccc(C#N)n1 CN1CCN(C(=O)NCc2nc3cc(Br)ccc3s2)c2ccc(Br)cc21 C1(N(C(=O)CCC2CCOC2)C)CCCCN(C(=O)CC2CC(=O)C2)C1 C1(NC(C(C)NC(C)=O)=O)CCCC12CCN(C(C1C3CC4C(C3=O)C14)=O)CC2 c1(N(C2CCC2)C(c2c(OC)ccc3c2CCC3)=O)ccc2c(c1)CCN(C)C2 C1(C)(C(=O)NC(CC#C)CC)CCN(C(c2cnc(OC)s2)=O)C1 CC1C(=O)N(CC(=O)NCC2CCN2C(C2CCS(=O)(=O)N2)=O)C(=O)C1C c1(SC)ccsc1C(=O)NCCC1CCN(C(C2(CC(C)=O)CC2)=O)C1 CCC(CC(=O)NC1CC(F)CN(C(c2ccc(C3CC3)cc2Cl)=O)C1)C(C)C C1(C(=O)NCCN(C(c2c(Cl)nc(OC)s2)=O)CC2CC2)CC2CCC(C1)S2 CC1CCN(C(C2CC2CC(=O)NCCOCC(F)F)=O)CC1 N1(C(c2nccc(C)n2)=O)CCC(NC(c2ncoc2C2CC2)=O)C(CO)C1 S(=O)(=O)(c1ccc(N2CC(C)CCC23CC3)cc1Br)N1C(C)CN(C)CCC1 C1(CNC(C2CCC(N(C)C)CC2)=O)N(C(C2CC2(F)F)=O)CCC1(C)C C12(C)CC(CCO1)NC(=O)CC1(OC)CN(C1)C2=O.c1(CC)ccc(O)c(C)c1 CN1CCC(C)(C(=O)NC2CC(C(F)C(=O)Nc3cccnc3)C2)C1=O N1(C(CN(CCOC)C)=O)CCCC(O)(CNC(c2ncn(C(C)C)n2)=O)C1 C(C(O)(CNC(=O)Nc1ccc(C2CCC2)nc1)CO)OC C(=O)(C(C)(C)CNC(C1(O)CCCCC1)=O)NC(CC(=O)NC)C1CC1 c1(C(=O)NC2CCC(NC(CNC(CCC)=O)=O)CC2)cnc(C)[nH]c1=N C1(CC)CN(C(=O)C2=COCCO2)CCN1C(=O)C(C)NC(=O)COC c1(OC)ccc(NC(=O)CN2CCC(C)CC2)nc1.C12CC(O)(C1)CN(C)C2=O Cn1cc(CNC(c2nnnn2CC2CC2)C2(C)CCCO2)nn1 c1(CC(=O)N(C)C)ccc(-c2c[nH]c(=NCc3cc(C(=O)O)ccc3F)s2)cc1F c1(CNC2CCCC(CC)C2)ccc(Br)cc1C(F)(F)F.C12CN(CCO1)C2=O Cc1cc(C(N2CC(NC(c3ccco3)=O)CC(O)C2)=O)ccc1Cl N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C(n2cnc(C#N)n2)C)CCC1C c1(C(=O)NC2C(NC(CC3CC(=C)C3)=O)CC2)cccc2nonc12 C1(CN2C(C(=O)NC3CC(C(N)=O)C3)CCC2)CCS(=O)(=O)CC1 C1(NC(C2C(CCC)C2)=O)CN(C(=O)CC2CCOCC2)CC12CC2 Cn1nccc1C(=O)C(=O)NC(C)(C(=O)N1CCC(C(=O)OC)C1)c1cccs1 c1(C(=O)NC)cccc(CCN(Cc2nc(C)cs2)C)c1.C(=O)(C(C)CC1CC1)N N1(c2nc(C)nc(Cl)c2)CC2CCCC(NC(C3(F)CCOC3)=O)C2C1 C1(NC(C2(OCC)CC2)=O)CCCCC12CCN(C(c1ccsc1OC)=O)C2 C(=O)(CCC(=O)N(C)CC1CCN(C(C2CCC(=O)N2C)=O)C1)NC CN1CCCc2cc(CC(=O)NCC3CC3NC(c3cn(CCO)nn3)=O)ccc21 c1(C(=O)NCCC2(OC)CN(C(C(CCC)CC)=O)C2)cnn2c1CC(C)CC2 C#CCC(C)(CC)C(=O)NC1CCCCC1NC(c1ccc(C(C)C)c(C)c1)=O C1(NC(C(COC)NC(C)=O)=O)CCC(C)N(C(=O)Cc2n[nH]c(C)n2)C1 N1(C(Cn2c(C)csc2=O)=O)CCC2(CC1)CC2NC(C1CCCCN1C)=O CP1(=O)CC(NC(c2ccccc2CCc2ccccc2)=O)C(O)C1 N1(C(c2ccc(Cl)c(I)c2)=O)CCC2C1CCCN2S(=O)(=O)CCC(F)(F)F C1(O)(CN(C)C(C2CC3(CC3)CO2)=O)CCN(C(C2Cc3nncn3C2)=O)CC1 C1(c2ccno2)(C(N(CCCN(C(c2c(CC)noc2)=O)C)C)=O)CCOCC1 C12(C(=O)NCCCCC(C)NC(CNC(=O)OC)=O)CCCC1OCC2 c1(CCOC)n[nH]c(=NCC2CC(NC(=O)CC3CC(O)C34CCC4)C2)s1 C(C(O)CC(=O)N1CCOCC1CN(C(=O)CCc1csnn1)C)N(C)C Cc1cc(C)c2nc(N3CCN(C(c4ccn(C(C)C)n4)=O)CC3)sc2c1 c1(C(N2CCC(O)(CN(C(C(C)C(F)F)=O)C)CC2)=O)nccc2ccn(C)c12 N1(C(C2CC2c2ccccc2)=O)CCCCC(NCc2sc(O)nc2O)C1 C=C(C)C1OCCCC1C(=O)N(CCCNC(=O)C=CS(C)=O)CC1CCCC1 N1(C(c2cc(C)c(-c3cccc(F)c3)s2)=O)CCC2CCC(=O)C1C2 C(=O)(C(C)CCCC(C)=O)NC(CC=CC)C(=O)N(CC(O)CF)C C(CCCC(C)NC(c1nc(Br)sc1C)=O)NC(C(C)OC)=O c1(C(=O)NCC2CC(NC(=O)COC3CCCC3)C2)cccc(F)c1F c1(C(=O)OC)cn(C)nc1C(=O)NCC1CCC(NC(=O)Cc2cncs2)C1 CCC(CC)CC(=O)NC(C)(CNC(c1ccnc(O)c1Br)=O)CO C1(CCC)CN(C(=O)CCc2nc(CC)no2)CCN1C(=O)CC1CCCO1 N1(C(CCN2C(C)CCCC2)=O)CCN(C(c2ccnnc2S)=O)C(CF)C1 n1(CC)nc(C(=O)NC2CN(C(=O)C(C)CCOC)C2)c(Br)n1 C1(NC(C2(COC(C)C)CC2)=O)C=CCN(C(=O)C#CC(=O)N(C)C)C1 CC1(C)CN(C(=O)Cc2ccc(Cl)cc2)CC1CNC(C1CCCC2(CC2)C1)=O C(=O)(N=c1ccn(CC2CC2)[nH]1)C1(CO)CCN(C(c2cn(CC=C)nn2)=O)C1 CC1(C(=O)NCCOC2CCN(C(=O)CCc3ccccn3)C2)CCC(=O)NC1 C(=O)(CCCC(C)NC(c1ccc(C#N)cn1)=O)NC1(c2nc(C)[nH]n2)CC1 C1(OC)CC(NC(C2(c3ccc(Cl)nc3)CC2)=O)CN(C(c2cscc2Cl)=O)C1 N1(C(c2ncn(CC)n2)=O)CCOCC1CN(C)C(C1(CC)CCCO1)=O C1(CC(=O)NC2CN(C(c3cc(O)ccc3F)=O)CC2O)CC2CCC1CC2 c1(OC)ccc(C(N2CC=CC(NC(c3nnn(C(C)(C)C)n3)=O)C2)=O)nc1Cl CC1CCCC(c2nnnn2C)(NC(C)(C)C)C1.C1CCC(=O)N1.C1C(=O)OC1 N1(C(CCN(C)CC)=O)CCC(NC(=O)C(c2cc(C)cc(C)c2)C)C(C)(C)C1 N1(C(C(=O)NCc2csc(Cl)c2)=O)CCC(O)CC12CCC2 c1(CC)onc(C(N2CC(C(C)(C)O)(CNC(=O)C(C)C3CCOC3)C2)=O)c1C N1(C(COCCCC)=O)CC2CCN(C(c3ccncc3C)=O)CC2C1 N1(C(C2CC(C#N)C2)=O)CCN(C(=O)CCc2ccoc2)C(C2CCC2)C1 C1(C(N2CCC(c3ccc(C#N)cc3)CC2)=O)Cc2nccnc2C1 N1(C(c2ccc(OCCOC)nc2)=O)CC(NC(C2CCC2(F)F)=O)CC(C)C1 N1(C(=O)NCC(C#C)C)CCC(C2CCOCCN2)CC1 c1(-c2n(CCC(C)C)nc(Cn3cncn3)n2)cc2c(F)cccc2[nH]1 c1(C(=O)NCCC(C)N(C(CC(=O)NCC#C)=O)C)sc(C(C)C)nc1C CCCC(C)(C)CC(=O)N(C(C)CNC(c1nncn1CC)=O)CC C(C)(c1ccccc1C)=CC(=O)NC(C1CCN(C(C(C=CC)O)=O)C1)C N1(C(C(CC=C)CC)=O)CCCC(C2CN(C(c3ccnn3C)=O)C2)C1 c1(CNCC(C)Sc2ccccc2OC(F)F)ncnc(OC)c1Cl C123CC(C1)(OC2(C)C)COC3=O.C1(COC(C)(C)C)CC2OCCC2O1 Nc1c(C(N2CCC3(CC2)CC3NC(C2CC(F)C2)=O)=O)cnc(Cl)c1F n1(CCOC)nccc1C(=O)NC(CNC(=O)Cc1cc(C(F)(F)F)n[nH]1)CO c1(C(C(N2CCC(C)(CNC(CSCC#C)=O)C2)=O)C)ccc(F)c(F)c1 C1(NC(=O)NC2(c3ccno3)CC2)C2CCN(C(=O)C=C3CCOC3)CC12 c1(C(N2CCCC(N3CCN(C)CC3)C2)C(=O)NCC(=C)C)ccc(OCC)cc1 Cc1nn(C)c2cc(N(C(=O)C(O)C(C)C)C(C3CC34CNC4)=O)ccc12 C1(C(=O)NCCNC(CCN(C(C)=O)C)=O)CC2(C1)NC(=O)NC2=O C(CCO)(CC(C)C)NC(C(c1cccnc1)NC(c1cc(CC)nn1C)=O)=O C1(OC)CN(C(=O)CCC2CCCC(O)C2)CC1NC(=O)CCSC(F)(F)F C1(NC(C=CCCCCC)=O)CC2(C1)CC(NC(=O)C1=NNC(C(F)(F)F)C1)C2 C1(C(=O)NCC2(O)CC3C=CC2C3)CN(C(=O)C=Cc2ccoc2)CC12CC2 c1(CN2C(C(N3CCC(CCCO)CC3)=O)CSCC2)ccc(Cl)c([N+](=O)[O-])c1 c1(CC)ccc(O)cc1C(N1CCC(NC(=O)CCC2(C)CC2)C(O)C1)=O C=CCC(CNC(=O)CC1OCCO1)C(=O)Nc1cncc(N(C)C)c1 C1(C(=O)NCCC2(O)CN(C(CC3C(CC)C3)=O)C2)CC2CCCCC12 CCCC(C(=O)OC)C(=O)NC1CCCCC1C(N1CCC12CC(O)C2)=O c1(OC)cccc2cnc(NC(C3(C)CCCN3Cc3cnccc3Br)=O)nc12 C(=O)(C(CCOC)NC(=O)CC(CC)SC)NCCCOCC#C C1(NC(c2nc(C(C)OC)sc2)=O)CCCC12CN(C(=O)CC1CSC1)C2 c1(CC(=O)NC2CC(NCc3ccc(F)cn3)C2)cccc(C(F)(F)F)c1 N1(C(C(CCC)C)=O)CC2(C1)OC1(C)CC2(NC(=O)Cn2cnccc2=O)C1 C1(NC(N=c2ccn(CCCOC)[nH]2)=O)CCC2C(CC1)C2(F)F c1(C(=O)NC(CC)CNC(c2ccn(C)c(=O)c2)=O)ccnc2c1nnn2C CC(C)C(CNC(C1(C)CC1(F)Cl)=O)NC(=O)CC1C=CCC1 c1(C(=O)NC2CCN(C(C(C#N)=CC(C)C)=O)CC2C)cn2cc(C)ccc2n1 C1(NC(C(CC2CCC2)NC(c2[nH]ccc(=N)n2)=O)=O)CCCC2(CC1)CC2 C1(C(=O)NC2(CNC(c3cnc(C(F)(F)F)s3)=O)CC2)CC2CSCC(C1)C2 C(=O)(C1=Cc2ccccc2C1)N1CC(C(C(=O)OCC)N(C)CCOCC)(OC)C1 N1(C(c2c(CC)cccc2)=O)CCC(OCCNC(c2ccc[nH]2)=O)C(C)(C)C1 C1(NC(c2n(CCC)nnn2)c2ccno2)CC(C)(C)C1CC N1(C(CC2C(C)CCN(C(c3ccn(CCC)n3)=O)C2)=O)CCC2(CCCC2)C1 c1(C(=O)NC2CC(C)CN(C(=O)CCCCNC(N)=O)C2)nnn2c1CCCC2 C#Cc1cc(F)c(C(N2CC(CNC(c3occc3C)=O)C3(CC3)C2)=O)c(F)c1 c1(C(C)C)[nH]ccc1C(=O)NC1CC1NC(=O)Cn1cccn1 c1(CC(C)N(CCC)C(=O)NCc2ccc(Cl)o2)cccc(F)c1 Cc1nc2c(s1)CCCC2C(=O)N(C1CN(C(=O)C(=O)Cc2ccccc2)C1)C c1(OC)ccc(CC(=O)NC2CC3(C2)CN(C(C2CC(F)C2)=O)C3)cc1OC C1(CNC(c2ccccc2N2CCCC2=O)=O)CN(C(=O)C(F)F)C2CC12 N1(C(C=CCNC(Cc2c(C)cnn2C)=O)=O)CCNC(=O)CC1C C12CC(C1(C)C)NC(=O)C2.C(=O)(CN(C)C)N(CC=C)CC=C CCC(C)CC(C)C(=O)NCc1nc(CNC(=O)C(=O)NOC)cs1 Cc1cc(C(=O)NCCCC(C)(C)NC(c2cc(CCCO)on2)=O)ccc1Cl C1(N(C)C(c2cn[nH]c2)=O)CCCN(C(c2cccc(C(N)=O)c2F)=O)CC1 c1(NC(Cc2cccc(C)n2)=O)ccc2c(c1)CN(C(=O)C(O)CC(C)C)CC2 N1(C(c2ccc(SC)s2)=O)C2CCC1CC(NC(C13CCC(CC1)CO3)=O)C2 C1(C(=O)NC2CCOC(C(=O)N(CC3CC3)CC3CC3)C2)CC2C(C1)C2(F)F CC(C)(COC(=O)CCNS(C)(=O)=O)C1CCCC1 C1(C(N2CC=CC(NC(c3c(CC)nccn3)=O)C2)=O)(OC)CCC(C)(C)CC1 N1(C(c2nnn(C)n2)C)CCC(NC(=O)CCC2NC(=O)NC2=O)C(C)C1 c1(C(N2C3(CNC(c4cnc(C)[nH]4)=O)CCC3CC2)=O)nn2c(c1C)OCCC2 C(=O)(CCCC(F)F)NCC1(O)CCN(C(C(C)OCCC(C)C)=O)C1 Cn1nncc1C(=O)NC(CNC(c1cn(CC(F)(F)F)nn1)=O)CO C=C1CCN(C(=O)C(C)NC=O)C(C(=O)NC(c2ccnn2C)C)C1 N1(C(CCC)=O)CCCCC1CCNC(C1(c2cnn[nH]2)CCCO1)=O c1(CC(=O)NC2C(NC(c3c(C)nc(CC)s3)=O)CC2)ccc(O)c(C)c1 c1(C(N)=O)c[nH]c(=NC2CN(c3ccc(Cl)cc3)C2)cn1 c1(C(=O)NC(CNC(c2c(CCC)occ2)=O)(C)C(C)C)cc2ncccc2s1 c1(C(=O)NC2CCN(C(CC(C)OC)=O)C2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 c1(C(=O)NCC(CN(C(C(N2CCSCC2)C)=O)C)O)ccc([N+](=O)[O-])s1 c1(C(=O)NC2CCC(N(C(C(C)CO)=O)C)CC2)cc2c[nH]cnc-2n1 C1(CCC)CC(C(=O)NCC2(C(C)(C)C)CCN(C(=O)C(O)C3CCC3)C2)CCO1 N12CCCC(C1)C2=O.C1(n2cc(CCCC(=O)O)nn2)C=CCC(C(=O)O)C1 N1(C(CCC(C)(C)F)=O)CCC(O)(C2(NC(=O)C=Cc3cncs3)CC2)CC1 c1(OC)cc(C(=O)NC2(CNC(C3CCC34CCC4)=O)CC2)cc(C)n1 N1(CC)CCc2nc(NC(=O)CCCn3cc(-c4ccc(F)cc4)nn3)sc2C1 C(N=c1[nH]c(=NCCC(C)CO)[nH]c2ccc(Cl)cc12)c1n(C)nc(CC)c1Cl N1(C(CC(CCCC(C)C)C)=O)CCCC2(C1)CN(C(C1CC(F)C1)=O)CCO2 c1(CC)cccc(C(=O)NCC2(O)CCCN(C(C3CC(C)(C)CO3)=O)C2)c1O Cc1nc(Cl)[nH]c(=NC2CCC(NC(=O)CCN(C(=O)CO)C)CC2)c1Cl c1(C(=O)NC(C(=O)NC)C)ccnc(CNC(=O)CC(C)C2CC2)c1 c1(C(=O)NCCCCN(CCCNC(C(CCC)OC)=O)C)ccn(C)c(=O)c1 c1(C(=O)NC(C)CCCNC(=O)Cc2ccc3c(c2)CC3)ccc(C#N)cc1F C1(NC(C(C)(C)c2ccsc2)=O)CCCCC1CNC(C1(CF)CCOCC1)=O c1(C(=O)NCC(C2CCN(C(C3(CCF)CC3)=O)CC2)C)ccc2sccc2c1 c1nc(C(C(=O)NC2CCC2)N(c2ccns2)CC2CC2)n[nH]1 c1(C(N2CC(NC(C3(CC#C)CCOC3)=O)C(OC)C2)=O)ccc(F)cc1OC N1(C(C2C(CC)CCC2)=O)CCCC(CCNC(=O)CCc2cccn2C)CC1 CC(C(=O)NO)NC(=O)COCCNC(=O)C(C)CO C1(C(=O)NC(Cn2cc(CCC(C)=O)nn2)C)CCC(F)(F)CO1 C1(C(N2CCC(C(CNC(C=CCCC)=O)(C)C)CC2)=O)CC2(CC(=O)N2)C1 Cc1ncsc1CCC(=O)NCC(F)CNC(C1CSC1)=O c1(C(N2CCC(C(C)NC(=O)CC(C)(F)F)C2)=O)ccc(C#N)n1C C(=O)(CC(C)(C)C)N(CC(C)NC(c1n[nH]cc1Cl)=O)C C1(NC(C2(C)N(C)CCC2)=O)CN(C(c2c(N)cc(F)cc2F)=O)CC(C)(C)C1 C1(NC(c2c(COC)ccs2)=O)CCCC(NC(c2coc(CF)n2)=O)CC1 C1(CNC(c2c(C)nc(C)[nH]2)=O)CC2CCC1N(C(c1cccc(O)c1)=O)C2 c1(-c2scc(CCNC(N3CCCC3c3ccco3)=O)n2)ccc2c(c1)OCO2 C1(C(C)C)N(C(=O)C(CC(=O)O)NC(=O)OC(C)(C)C)CC12CCCCC2 c1(C(=O)OC)cccc(Cl)c1NC(C1CCN1Cc1cnc(OC)c(C)c1)=O CC(O)C(F)(F)C(=O)N1CC(O)(CCNC(=O)C(F)(F)C(O)C2CC2)C1 C1(C(=O)NC2CC(F)(CNC(c3cnc(C)o3)=O)C2)CCn2ccnc2C1 C(=O)(CCCCCCn1cc(C(c2ncc(C(=O)OC)s2)(C)C)nn1)NC C(=O)(C(C)(C)C(=O)N1CCCC(CN(CCCC2(O)CC2)C)C1)OC Cc1cc(NC(=O)CNC2CCC2c2nncn2C)cc(C)c1I C1(C(=O)NCC(O)CN(C(=O)CC2CC23CC3)C)(OC)CCC(F)(F)CC1 C12(C(=O)OCC)CCCC1N(C(=O)Cc1ccc3c(c1)CC3)CC2.C(CC)=CC=C c1(C(=O)NCC2CCN(C(C3CC(CC)C3)=O)CC2)c(C2CC2)cccc1F C1(CCN(C(CCC#C)=O)C)CCCCN1C(C1CC(OC)(OC)C1)=O C1(C(=O)NCC(C)C(=O)N(CCCF)C)CCCOCC1 N1(C(c2ccc(CC)s2)=O)CC2CCOC2(CNC(=O)C=CC(C)CC)C1 C1(NC(CNC(=O)NC)=O)CN(C(C2CCC2NC(=O)C(F)(F)F)=O)CC12CC2 CCCCC(O)CC(=O)N(C(C)CCNC(c1cc(C(=O)C(C)C)c[nH]1)=O)C C1(NCCC(C(=O)NC)N(C)C)CN(C(c2c[nH]c(C(N)=O)c2)=O)CC12CC2 C1(C2(O)CCN(C(=O)Cc3ccc(F)cc3)CC2)(NC(C(CC(C)C)F)=O)CC1 c1(-c2ccc3nc(C)sc3c2)ccc2c(c1)CC(=O)N(C)C2 n1(C(C)C)ncc2c(NC3CC(NC(C4(CF)CC4)=O)C3)ncnc12 C1(CCC(=O)NCC2C3CN(C(=O)CCOC4CC4)CC23)CC2(CCC2)C1 c1(CC)cc(F)ccc1C(N1CCN(C(C23CC(F)C2C3)=O)C(C(F)F)C1)=O c1(N(CC(N2CCN(C(=O)C=Cc3ncc[nH]3)CC2)=O)C)ccnc2ccccc12 C(CCC(=O)NCCC(C)CCO)(C(C)C)NC(c1cc(OC)ncc1)=O c1(CC(N2CC3(NC(C4(F)CCCCC4)=O)CC2C3)=O)ccc2nc(O)[nH]c2c1 CCCC(C)CCCNC(c1ccncc1)C(C)C CCCCC(C)CCC(=O)N1CCC(CC)CC1.c12cn(nn1)CCC(=O)NC2 N1(C(CCC)=O)CCOC(Cn2cc(C3CCN(C(=O)CC(O)CC)C3)nn2)C1 C1(CNC(CN2CC(C)(C)C2)=O)CCCC12CCN(C(c1ccsn1)=O)CC2 C1(C(=O)Nc2c(OC)nn(C)c2)CC(C)CN(C(=O)C=Cc2cc[nH]c2)C1 C12(NC(CN3CC(C)(OC)C3)=O)CCCC1(F)CN(C(=O)C=CC(C)(C)SC)C2 c1(C(=O)OC)cc(O)ncc1CNC(c1ccc(CN2CCCC2)cc1)=O c1(C(=O)NC2(C)CN(C(C3C(C)(COC)C3)=O)C2)ccc2occ(C)c2c1 c1(C(C(=O)NC(c2ccc(F)s2)C)F)cccc(Cl)c1F c1(COC)nc(C(=O)NCCNC(C2CC(C(C)C)C2)=O)co1 N1(CC(=O)NC(CN(C)C(C2(C(F)(F)F)CC(F)C2)=O)C2CC2)CCCCCC1 C1(C2(O)CN(C(c3ccsc3)=O)C2)(CNC(C2(C#N)CCCO2)=O)CC1 CC1(C)CCC(C)(NC(=O)CC2CN(C(C3CC(=C4CC4)C3)=O)C(C)(C)C2)CC1 c1(COC)cc(C(N2CCCC2C(C)(C)NC(c2ccncc2)=O)=O)c(C)o1 NC1CCCS(=O)(=O)C1CC(=O)N1CC1.c1(CN2CCCC2)cccs1 N1(C(c2n(CC)ccn2)=O)CCN(C(=O)CCC#N)C(COC)C1 C1(C2CCCN(C(c3coc(C(C)C)n3)=O)C2)(NC(C(COC)C)=O)CC1 c1(C(=O)NC(C(=O)OC)CC2CC(F)(F)C2)ccc(N)cc1-c1ccccc1 C1(F)(CNC(C(C)=C2CC2)=O)CN(C(=O)CC(C)C2CCCO2)C1 C(C(C)(C)C(=O)N1CCC(NC(C2CCCO2)=O)C1)N(C)C CCCC(C)(CC)C(=O)N1CCCC(N(C(=O)C=Cc2ncc[nH]2)C)CC1 Cc1ccc(C=CC(N2CC3CC(C2)C3NC(c2nccn2C)=O)=O)c(C)c1 Cc1ccc(C)c(SCC(=O)NC2CN(C(C3CC4CC4C3)=O)CCC2O)c1 C1(NC(=O)CC(F)(F)F)CCN(C(C2CCCCO2)=O)C12CC2 C1(CNC(C=CC(C)(C)NC(C=CC)=O)=O)CC12CCCCC2 c1(C(=O)NCC(C)N(C)C(C2CCC(=O)N2C2CC2)=O)cc([N+](=O)[O-])cnc1N N1(C(C2N(S(C)(=O)=O)CCC2)=O)CC2=C(C1)CN(C(=O)C(C1CCOCC1)F)C2 c1(C(=O)NC(C(C)NC(C=CCC)=O)CO)cc2c(=O)cc[nH]c2s1 c1(C(=O)NC2(CCC(=O)Nc3cccc(SC)c3)CCCC2)[nH]ccc(=O)c1C C=CC(C)(C)CC(=O)N1CCC(NC(=O)Cc2cnsc2)C1C C1(C(N(C(C)C)C(c2ccco2)C)=O)CCN(c2ccc(OC)nn2)CC1 N12C(CC1C)C(=O)N1CC(C1)C2=O.C1(CCOCC)(CO)CC1 CC(CC(C)(C)C)C(C(=O)NC1CCOCC1)N1CCCCC1C1CC1C(F)(F)F C1(CNC(C2CCC(C(C)(C)O)CC2)=O)CC(O)C12CCC2 S(=O)(=O)(c1cc(C)c(Cl)c([N+](=O)[O-])c1)CNCCOCCOCCCNC(CCCC)=O c1(C(N2CC(C)(NC(Cc3c(OC)nc(Cl)cc3)=O)C2)=O)csc(S(C)(=O)=O)c1 c1(OC)cccc(=NC(=O)C2CC3(C2)CC(C(N2CCCC(Br)C2)=O)C3)[nH]1 N1(C(C2CCN(C(C3CC3c3ccco3)=O)C2)=O)CCCC(OCCO)C1 N1(C(c2c(C)cccc2Cl)=O)CCCN(C(=O)C(F)C2CCC2)CC1CO C1(C(=O)NC(C2N(C(c3ccc(C)o3)=O)CCC2)(C)C)CC2(CCCCC2)C1 Cc1c(CC(N2CCC(C)C2CNC(=O)C(c2ccc(F)cc2)O)=O)ncn1C C1(CNC(C2(CC(C)=O)CCCC2)=O)CC(C)N(C(c2cc(C)c(C)o2)=O)C1 C1(CNC(CN(S(CC)(=O)=O)C)=O)CCN(C(=O)Cc2cc[nH]c(=N)c2)CC1C C(CCCC(=O)NC1(CCNC(c2cc(C)cc(Cl)c2)=O)CCC1)(OC)OC C1(C2CC2)(C(=O)NC(c2nccc(O)n2)C)CN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 c1(C(N2CC3C(CNC(C4OCCN(C)C4)=O)C3C2)=O)ccc(=O)n(CCO)c1 N1(C(c2c(OCC)ccc(F)c2)=O)CCCCCC(NC(=O)C(C(C)C)SC)C1 C(CC(O)C(=O)NC1C=CCCC1C(=O)NOCCN(C)C)N(C)C c1(CCC(=O)NC(CC)CN(C(=O)CC2COCCO2)CC)cncc(F)c1 c1(OC(C)C(N2CCC(CNC(=O)CN(C)C3CC3)CC2)=O)cccc(CO)c1 N1(C(C(CC=C)CC)=O)CC(NC(=O)CCCCC(C)=O)C2(CCC2)C1 c1(C(N2CC(N(C(C(COC)C)=O)C)C3(C2)CC3)=O)cc2c(Cl)nccc2s1 C#CC1CC2(CC2)CN1C(C1(C)CCCN1C(=O)CC(C)CC)=O C1(NC(CC(C)NC(N)=O)=O)CN(C(=O)CC(C)(C)c2ccccc2)CC1F C1(CNC(CCCCCC)=O)CN2CCCCC2CN1C(=O)CSc1cccs1 C1(NC(COCC)=O)CC2(NC(c3cccc(F)c3Br)=O)COC1C2 C(=O)(C#CC1CCOC1)N1CCC(CC)(NC(c2cc(C(=O)NC)c[nH]2)=O)CC1 c1(C(=O)OCC)ccnc(N(CCCCN(C)C(c2n[nH]c(O)n2)=O)C)c1 c1(NC(C(C)N(C(C2(COC)CC2)=O)C2CC2)=O)ccn2ccnc2c1 CC1CC(=O)CCC1C(=O)NC1CC(C)N(C(=O)C=CC2CC2)C1 N1(C(C2(OC)CC(CF)C2)=O)CC(NC(c2cc(C)nc(O)c2)=O)C2(CC2)C1 Cc1nc(C(=O)NCCCOCCCO)c2c(C)c(C)sc2n1 C(CCC(C)C(=O)N1CCC(C(=O)NCc2ccnc(CO)c2)C(C)C1)OC C(=O)(CC(O)CC(C)C)N1CCC(COC)(NC(=O)C(C)n2ccnn2)C1 c1(C(N2C(CNC(C=C(CCC)CCC)=O)CC2)=O)ccc(C2CC2)nc1O c1(C2C(C)(COCC)C2)nc(-c2ccoc2)nn1Cc1nncn1CC c1(NC(=O)NC(CC#CC)C)ccc(NC(=O)OC(C)(C)C)cc1Br c1(C(=O)NCC(C)N(C)C)ccc(CNC(=O)C(N)=O)o1 C1(C(=O)NC2C3CCC2CN(C(c2ccno2)=O)C3)CC2(CO1)CC(F)(F)C2 c1(NC(C2C=CC(NC(c3nc(C)sc3C)=O)C2)=O)ccc2ncnc(O)c2c1 N1(C(C=CC)=O)CSCC1C(N1CCCC1CSC)=O Cc1nccc(Cl)c1C(=O)NCC1(CNC(C2CCC(=O)N2)=O)CC12CCC2 c1(C(N2CC(NC(C=Cc3scc(C)n3)=O)(CO)C2)=O)cncn(C)c1=O Cc1cccc2oc(C(=O)NC3CN(C(=O)CCc4ccsc4)C3)cc12 N1(C(CC(C)(C)OC)=O)CCC2CC2N(C(c2cnnn2C2CC2)=O)CC1 C1(C(=O)NCCCCNC(C(C)NS(C)(=O)=O)=O)CCOC(=O)CC1 c1(C2C(COC(Cc3c(Br)cn(C)n3)=O)C2)cc(F)cc([N+](=O)[O-])c1 N1(C(C(CC)(C)O)=O)C2CCC(C2)C1C(=O)NCC1CCCN(C)C1 c1(CN(C(C)=O)C)n[nH]cc1C(=O)NC(C)C(c1ccccc1)C c1(CCC(C)C)ccc(S(=O)(=O)NC2CCC3(CCNC3)CC2)cc1 c1(CNCCC2C(=O)OCC2)cc(C(F)(F)F)ccc1O CCCC(CNC(=O)CN1CCOC1=O)C(=O)NCCC1CC2C=CC1C2 c1(C(=O)NCC2CCC(C(NOCCOC)=O)C2)nccc(C)c1F C(C)(C(C(=O)N(C(C)C(C)C1CC1)C)C(C)C)NC(COCC=C)=O C1(C(N2CCC(CCN(C)C(C3CC3C#N)=O)CC2)=O)CC2(CCCCC2)C1 c1(C(N2CCC(CC=C)(NC(=O)CCC(=O)NCC)C2)=O)sc2cncn2c1C c1(C(N2CCC3NCCC23)C(=O)OC)ccc(F)cc1F C1(CCNC(C(C)(C)C2CCOC2)=O)CCN(C(=O)CC2(C#N)CC2)CC1 N1(C(c2c(C)csc2)=O)CCC(NC(c2nccc(C(F)(F)F)n2)=O)C(C)(C)C1 C1(C)(CC)NC(=O)N(CC(=O)NC2CC(CCNC(c3cnn[nH]3)=O)C2)C1=O C(=O)(C1CCCn2nccc21)N1C2(CN(C(=O)OC(C)(C)C)C2)SCCC1 C#CCC(C(=O)NCC1CC1CC(=O)NCC(CO)C(C)C)C1CC1 Cc1cc(C(N2CC(NC(=O)Cn3nc(C)cc3C)C3(CC3)C2)=O)c(C)c(C)c1 N1(C(C(C)Cc2cnc[nH]2)=O)CCCOC(CNC(=O)C(C)(C)N2CCCC2)C1 c1(C(=O)NC2C3CCN(C(Cc4cn(CC)nc4)=O)C3C2)ccc(S(C)=O)cc1 c1(OC)c(C(=O)NCCC2(OC)CN(C(=O)CC3CC(F)C3)C2)ccnc1F C(=O)(C1CCOc2ccc(Cl)cc21)NCC(CC(C)C)NC(c1cncn1C)=O c1(C(N(C)CC2CCSC2)=O)coc(CNC(=O)CN2CC3CC3C2)n1 N1(C(c2cc(C)c(Br)o2)=O)CC2CC1CN2C(c1cccc(N(C)C)c1)=O N1(C(C2N3C(C)CN(CC3)C2)=O)CC2CCCC(C1)N2C(=O)CCC1CC1(Cl)Cl CC(CF)CC(=O)NC1CN(C(C2(n3cncn3)CC2)=O)CC1F c1(NC(C2(COC)CN(C(=O)CCC3CCCCO3)C2)=O)ccc2nccn2c1 C1(OC)CN(C(=O)C(C2CC2)SC)CC1NC(c1cc(C(F)(F)F)n[nH]1)=O c1(OC)ccc(C(=O)NCCN(C)C(C2C(c3nc(=N)[nH][nH]3)C2(C)C)=O)c(F)n1 S(=O)(=O)(c1c[nH]c(C(N2CCC(NC(C3CC(CF)C3)=O)C2C)=O)c1)NC c1(C(=O)NCC(CC)NC(C2C3CCC23)=O)ccncc1Oc1ccccc1 c1(C(=O)NC2CCN(C(=O)Cc3ccno3)CC2O)ccnc2cc(Cl)ccc12 O=C(C(O)Cc1ccco1)NC(CCO)C1CCCC1.C12CC1C2.C(=O)N c1(C(C(=O)Nc2c(C)cc(F)cc2)N(C2CCC(C)C2)C)ccc2c(c1)CC(=O)N2 c1(C(N2CC(NC(CN3CCC(C)C3)=O)CC2(C)C)=O)cc(S(C)(=O)=O)co1 C1(CNC(c2c(CC)cns2)=O)N(C(=O)CC2CCCOC2)CCCC1(C)C N1(C(C(C)SCCCC)=O)CC(C(=O)NCc2oc(C)nc2C)C(F)(F)C1 CC(C)CC(C(=O)N1CCCC(NC(C2(C)CCCNS2(=O)=O)=O)CC1)C(N)=O N1(C(c2cccc(Cl)c2O)=O)CC2(CCCN(C(c3cnn(CCO)c3)=O)C2)C1 C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC(C)CCCNC(=O)C(C)N(C)C c1(CNC(=O)CC2CCC2)nc(CNC(=O)C(c2ccc(Cl)s2)=O)cc(O)n1 c1(CCC)cc(C(=O)N(C(C)C(=O)N(CCCCO)C)CC)no1 N1(C(C(CC)n2ccnc2)=O)CC(NC(C2CC(OC(F)F)C2)=O)C(C)C1 C1(NC(COC2CN(C(CC)=O)C2)=O)CCOC2(CCCC2)C1 c1(CC(=O)NC2(C)CN(C(CCCOCCC)=O)C2)ccc(O)cc1Cl c1(C(N2CC(C(C)NC(C3CCC(F)C3)=O)OCC2)=O)cccc(C#CCO)c1 c1(C(=O)NCC(C)N(C)C(C2CC2(C)Br)=O)cccc2c1OCC2(C)C c1(C(=O)NC(CNC(C(C)(C2CC2)NC(C)=O)=O)(C)CO)ccn(C)c(=O)c1 N1(C(N)=O)CCCc2c(NC(CN3CC(c4c(C)ccnc4)C3)=O)cccc21 c1(NC(C(C2CCN(C(C3CCCS3)=O)CC2)C)=O)ccc2ccncc2c1 c1(C(=O)NCC2N(C(C(COC)OC)=O)CC=C2)ccc2c(c1)CC2 C1(NC(C2CC(=O)NC2)=O)CCC2CCN(C(c3cnc[nH]3)=O)C12 C12N(CCC1(C)C)C(=O)C(=O)NC2.C(CN=[N+]=[N-])OCC(=O)NCCCOCC C1(CNC(c2cc(Br)cs2)=O)CC2(CCC2)CN1C(C1CCCO1)=O CCCCC(C(=O)NC(c1cnn(C)c1)CC)NC(c1cccc(C)c1)=O Cc1cccc(C(N2CCC(CNC(C3(C(N)=O)CCC3)=O)C2)=O)c1I C1(CCNC(C(C(C)O)(F)F)=O)CCN(C(C2CC(=O)CCO2)=O)CCC1(F)F c1(C(=O)OC)cc(C)n(CC(N2CC(CNC(=O)CC(C)C)CC2C)=O)n1 Cc1cc2cc(CNC(NC3CCc4ccc(F)cc43)=O)ccc2n1C C1(F)(C(=O)NC(C)C(C)n2cccn2)CCN(C(=O)CC2CCC=CCC2)CC1 C1(O)(CNC(C(C(C)C)O)=O)CCCN(C(C2CCC(O)CC2)=O)C1 Cc1ccc(C(=O)NC(CCCO)C(=O)O)c(OCCN=[N+]=[N-])c1 C(=O)(C1=CCS(=O)(=O)C1)NCCC(C)N(C)C(c1nncn1C)=O Cc1cc(C(=O)NC2CCC(NC(=O)CC3CCCO3)C2)cc(Cl)c1Br S(=O)(=O)(c1ccccc1[N+](=O)[O-])NCCCC=C N1(C(c2cccc(OC)n2)=O)CCC(C2(O)CN(C(=O)C(C)CN(C)C)C2)CC1 C1(NC(C(CC)O)=O)CCCCCN(C(C2(C)CCC2)=O)C1 C1(c2ccccc2)(C(=O)NC(C)CCCNC(C2CC2F)=O)CCN(C)C1 N1(C(C(C(C)NC(C(CC)COC)=O)C)=O)CC2CCC(C1)O2 Cc1ccc(C(=O)Nc2cccc(NC(C3(C(F)(F)F)CCC3)=O)c2)cc1 C1(C(N2CCC(OC(C)C)C2)=O)(NC(=O)C(C2CC2)N(C)C)CCCC1C CC(CCC(=O)N(CCCNC(c1cc2n(n1)CCC2)=O)C)S(C)(=O)=O N1(C(Cc2nc(CC)sc2)=O)CCOC2(CCN(C(=O)CCNC(=O)CO)C2)C1 Cc1cc(CNC(=O)NCc2n[nH]c(=N)o2)[nH]n1 c1(C(=O)NCC(C)N(C(c2c(CC)cno2)=O)CC)ccc2ccncc2n1 C1(C)(C(=O)NCCN(C(=O)Cn2nc(C)c(Cl)c2C)CCC)CC(C)OC(C)C1 C1(C(=O)NCC(=O)N(CC)CC)CCCN(C(c2csc(Cl)c2)=O)C1 Cc1ncc(C(=O)NCc2cn(CC(=O)NC3(CF)CCCC3)nn2)s1 c1(N(S(CCC)(=O)=O)CC(=O)OCC)c(Cl)cc(S(=O)(=O)N2CCCC2)cc1Cl C1(F)(CNC(c2c(CC#N)ccs2)=O)CCN(C(=O)CC2C=CCC2)CC1 N1(C(c2cnc(C(=O)NC3CC(C(=O)OCC)C3)nc2)=O)CCC(F)(F)CC1.OCC N1(C(c2cnn(C)c2F)C(=O)NCC(F)F)CC2CCCC(C2)C1 CC(C)(CNC(c1ccoc1Br)=O)Cn1cccn1.c12n[nH]cc1CC(=O)N2 C#CCC(C)(C(=O)NC(C1CCCCC1)C)NC(=O)C(CCC)OCC CC1CCCC(C(=O)NC(c2ccnn2C)C(=O)N2CC(Cn3ccnn3)C2)CC1 C(CCN(C)C(c1cc(C(C)C)ccc1N)=O)(C(C)(C)C)NC(CCC)=O Cc1cc2ccnc(NCc3ccc(C4CCCCC4)cc3)c2cc1Cl c1(C(=O)NCCCN(C)C(C2CC(C)(C)O2)=O)cc2c(cc1Cl)NC(=O)CO2 C1(CC)C(NC(c2c[nH]nc2-c2ccn(C)n2)=O)CCN1C(=O)Cc1ccco1 CC(C)CCC(O)C(=O)NC1CCCCC1CC(=O)NCC(O)CNC(N)=O C(C(C(=O)NC1CCC2(CCCC2)C1)C(C)(C)C)NC(COC(CC)C)=O c1(CC(=O)NC2CC(NC(c3cncc(C(F)(F)F)n3)=O)CC2O)c[nH]ccc1=O C(=O)(C1=C(C)CCCC1(C)C)N(CCC)Cc1ccc(SC)cc1 N1(C(C(C)CC2CCCC2)=O)CCN(C)CC1C(=O)NCC1CC(O)C1(C)C N1(C(C2C(C)CC(=O)N2)=O)CCCCC(CNC(=O)CC2(C)OCCO2)C1 c1(C2C(NC(N(C)Cc3ccc(C(=O)OC)[nH]3)=O)C2)cccc(Cl)c1Cl c1(COCc2[nH]c(=N)sc2)ccc(NCCC(=O)NC(N)=O)cc1 C1(NC(c2c(COC)cco2)=O)CCN(C(c2cc[nH]n2)=O)C1C(C)(C)C c1(C(=O)NC(C2CCCN(C(=O)OC)C2)C)nc2ccc(Br)cn2c1F C1(CNC(CC2N(C)CCC2)=O)(CO)CCN(C(=O)CC2(N(C)C)CCC2)C1 c1(C(=O)NCc2ccc(CCNC(C3CSC3)=O)cc2)ccc2ncccc2c1 C1(N(C(c2cc(COCC)sc2)=O)C)CN(C(=O)CSC(C)(C)C)CCC1C N1(C(CC(CC)O)=O)CCC2(CNC(c3[nH]c(O)nc3C)=O)CCCC12 C#Cc1ccc(NC(=O)NCC2CC23CC3(F)F)c(F)c1 C#CCC(C)(C(=O)N1CCSCCC1C)NC(=O)CC1(C#N)CC1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(N(C(=O)CC2(N(C)C)CC2)C)C2(C1)CC2 CC1(C)CCC12CN(C(C1CCCCC1NC(=O)CC1C=CCCC1)=O)C2 C1(C(=O)NCCC(C)(C)NC(=O)CCc2ccc(F)cc2)C=CC=CC=C1 c1(C(CNC(C2CCCC2O)C(=O)NCc2ccco2)N(C)C)ccccc1Cl CON(C)C1CN(C(C2CC2CNC(=O)C(C)C(=O)OC)=O)C1 C1(C(=O)NC2CCN(C(=O)OC(C)(C)C)C2C2CC2)CCCCNC1=O c1(C(N2CCC(CNC(Cn3c(C)ncc3)=O)C2)=O)snc2ccccc12 c1(C(=O)NCc2ccc(OC)c(OC)c2)c[nH]c2ccc(C3=CCCCO3)cc12 C1(CNC(Cc2c(C)occ2)=O)CN(C(=O)CC2CCCOC2)CC(C)(C)O1 c12ccc(cn1)CN2C(Cc1ccccc1)C(OC)OC.C(=O)(COC)OCC C1(NC(c2c(CCC)nco2)=O)CCC(NC(c2n[nH]c(C)c2Cl)=O)CC1 c1(C(N2C(C(=O)NC3C=CCCC3)CCCC2)=O)cc(F)ccc1F c1(OC)cc(I)c(CNC(C2CC(O)C(O)CN2)=O)cc1OC c1(C(N(C)CCOCCNC(=O)CC#N)=O)cncc2sccc12 c1(CC)ccc(C(N2CCCCC2c2nc(=O)o[nH]2)=O)c(OC(C)C)c1 Cc1ccc(C(N2C3CCC2C(F)C(NC(C2CCCC2)=O)C3)=O)c([N+](=O)[O-])c1 N1(C(C2CC(CN=[N+]=[N-])OC2)=O)CCc2sc(-c3nn[nH]n3)cc2C1 C(C(C)CC(=O)NCCC(C)NC(c1cn(C)c(O)n1)=O)OC C=CCCCS(C)(=O)=NC(=O)C(CNC(=O)CNC=O)C(C)C c1(C(=O)NCC(CNC(C2(OCC)CCOC2)=O)O)ccc(P(C)(C)=O)o1 c1(N2CCCC(C(C)NC(C(C)NC(COC)=O)=O)C2)cccc(F)c1[N+](=O)[O-] C1(C(N(CCN(CCC)C(c2ccsc2)=O)CC)=O)CCCN1C(=O)C(C)C c1(C(N(C)CC2CCCC(NC(CSC)=O)C2)=O)cnc2n[nH]c(C)c2c1 c1(C(=O)OC)nc(Br)ccc1NC(C1CC(F)CN1Cc1cc(Br)co1)=O c1(C(=O)NCCC(C)N(C(=O)CN2CC(=O)NC2=O)C)cccc(N)c1Br c1(NC(c2c(-c3cn(CCOC(C)(C)C)nc3)csc2)=O)cnc2sccc2c1 N1(C(C(c2cnn(C)c2)C)=O)C2CCCC1CC(NC(C1C3CN(C)CC13)=O)C2 C1(CC(=O)NCC2(N(C(C=CC)=O)C)CC2)CCCC(C)(C)C1 C12(C(=O)NCC(C(C)C)NC(=O)CCc3nnc(S)n3C)CC=CCN1CCC2 N1(C(CCCCC(CC)C)=O)CCC(C2CCCN(C(=O)C(C)CSC)C2)C1 C(=O)(C(C)CC(F)F)N1CCC(N(C(=O)Cc2cccc(C3CC3)c2)CC)C1 N1(Cc2ccnn2C)CC(=O)Nc2cc(C3CC3)ccc21.C12CCN1C(=O)N2C c1(NC(C(C2CN(C(c3cnc(C)s3)=O)C2)O)=O)c(C(N)=O)cccc1Br Cc1cnc(NC(=O)NCc2cccc(CSc3nccn3C)c2)cc1I CC1=NOC(C(N2CC(C(N)=O)(CNC(=O)C(F)C3CCC3)C2)=O)C1 c1(NC(C2C3CN(Cc4ccc(OC)nc4)C2C3)=O)cnc(Cl)cc1C c1(N(C(c2c(SC)occ2)C(=O)NC2CCN(C)C2)CC(=O)NC)cccc(O)c1 N1(C(C2(O)C(C)(C)C2)=O)CCCC(F)(CNC(=O)CCN2CCP(C)(=O)CC2)C1 c1(C(N(CC(C)NC(CCC(C)SC)=O)C)=O)cccc2ncnn12 c1(OC)cc(C(=O)NC2CN(C(c3ncccc3F)=O)CC2C)c(Cl)cc1Cl c1(OC)ccnc(CCC(=O)NCC(C)CN(c2ccc(F)cc2)C)n1 Cc1cc(C(N2CCN(C(C3CC3CC(C)C)=O)CC2C2CC2)=O)c(C)cn1 CC(C)CCCOCC(=O)NC(C1CCN(C(=O)Cc2ccsc2)C1)C N1(CC(=O)N(CCNCc2ccc(C(=O)O)o2)CC)CCC(F)C1 C1(NC(CC2C(C)(C)C(NC(=O)Cc3ccco3)C2)=O)CCC(C#N)CC1 N1(C(C2OCCN(C(CSCCCC)=O)C2)=O)CCC(CO)C1(C)C N1(C(C(CC=C)OC)=O)CCCC(F)(CNC(c2cnccc2Br)=O)C1 C12(C(=O)NCC(C#C)C(C)C)CC(CN(C(=O)C(C)(O)C3CCC3)C1)C2 C1(NC(CCC2CCC(=O)NC2)=O)CCN(C(c2ccc(O)cc2)=O)CC1F C#Cc1ccc(NC(=O)COC2CN(C(c3cc(C)c(C)s3)=O)C2)c(C)c1 c1(CC)[nH]nc(C(N2CC(CNC(c3scc(OC)c3OC)=O)C(C)C2)=O)c1C C#CCC(C)(C)C(=O)N1CCC1CNC(c1cnn(CC)c1Cl)=O c1(C(=O)NCCCC(C)NC(COCCOCC)=O)cc(Cl)c(C(F)F)cc1F N1(C(C(F)=CCC)=O)CCC(NC(c2cc(OCC(F)F)ccn2)=O)C1CC C1(C(=O)NC(CNC(c2c(C)nco2)=O)C(C)(C)C)CCC2(CC1)CC2(F)F c1(CC)c(C(=O)NCCC=CCNC(C2CCCN2CC)=O)cnn1C(C)C C(C)(C)(CC(=O)N1CCOCC1CN(C)C(C1CCC=CN1C(C)=O)=O)SC C(=O)(C1=CC(C)(C)C1)NCCNC(c1n(C(C)C)ncc1)=O c1(C(=O)NC2(C)CCN(C(C3CC3C#N)=O)C2)ccc(S(N)(=O)=O)o1 C(=O)(C(C)(C)C1CCCC1)NCC.CC(C(=O)N(C)C)N(C)C(=O)OC(C)(C)C N1(c2cccc(CNCC3CC(OCC)C34CCC4)n2)CCS(=O)(=O)CC1 N1(C(CC(CCC)NC(C2CC(C3CC3)=NO2)=O)=O)CCC12CCC(C)CC2 C1(COC)(CNC(=O)CC2CSCCO2)CCCN1c1ncns1 C(=O)(CC(C)(C)C(=O)OC)NCCC(C)NC(c1ccc(N(C)CC)cc1)=O c1(C(N(C2CCN(C(C3(COC)CCC3)=O)CC2)CCC)=O)cc(C)sc1C C1(C(N2CCN(CCCOCC)CC2)=O)CNC(=O)CN1C(c1nc[nH]n1)=O C1(C(=O)NCc2n(C)ncn2)CC2(CCN1C(C1CCC3CC13)=O)CC2 c1(C(=O)NCC2(CCNC(C3(F)C(C)OCC3)=O)CC2)cccc2c1NCCC2 N1(C(=O)C2CC2)CCC2CCN(C)C2C1.C1C(=O)NCC2(CC2)C(=O)N1C N1(C(C(C)C2CCC2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CC12CCCCC2 N1(CC)C(=O)CCC1C(=O)NC1CCCCC1NC(c1c[nH]nc1C(C)(C)C)=O C1(C(N(C2CCCN(C(=O)CSc3n[nH]c(O)n3)C2)CC)=O)COCCOC1 C=CCC(C)(C)C(=O)NC1CCCC(CC(=O)NCCCOCC)C1 C(=O)(C(O)C(C(C)C)OC)NCC(CC)NC(C1CC(C(C)=O)C1(C)C)=O N1(C(C2CCC(C(C)C)CC2)=O)CCC2(NC(c3ccc[nH]3)=O)CCCC12 Cn1cc2c(C(=O)NCC3CCC3NC(c3ccc(C#N)o3)=O)cccc2n1 C1(CNC(CSCc2nc(C)sc2)=O)CC(C)(C)CN1C(c1ccccn1)=O C1(NC(c2c(N(C)C)cccc2)=O)CC2(NC(=O)CCc3ccon3)COC1C2 n1(CC(=O)NC2C(C=C)CN(C(=O)COC(F)F)C2)cc(C)c(O)nc1=O c1(C(=O)NCC2CCCCC2NC(c2ccoc2Cl)=O)cc2sccc2cn1 c1(C(N(C)CCOCCNC(=O)CC2(C)CC2)=O)nncc2c1CCCC2 C1(C(=O)NCCCCN(C(C(CCC)OC)=O)C)CCc2cn(C)nc2C1 C1(C(=O)NCC2C(NC(c3cncc(CC)c3)=O)CC2O)CCn2ccnc2C1 c1(C(N2C(C(N(C3C(C)CC3)C)=O)CCC2)=O)cc(O)cc(=O)o1 N1(C(C2C(NC(c3cc(C)c(C)nn3)=O)COCC2)=O)CCc2ccsc2C1 c1(OC)ccc(O)cc1C(N1CC(O)(C(C)NC(=O)CC2CCCOCC2)C1)=O CCN=C(NCc1cccn1C)N1CCCC(CCCc2ccc(Cl)cc2)C1 CC1CN(C(=O)OC(C)(C)C)CCC1NC(=O)NC1CCN2CCC1C2 C1(C(N2CCC(CN(C)C(c3ccsc3)=O)C2)=O)CC(=O)N(CC2CC2)C1 c1(C(N2CCN(S(Cc3ccc(C#N)cc3)(=O)=O)CC2)=O)ccc2nsnc2c1 C1(NC(C2(OC)CC2)=O)CC2CCC1C(NC(=O)CC1=CCOCC1)C2 CC(C)C(O)CNC(=O)CSCCNC(=O)C(c1ccccc1)F C(=O)(CC(C(F)F)C(C)(C)C)NCc1ccc(-c2ncc(C)[nH]2)nc1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC2CCC12CNC(=O)CNC(c1ccco1)=O N=c1nc2ccc(C(=O)NC3CCC3NC(c3cncc4nc[nH]c34)=O)cn2[nH]1 CCC(C)(CO)C(=O)NCC(C(C)(C)C)NC(=O)CCc1ccccc1C#N c1(C(N(CCNC(C2COC(=O)O2)=O)CC)=O)ccc(OC)cn1 C1(C)(CNC(C(CC)F)=O)CCCN1C(=O)C(C)Oc1cccc(F)c1 c1(C(=O)NCCC(N2C(CNC(C=CC)=O)C(C)CC2)=O)nc2ccccc2s1 Cc1ccc(C(N2CCCCC2C(=O)NCC2C(CO)C2(C)C)=O)nn1 c1(CCNC(C2N(C(CC=C)=O)CCCCC2)=O)c(C)c(O)nc2ccccc12 C(=O)(C#CC1(C)CCCO1)NC1CC2N(C(C3CCC(OC)C3)=O)C(CCC2)C1 c1(CNC(C(=O)N(CC(c2cnn(C)c2)O)C)=O)ccc(C#N)c(I)c1 C(=O)(CCCCN1CCCC1)N(C1C=CCCC1CNC1CCN(CC)C1)C C(C(=O)N1CC2(C1)CC(=O)N2)(C(C)C)SCC.n1(CC)cc(CO)nn1 C#CC(C1CCc2ccccc21)NC(=O)C1CCCc2nccn21 C1(CNC(C2(SCC)CC2)=O)CN(C(c2cn(C(C)C)nn2)=O)C(C)(C)C1 n1(CC)ncnc1C(N1CC(F)(CNC(=O)Cc2cnsc2)C1)=O CN(OCC(F)(F)F)C(=O)OCc1nc(CCCN(C)C)n[nH]1 c1(C(=O)NC2CCN(C(C=CCC)=O)CC2F)cnc2[nH]cc(C)c2c1 c1(CNC(N(CCCCN2CCOCC2=O)C)=O)ccc(Cl)c(F)c1 c1(OC)cc(C(=O)NC2CCCC2CNC(C2CC3CC3C2)=O)ncn1 Cc1cc2[nH]c(C(=O)NC(C)CCN(C(=O)Cn3cnnc3O)C)cc2o1 CN=c1[nH]c(=NCC2CCCN2C)[nH]c(=NCC(C(C)C)Oc2ccccc2)[nH]1 C(=O)(C(C)CC(N)=O)N(C1CCN(C(=O)C(COC)OC)CC1)CCC c1(SC)cc(C(N2CCN(C(C3(C4CCCO4)CC3)=O)C(C)C2)=O)ccc1N c1(CN(C(=O)NC2CCC(N3CCOCC3)C2)CC)cc(F)ccc1F c1(OC)ccc(CN(c2ccc(C3SCCS3)cc2)C(C2CCCCC2)=O)cc1F CC1=C(C(=O)N2CC(NC(C3(C)CCCNC3=O)=O)CC(F)C2)CCCC1 S(=O)(=O)(c1c[nH]ccc1=NCC1CCCC(C)O1)NCC1(OC)CC1 N1(C(C(CNC(=O)CCc2ccoc2)N(C)C)=O)CCOCC1CO c1(OC(C)C)ccc(Cl)cc1C(=O)NC1CCC(NC(c2occc2Br)=O)C1 C=CC(C)(O)C(=O)NCCN(C(=O)CCCNC(c1cccs1)=O)CCC c1(CC)ccc(OCC(=O)NCCNC(=O)C(C)Sc2ccccc2)c(OC)c1 CC(CN(C(=O)Cc1cc[nH]c1)C)C(=O)NCc1[nH]nnc1C1CC1 N1(c2c(C#N)cnc(C)n2)CC2CCN(C(c3cc(Cl)n(C)n3)=O)CC2C1 CN1CCC(C)(C(=O)N(CCCNC(=O)CSCCCc2ccccc2)C)CC1 n1(CC)cc([N+](=O)[O-])c(C(=O)NC(C)CN(C(=O)CC2CN(C)CC2O)C)n1 c1(CNC(C2(CC#C)CCN(C(C3CC4(CCC4)C3)=O)C2)=O)ccc(C)c(F)c1 C1(C(=O)NCc2cocn2)CCN(C(c2cncc(CO)c2)=O)CC1O CC1CCN(C(=O)CCn2ccccc2=O)CC1NC(=O)CC(F)(F)F N1(CC)CCCC(OCF)C1.c1(C(C(=O)Cn2nnnc2C)=O)oc(CNCC)nc1C Cc1cc([N+](=O)[O-])ccc1CN=c1cc(NCCn2cc(C3CC3)nn2)nc[nH]1 CC1CN(C(c2cccc(Cc3ccccn3)c2)=O)CC1NC(=O)C(Cl)=CCl c1(C(N(CC(=O)NC(C#C)C(C)C)C(C)C)=O)cn2ccccc2n1 C1(NC(C(Cn2cc(COC)nn2)F)=O)CC(CO)C12CCC2.C1CO1 C1(CNC(c2cc(C)ncc2)=O)CN(C(C2C3CNC(=O)C23)=O)CC(C)(C)O1 S(=O)(=O)(c1ccc(NCc2cc3cccc(F)c3o2)c(Br)c1)NCC1(CC)CC1.C1CC1 Cc1cc(S(C)(=O)=O)ccc1NC(C1C2CN(C(=O)CC#N)CC12)=O C1(CC(=O)NC2C(NC(CNC(=O)OC(C)(C)C)=O)C2)CC12CC2 c1(C(N2C(C)CC(NC(=O)Cn3cncn3)C2)=O)ccc(O)c(Cl)c1 CC(CC(C)(C)C)C(=O)N1CCCCCC1CNC(C12CC(C(C)(C)C)(C1)C2)=O Cc1nc2ncnn2cc1C(=O)NCC12CCCC1N(C(=O)C=CCF)CCC2 c1(NC(c2ncc(C(=O)OCC)cn2)=O)nccc2nc(C)ccc12 N1(C(c2ocnc2C2CC2)=O)CC(C2CCCN(C(c3cnns3)=O)C2)C1 C(CC(=O)NC1CC(CCNC(=O)C(C2CCCC2)NC(C)=O)C1)OC Cc1ccc(C=CC(=O)NC2CCC2CNC(=O)CCc2cccnc2C)o1 C1(CC(=O)N(CCCN(C(C2(C)CN(C)C(=O)C2)=O)C)C)CCC2(CCC2)CO1 C1(C(N)=O)CCCN(C(=O)CCCCc2nn[nH]n2)C1Cc1ccccc1C(=O)O c1(NC(C2CC23CCN(Cc2cc(O)cc(O)c2)C3)=O)cnc(Cl)cc1Cl C(=O)(C(C)(C)C)NCCC(=O)NCC#CCNC(CCNS(CC)(=O)=O)=O N1(C(c2ccc(C)cc2-n2cc(C(C)(C)F)nn2)=O)CCCC2(COCCN2)C1 Cc1cc(C(N2CCCCC2CNC(C2CC(n3cccn3)C2)=O)=O)nc(C)c1 CCCCC(CC)CCC(=O)N1CC(NC(C2(C)CC(=O)N(C)C2)=O)C1 C1(C(N2CC(F)(CNC(C3(NC(C)=O)CCCC3)=O)C2)=O)CCCC(C)(C)C1 N1(C(c2c(C)[nH]cc2)=O)CCN(CC(=O)NOC2CCN(C)CC2)C(=O)C1 CCC(CC(=O)N1CC(CCO)(NC(C2CNC(=O)O2)=O)C1)OC c1(C(CC)C)ccc(C(=O)NC2CN(C(=O)CC3OCCCC3(C)C)C2)c(O)n1 C1(C(N2CC(NC(CN(C)C)=O)C(O)C2)=O)CCC(C2CCC2)CC1 c1(C(=O)NCCCNC(COC2C(C)CCCC2)=O)ccc2c(c1)C(=O)CCO2 C1(C(N(CCC(=O)OC)C)=O)CCCC(NC(=O)Cn2ncn(C)c2=O)CC1 c1(CC(=O)NC(CC(C)NC(c2cnc(CC)s2)=O)C)ccc(C(C)(C)C)cc1 c1(CC(=O)N(C2CCC(NC(C3CC=CC3)=O)CC2)C)cccnc1O c1(-n2c(C(=O)NC(C3CCN(C(=O)OC)C3)C)cnc2)ncccc1Cl N1(C(c2c(C)snc2)=O)CCC2(CCC(NC(=O)Cc3cccc(Cl)c3)C2)CC1 C1(C(N2CC(N(C(CC(C(C)C)O)=O)C)C(O)C2)=O)CCC(=C(F)F)CC1 Cc1cc(NC(=O)C(N2CCC(C)(N)C2)=O)ccc1C(N1CCOC(C)C1)=O n1(CC(=O)NC2CN(C(C(C)CO)=O)CC(F)C2)c(S)nc2ccccc2c1=O N1(C(C(COC)N(C)C)=O)CCC(CNC(c2cccc(=O)n2O)=O)C1(C)C c1(CCC)ccccc1C(=O)NC1CCC(N(C(=O)CC2CC=CC2)C)CC1 c1(C(=O)O)ccc(C(F)(F)F)cc1[N+](=O)[O-].CCC(O)CC=O.C1CCOCCN1 C1(CCNC(C2CC2(Cl)Cl)=O)CN(C(c2cccc(=O)o2)=O)CCS1(=O)=O C12(CNC(CCC=CC)=O)CCC1CCN2C(c1cccc(Br)c1N)=O C(C(=O)N1CCC(CNC(=O)CC2CCCSC2)C1)(C(C)(C)C)OC C1(C(N2CCC(NC(=O)CC34CCCN3CCC4)C2)=O)CCc2ccccc2O1 c1(NC(c2ccn(C)c2)C)ncc2n1CCC2 N(C1CSCc2ccccc21)c1ncnc(NCCCCc2scc(C)n2)c1C C(=O)(C(C(C)(C)C)NC(=O)C=CC(F)F)NC(CC(=O)NC)C N1(C(C=Cc2ccc(CC)o2)=O)CC2(C1)CN(C(c1cc(=O)cc[nH]1)=O)CCO2 N1(CC(C)OC(F)F)C(=O)C2Cc3ccoc3N2C1=O c1(C(CCC)C)ccccc1COC(c1cnc(-c2cnccn2)s1)=O C1C(C(C)(C)C)NC(=O)N1C.C1(Oc2ccccc2)CCC2CC12.C(CO)SCC C1(C(=O)NC2CCC(NC(c3c(C)oc(CO)c3)=O)CC2)CCC(N=[N+]=[N-])CC1 C(C(C(=O)N1CCC2(CCC2)C1)C(C)C)NC(CC(OCC)OCc1ccccn1)=O Cc1ccc(C(=O)NCC(CO)NC(=O)C#CC2CC2)c(F)c1Br C1(CN(C(=O)NC(CC2(OCC)CC2)=O)C)CCCO1 c1(C(=O)NCCC(C)NC(c2cn(C)nc2Cl)=O)ccc(P(C)(C)=O)o1 C(=O)(C(C)(COC)OC)NCC1CCC(NC(C2(C)CC(=C)C2)=O)C1 C1(C(=O)NCC2CC(N(C)C)C2)CC(N=[N+]=[N-])CN1C(c1ccc(C#N)o1)=O N1(CC(CCOC)NC(=O)OC(C)(C)C)CCC(C(=O)OC(C)(C)C)CC1(C)C C1(C(N2C3CN(C)C(C3)C2)=O)C2CCCC1CN(C(=O)C(N)=O)C2 c1(NC)cnc(C(=O)NCC2CCN(C(C3CCC(OC)C3)=O)CC2)cn1 Cc1ccc(SC(C)C(=O)N(C(C)CNC(=O)CSc2nncs2)C)cc1 C1(NC(CCn2ccc(C)n2)=O)CCC(C)N(C(=O)COc2cccc(F)c2)C1 N(C1c2ccccc2CC1NC(=O)CC(C)CF)C(C(=Cc1ccco1)C)=O C1(CNC(CCC#C)=O)CN(C(c2nn(C)cc2Br)=O)CC1C(F)(F)F c1(NC(CC=C)=O)cccc(C(=O)NC(c2ccncc2)c2nnnn2C)c1 c1(C(=O)NCCn2cc(CNC(CC(C=C)C)=O)nn2)cc(Cl)cc2c1OCC2 N1(CC(=O)Nc2ccc3[nH]cc(CCC(N)=O)c3c2)CCCC2(CCCCN2)C1 C1(C(=O)NC2CC(C(C)C)C2)CCN(C(=O)Cc2ccsn2)C(C)(C)C1 C1(CC)CCCC(NC(=O)C(=O)NCC(n2c(C(=O)N)ccn2)N(C)C)C1.C1CC1 Cc1nn(C2CC2)cc1C(=O)N(C)CC1CCN(C(=O)CCC2CCCCO2)C1 c1(C(N(CC(=O)O)Cc2cn(-c3nccc(C)n3)nn2)=O)c(F)cccc1Br C1(NC(c2c(CC)c[nH]c2)=O)CCN(C(C2(C)CS(=O)(=O)C2)=O)CC(C)(C)C1 c1(C(=O)OCC(=O)NC)ccc(S(=N)(=O)C(F)(F)F)cc1 c1(C(=O)NC2COCCN(C(=O)C(C3CC3)C3CC3)C2)cc2c(Cl)nccc2s1 c1(CC(C)C(=O)N2CC(CCCCNC(=O)COC3CCC3)C2)ccc(F)cc1 C(=O)(CCCCCNC(c1c[nH]c(=N)o1)=O)N(C1CC(O)C1(C)C)C c1(OC)cncc(C(N2CCN(C(C3CC3C(F)F)=O)CC2C)=O)c1C n1(CC)ncc(Br)c1C(=O)NCCn1cc(C(N2CCOC2=O)(C)C)nn1 C1(C(N(C(C(=O)NC(c2ccn(C)n2)C)C)C2CC2)=O)CC2C(C1)C2(F)F C1(C(N2CCCC(C(C)C)C2)=O)CC2CCN(C(=O)CC3CCN(C)CC3)CC12 C(c1cc(C)cc(C)c1)=CC(=O)NC(C1CN(C(c2ncc(NC)nc2)=O)C1)C C12(C(=O)NC3CCCN(C(Cn4nnc(=N)[nH]4)=O)C3)CCCN1S(=O)(=O)CC2 C1(NC(C2(SC)CCC2)=O)CCCN(C(c2c(C)nc(COC)s2)=O)CC1 c1(C(=O)NC(C)CNC(=O)CCC2CC2(F)F)cnc2n1C(C)CCC2 C1(OC)CC(C(=O)NCC(C)(C)NC(=O)CCCc2nncn2C)C12CCC2 N1(C(CC=C=C)=O)CCC(NC(=O)C(F)=C(C)C2CC2)C(C)(C)C1 C(CCCCC(=O)N1CC(NC(=O)CCCn2cccn2)CC1C)OCC N1(C(C2N(CC)CC2)=O)CC2CCC(C1)N2C(C1(C2CCCO2)CCOCC1)=O C1(C(=O)NCC(C)NC(CCc2cnc(C)o2)=O)CCN(S(=O)(=O)N(C)C)C1 CC(C)C(F)(F)CC(=O)N1CCCC1CNC(=O)C(n1ccc(Br)n1)C C#CC1CCN1C(=O)C(Cc1cnc[nH]1)NC(c1sccc1F)=O c1(NC(C2N(C(C(CC=C)C)=O)CC(OC)C2)=O)ccc(F)c(CO)c1 c1(C(=O)OC)cn(CC(=O)NCC(C)N(C(=O)CCN2CCOCC2)C)nn1 N1(C(C2OCCN(CC)C2)=O)CCCC2(NC(=O)CC3(OC)CC3)CCCC12 N1(C(c2cnc(C)n2C(F)F)=O)CCCC2CCC12Cc1nn[nH]n1 C(=O)(C1CCCc2ccccc21)N1C(CC(=O)NC2(C(=O)OC)CC2)CCC1 CC1(C)C(C(=O)NCc2ccco2)CCN1C(=O)CC1CCSCC1 C(=O)(C(F)(F)C(C)O)N1CCC(CC(=O)NCC(COCC)(C)C)CC1 C1(C(=O)NCC(C)CNC(c2ccn(CC(F)(F)F)n2)=O)CC2OC(=O)OC2C1 O=S(=O)(c1cnc(C2CC2)[nH]1)NCCn1cccn1 c1(C(=O)NC(CNC(C(C)N(C(C)=O)C)=O)C(C)C)cc(Cl)ccc1C(F)F C1(NC(C=C(CCN(C)C)Cl)=O)(CF)CCN(C(=O)CC2CC(C)(C)C2)C1 C(CCCCC(=O)N1CC2CC2(NC(C2CCN(C3CC3)C2=O)=O)C1)N(C)C c1(C2CC(NCc3ccc(-c4onc(C(=O)NC)n4)s3)C2)ccccc1C N1(C(C2CCN(C(c3cccc(CC#N)c3)=O)C2)=O)CCC2OCCC2C1 c1(C(N(CC(C)(C)NC(C2C3C4CCC(C4)C23)=O)C)=O)c[nH]c2nc(F)ccc12 C1(CNC(CNC(C)=O)=O)(CO)CCN(C(C2C(C=C(C)C)C2(C)C)=O)C1 c1(NC2CN(C(C)C)C2)[nH]c(=NC(C)Cc2ccco2)nc2c1cnn2C C12(C(=O)NC(C)C(=O)N3CC(OCF)C3)CCCN1S(=O)(=O)CC2 c1(C(N2CCCN(C(c3nccc(CC)c3)=O)CC2)=O)cccc2c1OCC2 Cc1ncc2c(n1)CCC(NC(=NCCCCl)NCCN1CCN(C)C(C)(C)C1)C2 N1(C(C2(SC)CCC2)=O)CCN(C(c2csc(C)c2C)=O)C2CCCCC2C1 Cc1nc(C(=O)NC2(CNC(=O)CC3(C)CC3(F)Cl)CCCCC2)c(C)o1 C1(CCNC(C2(c3cccnc3)CCCC2)=O)COCCN1C(C1CC1CF)=O c1(C(=O)NCCN(C(=O)C(C)=C(C)C)CC)ccc(-n2cccc2)c(F)c1 c1(C(C(=O)NC2CCC2)N(C(C)Cc2cnn(C)c2)C)ccnc(F)c1 c1(C2(CN(CCCCCN)CC)CCC2)ccc(Cl)cc1F c1(CSCC(N2C(CNC(C=CC)=O)CCC(C)C2)=O)nc2ccccc2s1 C(=O)(CC(C)(C)C)NCC(CC)(C)NC(c1cc[nH]c1C1CC1)=O C1(C(N2CCC(NC(c3c(C)ccs3)=O)(CF)C2)=O)CCCCN(C)C1=O C1(C(=O)NC2(CNC(C(=O)NC3CC3)=O)CCOC2)CC2(CO1)CC(F)(F)C2 c1(CC)nn(C)c(C(=O)N2c3nc2cc(O)n3)c1Cl.C12(C(=O)NC)CC(N)(C1)C2 c1(OC)ccc(NC(=O)NC(c2c(N(C)C)cccc2F)C)c(Cl)n1 c1(C(CNC(C(COC)(C)C)=O)NC(C2CCCN(C)C2)=O)cc(F)cc(Cl)c1 c1(C(=O)OCC)sc(CCc2cccc(SCC)c2)nc1C.C#CCNC(=O)OC C=CC1CN(C(c2cc(=N)[nH]c(Cl)n2)=O)CC1NC(C1(O)CCCCCC1)=O C#CCC(C)(CNC(C1CC(C)CN(C(=O)CNC=O)C1)=O)CO c1(C(N(C2CC(NC(c3scc(C)c3Cl)=O)C2)C)=O)ccc(F)cc1OC(F)F CCC(C)(CNC(=O)C(C1CCCC1)OC)NC(c1cc(CCOC)on1)=O C1(C(=O)NC2CC3CN(c4nc(C)c(Br)cn4)CC32)CCCC(C)(C)CC1 C1(NC(CNC=O)=O)CCN(C(C2(F)CCCC2)=O)CC1F C1(F)(CNC(C2C=CCC2)=O)CCN(C(=O)CC2COCCO2)CC1 N1(C(C(CCC)NC(C)=O)=O)CC2CCCC2(C(=O)NCC(C)(C)C(C)C)C1 c1(C(N2C3C(C(=O)Nc4cncc(SCC)n4)C(C3)C2)=O)c(C)ccc(Br)c1F N1(CCC)CC(C(=O)NC(CNC(c2sccc2F)=O)CC(C)C)CC1=O c1(C(=O)NCCCCCNC(c2n(C)ccc2)=O)c(Cl)csc1Cl c1(C(=O)N(C(CC2CC(F)(F)C2)CO)C2CC2)ccc(Cn2cccn2)cc1 c1(CNC(C(CNC(CCN(CC)CC)=O)(C)C)=O)ccc(F)nc1C CCC(CC)OC(CN(C(CN)=O)C(C)CSC)=O.C1CN1 C(=O)(C#CC(C)(C)CNC(=O)C(C(C)OC)N(C)C)N(CCC)CC Cn1ccc(C(=O)NC(C)(C)CCNC(=O)CC2CCCS(=O)(=O)C2)cc1=O C1(C(N2C(C(N(C(C(=O)OC)C)C)=O)CC2C)=O)C2CCC(F)C12 CCC(CC)C(C(=O)N1CCC1C(=O)NCCC(O)CCO)OC N1(C(C(CC)C#N)=O)CCC2C(NC(=O)CC3(C)CCOC3)C2C1 N1(C(C2(CNC(c3n(CC)nc(C)c3)=O)CC=CC2)=O)CCC(F)(C#N)C1 C1(C(=O)NCCCCCCN(C(=O)COc2ccsc2Cl)C)CCCCNC1=O Cc1ccc(C(=O)C(=O)NC2(CCNC(=O)C(C)c3ccsc3)CCC2)cc1 C1(N=c2[nH]nc(C3CC3)o2)(CNC(c2cc(CC)c(C)s2)=O)CCCCCC1 c1(CC)cc(C(=O)N(C2CCCN(C(C3CC(F)C(=O)N3)=O)C2)C)sc1C c1(OCCC(c2n(CC=C)nnn2)N)ccc(C(N)=O)cc1.C12(C)CCCC1C2 c1(C(=O)OC)ccc(C(c2c(CC)cccc2)=O)c(F)c1 C(CN=c1[nH]c(=NCCC(C)CC)[nH]c2c1CCC2)c1c(C)nn(C)c1 C1(NC(c2ccc(Cl)c3occc23)=O)CCOC12CCS(=O)(=O)CC2 C#Cc1ccc(C(N2CCN(CC(C)NC(=O)C(C3CC3)OC)CC2)=O)c(F)c1 N1(C(CCC=CC)=O)C2CCC1CN(C(c1cncc(C(F)(F)F)c1)=O)CC2 C1(C)(CC)CCN(C(C2(NC(=O)Cc3c(C)noc3C)CCCCC2)=O)C1 c1(NC2C(C=C)CN(Cc3ccccc3)C2)ncnc2c1ccn2C N1(C(=O)OC(C)(C)C)CCCC1CC(=O)NCC1C(C(=O)NCCC(O)CO)C1 CCCCCCC(=O)NCCC1CCC(NC(c2cc3sccc3[nH]2)=O)C1 CC(C)C(C(=O)NCC1(NC(=O)CC2CCOC2(C)C)CCC1)c1ccn(C)n1 C(=O)(C1=CC2CCC=CCCC12)N1CC(CCNc2ccc(OCC)nc2)C1 C1(C(N2CCc3ccc(O)cc3C2)=O)COC2(CCN(Cc3nccs3)CC2)C1 N1(CC(CC(C(=O)NCC(CC)(C)OC)COC)=O)CCCCS1(=O)=O C1(C(=O)NC2CC(OCC)C2)CCCN(C(=O)NC(CSCCCC)C2CC2)C1 c1(N2CC(C(C)O)C2)nc2ccc(S(=O)(=O)N3CCC(CC(C)O)CC3)cc2s1 C1(NC(CN(CCC)C)=O)CCCC(NC(c2ccc(=O)n(C(C)C)c2)=O)CC1 C1(CNC(Cc2c(C#C)cccc2)=O)CCCC2(CN(C(=O)C(CC)OC)C2)O1 CCCC(CC)NC(=O)C(C)CNC(C1(C(F)(F)F)CC1)=O CC1C2CCC(C2)C1C(N1CC(C(N2CCN(CC(N)=O)CC2)=O)C(F)(F)C1)=O C1(C(=O)NCC(CNC(CC2C(C)CCO2)=O)F)CCC(C(F)(F)F)CC1 CCC(C)C(C(=O)N1CC(OC)C1)N(C)C(c1cc(C(C)C)[nH]n1)=O C=CC(C)CC(=O)NC(C)(C)CC=CC(=O)NCC(C)O c1(C(c2nnnn2-c2ccccc2C)NC(CC)CSC)cc(Cl)cc(Cl)c1 S(=O)(=O)(c1ccc(=O)n(C)c1)NC(N1CCC(n2cc(NC)nn2)CC1)=O N1(C(c2cc(OC)ns2)=O)CC(NC(C2(F)CC2)=O)CC2(CCC2)C1 C1(NC(C2C(C)CCC2)=O)CC2(C1)CC(NC(=O)C=Cc1ccc(O)cc1)C2 C=CCC(C)(CC)C(=O)NCCCN(C(C1CCS(=O)(=O)C1)=O)C(C)C C(=O)(C(C(C)CC)N(C(=O)CCN(C)CCO)C)N(CCC#C)CC C1(CNC(c2ncn(CC)c2)=O)CCCCN(C(c2cn(C)nc2C2CC2)=O)C1 C1(NC(C2N(C(c3cc[n+]([O-])cc3)=O)CCC(=C)C2)=O)CCc2nn[nH]c2C1 C1(C(=O)NCC2CN(C(CCOC)=O)C2)CCCN(C(C)C)C1 N1(C(C=C(C)C(F)F)=O)CCC(C(C)NC(C2COC(=O)N2C)=O)CC1 c1(C(N2CC(COC)(NC(c3cc(C)n(C)n3)=O)C2)=O)cnn(C)c1S(N)(=O)=O c1(C(N2CCC(N(CCC)C(c3n[nH]cc3C)=O)C2)=O)cnn(C2CC2)c1C C=C=CCC(=O)N(CCCNC(C1CC1c1ccccn1)=O)CCOC N1(C(C(COC)(F)F)=O)CCCC2C1CCN2C(C1CC(F)(F)C1(F)F)=O CCC(C)CCCC(=O)NC1(COC)CCN(C(c2cc(F)c(C)cc2Cl)=O)C1 c1(CCOC)nc(-c2ccn(CC(F)F)n2)n(C2CC2)n1 c1(CCC(=O)NC2CC(O)(CNC(=O)C=CC(=O)NC3CC3)C2)cccc(Cl)c1 c1(C(=O)OC(c2cc(C)nn2C)C)ccc(F)c(CC#N)c1 c1(NC)ccc(C(=O)NCC(CC2CC2)C(=O)NCC2CC(=C3CCC3)C2)cc1 CCCS(=O)(=O)CC(=O)N1CC(C(F)(F)F)OCC1CNC(c1ccnn1C)=O c1(CC)nc(N2CC(CNC(=O)C(F)(F)C(C)O)(OC)C2)cc(C#N)n1 c1(C(N(CC)Cc2nccs2)=O)ccc(Br)c2cccnc12 c1(C(C(C)NC(=O)Nc2ccc(N3CCOCC3)nc2)=O)ccc2c(c1)OCCO2 S(=O)(=O)(c1cc2ccccc2s1)N1CC2C(CNC(c3nc[nH]n3)=O)(C2)C1 C(=O)(C1=NOC2COCC12)NCCn1cc(C(=O)NCc2c(C)nn(C)c2)nn1 CS(=O)(=O)C1(C(=O)NCC2(F)CCCN(C(C3CC4(CCC4)C3)=O)C2)CCC1 N1(CCN(C(CCN(C(CCC)C)C)=O)CC(C)O)CCOCC1.C(=O)(C=CCF)N c1(C(=O)NC(C)CCCNC(c2ccc(C3CCC3)cc2)=O)cc(O)cc(F)c1 C1(NC(C(C2CCN(C(C3(Cl)CC3)=O)CC2)C)=O)CC(=O)N(C)C1 C1(N(C)C(c2cc(C(F)F)no2)=O)CCCC(NC(c2cccn2C)=O)C1 N1(C(C2(C=C)CN(C(c3cc4cc[nH]c4cn3)=O)C2)=O)CCn2c(C)cnc2C1 c1(C(N(C2CCC(NC(c3ncsc3C3CC3)=O)C2)C)=O)c(F)cc(Cl)cc1F N1(C(CSCC)=O)CCCC(C(=O)N(CC(C2CCC2)OC)C)C1 N1(C(CCN(C(C)=O)C)=O)CCC(C(F)(F)F)C(NC(=O)CCn2cccc2)C1 N1(C(=O)Nc2c(OC)noc2C)CCSC(c2ccccc2)CC1 CC1(C)CC(CNC(C2CNC(=O)N2)=O)CN1C(=O)CNC(c1ccsc1)=O c1(C(N2CCCC(NC(=O)CSc3nncs3)C2)=O)ccc2snnc2c1 c1(C(N(CC(C)NC(=O)C(C)(C)CCSC)CC)=O)ccc2c(c1)N(C)CC2 C12(C(=O)OC)CCC(C(N3CCC(NC(=O)C(C)N(C)C)C(O)C3)=O)(CC1)CC2 CC(C)C(C(=O)NC1CCC1NC(C1CC1c1ccoc1)=O)NS(N)(=O)=O c1(NC(C)CNC(C2CCc3nnnn3C2)=O)ncnn2c(Br)ccc12 N1(C(C2(C)CC(C)C2)=O)CCCC(n2cc(-c3ncccn3)nn2)C1 N1(C(C(CCC)OC)=O)CCN(C)CC1C(=O)NCc1c(C)cnn1C CC1=NOC2(C1)CC(C(=O)NCCC1(O)CN(C(c3ncsc3C3CC3)=O)C1)C2 c1(OC)nc(=NCCN2CCN(C(=O)CCC=C(C)C)CC2=O)[nH]cc1C c1(C(=O)NC(C(N2C(C(CSC)(C)C)CCC2)=O)=O)ccc(-c2ccon2)cc1 C1(CNC(C2C(C)CCC2)=O)CN(c2cnc(C#N)cn2)CCCO1 c1(CCCNC(=O)CCC2CCCOC2)cccc2c1OCO2 C(C(C(=O)N1CC(CN=[N+]=[N-])C1)C(C)(C)C)NC(CC(C)C1CCCC1)=O C1(C(=O)NC2C3CCCC23)CC(F)CN1C(=O)CC1CC(C2CC2)C1 C(C(C)(C)C)C1(C(N(C(C)C(=O)NC2(C3CCCO3)CC2)CCC)=O)CC1 C1(CNC(C(CCSC)NC(=O)CCCn2cncn2)=O)CC2CCC(C1)C2 c1(C(=O)NC2CCCCN(C(C(C)CC(F)F)=O)C2)cc2cnccc2o1 N1(C(C(CC=CC)NC(C2CC(F)C2)=O)=O)CCC2(CC(CO)C2)C1 C1(C(N2CC(CCNC(c3c(C#C)cn(C)n3)=O)C2)=O)CCc2cnc(C)n2C1 c1(C(N(CC=CC(=O)N(C(C)CSCC)CC)CC)=O)cc(SC)ccc1N C12(NC(C(F)=C(C)C)=O)CCCC1CN(C(=O)COC1CCCCC1)C2 CCC(C)CCCCC(=O)NCC1N(C(c2cccc(N)c2)=O)CCCC1(C)C C1(NC(c2ncccc2C2CC2)=O)CCN(C(=O)CC2CCCCC2)C1C1CC1 N1(C(Cc2n(C)cnc2)=O)CC2CCC(CNC(C3CC(=C4CCC4)C3)=O)C2C1 c1(C(N2CC(C)C(N(C(=O)C=CC3CCCC3)C)CC2)=O)cccc2c1CCN2 c1(C(=O)NC2CCCCCN(C(c3cc(C)sc3)=O)C2)nc(C)n2c1CCCC2 N1(C(c2c(C)ccs2)=O)CCC2(CCCN2C(=O)CC(C)CC(C)C)CC1 N(C1C(=O)Nc2cc(Br)ccc21)C(=O)NOC1CCOC1 N1(C(CC2CCC(NC(=O)CCN3CCOCC3)C2)=O)CCC(O)CC12CC2 CCC(CC(=O)NCCN(C(=O)CC1CCCCC1)C)CC(C)C CC(C)C(F)C(=O)N(C(C)(C(=O)NC(C1(O)CCC1)C)C1CC1)C c1(CC(C)NC(Cc2c(C)nc(CS(C)(=O)=O)s2)=O)cccc(F)c1C(=O)O N1(C(Cc2c(OC)cccc2)=O)CC2CN(Cc3ccc(C#N)s3)C2C1 C1(CNC(C2C(NC(C3CCC3)=O)CC=CC2)=O)CCC2COCCC2O1 C(=O)(CCCCC(=O)N1CCC(C(=O)NC2(C)CCOC2=O)C12CC2)OC C1(c2scc(C(=O)NC3CC(NC(c4cc(OC)n[nH]4)=O)C3)n2)CCCN(C)C1 C1(C2CC2)(C(N(CC)Cc2ccncc2)=O)CN(C(c2cc(C(F)F)[nH]n2)=O)C1 c1(C(N2CCC3(CN(C(=O)CC4CSCCS4)C3)C2)=O)cc2n(n1)CCCC2O c1(OC(C)C(=O)N(C)CCN(C(=O)C(C)NC(C)(C)C)C)ccccc1F CCCCCS(=O)(=O)CC(=O)N(C)CC1CCN(C(C2CCCC(C)(C)O2)=O)C1 c1(OC)cc(CC(=O)NC2CCCN(C(=O)CSC3CC3)C2C)ccc1C c1(C(=O)NCCN(C)C(C2CC=CCC2)=O)c[nH]nc1OCC(F)(F)F N1(C(CCc2nc(C)sc2)=O)CCC(C)N(C(=O)CN2CCCC2CO)CC1 CCC(C)CCCC(=O)N1CCC(C(C)(C)CN(C(=O)C(O)C(F)(F)F)CC)CC1 N1(CC(=O)N(CC(=O)OC)CC2CC2)CCC(C(c2nnnn2C)NCC)CC1 c1(NC(C2CC(NC(c3ccc(C(C)N)cc3)=O)C2)=O)nc2cc(F)ccn2n1 C(=O)(CCC(CF)CF)N1CC(NC(c2ccc(C)c(C)c2)=O)C(C(F)F)C1 N1(C(CNC(=O)OC(C)(C)C)=O)CCCCC(COC(=O)CC2(C)OCCO2)C1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCC(C)(C(N2CC(c3noc(C4CC4)n3)C2)=O)C1 CC(C)C(O)C(C)C(=O)N1CCC(O)(CNC(c2ccc(O)nc2Cl)=O)C1 C=C1CCN(C(=O)C(C2CCCC2)OC)C(C(=O)N(CC(O)COC)C)C1 C1(C(N2C(CN(C)C(c3ncsc3C3CC3)=O)CC(F)C2)=O)CC(=O)NC(=O)C1 C1(C(N2CC(C)(NC(c3cc(C(C)C)on3)=O)C2)=O)CCc2nnnn2C1 c1(C(N2C(C)(C(=O)NC)CCC2)=O)ccc(O)c(CO)c1 CCC(C(C)(C)C(=O)NNc1nc(O)c2cnn(C)c2n1)NC(C)=O N1(C(CN2CCC(C)C2)=O)CCC2CCN(C(C3CCC(C)CC3)=O)C2C1 N1(C(C=CC=CCC)=O)CC(CNC(C2(C)CC2(F)F)=O)C(F)(CO)C1 C1(CCNC(C(=O)N(CCC(=O)OC(C)(C)C)C2CC2)=O)CCC2(CC2)CO1 N1(C(c2cnc(O)n(C)c2=O)=O)CCCC2(NC(=O)CC3CCCC3)CCCC12 c1(C(=O)NC)c(NC(c2ccc(OC)nc2)=O)cnn1C1CCCC1 C1(OC)CC(CCNC(=O)C(C)C(C)C)N(C(=O)CCCc2csc(C)n2)C1 CCCCCCCC(=O)NC1CCOCC1NC(c1c(SC)nc(O)nc1C)=O n1(CCC(N2CCCC2CSC2CCCC2OCCC)=O)cnc(C#N)n1 c1(C(=O)NC(C(CO)NC(c2c[nH]c(=NC)s2)=O)C)cccc2c1OCC(=O)N2 CCCC(C(=O)NC1CCC(N(C(=O)C#CC2CC2)C)CC1)N(C)C c1(NC(C)CNC(=O)COCCOCCO)ccc(NC(=O)CSC(F)(F)F)o1 Cc1cc(C(=O)NCCC2(NC(C3CN(C)C3)=O)CCC2)no1 c1(CNC2CN(C(c3cc(F)c(F)cc3O)=O)C2)c[nH]c2cc(F)c(F)cc12 C(=O)(C(C)(CC)CC)N1C(CCCNC(c2c(CC)non2)=O)CCCC1 C(=O)(C1CCc2cccnc21)N(C)CC1(CNC(c2cc3n(n2)CCO3)=O)CC1 c1(NC2CCC(NC(c3ccc4nc[nH]c4c3)=O)C2)ncc2c(Br)cccc2n1 C1(C(=O)NCCCCN(C(CCC(C)c2ccccc2)=O)C)CC2(CC2)CN1C C(=O)(C1=CCOCC1)NCC(CNC(C(C(C)C)c1ccccc1)=O)CO c1(C(N2CCOC(C3CCOCC3)C2)C(=O)NCC2CC2)n[nH]c2ccccc12 C1(O)(CCNC(CCC(=C)C)=O)CCCN(C(c2c(C(C)=O)cnn2C)=O)C1 c1(CC)cscc1C(=O)NCCCNC(=O)C(CC)C1CCOCC1 c1(C(N(C(CNC(CCCN(C(C)C)C)=O)C)C2CC2)=O)ncccc1Br Cc1cccc(C(N2CC3(C2)CN(C(c2cc(C)n(CCO)n2)=O)C3)=O)c1N C1(N(C(C2CCC(C(F)(F)F)CC2)C(=O)NC)C)CCc2cc(Br)ccc2C1 c1(C(N(CCN(C(=O)CC2CCCO2)CC)CC)=O)ccc(NC(N)=O)cc1 CC(C)C(C#N)C(=O)N1CCOCC1CC(=O)NCC1SCCS1 N1(C(C)=O)CC2CC(NC(c3cc(Cl)sc3Cl)=O)C1C2 c1(CNC(C(C)N2CCC2)=O)csc(CNC(c2nnn(C)n2)=O)n1 c1(-c2nc(C(=O)Nc3cc(OC)c(Cl)cc3)sc2)ccc2sc(C)nc2c1 C1(NC(c2c(CC)scc2)=O)CC2CC(NC(c3cn(C)cn3)=O)C2C1 C=CCC(C)(C)C(=O)NCC1CCCN1C(c1cc(C(=O)OC)oc1C)=O c1(C(=O)NCC(CC)NC(=O)CC2COC(=O)C2)ccc2sccc2c1 N1(C(C2CC(=C)C2)=O)CCC(F)(C(=O)Nc2cc(C)on2)C1 Cc1oc(C2CC2)nc1C(N1CC(O)CC1CNC(=O)C(CCO)N(C)C)=O CCC(C)(CC)C(=O)NCc1cc(O)nc(CNC(=O)CCc2cc(C)no2)n1 c1(CC(=O)NCC(F)CNC(c2ccc(F)c(O)c2F)=O)ccc2c[nH]nc2c1 C1(C(N2C(CCN(C(C(COC)OC)=O)C)CCCC2)=O)CCC(O)CN1C C(=O)(C(F)C(F)(F)F)NCC1(COC)CCCN1C(c1ccn2ccsc12)=O c1(N(CC#CC)C)nc2ccccc2nc1NC1CC1OC(C)(C)C c1(CNC2CCC(NC(c3c(C)c(Cl)ncc3)=O)C2)ccncc1[N+](=O)[O-] N1(C(C(C(CC)C)O)=O)CCN(C(=O)C2=CCCCO2)C(C)C1C N1(C(C(C)c2cc[nH]n2)=O)CCC(C(=O)NCC2CC2Cl)C1(C)C c1(C(N2CC(CNC(CC(=C=C)C)=O)OCC2)=O)cnc2c(F)ccc(F)c2c1 c1(C(=O)OCC(N2CCCC2)C)noc2ncccc12 C1(NC(=O)OC(C)(C)C)(CNc2ccnnc2)CC12CCC2.C12CC(C1)CC2=O C(=O)(C1=NOC(C)C1)NCc1cc(C(N2C(CC)CC(C)C2)=O)on1 Cc1n[nH]c(C)c1CCC(=O)NCCCNC(=O)CC1CCN(CC(F)F)CC1 CCC(C)CC(C)C(=O)N1CCC2(C1)CN(C(=O)CC1CC(OC)C1)C2 C(C(=O)N1CCCC(N(CCO)C(C23CC(C)(C2)C3)=O)CC1)(C(C)(C)C)N(C)C CC1(C)c2[nH][nH]c(=NC(=O)c3c[nH]c(=N)s3)c2CN1Cc1ccc(CO)cc1 N(C(=NCCC1CCS(=O)(=O)CC1)NCCF)CC C(=O)(C=CS(F)(F)(F)(F)F)NCC1N(C(CCOCCCOC)=O)CCC1C C(CCCCCC(=O)NCC1CN(C)CCO1)NC(CSCC#C)=O c1(C(=O)NC(CCN(C(C2N(CC)CCOC2)=O)C)C(C)C)cc(O)cc(Cl)c1 C(CCCC(=O)NCC1CC(C(N2CCC2(C)CCO)=O)CO1)N(C)C C1(CNC(=O)Cc2cnns2)COCCN1C(c1cc(-c2ccco2)no1)=O CC1CC2(CCN(C(C3CCCCCC(=O)C3)=O)CC2)CN1C(=O)C(N)=O c1(CC(C(=O)NCCCC(C)NC(C2(CC)CC2)=O)C)cccc(F)c1 N1(C(c2c(C)c[nH]n2)=O)CC2CCC(NC(=O)C(C)NC(c3ccco3)=O)(C2)C1 O=C(CS(=O)(=O)CC1CCCO1)NCCC1(CNC(=O)C(F)(F)CO)CC1 C1(C(=O)NCC(NOCC)=O)(NC(C2CCCN2C2CC2)=O)CCCCC1 c1(C(=O)NCC2N(C(CCc3cc(C)[nH]n3)=O)CCCC2)c(N)sc2c1CCC2 N1(C(C(C)N(C(C23CCC(C2)C3(C)C)=O)C2CC2)=O)CCCC2NC(=O)CC12 Cc1nn(C)c(C)c1C(N1CCCCC(N(C)C(c2csc(C(F)F)c2)=O)C1)=O C1(N(C(=O)C(c2cccs2)SC)CC)CCN(C(C2CC(F)(CO)C2)=O)C1 C1(CN)CCCC(C(=O)NC2CCN(CC(F)(F)F)C2)O1 c1(CC)cnc(Cl)nc1NC(C1CN(C(=O)C(C)NC(C)=O)CCO1)C c1(OC(C)C(=O)NC2CN(C(=O)C(C)(C)CO)CCC2C)cc(F)cc(F)c1 CS(=O)CCC(O)C(=O)NC1CC2(C1)CN(C(c1ccc(Br)s1)=O)C2 C1(C(=O)NC2C(NC(C3CN4CCC3C4)=O)COCC2)CC(C2CC2)=NO1 c1(C(N2CCCC(O)(C(=O)OC)C2)C(=O)NCC)csc2ccccc12 N1(C(C(C)=CC2CC2)=O)CCC2(CC1)CC(C)N(C(=O)C=CS(C)=O)C2 c1(CC(=O)NC(CN(C(C(C(=O)OCC)F)=O)C)C)cccc([N+](=O)[O-])c1 c1(C(=O)NCC(C(=O)NC2CN(C(=O)OC)C2)OC)n[nH]c(C)c1Cl N1(C(C2(C#N)CC23CCCC3)=O)CCCC2(CCCN2C(=O)CCCC(F)F)C1 c1(C(N(C(C)CN(C(=O)CSC2CCCO2)C)C)=O)cccc(C(F)(F)F)c1 CC1=NN(C)C(=O)C1CC(=O)NC1CC2(C1)CN(C(c1csc(CO)n1)=O)C2 O=C1CC2C(=O)NC1=C(F)C=CC=C2NCCCCNC(=O)C[SH](F)F c1(C(N2N3CC2(C)C3)=O)ccc(C(=O)OC)s1.c1(CC(=O)N)ccc(C(C)=O)s1.CC C1(C)(CNC(Cc2c(C)cco2)=O)CCCN1C(=O)CCN(C)CCO N1(C(c2cccc(OC)c2)=O)CCCC2C1CCCN2C(C1CC(Cl)(Cl)C1)=O C(CNC(c1[nH]c(C)cc1C)=O)(CC)(CC)NC(C1(OCC)CCOC1)=O N1(C(c2c(N)nccn2)=O)CCCC(CC(=O)NC2CCOC2)CC1 c1(C(C)C)ccccc1CC(=O)NCC(O)CCNC(=O)C(C)OCC1CC1 N1(C(CCS(C)=O)=O)CC2CCC(C1)C(NC(=O)COc1cccnc1)C2 c1(C(=O)NC(C(C)NC(C(CC)CCOC)=O)CO)cccc2c(C#N)c[nH]c12 c1(C(N(CCN(C(=O)C(c2ccccc2Cl)=O)CC)CC)=O)ccc(NC)cc1 c1(OCCC(=O)NC(CC)CNC(=O)C(F)(F)C(F)F)ccc(Cl)cc1[N+](=O)[O-] N1(C(c2c(CNC(c3cnc(CC)o3)=O)noc2)=O)CC(C)(C)C1COC C(C(=O)NC(C)Cn1cc(C2CC2C(=O)O)nn1)(C(C)C)N(CC)CC C1(C(C)C)CN(C(=O)C(=O)N(C2CC2)Cc2ccc(F)c(Br)c2)CCC1C(F)(F)F N1(C(c2c(CC)occ2)=O)CCN(C(c2ccc(Br)c(N)n2)=O)CC1CC CC(C)(C(=O)NC1CCCC1CNC(c1cc(Br)co1)=O)C1CCCCC1 c1(C(=O)NCC(CC=C)NC(C23CC2COC3(C)C)=O)cc([N+](=O)[O-])cn1C C(=O)(CCCCC(C)C)NCC1CCN(C(CC(C)(C)OC)=O)CC1C Cc1nn(C)c(N2CCOCC2)c1CNC(=O)NC1CC(Cc2ccncc2)C1 N1(C(c2c(C)occ2)=O)CCN(C(=O)CC#N)C(c2ccncc2)C1 c1(NC(CC(CNC(C(CC)OCC)=O)O)=O)ccc2occc2c1 c1(C(=O)NCC(CNC(c2n(CC)cc(Cl)c2)=O)(C)C)cc(F)ccc1N N1(C(C2C(C)(C)C2)=O)C2CCC1CC(COC1CCOCC1)C2.C1(=O)CCCN1 c1(C(N2CCC(NC(CSC(C)(C)C)=O)C(F)C2)=O)cnc2c(c1)COCC2 N1(C(c2c(N)nccc2)=O)CCCC2(NC(c3cc(Cl)no3)=O)CCCC12 Cc1nn(C)c(F)c1C(=O)NCC(C(C)C(C)C)NC(=O)CN1CCCCC1=O c1(C(=O)NCC(=O)N(CCCCN(C(C2(CC#C)CC2)=O)C)C)cccc(F)c1 c1(C2C(C)C2)cc(=NC(=O)C(=O)NCCc2nccs2)[nH][nH]1 C1(NC(c2c(F)cc(F)cc2F)=O)CC2CC1CN(C(=O)C(O)C(F)(F)F)C2 c1(C(N(CC(CN(C(=O)CSC(F)F)C)O)C)=O)cnc2ncc(Cl)cn12 C1(CNC(=O)C=CCF)CN(C(c2cccc(-n3cncn3)c2)=O)CC12CCC2 C(=O)(CC(C(F)(F)F)n1cccn1)NC(CN(C(CCCC(C)C)=O)C)C N1(C(c2c(CCC)nco2)=O)CC2(CCC(C(=O)NC(c3cncnc3)C)O2)C1 N1(C(c2n(C)nc3c2CCC3)=O)CCCCc2ccc(Br)cc21 N1(C(C(C2CC2)OC)=O)C2CCC(C2)C1CC(=O)N1CC1 CN1CCC(C(=O)NCC2(CNC(=O)CCSCC(N)=O)CC2(F)F)C1=O c1(C(C2CC2)NC(C2SCCN(C(CCCC=C)=O)C2)=O)cccc2ccccc12 c1(C(N(CCCCNC(c2c(CC)n(C)nc2)=O)C)=O)ccc(OC)cc1O c1(C(N2CCC(CNC(C(C)C(F)F)=O)C2)=O)cc(F)c(F)c(C#N)c1 c1(C(N(CCNC(C(C)(CO)OC)=O)C)=O)cc2ccncc2[nH]1 C1(C(=O)NCC(C)NC(=O)C2CC2)CCN(CCO)C(=O)C1 C(=O)(C1Cc2ccccc21)N1Cc2c(ccc(CNC(C3CC(F)(F)C3)=O)c2)C1 Cc1n[nH]c2cnc(C(N3CCCN(CCNC(=O)CC(C)F)CC3)=O)cc12 C(=O)(C(CC)CCOC)NC(CN(C(C1(CCCC)CCCC1)=O)CC)C C(=O)(C(C)(C)C(C)C)N1CC(CCNC(c2cc(SC)n(C)n2)=O)C(C)C1 N1(C(C=CC(N)=O)=O)C2CCC1CN(C(=O)CCCC1CCOCC1)CC2 C(CC1CCc2ccccc21)NC(C(=O)OC)C(C)(C)C c1(C(N2CC3C(NC(C(CC)CC4CCCC4)=O)(CC3)C2)=O)ccc(S(C)(=O)=O)[nH]1 CC(C)CC(O)C(=O)N1CC(CNC(c2ccsc2C(F)F)=O)CC1(C)C N1(C(c2cc(C)on2)=O)CC2CC1CCC2NC(=O)C(F)(F)c1nccs1 C(C(F)(F)C(F)(F)F)OCCC(=O)NCC(C1CC1)NC(C1(C)CC1)=O CC(C)=C=CC(=O)N1CCC(CF)(NC(=O)CCC2CCN(C)C2)C1 C1(SCC(=O)NCCN(C)C(C2CCOC2c2ccnn2C)=O)CCS(=O)(=O)C1 O=[N+]([O-])c1n[nH]c2c(N3CCOC(Cc4ccc(F)cc4F)C3)nccc12 C1(COC)(CNC(C2C3CCC23)=O)CCN(C(C2CC2C)=O)CC1 c1(C(=O)NC2C(CNC(C3CN(C)C3)=O)CC2)cn(C)nc1C1CCOC1 N1(C(c2c(CC)nns2)=O)CC2CCCC2(NC(=O)CCc2csc(C)n2)C1 c1(OC)ccc(Br)cc1C(=O)NC1CCC1CNC(=O)CCC(C)(C)C C1(=CC(=O)NCCC2CCCN(C(CS(CC)=O)=O)C2)CC2CCC(C1)N2C C(C(=O)NNC(=O)C(C)(C)CCCCNC(c1ccc(CSC)cc1)=O)=CC CCC(C)(CC)C(=O)N(CCCNC(c1c[nH]c(C(N)=O)c1)=O)CCO N1(C(c2c(NCC)scn2)=O)CCC(CCOC)(NC(C2CC(C)=NO2)=O)C1 C(=O)(C1=C(Cl)CCC1)NCC(CC(=O)NC(CCN(CC)CC)C)C c1(CC(=O)NC2CCC(NC(c3c(C)con3)=O)CC2)ncn2c1CCC2 NS(=O)(=O)c1c[nH]c(C(N2CCOCC2CNC(=O)C(F)CC2CC2)=O)c1 N1(C(c2ccc(CNC(c3ccc(CC)[nH]3)=O)cc2)=O)CCSC(C)CC1 CC1=C(C(=O)NC2CCCCC2NC(=O)C(=Cc2cn(C)cn2)F)CCO1 CC1(C)CCCC1C1CCN(S(=O)(=O)c2ccc(N3CC(CCO)C3)nc2)C1 C1(NC(CSC(C)C)=O)CN(C(c2csc(Cl)c2)=O)CCC1O Cc1cc(F)ncc1-c1cn(CC2(NC(c3ccccc3)=O)CC(F)(F)C2)nn1 C1(C(N2CCC(CCC(=O)NCC3CC[Si](C)(C)C3)CC2)=O)(CC)CCCCC1 C1(OCC(C)C)(CNC(=O)COC2CCC(N)CC2)CC2CCC1C2 CCC(CC(=O)N1CCC2(CC(NC(c3ncc(F)c(OC)n3)=O)C2)C1)C(C)C C=CCC(C(=O)N1CCC(N2CCN(C(C3(O)COC3)=O)CC2)C1)NC(C)=O C1(CNC(C(C=C)O)=O)(NC(c2cnn(C)c2COC)=O)CCCCC1C c1(C(=O)NC2(CN(C(=O)C=CC(=O)N(C)C)C)CC2)cnn(C)n1 O=C(CC1=CCCC1)NCC1CCCN1C(=O)Cn1nccn1 C1(=CCNC(c2cnc(NC(C)=O)o2)=O)CCN(C(=O)CCC2CC2)CC1 N1(C(C2C(COC)C2)=O)CC2CC(NC(c3cccc4cc[nH]c34)=O)CC1C2 c1(-c2scc(C(=O)NCC(CN(C(CSCC=C)=O)C)O)n2)ccc(F)cc1 C1(Cl)(C(=O)NCCN(CCC)C(c2cnoc2-c2ccccc2)=O)CC1(F)F C1(CNC(c2cncc(F)c2)=O)CC2(CCC2)CN1C(c1cc(Cl)nnc1O)=O C1(NC(c2cc(COC)cc(F)c2)=O)C[SH](=O)(C(F)(F)F)CC1COCCO C1(NC(=O)CC2CCCCO2)CC(CNC(=O)CCN2CCCC2)C(O)C1 CN1CC2(CCN2C(C2CCC(O)CN2C(C2CCCC2F)=O)=O)C1 C(C(COC)CC(=O)N(C(C)CN(C(=O)C=Cc1cccc(CO)c1)C)C)OC N1(C(C(C2CC2)NC(C(C)OC(C)=O)=O)=O)CCN2CCC1CC2 Cc1sc(=O)n(CCC(=O)NCC2C3CC3CN2C(=O)CN2CCCC2=O)c1C c1(CCN=C(NC(C)C2CC2)NCC2(N(C)C)CCC2)cccc2c1OCCO2 C1(NS(CC)(=O)=O)CCCC(C(N2CCC(N(C(=O)C(F)F)CC3CC3)C2)=O)C1 c1(CC)cccc(C(N2CCC(C)C2C(=O)NC(C2(OC)CCC2)C)=O)c1 c1(C(N(CCOC)CCNC(=O)CN(C(=O)C(C)C)C)=O)cc(F)c[nH]1 C(CC(O)C(=O)NCCC(O)C(F)F)NC(c1cnccn1)=O C(=O)(C(C#N)C(C)C)NCCN(CC(C)O)C(c1oc(C)c(Br)c1)=O CCC(O)C(C)C(=O)N1CCC(NC(=O)COCCOCCO)CC1 c1(C(N2C(CCNC(=O)C(F)C3CCOC3)CCC2)=O)ccc(O)c([N+](=O)[O-])c1 c1(OC)ncc(Cl)c(=NC2CCN(C(=O)CC3C=CS(=O)(=O)C3)C2)[nH]1 Cn1ccc(=O)cc1C(N1CC2CCC2(CNC(c2cc(Br)cnc2Cl)=O)C1)=O C(=O)(CCC1=CCCCC1)N1CCC(CC(N2CCC(C#C)C2)=O)C1(C)C c1(CC(=O)N(CCCNC(=O)CSc2cn[nH]c2)C)cnc2cccnn12 CC(C)CC(CNC(C1CC(CCNC(C2CCC2C#N)=O)C1)=O)N(C)C c1(NC(C2C(O)CCN2Cc2ncccc2C(F)(F)F)=O)ccc(F)c(Cl)c1F N1(C(CCOCC#C)=O)CCCC(CC(N2CC(O)CC2CC)=O)CC1 CS(=O)(=O)CCCCCN=c1[nH]c(NC2CC3CC4C(C3)C24)nc2c1CCCC2 c1(C(N2C(c3ccc(C)o3)COCC2)=O)ccc(C)c(C#N)c1 N1(C(c2c(C)onc2)=O)CCOCC(CNC(=O)Cc2ccccc2)C1 Cc1cc(C(=O)NC2CCCN(C(C3CC4CC4C3)=O)CC2)nc2[nH]nc(O)c12 C1(C(=O)NC(CCC)CC)CN(C(=O)Cn2ccccc2=O)CC1(C)C N1(C(COC2(C)CCCC2)=O)CCC(O)(CNC(C23CC(C#N)(C2)C3)=O)CC1 N1(C(c2n(CC)c(O)nc2)=O)CCC2CN(C(=O)CC3CCC(C)CC3)CCC12 N1(C(CCc2c(C)noc2)=O)CCC2(CNC(C3CC(C4CC4)C3)=O)CCCC12 C(=O)(CC(C(F)F)n1ccnc1)N1CCC(C(C)Nc2ncncc2Cl)C1 C1(NC(C2(C)CSC2)=O)CCCCN(C(=O)CCCNS(C)(=O)=O)C1 c1(C(=O)NC2CCN(C(C(C(C)(C)O)F)=O)C2(C)C)cccc2c1CCN2 CCC(C(=O)NCCOCCNC(=O)CCCN1CCCC1)C(C)(F)F c1(C(=O)Nc2ccc(SCC(=O)C3CC3)cc2)c[nH]c2ccccc12 c1(NCCNC(CC2CCCC(C)C2)=O)c(Br)cccc1[N+](=O)[O-] c1(OC)cc(C(=O)N(C)CC2CCCN2C(C2CCSCC2)=O)cnc1O Cc1nc2c(O)cc(C(=O)NCCN(C(C3CC3F)=O)C(C)C)cc2n1C N1(CCNC(=O)Cc2cccnc2)CCC(NC(=O)CC2CC(F)C2)CC1 c1(OC)cccc(OCCC(N2CCCC2CCNc2ccccc2)=O)c1 CCCCCCCCC(=O)N1C(C(=O)Nc2cc(Cl)ncc2Cl)CCC1C C#CCCCCCC(=O)NC1CN(C(c2cc(N)c(F)cc2F)=O)CC1OC C1(CC(N2CC(CCC)C2)=O)CN(C(=O)Cc2scnc2C)CC12CC2 C1(CC)COCCN1Cc1cccc(N(C)CC2CCCCN2CC)c1 c1(C(N2C3CN(c4cc(C#N)ncn4)CC32)=O)cn2cccc(C(F)(F)F)c2n1 C=CCC(C(=O)N1CCCC1CCNC(=O)C(C)(C)n1ccnn1)NC(C)=O C(=O)(C(F)(F)CC(C)C)NCC(CNC(c1cc(OC)n(C)n1)=O)CO CCCCC(CC)C(=O)NC1CCSC12CN(C(c1ncccc1SCC)=O)C2 CC12CCN(C(C3CC3C3CCCO3)=O)C1CN(C(=O)Cc1c[nH]c(=N)[nH]1)C2 N1(CC(=O)N(CC=C)CC)CC(NC(=O)Cc2ccc(C(N)=O)cc2)CCC1C Cc1cc(C(N2CCCC(CN3CCCC3)C2)=O)ccc1-n1cncn1 Cc1ccc(CN2CC(O)CC2C(=O)NC(c2ccsc2)C2CC2)cc1O c1(C(N2CC3C(N(C(CC(COC)(C)C)=O)C)C3C2)=O)ccc2ncnn2c1 Cc1ccc(C(=O)NCC(C)NC(=O)COCc2nccs2)n1C N1(C(=O)NCCCC)CCC(C(=O)NC2CN(C(=O)C(C)(C)n3ccnn3)C2)CC1 C1(C)(C)C(=O)NNC(=O)c2ccccc2N1.c1(OC)ccc(N(C)C)cc1 C1(C(=O)NC(C)(C)CCNC(=O)C(C)(C)F)CC2CCCN2C(=O)N1 Cc1nc(C(=O)N)ccc1C#N.N1(CC)CCCOCC1.c1(C2C(=O)NCC2)ccnn1C c1(CNC(=O)COC2CC(NC(c3ccc(C4CC4)s3)=O)C2)ncccc1F CON1CCC(C(=O)N(CCC(N2CC3(C2)CN(C)C3)=O)CCCO)CC1 C(C(CNC(=O)C=CC1CCC1)CO)NC(C1C(C)(C)C1)=O S(=O)(=O)(c1ccc(-c2cncnc2)c(C)c1)NCCN(C(C)C)CC N1(C(C=CCCC)=O)CC2(CC(NC(=O)C(O)CCCc3ccccc3)CO2)C1 CC(C(=O)N1CC(O)(C(C)NC(=O)CCc2cccc(OC(F)F)c2)C1)C(F)F c1(C(=O)NCC2(F)CN(C(=O)CCn3cccn3)C2)ccc2[nH]ccc2c1F c1(CC(N2CCC(NC(=O)Cn3cncn3)C23CC3)=O)csc2cccc(F)c12 c1(C(N2CCN(C(c3cc4sccc4s3)=O)C(CO)C2)=O)ccc2cnsc2c1 c1(C(=O)NCC(=O)NCCCN(C(=O)CC2(O)CCOC2)CC)ccncc1 N1(C(COCCOC)=O)CCC2CCN(C(c3nn(C)cc3S(N)(=O)=O)=O)CC12 c1(C(=O)NC(C)(CNC(=O)C(F)n2cccn2)CO)occ2c1CCOC2 CC1(NC(=O)Cn2c(O)nnc2O)CCCCC1C(=O)NCc1nc(CO)n[nH]1 c1(CC)occ(C)c1C(N1CCC(COC)(NC(=O)CC2COCCO2)C1)=O CCCCCC(O)CC(=O)NCCCN(C)C(c1c(Cl)c(CC)nn1C)=O N1(C(C(CCCC)O)=O)CC(NC(=O)C=Cc2ccc(SC)s2)CCC(O)C1 C1(C)(CNC(C2C(CC)OCC2)=O)CCCC1NC(c1cnn(C2CCC2)c1)=O C1(C(=O)NCCN(C(c2c(Cl)cn(C)n2)=O)C2CC2)CC12CCSCC2 N1(C(CCc2ccc(C#C)cc2)=O)CC2CCN(C(c3nc(C)nn3C)=O)CC12 CC(CC(F)(F)F)C(=O)NC1CC2CCC1CN2C(C1CC(F)(CF)C1)=O C1(NC(C(CCOCC)NC(C2CCCO2)=O)=O)CCC2(CCC2)C1 c1(C(=O)NC(CN(C)C(C2CC3C=CC2C3)=O)(C)C)ccc2[nH]c(=O)cnc2c1 C1(C(N2C3(C)CC(CNC(=O)Cc4ccsc4)(C2)C3)=O)CC2(C1)NC(=O)NC2=O N1(C(C(C)SC)=O)CCC(C(C)C(=O)NC(C)Cc2cc(C)[nH]n2)CC1 N1(C(Cc2noc(C)c2C#N)=O)CCN(C(c2cnco2)=O)CC2CCCCC12 c1(C(c2ccc(C)cc2)Nc2n(C(=O)OCC)ncc2)ccc2c(c1)OCCO2 Cc1ccc(C(CO)NCc2ccc(Oc3ccc(Cl)cc3)nc2)c(C)c1 c1(C(N2C3CC(NC(CCCCC=C)=O)CC2CC3)=O)ccc2c(c1)CNC(=O)N2 C1(C)(CNC(COC)=O)CCCN(C(C)=O)C1 N1(C(c2c(CC)con2)=O)CC2CC(C1)N2C(=O)CCc1nc(C)cs1 N1(C(C(C(C)C)SCC)=O)CCCC(CNC(=O)C(O)CC(N)=O)(COC(C)=O)C1 CC1CN(C)C(C)CC1NC(=O)CCN(CCO)C(C1CCCO1)=O C12(COC)CC(CNC(=O)CC3CCCNC3=O)(CN1C(=O)C#CC(C)(C)C)C2 C1(C(N2CC(O)(CCc3cn(-c4ccc(Cl)nc4)nn3)C2)=O)CCCCCCC1 N#Cc1ccc(NC(C2CC23CCN(Cc2cccc(F)c2I)CC3)=O)c(F)c1 Cc1ccc(CC(C)C(=O)N(C(C)CN(C(=O)CSCc2cscn2)C)C)cc1 c1(C(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)cc2c(F)cccc2s1 C(C(N=[N+]=[N-])C(=O)N1CCN(C(=O)Cc2ccc(Cl)cc2C)C(CO)C1)OCC C1(CNC(CCOC)=O)CCCC2CN(C(C34CCC(CC3)C4)=O)CC12 C1(NC(C2C(C(C)C)C2)=O)(CNC(=O)CSc2ccccc2F)CCOCC1 C12CCCCC1NC2=O.C1(COCC)(NC(C2CN(C)C2)=O)CCCCC1 C1(C(=O)NC2CC(C)(NC(c3cnc(Cl)s3)=O)C2)CN2CCCN1CC2 c1(C(=O)NC(CNC(C(CC)SC)=O)C2CCC2)cc2c(c([N+](=O)[O-])c1)OCO2 c1(C(N2CCN(CCNC(C(C)(C)OC)=O)CC2)=O)sc2nccn2c1C N1(C(C#C)C)CCN(C(=O)CC=CCNC(c2ccn(CC(C)C)n2)=O)CC1 N1(C(C2N(C(c3cc(C)sc3C)=O)CCCC2)=O)CCc2c(C)cccc21 C1(C(=O)N(C(C)C(=O)NCCOCCc2ccsc2)C2CC2)(OC)CCOC1 Cc1cn2c(n1)C(C(=O)N1CCCC(c3nc(C)c(C)[nH]3)C1)CCC2 C(=O)(CS(=O)c1cccc(OC)c1)NCCN(C(c1c(CC)c(C)sc1)=O)CC c1(C(=O)Nc2cccc(CNC(=O)C=C3CC3)c2)cnc2cc(Br)ccc2c1 N1(C(c2c(OC)c(F)c(Br)cc2)C(=O)NC2CC2)CCc2ccc(C#N)cc2C1 Cc1ccoc1C(=O)NCC(C)(C1CCC1)NC(c1cnn(CCF)c1)=O C(CCC(C)(C)C(=O)NC(CO)C(C)O)NC(c1n(CC)nc(C)c1)=O N1(C(C2C=CCN(C(c3cc(C4CC4)[nH]n3)=O)C2)=O)CC(F)(F)CC1CO C(=O)(C1OCCc2ccccc21)NCCC(=C)CNC(=O)CCC(=O)NCC CC1CC(C(=O)NCCCOCCNC(=O)C2=C(Cl)CC2)C1(C)C C(C)(C(=O)N1CC(C)(NC(=O)CC2CCCOC2)C1)(C(C)C)OC S(=O)(=O)(c1ccc(C#N)cc1C)Nc1c(C(=O)NCC)nccc1 c1(C(=O)NCC(C2CCC2)NC(=O)CC2CCSC2)cscc1Cl N1(C(Cc2c(C)ccs2)=O)CCC2(CCN(C(c3cc(CF)on3)=O)C2)C1 CCC(C)(CNC(=O)C(C)CN(C)C)C(=O)N(CCCC(C)(F)F)C Cc1nnn(C)c1C(=O)NCCC1CCC(NC(=O)C=C2CCOCC2)C1 CCC(C)CC(=O)C(=O)N1CC2CC(NC(=O)C(CC3CC3)OC)C1C2 c1(N(CCOC)C)ccc(Br)c(S(=O)(=O)N2CC3OCCOC3C2)n1 CC1=C(C(=O)NCC2CC(NC(c3cc(C(N)=O)ccn3)=O)C2(C)C)CCC1 C1(CC(=O)N(C)CCOCCCNC(C2CC(F)(F)C2)=O)OCCC1(C)C C1(NC(Cc2n(C)ncc2)=O)CCCCN(C(=O)CCC2CC2(F)F)C1 N1(C(c2c(CC)ncs2)=O)CCCN(Cc2cc(F)c(F)cc2I)CC1C C(CN=c1[nH]c(=NCCC2CSCCO2)[nH]c2c1CSC2)(C1CCC1)OC c1(NC(CCN(C(Cc2nc(C)oc2)=O)C)=O)cccc(F)c1O C=CC1CN(C(c2cc(O)nn2C)=O)CC1NC(c1sc(CCC)nc1C)=O N1(C(C(C)=CC)=O)CCC(C(C)CNC(=O)C(CCC)OCC)CC1 C(CC(O)C(F)(F)F)NC(C(CN(C)C)NC(C1SCCS1)=O)=O c1(CN(C(C(=O)N(CCC)CC)C)CCO)cccc(-c2cnccn2)c1 C=CC(C)(C)CC(c1nnnn1C)NCCC12CCC(CC1)OC2 c1(C(C)C)n[nH]cc1C(=O)NC1CC1CNC(=O)CSc1nc[nH]n1 C1(NC(CSCC)=O)CN(CC)CCC1(C)C.C1(=O)C=CCOCCN1 c1(OC)c(C)cc(C(N2CCC(NC(c3csc(CO)n3)=O)C(O)C2)=O)cc1C c1(CCNC(C(c2cnn(C)c2)NC(CCc2onc(C)n2)=O)=O)noc(=O)n1C C1(C(=O)O)CN(C(=O)Cc2csc(Br)n2)CC(C(F)(F)F)O1 C1(C(=O)NCC(CC)(CC)NC(C(CCC)=CCC)=O)CCC2(CCC2)O1 C1(NC(C2N(C(C3N(C)CC(F)C3)=O)C3C(C2)C3)=O)CC2(CCOC2)C1 C1(C(N2CCC(=C)CC2)=O)CC(F)(F)CN1Cc1ncn(C)n1 C1(C(=O)NCCC2(CNC(=O)CNc3nccs3)CC2)CCn2cncc2C1 C12(NC(c3cc(C)c(C)[nH]3)=O)CCN(C(c3cc(CN(C)C)c[nH]3)=O)CC1C2 n1(CC(=O)NC(CCCC)CNC(=O)CN(C)C)ccc(O)nc1=O C12(C(N)=O)CCCC1(C(N1CC(O)(CNC(c3cc(Cl)ns3)=O)C1)=O)C2 O=C(C(F)C(F)(F)F)NCC1CCCC1NC(=O)C=CC(=O)Nc1ccccc1 Cc1oc(C(C)C)cc1C(N1CCC(NC(=O)CC2CC(F)(F)C2)C1C)=O Cc1cc(C(=O)NCCN(C(=O)CP(C)(C)=O)C2CCCC2)n(C(F)F)n1 N1(CC(c2n[nH]c(CO)n2)(C)C)CC2(CCCN(CC3(C)COCCO3)C2)C1 C1(CNC(C(Cc2ccc(C)cc2)(C)O)=O)CCC2(CCOCC2)C1O c1(NC(C(CC#CC)NC(c2cc(C)c[nH]2)=O)=O)cccc2ccoc12 Cc1no[nH]c1=NC(=O)CC1CCCN1Cc1c(C)[nH]c2ccccc12 N1(C(C(CN(C)C)O)=O)CCCC(CNC(=O)CC2(C#N)CCC2)C1 C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)CN(S(C)(=O)=O)C)CC2(CC2)C1 c1(OC)ccccc1C(C)Nc1ccc(C(=O)OC)cc1.C1(=O)CN1C c1(C(=O)Nc2c(C(C)NC(C3CC(OCC)C3)=O)noc2)ccc(C)cc1 N1(C(C)C(N2CCCC(O)CC2)=O)CCC(O)C(NC(C2CCC(O)CC2)=O)C1 c1(C(=O)NCC2CC(CNC(C(C)SCCCC)=O)C2)cocc1C c1(NC(C2C(CNC(CC(C)C3CC3)=O)C2)=O)cnn2c1CCCC2 c1(C(=O)Nc2c(OC)nsc2)cccc2c1NC(=O)CC2 CN1CCC2CC1CN2C(=O)C(c1ccccc1F)c1ccccc1 N1(C(CN(C(CN(C(C)C)C)=O)C(C)C)=O)CCC(CO)C(C)(C)C1 C(C)(C)(CC(=O)N(C1CN(C)C1)C)NC(c1c(OC)n[nH]c1)=O N1(C(c2ncccc2C2CC2)=O)CC2CCC(C1)N2C(c1ccc(O)cn1)=O N1(C(CSCCCC)=O)CCOC2CCN(C(C3C4CCCCC34)=O)CC12 c1(CC)nc(C(=O)NCC2CCC2NC(=O)C=C(Cl)Cl)cs1 C(CC(C)C)(C(=O)NCCc1cn[nH]c1)NC(C1CCC(C)(CC)O1)=O c1(N2CCC(C)(CNC(C(CC)OCC)=O)C2)ncc2cccnc2n1 N1(C(c2n(C)cnc2)=O)CC2(CCN(C(=O)CSCCC#N)CC2)C1 Cc1nc(C(=O)NCCN(C(c2ccnc(C(F)F)c2)=O)C2CC2)c(C)o1 N1(C(C=CC=CC)=O)C(C(=O)NCc2cncc(F)c2)CCC1C c1(NC)nc(C)ccc1C(=O)NCC12CC(CO1)N(C(=O)CSC(F)(F)F)C2 C(=O)(C(C)C(O)CC(C)C)NC1CN(C(CC2(OC)CCC2)=O)CC(C)(C)C1 c1(CC)ccc(C(=O)NCC(C(=O)NCCOc2ccncc2)N(C)C)[nH]1 C(=O)(C(O)COC)NCCN(C(C1CC(=C)C1)=O)C(C)C.c1(C=O)ccccc1 C1(NC(c2c(C)nn(C)c2)=O)CC2CC1CN2C(c1ncoc1C(C)(C)C)=O c1(C(=O)NC(CC=C)CNC(c2ccc(SC)s2)=O)cc2sc(Cl)cc2[nH]1 CCC(O)(CC)CN(C)N1CCOC(CCSc2ccccc2)C1 Cc1ccc(C=CC(=O)NC(CNC(=O)C(C(C)C)NC(C)C)CC(C)C)cc1 C12(NC(C3C(C)CCC3)=O)CC1CN(C(c1ccc(C3CCC3)nc1)=O)C2 Cc1n[nH]cc1N(C(CC1CCCO1)C(=O)NCCCOCC1CC1)C N1(C(C2(NC(c3ccn(CC)c3C)=O)CCOCC2)=O)CCC2CC1C(=O)O2 c1(CNC(C(c2cnn(C)c2)NC(C2CC(SC)C2)=O)=O)cncc(Cl)c1 C(=O)(C(C)(F)C(=O)NCC1CCCC1NC(c1ccc(C)cc1)=O)OCC c1(N(C(C(=O)NCCCSC)c2ccco2)C)cc(-c2ccccc2)no1 C1(NC(=O)C(F)C2CCC2)COC2CN(C(c3cn(C4CC4)nn3)=O)CC12 N1(CCCCNC(c2sccc2Cl)=O)CCCN(C(C2CC2F)=O)CC1 Cc1ccc(CNC(C2CCC2CNC(C2CC(=O)NC2(C)C)=O)=O)c(F)c1 N1(C(C(CC)OC)=O)CCC(CNC(=O)COc2c(C)ncnc2C)(OC)CC1 N1(C(=O)C(c2c[nH]c3ccccc23)c2ccccc2)CCCCC2C1C2(F)F C(=O)(C1CCc2nnc(C)n21)NC(CC)(CNC(c1cccc(C)c1Cl)=O)CC C=CCCCCN(C(=O)CN(C(=O)Cn1nccc1C)C)C C(=O)(C(CC(C)C)N(C(=O)C=Cc1ccc[nH]1)C)NCC(CC)(C)CO C1(NC(c2c(C)ncs2)=O)CC2CC(C1)N(C(c1ccccn1)=O)C2 N1(C(C(=O)NCCC)CCC2(C#N)CC2)CCOC(C)(C(F)F)C1 C1(NC(c2c(OC)scc2)=O)CCCN(C(c2ccc(C)cc2F)=O)CC1 N1(C(=O)NCC#C)CC2CCC(C1)N2C C1(CC(=O)NCCCC(C)NC(C(CC)C)=O)CC2(C1)CC1(CCC1)C2 C1(C(N2CCN(C(c3cn[nH]c3)=O)C(CC(F)(F)F)C2)=O)Cc2ncccc2N1 N12CCC3CCCC13C2=O.C(CC(O)C(F)F)NC1(c2ccccn2)CC1 Cc1cnc(N2CCC(C(=O)NCCC3CCCC3)C(O)C2)nc1C CC1CCCC1(c1nnnn1C(C)(C)C)NCC12CCN(CC1)CC2 N1(C(c2cc(C)n(C(C)C)n2)=O)CC(C)(C)CC1CNC(C1CCCC1O)=O c1(OC)cccc(C=CC(=O)NCC2(NC(=O)C(C)n3cccc3)CC2)c1 N1(C(C(C2CCCO2)OC)=O)C2CCC(C(=O)NCc3cc(C)c(C)s3)C1CC2 c1(NC(C23CC(N(C)C(c4ccccc4C#N)=O)(C2)C3)=O)ccc(I)cc1[N+](=O)[O-] c1(C(=O)NCC2N(C(C3CCC(C)O3)=O)CC2)ccc(Cl)cc1[N+](=O)[O-] N1(C(C(OC)OC)=O)CC(C)C(C)(CNC(C2CC(=O)NC(=O)N2)=O)C1 c1(C(N2CCC(CN(CC3CC3)CC3CC3)CC2)=O)cc2ccc(Cl)cc2o1 C1(CNC(C=C(C)C(F)F)=O)CCN(C(=O)CCc2cocn2)CC1C n1(C2(C(=O)NCC3(CNC(C4CCCO4)=O)CCC3)CC2)cc(Br)nn1 CC1CN(C(C2CCC3(CC3)C2)=O)CCN1C(=O)C(c1ccc(Cl)s1)C C1(C(=O)NC2C(N(C)C)COC2)CC2CCC1N2C(c1ccccc1C1CC1)=O C1(C(=O)NC23CC(NC(CC(n4ccc(C)n4)C)=O)(C2)C3)CCC(O)CC1 C1(NC(C2(C)CCCC2)=O)C2CCC1CN(Cc1cccc(-n3ccnc3)c1)C2 C(=O)(CCCCC(=O)N1CCC(N(C(=O)C(C)CC(C)C)CCO)CC1)OC C(=O)(C(C)C(F)(F)C(F)F)N1CCN(C(c2[nH]cc(C)c2C)=O)C(CC2CC2)C1 c1(COC(N2CC(CCC=C)(COC)C2)=O)c(C#N)cnn1-c1ccc(F)cc1 O=S(=O)(c1ccc(F)c(F)c1)N1CCc2cccc(-c3ccc(F)nc3F)c2C1 N1(C(C2(F)C(C)C2)=O)CCC(C)(C)C(NC(c2ccc(-c3ccco3)s2)=O)C1 n1(CCOC)ncc(C(N2CCN(C(c3sc(F)cc3Cl)=O)CC2)=O)c1C c1(C(=O)NCC(=O)N(C(C)CNC(=O)CC2CC2CC)CC)cccc(C#N)c1 C1(C(C)(O)CNC(c2cc(Cl)no2)=O)CCCN(C(c2ccc(O)cn2)=O)C1 N1(C(c2c(Cl)ncc(C)c2)=O)CCC2CN(C(=O)C=CCBr)CC12 N1(CC2CC(OC)(OC)C2)C(=O)CN(CC(C)CN(C)C)C1=O C1(COC)(CNC(c2cc(OC)ncn2)=O)CCCN1C(C1CCCC(C)C1)=O c1(C(=O)NCC(CNC(CC(CCCC)O)=O)C)ccc2c(c1)N(C)C(=O)CC2 C1(NC(C(CC)OCC)=O)CN(C(=O)CNC(=O)CC)CC2(CC2)C1 N1(C(c2c(CC)noc2)=O)CCCN(C(C2CCS(=O)(=O)N2C)=O)C(C)C1 c1(C(C)NC(=O)C(=O)NC2CC23CCNC3)ccc(F)c2ccccc12 C1(CNC(C(CNC(CCOCC)=O)CC2CCCC2)=O)CC2CCCC2C1 C(CS(=O)(=O)Cc1cn(CCN2CCOCC2)nn1)NC(C1CCC=CO1)=O N1(C(c2nocc2C)C(=O)NC(CC)C)C2CCC1CC(C(=O)NC)C2 Cc1cc(C(N2CCN(C(=O)CC3OCCC3(C)C)C(CCO)C2)=O)ccc1Cl N1(C(C2(C)C(C)(C)C2)=O)CCC2(CCCCN(C(c3n[nH]cc3Cl)=O)C2)C1 CC1(C(=O)NCCC2(O)CCN(C(C3(CO)CCC3)=O)C2)CC=CCO1 C(=O)(C1=COCC1)NC(CCNC(c1c(C)occ1)=O)Cc1ccccc1 N1(C(CC2CCC(C)C2)=O)CC2(CNC(c3cc[nH]n3)=O)CC1CCO2 c1(C(C)C(N2CCOC(CNC(=O)CC3CCC3)C2)=O)ccc(F)c(F)c1 CCCCCCCC(=O)NC1CN(Cc2cccc(I)c2F)C1 O=C1NC2(CCO1)CN(C(=O)Nc1cccc(C(=O)C3CC3)c1)C2 N1(c2ncc(C(=O)OCC)s2)CC2CCCC(NC(=O)Cc3csc(S)n3)C2C1 C1(C(N(CC(CO)(CO)NC(c2cc(C(N)=O)n[nH]2)=O)C)=O)CCCNS1(=O)=O c1(C(=O)OC)ccc(C(N2CCC(NC(c3cc(Cl)c(C)cn3)=O)C2)=O)c(F)c1 C1(C(=O)OC)CN(C(c2cnn(C)c2Cc2ccccc2)=O)CC12CCC2 N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C1C(=O)NCC(C)(C)OC(C)C C(C1CSc2ccccc21)NC(=O)Nc1cc(NC(C)CN2CCOCC2)ncn1 C(CCNC(C1CN(C2CCOCC2)C1)=O)(C(C)C)NC(C1C(=C)CC1)=O c1(C(=O)OCC)cccc(CC(N2CC(O)(CNC(C3CC(C)=NO3)=O)C2)=O)c1 CC(C)(C)CCC(=O)NC1CC(NC(C2(CCO)CC2)=O)C(O)C1 N1(C(C(C)=O)=O)CCC(F)(CNC(c2cnc(O)c(Br)c2)=O)CC1 CC1COCCC1NC(=O)C(c1ccccc1)NC(=O)Cc1ccoc1 C1(C(=O)NCC2(C(=O)NCCC(C(C)C)O)CC2)CC2CCC(C1)O2 C1(CNC(c2nc(C)oc2)=O)CN(C(=O)CCN2CCC(F)C2)CC(C)(C)O1 CCCCC(O)C(C)C(=O)NCC1(O)CN(C(c2ccccc2OCCC)=O)C1 c1(CCCC)nc(C)c(C(=O)NCC(C)(C)CN(C)C(c2cnc(O)n2C)=O)s1 C1(CC=C)(NC(=O)CC(C)(C)O)CCN(C(=O)CC(c2ccc(CC)cc2)C)C1 N1(C(Cc2c(C)cccn2)=O)CC2CC1CCC2NC(c1c(C)nn(C)c1Cl)=O Cc1noc2nc(C(=O)NCC3CN(C(=O)C(C)(O)C4CCC4)C3)ccc12 N1(C(C2C3(CN(C(C(C)Cn4cccn4)=O)C3)C2)=O)CCc2ccc(F)cc2C1 c1(C(=O)NC2CCN(Cc3cc(C)ncc3)CC2F)cnn2ccncc12 N1(C(Cc2c(C)nc(C3CC3)s2)=O)CCN(C(C2OCCN(C)C2=O)=O)C(C)C1 Cc1ccc2occ(C(=O)NC3CC3NC(c3cc(CF)on3)=O)c2c1 c1(C(=O)NC2N(C(CNC(=O)OC)=O)C3C(C2)C3)ccc2c(c1)NC(=O)CC2 O(N=C1CCCCCC1)CC(N1C(C)CC(NC(C2(C)CCNC2=O)=O)C1)=O c1(-c2cc(SC)c(F)cc2)cc(C(=O)NCCN(C)C)c2cc[nH]c2c1 CN1CCC(NC(C2(n3cc(C(N4CCOCC4)=O)nn3)CC2)=O)C1=O C1(O)(CN(C(=O)CC2CC(CF)C2)C)CCN(C(C2CC(F)(F)C2)=O)C1 N1(C(C2C(CC)N(C)CC2)=O)CC(CNC(C2CC(O)C2)=O)OC2(CCC2)C1 C1(C)(OC)CCN(C(=O)CCC(C)NC(=O)CC2OCCCO2)C1 N1(C(C(C(C)C)C#N)=O)CC(CNC(c2cnc(C3CC3)[nH]2)=O)CC(C)(C)C1 c1(OC)ccc(O)c(C(=O)NCCC2CCCN2C(=O)CN(C2CCSC2)C)c1 c1(C(=O)NCCCN(C(C(C(C)C)O)=O)C)cn2c(n1)CCC2 C=CCC(C(=O)N1CCN(CCCCNC(c2cscn2)=O)CC1)OC c1(C(=O)NC2CC3(C(NC(CCC=C)=O)C3)C2)cnc2c(=O)[nH]cc(CC)c2c1 N#Cc1ccc(NC(N2CCOCC2c2nc(C(F)(F)F)n[nH]2)=O)cc1Cl N1(C(CC=C=C)=O)CCCC(CN(C(=O)CCOCC(C)C)CC)C1 O=S(=O)(c1ccnn1C1CCCCC1)Nc1ccc(Cl)cc1N1CCSCC1 N1(C(C2(C(C)C)CCC2)=O)CC(C)OC2(CCN(C(C3CS(=O)(=O)C3)=O)C2)C1 C(c1ccc2nc(Nc3ccc4[nH]ccc4c3)[nH]c2c1)=CCCC c1(OC)ccc(CNC(C2(F)CN(Cc3ccc(Br)cc3O)C2)=O)cc1Cl c1(C(=O)NCC#CCNC(c2ccc(OC)s2)=O)cccc2cccnc12 Cc1cc2c(C(N3CCC3CNC(C3(O)CN4CCC3CC4)=O)=O)cccc2[nH]1 c1(-c2ccn(CC(C)C)n2)nc(C(C2CC2)N(C)C)nn1C1CCSCC1 C(C)(N=c1[nH]c(Cl)ncc1Br)C1N(C(C(CCC)CCC)=O)CCCC1 c1(C(N2CCC(C)(CNC(CC3C(C)OC(C)C3)=O)C2)=O)nn(C)cc1[N+](=O)[O-] C1(C(N(C(C(=O)NC(C)C2CC2)(C)C2CC2)C)=O)C2CC(=O)CC12 c1(C(N2CC(CCNC(C3(CO)CCCO3)=O)(OC)C2)=O)ncc[nH]c1=O c1(C(=O)OCC(CC)(CC)OC)cc(-c2ccc(C)cc2)nc2onc(C)c12 CC1=C(C(=O)NCC2CCCCC2C(=O)NCC2OC(=O)CC2(C)C)COCC1 N1(C(c2n(C)ncn2)=O)CC2(CC(NC(=O)Cc3noc4ccccc34)CO2)C1 C1(CCC)CN(C(=O)C(O)C2CC2)CCN1C(C1CN(C2CCC2)C1)=O Cc1cc(C(=O)NC2CN(C(C3CCN(C)C(=O)C3)=O)CC2C)c(N)c(C)c1 c1(C(=O)NCC2C(NC(c3c(COC)nn[nH]3)=O)C2)c(C)sc2ccccc12 CC(C)(C)C(=O)NCC(=O)NCC1(CCNC(=O)CNS(N)(=O)=O)CC1 C(=O)(C1OC(=O)c2ccccc21)NCC(CC=C)NC(=O)C1=CCC(C)(C)CC1 c1(C(N(C2CCC(NC(c3cc(CC)on3)=O)CC2)C)=O)cc2ncccc2s1 N1(C(C(C)Sc2ccccc2)=O)CC2CC2(CNC(=O)Cn2cccn2)C1 C(=O)(C1CCCc2nn[nH]c21)NC(CNC(c1cncc(OC)n1)=O)CO CS(=O)(=O)C1CC(C(=O)NCC2(O)CCN(C(C3CC(C#N)C3)=O)CC2)C1 C12(NC(c3cc[nH]n3)=O)CCC(CC1)N(C(=O)C(CC(F)F)C1CCC1)C2 c1(C2N(Cc3cn(C4C(=O)NCCC4)nn3)CCC2)ccc(Cl)c(Cl)c1 C1(C(N2CCC(C)C2C(=O)NCC(F)(F)Cl)=O)CC2CCCC2C1 C(=O)(CC(C)CC(F)(F)F)NCCC1OCCN(C(c2c(OC)n[nH]c2)=O)C1 C1(C(N2CC(C3(NC(=O)C(C)CC4CCCO4)CC3)C2)=O)(OC)CCCCCC1 N1(C(C2(C(F)F)CC2)=O)C2CCC1CC(NC(C13CC(F)C1C3)=O)C2 c1(OCC(C)C)ccc(C(N2CCC(N(C(=O)COCC3CC3)C)CC2)=O)cc1 N1(C(C2CCN(C(=O)NC)C2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)CC12CCC2 c1(C(N)=O)ccc(F)c(C(=O)NC2CCN(C(=O)CSc3ccncc3)CC2)c1 C(C(C(=O)NC(c1nc[nH]n1)C1CC1)NC(=O)CC1(C)CCOC1)N(C)C C(C)(C(=O)NCCOCCN(C)C(C1(F)COC1)=O)SC c1(OC)ccc(CC(=O)NCCCCC(C)NC(c2c[nH]c(CO)c2)=O)c(Cl)c1 c1(C(=O)Nc2cn(C)c(CNCc3ccc(C(=O)O)s3)c2)cc(F)ccc1[N+](=O)[O-] C(=O)(C1=NOC(C)(C)C1)N(C(CCc1n(C)cnc1)=O)C(c1ccccc1)C(N)=O C(N=c1cc(N2CCOC(C)CC2)nc(C)[nH]1)c1ccc(OC)c(OC)c1 c1(C(=O)NCCCN(C(=O)CSC(F)(F)F)C(C)C)cc2ncn(C)c2cn1 C1(C(C)C#N)CCN(C(=O)CC2CCCN2C(=O)C(C)c2ccsc2)CC1 C(=O)(CCCC(=O)N(C)C)N(CCCCNC(C12CCC1CC2)=O)C N1(C(Cc2ccc(C)nc2Cl)=O)CC2CN(C(C3C4CCN3CC4)=O)CC2C1 C1(C(=O)NC2CCCC(CO)C2)CN(C(c2cc(O)nc(O)n2)=O)CC1(F)F CCCCCCCCC(=O)NC1COC2(C1)CN(C(C1(C)CC(F)C1)=O)C2 C#CCCCCCCC(=O)NC1CN(C(C2CC(N3CCCC3)C2)=O)CCC1C c1(C(=O)OCC(N2C(C(N)=O)CCCC2)=O)nnc2ccccc2n1 c1(C(=O)NCCCC(CO)NC(C2CCC(CC)O2)=O)cc(C)cc(F)c1 C(=O)(C(C)(C)C(C)C)N1CCC(CCN(C(C(CC)COC)=O)C)CC1 CC1(NC(c2nnnn2C2CCCC2)C2(CF)CC2)CC(O)(CO)C1 C1(CCCNC(Cc2cc(C(C)C)no2)=O)CCN(C(=O)C#CC2CC2)CC1 C(=O)(CC(O)CC(C)(C)C)NCC(CC)(CC)NC(C12COCC1C2)=O c1(C(=O)NC2CC(CNC(C=C3CCN(C)C3)=O)C2)ccc(F)c(S(N)(=O)=O)c1 C1(NC(C(CC)(F)F)=O)CC2CC(NC(=O)CC(C)n3cccc3)CC2C1 C1(CCO)CCCN(CC2COCCN2Cc2ncc(-c3ccccc3F)o2)C1 Cc1cnc(C)c(C(=O)NC2CCOCC2NC(=O)C2=CCCSC2)c1 C1(C(=O)NC2(CCNC(C(C)C(C)(C)C)=O)CCOCC2)CCn2ncnc2C1 c1(CNC(=NCC(C)C)NCC2CCCCS2)cn(C)c2ccccc12 c1(C(=O)NC(c2ccsc2)C)ccc(CNC(=O)C(O)CN2CCCC2)cn1 C1(CC(=O)NC2CC3CN(C(=O)CC4(CO)COC4)CC23)CC2(CCC2)CO1 CCCC(CNC(=O)C(C)=C(C)CC)C(=O)N(C)Cc1cc(C)on1 S(=O)(=O)(c1cnoc1C(C)C)NC(c1ccc(C)cc1)CCO CC(O)(CNC(C1CCC1c1nc[nH]n1)=O)CNC(=O)Cn1cccc1 CC1=NNC(=O)C1CC(=O)NCC1(O)CCN(C(=O)CCc2cnn(C)n2)C1 C=CCC(C)(CC=C)NC(c1nnc(-c2cc(C)ccc2C)o1)=O Cc1nc(C)c(C(=O)NCCCOCC(C)(C)NC(C2C(C)C2(F)F)=O)o1 c1(C(N2C(CNC(c3nc(C)oc3C)=O)CCC2)=O)cccc2c(C)ccnc12 N1(C(Cc2c(C)scc2)=O)CCC(C(=O)NC2C(C)C2(C)C)C12CC2 N1(C(c2cc(C(C)=O)sc2)=O)CC2CC(NC(=O)CN(C)C)C(C2)C1 N1(C(c2[nH]cc(C)c2)=O)CCC(N(C(c2ccc(CO)cc2)=O)CC2CC2)CC1 Cc1cc2c(C(N3CC(NC(C4COCCO4)=O)C(F)C3)=O)cccc2[nH]1 c1(C(=O)O)cnc(NCCCOC2CCCCO2)c([N+](=O)[O-])c1 C1(CNC(c2occ(C)n2)=O)CCCCN1c1nccc(C(C)(C)C)n1 C1(NC(c2ccc(CCC)cc2)=O)CC(F)CN(C(c2cc(C)cc(C)c2)=O)C1 N1(C(CCCN(C)C)=O)CC(=O)CC1C(=O)N(C)Cc1cnn[nH]1 C12(C(=O)NC3C(CC)N(C(C4COCCOC4)=O)CC3)CCC(CC)(C1)OC2 CCCC(CCC)C(=O)N1CCC(NC(=O)C(C)(C)OC2CCCC2)C1 N1(C(c2n(COC)nc(Br)c2)C(=O)NCCCOC)CCCC(C)(COC)C1 C1(C#N)(C(=O)NCCc2cn(CCN(C(=O)NC)CC)nn2)CC=CC1 c1(C(N2C(CNC(=O)C#CC3CCC3)CCCC2)=O)ccnc2ccc(Cl)cc12 C1(CC)CN(C(=O)Cc2nccs2)CCN1Cc1ccc(Br)cc1C c1(C(N2CCC(OCCNC(Cn3nnc(C)n3)=O)C2)=O)cnc(S)n1C c1(C(C(=O)N(C(CNC(C2(COCC)CC2)=O)C2CC2)C)O)ccccn1 c1(OC)cccc(CN2C(C(=O)NCc3c(Br)cccc3Br)CC3CC23)c1Cl c1(C(N2CC(NC(c3nn(C(CC)C)c(C)c3)=O)C2)=O)cc2n(n1)CCCC2=O c1(NC(C(Cc2cccnc2)NC(=O)OC(C)(C)C)=O)coc2cc(O)ccc12 c1(C(=O)NC2CN(C(C=CC)=O)CC2(C)C)c[nH]c2ccc(Br)cc2c1=N C(CCN=C(NCc1ccon1)N(C)CC1CCOC1)OC C12(NC(C=CC(=O)NC3(c4ccccc4)C(N)CCC3)=O)CC3CC(C1)CC(F)(C3)C2 c1(OC)cc(F)cc(C)c1C(=O)OC1CCCC1n1cnnc1 c1(NCC(N2CC3CN(CCO)CC3C2)=O)ncccc1S(=O)(=O)N(C)CC c1(NCC(CC=C)(C)C)ccc(S(=O)(=O)N)c(Br)c1.S(C)(=O)(=O)N(C)CC N1(C(C2(C)COC(=O)C2)=O)CC2CC(NC(=O)CCSc3ccccn3)C1C2 CC1CCN(C(=O)CC(C)(C)CNC(C2(C#N)CC23CCC3)=O)CC1C c1(OC)ccc(C(=O)NC2C3CN(C(=O)C(C)CF)CC23)cc1[N+](=O)[O-] C1(OCC(N2C(CSC)CC(NC(C(CC)SC)=O)C2)=O)CCCC(C)C1 c1(C(=O)NCCN(C(=O)C(C)CO)CCC)csc2c(OC)cccc12 CN(S(N)(=O)=O)CC(=O)NCCN(C(=O)CC(=O)OCC(F)(F)F)CCOC C1(C2CC2)(CC)CN(C(=O)C(=O)N(C(c2ccccc2)C(C)C)CCN(C)C)C1 C#CC1(F)CCN(C(C(=O)NCCCC2CC2)C2CC=CC2)CC1 CCC(CC)C(C)C(=O)NCC(c1ccc(F)cc1)NC(C12CC(CO1)C2)=O O=C1NCC2(CCN(C(=O)C(C3CCCC3)NC(C3CCC(=O)CC3)=O)C2)O1 C1(O)(CN(C(COC)=O)C)CCCN(C(C2CCC2(F)F)=O)C1 C(CC(F)(F)CO)NC(=O)CC1(NC(C2(C3CCCCO3)CC2)=O)CCC1 C1(CNC(C=C(CCC)C)=O)CC2CCC1N2C(C1(OC)CCS(=O)(=O)C1)=O Cc1nnc2c(C(=O)NCCCNC(C3CC(C)CCO3)=O)cccn12 c1(OC(=O)NC2CCN(C(C)=O)C2c2ccccc2)nc2ccc(C#N)cc2o1 C(CCCC(=O)N1CCN(C(CNC(c2csc(C)c2C)=O)C(F)F)CC1)OC C1(C(=O)NC(CNC(c2c(CC)ccs2)=O)CO)CCc2c[nH]nc2C1 c1(C(=O)NCC(CNC(c2c(OC)noc2C)=O)O)cc2sccc2[nH]1 N1(C(CCCOCCOC)=O)CC2(CC(CNC(C3CC4CCCC4C3)=O)C2)C1 N1(C(CC(C)(C)C)=O)C2CC1CN(C(C1(O)CCSC1)=O)C2 C(=O)(CC(C)CC(C)(C)C)N(CCN(C(=O)CCC1CCCN1C)C(C)C)C C1(C)(C(=O)NC(c2ccccc2)C(=O)NCC(C)(C)c2cnsc2)CC=CCC1 C1(NC(C(CC)N(CC)CC)=O)CCN(C(=O)CCOCCCOC)C1C(C)C Cc1cc(NCC=CC2CCCC2)ccc1[N+](=O)[O-].c12ccnc(c1)CNC2=O CC1(C)OCCC1C(=O)NC1CCC(CNC(C2COCCO2)=O)CC1 c1(C(=O)OC)[nH]c(N(C(=O)Cc2cc(-c3ccc(Cl)cc3)on2)C)nc1C(C)C CC(C)CC(CC(=O)NCC(c1nccs1)C)NC(C1(F)CCOC1)=O CC1CC(NC(=O)C=Cc2ccncn2)CN(C(=O)C(c2ccc(Cl)s2)C)C1 C1(CNC(C(F)=CC)=O)CN(C(c2cc(C)ncc2C)=O)CCC1(C)C N1(C(C(C)(C)c2cncs2)=O)CCC(O)(CCNC(=O)COC2CC2(F)F)CC1 c1(NCC)ccc(C)cc1C(N1CCC(NC(c2c(C)ncn2C)=O)C(C)C1)=O C(=O)(C(CC(F)F)N(C)C(C1CC(C)CO1)=O)N1CCC(CCCC)C1 O=C(C1CCOc2ccccc21)NCC12CC1CN(C(=O)C1=C(Cl)CCCC1)C2 c1(C(=O)NC2(CCNC(C3C(C(C)C)OCC3)=O)CC2)ccnc2ccnn12 Cc1c(NCc2nnc(C3CC3)o2)ncnc1N(CC=C1CCSCC1)C c1(NCC2CN(C(C3C(C)CC(=O)NC3)=O)C2)ncc([N+](=O)[O-])cn1 C1(CCNC(C(C=C)C)=O)CC(OC)CN1C(c1cc(C)c(C)s1)=O c1(OC)ccc(CC(=O)NC2CC(F)(CNC(=O)CN3CCCCC3C)C2)cc1 c1(-n2ncc(C(N3CC(OCCNC(C(CC)O)=O)C3)=O)n2)cccc(Cl)c1 C(=O)(CCC(=O)NCCOCCCNC(c1cc(Cl)ns1)=O)OC CCCCCC(O)C(=O)NCC(O)CNC(C1(Cl)CC2CCC1O2)=O N1(C(COCC)=O)CC(C(=O)Nc2c(C)cc(Br)cc2Br)CC2OCCC12 c1(SCC(N2C3CN(C(c4nc(N(C)C)oc4)=O)C(C3)C2)=O)ncnc2[nH]cnc12 c1(-c2n(OCc3nc(-c4c(O)ncc(Br)c4)on3)ccn2)cnn2c1CCCC2 C(=O)(C1CCc2nnc(C)n21)N1CCC(NC(c2c(C)[nH]cc2)=O)(CO)C1 Cc1cccnc1CCNC(=O)C=CCC1(NC(C2CCOC(C)C2)=O)CCC1 O=C(CS(=O)(=O)C1CCCC1)NCCCC1CCCCN1C(c1ccc(Cl)[nH]1)=O Cc1cc(Cl)ncc1CC(=O)NC1(C)CC(NC(=O)C(c2ccccc2C)C)C1 c1(CC(N2C(C)CC(NC(C3(O)CC(C)(C)C3)=O)C2)=O)ccc2ocnc2c1 CCCCS(=O)(=O)CC(=O)N1CC(NC(c2coc(C(C)OC)n2)=O)C(F)C1 CN1CC=C(C(=O)N2CCC(C3CC3)(CNC(c3ccc([N+](=O)[O-])[nH]3)=O)C2)C1 c1(OC)cc2c(cc1NC1CCc3c(cnn3CCO)C1)NC(=O)CC2 c1(C(=O)NC(C)CC(C)NC(C2(Cl)CC2)=O)c(F)ccc2occc12 C1(C(N(C)OC2CCCC2)=O)CC12CCN(C(=O)C=Cc1ccncn1)C2 N1(C(C2(C)CCC(C)C2)=O)CCC(CO)(NC(=O)CCC2CCCCO2)CC1 C1(C(=O)NCC2COCCN2C(C2CC2F)=O)CCCC(F)(F)C1 c1(C(N2CC(C)(CNC(=O)C=C3CCC3)OCC2)=O)cnc2n1CCOC2 C(CCCC(F)(F)F)c1cn(C(C)C(C)(C)c2ccccc2)nn1.c1(CN)cccs1 c1(C(C(N2CCC(CNC(C(CC=C)OC)=O)C2)=O)(F)F)ccc(F)cc1C CC1CC2(CCN(C(=O)CCCF)CC2)CN1C(=O)C=CCCCCCCCO c1(OC)cc(C(=O)NCCCCCNC(=O)C(n2nnnc2C(C)(C)C)C)[nH]n1 c1(N(CCOC)CCNC(c2nc(C)no2)=O)ccc([N+](=O)[O-])cc1 C12(NC(C=CC=CC)=O)CCCC1N(C(c1ccnc(OC)c1Br)=O)CCC2 C(CN=c1[nH]c(=NC2CC(N3CCOCC3)C2)c2ccccc2[nH]1)OC C12(C(=O)Nc3c(OC)cccc3)CC(CN(C(=O)OCc3ccccc3)C1)C2 C1(C(=O)NCC(CNC(C(C)OCCC(C)C)=O)O)CCCCN(C)C1=O CC1CC(N(C(Cn2c(CC3CCCC3)nnn2)=O)C)CN1C(=O)COCO C1(NC(C(Cc2ccoc2)NC(C2CC3C=CC2C3)=O)=O)CC1C1CCOCC1 N1(C(C2(CC=C)CC2)=O)CCOC2(CCCN(C(C3CC3F)=O)C2)C1 CC1CC(NC(=O)CC2(N3CCCC3)CC2)CN1C(c1ccc(C2CCOC2)s1)=O N1(C(Cn2cnc(=N)[nH]2)=O)CCOC2(CCC(NC(C3CCOCC3)=O)CC2)C1 N1(C(C(C(CC)C)N(C(=O)CN2CC=CC2)C)=O)CCC(C)(C2CC2)C1 CON1CC(C(=O)NCCCN(C(=O)CCn2cc(C)cn2)CCO)CC1=O C1(C(N2CC(CCC=C)(C(N3CCC3C(N)=O)=O)C2)=O)COCC(C)O1 C(=O)(CC(C)(C)O)NCCCN(CCCNC(C(c1nc(C)sc1)=O)=O)C CC1(CC(=O)NCCCO)CCN(C(=O)CCc2ccccc2O)C1 CC1=C(C(=O)N(CCCS(C)(=O)=O)CC(O)C(C)C)COCC1 c1(C(N2C(CN(C(CCCNC(C)=O)=O)C)CCC2)=O)cc2c(=O)cc[nH]c2s1 C1(C(=O)NC(C(C)NC(=O)C(C2CCCCC2)O)CO)Cc2cccnc2C1 Cc1cc(NCc2cn(C3CCC(C(=O)Nc4n[nH]cc4Br)C3)nn2)cc(C)c1 C(C(CC(C)C)NC(c1cc(-c2ccccn2)ns1)=O)NC(C(C)(C)OC)=O N1(C(CSC(C)C)=O)CCC(CO)(CNC(C2C(CO)C2(C)C)=O)C1 N1(C(C(CC=C)OC)=O)CCC(C)(CCNC(c2cncc(C)c2)=O)CC1 C1(NC(c2cc(C)ncc2)=O)CC2CC1CN(C(c1cc(C)c(Br)o1)=O)C2 c1(C(=O)NC2(C3CCCO3)CC(=O)C2)cccc(C2CCC2)c1 C1(SC)CCC(NC(=O)C(=O)NCC(c2ccccc2)=O)CC1 O=C(CCCCCn1cnnn1)N1CCC(F)C(CO)C1 C1(C)(OC)CCCN(C(=O)C(C(C)C)NC(=O)COCC2CCCO2)CC1 c1(C(=O)OCC)cnc(Nc2c(CC(N3CCC(SC)CC3)=O)scc2)nc1C C(=O)(CCCC(C)CC)N1CCCCC(NC(CCCC)=O)C1 N1(C(=O)OC)CCCN(C(c2cnc(C(F)(F)F)s2)C(=O)NCCCF)CC1 c1(CC)ccc(S(=O)(=O)NC(C(N2CC(C(N)=O)C(CC(=O)OC)C2)C2CC2)=O)cc1 CC1(C)CN(C(=O)C(C)(C)C2CCN(C3CCN(C)CC3)C2)CCO1.CO CC1=NOC(C(C(=O)NCc2ccco2)N(C)CC2CCCOC2)C1 C1(C)CC(=O)NC1.C(=O)(CCSCC(N)=O)NCC(C)NC(c1ccoc1)=O C12(C(=O)NCCN(C)C(c3ccoc3C(F)(F)F)=O)CCC(C)(CO1)C2 c1(CC(=O)NCC(CN(C(C2CC(C)C2)=O)C)C)cncnc1 N=c1[nH]c(=NCc2cncs2)[nH]c(=NCCN2CCC3CCCCC3C2)[nH]1 c1(CCCCOCCOC)nc(COC)nn1-c1cccc(C(F)(F)F)c1 CC(CN(C)C)CCC(=O)NCC1(O)CCN(C(=O)CC(C)c2ccccc2)C1 C1(NC(C(C)COc2ccc(F)cc2)=O)CCN(C(=O)C(=O)N(C)C)CC(O)C1 Cc1ccc(-c2nn[nH]n2)cc1C(C)NCCc1cn[nH]c1 C1(NC(C2CC3CCC2C3)=O)CCCCC12CCN(C(=O)C(C1CC1)C1CC1)C2 C1=CCCn2cc1nn2.C(Cc1ccccc1)(C(=O)O)NC(C1(CO)CCCO1)=O Cc1nc(NCCCOCCNC(C2CC3CCCC23)=O)cc(C#N)n1 c1(C(=O)NC(C(C)NC(=O)CCCc2cnn[nH]2)C)ccc2cnoc2c1 C1(NC(CCSC)=O)CCN(C(=O)Cc2cnc(C)nc2O)C12CC2 C(C(C)(C)C(=O)NCC(C)N(C)C(C1CC(=O)N(C)C1)=O)OC(C)C C1(NC(CNC(CC)=O)=O)CC2CC(NC(=O)C(C)(C)C(N)=O)C1C2 N1(C(C2N(C(c3nc(C)sc3C)=O)C(C3CC3)CC2)=O)CCS(=O)(=O)CC1.C(C)C N1(C(=O)Cn2cc(-c3ccccc3)cn2)CCN(C(c2cc(CO)[nH]n2)=O)CC1 N1(C(C=CSC)=O)CCC(CC(C)NC(c2cccc(C(=O)OC)c2)=O)CC1 C(=O)(C1=CCOCC1)N1C(C(=O)NCc2c(C)cccc2)CCCC1 N#Cc1cnn(CC(N2CCCOC(CNC(=O)CC3CCCCO3)C2)=O)c1N c1(CCC(=O)NCC(C)NC(=O)CCSC(F)(F)F)nnc(C(F)F)o1 c1(CCC)cnc(N(C(C2CNCC(O)C2)=O)Cc2occc2Br)nc1 c1(N2CC(c3scc(C)n3)OCC2)nc(N(C)C)cc(N2CCC(C(F)(F)F)C2)n1 CC(C)(CC(=O)N1CC(F)(F)CC1CCNC(c1ccc([N+](=O)[O-])o1)=O)C(F)F C1(NC(CCCCC#C)=O)CN(C(=O)Cn2cncn2)C2CCCC12 C1(C(=O)NC2(C=C)CCC2)CC(=C)CCN1C(=O)CN(C(=O)COC)C CC1CCc2nc(CNC(=O)N(C)Cc3cccnc3Cl)sc2C1 CC1(C)CCC(C(Cc2cnc[nH]2)C(=O)N2CCC(c3nccs3)C2)CC1 C(C#Cc1cn(C(c2cccc(F)c2)CCO)nn1)NC(CC(C)C)=O C=CCC(CC=C)C(=O)NCC(C1CC1)NC(C1(C)CCCCNC1=O)=O CC1CC(CNC(=O)CONC(C2CC(=O)C23CCC3)=O)CC(=O)N1 C1(CCNC(C2CC(C(C)C)C2)=O)CC(F)(F)CN1C(=O)C1=CCCSC1 C#CC1CCCC(CNC(=O)C(CC=CC)NC(=O)Cc2ccc(F)cc2)C1 C1(CC)CCC(C)N(C(C2CCN(C(c3ncccc3C)=O)CC2)=O)C1 C1(C(=O)NCC23CC2CN(C(=O)C2=COCCC2)C3)CC(C2CC2)=NO1 c1(C(N2CCC(CCNC(C(C)=C(C)C)=O)C2)=O)ccnc(C)n1 n1(CC(=O)NCC2(F)CCN(C(C3CC3C3CCCO3)=O)C2)cnc([N+](=O)[O-])n1 C(=O)(CC(CC=C)NC(c1ccccc1C(N)=O)=O)NCCC=CC=C c1(NC(C(N2CCC(CC(=O)Nc3ncn(CC#C)n3)C2)=O)=O)ccc(C)cc1 CN=c1cc(C(=O)NC(CC(C)C)C(=O)NCC(O)CC(C)C)cc[nH]1 CCC(CC(=O)NC1CN(C(c2ccc(SC)cc2Cl)=O)CC1(C)C)C(F)F c1(C(=O)NC2C(CNC(=O)CCOCC(F)(F)F)CC2)cc2n(c1)CCSC2 C(=O)(C(C)(C)CS(N)(=O)=O)NC1CCN(C(C)C(=O)NCC2CC2)C1 C1(C(=O)NCC(CC)N(C(=O)CCOCCOC)C)CCC(C(N)=O)C1 C1(NC(C(C)NC(C)=O)=O)CCN(c2ncnc3sccc23)CC1(C)C c1(NCCCCCN(C)C)ccc(N)c([N+](=O)[O-])c1 Cc1nc(CNC(Cc2ccccc2Br)CO)nn1C.C1(c2nccs2)C(=O)N1 OCCC(N=c1nc(N2CCc3nocc3C2)c2c([nH]1)CCS2)C1CCOCC1 c1(C(N(CCNC(C2(OCC)CCCC2)=O)CC)=O)ccc(Cl)c(F)c1O C(=O)(CC(F)(F)C(F)F)N1CCCC(CN(C(=O)CCN(S(C)(=O)=O)C)C)C1 CC(C)C(F)(F)CC(=O)NC1CC(CO)N(C(C2CC(C)N(C)C2)=O)C1 Cc1[nH]c(=N)nc(O)c1CCC(=O)NC1CC1NC(c1cc2ccncc2o1)=O C1(C(=O)NCC2(N(C)C)CC2)(COC)C=CCN1C(c1cc(=N)[nH][nH]1)=O Cc1cc(C(=O)N(CC(=O)NC2CCSC2)C)cnc1O c1(CC(C)C)cnc(C(N2CCC(C(C)(O)CO)C2)=O)s1 N1(C(C(c2cnn(C)c2)OC)=O)CCN(C(=O)CCn2ccnn2)CC(CO)C1 N1(C(C(n2cc(CNC(c3cc(Cl)nn3C)=O)nn2)C)=O)CCC(O)(CO)CC1 c1(C(=O)NCC2(NC(C(CC)C(C)C)=O)CCOC2)c[nH]c(=N)c2[nH]ccc12 c1(C(C(=O)NC2CCCCC2)N(C2CCSC2)CC)cnc(Cl)cc1 CCC(CC)CCC(=O)NCCC1CCCN(C(c2cc(CO)[nH]n2)=O)CC1 c1(OC)ccc(C(C2(O)CN(C(C)=O)C2)C)cn1.C(=O)(CCOCCOC)NC c1(CNC(C2CCC3CC3CC2)=O)cnc2n1CCOC2 C(=O)(C(C(=O)N1CCC(c2cn(-c3occc3N(C)C)nn2)C1)OC)OC N1(CC(=O)NCC(=C)CCNC(=O)C2=CC(C)(C)C2)C(=O)NC(C)(C2CC2)C1=O CCCN=C(NCC(C)Oc1ccccn1)NCC1CC12CCC2 C(=O)(C(C)C(O)C(C)CC)N1CCC(CCNC(COCCCC#C)=O)CC1C N1(C(C2C(C)OCCC2)=O)CCC2(CCC(CNC(c3coc(Cl)c3)=O)O2)CC1 Cc1ncc(C(=O)NCC2(CNC(c3n[nH]c(C)c3O)=O)CCOCC2)cn1 N1(C(CN(C)C)=O)CC(F)(F)CC1CCNC(C1CC(O)C1)=O N(C(=NCCCOC1CCC1)N1CCCC(C(=O)OC)CC1)CC#CC C#CCCCCCCC(=O)NC(c1ccc(OC)c(Br)c1)CCCCC N1(C(c2c(C)cccn2)=O)CCCC2(NC(=O)CCOCCOCCO)CC2C1 N1(C(=O)OC(C)(C)C)CCc2c(C(=O)OCC(N3CCCCC3)=O)n[nH]c2C1 C1(O)(C(C)NC(C2CC(CCO)C2)=O)CCN(C(=O)C(C)(C)c2cccnc2)C1 C(CCCC(=O)NCc1ccc(C(C)NC(=O)C=C2CCN(C)C2)cc1)OC CC(C)CC(F)C(=O)NC1CCCC(CNC(C23CC(F)(C2)C3)=O)C1 c1(CCC(=O)NC2(C)CCN(C(c3c(C)coc3)=O)C2)ccc(F)cc1Cl N1(C(Cc2c(C)occ2)=O)CCC(NC(C2(c3ccccc3Cl)CC2)=O)CC1C C(=O)(C1CCCn2cnnc21)N1CC(=O)N(Cc2ccn3cnc(C)c3c2)C1=O C1(CNC(C2(C)CCN(C)C2=O)=O)CN(C(=O)Cc2ccsc2)CC(C)(C)C1 c1(C(C)O)ncc(C(=O)NC(CNC(=O)CC2(CO)CC2)CO)s1 N1(C(C2C(C)(C)C(CNC(=O)Cc3cccnc3F)C2)=O)CCOC2COCC12 CC1(C)CCC=C1C(=O)NC1CN(C(c2cc(Br)sn2)=O)CC12CC2 c1(-n2c(-c3sc(C)cc3Cl)nc(CSC)n2)ccc(Br)cc1C CCC(CC)C(C)C(=O)NC1(CNC(=O)C=Cc2ccc[nH]2)CCOCC1 C1(CNC(=O)C=Cc2ccco2)CCN(c2ncc(I)cn2)C12CC2 C1(C#N)(C(N(CCN(C(C)C)C(c2cn(CC(F)F)cn2)=O)C)=O)CCCOC1 C1(N(C(=O)CC2CC23CC3)C)CCN(C(c2cc(C3CC3)ns2)=O)CC1 c1(OCC)oc(C)nc1C(N1CC(CO)(NC(C2CNC(=O)N2)=O)C1)=O c1(CC)noc(C(N2CC(NC(=O)CCn3ncn(C)c3=O)C(O)C2)=O)c1C C1(N(C)C(C2CC2C(F)F)=O)CN(C(=O)CCc2cccc(Cl)c2)CC1O CCCC(F)C(=O)NC1CCCC(CN(C(=O)C(C)N(C)C(C)=O)C)C1 c1(C(=O)OCC(C2(CC(=O)OC)CC2)OC)cnc2c[nH]nc2c1 C1(C)(NC(C(CC2CC2)OC)=O)CCCN(C(=O)CN2CCC(N(C)C)CC2)C1 c1(C(N(C)CC2CCCN2C(=O)CCOC2CC2)=O)c(Cl)ccc(Br)c1F CCCCC(C)CCC(=O)N1CCC(CC(N2CC(OC)CC(F)C2)=O)CC1 C1(C=O)CC2CCC1C2.c1(C=O)ccc(C(N)=O)[nH]1.CC(C)N1CCN1C N1(C(c2c(SC)n(C)nc2)=O)CCN(C(=O)Cn2cncc2C)C(C)C1C C1(O)(C(N2CCC(C3CCCCN3C(C34CCC3C4)=O)CC2)=O)CCOCC1 C(=O)(CS(=O)CC)NC(C(C)NC(c1c(CCC)nco1)=O)(C)C CC1(C)CC2C(CO1)C1=NNC=CCN(CC1)C(=O)C1CCN(C2=O)O1 N(C(=NCc1ccccc1)N1CCC(C)(C(=O)OCC)C1)C(C#C)C1CCC1 CC1CN(C(c2cc(CO)[nH]n2)=O)CC1NC(c1csc(C2CCCCO2)n1)=O c1(OCCC(N2CC3C(CNC(COC)=O)(C3)C2)=O)ccccc1C#N N1(CC(=O)N(C)CC2CN(C(CNC(CCC)=O)=O)CC2O)CCN(C)C(=O)C1 C(=O)(C1=CCOCC1)NC12CC(NC(COc3cccc(N)c3)=O)(C1)C2.C1CC1 C1(CC(=O)NCC(CC)N(C(c2c(C)cc(CC)o2)=O)C)OCCCC1(C)C c1(C(=O)Nc2cccc(CNC(=O)CSC(F)F)c2)cc2c(nn1)CCOC2 n1(CC(=O)NCC2N(C(C(CC)CCOC)=O)CCCC2)nc2c(n1)CCCC2 CN(CCS(=O)(=O)c1cccc(N)c1)Sc1ccc(F)cc1 CC(C(=O)N(C)CCn1ccnc1)NC(=O)C(F)n1ccnc1 C#CCCCCCC(=O)NCC1(C)CCCN(C(C(=O)NC(C)C)=O)C1 c1(C(=O)NCC2CC(NC(c3cnn(CC)n3)=O)C2)c(C)cc(Cl)cc1C c1(C(=O)NCC2C(NC(C3(C(C)C)CCC3)=O)C2)cnc2cc(Br)ccn12 c1(C(=O)OC)ccc(S(=O)(=O)Nc2cccc(Cl)c2C)cc1[N+](=O)[O-] Fc1cc(Br)c2ncnc(N3CCOC(c4ccoc4)C3)c2c1 Cc1c(C(=O)NCCCCC2CN(C(C3CC4CC4C3)=O)C2)cccc1Cl c1(CC)cc(OCC(=O)NCC2CN(C(C3CCCC3)=O)CCO2)ccc1Cl CC12CC(NC(c3cccc(Cl)c3Cl)c3nn[nH]n3)(C1)C1(CNC1)O2 c1(C(=O)NCCC2N(C(c3ccc(C#N)[nH]3)=O)CCC2)cnc(O)c(F)c1 N1(C(CCC(=O)N(C)C)=O)CCCN(CCNC(c2ccc(Cl)[nH]2)=O)CC1 N1(C(C2N(CCC)CCC2)=O)CCC(C(=O)NCc2nnnn2CC)C1C Cn1cnc2c(C(=O)NC3(CNCC4(c5ccno5)CCC4)CC3)ncnc12 c1(C(=O)NC(C2CCCCC2)(CNC(CN2CC(C)C2)=O)O)ccnnc1O C(CCC(C)C)(C(=O)NCc1sccc1C)NC(Cc1c(C)n[nH]c1)=O C1(NC(CCCOC(C)C)=O)CN(C(=O)Cc2nnc(O)s2)CCC1O c1(C(N2CCN(C(C34C(C)OC(CO)(C3)C4)=O)CC2)=O)cccc2c1OCC2C c1(C(N2CC(c3cn(CC)nn3)(N=C(C)C(F)F)C2)=O)cnn(C2CCC2)c1C C1(C(C(=O)NCC)N(CC)CC2CCN(CC(F)F)C2)CCOCC1 C1(OC)(CNC(c2ccco2)=O)CCN(C(=O)COc2ccc(C(N)=O)cn2)C1 CCCC(O)(CCC)CC(=O)N(CC)CC1(C)CN(C(=O)C(C)O)CC1C C1(NC(CC=CCCCCC)=O)COCCC1C(N1CCCC(CCCO)C1)=O n1(CCC(=O)NC2CCCC2NC(C2CCCN2CC(F)F)=O)cnccc1=O c1(NC(CC2N(Cc3cc(C)[nH]c3C)CCC2)=O)ccc2n[nH]cc2c1 C1(NC(c2c(C)cnnc2)=O)CN(C(=O)Cc2ccc(CO)cc2)CCC1CO C12(NC(c3c(OC)cccc3)=O)CCCCCC1N(C(=O)Cn1cccn1)CC2 C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(=O)COCCCF)CC1F C(=O)(C1CCCc2scnc21)N(CCCNC(c1nccc(OC)c1)=O)C(C)C C1(C(=O)NC(C)CC(C)NC(C2(C)CC2)=O)CC2(CCCCC2)C1 N1(C(c2c(C)cno2)=O)CCC2(NC(C3CCCSS3)c3ccccc3)CCCC12 N1(C(c2n(CC)cc(Cl)c2)=O)CCCC2(CCN(C(c3ccccc3O)=O)C2)C1 c1(C(=O)OC)ccnc(CNC(=O)N(c2ccccc2Br)CCO)c1 N1(C(COC(CC)C)=O)CCC(C)(C)CC1C(N1CCN(C)C(=O)C1)=O C(CC(C(=O)NCC(C)(O)CCO)NC(C1CCC(=O)NC1)=O)OC Cc1cn2c(C(=O)NC3CCC(NC(C45CCC4C5)=O)CC3)c(C)nc2s1 CCCCCCC(CC)NC(c1ccc2cncn2c1)=O N1(C(C(C)c2cccs2)=O)CC2CC2(CNC(=O)CC2CC2)C1 N1(C(COC(CC)C)=O)CC(C2CN(C(C3(CO)CCC3)=O)C2)C1 c1(C(=O)OC)ncc(F)cc1NC(C1CC(O)CCN1C(c1nc(Br)cs1)=O)=O C1(CC)CCN(C(=O)CC=C(Cl)Cl)C1C(=O)NOC(c1ccccn1)C c1(CCC(=O)NC2C(OC)CN(C(=O)Cc3ncc(C)[nH]3)C2)ccc(C)c(Cl)c1 c1(C(N2CCN(C)C(CNC(=O)CCS(N)(=O)=O)C2)=O)cccc2c1OCO2 N1(C(C2C(OC(C)=O)C2)=O)CC2CC(C(=O)NCCOCCCO)C(C2)C1 N1(C(CCc2cc(C)no2)=O)CC2(CC2)CC1CNC(C1CC(C)(C)CN1C)=O c1(C(=O)NCC2(NC(C3C(C)(C)C3)=O)CC2)cccc2c1OCCC2 N1(C(C2C(OCC)C2)=O)C2CCC1CC(CNC(=O)C(O)C1CCC1)C2 c1(CNC(N(OCC)C)=O)cccc(C)n1 c1(C(N(C2CN(C(c3cnc(C(C)C)s3)=O)C2)C)=O)ccccc1F C#Cc1ccc(CC(=O)NCC2CCCCN(C(=O)C(O)c3cnc[nH]3)C2)cc1 c1(C(N2C3CN(C(CCC(C)C#N)=O)C(C3)C2)=O)cc2ccncc2s1 N1(C(COCC=C)=O)CC(NC(c2cnn(C)c2)=O)CC1CO C(=O)(C(C)(O)COC)NCC(n1cc(CCCC=C)nn1)C c1(CN2C(c3cccc(C)c3)COCC2)cccc2c(C(=O)O)n[nH]c12 C1(CC)CN(C(=O)CC(Cl)Cl)CCC1NC(=O)CC1=CCCC1 c1(C(=O)NC(CC(C)NC(c2c(COC)scc2)=O)C)c(F)cc(C#N)cc1F c1(CNC2CC(N(C)C)C2(C)C)ccc(O)cc1C#N C(CCCCCC(=O)NC1C2CCN(C(=O)C3=CCOC3)CC12)SC c12conc1CC(=O)NC2.C1(CNC(C2C(C(C)C)CC2)=O)C(CO)C1(F)F n1(CC#C)ccc(CNC(C(F)(F)F)C2CC2)c1 C1(C)(COC)CC(NC(=O)C(C)(C)C(C)C)CN1C(=O)C=Cc1sccc1C C(=O)(C1CCCc2sccc21)NCC(C)(C)NC(C1C(COC)(COC)C1)=O C1(NC(=O)OC(C)(C)C)CCN(N2CCN(C(N)=O)C(C(N)=O)C2)CC1 c1(CN2CCN(c3cc(OC)c(F)cc3)CC2)c(F)ccc(Br)c1Cl c1(OC)cccc(CNC(=O)NC(c2cccc(OC)c2)C(O)SC)c1F c1(C(=O)NC(C2CCCN2C(=O)CCOCC2CC2)C)ncccc1F CC(CC(=O)N1CC(F)(F)CC1C(=O)NS(C)(=O)=O)CC(C)(C)C c1(C(=O)NCCC2CC(CNC(CN(S(CC)(=O)=O)C)=O)C2)c[nH]cc(C)c1=O C1(CNC(c2ccn(CC)n2)=O)CCC(C)N(C(c2cc(C(F)(F)F)no2)=O)C1 CC1CCC(C(=O)NC2CCC(=O)N(C)C2)CN1C(=O)CCC1CCCO1 N12CC3C(C3C1)C2=O.c1(CNC(C2CCN(C)C2)=O)cccc(F)c1 C(=O)(C(F)C(C)(C)O)N1CCC(C(C(C)C)NC(=O)CC(C)(C)C2CC2)CC1 Cc1c(C(=O)NCC23CC(NC(=O)CC4CCC5CC45)(CCO2)C3)nn(C)c1N c1(OCCOC)cccc(C=CC(=O)NC2CN(C(C3C=C3C)=O)CC2SC)c1 Cn1cc(C(N2CCCOC(CCNC(c3cc(Cl)cnn3)=O)C2)=O)ncc1=O C12(NC(c3ccc(OCC)nc3)=O)CC(C(F)(F)F)CC1CN(C(=O)NCC)C2 n1(CC(=O)NCC(C2N(C(CC(C)F)=O)CCCC2)(C)C)cc(Cl)c(O)nc1=O Cc1nnsc1C(=O)NCC1(CNC(c2cccnn2)=O)CCC1 C12(C(N(CC(CN(C(c3c(C)cno3)=O)C)O)C)=O)CCC(CC1)C(C)O2 Cc1cc(CNC(=O)CC=CCNC(C2CC3CCC2O3)=O)nc(C)c1 CCCCCCC(C)(CC)C(=O)N1CCCC(N(C(=O)CCCC)CC2CC2)C1 N1(C(=O)CCC2CCCC(O)C2)CCN(C(c2cc[nH]n2)=O)C2(CCC2)C1 N1(C(C(C)NS(CCCC)(=O)=O)=O)C2CCC(C2)C1CNC(=O)COC1CC1 N1(C(c2[nH]cc(S(N)(=O)=O)c2)=O)CCC2(CCCN(C(=O)CCC3CCC3)C2)C1 N1(C2CCCN(C)C2=O)CCC2(CCC2)C(NC(=O)CCc2ccncc2)C1 C#CCCCCCCC(=O)N(CCC(C(C)(C)C)NC(c1nn(C)cc1Cl)=O)C S(=O)(=O)(C1(c2ccc(-c3nc(C4CCCC45CCC5)no3)cc2)CCC1)N(C)C C(CCCC(=O)NC1CN(C(=O)CN2CCCS2(=O)=O)CC1C)N(C(C)C)C C1(CNC(CC2N(C(Cc3cc(OC)no3)=O)CCC2)=O)NC(=O)OC1(C)C C1(C(=O)NC(C(C)C)CNC(=O)CCc2ccsc2)OCCC1(C)C c1(CC)ccc(O)c(C(=O)NC2CC(C)CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)c1 OC1C(c2nc(-c3cc(Br)cs3)no2)COC1O Cc1cccc(C(=O)N(C2CCN(C(=O)CC(C)C)C2)CCO)c1[N+](=O)[O-] C1(NC(c2ncc(C)c(Cl)c2)=O)CCOC12CCN(C(C1CSCCS1)=O)CC2 C1(=O)CCCC(=O)N1.C1(C(N2CC(=C(F)C(=O)O)C2)=O)(CC)CCCO1 c1(C(C)C)ccc2occ(C(N3CCC3C)=O)c2c1.c1(C(=O)NCC=CC#N)cc[nH]c1 C1(CCC(=O)N2C(C(N)=O)CC2)(NC(=O)CC2OCCCO2)CCCC1 c1(C(=O)NC(C)CNC(=O)C2=NOC(C)C2)sccc1S(=O)(=O)NC(C)(C)C CN1CCC(C)(C(N2CCC(O)(CNC(c3cn(C)nc3O)=O)CC2)=O)C1=O N1(C(CCC(C)(C)NC(C(C)OCCC(C)C)=O)=O)CC2(CO)CCC1CC2 C1(OCC)CCC(c2nnnn2CC2CCOC2)(NCc2nncs2)CC1.CCO CC1CC(C(N2CCC(F)(CNC(C3CCN(C)CC3)=O)CC2)=O)CCN1C c1(C(=O)NC2CCCC(N(C(C(F)=CC)=O)C)C2)[nH]c(C)c(C(=O)OC)c1C CC1CC(C(=O)NCc2nccs2)N1C(=O)Cc1cnoc1 c1(OCC)ccc(Cl)c(C(N2CCN(C(c3nccn3C)=O)C(CO)C2)=O)n1 Cc1cc(C(=O)NCCCC(C)NC(=O)Cc2ccc(F)cn2)c(C)s1 C1(C(=O)NC2C(CNC(Cc3c(C)ncc(Cl)c3)=O)C2)CCCCC12OCCO2 C(=O)(CS(=O)(=O)CCOC)N(C1CCN(C(c2ncc(F)cn2)=O)C1)CCC CCCCC(C)C(=O)NCC(O)CNC(C1(c2ccc(O)nc2)CCC1)=O C12(CNC(C(C)SCC)=O)CC(NC(C3CCCN3N=O)=O)(C1)C1(CCC1)O2 C(=O)(C(C(C)CC1CCOCC1)N(C1CCSC1)C1CC1)NC(C(=O)OC)C N1(C(c2c(COC)scc2)=O)CC(NC(=O)CC2CC=CC2)CC12CCCC2 CS(=O)(=O)c1cccc(NC(=O)Nc2cccc(C3OCC3(F)F)c2)c1F CC1CN(C(c2n[nH]cc2C2CCC2)=O)CCN(C(=O)CCC(C)(C)C)C1 C(=O)(C(CCCC#N)N(C(C(=O)OC(C)(C)C)Cc1cnco1)C)OCC C(=O)(CC1C(=O)Nc2ccc(Br)cc21)N1CC(NC(C2CC(F)C2)=O)C1 c1(C2(C(N(CCNC(C(F)=CC)=O)CCC)=O)CCC2)ccccc1Br c1(C(N2C(CN(C(C3(OC)CC(CF)C3)=O)C)COCC2)=O)cccc(O)c1F Cc1cccc2cc(C(=O)NC3(CNC(=O)C(C)(O)C4CCC4)CCOC3)oc12 c1(C(=O)NCC2CC(C)N(C(=O)CCc3ccsc3)C2)c(F)cc(O)cc1F C1(CC(=O)NC(CN(C(=O)CCCc2ccncc2)C)(C)C)CCS(=O)(=O)C1 C=CC1(NC(c2nnnn2CCOC(C)(C)C)C2CC2)CCCCC1 c1(CC(=O)NCC2N(C(C(C=CC)O)=O)CCC2)c(F)cccc1F c1(CC)cc(C(=O)NC2CC(NC(=O)C=CSc3nc[nH]n3)C2)n(C)n1 c1(C(N2CCN(CC3CN(C(c4ccsn4)=O)C3)CC2)=O)n[nH]c2c1CCCC2 C(CC(C(=O)N1CCCC(N(C)C)C1)NC(=O)C(C)OCCOCC)=CC N1(C(CC(C(C)C)OCC)=O)CCC2(CC1)CN(C(=O)CCCN1CCCC1)C2 C1(CC(=O)NCC(C)CN(C(=O)Cn2ncc(O)nc2=O)C)CCC2(CC1)CC2 c1(CC(=O)NC2CN(C(C(F)OC)=O)CC2C)c(C)cc(Br)cc1C C1(C(=O)NCCN(C(=O)CCCN2CCCC2)CCOC)CCC2CC12 C1(NC(C(C)OCC=C)=O)CCN(C(=O)Cc2ccc(Cl)c(C)c2)CC1O c1(C(=O)NC2CCCCC2CNC(C23CC(F)(C2)C3)=O)cccc2cnccc12 C1(C(N2C(CC)C(NC(=O)CCC(N)=O)CC2)=O)CC2CC(O)C(C1)C2 c1(C(=O)NCCCCC2(NC(C3CCC(C)S3)=O)CC2)cnc2c[nH]nc2c1 c1(C(N(C(CC)C)CC)=O)cc(CNC(c2ccc(CO)nc2)=O)nn1C N1(C(c2c(C)nc(C)o2)=O)CCC(C)N(C(=O)CCN2CCCCC2C)CC1 C1(CC)C(=O)NCCN1C(=O)C(c1cnsc1)NC(=O)CSCCC(C)C C1(C(=O)NC(c2ccccc2O)C)(CC)CCCN1C(=O)CC1COCC(C)O1 CC(C)CC(C)C(c1nnnn1CCC1CC1)NCCCc1ncn(C)n1 C1(C(=O)NC2(C)CCN(C(c3cccc(=O)o3)=O)CC2)CCCCC12CC2(F)F N1(C(CC2CC(OC)C2)=O)C2CCC1CN(C(c1conc1C1(C)COC1)=O)C2 Cc1nccc2c(=O)c(C(N3CCc4scc(Cl)c4C3)=O)c[nH]c12 O=C(C1=CCCCO1)NCC(CC(=O)N1CC=CC1CF)C1CCC1 C1(NC(c2c(OC)n[nH]c2)=O)CN(C(=O)C(C)C2CC2)CC1N=[N+]=[N-] CC1=C(C(=O)NCC2CC2CC(=O)Nc2ccsc2C)CCC1 N1(C(CN(C(CC(=O)NCC#C)=O)CC)=O)CCN(C)CC1C N1(C(C(CC)O)=O)CCCN(C(=O)COCc2ccnn2C)CC1 C1(C(=O)NC(C)CC(F)(F)F)(OC)CCN(C(c2cccnc2)=O)C1 Cc1ccc(C=CC(N2CCC(NC(=O)Cn3nnnc3C)C(O)C2)=O)cc1C CCCC(CCC)CC(=O)N1CCC(C(F)C(=O)NCCNS(=O)(=O)CC)C1 C1(C(=O)NCCC=CC(C)(C)C)CC(NC(=O)CC(=O)NC2CC2)C12CCC2 N1(C(CN2CC(=O)NCC2)=O)CC2CCC2(CC(=O)NC2CC3CCC(C2)O3)C1 CC(C)CCC(=O)Nc1ccccc1C(F)(F)F.C12CCN(CC1)CC(=O)N2 CC1CN(C(c2ccn(CCO)c(=O)c2)=O)CCC1N(C(=O)CC(F)(F)F)C N1(C(C(C(C)O)N(C)C)=O)CC2(C1)SCCC2NC(=O)CCCc1nccs1 C12(NC(c3cccc(C)n3)=O)CCOCC1CN(C(C1(Br)CC13CCC3)=O)C2 N1(C(Cc2c(C(C)C)con2)=O)CCC2(C1)CN(C(=O)Cc1ccnnc1O)C2 CC1CC(NC(=O)C(=O)NCC(F)(F)F)CN1C(=O)CC=C(Cl)Cl C#CCC(C(=O)N(C)CC1CCN(C(=O)COc2cccnc2)C1)C1CC1 C(C(C)(COC)C(=O)NC(CC(=O)NCCC1CC(C)(C)CO1)C(F)F)OC C1(S(C)(=O)=O)(C(=O)NCCC(C)N(C(C(C(=O)OCC)OC)=O)C)CCCC1 CCCCCCCC(=O)N1CC2CC1C2NC(c1csc(C(C)OC)n1)=O C1(C)(CC)CCCN(C(C2(NC(c3cc(C)nc(C)n3)=O)CSC2)=O)CC1 C(=O)(C(C1=C(C)C=CCC1(C)C)N(C)Cc1ccc(F)cc1F)NC(CC)(C)C c1(N2C(CSC)CCCC2)ccc(S(=O)(=O)NC(C)CCSC)c(Br)c1 C(=O)(C1=C(F)CN(C(c2cnccn2)=O)CC1)N1CCC(C(C)(C)C)CC1 C(CC1CCCCO1)(C(=O)NCCCSCC)N(CCC)C(C)C c1(C(=O)NCC(CC(C)C)NC(=O)C(C)C2CCCC2)cccn2[nH]c(=N)nc12 C1(CNC(c2occc2Br)=O)CN(C(=O)C(F)F)CCC1(F)F C1(O)(CN(C)C(C2CCOC2)=O)CCN(C(=O)CSCc2csc(=N)[nH]2)CC1 C1(C)(C(N2CCC(N(C(C(C)OCCCC)=O)C)CC2)=O)CCCCNC1=O Cc1cccc(C(N2CCC(C)(C)C2CNC(=O)CC(C)n2ccnc2)=O)c1Cl N1(C(C(C)N(C)C)=O)CC2C(CNC(c3cccn3Cc3ccccn3)=O)C2C1 C1(CNC(CCNC(C)=O)=O)CC(O)CN1C(c1cnc(S)n1C)=O N1(C(C)=O)CC2CCC(C1)N2C1CCN(c2cccc(OC3CCCC3)c2)CC1 C1(NC(C(C2(C)CC2)NC(CCC=CC(C)C)=O)=O)CN(C)CC1C N1(Cc2cn(CCC)nc2)CCN(C(c2ncc(C(=O)OC)[nH]2)=O)C(C)C1 c1(CC)c(C)cc(C)cc1C.c12cc(cc(C)n1)C(=O)Nc1cccc(c1)NC2 N1(C(CCc2c(C)nn(C)c2)=O)CCC(NC(=O)CNS(N)(=O)=O)CC1C C1(NC(C=CC(N)=O)=O)CN(C(=O)CC2CCCCC2)CCC1C(F)(F)F C(=O)(C(C)C(O)C(C)C)NC1CC=C(C(=O)NCC(=O)NC)C1 c1(C(=O)NCC#CCNC(c2nc(C)oc2)=O)cc2cccc([N+](=O)[O-])c2[nH]1 C1(F)(C(N(CCC(=O)NCc2nc(C(C)C)n[nH]2)CC)=O)CC=CCC1 CCCCC(C(=O)NCCn1nc(C)nc1C)NC(c1coc(COC)n1)=O c1(C(C)(C)C)n[nH]c(=NC2CN(C(c3cccc4nc(O)[nH]c34)=O)CC2C)s1 c1(C(=O)NCCCN(C(CSCC)=O)C)ccn(Cc2ccncc2)c1C c1(CN(C(c2cnc(C)[nH]2)C(=O)NCC)C)ccc(OCCO)cc1 C(=O)(C(C)C(C)NC(=O)CC1CCC(NC(=O)Cn2ccnc2C)CC1)OC c1(C(C)C)ccc(-n2nc(CCOC(C)C)nc2-c2coc(C(C)C)n2)cc1 C#CCCC(O)C(=O)N1CCC(C(C)(C)NC(=O)CNc2ccc(Cl)cc2)CC1 c1(C(N2CCC(O)(C(CNC(CCOCCC)=O)C)C2)=O)cccc(F)c1SC N1(C(CC)C)CCN(C(=O)CN(C(=O)C2=CCSC2)C2CCC2)CC1 C1(C(N2CCC(N(C(=O)CCc3nnc(S)n3C)CC)C2)=O)CCN(C)C(C)C1 N1(C(C2(C)N(C(C)=O)CCC2)=O)C2CCC1CN(C(=O)CCc1ccon1)C2 C(=O)(C(CNC(C1(F)CCCC1)=O)CC1CC1)NC(COC)C1CC1 Cc1cnc(C(N2CCN(C(=O)CC(C)F)C(C)C2)=O)cc1Cl C1(CC(=O)NCc2n(CCC)ncn2)CC(F)CN1C(=O)C(C)C(F)F Cc1ccc(OCC(=O)NC2(C)CCN(C(c3[nH]c(C)c(C)c3C)=O)C2)cc1C CCCC(C)C(=O)N1CC(C)(NC(c2ccc(OCC(F)(F)F)cn2)=O)C1 C1(CC(=O)N(C(C)CCNC(=O)COC2CC(F)(F)C2)C)CCCC12CC2 C(=O)(C(OCC1CC1)NC(=O)C(C)=CCN(C(=O)C(C)OC1CCCC1)C)OC C1(C)(CNC(C(C=CCCC)O)=O)CN(C(=O)Cc2nc(C)sc2C)C(C)(C)C1 C(=O)(C1=CCC(NC(=O)CCCC2CC2)C1)NC(CC)Cn1cncn1 C1(C(=O)NCC(C)N(C(=O)C(C)N(C)Cc2ccccc2)C)COC(C)(C)C1 c1(C(N2C(C(N3CCOCC3C3CCC3)=O)CCCC2)=O)cccc(F)c1O n1(-c2n(C)nnc2)nc(-c2ccnn2C)nc1C1CCN(CC(F)(F)F)CC1 c1(CC(N2CC(n3cc(C4CCC4)nn3)C2)=O)ccc(O)c([N+](=O)[O-])c1 C1(C(=O)NC2CN(C(C(C=C)O)=O)C2)(CCF)CCOCC1 CC1CC2(CCCN(C(C3CC(C)(C)C3C(=O)O)=O)C2)CO1 N1(C(C2(C)CC2)=O)C2CCC1CN(C(C1CCC(=O)N1Cc1ccccc1)=O)C2 c1(OCC)ccc(C2CC(NC(c3cn(C)nc3Br)C)C2)cc1 C(#Cc1ccccc1)CCC=CCSC1CCC2C3C=CC(C3)C12 C(=O)(C#CC1(C)CCCO1)NC1C(C(=O)NC(CC=C)CC(F)F)CC1 Cc1cc(C(=O)N(CC(=O)NCC2(O)CCCCC2)CC2CC2)cnn1 N(C(=NCC(C)(C)OC(C)C)N1CCc2cccc(C)c2C1)C(CC)C c1(CNC(C2C(NC(c3c(C(C)C)ocn3)=O)COC2)=O)ccc(O)nc1 NC(=NCCCF)NC1CC1(C)C(F)F.Cc1cnc(CC)c(C)c1 N1(C(C(C)N=[N+]=[N-])=O)CCC2(CCC2)C(NC(=O)C(C)Cc2ccccc2)C1 C#Cc1cc(NC(=O)CCCCCNC(c2c(C)nn(C)c2C)=O)cc(F)c1 c1(OC)nscc1COC(c1conc1C(C)NC(=O)C(C)OCCC(C)C)=O C1(CNC(c2cnn(CCCC)c2C)=O)CN(C(=O)C2CC2)C2COCC2O1 N1(C(CS(C)(=O)=O)=O)Cc2ccccc2CC1CC(=O)Nc1ccc(C#N)nc1 C1(NC(c2n(CCC)ncc2)=O)CCC2(CCCN2C(=O)C=CS(C)=O)CC1 CC1(C)CC(NC(c2csc(-c3cnc[nH]3)n2)=O)CN(C(=O)CC=C(Cl)Cl)C1 c1(C(N(CCNC(=O)CC(C)(C)O)CC)=O)cc2c(s1)CCC(C(C)(C)C)C2 c1(OC)cc(C(=O)NC2CCCC2NC(c2cc(O)ncn2)=O)cc(Cl)c1O c1(C(C(=O)NCCCC(C)NC(=O)C(CO)NC(N)=O)=O)ccc(Cl)cc1O N1(C(C2(CC)CC2)=O)CCCC1C(C)NCCN(CC(F)F)CCO C=Cc1cnn(C)c1C(N1CCC(CNC(c2cccnc2OC(F)F)=O)C1)=O c1(N(C)CC)ccc(CNCC2CC2c2ccc(Br)s2)cc1 Cn1ncc2c(NCC3COCC3O)nc(N3CCC(F)(F)C(C#N)C3)nc12 C1(C(N2CC(N(C(=O)C(=O)C3CCCC3)C(=O)C(C)C)C2)=O)OCCC1CC C=CCCCCC(=O)NCC(O)CC(=O)N(C1CC1)CC1CC1 C(=O)(C(C)C(F)(F)F)NCC(C)(CO)NC(c1n(C=C)ncc1)=O n1(CC(=O)NCCCN(C(C2C(=C)CC2)=O)C)c(=O)n(C)c2ccccc12 Cc1cnc(C(N2CCOC(CNC(c3cnc(O)s3)=O)C2)=O)c(F)c1 C1(=O)C(C(C)C)C(=O)NCC2CN1C(C)(C)C2.C(C)(C)(C)OCC C1(C(=O)NCC(C=C)O)CN(C(=O)CC(C)C(C)C)CC(C)O1 C1(NC(CC2CCN(C(CC(C)(C)O)=O)C2)=O)CC12CCCCCC2 n1(CC(C)C)[nH]c(CC(=O)N(CC(C)NC(c2cc(Cl)on2)=O)C)cc1=O C1(C(=O)NCC(C2CC2)NC(c2ccn(CC)n2)=O)(CC2CC2)CCCOC1 C(C(C)(C)C(=O)N1CCCC(CNC(c2cn[nH]c2)=O)C1)OC Cc1cccc2c(C(=O)NC3(CNC(c4n[nH]c5c4CCOC5)=O)CC3)csc12 C1(NC(c2c(C)nc(COC)s2)=O)CCC(O)CN(C(c2cc(C)c(C)s2)=O)C1 N1(C(C(n2cc(C3CCOC3)cn2)=O)=O)CCCC(CNC(c2cnn[nH]2)=O)C1 N1(C(C2CCC(SCC)CC2)=O)CC(OC)C(C(C)C)C1.C12CC3(C1)CC3CN2 CCC1=C(C(=O)N2CCC3C(CCN3C(=O)C3=NNC(=O)C3)C2)SCCO1 C1(NC(c2c(CC)ncs2)=O)CCCCC12CCN(C(=O)CCCSC)C2 c1(C(C(=O)NCCC(C)NC(C(C=C)O)=O)(F)F)ccc(F)c(F)c1 C1(NC(=O)CCc2cnoc2)CC(C2CCN(C(c3ccnc(O)c3)=O)CC2)C1 c1(CC(=O)NC(CN(C(C(C2CCC(=O)N2)C)=O)C)C)cccc(Cl)c1 N1(C(C2C(C=C)OCCC2)=O)CC(CNC(c2conc2CC)=O)C2(CCC2)C1 N1(C(c2c(OC)c(C)sc2)=O)CCC12CN(C(=O)C(C)(C)n1cccn1)C2 c1(C(=O)NC2(CCOC)CCN(C(C3CC3C)=O)C2)nccc2c(C)cccc12 c1(C(=O)NC2C(CNC(c3cc(C)n(C)c3C)=O)CC2)cnc2ccncc2c1 C(=O)(C1=CCCCC1)NCC1N(C(C(CC)(O)c2cccc(Cl)c2)=O)C2C(C1)C2 c1(NC(c2c(C)n(-c3ccc(Cl)c(F)c3)nc2)=O)sc2ncccc2c1N Cn1ncc(C(=O)NCC(C)CC(=O)N2CCOCC2C(F)F)c1Cl c1(CN(C(=O)CC(F)(F)F)C2(CC(c3n[nH]c(=N)s3)=O)CCCC2)ccc(F)cc1 C1(NC(COCC#C)=O)CC(CNC(=O)CCc2cscn2)CC1O c1(C(N2C(C3CCN(C(C(CC)OC)=O)CC3)CCC2)=O)ncn2c1COCC2 C12(N(C(C(c3ccc(F)cc3)C)=O)C3CC3)CC(C1)N(C(C1CCCN1N=O)=O)C2 Cc1cc(OCC(N2CC(C(N)=O)(CNC(C3CC3c3ccsc3)=O)C2)=O)no1 Cc1c(Br)sc(C(=O)NCCCC2CCCCN2C)c1C c1(C2(O)CN(C(=O)NC(c3nc[nH]n3)C)C2)cccc(Cl)n1 C(CCNC(=O)C(c1ccccc1)C)(C(=O)NCCn1cncn1)OC C1(C(=O)NCCc2ccncn2)CCN(C(=O)CN2CCCC2)O1 N1(C(C2(CC#C)CCC2)=O)CCn2nc(C)c(CNC(=O)C(C)=CCC)c2C1 N1(C(C(CCCC)N(C)C)=O)CCC2CCN(C(=O)C(C)CCCC)C2C1 c1(NC(N2CC(CC)N(C)CC2)=O)ccc2c(c1)CC(C)(C)C2OC C1(NC(CC(C)OC)=O)CN(C(=O)C=CCCC(C)C)CC1C(F)F c1(NC(C2CCC(CC(=O)NCc3cnc(C)s3)CC2)=O)ccc(Br)c(I)c1 C1(CNC(=NCC)NCc2ccc(P(C)(C)=O)cn2)CC2CCC(C1)S2(=O)=O CC(N=c1cc(NC(c2ccccc2F)C)nc(C(C)C)[nH]1)c1ncn(C)n1 n1(CC)ncc(C(=O)NC23CC(CNC(c4cc(C)n(C)n4)=O)(C2)C3)c1C1CC1 CC(C)(CCNC(c1cnc2n1CCC2)=O)C(=O)N1CC(OCCO)C1 N1(C(C(C2CCC(=O)N2)C)=O)CCC(CO)C(NC(=O)Cc2cnn(C(F)F)c2)C1 N1(C(C(CCCC)NC(C23CC(F)(C2)C3)=O)=O)CCCN(CC)C(=O)C1 N1(C(c2cc(CC(C)C)nn2C)=O)CCN(C(=O)CC2CCCCO2)CC1CF c1(C(=O)NC(CC)CN(C)C(c2ccnc(O)c2F)=O)n[nH]c2c1CCOC2 C1(CC(=O)NCCCCNC(c2ccnn3ccnc23)=O)CCn2cncc2C1 C1(C)(CC)C=C(C(=O)NCC2(NC(c3cc(CCCO)on3)=O)CCCCC2)C1 c1(C(=O)NC2C(C)N(C(=O)CN3CCC(C)(O)C3)CC2)ccc(Cl)cc1Cl c1(-n2c(CC3COC(=O)C3)nc(C(C)OCC)n2)ccc(Br)c(F)c1 C1(C(=O)NCC(F)(F)C(N)=O)(CC)CCCN(C(=O)C(C)C2CC2)C1 c1(C(=O)NCCNC(=O)CN2CSCC2=O)cnc2c(Br)c[nH]c2c1 CCC(O)C(C)C(=O)NCCCCCC(=O)N(C1CCCC1)C C1(C(=O)NC(CC)C(=O)OC)CCCN(C(=O)CN(CC)CC2CC2)CCC1 CC(CNC(=O)CC1(C)CC1)CCC(=O)NC1CCC(C(N)=O)CC1 C1(C(C)C)CN(C(c2cnn3c2CCC3)=O)CCN1C(C1CCCCO1)=O S(=O)(=O)(CCC(=O)NC1CC(C(F)(F)F)(OCC)C1)N(CCCC)C1CC1 C(=O)(C(C)(CC)C(=O)N1CC(NC(=O)CNC(=O)OC)C(C(F)(F)F)C1)OCC CC1(C)CCCC(C(N2CCCC(O)(CNC(c3csnn3)=O)C2)=O)C1 C1(CC=C)(C(=O)NCCCSC)CCN(C(=O)CSc2cn[nH]c2)C1 S(=O)(=O)(c1cccnc1NCC1CCSC1)N(C)Cc1ncc(Br)cn1 c1(C(=O)NC2CC(C)(C)N(C(=O)CCC3CCOC3)C2)c(F)ccc(F)c1F c1(C(=O)NCC2N(C(CC3CCN(C)C3)=O)CCOC2)ccc2c(cnn2C)c1 CC1CN(C(=O)Cc2ccc3c[nH]nc3c2)CCCN1C(=O)CC1CCOC1=O Cc1cc(C(=O)NC(C(=O)N(CC(C)CO)C)c2cccs2)n(C)n1 C1(OCC)CCCCCC1NC(=O)CC1CCN(C(c2cc(C)ns2)=O)C1 C(CCN=C(NCC(=O)Nc1cc2c(s1)CCC2)NC1Cc2ccccc21)SC c1(C(N2CC(CN(C(=O)CCc3ccncn3)C)C2)=O)ccc(F)cc1[N+](=O)[O-] C1(NC(CN(C(=O)C(C2CC2)C2CC2)CCC#C)=O)CC(N2CCCC2)C1 C(C(C)C(C)C(=O)N1CCN(CC(C)(C)NC(c2ccc(F)cn2)=O)CC1)OC CCCC(CC(C)C)C(=O)N1CC2(CCN(C(=O)C=C3CC3)C2)C1 c1(C(=O)NCC2CC(NC(C(C(C)C)C)=O)CC2O)ccc(F)cc1[N+](=O)[O-] N1(Cc2c(Br)ccc(OC)c2C#N)CCc2c(-c3sc(-c4nn[nH]n4)nc3C)csc2C1 c1(C(c2n(C(CC)C)nnn2)NCCn2ccnc2C)c(F)cccc1F CCC(CNC(C1CCN(C)C1C)=O)(CC)C(=O)NCCC(C)SC N1(C(c2ccc(OC)s2)=O)CC(NC(c2c[nH]cc(C)c2=O)=O)CC(C)C1 C1(C(=O)NC(c2ncccn2)CC)CN(C(C2(C#N)CCCO2)=O)CC1(C)C c1(C(=O)NC(C2CN(C(c3c(CC)occ3)=O)C2)C)ccccc1P(C)(C)=O C1(NC(C(CC)=CC)=O)CCN(C(=O)C(C)N(CC(F)(F)F)C)C1C C1(C(C)C)(C(=O)NC2CCCC2CNC(=O)Cn2cnnc2O)CNC(=O)C1 c1(CCC(=O)C(C2(OC)CC2)=O)cccc(Br)c1.C(C)(CC(C)N)N Cc1cc(C#N)sc1C(N1CC2CC1C2NC(C1(C)CCN(C)CC1)=O)=O N1(C(Cc2ccn(CC)n2)=O)CC(=O)NCC1C(=O)NCC1CCCS1 C1(NC(C(C2CC2)OC)=O)(CF)CCN(C(=O)C(C)Cc2ccco2)C1 C1(COC)CN(C(=O)CC2(O)CCCN(C)C2)CCN1C(=O)CCCNC(C)=O CCC(C)(C)C(=O)C(=O)NC(CC1CCC1)C(N1CC2(C1)CN(C)C2)=O Cc1ncc(NC(=O)CCC2CCCCN(C(c3c[nH]nc3Cl)=O)C2)cc1Cl Cc1occc(=O)c1OCC(=O)NC1CN(C(=O)C(O)C(F)F)CCC1CO CC1CC2(CCN(c3nc(N4CC5CC5C4)c4sccc4n3)CC2)C(=O)N1 C12(NC(C3CC(NNS(C)(=O)=O)C3)=O)CC(CNC(CC(C=C)C)=O)(C1)OC2C C1(C(=O)Nc2cccc(CNC(=O)CCc3ncc[nH]3)c2)CCC(F)(F)CC1 N1(CC)CCC(NC(=O)N(CCC(N)=O)C(c2ccccc2)CO)C1 Cc1[nH]ccc(=NC(=O)C2CC(O)CCN2Cc2ccc([N+](=O)[O-])s2)c1F c1(C(CC)O)nc(C2CC(C(C)(C)C)CCO2)n(CCOc2ccccn2)n1 CCCCC(F)C(=O)NCC1CC2(CC2)CN1C(c1ncc(F)cc1F)=O N1(C(CCC#C)=O)CC2CC1CCC2NC(=O)C=Cc1ccccc1Br C1(C)(C(N(C2CCN(C(=O)CCNC(C)=O)CC2)CCC)=O)CCCS1(=O)=O CC1(C(=O)NCC=CCNC(=O)C(F)OC(F)(F)F)CCCOC1 Cn1ccnc1C1CC1C(=O)NCC(C1CCCCC1)NC(C1CC1CF)=O Cc1ccc(Br)c(C(=O)NC(C(C)NC(c2c[nH]nc2C)=O)C(C)C)n1 C12(C(=O)NCCN(C(c3ccc(C(C)C)cn3)=O)C)CCCCC1OCC2 C(CC(C)CCNC(c1cncc(C2CC2)c1)=O)NC(C(COC)NC(N)=O)=O CS(=O)c1cccc(C(=O)NC2CC(CNC(=O)C=Cc3ccncn3)C2)c1 c1(C(=O)NC(CNC(C(CC(C)C)(F)F)=O)CO)cnn2c(Cl)cccc12 Cc1nc(=NC2CCC3CN(C(c4ccnn4CCF)=O)CC23)s[nH]1 C(C(C(=O)NC1CC1CNC(C1(OC(C)C)CCC1)=O)c1ccccc1)SC Cc1ccc(C)c(CN2CC3(CN(C(C4CC(=O)N(C(C)C)C4)=O)C3)C2)c1 C(=O)(C(F)(F)C(C)(C)O)N1CCC(CNC(CCCC(=C)C)=O)(OC)CC1 C=C(C)C(O)CC(=O)N(C1CCCN(C(=O)Cc2sccc2C)CC1)C N1(C(C2CCCN(C)C2)=O)CCCN(CCNC(=O)CC(C)(F)F)CC1 N1(C(CN2CCC(C)C2)=O)CCN(CCNC(=O)CC(=O)OC(C)(C)C)CC1 N1(C(=O)OC(C)(C)C)CCCC(C)(CNC(=O)C(C)(C)CCCl)C1.C1CO1 C(N=c1[nH]c(Cl)ncc1F)C1CCN(C(=O)C=CCn2cncn2)C1 c1(CNC(C2(F)CCN(C(=O)CSc3nn[nH]n3)CC2)=O)c[nH]c2ncccc12 C1(NC(Cc2ccc(C)cc2)=O)CCSC12CN(C(c1cnc(S)[nH]1)=O)C2 N1(C(c2c(C)nc(O)cc2)=O)CCC(C)(C)C(C(=O)NOC(C)(C)CO)C1 CN1CCOC(C(=O)NCC2CN(C(c3scnc3C(F)F)=O)CC2O)C1 Cc1cccc(C(CNC(=O)Cc2nccn2C)NC(c2ccncc2F)=O)c1 C1(OC)CC(F)CN(C(C2CC(CNC(=O)C(O)c3ccsc3)C2)=O)C1 C12(C(=O)NCc3nc(CNC(C(CSC)C)=O)sc3)CCC(CC1)CC2 Cc1cnnc(O)c1C(=O)NCCN(C(=O)COC1CCOC1)CC1CCCC1 C1(CNC(C(CC)O)=O)CN(C(c2cc(C)c(CO)cn2)=O)CC(C)(C)O1 N1(C(CCN(C)C)=O)CCCC1CNC(C1CCOC1)=O c1(C(N2C(CNC(CN(C3CCSC3)C)=O)CC(O)C2)=O)cc2nc[nH]c2cc1F C1(CNC(c2c(CC)con2)=O)CC(COC)CN1C(c1cn(C)nn1)=O C1(O)(C(C)NC(CNC(=O)NC)=O)CN(C(=O)Nc2ccn(C)n2)C1 C1(C(N2C3CC(CNC(CSCC=C)=O)C(C3)C2)=O)Cc2ccccc2NC1=O C1(NC(=O)NC2C(C)CCC2)CCN(C(=O)OC(C)(C)C)CC1 c1(CN2CCN(CC(=O)Nc3c(C)ccc(O)c3)CC2)ccc(F)c(F)c1Cl N1(C(CCCN(C(C)=O)C)=O)CCC(NC(c2n[nH]cc2Br)=O)CC1C C1(CNC(=O)Cn2nnc(=O)[nH]2)CN(C(=O)CC2CC2(Cl)Cl)CC1O C(=O)(C1=NN2CCC(C)N=C2N1)NCCN(C(c1ccc(CC)c(Cl)c1)=O)CC C1(NC(c2cnc(C)[nH]2)=O)C2CC3CN(C(c4ccccc4Cl)=O)C1C3C2 C1(C(N2CCN(C(CN3C(C)CC3)=O)CC23CC3)=O)COc2ccccc2O1 N1(C(c2ccc(OC)cc2)=O)CC2(CNC(=O)C(C3CCCO3)OC)CCC1C2 C1(C(=O)OC)CC2(CCC2)CO1.C1(C)CCC(=O)N(C2CC2)CC2CCCN12 C1(C(=O)NCCOCCNC(c2cnc(CCCC)s2)=O)CCCCC1C1CC1 C1(N(C)C)CCCN(C(C2CCC(NC(C3CCCO3)=O)C2)=O)C1 c1(C(N2CCN(c3cccs3)CC2)C(=O)NCC=C)ccc(CC)c(F)c1 C1(C(N2CC(OCC(=O)NC(C3(O)CN(C(N)=O)C3)C)C2)=O)CC1C1CCCC1 c1(NC(c2ccc(-c3cc(C)c(F)c(F)c3)nn2)=O)c(Cl)cccc1[N+](=O)[O-] C=CCC(C)C(=O)NC1CCN(C(c2ccc(-c3cnco3)cc2)=O)C1C1CC1 Cc1cc(C(N2CC(CNC(=O)CCCCCF)C(F)(F)C2)=O)c(Cl)cc1F C1(NC(C(C)NC(N)=O)=O)CC2CCC(C1)N2C(C1CC12CC2)=O C1(NC(COCC#C)=O)CCCCCCC1NC(=O)C(C)CSC N1(C(c2c(CC)c[nH]n2)=O)CC2CCC1CN2C(c1cnc(C(C)OC)s1)=O C=CC1CCCC(N=c2ccnc(NCc3ccccc3C3CC3)[nH]2)C1 CC(CC(=O)NCC1CCN1C(=O)CCNc1ccccn1)N(C)C C(=O)(C(O)CC(N)=O)NCC1(OC)CCN(C(=O)C(C2CCOCC2)O)C1 C12(C(=O)OCC)CCCC1CCN2CC1CC1c1ccsc1 Cc1ncc(Cl)c(C(=O)NCCC2(CNC(=O)CCC(C)(F)F)CC2)n1 Cc1cn(CC(=O)N(C(C)CN(C)C(C2(C(N)=O)CC2)=O)C)nc1C(F)F N1(C(c2c(CC)nc[nH]2)=O)CC2CCCC(C1)N2C(=O)C(C)OC Cc1cc(C(=O)NCC(C)N(C)C(c2cnsc2)=O)c2c(C)noc2n1 Cc1noc(-c2cn(CC(N3CC(C)(NC(=O)Cc4cccn4C)C3)=O)cn2)n1 c1(CCC(N2CCC(NS(CC(=O)OCC)(=O)=O)CC2)=O)ccc(C)c(C)c1 C1(CCC(=O)NC(CC)CN(CC)CC)CCN(C(C2COCCO2)=O)C1 N1(C(c2nc(CC)sc2Br)C(=O)NC2CCOCC2)CCOC(C2CC2)(CC)C1 N1(C(c2nccc(OC)c2F)=O)CCCC12CCN(C(c1ccc(O)nc1)=O)C2 C1(CC)CC(C(=O)NC(c2nn[nH]n2)C2CC2)CCN1C(c1cc(F)cc(F)c1)=O c1(C(=O)NCC(C)(F)CNC(C2CCCCCCC2)=O)cnc2ncccn12 c1(C(N2CCC(O)(C(CNC(CSCC)=O)C)C2)=O)cc2c(=O)[nH]ccn2c1 C=CC(F)(F)C(=O)NCCC1(CNC(c2c(Cl)n[nH]c2C)=O)CC1 CC1CCCCCN1CCNC(c1ccc(OC2CC2)cc1)=O c1(CCC(N2C(C(C)N(C(=O)C(N)=O)C3CC3)CCC2)=O)ncc(C(C)(C)C)o1 N1(CC(=O)NC(C)CCNC(=O)CC2CCCN(C)C2)CCN(C)C(=O)C1 C1(C(=O)NC(C)CNC(C23CC(F)CC(F)(C2)C3)=O)Cc2cc(Cl)ccc2O1 c1(C(N2CCC(N(C(=O)CC3CCCC3)C)C2)=O)cnc2c(c1)CCCC2 N1(C(=O)Oc2ccccc2)CC2(CCC(NCc3ncc(N(C)C)nc3)C2)C1 c1(C(N(CCC)CCNC(C2CCCSC2C)=O)=O)ccc2c(c1)CCCC2=O N1(c2n(CC(C)C)c(CSC3C=CCC3)nn2)CCCC2CC1C2(C)C NC1(C(=O)NCc2cn(CCO)nn2)CCC2CCCC12 c1(C(c2n(C(C(=O)OC)C)nnn2)NCCCCC2CC2)ccc(C#N)nc1 N1(C(=O)CSCC(F)(F)F)CC2CCCC2(Nc2ncnc3c2CCO3)C1 N1(C(c2cnc(-c3ccccc3)[nH]2)C(=O)NCCCSC)CCOCC1C#N c1(C(N(CC(CC)NC(c2ccccc2OCC)=O)C)=O)cc(OC)cc(Cl)c1 C(C(C)C(=O)NC1CC(C(C)O)C1)NC(C(C)OCCCC)=O c1(C(=O)NCC(CNC(=O)CCC(=O)c2cccs2)F)cncc(F)c1Cl CC1CCC(C)(C(=O)NCCCCC(=O)N2CC(C(C)(C)C)C2)C1 c1(C(=O)NC(C)CNC(c2cscc2Cl)=O)ccc(N)c2ncccc12 N1(S(C)(=O)=O)CCCC(C(=O)NC2CCC(NC(C3CC(C)(O)C3)=O)CC2)C1 N1(C(=O)OC(C)(C)C)CCCOC(CNC(C2(CCF)CC(O)C2)=O)C1 N#CC1(C(=O)NCC(O)CNC(=O)CC2C=CCCC2)CC12CCOCC2 CCC(C)(COC)C(=O)NC1COCC1C(=O)NCC(=O)N(CC)OC C(=O)(CCCN=[N+]=[N-])N1CC(C(C)NC(Cc2cccc(OC)c2)=O)OCC1 C1(C)(C(=O)NC(C)CNC(C2(Oc3cccnc3)CC2)=O)CCCOC1 c1(C(N2CCC(C)C(CNC(=O)CSCCN(C)C)C2)=O)cc2ncccc2[nH]1 Cc1ccc(NC(CNC(=O)C(C2CCCCC2)O)C(C)C)cc1N C12(C(N3CC(CNC(c4cc(C)oc4)=O)OCC3)=O)CC1COC2(C)C C1(NC(c2cnc(C)nc2)=O)COCCN(C(=O)Cc2ccc(Br)cc2I)C1 c1(C(N(CCOCCCNC(CCC(=C)C)=O)C)=O)cc(CC)ccc1F N1(C(C(CCOC)C)=O)CC2CC(NC(=O)Cc3cscn3)C1C2 N1(C(c2c(C)scn2)=O)CCC(c2n[nH]c(CNC(=O)C(C)(C)C)n2)CC1 CCCCCCC(C)NC(C1(F)CCCN(C(C2(O)CCCCCC2)=O)C1)=O c1(C(=O)Nc2c(C(N3C4C(C(=O)OC)C(C4)C3)=O)nc[nH]2)c(F)cc(Br)cc1F CC1(P(C)(C)=O)CCCN1C(c1c(SCC#N)cccc1)=O Cc1cc(Br)ccc1C(N1CCOC(CC(=O)NCC2(C)CCCC2)C1)=O S(=O)(=O)(c1ccc2nc(O)[nH]c2c1)N1CC(N(c2nc3ccc(C)nc3s2)C)C1 C=CCCC(CO)NC(c1cnn(CCNC(=O)CCC2CCC(C)O2)c1)=O c1(OC)ncc(Cl)cc1NC(N1CCC1C1CCCOC1)=O CCC(C)(C#N)C(=O)NC1CCCN(C(C2(c3ccc(OC)cc3C)CC2)=O)C1 N1(C(=O)NCC(=Cc2ccccc2)C)CCN(C2CCCC(C)C2)C(C)C1 CC1Cc2cc(CC(=O)NC3CC4CC(NC(=O)C=CCF)CC34)ccc2O1 Cc1ccc(F)cc1CNC1COC(c2ccccc2)C1 Cc1c(C(N2CCC(CCC(=O)NCC(F)C(C)(C)O)CC2)=O)cccc1C#N N1(C(c2c(OC)cccn2)=O)CC2(CCN(C(c3c(OC)ncnc3C)=O)CC2)C1 CCC(C)(C#N)C(=O)N1CCC(O)C(N(C(=O)Cc2ncn3c2CCC3)C)C1 n1(CCC#C)cc(CN2CCC2C(N)=O)cn1 Cc1nc(NC(N2CCC(n3cnc(C(N)=O)n3)C2)=O)nn1-c1nc[nH]n1 CCC(F)(F)CC(=O)NC1CC(NC(C2(SC)CC2)=O)C12CCC2 c1(OC)cc(C=CC(=O)NC2CN(C(=O)C(C)O)CC(F)(F)C2)ccc1O N1(C(C(C)Cn2cccn2)=O)CCC12CN(C(C1CC1)=O)C2.c1(C(O)CC)csc(=N)[nH]1 c1(C2(C(N3CCC(CCCc4nc(CCC)on4)C3)=O)CC2)ccccc1F N1(C(C(CSC)O)=O)CCCC(CN(C)C(c2cc(C)sc2C)=O)C1 Cc1cnc2nc(C(=O)NC(C3CCOC3)CNC(=O)CC(F)(F)F)nn2c1 C(CN=c1[nH]c(=NCCCC2CCCC2)c2ccccc2[nH]1)OCC c1(CC(=O)NC2CC(NC(C(CC)OC3CCCC3)=O)C2)cccc2sccc12 n1(CC(=O)NC(CCC)CNC(=O)CCOCCC(C)C)nc(C)oc1=O N1(C(c2cc(CC)n(C)n2)=O)CCCC(F)(C(=O)NC2CN(C)NC2=O)C1 c1(C(N2CCC(O)(C(CNC(c3c(C)coc3)=O)C)C2)=O)cnc2[nH]ccc2n1 C(C)(C)(CCC(=O)NC1CCC1C1CC1)NC(C)=O N(C1CC(NC(=O)C(O)CCSC)c2ccccc21)c1nccc(OCCC)n1 c1(C(N2C(C(=O)Nc3cc(OC)ncc3F)CC(O)C2)=O)ccc([N+](=O)[O-])cc1C c1(CN2C3(CCC3)CC2=O)conc1C.C1CC1.CCO Cc1ncnc(C(=O)NC2C3CCC2N(C(=O)C(C)OCC2CCCO2)C3)c1C C(=O)(CCCC(N)=O)N(CCCCN(C)C(C1CN(C(=O)OC(C)(C)C)C1)=O)C C1(C(=O)NCc2c(OC)c(C)ccc2)CC12CCCc1ccccc12 N1(C(CN2CC(NC(=O)C(=O)NCC(O)CC(F)(F)F)C2)=O)CCc2ccccc21 c1(-c2nnccc2)nc(C(C)Cn2cncn2)n(C2CC(C(F)(F)F)C2)n1 Cc1ccc2c(C(=O)NCCC(C)(C)NC(c3coc(N(C)C)n3)=O)c[nH]c2c1 c1(N2C(CC)CN(Cc3ccc(C)s3)CC2)ncc2[nH]ncc2n1 Cc1nc(C(=O)N(C)CC2CCCC(NC(=O)CC(C)(C)C#N)C2)c(=O)[nH]c1C C1(CC=C)(NC(=O)COC2CC(F)(F)C2)CN(C(=O)C(C2CCOCC2)C)C1 C#CCCCCCC(=O)N(CCCNC(c1coc(-c2ccsc2)c1)=O)C N1(C(C=Cc2ncc(C)[nH]2)=O)CC2CC(C1)N(C(=O)COc1ccccc1F)C2 N1(C(c2c(CC)csc2)=O)CCC2CN(C(=O)C=CCOC)CC12 c1(CC)cc(C(=O)N(C2CCN(C(C3CCS(=O)(=O)N3)=O)C2)C)ccc1C c1(OC)sc(C(=O)NCCC(C)NC(=O)C(O)CCSC)cc1Br CC1(O)CCN(C(C2CN(C(C3CCN(C(=O)C4CC4)CC3)=O)C2)=O)CC1O C(=O)(C(CC(C)C)C(C)C)OC.C1CN=C2NN=C(S2)CC(=O)N2CCCC1C2 C(=O)(C(C)CC(=O)NCC1CC1CC(=O)NCc1c(C)n[nH]c1C)OC c1(C(=O)NC(C(=O)N(C)Cc2nnc(C)s2)CN(C)C)cccc2c[nH]nc12 C1(C(NOCC(=C)C)=O)C2CN(C(C3CC3F)=O)CC12 Cc1ccc(C(N2CCOCC(NC(c3cc(C(C)(C)C)n[nH]3)=O)C2)=O)c(C)n1 c1(C(N2CCN(C(Cc3cc(C)sc3C)=O)C3C2C3)=O)cccc2oc(=N)[nH]c12 N1(C(C(C)O)=O)CC(CCNC(c2ocnc2C(F)(F)F)=O)C(C)C1 c1(C(=O)NC2CC3CCC2N(C(=O)C(F)F)C3)c[nH]c2ccc([N+](=O)[O-])cc12 c1(C(=O)NC2C(n3cc(C(C)O)nn3)COC2)cccc2ncnc(O)c12 c1(CC(=O)NCc2ccc(C(C)C)cc2)cccc(Br)c1F C#Cc1cc(C(N2CC(NC(C3CC(C)(C)C3)=O)C3CCCC23)=O)cc(Cl)c1 C1(NC(CSCCN(C)C)=O)CC2(CCC(NC(=O)C(F)=C3CCC3)CC2)C1 Cc1cc(Cl)cc(C(=O)NCCC2CCN(C(c3cccnc3S)=O)C2)c1C N1(C(C=CC(=O)OCC)=O)CCC2(C(=O)NCC(C)(C)CCCCC)CCCC12 N1(CCC=CCC)CCN(C(c2ccc(Cn3ccnn3)o2)=O)C2CC12 C#CC1CN(C(C2CC(=C3CC3)C2)=O)CCN1C(c1cccc(CCC)c1)=O C1(CC(=O)OC)CN(C(=O)C(=O)Nc2c(C)cc(C)cc2C)CC(C)(C)O1 c1(C2C(C(N3CC(CC(C)NC(CC(C)(C)OC)=O)C3)=O)C2)c(Cl)cccc1Cl CCCCC(CN=c1[nH]c2cc(Br)cnc2s1)NC(=O)C(C)C1CCCO1 C=CCC(C)(C)C(=O)N1CCC(CCNC(=O)CC2CCCC(C)C2)CC1 c1(C(N2CCN(C(CCCCCSC)=O)CC(O)C2)=O)cc2n(c(=O)c1)CCS2 N1(C(C(C)OCCCC)=O)CCOCC1C(=O)NC(C)CC(=O)OCC C(=O)(C1=C(C#N)CCC1)N1C(CCCNC(CC2(OC)CCCC2)=O)CCCC1 C1(C2CCN(C(C3CC3C3CCCC3)=O)CC2)(NC(C(CC)=CCCC)=O)CC1 c1(C(N2CC(CO)CC(C)C2)C(=O)NCC)ccc2n[nH]cc2c1 c1(C(=O)NCC2CCCC2NC(C23CC(C(F)F)(C2)C3)=O)ccccc1[N+](=O)[O-] c1(C(=O)NCC2(NC(CC3C(C)=NOC3=O)=O)CC2)ccc2nc(CO)[nH]c2c1 N1(C(c2ccc(C)cc2)C(=O)NC)CCC2(CCCCCC2)CC1 C1(CNC(C2(CCC)CCC2)=O)CCCN1C(C1CC1c1ccnn1C)=O c1(C(=O)NCC2(NC(=O)C(F)F)CCCC2)ccc(OC(F)F)c(Cl)c1 C1(NC(C2CCCO2)=O)(CF)CCN(C(=O)CCc2nccs2)C1 Cc1cnccc1-c1ccc(C(=O)NCCC2CC(N3CC(O)C3)C2)s1.C(=O)N C(=O)(C1CCCn2nccc21)NC(C)CCCCNC(C1(O)COC1)=O N1(C(=O)Cc2cc(Br)cs2)CCCC(C2CN(S(=O)(=O)CC3CC3)C2)C1 C1(F)(CNC(=O)Cn2nccn2)CC(NC(C2CC2F)=O)C1 C1(NC(c2occ(C)c2)=O)CN(C(=O)C(C)NC(C)(C)C)CC12CCOCC2 N1(C(CCSC)=O)CCC(C2CC2)C1C(=O)Nc1nc(C)ccc1I c1(C(=O)NCC23C(CN(C(C4(CC)CC4)=O)C2)C3)cc(F)c([N+](=O)[O-])c(F)c1 C(CC(C)(O)C(=O)N1CCC(Cn2cc(CC(C)(C)O)nn2)C1)N(C)C N1(CC(=O)NC2CCN(C(CC=C=C)=O)C2(C)C)CCCCC(OC)C1=O C1(C(N2C(C)(CNC(=O)Cc3ncc(C(F)(F)F)[nH]3)CCC2)=O)CCCCC(=O)C1 c1(C(=O)NCC(C)(O)CNC(=O)C2=CCCS2)ccc(Br)cc1OC(F)F N1(C(Cc2ccn(C)n2)=O)CCCC2(CCN(c3nc(Cl)c(C#N)s3)CC2)C1 C(c1ccco1)=C(C)C(=O)N(C1CCN(C(C2CCCN2C(=O)C2CC2)=O)C1)C CCCCS(=O)(=O)CC(=O)NCCC1CN(C(=O)C(CCO)N(C)C)CC1C c1(C(=O)NC2CC(C)N(C(=O)Cc3cccnc3Br)C2)ccc2c(c1)CCN2 c1(C(N2CC3CCCC3(CSC)C2)C(=O)NCCCSC)cccc2sccc12 C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1(CNC(C(C)=C(CC)C)=O)CC12CCC2 CC(C(CO)NC(C1(C)CCC1)=O)NC(C1(C)C=CCC1)=O N1(C(COCCCC)=O)CCCCC1CCNC(=O)C(CCO)N(C)C C1(NC(=O)NC2(Cc3ccc(C#N)cc3)CC2)CCOCC12CCCC2 C(=O)(CC(O)CCCC)NC1(CC=C)CN(C(=O)Cc2cccc3c2OCO3)C1 C1(C2N(C(=O)CCC3CCCC3)CC2)CCN(C(c2cnsn2)=O)CC1 c1(CC)nc(C(=O)N(C(C)C(=O)NC(CO)C(C)O)C)co1 CC1CC(NC(=O)Nc2cccc(N(C)C(N)=O)c2)CN1C1CC1 C(C)(C(C(=O)N1C(C(=O)NCC2CSCCO2)CCC1C)N(C)C)OC C1(CCOC)CCN(C(C2(CCOC(c3coc(C(F)F)c3)=O)CC2)=O)CC1 C(c1cnc(O)nc1C)=CC(=O)NC1CCN(C(CSCC(=O)OC)=O)C(C)C1 C(=O)(CCCCC(=O)OC)NCC(CC)NC(=O)CCc1cnc(C)nc1O c1(C(C)NC(C2C(C(N3CCC(CC(=O)OC)CC3)=O)C2)=O)ccc(F)c(F)c1 c1(C(=O)NCC2C(NC(C(C=C)(C)C)=O)CCCC2)cc2oc(Br)cc2[nH]1 O(P(=O)(CNC(=O)NC(C1CCCCO1)C1CCC1)OCC)CC C1(CNC(C(Cc2cn(C)nc2)O)=O)CC2(C1)CN(C(=O)CSC1CC1)C2 C=C(C)C(CC(=O)N1CC2(NC(=O)CCSc3nnnn3C)CCC1C2)OCC c1(CNC(=O)OCC)cc(=NCc2ncc(C(=O)OC)s2)[nH]c(C(F)F)n1 N1(C(=O)CN(C2CC2)CC2CCCCO2)CCN(C(=O)CC23CCCC2C3)CC1 CC1CC(c2ccoc2)CN1C.c1(O)ccccc1C(c1ccccc1)=O c1(NC(=O)Nc2scc(C3C(CCC)C3)n2)ccc2c(C)[nH]nc2c1 CC1CN(C(=O)CC2CCCC3CC23)CC(C(N2CC(CC34CC(C3)C4)C2)=O)O1 C1(C(N(C)CCOCCNC(c2csc(CO)n2)=O)=O)CCc2[nH]nc(O)c2C1 C(C(C)(C)C(=O)N(C)CCc1ncon1)N(C(C(CC)n1cncn1)=O)C N1(C(C(C)=C2CCCC2)=O)CCC(C)(CNC(c2coc(C(F)(F)F)n2)=O)CC1 n1(CC)cnc2c(N(CCCC(C)C)C)[nH]c(=NCC3CC4CCC(C3)S4)nc12 N1(C(Cn2c(=O)ccc(C)n2)=O)CCN(C(=O)CCCCCF)C(C)CC1C c1(CN2C(=O)NCC2CCNCC(c2ccco2)O)cc(Cl)ccc1OC(F)F c12scnc1CN(CC1CCCO1)C2=O.C(C(C)CNC)N(C)CC C1(C(CNC(C(CC)OCC)=O)F)CCN(C(=O)C=Cc2ccsc2)CC1 c1(NC)ccc(C(N2CCCN(C(c3snc(Cl)c3Cl)=O)CC2)=O)cc1F c1(C(N2CCCC(C)(NC(c3c(CC)cccc3)=O)C2)=O)cccc2nonc12 C12(C(=O)NC3(C(C)O)CC3)CC1CCN2C(c1ccnnc1)=O C(=O)(CCCC(F)(F)F)NCCOC1CCN(C(C(C)Cn2cccn2)=O)CC1 C1(CCNC(C=C(C)C)=O)CCN(C(=O)C(N2CCC(C)C2)=O)CCC1(F)F C(=O)(C1COc2ccccc21)N1CCN(C(COCCC)=O)CC(O)C1 C(CCCCC(=O)NC(c1ccnn1C)C(N1CCC(n2cncn2)C1)=O)OCC c1(C(=O)NC(CCCC)CNC(=O)CN2CCCC2C)cc2ccnc(Cl)c2[nH]1 n1(CC#C)cccc1C(=O)NC1COCC1NC(c1nnc(C(C)(C)C)s1)=O C1(CC(N2CC(O)(C(C)NC(c3ccc(=O)oc3)=O)C2)=O)CCC(F)(F)CO1 C1(C(C(=O)N(C(COC)COC)C)F)CCN(C(=O)C(C)=C(C)C)C1 N1(C(C(C(CC)O)(C)C)=O)CCC(C2(NC(c3cocc3C)=O)CCC2)CC1 Cc1nsc(NC(=O)COc2ccn(C)n2)c1C#N N1(C(c2ccc(CO)o2)=O)CCCC(CC(N2CC(CO)C(O)C2)=O)C1 CC1(C)CCC(C(=O)NCC2(O)CCN(C(C3CCCC(C#N)C3)=O)CC2)CO1 C12(C(N(CC(C)SC)C)=O)CC1CCN2C(=O)CCC1CCC1 C1(N(C(C(C)(C)OC)=O)C)CCN(C(=O)CC2(OC)CCOCC2)CC1C C(CCCCC(=O)NCC1CCN(C(C2CC=CC(O)C2)=O)C12CC2)OC c1(C(C)(C)C)cccc(C(=O)NCC2CC(NC(=O)CCCC#N)C(O)C2)n1 N1(C2CCN(C(c3ccc(O)nc3)=O)CC2)C2CCC1CN(C(C1CCO1)=O)C2 c1(N2C(=O)CC(=O)NC(=O)CC2)ccc(C)c(C)c1.c1(CC)nc[nH]c1NC C1(C(=O)NCC(C2CC2)NC(=O)CCOCC(F)F)CN2CC3CC2(CO1)C3 C1(C(=O)NC(CNC(CCOC(C)C)=O)(C)C)CCN(S(N)(=O)=O)CC1 C12(c3onc(CC(n4nc(C)c(Cl)c4)(C)C)n3)CC(CN(C(C)(C)C)C1)C2 N1(C(C(CC)N(C(=O)OC(C)(C)C)CC)=O)CCc2nc[nH]c(=O)c2C1 C#CCCCCCC(=O)N(CC(C(=O)N(CCCO)C)OC)CCCO C(=O)(C1=CCC(F)(F)CC1)NCCC1(CNC(C2CN(CC)C(=O)C2)=O)CC1 CCC(C)CCCCC(=O)NC1CCC(F)(CNC(=O)CN(C)C(=O)OC)C1 n1(CCC(N2CCC(CC)(CC)CC2)=O)ccc2cccnc12 c1(N(C)CC2CC(SC)C2)cc(C)[nH]c(=NCCN(S(C)(=O)=O)C)n1 c1(Cn2cc(-c3c(OC)cccc3C(=O)OC)nn2)cc2c(ncn2C)s1 Cc1ccc(=O)n(CC(=O)NC2CC2NC(C2(C)CCN(C)C2)=O)n1 C1(C(=O)NCc2c(N(C)C)cccc2)CC(F)CN(C(c2cnsn2)=O)C1 c1(CC(N2C(C(C)NC(c3n(CCC)ncc3)=O)CCC2)=O)cccc(C)c1Cl c1(CC(=O)OC)cccc(-c2cccc(C(=O)OC)c2)c1.N12CCOC(C1)C2=O c1(C(=O)NC(C)CNC(c2cccn2Cc2cccnc2)=O)nc(=N)cc[nH]1 C(CC(C(=O)NCC1CC1Cl)NC(c1cc(C(N)=O)[nH]n1)=O)OC c1(C(N2CCC(C(F)C(=O)NC3CC(F)C3)C2)=O)ccnnc1O c1(CNC(=O)CN2CC3CC3C2)nc2c(s1)CN(C(=O)CCn1cnnn1)CC2 N1(C(c2n(CC)ncn2)=O)CCN(C)C(CNC(c2ccc(=O)n(O)c2)=O)C1 N1(C(C2C(CCC)C2)=O)CCOC2(CCC(NC(C3(Cl)CC3(F)F)=O)CC2)C1 C1(C(=O)NCC(CNC(CSc2cccc(OC)c2)=O)CO)COCCC1(F)F c1(CC)ccc(C)cc1C(=O)N(CC(C)NC(=O)CC1CCCCC1O)CC CC1CCN(C(=O)CCC2CCN(C(c3cocc3C(N)=O)=O)C2)CC12CCC2 N(C1CCCc2cnn(CC(=O)OC)c21)C(=O)Oc1cccc(COC)c1 C(=O)(CC(CC)C(C)C)NCCN(CCC)C(c1cc(C)oc1C)=O Cc1cc(=N)[nH]c(=NCCCc2ccc(C(=O)OC(C)(C)C)cc2)[nH]1 CC(C)(C)C(CC(=O)NCCNC(c1ccc(C(F)(F)F)c(N)c1)=O)C(F)F c1(C(=O)NCCC2(NC(=O)C=CC3CCC3)CC2)ccc(=O)n(CCO)c1 c1(CNC(C2N(C(CC3CC(=O)C3)=O)CC2)=O)cccc(Cl)c1 c1(C(=O)NC(CNC(COCC=C)=O)C(C)C)c(C)nn(-c2ccccc2)c1Cl N1(C(C(C)S(C)(=O)=O)=O)CCN(C(=O)Cc2cnc(C3CC3)[nH]2)C2(CC2)C1 C(C)(CC(C)NC(c1coc(CS(C)(=O)=O)n1)=O)NC(C(C)=C1CCCC1)=O C1(NC(C2C(NC(CCN(C)C)=O)CCO2)=O)CCC(F)(F)C1 c1(C2(NCc3cn(CC(C)O)nn3)CC2)ccc2c(c1)CCCO2 c1(NC(c2nnc(CO)s2)C)cc(S(=O)(=O)N(C(C)(C)CCO)C)ccc1C#N C=C1CCC(C(=O)NCC2(O)CC(C(N3CCC(C)(O)C3)=O)C2)CC1 CC1C(NC(=O)Cn2ncnn2)CC2CCC1N2C(C1(F)CCC(=O)CC1)=O C=CCCCCCCC(=O)NC(CO)C(N1CCc2cncnc2C1)=O CCC(C(=O)NCCC(=O)N(C)C1CC1)N(C)C(C1CCC(=O)O1)=O c1(N2C(C)CC(CNC(c3c(C)noc3C(F)F)=O)C2)ncnc2c1SCCC2 c1(OC)cc(N)c(F)cc1C(=O)NCC(C)N(C)C(c1occ2c1CCCC2)=O C1(C(C(=O)NC)N(C2CCCN(Cc3ccccn3)C2)CCO)CCCOCC1 c1(C(=O)NCC2(NC(CC3CCCC(C#N)C3)=O)CCC2)nc2c(s1)COCC2 n1(CC(=O)OCC)cc(NC(C)(Cc2cn[nH]c2)C(=O)OCC)c2ccccc12 C1(C(=O)NC(CCC)CO)CCCCC1C(=O)Nc1ccc(-n2cncn2)cc1 N1(C(=O)CC2CCCN2Cc2cncnc2)CCC2(CCCOC2)C1 N1(C(C(C)CN2CCOCC2)=O)CC(CNC(=O)C(F)=C2CCCC2)C(C)(C)C1 CCC(C)(O)C(=O)N(C)CC1CCCCN1C(c1csc(COC)n1)=O C1(NC(C2(COC)CCCC2)=O)CCC(CNC(C2(C)CC3CC3C2)=O)CC1 C1(CNC(c2cc(F)n[nH]2)=O)CCN(c2nnc(C(F)(F)F)s2)CCC1(F)F Cc1cccc(C(=O)NC(C)(CNC(=O)C(F)=CC2CC2)CO)c1Br c1(CSC)ccc(C(=O)NCCCCC2CCCN(C(=O)CC(C)C#N)C2)cc1 c1(SC)nc(O)c(C(N2CC(NC(C3(CCOC)CC3)=O)C(C)C2)=O)cc1C#N CC(O)CCC(=O)N(C)CC1COCCN1C(c1csc(-c2ncc[nH]2)n1)=O N1(C(Cc2c(C)noc2Cl)=O)CC(CNC(=O)C=Cc2cccnc2)CC1(C)C c1(OC)ccc(CC(=O)N(c2ccccc2)CCNC(=O)CNC(C)=O)cn1 c1(CNC(C(CC)n2cncn2)=O)c(F)c(F)c(F)c(F)c1F c1(NC(C)=O)ccc(C(=O)NC2CN(C(C3CCC(C#N)C3)=O)C2)cc1Cl C1(c2ccccc2)(NC(CCSC)=O)CCN(C(=O)CCC2CCN(C)C2)C1 Cc1ccc(NC(C2CCN(C(c3ncn(C)c3C)=O)C2C)=O)c(C)c1O c1(NC(C)C(=O)OCC2CN(C(=O)OC(C)(C)C)C2)ccc(Br)cc1 c1(CN(CC(F)(F)Oc2ccccc2)C)csc(Cl)c1Cl N1(C(c2cncc(C)c2)=O)CC2ON=C(CNC(c3cnc(C(C)C)s3)=O)C2C1 n1(CC)cnc2[nH]c(=NCCS(=O)(=O)CC)[nH]c(=NC3CCCc4cnccc43)c12 CCC(CC)C(=O)NCC(N1CCCC1C(=O)NCCC1(C)CC1)=O C12(CC(N3CCC(C)(C(N(CCC#N)C)=O)C3)=O)CC3CC(CC(C3)C1)C2 C1(C)(CC)CCC(NC(=O)CN(C(=O)C(C)CO)CC(C)C)CC1 N1(C(CCC(C)=O)=O)C(C(=O)N(CCC(F)(F)F)C)CC2CC12 C1(C)(CN2CCOCC2C)CC2CCC1C2.c12nnc(s1)CNC(=O)NC2C C1(CSCCCn2nccc2CNC(C(=O)N(C)CC)=O)CC2(CCOC2)C1 N1(C(C2CCCN(CC)C2)=O)CC(NC(C2CSC2)=O)CC12CCC2 CCC(CC)CC(F)C(=O)NCc1cccn2ccnc12 N1(C(c2c(Cl)cn(C)n2)=O)CCC(CO)C(NC(=O)C(C)(C)c2ccno2)C1 c1(C(N(CC(C)O)CCNC(c2c(C)csn2)=O)=O)nc(C)c(C)[nH]c1=O c1(OCC)cncc(C(N2CCC(CCN(C(=O)CSCC)C)CC2)=O)n1 C(CC(=O)NC1COCC1C)(CC(C)C)NC(c1c(C)cc(CC)o1)=O c1(C(=O)NC(C(C(C)C)NC(=O)CCc2cnn[nH]2)C)cnc(O)c([N+](=O)[O-])c1 N1(C(C2OCCN(CC)C2)=O)CC2(C1)CN(C(=O)Cc1cc(OC)ccc1Cl)C2 C1(NC(C(C)Oc2ccc(Cl)cc2)=O)CC2CCC1N(C(C1(C)COC1)=O)C2 C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CC=CC(NC(C(C)n2cncn2)=O)C1 CCCCC(O)CC(=O)N1CC(NC(c2[nH]nc3ncccc23)=O)C1 C(=O)(CCCCCC#N)N1CCC(CC)C1C(=O)NCC(C)C(=O)OC c1(C(=O)NCC(N2C(C(=O)NCC(=O)OC)CC2C)=O)cc(C)cc(C)c1 c1(COC)nccc(=NCC2(CNC(c3nc(C)ccc3OC)=O)CCCC2)[nH]1 C(=O)(C(C(C)NC(=O)Cc1ccnn1C)C(C)C)N(C(CCCC)C)C c1(OCC(=O)NC(CC=C)CNC(=O)C(N2CCSCC2)C)ccc(Cl)c(F)c1 c1(N2CC(C)C(C(C)(C)O)C2)ncc(S(C)(=O)=O)cc1Cl Nc1c(Cl)cnc(C(=O)NCCCCNC(C2CCOC2C2CC2)=O)c1Cl N1(C(C2(C)CCC2)=O)CC2(C1)CN(C(c1coc(CC3CC3)n1)=O)CCO2 CCCCC(O)C(=O)NC1CN(C(=O)COC2CCCCC2)CC1CC(C)(C)C c1(C(=O)NC(C2CCCN(C(c3cc(Cl)ccn3)=O)C2)C)cc[nH]c2nccc1-2 c1(CC(=O)N(CC(C)O)CCNC(=O)CCn2cncn2)cccc2ccoc12 c1(C(=O)NCC2CC(NC(C3(OC)CCOC3)=O)C2)cc2cc(C)cc(C)c2[nH]1 c1(C(=O)NC(CNC(C(C=C)CC)=O)Cc2ccccc2)ccc(N)c(F)c1 C1(C(N2CCC(CNC(=O)CCn3ccnn3)C2)=O)CCN(C2CCSC2)CC1 c1(C(N2C(C(=O)NCc3ncn(C)c3)CC(F)(F)C2)=O)ccc(F)c([N+](=O)[O-])c1 Cc1cc(C(=O)NC2(CCNC(=O)Cc3nnc(C)o3)CC2)c2n[nH]cc2c1 C(c1cncnc1O)=CC(N1CCC(C(=O)NCCc2ccco2)(CO)C1)=O Nc1cncc(C(=O)NCC2CC(O)CN2C(C2CC2Cl)=O)n1 N1(C(c2n(CCC)ncc2)=O)CCCCCCC1C(=O)Nn1cnnc1C N1(C(C2COCCN(C(c3ccc(OC)o3)=O)C2)=O)CCc2ccc(Br)cc2C1 C(CCCC(=O)NC1CCN(CCNC(C2C3CN(C)CC23)=O)CC1)(OC)OC C1(C(N(C2(C(=O)NCCN3CCC(CO)C3)CC2)C)=O)CCCC1C1CC1 C1(NC(CC(=O)NCC#C)=O)CCCCN(C(=O)Cc2cncn2C)C1 N1(CC(=O)NC(C2(O)CN(C(C3(C)CCOCC3)=O)C2)C)CCCCCC1=O C(=O)(C(C(C)NC(c1cc2ccccc2o1)=O)C(C)C)NCCCCC=C Cc1sc(CN=C(NC2(C)CCCS2=O)NC2CCCC2)nc1C1CCCCC1 CN1CC(CNC(=O)CN(C(c2csc(Cl)n2)=O)C2CC2)CC1=O CC(C)CCCCCC(=O)NCC(CO)Nc1ncc(C#N)cc1Cl c1(CC)ccc(CC(=O)NC(CNC(=O)C(C)C(C)O)CC(C)C)c(C)c1 CC1CCCC(CNC(=O)CC(O)CNC(=O)CN(CC(C)(C)C)C)C1 c1(C(=O)NCCN(C(Cc2c(C)nsc2)=O)C(C)C)ccc2cnc(C)n2c1 N1(C(CSSC)=O)C(CNC(=O)COc2cccc(OC)c2)CC2COCC12 C1(NC(CC2C(C)(C)C2)=O)CN(C(=O)C=Cc2nccs2)CC1N=[N+]=[N-] Cc1c(N)c(C(=O)NCC2(C)CCN(C(=O)CSCCC(C)C)C2)nn1C C(CC(C(=O)N1CC(CNC(=O)CCc2cnc(O)[nH]2)C(O)C1)NC=O)SC c1(CC)c(C(=O)NC2(CNC(C3CCCC3SC)=O)CC2)cccc1F C(CC1CC1)(C(=O)NOCCN(C)C)NC(CN(C(C)=O)C)=O CCC(C)C(C(=O)NCC1(O)CN(C(C2CC(F)(F)C2(C)C)=O)C1)OC c1(C(N2CCN(C(=O)CC3CCOCC3)C3C2C3)=O)ccc(I)cc1[N+](=O)[O-] C(=O)(C(CCCC#N)NC(=O)OC(C)(C)C)N(C1CCCN(C(=O)C2CC2)C1)CC N1(C(COCCN(C)C)=O)C2CCC1C(NC(C1CC=CCC1)=O)C2 CC1CN(C(=O)CC2CCC(C)O2)CCN(C(c2c[nH]c3nccc-3c2)=O)C1 N1(C(Cc2c(C(=O)OC)csc2)=O)CCN(C(c2cc(C)c[nH]2)=O)C(C(C)C)C1 N1(C(C2CC(C(C)C)C2)=O)C2CCC1C(C)C(NC(C1CC3(C1)CC3(F)F)=O)C2 c1(C(=O)NC(CC)(C)C(=O)OC(C)(C)C)cc(C(F)(F)F)cc(N)c1 C(=O)(C(C)(O)CC(C)C)NC1(C)CCN(C(C2(COC)C=CCC2)=O)CC1 c1(CN2CCC3(CN(C(c4ncc(C)c(Cl)c4)=O)C3)C2)c[nH]c2cccc(C)c12 c1(CC)nc(C)c(C(N2CCC(C)(NC(C3CCCC3(F)F)=O)CC2)=O)c(C)n1 CC1CC(C(=O)N(C)Cc2cnn[nH]2)CN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(NC(c2ccnc(C3CC3)n2)=O)CN(C(c2cscn2)=O)CCC1C(F)(F)F c1(C(C(N2CCC(NC(=O)C(C)(COC)OC)CC2)=O)OC)ccc(F)c(Cl)c1 C1(C(=O)NCC(CC)(C)O)CCN(C(C23CCCN2CCC3)=O)C12CCC2 C(=O)(C1=CCCCCC1)NCC(=C)CCNC(c1cccc(F)c1C(C)C)=O C1(O)(C(=O)NCC(CNC(COCC=C)=O)OC)CCCC(C)(C)C1 CCC(C)C(C(=O)NCc1cc(C)cs1)N(C)C(c1cncc(C)c1)=O N1(C(CCN(C(C=CCCCCC)=O)CC2CC2)=O)CC(=O)N2CCCC2C1 c1(CN2CC3(C(C(=O)Nc4nccc(I)n4)C3)C2)cnn2c1CCCC2 c1(C(N2CCCN(C(C3N(CC)CCOC3)=O)CC2)=O)c(C)ncn(C)c1=O C(=O)(CC(CNC1CCCC(N)CC1)CC(C)C)N(C(CC)CC)C C1(NC(C2CCN(C)CC2)=O)CN(C(=O)COC2CCCCC2)CCC12CCC2 S(=O)(=O)(c1cccc2nccnc12)N1C(C)CCC1C(=O)NCc1cncs1 c1(C2C(C(=O)NCC3C(NC(c4c(C)noc4)=O)COC3)C2)ccncc1F C#CCCC(O)C(=O)N(C1CCN(C(C2CC=CC2)=O)C1)CC C#CC1COCCN1C(=O)C(C)CNC(=O)C(C)(C)C(F)F C12(CC(=O)NC3CC4CC3N(C(C3(O)COC3)=O)C4)CC3CC(C1)CC(O)(C3)C2 C(CCCC(=O)N1CCCC1CN(C(=O)Cc1nccs1)C1CC1)N(C)C c1(OC)ccc(Br)c(C(N2CC3CN(c4ncnc5n[nH]cc45)C3C2)=O)c1F C1(C(=O)NCC(C)(O)CNC(C2(C)CC(C#N)C2)=O)CSCC(=O)N1 C(N=c1cnc(C(C)(C)C)c[nH]1)c1c(OC)cnc(Br)c1 C(=O)(CC(C)(C)C(F)(F)F)NCCCNC(c1n(C)ncc1C(F)F)=O c1(OC)ccccc1CC(=O)NCC(C1CCC1)NC(=O)Cn1nccn1 CC1C(=O)Nc2ccccc2N1C(C1(c2ccc(Br)nc2)CC1)=O c1(C(=O)NC(CNC(C(CC)OCC)=O)CC)cc2c(cn1)COCC2 N1(C(C(CO)NC(N)=O)=O)CC2CC1CN2C(=O)CSCC1CCCCO1 c1(NC)cc(Cl)ccc1C(=O)NC1CCN(C(=O)CC2COCCOC2)C1C c1(C(C(N2CCCC(CN(C(CCC#C)=O)CC)C2)=O)O)ccc(F)c(Cl)c1 C1(NC(c2ncc3cc(Cl)ccn23)=O)CCC2(CCN(C(c3ccns3)=O)C2)C1 Cc1ncc(C(=O)NCc2cn(CC(N3CCC(N(C)C)C3)C)nn2)cn1 N1(C(c2c(OC)ccc(F)c2N)=O)CC(CO)C2(C1)CN(C(=O)CC(F)(F)F)C2 C1(C(=O)Nc2cnc(C)c(F)c2)Cc2cc(O)ccc2CN1Cc1cccn1C C(=O)(C(C)(CO)NC(=O)CN1CCNC1=O)NC(CC(=O)OCC)C c1(NCC(c2ccc(Cl)cc2)C)c(N)cccc1[N+](=O)[O-] C1(CC)CN(C(=O)C(O)CF)CCN1C(c1cc(C(C)(C)C)oc1C)=O c1(C(N2C(CN(C(C3C(OC)CC3)=O)C)CCC2)=O)cc(C)c(O)c([N+](=O)[O-])c1 N1(C(COC(C)=O)=O)CCCC2CC(N(C(=O)CCCc3ccsc3)C)CCC12 Cc1cc(Br)ccc1CC(=O)NC1CCC(CC(=O)Nc2cncnc2O)CC1 C1(C(=O)NC2C(OC)CN(C(c3sccc3Cl)=O)C2)CN2CCN1C(C)C2 CC(C)(CCC(=O)N1CC(NC(=O)C=CCOC2CCOCC2)C1)[N+](=O)[O-] C1(CNC(c2cncc(Cl)n2)=O)CC2(CC2)CN1c1cc(C2CC2)ncn1 CC(C)(CC#N)C(=O)NC1CCC(F)(CNC(=O)C(Cl)=CCl)C1 c1(C(=O)NCC2CCC(NC(C3CC(C#N)C3)=O)C2)ncc(F)cc1F N1(C(COC(C)C)=O)CCN(C(c2sccc2C(F)F)=O)C2(CC2)C1 C1(CC)CN(C(=O)C(c2cccc(Cl)c2)(F)F)CCN1C(=O)CSC(F)F c1(C(=O)OC)cc(S(=O)(=O)NCCCCN2CC(N)C2)c(Br)cc1Br c1(COC(N2CCC(CC)C2C(=O)NCC)=O)sccc1S(=O)(=O)CO.C(C)(C)C N1(C(C2C(=C)CC2)=O)CC2(CCN(C(C3(CCN(C)C)CC3)=O)CC2)CC1C c1(C(N2CCC(OCCNC(C(CC)OCC)=O)C2)=O)oc(C2CC2)nc1C c1(CC(=O)N(C(CN(C(CCSC)=O)C)C)C)ccnn1C CC(CNC(=O)CC1CC=CC1)CN(C(=O)C(C)c1ccon1)C C(=O)(C1CCc2cccc(F)c21)NC1CN(C(C(CCC)C)=O)CC1C C1(NC(c2cc(C)c(C(F)F)cn2)=O)CCN(C(c2ccon2)=O)CC12CCC2 CC(C)(C)CCCCC(=O)NC1CCC1NC(c1c(O)ccc(F)c1Br)=O CC(C)CC(C)(O)C(=O)NCCCCCNC(C1Cc2cccnc2C1)=O C1(CC(=O)NC2CC(F)(F)CC2NC(c2cccnc2O)=O)CC2(CCC2)CO1 C1(C)(NC(C2(CNC(c3ncccc3C)=O)CC(=C)C2)=O)CCC(=O)NC1=O C1(CNC(C#CCNC(C(CO)N(C)C)=O)=O)CC(=O)NC1=O N1(C(C2(F)CCCCC2)=O)CCC(c2n[nH]c(CNC(C3CC(O)C3)=O)n2)CC1 S(=O)(=O)(c1cccnc1Cl)N1CC(CNC(=O)Cc2ccc(F)c(Br)c2)OCC1 N1(C(C(CC)CC)=O)CCCC(CNC(C2CCCC3(CC3)C2)=O)CC1 C1(N(C(N(C2CCN(c3nc(=N)[nH][nH]3)C2)C)=O)CC2CCOCC2)CCCC1(C)C Cc1nc(C2CC2)ncc1C(=O)NCC1CC(C)(C)CN1C(c1coc(Br)n1)=O CC1CCC(C)N1CCC(=O)NC1(C(=O)NC2C3CCC2CC3)CCCC1 CC#CCC(C(=O)NC(C)CC(=O)OCC)NC(=O)CC1=CCCC1 N1(C(=O)NC(C)Cc2cncs2)CCCCC1c1nccn1C N1(C(C(C)NS(C)(=O)=O)=O)CC2(CCCC2NC(c2ccc3[nH]ccc3c2)=O)C1 CC1CCOC(C(=O)NCC2(C)CCN(C(=O)Cc3cncn3C)C2)C1 C(=O)(CCCCC(N)=O)NCC(=O)NCC(C)C1CCC1 O=C(N=c1nc[nH]n1-c1ccccc1)N1CC(c2cncc(Br)c2)(O)C1 c1(CC(=O)NCCC2COCCN2C(=O)N2CC2)ccnc(F)c1F c1(CC(N2CCC(Cc3nnc(C)o3)CC2)=O)ccc(Cl)c(Cl)c1C c1(NC(C)=O)cc(C(=O)NC23CCC(C(=O)NC4CC(O)C4)(C2)OC3)ccc1F c1(C(N2CC(N(C(c3c(OC)c(Cl)sc3)=O)C)C2)=O)cccc2c(C)ccnc12 c1(C(N2C(CN(C(c3ccn(CCOC)n3)=O)CC)CCC2)=O)nc(C)n(C)n1 C(=O)(CC(C(F)(F)F)NC(=O)C(C)OCCN(C)C)N(CC(c1ccccc1)C)C c1(N(C(CC2CCOC2)C(=O)NCC(F)F)CC)ccccc1N(C)C C1(C(=O)NCC(CC2CC2)OC)C(C)CCN1C(C1CN(C)C(=O)N1)=O CCCC(C)(C)C(=O)NC1(CC(=O)Nc2ccc(Br)cn2)CCC1 C1(CC(=O)NC2CCN(CCNC(=O)COC3CCCC3)CC2)CC2(CCC2)C1 C1(c2ccccc2)(C(=O)NCC(CN(C(C=C(C)C(F)F)=O)C)C)CC(F)C1 Cc1ccc(C2CC2NC(C2(Br)CC2)=O)c(Cl)n1 C1(C(=O)NC(C(=O)N(CC)CC)C)CC12CCN(C(c1nccnc1C)=O)C2 C(=O)(CCCC(C)NC(=O)CS(=O)(=O)NC)NCCC(CC)CO CC12CN(C(=O)CCN3CCC3)C(C(=O)NC3CNC(=O)C34CC4)(C1)C2 N1(C(C(C)n2cnnn2)=O)Cc2ccccc2C(NC(c2ccnnc2S)=O)C1 c1(CC(=O)NC(C2CCCN2C(=O)CC2CCNC(=O)C2)C)cccc(F)c1 c1(CSCC(=O)N(C2CCN(C(=O)C(c3ccccc3)=O)C2)CC)cnn(C)c1 C1(OC)CC(NC(C2CCC3CC23)=O)CN(C(c2cnn(C)c2)=O)C1 C12(CNC(C3(CC(C)C)CC3)=O)CC1CN(C(=O)CCN(c1ccccc1)C)C2 N1(S(CC)(=O)=O)CCC2(CCCC2N2CCC(c3ccc(F)c(F)c3)CC2)CC1 C1(C(N(C)OC2CCCC2)=O)CC1C1CCOC1.C12(CCC1)CC(=O)N2 Cc1cc([N+](=O)[O-])cnc1N1CCN(C(=O)C#CC2CCCCO2)CC(O)C1 CC1CN(C(=O)Cc2cc(N)ccn2)CCN1C(c1cc(Br)nn1C)=O C(=O)(C(C(C)C)C1CC1)NC(CC(=O)Nc1cn(CC#C)nc1)C1CC1 c1(C(=O)NC2C(NC(C3C(C)C3C)=O)CC(F)(F)C2)nc(O)nc(O)c1F CC1C=C(C(=O)N2CC(N(C(c3cnn(C4CC4)c3)=O)OC(C(C)(C)C)=O)C2)C1 C1(c2nnnn2C(C)C)(Nc2ccc(C)c(C3CC3)c2)CC(C)(C(C)C)CC1C O=C1CC(CC(=O)N2CCC(NC(c3ccnn3C(F)F)=O)C2)c2ccccc2N1 N1(C(c2cc(OC)n(C)n2)=O)CCN(C(=O)NC(C(=O)OCC)C)C(C)C1 c1(N(CCCOCCCC)C)nc(N(C)CCC2CCCC2)nc2c1SCC2 c1(CCCC)ccc(C(=O)NCC2CC2NC(C2(C3(C)CC3)CC2)=O)cc1 N1(C(c2cccc(C)c2C)=O)CCC2(CCCN2C(C2CC2F)=O)CC1 C(c1ccccc1F)=CCC(N1C(C(C)NC(CCN(C)CC)=O)CCCC1)=O C1(C(=O)NCC(C)(C)OCCO)C2CC(O)C(C2)N1C(=O)Cc1ccc[nH]1 c1(C(N2CCC(O)(CN(C(CC(=O)NCC)=O)C)C2)=O)cc2c(Cl)cccc2s1 Cc1cc(C(N2CCOCC(NC(=O)CC3(CO)CCC3)C2)=O)c(C)nc1C N1(C(C2CCC(=O)O2)=O)CCC2(CCCCC2NC(c2cc3cscc3s2)=O)C1 C(C1=CCSC1(C)C)OC(c1cnn(CC)c1C(F)(F)F)=O N1(C(c2c(SC)snn2)=O)CCOCC1CCNC(=O)Cc1ccn(C)n1 C#CCC(C)(C(=O)N1CCSC2CCC12)NC(c1nc(CC)oc1C)=O C1(NC(C=CSC)=O)CN(C(C2CCCC(=O)N2)=O)CCC1C C1(CC)CN(C(=O)C(CC2CC2)NC(=O)COCC(=O)OC)CCS1 CC(CC(=O)NCc1cc(C(=O)NCC(F)Cl)no1)n1ccnc1 C(=O)(C(C)S(C)(=O)=O)NC1C(C)N(C(=O)CC2CCC3CC3C2)CC1 c1(CC2C(C(N3CCC(OCC#C)CC3)=O)C2)ccc(O)c(C)c1O Cc1nn(C)c(C(=O)NCCC2CCCN(CC(=O)NC3CC3)C2)c1Cl c1(OCC)c(C(N2CCC(NC(c3ccc(C)c(O)c3)=O)CC2)=O)cccc1F C(=O)(CCC(=O)NCc1ccc(CC(C)NC(C2CCC3(CC3)C2)=O)cc1)NC C(=O)(C1=CCCC(C)(C)C1)N(CCNC(c1ccc(SC)cc1)=O)C1CC1 c1(C(N2CC(OC)C(NC(=O)CN3CC4CC4C3)C2)=O)cccc(N=[N+]=[N-])c1 C1(OC)(OC)CC(C2CCN(C(CCC3(C)CC3)C(=O)NC3CC3)C2)C1 C(=O)(C1=NOC(C)C1)OCCN(c1ccnn1C(C)(C)C)C(C)=O c1(C(N(C2CCN(C(CCC#CC)=O)C2)CCO)=O)cc(C)c(C)nc1C Cc1cnn(CC(=O)NCC2(CCNC(C3CCCS3)=O)CC2)c(=O)c1 c1(C(=O)NC2C(C(N3CCN(C(CCC)=O)CC3)=O)CCC2)nccc(C)c1Br N#Cc1cccc(S(=O)(=O)NC2CN(Cc3cccnc3Cl)C2)c1 c1(CC)ccc2occ(C(=O)NCC(CN(C(C3(OC)CCCC3)=O)C)O)c2c1 Cc1cc(C(N2CC(n3cc(C(O)CC(C)C)nn3)C2)=O)ncc1C#N c1(OC)ccc(C=CC(N2CCCC3(NC(c4cnc(=N)[nH]c4)=O)CC23)=O)cc1 N1(C(C2CCC(OC)CC2)C(=O)OC(C)(C)C)CCCC1C1CCCN1C(C)=O C(=O)(CCC(C)(F)F)NCC1(C(N2C(C=C)CC2)=O)CC(=C)C1 C(=O)(C1Cc2c(Cl)cccc21)N(CCNc1cc(CC)nc(C)n1)C C(C(C)(C)CNC(=O)C(COCC)OC(C)(C)C)NC(C(C)NS(CC)(=O)=O)=O c1(C(N2C(CNC(c3cc(C(C)=O)sc3)=O)CCC2)=O)n[nH]c(C)c1C C(C)(CCC(C)(C)O)(c1nnnn1C(C)C)NCC(CCO)SC O=C(CC(C(F)(F)F)NC(C12CCCC1C2(F)F)=O)Nc1cccc(Cl)c1 c1(CNC(C(c2ccc(Cl)s2)N(CC(=O)NC)C)=O)ccccc1 C1(C(N2C(C)CN(C(=O)C(C)(C)c3cncnc3)CC2)=O)CCn2ccnc2C1 c1(CN2CC(NC(c3cn(C)nc3)=O)C(F)C2)cc(C#N)ccc1[N+](=O)[O-] C=CC1(C(=O)NCCCCS(C)=O)CCN(C(C2CC=CC2)=O)C1 CC1CCN(C(C2CCCCC2)=O)C1CNC(=O)C(C1CCOCC1)O c1(C(=O)NC2CN(C(c3cc(F)cc(Cl)c3)=O)CCC2F)ccnn2ccnc12 CC1CCN(C(C2COC(C)C2)=O)CCN1C(c1ccc2nn[nH]c2n1)=O C(=O)(C1=C(CC)OCCS1)NCC1(F)CCC(NC(CC(C=C)CC)=O)C1 c1(CC(=O)NC(CNC(C(C(C)C)(C)C)=O)(C)CC(C)C)cccc([N+](=O)[O-])c1 C#Cc1ccc(C(=O)NCC2CCCN(C(=O)C3=NOCC3)C2)nc1 c1(C(N2CC(C)(CC=C)C2)C(=O)NC2CCCC2)ccc2ccc(F)c(F)c2n1 N1(C(c2c(C)scn2)=O)CC2CCCC1C2CNC(c1cccnc1C1CC1)=O c1(C(=O)NC2CN(C(C(CC(C)C)(F)F)=O)CC2O)ccc2c(c1)CC(C)(C)C2 C(=O)(C1=CCC(C)CC1)NC1C(OCc2ccc(OCCC)cc2)CCCC1 CC1CCC(CNC(c2cccnc2CNC(C2CCCOCC2)=O)=O)CC1 N1(C(C(=O)NC(CC)(C)C)C)CCOC(C)(CNC(C2(C(N)=O)CC2)=O)C1 C#CC1(C(=O)NCCCCS(C)=O)CCN(C(c2ccccc2C)=O)CC1 N1(C(C(C)(C)NC(=O)OC)=O)CCCC(CN(C(=O)Cc2ncccc2C)C)C1 C1(C(=O)NCC(C)CN(C(=O)CC2CNC(=O)C2)C)CCCS(=O)(=O)C1 C1(OCCC)CCN(N2CCN(C)C(C(F)F)C2)C1 c1(C(=O)NC2C(NC(CCC#CC)=O)CC2)cc(S(N)(=O)=O)sc1C C1(C2CC2)(CNC(C(=O)N(CC(C)N)C)=O)CCNC1 c1(C(N2C(CC)CN(S(=O)(=O)c3ccsc3)CC2)=O)cc(Br)c(O)c(Br)c1 C#CC1(NC(C2CC2CNC(=O)C(C)=NOCC#N)=O)CCCOC1 Cc1ncc(S(N)(=O)=O)cc1C(N1CCC2(NC(=O)Cc3csnn3)CC2C1)=O N1(C(C2CCOCC2)C(=O)NCCSC)CCC(O)CC(C)C1 N1(C(c2c(CC)cccc2)=O)CCC2(COC(CNC(=O)C(F)C3CCC3)C2)C1 N1(C(C(CCCCC)O)=O)CCC2(CCCCN(C(=O)C3=CCCOC3)C2)C1 C1(NC(=O)CC(C)CF)(CC)CCN(C(=O)COc2cccc(CCC)c2)CC1 c1(OC)ccc(C)cc1C(=O)NC1(CNC(c2ccoc2C(C)C)=O)CCOC1 C1(O)(C(N(CC(C)NC(=O)CSc2ccccn2)C)=O)CCC(C)(C)CC1 c1(C(N2CCC(CCNC(c3c(C)ccs3)=O)C2)=O)c[nH]c2ccncc2c1=O C1(C(N(CCCCNC(C(CC)(C)COC)=O)C)=O)CCc2cncn2C1 CCCCC(O)CC(=O)NCC(CC(C)C)NC(=O)CC1CC2CC1C2 c1(C(N2CC(NC(c3cnn(C(C)C)c3F)=O)C(C)C2)=O)cccc(F)c1F N1(C(c2nc(C)c(Br)cn2)=O)CCC2(CCCN(Cc3c(C)nn(C)c3C)C2)C1 c1(CC(N2CCC(O)(C(C)NC(C=C(CCC)C)=O)C2)=O)nc2ncccn2n1 C1(C(=O)NCC2(C(N)=O)CN(C(=O)CC3CC4CC4C3)C2)(COC)CC=CCC1 C12(C(=O)NC34CC(CNC(C(C(=C)Cl)(C)C)=O)(C3)C4)CC(CO)(C1)OC2(C)C c1(C(=O)NC2CN(C(CC)=O)C2)cc(CC)c(C)s1.C12COC(C1)CNC2 Cc1[nH]nc(Cl)c1C(=O)NC(CNC(C1CCOC(C(C)C)C1)=O)C1CC1 Cc1onc2ncnc(SC)c12.N1(c2n(CCO)c(O)nn2)C2COC3C2OCC13 N1(C(C2CC(C)(CC)C2)=O)CCC(CC(C)NC(=O)CSCc2cscn2)CC1 C(=O)(C(CCCOC)N1CCCC(C)C1)NC(C(=O)NCC)C C1(CC=C)(NC(=O)Cc2cn(C)cn2)CCCN(C(C2CCCCN2C)=O)C1 O(S(=O)(=O)c1cc2cc(Cl)ccc2o1)c1cc([N+](=O)[O-])c(Br)cc1 n1(CC(=O)NC(C2CCN(C(C3(C)CC(F)C3)=O)C2)(C)C)ccc(C2CC2)n1 C1(CNC(C(C)N(C(CCN(C)CC)=O)CC)=O)CC2C=CC1O2 N1(C(c2ccc(OC)s2)=O)CCCC(N(C(=O)CCc2nnc(S)n2C)C)CC1 c1(C(=O)NC(CCNC(c2c(C)con2)=O)C(C)C)cc2c(s1)CCCC2 O=C1NC(=O)N2CCN(CC(=O)NCc3ccc(F)cc3Br)CC12 C1(NC(C(C)OCCC=C)=O)CCOCC1NC(=O)CCc1cc(C)nn1C C(=O)(CC(=O)NCCN(C(C1CC(OC)C1)=O)C1CC1)NCC#C N1(C(c2c(C)coc2C)=O)CCC2(CCCN(C(C3CCC=CCCC3)=O)C2)C1 c1(CNC(=O)CC2C3CCCC3N2C(C2(C)CC(C)C2)=O)cnn2ccccc12 C(=O)(CCCC(C)S(C)(=O)=O)N1CC2CC(CN(C(CS(=O)(=O)NCC)=O)C2)C1 CCC(CCC(=O)NC1CC12CCN(C(c1cc(COC)[nH]n1)=O)C2)OC c1(NC2CCN(CC)C2)ncc(C(c2nnnn2-c2ccccc2)NC(C)=O)o1 C1(O)(CNC(CCN(CCCCC)C(C)C)=O)CC(NC(C2CC2F)=O)C1 Cc1[nH]cc(C(=O)NCC2COC(CNC(=O)C3=COCCC3)C2)c(=O)c1Cl C1(CN(C(=O)CCCCO)C)COCCN1C(c1scnc1C(F)(F)F)=O c1(C(=O)NC2CC(C(F)CO)C2)ccc2c(n1)COCC2 CC1CCC(NC(=O)CCC(C)(C)C)CN1C(c1cccc(-n2cccn2)n1)=O O=C(CCS(=O)(=O)c1ccccc1)N1CCC2(CC1)CCN(C(C1CC1F)=O)C2 C=Cn1nccc1C(=O)NCC(CO)NC(c1csc(CC(F)(F)F)n1)=O N1(C(C=CCN(C(C23CCC(OC)C2C3)=O)C)=O)CCc2c(O)noc2C1 Cc1ccc2c(c1)CC(C(N1CCC(O)(CNC(=O)CCP(C)(C)=O)C1)=O)O2 C(=O)(C1=CCS(=O)(=O)C1)NC(CCN(C(C(COC)NC(C)=O)=O)C)C C1(CC(=O)NC2CCC2C(=O)O)CN(C(=O)Cn2cnnc2)CC12CC2 c1(C(N2CC(C)N(C(c3ccc(S(C)(=O)=O)s3)=O)CC2)=O)cccc2nccn12 c1(OC)ccc(Cl)c(C)c1C(N1CCC(CNC(=O)CS(C)(=O)=O)C(C)C1)=O Cc1ccc(Br)cc1CCC(=O)NC1CCCC(NC(=O)C2CC2)C1 Cc1csc2c(N3C4CCC3CC(NC(c3cc(Cl)cnc3F)=O)C4)ncnc12 C1(C)(COC)CCCN1C(=O)CCCn1cc(-c2nc(C)c(C)[nH]2)nn1 c1(CC)oc(C)cc1C(=O)NCC(C1CCC1)NC(=O)CCNC(=O)CO CC1(C)C2CC(C(N3CC=CC(NC(c4sccc4OC(F)F)=O)C3)=O)CC12 C1(CNC(c2cc(CC)[nH]n2)=O)CN(C(=O)C(C)N=[N+]=[N-])CC1N(C)C C#CCC(C)(C(=O)NC(c1ccncc1F)C)NC(=O)CC(C)C1CC1 C(=O)(C(C(=O)NC1CC(C(=O)NC2(c3ccccc3)CCOC2)C1)OC)OC Cc1cn2c(n1)CN(C(c1conc1CNC(C1CCC(C#N)CC1)=O)=O)CC2 CCCCS(=O)(=O)CC(=O)NC12COC(C1)C(NC(=O)C(F)(F)C(C)O)C2 N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(c3ccnc(Cl)c3)=O)CC2)C1 c1(C(C(=O)NCCOCCCNC(C2CCCC(=O)O2)=O)O)ccc(Cl)cc1 c1(C(N2CCC(C)(NC(C3CCC(C(=O)OC)C3)=O)C2)=O)n[nH]c2ccccc12 CC(C(F)C(=O)NCCOCCNC(c1ccnc(OC(F)F)c1)=O)C(F)(F)F CN1CCC(C(=O)NC2CCC(CCC(=O)NCCCc3cnn[nH]3)C2)C1 N1(C(CC2CC(C)(C)OC2)=O)CCOC2(C1)CN(C(=O)Cn1ccc(=N)[nH]1)C2 c1(C(C2CC2)NC2CCC(COC)CC2)c(C)cc(Cl)cc1C C(=O)(C(CCCOC)NC(=O)C(C)NC=O)N(C(C(=O)N(C)C)C)C.CO N1(C(c2c(CCC)occ2)=O)CC2CCCC(C1)N2C(C1CCCC(C#N)C1)=O CC1CN(C(C2CC2c2ccccn2)=O)CC1(C)C(=O)NC(C(N)=O)C1CC1 c1(C(N2C(CN(CCC)CCNC(=O)OC(C)(C)C)CCC2)=O)cncc(Cl)n1 N1(C(c2cccc(SC)c2)=O)C2CCC1CN(C(=O)Cc1csc3nccn13)C2 N1(C(C(C2CC2)SC)=O)CC2CC1CN(C(=O)Cc1csc(Br)c1)C2 C(C(=O)N(C)CCNC(=O)CCOCCCOC1CC1)(C1CCOC1)OCC c1(OCC(N2C(C)C(NC(C3C4CCC3CC4)=O)CC2)=O)ccccc1C#N C1(F)(C(C)NC(c2cccc(N)c2)=O)CCN(C(C2(C(F)F)CCCO2)=O)CC1 C(=O)(CCCC(F)(F)Br)N1CC(O)(CCNC(CCC(=C)C)=O)C1 C12(CNC(c3c(Cl)c(C)n(C)n3)=O)CCCC1CN(C(=O)C(C)N1CC(C)C1)C2 N1(C(CC(C)c2ccccc2)=O)CCC(NC(c2c(Cl)cncc2Cl)=O)C(F)C1 C(CC(C)(C)C(=O)N1CC(CNC(C2(CO)CCCC2)=O)CC1(C)C)OC N1(C(CCOC)=O)CCC2(CCCC(CNC(=O)C(O)C3CC3)O2)CC1 N1(C(CCSC)=O)CCC2(CC2)CC1C(N1CC(C)(C)C12CCC2)=O Cc1ccc(S(N)(=O)=O)cc1C(=O)NCCn1nc2ccccn2c1=O c1(NC)nccc(C(N2CC3(CCC3CNC(C3CC3F)=O)C2)=O)c1F C(=O)(C1CCCc2c[nH]nc21)NCC12N(C(C(C(C)C)F)=O)CC(C1)C2 c1(C(N(CC(C)NC(=O)Cc2cncs2)C)=O)cccc2c1oc(=O)n2C C(=O)(CCCC(CC)NC(c1cnc(=N)[nH]c1)=O)NC(CCC=C)CO N1(C(C(C2CC2)SC)=O)CCN(C(=O)CC(C)c2cnn(C)c2)C(CCO)C1 c1(COC)cccc2c(C(=O)NC(=O)C3CC3)coc12.C12(CC1)NC(=O)CS2 CC1CN(C)CCC1NC(=O)C(C(C)(C)O)NC(C1CCC(CO)CC1)=O CC1CN(C(c2ccc(CNC(c3ccc(F)cc3)=O)cc2)=O)CCCO1 Cc1ncncc1C(=O)NC(C)C(c1ccccc1)NC(=O)CN(C)C(N)=O C1(C)(C(N2CC(OC)(CNC(C3CC34CC4)=O)C2)=O)CCCCCC1 C(=O)(C(C)CCCC(C)C)NCCN(CCCCCC)C(=O)C=CC1CCCC1 c1(C(=O)NC)cncc(C=CC(=O)NCC2CC(CNC(C3(C)CC3)=O)CO2)c1 N1(C(CCN(C)CCO)=O)CCCC12CCCN(C(=O)Cn1cnnc1O)C2 N1(C(C(COCC)C)=O)CCN(C(=O)C=CCOCc2ccccc2)CC1CO Cc1cc(=NC2CN(C(C3CCCC3O)=O)Cc3ccccc32)[nH]c(Cl)n1 N1(C(C2C(COC)(CO)C2)=O)CC2(CCC(NC(=O)CC3(C)CC3)CC2)C1 C(C(O)CC(=O)NCC(c1ccccc1)O)N(C(=O)COCC1CC1)C c1(C(=O)NC2CCC(NC(c3ncccc3F)=O)C2)[nH]cc2c1CCC2 C(C(C)(C)C(F)(F)CC)NC(C#C)(C)C1CCOC1 N1(C(C2C(OC)(OC)CC2)=O)CCOC(C(N2C(C(N)=O)CC2C)=O)C1 Cn1ncc(C(=O)NCCC2COCCN2C(=O)CC=Cc2ccccc2)c1N c1(C(=O)OCC)nnc2n1CCN(C(c1c(I)ncn1C)C(=O)NC1CCC1)C2 C(C)(C)(CCC(=O)NCC1CC(NC(=O)CC(C)c2ccccc2)C1)OC c1(C(N2CCC(C)(NC(c3ncc(Cl)s3)=O)C2)=O)ccccc1[N+](=O)[O-] N1(C(C(C)OCCCC)=O)CCCCC(C(=O)NC2(c3cc[nH]n3)CC2)C1 C#CCC(CC(F)F)C(=O)NCc1cn(CCNC2CC(NS(C)(=O)=O)C2)nn1 C1(NC(c2cccc(C)c2F)=O)CCC2CN(CC3CC(C)C3)CC2C1 C(CCCCCC(C)C)NC(C(CC)NC(C1CCC2(CCC2)C1)=O)=O N1(CC(=O)Nc2ccc(-c3nnc(CC)o3)cc2C)CCn2c(C)nnc2C1 N1(c2nc(C)c([N+](=O)[O-])cc2Cl)CCC(=O)N2CCCCCC12 c1(N2CCC(NC(c3cc(C(F)F)[nH]n3)=O)C23CCC3)nc2cccc(F)c2o1 C1(CNC(C2(COC)CCNC2=O)=O)CCN(C(=O)COC(C)=O)CC1C C1(C)(CNC(C(F)OC)=O)CN(C(c2cscc2Cl)=O)C(C)(C)C1 C1(C(=O)NC2C(CNC(C3(C)COC3)=O)COC2)Cc2nccn2C1 CON1CCC(N=c2ncnc3[nH][nH]cc2-3)CC1.C(C)(C)C Cc1cc(C(N2CCCC(c3nnc(O)o3)C2)=O)c(C)o1 O=C(C1CCCc2nn[nH]c21)NC1CN(C(c2ccoc2Cl)=O)C1 c1(C(N2CCCC(n3cc(CCS(CC)=O)nn3)C2)=O)cnn2c1OCC2 Cc1cc(C(N2CC(NC(C3CCCC4CC34)=O)CC2C)=O)c(O)nn1 c1(C(=O)NCC2(F)CC(NC(c3c(C)nc(COC)s3)=O)C2)c(C)ccnc1C Cc1nc2c(s1)C(N(C)C(C(=O)NC1CCCC1)C1CCC1C(F)(F)F)CCC2 CC(Cc1ccccc1)C(=O)N1CC(C(N)=O)(CNC(=O)Cc2ncccn2)C1 c1(C(=O)NC2(CNC(COc3cn(C)nc3)=O)CC2)ccnc(Cl)c1O C1(NC(=O)C=CC(N2CCOCC2)=O)CCCCCN(C(c2ccsn2)=O)C1 c1(CC(=O)NC(C2CCN(C(=O)C(C)CO)CC2)C)ccccc1N Cc1ccnnc1C(=O)N(C)CCN1CCN(C(C2CN(C)C(=O)N2)=O)CC1 N1(CC(C)(C)NC(C(c2cccs2)SC)=O)CCN(C(C2CCCS2)=O)CC1 c1(C(=O)NC2CC(NC(c3ccc(C)nc3)=O)C23CCC3)ccc2n[nH]cc2c1 C#CCCN=C(NCC(CC=C)C(C)C)N(C)CCC1CCCO1 C1(C(N2CC(CNC(C(C(C)C)OC)=O)OCC2)=O)CCc2ccnn2C1 CC(C)C(C(=O)NCC1CCCN(C(C2(N(C)C)CC(O)C2)=O)C1)c1cnn(C)c1 CCC(C#N)(CC)C(=O)NCC(F)CNC(c1cccc2nn[nH]c12)=O C1(NC(c2ccc(CC)s2)=O)C(CNC(c2c(Cl)cnn2C)=O)CCC12CCC2 C1(C(N2CC(CN(C(CC(C)c3ccccc3)=O)C)C2)=O)CC(N=[N+]=[N-])C1 N1(C(C(C)OCCC=C)=O)CC2CC(C1)C2NC(=O)CCc1cncc(F)c1 C(N=c1[nH]c(C)nc(C)c1C)C1CCC(NC(c2cc(CSC)c(C)s2)=O)CC1 C(N=c1nc2sccc2c(NC2CCCc3occc32)[nH]1)C1CCN(CCF)C1 n1(CCNC(Cc2ccc(CC)cc2)=O)c(C)c(Br)c2ccccc12 c1(OC)cc(C)nc(N2CCCC(CNC(=O)CCC(C)(F)F)C2)n1 c1(OC)ncc(Cl)cc1C(N1CC(NC(=O)C(C)c2ncco2)C(C)C1)=O C(CNC(=O)C(N1CCCCC1=O)C)(C(C)(C)C)NC(c1c(C)[nH]cc1)=O c1(COCC)ccc(OC(=O)C(CC)S(=O)(=O)CC)cc1.c12nsc(n1)S2 c1(CN2CCC3(CC2)CN(Cc2cc(C)[nH]c2C)C3)c[nH]c2cc(C#N)ccc12 c1(C(=O)NCCC2(NC(C(CC)N(C)C)=O)CC2)cccc2nncn12 Cc1cccc(C)c1C(O)C(=O)NCCOC1CN(C(C2CC2(C)C)=O)C1 CC1CN(C(c2cc(Cl)cnc2O)=O)CCC1CNC(=O)CSc1ccncc1 N1(C(C(C)N(C(C2CCCC2)=O)CC)=O)CC(C)C(C)(CO)C1 c1(SC)nc(Cl)c(C)c(=NC2CC23CC(NC(C2CCCC4(CCC4)O2)=O)C3)[nH]1 C(=O)(C(CC)(CO)OC)N1CCC(C(N(C(CC)C2CC2)C)=O)(CC)C1 C1(OC)CC(CC(=O)NC(C)COC2CCC(C)CC2)N(C(C)=O)C1 Cc1nsc(NCC2C(C)CCCN2C(=O)CC2CC3CC3C2)c1C#N Cc1csc(C(C(=O)NC2CCCC2)N(CCC2=CCCC2)C)c1C c1(C(=O)Nc2cccc(-c3c(C)nc(F)cc3)n2)cc(F)c(F)c(Cl)c1 N1(C(c2ccccc2F)=O)CC2CC2(CNC(C2(n3cncn3)CC2)=O)C1.C c1(C(N2C(C)(CNC(C(=O)NCC)=O)CCC2)=O)ccsc1S(C)(=O)=O c1(OC)ccc(CCC(=O)N(CC(C)NC(=O)CC2CC=CCC2)C)cn1 C1(NC(C(N2CCC(C)C2)=O)=O)C2CN(C(c3cnc(C(F)F)nc3)=O)CC12 N1(C(C(CC)(C)Br)=O)CCCC(N2CCCC2=O)CC1 Cc1nc[nH]c1CCNC(C1(C2CCCN2C(=O)CC2CCOC2)CC1)=O c1(CNC(=NCCOCC)NCC(C)C(F)F)nc(C)c(S(C)(=O)=O)s1 N1(C(C2CCC(C)CC2)=O)CC(C)N(C(C23CCC(F)(CC2)CC3)=O)CC1C CC1C2CCC(C2)C1C(=O)NOCc1ccc(O)cc1.C1C(C)C(F)C(=O)N1 C12CN(CC1n1cccn1)C2=O.c1(C(N(C)C)C2CC2)cn(CC(=O)O)nn1 C1(C(=O)NC(CC)CC)CN(CC(C2CCOCC2)C)CC1C N1(C(C(COC)C)=O)CCC2(CCCC2NC(=O)C=CCCC=C(C)C)CC1 Cc1nc(CCC(=O)NCC2COC(CNC(=O)CCCNC(N)=O)C2)[nH]c1C C1(C2CC2)(C(=O)NC(C=C)CO)CN(C(c2ccc(O)cc2F)=O)C1 N1(C(C(C2CC2)OC)C)CCC(C(N2CC(C)(C)C2)=O)CC1 CC(C)(C#N)CC(=O)N1CCC(O)(CCNC(=O)CNC(C2CCOCC2)=O)C1 c1(SC)cc(F)ccc1C(=O)NCC1CCN(C(=O)C=Cc2cc[nH]n2)C1 C(C(F)(C(=O)N1CCN(C)C(C)C1)C(C)C)NC(C1=C(C)OCC1)=O Cc1[nH]ccc1C(N1C(C(N2CC(OCC(N)=O)C2)=O)CC1C)=O C(=O)(CCCC(C)C)N1CCC(CC=C)(NC(=O)CCCN2CCOCC2)C1 Cc1cc(C(=O)NC2CCC3CCN(c4nnc(C)o4)C2C3)n2ncnc2n1 c1(C(N2C(C(=O)NC3(C)CCC(C)C3)CCCC2)=O)cnn2cccc2c1 c1(C(N2C(CNC(C(C)(C3CC3)OC)=O)CC2)=O)c(F)cccc1Cl c1(C(N2CCOCC(NC(CNC(C)=O)=O)C2)=O)csc2ccc(F)cc12 O=C(C1=CCCCO1)NCC1CC(F)CN1C(=O)Cc1cccnc1 CC1C(NC(=O)CCOC2CC2)CC2CCC1N2C(=O)C1=NOCC1 c1(N(C(=O)C(n2nnnc2C2(c3ccno3)CCC2)C)C(C)=O)ccccc1 n1(CC)cc(NC(=O)C(Cc2cnc[nH]2)NC(C2CC(=O)CCO2)=O)c(C)n1 C(=O)(C1=CCC(C)(C)CC1)N(CC(C)NC(c1cccc(OCOC)c1)=O)C c1(OC)cc(C(=O)N(C)CC2(NC(=O)CCc3c(C)noc3C)CC2)cc(Cl)c1 c1(C(N2C3CN(C(C(COC)C)=O)C(C3)C2)=O)cnn2cc(C)cnc12 c1(NC(C(C)OCCC#C)=O)ccc(C)cc1SCC CON(CCC(=O)N1CC(O)CC12COC2)C(=O)CN1CCCCC1C c1(OC)ccc2c(c1)CCCC2C(=O)N(C(C)CNC(=O)Cc1cc[nH]c1)C CC(C(C)C(=O)N1CC(NC(c2ccnnc2O)=O)CCC(O)C1)S(C)(=O)=O C1(CNC(CCn2ncc(C)c2)=O)CCCN(C(=O)CN2CCSCC2)C1 c1(OC)ccc(I)c(NC(C2CN(C(C3(OC)CCC3)=O)C2)=O)c1 c1(C(=O)NCC(C2CC2)NC(C(C)SC)=O)ccc2cccc(O)c2c1 N1(C(=O)CNc2ccccn2)CC2CN(C(c3cn4cnnc4cn3)=O)CC2C1 Cc1cc(C(N2CCOCC2)CNCC(=O)NC2(C#N)CCCC2)ccc1F c1(OC(C)C)ccc(C(=O)NC(C)(CNC(=O)CC23COCC(C2)C3)CO)cn1 C1(C(N2CCCC(c3cc(OC)c(F)cc3)C2)=O)COc2ccccc2O1 CCC(CCCC(=O)N1CC2CC(C1)C2(C)C)NC(=O)Cn1nnc(C)n1 c1(C(=O)NC(C)CCCNC(C2CC2C#N)=O)cc2n(n1)CCN(C)S2(=O)=O c1(C(=O)NCC(C)N(C(C(CCCC)NC(N)=O)=O)C)cc(C)ccc1[N+](=O)[O-] N1(c2ncc(C(=O)OC(C)(C)C)nc2)CCC2C1C2(F)F c1(OC)ccc2[nH]c(C(N3CCCC(O)(CNC(C4CC4(F)F)=O)C3)=O)cc2c1 N1(C(CCC=CC(C)C)=O)CCC2(CC1)CC(CNC(c1c[nH]ccc1=O)=O)C2 n1(CC(C(=O)CCCC2CC2)=O)nc(O)ccc1=O.CCCC(=O)N CC1CN(C(c2cccnc2N)=O)CCN1C(=O)CCc1ccc(Cl)s1 S(=O)(=O)(c1cccnc1)NC(=O)OC(C)(C)C.CC1CCC2CC1CN2 c1(OCOC)cccc(C#N)c1NC1CCC(C)C(C)C1 N1(CC#CC)CCc2c(C)cc(C)cc21.C1(=O)C(C)(C)CCN1 c1(OC)ccc(CN2CC(NC(C3CC3(F)F)=O)C(C#N)C2)cc1O C1(NC(C2CC(OCC)C2)=O)CCCC(NC(c2cn(C(C)C)nc2C)=O)CC1 C1(C(=O)OC)C(C)CCN1C(=O)C#CCNC(C1CC(F)CN1C)=O c1(N2CCC(CCSC)CC2)cc(C)nc(NCC2CC23CC3)n1 c1(C(=O)NC(C)CN(C)C)ccc(Cl)nc1NC(C1CC1C)=O C1(CCNC(CN(C2CC(C#N)C2)C(=O)OC(C)(C)C)=O)COC(C)(C)C1 CC1(C)COC(CC(=O)NCCCCNC(=O)C(c2ccccc2)C2CC2)CO1 C1(CNC(C2C(=C)C2)=O)CC2(CC2)CN1C(=O)C=Cc1ncc[nH]1 N1(C(C(C=C)OC)=O)CCC(F)(F)C(CNC(c2c(C)noc2C)=O)C1 C1(NC(Cc2c(C)noc2)=O)CCS(=O)(=O)C12CN(C(=O)C(C1CCC(=O)N1)C)C2 Cc1nc(N2CC(C)(NC(=O)CC(c3ccccc3)N(C)C)C2)c2cc[nH]c2n1 c1(OC)ccc(C2(C(=O)NC(C)CNC(C3(C)CC=CCO3)=O)CC2)cc1OC N1(C(C2CCC(CC)O2)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC(O)C1 C1(NC(CNS(N)(=O)=O)=O)CC2COCC2N1C(c1cccc(C(N)=O)c1)=O N1(C(CSC(C)C)=O)CCC(CCC(=O)NCCC(N)=O)C1 N1(C(C(C)(C)SC)=O)CCC(C)C(NC(c2ccc(C(F)F)cc2Cl)=O)C1 C1(C(N2C(CNC(c3ccc(OC)cc3F)=O)C=CC2)=O)CC(C)(C)OC1(C)C C1(NC(=O)CN2CCC(C(F)(F)F)CC2)CC2CCC(C1)N2C(=O)C1=NOCC1 c1(OC)ccccc1CN(CC(c1nnn(C)n1)(C)C)Cc1cccs1 C1(C(N)=O)CC=CCC1C(N1CC(C(=O)Nc2ncc(-c3ccccc3)[nH]2)C1)=O n1(CCC)nnnc1C(c1cnco1)NC1(C)CC(O)C1 N1(C(=O)CC2CCN(C(c3ccc(Cl)c(I)c3)=O)C2)CCC2(CCCNC2=O)CC1 N1(C(C(CC)NC(C)=O)=O)CCN(C(C2COCCOC2)=O)C(c2cn[nH]c2)C1 c1(OC)ccc(C(N2CCCC2(C)C(=O)NC(c2ccno2)C)=O)c(O)c1 c1(C2(C)CCCC2)cccc(NC(c2ccncc2-c2ccnnc2)=O)c1 c1(OC)cc(CNC(=O)CCC2CCCN2C)ccc1-n1cnnn1 C1(C(=O)NC(CSC)(C)CO)CC2C=CC1N(C(c1ccc(C)cc1F)=O)C2 c1(C(N2CCCC(CNC(CC(C)C3CC3)=O)C2)=O)coc2c1C(=O)NCCC2 N1(C(C2C(C)(COC)C2)=O)CCCCC12CN(C(=O)Cc1cccc(C)c1C)C2 Cc1ccc([N+](=O)[O-])cc1C(=O)NC1C2CC1N(C(C1(F)CC1C)=O)C2 C(=O)(C(=O)C(C)(C)C)NC(C)CCC(=O)N1CCOCC1CCO c1(CN(C)C(c2ncc[nH]2)=O)ccccc1-c1nc[nH]n1 N1(C(c2c(N)cc(Cl)nc2)=O)CC2(CCC2)CC1CNC(=O)CCn1cncn1 N1(C(C(COC)(C)C)=O)CCCc2cccc(NC(=O)Cc3cc(C)no3)c21 N1(C(C(C)SC)=O)CCCC1(C)CNC(C1CCC(C(C)(C)O)CC1)=O c1(NC(c2scc(C(=O)NC(c3ccccn3)CC)n2)=O)c(Cl)cc(Br)cc1Br C(=O)(CC(F)(F)C(F)F)N1CCC(CC(=O)NC(c2c(C)cccc2)CO)C1 C1(CC(=O)N(C(CNC(c2coc(CO)c2)=O)C2CC2)C)SC2=NCCN2C1=O c1(C(=O)NCCN(C(=O)CCF)CCC)cc(Cl)c(OC)cc1Cl c1(CC)cc(C(N(C2CN(C(=O)C(C)(C)N(C)C)CC23CC3)C)=O)ccc1Cl Cc1cccc2nc(N3CCOCC(NC(=O)C(C)(F)C(C)(C)F)C3)sc12 C#Cc1ccc(C(N2CCC(CN(C(=O)CC(C)C(F)F)C)C2)=O)cc1C C1(C(=O)NCCC(=O)NCC)CC=CCN1C(c1csc(C)c1C)=O N1(C(CNS(NC)(=O)=O)=O)CC(C(=O)NC2CCCN(C)C2=O)CC1(C)C C1(C(=O)NC(C)CNC(=O)Cn2cccc2)OCCC1C C1(NC(c2c(C)oc(SC(F)(F)F)c2)=O)CCN(C(C2CC(F)(F)C2)=O)C12CC2 C1(C2CC2)(NC(C2C(CC)CCC2)=O)CCN(C(c2cccc(C(C)C)c2)=O)C1 n1(CC=C)cc(C(=O)NC2CCCC2CNC(=O)COC2CCCC2)nn1 C1(C(N(C2C3CN(C(c4c(CC)cccn4)=O)CC32)C)=O)CCCC2(CC2)C1 c1(NC(=O)NCC(=O)NC2CC2)cnnc(O)c1Cl C1(C(N2CCC(OC(C)C)C2)=O)CC12CCC(F)(F)CC2 C(=O)(C1CC(=O)Nc2ccccc21)N1CCN(CCCC#C)CC1 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)CSc2ccc(F)cc2F)C2CC12 c1(CC)ncccc1C(=O)N(C1CCN(C(=O)CC2CCCC(O)C2)CC1)C CN1CCCC(CC(N2CCC(O)(CN(C)C(c3nnn(C)n3)=O)C2)=O)C1 C(=O)(C(Cc1cccs1)NC(=O)CCc1nncn1CC)NC(C=C)C1CCC1 CCC(C)CC(C(=O)Nc1cc(C)cc(C)c1C)NC(c1cn(C)nn1)=O C(=O)(C(C)(C)n1cc(Cl)cn1)NCCN(C(C1C(C(=O)OC)C1)=O)C1CC1 c1(C(c2nnnn2-c2ccc(F)cc2)NCC(=O)NC)cc(Br)ncc1F C(=O)(C1CCCCc2ccccc21)N1CC(CCNC(C2CC(C)(C)C2)=O)C1 C1(CCSC)(C(N2CC(NC(C34CC(CO3)C4)=O)C(O)C2)=O)SCCCS1 c1(C(=O)NCC2(COC)CCCN2C(=O)C(C)CC2CC2)cc2cccn2cn1 C1(CC(C)NC(C2(N(C)C)CC2)=O)CC2CCC(C1)N2C(c1ccc(=O)n(C)n1)=O c1(OC)c(Cl)cc(Cl)c(OC)c1C(N1CCOC(C(=O)NC2CCCN2C)C1)=O S(=O)(=O)(c1ccc(Cl)s1)N1CC(CC(N2CCCC3(COC3)C2)=O)OCC1 CCC(C)(COC)C(=O)NCC1(O)CCCN(C(=O)CCC(N)=O)C1 C(=O)(C(C)(C)CC(C)C)NC(C1CCCC1)CNC(C1CN(CC)C(=O)C1)=O c1(OC)cc(C(N2CC(NC(C3CN(C)C3)=O)C3CC23)=O)c(N)c(C)c1 Cc1cc(=NCCCCc2ncc[nH]2)[nH]c(=NCC(C)OC(F)F)[nH]1 CC1COc2c(C(N3CC4CC3(CNC(=O)C(F)(F)C(C)O)C4)=O)cccc21 C=CC(C)(O)CC(=O)NC(C(=O)Nc1ccc(C)cc1)C(C)OC c1(CC(=O)NCC2C(NC(C(C)=C3CC3)=O)CCCC2)cccc2cnccc12 n1(C(=O)OC(C)C(=O)NC2(C(=O)OC)CC2)c2ccccc2c2ccccc12 CON(CCC(=O)NC1CCC=CCC1)C(=O)C(C)CCCOC C1(CNC(=O)Nc2ccc(OCC)cc2F)COc2ccccc2O1 N1(C(C(OC)OC)=O)CC(C)N(C(=O)CCc2cc(Cl)cc(Cl)c2)CC1C c1(CNC(=O)CN2CCN(C(C3SCCS3)=O)CC2)cccc[n+]1[O-] c1(CNC(C(C2CCC2)NC(C=CCC)=O)=O)c(F)cccc1F CC(CC(F)(F)F)NC(=O)CC1CCN(C(C2CC2F)=O)CC1 c1(C(N(CC(=O)NC(CCC)CO)C(C)C)=O)nnc(S)n1C n1(CC)ncc(C(N2CCC(N3CCN(C(=O)CP(C)(C)=O)CC3)CC2)=O)c1Cl CCCC(C(=O)N1CCC1c1cn(CCC(F)(F)C(C)C)nn1)C(C)C N(C1CN(C(=O)C2=CCSC2)CCc2ccccc21)C(=O)C=CI c1(C2C(CNC(CN(C(=O)C(C)C)CCOC)=O)C2)ccc(F)cc1 c1(C(=O)NC2(CCNC(c3cn(CCOC)nc3)=O)CCC2)nc(C)ncc1Cl Cc1[nH]nc2c1CC(C(N1CCN(C(c3cnc(O)nc3O)=O)CC1C)=O)CC2 N1(C(CCNS(CC)(=O)=O)=O)CCCC2(NC(=O)CCC(=O)NC)CCCC12 Cc1cc(NC(=O)CN(c2ccoc2)C)ccc1NC(=O)CC1CCCC1 C1(NC(CC=C)=O)CCN(C(c2ccc(-c3nn[nH]n3)c(Cl)c2)=O)CC1(C)C CC1(C(N2CCOC(C(=O)NCCc3ncccn3)C2)=O)CCCC1O CCCC(C(=O)N(C1CCC1)CCN(C)C)NC(c1ccsc1C#N)=O N1(C(C)=O)C(CNC(=O)C(C)Cc2ccncc2)CC1C c1(C(N2CCCC(CNC(c3nnc(C)s3)=O)C2)=O)ccc(=O)n(C)c1 N1(C(C2C(C)CC(=O)N2)=O)CCC(NC(c2ccc3c(c2)CC3)=O)C(C)(C)C1 N1(C(C(C)C(C)(F)F)=O)CCCc2ccccc21.c1(N)cc(=O)n(-c2ccccc2)[nH]1 c1(C(=O)NC2(C)CC(NC(CC3CCC(C)C3)=O)C2)ccc(O)nc1Cl C12(C(=O)NC(C)Cc3nn[nH]n3)CC(C)(CN1C(=O)CN1CCC(=O)CC1)C2 n1(CC)ccc(CC(=O)NC2(C(=O)NCCNS(=O)(=O)CC)CC(O)C2)n1 c1(N2CCC(C)(C(N3CCC4(CC3)CC4(F)F)=O)C2)[nH]cnc2nc(Br)cc1-2 C(=O)(CCCCC(=O)NC1CCC(N(C(=O)CC2C=CCC2)C)CC1)NC c1(CC)nccn1C(C)CC(=O)NC(C)CC1CN(C(=O)C(C)C2CC2)C1 C1(CNC(c2n(C)nc(C(F)(F)F)c2)=O)CN(C(C2CNC(=O)C2)=O)CC1(F)F C1(C(=O)Nc2n(CCC)ccc2)CCCCCN1CCNC(=O)NCCC(C)C CCCC(C)CC(=O)NCC(=C)CCNC(=O)C(C)OCCOC C1(C(N(C)CC2CCCN2C(=O)CCC2CCCCO2)=O)CC2CCC1C21CC1 N1(C(C2CCC(CC)O2)=O)CC(=O)NCC1C(=O)NC1(C)CCOC1=O c1(C(=O)NCC2CC(NC(CC(OCC)OCC)=O)C2)cnc(C2CC2)cc1C c1(NC(c2ncc(CCC(=O)OCC)s2)=O)cccc(Cn2cncn2)c1 C1(CC=C)(NC(c2coc(C(F)(F)F)n2)=O)CN(C(=O)COC)C1 C(c1ccccc1C#N)=CC(N1CC(NC(=O)C=CC2CCCO2)CC(C)C1)=O N1(C(=O)NC(CC#C)C(N)=O)Cc2ccc(C)c(Br)c2C1 CC1C(NC(c2n[nH]cc2Cl)=O)CCCN1C(C1CCN1C(=O)OC(C)(C)C)=O c1(C(N2CC(C)C(CNC(c3ccco3)=O)C2)=O)ccc(=O)n(CC(C)O)c1 c1(NC(=O)NC(C)CS(C)=O)ccnc(O)c1 C1(C(N2C(CNC(C=CC)=O)C=CC2)=O)CCC2(CCC2)O1.c12cccc(c1)S2 C1(NC(=O)CCC(F)F)CC(F)CN(C(c2cncc(C3CC3)c2)=O)C1 c1(C(=O)NC(CCOC)CNC(=O)C=CBr)nnn(C2CC2)c1C(F)F C12(CNC(COC(CC)C)=O)CC(CN1C(c1cc[nH]c1C1CCC1)=O)C2 CN1CC=C(CC(=O)N2CC(NC(=O)C(O)C3CC3)C(C)(C)C2)CC1 C(=O)(C(C#N)C(C)(C)C)N(CCNC(C1CCCC12CC2)=O)CC c1(C(C(=O)NCCCC)N(CCCO)CCOC)cccc(OC)c1 C1(NC(C(C(C)C)NC(C)=O)=O)CC(C)CN(C(C2CCCN2C(C)C)=O)C1 N1(C(C)=O)CCC(Nc2cccc(F)c2Br)c2cc(F)ccc21 C1(OC(c2cc(OC)cc(C(F)(F)F)c2)=O)CCc2nc(C)nn2C1 C(CNC(c1c(C)nsc1C)=O)(CC(=O)NCC(C)S(N)(=O)=O)OC C1(C(=O)NC(C(C(=O)OC)C)C)N(C(c2csnn2)=O)CCCC1(C)C C(=O)(C(O)C(C(C)C)OC)NCC1CC(O)(CNC(CCC(C)OCC)=O)C1 N1(C(C(CC)OCC)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)C(C)C1 c1(NCC(c2cccc(Cl)c2)COC)[nH]c(=NC2CCSC2)nc2scnc12 C1(C(=O)NCC2CCCO2)CCC(C(N2CC(C(=O)NC3CC3)C2)C)O1 C1(CCNC(c2noc(CC)c2C)=O)CN(C(C2CCCS2)=O)CCS1(=O)=O C(=O)(C1CC(=O)Nc2ncccc21)N(C(=O)CCCC1CCCCC1)C(C)C C(c1ccc(Cl)cc1F)=CC(=O)NC1(CCNC(C(CC)(C)CC)=O)CCC1 N1(C(CSCC#C)=O)CC2CS(=O)(=O)CC2(CNC(c2ccnnc2C)=O)C1 c1(OCC(=O)NCCNC(=O)C(=O)NC2(C(=O)O)CC2)ccccc1 c1(C(=O)NCC23C(CN(C(CC4CC(OCC)C4)=O)C2)C3)ncc(N)cc1C Cc1nc(CNC(C2(NC(C3CC3C(N)=O)=O)CC2C)=O)no1 C1(CN(C(=O)Cn2ccnc2C)CC)CCCCN1C(=O)Cn1cnnc1O CC(C)CC(C(=O)N(C)CC1CCCCO1)NC(=O)C(F)C(C)(F)F C1(C(=O)OC)CC12CCN(C(C1(C)CCN(C(c3sc(Br)nc3C)=O)C1)=O)CC2 c1(SC)ccc(C)c(C(=O)NC(C)(C)CCNC(C2(CO)CCOCC2)=O)c1 c1(C(=O)NCC2(C)CCCN(C(C3OCC(C)C3)=O)C2)cn2cc[nH]c(=O)c2n1 C1(C)(NC(c2scc(C)c2)=O)CCN(C(C2CCCC2C(C)C)=O)CC1 C(=O)(C(C)Cc1ccco1)NCCC(C)N(C(C1CC(C)C1)=O)C C#Cc1cncc(C(N2C3CCC2C(CNC(=O)CC2(C)CCC2)C3)=O)c1 C=CC1CN(C(c2csc(-c3cnc[nH]3)n2)=O)CC1NC(C1(C)COCCO1)=O c1(N(C)C)cc(-c2ncccc2C(N2CCC23CCNCC3)=O)cc(C#N)c1 c1(C(=O)NC2C(NC(CCC=C=C)=O)CCOC2)nccn(CC(F)(F)F)c1=O C(C(F)(C(=O)N(CC(C)(C)COC)C)C(C)C)NC(c1c(C)cc(CC)o1)=O CCC(CC)OCC(=O)NCC(C)CNC(C1CC(OC(F)F)C1)=O C1(C(N)=O)(CC)CCCN1C(=O)Cc1cc[nH]c1.C12CC1C(=O)NC2 N1(C(C2(C(=O)OCC)CCO2)=O)CC2CN(C(=O)CC(C)C(F)(F)F)CC(C1)O2 C12(CNC(C3(N(C)C)CCC3)=O)CC(CO1)N(C(C1CCCS1)=O)C2 C12CCC(C1)C(=O)N2C(c1c(C(c2cnoc2C)=O)c[nH]n1)=O.CO N1(C(CCOC)=O)CCC2(CC2C(=O)NCCc2ccn(C(C)C)n2)C1 N1(C(C2N(C(C)=O)CCC2)=O)C2CCC1(CNC(=O)C=Cc1ccc(C)s1)CC2 c1(C(=O)NCC#CCNC(c2cnc(C(C)(C)C)s2)=O)cscc1C#N c1(C(=O)NC2C(C)CN(C(C3(C#N)CC=CC3)=O)CC2)ccn2c1CCCC2 Cc1cccc(C(N2CCCC2CN(C)C(C2CC3CC2CO3)=O)=O)c1C Cc1cc(NC(=O)CN2CCC(C)(N(C)C)C2)c(C(=O)O)cc1C C(=O)(C1=COCCC1)N1CCCC(N(C(CCC=C(C)C)=O)C)C1 c1(C(C(=O)N(CCC)CCN)O)ccc(OC)cc1.C1(=O)CCSCC1=O.CC C(=O)(C1=CCN(C(=O)CCCCC#N)C1)N(C(C)CS(C)=O)C C=C(C)CCC(=O)N1CC(F)CC1CN(C(=O)C(C(C)C)c1ccn(C)n1)C c1(C(=O)NC2CC(CNC(C(CC)SC)=O)C(O)C2)c(C)cc(C#N)cc1C C(N=c1ccnc(N2CCCC(OCCNCC)C2)[nH]1)C1(N(C)CC)CCOC1 c1(C(=O)NC(CCCNC(CCC(=O)NCC)=O)C)ccc(C#N)c(OCC)c1 Cc1c(C(=O)NCC(O)CCNC(=O)CC2CC(C)C2)nnn1-c1ccccc1 C1(NC(COC(C)C)=O)CC2CC1N(C(=O)Cc1cccnc1)C2 c1(C(=O)NC2CN(Cc3c(C)n(C)nc3)CC2(F)F)ccc2cnccc2c1 C1(NC(c2c(C)ncs2)=O)CC2CC1CN2C(=O)C(C)(C)C(=O)N1CCOCC1 C(=O)(C1CCCn2ncnc21)N1CCCC(NC(CC=CC=C)=O)(CO)C1 O=C(CC1NC(=O)c2ccccc21)NCCC1(O)CCN(C(c2cocn2)=O)C1 c1(OC)ccc(C)cc1C(=O)N(CC(O)CN(C(=O)CC1CNC(=O)C1)C)C c1(C(=O)NCC(CC=C)NC(=O)Cc2nonc2C)ccc2c(c1)NCC2 c1(C(=O)NC(C2CN(C(c3c(C)cc[nH]3)=O)CCO2)C)nc(C)n(C)c1C C(=O)(C(C)(C)F)NCCNC(=O)NC1CN(C(C(C)C2C(C)C2)=O)C1 c1(C(N2CCC(OC)C(OC)C2)C(=O)NC(CC)(C)C)ccc2c(Br)cccc2c1 c1(C(=O)NC2CCCCN(c3c(C#N)nccn3)C2)ccc2c(c1)CCCS2 C1(C(=O)NCCN(C(=O)C(F)CC2CCC2)C)CCOCC12CCCC2 C1(NC(c2nccc(CC)c2)=O)CN(C(=O)CCc2ccc(C)s2)CC1(C)C C1(C(N(CC(CC)(C)OC)C)=O)CC2(CC(NC(=O)C(C)N3CCCC3)C2)C1 CC1CN(C(=O)CC2CC3CC3C2)CCCN1C(=O)CNC(=O)C1CC1 N(C(=NCCCCl)NCC(C)C1CC1)CC(=O)N(CCOC)C1CC1 Cc1cc(C(N)=O)cc(C(=O)NC2CC(NC(c3ccc([N+](=O)[O-])[nH]3)=O)C2)c1 c1(CC(N2CC3(CC(NC(COCC(=O)NC)=O)C3)C2)=O)nc2ncccn2n1 C(=O)(CC(C)C(C)(C)NC(c1cn2c(n1)CCC2)=O)NC(c1ncc(C)o1)C CN1CCCCc2cc(NC(N3CCSCC3c3ccccc3)=O)ccc21 C=CCCC(CO)NC(CCCC#N)c1nnnn1CCOCC C=Cc1cc(C(=O)Nc2ccc(NC(c3cncnc3)=O)c(C)c2)cc(F)c1 CC1CN(C(c2c(NC(C3CCN(C4CC4)CC3)=O)ncn2C)=O)CC(C)S1 c1(OC)cc(-c2nccn2-c2ncn(C)n2)cc(-c2cnn(C)c2)c1OC c1(C(=O)NC2(C)CN(C(=O)CCNC(c3ccoc3)=O)C2)cc([N+](=O)[O-])c[nH]1 Cc1nc(C(=O)NCC(CNC(=O)CC2CCOCC2)S(C)(=O)=O)cn(C)c1=O N1(C(C(C)SC)=O)CC2(CCN2C(c2cnn(C)n2)=O)C1 C=CCCC(C(=O)NCC1(CC2CC2)CC1)NC(=O)CC1CN2CCC1CC2 C1(C(=O)NC(CC(C)C)CNC(=O)CCCF)CC2C(C1)C2(C)C Cc1nc(NC(c2cccc(-c3cnn(CCO)c3)c2F)=O)cnc1C#N c1(CC)c(C(=O)NC(C)(C)CCCNC(c2nc(C3CC3)sc2C)=O)ccn1C C=CC1(C(=O)NC2CC2NC(c2cc(CC)ccn2)=O)CCCCC1 CCCCC(CNC(=O)CCCF)NC(C1(c2ccccc2)CC1(Cl)Cl)=O c1(C(N2CC=CC2CNC(C2CC(O)C2)=O)=O)cc(Br)c2nccn2c1 C12CC3(C1)CC(C3)NC(=O)O2.C1(C(=O)OC)CCCC(=O)N1C(=O)C1CC1 CC(CC(=O)NCC1C=CC(NC(=O)C(C)(C)c2cnsc2)C1)NC(N)=O C1(CC)(NC(c2ccc(-c3cnc(C(F)(F)F)nc3)o2)=O)CCNC1=O CCC(CC(=O)NCCCCCCNC(=O)COCc1ccnc(O)c1)C(F)F Cc1coc(C)c1C=CC(=O)N(C1CN(C(c2ncsc2C2CC2)=O)CC1O)C N1(C(CNC(=O)OCC)=O)CCC(C(=O)NCc2nn(C)c(=O)o2)C(C)(C)C1 N1(C(C(C)n2cncn2)=O)CC2(C1)SCCC2NC(=O)Cn1ccc(C2CC2)n1 CCC(CC)C(C)C(=O)NC1(C(=O)N(CC(=O)OC)C2CC2)CCC(C)(C)C1 N1(C(c2n(CC)nnc2)=O)CC2(C1)CN(C(c1cc(C3CC3)[nH]n1)=O)C2 CCC(CC)CC(=O)NC(CC(=O)N(C)Cc1c(C)noc1C)C(F)F C1(CC)CN(C(=O)CSc2nncs2)CCC1NC(=O)CC1CCC(F)(F)CC1 c1(-c2c(C)cc(C(=O)NC(C)C(F)(F)F)nc2)ccc([N+](=O)[O-])cc1 N1(C(CCC(C)OCC)=O)CCN(C(=O)C(C)(C)CC)CC1C1CC1 C#CCC(C(N)=O)NC(C1(CF)CCN(C(=O)CCSCC)C1)=O C(=O)(NNC(=O)Cn1ncc(Cl)c1C)c1c(-c2cn(CC)nc2)cccc1 c1(C(=O)NC(CN(C(C(C)NC(C2CCC2)=O)=O)C)(C)C)cc(Cl)c(N)c(Cl)c1 N1(C(C2C(C)C2)=O)CCC2(CCCN(C(c3cc4cccnc4cc3O)=O)C2)C1 N1(C(C2CCN(C(C(CC=C)(C)CC)=O)CC2O)=O)CC2(C1)OC(=O)NC2C c1(NCc2ncc(CC)[nH]2)cc(N(C)CCc2ccc(C)cc2)ncn1 N1(C(c2cc(CCOC)on2)=O)CC2(CCCC2NC(=O)CN(C)C(C)=O)C1 c1(C(N2CCC(C3CCN(C)C3)C2)=O)ccc2c(c1F)NC(=O)CO2 Cc1cc(C(N)=O)cc(C(=O)NCC(C)N(C)C(C2CC(O)C2)=O)n1 c1(CC(C(=O)NC(C)CCCNC(c2ncncc2Cl)=O)O)c(F)cccc1Cl O=C(CCC(F)(F)Cn1cc(COC2CCCC2O)nn1)NC1CCCCCC1 CC(C)CC(O)C(=O)N(CCNC(=O)C(c1ccccc1Cl)O)C1CC1 C(=O)(CCCC(CC)NC(=O)CSCCOC)NCCS(CC)=O c1(N(C)CC2CCC(=O)N2)nc(N2CCC(C(F)(F)F)CC2)nc2c1ncn2C Cc1ccc(C(=O)NC2CCN(C(C34CC(C3)S(=O)(=O)C4)=O)C(C)C2)cc1C CCCC(C(O)C(=O)NCCc1cccs1)NC(=O)Cn1ncn(C)c1=O C(=O)(C1=CCCN(C(=O)CCOCC(C)C)C1)N1CCC(CC(=O)OC)C1 S(=O)(=O)(c1ccc(N(CCC(N)=O)C)c(Cl)c1)NC1CC(C)N(C)CC1 c1(NC(=O)CC2(O)CCCOC2)ncnc(Cl)c1Br.N12CCN(CC1)C2=O c1(C(=O)NC2(C)CCCN(C(=O)CC3CN4CCC3CC4)C2)cccc([N+](=O)[O-])c1 C1(CC(=O)OC)CCC(NC(=O)NC2CN(C(=O)CC(C)C)CC2F)CC1 Cc1cccc2c1N(C)C(=O)C2NC1CCOC2(CCOCC2)C1 C1(C2CCN(C(C3CCCN3C(C)C)=O)CC2)(NC(CS(=O)(=O)NC)=O)CC1 N1(C(C2C(C)(C)CCC2)=O)CC2CC1CCC2NC(c1cc(C2(C)CC2)on1)=O c1(C(N2CCC(NC(C3(CC=C)CCC3)=O)C(F)C2)=O)ccc2nc[nH]c2c1F C1(CNC(Cc2c(C(N)=O)cccc2)=O)CC2(CC2)CN1C(C1CCSCC1)=O c1(C(=O)OC)ccc2c(c1)N(C(=O)NCC(COC)C(C)C)CC(=O)N2 c1(CC)cc(C(=O)NC2CC(CCNC(C3CCNC3=O)=O)C2)oc1CC C=CC1CN(C(=O)Cc2ccc(Cl)cc2)CC1NC(=O)C=CC1CCOCC1 C12=NC(C)=CC(=NC(C)CNC(=O)N3CC(C)N1CC3C)N2.C(C)(C)(C)OCC C(CN=c1nc(-c2ccc(C)cc2)[nH]s1)=CCNC(C(C1CCCC1)OC)=O CC(CC(N)=O)C(=O)NC(c1ccccc1)c1nc(CCc2ccccc2)no1 C(CCCCCC(=O)NCC1CN(C(C2(F)CCOCC2)=O)CC1C)SC c1(NC(C2C(NC(C(=O)NCCOC)=O)CCC2)=O)ccc(Cl)cc1C N1(C(c2cc(Cl)ccc2F)C(=O)NCCC2CC2)CCCc2[nH]ccc2C1 c1(C(N2CC(OC)C(NC(=O)C(F)F)C2)=O)nc(C)n2ccccc12 N1(C(c2ccc(SC)cc2)=O)CC(NC(=O)C(C)Cn2cccn2)C(C)(C)C1 c1(C(=O)OCC)coc(C(=O)NCC(C)N(C(=O)C=CSC)C)c1 N1(C(C2ON=C(C)C2)=O)CCCC(C(N(C)Cc2ccc(N3CCC3)nc2)=O)C1 N1(C(c2ccc(F)c(C)c2Cl)C(=O)NCCCSCC)CCCC2(CCOC2)C1 C1(CNC(C2(CC)CCCCC2)=O)CN(C(C2OCCO2)=O)CCC1C(F)(F)F Cn1cc(C(=O)NCC(C)(C)CC2CN(C(=O)CC3CC3C(F)(F)F)C2)cn1 C(=O)(C(C)(O)CNC(=O)C(C)N(C(C1(C)COC(=O)N1)=O)C1CC1)OC O(NC(=O)C1=NOC(CNC(c2ccon2)=O)C1)CC(C)C C1(CC(=O)NC(CCC=C)C2CC2)C2CCCC2N1C(=O)CC1CSCCO1 N1(C(CSc2ccc(OC)cc2)=O)CC2CC(C)N(C(=O)C(C)(F)C(C)(C)F)C2C1 C=CC(C)(CCOC)C(=O)N1Cc2occ(C(=O)NCC3(CO)CC=CC3)c2C1 c1(C(N2CCC(NC(C3CCOC3=O)=O)(CF)C2)=O)cc(F)ccc1Br C#Cc1cn(C)nc1C(=O)NCCC1CCCN(C(=O)CCc2cc(C)on2)C1 CC1(CNC(c2cnc(C3CC3)s2)=O)COCCN(C(c2csc(=N)[nH]2)=O)C1 c1(C(N2CC(CCNC(c3n(C)cc(C(N)=O)c3)=O)C2)=O)ccc2[nH]ccc2c1 c1(C2C(C(N(CCCN(CC=C(C)C)C)C)=O)C2)cccc(C)c1 Cc1nc(N2CCC(C(C)NC(=O)CC3CC3(Cl)Cl)C2)cc(Cl)n1 c1(C(N2CC(C3CN(C(C4(O)CC4)=O)CCO3)C2)=O)ccc(Cl)c(C(F)F)c1 C1(NC(C2C=CC(NC(CC(COC)C)=O)C2)=O)CCCCCC1C(=O)OC Cc1cc2c(cc1C(N1CCC3(CC1)CC3NC(c1ocnc1C)=O)=O)OCO2 c1(N2CCC(C)(NC(C3CC3(F)F)=O)C2)ncnc2scc(Br)c12 C1(NC(c2cccnc2-n2cccn2)=O)CCCN(c2ccccc2F)C1 C(=O)(N=c1ccn(C2CC2)[nH]1)C1(C2N(C(C(n3ccc(C)n3)C)=O)CCC2)CC1 C(=O)(C(Cc1ccccc1)CC)NCC1C(NC(C=CC(CC)C)=O)C1 CC1CN(C(C2(C)CCC(C)C2)=O)CC1CCNC(C1(C(N)=O)CC1)=O N1(C(C(C)OCCC#C)=O)CCN(C(c2cccn2CCOC)=O)CC1C(F)F c1(C(=O)NC2(CC(=O)Nc3ccnc(Cl)c3)CCC2)ccc(Cl)cc1Cl N#Cc1cc(C(=O)NC2CN(C(c3c[nH]nc3C3CC3)=O)CC23CC3)ccc1Cl c1(OC)cc(N)c(C(N2CCC(C(F)(F)F)CC2)=O)cc1OC C1(NC(c2nc(NC=O)sc2)=O)CCC(C2CC2)CC1 c1(C(N2CC(CN(C(C(C)CF)=O)C)C2)=O)nccnc1Cl c1(C(N(CCCCN(C(CC2C(C)C2)=O)C)C)=O)ccnc(F)c1F C1(COC)(NC(c2cnc(O)cc2C)=O)CCN(C(=O)C(COC)N(C)C)CC1 c1(C(=O)NC2CCCC(CNC(C(F)=CC)=O)C2)ccc(OC)c(F)c1N Cc1cncc(C)c1C(=O)NCCCC(=O)NCC(C)C(C)(C)C CCCC(CNC(C1CC(=O)CC(=O)C1)=O)C(=O)N1CCSCC1C1CC1 N1(C(CC=C(C)C)=O)CCCC1C(C)(C)CNC(C1CC1c1ccccc1)=O c1(OC)cc(F)c(C(N2CCC(O)(CNC(c3nnn(C)c3N)=O)C2)=O)c(Cl)c1 N1(C(c2ccc(Br)c(C)c2F)=O)CCC2(CC1)CCN(C(=O)C(O)C(C)C)CC2 C1(CNC(C(C)=C2CCCC2)=O)C2CN(C(C3(C)CCCCO3)=O)CC12 c1(CC)nc(CCNC(=O)C(=O)N(c2ccccc2)CCC#N)cs1 C(C(=O)NNC(=O)C(C)(C)S(C)(=O)=O)(C(C)(C)C)N(c1nn(C)cc1Cl)C C=CCCC(C(=O)NC1CC(CC)C1)NC(C1CC(F)C(=O)N1)=O c1(CC)ccnc(N2CCN(C(=O)CC3CCC(C(=O)NCC4CC4)O3)CC2)c1 N1(C(c2cnc(COC)s2)=O)CCC(N(C(c2cc(C3CC3)on2)=O)CC)CC1 C1(N(C)C(C2(C)CCCN2)=O)CCCN(C(c2ccc(-n3cncn3)cc2)=O)C1 C1(NC(Cc2nnc(C)o2)=O)CCCCCN(C(=O)CN(C)C)C1 Cc1nc2cc(C(N3CCCCC(NC(c4sncc4C)=O)C3)=O)cc(O)c2o1 C(CC(=O)N(CC(O)C1CCC1)C)N(C(=O)C(=O)N(C)C)C(C)C Cc1ccc(Br)c(CNC2(CC(=O)Nc3cnc(Br)c(F)c3)CCC2)c1F c1(C(=O)NC2COCCN(C(C3(CC(C)C)CC3)=O)C2)ccnc2ccnn12 C1(CNC(=NCCC)NCC(c2cnn(C)c2)C)CC2(CO1)CC(OC)(OC)C2 c1(C(N2CCC(CCC)C2)=O)cccnc1CNC(C1CC(=O)C1)=O C12(C(=O)NC(CC)(C3CC3)C3CC3)CCCC1CN(C(=O)Cc1ccns1)C2 C(=O)(CCCC(C)CC)NCCC1CCCN(C(CC2(OC)CCCC2)=O)C1 C1(CNC(C2(OCC)CCC2)=O)CN(C(=O)COc2ccncc2)CCCO1 C1(NC(c2n(CCC)nc(C)c2)=O)CN(C(=O)C(C)=CC2CC2)CC2CCCC12 c1(-n2cc(CN(C(C3CCC3)C)CC)nn2)cccc2n[nH]cc12 c1(C(=O)OC2CC2C(c2ccccc2)=O)ccc(C(F)(F)F)c(F)c1 c1(C(=O)NC(CNC(c2nc(CC)oc2)=O)(C)C2CC2)cnn2ncccc12 C1(NC(c2c(CC)scc2)=O)CC2(CCN(c3cc(C(C)(C)C)ncn3)C2)C1 N1(C(C(c2ccccc2F)C)=O)CCC(CNC(C2(C)CC2(Cl)Cl)=O)CC1C Cc1sc(C(N2CC(NC(C3(CF)COC3)=O)CC(O)C2)=O)cc1[N+](=O)[O-] c1(CC(=O)NC(CNC(c2nc(C)n(C)c2C)=O)C(C)C)ccc(F)c(Cl)c1F N1(C(c2c(C)cccc2)=O)CCCCCC(NC(c2ccncc2F)=O)C1 N1(C(C(N(C(=O)COCc2ccn(C)n2)C)C2CC2)=O)CCC(N=[N+]=[N-])C1 CCC(CNC(c1cc(Cl)cs1)=O)(CC)C(=O)NC(c1ccccc1)C C1(NC(Cc2n(C(C)C)ncc2)=O)CCC2(CCN(C(C3CC=CC3)=O)CC2)C1 Cc1cc(C)c(C(=O)NC(C)CC(C)NC(C23CC2COC3(C)C)=O)c(N)c1 c1(C(N2C(c3ccc(OC)cc3)CNCC2)=O)nn2c(c1Br)CCC2 c1(OC)ccc(F)c(CNc2cnc(F)cc2C(=O)Nc2cc(Cl)nc(C)n2)c1 O=C(C(=O)N(C(C1CCCC1)CO)C1CC1)NCC1CCCO1 C1(CNC(C2CC(NC(c3n(C)cnc3)=O)C(O)C2)=O)CC2C(C1)C2(F)F c1(SC)ccccc1CC(=O)N(C1CCCC(N(C)C(c2ccc(Cl)o2)=O)C1)C c1(C(N2CC(NC(C(CC)NCC)=O)(COC)C2)=O)cnc2cc(C)ccc2c1 C1(NC(C2CCC(C)C(C)C2)=O)CCCC2CN(C(=O)C(C)(C)CCC#N)CC12 c1(CNC(CCN(C(C2CC(=O)CS2)=O)CC)=O)cnc2n1CCC2 Cc1cc2scc(CC(N3CCC(C)C(NC(=O)CSc4cccs4)C3)=O)c2s1 N1(C(C(c2cccnc2)NC(c2cc(C)cc(O)c2)=O)=O)CCCC2(CCC2)C1 c1(C(c2n(CCOC)nnn2)NC2(c3nccs3)CC2)cccc(Br)c1Cl c1(C(N(C2CCN(C(c3nc(=N)cc[nH]3)=O)C2)CC)=O)cc([N+](=O)[O-])oc1C C(N=c1[nH]c(Cl)ncc1F)c1nc(NC(CC(C)N(C)C)=O)sc1 C1(C(N2CC(CNC(CCc3c(C)n(C)nc3)=O)C2)=O)CNC(=O)CC1C c1(C2C(C(N(CC)CC3(C(F)(F)F)N=N3)=O)C2)c(F)cccc1F c1(CN2CC(C)(C(N(C3CCS(=O)(=O)C3)C(C)C)=O)C2)cc(F)c(O)cc1F C1(C)(C(=O)NCC(CCCC)NC(=O)C(=O)NC(C)C)CCN(C)C1=O C12(C(=O)NC(c3nc(CC)on3)C)CCCC1CCN2C(C1CCS1(=O)=O)=O C1(C(N(CCNC(CC2(C=C)CC2)=O)CCC)=O)CCc2ccc(F)cc2C1 c1(OCC(=O)OCC)cccc(CC(=O)NCC(C)CNc2csc(O)n2)c1 C(=O)(CC(C)CNC(c1ccc(O)nn1)=O)NCCCc1onc(C)n1 N1(C(C2CC(C)(C)OCC2)=O)CCC2(CCC2NC(=O)Cn2ccnn2)CC1 c1(CC)ncnc(CC)c1C(N1CCC(N(C(=O)C(CC)C2CCC2)C2CCC2)C1)=O CC(C)C(CCN(C)C(c1cc(Br)c[nH]1)=O)NC(=O)Cn1ccc(C(F)F)n1 CC(C)(CN=c1ccc(Br)c(S(=O)(=O)N2CCOC(CCF)C2)[nH]1)NC C1(CC(=O)NC(C)(C)C)CCCCN(C(=O)C#CC2CC2)C1 n1(CC)nc(C)c(C(N2CC(NC(=O)Cn3cncn3)CC(C)C2)=O)c1C(F)F c1(CC)oc2ccccc2c1C(=O)N(C)CCN(C)C(c1ccnc(Cl)c1)=O C1(F)(CNC(C2(OC)CCC2)=O)CCCN(C(=O)C(F)C(C)(C)O)C1 C1(C(N2CC(NC(C3C(C)=C3)=O)C(C)C2)=O)CCC2C(C1)C2(F)F c1(C(=O)NC(CNC(C=CCC)=O)CC)ccc(OC(C)(C)C)cn1 Cc1nc(C#N)ccc1C(N1CCC(C(C)NC(c2cnccc2Cl)=O)CC1)=O C1(N(c2ccc(N3CCNC3=O)cc2)C(C(=O)N)=O)CCCCN(C2CCC2)C1=O.C c1(C(=O)NC(CNC(c2cc(C(N)=O)[nH]n2)=O)C2CC2)cc2c(nn1)CCOC2 N1(C(=O)Cc2ccc3c(c2)OCO3)CCC2CN(C(C3(F)CC3)=O)CCC12 C(=O)(C1=C(Cl)CCC1)N1CC(CCNC(c2c(CC)ccs2)=O)C(C)C1 c1(C(C)C(=O)NC2(CF)CCN(C(=O)Cn3cnnn3)C2)noc2ccccc12 C(CC(C(C)(C)C)NC(=O)CNC(=O)CN(C)C)N(C(C(CC)(F)F)=O)C C1(NC(C(C)CC2CC2)=O)CN(C(c2cccc(C(C)(C)C)c2)=O)CC12CCC2 Cc1nn(C)c(N)c1C(=O)NCC1CC(C)N(C(=O)C=Cc2ccncn2)C1 c1(C(N2CCC(n3cc(CCCSCC)nn3)CC2)=O)ccnc(OC)c1Br C(=O)(C(F)CC(C)(C)C)NCC(C1CCOC1)NC(c1cncc(CC)c1)=O Cc1cc(C(N2CCC(CNC(C3CCC(=O)NC3)=O)C2)=O)ccc1Br c1(C(C)C)ccc(N)c(C(=O)NC2CN(C(=O)CN(C3CCSC3)C)CC2C)c1 c1(SC)cccc(-c2nc(C)c(C(=O)NCCCOC(C)(C)C)s2)c1F N1(Cc2cn(CCNC(CCCCN(C)C(C3CC3)=O)=O)nn2)CCC(C#N)CC1 C1(CC#C)(C(N2CC3(NC(c4ncccc4Cl)=O)CC2C3)=O)CC=CCC1 c1(C(=O)NC(C2CCCN(C(c3ncccc3Br)=O)C2)C)cc(I)cnc1Cl C(=O)(CCCC(C)(C)C#N)N(CCNC(c1cn2c(n1)CC(C)CC2)=O)C1CC1 c1(C(C)OC)nc(C)c(C(=O)NC(CO)C(C)NC(c2cccc(Cl)c2)=O)s1 C1(NC(C2C(C(=O)NCC(C)C)C2)=O)C2CN(C(=O)CN(S(C)(=O)=O)C)CC12 c1(C(=O)Nc2c(NC(c3cccc(Cl)c3)=O)cc(Cl)cc2)c(O)ccc(Cl)c1O c1(OCC)ccc(CCNC(=O)N(C2CC2)CC2CNC(=O)CO2)cc1OC C1(NC(c2cc(CC)on2)=O)C2CC1CN(C(C1CCC(F)C1)=O)C2 N1(C(C(C)O)=O)CCCCC1c1cn(Cc2nccs2)nn1 C(=O)(C(C)CC(=O)NC(CC1CC1)C(=O)Nc1cnc(OC)cc1C)OC c1(C(=O)NC(C2OCCN(C(CC=C)=O)C2)C)cc(Br)ncc1OC c1(C(=O)NC2(CNC(CC3(C)CC3(F)Cl)=O)CCCC2)ccc2[nH]c(=N)[nH]c2c1 C1(CCNC(=O)CC2CC3CC3C2)COCCN1C(=O)CCN1CCCCC1=O N1(C(C2(C(C)C)CC2)=O)CCC(NC(=O)Cc2cccnc2Br)C(O)C1 C1(C(=O)NC(CC)C(C)(C)O)CCCCCCN1C(=O)CC1CCC(O)C1 c1(OC)ncc(C(C(=O)NC(C)C)N(C)Cc2ncsc2C)cc1Cl N1(C(CCOC(C)=O)=O)CC2(CCCCN(C(=O)CC3CC3(Cl)Cl)C2)C1 c1(C(=O)NC23CC(C(=O)Nc4ccc(C)c(O)c4)(C2)C3)cc(Br)c(O)cc1O C=C(C)CC(C(=O)N1CCC1COC)NC(C1CC2CCC1CC2)=O Cc1nc(NC(=O)NCC2CCC3(CC3)C2)c(C)o1 C(CCCCC(=O)NCc1cc(=O)cc[nH]1)N(C(=O)Cc1ccc(F)cc1)C C(=O)(CCCC(=O)N1CCC(COC)(NC(c2ccc(C(C)=O)[nH]2)=O)C1)NCC C1(C(=O)NC2CN(C(Cn3nc(C)c(C)c3C)=O)C2)CC2C=CCC(C1)C2 C#CCC(CC(F)F)C(=O)NC1CCOC1C(=O)N(C)Cc1cccc(O)n1 c1(CNC2C(C(=O)NCc3cnc[nH]3)C2)ccc(Br)nc1Br c1(CC(=O)N(CCNC(CSCC=C)=O)CC)cnn(C)c1 C(=O)(C1CCc2nccn21)NCCCN(C(C1CN(C(C)C)C(=O)C1)=O)C(C)C N1(C(C(C)OCC=C)=O)CC(C(=O)Nc2cnccc2SC)CC1(C)C C1(C(=O)NC2C=CC(C(=O)OC)C2)(CCl)CCCN(C(=O)C(C)CC2CC2)C1 c1(C(=O)NCC2CCCC(NC(CSCC=C)=O)C2)nc(C)[nH]c2nccc1-2 N1(C(C2(CN(C)C)CC2)=O)CCC2C(C1)CN2C(=O)CSCC1CCCO1 c1(C(N2CCCCC2COC)C(=O)NCCOC)ccc2c(c1)C(=O)NCCO2 C1(CNC(C(c2ccccc2)OC)=O)C2CN(C(=O)C(c3cccnc3)C)CC12 c1(CC(=O)N(CCNC(C2(C)CCOC2)=O)CC)cnn2c1OCCC2 CCCCCCC(=O)NC(CN(C(=O)CC1CCCC(C)(C)O1)CC)CC C12(C(=O)NCCN(C(=O)CSc3ccc(C)cc3)CC)CC3CC1C2C3O c1(CCOC)nsc(N2CCC(C(C)OC)C2)n1.C12CC(C)(C1)NC2=O c1(CN(C)C(C2C3CC2N(C(=O)C(F)C2CCC2)C3)=O)ccncc1F c1(C(=O)NCCCCNC(C2(C#C)CC2)=O)cn(C(C)(C)C)cn1 N1(CC)CCOCC1C(=O)NC1CN(C(c2csc(-c3ccc(C)cc3)n2)=O)C1 C#CCC(C)(C(=O)NCc1ncnn1CC)NC(=O)C1CC1 c1(OC)ccc(F)cc1C(N1CC(O)(CNC(=O)Cc2nncn2C)C1)=O Cc1nc2sccn2c(=O)c1CCN=c1ccnc(N2CCC(C3CCC3)C2)[nH]1 Cc1cc(Br)sc1C(N1CCC(C)C1CNC(c1cocn1)=O)=O c1(CC(=O)NC(C)CCNC(=O)CCN2CCN(C)CC2)cc(F)ccc1F c1(C(N(C)CC2CN(C(C(COC)OC)=O)CC23CC3)=O)cc(OC)cc(N)c1 C(=O)(C(=O)C(F)(F)F)NCC1C(NC(c2c(CC)c[nH]c2)=O)CCC1 Cc1cccc2c(=O)c(C(=O)COC(c3cn(C4CCCCC4)nn3)=O)c[nH]c12 c1(CC)cccnc1C(=O)NCc1ccc(C(=O)NCC(F)Br)o1 c1(OC)nc2ccccc2cc1CC(=O)Nc1cn(CCN2CCNCC2)nn1 CC1CC2CN(C(C3CCCN3C)=O)CC2N1C(=O)CCCC(N)=O c1(N2CC(CCOc3ccc(NC(C)=O)cc3)C(C)C2)nccc(C#N)n1 N1(C(C=CCN(C)CC)=O)CCCC(O)(CNC(=O)CCOC2CCCC2)CC1 C(C(=O)NCCC1CC1)(C(c1ccccc1)OC)N(C1(COC)CCSC1)C Cc1csc(=O)n1CC(=O)NCCC1CCC(NC(=O)CN2CCCCC2=O)C1 c1(CC(=O)NCCC(CCNC(C(C)(C)OC)=O)C)cnn2c1CCCC2 C1(NC(C2(C)N(C)CC(O)C2)=O)CC2CC1CN(C(C1CCC1C(C)(C)C)=O)C2 CC(=O)CCCC(C)C(=O)N1CCC(N(C(=O)C(C)CF)C)CC1 CCCCC(F)C(=O)NCC(CO)(CO)NC(c1cccnc1N(C)C)=O Cc1cc(O)ccc1NC(C1CN(C(C2CCC(=O)CC2)=O)CC1F)=O C(=O)(C(C)(O)Cc1ccccc1)NCC1CN(C(CC2CC(COC)C2)=O)C1 C1(C)(C(N2CC(C)(NC(CCC=CC(C)C)=O)C2)=O)CCCCC1(F)F c1(C(=O)NC2CC(C)N(C(c3cnc4[nH]cncc3-4)=O)C2)c(N)cc(Cl)cc1F CC1(C)OCCN2C(=O)N(C3CC3(c3cccc(F)c3F)C)CC12 CCCC(CC(C)C)C(=O)NCCC1CCN(C(=O)C(C)(CC)CC)C1 N1(C(C2CCN(C(C)C)C2)=O)CC2(CC2C(N2C3COCC2C3)=O)C1 c1(C(=O)NC(C2(O)CCN(C(c3c(C#C)c[nH]n3)=O)C2)C)ccc([N+](=O)[O-])nc1 c1(CC(N2CCC(C)(NC(C3CCCCN3N=O)=O)C2)=O)n[nH]c2ccccc12 CC1=CC(C(=O)NCC2CC(C(=O)NCC(C)C#N)CO2)SC1 c1(C(=O)NCC(C)(C2CCC2)NC(C(c2ccccc2Cl)C)=O)cnc(S)n1C N1(C(C2(CC)CC2)=O)CCN(CCNC(C2CCC(=C3CCC3)CC2)=O)CC1 C(=O)(CCC(=O)C(C)(C)C)NCC=CCC(NOCCCC)=O c1(CC)ncc(C(=O)NC(CNC(=O)C(C(C)C)NC(C)=O)(CC)CC)cn1 c1(-c2n(CCC)nc(Cn3ccnn3)n2)cc(Cl)ncc1F CN=S1(=O)CCN(C(c2c(C)cc(=O)oc2C)=O)CC1 c1(C(C)C(=O)NC2CCC2NC(c2n[nH]cc2C2CC2)=O)ccc(C#N)cc1 N1(C(CCOCC(C)C)=O)CCC2(CCC(NC(=O)C3=CCC(C)CC3)C2)C1 c1(C(c2nnnn2CC)NCCCC(=O)NCCC)c(Cl)cncc1Br N1(C(c2cc(OC)ncc2)=O)CCCC(C)(C(N2CCC3CCC23)=O)C1 C(=O)(CCNC(=O)NCC(C)(C)S)OC(C)C.C(C)(C)(C)OC=O C(=O)(C1=C(Cl)CCC(C)C1)NC(CN(C(c1cn(C)c(=O)nc1O)=O)CC)C c1(CNC(C2C(C3N(C(CC)=O)CC(C(F)(F)F)OC3)C2)=O)cc([N+](=O)[O-])cn1C S(=O)(=O)(c1ccc(NCC23CC(NC)(C2)C3)cc1Br)NC(COC)=O C1(NC(c2c(-n3cc(CCC(C)O)nn3)cccc2)=O)CCc2ccccc2C1 N1(C(Cc2ccc(C)cc2)=O)CCC(CNC(C23COCC(C2)C3)=O)C(F)(F)C1 C1(N(C(c2cnc(C(C)C)nc2)=O)CC)CCCN(C(c2cc[nH]c2)=O)CC1 C(=O)(C(C)(C)C1=CCN(C(=O)CC2CCC(C)(C)C2)C1)NCC1CC(C)OCC1 c1(C(=O)NC(C)CNC(C2(c3cc[nH]n3)CC2)=O)ncccc1Br N1(C(CCN(CCC)C)=O)CCCC(C(C)NC(c2nccc(C)n2)=O)C1 c1(NC(C23CC(n4cc(CCC(CC)O)nn4)C2C3)=O)ncc2c(n1)CCCC2 CCCCC(CC)CCN=c1[nH]c(N2CC(C)CC(C)(C)C2)nc2ccsc12 N=c1cc(C(=O)NCC2(CCNC(=O)CCOC3CC3)CC2)cc[nH]1 N1(C(CSCC(C)C)=O)CCCC1CC(=O)NC(C)CCNC(N)=O c1(CCCNC(=NC)NC(c2ccc(Br)o2)C)nnc2n1CCCCC2 c1(C(=O)NCCOCC)ccc(CC(C)C(=O)NC2(Cn3cncn3)CC2)cc1 c1(C(N2CC3(CN(C(c4nnn(CC)c4C)=O)C3)C2)=O)c[nH]c(C)c(Cl)c1=O CC1CCCCN1CC(N1CC(CO)(NC(=O)CNC(=O)C2CC2)C1)=O C(=O)(C(CNC(=O)CC1CCC(=O)NC1)CC(C)C)NC1CC(C#C)C1 C1(C2CCC2)(CNC(C(C)OCCC=C)=O)CCN(C(C2(CO)CCC2)=O)CC1 C(=O)(CC=C(Cl)Cl)NC12CC(C(=O)OC)(C1)C2.C12(C)CCN1C2=O c1(CC)cc(C(=O)NC(CNC(C2CCCS2(=O)=O)=O)C(C)(C)C)ccc1C c1(C(=O)NCC2(O)CCN(C(c3n(C)ncc3C#N)=O)C2)ccsc1S(N)(=O)=O c1(C(=O)NC23CC(CNC(C(CC)(C)O)=O)(OC2)C3)cc(Cl)cnc1OC c1(COc2ccn(C)n2)ccc(C(=O)Nc2nc(C(F)(F)F)n[nH]2)cc1 n1(CC)nccc1CNC(=O)COC1CCN(C(c2ccns2)=O)C1 C(CCc1ccccc1Br)(C(C)(C)C)NC(C(=O)N(CCCF)C)=O C(=O)(C(C#N)(CC)CC)NC(CN(C(c1ccc(CC)o1)=O)CC)C C1(CC(N2CCC(CNC(c3on(C)c(=O)c3)=O)C2)=O)CCn2cncc2C1 Cc1ccc2c(=NCCOCC3CC3)[nH]c(=NCC3CCOC3C)[nH]c2c1 CC(C(C)C(=O)NCC1CCCC1CF)NC(c1[nH]ccc1C1CC1)=O C1(NC(CCCCN(C)C)=O)CC2CCC1(Nc1nnc(CO)c(CO)n1)C2 C(=O)(C1CCCc2ccccc21)N1CC(CCNC(c2c(COC)ccs2)=O)C1 C(C)(C(C)(C)CO)NC(CCOCCN(C)C(c1cc(CCO)on1)=O)=O c1(CN2CCC(O)(C(N3CCC(CO)CC3)=O)CC2)cccc2c1CCNC2 C12(C(=O)OCC)CCN(C(=O)Nc3cc(SC)nn3C)CC1C2(F)F CC(CCO)C(=O)N1CCC(O)(C(C)NC(=O)C(c2ccc(N)cc2)(C)C)C1 O=C(O)C(CNCC(c1cnn(C2CC2)c1)CC1CCC1)Cc1n[nH]c(O)n1 C1(NC(CC=C=C)=O)CC2CC(C1)N(C(=O)COC1CCN(C)CC1)C2 C1(NC(COC2(C)CCOCC2)=O)CC2(C1)CN(C(C1CCC(C3CC3)C1)=O)C2 c1(C(C)NC(=O)NCC2C3CC3CN2C(=O)OC(C)(C)C)ccc(F)cc1F C1(c2n(CC=C)nnn2)(NCC2CCOCC2(C)C)CCC(C)(CC2CC2)CC1 c1(C(=O)OC)cc(C)cc(S(=O)(=O)Nc2c(C)c3cnc2C=CN3CC(C)C)c1 C1(NC(c2c(CC)scn2)=O)CCC2CCN(C(c3ccc(O)c(Cl)n3)=O)C1C2 Cn1cc(C(=O)NC2CCCC(NC(C3CC3C(C)(C)C)=O)C2)c(C(C)(C)C)n1 N1(C(CC=CCC)=O)CCC(CO)C(NC(C2CCCN2C(=O)C(F)(F)F)=O)C1 C1(CNC(C2(C)ON=C(C)C2)=O)CN(C(=O)COCP(C)(C)=O)CC(C)(C)O1 C1(C(N2CC(NC(Cc3c(C(C)C)cccc3)=O)C2)=O)CCc2nc(O)[nH]c2C1 n1(CC(N2C(CNC(C3(C)COCCO3)=O)CCC2)=O)ccc2ccc(F)cc12 c1(SCC)cccc(C(=O)NCCC(CC)(CC)NC(=O)C(C(C)C)N(C)C)c1 CC1CCC(NC(c2ccc(C#N)o2)=O)CN1C(C1CCC(=O)N1C)=O c1(CNC(CC2(OCC)CCC2)=O)cc(C(=O)NC2C(CO)CC2O)on1 C#CCC(CC#C)C(=O)N1CC(COC)(NC(=O)C(O)c2ccco2)C1 C(=O)(C1=CCC(C)CC1)NCC1CC(NC(C(CCC)CC)=O)C1 CC(CCCCNC(=O)Cn1cnnc1)NC(=O)C(O)CN1CCCC1 Cc1cc2[nH]c(C(N3CCCCC(NC(c4nocc4Cl)=O)C3)=O)cc2o1 C(c1cccc(F)c1F)=CC(=O)NC1CC(NC(Cn2ccc(C)n2)=O)C(O)C1 c1(C(=O)NC2C(O)CCN(S(C(C)C)(=O)=O)C2)cccc2nc(O)oc12 Cc1ccncc1CC(=O)NCC1CCC(NC(=O)CCC(C)C)CO1 C(=O)(C(O)CC(C)(C)C)N1CC(C(C)C)C(C(=O)NC2CC3(CCCCO3)C2)C1 N1(C(C(C2CCCOC2)OC)=O)CCN(C(c2ccc(CC3CC3)nc2)=O)CC1 c1(CC)cccc(C)c1C(=O)NCC(C)(O)CNC(c1ncc[nH]c1=O)=O c1(-c2n(CCCCC)nc(CCCN(C)C)n2)ccnc2c1CCO2 c1(C(N(CC(CNC(c2c(C)nco2)=O)C)C)=O)ccc(O)c([N+](=O)[O-])c1 C(=O)(C1COc2ccc(F)cc21)N1CCC(N(C(c2c(CCC)[nH]cc2)=O)C)C1 C(c1ccc(Cl)cc1)=CC(=O)NC1C(CNC(CC(C)c2ccccc2)=O)C1 C1(CC(=O)NCc2ccc(NC(C)=O)s2)CSc2ccccc2NC1=O N1(C(c2cc(CC)on2)=O)CCC2CCN(C(c3ccn4cncc4c3)=O)CC12 C1(CNC(=NCCSC)NCC2CC3C(C2)C3(F)F)CC2(C1)CC(F)(F)C2 C1(CNC(CC2NC(=O)OC2)=O)CCC2(CO1)CC(NC(=O)COC(F)(F)F)C2 c1(C(=O)NC2CN(C(C(C(C)C)c3ccc(Cl)cc3)=O)C2)cncn(C)c1=O Cc1ccsc1C(=O)N(C(C)CCNC(C1(c2cc[nH]n2)CCC1)=O)C c1(OCCCC(=O)NCC(CC)NC(C2CCC(=O)NC2)=O)ccc(SC)cc1 C1(CNC(COCCC=C)=O)CN(C(=O)Cc2ccc(OC)cn2)CCC1(F)F CC(C(=O)NC1CCCN(C(c2ccc(C#N)[nH]2)=O)CC1)C(C)S(C)(=O)=O c1(CC(=O)NCC2(F)CC(NC(c3c(C)nsc3N)=O)C2)nc2ccccc2s1 c1(COC)cc(C(=O)NCC2(C(=O)NCc3cnn(C)c3C)CCCC2)c(C)o1 Cn1nc(C(=O)NC(CNC(=O)CCc2cccc(Cl)c2)CO)cc1C(C)(C)C C1(NC(=O)C(O)C2CCC2)CCCC1C(=O)NCCCc1ccsc1 C1(C(=O)NCCC(CNC(C(C(=O)OC)(C)C)=O)(C)C)CCc2c(ncn2C)C1 c1(C(=O)NCC(C2CC(F)(F)C2)OCC)cccc(C2(C)CC2)c1 Cc1ccccc1C=CC(N1CC(c2ocnc2CNC(C)=O)C1)=O Cc1cccc(C(=O)N(C)CCOCCN(C(=O)CC(C)n2cccn2)C)c1C Cn1ncc(C(N2CC(NC(=O)C(C3CCCOC3)N3CCCC3)C2)=O)c1F N1(C(=O)CCC2CCCC2)CCC2(CC1)OCCO2.c1cccnc1 Cc1ncncc1C(N1CCC(C(=O)N(C2CCCC2C)CCO)C1)=O c1(C(=O)NC2CCN(c3cc(CC)ncn3)C23CCC3)cccc2cccnc12 C12CC3CN(CC13)C2=O.c1(CNC(=O)OC(C)(C)C)ccc(N)cc1O N1(C(C2(O)CCOCC2)=O)CC2CN(Cc3cc(Cl)c(Cl)cc3F)CC2C1 c12ccsc1OC2=O.C1(N(CCCC)C(C)=O)CCOC1 N1(C(C(C)(O)C2CC2)=O)CCN(C(=O)C=CC2CCC2)C(c2cn[nH]c2)C1 N1(C(C=C(CCN(C)C)Cl)=O)CC(NC(=O)Cc2ccc(C(F)(F)F)s2)C(O)C1 N1(c2ncc(C#N)cc2Cl)CCC2CCC(C1)N2C(C12CC3CC(CC1C3)C2)=O c1(C(=O)NC2C3OCC(NC(CCC(=C)C)=O)(C3)C2)c(F)cccc1[N+](=O)[O-] N1(C(c2[nH]cc(CN(C)C)c2)=O)C2CCC1CN(C(=O)CN1CC3CC3C1)C2 C1(CCC(=O)NCC2CCCN2C(=O)CSc2cccc(F)n2)NC(=O)NC1=O c1(C(=O)NCC2(C)C(NC(CNC(CC)=O)=O)CCC2)ccc2ncccc2n1 C=C(F)C1(CC(=O)NC2(CNC(=O)Cc3cnsc3)CCCCC2)CCOCC1 CCCCCCCCCCCNC(=O)CC1(Nc2cccc(OCC)c2)CCC1 Cc1ncc(Br)c(C(=O)NC23CCC(CC2NC(c2ccc[nH]2)=O)C3)n1 Cc1c(C(N2CCCC3C2CCN3C(C2CCC=CO2)=O)=O)oc2ccccc12 N1(C(c2n(C)ncc2Cl)=O)CCC(CC(N)=O)(NC(=O)CC23CCCC2C3)CC1 S(=O)(=O)(c1ccoc1)N1CC(C(=O)OC)C1C c1(SCCC(=O)NCCC(=O)N(CC(=O)OCC)CC=C)oc(C)nc1C#N C(CCSC)(C(=O)NC1(CO)CN(C(c2cccnc2C(F)(F)F)=O)C1)OC C(=O)(CC(C)CC(C)(C)C)NCCCN(C(Cc1c(C)cccc1)=O)C1CC1 C1(C(=O)NC2CCN(CCOC)C2)CN(C(C2CC(=O)OC2(C)C)=O)CCN1C c1(SC)cc(C(N2CCOC(CN(C(=O)COc3cnn(C)c3)C)C2)=O)nn1C C1(N(C(=O)C=CC2CCCO2)CC)CCN(C(=O)CCc2ccsc2Cl)CC1 N1(C(C(C=C)CC)=O)CC(CNC(c2ocnc2C)=O)C2(CCC2)C1 CCC(O)CC(=O)NC1CCN(C(=O)CCCc2ccncc2)C1 C12(CNC(C(COCC)n3cc(C4(OC)CCOC4)nn3)=O)COCC1C2(F)F C=CCC(CNC(C1CC(=C2CC2)C1)=O)NC(C1(SC)CC1)=O c1(N2CCCC(CC)(CO)C2)nc(=NCCOCC(C)C)[nH]c2cccc(F)c12 C1(NC(C(C2CCOCC2)C)=O)CCC2(CC1)CC(NC(=O)C(=O)C(C)(C)C)C2 N(C1CCOc2ccc(Cl)cc21)CCc1nc(CN=[N+]=[N-])sc1.C1(=O)CN1C(N)=O c1(CCC(=O)N(CC(CC)NC(=O)CC2(COC)CC2)C)cccc(OC)c1 C1(N(C(CC)C(F)(F)F)C(c2c(O)cccc2F)=O)CCNCCC1C c1(C(=O)NC2(C3N(C(C(CCC)OC)=O)CCC3)CC2)ccc(OC)cc1O CCCCC(C)(F)C(=O)NC1CCCN(C(c2cc(C#N)oc2C)=O)CC1 Cc1noc(C)c1CC(C)C(N1CCC(C(C)NC(c2cccn2C)=O)CC1)=O n1(CC)ccc(=NC(=O)C2CCN(C(=O)C(C)NC=O)C(C)C2)[nH]1 C1(OCc2c(OC)cccc2)CCCCCC1C(=O)OC(=O)CC(O)C(C)C C1(C(N(CCC(=O)OC)CCC)=O)CCC(n2cc(Cn3ccnc3)nn2)C1 C1(CNC(C2(SCC)CC2)=O)(NC(=O)Cn2nccn2)CCCCC1 c1(C(=O)NC2C(NC(CC(C)NC(N)=O)=O)CCCC2)nccc(Cl)c1F C#CCC(C)(CC)C(=O)N1CC(C(=O)N(C)OCC(F)(F)F)C2(CC2)C1 C(CC1=CCN(C(c2ccon2)=O)CC1)NC(c1cn(C2CCC2)nn1)=O N1(C(c2ccc(CN(C)C)o2)=O)CC(NC(c2ccncc2F)=O)CC(C)(C)C1 N1(C(C(n2cnc(C#N)n2)C)=O)CC(NC(c2coc(O)n2)=O)C2(CCC2)C1 C(CNC(c1cn(CC(N)=O)nn1)=O)(C(C)(C)C)NC(c1c(C(C)C)nns1)=O n1(CCN(C)C)cc(CCC2CCCN2C(=O)C(O)CN2CCOCC2)nn1 S(=O)(=O)(c1cnc(N2C3CCC2CC(F)C3)c(Cl)c1)N(C(c1onc(C)n1)C)C N1(CC(=O)NC(CCNC(C2C(CCOC)C2)=O)(C)C)CCCCCC1 CCC(O)CC(=O)NC1(CC(=O)NCC2C=CCC2)CCC1 c1(CCNC(=O)CC2COCCN2C(C2C3COCC23)=O)cccc(Cl)c1Cl c1(CN2C(C(C)O)CCC2)cn(-c2cn(C(C)C)nn2)nc1-c1ccccc1 CC1CC(NC(=O)COC2CCC2)CN(C(=O)CC2CCC=CCC2)C1 Cc1cnc(C(N2CC3(CCC3)CC2CNC(=O)CC(C)C(C)C)=O)cc1C#N C1(C(=O)NC2CC2)CCN(CC2N(C(CCSCC)=O)CCC2)CC1 N1(C(CN2C(C)CCC2)=O)CCCOC(CNC(C2(C3CCC3)CCC2)=O)C1 N1(C(Cc2cc(C)on2)=O)CC2(CCCN(C(c3sc(C4CC4)nc3C)=O)C2)C1 c1(C(=O)NCC2N(C(c3c(OC)noc3C)=O)CC2)nc2ccccn2c1F Cc1c[nH]c2ncc(C(N3CC4C(CNC(=O)CCC(=O)N(C)C)C4C3)=O)cc12 c1(OC)cc(C(=O)NCCC(C)NC(C2SC3C=CC2CC3)=O)cc(OC)c1C C1(CNC(c2c(C)cncc2)=O)CN(C(C2Cc3nccn3C2)=O)CCN1C c1(C(=O)OCC)c(C)[nH]c(C(=O)Nc2onc(C)c2C)c1C.N12C(CC3CC13)C2 c1(C(=O)NCc2ccc(C(=O)NCC(=C)CC)cn2)cn(C)c(=O)n1C N1(C(CCC=C)=O)CCCCCC1C(=O)NC1C(O)CC1O Cn1ncc2c1C(NC(N1CCOC(C(F)(F)F)(CN)C1)=O)CCCC2 CCC(C#N)C(=O)NC(C1CCN(C(c2n[nH]c(C3CC3)n2)=O)CC1)C N1(C(CCN(CC)CC)=O)CCC(NC(C2CC(F)(CO)C2)=O)C(CO)C1 C=CC1CCN(C(C2CN(C(C3CCCSC3C)=O)CC(C)O2)=O)CC1 C1(CC(=O)NCCC(=O)NC)CCCCN(C(=O)CC2(C)CCOC2)C1 N1(C(CSS(C)(=O)=O)=O)CC2CCC1CN2c1nc(C(F)(F)F)ccc1C#N c1(C(N2C(C)CN(C(c3cc(Br)c[nH]3)=O)CC2)=O)ccc([N+](=O)[O-])cc1I N1(C(C(F)OC)=O)CCC2(C1)CN(C(=O)CCc1ccc(O)nc1)C2 S(=O)(=O)(c1ccc(F)c(C(=O)NC2CCSC23CN(C(=O)C(O)CF)C3)c1)NC C12(CNC(C(C3CCOCC3)OC)=O)CC1CN(C(c1nc(=N)cc[nH]1)=O)C2 Cc1cc(C(=O)NCC2(C)CCC(NC(c3cc(N(C)C)ccn3)=O)C2)cnn1 c1(OC)cc(C)c(S(N)(=O)=O)cc1C(=O)NCC1COCC(C)O1 C12(C(=O)NCC(CCOC)O)CC(CO)(CN1C(C1CC(C)C1)=O)C2 C(CC(C(=O)NC1CC(F)(F)C1)NC(=O)CCc1cnoc1)N(C)C N1(C(C(COC)COC)=O)CC(C(=O)NC2C(O)CC2O)CC(C)(C)C1 c1(CC(N2C(CCC#C)CCCC2)=O)nc2ccccc2n1C N1(C(=O)NC2CN(C(C3CC(O)C3)=O)C2)CCC2CC2C1 C1(C(=O)NCC#CCNC(c2cncc(COC)c2)=O)CC(C(C)C)=NO1 C1(NC(c2c(CNC(c3cnn[nH]3)=O)occ2)=O)CCCC2(CC1)CC2 CCC(CC(=O)N1CC(O)CC1C(=O)NC1(C)CCOCC1)SC c1(NCC(CO)OC)nc(=NC2COC3(CCCC3)C2)[nH]c2c(C)nn(C)c12 CC(C)C(C(=O)NCC1(F)CCN(C(c2ccc(=O)oc2)=O)C1)c1cnn(C)c1 c1(C(N(CCCCNC(=O)CC2CCC2)C)=O)c(F)cc(F)c(F)c1F c1(C(=O)NCC2N(C(COCc3onc(C)n3)=O)CC2)ccc(S(=O)CC#N)cc1 C1(CNC(CN(CCC#C)C)=O)CCCC2(CN(C(=O)C(C)CS(C)(=O)=O)C2)O1 NS(=O)(=O)c1coc(C(=O)NC2COCCC2NC(=O)CC2CCCOC2)c1 C1(CN(C(=O)CCC2CCCOC2)CC)COCCN1C(=O)CCSC N1(C(C(F)OC)=O)CCC2C(NC(c3cc(CC(C)C)[nH]n3)=O)C2C1 C(=O)(C(Cc1cccc(Cl)c1)CCCO)OCCC=CCCC Cc1nc(NC2CC(NC(c3cnc4ccccn34)=O)C2)c2cnn(C)c2n1 C12(C(=O)NCc3c(CCNC(c4cc(C)ncc4)=O)ocn3)CCCC1C2(F)F N1(C(COCCCCOCC#C)=O)CC2CCC(C1)N(C(=O)C1=C(C)OCCC1)C2 C1(C(=O)OCC(F)(F)F)COCCN1C(=O)C(C)Oc1ccc(C(=O)NCC)o1 C1(NC(C(CC)C#N)=O)C2CCCN(C(c3cnnn3C)=O)C2C1(C)C N1(C(C(C(=O)OC)F)=O)CC(C)(C)CC1C(=O)NCCCCS(C)=O c1(OC)ccc(C(C(=O)O)NC(=O)NCC2CCC3CC3C2)cc1OC C1(CNC(C(C2CCCC2)NC(c2c(C)nsc2)=O)=O)CC(=O)N(C)C1 CC(C)CCC(=O)NC1(CO)CN(C(=O)C(N2C(C)CCC2C)C)C1 c1(C(N2CC(CC(=O)NCC3(C#N)CC3)(OC)C2)=O)nn(C)cc1C C1(C(=O)NC2C(C)CN(C(c3cn(C)[nH]c3=N)=O)C2)CCn2ccnc2C1 C1(O)(CC(N2CC(N3CCN(C(C4CC5(CC5)C4)=O)CC3)C2)=O)CCCCC1 c1(C(=O)NC(C2CCN(C(=O)C(N)=O)C2)C)ccn2nnnc2c1 C(=O)(CC(C)C(C)C(C)C)N(CCC1(C(=O)OC(C)(C)C)CCN(C)C1)CC Cc1cccc(C(=O)NCC=CCC(N2CCOC(C(N)=O)CC2)=O)c1O C(CCC(C(=O)NCCC(=O)NCC(C)C)NC(=O)Cc1cccnc1C)OC C(=O)(C1CCCc2c[nH]nc21)NCCCOCCN(C)C(c1cccnc1Cl)=O c1(C(=O)NCC(O)CCNC(=O)C(O)c2ccsc2)cccc2nc(CO)[nH]c12 CC1CN(C(C2CCC(C)CC2)=O)CCC1N(C(=O)COC(F)F)C c1(C(N2CCC(NC(C(CC)NC(N)=O)=O)C2C)=O)ccc2c(c1)COCO2 C(=O)(CCCN(C)N=O)N1CC(C(=O)NCC#CCOC)C2(C1)CC2 N1(C(CC2N(C(C)=O)CCCC2)=O)CC(C2CN(C(=O)C(C)C(C)(C)C)C2)C1 c1(-c2ccn(CCOC)n2)nc(C2CN(C)CCO2)n(CCCN(C)C)n1 c1(CC(=O)NC(C(=O)NCc2onc(C)n2)C2(O)CCC2)c(C)n[nH]c1C c1(C(=O)NC2CCCC2NC(C2CCCCC2(F)F)=O)ccc2sncc2c1 c1(C(=O)NC23CC(NC(CN4CC(C)C4)=O)(C2)C3)ccc2c(c1)C(=O)N(C)C2=O C(C)(CCCCNC(=O)Cc1nccc(OC)n1)NC(C1(CC)CCCC1)=O N1(C(C(C(C)C)OC)=O)CCN(C(C2C=C(C)CS2)=O)CC12CC2 C1(C(=O)NCC(CNC(C2(C(N)=O)CCC2)=O)O)CC12CCOCC2 C12(NC(CC(C)(C)C3CC3)=O)CC3CC(C1)CC(NC(=O)C(O)C1CCC1)(C3)C2 N1(C(C(C)CC(N)=O)=O)CCN(C(C2CC(O)CN2C(N)=O)=O)C2(CC2)C1 N1(C(CC2(OC)CN(C(C3CC4CC(=O)C3O4)=O)C2)=O)CCC2(C=CCO2)C1 CCCC(CC(C)C)C(=O)NC(c1ccccc1)C(=O)N(CCCO)C C(CC(O)C(=O)NC1CCC(NC(=O)CC2(C)CCOC2)CC1)SC C(C(C)(O)CC(=O)N(C1CCN(C(c2cc(Cl)cn2C)=O)C1)CCO)OC C1(C(N2CC(CC)N(C(c3cc(F)n(C)n3)=O)CC2)=O)CC12CCC1(CC1)CC2 C(C(O)CCNC(c1sncc1Br)=O)NC(C=C(CC)C)=O CON(C)S(=O)(=O)c1ccc(C(=O)N(C2(C)CCS(=O)(=O)C2)C2CC2)cc1 N1(C(CC(C)F)=O)CCN(C(c2cc(O)cc(Cl)c2)=O)C(C)C1C O=S1(=O)CCC(n2nc(-c3cscn3)nc2C23CC(C2)C3)C1 C(c1c(C)noc1C)=NC1(c2n(CCSC)nnn2)CC(C2CCOC2(C)C)C1 C1(C)(CCC)CCN(C(=O)CC2C3CN(C(c4cn(C)nc4C(C)C)=O)CC23)C1 C1(C(N(OC)C)=O)CCCC1.N12CC(C1)OC2=O c1(Cn2cc(C(CCC)NC(=O)Cc3sncc3Br)nn2)ccccc1[N+](=O)[O-] c1(C(=O)NC2CCCN(Cc3n(C)ccc3)CC2)cccc(S(N)(=O)=O)c1 CC(C)CC(C)(C)C(=O)NCC(F)CNC(=O)C(C(C)(C)C)NC(=O)OC CC(O)(CNC(=O)CNC(=O)CC1CCC1=O)Cn1cccn1 C(=O)(C1=C(Cl)CCC(C)C1)N1C2CC(CN(C(CSC(C)C)=O)C2)C1 N1(C(C2(CCC)CC2)=O)CCC(CNC(c2cc(CC)c(CC)o2)=O)(CO)C1 C1(NC(C(CC)C)=O)CCN(C(=O)CCC2(C)CC2(F)F)CC1O C1(CCO)(NC(=O)C(=O)NCC(F)(F)F)CN(C(=O)Cc2ncc(Cl)s2)C1 Cc1cc(C(N2CC3(C2)CN(C(c2ccsc2)=O)CCO3)=O)c2n[nH]cc2c1 C1(CC(=O)N(C2CCC(NC(C3(C)CC(=C)C3)=O)CC2)C)CCC(F)(F)CO1 C(C(C(=O)N(CC(C)(C)CNC(=O)C=C(C)C)C)OC)OC C(=O)(CC(C(F)(F)F)NC(C1CN2CCC1CC2)=O)Nc1c(CC)n(CC)nc1 c1(C(N2CC3(CN(C(C(CC(C)C)F)=O)C3)C2)=O)cc([N+](=O)[O-])c(N)cc1F C=CC1(C(=O)NCCC(Cl)Cl)CCN(C(C2CCOC(C)(C)C2)=O)C1 CC(C)C(O)C(C)C(=O)N1CC2(CO)CC1(C(=O)NCC13CC(CN1C)C3)C2 N1(C(c2cnc(C)s2)=O)CCCC(N(C)C(c2ccc(-c3cnc[nH]3)cc2)=O)C1 Cn1nc(C2CC2)cc1NC(C1CCN(C(=O)C(N2CCCCC2)=O)C1)=O C(=O)(C1=CS(=O)CCC1)N(C)CCN(C(=O)C(c1cc(Cl)cc(Cl)c1)O)C c1(C(=O)NC2CCC2NC(c2ocnc2C(F)F)=O)cnc(C2CCC2)nc1O Cc1cc(C(=O)NCC2CC(O)CN2C(=O)Cc2cnnn2C)ncc1Cl C(=O)(CCCCCCNC(N)=O)NC1C(OC)C(C)(C)OC1 C1(CNC(C2CN(CC)C2)=O)CC(NC(=O)Cc2ccc(C(N)=O)cc2)C(O)C1 C1(CC(N2C(CNC(c3c(C(C)C)[nH]cc3)=O)CCCC2)=O)CCCC(C)(C)O1 Cc1ccc(C=CC(=O)NCCOCCCNC(C2CCC(C(N)=O)CC2)=O)s1 Cc1c(O)ccc(C(N2CCCN(C(c3occ4c3CCOC4)=O)CC2)=O)c1C C(=O)(C1CCCc2nnn(C)c21)NCCC1(NC(C2ON=C(C(C)C)C2)=O)CC1 C(C)(C)(C(F)(F)F)OCC(=O)NC(CC)CNC(=O)CSC1CCOC1=O c1(C(=O)NCC2(O)CCN(C(C3CC(=O)NC3)=O)C2)ccc(C#N)cc1 c1(C(N2CCCC(C(=O)NCC3CC[Si](C)(C)C3)C2)=O)ccc(F)cc1I c1(C(=O)OC)cccnc1NC1CCOCC1C N1(C(CCCC)=O)CCC(CNC(c2ccc(CCF)cc2)=O)C12CC2 Cc1cnc(F)c(C(=O)NC2CCCC2CNc2nccc(C)n2)c1 CC(O)C(C(=O)NC1CC1CNC(c1ccsc1C(F)(F)F)=O)N(C)C N1(C(C(C)N2CCC2)=O)CCC(O)(CNC(C23CC(O)C2C3)=O)CC1 C(C)(CC(=O)N(CC(=O)NCC(C)(C)C1CCOC1)C)SC N1(C(c2ccccn2)=O)CCn2ncc(-c3c(O)cccc3O)c2C1 c1(SCC(=O)OCC2CCN(c3cccc(OC)c3)C2)ncnc2[nH]cnc12 N1(C(c2ccc(CNC(C(C)(C)n3cncn3)=O)cc2)=O)CCC2CCC(O)C1C2 C(=O)(C(O)CC(N)=O)N1CCC(CCCNC(CC2(C)CCOC2)=O)CC1 c1(Nc2oc3ccc(C)cc3c2)nc2cc(Br)ccc2cc1C(=O)O C#Cc1ccc(C(N2CCCCC(C(=O)NC3CCOC3=O)C2)=O)nc1 c1(-n2ncc(C(=O)NC3C(NC(C(C)=C(CC)C)=O)CCC3)c2)ccc(Cl)cc1 C(=O)(C1CCCc2c(O)cccc21)N(C(C)CNC(=O)C1=CCCOCC1)C c1(C(N2C(CNC(CCn3c(C)ncc3)=O)CC2)=O)cccnc1S C1(C)(CCCOC(NOCC(=C)Cl)=O)NC(=O)NC1=O N1(C(c2cn(CC)nn2)=O)CCN(C(=O)C(O)CSC)CC1c1ccccc1 CC(C)C1=NOC(C(N2CCN(C(=O)CSc3ccccc3)C(CO)C2)=O)C1 c1(NC(C)C)csc(Cc2ccccc2)n1.C12CN(C1)C(=O)C(=O)NCC2C C1(NC(C2(C)CC2(Cl)Cl)=O)CC2CC1N(C(=O)C(O)Cn1cncn1)C2 C1(NC(c2c(O)ccc(CC)c2)=O)CN(C(=O)C(C)(O)C(C)(C)C)CC12CCC2 C1(C(N2CCC(CN(C(c3nn[nH]c3Cl)=O)CC)C2)=O)CCC2(CCC2)O1 C(=O)(C(CC(CC)CC)N1CCC(CF)C1)N(CC=C)CC=C C1(C2CCCO2)(C(=O)NCC(CNC(C(c2cn(C)nc2)=O)=O)(C)O)CCCO1 c1(CC(=O)NCC2(CC(=O)Nc3n(C)ncc3)CCC2)ccc2cc[nH]c2n1 C1(C(C)=O)CC1(Cl)C(=O)NCC(C1CCCC1)NC(=O)CCC1CC1 N1(NC(C(N2CCCC(NC(C)=O)C2)c2nc(Br)cn2C)=O)CC(C)OC(C)C1 c1(C(=O)NC2CC2NC(C2CCSCC2)=O)coc2ccc(F)cc12 N1(c2ccc(C#N)cn2)CCC2(CCCC2NC(C2CN3CCN2CC3)=O)CC1 C1(CNC(c2ccc(SC(F)(F)F)cc2)C(C)C)CN(C)CCO1 c1(C(=O)NCC2(F)CC(NC(C3CC3CF)=O)C2)cccc2c1CCC2 c1(C(c2c[nH]nc2CO)=O)cc(-n2cc(-c3cc(F)nc(F)c3)nn2)cc(F)c1 c1(C(=O)NCC2CN(Cc3ccns3)CCCO2)n[nH]c2ccc(F)cc12 C1(C)(COC)CC(NC(=O)CC(C)(C)O)CN1C(c1ccc(NC=O)cc1)=O N1(C(C(=O)NCC)=O)CC2(CCCN(C(=O)Cn3cnc(Br)n3)C2)C1 C=CCC(CC=C)C(=O)NC1(COC)CCN(C(=O)CCc2nc(C)no2)CC1 C1(C(=O)OCC2CCCCC2)CCC(NC(=O)OC(C)(C)C)CC1 CP(C)(=O)CN1CCC(c2nc(C3CCCNC3)no2)C1 C#Cc1nccnc1NC(C1CC1NC(=O)C(CC)NC(C)=O)=O c1(C(N(CCNC(c2c(C)nc(O)[nH]2)=O)C)=O)ccc2ccccc2c1[N+](=O)[O-] CCCCC(CC(=O)NCC(C)C(C)(F)F)NC(=O)CSCCOC N1(C(CC)=O)CCN(C(c2ccc(CC3CC3)s2)=O)C(CC(F)F)C1 C(=O)(C1=CCCCC1)N1CC(=C(CNC(CC2C(C)C2)=O)F)C1 CCCC(C(=O)NC1CC2(C1)CC2C(=O)NCC1(CN(C)C)CC1)C(C)C c1(CC(CC)NC(=O)C(C)OCC2CC2)cccc(S(=O)(=O)CC)c1 C#Cc1cc(F)ccc1CNC(=O)CC(C(C)C)c1ccccc1 CCCC(C)(O)CC(=O)N1CCC(CC(=O)NC2CCN(C3CC3)CC2)C1 C1(NC(C2CC23CCCC3)=O)CN(C(C23CCC(F)(CC2)C3)=O)CC12CC2 n1(CC(=O)NC2C(n3cc(COCC)nn3)CCC2)c(C)ccc1C c1(-c2cn(CCC(=O)NC3(C=C)COC3)nn2)ccc(N)cc1C(=O)O N1(C(C(C(=O)OCC)F)=O)CC2COCCC2(NC(c2cc(Cl)ccc2Cl)=O)C1 CCC(C)C(C(=O)NCC(C)N(C)C(c1ccn2ccsc12)=O)OC c1(C(=O)NC2CN(C(CC(CC)C3CC3)=O)C2)cc2cc(N)ccc2[nH]1 CC(C)CCC(C(=O)NC1CCC(=O)NC1=O)NC(=O)CC1CSCCO1 O=S(=O)(C1CN(CCc2ccncc2Br)C1)N1CCOCC1 N#Cc1[nH]c(=NCC2CN(C(C3(C4CCOCC4)CC3)=O)CCO2)sc1Cl c1(C(=O)NC2CN(C(CC(=O)OC)=O)CC2F)ccc(Br)cc1C(C)C C1(C)(CNC(c2ccc(OC)cc2OC)=O)CC(F)(F)CN1C(=O)CNC(N)=O Cc1n[nH]cc1CN(C(C(C)(C)SC(C)C)=O)C.C12CCCN1C(C)(C)CN2 N1(C(c2c(C)c(N)cnc2)=O)CC(NC(=O)CC(O)C2CCCC2)C2CCCC12 C1(C)(CCNC(COCc2ncc(C)o2)=O)CCN(C(C2CC2C(F)(F)F)=O)C1 Cc1nc(C2CC2)sc1C(=O)NC1CC(F)(CNC(=O)CC(F)(F)F)C1 N1(CC(=O)NC2(C(=O)NCc3n(C)cnc3)CC2(C)C)C(=O)CNC1=O Cc1oc(CNC(C2CCOC(C)C2)=O)nc1C(=O)NCCC12CC(CO1)C2 CCCC(C)(C)C(=O)N(C1CCCN(C(=O)CC(C)CC)CC1)C C1(CCC(N2CC(=CCC)C2)=O)CCC(NC(=O)C(C)OCC2CC2)C1 C1(C(=O)NC(CC)(C)C2CC2)CC1C1CN(C(=O)Cc2cncc(C)c2)C1 N1(C(CC)C)CCCC(NCc2c(-c3ccc(F)c(F)c3)nn(C)c2Cl)CC1 c1(C(=O)OC)ccc(O)c(NCC23CC2CN(C(c2ncc(Br)cc2F)=O)C3)c1 c1(C(=O)NC2CCCN(C(CC3C(CC)C3)=O)C2C)c[nH]c2cnccc12 N1(C(C=C(C)c2cccs2)=O)CCCCC(NC(=O)C(C)Sc2nncn2C)C1 c1(C(=O)NC2C(NC(C(CC)(C)COC)=O)C2)cc(C)nc2ccc(OC)cc12 C12CCC(C1)NC2=O.C1(CC(=O)OC)CCCC1NC(C1COCOC1)=O C1(C(=O)NCC2CCC(NC(C=CC=CC)=O)CC2)CCC2CC2CC1 C1(C(=O)NC(C(=O)NCCCc2cccs2)C2CCC2)C2CCC(F)C12 N1(Cc2cccc(OCC=C)c2)CC(C(N2CCCC2CCC)=O)CC(F)(F)C1 N1(C(c2cc(OC)ncc2)=O)CCN(C(=O)C(CC(C)C)SC)CC1C(F)F C1(C)(C(=O)NCCCC(C)NC(C(C)OCCC(C)C)=O)CCCCO1 C1(NC(c2cnc(C3CCC3)s2)=O)CN(C(C2CC2F)=O)CC1C(F)F c1(C(=O)NC2CCC(NC(C(C)SC)=O)CC2)cc(C)nc2[nH]nc(O)c12 C1(NC(c2c(C)oc(Br)c2)=O)CN(C(=O)C=Cc2ccc[nH]2)CC12CCC2 C(C(COC)CC(=O)NCC(C(C)C)NC(C1(CO)CC1(F)F)=O)OC N1(C(c2nc(C)sc2)=O)CCC(=O)NC2CN(C(C3CCSC3)=O)CCC12 CC(C)(C)C(C#N)C(=O)NCCNC(C12CCC(N=[N+]=[N-])C1C2)=O c1(OC)ncc(S(=O)(=O)NC(Cc2ccccc2C)C(C)C)cn1 C(=O)(C(CC1CC1)NC(c1csnn1)=O)N(CC(C)O)C c1(-n2cc(C3(N4CCCC4)CC3)nn2)cc(F)cc(Cl)c1.C12(CCCCO1)C(=O)NC2 c1(CCC)cccc(C(=O)NC2CC23CC(NC(C2CC2CF)=O)C3)c1 CC(C)(O)C(F)C(=O)NCC1CCCC1C(=O)NCC(CO)OC N1(c2c(C)c(F)ccc2)CCN(N2CC(N(C)C)(CO)C2)CC1 N1(C(C2CC(CCC)C2)=O)CCC2(CC1)CC2(CO)C(N1CC(=O)N(CC)C1)=O N1(C(C2CC(C)=C(C)CC2)=O)CC2OCCN(C(=O)CN3CCCC3=O)C2C1 N1(C(c2ccc(CC)cc2)C(=O)NC(C)(C)CC)CCCC2(CC(=O)N(C)C2)C1 C1(C(N(C)Cc2ccoc2)=O)CCC2(CC2)N1C(=O)CCN1CCCC1 c1(OC)cc(=O)n(C)cc1C(=O)Nc1cc(C)c(NC(=O)N(C)C)nc1C c1(-c2n(C)cc(NC(C3C(C(=O)OC)C34CC4(F)F)=O)n2)ccc(C)c(F)c1F N1(C(C(C(C)(C)O)F)=O)CCN(C(c2coc(Br)c2)=O)C2CCCC12 N1(C(C(c2ccccc2)C)=O)C2CCC(C2)C1CC(=O)N(CC(C)C(C)(C)C)C O=C1CCN(CCC2CCC(F)(F)C2)C(=O)N1Cc1csc2c1CCCC2 Cc1n[nH]c(C)c1S(=O)(=O)N1CCCC(C(=O)NCCC(C)N2CCCC2)C1 C1(CC(N2CCC(CCCC)C2)=O)CCCCN1C(C1CC1[N+](=O)[O-])=O C1(C(=O)N(CCO)CC2CC2)CCN(C(=O)c2c[nH]c(=S)cn2)O1 C=CCC(C(=O)N(CC(CC)NC(=O)Cc1ccoc1)C)c1ccccc1 C1(CSC)C(C(=O)NCC2CC3(CC3)C2)CCN1C(=O)CCCCN(C)C n1(CCCC)nc(C)c(C=CC(N2CCC(F)(CNC(=O)C=CSC)CC2)=O)c1Cl c1(C(=O)NCC(CNC(C(C)OCCOCC)=O)C)nn(C)cc1SC CCC(C)(CC)NC(=O)CN(CC(C)C)C(=O)COC1CCOC1 CCCCC(CCCC)C(=O)N1CCC(O)(CN(C)C(c2ccccn2)=O)C1 C1(C(=O)NC2(COC)CCN(C(=O)Cn3nnnc3C)C2)OC2CCC1CC2 c1(C(N2CCC(C(C)NC(C3(O)CC(C)(C)C3)=O)C2)=O)cc(Cl)cnc1O c1(SCCC(=O)NC2CC2)ncnc(OC)c1Br CC1(NC(=O)C2=C(Cl)CC2)CCC(NC(=O)CS(=O)(=O)N2CCCC2)CC1 Cc1cccc(OCC(=O)NC2CN(C(C3CCOC3(C)C)=O)C2)c1C N1(C(c2cc(C(=O)OC)sc2)=O)CCC(O)(CNC(C2COCCO2)=O)CC1 C1(OC)CN(C(C2(C)C=CCC2)=O)CC1NC(=O)C(C)(F)c1ccccc1 N1(C(c2cnc(CNC(C=Cc3n(C)cnc3)=O)nc2)=O)CCCC(O)CC1 c1(CN(C)C)ncc(C(=O)NCC(C2CCCC2)NC(=O)Cc2nc[nH]n2)[nH]1 C(=O)(C1CCc2c[nH]nc21)N1CCCC(N(C(C(C(C)(C)C)OC)=O)CC)CC1 N1(C(c2c(C)ncn2C)=O)CCCCC(NC(C2CCOC(C)C2)=O)C1 C12(CNC(Cc3nc(CC)sc3)=O)CC(NC(C3CCC(C)NC3=O)=O)(CCO1)C2 CC(N=c1[nH]c(N2Cc3ccccc3C(F)(F)C2)nc2ccccc12)c1ccns1 N1(c2n(CCCOC)c(C3CCCCN3C)nn2)Cc2c[nH]nc2CC(C)C1 C1(C(C)C)CCC(C(N2CC(C)(C)C2c2cn(Cc3cnn(C)c3)nn2)=O)CC1 N1(C(=O)CSC2CC2)CCC2CCCC(C1)N2C(=O)CN1CCS(=O)CC1 c1(C(N2CCCC(NC(C3C(OC)CCCC3)=O)C2C)=O)c[nH]c(C)c(Cl)c1=O CC1(CC(=O)NCC2(C)CCCN2C(=O)CCn2cccnc2=O)CC(F)(F)C1 C1(CN2C(NC(=O)OCCC(=O)O)CCC2)CCN(c2cncs2)C1=O C1(CCCC)CN(C(=O)CS(=O)(=O)NC)CCN1C(=O)CN1C(=O)CN(C)C1=O c1(CNC(Cc2ccc(C)o2)=O)ccc(C(=O)NCCNS(N)(=O)=O)nc1 n1(CC)cnc2nc(=NC3CCCC(C)(C)C3)[nH]c(NCCCn3ccnc3)c12 C(N=c1cc(Cl)c(O)n[nH]1)C1(C(=O)Nc2c(F)cc(C)c(C(F)(F)F)c2)CC1 C1(CC=C)(NC(=O)CC(C)OC)CCN(c2ccnc(-c3nccs3)n2)C1 c1(NCC)ncccc1C(N1CCOCC1CNC(=O)C=CCF)=O N1(C(CCCNC(C)=O)=O)CC2(CCC2)CC1CNC(C1(C)CCC(O)CC1)=O c1(CNC(N(C2CC2C2CC2)C)=O)cnccc1C(C)(C)C c12ccc(nn1)OCC(=O)NC2.C1(C(N)=O)COCC1C(N1CC(OCF)C1)=O C1(OC)CN(C(=O)Cc2cccc(O)c2)C(C)(CNC(=O)C=CCN2CCC2)C1 Cc1cc2c(cc1C(N1CC(NC(C3CC(O)CN3C(N)=O)=O)C1)=O)OCO2 c1(CC(=O)NC2CCN(Cc3cnn(C4CC4)c3)CC2)c(O)ncnc1O N1(C(=O)Cc2cnn(C(F)F)c2)CCN(C(c2cnccn2)=O)CC1 CCC(CCC(=O)N1CC(C(C)OC)C1)NC(=O)CCCc1ccc(C)cc1 CC1(C)C(NC(c2ccc(F)cn2)=O)CC1CC(=O)NCCc1cccnc1F C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CC(CNC(C(=C(C)C2CC2)F)=O)C1 C1(C(=O)NC(C2CCCC2)CNC(c2cccc(F)c2O)=O)CC2(CCOC2)C1 N1(C(CCSCCCC)=O)CCCC(CNC(C2CCSCC2)=O)C1 N1(c2snc(CCOC)n2)C2CCC1CC(NC(=O)CCC1CCC(C)O1)C2 c1(CCCC(N2CC(F)(CNC(c3occ(C)c3)=O)C2)=O)ccc(O)cc1 C1(CNC(C2C(C)C2)=O)CCCCCN1C(C1CCCC1F)=O C1(C(=O)NC(C2CCCN2C(=O)CCCC(F)(F)F)C)COc2ccccc2O1 N1(C(CCN(CC)CC)=O)CCC(C)C(NC(=O)C=CC(=O)N(C)C)C1 CC(CNC(C1CCC(=O)C1)=O)CC(=O)N1CCC1 c1(C(=O)NC(CC=C)CNC(c2c(C)nn(CC)c2C)=O)sc2cncn2c1C N1(C(C(C=C)C)=O)CCCC2C(NC(=O)CC3CCCC(C)O3)C(C)(C)C12 CC1CC(C(=O)NCC2(O)CC3CCC2O3)CN(C(=O)C(F)C(F)(F)F)C1 Cc1ccc(CNC(c2cnn(CCNC(c3ccc(=N)[nH]c3)=O)c2)=O)cc1 O=C(CN1CCCC(F)C1)NN1C(=O)NC2(CCCCC2)C1=O c1(C(=O)NCc2c(C(=O)NCCC3=CCCCC3)occ2)cnn2ccccc12 C(=O)(C(C)CC(=O)N1CCN(C(C2CC2OC2CC2)=O)CC1)OC N1(C(C(n2ccc(C)n2)C)=O)CC2(CCN2C(c2cnn3c2CCC3)=O)C1 C(CC(C)C)(C(=O)NCC1CCN(C(C2CN(C)CCO2)=O)C1(C)C)OC N1(C(C(N2CCSCC2)C)=O)CCN(C(c2cc(Cl)ns2)=O)CC1C1CC1 C1(C(=O)N(CCO)CCO)CCC2(CN(Cc3ccnc(O)c3)C2)O1 CC(C)CC(CCC(=O)O)NC(N1CC2CC2C1)=O N1(C(C2CC(SC)C2)=O)CC2CCCC(NC(C3CCC3)=O)(C2)C1 c1(C(N)=O)cnccc1C(=O)NCC1CC1CNC(=O)C=C1CC1 C1(C(=O)NC(C2CC(NC(=O)CC=CC(C)(C)C)C2)C)CCCC(O)C1 c1(C(=O)NC2CC(C)(NC(CCCC#C)=O)C2)cc(F)c(C(F)(F)F)cc1F C(=O)(CC1c2ccccc2C(=O)N1C)N1C(CC=C)CCCC1 C1(NC(CCCC=C)=O)CCN(C(=O)Cc2csc3nccn23)CC1O c1(C(N2CCC(N(C(=O)Cc3cnc[nH]3)CC)C2)=O)cccc(C(F)(F)F)c1N c1(C(=O)O)c(NC2CC(F)(F)C2N)ccc(Br)c1F CC1(C)CCN(C(=O)CCCn2cncn2)CC1CNC(=O)C(C)(C)C#N C12(C(=O)NC(c3cccs3)CC)CCC(CC1)N(C(C1CC1C(C)C)=O)C2 Cc1nn(C)c2c(NCc3c(F)cccc3Br)nc(=NCC3(C)CC3(F)F)[nH]c12 C(=O)(C(C(C)NC(=O)CSCC1CCCO1)C(C)C)Nc1c(C)c(F)ccc1 C1(OC)(CNC(C2(C(=O)NCCc3csc(Cl)c3)CCC2)=O)CCC1.SC N1(C(C(CC#C)(C)C)=O)CCCN(C(c2ccc(C3(CC)CC3)cc2)=O)CCC1 CCCC(C(O)C(=O)NC12CC(F)(C1)C2)NC(c1cn(C)nn1)=O C12(CNC(C)=O)CC(C)(C1)OC2C.N12CCCC(C1)CC(=O)N1CCCC(C1)C2=O CC1OC(C)Cc2c(C(N3CC(CNC(=O)C#CC4CCOCC4)C3)=O)n[nH]c21 c1(C(=O)NC(C)C(CO)NC(C2(C)CCC(=O)NC2)=O)cc([N+](=O)[O-])cn1C C1(NC(c2cccc(SCC#C)c2)=O)CCN(C(=O)CC#N)C(C2CC2)C1 N1(C(C(=O)Nc2cc(OC)cc(OC)c2)=O)CCSC2(CCCC2)C1 c1(C(=O)NCC2(O)CCN(C(C(CC)SC)=O)CC2)ccc([N+](=O)[O-])nc1 C1(NC(c2cc(C(C)=O)sc2)=O)CCN(C(C2C=CC=CC=C2)=O)CCC1CO C1(NC(CC(=C)C)=O)CCN(C(c2cccc(NC(=O)OC)c2)=O)CC1O C1(OC)CCCCC1C(=O)NCC1(CNC(C2(N(C)C)CCCCC2)=O)CCC1 c1(C(=O)NCC(Cn2cc(-c3cncn3C)nn2)OC)nn(C)c(C)c1Br CCCCC(O)C(=O)N(CC(C)C(=O)NCc1n[nH]cc1C1CC1)C CCC(CC)C(F)C(=O)N1CC=CC(NC(c2cncc(F)c2)=O)C1 N1(C(CCC2CC(OC)C2)=O)CCC(CCC(=O)N(C)Cc2ccco2)C1 CN1C(=O)CCCC1C(=O)NCC1CCN1C(c1nn[nH]c1C(F)(F)F)=O C(CN=c1nc(N2CCCC(C)(CO)C2)cc[nH]1)NC(=O)NC C1(NC(=O)NCC2(c3c(OC)nccc3)CCOCC2)Cc2n[nH]cc2CC1C C#CCCCC(=O)NC1COCC1CNC(=O)CCN1CCCCC1=O C(=O)(C1=NOC(C(=O)OC)C1)N(C(C)CNC(c1ccccc1C(C)(F)F)=O)CC C1(CNC(c2c(C)csn2)=O)CC(C(=O)NCCc2ccc(F)cc2)C1(C)C N12CCC(C(F)F)(C1)CNC(=O)C2=O.c1(C(=O)OC(C)(C)C)ccn(C2CC2)n1 N1(C(Cc2nc(COC)sc2)=O)CCC(C)C(CNC(c2csc(C#N)c2)=O)C1 C#CC1(NC(=O)CC(C(C)(C)C)NC(=O)C=Cc2ccc(C)o2)CCC(C)CC1 c1(OC)cc(Br)ccc1CC(N1CC(F)(F)CC1CNC(=O)C#CC(C)C)=O Cc1ccc(C(C)OC(c2ccc(-c3ccccc3C)cc2)=O)cn1 c1(CCNC(c2cn(C(C)(C)C)nc2)=O)ccc(CNC(=O)C(N)=O)cc1 C(=O)(C1=C(C#N)CCC1)NCC(C(=O)NC1(C)C(C)CCC1)N(C)C N#Cc1nc(=NC2CC(CNC(C3CC3Cl)=O)C2)c2ccccc2[nH]1 c1(-c2scc(OC)c2)cc(S(=O)(=O)Nc2cc3cccc(Br)c3o2)ccc1C C1(C(=O)NC(c2ccncn2)C)CCN(C(=O)CCCC2CCCC2)O1 C(=O)(C1CN(C)C(=O)c2ccccc21)NC(c1ccc(OC)cc1)CO N1(C(C2(C(C)C)COC2)=O)CCC(O)(C(C)NC(c2coc(C(F)F)n2)=O)CC1 c1(C(=O)NCC2(OC)CN(C(=O)C(C)OCC(F)(F)F)C2)ccnc2ncnn12 C(=O)(CC1=NNC(=O)C1)N1CC2C(CNC(c3ccc(=N)[nH]c3Cl)=O)C2C1 C1(SCC)COCCN1C(c1cncc(C2CC2)c1)=O.c1(C(N)=O)cc(C(=O)N)c[nH]1 Cc1nc2cccnn2c1C(=O)NC1CN(C(=O)C(=O)CC(C)C)CC(C)(C)C1 CS(=O)(=O)c1cc(C(N2CC(NC(=O)Cc3cn[nH]c3)C2)=O)ccc1F C(=O)(C(=O)C(C)(C)C)NCC(CC=C)NC(C1CC(=O)N(OC)C1)=O c1(C(C)C)ccc(C(=O)NCCC2CCC(NC(=O)CCCc3cnn[nH]3)C2)o1 N1(C(c2nc(C)oc2)=O)CCN(C(=O)CC2CCN(C)C2=O)CC(CO)C1 C1(NC(CN2CCC(C)C2)=O)CC1C1CCN(C(=O)C(C)(C)C(C)(C)O)CC1 c1(CC(=O)N(C2CCN(C(=O)COC3CCCOC3)CC2)CC)nc(C)sc1C C1(C)(CNC(C(C)=C(C)C)=O)CN(C(=O)CC2CC3(CC3)C2)C(C)(C)C1 c1(C(c2nnnn2CCC)NCCCC2CC(=C)C2)cccnc1OC(C)C CC1(C)CCN(C(=O)CC2CC3(C2)CN(C(=O)C(O)C(F)(F)F)C3)C1C1CC1 c1(CC(=O)NCCC2CCC(NC(c3ccccc3)=O)C2)ccc2c[nH]nc2c1 C(=O)(CCCC(C)(C)C)N(C1CCN(Cc2ccccc2I)CC1)CCC CC(C)C(C#N)C(=O)N(C)CCN(C)C(c1c(C#N)cnn1C)=O C1(CC=C)(C(=O)NC2CCCC2CNC(=O)CSC2CCOC2=O)CCCC1 C(C)(C(C(=O)NCC(F)(F)C(F)F)C(C)C)NC(CCCCOC)=O c1(-c2nc(C)sc2)ccc(NC(=O)C(N2CC(O)CC2C2CC2)=O)c(F)c1 c1(CC(=O)NCC2(O)CCN(C(Cc3n(C)nnc3)=O)C2)cc(Cl)cc(Cl)c1 c1(C(C(=O)NC(CCOC)CNC(c2coc(N(C)C)n2)=O)O)ccccc1Cl CCC(C(=O)N1CCN(C(C2CC3(CCCCO3)C2)=O)C(C)C1)C(C)(C)CC c1(C(=O)NC(C(=O)NCCSCC)C(C)(C)O)cccc2ccnn12 n1(Cc2cc(C)on2)nnc(C(=O)NC(C)(CNC(=O)C(C)O)C2CC2)c1C c1(OCC)ccc(C(=O)NCC(F)CNC(C2CCC(=O)NC2)=O)c(F)c1F C1(C(N(C2CCN(C(c3cc(Br)sn3)=O)C2)C)=O)CC12CCC2 CCC(CC(=O)NCCC(=O)N(C)C)N(C(=O)C(C)CO)C C1(CNC(C(C2(O)CN(C(c3cc(OC)no3)=O)C2)F)=O)(CO)CC(F)(F)C1 c1(COC)nc(CCOC(=O)CCC2CCCN2CC(F)F)no1 N1(C(c2ccc(CN)cc2)=O)CCn2ccnc2C1 C1(C(=O)NCC2(O)CCN(C(C3CN(C4COC4)C3)=O)C2)(OC)CCCCCC1 CCCCC(O)C(=O)N1CCC(C(=O)Nc2oc(C)nc2C#N)CC1 Cc1cc(NC(=O)C(CNC(=O)C(F)F)N(C)C)c(F)cc1F C1(C(=O)NC(CC=C)CO)CN(C(C2CCC(=O)O2)=O)CC12CCC2 N1(C(C2CCN(C(=O)NC)CC2)=O)CCC(NC(C2(CF)CC2)=O)CC1C C=CC1OCCCC1C(N1CC(CNC(c2cc(CO)on2)=O)C1)=O C1(CC)CC(NC(C2(NC(=O)C=CC3CCOC3)CC(F)C2)=O)CCO1 N1(C(C(C=C)O)=O)CCN(C(=O)CCn2nc(C)cc2C)C(CC)C1 N1(C(c2cc(OC)no2)=O)CCN(C(c2sccc2Cl)=O)CC1C1CCC1 CON(CCC(=O)NC1C2CCCCC12)C(=O)c1ccc(N)cn1 c1(NC(c2cc(OC)cc(CC)c2)=O)nc2c(s1)CCC2C(=O)OC N1(CC(=O)N(C(C)C)CCNC(=O)CC2C(C)C2(F)F)CCC(CO)CC1 N1(C(=O)CC2CCCN(C(c3cc(=O)cc[nH]3)=O)C2)CCN2CC(F)CC2C1 N1(C(C(C)n2cncn2)=O)CC(NC(=O)CCc2ccccc2)C2(COC2)C1 C1(C)(CCC(=O)N(C)CC2(COC)CC2)CN(C(c2ccncc2)=O)C1 c1(NC(N(CC(C)CN2CCCC2)C)=O)sc(N2CCCC2)nc1Cl C1(N(C(C2C(=C)C2)=O)CC)CCN(C(=O)Cc2cnc(C(C)(C)C)[nH]2)C1 n1(CC(=O)NC2CC(N(C)C(C3CC3(C)C)=O)C2)nc(C2CC2)cc1C(F)F Cc1coc(C2CC2)c1C(=O)N(CC(O)CN(C)C(C1CCN(C)C1=O)=O)C c1(C(C)(C)C)ccc(C(=O)NCC2(NC(c3[nH]cnc3C#N)=O)CC2)cn1 CCCC(C(=O)NCC1CC(F)(F)CO1)NC(c1c[nH]c(C)c1)=O c1(C(=O)NCC(CC)(C)NC(C2(F)CCOC2)=O)cc(C)c(C)cc1Cl N1(C(C2C(C)CC2)=O)CCC(C2CCN(C(c3ccc(C4CC4)cc3)=O)C2)CC1 c1(SCC)ccc([N+](=O)[O-])cc1C(=O)NC12CC(CNC(C3(CO)CC3)=O)(C1)C2 C(C(C(=O)N1CC(N2CCC2)C1)NC(=O)C(C)(C)C)OCC(=O)N(C)C c1(CC)ccc(C(=O)NCCN(C(=O)CS(=O)(=O)NC2CCCO2)C)cc1CC C(CN(C(=O)CN1CCS(=O)CC1)C)(CO)(CO)NC(C1CCN(C(C)=O)C1)=O c1(C(N(C2CCCC2)CCNC(c2cc[nH]c2)=O)=O)cccc(OC(F)(F)F)n1 c1(CC)nn(C)c(CC(=O)NCC2(NC(=O)CCCc3csc(C)n3)CC2)c1Cl N1(C(c2n(C(CC)CC)ncc2)=O)CCC(N(C(=O)COCC(=O)NCC)C)C1 C1(C(N2C(C(C)NC(C3(C=C)CCC3)=O)CCC2)=O)CC(C2CC2)=NO1 CS(=O)CCCCc1nc(-c2cccc(N3CCCC3)n2)nn1C(C)C1CC1 C1(COC)(CNC(=O)Cc2n[nH]c(=N)s2)CCCN1C(c1ccn(C(C)C)n1)=O C(=O)(CC(C(N)=O)c1cn(C(C)CN2CCCC2C)nn1)OCC O=C(NNc1ccc(F)c(F)c1F)N(c1ccncn1)C1CCCC1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC(C)CC1CN(C(C2CCCCC(=O)N2)=O)C1 c1(C(=O)NC2CCCN(C(C(C(C)O)N(C)C)=O)C2)ccc(N)cc1Br n1(C(C(=O)NC(CNC(C2(CC)CCC2)=O)(C)C2CC2)C)c(C)cc(O)cc1=O C(=O)(C1=CC2CC(C1)CC2O)N1CC(NC(=O)Cn2cccn2)C1 C(C(COC)CC(=O)NCCCC(C)NC(c1cccc[n+]1[O-])=O)OC C1(C(=O)NC(CN(C)C(C2CCCOC2)=O)(C)C)CC2(CCC(CN)OC2)C1 C1(NC(c2cn(CCC(C)C)nn2)=O)CC2CC1N(C(c1cnco1)=O)C2 c1(C(N(CCC2CCN(C(=O)C(C)NC(C)=O)CC2)CC)=O)c(F)cccc1F C(C(COC)CC(=O)N1CCN(C(=O)CCC(=O)NCc2nccs2)C(C)C1)OC Cc1ccc2oc(C(N3CCC(C)(NC(=O)CC4CCCN4C)C3)=O)c(C)c2c1 C1(CC(=O)Nc2c(C)ccnc2)CN(C(C2CCOC2)=O)C(C)(C)C1 c1(C(=O)NCC2(C)N(C(c3c(CC)noc3)=O)CCC2)ccc(C)nc1N Cc1ccnc(-c2cn(CC(C)NC(c3ccc(C)s3)=O)nn2)c1 C1(C(=O)N(CC(O)CCO)C2CC2)CC2C=CC1O2 c1(CC)nc(C(=O)N(C(C)C(=O)NCC2CC(CN=[N+]=[N-])C2)CC)cs1 C=Cn1nncc1C(=O)N(C1CN(C(C2(C)CCOC2C)=O)C1)C C1(=CCNC(C2CC2F)=O)CCN(C(=O)CCC2CCOCC2)CC1 C(=O)(CCCN(C)C(c1scc(I)c1C)=O)NC c1(C(=O)NC(C)CC(C)NC(C2(O)CCSC2)=O)ccc(Cl)cc1O c1(OC)c(CC(=O)NCCOc2ccc(F)cc2Cl)cccc1F c1(CC(N2CCC(OCCNC(Cc3ccn(CC)n3)=O)C2)=O)cccc(F)n1 c1(NC=O)ccc(C)s1.C1(N(C(=O)C=CC(C)C)C(C)=O)CCCC1O C1(COC)(CNC(C2CC2c2cncn2C)=O)CCCN1C(c1cscn1)=O C(=O)(CS(=O)(=O)CCOC)NCC(CCCC)NC(c1cc(C)cc(N)c1)=O C1(CNC(c2nn(CC)c(O)c2)=O)CCCCN(C(=O)C(C)C(C)(C)C)C1 C1(NC(=O)CC2CSC2)CCN(C(c2ccn3nncc3c2)=O)CCC1CO C=CCC(C(=O)NCC(C)NC(c1ccc(SC)s1)=O)OC C1(C(=O)NCC(CNC(=O)Cn2cccnc2=O)OC)COCC2(CCC2)O1 C1(CCC)CN(C(C2CCC(=O)NC2)=O)CCN1C(=O)Cc1ccc(Cl)nc1 C1(NC(=O)C=CC(F)(F)F)CCCC12CCN(C(C1CC3(C1)CC(F)(F)C3)=O)C2 c1(OC)ccccc1-c1cc(CNC(C2CCC(CNC(=O)CO)CC2)=O)on1 c1(C(=O)NC2CCN(C(c3ccc(CC)o3)=O)C2)cnc(OC)nc1C Cc1ccnn1C(C)C(=O)N(CC(C)NC(=O)C(c1cccn1C)=O)C N1(C(C2ON=C(C)C2)=O)CC(NC(c2sccc2Br)=O)CC1(C)C c1(C(=O)NCC(C)N(C(C(=O)NCC)=O)C)cccc(-c2noc(C)n2)c1 c1(CC)cccc(OCC(N2CCCC(C(=O)N(c3ccccc3)C)C2)=O)c1 c1(C(=O)NC(CNC(c2c(C(C)C)nns2)=O)C2CCC2)ccc(N)c(Cl)c1O C1(NC(CCNC(N)=O)=O)CCCC(NC(C2CCC(C(N)=O)C2)=O)C1 C#CCCCCCC(C(=O)NCCSC)N1CCCC2(C1)OCCCO2 Cc1ccc(CC(=O)NCCCC(C)NC(C2(c3ccno3)CCC2)=O)cn1 C(N=c1cc(C)nc(Cl)[nH]1)C1CCCC(NC(c2c(C)ccc(OC)c2)=O)C1 N1(C(c2c(SCC)nccn2)=O)CCC(CNC(=O)C=Cc2cc[nH]n2)C1(C)C C(=O)(C(C)(CC)C(F)F)NCC1C(NC(c2c(CC)c(OC)ccc2)=O)C1 C(=O)(C(F)CC(C)(C)NC(C1COCOC1)=O)NC(c1ncc(C)o1)C c1(C(=O)NCC(C)NC(C2C(COC)(COC)C2)=O)cc2n(n1)CCC2 C(=O)(C(C)P(C)(C)=O)N(CC)CC1CCCN(C(c2snnc2C2CC2)=O)C1 CC1(C)CC(NC(c2ccoc2)=O)CCN(C(c2cnc(-c3ccco3)s2)=O)C1 N1(C(c2ccc(C)o2)=O)CCN(C(c2ccc(CN(C)C)cc2)=O)C2CCC12 C1(CC=C)CCCC1N=c1cc(C(C)C)nc(-c2cccnc2)[nH]1 c1(NC(c2c(Cl)ncc(-c3scc(OC)c3)c2)=O)cc(OC(F)(F)F)ccc1F C(=O)(C(C#N)CNC(c1cc(CNC(=O)OC(C)(C)C)cs1)=O)OC c1(OC)cccc(NC(C2CC(NC(=O)Cc3cccs3)C2)=O)c1OC N1(C(c2cncc(F)c2)C(=O)NC(CC)C)CCC(C)C2(CCCCC2)C1 N1(C(c2scc(C#N)c2)=O)CCC(C2CCN(C(C3(CF)CC3(F)F)=O)CC2)C1 Cn1ncc(C)c1NC(C1CCN1C(c1cccc(Cc2cccs2)c1)=O)=O c1(C(=O)NCCCCCCN(C(C=CC)=O)C)ccc(C)c(S(C)(=O)=O)c1 C(C)(CC(=O)N1CCC(NC(=O)Cc2ccsc2Br)C1)OC C1(C(=O)NCCN(C(C2CCN(C)CC2)=O)CCOCCO)CCOC(C)(C)C1 c1(CCC(=O)NCC(CNC(C(C)=C2CCC2)=O)(C)C)cc(Cl)cc(Cl)c1 C12(C(N(C3(C(=O)NCC(C)SC)CC3)CC)=O)CCC(OC)C1C2 Cc1nn(C)c(C(=O)NCC2CC3(CC(NC(c4ncoc4C)=O)C3)C2)c1Br C(CN=c1[nH]c(=NCC2(CO)CCCO2)[nH]c2c1CSC2)OCCCO C(c1ccc(F)cc1)=CC(=O)NCC(C)(CO)NC(c1csc(C(N)=O)n1)=O N1(C(CCSCC)=O)CCOCCC1C(=O)NCCn1ccnc1C c1(C(=O)NCC2N(C(c3scc(C)c3Cl)=O)CCCC2)nnc(O)nc1O Cc1cc(C(=O)NC2CCCN(C(c3cc(C(F)F)cc(F)c3)=O)C2)ncc1F Cc1oc(-c2ccccc2)nc1C(=O)NCC(C)NC(=O)CC1COCC1O Cn1cc(Br)c(CC(=O)NCCCNC(C2(O)CCOC2)=O)n1 C1(NC(C(C2CN(C(Cc3n(C)ccn3)=O)C2)OC(F)F)=O)CCC(=O)NC1=O c1(C(=O)NC2C(C(N3CC(SCC)C3)=O)COCC2)cccc(C#N)c1C Cc1cccc(C(=O)NCC2CCC(C(=O)NC3CCCSC3)CC2)n1 c1(CC)cc(C(=O)NCC2(NC(=O)CNC(c3cscn3)=O)CCC2)cs1 N1(C(C=Cc2c(C)coc2C)=O)CCC2(C1)CN(C(=O)CCC(F)F)CC(C)O2 N1(C(c2c(C)ncc(C)c2)=O)CC2CCN(C(=O)CSS(C)(=O)=O)CCC2C1 C=CCCCCCCC(=O)N1CC2CC1CN2C(=O)C=CCN1CCOCC1 c1(C(N2CCC(CNC(=O)CC3CCCCC3)(CO)C2)=O)cnn2c1OCCC2 N(C(=NCc1cn(C)nn1)N1CCC(OCC(C)(C)C)C(C)C1)CC(=O)NC c1(C(=O)NC(CN(C(C(CC)(C)CO)=O)C)C)ccnc2ccccc12 C(=O)(C(C)(F)C(C)(C)F)NCC(CC)NC(C1(C2CC2)CC1)=O Cc1cc(C(N2CC3CC2CN3C(c2cccnc2SC(F)F)=O)=O)cc(N)c1 Cc1ccc(C=CC(N2CCC(F)CC2C(=O)NCCCS(C)=O)=O)cc1 c1(C(C(=O)OC)N(CC(O)C(=O)NCCOCC2CC2)C)cn2ccccc2n1 Cc1cc(C(N2CCN(C(C3CCCC(F)C3)=O)CC2)=O)c2c(C)n[nH]c2n1 C(C(C)(C)N=c1ccc([N+](=O)[O-])c(C)[nH]1)NC(c1c(C)n2c(s1)ncc2)=O CC1=C(C(=O)NCC2(CCNC(=O)C3=COCCO3)CC2)Cn2ncnc2N1C C1(NC(C2CC(C)OC2)=O)CN(C(c2cnccc2Cl)=O)CCC1C(F)(F)F C(=O)(C(C(=O)NC(Cc1cn[nH]c1)C(=O)Nc1cccnc1O)OC)OCC Cc1ccnc(C(N2CCC(NC(C3(n4cccn4)CC3)=O)C2)=O)n1 C#CCC(CC(F)F)C(=O)NC(C(=O)NC1CCN(C(N)=O)C1)C1(C)CC1 c1(C(C(=O)N2CC(CNC(Cc3cnc(C)[nH]3)=O)C2)(C)O)ccc(F)cc1 c1(C(=O)NC(C(C)C)(C)CNC(=O)C=C2CCN(C)C2)cn2cccnc2n1 C1(CCNC(C2CC(n3cnnc3)C2)=O)CCN(C(=O)CCCc2ccsc2)C1 n1(CC)cc(C(=O)NC2C3CCN(C(=O)CCc4nc(C5CC5)no4)C23)c(C)n1 C1(C(=O)NCC#C)CC(F)CN1C(C1CC(=O)CS1)=O C(C[SH](=O)=O)O.C1(NC(CNC(C)(C)C)=O)CC(NC(=O)CSCC(N)=O)C1 N1(C(C(CC)(C)F)=O)CC2CCC1C(CNC(C1CC(=O)N(C(C)(C)C)C1)=O)C2 c1(CNC(C(CC=C)C)=O)ccc(CNC(=O)COCC2CCOCC2)c(F)c1 C(=O)(C(CC(F)F)C1CCC1)NCC1CCC(NC(c2nnc(C)s2)=O)CC1 c1(-n2c(C3CCCC3)nc(C(C)OC)n2)cc(Cl)ccc1C N#Cc1cccc(C(=O)NC2CCCCC2CNC(=O)COCCCN(C)C)c1 c1(OC(C)C(=O)N(C2CCN(C(C3CCCC3)=O)CC2)C)ccc(Cl)cc1Cl N1(C(C2CCOC2)=O)CC2CCCC(C1)N2Cc1ncsc1Br C(=O)(C1CCCn2ccnc21)NCC(CNC(c1nccc(OC)c1F)=O)(C)C Cc1ncc(C(=O)NCC2CN(C(C3(C)CCCS3(=O)=O)=O)CCCO2)c(O)n1 C1(NC(c2csc(Br)c2)=O)CN(C(=O)CCCF)CC1F C1(CC)CCC(CNC(C2CCC(NCc3cnn(C)c3C)C2)=O)CC1 c1(COCC)nc(N2CC(C(C)NC(=O)CCCc3cccs3)C2)cc(C)n1 C1(C(N(CCCCCC)C)=O)CC(NC(=O)C(C2CC2)SC)CCO1 N1(C(c2c(C)nn(C)c2)=O)CCC(C)(CN(C)C)CC1.N12CC3C(C3C1)C2 C1(C(N2CCN(C(c3nc(C)c(C)[nH]3)CCC)CC2)=O)CC2(CC2)CN1C C1(CNC(CNC(CCCCC)=O)=O)C(C2CC2)CCN1c1ncc(C)c(O)n1 c1(OC)nc(N2CC(NC(C3CC4C=CC3C4)=O)C3(CC3)C2)ncc1C c1(C(N2CC(CN(C(=O)C(O)C3CC3)C)C2)=O)cn2ccccc2n1 c1(CC(=O)NC(CNC(=O)Cc2c[nH]nc2O)CO)c[nH]c2cnccc12 C1(C(N(CCCOC)C)=O)CC(C)CN(C(=O)Cn2cc(C#N)cn2)C1 N1(C(C(C)OCC2CC2)=O)CC2CC(C(=O)NCC3C(C)(C)C3(C)C)(C2)C1 N1(C(c2nc(N(C)C)oc2)=O)CC2CC2(NC(C2CC(C(F)(F)F)CO2)=O)C1 c1(CNc2cn(C)c(C(=O)NCCF)n2)cccc(C(F)(F)F)c1Cl Cc1noc(C(=O)N(C(C)CN(C(=O)CCc2cc(Cl)cs2)C)C)c1C C12(NC(c3cc(O)ccc3F)=O)CCN(C(=O)Cc3c(O)ncnc3O)CC1C2 CC1CC(C(=O)NCCOC2CN(C(c3ccncc3)=O)C2)CCS1(=O)=O C1(NC(C2CC(O)C2)=O)COCCN(C(c2cc(C(F)(F)F)cc(Cl)c2)=O)C1 N1(C(C(CC)(C)CO)=O)CC2CC(C1)C(CO)C2NC(C1CC2CCC1O2)=O c1(OC)ccc(C(=O)NCC2(NC(=O)Cc3ccn(C)n3)CCOC2)c(OC)c1 C(=O)(CCCC(N)=O)NCC(C)(CO)NC(COC(c1nnc(S)n1C)C)=O N1(C(CSc2n(C)cnn2)=O)CCN(C(=O)Cc2nc[nH]n2)C(CC(C)(C)C)C1 Cc1cn2c(C(=O)NC(c3cccc(N4CCOCC4)c3)C)c(Cl)nc2s1 C1(NC(CNC(CC)=O)=O)CCOC(CNC(c2ccc(-c3cccs3)[nH]2)=O)C1 Cc1cccc(C(N2CC3CCC3(CNC(=O)CC(F)(F)F)C2)=O)c1O C1(C(=O)NCCC(=O)OCC2CCCO2)CC(C2CCC2)C1 C1(C(=O)NCCCCNC(c2c(C)cc(F)cc2)=O)CCC2CC1C2(C)C c1(CCC(C)NCC2OCCN(C)C2c2ccccc2)ccc(Br)cc1F c1(SC)ccc2c(c1)OCCO2.c12nnc(-c3ccc(Br)s3)n1CCN2CC CC12COCC1(C)CN(C(=O)C(c1ccccc1)NC(c1cc(C#N)cs1)=O)C2 Cc1cc(C)n(CC(=O)NCC(C(C)C)NC(=O)Cc2ccc(F)cn2)c(=O)n1 C(=O)(CC(=O)NCC1(C(=O)NCCn2cccn2)CCC1)NCC C1(c2cn(CCNC(C3CC(CCO)C3)=O)nn2)CCC2(CCCC2)C1 C1(C(=O)NCCCc2ccncc2)C2CN(C(=O)CC3COCCO3)CC12 C1(CC(=O)NC2CC(C(C)C)C2)C2CCCC2N1C(c1ccn(C)n1)=O n1(CCC(N2CCN(C(C(CC)F)=O)C(C)C2)=O)c(=O)n(C)c2ccccc12 c1(C(N2CC(O)(CNC(CC(C)C)=O)C2)=O)ccc(Br)c2ncccc12 N1(C(CC2ON=C(CC)C2)=O)CC(CNC(=O)C2=CCCC2)OC2CCCC12 c1(C(=O)NCC(CCC)C(=O)NC2CCc3nncn3C2)cc2cccnc2[nH]1 c1(CSC)ccc(C(N2CCCC2C(C)(C)NC(=O)C=CI)=O)o1 C1(NC(C(CC)OCC)=O)CN(C(c2ccc(CN(C)C)o2)=O)CC1C1CC1 Nc1ccccc1C(=O)CCC(=O)N1CC(NC(=O)COCc2ccccc2)C1 C=CCC(CC)N=c1[nH]c(N2CCOC3(CCSCC3)C2)nc2c1COC2 C(C(C(C)(C)C)NC(=O)CCC1CCCN(C)C1)OCC=C C(=O)(C(C(C)C)C(C)C)N(C1CCN(C(c2ccc(CC)c(Cl)c2)=O)C1)C C1(CNC(COCCN(C)C)=O)CC2(CCN(C(=O)CCc3cc[nH]n3)C2)CO1 c1(C(=O)NCC(C)NC(C23CCC(C2)C3)=O)cn(C)nc1-c1ccccc1 c1(OC)cccc(C(=O)N(CCNC(=O)COc2cccc(C)c2)C2CC2)c1F Cc1ncnc(C(=O)NCCOCCC(=O)NCCC2CCC3(CCC3)O2)c1C C1(CC)(NC(=O)CC=Cc2ccccc2)CCN(C(C2CCOC2=O)=O)CC1 c1(C(C)C)c(C(=O)NC2(C)CC2(C)C(C)C)cnn1-c1ccccc1 O=S(=O)(C1Cc2ccccc2C1)N1c2ccc(Br)cc2CCC1C(F)(F)F C1(C)(C(N(C)CCNC(C2CCCC3(CCCC3)O2)=O)=O)Cc2ccccc2C1 c1(C(=O)NCC2N(C(C(Br)=C(C)C)=O)CC2)ccccc1C1CC1(F)F C(=O)(CCC(F)(F)F)N1CC(CCNC(C2C(CC(C)C)C2)=O)C(C)C1 C1(C(C(=O)NCC(=O)OCC2CC(C(=O)NCC(F)(F)F)C2)F)CCOCC1 c1(-c2n(C)c(CSc3nccc4c3CCCC4)nn2)cc(O)c2cnn(C)c2c1 N1(C(COCCC)=O)CCN(C(C2CCCC3(CC3)C2)=O)CCC1C O(C=CC(=O)NCCc1ocnc1CNC(=O)C(O)Cc1ccccn1)CC Cc1cc2c(C(=O)NCC3C(C)CCN3C(C3CN(C(N)=O)C3)=O)cccc2[nH]1 CC(O)C(C)(C)C(=O)NC1CC(CCNC(=O)COc2cc(F)cc(F)c2)C1 c1(CC)[nH]nc(C(=O)NC(c2cnn(C)c2)C(=O)NCc2ncsn2)n1 C(C(=O)NCCC1COCC1O)(C(C)CC)NC(C(CC#C)C1CC1)=O CCC(CNC(=O)C(CCSC)OC)(CC)NC(=O)Cc1n[nH]c(C)n1 C1(CCN(C(C(CSC)C)=O)C2CC2)CCCCN1C(=O)CCN1CCC1 CC1CN(C(C2(C)CCN(C(C3CCC(=O)N(C)C3)=O)CC2)=O)c2cccnc21 CC(C)C(F)(CNC(c1ccncc1F)=O)C(=O)NCCC1C=CCC1 N1(CC)CCCN(C(c2ccoc2C)C(=O)NCC2CC2)CC1=O C1(C(C(=O)NCCC)N(C)CCc2cccc(Cl)c2)CCOC2(CCC2)C1 N1(C(CCC2N(C(c3ncn(C(C)C)c3)=O)CCCC2)=O)CC2CCCC2C1 CCC(C)CCCCC(=O)NC1CN(C(c2cc(Cl)c(Br)cn2)=O)C1 Cc1nc(NCc2ccc3ncoc3c2)cc2nncn12 N1(C(C(C=C)O)=O)C2CC1CN(C(=O)CC(C)NC(N)=O)C2 C1(OCC)CCCN(C(c2ccc(C(F)(F)F)o2)C(=O)NC(C)C)C1 C1(CC(N)=O)(NC(CCCCOC)=O)CCN(C(c2ccc(CO)cc2F)=O)CC1 C1(C(N2CC3CC(CO)C(C3)C2)=O)C(C2CC2)CCN1C(c1ccc(O)cn1)=O Cc1c(F)cc(C(=O)N(C2CCCN(Cc3cccc(Cl)c3)C2)C)c(F)c1F C1(CC)(CC)NC(=O)N(CC(N2CC(NC(=O)COC(C)C)CCC2C)=O)C1=O n1(CC2CC(n3cc(CCn4ncc(N)c4)nn3)C2)c(O)nc2ccccc12 c1(CC(C)N(S(=O)(=O)Cc2ccccc2F)C)ccc(F)cc1F C(=O)(C1=CCCCCC1)NCC1(C)N(C(CCn2ncn(C)c2=O)=O)CCC1 N1(C(C=CCC)=O)CCCC(C(N2CC(C)(C)C2C(C)C)=O)C1CC C1(C(=O)NCC(CC=C)NC(c2ccccc2CSCC)=O)C2CCCCC12 C(=O)(CCCC(=O)N1CCN(C(=O)C(F)=C2CCCC2)CC1C1CCC1)OC c1(-c2c(C)ccc(CO)c2)cnn2cc(C(=O)Nc3nccc(Br)c3F)cnc12 c1(-n2cc(CC(CO)NCc3ccsc3Br)nn2)ccc(Br)cc1 C=CCC(CC(C)C)C(=O)NCCCCC1CN(C(c2cc(N)cc(N)c2)=O)C1 Cc1c(C(=O)NC(C)(C)CNC(C2(CCN(C)C)CC2)=O)cccc1F C12(OC)CCC(C(=O)NCC3CN(C(C4CC(F)(CO)C4)=O)CC3C)(CC1)CC2 C1(O)(C(CC(CCO)c2cncn2C)C)CCCCC1.C(=O)(C(=O)N)N N1(C(CC=C)=O)CCCCC1CNC(=O)CCNC(c1ncc[nH]c1=O)=O C1(O)(CNC(C(C)(c2ccccc2)N(C)C)=O)CCN(C(C2CCOC2)=O)CC1 c1(C(=O)NC(C2CCCC2)CC)c[nH]c2cccnc12 c1(C(=O)NC2CCN(C(CC#C)=O)CC2O)ccc2nc(Cl)ccc2c1 S(=O)(=O)(c1ccc(C)c(C)c1)N1CC(C)CC(NC(CCCCCCCC)=O)C1 N1(C(C2(C(C)(F)F)CCOCC2)=O)CCCN(C(c2cc(Cl)cnn2)=O)CC1 CC1CCc2[nH]nc(C(N3CC4CC(C3)N(C(=O)CCN3CCCC3)C4)=O)c2C1 C1(COC)(NC(=O)CC(C)N(C)C)CCN(C(=O)COc2ccc(F)cc2)C1 C1(C(=O)NCC(C)(C2CC2)NC(c2cc(Cl)ns2)=O)CN2CCCCC2CO1 C#CCCCCCC(=O)N1CCC2CN(C(c3cc(F)ccc3OC)=O)CC12 CC(C)C(C(=O)NCCC1COCCN1C(c1csnc1Cl)=O)N(C)C CCCCCCC(=O)NC1CS(=O)(=O)CC1NC(c1cnn(CCC#N)c1C)=O C1(CC)(CC)CCN(C(=O)C(C)N(C(=O)CC2=CCCC2)C2CC2)CC1 CC(CCCCNC(C1C(C)(C)C1(C)C)=O)NC(=O)Cc1c(Cl)cnn1C N1(C(C2CCC=CO2)C(=O)Nc2ccc(OC)cc2)CC(OC)CCC1C CC1CC(C(N2CCC(NC(=O)CCCCCN(C)C)C2)=O)CC(=O)N1 Cc1ccc(CC(=O)NCC(CC(C)C)NC(C2CC3CCCCC23)=O)c(F)c1 C(=O)(CC(C(F)(F)F)NC(C1CC(CF)C1)=O)N(C(C)C)Cc1ccco1 C1(C(N(CCCOC)C)=O)CCN(C(=O)COC2CC2)C1C(C)C N1(C(c2c(OC)csc2)=O)CCCC2C1CCN2C(=O)C(N1C(=O)CCC1=O)C c1(C(N2CCC(N(C)C(c3ccc(O)c(Cl)n3)=O)C2)=O)ccc2c(c1)NC(=O)C2 C1(CN=c2nc[nH]s2)(Nc2sc(C(=O)OC)c(C)n2)CC(O)C1(C)C CCC(CC(=O)NCC(C1CCCCN1C(=O)Cn1nccc1C)(C)C)OC C(C(O)C(F)(F)F)N(CCS(=O)(=O)CNC1CCC(OC)C1)C.C(C)(C)(C)OCC(=O)O Cc1nn(CC(=O)NC2CCCC2NC(C2(c3ccc(O)cc3)CC2)=O)cc1Cl c1(C(=O)NC(CC=C)CNC(=O)C(COC)N(C)C)cc(COC)ncn1 C1(O)(C(C)NC(c2c(OC)c[nH]n2)=O)CCN(C(C2CCC(CO)CC2)=O)CC1 c1(C(=O)NCC(CNC(C2(C(C)C)CNC(=O)C2)=O)O)nc[nH]c2nccc1-2 Cc1nc(C(C)C)nc(O)c1C(=O)NC1CCC1CNC(C1(CO)CC1(F)F)=O c1(-n2c(CCCOCCOC)nc(-c3ccnc(Cl)c3)n2)ccc2nncn2n1 C1(CC)(NC(=O)C(O)Cc2cnc[nH]2)CCN(C(C2CC(=O)NC(=O)N2)=O)CC1 Cc1cccnc1CCC(=O)NCC1(F)CCN(C(=O)CN(C)S(N)(=O)=O)C1 C1(C(=O)NC(C2CN(C(=O)Cn3ccc(O)nc3=O)C2)C)CCn2nncc2C1 N1(C(C=C(C)c2cccnc2)=O)CCC2CC2(NC(=O)CS(N)(=O)=O)CC1 C1(NC(=O)C=C(Cl)Cl)CCCC2CN(C(C3CCCC4CCCN34)=O)CC12 C1(CC=C)(NC(c2ccoc2)=O)CCN(C(=O)C(CC)c2ccccc2)C1 N1(C(C2COCCN(c3cccc(CC)n3)C2)=O)CCCc2nc(C#N)ccc21 N1(C(c2cc(C)on2)=O)CC2(C=C(C(=O)NC3CCOC(C(C)C)C3)CO2)C1 Nc1cc(C(=O)NC2CCCN(C(C3CC(CC4CC4)C3)=O)CC2)cc(O)c1 C1(C(=O)NC2(C=C)CCCC2)CC12CCN(C(C1CC(=O)C13CCC3)=O)C2 C(=O)(C(C)(F)C(C)(C)F)NC1CN(C(c2ncc(C)cn2)=O)CC1(C)C CC1(NC(=O)Cc2nc(C3CC3)nn2C)CCN(C(C2CCCC23CC3)=O)CC1 N1(C(C(C(=O)NC)(C)C)=O)CCC2(CC1)CC(C)N(C(=O)C=CC=C(Cl)Cl)C2 c1(CN2C(C(=O)OC)CC(O)(C(F)(F)F)C2)cc2cnccc2o1 c1(SC)cn(C)nc1C(=O)NC1CCCC1NC(c1ccnc(C2CCC2)c1)=O Cc1ccc(I)c(C(=O)NCCC2CCCN(c3nc(C)cc(C)n3)C2)c1 C=CC(C)(C)CC(=O)NCCC1C(C)CCCN1C(=O)Cc1cn2ccsc2n1 CCC(CCC(=O)NCCCC(CO)NC(C12CC(C)(CCO1)C2)=O)OC C1(NC(=O)CC2CC=CCC2)CCOCC1NC(=O)C(O)(C1CC1)C1CC1 c1(C(N2CC=C(C(=O)N(C3CCCOC3)CC)C2)=O)cccn2ccnc12 C(C(F)(F)CCC(=O)NC1CCSCC1)n1cc(C2COC(C)(C)O2)nn1 C(C(O)C(=O)NC(CC1CCOCC1)C(=O)NC1CC(O)C1)SC O=C1CCC(C(=O)N2CCC(N(C(=O)Cc3cccc(F)c3)CCO)C2)=NN1 C(=O)(C1=Cc2ccccc2C1C)NCCN(C(C(CC)CC1CCCC1)=O)C c1(CC)nn(C)c(C(=O)NCCCC(C)NC(C2(COC)CC2)=O)c1Cl C1(NC(CSC)=O)CCCC12CCN(C(c1nc(N)cc3ccccc13)=O)CC2 c1(C(N(c2ccc(C)nc2)C2CCCC2)=O)cc2c(=O)[nH]ccn2n1 c1(NC(c2n(CC)nnn2)(C)CSc2nncs2)ccc2ncccc2c1 c1(C(N2CCCC2)=O)cc(CNC(=O)C(C)(C)C(N)=O)c(F)cn1.CO c1(C(=O)NCC(N(C(=O)C(F)n2cccn2)C)C2CC2)cc(Cl)on1 c1(OC)cc[n+]([O-])c(C(N2CCC(NC(c3coc(C)n3)=O)C2C)=O)c1 C(=O)(C(n1nnnc1C)=C(C)C)NC(C1N(C(CC(=O)NCC#C)=O)CCC1)C N1(C(C2N(CCCC)CCCC2)=O)CCCN(C(=O)Cc2cnsc2)C(CO)C1 C=CCC(CNC(=O)CCc1ccc(C)o1)C(=O)NCC(COC)C(C)C c1(CC(=O)NCC2N(C(C(C)CSC(F)(F)F)=O)CC2)coc2ccccc12 CCCC(O)CC(=O)N(CC(C)(C)CNC(c1cc(OCC)n[nH]1)=O)C C12(NC(c3cnn(CC(F)F)c3)=O)CCCC1CN(C(=O)COCC1CCC1)C2 N1(C(C(CCC)C#N)=O)CC(C2CCCN(C(c3ccnc4[nH]cnc34)=O)C2)C1 C(=O)(C(O)C1=CCCCC1)N(CC(=O)NC1C2(CC(OC)C2)C1)C n1(CC)nc(C(N2CCCC2C(C)(C)CNC(=O)COC(F)(F)F)=O)ccc1=O C(=O)(CS(=O)c1cccc(OC)c1)N1CCCC(C(=O)O)(CC)C1 C1(CNC(Cc2ccc(C)nc2)=O)CCC2(CCC2)C1NC(=O)CC(C)(F)F CC1(C)CC(CC(N2CCC(CCF)CC2)=O)CN1C(=O)C1=NNC(=O)C1 c1(C(=O)NC2CC(F)(F)C2)cc(Br)ccc1F.C12CCC(C1)Cn1cc(nn1)CN2 C(=O)(C(C(C)C)[N+](C(C1CCCC1)=O)([O-])NC)NCCCN(C(=O)C(C)C(C)O)CC C1(CO)(NC(=O)NCC(C)OCC=C)CCc2cc(Br)ccc21 c1(OC)ccc(OCc2nc(CC3CSC3)n(Cc3ccccc3)n2)cc1 CC1(C)OCC(CNC(C23CC(NC(c4cnco4)=O)(C2)C3)=O)O1 Cc1cc(-c2nn[nH]n2)c(C(=O)NNC(c2ccc(F)cc2Cl)=O)c(O)n1 C1(O)(CNC(=O)COCCOc2ccccc2)CCN(C(=O)C2=CCCCC2)CC1 Cc1ccc(Cl)c(C(=O)NC2CCN(C(C3NC(=O)OC3(C)C)=O)C2)c1O C1(C2CCN(C(=O)CCC3CC3)C2)(NC(=O)CC2CCOC2)CC1 C1(NC(C(CSC)C)=O)CCCN(C(=O)CCc2ccsc2Cl)CC1 c1(C(=O)NCC(C(C)(C)C)NC(c2c(C(C)C)ocn2)=O)nnc(O)cc1O c1(NC)nc(C)ccc1C(=O)NC(C)CNC(C1(c2cccc(F)c2)CC1)=O C(=O)(C1Cc2ccccc21)N1C(CCNC(c2ccc3c[nH]nc3c2)=O)CCC1 C1(CCN(C(=O)C(O)C2CCC2)C)CCCCN1C(=O)COc1ccsn1 C(=O)(C1=CCCOCC1)NC(CC)CCC(=O)N1CCN(C2C(=O)NCCC2C)CC1 C=C1CC(C(=O)NOCC2(C)CC2)(CNC(c2ccnn2C)=O)C1 N1(C(c2c(C)scc2)=O)CC2CC(C)N(C(=O)C3=CCCC3)C2C1 N1(C(c2c(CCC)nns2)=O)Cc2ccc(CNC(C3CC(OC)C3)=O)cc2C1 C(=O)(CCC(=O)NN(C)C)NCC(CNC(C(C=C=C)C)=O)S(C)(=O)=O n1(CC(=O)NC(CN(C(=O)C(N2CCSCC2)C)CC)C)cnc(Br)c1 N1(C(CC(CN(C)C)O)=O)CCCC(C)(NC(=O)C(C2CC(F)(F)C2)O)C1 N1(C(CC=CC=C)=O)CCCN(C(=O)C(N2CCC(C)C2)=O)CC1CO C1(NC(C2CC(=C)C2)=O)CC12CCN(C(C13CCC(=O)N1CCS3)=O)CC2 C(=O)(CCCS(C)(=O)=O)N(C)CC1CCN(C(C(C(C)C)SC)=O)C1 C(=O)(C(C(=O)N1CCCN(C(=O)CS(N)(=O)=O)CC1C)C(C)(C)C)OCC Cc1nc(C(N2CCC(NC(=O)CCc3ccn(C)n3)C2)=O)c(C(F)(F)F)[nH]1 c1(CC(=O)NCC2CCN(C(C(CCN(C)C)O)=O)CC2)cccc2sccc12 C1(CNC(=O)CC2CC2(Cl)Cl)CCC2(CCN(c3cc(C(F)F)ncn3)CC2)CO1 CC(=O)CCCC(=O)NC(CCC1CCC1)C(N1CC(CO)CC(C)C1)=O c1(NCCc2cccc(OCC)c2)nc[nH]c(=NCC(C)(CO)OC)c1C C1(C(=O)NCC2CC(CNC(C3C(CC(=O)OC)CCO3)=O)C2)CCSC(C)C1 CC(CN(C)C)CCC(=O)N1CC(O)C(O)C1CNC(c1coc(C(N)=O)c1)=O c1(C(=O)NC(C(C)C)CNC(=O)Cn2nccn2)ccc(S(N)(=O)=O)cc1N N1(C(Cn2ncc(C#N)c2)=O)CCC2C(CCN2C(=O)CCNC(C2CCC2)=O)C1 C1(CC=C)(NC(=O)CC2CCNC2=O)CCN(C(=O)C(O)CCSC)C1 C1(NC(c2c(OCC)ccs2)=O)CCCN(C(c2csc(-c3nc[nH]n3)n2)=O)C1 c1(N(C2C3CNCC23)C(c2cc(OC)c(F)cc2)=O)ncnc2c1CCC2 CC1CC(=O)NCC1C(N1CC(O)(C(C)(C)CNC(C2CCN2S(C)(=O)=O)=O)C1)=O c1(C(N2CC(NC(Cc3cnc(C)[nH]3)=O)(CO)C2)=O)cccc(SC(F)(F)F)c1 c1(NC(CN2CCN(C(c3nc(C)nc(Cl)c3)=O)CC2)=O)ccn2c(O)nnc2c1 c1(C(=O)NCC(C)NC(c2cncc(-n3ccnc3)n2)=O)ccc2nsnc2c1 N1(C(C(CC)OC)=O)CCCN(C(C(C(=O)OC)C2(C)CC2)=O)CC1 c1(C(N2CC(F)(CNC(=O)CC34COCC(C3)C4)C2)=O)cc(O)nc(O)n1 Cn1ccnc1C(=O)NCCCCCNC(C1CC(CC2CC2)C1)=O c1(C(C)C)ccc2c(c1)OC(C)CN2CC(C)OC1CCOC1 S(=O)(=O)(c1ccc(C(=O)NC2(CN(C(=O)C(CO)C(C)(C)C)C)CC2)cc1)NC c1(CNC2CCCN(C(=O)OCC)C2)ccc(Br)cc1Cl C1(C(N(C(CN(C(C)=O)C)C)C)=O)CC2(CC(NC(C3(Cl)CCC3)=O)C2)C1 Cc1cc(C)c(CNC(C2CCN(Cc3cccnc3F)CC2O)=O)cc1C CC(C)CCCC(C)CNC(C1C2CC3C(C2NC(C2CC2C2CCCO2)=O)C13)=O c1(C(CNC(C(CCC)=CCC)=O)NC(C2COC(=O)O2)=O)ccc(F)cc1F O=C(C1CCc2nccn21)N1CCC(CC(=O)N2CCC(CO)O2)(F)C1 C1(C(=O)NCCOCC(=O)NCC2C(C)(C(F)F)C2)Cc2ccccc2C1 CN1CCC(C)(C(N2CCCC(n3cc(CCNS(C)(=O)=O)nn3)C2)=O)CC1 N1(C(=O)Cc2cccc(F)c2)CCCC(NC(C2(CF)CCC2)=O)CCC1 CCCCC(O)CCC(=O)NCC(C)(C1CCC1)NC(=O)CC(C)(O)C(F)(F)F c1(C(C(=O)NC2CC(C(=O)OC)C2)N(CCCC)C)cnc(C)nc1 N1(C(C2CC(CCC)C2)=O)CC(C(=O)NCC2CC(CC3CC3)C2)C(F)(F)C1 N1(C(c2ccc(COC)o2)=O)CC(C)(C)CC1CNC(c1ncsc1C)=O N1(C(c2c(C)nc(C)nc2C)=O)CCC(NC(=O)COCC(C)C)CC(C)(C)C1 c1(C(n2ccnc2-c2cnn3ccccc23)C)ccc(N=[N+]=[N-])cc1 C1(NC(C2N(C(C)(C)C)CC2)=O)CC=C(C(=O)NC2(C)CCOC2=O)C1 C(=O)(C(CC(F)F)N(C)C(C1CCCCN(C)C1)=O)NC1CC(OC(C)C)C1 C1(C(=O)NCC(=O)NCCOCCCNC(CCCC)=O)CCCCC1 C1(C)(C(N2CC(CN(C(c3c(C)cc[nH]3)=O)C)OCC2)=O)CCCCNC1=O Cc1nn(CC(N2CCOCC2CNC(c2cc(F)cs2)=O)=O)c(C)c1Cl c1(C(=O)NC2C(C(N3C(C(N)=O)CCCC3)=O)CCC2)ccc(O)cc1O N1(C(C2C(C=C)C2)=O)CCCC(CCNC(=O)CC(C)(C)OC(C)=O)C1 CC1CCCN(C(=O)Cc2cnsc2)C1CNC(c1ncccc1N)=O CCC(CNC(=O)C(C)C1CC1)(CC)NC(c1cc(C2(C)CC2)on1)=O N1(C(c2c(CC)nns2)=O)CCCCC1CNC(c1cc[nH]c1-c1ccccc1)=O N1(C(COC(C)C)=O)CCOCC(C)(CNC(=O)COc2ccn(C)n2)C1 N#Cc1ccc(NC(C2CC2NC(c2ccc(F)c(F)c2Br)=O)=O)c(C#N)c1 Cc1cc(C(N2CCC(C(C)NC(c3nocc3C)=O)C2)=O)c(N)s1 n1(CC)nc(C(=O)N(C)CCOCCC(=O)NC2(C(N)=O)CCCC2)cc1C C1(NC(C(F)=CCC)=O)CCC(C)N(C(c2ccnc(OC(C)C)c2F)=O)C1 c1(C(N2CCC(C(C)NC(C3CCC(=C)CC3)=O)CC2)=O)cc2cc[nH]c2cn1 CN1CC(CC(=O)NCC(O)CNC(C2(C3CC3)CCC2)=O)C(O)C1 c1(C(N)=O)ccc(F)nc1NC(C1CCCN(Cc2cn[nH]c2)CC1)=O C12(NC(COCCOC)=O)CC(C1)N(C(=O)COCCC(C)C)C2 C(=O)(CC1=CCOCC1)N1C(C(=O)NCC2(C=C)CCC2)CCC1C c1(CC(=O)NC2(C)CC(NC(C3C(C)(COC)C3)=O)C2)cccc(F)c1 C1(C(N2CC(F)(CNC(C3CCCCO3)=O)C2)=O)Cc2cc(Cl)ccc2O1 Cn1ncc2c(C(N3CC(NC(c4nsnc4O)=O)CC(O)C3)=O)ncnc12 C(c1ccc(O)cc1)=CC(=O)NCCCN(C(C1(C)CCC(C)C1)=O)C NC1COC2(C(=O)NC(Cc3ccccc3)CCCO)CC1C2 c1(C(=O)NCCCN(C(C2CCCN(C(C)=O)C2)=O)C)cncc(Cl)c1C N1(C(c2c(CC)nc(C)[nH]2)=O)C(CNC(=O)CC(CC)C(C)C)CC2COCC12 C(=O)(C1CCCn2cnnc21)NC(CNC(c1c(OC)c[nH]n1)=O)(C)C1CCC1 c1(C(=O)NCCN(C(=O)C(C)C#N)CCOC)c(OC)ccc(Cl)c1Cl C1(C(=O)NCC(CN(C)C(c2ccnn2C2CC2)=O)O)CCN(CC(F)F)CC1 C(C)(CNC(C1CCN1Cc1ccccc1)=O)(CO)NC(CSC)=O c1(C(=O)NC(CN(C(=O)Cc2cnc[nH]2)CC)C)[nH]c(C)cc1C c1(SC)cc(C(=O)N(C)CC2(O)CCN(C(c3[nH]c(C)nc3C)=O)C2)ccc1F N1(C(=O)CCCc2cnccn2)CCC2(CCN(C(C3SCCS3)=O)C2)C1 C(C)(C)(CCC(=O)N(C)OC1CCCC1)NC(C(C(C)C)C#N)=O C1(C)(CC)NC(=O)N(CC(=O)N(C)CC2CCCN2C(=O)C=C(Cl)Cl)C1=O c1(OC)ccc(Cl)c(C(=O)NC(C)C(C(C)C)NC(c2nncs2)=O)c1 c1(CCC(N2CC3C(NC(C(C)(O)C4CC4)=O)(C3)C2)=O)ccc(Cl)c(F)c1 C(=O)(CC1OCc2ncccc21)NCCC(C)NC(c1cnc(CC(C)C)s1)=O C1(NC(c2cc(CC)ncn2)=O)CN(C(C2(CF)CC(F)(F)C2)=O)C(C)(CC)C1 c12ccc(cc1)CO2.N1(C(C2(F)C(C)C2)=O)CCOC(c2nccs2)C1 Cc1cc(CNc2ccnc(C(N)=O)c2)sc1Br.C12(CCC1)CC(=O)N2 C1(CNC(CCCn2cc(CCCC(C)O)nn2)=O)CCCC2(C1)OCCO2 C(CCN=C(NCC1(O)CCCC(C)C1)N1CN(C)C(=O)C1C)OC C#CC1C(C(=O)N(C(C)CNC(C2(CCN(C)C)CC2)=O)C)C1(C)C C1(OCC)CCCN(C(=O)C(C(C)C)N(c2cccc(Cl)c2)S(C)(=O)=O)C1 CC1CN(C(c2ccccc2-c2nc(S)n[nH]2)=O)CCN1C(=O)Cn1ccnn1 c1(OC(C)C)ccc(C(N2CCN(S(=O)(=O)CC#N)CC2C(C)C)=O)cc1Cl c1(C(N2CCC(CNC(CC(C)SC)=O)C2)=O)ccc([N+](=O)[O-])c(C)n1 c1(OC)c[nH]c(C(N2CCC(NC(c3ccc(F)o3)=O)C(F)C2)=O)cc1=O C(=O)(CC(C(C)C)C(C)C)NCC(=C)CCNC(=O)CCN1CCN(CC)CC1 CC1CN(C(C2CCN(C(c3cc(Br)c[nH]3)=O)CC2O)=O)CCN1C c1(OC)cncc(C=CC(=O)NCC2C=CC(NC(C3(F)CC=CCC3)=O)C2)c1 C1(NC(c2ccc(COC)s2)=O)CCCCC1C(N1CC(OC(=N)O)C1)=O C1(CC#N)CN(Cc2ccc(Cl)cn2)CCN1C(c1ccc(O)c(F)c1)=O C(C1=CCCOC1)N(C)CC1CCC(C)(C)C1 Cc1ccnc(O)c1C(N1CC(CC(=O)NC(c2cccc(O)c2)C)C(C)C1)=O C(=O)(CCCCCNC(=O)C=CCN(CC)CC)NCCC(CCC)C1CC1 c1(C(N2CC(CCNC(COCC)=O)OC(C)C2)=O)nccn2ccnc12 CN1CCCC(C(N2CCC(C)(NC(=O)C=Cc3cnc[nH]3)C2)=O)C1 C1(O)(C(=O)NCCC(C(=O)N(C(CC)CC)C)O)CCC(C)CC1 C1(CC)(NC(c2ccc(=O)n(CCF)n2)=O)CCN(C(=O)C(C)CC(C)C)CC1 C1(CC(=O)NCC(C2CCCCC2)NC(C(COC)O)=O)(CO)CCOCC1 C1(NC(C)=O)CC2C(NC(=O)CCn3cncn3)C2C1 N1(C(CN2C(C)CCC2)=O)CCC2(CC1)CC2NC(c1cc2nc[nH]c2cn1)=O C(CCN(C(=O)Cc1ccc(COC)cc1)C)(C(C)C)NC(CCSC)=O CC1CN(C(c2ccnc(C3CC3)c2)=O)CC1NC(=O)C(N1CCSCC1)C C(=O)(C1=NOC(C)(C)C1)NC(CCNC(c1c(C)cc(CC(C)C)o1)=O)C c1(C(N2CCC(CC#C)(C(=O)NC3CCC(O)C3)C2)=O)cccc(F)c1O C1(CC(NOCC=C)=O)CCCN(C(c2ccc(COC)cc2)=O)CC1 C1(NC(Cn2ccc(C)n2)=O)CN(C(=O)CC2CC3(CCC3)C2)C2CCCCC12 C(C)(C(CC(=O)NCCN1CCCCCC1=O)NC(=O)Cc1ccnn1C)OC c1(CCC)cccc(CNC(C2CC3CCC3C2)c2n(CC3CCC3)nnn2)c1 C=CC1CN(C(c2c(C)coc2C)=O)CC1NC(=O)COCc1nccn1C CC1=C(C(=O)NCCC2CCC(NC(C3CCN(C(N)=O)CC3)=O)C2)CCO1 C1(C(=O)NCCCC2(NC(C3CSCCS3)=O)CC2)CC2(CC2)C1 Cc1c(C(=O)NCC2(CS(C)(=O)=O)CCCO2)cccc1O c1(C(N(C(C)CNC(=O)COCC2CC2)C)=O)cc2ccc(F)cc2o1 c1(C(=O)NCC(C)NC(c2[nH]ccc2C2CC2)=O)cn(CCN(C)C)nn1 c1(CC(=O)NCC2OCC(CNC(=O)C=CBr)C2)cc(Cl)ccc1O C(=O)(CS(C)(=O)=O)NC1(C)CC(C(=O)NCc2ccc(C(N(C)C)=O)cc2)C1 Cc1nn(C)cc1CCNC(=O)CCC1CCC(NC(=O)COC2CCOC2)C1 C1(C(C)NC(C2(CC)COC2)=O)CCN(C(c2ccncc2C)=O)CC1 C1(C(N2C3C(NC(C4C(C)(C)CCO4)=O)C(C3)C2)=O)CC2CCC(C1)C2 C(CC(=O)NCC1CC(=O)N(C)C1)(C(F)(F)F)NC(c1c(C(C)(C)C)con1)=O N1(CC(C)NC(N2CCCCC2)=O)CC2(C)CC1CC(C)(C)C2 CC1CCC(C)N1CCCNC(=O)NCC1(c2ccc(Br)cc2)CCCCC1 C1(CC=C)(NC(c2occ(C)c2C)=O)CCN(C(c2scc(OC)c2OC)=O)C1 N1(CC(=O)N(CC(C)NC(c2ncc(Cl)cc2F)=O)CC)CCn2ccnc2C1 Cc1scc(C(=O)NC2CCN(C(c3cccc(CO)c3)=O)C2C)c1C C1(CNC(=NCC=C)NCC(=C2CCCCC2)F)CCC2(C1)CC2(F)F CC(C)CC(CCO)NC(=O)C(C)(C)C1CCN(C(C23CCCC2CCC3)=O)C1 C(=O)(CCCCc1cnc[nH]1)NC(C(C)NC(C(C)CN(C)C)=O)(C)C c1(C(N2CC(O)(CCNC(C3CC(=C)C3)=O)C2)=O)ccn2cc(C)nc2c1 c1(C(N2CCC(C#N)(NC(=O)CC(F)(F)F)C2)=O)cc([N+](=O)[O-])ccc1Cl C1(CCC)CN(C(c2c[nH]c(=N)s2)=O)CCN1C(=O)Cn1nccn1 c1(NC(N2C(C(C3CC3)OC)CCCC2)=O)ccc(C2CC2)c(C)c1 N1(C(C(C)(C)NC(=O)OC)=O)CC2(CCCCN2C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CNC(c2n[nH]c(CC)c2Cl)=O)N(C(c2cnc(CC)s2)=O)CCCC1(C)C CCCNNC(=O)CCCCCCCC.C(=O)O c1(C(=O)NC2CN(C(c3c(OCC)scc3)=O)C(C)CC2)cccc2c1NCC2 c1(OC(C(=O)NCC(CC=C)NC(=O)CCOCC)CC)ccc(C)cc1 N1(C(C2CCC(CC)O2)=O)CCC(O)(C(C)NC(=O)C=C(C)C(C)C)CC1 c1(OC)cccc(C(CNC(=O)CSC)NC(C23CC(F)(CO2)C3)=O)c1 c1(OC)ccc(NC(=O)C(O)C2CN(C(c3cc(C)sn3)=O)C2)c(O)c1 C(=O)(CC(N=c1[nH]c(N(CC(C)(F)F)C)nc(=N)[nH]1)c1cccc(OC)c1)NC C1(C2CCN(C(=O)C(C)(O)C3CCOC3)CC2)(NC(CSCC)=O)CCC1 c1(C(N(C)CC2OCCN(C(CCC=C)=O)C2)=O)ccn2ccnc2n1 Cc1oc(C2CC2)nc1C(=O)NCCC(C)CCNC(C1CCS(=O)(=O)N1)=O N1(C(C=CC=CCC)=O)CCC2CCC(C1)N2C(c1cnc(OC)c(C)c1)=O c1(CC(=O)NCCCN(C(=O)CSC2CCOC2=O)C)cccc([N+](=O)[O-])c1 C1(C(=O)OC(C2CCCCC2)C)CC2(CO1)CC(F)(F)C2 C12(C(=O)NCC(CO)OC)CCCC1CCN2C(=O)C(C)c1cc[nH]n1 c1(C(=O)NC2(CCNC(=O)C=CC3CC3)CC2)ccc2ncnc(O)c2c1 C(=O)(C1=CCOC1)NCC1CN(C(CN(C)Cc2cccc(Cl)c2)=O)C1 CCCCC(C)(F)C(=O)NC(CO)C(C)NC(c1cc(C)nn1CCC)=O CC1CN(C(=O)CCCc2ncco2)CCCN1C(c1ccsn1)=O c1(OC)cc(C)c(C(N2CC(NC(=O)CCC=CC(C)C)C(C)C2)=O)cn1 C12(C(NOCC(=O)N(C)C)=O)CCN(C(C3CCC(F)(F)C3)=O)CCC1C2 n1(CCC)nc(C)c(C(N2CCOCC(CNC(C3CCC3CF)=O)C2)=O)c1C C(CC(=O)NC1CN(C)CC1(C)C)(C(F)F)NC(CC1(NC(C)=O)CC1)=O C1(C(N(C)C[Si](C)(C)C)=O)(NC(c2ccc(CC)[nH]2)=O)CCC(C)(C)C1 CCC(C)CC(=O)C(=O)NCC1CC1NC(c1ccccc1F)=O c1(N(C(C)=O)C)nc(CNC(=O)Oc2ccccn2)cs1 N1(C(c2c(CC)nn[nH]2)=O)CC=C(C(C)(C)C(=O)NC2(C)CC2(C)C)C1 c1(C(=O)NCC(C2CCCCC2)NC(=O)C2=CCCS2)ccccc1OC(F)F c1(NCCOCCNC(Cc2cc(C)[nH]n2)=O)c(C#N)cccc1[N+](=O)[O-] c1(COCCCNC(=O)NCc2cccc(OC)c2)ccn(C)c(=O)c1 c1(C(C(C)C)=O)ccc(C(=O)NC2CCC2)cc1.c12cn(nn1)CCCS2 C1(C(=O)NCCC2CCCCC2)(OC)CCN(C(=O)CC(O)CN(C)C)C1 C(=O)(CC(C(C)C)NC(C1CCCCN1CC)=O)NC(c1ncc[nH]1)CC N1(C(CP(C)(C)=O)=O)CCCC2CN(C(=O)CC3CC4CC4C3)CC12 C(CNC(c1c(C)nn(CCO)c1C)=O)(C(C)C(C)C)NC(c1c(C)noc1)=O N#Cc1c(NC(c2n[nH]cc2NCc2c(Cl)cc(Cl)cc2Cl)=O)cc(F)cc1F c1(C(=O)NCC2(CNCc3cc(COC)no3)CC2(F)F)cc(F)ccc1C C1(NC(CC(C=C)CC)=O)CCC2(CC1)CN(C(=O)CCCS(C)(=O)=O)CCO2 C1(C(=O)NC(CN(C(c2cc(C(F)(F)F)on2)=O)CC)C)CC(=O)NC(=O)N1 c1(C(N(C2CCC(NC(CC(=C=C)C)=O)C2)C)=O)ccc(S(=O)(=O)NCC)cc1 C(Cc1ccoc1)(C(=O)OC)NC(C(C1CCC1)NC(C1(Cl)C(C(=O)OC)C1)=O)=O c1(OC(C)C)cccc(C(=O)NCC2CCC(NC(=O)CN(C)S(N)(=O)=O)C2)n1 c1(C(C(=O)NCCN(C(=O)CCn2c(C)csc2=O)CC)(F)F)ncccc1F C1(C(N2CCN(C(C=NOC)=O)C(c3ccccc3)C2)=O)CCc2ncsc2C1 N1(C(c2c(C(=O)OC)csc2)=O)CC(CNC(C2CN(C)CCO2)=O)C(C)C1 CCCC(C(=O)NC)NC(=O)CC1CCC(NC(C2CC2Cl)=O)C1 N1(C(CCOCC#C)=O)CCC(CC(N)=O)(NC(c2cnc(Cl)cc2Cl)=O)CC1 N1(C(C(C)NC(=O)NC)=O)CC2(CC(NC(=O)CCC(=O)NC)c3nccn32)C1 C#Cc1ccc(C(N2CCCCC2CN(C)C(C2(F)CCOCC2)=O)=O)c(F)c1 N1(CC(=O)NCC2(c3ccsc3)CC2)CCCCC1C(=O)O C1(NC(C(C)Oc2ccccc2Cl)=O)CCCCN(C(=O)CC2(O)CC2)C1 CC1CN(C(C2CC(O)CN2C(N)=O)=O)CC1CCNC(=O)CCCC1CCC1 C1(COC)CN(C(C23CCCC2CCC3)=O)CCN1C(C12CCC(CO)(CC1)C2)=O n1(CC(N2CC(OC)C23CCC3)=O)c(C)nc2cc(F)c(F)cc12 C(=O)(C(C(C)CC)N1CCC(=C)CC1)NCCCC c1(CC)ccccc1-n1cc(C(C)N(C)C(c2csnc2Cl)=O)nn1 c1(Sc2nnc(SCC(C34OC(C)(C)C(C3)C4)C#N)o2)nc2ccccc2[nH]1 c1(C(=O)NC2CC(NC(c3ccc(C(C)=O)cc3)=O)C2)coc2cccc(O)c12 C1(C(N(C(C)CNC(=O)Cc2csnn2)C)=O)OCC2CCCC12 c1(C(=O)NC2(C)CCN(C(C3(O)CC3)=O)CC2)c(Br)ccc2ccccc12 c1(C(=O)NCC(=O)N(CCCNC(C(C)SCC)=O)C)ccc(Br)o1 c1(C(=O)NCC2C(CNC(CC3N(C)CCCC3)=O)C2)ncnc2ccsc12 c1(C(=O)OC)ncc(C(=O)NC2CCCC2NC(=O)C(C)C#N)s1 N1(C(CCCC#N)=O)CC2COCCC2(NC(C23CC(F)(C2)C3)=O)C1 c1(CC(=O)Oc2cc(C(=O)NC)c(C)cc2)cccc2ccncc12 N1(C(C2C(CC)C2)=O)CCC(C2CC2)(CNC(=O)C(c2ccccc2Cl)C)C1 c1(C(=O)NCC2N(C(C(CSC)(C)C)=O)CCC2)ccc(O)nc1Cl n1(CC)ncc(C(=O)N(C(C)CN(C)C(c2ccccn2)=O)C)c1Br c1(-c2cncc(C)c2)ccc2c(c1)COC21CN(Cc2ccc(Br)c(O)c2)C1 N1(C(C(n2c(C)ccn2)C)=O)CC(O)CC1C(=O)N(C1CC=CC1)C CCCCCCCCCC(=O)N(C)CC1CCN(C(c2cnn(C)c2F)=O)C1 C1(C(=O)NCC(CCNC(c2cc(C3(O)COC3)on2)=O)O)CC2C(C1)C2(F)F N1(S(CCC)(=O)=O)CCC2(CN(C(c3cc(O)ccc3O)=O)C2)C1 N1(C(C(C(CC)C)C)=O)CCOCC12COCCN(C(=O)CC1CC=CCC1)C2 C1(CNC(N(C)CC2CCCCC2)=O)CCCC1(C)C C1(O)(CN(C(=O)CCCNS(C)(=O)=O)C)CN(C(=O)CCc2cn[nH]c2)C1 C(CCC)(CCCNC(c1ncnc(OC)c1F)=O)NC(C1(C#C)CCC1)=O CC(C)CCCCC(=O)N(CC(=O)Nc1ccsc1C)CCO c1(CNC(C2C(C)C2)=O)ccc(S(N)(=O)=O)c(Cl)c1.C12CC1CNC2=O C(C(=O)N=c1ccn(C(C)CC)[nH]1)=C1CN(C(C2CC(CCC)C2)=O)C1 C12(CNC(C(C3CC3)OC)=O)CCCCC1N(C(C1CCSCC1)=O)CC2 C12(CC(=O)NCC3CCN(C(CCC4N(C)CCC4)=O)CC3)CCC(CC1)OC2 N1(C(CCN(C(CCC#CC)=O)CC2CC2)=O)CC(C)SC(C)C1 C(=O)(C(CC(C)(C)C)OC)N1C(C(=O)NCC(CCC=C)O)CC(=C)CC1 N1(C(C2CCN(CC)C2)=O)CC2(C)CN(C(C3CCCCC3(F)F)=O)CC2(C)C1 CC(=O)CC(C)(C)CC(=O)NCC1CCCCC1NC(C1CCCC(F)C1)=O c1(OCC(=O)NCCNC(c2c[nH]c3cccnc23)=O)ccc(F)cc1Cl N1(C(C#CC2(CC)COC2)=O)CC2CN(C(C3CCS3(=O)=O)=O)CC(C1)O2 C1(CNC(=O)Cc2cccnc2)CCN(Cc2ncccc2Br)CC1(F)F C(c1ccc(Cl)cc1F)=CC(=O)NCCCOCCNC(C1CC2CCC2C1)=O c1(C(=O)NCCN(C(=O)C=CC(F)(F)F)CC)cnnc(O)c1 c1(C(N2CCCC3(NC(C4CCC(C)C4)=O)C(C2)C3)=O)cccc(P(C)(C)=O)c1 CN1CCN(Cc2ccc(OC(F)F)cc2)CC1.C12CCCCC1NC(=O)CC2 Cc1ccc(CC(C)C(=O)N2CC(C)(NC(=O)CNC3CCS(=O)(=O)C3)C2)cc1 Cc1cc(O)nc(C)c1C(N1CC2CN(C(=O)CCNC(N)=O)CC2C1)=O C(CCCCCCCCN1CCCCC(N)C1)N(C)C c1(NC(C)(CNC(=O)C=CCF)Cn2cccn2)ncnc2cc(Br)ccc12 N1(C(=O)Cc2cc(O)nc(O)n2)CC2CN(C(=O)C(F)n3cccn3)CC2C1 O=S(=O)(c1cccc(=NCC2CCC23CCOCC3)[nH]1)NC1CCCSCC1 C1(Cc2csc(CC)n2)CCCC1N=c1[nH]c(N(C)CC)nc(=NC)[nH]1 C1(C(=O)NCC2CC2C2CC2)(COC)C=CCN1C(C1CCC(=O)NC1)=O c1(C(=O)NC2CC(=O)N(C3CCC3)C2)ccc(Br)nc1Cl CC1(C)CC(C(=O)NC2CCCSC2)CN(C(c2cc[nH]n2)=O)C1 CCC(C)(C)C(O)C(=O)N1CCOCC1CCNC(=O)C(C)(C)c1cscn1 C1(NC(=O)C(F)C(F)(F)F)CN(c2ccc3nnnn3n2)CCC12CCC2 Cc1[nH]c2ccccc2c1CC(N1CCC(C)(C(=O)NCCC(C)(C)O)C1)=O NS(=O)(=O)CCC(=O)NCc1cc(O)nc(CNC(C2C3CCC(=O)C23)=O)n1 c1(C(=O)NC(CC(=O)N(CC)Cc2ncc[nH]2)COC)ccc(C)c(F)c1 C(=O)(CCCCC(C)C)NCC1(CNC(c2ccc(CNC(C)=O)s2)=O)CCC1 C(C#CC(=O)NOCC)NC(CCCC)=O c1(C(N2CC(CN(C(CCCOCC)=O)C)C2)=O)sc2nc(C)nc(N)c2c1C c1(OC)ncccc1NC(=O)CCC1CCCN(C(=O)C(O)CC2CCCC2)C1 c1(NCc2cc(OC)c(OC)c(O)c2)ccc(S(=O)(=O)C(C)C#N)cc1 N1(C(CC(CCC)NC(=O)C=Cc2cnccn2)=O)CCOCC(C)(F)C1 c1(NC(N(CCCC)CC(C)OC)=O)nc2ccc(S(C)(=O)=O)cc2s1 c1(C(N2C(C(C)NC(c3ccc(C)cc3)=O)CCC2)=O)cc2occc2s1 c1(OC)cnc(C(=O)NC2C=CCN(C(c3csc(C4CC4)n3)=O)C2)cn1 Cc1nc(=NC(=O)N2CCC3(CCN(C)C3)C2)n(-c2ccc(F)c(F)c2)[nH]1 c1(-n2c(C3ON=C(C(C)C)C3)nc(CCCO)n2)ccc2c(cnn2C2CC2)c1 C1(C(=O)NC(COC(C)C)C(=O)NCCC2CC(C)(C)C2)CCCC(=O)N1 c1(C(=O)NC2(c3ccccc3)CC(CNC(COC)=O)C2)cc(C)c(Br)cc1C CC(C)C(C#N)C(=O)N1CCCCC1CCc1cn(CC(N)=O)nn1 c1(CC)ccc(Cn2ccnc2CNC(=O)C=CCCC(C)C)cc1 N1(C(=O)NCCc2c(F)ccc(OC)c2)CCC2CCN(C)CC12 C1(NC(COCCOC)=O)CN(C(c2cccc(Cl)c2C)=O)CC2CC12 c1(C(=O)NC2CCN(C(C3(CC#C)CC3)=O)CC2CO)ccn2cnnc2c1 C(=O)(C1Cc2ccc(F)cc21)NCCN(C1CCCC1)C(c1c(C)cno1)=O CCCC(C)CC(=O)N1CCOCC1(C)c1cn(CCSc2cnn(C)c2)nn1 Cn1ncc2c(CNC(c3cnn(C4C(CN)CC4O)c3)=O)ccnc12 C(CC(=O)N1CC(n2cc(CCCS(N)(=O)=O)nn2)CO1)SC(C)(C)C c1(C(C)NC(C2CC(NCc3ccn(C)c(=O)c3)C2)=O)cccc2ncoc12 C12(N(C)C)CCC1CN(C(C1COCCN(C(c3ccc(F)c(Br)c3)=O)C1)=O)C2 N1(C(CSCC=C)=O)CCN(C)CC1C(=O)N(C)Cc1ncc[nH]1 c1(OC)ccc(C(=O)NC2CCCCC2NC(=O)COCC2CCCCC2)cn1 C1(C2CCN(C)CC2)(C(=O)NCC2C(NC(c3ccc(OC)nn3)=O)C2)CC1 C1(c2c(OC)cccc2)CN(C(=O)CC2COC(=O)C2)CCN1C(C)=O C12(CNC(c3c(OC)nsc3)=O)CCCCC1N(C(c1cc(CO)on1)=O)CC2 c1(NC(CC2C(CNC(Cc3c(C)ncs3)=O)C2)=O)cc(OC(C)C)cc(F)c1 c1(C(N2CC(CNC(CC3CC(OCC)C3)=O)C2)=O)c(C)nn(C2CCC2)c1C CC1(CNC(c2c(Br)noc2C2CC2)=O)CCC(NC(C2CC2F)=O)CC1 c1(C(N2CC(NC(C3(COC)CCCC3)=O)C(OC)C2)=O)cc(OC)ncc1F N1(C(C=C(C)c2ccco2)=O)CCN(C(c2csc(=N)[nH]2)=O)C(C(C)(C)C)C1 c1(C(C)C)nocc1C(=O)N(CC(C)O)CCNC(=O)CCNC(=O)C(C)(C)C C(C(C)(C)C)OCC(=O)NCC1(CN(C)C(C2CC2F)=O)CC1 Cc1cc(C(=O)N(CCCCCC(=O)NCCC2CC(C)(C)CO2)C)cnc1C c1(N(C)CC2CCN(C(=O)CCc3cscn3)C2)cnn2c1CCCC2 N1(C(COC(CC)C)=O)CCCCCC1C(=O)NCc1c(C)nn(C)c1C C(=O)(C1=C(C)OCCS1)NC(C(=O)NC1CN(CC)CC1C)CN=[N+]=[N-] N1(C(CC(C=C)C)=O)CCC(C2CC(NC(=O)CCc3ccnc(C)n3)C2)CC1 C1(NC(=O)C=CC2CCOCC2)CCC12CCCN(C(c1coc(CO)c1)=O)C2 c1(OC)cncnc1C(=O)NCC1(NC(=O)C(C)c2ccco2)CC1 CC1CCC(C)(C)CN1C(=O)C(C1(O)CCC1)NC(=O)CC1CC2CC2C1 c1(CC)ncccc1NC(C1CC(O)CN1C(c1cc(Cl)cn1C)=O)=O c1(NC(=O)Nc2n(C(C)C)cnc2)ccc(C(F)(F)F)cc1N C1(CCCC)CN(C(C2CC2C)=O)CCN1C(=O)COCCc1cccc(F)c1 c1(C(N(C)CC2CCCN(C(C(CC=C)(F)F)=O)C2)=O)ncnc2c1CCC2 Cc1ccc(N)cc1C(N1CCN(C(c2ccc(=O)n(C)c2)=O)C(C2CC2)C1)=O CCCC(C(=O)OC)NC(=O)CC1CCCN1C(c1ccc(COC)cc1)=O N1(C(C(C)N(C)Cc2ccccc2)=O)CCC2(CCN(C(=O)CC(F)(F)F)C2)C1 c1(CC)nc(C)n(C)c1C(=O)NCC1CC(OC)CN1C(c1cc(CC)[nH]n1)=O CC1CC(CNC(=O)C(c2cccc(O)c2)C)CCN1C(=O)CCC1CCOC1 C(=O)(C1Cc2ccccc21)N(CC(C)CNC(=O)Cn1cnnc1)C CC1(C)C(=O)CC1C(N1CC(O)CC1C(=O)NCCOC(=N)O)=O N1(C(C2N(CC)CC2)=O)CCCCC1CCC1CCCN1C(=O)CC1(C)CC1 C1(NC(c2c(C)nn(C)c2Cl)=O)CN(C(c2ccn(C)c2)=O)CC2CCCC12 c1(CNC(CC2CCN(C(c3cc(C)[nH]c3)=O)C2)=O)n[nH]c2c1CCC2 c1(OCC(N2C(CNC(c3c[nH]cc3C3CC3)=O)CC2)=O)ncnc2[nH]cnc12 CCC(CC(=O)N(CC(C)CNC(c1cccn1C)=O)C)C(C)C c1(C(CNC(C2(C)CC(C)C2)=O)NC(C(CC)NC(N)=O)=O)ccccc1F N1(C(c2c(C)coc2C)=O)CC(C)(C)CC1CC(=O)NC(c1c(C)n[nH]c1C)C N1(C(C(CC)n2cccn2)=O)CCC(C2CCCN(C(=O)CCCF)C2)CC1 Cc1cc(CNC(C23CC(NCc4ccc(C)o4)(C2)C3)=O)cc(C)c1 c1(C(=O)NCCCCCN(C(C2(OCC)CCC2)=O)C)cc(C)nnc1O Cc1ccc(C)c(CN2CCC(n3cc(CC45CCCC4(C(=O)O)C5)nn3)CC2)c1N c1(C(N2CCC(C(C)NC(=O)Cc3cocn3)C2)=O)cnccc1Cl C12(C(=O)NCc3ccc(NC)nc3)C(NC(=O)CSCC(C)C)C3CC1C2C3 N(C(=NCCc1c(Cl)cccc1Cl)NCC(F)F)C(COC)C1CC1 CCCCC(F)(F)C(=O)NCC(F)CNC(=O)CCNC(=O)CO C1(NC(C2(C)CC2(F)F)=O)CCC2(CC1)CN(C(=O)CCc1n[nH]c(=N)s1)C2 C1(OC)CC(CC(N2CCC(=CCNC(c3cccnc3Cl)=O)C2)=O)C1(C)C c1(C2N(C(C(=C)C(C)C)=O)CCC2)ccc(F)cc1OC c1(COCCCN(S(C)(=O)=O)C)cn(CCC(=O)Nc2c[nH]c(C(=O)O)c2)nn1 N1(c2c(OC)c(Cl)ncn2)CCC2(CCC(NC(C3(C4CC4)CCC3)=O)CC2)C1 c1(C(=O)NCCN(C(C(C)OCCC)=O)CC2CC2)cc(=O)n(C)cc1Br c1(-c2c(C(=O)NC3C(CNC(Cc4ccn(C)n4)=O)C3)cno2)cccc(N)n1 CCC(CNC(C1CC1C1CCCCO1)=O)(CC)NC(c1ccc(CSC)o1)=O CC(C)CC(C(=O)NCC1(C(C)C)CC1)N(C)C.C12CCC(O1)CNC(=O)C2 c1(-n2c(C3CC34CC4)nc(CCn3nccc3)n2)cc(C(F)(F)F)ccc1F n1(CC(CC(=O)OC)C)c(-c2cccc(SC)c2)csc1=Nc1ccnc(Cl)c1 C1(c2cn(Cc3cnc(C)o3)nn2)CCN(C(=O)CC2C=NN(C)C2=O)CC1 Cc1ccc(C(=O)NCCC2(NC(C3CCC(C)S3)=O)CCOCC2)c(F)c1 c1(C(C(=O)NCC(CNC(C2CCC=CCC2)=O)CO)(F)F)cc(F)ccc1F N1(C(C2(F)CCOC2)=O)CCC2(CC1)CC(N(CCO)Cc1ccccn1)CO2 C1(NC(c2ccc(OCC)c(Cl)c2)=O)C2CCN(C(=O)CCC(C)=O)CCC12 C12COCCN(C1)C(=O)OC2=O.N1(CC)CCOCC1CC(=O)NC(C)(C)C Cc1ccc(F)cc1C(F)(F)C(=O)NCC1CCN(C(c2cnc(S)nc2)=O)CC1 CC(C)CC(C(=O)NC(C)C(C)(C)C(=O)N1CC2CC2(CO)C1)C(N)=O c1(C(C)C)ncc(C(=O)NC2(CNC(=O)C(C)(C)C3CC3)CCCC2)n1C N1(C(CCC)=O)CCCC(C(N2CC(OC)C(NC(C3CCCCO3)=O)C2)=O)C1 C(=O)(C1COc2c(C)cccc21)NC(CN(C(Cc1ccc(C)nc1)=O)C)C c1(C(=O)NC(CNC(C=CC=CC)=O)CC(F)(F)F)cc(S(N)(=O)=O)co1 c1(C(=O)NC(CCNC(c2cc(C(C)=O)oc2C)=O)C)cc2c(cn1)CCCC2 c1(NC(C(N(C)C(C2CCCSC2)=O)C2CC2)=O)ccc2ccoc2c1 N1(C(C=NOC)=O)CC(OC)CC(NC(C2(C)CCCC2OC)=O)C1 c1(C(=O)NCC(C2CCCC2)NC(c2scc(OC)c2)=O)cncc2[nH]ccc12 N1(C(Cn2ccc(C)n2)=O)CCCN(C(=O)C(N2CCC(O)CC2)C)C(C)C1 C(=O)(C1=NOC(C)(C)C1)NCC(C(C)C)NC(C1CCC(C)C1)=O N1(C(C(C(C)C)O)=O)CC2CC(NC(=O)CC3CCC(C)C(C)C3)CC1C2 c1(CCCC(=O)Nc2cn(C)c(C(N3CCOC4CC34)=O)c2)ccc(Cl)cc1Cl c1(C(=O)NC2C3(CN(C(C4C(CC)OCC4)=O)C3)CC2)cnc2ccccc2n1 N1(C(CC(=O)NCC)=O)CCN(C(=O)C(S(C)(=O)=O)C2CC2)CC1C(C)C c1(C(=O)NC2CC(C)(NC(c3nc(C#C)sc3)=O)C2)ccc([N+](=O)[O-])c(Cl)c1 O=C(C1CCCc2ccnn21)NCC1CC2(CC2)CN1C(=O)C1=C(Cl)CC1 C1(NCc2n(C)ccn2)CC(F)CN(C(=O)OCc2cccc(C(C)(C)C)c2)C1 C1(C(=O)NCC2(NC(C3CCCNC3=O)=O)C(C)CCCC2)CC2CCC1CC2 n1(CC)cnc(C(=O)NCCCCNC(=O)C(C)C2CCOC2)n1 N1(C(C(CC)C#N)=O)CCCCC(NC(=O)CNC(c2csc(Br)c2)=O)C1 C1(C(N2C(C(C)NC(c3c(C)n[nH]c3)=O)CCC2)=O)CCCN(S(N)(=O)=O)C1 C1(C)(C(=O)NCC(C)NC(C2(C)CCC23CCC3)=O)CCN(C(=O)OC(C)(C)C)C1 CCC(CCC(=O)N1CC(C)C1(C)C)NC(=O)C(COC)OC S(=O)(=O)(C1CCOCC1)N(C1CCNCC12CC2)C(C(COC)N(C)C)=O c1(C(=O)NCC(=C)CCNC(=O)C(c2ccccc2)C)c(C)nn2c1CCCC2 c1(C(=O)NCCOCCNC(c2cc(C)on2)=O)nn(C)c2c1CSCC2 C(=O)(CC(C)(C)CC(F)F)NCC(CNCc1cn(CC(CC)O)nn1)C(C)C c1(C(N2CC(C(=O)NCC(C)(C)SC)(COC)C2)=O)cc(C)c(C)[nH]1 N1(CC)CCCN(C(=O)C(CNC(=O)CSc2nc[nH]n2)OCC)CC1=O C1(CN(C(Cn2c(C)ccn2)=O)C)CN(C(=O)CC(C)C2CCCC2)CCO1 N1(C(C(C)=CC(C)(C)C)=O)CCC(C(=O)NC2CCCC3(CCC3)C2)C12CCC2 C1(NC(C(C)NC(=O)NC)=O)CCCCC1NC(c1occc1C)=O C1(CNC(C=C(C)C)=O)CCN(C(=O)CC2CSC2)CC1C c1(N(C)C)nc2cccc(C(=O)NCCCCn3ccnc3)c2o1 C1(C(=O)NC(CCOC)CNC(=O)CN2CC(C)(C)C2)CSCC(=O)N1 C(=O)(C#CC1CCCCC1)N1CC(C(NOCCOC)=O)N(C)CC1 N1(C(CCc2c(C)cccc2)=O)CCCN(C(=O)CC#N)C(c2ccccc2)C1 C1(CN(C(C(COCC)O)=O)CC)CCN(C(=O)C2=CCSC2)CC1 C1(C(=O)Nc2ccsn2)C=CCN(C(=O)COC2CCCOC2)C1 c1(CC)cccc(C(N2CCCC(CNC(=O)C(C)c3ncco3)C2)=O)c1 c1(CN(C(CCN(C(C=CC(CC)C)=O)CC)=O)C)nc(C)ns1 c1(CNC(c2ccn(CC)n2)c2nnnn2CCC2(C)CC2)scc(C)c1C C1(C(=O)NCC2(CN(C(=O)CC3(O)CCOCC3)C)CC2)CCC2(CCC2)CC1 C1(C(N(CCOCCOC)C)=O)CN(C(C2CCCC3CC23)=O)CC1(C)C c1(C(N(C2CCCC(NC(=O)C(C)(C)C3CCC3)C2)C)=O)cnn2c1CCC2 CS(=O)(=O)C=CC(=O)N1CCCCC(CNC(=O)C2=CCC2)C1 C1(CC(=O)N(CCCC)CCCO)CC(F)CN1C(C12CSCC1C2)=O c1(C(=O)NCC2(OCC)CN(C(=O)C(C3CC3)OC)C2)cc(C)c(Cl)s1 S(=O)(=O)(c1cc(Br)c(F)cc1Cl)NC(c1cc(Cl)cs1)=O c1(C(N2CCC(CC=C)(NC(=O)C(O)C=CC)C2)=O)cc(N)c(Cl)c(O)c1 c1(N(C)CC2N(C(C3(OC)CCCOC3)=O)CCC2)ncc(Br)cc1C#N c1(C(=O)NC2CC(F)(CNC(c3cc(C)c(O)cc3)=O)C2)cnc2c[nH]nc2c1 c1(CCN(C)C)cn(CC(F)CCNC(c2cnn(CC(F)F)c2)=O)nn1 C#Cc1cccc(C(=O)NC2CC2NC(C2CCCCC(F)(F)C2)=O)c1Cl c1(C(=O)NC(CCCNC(C(C)(C2CC2)OC)=O)(C)C)cnc2sccn12 C1(C(=O)NCCN(C(C(C)Sc2nncn2C)=O)C)CS(=O)(=O)CC12CC2 c1(C(=O)NC2CC(NC(c3ccc(C)nc3O)=O)C2)ccn2ncnc2c1 C(=O)(C(C)(CO)NC(=O)COc1ccccn1)N(C)CC1(O)CCC1 C1(C(N2CC(CN(C(c3c(C)nc(CCC)s3)=O)C)C2)=O)COC2COCC12 CC(C)(CNC(c1ccoc1C1CC1)=O)CC(=O)NCCCCF CC1CC=C(C(=O)NC2COCCN(C(c3cc(CN(C)C)c[nH]3)=O)C2)CC1 C1(OC)CC(NC(c2cc(C)cc(Cl)c2)=O)CN(C(=O)CCc2ccncc2)C1 CC1CC(=O)NC1C(=O)NCC1(C)CC(NC(c2[nH]ncc2C#N)=O)C1 N1(C(CNC=O)=O)CCCC(CCNC(c2coc(C(F)F)c2)=O)C1 C(=O)(CC(C)(C)C)NC1CCCC(CN(C(CCc2onc(C(C)C)n2)=O)C)C1 c1(C(=O)NCC2(C)N(C(c3cnc(C(C)O)s3)=O)CCC2)c(F)ccc(N)c1F C1(C(=O)NCC(=O)NCCC)CCN(C(C2CCC2OC)=O)C12CCC2 C1(COC)CN(C(c2cccc(F)c2Cl)=O)CCN1C(c1cscc1Cl)=O C(CCCCC(=O)NCC(C)CNC(C1(S(N)(=O)=O)CC1)=O)OCC C12(C(N3CCC(OCC(N4CC(C)(OCC)C4)=O)C3)=O)CCC(OC)C1C2 c1(C(=O)NC2CC2)cc(N2CC(C)(OC)C2)nc(C)c1.C(=O)(C(=O)NC)NCCOC C1(NC(COCCOC)=O)CN(C(=O)CCN2CCNC(=O)C2)CC1C1CC1 N1(C(C2N(C(C3C(C(C)(C)C)CC3)=O)CC=CC2)=O)CCC2(CC1)CC2CO C1(CNC(Cc2cc(C)no2)=O)CCN(C(c2cn(C)nc2Br)=O)CC1C c1(CC(C(=O)NCC(C)C#N)NC(C2CC(C)(O)C2)=O)cnn(C)c1O C1(N(C(C2(CCNC(C(C)CC3CC3)=O)CC2)=O)C2CC2)CCOCC1C N1(C(CC2CCN(C)C2)=O)CCC2CN(C(=O)C(N)=O)CC2C1 C1(NC(c2ccoc2Cl)=O)C2CN(C(C3CC(CCO)C3)=O)CC12 C1(C(N2C(CS(C)(=O)=O)CC2)=O)CN(CC2CCC2)CCO1 N1(C(c2c(OC)cncc2)=O)CCC2CCC(NC(=O)C(F)C(C)(F)F)C1C2 CC1(C)C(NC(=O)CN2CCC(F)CC2)CC1C(=O)Nc1ccc(CCF)cc1 C1(C(=O)NCCCN(CCCN2CCCCCC2=O)C)CC2(CCC2)CCO1 c12cc3c(cc1CNC(=O)C(=O)N2)OCCO3.N1(S(C)(=O)=O)CCOC(O)C1 N1(C(c2[nH]c(=NCC)sc2)=O)CC2CN(C(=O)C(CO)NC(N)=O)CC2C1 N1(C(COC(CC)C)=O)CC2CC(NC(c3sc(C4CC4)nc3C)=O)CC1C2 C1(C(N(CC(CNC(CCNC(CC(C)C)=O)=O)C)C)=O)Cc2nnsc2S1 n1(CC)nc(C)c(CC(N2CCC(O)(C(C)NC(c3cnc[nH]3)=O)CC2)=O)c1C c1(CNC(C2(CC)CCN(C(c3coc(C(N)=O)c3)=O)C2)=O)c(C)nn(C)c1C c1(C(=O)NCC(CC)NC(c2cnn(C)c2Cl)=O)c(C)sc2ccc(F)cc12 C1(NC(c2ncnc(C)c2C)=O)CN(C(C2CCC2)=O)C2(CCCOC2)C1 N1(CC(=O)NCCCCCCNC(C2CCN(C)C2)=O)CCCCC(O)C1=O Cn1c(=O)c2c(Nn3ccc(NC(=O)OC(C)(C)C)cc3=O)ccnc2n(C)c1=O c1(C(=O)NCCCC(C)(C)NC(C(C)SC(C)C)=O)ccc(=N)[nH]c1Cl c1(C(c2ccc(F)cc2)C#N)cccc2c1N(C(C1CCCO1)=O)CCC2 c1(NC(=O)NC2CC(=O)N(C)C2c2nccn2C)c(C#N)sc2ncccc12 C1(CC)(CC)CC(NC(=O)CCSCC(N)=O)CN1C(=O)C(CC)C(C)C N1(C(C(C(C)C)OC)=O)CCC2(CC1)CN(C(=O)CCCCCSC)C2C(C)C CC#CCCCC(=O)NCC1(CNC(=O)C(C)Oc2cc(F)cc(F)c2)CCC1 C(CN=C(NCCOc1ccc(Cl)c(F)c1)NCC1CCN(C)C1C)OC Cc1nc2c(s1)C(N(C)C(C1CCCC(F)(F)CN1)=O)CCC2 c1(C(=O)NC2C=CCN(C(CCC(C)SC)=O)C2)cc(N)c(Cl)cc1C C1(CNC(=O)CCNC(C2CSC2)=O)CCCCN1C(=O)C=Cc1ccco1 c1(C(=O)NCC23C(CN(C(CCC45CC(C)(C4)C5)=O)C2)C3)cc[nH]c2nccc1-2 c1(C(=O)NC2CCC(F)(CNC(=O)C(F)CC3CC3)C2)ccc2c(c1)OCCO2 C1(NC(CSC)=O)CCCCC12CCN(C(=O)C(Cl)=CCl)C2 c1(C(=O)NCC(C2CCCCC2)NC(CCOC)=O)n[nH]c2ccc(Br)cc12 c1(C(=O)NCC(C)(CNC(=O)C(C)Cn2ccnc2)OC)c(C)ccnc1O c1(C(=O)NC(C(CO)NC(CCCOC(C(C)C)=O)=O)C)cnnc(C2CC2)c1 C#CC1(C(=O)Nc2ccc(O)c(CO)c2)CCN(C(=O)C(C)N(C)C)C1 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NCC1CCN(C(c2c(C)con2)=O)C1 c1(C(=O)NC2CC(N(C(C(C3CC3)SC)=O)C)C2)ccc2nccn2c1 c1(C(=O)NCC(CO)NC(C(CCC)F)=O)ccc(O)c(OC)c1 C(=O)(CCCCC(F)F)NCC1N(C(CCC(=C)Cl)=O)CCC1C Cc1c(C(=O)NC2CN(C(=O)C=Cc3cocn3)CC2C)cc(F)cc1Br C1(C)(CNC(C2(Cl)C(C(C)=O)C2)=O)CCC(NC(=O)Cc2cc(C)sc2C)CC1 c1(C(=O)NC2CC3N(C2)C3)cnc2ncccn12.C1(CC(=O)OC)CC=CCC1 C1(NC(C2(CC)CC2)=O)C=CC(CC(=O)NC(C2CCOC2)CO)C1 C(=O)(C1CNC(=O)c2ccnn21)NCCN(C(c1cc(C)c(C)[nH]1)=O)C c1(SC)ccc(C(C(=O)NCCSC)N(C2CC(OC)C2(C)C)C)c(C)c1 c1(C(=O)NCC2C(C(=O)NCCCc3cc(C)no3)CCC2)ncncc1C c1(C(=O)NC2CN(C(CC3(OC)CCC3)=O)C3C2C3)cc2c(C)ccc(F)c2[nH]1 Cc1n[nH]cc1C(c1cn[nH]c1)NCc1nnnn1C1CCOC1 C1(CC=C)CCCN(C(=O)CCCC2(NC(C3(F)CC=CCC3)=O)CCC2)C1 O=C(CS(=O)(=O)CCCc1ccccc1)NC1C(C2CC2)C1(F)F C1(NC(C2(SC)CC2)=O)CC1C1CCN(C(c2cccc([N+](=O)[O-])c2)=O)CC1 c1(CN2CCN(C(C3CCC(C)CC3)=O)CC2)c(Cl)ccnc1Br N1(C(c2nccnc2Br)=O)Cc2[nH]nc(-c3cccc(F)c3O)c2C1 Cc1ccc(Br)c(F)c1C(=O)NC1CN(C(=O)C(C)(F)F)CC2(CC2)C1 C1(CC)(CO)CCCN(C(=O)C(C)(C)CNC(=O)C(CO)N(C)C)C1 C1(C(=O)OCC(C)C)CCSC(C)C(=O)N1.CCCC(C)=CC(=O)OC(C)C CCCC(CC)CCC(=O)NC1CN(C(c2ccc(F)c(F)c2N)=O)CC1CC c1(C(=O)NCC=CCNC(C2CN(CC)C2)=O)ccc(O)c(F)c1 c1(C(=O)NC2(C)CC(NC(c3cc(CCC)[nH]n3)=O)C2)ccc(C)c(C)c1N N1(C(c2c(C)cco2)=O)CCC(NC(c2cc(=N)[nH]c(=N)[nH]2)=O)CC1C c1(N2C(=O)CC(C(=O)NC(C#C)C)C2)cccc(Cl)c1Cl Cc1nc(C)c(F)c(=NCC2CC(NC(=O)C(c3ccc(F)c(F)c3)O)C2)[nH]1 C(=O)(CCCCCN=[N+]=[N-])N(C(C(=O)NC(CC(=C)C)CO)CC(F)F)C c1(C(N2CC(N=[N+]=[N-])C(O)C2)=O)ccc2c(n1)CN(C(=O)CC1OCCO1)CC2 C(=O)(C(C(CC)C(C)C)N(C1CSC1)C)NC(C(=O)OC)CC(C)C C1(CNC(=O)COC2CC2)CC2CC(C1)N(C(c1ccc(CC3CC3)cc1)=O)C2 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)NCCN(C(CN(CC)CC)=O)C(C)C c1(OC)cccc(OC)c1C(N1CCCC(NC(c2cc(C(N)=O)[nH]n2)=O)C1)=O N1(C(CCc2nc(C)sc2)=O)CCC(NC(c2cc(CF)on2)=O)C(CO)CC1 Cc1cc(N2CC3CN(C(=O)CC4OCCC4C)CC3C2)c(C#N)cc1[N+](=O)[O-] Clc1cnc(CCNC(c2cnc(-c3cccs3)[nH]2)c2nnnn2CC(F)F)s1 CCC(O)C(=O)NCCn1cc(C(=O)NCC(c2ccccn2)C)nn1 C(C1CN(C(c2c(C#N)ncn2C)=O)CC1C(N1CC=CCC1)=O)=CC c1(C(N2CCCCC(CNC(c3c(C)scn3)=O)C2)=O)csc2c1CCCC2 CS(=O)c1cccc(NC(=O)NC2(c3ccncc3)CC2)c1 c1(C(C2CC2)OC(C)(C)C)nc(-c2cccc(Cl)c2)nn1C1CSC1 Cn1cc([N+](=O)[O-])c(C(=O)NC2CCC(F)(CNC(=O)C(F)CC3CCC3)C2)n1 N1(C(CC2C(C)(C)OCC2)=O)CC(NC(c2cscc2Cl)=O)CC1(C)C N1(CC)CCC(NC(c2cc3c(Cl)cncc3o2)=O)CC(C)(C)C1 Cc1ccc(CC(=O)NCCC2(C(=O)NC3CCCSC3)CCC2)o1 C1(CNC(CCC)=O)(OCC)CN(C(=O)CNS(=O)(=O)NC)C1 N12CCC(C)N(CC1)C(=O)c1cc(N)ccc1C2=O.C1(NC)CNC(=O)C1 c1(C(=O)NCCN(C(CC2CCCC(OC)C2)=O)C)cc(C)cc(O)c1 CCC(CCN)C(=O)NCC(c1cnc[nH]1)C c1(C2(CNC(C(C)(C)C)c3cncs3)CCC2)cc(F)c(F)cc1 C1(NC(C(CNC(c2cc(COC)[nH]n2)=O)N(C)C)=O)CCCC(OC)C1 c1(NC(c2noc(Cc3ccc(F)cc3)n2)=O)cccc2nc(O)ccc12 N1(C(c2c(C)nc(CC)s2)=O)CCCC2(CCN(C(=O)C(F)CC(C)C)C2)C1 c1(C(N2CCC(NC(c3cccc4cncn34)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl c1(C(=O)NCC2C(CNC(C=CCOC)=O)C2)c(C)nsc1Br c1(OCC)ncccc1NC(=O)C(C)(C1CC1)N(C(=O)C(C)NC(=O)CC)C CCCC(C)(O)C(=O)NCc1cc(O)nc(CNC(=O)CC2CC23CC3)n1 c1(C(N2CCC(C3(NC(C(C=C)O)=O)CC3)C2)=O)cccc2cc(O)ccc12 C(=O)(C(C)(O)CC(C)C)N1CC(C2CN(C(C(C=C)OC)=O)C2)OCC1 CC1(C(N2CCC(CNC(c3ccc(-c4ccccc4)o3)=O)C2)=O)CC=CCC1 N1(C)CCCC1C1CCCCN1C(=O)NCC1CC(OCC=C)C1.C(C)(C)(C)ON c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC(C)CN(C)C(C1(F)CCCOC1)=O c1(C(=O)NCC(CN(C(C(C(C)C)C)=O)C)O)c(F)cc(O)cc1F C(=O)(CCCC(=O)N1CCC(CNC(c2cn[nH]c2)=O)C1(C)C)OC Nc1cc2c(cc1C(=O)NCCN(C(=O)CCF)Cc1ccccc1)CCC2 C(=O)(C1=CCS(=O)(=O)C1)NCC1CC(CNC(CCS(N)(=O)=O)=O)C1 N#Cc1nc[nH]c1C(N1CCCC1C1CCN(C(=O)C(=C2CCCCC2)F)C1)=O c1(C(=O)NCCN(C(C(CC)OC2CCCC2)=O)C)ccc(Br)c(F)c1 Cc1c(C(=O)NCC2(NC(c3csc(Cl)n3)=O)CCCCC2)nn(C)c1N CC1(C)C2CC(C(=O)NC3CCC(NC(=O)C=Cc4ccc(C(F)F)o4)C3)CC12 c1(NC(N2CCC(Oc3ccc(F)cc3)CC2)=O)nc2ccc(F)cc2s1 c1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)CCC2)sc(=O)n(C)c1Cl c1(C(=O)NCCCNC(CN(C(COCCC)=O)C)=O)cccn2c(C)cnc12 C1(NC(COCCC)=O)(CO)CCN(C(=O)C(c2ccc(COC)cc2)C)CC1 C1(C)CCCCNC(=O)c2cc([nH]n2)C(=O)NCC(=O)N1.C(C(C)(C)C)OCC C1(CC(N2CC(NC(C3CCC4CC34)=O)C2)=O)CCCC2(CCC2)O1 c1(C(N2CC(C)(CC(N3CC(CC45CC(C4)C5)C3)=O)C2)=O)cccc2c[nH]nc12 c1(C(=O)NC2(C3N(C(C=CCC)=O)CCCC3)CC2)cc(COC)cc(F)c1 N1(C(c2nc(N)c(O)cc2)=O)CCC2(CCCC2NC(C23CCCC2C3)=O)C1 C(C)(C)(CCC(=O)NC1CCC1CNC(=O)CCCCc1ccccc1)OC C1(CNC(C(c2cncc(F)c2)C)=O)CN(C(=O)CC(C)(C)C#N)CCCO1 c1(OCC)cc(C(N2CC(CC(C)NC(C3CC3(C)C)=O)C2)=O)[nH]n1 CC12CN(C(C3CCCCO3)=O)CC1(C)CN(C(C1CC(n3ccnn3)C1)=O)C2 c1(C(N2C(CNC(c3c(OC)scc3)=O)CN(C)CC2)=O)sc([N+](=O)[O-])cc1Cl c1(CNC(c2ccc(NC(C3CCC(=O)NC3)=O)cc2)C)cc(Cl)ccc1Br c1(C(N2C3CC(NC(CCCC)=O)C(C)C2CC3)=O)cccc(S(=O)(=O)CC)c1 n1(CC(=O)N(CC(C)NC(=O)CC2CCCC2)C)ccnc1 N1(C(C2CCC(CNC(C=C(C)c3ccccc3)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(=O)Nc2ccccc2COc2ccccc2)CCN2C(CNS2(=O)=O)C1 C1(CC(=O)NCCc2c(CNC(=O)Cc3cccs3)nco2)COC2CC1C2 NC(=O)CCC(=O)N1CCN(C2CN(C(=O)CCC3CCCO3)C2)CC1 C(=O)(C(C(C)C)SCC)N(CCC)CCNC(=O)CC(C)C1CC1 C(=O)(C(C)(CO)NC(C)=O)NCCCN(C(=O)CCC1CCCCC1)CC CC(C)CS(=O)(=O)CCCN1CCC(NC(=O)Cn2cnnn2)CC1 S(=O)(=O)(CCC1CCc2ccccc21)N1CC(C#N)(CC)C1 c1(CC(=O)NC2CCN(C(C(C)OCCCC)=O)C(C)C2)noc2ccccc12 c1(NC(=O)OCCCSc2nncc(OC)c2)ccc2oc(=O)oc2c1 C1(CNC(C(CNC(c2cc(C)c(C)s2)=O)(C)C)=O)CC2CCCC2C1 C1(COC)CN(C(C2CC(O)C2)=O)CCN1C(=O)C(C)Nc1ccc(CO)cn1 c1(C(N2CCN(C(CCC=C)=O)C(C3CC3)C2)=O)ccc2c(c1)nc(O)n2C C(=O)(C1=Cc2cc(F)ccc2OC1)N(C1CN(C(c2ccc(C)n2C)=O)C1)C c1(N2CCC(c3nccc(OC)c3NCC3CC3CF)C2)ncc2n1CCCC2 Cc1nc(=NC2(CO)CCCN(C(c3ccnn3Cc3ccccc3)=O)C2)s[nH]1 C(=O)(C1=CCC(NC(=O)Cc2cccc(C#N)c2)C1)NC(C)CCCCO CC(CCC1CCCC1)N=c1[nH]n2cc(COCCCC#N)nc2s1 C1(CNC(C(CC)C)=O)CC2(C1)CN(C(=O)CC1(c3ccon3)CCC1)C2 c1(C(N2C(CNC(C(C)CC3CCCO3)=O)CC2)=O)cccc2nsnc12 N1(C(C2C(CC)CCCC2)=O)CC2CN(C(=O)Cc3cccc(C)c3)CC(C1)O2 C(CC(=O)NCCCN1CCCC1=O)(C(F)F)NC(C1(CCCC)CCC1)=O C1(NC(Cc2c(C)cccn2)=O)CN(C(=O)CCOC(C)CC(C)C)CC12CC2 Cc1cnc2cc(C(=O)NC3CN(C(=O)CCc4cccnc4)C3)nn2c1 CP(C)(=O)c1ccc(C(=O)NCC2CCCC2NC(C2CCCCCC2)=O)o1 C1(NC(C2N(C(CC)=O)CCCC2)=O)CCN(c2nnc(C#N)s2)CC1(C)C c1(C(N(CC(CN(C(c2c(C)ccc(C)n2)=O)C)O)C)=O)cccn2nnnc12 c1(C(N2CCN(C(C34CC(C)C3C4)=O)C(COC)C2)=O)ccc2c(c1)CNC2=O C1(C(=O)NCCN(C(c2c(SC)csc2)=O)Cc2ccccc2)CCN(C)C(=O)C1 C(=O)(C(C(C)(C)C)C1CCC1)N1CC(OC)C(NC(c2ncn(C(C)C)n2)=O)C1 C1(NC(CCCOC)=O)COCCN(C(=O)CC2CCCCCC2)C1 C=CC1CN(C(=O)C(=O)NCCOC)CC1NC(=O)Cc1csc(C)c1 c1(C(N2CC3C(NC(C4N(C(C)=O)CCOC4)=O)(C3)C2)=O)c(F)cncc1Br C1(NC(COCCCC)=O)CCCC1CNC(C1(OC)CCCC1)=O C1(C(=O)NC2(CNC(c3ccoc3C3CC3)=O)CC2)CCCCC1O c1(Cc2ccc(CNC3C(C(=O)NSC)C3)o2)nc(Cl)ccc1Cl CCC1=NOC(C(=O)NC2CCCCC2C(=O)N(C(C2CCC2)C)CC)C1 c1(N2CC(O)(CNC(C3CCC(N=[N+]=[N-])C3)=O)C2)nc(Cl)nc2sccc12 C1(C(N(C(CN(C(c2c(CC)ocn2)=O)C)C)C)=O)CNC(=O)CC1(C)C C(=O)(C1NCCc2c(C)cccc21)N1CCC(CO)=C(C)C1 c1(CCC(=O)NCCN(C(C(F)OC)=O)C(C)C)cc(F)cc(F)c1 Cc1cc(Cl)c(C(=O)NCC(C)N(C)C(c2cccc(C(=O)N(C)C)c2)=O)cc1C N1(C(c2nc(C(C)NC(=O)CC3CCCC3O)oc2)=O)CC2C(C1)C2(C)C C(=O)(CC(C)(C)CNC(=O)CS(=O)CC)NCCCOCC#C c1(OC)noc(C)c1C(=O)NCC(C)NC(C1CCCS1)=O C(=O)(CCCCC(F)F)N(CC(C)NC(CC(CC)C(C)C)=O)C c1(C(=O)NCCCOCCNC(=O)Cc2ccnnc2O)c(F)cc(F)cc1Cl C(=O)(CCCS(C)(=O)=O)N(CCCNC(c1nc(C)n(C)c1C)=O)C C1(NC(CNS(CCCC)(=O)=O)=O)CCN(C(=O)CC2CC(C)C2)CC1O C1(c2nnnn2C(C)(C)C)(Nc2cccc(OC)c2Br)CC2CC(OC)CC12 c1(NC(C2N(S(CCCC)(=O)=O)CC=C2)=O)cc(F)c(Br)cc1[N+](=O)[O-] C(C(CC(=O)N1CCC(OCCF)C1)NC(c1cc(C(C)=O)on1)=O)OC N1(C(c2cc(OC)nn2C)=O)CCC(NC(=O)CC(C)C(F)(F)F)C(F)(F)CC1 c1(SCC(=O)NCC2N(C(CCC=C)=O)CC(O)C2)ccc(C#N)cc1 Cc1cc(Cl)ccc1OCC(=O)NCC(CO)NC(c1csc([N+](=O)[O-])c1)=O N1(C(Cc2cnc(C)s2)=O)CC(NC(=O)C(C)Cc2cccnc2)C2CCCC12 c1(C(=O)NCC(O)CNc2ncc(I)cn2)cccc(O)n1 C12(NC(CCS(N)(=O)=O)=O)COCCC1CN(C(=O)C=Cc1ccoc1)C2 CCC(O)C(C)C(=O)N1CC(C(C)NC(=O)CCNc2ccccn2)C1 N1(C(c2c(C)ccnn2)=O)CCN(C(=O)CSC2CCS(=O)(=O)C2)CC1C C1(CNCC(C2(OC)CN(C(=O)OC(C)(C)C)C2)(F)F)CC2CC(=O)C1O2 C1(CCNC(c2c[nH]c(=N)s2)=O)CN(C(C2N(CC)CCC2)=O)CCO1 Cc1conc1N(C(=O)C(C)SC(F)(F)F)C(C(=O)OCC1CC1)=O c1(CNC(=O)NCCCOc2c(C)cc(Cl)cc2)cc(F)c(C(F)(F)F)cc1F c1(C2C(C(=O)NCC3(CN(C)C(C4(C)CC4(C)C)=O)CC3)C2)cccc(Br)c1 C1(CC(N2CCC(c3cn(CCC45CC(CO4)C5)nn3)C2)=O)CC2CCC1CC2 N1(CCC(=O)NC(CC)CNC(C2(CO)CC2(F)F)=O)CCC(C)CC1 Cc1ccc2cc(C(N3CC(CNC(=O)C(C)(C)CO)N4CCC3C4)=O)cn2c1 C1(CNC(C2(C(=O)NC)CCC2)=O)(OC)CCN(C(=O)C(C)CC2CC2)C1 N1(C(C(C)SC)=O)CC(C(=O)OC(C)(C)C)C(F)C1.C123CC(C1)(C2)NC3=O c1(C(=O)NCC2CC(F)(CNC(c3ccnn3C3CC3)=O)C2)ccc(Cl)cc1Cl c1(N(C)C)ncc(C(N2CCC(NC(=O)OC(C)(C)C)C2C(C)(C)C)=O)cn1 C(CC(C)(C)C(=O)N1CCC(CCCCNC(C2(C)CCC(C)C2)=O)CC1)OC C1(F)(C(=O)NC2CN(C(C(C)O)=O)CC2C(F)(F)F)C(C)(C)C1(C)C Cc1ccc2nc(C)c(C(=O)NC3CN(C(C4CC4CN(C)C)=O)C3)cc2c1 c1(OCC)ncc(F)c(N(C(c2ccccc2F)=O)CC2CCCN2)n1 N1(C(CNC=O)=O)CCCC2(CCCN2C(=O)CN2CC=CC2)C1 N1(C(c2c(C)cc(C)nc2)=O)CC(C2CCCCN(C(C3(C)CC(F)C3)=O)C2)C1 CC1=C(C(=O)N2CC(O)(CN(C)C(c3cc(C(C)C)no3)=O)C2)CCC(C)(C)C1 C1(C(N2CC3C(CC)(C3)C2)=O)CC(NC(=O)CCCOC(C)(C)C)C12CCC2 CC1(C(=O)NC2CC2NC(=O)CSCCN(C)C)CCc2ccccc2C1 c1(C(=O)N)cc(F)cnc1Cl.C1(COC)CCCN1C(=O)CC1CC(C)=NO1 C1(CC(NOCCC=C)=O)CCN(C(=O)C(c2cncnc2)C)CC1 Cc1nc(C(C)C)oc1C(=O)NCC(C1CCCC1)NC(C1(S(N)(=O)=O)CC1)=O N1(C(C(=O)NCC)=O)CC2CN(C(c3cc4cccnc4[nH]3)=O)CC(C1)O2 C1(CN(C(=O)CC2CC3(CC3)C2)C)COCCN1C(=O)CC1CSC1 N1(C(Cn2cccc(C)c2=O)=O)C2CCC1CN(C(C1CC=CC(O)C1)=O)CC2 C1(CC)C(C(=O)N(C(C)C(C)(C)C)C)CCCN1C(=O)C(N)=O C(=O)(C1CCNc2c(C)cccc21)N(CCNC(C(CCCCCC)CC)=O)C N1(C(C2CCN(C(CC(CCC)(C)O)=O)CC2O)=O)CCC2(COC(C)C2)C1 Cc1cc(F)cc(C)c1C(=O)NCCN(C(=O)CC1CCC(C)C1)CC1CC1 N1(C(c2c(OC)csc2)=O)CCC(NC(c2ccnn2C(C)(C)C)=O)C(CO)C1 C1(C(=O)NC(C2C(C(=O)OC)C2)C)C(C)CN1C(=O)C(O)CN(C)C c1(OCC(=O)NC(CN(C(C(CCC)OC)=O)CC)C)cccc(Cl)c1C c1(OCCCC)cc[nH]c(=NCCCN(C2CC23CCOC3)C)n1 Cc1ccc(Br)c(C(=O)NC2CCC2NC(=O)CC2C=NN(C)C2=O)c1N c1(C(=O)NCCCN(C(=O)C=C2CCC(C)CC2)CC)ccc(Br)nc1N C1(CC(=O)N(C)CC2CC2(F)F)C2CCCC2N1C(c1cc2occc2[nH]1)=O C1(NC(CC2CC(NC(COCC=C)=O)C2)=O)(CO)CC(C)CC(C)C1 CC1CC(NC(c2cn(-c3cnn(C)c3)cn2)=O)CN(C(=O)CCCC(F)F)C1 C12(CCC(=O)N1)C(=O)N(C)CCN(C)C2.C1(C(=O)OC(C)(C)C)CC1F c1(C(=O)NCCN(C(c2sc(C#N)cc2Cl)=O)CC)cnn2c1OCCCC2 c1(C(=O)NC(c2cn(-c3cccnc3)nn2)(C)C)nn2cccnc2c1Br C1(C(=O)NC(CCC)c2nn[nH]n2)CC(C)CN(C(=O)CC=CCCCCC)C1 c1(C(N2C3(CNC(C4C=CCC4)=O)CCC2CC3)=O)ccn2nccc2c1 C(C(C)CN=c1[nH]c(=NCC2(C(C)CCO)CCC2)[nH]c2c1COCC2)OCC c1(C2N(C(c3nc(OC)c(C)s3)=O)CCC2)ccc2cccnc2n1 C1(C(N2CCC(NC(C3N(Cc4ccc(C)o4)CC3)=O)C2)=O)NC(=O)OC1(C)C C1(CCN(C)C(c2ccc(F)cc2)=O)CCN(C(=O)Cn2c(O)nnc2O)CC1 C1(C(N2CCN(C(C(C(=O)OCC)F)=O)CC2C)=O)CCCC1S(C)(=O)=O C1(CC(N2C(C(C)NC(=O)CSC(=N)N)CCC2)=O)CCCCN1C C1(CNC(c2c(C)coc2C(C)(C)C)=O)CN(C(=O)COC(F)(F)F)CC1(F)F Cc1[nH]nc2ncc(C(=O)NCCC3CN(C(=O)C(C)CS(C)(=O)=O)C3)cc12 N1(C(C(CCOC)OC)=O)CCN(C(C2CCN(OC)CC2)=O)CC(C)(C)C1 C1(NC(C(c2ccc(C)o2)C)=O)C=CCC(C(N2CC=CC2(C)CO)=O)C1 C(c1cccc(CO)c1)=CC(N1CCCC(N(C(c2c(CC)non2)=O)C)C1)=O N#CC1CCCN(C(=O)CCCNC(c2csnc2Cl)=O)C1 c1(CC(=O)NCC(CN(C(c2cnn(C3CC3)c2)=O)CC)(C)C)c(C)cccc1C N1(C(C2=CC(C)C2)=O)CC2N(C(C3CCc4nnnn4C3)=O)CCC2(C)C1 c1(C(N(CCOC)CCNC(c2sccc2Br)=O)=O)cn2cc(C)c(C)cc2n1 CCCCCCC(C)C(=O)N1CCC(CNC(=O)CC2CCCCCC2(F)F)C1 C(=O)(C#CC1CCCCC1)N1C2CCN(C(c3c(C)ncn(C)c3=O)=O)CC2C1 C(=O)(C(O)CC(C)(C)C)N(C)CC1OCCN(C(C(COC)C)=O)C1 c1(C(=O)NCCC(C)NC(=O)C(C)(C)c2ccsc2)cc2ccc(O)nc2s1 c1(C(=O)NC(CC)CNC(c2cnn(C)c2SC)=O)cc2c(s1)CN(C)CC2 C12(CNC(C3(C)CC3)=O)CC(NC(=O)Cc3cccnc3Cl)(CCO1)C2 n1(CC)nc(C(=O)NCC(C23CCC(CC2)C3)NC(=O)CC2CCOC2)cc1C c1(C(N2CC(NC(=O)CCCN3C(=O)CNC3=O)C3C2C3)=O)ccn2ccsc12 N1(C(C)=O)CCC2(CC1)CC(N1CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)CC1)CO2 C12(CNC(c3c(CC)csc3)=O)CC(NC(=O)C(COC)N(C)C)(CO1)C2 C=CCC(C)(CC)C(=O)NC(C)(C)CN1CCN(C(=O)C(C)(C)C(C)(F)F)CC1 C(=O)(C#CC1CCCCC1)NC(COC)C(=O)N1CC(C)(C)C1 C1(N(C(c2c(C)cc(C)o2)=O)C)CCN(C(c2cnccc2C(F)F)=O)CC1C CCCC(CCCO)C(=O)N1CCCC(O)(CNC(=O)COc2cccc(O)c2)C1 C12(C(N3CC(N(C)C)C3)=O)CC1CN(C(c1ccc(=O)oc1)=O)C2 c1(C(=O)NCC2CN(C(c3c(CC)c[nH]n3)=O)CC2(C)C)cc(F)c(C)cc1Cl C12(NC(CC(C)(C)C(F)F)=O)CCCC1N(C(=O)CSc1nncs1)CCC2 N1(C(C(C)O)=O)C2CCC1CC(CNC(c1cncn1-c1ccncc1)=O)C2 C=C(C)CCCC(=O)NC(C)(CNC(=O)C(C)C=Cc1ccccc1)C1CC1 N1(CC(=O)NCC(C2CCOC2)NC(c2ccccn2)=O)CCCOC1=O Cc1nn(CC(C)C)c(Cl)c1CN(C(Cc1cccs1)=O)C(c1ccco1)C1CC1 N1(C(=O)NCCCCc2scc(C)n2)CCOC2(CCCOC2)C1 c1(OC)cc2c(cc1C(C(=O)NC1(C)CC1)N(C(COC)CO)C)CCC2 N1(C(C2CN(C(C)C)C2)=O)CC2CCC1CN2C(C12CCC(CC1)C(C)O2)=O c1(Nc2c(NC(C(CCC)C)=O)cnc(F)c2)ccnc2ccnn12 C1(N(C)C(c2cc(CO)[nH]n2)=O)CN(C(C2CCCO2)=O)CC1O c1(OC(C)C(=O)N(C2CCN(C(=O)CNC=O)C2)CCO)ccccc1Cl Cc1ccncc1CC(=O)N(CCC(C(C)C)NC(=O)C(C)(C)O)C c1(CC(N2C(n3cc(CC(C)(C)C(=O)O)nn3)CCC2)=O)ccc2c(c1)CC2 c1(CC)cc(C(=O)NCCC2CN(C(=O)CC3CCC(C4CC4)O3)C2)no1 c1(C(=O)NCCC2(NC(C3OCCC(C)C3)=O)CC2)cc(F)c(C(F)F)c(F)c1 C1(c2nnnn2C)(C(c2nnnn2C)CC)CCNC1.c1(N)[nH]nnc1C N1(C(C=CC(C)C)=O)CCCC(N(C)C(C2CCOC2C)=O)CC1 O=S(=O)(c1ccc(NCC2CCC=CCC2)c(Cl)c1)NC1CCn2cnnc2C1 C(=O)(C1=C(SC)CCCC1)NC1CCN(C(C=CC(CC)C)=O)C1 c1(C(C(=O)NCCCOC)N(C2CCCC(C)C2)C)noc2c1COCC2 c1(CNc2nc(C)nc(N3CC(CO)C4(CCC4)C3)c2)ccc2c(c1)CCC2 C1(CN(C(=O)C(=O)N(C2CCCOC2)C2CCSC2)C)C2CCCCC12 N1(C(C2C(CC(C)C)C2)=O)CCC(O)(C(=O)OC(C)(C)C)C1 C1(C(C)C)CCC(CCCC(=O)NCCNC(=O)OC(C)(C)C)CC1CCC c1(NC(C2C=CC(Nc3ncncc3F)C2)=O)cc(F)cc2[nH]ccc12 C(c1csc(C(F)(F)F)c1)=CC(=O)NCCCC1(NC(=O)CC2CC=CC2)CC1 N1(C(C2(C)CC2(Cl)Cl)=O)CC(NC(=O)CSCCC(F)(F)F)C(C(F)F)C1 C(=O)(CC(C)(C)Sc1ccccc1)NC(C)CCNC(=O)C(C)NC(=O)N(C)C N1(C(=O)OC(C)(C)C)CC(NC(=O)NCC2CC=CCC2)COCC1(C)C C1(C(=O)NCC2CN(C(CNC(C3CCCCC3)=O)=O)C2)CCC12CCCO2 c1(C(=O)NC(CC(C)C)CNC(=O)C(=O)NCCC(N)=O)ccc2sncc2c1 C1(C(=O)NCCOCC(=O)OC)(NC(c2ccncc2Cl)=O)CCC(C)(C)C1 c1(CC)ncc(C(=O)NCC(C)(F)CNC(=O)Cc2ccc(O)c(C)c2)c(C)n1 CCCCCCCCCC(=O)N1CCC(CNC(c2c(C)cc(C)oc2=O)=O)C1 C=CC1(C(=O)NCCN2CCN(C(=O)CC(CC)SC)CC2)CCCC1 C1(NC(CCCCC#C)=O)CCCOC12CCN(C(C1CCC(C)CC1)=O)CC2 N1(C(C2N=C(C)SC2)=O)CC2CCCN(C(c3ncc(C(F)(F)F)s3)=O)C2C1 CC1CN(C(=O)COC2CCCOC2)CC(C)N(C(=O)C=Cc2ccoc2)C1 c1(C(=O)NC2CCCCN(C(C3(C)CCCCC3)=O)C2)cc(O)c2ccsc2c1 c1(C(=O)NC2CCC(CNC(C3(O)COC3)=O)C2)cc2n(n1)CCOC2 n1(C(=O)NC2CC(CC(N3CC4CCCCC4C3)=O)C2)ccc2ccccc12 C1(NC(C2CC2c2cnc[nH]2)=O)CCCN(C(c2ccccc2Br)=O)C1 S(=O)(=O)(c1c(F)c(F)c(F)c(F)c1F)N1CC(C(=O)NCC(C)(C)F)C(O)CC1 c1(-c2nc(CCCN(C)C)nn2C2CCS(=O)(=O)C2)occ2c1CCOC2 c1(OC)cscc1C(N1CC(CCNC(c2ccns2)=O)(OC)C1)=O c1(C(N2CCC(NC(C3(CC)CCOC3)=O)C(O)C2)=O)c(Cl)cnc(OC)c1Cl C1(NC(C(=O)NC(c2ccc(CC)cc2)c2cccs2)=O)COC2(CCC2)C1 c1(C2(C(=O)NC(CCOC)CNC(=O)CC(C)C)CCCC2)cccc(F)c1 c1(OC)ccccc1C(=O)NC(C)C(C1CCCCC1)NC(c1cc(Cl)no1)=O C(CCC(C)(C)CO)NC(C(CN(C(C(C)=NOCC#N)=O)C)C)=O c1(C(N2CCC(O)(C(C)CNC(=O)Cc3cnccn3)C2)=O)c(N)cccc1Cl C1(C(=O)NCC2CCC2)CC2CCCCC2N1C(c1cnc(C(F)(F)F)cn1)=O C1(C(CNC(C2(CF)CC2)=O)NC(CNC(CCC)=O)=O)CCCCC1 CCCC(C(O)C(=O)NC(C)CCOCC)NC(C1CCC(C2CC2)C1)=O CC1CCC(C(=O)NC2(C#N)CCCCC2)CN1C(=O)COCC1CCCC1 Cn1cnc2sc(C(=O)NC3CN(C(=O)CCC4CC4)CCC3CO)cc12 C1(C(N2CCCC2=O)C)CCCN(N2CCC3CNC(=O)CC3C2)C1 c1(C(=O)NC23CCN(C(CC4(C=C)CCC4)=O)CC2C3)cncc2c[nH]nc12 CC(CCN=c1[nH]c(N2CCN(CC(=O)NCCO)CC2)nc(=N)[nH]1)P(C)(C)=O C=CCC(CNC(=O)C=CC(C)CC)C(=O)NCC(O)CC1CCC1 CC1(C2CCN(C(C3(NC(C4CC5(CCO4)CC5)=O)CC3(C)C)=O)C2)CC1 c1(CC)cc(C(=O)NCc2cc(C(=O)N(CC(CC)N(C)C)C)co2)n[nH]1 c1(CN2CCC(n3cnc(OC4CCN(C)CC4)n3)C2)cc(F)cc([N+](=O)[O-])c1 Cc1cc[nH]c(=N)c1C(=O)N(C)CC1CCCN1C(=O)CC1CCCCCC1 N1(C(C2C(OCC)C2)=O)CCN(C2CCN(C(=O)CC3C(=O)ON=C3C)C2)CC1 c1(C(N2CC(OC)(CNC(=O)CN3CCCC3C)C2)=O)cn(C)c(O)n1 C1(OC)(CNC(N2CC(C)CC2CO)=O)COCC1(C)C C(N=c1nc(NC2CCCCC23CC3)c2c([nH]1)c(C)nn2C)C1CCC(OC)C1 CCC(C)(CC(=O)N(C)CCOCCNC(=O)Cc1cncnc1O)C(=O)OC n1(C(C)C)ccnc1C(=O)NC(C)C(CO)NC(=O)C(n1ccc(C2CC2)n1)C c1(C(N(C2CCN(C(c3ccc(CO)o3)=O)C2)CC)=O)cc(SC)ccc1Cl C1(CC(=O)NC(c2ccnc(OC(F)(F)F)c2)=O)CC2(C1)CN(CC1(C)COC1)C2 C1(CNC(CCC#C)=O)CCCCN(C(C2CCN2CC)=O)CC1 C(=O)(C(F)(F)C(C)(C)O)N1CC2N(C(c3n(CCC)ncc3)=O)C(C2)C1 C(=O)(C(CCCOC)NC(=O)CSc1nc[nH]n1)NC1CCCN(CC)C1 c1(C(=O)NC(C2CCN(C(CCCCSC)=O)C2)C)cc2oc(C)c(C)c2[nH]1 C(=O)(C1CCCc2nncn21)NC(C1CCCC1)CNC(C(C(C)O)N(C)C)=O CC(C(=O)N1CC(CCNC(=O)CCNC(=O)C=CCl)C1)CS(C)(=O)=O c1(C(N2C(CN(C(=O)C=CC3CC3)C)CCC2)=O)n[nH]c2c1CCC2 c1(OC)nc(Cl)cc(=NC(=O)CC2CCCN2C(c2cc(F)cc([N+](=O)[O-])c2)=O)[nH]1 N1(C(c2c(C)snc2)=O)CCCC(NC(c2conc2C2CCCO2)=O)C1 C1(CNC(C(CC#C)O)=O)CC2(C1)CN(C(=O)C(CC)CC=CC)C2 n1(CC)nccc1C=CC(=O)NC(C)CCNC(=O)C(C)Cc1cccc(Cl)c1 C1(COC)(NC(c2[nH]nnc2C)=O)CCCN(C(=O)COCCF)C1 C(C(C)(C)C#CC(=O)NC(C)CCSC)NC(COC)=O n1(CC(N2C(CNC(c3ccnn3C)CC)CCC2)=O)ccc(C)cc1=O c1(NC2C(C(F)(F)F)CCN(C(=O)CN3CCCCC3)C2)ncnc2scnc12 c1(CCN(C(C(=O)OC)C(C)C)CC=C)ccccc1Sc1cccs1 C1(C(=O)NC2CC(NC(=O)CSCc3ccc(Cl)s3)C2)CC2CCC(C1)O2 C1(C(N(CC(C)NC(=O)CCc2cccnc2F)C)=O)CCc2ccnn2C1 CC1(C)CCCC(C(=O)NCCC2CCCN2C(=O)C(=O)NCCC(N)=O)CC1 CN1C(=O)OCC1C(=O)NCc1ccc(CCNC(C23CC4CC2C3C4)=O)cc1 c1(C(=O)NCC(C2CCCN2C(=O)C(F)C2CCC2)(C)C)cnncc1O C1(CNC(C(CCC)C)=O)CC2(C1)CN(C(=O)C(C)CN(C)C)C2 N1(C(C23CCC(C(N4Cc5c[nH]nc5C4)=O)(CC2)C3)=O)CC(F)(F)C(F)(F)C1 C123CCC(CC1)(C2)NC(=O)N3.N1(Cc2cn(CC(CC)O)nn2)CC2CCC1C2 C(=O)(C(CCC)N(C)C)NC(C1CC(SC)C1)C(N1CC(=CC)C1)=O C1(COC)C=CCN1C(=O)Cn1cc(C(=O)N(C)C(C)C)nn1 C(=O)(C(C)(C)CC(=O)OC)N(CCCNC(c1cccc(CC)c1C)=O)CC C1(n2cccn2)(C(N(CC(C)NC(c2ccc(Cl)nn2)=O)C)=O)CCOCC1 C1(C(=O)NC(C(C(N2C(COC)COCC2)=O)C)C)CC(C)(C)CCO1 Cc1[nH]c(C(=O)NCC23CC(CO2)N(C(C2CCS(=O)(=O)C2)=O)C3)c(C)c1C C(=O)(C1CSc2ccccc21)NCC(CC)(CC)NC(=O)C(O)C(C)(C)C C(CC(=O)NCC1OCC2CCC1C2)(C(C)(C)C)NC(C(C)n1cncn1)=O Cc1c(C(=O)NCC(N2CCN(C(=O)C(c3ccccc3)C)CC2)=O)cnn1C Cc1ccccc1COCC(=O)NCC#CCNC(C1(C)CCCC1C)=O CCC(C)C(C(=O)NCC1(O)CC=CC1)NC(=O)C(O)CCSC C1(NC(c2cn(CCC(C)(C)C)nn2)=O)CCCC12CN(C(C1CSC1)=O)C2 C(=O)(CC(O)CNC(=O)C(N)=O)NC(c1cncs1)C n1(CC)nccc1CC(=O)NCC1(NC(=O)CCn2cc[nH]c(=O)c2=O)CCCC1 c1(C(=O)NCC23OCC(NC(C(C=C)CC)=O)(C2)C3)cccc(F)c1CSC C(=O)(C(CC(C)C)NC(=O)C(c1cnc(Cl)n1C)N(CCC(F)(F)F)C)OC C1(C)(NC(CCCNC(C)=O)=O)CCCN(C(=O)CCc2ccccc2O)C1 C1(NC(CCCn2c(C)nc(C)n2)=O)CC(C2CCN(C(C3(C)CC3)=O)C2)C1 Cc1ccc(C#N)cc1OCCCC(=O)NCC1(C)Cc2ccccc2C1 Cc1c(F)ccc(N)c1C(N1CCCC(NC(C2(C)CCCCO2)=O)CC1)=O N1(C(C(CC)F)=O)CCC(N=c2[nH]nc(O)s2)(C(N)=O)CC1 C(=O)(CCCCNc1ccco1)N(C(CC)CC)C C1(CC)CC(=O)N(C(C)C)C1.c1(C2c3nnnn3CCCN2)cc(C(C)C)no1 c1(C(N(C(C)CNC(=O)C=Cc2cccs2)C)=O)cc(C2CCCO2)n(C)n1 Cc1cc(OCCN(C)C)ccc1N(C)C(C1CCCC1C)=O c1(C(N2C(CNC(c3c(Cl)n[nH]c3C3CC3)=O)CCC2)=O)ccccc1F C1(NC(C2C(COC)CC2)=O)CN(C(=O)C=Cc2cccnc2)CC2(CCC2)C1 C(CC(C)(C)CNC(=O)C(C)(C)Cc1cnn[nH]1)NC(C(C)OC)=O N1(C(C2(C)CC=CC2)=O)CCCCC2(CCN(C(C3CN(C4CCC4)C3)=O)C2)C1 c1(OCC(=O)NC2CN(C(c3cnc(C)n3C(F)F)=O)C2)nc(O)nc(O)n1 Cc1cc(SCC(N2CC(F)(c3ccncc3)C2)=O)sn1 C1(OC)CC(NC(c2cnoc2C2CC2)=O)CN(C(=O)C(=C2CCCCC2)F)C1 C1(NC(c2ccc(CN(CC)CC)o2)=O)CN(C(c2sc(C)cc2C)=O)CC1O N1(C(c2ccc(C)nc2O)=O)CCC2CCN(C(c3cccc(CO)c3)=O)C2C1 c1(Cn2c(C(=O)NC(c3ccsc3)C)ccc2)ccc(Cl)cc1 N1(C(CNC(C(C)=C(CC)C)=O)=O)CC(C)(NC(C2(SC)CCC2)=O)C1 N1(C(C2(C)CCN(C(c3c(C)cc(N)cn3)=O)CC2)=O)CCN2CC(C)CC2C1 CC1(C)CC(NC(=O)Cc2cc(Cl)ccc2O)CN1C(C1C2CC3C(C2)C13)=O n1(CC(=O)NC2CC2c2nc[nH]n2)cc(C(=O)NC2(CC3CC3)CC2)nn1 N#CC1CC(CNC(=O)CNC(=O)CNC(=O)CCCn2ccnc2)C1 C1(CNC(Cc2c(C)nn(C)c2)=O)COCCN(C(C2CCC(=O)N(C)C2)=O)C1 C1(NC(C(C)(C)OC)=O)CS(=O)(=O)CC1N=c1ccc2c([nH]1)CCCC2=O C1(CC)CN(C(c2n[nH]c(C3CC3)n2)=O)CCC1NC(c1nn[nH]c1Cl)=O C(=O)(CCCC(CC)NC(=O)COC(C)(C)CC)NCC=CCCC C12(CC(=O)N(CCNC(CC3CCCC(OC)C3)=O)C)CCC(CC1)C2(C)C c1(C(N2C(C(N3C4CCC3COC4)=O)CC3CC32)=O)cccn2ccnc12 Cc1sc(O)nc1C(=O)N(CC(C)C(=O)NCC(CC1CC1)CO)C C1(NC(CC2N(C)CCCC2)=O)CC2CCC1CC2NC(=O)C=Cc1cnc[nH]1 N1(C(C(CCOC)C)=O)CCCCCC1C(=O)Nc1ccc(OC(C)C)cc1O CCC(CC(=O)NCC1CN(C(c2c(F)ccc(C)c2N)=O)C1)CC(F)(F)F N1(C(C(C(C)C)F)=O)CC2(CCCC2)C1C(=O)NCc1ccnc(F)c1 S(=O)(=O)(c1ccc(C#N)c(NC(CO)C2CC2)c1)NCCCSC c1(C(N2CCN(C3CN(C(CS(C)(=O)=O)=O)C3)CC2)=O)ccnc2c1OCO2 c1(C(C)C(=O)NC2(CNC(C3CC(Cl)(Cl)C3)=O)CC2)ccc(F)cc1 C1(C(C(=O)NCC(CC)(C)NC(c2cc(OCC)cnn2)=O)F)CCCN(C)C1 Cc1ccc(C(=O)NC2CC3CC(NC(C4CCCCC4(F)F)=O)C3C2)nc1O Cc1nsc2ncc(C(N3CCN(C4CN(CC=CCl)C4)CC3)=O)cc12 Cc1cc(C(N2CC3CC2CN3C(c2cc[nH]c3nccc2-3)=O)=O)cc(C)c1N C(=O)(CS(=O)(=O)C(C)C)NC(CC)CNC(c1coc(C(C)OC)n1)=O C(=O)(C=C1SCC(=O)N1C)NC1C(OC)CN(C(C2CC3(C2)CC32CC2)=O)C1 c1(C(N(C2CN(C(=O)CC3(C)CCS(=O)(=O)N3)C2)C)=O)cccn2cncc12 CC1(C)CC(NC(C2CCN2C(=O)C=CC2CCCC2)=O)C12CC2 C1(C#N)(SC)CN(C(C2CCCC2CNC(=O)C=Cc2ccsc2)=O)C1 c1(C(=O)NC(c2ccccc2)C(=O)NCC(C)(C)OC)ncccc1N c1(C(N(CC(=O)NC(C)CC2(O)CCC2)CC#C)=O)cc(C(F)F)[nH]n1 N1(C(C=CC=CC)=O)CCN(C(=O)CC2OCCCO2)CC1CCOC c1(OCC)ccccc1N(CCCC(C)O)C.c1(C2C(=O)N2)nc(CO)cs1 C1(CCC(=O)N(CC(=C)C)CC)CCCN(C(=O)C=Cc2cnn(C)c2)C1 CC1CN(C(=O)COCC2CCOC2)CC1NC(=O)C(c1cccc(F)c1)(C)C CCS(=O)CC(=O)NCC(C)CNC(c1cnc(C2(C)OCCO2)s1)=O C1(NC(C=CC(=O)OCC)=O)(CNC(c2ccncc2F)=O)CCCCC1C c1(C(=O)NC2CN(C(c3n(C(C)C)cnc3)=O)C(C)C2)ccc2oc(=O)oc2c1 C1(CC(=O)NCC(C2CC2)NC(c2cc(C)[nH]n2)=O)NC(=O)NC1=O CCN=c1[nH]cc(C(=O)NC2CCCN(C(C3CC(C(C)C)=NO3)=O)C2)s1 N1(CC)C(=O)CCC1C(=O)N(C)CC1CCN(C(c2nn(C)cc2SC)=O)C1 C1(CC(=O)NC2C(NC(N)=O)CC2)CCCCC1NC(c1cocn1)=O Cc1cccc(CCn2cc(CNC(=O)C(C(C)C)c3ccn(C)n3)nn2)c1F C1(CNC(C(C)NC(=O)CC2C=CCC2)=O)CN(C(C2CC23CC3)=O)CCO1 Cc1nnc2n1CCCC2C(=O)NCC1CN(C(C2(F)CCOCC2)=O)CCO1 C(=O)(CC1=CCCCC1)N(C1CC(NC(C(C=C)c2ccccc2)=O)C1)C N1(C(C2COCC(C)(C)C2)=O)CCC(S(=O)(=O)c2ccc(Br)cc2)CC1 C12(NC(C=COCC)=O)CCCCCC1N(C(c1cc3nc[nH]c3cn1)=O)CC2 c1(-c2cccc(NC3CC(C(=O)OC)CC3O)c2)n[nH]c2c1CCCC2 C(C(O)CC(=O)NC(C)Cc1cnn(C)c1)NC(C1(CC=C)CC1)=O N1(Cc2nnc(CC)o2)CC2CCC1C1CN(C(c3ccoc3Cl)=O)CC21 C1(NC(C(CC)CO)=O)CCC2(CC1)CCN(C(=O)C(C)CC(=O)OC)C2 N1(C(CCC(C)NC(c2ccccc2)=O)=O)CCc2ccc(Br)cc2C1 N1(C(c2ccc(C#N)cn2)=O)C2CCC1CN(C(=O)CCc1nc[nH]n1)CC2 C1(C(N2CC3C(C(=O)NCCN4CCC(OCC)C4)(C3)C2)=O)CC(C(C)C)=NO1 Cc1cc(F)oc1C(N1CCC(C(C)C(=O)N(CC(O)CO)C)CC1)=O c1(-c2ccc(CN3CCC(O)CC3)cc2)ccc(C(F)(F)F)c2ncccc12 C(CN=c1cccc(S(=O)(=O)NC(CC)C(C)Cc2ccccc2)[nH]1)N(C)CC N1(C(Cc2c(C)ncs2)=O)CC(CCNC(=O)Cc2cnoc2)OC(C)C1 c1(C(C)C)cccc(NCC2COCCO2)c1O C1(C(CO)N(C(N(C)C2CC2)=O)CCO)COC(C)(C)O1 C1(CNC(c2n(CC)ncc2)=O)CC(F)(F)CN1C(c1cnc(Cl)s1)=O N1(CCOC)CC2CN(CCCCNC(c3ncc(C(F)(F)F)cc3Cl)=O)CC2C1.S c1(CNC(C2CCN(C(=O)CC3(N4CCCC4)CC3)C2)C)c[nH]c2cc(N)ccc12 C(=O)(C(C)C(CC)CC)N(Cc1cccc(CNC(C(C=CCCC)O)=O)c1)CC N1(C(CC2C(C)CCO2)=O)CCC(NC(c2occ3c2CCOC3)=O)C12CCC2 C12(C(=O)NC(C3(O)CN(C(c4ccncc4N)=O)C3)C)CC(C1)C(C(F)(F)F)O2 C1(NC(CC(C)F)=O)CCN(C(c2cc(-c3cccnc3)no2)=O)C1C(C)(C)C CCCCCCC(C)NC(=O)C(C1CC1)N(C(=O)COCCCN(C)C)C Cc1nccnc1NC(=O)CCC1CCCN1C(=O)C1CC1 c1(C(N2CCC(F)(C(=O)NCCCOCC#C)C2)=O)ccc2n[nH]cc2c1 c1(OC)c(Cl)cc(C(N2CC(NC(=O)CCN(C)CCO)CC2C)=O)nc1Cl c1(CC(=O)NC2C(C(=O)NC(c3ccccc3)CN)C2)csc2c(Br)cccc12 C(=O)(CCCCCn1cncn1)N1C(CNC(=O)CC2NC(=O)NC2=O)CCC1 C1(NC(CC2(C)CC2)=O)CC2CN(C(C3Cc4cscc4C3)=O)CCN2C1=O c1(CC)ncsc1C(=O)NCC(C)(C)CN(C(=O)CCCc1ccc(C)s1)CC CC1(C)CC(C(=O)N2CCC(CO)C(NC(=O)C=CC(F)(F)F)C2)=NO1 C1(CN(C(CC2CC(OCC)C2)=O)C)CN(C(C2CCC(C)(C)O2)=O)CC12CC2 CC(CC(N)=O)C(=O)NCC1(C)CCCN1C(=O)CCc1cnc(C2CCC2)o1 Cc1cc(=O)n(CCC(=O)NCC2CCN(C(C3CC(C)OC(C)C3)=O)C2)cn1 Cn1c(CCC(=O)NC(C2CCN(C(C3CC4(F)CC3C4)=O)CC2)(C)C)nnc1S Cc1cc(NC(=O)C(O)CN2CCCC2)ccc1C1COC1 N1(C(C2C(SC)C2)=O)CCC(c2ccc(F)cc2)(CNC(=O)C2=C(Cl)CC2)CC1 CCC(CC)(C(N)=O)NC(C12CCC(CC1NC(=O)C(C)OCC1CC1)C2)=O C1(C(N(CCN(C(C(CC=C)C(C)C)=O)C)C)=O)CC12CCC(F)(F)CC2 C1(CNC(C2C(OCC)CC2)=O)CCN(CCNC(=O)COC(CC)CC)CC1 CC1=NN(C)C(=O)C1CC(=O)NCC1(F)CCCN(C(C2COC(=O)N2)=O)C1 CC(CC(C)(C)C)C(=O)NCCC12CCC(C1)N(C(c1cc(C(N)=O)c[nH]1)=O)C2 CC1CN(C(=O)CN2CCC2)CC(C)N(C(=O)C(=CC2CCCCC2)F)C1 C1(NC(CC(OCC)OOCC)=O)CC2CCCC(C1)N2C(C1CCC1(F)F)=O CC1(C)CC(CNC(c2nc(Cl)sc2Cl)=O)N(c2ccnc(CO)n2)C1 CC1(CC(N2CC3C(C(N)=O)C3C2)=O)CCN(C(C2CC3(CC3)CO2)=O)C1 C1(C(C)(C)COC(C)C)c2n(nnn2)CCN1.c1(CSC)cnc[nH]1 Cc1ccc(C(=O)NC2(C(N3CC(O)CCC3C)=O)CCOCC2)cc1C C1(CNC(c2cnc(C3CC3)[nH]2)=O)(CO)CCN(C(c2ccsn2)=O)CC1 N1(C(C2C(NC(c3c(C)ccc(F)c3)=O)CCOC2)=O)CC2(CNC(=O)OC2)C1 c1(OC(C)C)cc(C(=O)NC2CC2CNC(=O)C(=O)Nc2ccccc2)ccn1 c1(CC)ccc(C(=O)NC2(CCNC(=O)CCc3ccccc3F)CCC2)nc1 c1(OC(C(=O)NCC=CCNC(C2CC(OC)C2)=O)C)ccccc1Cl O=C(CCC12CC1=NN=NN1C(=CC=COC(CC)COCCN2)CC1)NF N1(C(C)C(=O)N(C)C(c2ccc(F)cc2)C)CCC2(CCCCC2)C1 C1(C(N2CCC(N(C(=O)CC3CCC(=O)O3)CCO)CC2)=O)CCCCCCC1 n1(CCC)c(CSCC(=O)Nc2cccc(N)c2)nnc1SC C1(C2CCOCC2)(CNC(COC(CC)C)=O)CCN(C(c2csc(C)c2)=O)C1 c1(C(N(C2CN(C(=O)CC3COC(C)(C)CO3)C2)C)=O)cccc2cc[nH]c12 N1(C(C=CCOC)=O)CCN(C(C2C(C)C2C)=O)C(c2ccc(SC)cc2)C1 c1(CNc2c(C(=O)NCC(C)OC)n[nH]c2)ccc2cc[nH]c2c1 C(=O)(CC(O)Cc1ccccc1)NCCCN(C(c1n(CC)ncn1)=O)C1CC1 c1(C(=O)NC2C(NC(C(C)(O)CCc3ccccc3)=O)C2)cnc2c[nH]nc2c1 c1(C(=O)NCC2CCN(C(CC3CN(C)C3)=O)CC2O)ncccc1S(C)(=O)=O C(CCCCC(=O)NC(C)(C)C(=O)N(C)Cc1cc(C)ccc1C)SC Cc1cc(C(=O)NC23CC2CN(C(=O)C(C)OCC2CC2)C3)c2c(C)n[nH]c2n1 Cn1ncc(C(N2CC3=C(C2)CN(C(C2CC(C)(C)C2)=O)C3)=O)c1S(N)(=O)=O N1(C(CC(CC)NC(=O)Cc2cnsc2)=O)CC2CC=CC1C2 N1(C(c2c(O)ccc(SC)c2)=O)C2CCC1CC(NC(C1CC(N(C)C)C1)=O)C2 c1(C(=O)NC(C(N2CC(CCC#C)C2)=O)C2CCCO2)nscc1C Cc1cnc(F)c(CNC2(NC(c3ccc(C(C)C)s3)=O)CC2)c1 C(=O)(C(C1(O)CCC1)NC(C1CC1(C)C)=O)NC1(C(C)O)CC1 c1(C(N2C(CN(C(c3c(C)con3)=O)C)CC(F)C2)=O)cc(Cl)nnc1O C1(NC(C2(COC)CC2)=O)(COC)CCN(C(C2C=CC2C(=O)OC)=O)C1 CCCCCCC(=O)N(C)CCOCCN(C)C(C1CCC1C(=O)OC)=O C(N=c1[nH]c(=NC2CCCSC2)[nH]c2c1COC2)c1ccc(S(CC)(=O)=O)s1 CC(C)CCC(O)C(=O)NC1CCCC1NC(=O)CSCCC#N N#Cc1cc(F)cc(C#N)c1OCc1noc(C(F)F)n1 N1(C(C2(CC#C)CCN(C(=O)Cc3csc(C)c3)C2)=O)CCC(CO)C(C)C1 N1(C(CC(=O)N(CCC(=O)NC)CC)=O)CCC2(CCCO2)CC1 S(=O)(=O)(c1c[nH]c2ccccc12)N(C(CS(CC)(=O)=O)CC(C)C)C(C)C CC(C)(CC(F)C(=O)NCC1CCC2(CC2)CO1)NC(c1cccnc1S)=O N1(CCS(CC)(=O)=O)CCC(=O)N(CC2CCN(CC(C)C)C2)C1=O c1(C(=O)NC2CCCC(NC(C=CC)=O)C2)cc(C(C)(C)C)ccc1N C1(NC(CC(C)NC(N)=O)=O)CCN(C(=O)C(c2cccc(F)c2)O)CC1O CC1(C)CCN(C(C23CC(CCO2)C3)=O)CC1NC(c1cc2ncccc2s1)=O C1(C(=O)NC(C)CCNC(=O)CC2CSC2)CN(S(=O)(=O)N(C)C)CCO1 N#Cc1cc2cc(C(N3CC4CC3CN4C(c3ccc(Cl)o3)=O)=O)[nH]c2cn1 CC1CN(C(=O)CSSC)CC1CNC(C1(C(=O)Nc2ccccc2)CC1)=O C(C(C)C(C)(c1nnnn1C1CC1)NCCc1nc(C(C)(C)C)no1)OC S(=O)(=O)(c1ccc(Cl)cc1)N(C)C(C12CCC(c3cc(F)cc(F)c3)(C1)C2(C)C)=O C12(NC(c3ccc4ccccc4c3)=O)CCCC1N(C(=O)CCOC1CC1)CCC2 N1(C(C2(C)CC(OC)(OC)C2)=O)CCCC2(NC(=O)CCn3cncn3)CC2C1 CCCC(C)CCCC(=O)NCC#CCNC(=O)OC(C)(C)C C1(N(C)C)(COC)CCCN(C(C2Cc3cscc3C2)=O)C1.C1(=O)C(C(C)C)N1 c1(N2CCC(CC)C2)nc(N2CCN(c3ncccc3F)CC2)nc2sccc12 C1(NC(c2cc(C(=O)OC)oc2C)=O)C(C)CN(C(=O)C2CC2)CC1C CCCCC(CC)C(=O)N1CC(NC(=O)Cc2c(Cl)cncc2Cl)C(CNC)C1 C(C(=O)NOCc1ccc(F)cc1)(C(C)O)NC(CS(CC)=O)=O C1(NC(c2c(C)ocn2)=O)CC2(C(=O)NCCCc3ccsc3)COC1C2 C1(CN(C)C(C2Cc3nccn3C2)=O)CN(C(c2ccon2)=O)CC12CC2 c1(CC)cc(N)c(C(=O)NCC2CCC(NC(=O)C(O)CC(N)=O)CC2)cc1F C1(CN(C(=O)CC2CCSCC2)C)CC(F)CN1C(C1CC=CCO1)=O c1(C(N2CCC(C(C)CNC(=O)C(C)C(F)F)CC2)=O)nccc2cc[nH]c12 CC1(C(=O)NCC2CC(NC(=O)Cc3ccc(Cl)s3)C2)CCCOC1 C#CCC(O)C(=O)NCCN(C1CCCCC1)C(c1cc(Cl)no1)=O C1(NC(=O)OC(C)(C)C)CCN(C(c2cc(C3CCCC3)no2)=O)CC1C(=O)O N1(C(C(=O)N(CCC)CCN(C)C)=O)CC(CC)(CO)C1(F)F c1(COC(C(=Cc2ccc(OC)cc2)C#N)=O)cc2ccnc(Cl)c2o1 N1(C(c2n(C=C)ncc2)=O)CC(NC(c2cc(O)cs2)=O)C2(CC2)C1 C#CC#CC(C)(C)NC(c1sccc1CNC(C1CCC(C)S1)=O)=O C(=O)(N=c1[nH][nH]c(C)c1C)C1C(O)CCN(Cc2c(OC)ccnc2F)C1 C1(O)(CN(C(=O)CCCNC(N)=O)C)CCCN(C(C2CCC3(CC3)C2)=O)C1 C1(NC(C(CC=C)(F)F)=O)CN(C(=O)CCc2cc(C)on2)CC(C)(C)C1 C(N=c1[nH]nc(Cc2ccc(Cl)cc2)n1C)c1c(C)cc(CC)o1 c1(OC)ccc(OCCCNC(=O)C(C)O)cc1.C(CC(C)(C)N(C)C)SCC c1(C(=O)Nc2ccc(C)c(C)n2)ccc2c(c1)CCNC2C1CC1 n1(CC(=O)NC2C3CN(C(C(C)C(F)(F)F)=O)C2C3)sc(=O)c2ccccc12 N1(C(=O)CC2CCOCC2)CCCC(C2CCN(C(C3(O)COC3)=O)C2)C1 C12(C(c3nnnn3CCCSCC)NC(CC=C)(C)CC)CCC(CC1)CO2 CC1CCN(C(c2nccc(Cl)c2O)=O)CC1CNC(=O)C(O)C1CCC1 S(=O)(=O)(c1ccncc1)Nc1c(C(=O)NCCCN2CCCCC2)cc(OC)nc1 N1(C(CCCCN(C)C(C2(CO)CC2)=O)=O)CCC(F)C(O)C1 CC(C)CCCC(C)C(=O)N1CCC(CNC(=O)C(F)(F)CN(C)C)C(O)C1 c1(C(C(=O)NCCC2CN(C(c3ncccn3)=O)CCO2)O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(CN(C(c2cc(C(C)C)no2)=O)C)O)cc(Cl)ccc1F Cc1csc2ncc(C(N3CC=CC3CNC(c3ccon3)=O)=O)n12 C(=O)(N=c1[nH][nH]cc1C)c1cccc(NC(C(CC)(C)O)=O)c1 CCC(CC)C(F)C(=O)NCC1CN(C(C2(C)CCCN(C)C2)=O)CC1(C)C c1(C(=O)NCC(C2CCC2)NC(c2cc(C(N)=O)oc2)=O)ccc2nncn2c1 c1(NC)ccc(C(=O)NC2CCC(NC(=O)CC3(O)CCCOC3)C2)cc1F N1(C(C(C)(c2ccccc2)OC)=O)CCC2C(C(=O)OC(C)(C)C)C1C2 C1(NC(CC(=O)NC2CC2)=O)CC2CCCC(C1)N2C(c1ccon1)=O C12(C(=O)NC(C)CNC(=O)CCNC(c3cccs3)=O)CC(C)(C1)C2 C(=O)(CCCC(=O)N(C1CCCN(C(=O)C(CC)N(C)C)C1)CCO)NCC C1(CC(=O)NCC2CC(C)(C)C2)CCCCCN1C(C1CCCOCC1)=O Cc1ccc(NC(C2CCC(O)CN2C(=O)Cc2cc[nH]n2)=O)c(C)c1 c1(C(N2C(CCC)CN(C(C3CC(C)(C)C3)=O)CC2)=O)nnc2n1CCCCC2 c1(C(N(C2CN(C(=O)CCOCC3CCCO3)C2)C)=O)cccn2nncc12 Cc1oc(-c2ccsc2)nc1CC(=O)NCC(CCO)OC(F)(F)F C(=O)(C1=C(CCl)N(CCCOC)C(=S)NC1c1nc[nH]c1C1CC1)OCC N1(C(=O)CCC2OCCO2)CC2(CCN(Cc3csc(-c4ccoc4)n3)C2)C1 C1(CCC(=O)NC(C(=O)NCCCOC=C)C2CCOC2)CCC(=O)C1 CC1=C(C)CC(C)(C(=O)N(C2CCN(C(c3cc(Cl)ccc3Cl)C)CC2)C)CC1 N1(C(C(CC=C)(F)F)=O)CCN(C(=O)CCC(C)SC)CC12CCC2 C1(O)(C(=O)NCc2c(C(C)C)ocn2)CCCN(C(=O)C(=O)N(C)C)C1 O=C1CCC(C(=O)NCc2ncc(C(=O)N(CCCCO)CCO)cn2)CN1 N1(CC(C)NC(=O)CC2(C)CCN2C(=O)CCN2CCOC2=O)CCOCC1 C1(CC)CCCC(CNC(=O)Cn2cc(CNC(=O)CCl)nn2)C1 CCC(C)C(CNC(=O)CC(C)(CC)NC(=O)CN(C1CC1)CC)CO c1(C(N2C(CNC(C3(C(F)F)CC(=C)C3)=O)CCC2)=O)c(C)ccnc1C N1(C(c2c(CC)noc2)=O)CCC(C(=O)NCC2CCC(F)C2)CC1 Nc1cc(Cl)nc(Cl)c1C(N1CCOC(CNC(C2CCCCCC2)=O)C1)=O c1(CC(=O)NC23C(CN(C(C(C)OCCCC)=O)C2)CC3)nc2c([nH]1)CCCC2 c1(NC(C2N(C(c3scc(C)c3Cl)=O)CC(C)C2)=O)ccc2ncn(C)c2c1 n1(C(C(C2CCOCC2)OCC)OC)cc(CCC(C)N)nn1 C1(CNC(C2C(C(C)C)(CC)C2)=O)CCN(C(C2CC3CC3C2)=O)C1(C)C C1(NC(c2cncc(OC)c2)=O)CC1C1CCCN(C(=O)CC(C)(C)OC)C1 C1(NC(C(NS(N(C)C)(=O)=O)(C)C)=O)CC2CC1CN2C(=O)CC(=O)N(C)C c1(C(C)NC(=O)CCc2cc(Cl)sc2Cl)ccc(S(C)(=O)=O)cc1 c1(C(=O)NC2CCC(NC(=O)CCC3CCCO3)CC2)cnn2c1CC(F)(F)C2 C(=O)(C1=CCCCC1)NC(C(=O)NCCC1CCCN(C)C1)CC1CCOCC1 c1(C(=O)NC2C(NC(C(c3cnccn3)C)=O)COC2)cc2ncccn2n1 c1(C(=O)NC23CC(CNC(=O)C(F)C(F)(F)F)(C2)C3)cccc2cc(F)ccc12 c1(NCCOC(C2(C(=O)OC)CC2C)=O)c(F)ccc(Cl)c1F CC1CN(C(c2nscc2Br)=O)CC1NC(c1cccc(Cl)c1)=O O=C(CCC(=O)c1cccs1)Oc1ccc(Cl)nc1 C=CC(CC)CC(=O)NC(CNC(=O)CCc1cc(C)on1)CO Cc1ccc2c(=O)c(C(=O)NC3CCC(NC(C45CCC4C5)=O)C3)c[nH]c2c1C C1(N(C(C2OCCN(C)C2)=O)C)CC2CCC(C1)N2C(=O)CCc1cccs1 c1(C(N2CCC(C3=NOCC3)C2)C(=O)NCCC2CC2)cccc2cnccc12 N1(Cc2c(CC)cccc2)CCC(NC(c2c(C)nn(C)c2Cl)=O)C(F)C1 c1(C(N(CC(C)N(C(=O)CCC2NC(=O)NC2=O)C)C)=O)ccc2n[nH]cc2c1 c1(C(N2CC(C3CN(C(C(COC)C)=O)C3)C2)=O)ccc2c(C)nn(C)c2n1 c1(CC)cc(=NCC(C)(C2CC2)NC(c2cccc(Cl)c2N(C)C)=O)[nH]cn1 CN1CCC(C(=O)NC2CC2NC(=O)CSc2ccccc2)C1 c1(C(=O)OCC2COC3CCCC3O2)ccc([N+](=O)[O-])cc1Cl CC1(C)CC(C(=O)NC2CN(C(=O)C(C)(F)C(F)(F)F)C2)CC(C)(C)O1 C12(C(=O)NC3(CNC(=O)Cc4cccs4)CCCC3)CCCC1C2(F)F c1(C(N(CCC(C)NC(=O)C(F)(F)CO)C)=O)c[nH]cc(Br)c1=O c1(NC(CNC(Cc2nc(CC)sc2)=O)C(C)C)nc(C(F)(F)F)cc(C)n1 N1(C(Cc2n(C)ncc2Br)=O)CC2CC1CCN2C(=O)CN=S(C)(C)=O N1(C(C2C(C)(C)C2)=O)CCC2CCC(NC(c3conc3C(F)(F)F)=O)C12 c1(OCC(N2CCC(NC(C(C)=C3CCCC3)=O)C2)=O)cc(C)ccc1Cl N1(C(C(C)SCC)=O)CC(CO)C2(C1)CN(C(c1ccncc1F)=O)C2 CCCC(C(=O)NOC(CC(C)C)C(=O)NC1CSC1)OC Cc1nc(C(=O)NCC2CCN2C(c2ccc3c(n2)CCO3)=O)ccc1C#N C1(F)(CNC(c2c(C(C)(C)C)[nH]cn2)=O)CCN(C(=O)CCC(=O)c2cccs2)C1 c1(C(=O)NCC2CCCC2NC(c2cnc(S)[nH]2)=O)ccc2c(c1)OCCCO2 N1(CC)CCN(CCC(N2CCC(NC(c3c(C)noc3C)=O)C2C)=O)CC1 c1(C(=O)NC2(CO)CCN(c3nnn(C)n3)CC2)ccc2cnnn2c1 N1(C(=O)C=CC2CC2)CCCC(CNC(=O)C(F)(F)Sc2ccc(F)cc2)C1 C1(NC(C2(C=C)CCC2)=O)CCC2(CC1)CN(C(=O)CCCCCCC)C2 C1(CC)CN(C(=O)C(C)SC(C)C)CCN1C(=O)C=CC1(C)CCOCC1 N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(C2CC2(F)F)=O)C2COCC12 N1(C(Cc2c(C)scc2)=O)CCC2CCN(C(C3CN(C)CC(C)O3)=O)CC12 C1(C(=O)NC(CC=C)C2CC2)(COC)CN(C(=O)CCN(C)C)C1 C(C)(C(C)(C)C(=O)N1CC2(CC2C(=O)OC)C1)NC(c1c(C)snc1)=O Cc1cc(C(=O)NCC(C)NC(C2CC3(C2)CC(F)C3)=O)c2c(C)noc2n1 c1(OC)ccc(C(N2CCC(CSc3ccc(SC)cc3)C2)=O)c(OC)n1 c1(C(N2C3CN(C(CCc4ccc(C)s4)=O)CC32)=O)cccc(F)c1C c1(C(=O)NC2CC(CCNC(C(C)SCCCC)=O)C2)cc(C2CC2)nnc1O N1(C(=O)C(F)CC2CCCCC2)CCCC(N2CCC2)CC1 Cc1cc(C(N2CCOCC2)=O)nc(O)c1.N12CC(C1)C2=O c1(OCC=C)cccc(CN2CC3CC3(C(=O)NCC3(CO)CCC3)C2)c1 C1(CNC(CC(C=C)C)=O)CN(C(C2CN3CCN2CC3)=O)C2(CCC2)C1 N1(C(c2cnco2)=O)CC2(C1)CCCN(C(c1cnc(Cl)s1)=O)CC2CO CN(C1CN(C(=O)CC2C=CCC2)CCc2ccccc21)C(=O)CCn1cnnn1 c1(OC)ccc(-n2cc(C3C(C)CCN3C(=O)Cc3cscn3)nn2)c(F)c1 c1(CN2C(CNC(C(C)Cc3ccccn3)=O)CC2)cc(Cl)ccc1F c1(C(N2C(C(N(C)CC3CCN(C)C3)=O)CC3CC32)=O)cccc2ccoc12 c1(C(COC(=O)C#CC2(C)CC2)OC)cnn2c(C3CCCCC3)cc(C)nc12 CC(=O)CCCCCCC(=O)N1CCCC(CNC(=O)CC2CCCS2(=O)=O)C1 n1(C(CC)(C)C)nnnc1C1(NC(C)C(C)n2cncn2)CCC1 C(C)(CNC(=O)Cc1sc(COCC)nc1C)(C(C)C)NC(C1C(C=C)C1)=O C1CC(=O)N1C.C(=O)(C(C)=CC(C)(C)C)N(CCCC)C CC1(C(=O)NCC2CC(NC(=O)Cn3ccccc3=O)C2)CNC(=O)C1 C1(C(=O)NCCCN(S(C)(=O)=O)C)CC12CCN(C(C1CCCC(C)(C)C1)=O)C2 N1(C(C(C)O)=O)CCC(CNC(c2ccc(F)c(Cl)c2F)=O)C(F)(F)CC1 C1(C(=O)NCC2CC(NC(C3(CO)CCCO3)=O)C2)CCC2(CCC2)CO1 C1(S(C)(=O)=O)(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CC2)CCC1 N1(C(c2cc(OCC)ns2)=O)CCC2(CCCC2NC(=O)CC2(OC)CC2)C1 C1(NC(c2ccccn2)=O)CC2CN(C(=O)CC3Cc4ccccc4N3)CC2C1 c1(C(=O)NCCCCC2CN(C(c3n(C)nnc3)=O)C2)ccc(C2CC2)cc1 C(c1cccc(F)c1)=CC(=O)NCC1CC2(CC2)CN1C(=O)CC(F)(F)F c1(C(N2CC(NC(=O)CCCOc3ccccc3)C2)=O)ccc(Br)cc1O S(=O)(=O)(c1ccc(CNC(c2cnc(C)nc2OC(F)F)=O)s1)NC c1(C(=O)NCC2C(CNC(CCC(C)OC)=O)C2(F)F)ncc2n1CCCC2 c1(C(C)NCc2cccc(-c3cccnc3)c2)ccc(N)c(Cl)c1 c1(CC)ccc(=NCc2ccc(OC(=O)NCC)cc2)[nH]c1 c1(C(N2CCC(C(C)NC(c3coc(C(F)F)n3)=O)CC2)=O)cc(F)ccc1F N1(C(CCC=CCC=C)=O)Cc2n[nH]cc2C1C(=O)N1CCC(F)C(O)C1 N1(C(CC(n2ccc(C)n2)C)=O)CCOCC1CNC(=O)C1=CCC1 N1(C(c2cnco2)=O)CCC2(CCCC2C(N2CCC3(CCCC3)C2)=O)C1 C1(n2cc(CCCC)nn2)CC2CCC1(NC(=O)C=CCF)C2 S(=O)(=O)(c1cccc(Br)c1)N(C)CC1CCCS1 c1(C(=O)NCC2(NC(C3CC(C)SCC3)=O)CC2)cc(F)c2cn[nH]c2c1 c1(NC(C(=O)NCC2CCOC2c2ccccc2)=O)ccc2nc[nH]c2c1 C(=O)(C1=CCCOC1)NC(C)CN(C(=O)CNC(c1cccc(F)c1)=O)C N#Cc1ccc(CC(=O)NCC=C2CCN(C(c3csc(O)n3)=O)CC2)cc1 C1(CNC(CCn2c(C)nc(C)n2)=O)CN(C(C2CCCOC2)=O)CC1(F)F C12(C(=O)NC(CC=C)CC)CC(CO)(CN1C(C1(C)CCCC1O)=O)C2 c1(CNC(C)Cn2cccn2)cccc(-c2cccnc2)c1F C#Cc1ccc(C(=O)NC(CC(C)C)C(=O)N(CCC=C)CC)nc1 CCC(C)C(C)C(=O)NCCCCCCN(C(=O)CCc1ncco1)C C(=O)(C1Cc2ccccc21)N1CCN(C(c2cccn(C)c2=O)=O)CC(O)C1 c1(C(=O)NC23C(CN(C(C4C(OC)CCC4)=O)C2)CC3)cnc(O)n(C)c1=O c1(C2N(C(=O)NCC3CCCCO3)CCC2)cccc(Br)c1 Cc1ccc(Cl)c(F)c1C(=O)NC1CCCC1CNC(C1(O)CCSCC1)=O C1(CNC(CCOCCN(C)C)=O)COC(CNC(=O)C(C)(C)C)C1 C1(CC(N2CCCC(O)CC2)=O)CNC2(CCC2)CO1.C1(N)CC1F Cc1cc(F)cc(Br)c1C(N1CC(C(C)NC(=O)C(F)n2ccnc2)C1)=O C1(C)(NC(=O)NC(C)CC(=O)NCC(CC2CC2)CO)CCOCC1 c1(CC(=O)NC(CNC(C=C(C)C(C)C)=O)C)cnc2c(C)cccn12 C1(C(=O)NC2CC3CC(C2)N(C(c2cc[nH]n2)=O)C3)CC2CC(O)CC(C1)C2 C(=O)(CC(C)C(F)F)NCC1CCC(C(=O)NC2C(OC)C(O)C2)CC1 N1(C(CC(CNC(=O)CCc2ccncc2)O)=O)CCc2cc(F)ccc21 C12(NC(CN=S(C)(C)=O)=O)CCCC1CN(C(c1cc3cnccc3[nH]1)=O)C2 CCC(C)(CC)C(=O)NC1C=CCN(C(=O)CCc2ccc[nH]2)C1 Cc1ccoc1C(=O)NC(C)(CNC(C1C2COCC12)=O)Cn1cccn1 C(CC(=O)N1CCC1C1CCOCC1)(C(F)F)NC(C1CC(O)(CC#C)C1)=O C1(NC(C(F)OC)=O)CN(C(c2ccn(CCC(F)(F)F)n2)=O)CC1C Cc1c(NC(=O)C(=O)NCCOc2cc(F)ccc2C)cc(C#CCO)cc1Br C1(OC)CC(CNC(c2cncc(F)c2)=O)N(C(c2cscc2F)=O)C1 c1(NC(=O)NC(C2Cc3ccccc3C2)CC)ncc(I)c2c1CCCC2 c1(C(=O)NCC(N(C(Cc2c(C)nc(C)s2)=O)C)C2CC2)ccc2sncc2c1 C=Cn1nncc1C(=O)NC(C)C(C)C(=O)N1CC(O)CC1CO C1(NC(=NC)NCC(c2ccc(C)c(C)c2)OC)CCn2ccnc2C1 C1(CCC(=O)N(CC#C)CC2CC2)CCCCN1C(c1nccn1CC)=O c1(C(=O)NC(CCNC(C(=Cc2cnc[nH]2)C)=O)C)ccc2[nH]c(C)c(C)c2c1 c1(C(N2CCCC(NC(CCCC(C)=O)=O)C(F)C2)=O)cn2cc(Cl)cnc2n1 CC1(C(N2CCCC(NC(c3csc(CO)n3)=O)CC2)=O)CC2CCC1C2 C(C(O)CC(=O)N1CCC(C2CCCCN2C(C2COC2)=O)CC1)N(C)C N1(C(C=C2CCN(C)C2)=O)CC2(NC(=O)COC(F)F)CCCC2(F)C1 c1(C(=O)NC(CC(C)C)CNC(C2COCC2(C)C)=O)ncn2c1CCCCC2 c1(C(=O)NC(C)CCNC(c2cnn(C3CC3(F)F)c2)=O)ccncc1Cl CCC(C(=O)N(C1CC(N(C(=O)C(SC)SC)C)C1)C)OC N1(C(Cc2c(C)ncs2)=O)CCC(F)(CNC(=O)C(N)=O)C1 C12(C(=O)NCC3(CCNC(COCCCC)=O)CC3)CCC(O)(CC1)CC2.C CC(C)(CC#N)NC(=O)NCc1csc(Br)c1 O=C(O)CCCCc1cccc(SCc2cc(-c3ccccc3)ns2)c1 C1(C(N2C(CNC(CC3C(C)CCC3)=O)CC(F)C2)=O)CCC(C)(C)CC1 c1(OC)ccc(C(=O)N(CCCNC(=O)CN2CCCCCC2)C)cc1Cl N1(C(c2cc(C)no2)=O)CC(C2(NC(c3cc(Cl)ccc3N)=O)CC2)C1 C#Cc1cccc(C(N2CC(NC(=O)CCOC3CC3)CC2(CC)CC)=O)c1F n1(C(=O)OC(C)(C)C)cnc2c(C(C)CO)ncnc12.C12(CCCC1)CC(=O)N2C C1(CNC(c2c(Cl)ncc(C)c2)=O)CCC2CN(C(=O)CC(C)(F)F)CCC2C1 c1(CC)ccc(Cl)c(NC(c2cncc(-n3c(COC(=O)OC)ncc3)n2)=O)c1 c1(C(=O)NC2CC(CNC(c3nc(COC)sc3)=O)C2)cnc2ccnn2c1C C(=O)(C(C)S(C)(=O)=O)N1CC(C)C(CNC(c2ccc(=N)[nH]n2)=O)C1 C1(C(=O)NCC(=O)NC(C(C)(C)CO)C2CC2)OCCCC1(C)C c1(C(N2CC(NC(CCC(=O)NC)=O)C(CC3CC3)C2)=O)cc(F)cc(Cl)c1 N1(C(C=CC)=O)CC(=O)N2CCOCC2(CNC(c2cc(S(N)(=O)=O)co2)=O)C1 N1(C(c2c(C3CN(C(C(CCC)F)=O)C3)ocn2)=O)CCCC(O)C1C.C C(C(CC(=O)N(CC(O)CO)C)OC)NC(CN(C1CC1)CC)=O CC(C)CCCC(=O)N1CCCOC(CCNC(c2cccc(Cl)c2O)=O)C1 Nc1cc(C(F)(F)F)cnc1C(N1CC(CNC(=O)Cc2nc(C3CC3)no2)C1)=O C1(NC(CC2C(CNC(C3N(CC)CCCC3)=O)C2)=O)COCCN(C)C1 CCCCC(C)(F)C(=O)N1CC(NC(c2ncoc2CC)=O)C(C)C1 C(=O)(CCCC(C)(F)F)NCCC1(NC(C(COC)N(C)C)=O)CC1 CCC(C(=O)NCC(F)CNC(=O)CNC(C1CCC1)=O)NC(C)=O c1(NC(C23C(CN(c4cc(COC)ncn4)C2)C3)=O)ccc(C(F)(F)F)c(F)c1 CCC(C)CCC(=O)NC(CO)CCCNC(c1nc(Cl)ccc1N)=O C1(CC(N2CC(n3cc(Cn4ncc(C)c4)nn3)C2)=O)CCC(F)(F)CO1 c1(CC)ncncc1C(=O)NCc1cnn(C)c1C(=O)N(C1CCOC1)C1CC1 C(=O)(CC(C)CNC(c1cc(COC)[nH]n1)c1nnnn1C(C)(C)CC)OCC C12(NC(C(C)SCC)=O)CC1CN(C(=O)CSc1ccccc1C)C2 C1(C(=O)NCC(CCOC)NC(C(CC#C)C)=O)CC2CCCC(C1)C2 C(CCCCC(=O)NC(C)CCCNC(=O)C(C1CC(F)(F)C1)O)SC c1(C(=O)NCC(C)CNC(=O)C(c2ccc(F)cc2)C)cccc2ccoc12 C1(NC(C(C)(C)O)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C#N)cc1F CC1(C)NC(=O)N(CC(=O)NC2(C)CCCN(c3nnnn3C3CC3)C2)C1=O c1(CNc2cc(NCc3c(O)nccc3)ncn2)ccn2ccnc2c1 c1(NC(CNC(=NC)NCCSc2ccco2)=O)ccc(Cl)cc1 c1(OC)ccnc(C(=O)NCCN2CCN(C(=O)C(C)C#N)CC2)c1F C1(C(=O)NCC2CN(C(=O)C=Cc3ccc(C)o3)C3CC23)(COC)CCCCC1 C1(C(N(C2CCOC2)CC#C)=O)CCN(C(=O)C2CC3C=CC2C3)O1 c1(C(=O)NCC2(F)CC(NC(C(C)C3CCCC3)=O)C2)cccc2c1CCO2 c1(C(N2CCN(C(c3ccn(C4CC4)n3)=O)CC2CF)=O)cccc2cncn12 N1(C(c2c(C)onc2)=O)CC2CC(NC(=O)C3=NOCC3)C(C2)C1 C=CCC(CC=C)C(=O)NC(C)CN(C)C(C1CCC(NC(C)=O)CC1)=O C1(C(=O)NC2CCCC(N(C(=O)CCOC3COC3)C)C2)CCc2n[nH]cc2C1 C12(CC(=O)NC)CCC1CN(C(=O)C(C)CC(N)=O)C2.ONC(=O)CCOC(C)C C(C(C(=O)NC1CC(SC)C1)N1CCCC1CC(=O)OC)SCC c1(SCC(=O)N(CCCNC(C2C3CCN2CC3)=O)C)nc2ccccc2[nH]1 CC#CCCCC(=O)NC(c1cccnc1)CCC1CCCO1 CCCC(C(=O)NC1CN(C(c2ccc(F)s2)=O)CC1c1cnn(C)c1)C(C)C c1(CC)c[nH]c(C(=O)NCC2CCCC2NC(c2cc(C(C)=O)c[nH]2)=O)c1 c1(C(=O)NCCNC(CC2C(OC)CC2)=O)cc([N+](=O)[O-])c2nsnc2c1 C(=O)(CC(F)(F)C(F)F)NC1C(C)CN(c2cc(C(N)=O)nc(Cl)n2)CC1 c1(NC(c2cc(C)n(-c3ccc(Cl)cc3)n2)=O)cc(NC(N)=O)ccc1F N1(C(c2ccc(C3CCC3)cc2)=O)CC2CN(C(C3CCCC34CC4)=O)CC2C1 C1(NC(=O)CC2CCCC2)CC(NC(c2ccc(CF)cc2)=O)C12CCOCC2 N1(c2cc(NC(CC3=NNC(=O)C3)=O)ncn2)CCC(C2(O)CC2)CC1 C(=O)(CC(O)C(C)CC)N(C1CCN(C(c2cnc(N(C)C)s2)=O)CC1)CCC CN1CCCCC(C(=O)N(C)CC2CCCC2NC(=O)CC(F)(F)C(F)F)C1=O c1(CC)[nH]nc(N2CCC2C(N2CCN(c3ncccn3)CC2)=O)c1F c1(C(=O)NC(CNC(c2cc(CCC)on2)=O)C)ncc([N+](=O)[O-])cc1C C1(NC(C2(CC(=O)OCC)CC2)=O)CCN(C(c2c(C)noc2CC2CC2)=O)CC1 N1(C(CC(C)(C)C)=O)CCC2(C1)CN(C(C1CCC(=O)O1)=O)CCO2 C1(CC)CCOC1C(=O)NC1CCC(CNC(=O)C=C(C)C(F)F)C1 C1(CC=C)CCN(C(c2cnc(C3CCCO3)s2)C(=O)NCC)C1 CC(C)CC(C)(C)C(=O)NC(C1CC(NC(=O)CCC2CCCCC2)C1)C c1(-c2c(OC)cc(F)c(F)c2)ccc2[nH]cc(C(N3CCOC(CO)C3)=O)c2c1 c1(OCCCC)ccc(C(=O)NCC2CC(O)CN2C(C2CC2C)=O)cc1 C1(NC(c2scc(OC)c2)=O)CCCC(C(=O)NC(c2ncc[nH]2)(C)C)CC1 N1(C(CSC)=O)CCC(O)(CCNC(n2ncc(Cl)c2C)=O)CC1 c1(C(N(C)CCN(C)C(c2ccn(C)n2)=O)=O)ccc(Cl)cn1 c1(C(N2C(C(=O)NCC3=C(C)CCC3)CCC2)=O)cccn2nccc12 CC12CCC(C(=O)NC3CC4CC(NC(c5ccoc5)=O)CC34)(CC1)CO2 C#CC1CCCN(C(=O)C(=O)NCC2CN(C(c3nc(Br)cs3)=O)C2)C1 Cc1ccc(C(=O)NC(C2CCCN(C(=O)C3=CC(C)(C)C3)C2)C)nc1C c1(NC(C)=O)ccccc1C(=O)NCCCCC(C)NCCNC(c1cscn1)=O C#CCC(CC#C)C(=O)NC1CC2CCC1N(C(C1CC1CC)=O)C2 CCCCC(CNC(=O)C(F)=C1CCCC1)NC(=O)C(C1CCCC1)OC c1(C(=O)NCC2CC2CNC(C2C3CCC2CC3)=O)ncnc(O)c1Br C1(CNC(c2c(CC)nn[nH]2)=O)CN(C(c2cn(C(C)C)cc2C)=O)CCO1 CC(=O)CCCC(=O)NCCN(C1CCCCCC1)C(C1CC2(CC(=O)N2)C1)=O c1(CCC(N2CCC(CNC(CNC(CCC)=O)=O)C2)=O)ccc2ocnc2c1 C(=O)(CCCC(F)(F)F)N1CC(NC(=O)C(=Cc2c[nH]cn2)F)C(O)C1 N1(C(C(CC=C)N(C)C)=O)CCN(C)C(CNC(=O)C(O)Cc2ccccc2)C1 C1(C(N2C3CC(CN(C(c4cc(C)n(C)c4)=O)C3)C2)=O)CCc2cnn(C)c2C1 c1(CNC(=O)Nc2nc(C)c(C#N)s2)ccc([N+](=O)[O-])cc1Br C12(C(N3CCC(OCC=C)C3)=O)CCC(NC(=O)C(O)C(F)(F)F)(CC1)C2 N1(C(c2cnc(C)[nH]2)=O)CCC(C)C(NC(C23C4CC(CC24)C3(F)F)=O)C1C CC#CCN=c1[nH]c2c(c(=NC(Cc3ccccc3)CCO)[nH]1)COCC2 C1(N(C)C(C2CC(O)C2)=O)CCCC(NC(c2cc(-c3ccco3)no2)=O)C1 c1(C(=O)NCC(C)OC)ccc(C(=O)NCCNC(=O)C(C)OC2CC2)cc1 c1(C(=O)NC2CCC(NC(c3ccc(C)cc3)=O)C2)cccc2[nH]ncc12 C(=O)(CCC=O)OCC.N1(CC)CCCC1CCCO N#CCCCC(=O)N1CCCC1C=CC(=O)NCCN1CCC2CC12 CCCCCCCC(O)CC(=O)N1CCC(O)C(O)C1 N1(C(C(C)(C)C2CCCCO2)=O)CC2CC1CN2C(=O)Nc1ccc(Br)cc1 C12(CNC(C3(CC)CC3(F)F)=O)CC(NC(=O)CC(C)C)C(CO1)C2 N1(CC(C)NC(=O)C(N)Cn2ccnn2)CCN(C)CC1.C1(C2CC2)CCOCC1 c1(NC(C2N(C(c3c(C)csc3)=O)CC(O)C2)=O)c(O)cccc1O N1(C(c2c(C)cn(C)n2)=O)CCC(C(=O)NCC(C)(O)C(F)F)CC1C(C)C N1(C(c2nc(CC)sc2)=O)CCCC2(CC(NC(C3CNC(=O)N3C)=O)C2)C1 C(c1ccoc1)=CC(=O)NC1CC(NC(c2csc(Cc3ccccc3)n2)=O)C1 C(=O)(CCCCCCC(=O)NC1(CNC(=O)Cc2ccoc2C)CCOC1)OC CCCC(C(O)C(=O)NC1CC2CCCC2C1)NC(=O)NC1CC2(CCO1)CC2 N(C1CCOc2ccc(Cl)cc21)C(C12CCN(C(C(C)(C)C)=O)CC1C2)=O CC1CN(C(=O)CN2CC(=O)N(C)C2=O)CCC1N=c1ccnc(C2CCO2)[nH]1 N1(C(c2sccc2Br)C(=O)NCC2CCOC2)CCCC2(CC(O)C2)C1 CCC(C)C(C)C(=O)N(CC(N1CC(F)(C(=O)OC)C1)=O)C1CCC1 C1(C(N(CC(C)(C)NC(CSCC)=O)C)=O)CCN(C(C)=O)C1 c1(CC(N2CCC(CNC(C(C(C)O)N(C)C)=O)C2)=O)c[nH]c2ccccc2c1=O N1(CC(N2CC(O)(CCNC(C(C)C(C)O)=O)C2)=O)Cc2ccccc2C1 n1(CC(=O)NCCC(C)NC(=O)CCc2ccc(O)nc2)ncc2cccnc12 C1(O)(CN(C)C(c2cc(CO)on2)=O)CCN(C(c2cnn(C(F)(F)F)c2)=O)C1 c1(CC)c(C(=O)NCCn2cc(C(=O)NC(c3nc[nH]n3)C)nn2)cnn1C c1(CC(N2C3C(NC(C(C)SC(C)C)=O)C(C3)C2)=O)ccc2[nH]ccc2c1 N1(C(c2c3ccc(OC)cc3[nH]n2)=O)CCC2CN(C(=O)C(C)N(C)C)CC2C1 C#CCC(CC(F)F)C(=O)N1CCC(C)(CCNC(=O)CCCn2cncn2)C1 C(C(C)(C)C(=O)NC(CNC(=O)C(C(C)C)SCc1ccccc1)C(C)C)SC c1(CC(=O)NC2C3(CCN(C(CSCCC#N)=O)C3)C2)ccc2cccnc2c1 c1(N(C2C3CCC2CNC3)C(C(C)(C)OC)=O)nc2c(s1)CCc1ccccc1-2 C1(NC(c2ccon2)=O)CN(C(c2scc3c2CCCC3)=O)CC2(CC2)C1 C12(CNC(c3cnc(C)[nH]3)c3nnnn3C3CC(F)(F)C3)CC(C)(CCO1)C2 CC1CCN(C(c2cc3n(n2)CCC3)=O)C(CNC(=O)CCS(C)=O)C1 Cc1ccc(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)C2CC2)c(Cl)c1Cl Cc1cc(Br)ccc1CN(C1CNCCC1C)c1nc(C2CC2)cs1 c1cc(C)ccc1OC.c1(SCC)cc(C(c2nnnn2C)NCC2CC2)no1 C1(NC(C(Cc2cnc[nH]2)NC(C2N(CC)CCCC2)=O)=O)CCCCC1C#N CCC(CC)C(F)C(=O)N(CC(=O)NC1CCCC1C#N)CC(C)C c1(C(=O)NCC2(NC(=O)C=Cc3ncc[nH]3)CC2)ccc2c(c1)CC2 CC1(C)CC(NC(=O)CN2OC(C)(C)CC2=O)CN(C(=O)CC2(C(F)F)CC2)C1 c1(C(=O)NCC2(F)CC(NC(C(CCSC)O)=O)C2)cccc2c1OC(C)C2 N1(C(c2cc(CSCC)on2)=O)CCN(C(C2(C#N)CC2C)=O)CC12CCC2 c1(OC)ccccc1CNC1CCC(C(=O)Nc2cccc(-n3cccn3)n2)C1 C(=O)(CCC(C)(C)F)NC(C(=O)NCC(C(=O)OCC)C)CCC1CCC1 CC1(CNC(=O)C(F)(F)CO)CCC(NC(=O)C=CSc2nc[nH]n2)C1 CCC1=C(C(=O)N2CCOC(CCCNC(=O)CSC(C)C)C2)CCCO1 C1(NC(C2C(C)(C)C2)=O)CCC2(CCN(C(c3conc3C(F)(F)F)=O)CC2)C1 c1(C(=O)NCCC2CC(NC(c3ccc(C#C)nc3)=O)C2)ccn2cnnc2c1 c1(C(CNC(C(CC)C)=O)NC(=O)CC(=O)N(C)C)cccc(C)c1 Cc1ccc([N+](=O)[O-])cc1-n1cc(CONC(c2ccc(S(C)(=O)=O)nc2)=O)nn1 C(=O)(C(C(C)CC)NC(c1cn(C)c(=O)n1C)=O)NC(CC(=O)OCC)C N1(C(CCC2(C)CC2)=O)CC2CC2C1C(N1CCC(C(=O)C2CC2)C1)=O O=C(C#CC1CCCC1)NCCC1(C(=O)Nn2cnnc2)CCCC1 c1(C(N(C)CC2CCCC(NC(C(F)=CCC)=O)C2)=O)cc(F)c(F)cc1O c1(C(=O)NC2C3(NC(=O)CC4CCCC4)CCC(C2)C3)cc(Cl)c(F)cc1O C12CCN(CC1)C(=O)N(CC)CCCNC2=O.C1(NCCN)CCOCC1 C1(CNC(c2cn(C3CC3)nn2)=O)CN(C(=O)CCC2CC2(F)F)CC12CC2 C1(CC(=O)NC2CC3(C2)CC3NC(=O)C=CCO)Oc2ccccc2NC1=O C(=O)(C1=NOC2(CCOC2)C1)N1CC(C)N(C(=O)CC(F)F)CC1 N1(C(CN(C(C)C)C)=O)CC2(NC(=O)C(C)C3CC3)CCC1CC2 CC1=C(C(=O)N2CCN(C(=O)CCc3ccc(C)o3)CC2C)CCCC1 C(=O)(C1CCCc2nccn21)NCC1=CCN(C(C2CCCN(C(C)=O)C2)=O)CC1 C1(Cc2cn(C3CC(C(=O)NCC4CC(CSC)C4)C3)nn2)CN2CCC1C2 C(CCCCCN=[N+]=[N-])NC(C(CCOCCO)NC(Cc1c(C)ncs1)=O)=O c1(C2C(NC(=O)NCCOCC)C2(C)C)cc(Cl)cc(Cl)c1 C1(N(C(=O)Cc2ccccc2F)C)CN(C(C2(C(C)(C)C)CCC2)=O)CC12CC2 N1(C(Cn2c(C)ccn2)=O)CCOCC1CC(=O)NCCC1(O)CCOC1 C=C(C)CCC(=O)NCCCOC1CCN(C(c2c(C)csc2Cl)=O)CC1 CN1CCN(C(=O)CCNC(C2CC3(CC(=O)C3)C2)=O)C(C2CC2)C1 c1(-n2ncc(NC(=O)NC(c3cnc(Cl)s3)CC)c2)cccc(O)c1 S(=O)(=O)(c1cc(NC2CCCC2)ccc1C)NC(C(c1ccc(F)cc1)OC)C C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(c2cnc[nH]2)=O)CC1O N1(C(c2c(Cl)c(C)n(C)n2)C(=O)NCc2cccs2)CCC2CN(C)CC12 N1(C(C(=Cc2cnc[nH]2)C)=O)CCC(CNC(C2(C(F)F)CCCC2)=O)CC1 CCC1=NOC(C(=O)NCc2c[nH]nc2C(=O)NC(c2cnn(C)c2)C)C1 c1(C(=O)NCC(CNC(C(C)CC(N)=O)=O)C)ccc(O)c2ncccc12 CC1(C)C2CCC1(CCNC(N1CCOC3CCC13)=O)CC2 C(=O)(C#CC1(C(F)(F)F)CC1)N1C(C(CNC(CC(=C)C)=O)(C)C)CCC1 c1(C(NOCCCC(=O)OC)=O)c(CNC(C2CCCC(=O)C2)=O)cnn1C c1(C(=O)NC2CCN(C(c3cccnc3Cl)=O)CC2F)cnc2cc[nH]c2c1 Cc1nc2c(NC3CCC3NC(=O)CCN(C)CCO)ncnc2s1 c1(C2(C(=O)NCC3(CNC(C(CC=C)N(C)C)=O)CC3)CC2)ccc(C)cc1F C#Cc1cnn(CC(N2CC3C(CN(C(=O)CNC(=O)C(C)CC)C)C3C2)=O)c1 Cc1nc(C)n(O)c1C(N1CCCC(CNC(=O)C=Cc2cocn2)C1)=O C1(NC(C(SC)SC)=O)CCN(C(c2ccc(NC(C)=O)cc2Cl)=O)CC1CO c1(C(N(CCCO)C)=O)ccoc1CNC(=O)C=C1CCCCC1 N1(C(C(C)CNC(=O)CCc2ccsc2)=O)CCC2(CCC2)C(O)C1 Cc1nnc(CC(=O)NC(C2CN(C(=O)C(C)(C)C3CCCO3)C2)C)s1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCCC(NC(c2nocc2C2CC2)=O)CC1 c1(NC(c2nnnn2C)CC)ncc(C)cc1S(=O)(=O)N1CC(C#N)C1.N1CCC1 C1(CNC(CC2CC(C)C2)=O)(CNC(=O)CCc2cccn2C)CCOCC1 N1(C(C2N(C(CC(C)(C)O)=O)CC(F)C2)=O)CCCC(O)(C(N)=O)C1 N1(C(CC2CC(SC)C2)=O)CCCN(CCNC(=O)C(F)CC2CCCC2)CC1 C(=O)(C1CCc2c[nH]nc21)N1CC(CC)N(C(c2cc[n+]([O-])cc2)=O)CC1 N1(C(C)=O)Cc2c([nH][nH]c2=NC(=O)C=CSc2cnn(C)c2)C(C)C1 N1(C(CNC(CC)=O)=O)CC2CC1C2CNC(C1CCOC1C)=O N1(C(CC2C(C(=O)OCC)C2)=O)CCCCC(CNC(=O)CCC(C)(C)OC)C1 c1(CC)nc(=NC2CCN(C(=O)CC(C)n3cccn3)CC23CCC3)s[nH]1 n1(C(C)C)c(O)nc(N2CCCN(Cc3nc[nH]n3)CC2)cc1=O CC(C)CCC(F)C(=O)N(C1CC1)CC1CCCN1C(c1ccc2c[nH]nc2n1)=O C1(CNC(C(CC)(C)C)=O)N(C(c2cnc3n2CCS3)=O)CCC1(C)C CCC(C(=O)N1CC(NC(=O)CN2CCOC2=O)C1)N1CCCC1=O c1(C(=O)NCc2nccc(C(=O)Nc3ncc(Br)nn3)c2)nc2ncccn2n1 S(=O)(=O)(c1ccc(C(=O)NC2CC2CNC(C2CC3(CSC3)C2)=O)cc1)NC CCC(C)CCC(O)CC(=O)NCCn1cc(CNS(=O)(=O)C2CC2)nn1 c1(N(C(C)C)C)ccc(CN2CCN(CC(O)C3CC3)CC2)cn1 CCCC(C(=O)N1CC(NC(c2cnoc2CC)=O)C(CO)C1)NC(N)=O N1(C(C)=O)CCCC(O)(CC(N2CCC(NC(c3nccn3C(C)C)=O)C2)=O)C1 C=CCC(C)C(=O)NC(CN(C(c1onc(Br)c1C)=O)CC)CC N1(C(Cn2cc(C(=O)OC)nc2)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1C Cn1nnc2c1CCC(C(=O)NCC1(C)CN(C(c3n[nH]cc3F)=O)CCO1)C2 C1(NC(=O)Cc2c[nH]nc2O)CCN(C(=O)C(C2CCCCC2)F)CC1O c1(OC(CC)C(=O)NC2CC2CNC(c2nccnc2N)=O)cccc(C)c1 CCCC(CC(C)C)C(=O)NCC1(F)CCN(C(=O)CCN2CCN(C)CC2)C1 CCCC(F)(F)C(=O)N1CC(C(=O)NCC2CC3(CC3)C(=O)O2)C2(CC2)C1 N1(C(C(CCC)N(C)C)=O)CCC2CN(C(c3ccc4c[nH]nc4n3)=O)CC2C1 c1(C(N2CCC3(C(NC(C=C(CCC)C)=O)C3)CC2)=O)cc2n(c(=O)c1)CCS2 N1(C(C(C)c2ncco2)=O)CC(NC(C2(C(C)(C)C)CCCCC2)=O)CC1(C)C C(=O)(C(CCC)C(=O)OC)N1C(CC=C)(C(=O)NC2CC(F)C2)CCC1 C1(CNc2c(OCCOC)cncc2)CCCCC1C1CC1 c1(C(C2C3CC4C(C3)C24)=O)ccc(C)c(NC(c2cc(C(C)OC)no2)=O)c1 CCCCCC(C)CC(=O)N(CCC(=O)NC(COC)CO)C1CC1 C(CO)(CCCCNC(=O)CSCc1nccn1C)NC(CN(CCC#C)C)=O c1(OC)ccc(C=CC(=O)NCC23CCC2CN(C(=O)Cc2cn[nH]c2)C3)cc1 CCCC(CC)C(=O)NCCCNC(C12CC(F)(C1)C2)=O CC(C)(CNC(=O)CC1CC2(CC2)CO1)CC(=O)N1CC=CC1C(N)=O Cc1cc(C(=O)NCc2ccc(Br)cc2C(F)(F)F)c(Cl)cc1Cl c1(C(=O)NC2C(CNC(CCSC)=O)COC2)ccccc1CNC1CCC1 CC1CN(C(c2ccn(CC(F)F)n2)=O)CCCN1C(c1cccc(N)n1)=O c1(C(C(=O)NCCCOC)N(C2CCS(=O)(=O)C2)CC)cnc2n1CCOC2 c1(C(=O)NC(CC)CNC(=O)CC2(C#N)CC2)cc(C)c2nc(C)cn2n1 C(=O)(C1Cc2ccc(F)cc21)NCC1CC(NC(=O)CCn2cccnc2=O)C1 c1(C2C(C)C2)ccc(C=CC(=O)NCC2CC(O)CN2C(=O)CC2(C3CC3)CC2)o1 Cc1cc(F)c(Cl)cc1NC(C1CCC(C(=O)Nc2ncc(F)cc2Cl)C1)=O C(CCC(C)CC(=O)NC12CC(C(=O)Nc3nc(Br)ccc3Br)(C1)C2)=C(C)C CCS(=O)(=O)c1ccc(CNCC2CCCN2S(=O)(=O)CCc2cn[nH]c2)cc1 N1(Cc2cccc(OC)n2)CC2CC1CN2C(c1cc(Br)ccc1C)=O C1(NC(c2cc(C)no2)=O)CCSC12CN(C(c1conc1C1CCCC1)=O)C2 CCC(C)CC(C(=O)NC1CC(CC(=O)OC)C1)NC(=O)C1=CC(C)(C)C1 C(CC(C)(C)C)(C(=O)NCc1ncc(C(=O)NCC2(C)CC2(Cl)Cl)cn1)OC c1(C(=O)NCC2(C)CCN(C(CC=CC=C)=O)C2)[nH]c2c(c1C)CCCC2 CCC(CC)CCCC(=O)NCC#CCNC(C1CC2(C1)CC(CO)C2)=O C1(C(N2C(CN(C(=O)Cc3ccon3)CC)CCCC2)=O)CCCC(=O)N1C c1(C(C(C)OC(C)C(C)(C)C)NCc2ccccc2)csc(C)c1C c1(C(=O)NC(CNC(C(c2cn(C)nc2)(C)C)=O)C(C)(C)C)cc([N+](=O)[O-])c[nH]1 C1(NC(C2CC(=O)N2)=O)CN(C(c2cc(F)c(Br)cc2Cl)=O)CCC1(F)F c1(C(N2C3(CNC(C4CCN(C)CC4)=O)CCC3CC2)=O)n[nH]c2ccccc12 CCCCC(O)C(=O)NC1(CC2CCCN2C(=O)C(F)CCC)CCC1 Cc1cc(O)c(F)cc1NC(c1ccc(CNC(c2cncnc2)=O)o1)=O n1(CCCNC(=O)NCCn2cc(Cl)cn2)cc(Br)cn1 N1(C(C(=O)NC(C)CCN)=O)CCN(CCCOc2cccc(Cl)c2)CC1 C(c1ccccc1C(F)(F)F)=CC(=O)NCCCN(C(c1cc(C)no1)=O)CC c1(OCC)cc(CC)ccc1F.c1(C2c3nnnn3N2)ccnc(OC)c1Br CCCCC(C(=O)N(CC(CC)NC(c1ccncc1N)=O)CC)ON=C(C)C C(=O)(CCCCC(N)=O)NC1(C)CCN(C(=O)CC2C(CN=[N+]=[N-])C2(F)F)C1 c1(-c2nccc(C(=O)NC(C3CCOC3)C)c2)c(O)cccc1F c1(C(N(CCC(C)NC(C(CC)OC)=O)C)=O)ccc([N+](=O)[O-])cc1 C1(NC(C(CCOCC)NC(=O)C=C(CC)CC)=O)CN2CCC1CC2 C1(c2onc(C)n2)(Cn2ccnc2C2CC(C)OC2C)CCCCC1 N1(C(C2CCC(COC)C2)=O)CCC2(C1)CN(C(=O)C=Cc1ccn(C)c1)C2 Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(O)C2CCCC2)c2occc2c1 CCCC(CCCNC(=O)CCSCC(C)C)NC(c1ccnc(COC)c1)=O C1(C(=O)NCC2N(C(c3c(N)c(O)nc(O)n3)=O)CC2)C2CC3CC(C2)CC1C3 C1(OC)CCC2(C(=O)NCC3CCCN3C(C3(n4cccn4)CC3)=O)CCC12 c1(C(N2C(CNC(CC(CC)C)=O)CCC2)=O)cc(OC)c2ncccc2c1 Cc1ccc2c(c1)CC(C(=O)NCCCN(C)C(c1cnc3[nH]cncc1-3)=O)S2 N1(C(CC(C)c2cccnc2)=O)CCC(O)(CNC(C2CC=CC(O)C2)=O)CC1 c1(N2CCC(CN(C)C)C2)cccc(S(=O)(=O)N2CCOC(CCF)C2)n1 Cc1c(C(N2CCC(CO)(NC(c3cccc(=O)o3)=O)C2)=O)cnn1C1CCC1 c1(OC)nccc(C(=O)NC2CC(C(=O)NCCOc3ccc(F)cc3)C2)c1Cl Cn1ncc([N+](=O)[O-])c1C(N1CC(NC(=O)CCn2cncn2)CC(C)(C)C1)=O Cc1nn(C)c(Cl)c1C=CC(=O)NCC1COC(CNC(=O)C=CCO)C1 N1(C(CS(CC)(=O)=O)=O)CCCC2(CCN(C(C3CCCC3S(C)(=O)=O)=O)C2)C1 N1(C(C2C(C(C)C)CN(C(C3(C(C)(F)F)CC3)=O)C2)=O)CCC(O)C(C)(C)C1 c1(NC(C2CN(Cc3cscn3)CCC2O)=O)cccc2cccnc12 C1(CNC(COCCSC)=O)CC(C)(C)CN1C(=O)CC1CCNC(=O)C1 c1(C(C)C(=O)NC2(CC(=O)N(C(C)C(N)=O)C)CC2)ccn(C)c1 C1(CNC(Cc2cn(CC)nc2)=O)C(C2CC2)CCN1C(c1cncc(C)c1)=O C1(C2CCCC2)(CNC(=O)C(C2(O)CCCCC2)c2ccc(Cl)s2)CC1 N1(C(C2(C)C(C(=O)OCC)C2)=O)CCC2(CC1)CN(C(=O)CSCCN(C)C)C2 C(=O)(CCCCSC)NC(C1(CNC(c2cc(CCCCC)[nH]n2)=O)CC1)C.C C1(CC=C)(NC(=O)CC2CCC2C2CC2)CCCN(C(=O)CCC(N)=O)C1 c1(C2(C(=O)OC)CC2)csc(=NCc2ccc(OC(F)F)cc2)[nH]1 c1(C(=O)NC(CC(C)NC(C2(SC)CCC2)=O)C)c(C)oc(Br)c1C c1(CCC(=O)NCC2C(CNC(CC(CC)O)=O)CCC2)nc2ncccn2n1 C1(NC(C(C(C)C)O)=O)CN(C(c2ccnc(C(F)F)c2)=O)CC1(C)C CC1(C)C(CC(=O)NC2CCCCCC2)CCN1C(C1CCCOC1)=O CC1C(=O)Nc2cccnc2N1C(=O)NCc1ccccc1C(F)F c1(C(=O)NC2CCC(C(N3CC(O)C(O)C3)=O)CC2)cc(F)c(Cl)c(Cl)c1 c1(OC)cc(C(N2CC(C(C)NC(C3(CO)CCC3)=O)C2)=O)ccc1Cl S(=O)(=O)(c1ccncc1Cl)Nc1c(CC(=O)OC(C)C)cccc1 CCCC(CNC(c1ncn(C)n1)=O)C(=O)NCC(C1CCC1)OCC c1(C(N2CCC(N(C)CCO)C2C)C(=O)NC)nc2c(n1C)CCCC2 c1(OCC)ccccc1C(=O)NC1CCC(NC(c2coc(C)c2)=O)CC1 CCC(C)(C)CC(=O)N1CC(NC(C2C(c3nc(C)no3)C2(C)C)=O)CC1(C)C C1(NC(c2c(OCCC)cccn2)=O)CCC(=O)N(CC(F)(F)F)C1 C1(C(=O)NC2CC(CNC(COCCC#C)=O)C2)OCCC1(C)C N1(C(C2C(C(N)=O)C2)=O)CCC2CN(C(C3(O)CCCC3)=O)CCC12 CCCCN=C(NCc1ccc(OC)cc1CC)NCC1(Cl)CCOCC1 CC(C)C1=NOC(C(N2CCC(C)(CCNC(=O)C(c3cncn3C)=O)C2)=O)C1 CC(F)(F)CCC(=O)N1CCC(NC(c2cnc(C3CC3)cn2)=O)C(O)C1 C(C(C)(C)C(C)(C)C)NC(C1C(CNC(C=CC2(C)COC2)=O)CCC1)=O Cc1n[nH]c(C)c1CNC(=O)C(CNC(C1CCCC1O)=O)CC1CC1 c1(CC)cc[nH]c1C(N1CCC(NC(c2cc(-c3cccs3)on2)=O)C1)=O [N-]=[N+]=NC1(C(N2C3CCC2COC3)=O)CCN(C(=O)C(C2CCOCC2)O)C1 c1(C(=O)NCC(C)NC(c2ccccn2)=O)ccc2cnsc2c1 C1(NC(CN(C(C)=O)C)=O)CN(C(c2cn(C(C)C#N)nc2C)=O)CC1O Cc1cc(C)c(NC(=O)CN2CC(N(C(=O)CCOCC(F)(F)F)C)C2)c(O)n1 C(=O)(C#CC(C)(C)O)N1C2C(C(=O)NCC(C3CCCC3)OC)C(C2)C1 C(=O)(CCCN=[N+]=[N-])NC1CC(CC(=O)NCCc2cc(C)on2)OCC1 c1(C(=O)NC(CCCC)CNC(=O)COCC(=O)OC)cc(F)cc(F)c1 C1(CCC)(C(=O)NCC2CC(CC(=O)NOCCCN(C)C)C2)CC(=O)C1 Cc1ccc(Cl)cc1NC(=O)NC12CC(NCc3cnc(Br)s3)(C1)C2 Cc1cnn(C)c1CC(=O)N(C1CCN(C(=O)COCC2CCCCO2)CC1)C C(=O)(C1CC(=O)N(C)c2ccccc21)NC1CN(C(COC(C)C)=O)CC(C)C1 CC1(C)OC(=O)NC1C(N1CCC1CNC(C1C2CCCCC12)=O)=O c1(C(=O)NC2CCC(CNC(c3c(C)n(C)cc3)=O)C2)cn(C)ccc1=O C1(=O)C(C)(C)C2CCN(C2)C(=O)C2(CC2)N1.C1(CC)CCC1OC c1(NC(CC(=C)C)=O)cc(C)n(NC(=O)OC(C)(C)C)c1C.C12CCN(C1)C2=O Cc1cc(N2CC(=C(F)CNC(C3CCCC34CC4)=O)C2)nc(Cl)n1 CCCCCCC(C(=O)Nc1cccc([N+](=O)[O-])c1)N1CC(C)C(C)C1C Cc1cc(C(=O)NCC2(CCNC(c3c(Br)nnn3C)=O)CC2)c(C)n1C c1(CC(=O)NCCC(CNC(C2=NOC(C)C2)=O)O)ccc2[nH]ccc2c1 C1(C(N2CCC(O)(CCNC(=O)CC3CCCOC3)C2)=O)(CC)CCOCC1 C1(C(N2CCC(COC)(NC(=O)CCSC(F)(F)F)C2)=O)CC2OC1C1CC21 c1(OC)ccc2[nH]c(=NC3CCCC(NC(=O)CCC4CCCO4)C3)oc2c1 C1(OC)(CNC(C2CCN(C)CC2)=O)CCN(C(=O)C=Cc2ccc(C)s2)C1 C(=O)(C1=C(Cl)CCC1)N(CC(CC)NC(c1cc(C)nn1C1CCC1)=O)C C(=O)(C(O)CC(F)(F)F)NC(C1CC=CCC1)C(=O)NCCC(C)(C)C(F)F C(=O)(C1CCc2cc(F)ccc21)NC1C2CCN(C(CC3CC(C)C3)=O)CC21 CC1CN(C(c2ccc(CNC(C3(F)CCCCC3)=O)o2)=O)C(C)C1C N1(C(=O)C=CCNC(C2CC(F)C2)=O)CC2(CCCC2)C1 N#Cc1cc(F)ccc1NC(C12CC1CN(C(c1cc(O)c(O)c(Cl)c1)=O)C2)=O CC1CC(NC(c2ccsc2Br)=O)CCN1C(c1ccccc1F)=O c1(OC)ccc(NCC(C)(C)CNC(C2CC(C)CCN2C(C)=O)=O)cc1Cl N1(C(C2CCCN(C(C3CC4CCC(C3)O4)=O)C2)=O)CCC2COCC2C1 N1(C(C(n2cnc(C#N)n2)C)=O)CCCCC12CN(C(=O)C(C)n1ccnn1)C2 C1(CNC(=O)COCC2CC2)CC(O)C(O)CC1C(=O)NCC(O)CC(F)(F)F c1(C(=O)NC(C(CO)NC(c2cc(CC)c(C)cc2)=O)C)ccc2nccn2c1 Cc1cccc(C(=O)NC2CCC23CN(C(C2COCCO2)=O)C3)c1Cl CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CCN1C(C1SCCCS1)=O C1(NC(=O)NCCc2n(CC)cnn2)CCN(C2CC2)CC1 CC1(C)CN(C(=O)C=Cc2ccc[nH]2)CCN(C(C2CC3(C2)CC(C)(C)C3)=O)C1 C1(O)(C(CNC(C2(C)CSC2)=O)C)CCN(C(c2c[nH]nc2C2CC2)=O)C1 C1(c2cn(N3CC(CS(C)=O)C3)nn2)CCC(F)(F)CC1 C1(NC(C2CCC(C)N2C(c2cccc(Br)c2O)=O)=O)CCCC2CCCCC12 C(=O)(C(C(C)CC)NC(C)=O)N1CC2C(C(=O)CN)C2C1.C1(CCC)(CNC)CC1 c1(CC)nc(CNC(=O)CC(C2CC2)NC(=O)OC(C)(C)C)c[nH]1 C1(C(N(C2CN(C(c3nc[nH]c4nccc3-4)=O)C2)C)=O)CCc2ncnn2C1 CC1(C(=O)NCCCN(C(C2CCOCC2)=O)C2CC2)CCOCC1 c1(C(=O)NCCCCCN(C)C(C2C(C)(C)C2(C)C)=O)cccc(N)c1F N1(C(C(CN(C)C)(C)C)=O)CCCC(N(C(=O)Cn2nnc(C3CC3)n2)C)CC1 C#CC(CC1CCOC1)NC(=O)NCC=C(C)C1CC1 N1(C(C(C)S(N)(=O)=O)=O)CCCC12CCN(C(C1CCC3(CC1)CC3(F)F)=O)C2 C(=O)(C(CCSC)NC(=O)CC1CCCNC1=O)N1CC(C)(COC)C1 N1(CCNC(C(COC)(C)O)=O)CCCN(C(=O)C=C2CCSCC2)CC1 N1(C(C2(C)CCCO2)=O)CCC(CO)C(NC(c2cc3sccc3s2)=O)C1 Cc1nn(CC(N2CC(CCNC(c3[nH]cnc3C#N)=O)C2)=O)c(=O)o1 c1(OC(CC(N2CCC(C(C=O)(C)C)C2)=O)CO)ccc2c(c1)CCC2.CCS N1(C(CN(CC)CC)=O)CC2CCN(Cc3cc(C(=O)O)cc(Br)c3)CC2C1 C12(C(=O)NC(C)CO)CCCC1N(C(c1ncccc1Cl)=O)CC2 C(F)(c1ccccc1)=CC(=O)NCC(C)CNC(C1(C#N)CCC1)=O C(=O)(C(F)(CNC(c1cscc1OC)=O)C(C)C)NC(CC)C(C)(C)C C1(NC(C2(C)CCCCC2)=O)CCN(c2ccnc(C(F)(F)F)n2)CC1O N1(C(c2c(F)ccc(C)c2)=O)CCC2CC1CN2C(c1cccc(F)c1)=O c1(NC(CNC(c2c(OC)cc(OC)s2)=O)C)nccc(C#N)n1 C1(C(=O)NCCN(C(c2cnc(OC)cc2C)=O)CC)CC(C)CC(=O)N1 CC1=C(C(=O)NC2CC(O)CN(C(=O)CCCN3CCCC3)C2)COCC1 C1(C(N2C(C(N(C3CC(CO)C3)C)=O)CSCC2)=O)CCC2(CC1)CC2 CCC(O)CCNC(c1ccc(-c2cccnc2)o1)=O C(=O)(C(F)(F)C1=CCOCC1)NCCCCCNC(C1C(C)C1C1CC1)=O N1(C2CN(C(c3c[nH]c(C(=O)O)c3)=O)C2)CCOCC(O)(C(F)(F)F)C1 N1(C(c2cn(CC)nn2)=O)C(C(N2CC3CCC3(C)C2)=O)CC2CCCC12 C1(C(=O)NC(C(=O)NC(C23CCC(CO2)C3)C)c2ccco2)CC2CCC2C1 C1(CC(=O)NCCN(C(C(n2ccc(C)n2)C)=O)CCCN(C)C)CCCCC1O C1(CNC(C2N(S(C)(=O)=O)CCC2)=O)CCC(CNC(C2CC23CCC3)=O)CC1 c1(NC(C(C2CCOCC2)C)=O)ccc(C(=O)NCC(C)(C)CC2CC2)nc1 C1(CC(N2CC(c3n(C)nnn3)(NCCO)C2)=O)CCc2ncc(Br)n2C1 c1(C(=O)NCC2N(C(C(c3cccc(Cl)c3)C)=O)CC(F)C2)ccc(=O)n(C)n1 C12(NC(CCCOC)=O)CCN(C(=O)Cc3ccncc3Cl)CC1C2 C(=O)(CC(C)C(C)C(C)C)NCC(C)N(C(c1c(OCC#C)nccc1)=O)C c1(C(=O)NC2CC(C)N(C(c3ccc(=O)oc3)=O)C2)cc(F)c2c(c1)CCC2 C1(C(C)O)COCCN1C(=O)CC(CC1CC1)NC(C1C2CCCOC12)=O c1(C(=O)NC(C2CCN(C(=O)CCc3nccn3C)C2)C)ccc(=O)oc1 N1(C(CC2CC(=C)C2)=O)CCCC2CN(C(c3ccc(C(C)C)o3)=O)CCC12 N1(C(Cc2c(OC)nccc2)=O)CCC(CNC(C2CCSC2)=O)C(F)(F)CC1 C(=O)(C1=C(C)OCCC1)N1C(C(NOCC)=O)CC(O)C1.c1ccccc1N C(=O)(CCCC(C)C)NCc1c(C(=O)NCc2c(C)ccnc2)c[nH]n1 C1(NC(C2CCCCO2)=O)CC2CN(C(C34CCCC(CO3)C4)=O)CC2C1 c1(C(CC)OC)ccc(CNC(=O)NCC2CC(F)(CN3CCCC3)C2)cc1 N1(CCN(C(c2cc(C)ns2)=O)C)CCN(C(=O)CC2CC3CCC2C3)CC1 N1(C(CSCCC)=O)CC2CCC1C(CNC(=O)C(N1CCCC(C)C1)=O)C2 C(=O)(CC(C)(C)CCC)N1CCCC(CN(C(C2CCC(=C)CC2)=O)C)C1 N12CC3(CCOCC3)C1c1cn(nn1)CCC2.C1(C=O)CC2(CCCC2)C1 C(C(C)(C)CN(C(=O)Cc1ccn(C(C)C)n1)C1CC1)NC(CN(C(=O)OC)C)=O C(=O)(C1=CCCC1C)NC(C(=O)NC1(CO)CC(OC)C1)Cn1cccn1 c1(CC)cc(N)ccc1C(N1CCC(CCCNC(=O)C2=CC(C)(C)C2)CC1)=O Cc1cc(F)cc(C)c1C(=O)NC1CCN(Cc2ccc(F)cc2Cl)CC1F CCCC(C(=O)NC(CC1CC1)C(=O)NC(C)(C)C(F)(F)F)C(C)C N1(C(CCN(CCC)C)=O)CCOCC1CC(=O)NCC1CC12CC2 c1(C(=O)NCC2(CC(=O)N(CC(C)C)C)CC2)cnn(CCF)c1 N1(C(c2cccc(CC)c2F)=O)CC2CC(NC(C3(F)CC=CCC3)=O)C(C2)C1 C(CC(=O)Nn1cnnc1C)N(C(c1ncnc(C)c1C)=O)CCO c1(C(=O)NCC(C)(C2CC2)NC(=O)COC2CCCOC2)cccnc1N C1(CN(CCC)CCC)CCN(C(c2c(C(C)C)cnn2C)=O)CC1.C(=O)(C(C)O)N CC1CC(C(=O)NC2(CNC(C3(CO)CCCC3)=O)CC2)CCS1(=O)=O c1(-c2ccc(OCCOCC)s2)ccc2[nH]nc(C(=O)NC)c2c1 C1(NC(c2c(C)nco2)=O)CCC12CN(C(=O)C(C)C(=O)N1CCOCC1)C2 c1(NCCSC2CCN(C(C)=O)C(C(=O)O)C2)ccnc2[nH]ncc12 c1(NC(C2CC(C(C)C(=O)O)C2)=O)cc(Cl)cc2c1OCC(=O)N2 c1(C(N(CCCCNC(CC2CC(OC)C2(C)C)=O)C)=O)cc(F)c(Cl)cc1Cl N1(C(CCC(=C)Br)=O)CCC(CNC(c2nccn2C(C)C)=O)C12CC2 Cc1cc(NC(=O)CC(C(F)(F)F)OC(F)F)cc(Cl)c1O N1(CC(=O)NCC(=C)C)CCC(C(=O)NOCCC2CC2)CC1 C1(C(=O)NCC2CN(C(C)=O)C2)(OC)CCN(C(c2cnsn2)=O)C1 CCC(CCC(=O)NC(c1nc(=O)o[nH]1)C)NC(C1CC1(Cl)Cl)=O C1(NC(COC)=O)CCCN(C(c2cc(C)c(C#N)cn2)=O)CCC1 CC1(C)CC(CNC(=O)CNC(c2ccsc2)=O)N(C(=O)C=C(Cl)Cl)C1 C1(CC(=O)Nc2ccc(C)cc2)CC2(C1)CN(C(C1CCCC(C#N)C1)=O)C2 C(C)(CCC(=O)N(C(C)C(N1CC(F)(F)C1CC)=O)C1CC1)SCC C1(NC(c2cccc(-n3cc(C(C=C)(C)O)nn3)c2)=O)CCC2(CC1)CC2 N1(Cc2cc(C)ncc2)CCC(O)(C(N2CCC(C(O)CO)CC2)=O)CC1 N1(C(CC)=O)CCC(C(=O)NC(C2CCN(C(=O)COC3CC3)C2)C)CC1 C1(C(=O)NC2(CNc3nccc(C)n3)CC2)CC2CCCCCCC12 C1(C(=O)OC)CC12CCN(CC(F)(F)CO)CC2 N1(C(=O)CCCC(F)F)CC(C2CN(C(=O)Cn3cc(Br)cn3)C2)C1 CC1(C(=O)NCCC2CC(C(=O)NCc3cccs3)C2)CCCC1 N1(C(C(=Cc2ccccn2)C)=O)CCC2CN(Cc3ccc(F)cc3Cl)CC12 CC(C(=O)N1CCC(CO)(NC(=O)Cn2nnc(C3CC3)n2)C1)C(C)(C)C C(c1ccc(F)c(F)c1)=C(C)C(N1CC2CCC1CN2C(c1cc(Cl)on1)=O)=O N1(C(c2cc(C3CC3)n(C)n2)C(=O)NCCSC)CCc2ncc(C)n2CC1 c1(SCC(=O)NCC(C)(C2CC2)NC(=O)CC2CCC2)cc(F)ccc1F N1(C(c2cnc(SC)nc2)=O)CC2CCC(C1)N(Cc1cc(O)cc(O)c1)C2 C1(NC(CCCC(CC)C)=O)CS(=O)(=O)C2CN(C(=O)C3=COCCC3)CC12 C1(NC(c2cc(C)cc(C)n2)=O)CCN(C(=O)C(C)OCC(C)C)CCC1CO N1(C(C(C)(C)NC(Cc2cc(C)n(C)n2)=O)=O)CCN(C)C2CC12 C1(C2CCOCC2)(C(=O)NCC2N(C(CCSC)=O)CCOC2)CC1(F)F C1(C(=O)Nc2c(C)cccn2)CN(C(=O)C(O)CC(F)F)C(C)(C)C1 c1(N2CCC(C(C)NC(c3csc(C4CC4)n3)=O)CC2)cc(=O)n(C)cn1 N1(C(C=CCC(C)(C)NC(c2cccc(OC)c2)=O)=O)CCCC12CCNC2=O C(=O)(CS(=O)(=O)C1CC1)N1CCC(F)(CNC(C(C=C)O)=O)C1 C1(C(N2CC3CC2(C(N2CCC2(CO)CO)=O)C3)=O)(CC)CC(C)(C)C1 CN1CCCCC1CC(=O)NC1(C(=O)NC2COC(C(F)F)C2)CC(O)C1 N1(C(CSc2n(C)cnn2)=O)CC2CC(CNC(=O)C3=CCCC3)CC1C2 c1(OC)cscc1C(c1nnnn1C(c1noc(C)n1)C)NCC1CCC1 C1(C(=O)NCC=CCNC(c2ccc(C3(C)COC3)o2)=O)CC1C1CCCC1 N1(C(c2ncc(C)cc2F)=O)C2CCC1CC(CNC(C1(CC3CC3)CC1)=O)C2 C1(CN(C(=O)Cc2cn[nH]c2)C)CC(F)CN1C(=O)CCNC(=O)CO c1(C(=O)NC2(C)CN(C(C3(C)CCCC3O)=O)C2)cnc(S(C)(=O)=O)s1 CCCCCCC(C)C(=O)NCCCCc1cn(CCCOC)nn1 C1(C(=O)NC2CC(NC(c3[nH]cc(C(C)=O)c3)=O)C2)CC2(C1)CC2F C(=O)(CC(C)CC)NC(CC)CNC(C1CCN(c2ccnc(Cl)n2)CC1)=O c1(-c2cnc(CC(=O)N(CCN(C)C)C)nc2)ccc(F)c2cccnc12 c1(C(N(C2CCCN(CC(=O)NC3CCOC3)C2)CC)=O)cc(C)cc(F)c1 C1(C(=O)NC(C#C)C(C)(C)C)CC2CC1CN(C(c1cc[nH]c3nccc1-3)=O)C2 C1(C)(NC(C(C)(C)CO)=O)CCCN(C(=O)C(=O)Nc2ncc[nH]2)C1 C(=O)(CS(=O)(=O)CC)NCCC(C)NC(c1ccc(C#C)o1)=O CC(O)(Cn1cc(Br)cn1)C(=O)NCCNC(=O)CCc1nc(O)n[nH]1 Cc1ccc(Cl)c(C(=O)NC2CC2CNC(c2cn(C3CC3)nc2C)=O)c1 c1(C(=O)NCC(CCCC)NC(=O)C(CCC)NC(C)=O)cccc2c1OCO2 C1(CCC)CN(C(=O)CSc2ccccn2)CCN1C(=O)C(F)n1cccn1 c1(OC)cc(C(=O)NCCC(C)N(C)C(=O)OC(C)(C)C)c(F)cc1F C1(C(=O)NCC2(COC)CCC2)CCOCC1NC(=O)C(O)CN(C)C C(=O)(CCS(N)(=O)=O)NCc1c(C(=O)NC(c2ccncc2)C)[nH]cc1 c1(CN(C(c2ncc(-c3c[nH]c(=N)s3)cn2)=O)CC)c(CO)cnc(C)c1O C1(C(=O)NC)CCS(=O)(=O)C12CN(C(c1cccc3oc(C)nc13)=O)C2 C#CC1(C(=O)NCCC(C)(CC)NC(=O)Cc2ccc(C)nc2)CCCC1 CC1CN(C(C2CCC3(CCC3)OC2)=O)CC2(CCOCC2)O1 c1(C(=O)NCCCCC(C)NC(=O)CCc2nc[nH]n2)cnc2[nH]nnc2c1 c1(C(=O)NC2C3CN(C(Cn4ccc(C)n4)=O)C2C3)cc(I)ccc1Cl N1(C(C2(NC(C3SCC(=O)C3)=O)CCC2)=O)CC2CCC(O)C(O)C12 c1(OC)ccc(CNC(=O)C(c2cccnc2)Nc2ncc(C)s2)cc1 CN1C(=O)CCC1C(=O)NC1(CNC(=O)CCCc2cnccn2)CCOCC1 N1(C(C2C(C)(CC)C2)=O)CC2CCN(C(=O)CC3(N(CC)CC)CCC3)C2C1 c1(C(N(CCCNC(=O)CNC(N)=O)CC)=O)ccc(OC(F)(F)F)cn1 c1(NC(CN(CCOCCOCC#C)C)=O)nnc(CC)n1-c1ccccc1C c1(C(C(=O)NCc2cccs2)N(C(C#C)(C)C)C)cscc1Br C1(C)(NC(C(C)C2CCCO2)=O)CCCN(C(c2cc(O)nn2C)=O)C1 c1(OC)cccc(OCC(=O)N(CC(C)N(C)C(c2ccc(C)n2C)=O)C)c1 c1(C(C)=O)nc(N2CC(CC(C)NC(c3csc(Cl)c3)=O)C2)c(F)c(Cl)n1 CCCC(C(=O)NC1CC(CCC(=O)N(C2CN(C(C)C)C2)C)C1)NC(N)=O C(=O)(CCC(CC)CC)N1C(CCC)CN(C(=O)C2=CCN(C)C2)CC1 C1(CCC)CCC(C(=O)NC2CN(C(C3(CO)CC(F)(F)C3)=O)CC2OC)CC1 N1(C(CSC(C)C)=O)CCCC(C2CCN(C(=O)C=CCOCC(F)(F)F)C2)C1 C(C(C(F)(F)F)N1CCN(C(C2CCCSC2)=O)CC1)NC(c1cc(C)[nH]n1)=O C1(C(N(CCC(C)NC(c2cc(F)n(C)n2)=O)C)=O)CC2(C1)CC2(F)F N1(C(C(c2ccc(OC)c(OC)c2)N)=O)CCC2(CCC(=O)NC2)C1 C(CC(C)(C)CC(=O)N(C1CN(C(=O)CCC(=O)N(C)C)CCC1C)C)OC C(=O)(C1CCCc2n[nH]cc21)NC1(C)CC(NC(c2ccncc2)=O)C1 c1(CC)cc(NC(=O)C(C2CCN(C(c3[nH]ccc3C)=O)C2)C)ccc1F C(CCN(C)C(C1CC12CCOCC2)=O)(C(C)(C)C)NC(C(CC)CC)=O C1(COC)(CNC(c2cnnn2C)=O)CCCN1C(=O)CC1CCOC1C C1(NC(C(C(CC)C)O)=O)CC2(CCN(C(c3nocc3C3CC3)=O)C2)C1 N1(C(=O)Nc2c(SCC(N)=O)cccc2)CC(O)CC2(CC2)C1 N1(C(CC2(OC)CCC2)=O)CCN(C(C2CC3CC3C2)=O)C(CF)C1 c1(C(N2CCC(N(C(C(C)=C3CCCC3)=O)C)C2)=O)ccn2ncc(C)c2n1 C12(C(=O)NC(COC)CCOC)CCC(NC(=O)C(C)=CC(C)(C)C)(CC1)C2 Cc1nc(O)ccc1C(N1CCC(C(C)C(=O)NC(c2cnn[nH]2)(C)C)C1)=O C1(CNC(c2cc([N+](=O)[O-])c[nH]2)=O)C(C2CC2)CCN1C(=O)Cc1ccco1 C(CC#CC)(C(=O)N1CC(C)(O)CO1)NC(CCC#CC)=O N1(C(C(C)C2CCCOC2)C(=O)NC2COC2)CC2CCC(C1)N2C CCC(C)(CCC(C)C)C(=O)NC1(CF)CCN(C(c2ccc(Cl)c(O)c2)=O)C1 N1(C(c2cnc(CCCC)s2)=O)CCC2(CCC2NC(C2CC(C)(C)C2)=O)CC1 C(C(CC1CCCC1)C(=O)N(CC(F)Cl)C)NC(C(C)NC(CC)(C)C)=O N1(C(c2c(C)ccnn2)=O)C(CNC(=O)CC2CCCCN2C)CC2CCCC12 N1(C(c2cn(CCC)nc2)=O)CC2(CCCC2)C1C(=O)NC(C)(C)CCCF CCS(=O)(=O)C=CC(=O)N1CCC(NC(=O)C(C)(C)NC(=O)C=COCC)C(C)C1 C1(C(=O)NC2CC2NC(C2(S(C)(=O)=O)CCC2)=O)(COC)CCCNS1(=O)=O C1(CCOC)(NC(c2cc(C3CC3)nn2C)=O)CCN(C(C2(C)CCOC2)=O)C1 c1(C(N(CC(O)CN(C)C(C2(C)CC=CC2)=O)C)=O)cccnc1N C(=O)(C(C)(C)CC(=O)N1CCC(O)(CN(C)C(c2cc(Br)n[nH]2)=O)C1)OCC c1(C(=O)NCC(C2CC2)NC(C(C)(C)OC(C)=O)=O)cccc2c1OCC2C C1(C(N2C(C(N3CCC(C(=O)OCC)C3)=O)CCC2)=O)CC2CCCC2C1 CCC(C(=O)NCC1CCC(C)CN1C(C1CN(C(C)C)C1)=O)C(F)(F)F CC1(C)CNC(=O)c2cc(C(=O)OCc3ncnn3C(C)(C)C)ccc2O1 C1(NC(C2C(C)OCCO2)=O)CCCCN(C(=O)CN2CCSCC2)C1 C(=O)(C(C)(C)CC(F)F)NCC1OCC(CNC(CC2(C=C)CCC2)=O)C1 CN1CC(C(=O)NC2CCC2CNC(C2CC(O)C2)=O)NC1=O c1(C(N2C(CNC(C(C)(C)C(F)(F)F)=O)CCC2)=O)ccc2c(c1)OCCN2 c1(C(=O)NCC(N(C(C(CC)OC)=O)C)C2CC2)ccc2occ(C)c2c1 Cc1oc(Br)cc1C(N1CCC(C)(NC(c2cc(C(F)F)cs2)=O)C1)=O c1(NC(C(Cn2cncn2)NC(Cc2nc(C)[nH]n2)=O)=O)cc(C)c(C)cc1C c1(C(=O)OC)cc(C(=O)NC(CO)C(C)NC(=O)C=CCF)c(F)cn1 c1(C(=O)NC2C(CNC(C3C(OC)C3)=O)CCC2)cnn(C(C)C)c1C C(=O)(CCCCC(C)(C)OC)N1CC(F)(CNC(c2c(CC)con2)=O)C1 C(N=C(NCC(F)F)N1CCC2C(C1)NC(=O)N2C)c1c(N(C)C)nccn1 N#Cc1cncc(C(=O)NC2CC3CCC2(C(=O)NCCC2COCCO2)C3)c1 C(CNC(c1cncc(Cl)c1)=O)(CCCC)NC(CC=C=C)=O c1(OC)c(C(N2CCC3(NC(C45CSC(C4)C5)=O)CC3C2)=O)cc(F)cc1F c1(C(=O)NC2CC(C)N(C(=O)C(=Cc3cccnc3)F)C2)ccnc2ccsc12 c1(OC)ccc2ccccc2c1-c1ccc2[nH]c(C(=O)NCC(=O)NC)cc2c1 N1(C(Cc2c(C)n(C)cn2)=O)CCC(O)(CCNC(C2CCCCCC2)=O)CC1 C(=O)(CCC(=O)N(C1CN(C(=O)C(C)CONC(=O)OC(C)(C)C)C1)C)NC Cn1ccc2ccnc(C(=O)NCC3CC(NC(=O)CNS(C)(=O)=O)C(O)C3)c12 C1(CNC(c2nc(C)[nH]n2)=O)CN(C(C23CCCC2OCC3)=O)CC1(C)C C(C)(CNC(=O)CCC1CC1(Cl)Cl)(CC(C)C)NC(c1ccc(C2(C)CC2)cc1)=O N#Cc1cc(S(=O)(=O)NC2C3CCCCC23)ccc1NC1CCN(CC(F)F)C1 c1(CN(C)CC2CCN(C(c3nccnc3Cl)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 CC(F)CC(=O)NCC1(O)CC(NC(c2c[nH]c(C(F)(F)F)c2)=O)C1 c1(NC2(CCNC(C3CCOC3)=O)CCC2)c[n+]([O-])ccc1[N+](=O)[O-] C12(CNc3cccc(CNCc4n(C)ncc4)c3)CNCC(=O)N1CCOC2 N1(C(C(C(C)C)SC)=O)CC2(C1)CN(C(=O)CCC(=O)NCC1CCCC1)C2 C(CCCCC(=O)NCC(C)(C)CNC(c1nnn2c1CCC2)=O)SC C1(CC(=O)NCC(C)(C2CC2)NC(c2cc(Cl)cnn2)=O)CCCC(C2CC2)O1 N1(C(C(C)(C(C)C)OC)=O)CC(C(=O)NCC(C)(O)CC(C)C)CC(C)(C)C1 c1(C(=O)NC2C(CN(C(C3C(C(C)O)C3)=O)C)CCC2)nn(C)cc1Cl N1(C(c2nccc(C#C)c2)=O)CCC2CCN(C(=O)CCC(C)C)CC2C1 N1(C(c2c(C)cc(F)s2)=O)CCN(C(c2ccc(C#N)o2)=O)CC1C1CC1 C(=O)(C1CCc2cc(F)ccc21)N(C(CNC(c1c(OC)cccn1)=O)C)C N1(C(C2CN(C(C)=O)C2)=O)CCC(C)C(CNC(c2cscc2Cl)=O)C1 c1(CN(C)C(C2(CF)CCC2)=O)cnn2c1CN(C(c1[nH]ncc1C#N)=O)CC2 c1(OC)cc(CO)ccc1C(N1CC2CC2(C(=O)Nc2ncc(C#N)s2)C1)=O Cc1ccc2c(C(=O)NCC(C3CC3)NC(=O)Cn3cccc3)ccnc2c1C CCC(C)CC(=O)NC1CN(NC(c2cc(Nc3nccs3)ccn2)=O)C1 c1(CC)cc(C(N2CC3CC2(CNC(C2CCCN2C(N)=O)=O)C3)=O)cc(O)n1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(N(C(C(C)OCC=C)=O)CCO)CC1 c1(CC(=O)N(C2CC(CO)C2)C)cncnc1O.C12CCCC1C(=O)NC2C c1(C(N(CC(C)(C)NC(c2cccc(N)c2)=O)C)=O)cc(Br)cn1C C12(C(=O)NC(CCCC)CNC(C3CCS(=O)(=O)CC3)=O)CCC(C)(CC1)OC2 N1(C(C2C(C#N)C2)=O)CCN(C2CCCC2NC(c2cc(Br)co2)=O)CC1 C(=O)(C=CS(F)(F)(F)(F)F)N1CC(NC(C(C)c2ccco2)=O)C1 C1CC(O)C(=O)N1.C(C)(CC(=O)NC1CCOC1C)SC C1(NC(=O)C2CC2)CN(C(C2CC(C(F)F)C2)=O)CC12CCOCC2 c1(OC)cncc(C(=O)NCCOCC(N2CC(O)C(O)C2)=O)c1.C1CN1 c1(C(C)C)c(NC(=O)Cn2cc(CCC(C)O)nn2)ncnc1Cl c1(C(N(C(c2cn(-c3cccc(C)c3)nn2)C)C)=O)ccnn2ccnc12 c1(C(=O)NCC2CN(C(c3c(C)nccc3)=O)C2)cc(S(=O)(=O)N(C)C)c(C)o1 c1(NC(c2ccc(OC)c(OC)c2Cl)C)ncnc2c(Br)cc(Cl)cc12 c1(OC)cc2ccc(C(=O)NC(CNC(C3CC3C)=O)C(C)C)nc2cc1OC CC1CC2(CCO1)CCN(C(N1CCCCC(CN)C1)=O)C2 CCC(C(=O)NC(C)C(=O)N1CC(c2ccncn2)C1)N.C(N)=O N1(C(C2OCCC(C)C2)=O)CCC(CNC(c2ncccc2Cl)=O)C(C)C1 c1(CC(C(=O)NC(C(C)O)CO)NC(=O)CCc2cnco2)ccccc1Br c1(C(=O)NC2(CC)CCN(Cc3ccc(OC)cc3)CC2)c(F)ccc(Cl)c1F C(=O)(C(CC(=C)C)OC)NC1CCC(C(N(CC=C)CC)=O)C1 N1(C(C(C)OC2CCOCC2)=O)CCC(NC(c2cc(O)ccc2F)=O)C(O)C1 c1(NC(=O)CNC(C2CCN(C3COC3)CC2)=O)ccc(Br)c(F)c1F C1(CC(N2C(Cc3cn(C(C)(C)C(=O)O)nn3)CCC2)=O)CCCCC1O c1(C(=O)NC2CCC(NC(CCC(C)OC)=O)C2)cc(C)nc(C(F)(F)F)n1 CC(N=c1nc(N2CCNC(=O)CC2)c2ccccc2[nH]1)c1ccccn1 N1(C(C2(C)CC(O)CN2C(=O)CC2CCC2)=O)CCc2nnnn2CC1 c1(NC(C2CC(NCc3c(C(=O)O)cccc3)C2)=O)ncc(I)cc1I n1(CC(=O)NC(C(C)NC(c2cc(C3CC3)[nH]n2)=O)C)ccc2cc(F)ccc12 CC(C)(C)CC(O)CC(=O)N1CC(F)CC1C(=O)NC1CCCCC1(C)C C1(NC(CC2CCN(C(C(CC)O)=O)C2)=O)CCC(=O)NC1(C)C c1(OC)cc(C(=O)NC2CN(C(=O)C(c3ccccc3)C)CC2F)ncn1 C(=O)(C1=CCCCCC1)NC1C(C(=O)NC(c2c(C)n(C)nc2)C)COC1 C1(C(=O)NCC2(C(=O)NC(C(C)(C)C)CO)CCC2)CCCCC(=O)N1 C1(NC(c2c(CC)nns2)=O)CCCN(C(c2sccc2F)=O)CC1 Cc1nn(C)c(C)c1CC(N1CCCC(C)(NC(=O)CCc2nc[nH]n2)C1)=O c1(C(N2CC(CN(C(C(C)SC)=O)C)OCC2)=O)cnc2ccnn2c1 C(=O)(C(C)S(N)(=O)=O)Nc1cc(CNCCn2cc(-c3nc(C)sc3)nn2)n(C)n1 C1(NC(c2c(OC)ncc(C)c2)=O)CN(C(c2ccco2)=O)CC12CCC2 CC(C)C(C(=O)NC1(CCNC(C2(F)CC=CCC2)=O)CC1)c1ccncc1 O=C(CCCCc1ccc(F)cc1)NC1CCN(c2ccccn2)C1 Cc1nc(Br)ccc1NC(c1c(N)cccc1F)=O.C12CC(CN1)CNC2 N1(C(C2(C)CCCNC2=O)=O)CCC2(CCN(C(c3cc(O)ncn3)=O)CC2)C1 C(CCCC(=O)NC(C)CCN(C(=O)Cc1ncc(C)o1)C)OCC C1(CC=C)(NC(c2ccc3c(c2)CC3)=O)CCCN(C(C2CC(C)CO2)=O)C1 N1(C(C2CCC(NC(c3ccoc3Cl)=O)C2)=O)CCC(O)(CO)C1 N(C1CN(C(=O)C(C)S(C)(=O)=O)Cc2ccccc21)C(c1cc(C)c(C)[nH]1)=O CCC(C)C(CC(=O)NC1CCn2nccc2C1)NC(c1cc(C)cc(C)c1)=O C1(NC(CN(C)S(N)(=O)=O)=O)C2CCC1CN(C(c1cccnc1Br)=O)C2 C(=O)(CCC(=O)NC(C)(C)CO)NCCCCC.C1(C#N)(C(=O)NCC)CC1(C)C CC(C(=O)N1CC2CC(N(C)C(c3coc(Br)n3)=O)C1C2)C(C)(F)F N1(C(c2cnc(C)[nH]c2=N)=O)CCC2CC2(C(=O)NCC2(O)CN(C)C2)CC1 C(=O)(C(C)(CC)CCCCCC)NCC=C1CCN(C(C2C(C=C)CC2)=O)CC1 N1(C(CC(C)C)=O)CCc2cc(C(N3CCC(C#N)C3)=O)ccc2C1 c1(C(=O)NCC(CN(C(=O)C=CCF)C)O)ccc(Oc2ccc(F)cc2)nc1 Cc1cc(Br)cn2c3c(nc12)CCN(C(c1ccncc1F)C)C3 C(=O)(C(C)(O)C(F)(F)F)NCC=CCNC(C(c1ccc(F)cc1)CC)=O Cc1cnc(Cl)nc1N1CCC(C)C(NC(c2cnccc2C#N)=O)C1 c1(C(=O)NCC2(C)C(C)CN(C(CC(C=C)CC)=O)C2)ccc2cccnn12 N1(C(CCC(CC)C)=O)CCC(C2(NC(=O)C(COC)N(C)C)CC2)CC1 CCC(C)(C)CCCC(=O)NCC(CCOC)NC(=O)CNC(C1CCCC1)=O C1(C)(C(=O)Nc2cc(C)ncc2)CCCN(Cc2ccc(C(N)=O)cc2)C1 c1(C(=O)NC2CCN(C(c3c(COC)ccs3)=O)CC2)[nH]nc2ncccc12 C1(C(=O)NC(C)C(C)NC(=O)CN2CCC(=O)NC2=O)CCC2(CC1)CC2(F)F N1(C(C2(C)CCCOC2)=O)CC2(CCC2)CC1CNC(c1ncc[nH]c1=O)=O c1(C2(C(=O)NC3C(NC(c4cccc(C)c4)=O)CCCC3)CC2)ccc(C)cc1F CC1(C)CN(C(=O)C2=C(Cl)CC2)CCC1NC(=O)C(C)(C)c1cnccn1 CC1(C)CCC(CNC(C2(Br)CC2)=O)N(C(c2cn3c(n2)CCC3)=O)C1 C1(CNC(=O)C2=CCCC2)CC2(CO1)CN(C(C1CCC(=O)N(C3CC3)C1)=O)C2 C1(CNC(c2c(CC(C)C)n(C)nc2)=O)C(C)CCCN1C(=O)Cc1cnoc1 C1(NC(c2cn(CCC)nc2C)=O)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 CCCC(C)(CC)C(=O)NCC1(O)CC(NC(=O)CSC)C1 C1(N(C(c2n(COC)ncc2)=O)C)CCCC(N(C(=O)C=Cc2cc[nH]n2)C)C1 Cc1noc(C)c1C(C)CC(=O)NCC(=O)Nc1ccc(C(N)=O)cc1 O=C(NNC(=O)c1ccc(Br)cc1)NC1CCN(c2ccccc2Br)C1 C(=O)(C(C)C(O)C(C)C)N1CCC(C(=O)NC2CC3(CCOC3)C2)(SCC)CC1 CC1CC(O)CN(C(C2CC(NC(c3c[n+]([O-])c(C)cn3)=O)C(O)C2)=O)C1 C12(C(N3CCCC(N(C(CN(C(C)=O)C)=O)C)CC3)=O)CCC(=O)N1CCS2 c1(C(=O)NC2CC(C)(NC(C(CC)NC(N)=O)=O)C2)c(OC)c(Cl)cc(O)c1Cl CC1CN(C(c2cc(F)n(C)n2)=O)CCCN1C(C1CCCCC12CC2)=O c1(C(=O)NC2(CNC(CC(CC)OC)=O)CCOC2)cc(Cl)ccc1N c1(SCC)ccc(NC(=O)CN2CC(C(=O)OC)C2)cc1 c1(C(=O)NCC2(F)CC(NC(Cn3c(C)cc(C)n3)=O)C2)ccnc2[nH]cnc12 c1(-n2ncc(CCNC3CCC(CCC(=O)OC(C)(C)C)C3)c2)cccc(Cl)c1 Cc1nccnc1-c1cn(CC(C)(C)CNC(C2CC2n2cncn2)=O)nn1 N1(CCNC(C2(CSC)CC2)=O)CCCN(C(C2C(F)(F)C23CCC3)=O)CC1 c1(SCC)cccnc1C(N1CCC(C(C)NC(C2CCCC(C)C2)=O)CC1)=O N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(C2(NC(C3CC4(C3)CC4F)=O)CC2)C1 C1(CNC(c2cccc(OC)c2F)=O)CCCC2(CCOCC2)O1 n1(COCC)nnc(C(=O)NCC(C)(C)NC(=O)C(C)SC)c1N N1(C(Cc2nc(C)sc2C)=O)CCC2C(CCN2Cc2ncc(C(F)(F)F)[nH]2)C1 N1(C(C=CCOCCOC)=O)CC=CC(NC(c2ccncc2)=O)C1 c1(C(=O)NCC(C(CC)C)O)cc2c(N(C)C)ncnc2n1C N=c1[nH]ccc(O)c1C(=O)NNC(=O)C1CC1 N1(C(C(F)=CCC)=O)CCC(NC(=O)CC2CC3(CCC3)CCO2)C(C)(C)C1 c1(OC)ccc(-c2cc[nH]n2)cc1.c1(C(=O)NC(c2n[nH]cc2)=O)cc(C)n(C)c1 N1(C(=O)NCC2CC2(Cl)Cl)CCC=C(c2ccncc2)C1 Nc1ccc(-c2cn(C3CCCC3NC(c3cnncc3O)=O)nn2)cc1F C1(CCNC(C(C)(C)N(C)C)=O)CN(C(=O)C=Cc2cocn2)CCS1(=O)=O N1(C(C2C(C(C)=O)C2)=O)CCC(C)C(NC(=O)CC2(O)CCOC2)C1C n1(C)cc(CCN(C)C(C2(c3cccs3)CC2)=O)nn1.c1(C(CC)N)ccc(Cl)o1 c1(C(=O)NCC(CC)(C)NC(=O)C(C)CSc2ccccc2)nnn(C)c1C c1(C(=O)NCC2C(C)CN(C(=O)CC3C=NN(C)C3=O)C2)ccc(O)c(Cl)n1 C1(C)(C(N2CC(OC)C2)=O)CN(C(c2nc(Cl)cs2)=O)CC1C C1(F)(C(=O)NCCCS(C)=O)CCCN(C(C2CC(C)(C)C2)=O)C1 Cc1csc(=O)n1CC(=O)NCC1CCCN1C(C1(C(F)F)CCOCC1)=O c1(CC(C)C)nccc(C(=O)NC(C2CCCN2C(=O)CO)(C)C)n1 C1(C)(C(=O)N)CCOCC1.C1(CC)C(C(=O)NCCOCC2CC2)C1C.C1CCO1 C1(NC(c2c(C)nco2)=O)CN(C(C2CCOC2(C)C)=O)CC2(CC2)C1 C(N=c1[nH]cncc1Cl)C1N(C(c2ccc(C(C)(C)C)nc2)=O)CCC1 N1(C(C(C)CO)=O)CCc2ccccc2C1CNC(=O)C(c1cnn(C)c1)O CC1(C)C(NC(=O)CCc2cccc(O)n2)CCN1C(=O)Cc1ccccn1 c1(C(N(CCC(C)NC(c2nccc(OC)c2)=O)C)=O)nccc2cnn(C)c12 c1(NC(C2(F)CCN(C(C(C)NC(C)=O)=O)CC2)=O)cccc2cc(Cl)cnc12 C(=O)(C1COCc2ccccc21)NCC1OCCN(C(CCC=C)=O)C1 CC1(CNC(C2CCCCS2(=O)=O)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)CC1 C(c1ccccc1Cl)=C(C)C(=O)NCC(O)CN(C(=O)C(C)(O)C(C)C)C C1(C(N(CC(=O)NCc2c(OC)nsc2)CC(C)C)=O)CCCCC(=O)C1 C(=O)(CC(CC1CC1)NC(=O)CCCn1cccn1)N(C1CCCC1)CC=C c1(OC)ccc(C(N2CC(N3CCN(C(C4CC4F)=O)CC3)C2)=O)c(F)c1 c1(C(=O)NCCN(C(CC)C)C)coc2c1CN(C(c1ccnnc1)=O)C2 N1(C(c2nccc(C)c2)=O)CC=C(CNC(=O)CC2CCC(C)(C)C2)CC1 C1(NC(c2c(C#N)cn[nH]2)=O)CCCCN(C(c2cc(C(F)F)cs2)=O)C1 C1(CNC(CCC=CC)=O)CN(C(c2cc(C)ccc2O)=O)CCC12CCC2 C(=O)(CC(C)C(=O)NCC1CCCN(C(=O)CC2CC(C)(C)CCO2)C1)OCC N1(C(C(C)n2cccn2)=O)CC2CC(C1)N(C(=O)CCc1cccs1)C2 CCC(C)(CCC(C)C)C(=O)NC1CC2CC1N(C(=O)CCC1CCCCC1)C2 C1(O)(CNC(=O)C2=CCCO2)CCN(C(=O)CC2(C(O)C(F)(F)F)CCC2)CC1 C1(CNC(CC2C(C)CCO2)=O)CCC2(CCC2)CN1C(C1CSCC(=O)N1)=O c1(C(N2CC(NC(c3n(CCC)nc(C)c3)=O)C2)=O)ccc2c(c1)C(=O)NC2 C(=O)(CC1=CCCCC1)NCC(C)(CO)NC(=O)CCC(=O)c1ccccc1 C(=O)(C1=CCCOC1)NCC(CC=C)NC(c1ccc(SC)cc1)=O N1(C(C(C2CC2)OC)=O)CC2(NC(c3cn(C4CC4)cn3)=O)CCCC2(F)C1 CC(C(O)C(=O)NC(C)(CCCl)c1nn[nH]n1)c1ccccc1F C(=O)(CCS(C)=O)NC1C(NC(c2ccc(CCC)[nH]2)=O)CCC1 c1(C(N2C(C)CC(CNC(C3(F)CCC3)=O)CC2)=O)cc(N=S(C)(C)=O)ccn1 C(Cc1ccccc1C(F)(F)F)(CC(=O)N1CCC(O)C1)NC(=O)C1CC1 CCCC(CC)C(C(=O)NCc1cccs1)N(C)Cc1ccccc1.C1C(=O)N1 Cc1cnn2ccc(C(=O)NCCNC(=O)CC(C)c3ccccc3)nc12 C1(C(=O)Nc2nc(COC)oc2)CC(C)CN(C(=O)CC2CCCC2)C1 CCC(CC(=O)N1CC2CC1(CNC(c1cc(C)nn1C)=O)C2)C1CCC1 c1(OC)cc(NC(C2(C)CN(C(=O)C=CC3CCCC3)C2)=O)c2ccccc2n1 N1(C(C2(CC)CCOC2)=O)CC2CC(C1)CN(C(c1nc3c(s1)COCC3)=O)C2 CCC(CCC(=O)N1C2CCC(C2)C1CC(N1CC2CC1(C(F)F)C2)=O)OC CC1CN(C(C2CN3CCC2C3)=O)CC(C(N2CCC(CF)CC2)=O)O1 C(=O)(C#CC(C)(C)CNC(c1ccn(CCC)n1)=O)N1CCC(O)(CC#C)CC1 C1(C(=O)NC2CN(CCC)C(=O)C2)CCN(C(=O)CC2(CO)CC2)CC1(C)C C1(CNC(NCCOCC)=NCCc2cccc(C#N)c2)CC2(CCOCC2)O1 C(=O)(CCC(C)C#N)NCC(CC)NC(c1cnc(-c2cccnc2)s1)=O c1(OC)cc(C(N2CCN(CCCNC(C3C(C)C3(F)F)=O)CC2)=O)cc(C)n1 N1(C(C(N2CCNC(C3CC3)C2)=O)=O)CCCCC1c1ccc(F)cc1 c1(CCC)ncoc1C(=O)N(CCN(C)C(C1CCC(CC)O1)=O)C(C)C c1(SCC)ncccc1NC(=O)CC1CCN(C(c2ccnn2CC2CC2)=O)C1 CC(F)(F)CCCC(=O)NCCC1(CNC(=O)Cc2c(F)cc(F)cc2F)CC1 c1(OC)ccc(C)cc1C(=O)NCC1(CO)CCN(C(=O)C(C(C)C)SC)CC1 C(=O)(CC1=CCN(C)CC1)NC1(CN(C(c2cnc(C)[nH]2)=O)C)CC1 N1(C(c2ccc(F)c(Br)c2F)=O)CC2CCCC(C1)C2C(N1CCC(O)C1)=O N1(C(c2c(C)sc(O)n2)=O)CC2(CCCC2)C1C(=O)NCC1CCC(C)C1 C(=O)(CCC(C)(F)F)NCC(CN(C(C(c1ccc(C)cc1)(C)C)=O)C)C c1(-c2scc(C(C(=O)C(C3CC3)C3CC3)=O)n2)cccc(Cl)c1.C1(C(=O)N)CC1CN C(=O)(CC(C)C(C)(C)C)N(CC(C)O)CCNC(C1CCC(C)(C)CC1)=O C12(CCNC(COc3c(C)cccc3)=O)CCC(C1)N(C(c1ccnn1C)=O)C2 C1(C(=O)NCc2c(C)cccc2)CC(F)(F)CN1C(=O)C(O)CN(C)C CN1CC(NC(c2cn(CCNC(C3(n4nccn4)CC3)=O)cn2)=O)CC12CCC2 C1(CNC(c2ccn(C(F)(F)F)n2)=O)C2CN(C(C3CC3F)=O)CC12 C1(C)(COC)CCN(C(C2CC(O)CN2C(=O)CC2OCCC2(C)C)=O)C1 c1(C(N2CC3(CCC(C(=O)NCC(C)(C)C)O3)C2)=O)cc(F)c2cc[nH]c2c1 N1(C(CCCC#C)=O)CC=C(CNC(c2cnc(C)nc2O)=O)CC1 C1(NC(=O)NC(c2c(C)nc(C)s2)C)CN(C)C(=O)C12CC2 C12(C(=O)NCCCCNC(CCOC(CC(C)C)C)=O)CCCC1C2(F)F c1(C(=O)NCC(N(C(c2ccnc(OC)n2)=O)C)C2CC2)ncc(C#N)cc1C CC1(C)CC=C(C(=O)N2CC3CC2CC3NC(=O)CCC=CBr)CC1 C(=O)(C1CCCc2scnc21)NCC1N(C)CCN(C(C2=C(C)OCC2)=O)C1 N1(C(C2C(=C)C2)=O)CC2CCC(C1)N2C(=O)C(C(C)C)NC(C)=O O=C1CC(C(=O)NCCN(CCOCCO)C(C2CCNC2=O)=O)CN1 CCC(C)(C)C(O)C(=O)N(C)CC1CN(C(c2[nH]nnc2C)=O)CCO1 c1(C(N2CC(CC(C)NC(CC(C=C)C)=O)C2)=O)cncc(O)c1Cl N1(C(C2CCN(OC)CC2)=O)CC23CCCCC2(C1)CN(C(c1ccco1)=O)C3 C1(C)(C(=O)NCCCN(C(=O)CP(C)(C)=O)CC)CC=CCC1 N1(C(CCC(=O)NC)=O)CC2C=CC1C(C(=O)NC1(CCF)CCC1)C2 c1(C(N(CC(=O)NCCN2CC3CC3C2)CCC)=O)ncccc1F c1(C(=O)NC(CC)CNC(=O)C=C(Cl)Cl)ncnc(OC)c1F C(CC(=O)NCC1CCCC(O)C1)(C(F)(F)F)NC(c1c(C)n(C)nn1)=O Cc1cn(C)nc1-c1cn(CCCCCCO)nn1.CC(N)=O c1(CNC(=O)NC(C2CCCCC2)C(C)OC)ccc(F)cc1O c1(C(N2CC(OC)(CNC(=O)CC3CC(C)=NO3)C2)=O)cccc2[nH]nc(O)c12 c1(CC(=O)NC2CCC(n3cc(C(C=C)(C)O)nn3)CC2)nn(C)c(C)c1Cl c1(CC)nn(C)cc1C(=O)N(CC(CC)NC(c1ccnn1C1CC1)=O)C n1(CC=C)ncc2c(O)nc(N3CC(C)(NC(=O)C(C4CC4)SC)C3)nc12 C1(C(=O)NC2CCCC2C(=O)NCCCS(N)(=O)=O)(OC)CCC(C)(C)C1 C1(CCNC(CC(=C=C)C)=O)CN(C(c2ccc(N)c(SC)c2)=O)CC(C)O1 C(CC(O)CNC(=O)CCC=C(C)C)NC(C(C1CCC1)OC)=O c1(OC)ccnc(CN2CCC(NC(=O)C(C)SC)CC2)c1 c1(C(=O)NC2CC(NC(C(N)=O)=O)C2)cnc(-c2ccccc2Cl)nc1 C(COC)(C(=O)NC(c1cnc(C)s1)C)NC(C(=O)OCC)=O c1(CCC(=O)NC23C(NC(C=CC=CC)=O)CC(CC2)C3)cnc2ccccc2c1 c1(C(=O)NCCC(C)(C)NC(C#CC2(CC)COC2)=O)ccc2sc(O)nc2c1 C1(CNC(c2c(N(C)C)cncc2)=O)CN(C(c2cc(Cl)cn2C)=O)CC12CC2 CC1CN(C(=O)Cn2cncn2)CC1NC(c1ccc(O)c(CO)c1)=O c1(C(=O)NC23CCN(C(C(=O)NC4CC4)=O)C2CCC3)cc(F)c(F)c(Cl)c1F c1(CC)nc(=NC(=O)N2CCN(CC(N3CCc4ccccc43)=O)CC2)n(C)[nH]1 C1(CN(C)C(c2c[nH]c(=N)o2)=O)CCCCN1C(c1ccoc1C(F)(F)F)=O S1(=O)(=O)c2ccc(Cl)c(c2)C(=O)N1.N1(C(C)C)CCOC(C(=O)OC(C)(C)C)C1 Cc1c(C(=O)NC2C(C(=O)NC3(C)CC3)C2)ccn1C1CC1.C(C)(C)O C1(CNC(=O)C=CC(F)(F)F)C2CN(C(c3n[nH]cc3F)=O)CC12 N1(C(C(CC=C)OC)=O)CCC2CC2(C(=O)NCc2cccc(C3CC3)n2)CC1 c1(C(=O)OCC)cc(C(N2CCOCC2CNC(C2CCC(=O)N2)=O)=O)[nH]c1C Cc1nc2ccc(C(=O)NCC(CO)NC(=O)CN3CCC3C)cc2s1 N1(C(C2CC(CCNC(C3C(CC)CCC3)=O)C2)=O)CCCC2(CC1)CC2 N1(C(c2ccc(C(C)C)cc2)=O)CC(C(=O)NC2CN3CCC2C3)C2(CC2)C1 N12CC(C3CCCN(C3)CC1=O)C2.CCC(CC)C(=O)NC1CCC(OC)C1 C(CC(CC)C(=O)N1CCCC(NC(=O)C2=CCOCC2)C1)=CC N1(C(C(CC)(C)C)=O)CC(CO)C2(CCN(C(=O)C(C)(C)CSC)CC2)C1 c1(N2CC(C)OC(C(N)=O)C2)ccncc1S(=O)(=O)NCc1cnoc1 C1(CNC(=O)COC2CCCCC2)CCC(SCC)CC1.C12(CCCC1)C(=O)N2 Cc1cccc(CCC(=O)NC(C2CCNCC2)C(N)=O)c1 C1(C)(C(=O)NCC2C(CCN(C)C(=O)OC(C)(C)C)CCCC2)C=CCC(=O)N1 N1(C(c2nc(CCC)oc2)=O)CC2C(NC(=O)C(F)=C3CCC3)C2C1 c1(C(=O)NC(CN(C)C(C2CCC(=O)O2)=O)(CO)CO)cnn2c1CCCC2 C12(C(=O)NCCC3(O)CN(C(Cn4ccc(C)n4)=O)C3)CC(CO1)C2(C)C Cc1oc(Br)cc1C(N1CCC(CNC(=O)C(F)=CC2CC2)CC1)=O CCC(CC)CC(F)C(=O)N1CC(C)(OCC(=O)NCc2cccc(Cl)n2)C1 C(=O)(CCCC(=O)NC(C)(C)C(C)NC(=O)CC1OCCC1(C)C)NC(C)C c1(N2CC(N3C(C(N)=O)CSC3)C2)ccc(C2CC2(F)F)cc1 C1(NC(c2c(C)ocn2)=O)CC2CCC1CN2C(=O)CCCOC(C)C N1(CCCC)C(=S)NC(c2cnn(C(C)C)c2C)C2=C1CC(C)NC2=O c1(C(=O)NCC(CC)NC(C2CC23CCCC3)=O)cc(N)cc(O)c1 C(N=c1[nH]cnc(NCC23CCCC2CCO3)c1C)C1CCN(CCCC)CC1 Cc1noc(C)c1NC(=O)CCC(C)c1ccc(Br)cc1 c1(C(N2CCCC(C(N)=O)CC2)C(=O)NC)cnc2n1CCOC2 c1(OC)cc(C)sc1C(=O)NCC1(NC(=O)CC=CCN(C)C)CCCCC1 c1(C(c2nnnn2Cc2cccs2)NC2(C)COC2)cc(Br)ccn1 C1(NC(C(C)N(c2ccccc2)C)=O)(CF)CCN(C(=O)C=Cc2ccc[nH]2)C1 CC1CN(C(c2cnn3cccnc23)=O)CC(C)N(C(=O)C#CC(C)(C)O)C1 N1(C(C(C)(C)OC(COC(C)C)=O)=O)CC(CN2CCCNS2(=O)=O)CC(F)(F)C1 C1(NC(C2C(C(C)(C)OC)C2)=O)CN(C(=O)CCC2(C)N=N2)CC1CC1CC1 c1(CCC)c(C(N2CC(NC(C3CC(C#N)C3)=O)C2)=O)nnn1C C1(NC(C(C2CCC2)OCC)=O)CN(C(=O)Cc2cnn(C)c2C)CC1C C=CC1(C(=O)N(CC(=O)NCC=CCSC)C2CC2)CCOCC1 N1(C(C2CC(C)(NC(Cn3c(C)cc(C)n3)=O)C2)=O)CCSCC(C)C1 c1(C(N2C3(CN(C(C#C)=O)C3)CC2)=O)cc(Cl)cc2cc[nH]c12 C1(NC(CSC)=O)CCC2(CCCN(C(c3ccc(C#N)c(O)c3)=O)C2)C1 C(c1sc2ccccc2c1Cl)=CC(N1C2CCC1CC(O)C2)=O C12(CC)CC(NC(=O)C(CCNC(=O)CC3CC3C3CC3)OC)(CO1)C2 CCC(CC)C(=O)NC12CC(CNC(c3cnc(C)[nH]3)=O)(C1)C2 N1(C(=O)C(F)(F)OC2CCCCC2)CCCCC1c1ccc(Cl)nc1 c1(C(N)=O)cc(C(=O)NC2CCC(NC(=O)C=Cc3cocn3)C2)ccc1F CC1CN(C(c2ncnn2C)=O)CC1NC(=O)CC1CC(C)OC1C Cc1nc(C(NC2CCCn3ncnc32)=O)c2ccccn12 C1(CNC(C(C)=C2CC2)=O)(NC(c2cc(F)cc(F)c2)=O)CC2CCC1C2 C(=O)(C1CCCc2ncnn21)NC1CN(C(c2ncn(CC)n2)=O)CC1O C1(NC(COCC(=O)NC)=O)CC(O)CN(C(=O)CCCOCCOCC)C1 N1(C(c2nc(OCC)oc2)=O)CCC(CO)C(NC(=O)C(C)=C2CCCC2)C1 C(CC1CCCC1)(C(=O)N1CCC(CO)C1)NC(=O)C=CCN1CCC1 C(=O)(CC(C)(C)C(F)F)NC1(C(N2CC(C(=O)OCC)C2)=O)CC1(C)C N1(C(C(CC)CC2CCCCC2)=O)CCC2CN(C(=O)C3=CCCCO3)C2C1 C(=O)(C1=NOC(CNC(c2cc(C)c(C)nn2)=O)C1)N(C)Cc1n(CC)cnn1 c1(NC(=O)CNC2(C)CCCC2)cnn(CCNC(CN(C2CCSC2)C)=O)c1 c1(NC(C2CCCOC2)CC)cccc2c1OCCC2O Cn1nc(C(=O)NC2CC(CNC(=O)Cc3ccon3)CC2O)cc1O N1(C(C(C=C)C)=O)CC2(C(=O)NCCc3cnc(C)[nH]3)CC1CO2 Cc1nc2[nH]c(C(=O)N(C3CCCN(C(=O)C(O)C(F)F)C3)C)cc2s1 N1(C(CC(c2ccccc2Cl)C)=O)CC(CNC(C2CC2C)=O)CC12CCC2 N1(C(c2c(CC)noc2)C(=O)NC2CCCCC2)CC(C)C(C)C1C CC1(CNC(C23CCC2C3)=O)CCN(C(=O)CCN2CCCCC2=O)CC1 C1(NC(CN(CC)CC)=O)CCOC2(CCN(c3ncnc4c3COC4)CC2)C1 N1(C(C(C)C)=O)CCCCC1C(=O)NCC=CCNC(=O)CCCn1cccn1 c1(C(N2C(CNC(CCCOC(C)C)=O)CC(F)C2)=O)ccn(C)c(=O)c1 C1(NC(c2c(C)cc(F)s2)=O)(CNC(C2CCC(F)C2)=O)CCC(F)(F)CC1 c1(CN2CCC(C(N3CCC4(CCOC4)C3)=O)C(O)C2)ccc2occc2c1 C(=O)(C(CC(F)F)NC(=O)C(O)C1CC1)N(C)Cc1cncnc1 c1(C(=O)NCC2C(C)CCN2C(=O)Cc2csnn2)cnn2c1C(=O)NCC2 CCCS(=O)(=O)C(C)C(=O)N1CCC(NC(c2ccc(S(N)(=O)=O)cc2)=O)C1 c1(C(=O)NCC(CC)NC(C2(F)CCOCC2)=O)cccc2[nH]ccc12 C1(c2nc(C(COC)C)nn2-c2cc(N(C)C)nc(Cl)c2)CN2CCCN1CC2 N1(C(C(CC)SC)=O)CCCC2(NC(=O)C(O)CCn3cncn3)CCCC12 c1(C(=O)NC2CC(C)N(C(=O)CC3CC4(CC4)CO3)C2)cc(=N)[nH]c(=N)[nH]1 Cn1ncc2c(O)nc(=NCC=CCNC(=O)CC3CCCS3(=O)=O)[nH]c12 CC1CN(C(c2cscc2F)=O)C(C)CN1C(=O)C=CCO c1(OC)n[nH]cc1C(=O)NCC1CC1CNC(=O)C(n1ccc(Br)n1)C C1(NC(Cc2c(C)ccs2)=O)CCCCC12CCN(C(=O)C(F)(F)C(C)O)CC2 N1(C(C(C)N2CCC2)=O)CCCC(C)(CNC(=O)CC2CC3CCC2O3)C1 Cc1ccc(O)c(CC(=O)NC2(C)CCN(C(C3(c4cc[nH]n4)CC3)=O)CC2)c1 C(=O)(C(C#N)C(C)C)NC(CN(C(C1(OC)CCCCC1)=O)C)C C=CCCC(C(=O)N(CC(C)(C)C)C)NC(=O)C(C)n1cncn1 CC1(C)CCC(=CC(=O)NCC2CC(NC(=O)Cc3cnoc3)C23CCC3)CC1 C1(C(=O)NCC(CC)(CC)NC(=O)C(C)c2cncs2)CCCCC(=O)N1 Cc1ccc(S(C)(=N)=O)cc1NC(=O)N(C(CO)C(C)C)C Cc1cc(C(=O)N(C(C)CNC(c2ncccc2Br)=O)C)ncc1F c1(OCCCC(=O)NC(C)CN(C(=O)CCc2cc(Cl)no2)C)ccc(F)cc1 c1(C(=O)NC2C(CNC(c3c(C)nn[nH]3)=O)CCCC2)csc(S(N)(=O)=O)c1 c1(C(=O)OCC)ccc2c(OC3CN(C(=O)OCC)C3(C)C)n(C)nc2c1 C1(CC(=O)N(C(c2ccccc2OC(F)(F)F)C(=O)O)C)CCS(=O)(=O)CC1 c1(C(=O)NC2CN(C(C3(C)C(C)C3)=O)CC(O)C2)ccc(F)c(C#N)c1 c1(OC)cnc(CN(C)C(N2CC(N3CCNC(=O)C3)C2)=O)cn1 c1(CCCC(=O)NCCNC(c2ccc(Br)cc2)=O)ccc(F)cc1 CCCCCCCC(=O)N1CCCCC1CNC(c1csc(C)c1Br)=O Cc1c(C(=O)Oc2ccc(CCCF)cc2)oc2c(Cl)cccc12 N1(C(C=CC)=O)CCCC1CNC(C1CC(CCO)C1)=O C1(NC(c2n(CC)nnn2)CC2CCOC2)CCC2(CCCC2)CC1 C1(NC(c2cc(C)on2)=O)COCCN(C(c2cncc(O)c2)=O)C1 C(=O)(C1=Cc2cccc(Br)c2OC1)NC1C(SC)CN(C(=O)CO)C1 c1(C(=O)NCC2(C)N(C(C(C)Cn3ccnc3)=O)CCC2)cccn2nnnc12 C1(CNC(COCCOCC#C)=O)COC(CNC(c2ccn(C(F)F)n2)=O)C1 CC1=C(C(=O)NCC2(C)CN(C(=O)CCn3ccnc3)CC2C)CCC1 c1(C(N2CC(CNC(CCNC(C)=O)=O)C(O)C2)=O)c(C)nn(C(C)(C)C)c1C C1(C(=O)NCC2OCCN(C(c3c(CC(C)C)onc3)=O)C2)CCOC(=O)CC1 C=CC(CCC)CC(=O)N(C1CCN(C(c2cn(C)cn2)=O)C1)CCO N1(C(Cc2ccc(C)o2)=O)CC2CCC2(CCNC(=O)Cc2c(C)cnn2C)C1 c1(C(C(=O)NCCCC)N(CC(C)(C)N(C)C)C)csc(-c2cccs2)n1 C1(NC(=O)C(C2CCCCC2)=O)CCN(C2CC2)CC1 C(=O)(C(C)(C)CCC(=O)NCC1(F)CC(NC(=O)CCC(C)CN(C)C)C1)OC c1(C(=O)NC2C(OC)CN(C(CC=CC=C)=O)C2)cc2ccc(F)cc2nc1O N1(CCCc2onc(C)n2)CCOCC(NC(=O)CC2CCCS2(=O)=O)C1 CN1C(=O)CC(C(C)(C)CNC(c2cc(-c3ccncc3)on2)=O)C1=O Cc1nc(C(OC(=O)C(C)NC=O)OC(C)C)c(C)o1 Cc1ccc(S(=O)(=O)N2CCCC(C(=O)Nc3cc(F)cc(Br)c3C)C2)c(F)c1 N1(C(c2c(C(C)C)cccc2)=O)CCC2(CCCC2C(=O)NCCCCCO)C1 Cn1ncc2c1CCCC2NC(=O)NC1COCCOC1 CN1C(=O)CCCC1C(=O)NCCC1CC(NC(=O)CNC(C2CCC2)=O)C1 c1(OC)cccc([N+](=O)[O-])c1C(N1CC2C(C1)N2C(=O)C(C(C)O)N(C)C)=O CCC(CC)CC(F)C(=O)N1CCN(C)C(C(=O)NC(c2cc(C)no2)(C)C)C1 C1(C(=O)NC(C(C)C)CNC(c2ccnn2CC#N)=O)CCC2CCC1O2 c1(CC(=O)NC(C)CNC(=O)C=CC2CCCC2)ccc2[nH]ccc2c1 c1(N(C(c2cc(C)co2)C(=O)NC2CCOC2)CC#CC)cccc(OCC)c1 C1(CC)CC(C(N2CCCC(CC(N3CCC(C)(C)C3)=O)C2)=O)CCO1 C12(NC(c3cnc(CNC(CC(C)(C)C4CC4)=O)nc3)=O)CCC(CC1)CC2 Cc1c(C(=O)NCCC2CN(C(=O)CCC3CCCOC3)C2)nn2c1CCCC2 CC1(C(=O)NC2CCCC(CNC(c3coc(Br)n3)=O)C2)CCCCO1 C1(OC)CC(CCNC(=O)C(C)CSC(F)(F)F)N(C(=O)Cc2[nH]cnc2C)C1 c1(CC)ccc(C(=O)NC2CC(NC(c3ccc(C(=O)OC)[nH]3)=O)C2)[nH]1 C(=O)(CC(C)CC(C)C)N(CC(CC)NC(c1cnncc1NC)=O)C CCC(CC(=O)N1CCN(C(C2CC(C)(C)CO2)=O)C(CCO)C1)C(C)(C)C N1(C(C2CCN(C(C(CC=C)(F)F)=O)CC2C)=O)Cc2cncnc2C1 C(C(C)(CO)NC(=O)C(CC1CCC1)OC)NC(CN(CCCC)C)=O CCCCCC(O)CC(=O)NC(C(=O)NCCc1cn(C)nc1C)C1(C)CC1 C1(C(=O)NC(C)(C)CCNC(c2cncn2C2CC2)=O)CC2CCC(C1)C2O c1(C2C(C(=O)OCC(C(=O)OC)C)C2)ccccc1F C1(CN(C(=O)CC2(O)CCC2)C)CCN(C(=O)CCc2cc[nH]n2)CC1 N1(C(c2cn(CC)nn2)=O)CCCC(C2(NC(=O)CCC=CC(C)C)CC2)C1 CCCCC(O)C(=O)N1CCSCC1CCNC(c1cccnc1NC(C)C)=O C(N=c1[nH]cc(C#N)c2ccsc12)C1N(C(CSC)=O)CCCC1C N1(C(c2c(NCc3cc(C)[nH]n3)ccs2)=O)CCN2CCCC2C1 CC1(CNC(C2CC2c2ccco2)=O)CC1(F)F c1(C(N2CCC(OCCNC(CC(C)OC)=O)C2)=O)ccc(NC(C)C)nc1 c1(C(=O)NCC(C)N(C(=O)CCc2cccc(O)c2)CC)cccc2c1CCC2 C1(CNC(c2nc(COC)sc2)=O)(NC(c2cn(C)nn2)=O)CC2CCC1C2 C1(NCc2c(C)cc(C(F)(F)F)s2)CC2C=CCC(C1)C2 CCC(CCc1ccccc1)C(=O)NCC(C)(CO)NC(=O)C(C)=C1CCC1 c1(C(N2CCC(NC(COCC)=O)C23CCC3)=O)cncc(P(C)(C)=O)c1 N1(C(CC(=O)NCC)=O)CC2CC1C2CNC(=O)CCC(=O)NC1CCCC1 c1(-c2nnc(C(CC)C)o2)nccnc1C Cc1ccc(C(CNC(C2CCCN2N=O)=O)NC(=O)C(F)(F)c2cscn2)cc1 C1(CC)CCN(C(=O)CS(C)(=O)=O)C(C(=O)NCC2(COC)CCCC2)C1 N1(C(CC(COC(C)=O)(C)C)=O)CCN(C(C2CC3(C2)CC32CC2)=O)CC(C)C1 c1(OCCOC)ccc(F)cc1C(=O)N(C)CCSc1ccccc1 N(C1CCOCc2c(Br)cncc21)Cc1cc(F)cc(OC)c1N N1(C(C(C=C)(C)O)=O)CCC2C1CCCN2C(=O)Cc1ccc(F)c(F)c1 c1(C(=O)OCC)c[nH]c(=NCCCC(C)NC(=O)C(F)C(F)(F)F)nc1C CC1CCCc2ncc(C(=O)NC(C)(C)C(C)NC(=O)CN3CCCC3=O)n21 N1(C(C2C(CC)OCC2)=O)CCOC2(CCCN(c3c([N+](=O)[O-])cnn3C)C2)C1 C(=O)(C1=NOC2(CCC2)C1)NCC(CCNC(c1c(N)cccn1)=O)O C1(C(=O)NCCOCCCN(C(=O)C(C)(C)c2ccccn2)C)(OC)CCCC1 C1(NC(c2c(OC)n(C)nc2)=O)CCN(C(=O)Cc2cn(C)cn2)CC(C)(C)C1 C1(CCN(C(=O)C(C)(C)C2CCOC2)C)CCN(C(c2cn(C)c(O)n2)=O)CC1 N1(C(C2CCC(=O)N2)=O)CCC(CO)(CNC(C2(C(F)(F)F)CCC2)=O)C1 N1(C(COCCCC)=O)CC(C)OC2(CCN(C(C3(CC)CCOCC3)=O)C2)C1 N1(C(C2CC(N(C)C(c3ccsc3C#N)=O)C2)=O)CCC(C)(C2CC2)C1 c1(C(N2CCC(OC)CC2C(F)(F)F)C(=O)NCC=C)csc2cc(Br)ccc12 c1(C(=O)NC2CCN(C(c3cc(SC)oc3C)=O)CC2)ccc2c(c1)OCCO2 c1(NCC(CC)C(C)(F)F)ncc(S(=O)(=O)N(C)Cc2cc(Br)cs2)cc1Cl c1(OC)ccc(S(=O)(=O)N2CC3(CCN3C(=O)Cn3nc(C)cc3C)C2)cn1 C1(NC(C2C(F)(F)C23CCC3)=O)CN(C(=O)C2CC2)CCC12CCC2 c1(CC(=O)NCC(CCNC(CC(C)CF)=O)(C)C)cccc2c1OC(C)(C)C2 C(CC(=O)N(C1(C#C)CC1)C)(C(C)C)NC(C1(CC#C)CCCO1)=O N1(C(C2(C)CSC2)=O)CC(C(=O)NCCC2(C)CCCO2)C(C)(C)C1 CCC(O)C(F)(F)C(=O)NCC(N1CC(O)CC1CC)=O c1(CC)ccc(CC(=O)NC(C)CC(C)NC(=O)C(CC)SC)cc1 C1(NC(CC2C(OC)CC2)=O)CCCC1NC(c1cc(C2CCOCC2)no1)=O C1(C(=O)OC)C2CN(C(=O)C(CCC3CC3)NC(=O)COc3cccnc3)CC12 CC(C)(CCCC(=O)N1CC2(CO)CC2(CO)C1)NC(c1cc(C2CC2)no1)=O C1(NC(C2CCOC2CNC(C2(O)CCOCC2)=O)=O)CC(=O)NC1=O c1(C(=O)NC(C2CN(C(C3CCOC(=O)CC3)=O)CCO2)C)cc2n(n1)CCO2 C(=O)(C1CC(=O)c2ccccc21)NCC1N(C(c2ncc(OC)cc2F)=O)CC1 N1(CCCNC(C(CSC)C)=O)CCN(C(=O)CC2CCC2(C)C)CC1 c1(C(=O)NCCCc2n(C)ncn2)ccnc(O)c1F.C12(F)CCN(C1)C2 C1(NC(C2N(CC)CCC2)=O)CC2(C1)CC2CN(CC(=O)NC)C1CC1 C1(F)(CNC(c2c(C)coc2)=O)CCN(C(=O)CC(C)(C)C)C1 c1(C(=O)NC23CC(CNC(C4CC4(F)F)=O)(C2)C3)csc2ncnc(O)c12 n1(C(c2n(CC(=O)NCC=C)nnn2)NCC=CCl)cc2ncccc2n1 C(C)(CCC(C)(C)C)N(CC(C)C)Cc1ccco1 c1(C(=O)NC2CN(C(c3ccnc(C(C)C)n3)=O)C(C)C2)cc(F)cc(Br)c1O C=CCC(CC=C)C(=O)NCC(CO)NC(c1ccn(C)c(=O)c1O)=O C12(NC(c3ncc(OC)nc3)=O)CCC(CC1)N(C(c1cn(C(C)C)cn1)=O)C2 CCC(C)CC(=O)C(=O)NCCC1(C(N2CC3CC3C3CC23)=O)CCCC1 C1(C(=O)NCC(CN(C(C(CCC)C)=O)CC)(C)C)Cc2nncn2C1 Cc1cc(C(=O)NC2CC(N(C)C(c3nnnn3C)=O)C2)[nH]c1C.C1C(=O)N1 C=CCC(C(=O)NCc1csc(CNC(C2CCN2S(C)(=O)=O)=O)n1)C(C)C C(=O)(CC(C)CNC(c1ncoc1C)=O)N(C1CCCCCC1)CC#C Cc1cccc2nc(N3CCN(Cc4nn(C)cc4Br)CC3)[nH]c12 C1(C(=O)NC2C=CC(C(N(C(CC(=O)OC)C)C)=O)C2)CC(C)(C)CN1C C1(NC(C2(CC(C)C)CCC2)=O)COCC1CNC(=O)CCC1CC1C(C)C n1(CC(=O)NC2CCCC(N(C(c3ccn(CC)n3)=O)C)C2)cnc([N+](=O)[O-])n1 N(C1CCCc2cc(CNC(=O)C(O)C(F)F)ccc21)C(=O)CCC(F)(F)F c1(C(N2CCC(N(C(C3CC(C)CO3)=O)CC)C2)=O)c(OC)ccnc1F N1(C(COCCCOC)=O)CC2CCC1CN2C(=O)C(c1ccc(F)cc1)(C)O c1(OC)cnnc(C(=O)NC2CCC2NC(c2cnn(C3CCCC3)c2)=O)c1 Cc1cc(NCC(F)C2CCC2)c(S(N)(=O)=O)c(F)c1 CCCCCCCCN(C(=O)C(CNC(c1ccc(C)cc1C)=O)C(C)C)C c1(NC(c2csc(C(=O)Nc3ncc(Br)c(O)n3)n2)=O)c[nH]c2nccc-2c1 C1(CNC(C(C)Cn2cccn2)=O)CN(Cc2cccc(Cl)n2)CCC1(F)F C(CCCCC(=O)NC1CC1NC(c1ccc(-c2ccccn2)nc1O)=O)=CC N1(C(CCCCC=C)=O)CC2CN(C(=O)C(F)=C3CCCC3)CCC2(CO)C1 N1(C(=O)NCCC(C(F)(F)F)N2CCOCC2)CCOc2cc(F)cnc21 N1(C(C=COCC)=O)CCC2(NC(=O)C=Cc3c[nH]nc3C)CCCC12 C1(NC(C2C=CC=CC=C2)=O)CC(O)CN(C(C2CC2c2cn[nH]c2)=O)C1 c1(C(N2CCC3(NC(C#CC4(C)CC4)=O)C(CC2)C3)=O)cc(F)cc([N+](=O)[O-])c1 C1(NC(c2cncc(CO)c2)=O)CC(O)CN(C(=O)CCC(F)(F)F)C1 c1(C(=O)NCC(CCNC(CCSC)=O)O)cc2n(n1)CC(C)(C)CO2 C(C(C)CC(=O)NCCCc1cc(C)no1)NC(c1cn(CC)nc1)=O C1(C)(CNC(C(c2cn(C)nn2)NC(C2N(CC)CCC2)=O)=O)CC2CC2C1 c1(C(C)OC)cc(Cl)n[nH]c1=NC(=O)c1cccc(CNC(C)=O)c1 C(=O)(C1=CS(=O)CCC1)NC1CC(CNC(c2ccc(C(N)=O)cc2)=O)C1 N1(C(CCc2cc(C)on2)=O)CCC2C(NC(C3CCCC34CCC4)=O)C2C1 N#Cc1ccc(N2CCC23CN(C(C2CC4(CC(=O)C4)C2)=O)C3)cn1 C#CCC(CC(=O)NCC1(C)CCC1)NC(C1CC(C)(C)CO1)=O c1(NCC(CC(C)C)NC(c2ccns2)=O)ccc([N+](=O)[O-])c(O)n1 N=c1nc(C2CC2)[nH]c(=NC2CCN(C(=O)CCc3cncs3)CC2C)[nH]1 c1(C(=O)NC2CC(F)(CNC(C3C(OCC)C3C)=O)C2)ccc(OC)c(F)c1F C1(NC(=O)C=Cc2ccsc2)CC(NC(c2csc3cncn23)=O)C12CCC2 c1(C(=O)NC2C(C(=O)OCC)CCC2)c(Cl)cnc(OC)c1C Cc1csc(C=CC(=O)NCc2cccc(NC(=O)CNC(=O)OC(C)(C)C)c2)n1 C=CCC(CCCCC)C(=O)N1CCC(CC(C)NC(c2cccnc2)=O)CC1 n1(CCC(=O)NCC(C2CCN(C(C(CC)O)=O)CC2)F)cc[nH]c(=O)c1=O N12CCN(C(=O)C1)C1CCN(CC1)C(=O)C=C(F)C2=O.C1(=CC)CCCCCC1 C12(NC(c3c(CC)nns3)=O)CCC(CC1NC(=O)CCCNC(N)=O)C2 C1(CCC)CCCC1C(=O)NC1(CCNC(=O)CN(C)C2CC2)CC1 Cc1ncc(C(=O)NC2CC(C(=O)N(CCCC(C)O)CC#N)C2)c(=N)[nH]1 C1(C(N2C3CCN(C(CC=C(C)C)=O)CC3CC2)=O)CSC(c2ccccc2)=N1 c1(C(c2nnnn2C2(C)CC2)NC(C(=O)NCC(C)C)C)cc(Cl)cn1C N1(C(C(C)N(C(=O)CSC(F)F)CC)=O)CCC(C(C)F)CC1 CON1CCC(CC(=O)NCCCCCCNC(C2CC23CCCOC3)=O)CC1 C1(CNC(CCSCC(C)C)=O)(OC)CCCN(C(=O)CCC2CCOC2)C1 C#Cc1cnn(C)c1C(N1CC2CC2(CNC(c2sccc2OC)=O)C1)=O N1(C(CNC(C)=O)=O)CC(NCc2ccc(I)c(Cl)c2)C2(CC2)C1 C1(C2CCCOC2)(NC(c2n(C(C)(C)C)nnn2)Cc2ccc(F)cc2)CC1 CCN=c1[nH]c(C)c(C(=O)NC(C)CN(C(=O)C=Cc2cccc(F)c2)C)s1 c1(C(N(CCCCCNC(C2CC23CC3)=O)C)=O)cc(C2CCCC2)nn1C C1(C(=O)NC2CCCCC2)COCCN(CC2CCCC2)C1 N(C(=NCCOC(=O)CC1CC1)NC1CC1)CC(c1cccc(Br)c1)OC C(=O)(CC(OC(=O)C(O)Cc1cn(C(C)C)nn1)OC)OC Clc1c(-c2nc(-c3ccn(-c4ccncc4)n3)no2)sc2ccccc12 Cc1ccc(OCC(N2CCCC(N(C)C(c3cnn(C)c3F)=O)C2)=O)nc1 C12(C(=O)NCCNC(=O)CSCCc3ccccc3)CCCC1OCC2 c1(C(N(C)CC2CCC3(CCCC3)O2)=O)ncnc2c1nc1n2CCOC1 c1(C(N(C2CC(NC(CC3(COC)CC3)=O)C2)C)=O)cc2c(F)c(C)ccc2[nH]1 N1(C(C=C(C)C2CC2)=O)CCC(NC(c2n[nH]c3c2CC2CC32)=O)C(F)(F)CC1 C1(C(N(C2CC(O)C2(C)C)C)=O)CCN(C(=O)C=CC(=O)NCC2CC2)CC1 C(=O)(C1=NOC(C)C1C)NC1(CC=C)CCN(C(c2c(F)ccc(F)c2N)=O)C1 Cc1cc(S(=O)(=O)N2CCCC(N3CCOCC3)C2)n(C2CC2)n1 C#Cc1cncc(C(=O)NCCCCC(C)NC(=O)Cc2conc2C)c1 N1(CCC(N2CC(C(C)NC(CCSCCC)=O)C2)=O)CCCC1=O C12(NC(CC3CCN(C(C)=O)CC3)=O)CCN(C(=O)Cc3[nH]cnc3C)CC1C2 C12(COC)CN(C(c3cncc(N)c3)=O)C(CNC(c3cocn3)=O)(C1)C2 CC1CN(C(=O)Cc2cnnn2C)CCN1C(=O)CC1CC(O)C1(C)C c1(C(N2CCOCC(NC(C(C(C)C)SCC)=O)C2)=O)[nH]c(C)c([N+](=O)[O-])c1C c1(C(N(CCOC)CCNC(=O)C=CC2CCOC2)=O)ccccc1COC c1(CNCC2(C)CCCO2)cncc(-c2ccc(CNS(C)(=O)=O)nc2)c1 C1(NC(C(C2CC2)OC)=O)CC2CC(NC(=O)CNC(=O)CC3CCCC3)C1C2 C1(OCC)(CNC(=O)C(=O)Nc2ccn(C)n2)CCOC1 CCC(C)(C)CC(=O)N1CCC(CC(=O)NCCn2cnc(CO)c2)C1 C1(C)(CC(=O)NCc2ncc(C)[nH]2)CCN(C(=O)C(F)(F)CO)C1 c1(C(=O)Nc2cc(C)c(F)cc2F)cn2cc(-c3ccc(C#N)s3)ccc2n1 C(c1nc(C)c(C)[nH]1)=CC(=O)NC1C(NC(C=Cc2c(C)ccs2)=O)CCC1 C1(CC(N2CC(C)(NC(=O)CCCCc3cnc[nH]3)C2)=O)COC(C)(C)CO1 N1(C(C2C(C#C)C2)=O)CC2(CCCC(C(=O)NCC3(C(=O)OC)CC3)O2)C1 C(=O)(C(CC(C)C)NC(=O)CCc1ccnn1C)Nc1cccc(C)n1 CCCC(C)(O)CC(=O)N(C1CN(C(=O)C(C)(C)Oc2ccc(F)cc2)C1)C C1(NC(CC)=O)CCc2n[nH]c(C)c2C1.c12cc(nc(C(C)C)n1)N1CCN2CC1 C1(C(N2CC(N(C)CC)C2)=O)CC12CCN(C(=O)C(C#N)CC)C2 C1(CN(C)C(C2CC2F)=O)CCCCN1C(=O)CCNC(c1ccccc1Cl)=O N1(C(CC(C=C)CCC)=O)CC(C2CCCN(C(=O)Cc3cn(C)nc3C)C2)C1 N1(C(CN(CC)CC)=O)CCCC2(NC(=O)CCNC(C)=O)CCCC12 CC1(C)CC(=O)OC1CCCO.c1(C(C(=O)O)=O)ccc(O)cc1 C1(NC(CNC(CCC)=O)=O)CN(C(c2cc[n+]([O-])cc2)=O)CCC1C(F)(F)F C(c1ccccc1)=CC(=O)NC(CNC(=O)CNC1CCC1)C1CCC1 C1(F)(C(N(C)CC2N(C(C3C(C)C3C)=O)CCOC2)=O)CC2(CCC2)C1 C1(NC(c2cc(C)on2)=O)CCCCC12CCN(C(c1c(C)nsc1C)=O)C2 C1(C(C)C)CC(C(N2CCC(NC(=O)COC3CCOCC3)C2)=O)CCO1 CC(C)C(C(=O)N(c1ccccc1Cl)C)Nc1ncc(Br)cn1 Cn1ncnc1CCC(N1C(C(=O)NCCC2CC2)CC1C)=O C(=O)(C1=COCCO1)NCC1CCN(C(C2(COC)C=CCC2)=O)C1 N1(C(C(C)OCC2CC2)=O)CCC(O)(C(C)CNC(c2ccoc2C(C)C)=O)C1 N1(C(CC2C(NC(C(c3n(C)cnc3)O)=O)CC2)=O)CC(CO)C2(CC2)C1 N1(C(c2c(C)ncnc2)=O)CC2CC3CC2C1C3NC(C1CCOCC1)=O C(=O)(C1CNC(=O)c2ccnn21)NCC(C)N(C(=O)CCC(=O)NC)CC c1(C(=O)NC2CC(NC(=O)C(CC(F)F)C3CCC3)C2)coc2c(Cl)cccc12 C(=O)(C(=O)N=c1ccn(CCc2ccccc2)[nH]1)N1CCC(CCNC)CC1 C1(C(=O)N(CC(O)Cn2cccn2)CCO)(NC(=O)Cn2cnnn2)CCSC1 c1(C(=O)NC2(CNC(CC(C)n3cccn3)=O)CC2)cc2occc2[nH]1 c1(CC(N2C(C)(CNC(C3C(C)CCC3)=O)CCC2)=O)ccc(F)c(Cl)c1 C(C(CNC(=O)Cc1nc[nH]n1)NC(=O)CCn1cccn1)OC N1(C(C(CC)F)=O)CCC2(CCN(C(c3ccnc(OCCOC)c3)=O)C2)C1 O=C1COC2(CN1)CN(S(=O)(=O)CC1CC(F)(F)C1)C2 CC1CCSC1C(=O)N(C1CN(C(=O)CSc2ccccc2)C1)C N1(C(=O)Cc2cc[nH]n2)CCC2CN(C(C3CC(F)(F)CS3)=O)C2C1 c1(NC(=O)C(F)(F)CC2CCOCC2)cc(N2CCNCC2)ccc1F N1(C(C(CC)CC)=O)CC2CCC2(NC(=O)Cc2cc[nH]n2)C1 c1(N2C(CNC(C3(CC=C)CCC3)=O)C(C)CC2)ccc2nccnc2n1 c1(NC(=O)CC2CCN(C(c3cc(Cl)cc(Cl)c3)=O)C2)ncnc2ncncc12 N1(CC)CCOCC1CC(=O)NC(C)(C)CCNC(=O)Cn1cc(Cl)cn1 N1(C(CN(C)CCO)=O)C2CCC(C2)C1CNC(=O)C=Cc1ccc(Cl)cc1 c1(C(CNC(=O)NC(CC=C)C)(C)O)cccc(Br)c1 C=CC1CN(C(=O)Cc2cnccc2C)CC1NC(c1sccc1CO)=O CC(C)C(O)CC(=O)NC1CC(F)(CNC(c2ccc(-c3csnn3)cc2)=O)C1 c1(CN2CC(C#N)C(NC(=O)C(Cl)(Cl)Cl)C2)c(Cl)ccc(Br)c1F C(=O)(CS(=O)(=O)CC(C)C)NCC(C)NC(c1ccc(OC(F)(F)F)cc1F)=O c1(C(N2CC3CN(Cc4cnc(Cl)cc4F)C3C2)=O)c(F)cccc1I C1(O)(CNC(CC2C(C(=O)OC)CCC2)=O)CCN(C(=O)C2=CSCS2)CC1 CCCC(C(=O)NC1CN(C(C2(C)CCC(=O)C2)=O)C1)C(C)C c1(CC)ccoc1C(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cncs1)C Cc1cncc(CC(N2CC(c3ocnc3CNC(=O)CCC(F)F)C2)=O)c1 C1(=CC(=O)NC(CCOC)CNC(c2cc(F)c[nH]2)=O)CCC(C)CC1 c1(NC(C)CCNC(c2n[nH]cc2Cl)=O)snc(Cl)c1C#N C1(C)(NC(C(C)(C)C2CCCCO2)=O)CCN(CC(=O)NCC2CC(=O)CO2)C1 c1(N(CCN(C)C)CCO)ncc2c(n1)CCCC2=CC(=O)O Cc1cc(C)c(C(N2CC(NC(C3(C)CC3(F)F)=O)C(C)C2)=O)[nH]1 c1(CNC(C2(CC)CCN(C(C3CCC3C(=O)OC)=O)C2)=O)nnn(C)c1C C(C(C)(CNC(=O)OC(C)(C)C)OC)NC(C1C(=C)C1C1(N=[N+]=[N-])CC1)=O N1(C(C2N(C(C(C)NC=O)=O)C3CC(F)C2C3)=O)CCC2(CCCC2)CC1 CC1CCC(NC(=O)CCCCC2CC2)CN1C(c1cnc(N(C)C)s1)=O CC1(C)CN(C(=O)CCc2cnc[nH]2)CC1NC(C1CC1c1cccs1)=O C(CCF)(C(=O)OC)NC(=O)NC1(COC)CCCC1 C1(NC(C(CCC)C)c2nnnn2CC2CCCO2)CN(C)S(=O)(=O)C1 N1(C(c2c(C)con2)=O)CC2CCCC(C1)N2Cc1ccc(Cl)cc1Cl Cc1cc(NC(=O)C(c2csc(C3CC3)n2)Nc2ccc(Cl)cc2Cl)ccc1Br c1(CNC(C2(C)CCCCO2)=O)nc(CNC(C2(C#N)CCOC2)=O)cc(O)n1 C1(CNC(C2CCN(C(C=CC=CC)=O)C2C)=O)CC2(CCC2)CO1 c1(C(=O)NCC(C)CC(=O)NCC(C)(O)C(F)(F)F)cccc(F)c1N c1(C(=O)NC2(c3ccccc3Cl)CCC2)c(O)nnc2c1COCC2 N1(CC(CCCC)=O)Cc2ccccc2SCC1C CN1CCC(C(N2CCC23CN(C(=O)C(Cl)Cl)C3)=O)CC1=O C1(NC(C(C)C2CCC2)=O)CC2CN(C(c3cccc(N4CC=CC4)c3)=O)CC12 C(C(CC(F)(F)F)C1CCCNC1)NC(C(CC)C)=O C1(C(C)(C)C)CCC(C(=O)NC(C2CCCC2)CNC(=O)C(Cl)=CCl)CC1 c1(CC(=O)NCC2(O)CCN(C(c3c(C)ccs3)=O)CC2)cnn2c1CCCC2 N1(CC(=O)NC2CCC2CNC(c2ccc(SC(F)(F)F)o2)=O)CCCS1(=O)=O CC1(C)C=CC(NC(C2CC=CCN2C(=O)CC2CCC(=O)C2)=O)CC1 N1(C(=O)CN2CCc3ccccc32)CCN(C(=O)Cn2cccc2)CC(O)C1 C12(C(=O)NC3CCC(NC(c4csc(C(F)(F)F)n4)=O)C3)CCCC1C2(F)F C(=O)(CC(C(F)(F)F)NC(c1cc(F)cnc1O)=O)NCCCC(C=C)(C)C N1(CCNC(c2ccsn2)=O)CCN(C(C2(C3CCCCO3)CCC2)=O)CC1 N1(C(CC(C(F)F)NC(C(CCC)(C)O)=O)=O)CCOC(C)(C)C1C c1(NCC2N(C(C(C)CCC(C)(C)C)=O)CC2)c(F)cc([N+](=O)[O-])cc1F c1(CN(C)C(c2ccc(NC(c3ccncc3O)=O)nc2)=O)ccccc1Br n1(CC(=O)NCC(CO)NC(C(c2cn(C)nc2)=O)=O)nc(O)ccc1=O C1(c2n(C)ncc2)CC(C(=O)Nc2cccc(CCCN(C)C)c2)CCO1 c1(C(N2CC(C(C)NC(=O)CCC3(C)CC3(F)F)C2)=O)nn(C)c(Cl)c1Cl c1(C(=O)NC(C)CNC(=O)C2=CSCCO2)cc2ncccc2cc1Cl C1(NC(c2cc(N)c(Cl)cc2)=O)CC2CC(NC(=O)CCC(=O)C3CC3)CC2C1 N1(C(=O)NCCCl)CC(N)(CO)C1.C1(N)CCCC1 CC(C)CC(C(=O)NC1CN(C(C2CCC(C)(C)OC2)=O)C1)c1ccccc1 C1(OC)C(NC(C2(CF)CCN(C(c3cc(C(N)=O)co3)=O)C2)=O)CC12CCC2 c1(C(=O)OCC2CN(C(=O)OC(C)(C)C)CC(OC)O2)ccc(F)c([N+](=O)[O-])c1 c1(C(=O)NCC2CC(NC(COC)=O)C2)sc2ccc(F)cc2c1C c1(C(C)C)nccc(C(N2CC(NC(c3ncccc3O)=O)C(C)C2)=O)n1 C(=O)(C(C)(O)CO)N(C(CC)CC)CC(C)Sc1ccccc1 C(C(CC(C)C)C(=O)N1CCC1CNC(c1c(N)ccc(F)c1F)=O)OC N1(C(C(C=C)O)=O)CC(CNC(c2cc3oc(C)cc3[nH]2)=O)CC(C)(C)C1 c1(C(C(=O)NCC(CNC(CCNC(C)=O)=O)C)(C)C)cccc(F)c1 N1(C(C(CC)(F)C(=O)C(=O)C=Cc2nccs2)=O)CCC2(CCC2)C(N)C1.OC c1(C(=O)OC(c2nc(C)[nH]n2)C)ccc(C)c(C)c1N N1(C(c2c(OC)nn(C)c2)=O)CC2=C(C1)CN(C(=O)C(C(C)C)n1cncn1)C2 CC(O)C(C)(C)CN=c1[nH]c2c(c(=NCCCc3cnn(C)c3)[nH]1)COC2 C(=O)(C1=COCCC1)NC1CCC(CNC(C(C)CCO)=O)CC1 CCC(O)(C(=O)NCC1CCN1C(=O)CCNC(C)=O)c1ccccc1 CC1CCCN(C(=O)C(C)(C)C)C1CNCc1ccc(-c2nnc(O)o2)cc1 C1(C(C(=O)NCCN(C(=O)Cc2ncc(C)o2)CC)C)CCC(=O)N1C N1(C(CCC(=C)Cl)=O)C2CCCC1CC(NC(=O)CSc1cccc(C)c1)C2 c1(NC(C(C)NS(CC)(=O)=O)=O)cc2cnc(C)nc2nc1O c1(C(N2CC(NC(C(n3cc(C)nc3)(C)C)=O)C2)=O)ccnc(Cl)c1Cl CCCCCC(O)CC(=O)NCC1C=CCN1C(=O)Cc1ccc(NCC)cc1 C1(CCC)CN(C(=O)C(O)C(C)CC)CCN1C(=O)C(C)CCOC C(CC(C)(C)C#N)(C(=O)NCCCOC(=N)O)N1C(c2cccc(C)c2)CCC1 c1(C(N(CCCNC(CC(C=C)CCC)=O)CC)=O)cncc(P(C)(C)=O)c1 C1(C(N(CC(CC)NC(c2cscc2OC)=O)C)=O)CCCN(C(C)C)C1 C1(CNC(c2c(C)noc2)=O)C2CC1N(C(=O)CSc1ccc(F)cc1)C2 C(C)(C(=O)NCCOCCNC(=O)C(C)c1cc[nH]n1)OCC(C)C C1(CN)CCCCN1S(=O)(=O)Cc1ccc(F)s1 C1(CNC(C=CC(=O)N(C)C)=O)C(C2CC2)CCN1C(C1CCC=CCC1)=O CC(O)(CC(F)F)C(=O)NCCCOCCNC(=O)CSc1cccc[n+]1[O-] c1(CNC(=O)NC(C2CCCCO2)C)ccc2ccc(O)nc2n1 C1(C(=O)NCC(C(=O)NCC2(C)CC(C)=NO2)OC)CCCC2CC12 Cc1cc(Cl)cc(C(=O)NCCN(C(=O)CCN2CCOC2=O)C2CC2)c1C c1(C(N2CC(CCNC(C3OCCC(C)C3)=O)OCC2)=O)ccc2nn[nH]c2c1 C1(COC)CN(C(C2CCN(C(C)=O)C2)=O)CCN1C(=O)CCc1ocnc1C c1(C(=O)NCCCOCCN(C(C(CC)C(C)O)=O)C)cc2cc(Cl)cnc2o1 C(=O)(C1=CCCCO1)N(CC(C)N(C(C(c1cccc(Cl)c1)CC)=O)C)C N1(C(C2(c3cccs3)C(C)C2)=O)CC2CCC1CN2C(=O)CCCC#N O=C(C1=CCCOC1)N1CC(C2CN(C(c3sccc3C3CC3)=O)CCO2)C1 c1(C(=O)OCC)cncc(C=CC(=O)Cn2cnc(C(F)(F)F)c2)c1 CC(C)(C)N1C2=CC=CC=CC(CC(C)CNC(=O)CNC(=O)CC2)NC1=O c1(OC)ccc(F)c(C(=O)NCCCCC(C)NC(C2CCCC2O)=O)c1N N1(C(C(CCCCC)O)=O)CCCC2(CNC(C3(Br)CC3)=O)CCCC12 N1(C(CC2CN(C(C3CC(F)(F)C3)=O)CC23CC3)=O)CCCC(C2CC2)C1 C1(C(=O)NCCC2(OC)CCC2)C(C)CCN1C(=O)CC1CC=CC1 C1(CNC(C2(C(=O)NC)CC2)=O)(NC(=O)CC2CCC2)CCC1 C1(CC)CCN(C(c2csc(C#N)c2)=O)C1CNC(C12CCCC1C2)=O CC(C)(C(=O)N1CC(NC(c2cccc(N(C)C)c2)=O)CC(F)C1)S(C)(=O)=O C(=O)(CCCN=c1nccc[nH]1)N1CC(O)(CNC(C(CC(CC)C)C)=O)C1 N1(C(c2cc(OC)no2)=O)CCC2(CC1)CC2NC(=O)CCC(C)N(C)C c1(C2CN(CC(=O)Nc3ccc(SC)cc3OC)C2)nc(OCC)cc(O)n1 C1(C(N2C(CNC(C(C3CCOCC3)OC)=O)CC(F)C2)=O)CCN(OC)CC1 C1(C)(C(=O)NCC(C)(C(C)C)NC(C(C(C)C)C2CCC2)=O)CCS(=O)(=O)CC1 N1(C(C2(CN(C)C)CC2)=O)CC(NC(c2ccc(C(F)F)cc2)=O)CC1(C)C c1(C(N2CCC(NC(CC(C=C)C)=O)C23CC3)=O)ccc2nc(C(F)(F)F)cn2c1 C(=O)(C#CC1CCCO1)N1CC(CNC(c2cc3ccccc3o2)=O)OCCC1 N1(C(CCOCC)=O)CC2CCC(CNC(c3ccc4nc[nH]c4c3)=O)C2C1 CCC(C(=O)NC(C(=O)NCCCN1CCOCC1)C1CCOC1)C(F)(F)F N1(C(C(C)(C)C(F)F)=O)CC2CN(C(=O)CC3CCCCC3O)CC2C1 N1(C(C)CC(C)(C)C)CCC(O)(Cn2nnnc2-c2ccc(Cl)c(F)c2)CC1 C1(O)(CNC(CNC(C)=O)=O)CCN(C(=O)C=Cc2nnn(C)n2)C1 C(CNC(=O)CN(C(=O)COC)C)(CC)(CC)NC(C1C(=C)C1)=O C(=O)(C(=O)N=c1cc(C)o[nH]1)N1CCC(COC)(CNC(C23CCC2C3)=O)CC1 CC1CCn2c(C(N3CCN(C(=O)C=CCO)CC3CC3CC3)=O)cnc2C1 C1(C(N2CCC(CC(=O)NCC3(N(C)C)CCCC3)C2)=O)CC(C2CC2)=NO1 c1(C(=O)NCC23CCC(NC(C(C)C(F)(F)F)=O)(C2)CO3)ccc2n[nH]cc2c1 C1(C(N2CCN(C(c3ncc(C)cc3F)=O)CC2CO)=O)CCCCN(C)C1=O N1(C(C(C)SCC)=O)CCCC2(NC(=O)C(=O)Nc3cccc(C)c3)CCCC12 C1(CC#C)(C(N2CC(N(C)CC)C2)=O)CCN(C(C2CCCCS2)=O)C1 Cc1c(C(=O)NC2CCN(C(=O)C#CC(C)C)CC2C)sc2ccc(Cl)cc12 c1(CC)cc(=NC(=O)C2CC3(CC3)CN2C(c2cc(C)nnc2O)=O)[nH]n1C CCCCC(CNC(=O)CCCCC1CC1)NC(c1nnc(S)n1C)=O S(=O)(=O)(c1c[nH]c(C(=O)NCC(F)CNC(c2cc(O)n(C)n2)=O)c1)NC c1(C2CCCN(CC(CC#C)O)C2)nc2ccccc2o1 C1(C(=O)NC2CC(F)(CNC(C=CS(C)=O)=O)C2)Cc2ccccc2O1 C(C(C)CCC=C(C)C)(c1n(C(CC)(C)C)nnn1)NCCCSc1cn[nH]c1 C(CCCC(=O)NC(CCc1cn(C2CCOC2)nn1)C(=O)O)N(C(C)=O)C CC1CCC(C)(c2cn(CCCC(=O)N3CCCC3c3ncon3)nn2)C1 Cc1cnn(C)c1C(=O)NCCC1CSCCN1C(=O)CCSC(F)(F)F C#CC1CC2CCC1N(C(C1(CCNC(=O)CCCCC(C)C)CCC1)=O)C2 N1(C(CN2CCC(OC)C2)=O)CCN(CCNC(=O)Cc2cnc(C)[nH]2)CC1 C(C)(CC(=O)NC1(CCC(=O)N2CC(OC(=N)O)C2)CCCC1)=C(C)C c1(CS(=O)(=O)NC2C(C(=O)OC)CC2O)cccc(Br)c1 c1(C(=O)NCCCCCNC(c2c(NC)cc(Cl)cc2)=O)cnn2ncccc12 N#CC1(C(=O)NC2CCC(NC(c3cc(Br)co3)=O)C2)CCC1 CC1(C)COCC1.N(C(=NCC1CC1)NCc1ccccc1)CC1CC=CCC1 C(=O)(C(C)CCC(C)(C)C)NC(CCOC)C(=O)N1CC(CN=[N+]=[N-])C1 c1(C(N2C(CNC(C3N(C)CCC3)=O)CCC2)=O)cccc2ccnn12 N1(C(c2ccc(OCCOC)nc2)=O)CCC(C2CCN(CC(N)=O)C2)CC1 c1(NC(=O)Nc2cccc(SCCCC)n2)c(C)nn(C2CCOCC2)c1C C(=O)(C(CC(F)F)NC(C1CC2(C1)CC21CC1)=O)NC(CN(C)C)CCO C(c1cccc(F)c1F)=CC(N1CC(C2(NC(c3c(C)nn[nH]3)=O)CC2)C1)=O Cn1cc2c(n1)C(C(=O)NCCn1cnc3ccncc3c1=O)CCC2 C(C(=O)NCCCCNC(c1c(C)nnn1C)=O)(C(C)C)SC CC1CC(C(=O)NC(c2ccccn2)Cc2ccncc2)CCS1(=O)=O Oc1cc(C(F)(F)F)ccc1CNc1cccnc1[N+](=O)[O-] N1(C(C(C)Cc2cccc(F)c2)=O)CCC(NC(=O)CCCCCF)C12CCC2 c1(C(=O)NCc2nccc(OCC)n2)c(Cl)ccc([N+](=O)[O-])c1Cl CCCC(C(O)C(=O)NCc1cnc(C)n1CC)NC(=O)C(C)(C1CC1)OC c1(C(N2CCC(NC(C(CCC#C)O)=O)C(C)C2)=O)ccc2nc(O)sc2c1 Cc1c(CN2CCOCC2C(=O)Nc2cc(F)cc(Br)c2)[nH]c2ccccc12 c1(SC(CC(CC)C)C)ccc(OC)c(S(=O)(=O)N2CC(N(C)C)C(C)C2)c1 c1(C(=O)NC2CCC23CN(C(C2CCCO2)=O)C3)nc2cnccc2s1 N1(C(C(C=C)C)=O)CCN(CCN(C(=O)C(C)C2CCCO2)C)CC1 c1(C(=O)NC2C(CNC(=O)OC)CCC2)cccc(NC(=O)CN(C)C(C)C)c1 CCCCC(O)CCC(=O)NCC1CC2CCC1N(C(C1(SC)CC1)=O)C2 CCCCCCCC(C)CNCC1CNC(=O)CO1 C1(CC)(NC(c2cc(C)nn2C)=O)CCCN(C(c2cnc(NC3CC3)s2)=O)C1 C(=O)(C1CCc2ccc(OC)cc21)N(CCNC(=O)C1=CCC1)CC N1(C(CC(=O)N2CCOCC2)=O)CCOC2(CCN(C(=O)CCOC(C)C)C2)C1 C1(CC(=O)NC2(C)CC(NC(c3ncc(F)cc3F)=O)C2)CCC(=O)NC1=O C(C(C(C)C)NC(=O)C=CBr)(c1ccccc1)NC(CCOCC#C)=O Cc1c(C(c2nnnn2C2CCOC2)NC(C)(C)C2(C)CC2)sc2nccn12 C1(C(=O)NC2CCC(NC(c3cc(Cl)sc3Cl)=O)C2)CC2(CCC2)CO1 N1(CC)CCC(NC(c2cc(-c3ccccc3)c[nH]2)=O)C1=O c1(C(=O)OC)cc(C(=O)NC2(C(N3CC(CC4CC4)C3)=O)CC2)n2c1COCC2 N1(C(C#CC(C)C)=O)CC2(CNC(=O)CCC3CCN(C)CC3)CC1CCO2 CC(C)(CCC(=O)NC1CC(NC(c2cnc(C(F)(F)F)s2)=O)C1)[N+](=O)[O-] c1(OC(CC)C)cc(C(=O)N(C)CCN(C)C(c2cc[nH]c2C)=O)ccn1 C=Cn1nncc1C(=O)NCC1(C)CCCC1NC(=O)C(=O)NOC c1(C(=O)NCCC(=C)CNC(c2ccc3c(c2)CC3)=O)cc(=O)c(OC)c[nH]1 C(=O)(C(C)(C1CC1)NC(=O)CN(C(=O)CNC(=O)CC1CCCC1)C)OC C=CCC(CC(C)C)C(=O)N1CC(CNC(=O)CSCC(=O)OC)CC1(C)C c1(CC(=O)N(C(CNC(C2(C(=O)NC)CC2)=O)C)C)cc(C)[nH]n1 c1(C(N2CCC(C#C)(O)C2)C(=O)NC2CCCCC2)ccc2c(C)[nH]nc2c1 CCC(CNC(=O)C(C)Cc1ccc(C)cc1)(CC)NC(C1CCN1S(C)(=O)=O)=O N1(C(C(COCC)n2cc(-c3ccccc3C#N)nn2)=O)CCC(F)(F)CC1 N1(C(CC2(OCC)CC2)=O)CC(NC(c2ccc(N3CCCC3)nc2)=O)C2CC12 C1(NC(C=CC=CCC)=O)CCCCN(C(=O)Cc2ccc(OCC)cc2Cl)C1 N1(C(=O)Nc2cc(C)cc(C)n2)CCOCCC1C1CCOCC1 Cc1c(CC(=O)NC2(C(N3CCC3(C)CCO)=O)CCSC2)cnn1C N1(C(CC=C=C)=O)CCC(C(F)F)(CNC(=O)Cc2ccccc2OC)C1 C1(CN(C(C(CC)=CCCC)=O)CC)CCCCN1C(C1C=CCC1)=O c1(C(c2scc(N3C4C(C4)C3=O)n2)=O)cc(F)ccc1F.c1(CCO)ccc(F)cc1 C1(CN(C)CC)CCN(C(C2(C)CN(C(=O)CC3CCC(C)(C)O3)C2)=O)CC1 c1(C(=O)NC(CCC)CNC(=O)Cc2ccn(C)n2)nccc2cc[nH]c12 C(=O)(C1=CCCN(C2(C(N(CC)OC)=O)CC2)C1)NCCCN(C)C C(=O)(N=c1ccn(CCF)[nH]1)C1OCCN(C(C(C)NC=O)=O)C1 C1(C(=O)NC(C#C)CC(C)C)C2CC3C(C2NC(C2CC(O)C2)=O)C13 N1(C(C(CCF)N(C)C)=O)CCOCC(C(=O)NOCC=CCl)C1 C#CC(CC)(CC)NC(=O)C(C)CN(C)C(c1cccc[n+]1[O-])=O c1(C(=O)OC)ccc(-c2nc(Cc3ccc(F)c(C(=O)O)c3)no2)c2ccsc12 N1(C(c2ccnc(OC)n2)=O)CCOC2CN(C(c3ccc(C)c(C)n3)=O)CC12 N1(C(C2CCCC(NC(CCC#C)=O)C2)=O)CCC(N(C)C)C1(C)C N1(C(c2oc(CC)c(C)c2)=O)CCCC2C1CCCN2C(=O)CN(C)C(C)=O c1(-c2n(C)nc(Cl)c2)nc(C2Cc3ccccc32)nn1Cc1c[nH]nn1 c1(C(=O)NCCC(C)N(C(CC=C(C)C)=O)C)noc2c1CC(C(C)(C)C)CC2 N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCCC(C2CN(c3nnc(C(N)=O)s3)C2)C1 C1(OC)CC2CCC1CC2C(N1CCCC1CN)=O.C(=O)(C(C)C(C)O)C(C)=O C(C(=O)NC(C)(C)C)(C(C)(C)C)n1cc(CN(CC(c2ccc(Cl)cc2)O)C)nn1 C1(C(=O)NCC2CC(C)(C)CN2C(=O)C2=CCCS2)C2CCC1(C)C2(C)C CCC1=C(C(=O)N2C3CN(C(=O)CC(c4ccccc4)N(C)C)CC23)CCCO1 C=C(C)CCC(C)NC(=O)C(C)=CCNC(c1cncc(O)c1)=O c1(C(N2CC(N(C(c3c(C)nc(CC)o3)=O)C)C2)=O)n[nH]c2cc(C)ccc12 c1(C(=O)NCC(CC)(C)NC(=O)CC2=CCCCC2)cnc2n1CCCC2 CC1CN(C(C2CCCC2(C)C)=O)CCC1CNC(=O)CC12CCC(CC1)CC2 C1(NC(C(C)N(C(C2CCC(F)CC2)=O)CC)=O)CN2CCC1(F)CC2 c1(C(=O)NCC2CCCCN2C(C2CC2c2ccccn2)=O)occ2c1CCOC2 n1(COC)cccc(NC(=O)C(CC2CC2)NC(=O)C(c2ccccc2)O)c1=O C1(C(=O)NCC(C)(C)NC(c2cccnn2)=O)CC2C(C1)C2(C)C c1(C(=O)NC2CN(C(c3c(C)noc3)=O)CC3(C2)CC3)cc2c([nH]1)CCCC2=O c1(CNC(=NCC(=C)F)NC(C2CCCO2)C)ccnc2[nH]ccc12 Cc1nccnc1CN1CCCC(C(C)NC(=O)CCC2CCCCO2)C1 N(C(=NCCN1CCC(C)C1)NC1CC(NC(=O)OC(C)(C)C)C1)C(C)C N1(C(CC(COC)C)=O)CCCCC(NC(=O)COc2cccc(OC)c2)CC1 C1(C(C)C)CCc2nc(NC(N3CC(N(C)C)CC(C)C3)=O)sc2C1 N1(C(CCC)=O)CC(NC(c2cccn(-c3cccs3)c2=O)=O)C(C#N)C1 C(c1cccs1)=C(C)C(=O)NC(C)CCN(C)C(C1CCOCC1)=O Cc1ccc(C(=O)NCC2(F)CN(C(c3ccc(Cl)nc3O)=O)C2)cc1CO c1(C(N(C2CN(C(C3=C(C)CC3)=O)CC2F)C)=O)ccc2nc[nH]c2c1 C1(C(=O)NCCC2(O)CCN(C(c3c(C)sc(O)n3)=O)C2)CC(C)CC(C)(C)C1 Cc1cc(CN2CC3CC2CN3C(C2CCCS2)=O)ccc1[N+](=O)[O-] N1(C(C2CC(CC)(CC)C2)=O)CCOCC1CCNC(=O)CCC1CCN(C)C1 c1(OCC(N2CC(NC(c3c(C)nc(CC)o3)=O)C(C)C2)=O)ccc(F)cc1O n1(CC(=O)N(CCC)CCNC(=O)CC2CCOC2)nnc(-c2ccsc2)n1 CC(C)(C)CC(F)C(=O)N1CC(C(=O)NCC2CCC3(CC3)CO2)CC1(C)C C(CC(C)(C)C)(C(=O)NC(c1nn(C)cc1O)C)NC(C(C)=CC=C)=O C(=O)(CCS(C)=O)N(C)CC1CCN(C(c2cncnc2)=O)C1 N1(C(CN(C(C)=O)C)=O)CCC2CCN(C(c3cnn(C)n3)=O)C2C1 C1(N(C)C)CC2(C1)CC2NC(=O)CCn1cc(-c2ccccc2F)nn1 Cc1nc(NCC2CC3(C2)CC(F)(F)C3)cc(=NC(C)c2nccc(O)n2)[nH]1 C1(COC)COCCN1C(C(=O)Nc1ccc(OC)cc1)C1CC1C C(=O)(C1CCc2nccn21)NCCOCCNC(c1ncsc1C(=O)NC1CC1)=O Cc1nnccc1C(=O)N(CCCCCNC(C1NC(=O)CC1C(F)(F)F)=O)C C1(C(=O)NC(CC)CNC(=O)C=C(C)c2cccs2)CCCCC(=O)N1 CC1(C)CCCN(C(=O)CC2NC(=O)NC2=O)C1C(=O)NC1CCn2cnnc2C1 c1(NC(=O)NCC(c2ccc(I)cc2)F)ccc(Br)c(Cl)c1F c1(CN(C(=O)Nc2c(OCC)nccc2)C)cccc(C)c1C c1(C(=O)NCC(C(C)C)NC(C2(C)CC(O)CN2C)=O)c(C(F)F)nn(C)c1C c1(OC)ccc(C(N2CCN(C(=O)CC3CC=CCC3)C(CO)C2)=O)nc1Br c1(C(N2CCC(CN(C(=O)Cc3cccc(Cl)c3)C)C2)=O)cc2cc(Cl)sc2[nH]1 N1(C(C(CC)Sc2ccccc2)=O)CCC2CCN(C(=O)C(F)(F)CC)CC12 CC(O)C(C(=O)NCC1(C(=O)Nc2ccc(CCF)cc2)CC1)N(C)C Cc1nn(C)cc1CC(N1CC(CC(C)NC(c2cc(C(F)F)ccn2)=O)C1)=O C12CCC(CC1)NC2=O.c1(OC)cc(C(=O)NCC(n2ccnn2)C)on1 CC1CC2(CC(NC(C3CC3CNC(c3ccncc3O)=O)=O)C2)C1 C12(CC)CN(C(=O)CC3CCC4CC34)C(CNC(c3c(F)cccc3Cl)=O)(C1)C2 CCCCC(CC(=O)N1CCOCC1CC(C)C)NC(c1ccc([N+](=O)[O-])[nH]1)=O N1(C(CC=C=C)=O)CCC2(CC1)CN(C(c1ccc(C)cc1)=O)C2 c1(C(N2CCOCC(NC(c3c(C)coc3C)=O)C2)=O)ccc(C)c(Cl)c1N N1(C(c2ccc(OC)c(Cl)c2Cl)=O)CC2CCCN(C(c3ccsc3)=O)C2C1 c1(C(N2CC3CCN(C(C(C)OCC)=O)C3C2)=O)cc2c(nc(C)n2C)[nH]1 c1(C(=O)NCCN(C)C(c2ncn(C)n2)=O)csc(Br)c1Br CN1CC2(CCC2)CCC1CNC(C1(C)CCNC1=O)=O c1(C(N2CC3C(NC(CNC(=O)OC)=O)(CCC3)C2)=O)[nH]c2ccccc2c1Cl C1(NC(=O)CC2CCCC2)CCN(C(C2(F)C3CCCC23)=O)CC1 N1(C(C(C)C(=O)N2CCOCC2)=O)CC2(CCN2C(=O)COc2ccn(C)c2)C1 C(=O)(CCCC(C)(C)C)N1CC(C(=O)Nc2c(-c3cn(C)nc3)cccc2)SCC1 CC1(CNC(C2CC3CCCC3C2)=O)CCN(C(=O)CN2CCCCC2=O)CC1 N=c1cc[nH]cc1C(N1CCCC(NC(=O)C(C2CCOCC2)O)C1)=O Cc1cc(=NCc2ccc(Cl)cc2C)[nH]c(=NCCC2CC(C)(C)CO2)[nH]1 CC1CN(C(C2CC23CC3)=O)CCN1C(c1ccc(O)c(F)c1)=O N1(C(C(N2CCC(C=C)C2)=O)=O)CCn2c(Br)cnc2C1 N1(C(C(C)CSC(F)(F)F)=O)CC2(CCCN(C(C3(F)CC3C)=O)C2)C1 c1(C(c2n(CCCSC)nnn2)NCC2(F)CC2)ccc(C)c(I)c1 C(=O)(CCC(=O)N(C)C)N1CCC(CCC(=O)NC(C)C2CC2)C1 CC1(C)CC(CNC(=O)CCNC(N)=O)CN(C(=O)CCn2cc(Cl)cn2)C1 C1(C(=O)NC(C)CN(C)C(c2ccc3oncc3c2)=O)CCC(S(N)(=O)=O)CC1 C1(NC(c2c(C)cccc2)=O)CCCN(C(=O)CCc2ccsc2)C1C C1(C2CCC2)(CNC(CC(=O)N(C)C)=O)CCN(C(=O)C=Cc2cscn2)CC1 N12CC3CC1CN3CC1CC(C1)CCC(CCCCC)C(C)NC2=O C(=O)(CC1CCCc2oc(C)nc21)NCC1N(C(c2onc(C)n2)=O)CCCC1 CCC(C(C)CN(C)C)(c1nnnn1C1CC1)NCc1cc(C)cc(F)c1 c1(C(=O)NC2CCCN(C(C(C)(C)OC)=O)C2)cccc(Br)c1Br N1(C(C2CCC(CC)CC2)=O)CCOC(C(=O)NC(C)(C)CN=[N+]=[N-])CC1 C1(OC)CC(CCNC(c2csc(CO)n2)=O)N(C(c2ccc(CF)cc2)=O)C1 C1(C(=O)NCc2cc(OC)nn2C)CC2(CCC2)CN1C(=O)CCC(C)C1CC1 N1(C(COCCOCC)=O)CCN(C(=O)CC2CC3CC3C2)C2COCC12 C1(=CC(=O)N(C(C)CCNC(=O)C=C(Cl)Cl)C)CCOc2ccccc21 C1(NC(C(C2CC2)OC)=O)C2CC1CN(C(=O)CC1CCCN(S(C)(=O)=O)C1)C2 CC(CC(=O)N(CC(O)CNC(c1cc2c[nH]cnc-2n1)=O)C)CC(F)(F)F C(=O)(CCCCCO)N1CC(CNC(Cc2cccc(OC(C)C)c2)=O)C(O)C1 N1(C(CCCCC)=O)C2CCC1CN(C(=O)C(C)Cn1cccn1)C2 C(=O)(C(C(CC)CC)C1CC1)OC(CC#C)CC#C c1(C(=O)NCC2(C)C(C)CN(C(c3ccc(F)cn3)=O)C2)ccc(S(C)(=O)=O)s1 N1(C(CC(C)OC)=O)CCC2(CC1)CC2NC(c1c(NC(C)=O)c[nH]c1C)=O C(=O)(C1=CCC(C)(C)CC1)N1CC(NC(C=Cc2c(C)ccs2)=O)C(C2CC2)C1 N1(CC(COC)O)CC=C(CNC(=O)CC(=O)Nc2nccs2)CC1 CCC(C#N)(CC)C(=O)NC1C(C)CN(C(=O)C(CO)N(C)C)CC1C c1(C(=O)NC(CNC(CC2(C)CCN(CCC)C2)=O)CO)cc(CC)ccc1N N1(C(c2cc(CC)nn2C)=O)CC(NC(C2CCC(C)(C)C2)=O)CC2(CCC2)C1 C(C)(N=c1[nH]c(=NC)[nH]c(=NCCC2COCCO2)[nH]1)c1c(OC)ccc(F)c1 CC1c2ccc(Cl)c(Cl)c2CCN1C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 C1(CNC(CNC(=O)NC)=O)(CO)CCN(C(=O)COC2CCC(C)CC2)CC1 C(=O)(C1=CC2(CCOC2)C1)NC1C2CC(NC(Cc3ncn(C)c3)=O)CC21 CC1C(C(=O)NC2CC(CCC(N3CCNC(=O)C3CCO)=O)C2)=NOC1C Cc1nscc1N(C)C(C1(NC(=O)COC(C)(C)C)CC1)=O C1(NC(C)=O)CCN(C(=O)C(C)CNC(=O)CC2CC2)C1 c1(N2C3CC(CC(NC(Cc4nnc(C)o4)=O)C3)C2)ncnc2ccc(O)cc12 C1(NC(C(C)SCC)=O)CCCN(C(=O)CCc2nc(O)n[nH]2)C1C N1(c2n(CCC(C)(O)C(F)(F)F)c(CC3CCC3)nn2)CCc2ccncc2C1 N1(C(CC2CN(C(C(CC(C)C)=O)=O)C(C)(C)C2)=O)CC2CCCC(C2)C1 c1(C(=O)NC2C(CNC(C3(OC)CCS(=O)(=O)C3)=O)C2)cc2c([nH]1)CCCC2 C1(C(=O)NC(COCCCNC(CC=CCC)=O)(C)C)CC12CC2(F)F c1(CNC(C(c2cnc(C)s2)N2CCC(n3cnnn3)C2)=O)cccc(Cl)c1 N1(C(Cc2cc(C)c(C)nc2)=O)CC(C)N(C(C2CC(=C3CCC3)C2)=O)CC1C c1(NC(C2C(C(=O)NCc3cccc(OCF)c3F)C2)=O)nc(O)ccc1[N+](=O)[O-] Cc1cc(O)nc(CNC(=O)CC2N(C(c3ccncc3O)=O)CCC2(C)C)n1 C=C(Cl)CCC(=O)N1CCC(C(N2CCC(F)(CO)C2)=O)C1CC Cc1nccc(N2CCC(CC(=O)N(N3CCCC3)C3CC3)C2)n1.C(C)C C(=O)(CCC(=O)N(C)CCOCCN(C(=O)C(C)Cc1c(C)n[nH]c1C)C)OC N1(C(C)C)CCN(C(=O)CC(C(F)F)NC(=O)C(=O)C2CCCC2)CC1=O C1(CC(=O)N(C(CNC(C2(C)CCOCC2)=O)C2CC2)C)CCCC(F)(F)C1 C1(C(=O)NCCCCCNC(c2c(C(=O)OCC)c[nH]c2)=O)C(C)(C)C1(F)F C(c1ccccc1Cl)=C(C(=O)NC1CC(CCNC(CCCC=C)=O)C1)C C1(C(=O)OC2(c3nnnn3C)CN(CC=C)C(CC)C2)CC(C)=CC(C)C1 C(N=c1cc(Cc2ccccc2)nc[nH]1)C1(CNC(CN=S(C)(C)=O)=O)CCCC1 c1(C(N2C(C(C(=O)NC(c3n(C)cnn3)CO)(C)C)CCC2)=O)ccc(Cl)o1 N1(C(C(C)CCc2cccc(F)c2)=O)CCCCC2(C1)CN(C(=O)C#CC1CC1)C2 C1(NC(C=CCN(C)C)=O)CCC2CN(c3cnc(C#N)cn3)CC2C1 c12coc(n1)CNC2=O.c1(C(=O)NC2(CC=O)CC2)[nH]nnc1C.CO C12(C(=O)NCC(C)N(C(=O)CCSC(F)(F)F)C)CCC1C2 c1(C(CN)=O)c[nH]c2cc(Cl)cc(Cl)c12.N1(C(=O)C2CC2)CCCC1 N1(C(c2nc(CC)oc2)=O)CCCC2(CCN(C(=O)CC3CCCC3C)C2)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)NC(C(=O)OC)C(C(C)C)OC c1(C(=O)NC2CC(NS(N)(=O)=O)C2)ccc2ncc(=O)[nH]c2c1 N1(C(Cc2c(C)cco2)=O)CC(N(C)C)C(CNC(=O)Cc2cnn(C)c2)C1 C(CCCCC(=O)N1CC(NC(c2cn(CCF)nn2)=O)C(SC)C1)OCC N1(C(C(c2cn(C)nn2)N(C)C)=O)CC2CCCC(C1)N2C(c1cnc[nH]1)=O c1(C(=O)NC(C2(F)CCCC2)C)ccc2c(c1)CC(C)O2 Cc1ccccc1CC(N1CCOC(CNC(C2CCCO2)=O)C1)=O Cc1ccc(CN=C(NCC(F)F)NC2CCOC(C)C2)cn1 c1(C(=O)NC2C(C)(C)N(C(=O)CCc3cncs3)CC2)cnc2sccn2c1=O C12(CNC(=O)C(O)C3CCCC3)CCC(CC1)N2C(=O)CCC[N+](=O)[O-] C(C(C)N=c1cccc(S(=O)(=O)NCCc2ccnc(Br)c2)[nH]1)OCCOC C(=O)(C(C)(C)C)NC(C)C(=O)NCC1(O)CC(C(=O)NC2(C)CC=CC2)C1 C1(CNC(C2(CC=C)CCN(C(C3OCCC3C)=O)C2)=O)CC2(CCC2O)C1 C1(CC)CN(C(c2ccn(C)c(=O)c2)=O)CCC1CNC(=O)CC1CSCCS1 c1(C(=O)NCC(C)N(C(C(c2ccc(C)s2)C)=O)C)cccc2nc(O)n(C)c12 C1(CC=C)(NC(c2cc(CO)[nH]n2)=O)CCCN(C(=O)CN2CCS(=O)CC2)C1 c1(CSC)cccnc1C(=O)NC1CN(C(=O)CC=Cc2ccccc2)C2CC12 C=C(C)CC(C(=O)NCC1CN(C(=O)CCc2cncs2)C1)NC(C)=O C(=O)(CC(C)C1CC1)NCCCOCCN(C(=O)Cc1csc(C2CC2)n1)C N1(C(C(CC2CC2)OC)=O)CC(C(N2CC=CC(OC)C2)=O)C(F)(F)C1 c1(C(=O)NCC23C(CN(C(c4cncc(C)c4)=O)C2)C3)cnc(C2CC2)nc1C C1(NC(Cc2ccc(C)nc2)=O)CC2CC1N(C(c1cc(Br)nn1C)=O)C2 N1(C(c2nc(C)c(C)s2)=O)CCN(C(c2cccnc2Cl)=O)CC1C c1(C(=O)NC(CCOC)CNC(C2CC3CC2CO3)=O)ccc(C)cc1F N1(C(C2CC(C)CC(C)(C)C2)=O)C2CCCC1CC(NC(c1c[nH]c(=N)o1)=O)C2 C1(NC(=O)CCNC(=O)COC2CCC2)CCCCC(=O)N1 C1(O)(CC(=O)NCC(C(=O)Nc2c(C)n[nH]c2)O)CCOCC1 CC1CC2(CCN(C(C3CC3F)=O)CC2)CN1C(C1CCC2(CC2)C1)=O c1(OCCNC(CCN(C(=O)C=C(Cl)Cl)CC)=O)ccccc1 c1(C(CC)C(=O)NC(c2cn(CCCF)nn2)(C)C)ccc(Cl)cc1 c1(C(=O)NCC2C(NC(Cc3n[nH]c(=NC)s3)=O)C2)cc(S(N)(=O)=O)cnc1C N1(C(CNC(=O)OCC)=O)CCC(N(C(=O)C(C)(C)CC)CCO)CC1 Cc1ccc(-c2cn(CCCCCCNC(=O)CCc3cnoc3)nn2)cc1 N1(C(C(C)N(C(C)=O)C)=O)CCN(C(=O)C(C)(F)F)CC1c1cccc(Cl)c1 c1(C(N2CCC(N(C(C3CCCC4CC34)=O)CC)C2)=O)c(C)ccc2cccnc12 c1(C(=O)NC(C2CN(C(c3cnc(C4CC4)[nH]3)=O)C2)C)cc(Cl)nnc1Cl N1(C(CC2(C)N(C(CCN(CC)CC)=O)CC2)=O)CC(C(C)C)C2(CC2)C1 c1(C(=O)NCC(CN(C(=O)C=Cc2ccc[nH]2)C)O)cnnn1C c1(-c2cc(OC)c(O)cc2)ccc2ncc(C(N3CCNC(=O)C3)=O)c(=O)n2c1 C1(NC(CCN(CCC(C)(C)C)C)=O)CN(C(C2CCOCC2)=O)C(C)(C)C1 C1(C)(C(=O)NCC=C)CC(O)CN1C(=O)C(F)C(C)(F)F c1(C(N(C2CCN(C(=O)C3=CCCS3)CC23CC3)C)=O)c[nH]c2ccc(F)cc12 CCS(=O)CC(=O)NCCC1(NC(=O)C(O)C2CC2)CC1 c1(C(=O)NC2C(NC(C(C)CSc3ccccc3)=O)CC2)n[nH]c2c1COCC2 c1(C(=O)NC2C(NC(c3n[nH]c(C)c3F)=O)C2)ccn2ccnc2c1 c1(C(N(CCNC(C(C)c2cccs2)=O)C)=O)c(F)cc(O)cc1F C=C1Cn2c(C(N3CCC4CN(C(C5CC5(F)F)=O)C4C3)=O)nnc2S1 Cc1ccc(C(N2CC(N(C(=O)CCCN3CCCC3)C)C3(CC3)C2)=O)nc1O C(C)(c1cnn(C)c1)=CC(=O)NCC(CN(C(C(CC1CCC1)OC)=O)C)O N#CC1=C(C(=O)N2CCOCC2C(=O)NCCCc2cnn[nH]2)CCC1 C(c1cccnc1C)=CC(N1CC2C(CNC(CC=C(C)C)=O)C2C1)=O C(=O)(CCC(C)(C)NC(c1cnc(Cl)n1C)=O)NCC(CC)n1cccn1 c1(C(=O)NCC2(C)CCC(NC(c3cc(C)[nH]n3)=O)C2)c(C)ccc(C)c1N C(CC(C)C)(C(C(=O)NC1CCOC1)N1CCC(C(C)C)C1(C)C)OC C1(C(=O)NC(C(=O)NC)C2CC2)C=CCCN1C(=O)CCC1CCCN1C N1(C(C2OCC(C)(C)OC2)=O)CCC2CN(C(c3cc(C4CC4)[nH]n3)=O)C2C1 CC1=C(C(=O)N2CC(CNC(C34CC(C(=O)OC)(C3)C4)=O)CC2C)SCCO1 N1(C(C=CCN(C)CC)=O)CC(C(=O)NCC2COC3(CCC3)C2)C(C)(C)C1 N1(C(c2c(C(F)(F)F)cc(C)o2)=O)CC(NC(C2C=CCS2)=O)CC(O)C1 O=C1CC(C(=O)NC(C2CCCN2CCSCCO)C2CC2)CCN1 c1(C(N2CC(NC(C3CCC(C(=O)OC)C3)=O)C2)=O)ccc(F)c(S(C)(=O)=O)c1 C#CCCCCCCC(=O)NC1C(C(=O)NC(c2ncccn2)C)C1(C)C CC1CN(C(C2CC23CCN(C(C2(CO)CCCC2)=O)C3)=O)CC1N=[N+]=[N-] C1(CCNC(C2(C(C)C)CCC2)=O)CCCN(C(=O)CC2CCCCO2)C1 C12CCCN(C1)CCC(=O)N2.c1(CC)nc(C(N)C(C)(C)C)cs1 N1(C(C(c2ccccc2)OC)=O)CCOCC1CCNC(C1(F)CCOCC1)=O c1(C(=O)Nc2cc(Cl)c(F)cc2F)cc2cccc(C(F)(F)F)c2nc1Cl C1(CNC(C2C(CC)C2)=O)CN(C(c2ccsc2Cl)=O)CCN1C O=C(C(F)C1=CCCCC1)NCCC1CCN(C(=O)CCc2cccnc2F)C1 CC1OCCN(C(=O)CC2C=CCC2)C1C(=O)NCC1C(CO)C1(C)C C1(NC(C2(CC=C)CCCCC2)=O)CN(C(c2occc2Br)=O)C2CCCCC12 N1(CC(=O)NC(c2cccnc2)C(=O)NC(CC#C)CO)C(=O)CCC1=O N1(C(Cn2nc(C)oc2=O)=O)CCN(C(C2CCC(F)C2)=O)C(C)C1 C=CCC(CC(F)F)NC(C1CC(N(C(=O)C=Cc2cscn2)C)C1)=O C1(NCC2(CCC)CCCNC2)CC2CCC(C1)N2C N1(C(c2c(C)scn2)=O)CCCN(C(=O)C2=CCC2C(F)(F)F)CC1C(C)C Cc1ccc(C)c(C(=O)NC2CCN(C(c3sc(C)c(C)c3C)=O)C(C)C2)c1C C(CNC(=O)CN1CCOCC1=O)(CC(=O)N(CC(F)F)C1CC1)OC c1(CNC(c2c(C)noc2C)CC)ncnc2scc(-c3ccc(Br)cc3)c12 C1(CC(=O)NCCNC(=O)CN2CC(CF)C2)CCOCC1 S(=O)(=O)(c1ccc(F)cc1)NCC(N1CC(O)(N(C(=O)CSC(C)(C)C)C)C1)=O C1(C(=O)NC(C(=O)NCC(=C)CC)C)CCC2(CC1)CC2 C(=O)(C(C)CCC(C)(C)C)N(C1(C2CCC2)CC1)C.C#CCC1C(=O)N1 c1(CC(=O)NCC2(F)CC(C(=O)OC)C2)ccc(NC(C)=O)cc1F.C12CC1N2 N1(C(=O)C(O)C(F)(F)F)CCC2CCN(C(=O)C#CC3CCC3)C2C1 c1(CN(C)C)ccc(NC(=O)NCc2csc(Br)n2)c(I)c1 N1(C(C)=O)CCCC(O)(C(N2CCCC(NC(=O)CCn3ccnc3C)C2)=O)C1 CCC1=NOC(CNC(=O)CCCN(C)C(c2ccnn2C)=O)C1 c1(OCC)cccc2c(N3CC(C)(C)CC3C(=O)NCCC3CC3)ccnc12 N1(C(c2cc(C(C)=O)c(C)o2)=O)CC2CN(C(=O)C3=CCSC3)CCC2(CO)C1 Cc1cc(CC(=O)NC(C)CCCCNC(=O)CC(F)(F)Cl)n(C)n1 C(=O)(CS(=O)(=O)C(C)C)N1CC(N(C(c2cc(SC)nn2C)=O)C)C2(C1)CC2 N1(c2ccnc(C)n2)CC2CCC1C(NC(c1cn(C)ccc1=O)=O)C2 N1(C(C2C(C)(C)C2(F)F)=O)CCCC(F)(CNC(C2(n3cccn3)CC2)=O)C1 c1(OC(C)C)cnc(C(=O)N(CCC(C)NC(=O)C=CCCC(C)C)C)nc1 c1(C(N2CCC(CC(=O)NC(CCCC)CO)C2)=O)cnc(Cl)c(F)c1 C(CC(=O)NC1CC(CNC(C23CCC2C3)=O)C1)OC c1(C(N2CCC(CNC(c3c(C)cc(O)nn3)=O)C2)=O)cc[nH]c2nccc1-2 c1(C(=O)NC2CCC(CCNC(C3(CC)CC3)=O)C2)cccc2occc12 C(CN=c1cc(C)nc(S(C)(=O)=O)[nH]1)C1CCN(C(C=CC=CC)=O)CC1 C(=O)(C(C)C(F)(F)C(F)F)OC(c1cc(C#C)c(C)cc1)=O.C1=CCN(C)C1=O N1(C(c2ccc(C#N)s2)=O)CCC2CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)C2C1 c1(C(=O)NCC(C)N(C(c2cc[nH]c2)=O)CC)csc(C(C)(F)F)n1 CCCCCCCCC(=O)NC1CCN(C(c2cnn3c2CCC3)=O)C1C N1(S(C)(=O)=O)CCCC(S(=O)(=O)C(N2CCC(c3nc4c(s3)CCC4)CC2)=O)C1 C1(NC(c2ccn(C)n2)=O)CC2CCC(C1)N2C(c1cncnc1C1CC1)=O c1(C(=O)NC(CN(C(c2c(C)[nH]nc2Cl)=O)C)C)cc2c(=O)[nH]ccn2c1 CC(C)CCCCCNC(=O)CC1CCCC(NC(=O)CC#N)C1 C(=O)(CN=c1cc[nH]cc1)NC(C1CN(C(=O)C(c2ccccc2)F)C1)C c1(C(N(CC(CC)NC(CN(CCC)C)=O)C)=O)cc(C)cc2ccoc12 c1(SC(C(=O)N(CC(N2CCCC2)C)C)C)cnn(C)c1.C12(CCC1)C(=O)N2 C1(CNC(C2C(NC(C=CCCC)=O)COC2)=O)CC[Si](C)(C)C1 C(C(C(=O)NC1CCC(CCNC(c2ncsc2C)=O)C1)NC(C)=O)OC C1(CC)CCCN(C(=O)C(F)C(C)(C)O)C1C(=O)NCc1nc(C)c(C)o1 c1(C(=O)NCC(CCCC)NC(=O)C=Cc2ccc(F)cc2)cc(C#N)oc1C N1(C(CCC(C)OC)=O)CCCC2(NC(c3n[nH]cc3Br)=O)CC2C1 CC1CCCC1(C)C(N1CCN(CCNC(C2CC(F)(F)C2)=O)CC1)=O N(C1CCCn2nccc21)C(C(CCNC(C1CCCC(CF)C1)=O)OC)=O CN1CCC(C(=O)NC2CC(n3cc(-c4cnn(C)c4)nn3)C2)S1(=O)=O c1(C(=O)OC)cc(C(N2CC(NC(=O)C(C)CC(C)C)C(C)C2)=O)ccc1C c1(C(=O)NC2(CO)CN(C(c3c(C)sc(O)n3)=O)C2)ccc(Br)c(F)c1 N1(C(c2c(C)[nH]cc2)=O)CC2(NC(C3CC=CCO3)=O)CCCC2(F)C1 N1(C(C2C(C(C)=O)C2(C)C)=O)CC(CNC(c2cc(C)oc2C)=O)CCC1C C1(C(CNC(Cc2ccn(C(C)C)n2)=O)(C)O)CCN(C(c2ccsc2)=O)CC1 C1(NC(C=CC)=O)CCC12CCN(C(c1ccc(OCCCCC)cn1)=O)CC2 N1(C(C(C)(C)NC(c2ccc(C#N)o2)=O)=O)CC2CC=CC1C2 C1(C(=O)NCC2(C)CC(NC(=O)CCc3ncccn3)C2)(CO)CCCCC1 C(c1cccc(Cl)c1)=CC(=O)NCC(=C)CCNC(C1(C(N)=O)CCC1)=O C12CCN(C1=O)C(CC)C(CCCc1ncc(CCN(S(C)(=O)=O)C)s1)C(=O)N2 Cc1ccc(C=CCC(=O)NC(C)C(CO)NC(C2CC2C(C)(C)C)=O)cc1 c1(OC)cc(CN(C2CCN(C(C)=O)C2)C)ccn1.c1(-c2nc[nH]n2)ccc(CN)cc1 c1(CN2C(C(=O)NCC(O)C(F)(F)F)CC(OC)C2)cc(Cl)ccc1C N1(CCNC(C2(C(C)NC(C(CC)SC)=O)CC2)=O)CCOC(C)C1 C1(CC(=O)NC2CC(O)(CNC(C3CC4(C3)CC(O)C4)=O)C2)CC2CCC1CC2 CC1(C)CN(C(C2CCCO2)=O)C(CNC(c2ccn3cncc3c2)=O)CO1 C1(NC(c2c(CC)c(F)ccc2)=O)CCCCN(C(=O)C=Cc2nccs2)CC1 c1(C(C)C)ccc(C(N)C(=O)NC(C)COc2ccc(Br)cc2)cc1 c1(C(N2CCN(C(C3ON=C(CC)C3)=O)C3C2C3)=O)cc(Cl)c(O)cc1C C1(C(=O)NC2C3CN(C(C4CCN(C(CC)=O)C4)=O)CC32)CCCCC1C1CC1 c1(C(=O)NCC2(c3ccc(F)cc3F)CC2)c[nH]c2ccncc2c1=O c1(CNc2nc(-c3ccc(F)nc3)sc2)cccc2ccoc12 C1(CC(=O)NCCCC(=O)N(CCC)C)CCCC(O)C1 C(=O)(N=c1[nH]nc(Cl)cc1Br)C1N(C(Cc2c(OC)cccn2)=O)CC(F)C1 C1(NC(c2ccn(C(C)C)c(=O)c2)=O)CC2CCC(C1)N2C(c1ccoc1Cl)=O CC1(C)CC(NC(=O)C(c2ccccc2Cl)O)CCN(C(=O)CCCCCF)C1 C1(CNC(c2cccc(Cl)c2)=O)COCCN1C(c1ncoc1C(F)(F)F)=O C#CCCC(O)CCNC(=O)CC(C)CNC(c1cc(Cl)n[nH]1)=O c1(N(CC(CC)CC)C)cc(C)c(S(=O)(=O)NCCCOCC(=O)OC)cn1 C(=O)(CC(C)CC(=O)N1CC2CCC(C1)C2NC(=O)C(C(C)(C)C)SC)OC CCC(O)C(C)C(=O)N1CCC(CF)(NC(c2cnn(C(C)CC)c2C)=O)C1 C(C(CNC(c1cc(Cl)c[nH]1)=O)C(F)(F)F)NC(C(C)COc1ccccc1)=O C1(CC(=O)NCCCCNC(CCc2cc(OC)no2)=O)CC(C(C)=O)C1(C)C C1(C)(CNC(Cc2c(C)noc2)=O)CCCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 Cc1cc(C)nc(SCC(N2CC(C)(NC(=O)C=CC(=O)NC3CC3)C2)=O)n1 c1(C(C(=O)NCC(CNC(c2ccc(F)s2)=O)CO)OC)ccccc1O Cc1ncc(CNC(c2nncn2C)c2nnnn2CC2CCOC2)[nH]1 c1(NC(C(C)Oc2cccc(C(C)=O)c2)=O)cc(I)cc(I)c1 c1(C(=O)NCCC2CN(C(C(C)CC3CCC3)=O)C2)ccc(O)c(N)n1 CCC(CC)C(C(=O)NCCN(C)C(c1csc(C(F)(F)F)c1)=O)OC C(=O)(CCCC(C)(C)C)NC(CCCNC(C=CCCC)=O)c1ccccc1 CC(CC(=O)NCCCN1CCN(C(C2CC2C)=O)CC1)CC(F)(F)F c1(C(=O)NCCN(C(CC)=O)CCCN(C)C)ccc(C(F)(F)F)nc1 Cn1cc(CCC(=O)NC2CCC(NC(=O)C(O)C(C)(C)C)C2)c2ccccc12 n1(CCOCCOCCOCCOC)cnccc1=O.C1(C(=O)OC)CC1C(=O)C C(=O)(C(CC(C)C)OC)NCC1(O)CCN(C(CCN(CCC)C)=O)C1 N1(C(c2c(C)n[nH]c2)=O)CCC2(COC(CNC(=O)CCC3CCC3)C2)C1 C=CCC(C)(C)C(=O)NCC1C(CNC(=O)CC2CCC3CC23)C1(F)F C1(CNC(c2c(C)scn2)=O)CN(C(c2[nH]c(C3CC3)nc2C)=O)CC12CC2 CC1N(C(C2(CNC(=O)Cc3ccsc3)CCCC2)=O)CCC1(C)C N1(C(C(C)c2ccsn2)=O)CCC(F)C(NC(c2conc2C(C)(C)C)=O)C1 O=C1CCc2nc(N(CCNC(=O)CSC3CC3)CC3CC3)ccc21 CN1CCC(C)(C(=O)NCC(C2CC2)NC(=O)CC2CC=CCN2C)CC1 C1(C(C)NC(=O)CCC2CC2(Cl)Cl)CN(C(=O)CCc2cn(C)cn2)CCO1 c1(C(c2nnnn2-c2ccc(N(C)C)cc2)NC(C)C)c(Br)c(Br)nn1C N1(C(c2n(C(C)C)nnc2)=O)CCOC(c2ccc(-c3nn[nH]n3)cc2)C1 C12(NC(C3COC4COCC34)=O)CCCN(C(=O)C=Cc3cocn3)CC1C2 N1(C(=O)Cn2ccnn2)CCCC(CO)(Nc2cc(O)ncn2)C1 Cc1cc(Cl)cc(C(=O)NCCCC(C)(C)NC(=O)CC2CCCCC2C)c1O N1(C(C2OCCN(C(C)C)C2)=O)CCCC2(NC(=O)C(C)O)CCCC12 c1(CC(N2C(C(=O)NC)CCC2)=O)cccc(C)c1F C1(CNC(C(CC)CO)=O)CCCN(C(c2nn(C)cc2C(=O)OC)=O)CC1 C1(C(=O)NC(C)(CNC(=O)CCn2cc(Cl)cn2)C2CC2)CC2CCC1CC2 c1(OCC2N(C(N(C3COC3)C)=O)CCC2)cccc(Cl)c1 c1(CC)ccc(NS(=O)(=O)CC(=O)OC2(COC)CCCOC2)cc1 c1(NC(C23C(CN(C(c4c(C(C)C)ccs4)=O)C2)C3)=O)cnc2c(c1)CC(=O)N2 c1(SC)c(C(N2CC(F)(CNC(C3CCCC(F)C3)=O)C2)=O)cnn1C Cc1sc(-c2cccnc2)nc1C(N1CCC1CNC(=O)C(C)CC1CCC1)=O c1(CC(=O)N(C)CC2(O)CN(C(COCC=C)=O)C2)ccc(CC(C)C)cc1 c1(NCC(C)C)cc(N2CCC(C(C)CN3CCCCCC3)CC2)ncn1 N1(C(C(CC#C)C2CC2)=O)Cc2occ(C(=O)NC(COC(C)=O)CO)c2C1 C1(n2cccn2)(C(=O)O)CCC(NS(CC2CCC(C)C2)(=O)=O)CC1 c1(CC)ccccc1CC(N1CCC(O)(CNC(=O)Cc2cc(CC)no2)C1)=O C1(C(N(CCN(C(=O)C=Cc2cnc[nH]2)C)C)=O)Cc2cc(Cl)ccc2O1 C1(CCC)(C(=O)O)CN(C(N2CCC(CC)C2)=O)CCC1O CCCCC(CC)CC(=O)NC1CC(CNC(C2CCCN(C(C)C)C2)=O)C1 c1(C(C)O)cncc(C(=O)NCC(C2CCCC2)NC(c2ccon2)=O)c1 C1(NC(C(C2(OC)CCCC2)(F)F)=O)CCN(C(C2CC(C)(O)C2)=O)CC1C C(CC(C)C(F)(F)F)NC(C(C1CN(C(Cc2ccc(C)o2)=O)C1)O)=O c1(C(=O)NC(CCN(C(CCC=CC)=O)C)C(C)C)cccc2c1CC(C)(C)C2 C1(CC(=O)NC(C(=O)OC)C)C2CCCC2N1C(=O)CC1CCCN(C)C1 c1(NCC(O)C(F)(F)F)cc(NCC2(C(F)(F)F)CC2)nc(C(F)(F)F)n1 CCC(CC)CCCC(=O)NC1CCC(NC(c2cnc(Cl)cc2N)=O)CC1 c1(NC(=O)NCC(c2ccco2)NS(C)(=O)=O)ccc2c(c1)CCCO2 c1(C(=O)NC2(CC(=O)NC(COC)C3CC3)CC2)ccnc(OCCN(C)C)c1 C1(C(=O)NCCC(N2CCCC2Cn2cnnn2)=O)CCOC(C2CC2)C1 C1(C(=O)NCc2nnc(CC)o2)CN(C)CCN1C(=O)Cc1ccc(O)cc1 CCCCCCC(C)C(=O)N1CCN(C(=O)Cc2cc(F)c(N)cc2F)C(C)C1 N1(C(C2CCN(C(C=C(C)C(C)C)=O)C2(C)C)=O)CCCC(C)(O)CC1 Cc1cc(C(F)F)nn1CC(=O)NC1CN(C(=O)C=CC2CCOCC2)C1 C1(NC(COCCOC)=O)C=CCC(C=O)C1.c1(C2CCC2)ncc[nH]1 c1(N(C2CCN(C(C(C3CC3)OCC)=O)C2)CCO)nc(Cl)nc2c1CCOC2 CCCCCC(CC)C(=O)NC1CCC2(CC1)CN(C(=O)C(C)C(O)CC)C2 C1(C(N(CC)CC2CCC2)=O)COC2(C1)CN(C(c1cnc3[nH]ncc3c1)=O)C2 C(=O)(C(F)CCC(C)C)N1CCCC(C)(C2C(NC(C=C(COC)C)=O)C2)C1 Cc1onc(C2CCCC2)c1C(N1CC(NC(=O)CCC2CCCCN2C)C1)=O CCCC(C)(CC)C(=O)N1CC(O)(C2CCCN2C(c2sccc2SC)=O)C1 C12(CC(=O)NC3C(NC(C4(C)CCOC4)=O)CC3)CCC(CC1)CC2 c1(C(=O)NCC2C(C(=O)NC(C3CCOCC3)C)C2)cc(C#N)cn1C C(=O)(CCCCCCNC(C1(NC(N)=O)CC1)=O)N(C(CC(C)C)C)C N1(C(C)=O)CCCC(CN2CCCC(C)C2)C1 N1(C(C(CCNC(CC2CC(=C)C2)=O)OC)=O)CCC2(CCOC2)C1 Cc1cccc(Cl)c1OCC(N1CC(NC(c2[nH]c(C)c(CO)c2C)=O)C(C)C1)=O c1(C(N(CC(N2CCC(CN=[N+]=[N-])C2)=O)C2CCC2)=O)ccccc1[N+](=O)[O-] CC1CN(C)CC(C(N2CCOC(C(C)NC(=O)CN3CC4CC4C3)C2)=O)O1 c1(C(=O)NCC(O)CNC(C2(n3ccnc3)CCCC2)=O)cc(=O)cc(Cl)[nH]1 N1(C(c2ccc(C)s2)=O)CCC(C2CCCN(C(=O)C(O)C3CC3)C2)C1 Cc1cncc(C)c1C(=O)NC(C)CC(C)NC(=O)CCc1ccc(F)nc1 c1(NC(C(CC#C)NC(c2cnn(C)c2CC)=O)=O)ccccc1N=[N+]=[N-] Cn1cnc(C(N2CCC(NC(=O)CN3CCSCC3)C(O)C2)=O)cc1=O c1(C(=O)NCC2(C)CCN(C(CN(CCC)C)=O)C2)cccc2c1NC(=O)CC2 c1(NC(c2c(NS(CC)(=O)=O)cnc(F)c2)=O)c(Cl)cc(C(F)(F)F)cc1Br C1(OC)CCCC(C(=O)N(C)CC2CCCN2C(=O)CCc2c(C)noc2C)C1 c1(OC)ccc(C)cc1CC(N1CCC(CNC(C2CCCO2)=O)C(C)C1)=O c1(C(C)(F)F)ccc(C(=O)NC2C3CCN(C(=O)COC4CCCC4)C23)c(O)n1 c1(C(C(=O)NC(C)C(N2CCCC2NCC(F)(F)F)=O)N)cccc(F)c1 CC1(CNC(C2(CO)CC2(F)F)=O)COCCN(C(=O)CCF)C1 CN1CCc2nc(C(=O)NCCC3CSCCN3C(=O)CCC(N)=O)sc2C1 c1(OC)ccc2c(C(=O)NC3CCC(NC(=O)CC4CCOC4)CC3)cnn2c1 c1(C(=O)NCCC2(C(=O)NCc3ncn(C)n3)CCCC2)cnn2c1OCC2 c1(C(=O)NC(C2CCCC2)CNC(c2n(CCCC)ncc2)=O)cc(F)n(C)n1 c1(OC)cc(C(=O)NC2CN(C(c3cc(C#N)c[nH]3)=O)CC2F)cc(F)c1F c1(C(=O)NCC(CNC(C2(C(N)=O)CC2)=O)CO)cccnc1-c1ccncc1 O=Cc1csc2cc(C(=O)NCCc3ccccc3Cl)ccc12 CC(CC(C)(C)C)C(=O)N1CC2(CC2)CC1CNC(=O)C(C)(F)F N1(C(CCC(=O)C2CC2)=O)CCC2(CO)CN(C(c3cccnc3)=O)CC2C1 Cc1nc2cc(C(=O)NC(C)(C)C(C)NC(c3cc4n(n3)CCO4)=O)[nH]c2s1 Cc1ccc(C=CC(N2CC(CNC(C3CC3(F)F)=O)C(F)(F)C2)=O)nc1 Cc1cccc(O)c1C(=O)NC1CN(C(C2(C)CCN(C)C2)=O)CC1C N1(C(=O)NCC=C)Cc2nnc(O)n2CC1C(=O)OC C1(OC)CC(C(=O)N(CCCNC(C2CC(CF)C2)=O)C)CC1OC.C1(C)CC1 n1(CCC(N2C(C(C)(C)NC(C3C(=C)CC3)=O)CCC2)=O)cc(Br)c(C)n1 N1(C(C(C=C)O)=O)CCCC12CCN(C(C1OCC3CCCCC13)=O)CC2 N1(C(CCCC(C)=O)=O)CC2(C1)OC1(C)CC2(NC(=O)CCC(C)N(C)C)C1 C1(F)(CNC(C2N(C(CCCOC)=O)CC=C2)=O)CCOCC1 N1(C(C(CC)(CC)CC)=O)CC2CCCC(C1)N2C(=O)Cc1ccc(F)cc1 Cc1cccc2c1CN(C(C1CN(C(c3cncn3C)=O)CCC1O)=O)C2 C(CC)(C(=O)N(C)CC=CC(N1CC(C)(F)C1)=O)OCC C1(CNC(CC(CC)CN(C)C)=O)CCN(C(=O)CCOC(C)=O)CC1(F)F C1(OC)CCCN(C(=O)CCC2CCCN2C(c2ccc(C)cc2)=O)CC1 C(CC(C)C(=O)NCCN(C(=O)C(C(C)C)NS(=O)(=O)C1CC1)C)OC Nc1nc2c(cc1C(N1CCC(NC(=O)C(F)=C3CCCC3)C1)=O)CCC2 c1(CCC(N2CCC2C(=O)OC(F)F)=O)nnc(-c2ccco2)o1 CC(C)CC(O)C(=O)NC(C(=O)NCc1nc2c(s1)CCC2)C(C)C CCC(C)CCCC(O)CC(=O)N1CCN(CC(F)F)CC1 N1(C(C(CC(C)C)F)=O)CCOC2(CCC(NC(=O)C=C3CCOCC3)CC2)C1 CC(F)(F)C(C)(C)C(=O)NCC1C2CN(C(=O)CCNC(c3ccsc3)=O)CC12 c1(OCC)c(CC(=O)NC2(C3CCCN3C(=O)C(F)OC)CC2)cccc1F CC(C(F)C(=O)NCC12CN(C(c3cc(C#N)c[nH]3)=O)CC1CCO2)C(F)(F)F N1(C(C=CC)=O)CCCC(O)(CNC(=O)CN(C2CCSC2)C)CC1 C1(NC(c2cc(C)oc2C)=O)COC2(CNC(=O)C(c3ccccc3)=O)CC1C2 C1(C(=O)NCCCCNC(c2cc[nH]n2)=O)CC2CCCCN2C1 c1(CNC(C2CC2C(=O)NC2C(C(=O)NCC#C)C2)=O)ccnnc1 c1(C(N2C(C3(NC(C4C(N(C)C)COC4)=O)CC3)CCC2)=O)cnn(CCO)c1N C1(CCCC)CN(C(=O)C2=CCCCC2)CCN1C(C1CCCN1C1CC1)=O C1(C(N2CCC(OCCNC(C(C)CC3CC3)=O)CC2)=O)CC2(COC(=O)N2)C1 C1(C(=O)NC2C(NC(CN(CC)CC)=O)CC2)CC2C=CC1C21CC1 CCCCC(CNC(=O)CC1CC(O)CN1C(c1ccncc1NC)=O)CCC N1(C(CC(C=C)C)=O)CC2(CCN(C(c3ccc(OCCF)cc3)=O)CC2)C1 N1(C(C(CC2CC2)NC(=O)C=CCF)=O)CCOC2(CCCC2)C1 S(=O)(=O)(c1ccc(Br)c(NC(=O)CS(=O)(=O)CCO)c1)NCC(C)C c1(C(N2C(CNC(C3CCc4nnnn4C3)=O)CC2)=O)ccc2snnc2c1 c1(C(N2C(C(C)NC(c3cncnc3)=O)CCC2)=O)ncnc2c1CCC2 Cc1cccc(Br)c1C(C(=O)NCCCC(F)F)NC(=O)CC(C)c1ccco1 c1(C(=O)NCC2COCC2O)cnc(-c2cccc(O)c2)cn1 CC1C2CC(C2NC(=O)CC2(O)CCOCC2)N1C(C1CCC(=O)O1)=O c1(NC(C(c2ccoc2)NC(=O)C2=NOCC2)=O)ccc(F)cc1O C1(C(=O)NC(CC=C)CO)(CC)CCN(C(=O)C(C)CNC(C)=O)CC1 c1(C(C(=O)NCCn2cc(C(c3ccccc3)(C)O)nn2)O)ccc(C#N)cc1 C1(CNC(=O)Cc2nc[nH]n2)CCN(C(C2CCCC2)=O)CC1(F)F C(CCCCC(=O)N1CC(F)CC1CC(=O)NC1(CO)CC=CC1)N(C)C N1(C(CN(C(C2C(C(C)=O)C2(C)C)=O)CC2CC2)=O)C(CO)CC2OCCC12 C(=O)(C(C)(C)CCCOC)N1CC(NC(C(CCOC)OC)=O)C(O)CC1 c1(C(=O)NCC2CC2CNC(C2CC3CCC2C32CC2)=O)cc(O)cc(F)c1F C(=O)(C(F)(F)C(C)O)NCC(C(=O)NCC1CCC(=C)CC1)C C1(C)(C(N(C)CC2(O)CCN(C(=O)CCC3CCCO3)C2)=O)CCC(C)(C)CC1 c1(CNC(C2(CCNC(CC3COCC(C)O3)=O)CCC2)=O)nn(C)c(=O)n1C N1(C(CCSC)=O)CC(C(=O)NCCn2nc(C)nc2C)C2(CCC2)C1 N1(C(c2cc(C3CCOCC3)[nH]n2)=O)CC(NC(C2(CO)CCC2)=O)CC(F)C1 N1(C(=O)NC2CC(NC(CC=C=C)=O)C2(C)C)c2ccccc2CC1C c1(NC(C2(C)CCCN2Cc2c(Br)ccnc2Br)=O)cc2ccc(Cl)nc2[nH]1 c1(C(=O)NC)ccc(COC(C)(C)C)c(Cl)c1.C(CNC=O)NC(=O)N CCS(=O)(=O)CCCCCNn1nnnc1C(c1cc(C)nc(C)n1)OC c1(OC)cc(C(=O)NC2CN(C(C3CN(C(=O)N(C)C)C3)=O)C2)cc2c1OCO2 C1(CNC(C2C(NC(C(CN(C)C)O)=O)CCCC2)=O)CC2CCCC2C1 C1(C(=O)OC)CCC(C(=O)NCCN(C(C(CO)C(=O)CO)=O)C)C1 c1(OC)ncccc1CN1CCCC1c1ccnc(Br)c1 N1(C(C2C(C)=C2)=O)CCC2(NC(c3ccc4c(c3)CCC4)=O)CCCC12 C1(NC(Cc2cc(C(=O)OC)sc2)=O)CCN(C(=O)C=Cc2nc(C)co2)CC1C N1(C(C(C2CCCC2)OC)=O)CCC(C)(NC(=O)C=Cc2cocn2)CC1 C(=O)(C(O)C(C)(C)CC)NCC1N(C(c2c(CC)nc[nH]2)=O)CCN(C)C1 CC1CN(C(c2cccnc2C(F)(F)F)=O)CCN1C(c1ccc(=N)[nH]n1)=O Cc1cccc(CC(=O)NC2CCOC(CNC(c3cc(C#N)c[nH]3)=O)C2)c1Cl C(=O)(C(O)C1=CCCCC1)N1CCN(C)CC1C(=O)NC1CN(C2CCC2)C1 C(=O)(CC1=CCN(C(c2cnnn2C)=O)CC1)NCCCC=C c1(-c2cc(C(N3CC(NC(CCc4cn(C)nc4)=O)C3)=O)n[nH]2)ccc(Cl)cc1 C1(OC)CCC2(C(=O)NC3CC(CCNC(c4cnc(O)o4)=O)C3)CC12 c1(OC)cccc([N+](=O)[O-])c1C(N1CC2CN(C(c3ccnc(O)c3)=O)C2C1)=O N1(C(CCSCC)=O)CCOC(C(=O)NCC2CC(CC)=NO2)C1 C1(NC(C(=O)NCC)=O)CN(C(=O)Nc2cnc(C(F)(F)F)cc2O)CCC1C C1(C)(CC)CCC(C(N2CC(=C(F)CNC(=O)CC3CCOC3)C2)=O)O1 N1(c2c(C)cccc2)C(=S)NC(c2sc(Br)c(Br)c2C)C2=C1CCN(OC)C2=O c1(C(N2CC(NC(CC(C)(F)F)=O)C(N(C)C)C2)=O)cc(Br)cnc1S O=C1C(NC(=O)N(CC(F)F)C2CC2)CCN1C1CC1 CN1CC2CCN(C(C3CCCCC3NC(=O)Cc3cncnc3)=O)CC2C1 CC1CN(C(=O)CC2CCCN2C(=O)C(F)=CC2CC2)C(C)CCO1 N1(C(c2ccc(SC)s2)=O)CCN(C(=O)C(c2ccccc2)C)C2CCCC12 C1(CNC(C2CC2CCC(F)(F)F)=O)CCCCN1C(=O)Cc1cc[nH]c1 N1(CC)CCN(C(=O)C(CN(C)C)NC(C2CC2(C)C)=O)CC1=O c1(C(=O)NC2(CCCNC(C(C)N(C(C)=O)C)=O)CC2)ccc2c(c1)C(C)CO2 CCCC(C(=O)NCC(C)(CO)NC(=O)CCc1cn(C)nc1C)C(C)C CCCC(C(=O)NCC(C)(C1CC1)NC(=O)Cc1nccn1C)N(C)C N1(C(C(C)OCCCC)=O)CC2(CNC(=O)CC(C)CC)CC1CO2 N1(C(=O)CC2CCN(C(C3CC4CCC3C4)=O)C2)CCc2nc[nH]c2C1 c1(C(C)=O)ncccc1NC(C1C(C)CN1C(C1CNC(=O)C1)=O)=O CCCCCCC(CC)NC(=O)NCc1cc2ccoc2cn1 N1(C(CCCC#N)=O)CCN(C(C2(CCF)CC2)=O)C(c2cc(F)ccc2F)C1 c1(CC)cc(C(=O)NC2CCC(NC(=O)CC3CCC(=O)NC3)CC2)c(C)o1 c1(C(=O)OC)cc(F)ccc1NC(=O)CC1CCN(Cc2ccc(C)c(Cl)c2)C1 O=C(C#CC1CCCO1)NCC1(CO)CCCN(C(=O)C(Cl)=CCl)C1 C(=O)(C1=CCC(NC(c2cc(C(C)C)no2)=O)C1)NCCCCC C1(NC(Cc2ccc(C)nc2)=O)CCCCN(c2ncc(Br)c(O)n2)C1 c1(C(=O)OC)ccc(C(=O)NCCOCCN(C(=O)C(C)S(N)(=O)=O)C)c(F)c1 c1(CC)cc(C(=O)NC2(C)CN(C(c3c(C)cc(C)oc3=O)=O)C2)cn(C)c1=O C1(CC)CN(C(c2ncc(OC)cc2F)=O)CCN1C(=O)CS(=O)CC CC1CCC2(CO1)CN(C(=O)C(O)CCNC(C1CCCCN1C1CC1)=O)C2 c1(CC)ccnc(O)c1F.c12nccnc1C(=O)NCCSCC(=O)NC2 c1(C(N2CCC(NC(c3cn(CCC)nc3)=O)(COC)C2)=O)nccc(N)c1Cl O=C1CC2C(C(=O)NC3(CCC(=O)NC4CC(CCF)C4)CCC3)C2C1 CC1CCN(C(=O)Cn2cc(F)ccc2=O)C(CNC(C2(C)CCN(C)C2)=O)C1 C1(C(=O)NC2CC(NC(C(C)CC3CCCO3)=O)C2)COCCOC1 CC(C)(C)C(CNC(C1(NC(c2n[nH]cc2Cl)=O)CCOCC1)=O)CO C(=O)(CC(C)(C)CNC(C1CC1c1ccco1)=O)N1C(CN(C)C)CCC1 c1(CC)cnoc1C(=O)NCC(C)(C)NC(=O)CCOCC1CC1 C(=O)(C1CCc2c[nH]nc21)N1C(CNC(C2CC(F)(F)CS2)=O)CC(O)C1 C1(NC(c2c(OCC)n[nH]c2)=O)CN(C(=O)Cc2cccc(C)c2F)CCC1F C1(NC(C(=O)NCC)=O)CC2CC1CN(C(c1[nH]ccc1COC)=O)C2 Cn1c(O)ncc(C(=O)NCC2CCC(NC(C3(C)CCCS3)=O)C2)c1=O C(c1ccc(S(C)(=O)=O)o1)=CC(N1CC2C(CNC(CCOCC)=O)(C2)C1)=O C1(NC(c2nnc3ccccn23)=O)CC2CCC(C1)N2C(C1CC12CC(O)C2)=O N1(c2ccnc(C)n2)CCC(O)(C(=O)NCCC2CCC(=O)N2)CC1 CC1CN(C(c2ncc(C(F)F)s2)=O)CC(C)N(C(=O)CCn2cncn2)C1 C#CC1CCCC(C(=O)NCC23CC(CN(C(=O)CCC4CCCOC4)C2)C3)C1 C1(OC)CC(CNC(c2cnn(CCO)c2)=O)N(C(=O)CC2CCCCO2)C1 CC1C(C(=O)NC2(CF)CN(C(c3ncn4ccccc34)=O)C2)=NOC1C N1(CCC(C)NC(CCC(=O)NC)=O)CC(CO)CCC1C c1(C(N2CC(O)(C(C)NC(=O)CC3CCCCC3F)C2)=O)cn2c(n1)COCC2 c1(NC(c2cc(CC)cc(C)c2)=O)cccc(Br)c1[N+](=O)[O-] Cc1nc2c(COC(C3(F)CCN(C(=O)OC(C)(C)C)C3)=O)ccnc2[nH]1 N1(C(c2c(C)nn(C)n2)=O)CC2CCC(CNC(C3(C(F)F)CCCC3)=O)C2C1 CC(=O)CCCC(=O)N1CCC(C(=O)NC2CN(C(C)COCC(F)(F)F)C2)CC1 N1(C(CC(=O)OCC)=O)CCCC1(C)C(=O)Nc1cccc(CCO)c1 c1(C(N2CCC(NC(C3CC(O)C3)=O)C2)=O)cc(F)c(Cl)c(Cl)c1 n1(CCC(=O)NCC2(C(=O)NC(C3CCCO3)(C)C)CC2)cnc(=N)[nH]1 c12cccc(n1)CN(C)C(=O)N2.c1(COC(C)C)nnc(-c2cccs2)o1 N1(C(CC2CC(CC)OCC2)=O)CCC2CC(c3cn(C4CC4)nn3)C2C1 S(=O)(=O)(c1cc(C)cnc1N1CC2CCC2C1)NC(C1CCCC1)COC c1(C(C(=O)N(CCCNC(CC=CCC)=O)CC)O)cccc(F)c1 C(=O)(C(CC(C)C)C(N)=O)NCC1N(C(CC(=C=C)C)=O)C2CCC1C2 CCCC(CC)CC(=O)NC1CCN(C(c2csc(C(=O)OC)n2)=O)CC1CO C1(CNC(c2cc(CC)c(C)s2)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CCC1C Cc1cocc1C(=O)NC1CCC(CCC(=O)N(CC(O)CO)CCO)C1 c1(CNC(=O)CN2CCCC(COc3ccccc3)CC2)ccc2nc[nH]c2c1 N1(C(C2CN(C(C)=O)C2)=O)CC(O)(C(F)C(=O)N(C)CC2CCCCO2)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC(NC(=O)CCOCC2CCC2)C(C)(C)C1 C(=O)(CC1=CCCCC1)NC(C1(C(N2CC(CCCC)N(C)CC2)=O)CC1(C)C)=O Cc1ccc(CNC(=NCCc2nccnc2C)NCCF)c(Br)c1 C1(NC(CCSC)=O)(CO)CCCN(C(=O)CCc2ccc(OC)c(OC)c2)C1 c1(C(=O)NCC2N(C(C3(C)CCCNS3(=O)=O)=O)CC2)cccc2c1OCCO2 C1(CN(C(=O)CC2CCSCC2)C)C2CN(C(C3CC4C=CC3O4)=O)CC12 c12ccc(cc1)CCC(=O)N2.N1(C(C=CCC)=O)CCCC1CC(=O)N(C)C.S C1(C(=O)Nc2ccns2)CC12CCN(Cc1ccc(-n3ccnc3)c(Cl)c1)C2 N1(C(C2C(OCC)C2)=O)CCC2CCC(C1)N2C(=O)CCSc1cncnc1 c1(OCC(=O)NCC(CC)NC(=O)Cc2ccco2)ccc(Br)cc1 C1(CNC(Cc2cncc(C)c2)=O)CCN(C(c2cc(=O)n(C)o2)=O)C12CC2 C1(C(C)NC(=O)CNC(=O)NC2CC2)CCN(C(c2cscn2)=O)CC1 c1(C(N2CCCN(C(COCC=C)=O)CC2C)=O)cc2c(cc1Cl)OCCO2 N1(C(C(c2ccccc2Cl)C)=O)CC2CC(C1)C2NC(=O)C=Cc1cocn1 N1(C(C(CC(N)=O)O)=O)CC2OCC(NC(=O)CCCC3CC3)C2C1 C1(NC(CNC(C)=O)=O)(CO)CCN(CC(N2CCOC(CN)C2)=O)CC1 c1(C(N(C2CCC(NC(=O)C(=C3CCCCC3)F)CC2)C)=O)ncnc(O)c1F c1(C(=O)Nc2ncc(OC)cn2)cccc(S(=O)(=O)N2CCNCC2)c1 C1(NC(c2ccnc(C)c2N)=O)CC2CC(C1)N(C(c1cnc(Cl)[nH]1)=O)C2 c1(CC(=O)NCC(C2CC2)NC(CNC(CCC)=O)=O)c(F)cccc1F C(CC(C(=O)NC(C)CC(N)=O)NC(c1csc(C)c1)=O)OC N1(C(C(CC)OCC)=O)CCC(C)(C)C(CNC(C2CCN(C3COC3)C2)=O)C1 c1(C(N2CC(CC(=O)NCC3(CCO)CC3)(OC)C2)=O)cnc(O)c(F)c1 c1(CC)nc(C(=O)NCC(CC)NC(C2C(F)(F)C23CC3)=O)c(Br)s1 Cc1ccc(C)c(C(=O)NC2CCN(C(c3c(C)ncn3OC)=O)CC2C)c1C c1(CC(=O)N(CCNC(C(F)=C(C)C)=O)C2CC2)cn2ccsc2n1 CCCCCCC(O)CCC(=O)N(C)CCOCCNC(c1ncccc1F)=O C1(COC)(NC(c2cscc2OC)=O)CCN(C(c2ocnc2C)=O)C1 C1(CC(N2CCC(OCC=C)C2)=O)CN(C(C2CCCN2C)=O)CC12CC2 C(=O)(C(CCOC)N1CC(O)CC1c1ccccc1OC)OCC C(CC)(CCCC(=O)NCC1(C)NC(=O)NC1=O)NC(c1ccn(CCC)n1)=O CC(C)(C(=O)NCC1CCN1C(=O)CSC(F)(F)F)n1cccn1 C1(NC(C=C(CC)CC)=O)CCCN(C(=O)CCc2ccc(C#N)cc2)C1C CC1CCCN(C(=O)CC(F)(F)Cl)C1CNC(C1CCCOC1C)=O c1(NC(C2CC(=C)CN2C(=O)C(C)OCOC)=O)cccc([N+](=O)[O-])c1F C(CC)(C(=O)NCC=CC(=O)NC1CC(C(=O)NC)C1)OCC C(=O)(C1CCOc2ccccc21)N1CCC2(CCCN(C(c3cocn3)=O)C2)C1 C1(NC(C2(CC)CC2)=O)CN(C(C2CCCC(O)CC2)=O)CC1N=[N+]=[N-] c1(C(N2CCCC(NC(C(F)(F)C3(OC)CC3)=O)C2C)=O)cnn2cccnc12 Cc1ccc(COC(C)CC(=O)NC2C3CN(C(=O)CSCC(N)=O)CC23)cc1 c1(NCC(=O)N(CCN(C(CC2(OC)CCCC2)=O)C)C)cccc(C)c1 Cc1c(Cl)ccc(C(N2CCC(NC(=O)C(F)(F)CO)C(CO)CC2)=O)c1O c1(C(CCO)NCCCC)ccccc1OC(CCN(CC=C)CC=C)=O C(c1nc(C)co1)=CC(=O)NCCCCN(C(CCc1cc(C)on1)=O)C C1(CNC(C(=O)NCc2scc(C(C)C)n2)=O)CN2CCC1(C)CC2 c1(OC)cccc2[nH]cc(CC(=O)N(CCC(C)NC(=O)CC(F)F)C)c12 c1(-c2cn(CCN(C(C3(OC)CCCOC3)=O)C3CC3)nn2)ccc(C#N)c(F)c1 c1(C(=O)NC2C(CC)N(C(c3ccc(Cl)cn3)=O)CCC2)ccn2ccnc2c1 C(=O)(C(CC)(CO)OC)NC(CCC(=O)NC(C(=O)NC)CC1CC1)C C(CC(C)(C)C(=O)NCC1CCC(=O)O1)NC(c1c(CC)nc(C)o1)=O CC(C)C(C)CC(=O)N1CC(NC(=O)CC(=O)N(C)C)CCC1C c1(C(=O)NC(CN(C(C(CC)c2cccnc2)=O)CC)C)snc(C)c1N N12CCOC(C)C1C2=O.C1(C(C)CNC(=O)COc2ccsc2)CC(=O)N(C)C1 N1(C(C(C)CCO)=O)CCC2(CC1)OCCCC2NC(=O)C(C)(C)C1CCCC1 C1(CNC(c2cn(C(C)(C)C)nn2)=O)CC2CC1CN2 C(CN=C(NC1CCC1)N1CCC(N2CCc3ccccc32)CC1)OCC C=CCCCC(C(=O)NCCc1ccccc1O)NC(c1cc(O)n(CC)n1)=O Cn1nc(-c2ccccc2)c2cc(C(N3CC(C)(CO)CC3(C)C)=O)sc12 c1(NC(C2CCC(NC(C3CN(C(=O)NC)C3)=O)C2)=O)ccc(C)c(F)c1 N1(CC(=O)NCC(CNC(CCOC)=O)F)CC(=O)N(C)C1=O C(=O)(CC(O)C(C)C)N(C1CCC(C)(CC)C1)N1CCC(c2nnn(C)n2)CC1 C1(CNC(C2CNC(=O)N2)=O)CCCC2(CN(C(c3sccc3CC#N)=O)C2)O1 C(=O)(C1c2ccccc2OCC1(C)C)NC1CN(C(CCCOC(C)C)=O)C1 N1(C(C=C(C)c2ccco2)=O)CCCC(F)(CNC(=O)CC2CCCN(C)C2)C1 c1(C(=O)NCC2(CNC(C3C4CCC(=O)C34)=O)CC2)cc(OC(F)F)ccc1F C1(NC(c2cc(C)on2)=O)CCN(C)C12CCCN(C(=O)C(C)OCC(C)C)C2 C1(CC)C(CC(=O)NOCCCF)CCCN1C(c1ncsc1C)=O c1(C(N2CCC(C)(CNC(C(C)(C)SC)=O)C2)=O)c(F)cncc1Cl C(=O)(C(O)CC(C)(C)C)NC1(CC)CCCN(C(=O)CSCC(C)C)C1 C1(CN(C(Cc2c(C)ocn2)=O)C)COCCN1C(=O)CC1CCC(=O)NC1 C1(C(=O)NC2COCCC2C(N2CCC3CC23)=O)(CC)CCCCO1 Cc1cc(C(=O)NC2CC(C)CN(C(c3cnccc3C)=O)C2)nc(O)n1 C1(NC(C(C)OC2CCCC2)=O)CCCN(C(c2ccncc2O)=O)CC1 C1(NC(Cc2c(C)nsc2)=O)CCCCN(C(=O)C(C)NC(C2CCC2)=O)C1 C1(CCC)(NC(=O)Cc2cccnc2)CCCN(C(=O)C(C)CCOCC)C1 C(C(=O)NC1(C(=O)N(C(C(N)=O)C2CC2)C)CC1)(C1CC1)SC c1(C(=O)NC2CCCCN(C(=O)C3CC3)C2)n[nH]c2ccc(Br)cc12 C1(CNC(N2C(C(=O)NCC)CCC2)=O)(O)CCC(C)CC1.SCC N1(C(C)C)CCCC(NC(=O)C(CCF)NC(=O)CC2CCC2)C1 C1(C(C)NC(CCCN(C(=O)OC)C)=O)CCCCN1C(=O)C#CC1CC1 C#CCCN=C(NCCc1ccc(C)cc1)NC1CCC(=O)NC(CC(C)C)C1 c1(C(N(CC(CN(C(C(CCC)OC)=O)C)O)C)=O)c(C)ccc2ncccc12 N1(C(C2CCCN(C)C2)=O)CCN(C(c2cnc[nH]2)=O)C(CO)C1 N1(C(CCCC=C)=O)CC(NC(c2c(C)cc(C)nc2S)=O)CCC(O)C1 c1(C(N2CC(CC)C(NC(=O)CCC#N)CC2)=O)cc(S(=O)(=O)N(C)C)c(C)o1 CC(C)C(O)CC(=O)N(CCCOCCN(C(=O)CC1COC(=O)C1)C)C c1(C(=O)NC(CC=CC)C(=O)N(CC(O)CC)C)ncc(C)cc1C Nc1cc(F)ccc1C(=O)NCC1CCN(C(=O)C2=CCSC2)C1 Cc1ccnnc1C(=O)NC1CCC(NC(C2(C)CCC(C)C2)=O)CC1 Cc1cccc([N+](=O)[O-])c1S(=O)(=O)N1CCN(CC(c2ccc(Cl)cc2)O)CC1 C1(C(=O)NC(CCSC)C(=O)NC2CN(C)NC2=O)CCC2CC1CO2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1(C(=O)NCC2(CCC)CCC2)CCOCC1 c1(CCCCC)cc(C(N2CCC(NC(=O)C(F)(F)CC)C2)=O)ccc1F C(CS(=O)(=O)CC(=O)NCc1c[nH]nc1C(N1CC2C=CCC(C2)C1)=O)OC C=CC(CCC)CC(=O)NCc1cccc(NC(=O)CCCCCOC)c1 c1(SCC(=O)NC2C(NC(=O)Cc3cccnc3)CCC2)cccc(C(F)(F)F)c1 C1(C(=O)NC(C(=O)OCC)CO)CC12CCN(Cc1ccc(Cl)c(Br)c1)CC2 c1(C(=O)NC2C(CNC(C3C(CCC)CCC3)=O)CC2)cnncc1NC C1(C)(NC(C(C)OCCC(C)C)=O)CCN(C(C2(C#N)CC=CC2)=O)C1 C1(NC(CSC)=O)CCOCC1NC(=O)CC1CCN(C)C1 N(C1CCc2ccc(F)cc21)C(N1CCN(c2ccc(C)cc2)CC1)=O c1(C(=O)NCCC2CCN(C(c3ccn(C)c3)=O)CC2)cc(F)cc2nn[nH]c12 CC1CC2(CC(C(N3CCC(C(N4CC5CC5C5CC45)=O)C3C)=O)C2)C1 c1(OCC)ccc(C(N2CCC(CO)(NC(=O)CC3C=CCC3)C2)=O)cc1OC N1(C(CCOC)=O)CCN(C(=O)C(=O)NCC(F)(F)F)C2CCC12 N1(C(c2cc(Cl)c(F)c(Cl)c2)=O)CCC2CCCN(C(C3CCC3)=O)C2C1 c1(C(N(C)CC2CCCN2C(C2(C)CC2(F)F)=O)=O)cc(Cl)cn1C c1(C(N2C(CN(C(=O)CC3CC(=O)NC3=O)CC)CCC2)=O)cc(C)ccc1Cl CC1(NC(=O)Cn2cccn2)CN(C(C2CCCS2)=O)C1 c1(NC(N(C2CCCC2)CCC#C)=O)nc2ccc(C#N)cc2s1 Cc1nc(C2CC2)ccc1C(N1CC(NC(=O)C(=O)CC(C)C)CC(C)C1)=O C(=O)(C1Cc2ccc(F)cc21)N(C1CCCN(C(c2nccc(CC)c2)=O)C1)C Cn1cc2cccc(CNC(C3CCCN(S(=O)(=O)CC4CCC4)CC3)=O)c2n1 N#Cc1ccc(NC(C2C3CCC(C3)N2C(c2cccnc2Cl)=O)=O)c(O)c1 C(=O)(CCCCCF)N1CCC(CC2CCN(C(c3ccc(C)cc3)=O)CC2)CC1 C1(C2CCCC2)(C(=O)NCc2cccc(NC(=O)CC3C=CCC3)c2)CCCCC1 C(C(CC)=Cc1cccnc1)(C(=O)NCc1nnn(C)n1)N1C(CC)CCC1 C(C1C(=O)N2CCC(C2)NCc2coc1n2)OCC.c12cn(nn1)C2.N(C)C.OC c1(N2CC(CNC(=O)C=Cc3ccncc3)C2)ncnc2sc3c(c12)CCC3 C1(OC)CC(NC(=O)C=CCO)CN(C(=O)C=CC(C)C)C1 CC1CC(NC(=O)C=CCN(CC(F)(F)F)C)CN1C(=O)CSC1(F)CC1 N1(CCC)CCCC(C(=O)NCC2(CNC(c3nnn(C)n3)=O)CCCC2)C1 C(c1ccc(C)cc1)=CC(N1CCC(O)(C(CNC(COCC#C)=O)C)C1)=O c1(C(=O)NC(C(=O)NC(c2cccnc2)C)c2ccoc2)cnc(Cl)nc1 N1(CCC)CCC(NC(=O)C(=O)NC2CCCC2c2ccccc2)CC1 N1(C(C(CC)(F)F)=O)CCN(C)C(CNC(c2cc(C3CCCC3)n(C)n2)=O)C1 c1(C(=O)NCC2C(CNC(CCC(C)OCC)=O)C2)ccc2c(c1)CCCO2 c1(C(N(CCCNC(=O)CC2CC(F)(F)C2)C)=O)cnc2c(F)c(F)ccc2c1 c1(C(=O)NC(CC)CN(C(=O)CCOCC(C)C)CC)ccc(C)cc1C1CC1 C1(C)(C(=O)OC(C)C(=O)Nc2cnn(C)c2)C=CCCC1 C12(NC(CCCOCCOC)=O)CCC(CC1NC(c1cncc(CO)c1)=O)C2 N1(C(C2CCC(C)(C)O2)=O)CCOCC(NC(c2c[nH]cc(Br)c2=N)=O)C1 C1(C(N2CC(F)(CNC(C(C)n3cccn3)=O)C2)=O)CCn2nncc2C1 C1(N(c2cnn(C)c2)CCOC)CCN(C2CCN(C(=O)OC(C)(C)C)C2)CC1 c1(N(CCOC)CCNC(=O)CCCOC)cc(C)c([N+](=O)[O-])cc1F c1(C(N2C3C(CNC(C4(COC)CC4)=O)C(C3)C2)=O)ccc2ccccc2c1 C1(C(CO)NC(CCN(c2ccccn2)C)=O)CCN(C(=O)Cn2cnnc2)CC1 c1(CNC(N2CC3CC3(NCc3ccc(C(F)F)cn3)C2)=O)cccc(F)c1 c1(C(N2CCOCC(NC(C#CC(C)C)=O)C2)=O)cc(Cl)cc(Cl)c1O c1(OC)nccc(Cl)c1C(=O)NCC1CCCN1c1nc(C)ns1 N1(CC)CCN(C(C2CN(C(c3cc(C)ncc3C)=O)C(C)(C)C2)=O)C(C)C1 c1(CNC(NC(C=C)C)=NCCC2CCN(C)CC2)c(F)cc(COC)cc1F N1(C(c2nccc(OC)c2F)=O)CCOC2(C1)CN(C(C1CCC(=O)N1C)=O)C2 C(=O)(CC(C)CC(F)(F)F)NC(CC)CN(C)C(c1cc(F)c[nH]1)=O c1(C(=O)NCCOCCNC(CCC#C)=O)coc2ccc(F)cc12 c1(C(=O)NC(C(=O)NCC(C)NC(=O)OC)C2CC2)cc(C)c(C)cn1 CN1N=C(CC(=O)N2CC3CCC2CN3C(c2cnn(CC3CC3)c2)=O)CC1=O C1(NC(=O)C(C2(O)CCCCC2)F)CCCN(Cc2ccccc2)CC1 c1(C(=O)NCCC2(NC(C3C(C)CCCC3)=O)CC2)ccn2c(O)nnc2c1 O=C1CC(CC(=O)NC2C3CN(C(C4(CO)CCCC4)=O)CC23)=NN1 c1(C(=O)NC2CCCC(N(C)C(c3cccc(N)n3)=O)C2)ccn2cnnc2c1 N1(c2ccc(C#N)cn2)CCC(CNC(=O)C=CC(N)=O)C(F)(F)CC1 N1(C(C=NOC)=O)CCC(C2CCN(C(=O)CCn3ccc(C)n3)C2)C1 C1(C(N2CC3CC2CC3O)=O)(CC)CCN(C(=O)CN2C(=O)CNC2=O)CC1 CN1CC(NC(=O)CN(C(=O)C=Cc2ccnn2C)CC2CC2)CC1=O c1(C(NOCC(n2cc(Cc3nccs3)nn2)C)=O)ccnn(C)c1=O N1(C(C(C)(C)c2nccs2)=O)CCC(CO)C(NC(c2cnns2)=O)C1 C1(CC=C)(NC(c2ncc(F)cn2)=O)CCN(C(c2cccn2C(C)C)=O)CC1 C12(C(=O)NCC(C(C)C)O)CCN(C(C3CC4(CCC4)C3)=O)CCC1C2 c1(C(=O)NC2CCC(NC(c3c(C)noc3C3CC3)=O)C2)ccc(N)c(F)c1F c1(CC)c(NC(CNC(c2sccc2C)=O)C(C)C(C)C)ncnc1Cl CC(C)C(C#N)C(=O)NCC1CCCC(CNC(=O)C(C(C)O)N(C)C)C1 c1(CNc2cccc(C(N3CCC(C(N(C)C)=O)C3)=O)c2)csc([N+](=O)[O-])c1 c1(C(N2CCC(N(C(CSCC=C)=O)C)C2)=O)c(C)cc(C)c(Br)c1C c1(C(=O)NC2CN(C(c3cnn(C(C)C)n3)=O)CC2C)cnc2[nH]c(O)nc2c1 N1(C(CCC2C(C)=NNC2=O)=O)CC2CC(NC(c3cnc(S)nc3)=O)CC2C1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C(C(N2CC(C)CC(C)C2)=O)CCC1 C1(F)(CNC(C2N(S(C)(=O)=O)CC2)=O)CCN(C(=O)C(F)CC2CC2)C1 c1(C(N2CC(N(C(=O)C(=O)NC3CC3)C)C(F)C2)=O)cccc(O)c1F C1(C)(CNC(CCCC#CC)=O)COCCN(C(C2CCCC(=O)N2C)=O)C1 c1(OC)cccc(OCCC(=O)NCC(C)N(C(=O)COCCSC)C)c1 CC1CCC(NC(=O)C(F)Cc2ccccc2)CN1C(c1ccc(O)c(Cl)n1)=O c1(C(=O)NCC2N(C(c3cnn(C)c3F)=O)CC2)cncc(P(C)(C)=O)c1 N1(C(CCOCC(C)C)=O)CC(NC(=O)CCCF)CC(C)C1 c1(C(C)(C)C)n[nH]cc1C(=O)NCC1(CNC(=O)Cn2nnc(=N)[nH]2)CC1 c1(OC)ncc(-c2ccnc(N3CCN(C(=O)C=Cc4cccs4)CC3)c2)cc1C C12CCC(C1)NC2=O.C(CN(C)C(C1CC1c1ccco1)=O)(CC)OC c1(C(=O)OC)ccc2[nH]c(C(=O)NCc3nc(=N)n(C)[nH]3)c(C)c2c1 Cc1ncnc(C(N2CC(C)(C(=O)Nc3c[nH]ccc3=O)C2)=O)c1C N1(C(C(CCC)C)=O)CCC(F)(F)C(NC(c2cc(OC)ccn2)=O)C1 Cc1cc(C(=O)NC(C)CCCNC(=O)COCC2CCCO2)nc(N(C)C)n1 CC(C)C(Cc1ccccc1)N=c1nc(N2CCCC(SC)C2)c2c([nH]1)CCC2 c1(C(C)NN2CCN(C(=O)NC3CCC(C)(C)CO3)CC2)cc(Cl)ccc1F CC(C)CC(C)C(=O)NCCCNC(c1ccc(C#N)n1C)=O C1(C(=O)NC2CC3CCC2(CNC(=O)C(F)(F)CO)C3)CC2C=CC1C21CC1 n1(C2CCCN(C(c3cc(C)[nH]n3)=O)C2)cnc2c1CCN(C(C1CSC1)=O)C2 C(=O)(C1(C)CCc2ccccc21)NC1CCN(C(C(C)OCC#C)=O)C1C N1(CC(=O)NC2(C)CCCO2)C(=O)NC(C)(c2ccc(F)cc2)C1=O Cc1oc(C#N)cc1C(=O)NCC(C)(C)CCNC(c1ccc(F)c(Cl)c1)=O C(=O)(NNc1cc(F)cc(Br)c1)NC(C)CCC1CCCCC1 CC1(CO)CCN(C(c2cc(C#N)c[nH]2)=O)CC1 c1(C(=O)OC)ccc(CC(=O)NC2(CNC(c3ccncn3)=O)CCC2)cc1F C12(NC(C3CCC(OC)CC3)=O)CCC1CN(C(=O)Cc1ccc(F)cc1Cl)C2 C1(C(C)NC(c2c(C)ccs2)=O)CCCN(C(c2csc(CS(C)(=O)=O)n2)=O)C1 C=C(C)C(O)CC(=O)NCC1CCN1C(c1cc(Oc2ccccc2Cl)ccn1)=O c1(NC(c2nnc(-c3cnc[nH]3)o2)=O)ccc(Br)c(Cl)c1 c1(OC)ccc(C(=O)NC2CN(C(C3OCC3(C)C)=O)C2)cc1OCCO S(=O)(=O)(c1cccnc1)NC(=O)CCc1ccccc1O C(CC(C)(C)COC)NC(CC1N(C(c2c(CCC)nco2)=O)CC1)=O C1(CN=C(NCC2C(C)C2)N2CC(N3CCCC3)C2)CCC2(CC1)CC2 c1(C(N2C3CC(NC(CC(C)C)=O)C(C3)C2)=O)cc2n(n1)CCCC2 N1(C(CCCCCCC)=O)C2CCC1C(C)C(NC(=O)C(C)CCCOC)C2 C12(C(=O)NC3CC(C#C)(O)C3)CCC(CN=c3ccc(N(C)C)c[nH]3)(CC1)CC2 c1(C2(C(=O)NCC(CCOC)NC(=O)OC(C)(C)C)CC2)ccc(F)cc1C C1(NC(C2C(C=C)CC2)=O)CN(C(c2ccncc2C)=O)CC2(CC2)C1 C(=O)(C1=CCCOCC1)N1CC2C(NC(C3CCC4(CC3)N=N4)=O)C2C1 N1(C(c2c(Cl)cn(CCC)n2)=O)CC2CC(C)N(C(=O)Cc3ncc(C)[nH]3)C2C1 c1(C(=O)NC2CN(C(C3(COC)CCCO3)=O)CC2C)ncc(F)cc1N CN1CCN(C2COCC2CNC(=O)NCCCC(=O)Nc2ccccc2)CC1 C1(CNC(c2nn(CC)c(C)c2)=O)CCCCCN1C(=O)C(C)Cc1ccco1 c1(CCOC(CCSCC(=O)OCc2ccccc2)=O)cccc(Cl)c1F C1(NC(c2cncn2C2CC2)=O)CC(CO)N(C(c2ncc(C(F)F)s2)=O)C1 N1(Cc2ccc(OC)cc2F)CCC2(CN(C(c3ccc(Cl)nc3Cl)=O)C2)C1 Cc1csc2ccc(C(=O)CC(=O)CN=c3cc[nH]cc3)cc12 C1(CCCC)CN(C(C2CCC(C(F)(F)F)O2)=O)CCN1C(C12CCC(C1)C2)=O c1(SCC(N2CC(=C(CNC(C3CCCSC3)=O)F)C2)=O)nc2ccccc2s1 S(=O)(=O)(c1ccc(Sc2ccoc2)c(F)c1)N(C)NC1(COC)CC1 CN=c1[nH]c(=NCCCCc2ncc[nH]2)[nH]c(=NC2CCC3CCC2C3)[nH]1 N1(C(C(C)OCc2cccc(Cl)c2)=O)CC(CNC(=O)C(C)(F)F)C(F)(F)C1 c1(C(N2CCCC(n3cc(-c4cccs4)nn3)CC2)=O)c(C2CC2)cccc1N c1(CNC2(c3n(CCCSC)nnn3)CCC(C(C)C)C2)cc(C)nnc1O CC(CC(=O)NC1C2CC1N(C(C1CC(CC(F)(F)F)C1)=O)C2)C(C)(C)C C12(CC(=O)N(CCCCCCNC(C3CCCO3)=O)C)CC3CC(CC(C3)C1)C2 N1(C(C2C(C)(C)NC(=O)C2)=O)CCN(C(c2csc3nnsc23)=O)CC(O)C1 N1(C(C(CC=C)OC)=O)CC(CNC(c2ncccc2COC)=O)CC1(C)C c1(C(=O)NCC(C(C)C)NC(CC(CC)C)=O)ccc(Br)cc1C(C)C c1(OC)c(C(N2CC(NC(C3COCCN3C)=O)CC2CO)=O)cc(F)cc1F n1(CCOC)nccc1C(=O)NCC(CO)NC(c1snnc1C(C)C)=O CC(C(=O)N1CC(C(=O)NCCNC(=O)CC2CC2)C1)C1(O)CCC1 c12ccc(C)n3cc1nc23.Cc1cc(Br)ccc1NC=O.c1(C)cccc(Cl)c1Cl C1(CNC(=O)C(c2ccccc2)F)CCCC(CNC(c2cc(CO)on2)=O)C1 N1(C(c2[nH]n(C)c(=O)n2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C1(C)C C(=O)(C(C)CCC(C)(C)C)N(CCOCC#C)CC.C1(=O)C(CCCC=C)N1 CCC(C#N)C(=O)N1CCC(c2ccccc2)(NC(c2ccsc2Br)=O)C1 CCCC(CC)CCC(=O)NC(CN(C(=O)CNC(=O)CCC(C)C)C)(CO)CO C12(C(N(C3CC(NC(=O)C(C)(O)c4ccccc4)C3)C)=O)CC(F)(C1)C2 c1(OCC(N2C(C)CC(NC(C3(C#C)CCCC3)=O)C2)=O)c(CC)cccc1C c1(C(N)=O)n[nH]c2c1CCN(C(C1CN(Cc3c(F)cc(F)cc3Br)C1)=O)C2 C1(NC(c2cn(CC)nn2)=O)CCCCC1N(C(=O)CCc1ccc(F)cc1)C c1(C(=O)NCC=CCNC(C2C(CCC)CCC2)=O)cc(N)ccc1SC c1(C(=O)NC2CC(F)(CNC(CCCC=C)=O)C2)cc(F)c(F)c(N)c1Cl N1(C(CC(C)CN(C)C)=O)CCC(NC(c2ccc(C(F)F)nc2)=O)C(CO)C1 c1(C(c2n(CCC)nnn2)NCC(C)Cn2ccnc2)nc(Br)c(C)cc1F C1(NC(C(CC)N(C)C)=O)CC2(C1)CC(NC(C1CCCN1C)=O)C2 n1(CC)cnc2nc(=NC(C)CC3CC3)[nH]c(NCCc3c(Cl)cccc3Cl)c12 N1(C(C(=O)N(C(C)C)CCO)=O)CCCNCCC1C C1(NC(c2cccc(NC)n2)=O)(CO)CCN(C(=O)C(C)=O)CC1 c1(C(N2C(C(=O)NCC=C)CCCC2)=O)cnc2onc(C)c2c1 C1(CNC(CC(C=C)C)=O)CC(C)CN(C(c2ncccc2Cl)=O)C1 c1(C(=O)NCC(CNC(c2csc([N+](=O)[O-])c2)=O)OC)ccc2nccn2c1 c1(C(=O)NC2CCC(C)N(C(=O)CP(C)(C)=O)C2)cc2ccccc2nn1 C1(N(C(=O)NCCC2CCN(C(=O)OC(C)(C)C)C2)C2CC2)CCC12CCNCC2 c1(C(=O)NCC2C(NC(C3C(C(=O)OC)C3)=O)C2)ccc2c3c(cccc13)CC2 N1(C(C=C(C)C)=O)CCN(C(C2CCCCC2O)=O)CC1c1ccccc1 Cc1cccc(-c2cncc(Cn3cnc(C(=O)O)n3)c2)c1 N1(C(C2COCCN(C(c3n(C)ncc3)=O)C2)=O)CCc2ccc(O)cc21 N1(C(c2ccc(OC)c(C)c2)C(=O)NC2CC2)CCC2(CC1)CC(OC)C2 c1(-n2cc(C(C)N(C(=O)C(C)N(C)C)C)nn2)ccc2nc(C(=O)O)oc2c1 c1(C(=O)NCC2N(C(CC(C=C)CC)=O)CCC2)c(OC)ccc2c1CCC2 C(CNC(c1occc1C1CC1)=O)(CCNC(=O)C(CSC1CC1)OC)OC c1(C(N2CCC(NC(C3(O)CN4CCC3CC4)=O)C2)=O)ccc(F)c2occc12 CN1CC=C(CC(=O)N2CCC(C(C)(C)NC(=O)CCc3nc(O)n[nH]3)C2)CC1 c1(NC(CC)CC(F)(F)F)ccc(S(=O)(=O)NCC(O)COC)c(Cl)c1 C(CCCC(C)NC(=O)CC(C)(C)C1CC1)NC(C(C)OC1CCCC1)=O C1(NC(=O)Cc2cnc[nH]2)CCC(NC(c2ccc(C3CCCO3)[nH]2)=O)CC1 C(=O)(C1=CC(C)(C)C1)N(CC(C)NC(c1ccc(CN2CCSCC2)cc1)=O)C C=CCC(C)(C)CC(=O)NCC(C)(CO)NC(c1ccc(F)c(CO)c1)=O CON1CC(C(=O)NC2CN(C(=O)CN3CCCCCC3)CC23CC3)CC1=O C1(CC)OCCC1C(=O)N(C(C)(C(=O)NCC(F)(F)Cl)C1CC1)C C(=O)(C(C)(C)CC(=O)N1CCCN(C(=O)COC(c2nccn2C)C)CC1)OC Cc1cc(C)n(C(C)CC(=O)NC(CNC(C2SCCCS2)=O)CC(C)C)n1 C1(C2C(C(NOCCC(C)(C)O)=O)C2)CCCN(C(C2(C#N)CC(=O)C2)=O)C1 CS(=O)(=O)c1ccsc1CNc1ncc(Br)cc1CO C12(CNC(CC3N(C(=O)OC)CCC3)=O)CC1CN(C(=O)C=C1CCC1)C2 c1(C(Cn2cc(C3CC(C(=O)O)(C(=O)O)C3)nn2)(F)F)cc(F)cc(F)c1 N1(C(CN(C(=O)C(F)CCC(C)C)CCOC)=O)CCCCC(C)(F)C1 CCCC(C(O)C(=O)NCCC#CCO)NC(=O)C(C)NC(=O)CC C1(NC(C(C(C)O)C)=O)CCCN(C(c2ccc(C3CC3)cc2Cl)=O)CCC1 C(CCCC(=O)N1CCCC1CCNC(c1c(C)cccc1F)=O)(OC)OC C12(C(N3CC(CNC(=O)CCCOc4cccnc4)C3)=O)CCCCN1CCC2 N1(C(CC)=O)CCC2(C1)CN(C(C1CCC(O)CN1C)=O)C2 n1(C(C)C)ncc(C(=O)NC2CC(CNC(=O)C(C)(C)c3cscn3)C2)c1Cl C1(C(N2CC3C(NC(C4(CSC)CCC4)=O)C3C2)=O)CCn2nccc2C1 c1(C(N2CCCC(O)(CNC(C(CCC)C)=O)C2)=O)ccc(C)c(F)c1F N1(C(C=CC(C)(C)SC)=O)CCOCC(C(=O)N(CCO)CC2CC2)C1 Cc1ncnc(C)c1CC(=O)N(C)CCNC(=O)CCCN1C(=O)CN(C)C1=O N1(C(CC(CNC(C(CCC(C)C)F)=O)C)=O)CCCC2(CCCO2)C1 N1(C(Cn2ccc(C)n2)=O)CCC(O)(CN(C(=O)CN2CCC2C)C)C1 N1(C(CN(C(C(CSC)O)=O)C)=O)CCC2(CCCOC2)C1 C1(CNC(c2cn(C(F)(F)CO)nn2)=O)(NC(c2cc(Cl)cs2)=O)CCCC1 c1(C(=O)NCC(C(=O)N(CCOC)CCF)C)ccnc(OC)c1 c1(C(=O)NC2CCN(C(C3CCCS(=O)(=O)N3)=O)C2)cnc2sccn2c1=O N1(C(C=CCCC)=O)CC(NC(c2ccco2)=O)CC12CCCC2 N1(CCC)CCc2cccc(C)c21.C(CCC(F)(F)F)c1cn(C(C(=O)NC)C)nn1 c1(C(=O)OC)ccc(C(F)(F)F)nc1N.c12cccc(c1)CN(C)C2 c1(CC2(C(=O)NCC#CCNC(c3cc(O)ncn3)=O)CC2)ccc(F)cc1 c1(C(=O)NCC(C)CNC(c2ccnc(NC(=O)OC)c2)=O)ccc(Cl)c(O)c1 c12ccn(c1)CCNC(=O)C1(CC1C)NC2=O.C1(C(C)C)(OC)CC1 N1(C(C#CC(C)C)=O)CCN(C(C2CN(C)C(=O)N2)=O)CC1c1nccn1C S(=O)(=O)(c1cccc2scnc12)N1C(C(N2CCC(CCO)CC2)=O)CSCC1 C(=O)(C(C)(CC)C(=O)N1CCC(F)(F)C(CNC(c2cc(C)co2)=O)C1)OCC C12(NC(c3ccn(C)c3)=O)CC1CN(C(c1ccccc1C1(C)CC1)=O)C2 c1(C(=O)NCC(CC)NC(c2ccc(-c3ccc(Cl)cc3)[nH]2)=O)ccc(O)nc1 CC1CC(NC(=O)CCc2cccc(O)c2)CN1C(=O)CCOC1COC1 N1(C(C(C2CC2)SC)=O)CC2C(CNC(C3CC(n4cnnc4)C3)=O)C2C1 C(=O)(CCC(C)SC)NCCNC(C1CN(C(Cc2nc(C(C)C)sc2)=O)C1)=O N1(c2snc(CC)n2)CC2CCC1CN2C(C1CCCC2CCCN12)=O Cc1ccc(C2CCC2COC(C2CCCC(=O)N2)=O)c(C)c1 N1(C(C(N(C)C(C23CCCC2C3)=O)C2CC2)=O)CC2(C1)CC(C)(O)C2 c1(C(N(CC(C)NC(=O)Cc2nc([N+](=O)[O-])n[nH]2)CC)=O)ccn2nccc2c1 C12(NC(c3cnc(CC)s3)=O)CN(C(C3(C)CCOCC3)=O)CC1CS(=O)(=O)C2 c1(C(N(C(=O)CCCCCl)C(C2CCCNC2)C)=O)cc2cc(Br)cnc2s1 C=CC1CCCN1C(C1CCOC1CNC(=O)CC(C)C)=O C1(NC(C2N(C(C=C(CC)CC)=O)CCOC2)=O)CCc2nncn2C1 c1(NC(CC)CC#N)ncnc(N2CCOC(COC)CC2)c1C N1(C(CCOCCC)=O)CCC(NC(=O)Cc2cc(OC)ccc2OC)C(O)C1 C1(CNC(C2(CC)CCCC2)=O)CCN(C(=O)CC2CCC(=O)N2)CC1C CC1(C)CCc2[nH]c(C(N3CC4C(NC(C5CC(F)(F)C5)=O)C4C3)=O)cc2C1 c1(C(N2CC(N(C(c3cnc(C(C)=O)s3)=O)C)C2)=O)nccnc1C(N)=O C1(CNC(c2c(C)n(C)cn2)=O)CN(C(C2(C)CC=CC2)=O)CC(C)(C)O1 n1(C(C)(C)C)ncc(CN(C2CCC(N)C2)C=O)c1Cl C(C(O)C(F)(F)F)C(=O)NCC(C1CCCC1)NC(=O)C=CC1CCCC1 C1(C(N2CC(NC(c3c(CC)cccc3)=O)C(OC)C2)=O)COC2(CCC2)C1 Cc1cnnc(O)c1C(N1CC2CC(NC(=O)CSS(C)(=O)=O)C1C2)=O Cc1cc(F)cc(C)c1C(=O)NC1CCCCN(S(=O)(=O)c2nccs2)C1 C1(O)(CCNC(C)=O)CCN(C(c2ccc(Cn3ccnc3)o2)=O)C1 c1(NC(C2CCCC(NC(c3c(C)c(F)ccc3)=O)C2)=O)nc(Cl)c(C)c(Cl)n1 N1(C(c2nc(C)[nH]n2)=O)CC(NC(C23CC(CN2C2CC2)C3)=O)CC(C)C1 C(c1ccccc1Br)=CC(=O)NC(C1CN(C(C2C(C)C2)=O)C1)C c1(C(=O)NCC(=CC(N2CC(OCC(=O)NC)C2)=O)C)cccn1C C1(C(=O)NCc2c(C)ncs2)COCCN(C(C2CCC(C)CC2)=O)C1 c1(C(c2ccco2)NC2CN(C(CNC(C)=O)=O)C2)cc2ccccc2o1 CCC(O)C(=O)NCCCCCNC(=O)CCNC(=O)C(C)(C)C CC(Cc1cccc(F)c1)CC(=O)NC1CCC1NC(=O)Cc1cscn1 C1(CCC)CN(C(=O)Cc2cocn2)CCN1C(=O)C=Cc1csc(C)n1 c1(SC)ncc(C#N)c(NC2CC(CC(=O)Nc3ccc(Cl)c(Cl)c3Cl)C2)n1 c1(OCCNC(c2nnc(C)s2)c2nnnn2C)ccccc1F N1(C(C2(OCC)CC2)=O)CCC(F)(CNC(c2cccc(C(C)C)n2)=O)C1 C1(C(C)CNC(C2CCN2S(C)(=O)=O)=O)CCN(C(=O)Cn2cnccc2=O)CC1 C1(c2nc(C(C)C)no2)(NC(C)=O)CCN(Cc2cnc(C)o2)CC1 N#Cc1cc(NC2CN(C(c3cnns3)=O)CC3(CCC3)C2)c([N+](=O)[O-])cc1F C(=O)(C(F)(F)C(O)CC)NCC1OCCN(C(C(CCC)N(C)C)=O)C1 CCC(CN(C)C)CC(=O)NC1(CNC(c2cc(OC)ccc2OC)=O)CC1 N1(C(C=C(C)C(C)C)=O)CC2CC(NC(=O)CC3CCC(=O)N3C)CC2C1 c1(OC)cc(C(N2C3CCC2CC(CNC(=O)C(C)CF)C3)=O)c(OC)cc1Cl C1(CCNC(c2c(C(C)C)ccs2)=O)CN(C(=O)C=Cc2ncco2)CCO1 c1(N(C)C)ccc(C(=O)N(C2CN(C(c3cccn3C)=O)CC2F)C)cc1 C1(NC(CC2(OCC)CCC2)=O)(CO)CCCC1.C1C(CC)OCC(=O)N1 CC1CC(CNC(c2[nH]c(=N)sc2C(F)(F)F)=O)CN1C(=O)C=C(Cl)Cl C#Cc1cccc(CC(=O)NCC2CC(C(=O)Nc3cnn(CCOC)c3)=NO2)c1 CN1CCC(C(=O)NC2(C3CCCN3C(=O)CS(N)(=O)=O)CC2)c2ccccc21 O=C(CC(CC1CC1)C(=O)O)Nc1ccc(Oc2ncccc2F)cc1 C1(NC(CC)=O)(CNC(c2ccn(CCF)n2)=O)CC2CCC1CC2 c1(C(=O)NC2C(NC(CCSCC)=O)CS(=O)(=O)C2)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N(C(C)CNC(=O)C(O)C(C)(C)C)C)=O)ccc2cc([N+](=O)[O-])ccc2n1 c1(C(=O)NCC2OCCN(C(c3cc(C)sc3)=O)C2)cc(O)c2sccc2c1 C1(C(=O)NCCCC(C)NC(CC(COC)C)=O)CCCC(C)CC1 C1(NC(c2cncc(SC)c2)=O)C(C)CN(C(=O)Cn2ncccc2=O)CC1C c1(C(=O)NCCC(CNC(=O)C(C2CC2)N(C)C)OC)cn(C)c(C)n1 N1(C(c2cc(OC)cc(OC)c2)=O)CC2(CCC(C(=O)NC3CN(C)C3)O2)C1 N(C1CCCn2nc(C)nc21)CC12CC(C(=O)OCC)(C1)C(C)(C)O2 c1(OC)cc(F)c(C(N2CCC(C3CCCCN3C(=O)CC3CC3)C2)=O)c(F)c1 C(=O)(C(C(C)(C)C)NC(=O)CC1CCC(C)(C)C1)NCc1c(C)con1 c1(OC(C(=O)NC(CC)CN(C)C(c2cc(F)n(C)n2)=O)C)ccc(F)c(F)c1 C(=O)(C(F)(F)C(F)F)N(C(c1nccc(N)c1)=O)CCC(F)(F)F.C12(O)CN(C1)C2 C(=O)(C(C)C(C)(C)C)NC(C(C1(O)CN(C(C2(C(C)=O)CC2)=O)C1)F)=O Cn1cnc2c(C(=O)NCCNC(=O)COC3CCCCC3)cccc12 N1(C(c2n(C(CC)C)ncc2)=O)CC2CC1CN(C(=O)CN1CCC(O)CC1)C2 CC(C)CCC(=O)NC1CC(O)(CNC(c2ccccc2-c2cncnc2)=O)C1 CC1CCN(C(=O)C(=O)Nc2cn(C3CC3)nn2)C1CSc1ccccc1Cl c1(N2CC(SC)CC3(C2)CC3)ncnc2ncc(Br)cc12 c1(CC)noc(CC)c1CC(=O)NC1CC(NC(c2c(C)cnn2C)=O)C1 CC(C)(CN=c1[nH]c(=NCCN2CCCCC2=O)[nH]c2c1CSC2)C(N)=O N1(C(CC(C)C)=O)CCC(NC(=O)Nc2ccc(Oc3nccs3)cc2)C(C)C1 c1(OC)nccc(I)c1CNC(C1CC1OC)=O.C12(F)CCC(CC1)C(=O)N2 c1(C(=O)NC2CCC(CCNC(C=C(C)C)=O)C2)c(C)sc(C)c1C#N C(=O)(C(O)C(C(C)C)OC)NC(CSCC)C(=O)NCc1ccc(C)c(O)n1 C#Cc1ccc(C(=O)NC(CNC(C2CC(C3CC3)=NO2)=O)CO)cc1 Cc1cc(C#N)ccc1C(N1CC(CNC(C2(C)CC2C)=O)C(O)C1)=O N1(C(C(C)C2CC2)=O)CCC(NC(=O)COC2CCC(F)(F)CC2)C(O)C1 c1(C(N2C(CNC(C3CCSCC3)=O)CCC2)=O)cnn2c(Cl)cccc12 c1(C(=O)NCC2N(C(CCC=CC)=O)CC(F)(F)C2)ccc(OC)c(S(N)(=O)=O)c1 CC1CN(C(C(=O)NCCCC2CC2)C2=NOCC2)C(C)(C)CO1 C1(C(N2CCN(CC(C)O)CC2)=O)(SCC=C(C)C)CC(C)(C)C1 C=CCC(C(=O)N1CCCC(N(C(c2cnc(O)c(C)c2)=O)CC)C1)C(C)C CC1CCN(C(=O)COCCCF)CC1NC(=O)C(C)(C)O C(C(O)CC(=O)N1CC(CO)C(O)C1)NC(c1ncccn1)=O C(C(C)CC(=O)NCC1CCC(F)(F)C1)NC(CNC(C)=O)=O N1(C(C(C2CCC2)OC)=O)CC(NC(=O)C(C)C)CC12CCCC2 N1(C(c2c(C)c(F)ccc2)=O)CCCC(NC(=O)Cc2ccsn2)C(F)C1 C1(CC=C)(NC(=O)COC2CC=CC2)CCN(C(C2(CF)CC2)=O)CC1 c1(-c2cnc(CC)[nH]2)nc(-c2ccc(C)cc2)nn1-c1ccnnc1 c1(-n2ncc(CN3CCC(C#N)C3)c2)nc2ccccc2o1 Cc1nn(CCO)cc1C(=O)NCC(C)N(C)C(C1CCC1(C)C)=O.S(C)(=O)(=O)NCC Cc1cc(C(=O)NCC2C=CC(NC(=O)CC3CC(C)C3)C2)cc([N+](=O)[O-])c1Cl CC(CC(=O)NCCc1ocnc1CNC(=O)C(O)CC1CCCC1)CC(C)(C)C N1(CCOCC)CCC2(CC1)COC(CN)C2.C1(C)(O)CCCC1 C1(O)(C(C)C)CCCN(C(=O)CC(C)(C)CNC(c2cccc(CO)n2)=O)C1 N1(C(c2ncn(CC)c2)=O)CC2CCN(C(C34CCC(C3)C4)=O)CC12 c1(C(=O)NCCC(C)NC(CCOCC)=O)c(C)ncn(C)c1=O N1(Cc2c(OC)cccc2)CCOC(C(N2CC(O)CC2CO)=O)C1 C(CCCNC(=O)CC1(CSCCOC)CC1)SCC#C.C(=O)(C(C)=CC1CC1)NC Cc1cc(C(N2CCN(C(c3cocn3)=O)C(C3CC3)C2)=O)cc(OC)n1.C1(C)CC1 c1(OC)ccc2c(c1)C(N(C=O)Cc1cc(Br)c(Br)cn1)CCC2 c1(C(C(=O)NC(C(C)NC(CCCc2scc(C)n2)=O)(C)C)C)cn(C)nc1C C12(NC(C3C(NC(C4C(C)(C)OCC4)=O)CCO3)=O)CCC(CC1O)C2 c1(CC)cccc(C)c1NC(=O)C(c1cccc(Br)n1)N1CCCC(CCF)C1 N1(C(c2c(C)nco2)=O)CCC(C2CC2)(CNC(=O)C=CC(F)(F)F)C1 N1(C(CC2(CNC(CC3CCCN(C)C3)=O)CC2)=O)CCCC(C2CCC2)C1 Cn1nc(C2CC2)cc1C(N1CC(CNC(=O)Cn2cnnc2)C2CC12)=O CCC(C)(CC(=O)N1CC(C)(NC(C2CC=CC(O)C2)=O)C1)C(=O)OC C(=O)(C1=CCCN(C(C2CCC(N(C)C)C2)=O)C1)Nc1cc(C)cc(C)c1 c1(N2CC(C(C)NC(c3cc(C)ns3)=O)OCC2)ncc([N+](=O)[O-])cn1 c1(C(=O)NC2(CNC(C34CCCC3OCC4)=O)CCOC2)ccc(F)c(O)c1 N1(C(C2CCN(C(c3cc(C)c(C)nc3)=O)C2C)=O)CC2COC(=O)C2C1 N1(C(C(C)Cc2ccccc2)=O)CC2CCC(NC(=O)C(C)C(C)O)CC2C1 C1(C(=O)NC2(CC=C)CC=CC2)CC(=C)CCN1C(c1nnc(S)n1C)=O C12(NC(CCCCC(CC)C)=O)CC(C)(C1)OC21CN(C(=O)C2=CCCCC2)C1 n1(CCC)ccc(=NC(C)(c2nnnn2CCCSC)C2CC2c2ccco2)[nH]1 N1(C(C(C)(C2(C)CC2)OC)=O)CCOC(CNC(=O)Cc2conc2C)C1 CCC(C)C(=O)C(=O)N(CC(=O)N(CCCC(CC)CC)C)C1CCC1 C1(CNC(c2c(C)nn(C)c2)=O)CCCCN(C(c2cc3c(s2)CCC3)=O)C1 C1(CC(=O)NCCCNC(=O)C(F)(F)C2(O)CCCC2)CC2COCC12 CC(CN=c1[nH]c(=NCC(C)(C)CC(C)C)[nH]c2c1COC2)c1ncc[nH]1 c1(C(=O)NC(CC(C)NC(c2c(C)c(O)ccc2)=O)C)cc2nc(Cl)ccc2o1 C(C(C(=O)NC1(C)CCC12CCC2)C(C)(C)C)NC(CCSCC)=O c1(C(=O)NC(CC)CNC(c2cc(O)no2)=O)ccc2ncnn2c1 C12(C(=O)NCC3CC(C)(C)N(C(C4CC45CCC5)=O)C3)CCC(C)(CC1)CO2 N(C1CCCOc2c(Cl)cccc21)C(CCCC1CCC(=O)N1)=O N1(C(=O)OC(C)(C)C)C2CCC1C1CC1(C(=O)Nc1ccc3nccnc3n1)C2 C(=O)(CCCC(=O)NCC1CCCCN(C(C2(C)CCCN2C)=O)C1)NCCC c1(-c2onc(C)n2)ccc(CNC(=O)NC2CC2c2ccco2)cc1 N1(C(c2sccc2C2CC2)=O)CC2CCC(C1CO)N2C(C1CCSC1)=O Cc1cc(C(C)(C)C(=O)N2CCC(NC(=O)C3=CCC3)C2)ccc1Br C1(C(N2CC(C)C(C(=O)N3CC=CCO3)C2)=O)CC1C1CCCC1 S(=O)(=O)(CC(=O)NCCOCC(=O)N(C1CCOC1=O)CC(C)C)NC C1(F)(C(=O)NC(C2CCN(C(c3ccon3)=O)C2)(C)C)CCCCC1 n1(CCCC)cc(C(=O)NCCOC2CCN(C(=O)Cc3cncn3C)C2)nn1 C1(C)(C(N(C)CCNC(=O)CCCCCC2CC2)=O)CCCNS1(=O)=O c1(CNC2CC3C(N)C3C2)cccn2cncc12 C(=O)(C(O)CCCCC)N1CCC(N2CCN(C(C3CC(CCC)C3)=O)CC2)C1 c1(C(=O)NC(CN2CCN(C(C(CCC)(C)O)=O)CC2)(C)C)cccc(N=[N+]=[N-])c1 C(=O)(CCC1=CCCCC1)N1CC(CCC)N(C(=O)C(F)C(F)(F)F)CC1 C(=O)(C(C)(F)C(C)(C)F)N1CCC(N(C(COCCCC(C)C)=O)CCO)C1 c1(C(=O)NC(c2n(C)ncc2)C(=O)NCC2COCC2(C)C)ccncc1O C1(CCCCN(C)C(C2CC(C#N)C2)=O)CCCN(C(c2ccc(O)nn2)=O)C1 c1(CNC(COC)(C(C)C)c2nnnn2CCCSC)c(F)cccc1Cl C1(C(=O)NC(C(N2CCC(CC3CC3)CC2)=O)C2CCOC2)CC(=O)C12CCC2 C1(C(=O)NCC(CC)(C)NC(c2cccnc2O)=O)CCn2c(C)cnc2C1 N#Cc1c[nH]c(C(=O)NCC(O)CNC(=O)CN2CCOCC2)c1 N1(C(C(CC2CCCC2)NC(CC2N(C)CCC2)=O)=O)CC2COCC2(C)C1 c1(C(N2C3C(NC(c4nnn(C)n4)=O)CC(C3)C2)=O)c[nH]c2cccc(C#N)c12 c1(N2C3CC(CN(C(c4cc(CC)n(C)n4)=O)C3)C2)ncnc2cccc(C)c12 C1(C(N2CCC(CC(C)NC(C34CCN(CC3)C4)=O)CC2)=O)CN2CCC1CC2 c1(NC(=O)OC(C(C)C)C)cncc(C=CC(=O)O)c1 C1(C(=O)NCCCN(C(Cn2c(CCC)nnc2S)=O)CC)CCN(C)C(=O)C1 N1(C(CSSC)=O)CCCCC(NC(=O)CCCc2ccc(F)cc2)C1 C=CC1(CC(N2CC(OCCO)C2)=O)CN(C(C2(SC)CC2)=O)C1 c1(C(=O)NC2(CO)CCCN(C(CC#N)=O)C2)cccc2ncsc12 c1(C(=O)NC2(CNC(c3ccc(C)nc3)=O)CCCC2)ccnc(C)c1O Cc1c(C(=O)NCC(C)(C)NC(=O)C(F)Cc2ccccc2)cnn1CC(C)C Cc1ccc(C(=O)NCC2CC2NC(c2cnn(C(C)(C)C)c2C)=O)nc1C C(=O)(C(C)(C)CC(F)F)N1CC(CC)(NC(c2c(OC(F)F)cccc2F)=O)C1 c1(C(=O)NCc2occ(C(=O)NC(C)COC(F)(F)F)c2)nnn(C)c1C C1(C(=O)NCCN(C(C)C)CCOCS)CC(=O)N1 c1(C(=O)NCC2CC(n3cc(CO)nn3)C2)cc(O)ncn1 c1(C(=O)NC(CCN(C(c2ccn(CC)n2)=O)C)(C)C)ccc2cn(C)nc2c1 c1(N2CC(OC)(CNC(=O)CCn3cc(Cl)cn3)C2)ccccc1[N+](=O)[O-] N1(S(=O)(=O)CC2CCC2)CC2CCN(Cc3c(Cl)cccc3Cl)CC2C1 C(=O)(CC1=NN(C)C(=O)C1)NC(CNC(c1cc(C)nn1C)=O)C CC(C)CCC(O)C(=O)N1CCN(CC(C)(C)NC(=O)CC(C)CF)CC1 C(CC(C(=O)N1CCC(NC(=O)NC)C1)NC(=O)CC(C)CC)=CC c1(N(C(C(=O)OC)COC(C)C)CC2CC2)ccccc1C n1(CC)ccnc1C(N1CCCC1C1(NC(c2csc(CC(C)C)n2)=O)CC1)=O c1(CC(N2CC(O)(CNC(C3(C)CCCOC3)=O)C2)=O)coc2ccccc12 C1(C)(CN(C2CCN2C2CCCC2)C)CN(Cc2nc(=N)[nH][nH]2)CCO1 Cc1c(C(=O)NCC=CC(=O)O)sc2nnc(S)n12 C(=O)(N=c1ccc(OC)n[nH]1)C12CCC(NC(C(CCCCC)C)=O)(CC1)CC2 c1(C(=O)NC(CC(C)C)C(=O)NC2CCN(C3CC3)C2=O)cc2cccnc2[nH]1 c1(-n2c(C)cc(C(=O)NCCNC(C(CC)SC)=O)n2)ccc(Cl)c(Cl)c1 c1(N2CCC(C3(NC(C4(O)CC5CCC4C5)=O)CC3)C2)ncc([N+](=O)[O-])cc1Cl C1(NC(C(C2CC2)OC)=O)C2CC(O)C1N(C(=O)CCc1ccc(F)c(F)c1)C2 CC1=C(C(=O)NCC(C)(C)OC(C)(C)CCNC(=O)C(C)N2CC(C)C2)CCC1 n1(CC)c(C)cc(C(=O)NCC2(CN(C(=O)C=[SH]c3ccccc3)C)CC2)c1C CC(C)C(C)(C)C(=O)NCC1CCN(C(=O)C(c2ccccc2)O)CC1C c1(NC2CC(c3cccc(Cl)c3)(C(=O)OCC)C2)cc(C#N)ccc1Cl NC(CCS(N)(=O)=O)C(=O)NC1C(c2ccccc2)C1(F)F C1(C(N(C)C(C2CC2)C2CC2)=O)C2CN(CC#CC3CC3)CC12 C(CNC(C1(C#N)CC(C)C1)=O)(CC(=O)NCC(N1CCCC1)C)OC c1(C(=O)NC2CC3(C(Nc4ncnc(OC)c4C)C3)C2)cccn2c(O)nnc12 C1(C(=O)NCCOC)CN(C(=O)C(C)CC(C)C)CC1(C)C C1(N(C)C)CN(C(c2ccnc(Cl)c2Br)C(=O)NCCC#N)CCC1C(F)(F)F CC1CC(NC(=O)C=CC2CCOCC2)CN(C(=O)CC(C)(C)N(C)C)C1 C(=O)(C(C)(C)CNC(c1ccc(C2CC2)n1C)=O)N1C(C(N(C)C)=O)CCC1 N1(C(CC=C)=O)CC2C(NCc3ccc(O)nc3)C2C1 Cc1oc(C2CC2)nc1C(=O)NC(C1CCCN1C(=O)C(C#N)C1CC1)(C)C CCC(CC)C(F)C(=O)OC(c1ccc(Cl)cc1)C(N1CCOC(C)(C)CC1)=O C1(N(C(=O)CNC=O)C)CN(C(c2c[nH]nc2C2CC2)=O)CC1F C1(CC=C)(NC(C2CC(F)C2)=O)CC2CCC(C1)N2C(=O)C(C)COC N1(C(CC=C)=O)CC2CCC(C1)C2NC(c1ccc(Br)c(C)c1C(=O)O)=O n1(CC(N2CC(NC(C3CC(OC)C3)=O)C(OC)C2)=O)cc2ncccc2n1 C(=O)(CCCCCCS(N)(=O)=O)NC12CCC(NC(C3CCN(C)C3)=O)(CC1)C2 C=CCC(C)(C)C(=O)N1CCC(NC(=O)CCC2CC(F)(F)C2)C1 N1(C(c2nc(C#C)sc2)=O)CCN(C(=O)Cc2nc(C)sc2C)CC(O)C1 C1(C(=O)NCC(C)(C)NC(C#CC2(C)CC2)=O)CCc2nc[nH]c2C1 n1(CC(=O)NC2CC3C(NC(C4(N5CCNC5=O)CC4)=O)C3C2)cnc([N+](=O)[O-])n1 c1(OCC)ccc(C(C(=O)NC2CC2)N(C(C)CC(C)(C)O)C)cc1 C1(CC)CCCCC1C(=O)N(C)CCNC(C1(Br)CC1)=O N1(C(CSC)=O)CC(OC(F)(F)F)C(NC(=O)CC(F)(F)F)C1 n1(CC(CC)O)cc(C(=O)NCC2C=CCN2C(C2CC(O)C2)=O)nn1 CC1CCC(C(=O)NCC2(C(C)NC(=O)CCCn3ccnn3)CC2)CC1 N1(C(=O)CCOCC(F)F)CCC2(CC1)CN(C(=O)COC1CCOC1)CC2CO C(C(C)(C(=O)N1CC(C(C(=O)NC2CCC2N(C)C)OC)C1)OC)OC N1(C(=O)NCCCN(C(=O)C(C2CC2)C2CC2)C2CCCC2)CCCC1=O N1(C(c2c(C)noc2)=O)CCC(O)CC1C(=O)NC(c1ccc(O)cc1)C c1(CC(N2C(CNC(CC3(C)CC3(F)F)=O)CC2)=O)ccc(Cl)cc1Br C(CC(O)C(=O)NC(c1nc[nH]n1)C1CC1)NC(C1(C(N)=O)CC1)=O c1(C(=O)NC2(COC)CCN(C(c3ccsc3Cl)=O)CC2)cc(C)cc(Cl)c1N C1(NC(C(=O)NC(C2CCC2)C)=O)CCCC(CN)C1 C1(NC(c2cnn(CCCC)c2C)=O)CCN(C(C2CC2(C)C(C)C)=O)CC1C N1(C(C)=O)Cc2ccccc2CC1C(=O)NCCC1CN(C(=O)CC(C)(C)O)C1 S(=O)(=O)(CCCC(F)(F)F)NC1CC2OCCC(C)C2C1 c1(CN2C(C(=O)Nc3ccccc3[N+](=O)[O-])CCC2)c[nH]c2ccc(Br)cc12 c1(SCC(=O)NCc2cn(C3C(=O)NCCC3)nn2)ccc2c(c1)C(=O)NC2=O c1(CNC(C2C(C)(CC)C2)=O)ccc(CCNC(c2cc(Cl)n[nH]2)=O)cc1 c1(C(N2C(C(=O)Nc3cccc(F)n3)CC(F)C2)=O)cc(Cl)c(F)cc1F CC(C)CC(C)(O)C(=O)NCCCCCNC(=O)C(c1cscn1)N(C)C CC(CC(=O)N1CC(C2=NOCC2)C1)C(C)(C)NC(=O)CCC1CC1(F)F c1(C2CCCN(C(C34C(C(=O)OC)CC(C3)C4)=O)C2)ccc(F)c(F)c1 C1(CC(=O)NC2CCC(NC(CC(C)CN(C)C)=O)CC2)Cc2ccccc2O1 C1(C)(C(=O)OC)C=CCN1C(=O)Cc1c(C)n[nH]c1C c1(CC)ccoc1C(N1CCCC1C(=O)NCC(=O)NCCOCC)=O C(=O)(C1=CCCCO1)N1C(CNC(c2c(CC)nc(C)[nH]2)=O)CC2CC21 c1(NC(=O)CC2CCN(C(C3CCCCC3)=O)C2)cc(Cl)ncc1Cl CC(CS(C)(=O)=O)C(=O)N1CC2CCN(C(c3ccc(C#N)o3)=O)CC12 c1(N(CCOCCOC)C)cc(NCC2CCCC(C)(C)C2)nc(CO)n1 C1(NC(C2CCCC(OC)C2)=O)CC2CN(c3cc(C(F)(F)F)nc(C)n3)CC12 N1(C(C)=O)CCC(NC(c2cccc(C3CC3)c2C)=O)C12CCC2 N1(C(CC(CN(C)C)O)=O)CC2CC(NC(=O)CSCC(N)=O)C1C2 N1(C(C2CN(CCC)C(=O)C2)=O)CC(C)N(C(c2ccnc(OC)c2)=O)C(C)C1 C12(NC(C(CC)CCOC)=O)CCC(CNC(c3snc(C)c3N)=O)(CC1)OC2 C#Cc1ccc(C(=O)N(C)CC2COCCN2C(=O)C(C)C2(O)CCC2)c(F)c1 C12(C(N(C)CCNC(c3cc(C(F)(F)F)on3)=O)=O)CC=CC(C1)OC2 C1(CCCNC(C2CC(C(F)(F)F)C2)=O)CCN(C(c2cc(F)n[nH]2)=O)CC1 CC1CC(NC(c2ccc(C3CC3)s2)=O)CN1C(=O)CC1CC2(CC2)CO1 C1(NC(N(CC(C)(C)OC)C)=O)CCC(c2ccccc2)CC1 C1(NC(c2cnc(COC)s2)=O)CC2CC(C1)CN(C(c1cc[n+]([O-])cc1)=O)C2 Cc1cc(C(=O)NC2(C)CC(NC(=O)CC3(C)CCCC3)C2)sc1C c1(C(C)NC(C(N2CC(C)C(N)C(C)C2)=O)=O)ccc2ccccc2c1 C1(C(N(CC(CNC(c2c(C)c[nH]n2)=O)(C)C)C)=O)CCCC(=O)N1 c1(NC(C=CC(C)NC(=O)CCCN2CCOCC2)=O)ccc(CCF)cc1 C1(C(=O)NC2CN(C(c3cccc(C)c3)=O)CC2F)CC(C)CCC1C(C)C c1(NC(C(C2CCN(Cc3nccs3)CC2)C)=O)cc(Br)c(O)cc1Br N1(C(C(n2cc(Cl)cn2)C)=O)CCC2C(C1)CN2C(c1onc2ccccc12)=O N1(Cc2c[nH]c(=N)o2)CCC(CC(=O)N2CCC2)CC1 CC12CCN(C(=O)CSCc3ccncc3)C1CN(C(C1CCCCC1)=O)C2 N1(C(CCOCC)=O)CCC2CCC(C1)N2C(c1cnc(C2CCC2)nc1O)=O c1(CC(=O)NC(c2ncc(C(=O)N(C)CC3(CC)CC3)s2)=O)ccccc1OC n1(CC(=O)NC(CCN(C(c2c(C)ccnc2)=O)C)C)[nH]cc2c(=O)ncnc1-2 C1(C(=O)NCC23CN(C(c4c(OC)nsc4)=O)C(C2)CO3)CC2(CC(C)=NO2)C1 C(=O)(C1CCCc2cncn21)NCC1CC(NC(CC(C=C)C)=O)C1 c1(Cn2cc(-c3cnc(CC)o3)nn2)cc(F)c(Br)cc1F C1(O)(CNC(=O)CONC(C2CC3CC2CC3O)=O)CC2CCC1O2 C(=O)(C1=CC2CCC(C1)C2)N(CC(CN(C(C1(OCC)CCC1)=O)C)O)C N1(C(=O)C=Cc2ncc[nH]2)CC2CCCC(C1)N2C(=O)Cc1ccc(F)c(F)c1 c1(C(C(=O)NC(C(=O)OC)C)N(C)CC2(OC)CCC2)cccc(F)c1Br C1(NC(C2CC(CCC(=O)O)C2)=O)C2Cc3cc(Cl)ccc3C12 CC1CN(C(c2cn(C)nc2C2CCCC2)=O)CCN(C(C2CCC2C)=O)C1 CC1(C)COC(CC(=O)NC(C(=O)NCCN2CCCC2)C2(C)CC2)C1 C(CC(C(C)(C)C)NC(=O)C=C1CCCCC1)N(C)C(C1(C)CCN(C)CC1)=O c1(CC(N2CC(CNC(CCCCC)=O)C(C)C2)=O)cc(Cl)cc2c1OCC2 CC1(n2cc(C(=O)NC3CC3)nn2)CCN(C(C2CCCN2CC(F)(F)F)=O)CC1 c1(C(=O)NC2C(NC(CSCCCC)=O)CC2)cc2c(s1)CCOC2 CC1CCC(CC(N2CC(O)(C(F)C(=O)NC(C)CC3CC3)C2)=O)OC1 c1(OC)ccc(OC(=O)C(O)CNC(=O)OC(C)(C)Cc2ccc(C)cc2)cc1 C1(CNC(C2C=CC(NC(c3scnc3Cl)=O)C2)=O)CC2CCC(C1)O2 N1(C(=O)CC2CCCCN2C(c2cn3c(n2)CCC3)=O)CC2(CCCCC2)C1 C1(NC(C(CC#C)C)=O)CN(C(=O)CSC)CCC1CO CC(C)CC(C)(C)C(=O)NC1CCN(c2cc(C(F)(F)F)ncn2)CC1F C1(CNC(C(CCCC)F)=O)CC2CCC(C1)N2C(=O)CC1COCC(C)O1 CC(C)CCC(F)C(=O)NC1CCCCC1C(N1CCC(N(C)C)CC1)=O C1(c2ccccc2)(CNC(C2(Cc3ccccc3)CC2)=O)CCCO1 C1(C)(C(=O)NC2CCN(C(Cc3c(C)ocn3)=O)C2)CCCNC1=O C(=O)(C(C(C1CCCCC1)OC)N(C1CCCN(C2CC2)C1)C)NCCC C1(CCOC)CN(C(C2CC2C)=O)CCN1C(C12COCC(C1)C2)=O N1(C(C(CO)OC)=O)CC2CC1CN2C(C1CC(C(C)C)=NO1)=O c1(C(N2CCCN(c3nnc(C(C)(C)C)o3)CC2)=O)ccc2c(c1)CCCS2 C1(CNC(C2C(C)OCCC2)=O)CN(C(c2cc(O)nc(O)n2)=O)CCN1C C1(NC(C(CC)=CC)=O)CN(C(=O)CSCC)CC12CCOCC2 c1(CC)nn(C)cc1C(=O)N(C(CNC(=O)CC1(O)CCOC1)CC)C C=C(C)C(O)CC(=O)N(C)CCN(C(=O)CCc1ccc(C)o1)C C12(NC(=O)CSc3n[nH]c(O)n3)CCCC1N(C(C1CC=CCC1)=O)CC2 C(=O)(N=c1c(Cl)c[nH]cc1I)C1CN(Cc2c(C)ccc(Br)c2)C1 C#CCC(C)(CNC(c1ccn(CCNC(=O)C(F)(F)CO)c1)=O)CO N1(C(C2C(C)C2)=O)CCCC(NC(c2ccn(C3CCCC3)n2)=O)CC1 C1(C(=O)NCC(C(C)(C)C)NC(=O)C(F)(F)c2cccnc2)(OC)CCCCC1 C1(NC(C2C(OCC)C2)=O)C(C)(C)CN(C(C2(F)CC=CCC2)=O)CC1(C)C C12(C(N3CC(Cc4nnn(C)n4)C3)=O)CC(C)(CCO1)C2 C(=O)(C(=O)N=c1cc(C)o[nH]1)NCCCN(C(CC(CCCC)O)=O)C c1(CCNC(=O)NCC(=C)CCNC(=O)OC(C)(C)C)cc(Cl)nn2ccnc12 C1(NC(Cc2n(C)ccn2)=O)CC2CN(C(=O)CC3CCCNC(=O)C3)CC2C1 c1(C(=O)NC2(CNC(=O)CCc3ncc[nH]3)CCC2)cc2c(s1)CCCNC2=O c1(C(N(C)CC2CCN(C(=O)CCc3ccsc3)C2)=O)ccc2c(c1)COC2=O Cc1nc(C(C)(C)C)ncc1C(=O)N(C)C.c12ccc(cn1)C(=O)OCC2 C(=O)(C(C)(C)CS(=O)(=O)N1CCCC(CS)C1)OCC Cc1ccc2c(=NCC(C)(C)N3CCOCC3)[nH]c(C)nc2c1 CC(C)CC(C(=O)N1CCC(Cc2ccccn2)CC1)NC(c1ccco1)=O c1(-c2n(C(c3ccccc3)C)ccn2)cc(-c2ccc(Cl)c(N)c2)c(O)c(Cl)c1 O=C(CC(Cc1ccc(I)cc1)n1ccnn1)N=c1ccn(C2(CO)CC2)[nH]1 N1(C(c2n(C)cc(Br)c2)=O)C2CCCC1CN(C(C1(C)CCCO1)=O)C2 C1(=O)C(CCF)N1.c1(C(N(C2CC(OCC)C2)C)=O)c[nH]cc1CC c1(C(=O)NC(CNC(C2CC2c2ccsc2)=O)C2CC2)ccc(O)cn1 c1(C(=O)OC)cc(C)c2c(c1)CCCN2C(=O)CSNN1CCN(C)C2(CCC2)C1 c1(OC)c(NCCCc2csc(C)n2)cc(Cl)cc1Br c1(CC)ccc(F)c(C(C(=O)NCC2CC2)N(C)Cc2cncnc2)c1 C1(NC(CNC(C(C)(C)C)=O)=O)CCC12CN(C(c1ccn(CCF)n1)=O)C2 C1(COC(C(C)OCCC=C)=O)CC2CCC1CC2 N1(C(c2n(CC=C)ccc2)=O)CCC(C)C(CNC(c2cnc(COC)s2)=O)C1 c1(C(N2CCC(C)(NC(c3c(Cl)cn(C)n3)=O)C2)=O)ccc2c(c1)CC(C)(C)O2 C#Cc1cc(C(=O)N(C2CCN(C(c3cc(O)nc(C)n3)=O)C2)CC)cc(Cl)c1 N1(C(C(CC)NC(N)=O)=O)CC2C(CC(=O)NCc3ccncc3F)C2C1 c1(C(=O)NC2(CO)CN(C(C3(C(=O)OC)CC3C)=O)C2)cccc2ccsc12 C12(CC(=O)NC(CC=C)CNC(C3CCOCC3)=O)COC(COC)(C1)C2 c1(C(=O)NC2C(C)(NC(C3C(OC)CCCC3)=O)CCC2)cccc2occc12 C1(CC)(NC(c2nccc(C)c2O)=O)CCCN(C(C2CNC(=O)N2)=O)C1 C=CC(C)(CC)C(=O)NCC(C1CC1)NC(C1(C(C)(C)OC)CC1)=O N1(C(C(COC)N(C)C)=O)CC(CNC(c2coc(CC3CC3)n2)=O)CC(C)C1 Cc1cccc(C(=O)NCC2CN(C(=O)CCC(C)C)CCCO2)c1F CCC(C)(CC)C(=O)N1CCOCC(C(=O)NC2CCC(C)C2)C1 Cc1c(NC(c2cc(Cl)cc(Br)c2N)=O)ccc(C(=O)O)c1C Cc1ccccc1C(=O)NC(C1CCCN1C(=O)C(CO)N(C)C)(C)C C(C1CN(C(C2CCC23CCC3)=O)Cc2ccccc21)NC(=O)Cc1cn[nH]c1 C1(C(=O)NCC(C(=O)NCC)(C)C)CN(C(c2n[nH]c(=N)[nH]2)=O)CC1(C)C c1(C(N2CC3CN(C(C(CCC)C)=O)C3CC2)=O)ccnc2c1ncn2C c1(C(=O)NCCC(=C)CNC(=O)CCC2CC2)cncc2ncn(C)c12 c1(C(N2CC3C(CN=[N+]=[N-])C3C2)C(=O)NCCCC)cccc(OC(F)(F)F)c1 c1(OC)cc(NC(=O)OC2COc3ccccc3C2)c2occc2c1 c1(C(=O)NC(C(N2CC(C(=O)OC)OCC2)=O)C)ccc(C)cc1O c1(C(=O)NCCC(C)NC(=O)CCn2ccc(=N)[nH]2)ccc([N+](=O)[O-])c(Cl)c1 c1(OC)cc(CC(=O)NC2COC(C3CCNCC3)C2)cc(Br)c1 N1(C(CCC=C=C)=O)CCC2(C(=O)NCC=CC3CC3)CCCC12 C=CCC(C)C(=O)NC(CCN(C)C)C(=O)NCCN(C)CCO NS(=O)(=O)N1CC(C(N2CC3(C2)CN(C(C2CCCO2)=O)C3)=O)C1 C(=O)(CC(C)(C)COC)N1CC(C(C(=O)N(CC(CC)CC)CCC)OC)C1 CC(C)CC(O)CC(=O)NC1CC2CC1N(C(c1cc(N)ccn1)=O)C2 c1(C(N2C(C3(NC(=O)CCn4ccnc4)CC3)CCC2)=O)cccc(CCO)c1 CC1(C)C(NC(=O)C(c2cccs2)NC(C23CCC(C)(C2)OC3)=O)CC1(F)F N1(C(CC(=O)OC)=O)CCC(NC(=O)C=Cc2ccc(C(N)=O)o2)C(C)C1 c1(C(=O)NCC2(F)CC(NC(C3CN(C)C(=O)N3)=O)C2)ccc2cc[nH]c2c1 C1(NC(C(C)O)=O)CN(S(=O)(=O)C2CC2)CC12CC2 CON(CCC(=O)N1CC2CCC1C(O)C2)C(=O)C(O)c1cnn(C)c1 C1(NC(c2ccncc2)=O)CN(Cc2cnc[nH]2)CC(F)(F)C1 C1(C(N(CC(CC)(F)F)C)=O)CC(F)(F)CN1C(=O)CC1CCOC1(C)C c1(CC)cc(C(=O)NC(C)(C)CCCNC(=O)CCC(C)OC)cn(C)c1=O c1(CC)occc1C(=O)N(C)CCOCCNC(C1COC(C)C1)=O N1(c2nc(C(=O)OC)nc(C)c2)CCN2CCCC2C1 c1(NS(CCNC(c2ncn(C)n2)=O)(=O)=O)cccc(N2CCCC2)c1 c1(C(=O)NCCCC(C)NC(c2cc3nc[nH]c3cn2)=O)ccc(C#N)nc1O c1(CC2N(C(=O)Nc3n(CC)ccc3)CC2)cccc2[nH]ncc12 Cc1cc(C(N2CC3CC(C2)C3NC(=O)CC2(O)CCOCC2)=O)nnc1C Cc1csc(C=CC(=O)NC2CN(C(=O)CCC3NC(=O)NC3=O)CC2C)n1 c1(C(=O)NCC2OCCN(Cc3scc(C)n3)C2)cc2cccnc2[nH]1 N1(C(c2cc(CC)nn2C)=O)CCN(C(c2ccc(SC(C)C)cc2)=O)C(C)C1 C1(C(C)NC(c2cnc(SC)s2)=O)CCCN(C(=O)CCn2cnnn2)C1 c1(C(C)C(=O)NCCOC2CCN(C(=O)Cc3cc[nH]c3)C2)ccc(F)cc1 c1(OC)ccccc1-c1oncc1C(=O)Nc1cc(C(=O)NCCO)cs1 CCC(C)CC(C(=O)NCCC#CCO)NC(=O)COC1(C)CCC1 c1(C(N2CCCC(NC(C3CN(c4ccncc4)C3)=O)C2)=O)cc(Cl)cnn1 c1(C(N2C(CC(=O)NC3(C#C)CCOC3)CC(O)C2)=O)ccc(C)c(O)n1 C1(C(=O)NC2CC3(CCC3)C2)CCCN(C(c2nc[nH]n2)=O)CC1 c1(C(CNC(=O)CC2(C)CC2(F)F)NC(CCCOCC)=O)ccccc1F N1(C(c2c(C)noc2C)=O)CC2CCN(C(c3cnc(Cl)c(F)c3N)=O)C2C1 Cc1nc2cccc(C(=O)NCC3(C)CCCN(C(=O)C(C)NC(N)=O)C3)c2[nH]1 C(CN=c1ccnc(Cl)[nH]1)OCCN(C)C(C1CCC2CCCCN12)=O c1(C(=O)NC2(C)CN(C(=O)Cc3sc(O)nc3O)C2)cc(Br)ccc1F S(=O)(=O)(c1ccc(Br)cc1Cl)N1CCC2CN(Cc3cccc(C(C)C)c3)CC21 C1(C(N(CC(CC)OC)CC)=O)C(C2CC2)CCN1C(=O)COCCF C1(CC(N2CCC(COC(C)=O)C2)=O)CC2(CC2)CN1C(c1cc(C)[nH]n1)=O C1(=CC(N2CCCC(NC(C3C4COCC34)=O)CC2)=O)CCCCCC1(F)F CC1CCC(NC(=O)CC2CC2(Cl)Cl)CN1C(c1cc(F)cc(F)c1)=O C=CC1(C(=O)NC(COC)CCO)CCN(C(C23CC(F)(C2)C3)=O)CC1 C(C(CC(=O)NC1CCCCN(C(=O)C2=CCCOCC2)C1)C(F)(F)F)N(C)C N1(C(c2ccc(N(C)C)cn2)=O)CC2CC(CNC(c3cc(N)ccn3)=O)C2C1 c1(C(=O)NC(CNC(CSCC(=O)OC)=O)(C)C)coc(C(C)(C)C)n1 Nc1cc(F)cc(C(=O)NCCC2CCCN(C(C3CCCCC3)=O)C2)c1F C1CC(C)N=C2N=CNc3[nH]c(cc32)C(=O)N1.C(CC(F)(F)F)SCC CCC(F)C(=O)NC1CC(CNC(c2ccsc2C)=O)C1 C1(C(=O)Nc2ccc(C(=O)O)c(CO)c2)Nc2ccccc2NC1=O C1(CNC(=O)CCc2ccon2)CCCC1NC(C1CCOCC1)=O CCC(C)C(=O)NCC(=O)N(C)CCOCCC(N1CCCC1C(C)O)=O N1(C(C2C(CCC)C2)=O)CC2CC1C2NC(=O)CCc1cn(C)nc1C C(=O)(C1=CCC2CCC1N2C(C1CC2CC(=O)C1C2)=O)N1C(C)(C(F)F)CCC1 C(CCC(C)CC(=O)N(C1CN(Cc2cc(F)cc(Br)c2OC=O)C1)C)=C(C)C C(=O)(C1CCc2ccccc21)N(C(C(=O)NCC=CCOC)CC(C)C)C C1(C(=O)NCC(C#C)OC)CN(C)CCN1C(=O)CCN1CCCC1=O N1(c2nccc(NC(c3cnccn3)C)n2)CC(C)OC(C)C1 C1(C2CC2)(CNC(c2c(C)oc(C)c2C)=O)CCN(C(C2(C)CCC(=O)N2)=O)C1 Cc1cc(Br)c(NC(C2CC3CC3N2c2ncc(Br)cn2)=O)cc1C c1(C(=O)NCC2N(C(c3n(C)ncc3)=O)CC(O)C2O)cnn2c(=O)cc[nH]c12 C(=O)(C(C)(C)CCC#N)N(C)CC1(O)CCCN(C(CNS(CC)(=O)=O)=O)C1 C1(CC(=O)NCC23CCC(C(=O)OC(C)(C)C)(CO2)C3)CC2(CCC2)CCO1 C(=O)(C(C)C(C)NC(c1sccc1OC)=O)N1C(C)(COC)CC1 c1(COC(C(c2ccc(F)cc2)NC(=O)OC(C)(C)C)=O)cncc(F)c1 C#CC1(NC(=O)COCC)CCOC1.C(CC)NC(=O)COCC(C)C C=CC(CCC)CC(=O)NCC1C=CCN1C(c1nnn(C)n1)=O c1(C(=O)NCCC2CCN(C(c3n(C)nc(Cl)c3)=O)C2)cc(Cl)cc(F)c1F C1(CNC(C(CC)n2cccn2)=O)CN(C(c2cnc(C3CC3)o2)=O)CC1(F)F CC1CCC(C)(C)N1C(C1CC12CC(NC(c1cocn1)=O)C2)=O c1(OCC)nc(NC2(CCNC(c3cncc(C)c3)=O)CCC2)ncc1Cl CC(CC(C1CC1)NC(=O)OC(C)(C)C)C(=O)NCC1(NC(N)=O)CCC1 C(=O)(C1=C(C2CCC2)N(CCC#N)C(=S)NC1c1cccc(F)c1F)OCC C1(N(c2nccc(Br)n2)C(c2cc(O)nc(Cl)c2)=O)CC12CCNCC2 C(=O)(CCCn1cncn1)N(C(C)C(=O)NCCN(CC)CC)CCC CC(CC(=O)NCC(C)(C)C)C(C)(C)NC(C1CC(=O)CCO1)=O c1(C(N2CCC(NC(C(CCC)(C)C)=O)C2CC)=O)ccc2c[nH]nc2c1 c1(C(N2C(CNC(=O)CC3COCCO3)COCC2)=O)cccc(C=C(F)F)c1 C1(C(=O)Nc2c(CC)ccs2)CC(C)CN1CC1(C#N)CCC1 C1(CC)CN(C(=O)C(F)(F)C2(OC)CCC2)CCC1NC(=O)CC(C)(C)CC C(=O)(CCCCCc1cccs1)NCCN(C(C(CSC)OC)=O)C1CCCC1 C1(C(C)(C)NC(c2cnc(C)[nH]2)=O)CCN(C(c2ns[nH]c2=O)=O)CC1 C(CC1=CCCCC1)NC(C(CCOC)NC(c1cnn[nH]1)=O)=O CC1(C(=O)N2CC3CC2CN3C(=O)C2CC2)CCc2cc(Br)ccc21 c1(CCOC)cc(Cl)ccc1C.C1CC(C)NC(=O)N1 c1(OCC)cnc(C(=O)NCC(CNC(c2ccnnc2S)=O)OC)c(Cl)c1 N1(C(C(=O)NCC(=C)F)=O)CCC(C)(Nc2ccccc2CC)CC1 C(=O)(C#CC1CCCO1)NCC(C)N(C(C(c1cccc(C)c1)=O)=O)C c1(CNC(CC(CC)C2CCC2)=O)ccc2c(c1)CN(C(C1CC(OC)C1)=O)C2 c1(OCC(N2C(CN(C(=O)CC3CCC34CCC4)C)CCC2)=O)ccc(Cl)cn1 C(=O)(C1=CCCC(C)(C)C1)N1CCN(C(C(C)CCO)=O)C(CCO)C1 Cc1ccc2c(=NCC3CC(C)N(C(C4CCCN4C(C)C)=O)C3)[nH]cnc2c1 CC(C)CC(F)C(=O)NCC1(CNC(C2Cc3nccn3C2)=O)CCC1 Cn1cc2c(COC(c3csc(Br)c3Cl)=O)cccc2n1 c12ccccc1S(=O)(=O)NC2=O.c1(CCOC)cccc(N(C)C)c1 CCC(CC(=O)NCCC(C)N(C)C(c1cc(F)cs1)=O)C1CC1 c1(C(N(C2CCN(C(C(C)CN(C)C)=O)C2)C)=O)cn2ccccc2n1 C1(NC(CN(C)C(C2(F)CC=CCC2)=O)=O)CC2CCCCCC12 C(=O)(CC1COc2ccccc21)N1CC(CN(C(CCC(=C)Cl)=O)C)OCC1 c1(C(=O)NCCNC(CC2(C)CC2F)=O)ccccc1NC1CCCCC1 C1(CNC(=O)C(Cl)=CCl)CN(C(=O)CN2CCOC2=O)CC(C(F)(F)F)O1 N1(C(CCN(C(=O)C(C2CCOCC2)=O)CC=C)=O)CCCC(CC)CC1 C(N=c1[nH]c(N2CCC3(CCCCC3)C2)nc2ccc(Cl)cc12)C1OCC(C)C1 C(=O)(C(C)(CC#C)NC(=O)CC1CC1(C)C)N(CC#C)CCOC c1(C(N2CCN(C(C)CNC(=O)CCn3cccn3)CC2)=O)cc([N+](=O)[O-])c[nH]1 C1(NC(C2(C)CCSCC2)=O)C2CCCC1CC(NC(C1CCC(F)(F)C1)=O)C2 S(=O)(=O)(c1ccc(Br)cc1N1CCC(n2cccn2)C1)NCC(CCC)OCC C1(NC(=O)C(F)Br)C2COCC1CN(C(=O)C(=O)C1CC1)C2 CC1CCN(C(C2CC2Cc2ccccc2)=O)CC1N(C)C(c1ccoc1)=O C1(CNC(c2ncn(C)n2)=O)CC2CCC(C1)N2C(=O)CC1CCC2(CCC2)O1 C1(NC(CCC(C)C)=O)C(CNC(=O)CCN2CCCC2)CCC12CCC2 C(=O)(C(c1cccs1)=Cc1ccccc1)N1CCC(CNC(=O)Cc2cscn2)C1 N=c1[nH]ccc(C(=O)NCCOC2CCN(C(=O)C(F)C(F)(F)F)C2)c1[N+](=O)[O-] N1(C(CC(COC)(C)O)=O)CC2CN(C3CCCc4ccc(F)cc43)CC2C1 C1(C(N(CC(CC)C)CC)=O)CCCN(C(=O)CCc2cnn(C)c2)C1 c1(C(N2CCN(C(c3nccc(N)c3)=O)CC2)=O)c(Cl)cc(F)cc1Cl CC1(C(=O)Nc2cc(I)ncn2)CCCN1C(c1ccc(Cl)o1)=O C(c1ccsc1Br)=CC(=O)NC(C1CN(C(C2C(C)(C)C2(C)C)=O)C1)C c1(CC(N2CCCC(NC(CN(C)C3CC3)=O)C2)=O)cc(O)nc(O)n1 c1(C(C)C)nc(N(CC(O)CNC(c2ccn(CC(F)(F)F)n2)=O)C)cc(Cl)n1 N1(c2ncc(SC)cn2)CC2CCC(C1)C2NC(=O)Cc1ccc(Br)nc1 Cc1c(C#N)nn(CCCNC(c2ccc(OC(F)F)cc2)=O)c1N CCC(C)(C)CC(=O)N(C(C)(C(=O)NCC(O)CNC(N)=O)C1CC1)C N1(C(C(C)C)=O)CCCCC1C(N1CC(C)(NC(=O)CC(=O)NC2CCC2)C1)=O N1(C(C)C)CCOC(C(N2CC(N(C)C(c3ccnn3C(C)(C)C)=O)C2)=O)C1 C1(CNC(c2n(CC)cnn2)=O)(NC(c2n[nH]cc2Br)=O)CCCCCC1 C1(C(=O)NCC(C(=O)OC)OC)CC2CC1CN(C(=O)COC(C)C)C2 CC(C)C(CCNC(C1(CO)CC(F)(F)C1)=O)NC(C1(CC2CC2)CCC1)=O C1(NC(C=Cc2ccc(C)o2)=O)CC2CCC(C1)N2C(C1CCCC12CC2)=O CC#CCCCCNC(=O)CC(C)CNC(C1CCNC1=O)=O C1(O)(CNC(Cc2c(C)con2)=O)CC2CCC(C1)N2C(=O)CCP(C)(C)=O CC1C2CC(CC1(c1nnnn1C1CCC1)NC1CC3(CCC3)C1)C2(C)C C1(C(N2C(CNC(c3ncc(C)nc3)=O)C=CC2)=O)CCOCC1(C)C c1(OC)nccc(C(=O)NCCOc2c(C)cccc2Cl)c1SC n1(CC)nnnc1C(C)(CCBr)NCC(=O)Nc1nnc(C(F)F)s1 C#Cc1cccc(C(=O)N(C2CN(C(=O)Cc3ccc(Cl)cn3)CC23CC3)C)c1 c1(OC)ccc(Cl)c(CNc2cccc(NC(c3ccoc3C(F)(F)F)=O)c2)c1 C12(CNC(c3cccs3)=O)CCC1CN(C(c1cccc(-c3cc[nH]n3)c1)=O)C2 C1(CC(=O)NC2CC(F)(CNC(CNS(NC)(=O)=O)=O)C2)CC2CCC1O2 N1(C(C)C)CCC(c2nnnn2C)(NCc2cc(Cl)ccc2F)CC1 C1(NC(CSCC#C)=O)CCOC(CC(=O)NCc2ccc(CC)cc2)C1 N1(N(C2CN(S(C)(=O)=O)C2)Cc2cccc(F)c2Cl)CCC(CC(=O)O)C(F)(F)C1 C(=O)(C(O)CCCNC(C1CCCN1CCC)=O)NC1C(CC=C)COC1 N1(C(c2cccc(CC)c2)=O)CCN(C)CC1C(N1CCN(C(C)C)C(=O)C1)=O c1(OCC)cc(C(=O)NC2CC(NC(=O)CC3(CO)CCCC3)C2)ccn1 Cn1ccnc1CCC(=O)N1CCC1CNC(c1csc(-c2cccs2)n1)=O c1(C(C(=O)OC)NCC2CCCN2C(=O)C(C)(C)C)[nH]c2ccccc2c1OC c1(C(=O)NC(CCCC)CNC(c2cn(CC)nn2)=O)cccc(C2CC2)c1Cl N1(C(COCCC=C)=O)CCC(CNC(c2ncsc2C)=O)C1 C(C)(CCC(=O)NCC1CCN1C(c1c(C(F)(F)F)coc1C)=O)OCC N1(C(Cc2nc(C)sc2)=O)CCN(C(C2CC(n3ccnn3)C2)=O)CCC1C N1(C(c2c(C)cc(N)cc2)=O)c2cccn2C(C)CC1C N1(CC(=O)NC2C(NC(c3c(OC)cnc(Cl)c3)=O)C2)Cc2ccccc2C1=O C1(C(C)NC(=O)CCCN(C)C)CCCN(C(C2CSCCS2)=O)C1.N1(CC)CCCC1 C1(NC(C(C)N2CCC2)=O)CC2CN(C(=O)CCCC3(C)NC(=O)NC3=O)CC12 c1(CCC(=O)NCC#CCNC(CCSCCC)=O)ccc(C)cc1C N1(C(C(CNC(C)=O)(C)C)=O)CCOCC(CNC(=O)C(F)=CC2CC2)C1 C(=O)(C1CCc2cccc(Cl)c21)NC12C(CN(c3c(C#N)cnc(C)n3)C1)C2 c1(CC(=O)NC2CCN(C(C3C4CCCCC34)=O)CC2)ccc2c(c1)COC2 C1(OC)C(OC)CN(C(C2CC3CCC3C2)=O)C1CNC(=O)C(C)(C)CCSC C12(CNC(CC(C)C)=O)CC1CN(C(C1CCCN(C(=O)OC(C)(C)C)C1)=O)C2 c1(C(=O)NCCC2CC(OC)CN2C(=O)C=CCF)c[nH]c2ncccc12 CCC1=NOC(CC(N2CC(O)(CN(C(=O)C=C(C3CC3)C3CC3)C)C2)=O)C1 CN1CC=CCC1CC(=O)NCC(O)C(=O)NCc1cnns1 C1(NCC2(C(N(C(C)C)C)=O)CC2)C2CN(C(C3CCC4CC34)=O)CC12 N1(c2c(C)c(N3CCC=C(Br)C3)ncn2)CCc2ccc(F)c(F)c2C1.CCC#N c1(OCC(C)NC(=O)NCCc2cccc(O)n2)ccc(F)cc1 Cc1cncc(F)c1C(=O)NCCCCC(C)NC(C12CCC(C1)C2)=O C(CC(C)(C)CNC(=O)Cc1ccccc1Cl)NC(C1CN(C(C)=O)C1)=O c1(CC)nnc2cc(NC(C)CCNC(=O)C3=CCCC3)ncn12 c1(CC(N2C(CNC(C(C)CF)=O)C=CC2)=O)ccc(Cl)c(F)c1 c1(CCC)ccc(-c2cscc2C(N2CCN(CCC(F)(F)F)CC2)=O)cc1 C1(C(=O)NCCCN(C(=O)C=CCn2cncn2)C2CC2)(COC)CCOC1 C1(NC(c2cnc(C#N)s2)=O)CN(C(=O)Cc2cncs2)CC12CCOCC2 C1(NC(c2ccccc2)C(=O)NC)CC2CNC(OC(C)(C)C)CC12 N1(C(CCC(CCC)C)=O)CCCC1(C)c1cn(-c2cccnc2)nn1 C(CN=c1nc(N2CCN(C)CC2)cc[nH]1)C1N(Cc2[nH]nc(OC)c2Cl)CC1 Cc1c(C(=O)N(C)CCNC(C2NC(=O)CC2c2ccc(F)cc2)=O)ccn1C c1(CC)ncc(C(=O)NC2CCN(C(c3ccc(C#N)n3C)=O)CC2C)c(C)n1 C1(C(=O)NC2CC(NC(C3CCOCC3)=O)C2)CC2(C1)CC2F Cc1[nH]nc(Cl)c1C(=O)NCCC1CCCN(C(C23COCC(C2)C3)=O)C1 C(=O)(C1=C(C)CCCC1(C)C)NC1C2CC3CN(C(CCCOCC)=O)C1C3C2 C1(CC(=O)NC2(C(N(C)Cc3cnnn3C)=O)CCSC2)CCCC2CC12 CC(C)CC(C(=O)NCC12CCC(CC1)N2C(=O)CC1CCC(=O)O1)N(C)C c1(C(=O)NCCCN(C(c2c[nH]nc2C2CC2)=O)CC)cc2cccnc2s1 S1(=O)(=O)c2cc(ccc2Cl)C(=O)OC2CCN1CC2.CCC(C)OC(=N)O Cc1cc(C(N2CCC2CNC(c2cccnc2F)=O)=O)n(CC(F)F)n1 C1(C(=O)NCCOC2CN(C(C(COC)OC)=O)C2)Cc2cccc(F)c2O1 C1(NC(C2(C#C)CN(C(C3CC(=O)CCO3)=O)C2)=O)C2CCC(F)(F)C12 CC1CN2CCCC2CN1C(c1occc1CNC(C12CC(C)(CCO1)C2)=O)=O C(=O)(CCC(C)NC(=O)OC(C)(C)C)NC(C1(O)CCC1)C CC(F)(F)CC(=O)NCc1cn(CCNC(C2CCN(S(C)(=O)=O)C2)=O)nn1 N1(C(C=CC=CC)=O)CCC(CNC(=O)C(C(C)(C)C)NC(=O)NC)C12CC2 C1(CNC(c2cscc2C(F)F)=O)CCN(C(=O)C=C(Cl)Cl)CC1 N1(C(Cc2c(C)noc2)=O)CC(C)CN(C(=O)CCn2cnnn2)CC1C C(CC(O)(CC)CC)NC(C(CC)NC(C1C2CCC(=O)C12)=O)=O C1(CNC(CCCC=C)=O)CN(C(=O)CCCN2CCCCC2)CC(C(C)C)O1 C1(C(C)C)CN(C(=O)CC(F)(F)Br)CCN1C(C1CCCN1N=O)=O c1(OC)cc(NC(c2cncc(NC(c3cc(I)ccc3Cl)=O)c2)=O)c(Br)cn1 c1(OC)ccc(C#N)c(NC(C2CN(S(=O)(=O)c3cn[nH]c3)C2)=O)c1 CN1C(=O)c2ccc(C(=O)NCC3(NC(C4CC45CC5)=O)CCCC3)cc2C1=O c1(OC)ccc(Cl)c(C(=O)C(=O)NCC(C(=O)OC)Oc2ccc(Cl)cc2)c1N N1(C(c2cc(SC)oc2)=O)CC(C)N(C(=O)Cc2ccccc2CC#N)CC1C C=CCCC(CC(C)C)C(=O)N(C1CCN(C(C2(C)CC2)=O)CC1)C CC1CCN(C(=O)CCSC(F)(F)F)CC1NC(c1ccccc1F)=O c1(CC)conc1CC(=O)N(CCC(C)N(C1CCCCC1)C)CC.C1(=O)CN1 C(=O)(C#CC1CCC1)N1CCC(N(C(=O)Cc2ccccc2F)CCC)C1 c1(C(N(C2CCN(Cc3c(OC)cccc3)C2)C)=O)cc2nccnc2cc1F N#Cc1c(NC(=O)C(=O)NCCCCCCC2CC2)cccc1Cl c1(C(N2CCC2c2cn(CC3CC3CC3C4CCCC34)nn2)=O)ccn2cnnc2c1 C1(C(=O)NC2(CC(=O)NCC(CCC)OC)CCC2)COCCC1C C1(C)(CC)C=C(C(=O)NC(c2ccccc2)C(N2CCCCC2)=O)C1 N1(C(CCC=CCC=C)=O)CCC(O)(C2(NC(c3ccnnc3C)=O)CC2)CC1 c1(CC(C)NC(C2CCC3CC3C2)=O)cccc(Br)c1 c1(C(c2nnnn2-c2ccc(CC)cc2)NCC=CC)ccnc(Cl)c1Cl c1(C(=O)NC2C=CCN(C(c3c(C)cc(F)s3)=O)C2)c2ccccc2nn1C c1(COC)cncc(C(=O)N(C2CN(C(=O)Cn3ccsc3=N)C2)C)c1 n1(CCOC)cc(C(N2CCC(C)C2CNC(=O)C=CCOC)=O)c(C)n1 c1(C(=O)NCC2(O)CC(NC(c3c(C)csc3)=O)C2)cc2c(F)ccc(F)c2s1 Cc1cc2ccc(C(N3CC(CN(C(=O)C(C)S(C)(=O)=O)C)C3)=O)cn2c1 c1(C2(C(=O)NCCCCc3cn(CCOC(C)=O)nn3)CC2)ccc(Cl)cc1F CCCC(C(=O)N(CC(C)OC)C)NC(=O)CCC(=O)N(C)C Cc1nc(N)cnc1C(=O)NCC=CCNC(=O)CC1CCCS1(=O)=O O=C1CC(N=c2ccnc(N3CCSCC3)[nH]2)CN1c1ccc(Cl)cc1 c1(OC)ccc(Cl)cc1C(F)(F)C(=O)N(CC(O)CN(C)C(C1C(C)C1C)=O)C c1(C(=O)NC2CC(NC(c3cncc(C)n3)=O)C(O)C2)c(C)nn(C)c1F C(=O)(CC(C)(C)N(C)C(C1CS(=O)C1)=O)NCc1c(C)cco1 C1(NC(C(C)=CC)=O)CC12CCN(C(=O)C(O)C(C)C)CC2 CCCCC(O)C(=O)N1CCC(Cn2cc(CC(c3ccccc3Cl)O)nn2)C1 Cc1cc2c(C(N3CC(NC(c4cc(OC(F)F)ncn4)=O)C3)=O)cccc2o1 C1(C(N(CC(C)C)CCO)=O)CCCCC1(C)NC(c1ccc(F)cc1F)=O C1(=CCNC(=O)CCC2CCCOC2)CCN(C(=O)COc2ccsc2Cl)CC1 C12(NC(C(N3C(=O)CCC3=O)C)=O)CC(C)(C1)OC21CN(C(=O)C=CCF)C1 c1(SC)cc(C)c(C(=O)N(C)CC2CCCN2C(=O)C=Cc2cnc[nH]2)s1 c1(OC)ccc(CC(=O)NCCN(CC(C)O)C(c2cn[nH]c2)=O)cn1 C1(N(C(C2C(CCC)C2)=O)CC)CCC(NC(=O)C=COCC)CC1 C(=O)(C(C)(CNC(=O)C=C(C)C)CC)NCC1CCN(CCC)C1 C1(CNC(=O)C=CC(F)(F)F)CCCCCN1C(=O)C=CC1CCCO1 N1(C(C(CN(C)C)(C)C)=O)CC2CC(C1)CN(C(c1csnc1Cl)=O)C2 c1(NCCN2C(=O)NC(=O)C2)cc(N2CCOC(C(F)F)CC2)nc(C(C)C)n1 Cc1ccc2c(c1)SC(C(=O)NCCC1CCCN(C(=O)C=CBr)C1)C2 C1(C(N(C2CCN(C(C(C(C)C)N(C)C)=O)CC2)C)=O)CC(S(C)(=O)=O)C1 C1(CN(C(C(C)C#N)=O)C)CC(F)CN1C(=O)Cc1cc(Br)nn1C CCC(C)(C)C(=O)C(=O)N1CCCC1CCC(=O)NCC1CCCOC1(C)C Cc1cnccc1C(=O)NC1(CNC(=O)CC2CNC(=O)C2)CCCCC1 c1(C(=O)NCC(C)NC(C(C(C)(C)C)NC(=O)OC)=O)cc(F)cc([N+](=O)[O-])c1 c1(C(N(CCCNC(c2ccc(CC)cn2)=O)C)=O)cc2c(s1)CCC(C)C2 C12(NC(c3nn(CC)c(C)c3)=O)CCCC1N(C(c1cc(Cl)n(C)n1)=O)CC2 C(c1cnc(C)nc1O)=CC(=O)NC1CC(CNC(CCCCCOCC)=O)C1 C12(CNC(c3c(Cl)cn(C)n3)=O)COCCN1C(=O)CN(C(=O)CC1CC1)C2 C1(CCCNC(=O)CCc2cnoc2)CCCN1C(c1csc(CO)n1)=O Cc1cccc2nc(N3CCC(C(C)NC(C4CCC5CC5C4)=O)C3)oc12 C(CCS(=O)(=O)N1CCCC1CCOC(C)(C)C)N(C)C C1(CNC(C(C)SC(C)C)=O)CN(C(c2c(Cl)csc2Cl)=O)CCO1 C1(C(=O)OC)CN(C(=O)CC2(O)CCCN(C)C2)Cc2ccnn2C1 c1(OC)nccc(CNC(c2ccoc2C(F)(F)F)c2nnnn2C)c1Br CC(C)(F)C(C)(F)C(=O)N1CCC(O)(CNC(=O)CCSc2cccc(Cl)c2)C1 C1(CNC(CC2(COC)CC2)=O)CN(C(=O)CC2COCCOC2)CCC1(F)F c1(COC(=O)NC(CC(=O)NC2(C(=O)OC)CC2)C)ccc(C(F)(F)F)nc1C c1(OCCC)cc(C)cc(-c2ccc(C(N3CCCC(O)C3C)=O)nc2C)c1F N1(C(c2c(C)nns2)=O)CCN(C(c2cnsc2)=O)CC1CC(C)(C)C C1(C)(COC)CC(NC(=O)CCC2CCC2)CN1C(=O)Cn1nnnc1C c1(C(N(C2CCN(CC(O)COCC(C)C)C2)CC)=O)cnn(C(F)F)c1 C1(CNC(CC)(C)C(=O)OC)CCN(C(=O)OC(C)(C)C)C12COC2 N1(C(C(=Cc2ccccc2)C)=O)CCCC(CC(N2CCC(F)(CF)C2)=O)CC1 c1(SCC)cc(N)ccc1C(N1CC(N2CCN(C(=O)C(C)(C)CC)CC2)C1)=O C1(NC(c2c(Cl)nc(OC)s2)=O)CC2CCCC(C1)N2C(=O)C(C)=CC(C)(C)C C(=O)(CCCCN=[N+]=[N-])N1CCCC(C(=O)NC(C#C)(C)C)C1C C(=O)(CC(C)C(F)(F)F)NC(CNC(c1c(O)ncc(CC)c1)=O)(C)C1CCC1 C(CC(=O)N1CCCC(NC(=O)CCSc2nnnn2C)C1)(C(F)(F)F)OC C1(CNC(CCC2C(C)(C)C2)=O)CC(C(=O)NC2C3CCCOC23)=NO1 C(c1ccc(F)cc1)=CC(N1CCN(C=O)CC1)=O.N=c1[nH]cc(C)s1 C1(NC(c2cn(CC(C)O)c(=O)cc2)=O)CC2CCC(C1)N2C(=O)CC#N N1(C(Cc2c(CC)con2)=O)C2CCC1CN(C(=O)C(=CC1CCCC1)C)CC2 C(=O)(C1=CCC(C)CC1)NCC1(CO)CCCN(C(c2c(CC)ccs2)=O)C1 C(=O)(C1=C(C)CCCC1)N(C1CCN(C(COCC(=O)NC)=O)CC1C)C C1(CC)OCCCC1C(=O)NC1CC(NC(c2scc(C)c2OC)=O)C1 C1(O)(CC(=O)N(C)CC2N(C(c3c(CC)c(C)sc3)=O)CCC2)COC(C)(C)C1 N1(C(c2[nH]ccc2C2CC2)=O)CCCC(NC(C2CC2c2ccccc2)=O)C1 c1(CCC(N2C(CCNC(C(C)C)=O)CCCC2)=O)cccc(F)c1Cl c1(C2(OC)CCN(n3nc(C4CC4)n(C)c3=S)CC2)ccc(F)c(F)c1 c1(C(=O)NCC(=O)NCc2ccn(CC)n2)cc(C)n(C)c1 n1(COCC)nnc(C(N2CC(C(C)NC(=O)COC)C2)=O)c1N C(CCCC(F)(F)F)NC(C1(C(C)C)N(C(CC(CC)O)=O)CCC1)=O c1(NC(COCC=C)=O)ccc(NC(c2cc(C)n(CC)n2)=O)c(C)c1 C1(OC)CC2CC(NC(=O)CC3CCN3C(=O)CCC3CCOC3)C1C2 c1(C(=O)NC(CNC(C(C)(C)C#N)=O)(C)C2CC2)cnn2c1CCC2 c1(C(N2CCC(CNC(C34COCC3C4)=O)C2)=O)cc2ccc(Br)nc2[nH]1 C1(C(N(C2CCCN(C(=O)CC3(O)CCCOC3)C2)C)=O)CC(F)C(=O)N1C c1(OC)ccc(CN2CCN(C(=O)C(O)c3ccccc3)C(CC#N)C2)c(Cl)n1 C(=O)(CCC(=O)NC1CC(C)N(C(=O)CCCN2C(=O)CCC2=O)C1)OC CCCC(C)(C)CC(=O)NC(CC1CCOCC1)C(=O)NC1CCCCC1(C)C c1(OC)ccccc1C(C)CNC(C)Cc1c(C)noc1C N1(C(C)=O)CCC(NC(=O)C(N2CC3CC3(CO)C2)=O)c2ccccc21 C12(CNC(C3CN(C(C)=O)C3)=O)CCN(CC1)C2 C1(C(N(CC(F)Cl)C)=O)COCCN1C(=O)C=CC1CCCN1C c1(C(c2n(C(C)(C)C)nnn2)NCC2CCCCC2)ccc(C(C)(F)F)cc1 CC(=O)CC(C)(C)CC(=O)N1CC(CNC(c2cncc(C)c2)=O)CC1C Cn1cc(C(N2CCN(C(c3cnsc3)=O)CC2)=O)nc1-c1ccccn1 c1(SC)cn(C)nc1C(=O)NCC1CCCN1C(c1scnc1C)=O O=C(C1=CCC1)N1CCC1c1cn(CC2CCCOC2)nn1 C(C)(CNC(=O)C(F)F)(CC(C)C)NC(Cc1cc(C)on1)=O Cc1cc(C(=O)NC(CNC(C2C=CC=CC=C2)=O)C(C)C(C)C)ncc1C#N C(=O)(C(F)(F)CC(C)C)NC1CN(C(COCCOC)=O)CC1C(F)(F)F Cc1occc(=O)c1OCC(=O)NCc1ccc(CNC(C2CC2CF)=O)cc1 CC1CN(C(=O)C=Cc2ccn(C)c2)CCN1C(c1cc(C2CC2)no1)=O CC1(C)CC(CO)CN(C(=O)C=CCNC(=O)CC2(C)CCOC2)C1 CC(C)C(C)C(C)CC(=O)N1CCCC(NC(c2cc(CF)on2)=O)CC1 N1(C(c2c(C(=O)OC)cn(C)n2)=O)CCC(C)(C)C(CNC(C2CCCO2)=O)C1 c1(C(=O)NC2CCN(C(C(CC)SC)=O)C2C2CC2)cc2ccc(OC)cc2o1 N1(C(C2(CSC)CCOCC2)=O)CCC(NC(=O)C(C)=C2CC2)C(F)C1 C1(C(C)NC(=O)CCc2cnn(C)n2)CCN(Cc2cnc(Br)s2)CC1 c1(CC)scnc1C(=O)NC(CNC(=O)C(C)(C)c1cnn(C)c1)C(C)C c1(-c2ncc(COC(CC3C(C)CCC3)=O)s2)cccc(F)c1 N1(C(COCC(=O)OC)=O)CC(O)(C(C)NC(c2conc2C(C)C)=O)C1 C1(CCOC)CN(C(C2(C)CS(=O)(=O)C2)=O)CCN1C(=O)CC1CCCCC1 C12(C(N3CCN(C(C4C5CC(=O)CC54)=O)CC3)=O)CCC1CCCN2 C1(C(N2CCC(NC(c3cccnc3-c3ccccc3)=O)C2)=O)C2CC2C2CC12 C1(C(N2C(CCCC)CCC2)=O)CN(C(=O)Cc2ccsc2)CC1O C(CO)(C(=O)NCCC1(NC(=O)CC2CC2)CCC1)N(C)C C1(C(=O)NCC2(OCC)CCN(C(CC=CC=C)=O)C2)CCS(=O)(=O)C1(C)C CC(C)CC(C)C(=O)NCC1(F)CCCN(C(=O)CCc2ccn(C)n2)C1 c1(C(N2CCC(NC(C3(F)CC3(F)F)=O)C2)=O)ccc(-c2ccncc2)s1 C#CC1(C(N2CCC(O)(C(C)NC(=O)CCc3ccnn3C)C2)=O)CCCC1 Cn1c(C(=O)N)cc2occc12.c1ccccc1.C1COCC1 N1(C(CC(=O)NCC#C)=O)Cc2ccccc2C1CNC(c1nsnc1O)=O N1(CCCCCC)CCC(NC(C2CCOC(C(C)C)C2)=O)CC(C)(C)C1 C(=O)(CCCc1ccncc1)NC(C1(NC(C=C(CC)C)=O)CCC1)C N1(C(C(C)OCCC#C)=O)CC2CC(C1)N(C(C1C=C(C)CS1)=O)C2 N1(C(C(C)Oc2ccccc2)=O)CC2C(C1)C2(C)C c1(C2(CC)CC2)cccc(C(=O)NCC(C)(CO)NC(=O)Cc2ccn(C)n2)c1 N1(C(CCOCC(=O)OCC)=O)CCC2CCN(C(=O)CC3CCCOC3)CC12 c1(CC(N2CCC(c3ncc(C(=O)OC)s3)C2)=O)cncc(OC)c1 C(=O)(C(F)C(F)(F)F)NC1CCC(CCNC(c2c(CC)nc(C)s2)=O)C1 N1(C(CC(CC)CN(C)C)=O)CC2(CCN(C(=O)CCSc3nccn3C)C2)C1 N12CCC(C1=O)N(C)C1CC2C1.C1(SC)C(=O)NN=C1C CCCC(C)(O)C(=O)NC1CCC(NC(=O)C=Cc2cccc(Br)c2)C1 c1(C(=O)NCC(C)(CO)NC(Cc2n(C)nc(C3CC3)c2)=O)ccc(F)cc1F C1(NC(c2c(CC)nc[nH]2)=O)CCC(F)(CNC(=O)CCc2cncnc2)C1 CC1C2CCC(C2)C1C(=O)NC(C(=O)NC1(CF)CC1)C(C)O C1(NC(C(Cn2ccc(C)n2)C)=O)CCC2CN(c3ncc(I)cn3)CCC2C1 CC1(NC(=O)C2=COCC2)CCCN(C(C2(C3CCCCO3)CC2)=O)C1 CC1(NC(=O)CCc2nnc(O)nc2O)CCCCC1C(=O)NC1(CF)CC1 Cc1ncnc2c1CC(C(N1CC(Cn3cc(CSCCO)nn3)C1)=O)CC2 c1(CCNC(Cn2cc(CCN(C)CC)nn2)=O)ccc(Br)c(C)c1C C1(CNC(C(N2CCC(CCC(C)C)CC2)=O)=O)CCC2(CC1)CC2(F)F C1(C(=O)NCC(CO)NC(CCCc2onc(CCC)n2)=O)CCCCN1CC S(=O)(=O)(c1cc(-c2nnc(N(C(C(C)SC)C(F)(F)F)C)n2C)c(Cl)s1)N O=C(N=c1c(F)c[nH]cc1I)c1ccc(NC(=O)C2CC2)s1 N1(C(c2ccc(C)nc2)=O)CCC2C1CCN2C(=O)CC(N)c1ccccc1 C1(C(=O)NCCCOCCC(=O)NCC2CCC2)CC2CCC1(O)C2.C1CO1 c1(OC)nccc(C(=O)NC2CC2CNC(=O)Cc2ccc(F)cc2C)c1F C1(C2CC2)(NC(CSCCSC)=O)CCN(C(=O)C=Cc2cccs2)C1 c1(C(=O)NC(C2CCOC2)CNC(CN(C)C)=O)cc(O)nc2c1CCCC2 c1(CC)cccnc1C(N1CC(NC(=O)CCOCC(C)C)C2CC12)=O c1(CC)cc(C(=O)N(C2CCN(C(=O)CNS(=O)(=O)N(C)C)C2)C)oc1CC c1(C(=O)NCC2(C)N(C(CC3C=NN(C)C3=O)=O)CCC2)cc2cccnn2n1 C(C)(CCN=c1nc[nH]s1)NC(Cc1c(OC)ccc(F)c1)=O N1(C(c2n(CC)ccn2)=O)CC2CC(C1)N(C(=O)CCC(F)(F)F)C2 c1(OC)cc(S(N)(=O)=O)ccc1NC(C1CN(Cc2ccc(Br)nc2)CCO1)=O N(C(=NCC1CC1)N1CCC(C)(F)C1)C(C1(c2ccccc2)CC1)C C1(NC(c2c(CC)nc(C)[nH]2)=O)CCN(C(C2COCC2(C)C)=O)CC1F CC1Cc2cc(F)ccc2N1CC(=O)OCc1noc(-c2cccc(I)c2)n1 C(=O)(C(C)C(=O)OC)NC1C(NC(C2(CC)CCC2)=O)COC1 CC1CC2(CO1)CN(C(C1(CCNC(=O)CN3CCN(C)CC3)CCC1)=O)C2 C1(NC(COCC)=O)CCCC12CCN(C(=O)Cc1ccc(CO)c(C)c1)C2 N1(C(C=C(C)C)=O)CC2CCC1C(NC(c1csc(Cc3ccccc3)n1)=O)C2 c1(C(N(CC(=O)NCC(=O)NCCCC2CCCCO2)C)=O)ccc(CO)o1 c1(CC)nnc(C)cc1C(=O)NC1CCC1CNC(C1(CS(N)(=O)=O)COC1)=O CCCCCCC(C)(CC)C(=O)NC1CN(C(=O)C=CCN(C)CC)CC1C C(=O)(C(O)CCC(C)C)N1CCC(CCCCNC(C(C=C)C)=O)CC1 C(=O)(CCCCCCn1cc(CCCN2CCCC2)nn1)Nc1c(C)nc[nH]1 N1(c2nnc(-c3cncc(OC)n3)n2CCCOCC2CC2)CC2CC(C1)N(C)C2 Cc1cc(C(=O)NC2(CNC(C3C4CC5C(C4=O)C35)=O)CCOCC2)cc(C)n1 C1(CNC(CCC=C=C)=O)CCN(C(=O)Cc2ccc(Br)s2)C1(C)C Cc1oc(C#N)cc1C(=O)NCC1CC1NC(c1nn(C)cc1Cl)=O c1(C(C)C)nnc2cc(NC(C3CN(C(=O)Cc4ccco4)CCO3)C)ncn12 N1(C(CC(=C)C)=O)CCC(C2CC2)C1CNC(c1ccc(OC)cc1OC)=O C1(C)(C(=O)NC2CCN(C(C)=O)C2)CCCN(CC2CCCO2)C1 N1(Cc2ncc(C)c(Br)c2)CC2CC(CN(C(c3ccn(C(C)(C)C)n3)=O)C2)C1 C1(NC(C(Cc2cnc[nH]2)NC(C)=O)=O)CN(C(=O)C(C)C#N)CC12CCCC2 C1(NC(CC(=C)C)=O)CN(C(c2cccnc2C)=O)CC1CC1CC1 c1(C(N2CC(C)C(CNc3cc(=O)n(C)cn3)C2)=O)ccc2c(c1)CN(C)C2 CC1CCC(Cl)=C(C(=O)NC2CC(CCNC(=O)CN(C3CCCCC3)C)C2)C1 c1(NC(C2N(C(CN(C3CCC3)C)=O)C3CCC2C3)=O)ccc2ncccc2c1 O=CN1CCCC1C(N1CCOC(CC(=O)NCC2CC2(F)F)C1)=O N1(C(=O)OC(C)(C)C)CC2C(=O)CCC2(CNC(c2cccn3nnnc23)=O)C1 c1(NCCC(=O)NC2(NCCNC(COC)=O)CCC2)oc(C)nc1C#N CC(C)C(C(C)C)NC(c1c(CNC(=O)CC2CCOC2=O)nnn1C)=O CCCC(C)CC(=O)N1CC2CCC2(CC(=O)NCC2CC3(CCC3)C2)C1 C(C1=CCN(C(C2CN3CCC2CC3)=O)CC1)NC(C1CCCN1C1CC1)=O C1(C(=O)NCC(C)(C)NC(C=C(CCC)C)=O)CCCN1C(=O)OCC C1(C(=O)OCC)(C(C)C)CCN(N2CCCC(c3cccc(OCC)c3)C2)C1 C(=O)(C(C)C(F)(F)F)NC(CNC(c1ccc(OCC(C)C)nc1)=O)C1CCC1 CC(C)C(C(=O)N1CC2C(C1)C2(F)F)C(C)C.C(C(F)C=O)C1CNC1 c1(CC(=O)NC2CN(C(C(C)(C)C3CC3)=O)C2)ccc(Cl)c(Cl)c1 N1(CC2C(=O)CCCC2)CCC(=O)N(Cc2cc(Cl)cc(Br)c2)C1=O C1(NC(CN(C)C)=O)CN(C(C2(NC(N)=O)CCCCC2)=O)CC1O n1(CCCOC)cc(C(N2CCC(N(C(=O)Cc3ccno3)C)C2)=O)cn1 c1(CC(N2CCCCC(NC(CC(C)OC)=O)C2)=O)cn2cc(Cl)ccc2n1 c1(C(=O)CC)cc2nc(NC(=O)NCCc3cc(C(=O)OCC)no3)ccc2[nH]1 C1(NCC(CC2(C#N)CCOCC2)C(=O)OCC)CC12CCN(CC)C2 N1(C(c2ccc(N)cn2)=O)CCN(C(C2CCC(F)(F)C2)=O)CC1C(F)F C(=O)(C(F)C(=O)N(CC(O)CN(C(=O)CC1CC2CCC1O2)C)C)OCC Cc1c(C(=O)NC(C2CCCCC2)C(N2CCC(C)(F)C2)=O)c[nH]c1C#N C1(Nc2cc(OC)nc(C(F)(F)F)n2)CCCCCN(C(=O)CC(C)(C)C)C1 c1(C(=O)NC(CN(C(C=CCCC)=O)C)C)c(C)c(C)nn(C)c1=O c1(CCC)cc(C(=O)N(CCC(C)NC(=O)C=CC(C)CC)C)n[nH]1 CC(C#N)C(=O)NCCN(CCCN(C)C)C(c1ccc(-c2cccs2)s1)=O C1(C2CN(C(c3ccc(F)cc3Br)=O)C2)(NC(C(C=CCCC)O)=O)CC1 c1(C(C)C)nc2[nH]c(Cl)nc(NCc3ccnc(N(C)C)c3)c-2n1 CC1(C)OC(=O)NC1C(=O)NCC1CCOC1C(=O)NCC1(S(C)=O)CC1 c1(NC(N(C2C3CCCC23)C)=O)nc(C2CCC2)nc2ccccc12 C(=O)(C(=O)N=S(C)(C)=O)NCC(CNC(CCc1ccc(OCC)cc1)=O)CO C(=O)(CCCC(F)(F)F)N1CC(C)C(CNC(=O)Cc2nc(F)c(F)cc2F)C1 c1(CC(C)C)cc(C(=O)N(C2CCNC2)C)n[nH]1 C(C(=O)N1CCOC(CC(=O)NCCCOCC2CCC2)C1)(C(C)C)SC Cc1ncc(NC(=O)C(CC(C)C)NC(=O)CN2CCCC2=O)cc1C#N Cc1n[nH]c(C)c1C(C)C(=O)NCC1(F)CN(C(=O)CC2CCC(=O)O2)C1 C1(C(N(CC=C)CCOC)=O)CCCN(C(C2CC2c2ccccc2)=O)CC1 CCC(CCC(=O)N1CCCC(C(C)OC2CCCOC2)C1)OC.C1(=O)CO1 N1(C(COc2cc(C)on2)=O)CCOC(CCCNC(C2(C3CC3)CC2)=O)C1 C1(NC(CCC)=O)CCN(C(c2ccc(-c3ccco3)[nH]2)=O)CC12CCC2 C(CC(C)(C)CC(=O)N1CC(C)CC1C(=O)NCCN1CCCOCC1)OC N1(C(CCc2n[nH]c(=N)s2)=O)CC2(COC(CNC(c3nccnc3Cl)=O)C2)C1 C(c1ccc(C2CC2)cc1)=CC(=O)NC(C(C)C)(C)CNC(=O)C(F)CC1CC1 c1(C(=O)OC)cc(=NC(=O)C2CC(NCc3nc[nH]c3C(C)(C)C)C2)[nH][nH]1 C1(C(N(C2CCN(C(=O)CC3CC=CCC3)CC2)C)=O)CC(=O)N(C)C1 C(=O)(C(C)CC(N)=O)NC(CNC(C(Cc1ccccc1)NC(C)=O)=O)C1CC1 Cc1ncnc(C)c1C(N1CCN(C(c2cnc[nH]c2=N)=O)C(C(F)F)C1)=O C1(C(N2C3C(CNC(c4cccn4C4CC4)=O)C(C3)C2)=O)CC1C1CCCC1 c1(C(=O)NCC2CCN(C(=O)CN3CCS(=O)CC3)C2)ccc2n[nH]cc2n1 c1(C(=O)NC(CCNC(C(c2ccnn2C)C)=O)C)ccncn1 C(=O)(CC(C)C(F)F)N1CCC(CN(C(CCn2c(C)ncc2)=O)C)C1 CCCCCC(C)(C)C(=O)N1CCC(CCNC(=O)CN2CCCCS2(=O)=O)C1 N1(C(c2ncn(C)c(=O)c2)=O)CCC2(CCCC2CNC(=O)Cc2cn[nH]c2)CC1 C(=O)(CCC(CF)CF)N(CCC(=O)N(CC#C)C)CC C1(F)(C(=O)NCC(CNC(Cc2cc(OC)c(F)cc2)=O)F)CCC(F)(F)CC1 CC1(C)C(NC(=O)CC2CCCCC23CC3)CCN1C(c1cc(Cl)nnc1O)=O C(=O)(C(C)(CO)OC(=O)C(c1ccccc1)Oc1cccc(C)c1)OC N1(CC(=O)NC2CC2)CCN(CCCO)CC1.C1(O)CCOC1 N1(C(c2cnc(OC)c(Cl)c2)=O)CC2CCCC1(CNC(=O)C=C(C)C1CC1)C2 Cc1sc(C)c(C(c2nnnn2C2(C)CC2)NCCc2ccnn2C)c1Br c1(SCC(N2C(CN(C(c3cc(CCC)n[nH]3)=O)C)CCC2)=O)ccccc1O c1(C(N2CC(CNC(c3nncs3)=O)C2)=O)cnc2c(Br)cccn12 CC1CCC(C(C)(O)CNC(=O)NC(c2ccnc(O)c2)C2CC2)CC1 C(=O)(CCC(O)CN(C(C)(C)C)Cc1nc[nH]n1)OC c1(OC)cc(F)ccc1NC(c1ccccc1CN(CC(=O)NCC#N)C)=O C1(C)(CC(=O)N(CCNC(C)=O)C)CCN1C(c1[nH]ccc1C)=O C(=O)(C(F)C(C)(C)O)NCCCN(C(=O)C(C)Cc1ccc(Cl)cc1)C(C)C c1(OC)ccc(C(C)NCCOC(C)=O)cc1F.C1C(=O)N1 C(CCC(C)C(=O)NC1CCN(C(=O)CC2OCCOC2(C)C)CC1)OC C(=O)(CC(C)(O)C(F)(F)F)N(CC(C)NC(CCN(C(CC)CC)C(C)C)=O)C C=CCC(CNC(=O)C(C)NCc1cnn(CC(=O)OC)c1)NC(=O)OCC=C c1(C(=O)NCC=C2CCN(C(c3cc(C)nnc3)=O)CC2)cn2cccnc2n1 CCC(CC(=O)NCCN(C(C1(C#N)CC1(C)C)=O)C1CC1)CC(F)(F)F C1(NC(c2nc(C)[nH]n2)=O)CCN(C(c2cc3sccc3[nH]2)=O)CC1C c1(CN2CCC(CNC(c3ccnc(Br)c3)=O)CC2)cccc(Cl)c1O c1(C(N(CC=C)C)=O)ccc2c(n1)CN(C(C1Cc3ccccc3C1)=O)CC2 C=CCC(C)C(=O)N1CCC(N(C(=O)Cc2ccncc2Br)CCC)C1 CCC(C(=O)N(C)CC1CCN(C(=O)CCN(C)CCO)C1)C(F)(F)F C1(C(=O)NCC2CC(NC(C34CCOC3CCOC4)=O)C2)CC2CCCCN2C1 CN(C)S(=O)(=O)N1CC(C(=O)NC2(CNC(=O)CS(N)(=O)=O)CCOC2)C1 O=C1CC2(CN(C(c3ncc4sncc4n3)=O)C2)Oc2ccccc21 c1(C(N(CC#C)CC=C)=O)ccc2ncc(-c3ccc(OC)nc3)n2c1 C1(NC(C=CC(=O)OCC)=O)CC2CCC(C1)N2C(c1csc(S(C)(=O)=O)c1)=O CC1CCCn2c(CC(=O)NC3CC34CCN(C(c3cn[nH]c3)=O)CC4)cnc21 Cn1cccc(C(=O)NC(C)(C)CCC(=O)NCC2(C)CCOC2)c1=O N1(C(CCCC(=O)NCC)=O)CCOC2(CCN(C(C3CCOC3C)=O)CC2)C1 CC1(C)CCN(CC(=O)NC(Cc2ccco2)C(=O)NCCC2(O)CCC2)C1 CCCCC(C(=O)NS(C)(=O)=O)Cc1ccc(Cc2nn[nH]n2)c(C)c1 c1(NCC2N(C(c3nccc(C)n3)=O)CCCC2C)c[n+]([O-])ccc1[N+](=O)[O-] N1(C(c2cc(C)cc(N)c2)=O)Cc2ccc(Cl)cc2C1 C(=O)(C1CCc2snnc21)N1C2CC(NC(=O)CCCC3CCCC3)(C2)C1 Cc1cn(C)nc1C(=O)NCCC(O)CNC(=O)C(N1CCCC(C)C1)=O C12(C(=O)NC3(CC=C)CCN(C(=O)CCCN(C)CC)C3)CCC(C)(CC1)CO2 N1(C(C(C)SCC)=O)CCCC(C2(NC(c3cncc(Cl)c3)=O)CC2)C1 Cc1ccn2nc(C(=O)NC3CCN(C(=O)C4=CCCCCC4)C3)nc2n1 c1(-c2c(OC)cccc2F)ccc2[nH]nc(C(=O)NCCNC(C)=O)c2c1 N1(C(C#C)C)CCN(C(c2ccc(CNC(=O)C(F)C3CCOC3)cn2)=O)CC1 C1(C(N(C)CC2CN(C(=O)C(=O)NC3CC3)CCO2)=O)CC2CCC1C21CC1 N1(C(C(C)=C(C)C)=O)CCOC(C)(CNC(=O)CCC2CCCCC2)C1 N#Cc1cnc(NCC2CC(NC(C3CC3F)=O)C2)cn1 c1(CCC(=O)NCCC2(SC3CCCCO3)CC2)ccc(NS(C)(=O)=O)cc1F C1(COC(C(CC)(C)C)=O)CCN(CC2CC2)CC1F C1(C(=O)NCC2CC(OC)CN2C(=O)CCN(C)CCO)Cc2ccccc2C1 C(=O)(C(C)(C)CCSC)N(C1CCN(C(=O)CCC=CC(C)C)C1)CCC C1(CC)(CC)CCN(C(C2CCN(C(c3ccc(C)n3C)=O)CC2O)=O)CC1 C1(COC(c2ccc(C)nc2O)=O)CC(NC(=O)OC(C)(C)C)C12CC(F)(F)C2 C(=O)(CCC(=O)NCC1CCC1C(=O)NC1(CCO)CCOC1)NCC Cc1ncc(N)cc1C(=O)NC(C(C)NC(=O)Cc1ccc(F)c(F)c1)C(C)C C1(O)(Cc2cn(CCC=C)nn2)CCN(C(=O)CCSC(=S)SCCC)CC1 CC1(C)CCC(C(N2CCC2CNC(c2cc(CO)on2)=O)=O)C1.C(C)(C)(C)O N#Cc1cc(F)ccc1NC(c1ccc2c(c1)CNS2(=O)=O)=O C1(NC(C=CCC)=O)C(C)(C)CN(C(C23OCCCC2C3(F)F)=O)CC1(C)C c1(N2CCC(NC(COCc3cc(C)no3)=O)C2)nc2cccc(F)c2o1 C(=O)(C1=CCCC1)NC(c1cn(CCOCCOCC2NC(=O)OC2)nn1)C c1(C(=O)NCC(C(C)C)(C)NC(=O)C(C)c2cc[nH]n2)occ2c1CCOC2 c1(CC(C)C)cc(C(=O)NCCC(C)NC(=O)CC2COCC2O)n(C)n1 C1(NC(C(=O)N(C)CC2CCCS(=O)(=O)C2)=O)C2Cc3ccccc3C12 C1(NC(CCC=C)=O)CCOC(C(=O)NCc2cc(C)ncn2)C1 C1(CNC(c2ccc(C)c(CO)c2)=O)COC(C)(C)CN1C(c1ccoc1C)=O c1(CN2CC(F)C(=O)N3CCC(C3)C2(C)C)ccc(C)nc1.C1(OCC)CC(OC)CC1 CC1C(CO)CCCN1C(C1(c2ccc(C(F)(F)F)cc2)CC1)=O C(C1COC(C)(C)O1)=CC(=O)NC(C)CNC(=O)CC1CC(F)C1 c1(CCC)nc(C(C(=O)NCC2CC2)N(CCOCc2ccccc2)C)cs1 c1(C(N2C(CNC(c3c(OC)oc(C)n3)=O)CCC2)=O)cc(S(N)(=O)=O)c(C)o1 N1(C(C(CCC)OC)=O)CC2(C1)SCCC2NC(=O)CC1=CCOCC1 C(=O)(C1=NOCC1)NC(C1CCN(C(c2c[nH]nc2-c2ccoc2)=O)CC1)(C)C CC(C)CC(O)C(=O)NCCC(C)N(C)C(c1cnc(Cl)n1C)=O c1(C(=O)NCc2ncoc2C2(C)CC2NC(=O)C(F)OC(F)(F)F)ncccc1F N1(C(=O)CC2CC(F)C2)CCC(C(F)F)(CNC(C2(CCF)CCC2)=O)C1 C(=O)(CCC(C)(C)F)NCC(CO)NC(Cc1cc(C)on1)=O N1(C(C(C)(C)C2CCOCC2)=O)CCC(C)(CC(=O)NCC2CCOCO2)C1 N1(C(Cc2cc(OC)ncc2)=O)CC(NC(c2cc(F)n(C)n2)=O)CC(O)C1 C1(C(NOCC(=O)OC)=O)CCCN(C(=O)C(C2CC2)OC)C1 c1(C(=O)NC2C(NC(CC=CC=C)=O)CCC2)cc2ccc(C)cc2nc1C c1(OC)cc(C(N2CCC(CC(=O)NCc3nccnc3SC)C2)=O)cc(Cl)c1 Cc1cc(C(N2CC3CN(Cc4ccc(Br)cc4C)C3C2)=O)cnc1Cl C#Cc1ccc(C(=O)NCCCCNC(=O)C(CO)NC(N)=O)cc1 CCCC(C(=O)NC(C)CCCCNC(=O)COCc1ccc(F)cc1)OC CC(c1cnn(C)c1)=CC(=O)NC12CCC1CN(C(=O)COC1CCCC1)C2 N12CC3C(C3C1)CC2=O.C(COCC)(C(=O)OC)NC(C1C(=C)C1)=O C(=O)(C(C(C)C)c1cccnc1)NCC1N(C(c2nc(NC(C)=O)sc2)=O)CC1 C(=O)(C#CC1(C)COC1)N1CCC(C(N2CCC(CC#C)C2)=O)C1(C)C Cc1cccc(C(C)(C)CNC(COC2CCCC2)C(=O)O)n1 C(=O)(CCC(=O)N(C)C)N(C1CCCCN1C(=O)C1=NOCC1)CCC C12(NC(C(C)Oc3cccnc3)=O)CCC(CNC(=O)CNC(N)=O)(CC1)OC2 C1(CNC(=O)CCCF)CC2(CC(NC(c3ccncc3F)=O)CCS2(=O)=O)C1 CON(CCC(=O)N1CCOCC1C)C(=O)C1CC(=O)C1(C)C c1(C(N(CC(C)NC(=O)CC(C)c2ccco2)CC)=O)ncc(F)cc1F Cc1cc(C(c2nnnn2C2COC2)NCc2cc(C)[nH]n2)c(F)c(Br)c1 c1(CCNC(c2ccc(-n3cc(-c4cnsc4)nn3)cc2)=O)cc(Br)ccc1Cl CCC(C)(C)C(=O)NCC1(C(N2CC(C)(CO)C2)=O)CCCCC1 C1(C(=O)NC(CC(C)NC(c2c(C)c(C3CC3)on2)=O)C)CCC(N=[N+]=[N-])C1 c1(CN2CCC(CNC(c3c(C)nc[nH]3)=O)C2)ccc(C(=O)O)cc1Cl c1(OC(C)=O)ccc(NC(C2CCCCN2S(C)(=O)=O)C)cc1 c1(C(CC)=O)cc(C(=O)NCC2(NC(=O)CCSC)CCCCC2C)ccc1F N1(C(C2(COC)CCCC2)=O)CC2OCC(NC(=O)CC3CCCN3CC)C2C1 C1(CC)OCCC1C(=O)N(CC(O)CN(C)C(c1cc(O)cs1)=O)C CCC(C)(O)C(=O)NC(CNC(c1ccsc1OC)=O)CO N1(C(C(C=C)(C)O)=O)CC(CC(=O)NCc2nc(C)sc2C)CC1(C)C CC1(C)CCN(C(=O)C=CC2CCCC2)C1C(N1CC(F)(F)CC1CO)=O c1(OC)cc2c(cc1C(N1CC(NC(=O)C3=NNC(=O)CC3)C3CC13)=O)CCC2 C1(NC(c2n(CC)ncc2Br)=O)CN(C(C23CCC2CC3)=O)CCC1C C1(N(C(=O)CC(F)F)C)CCCN(C(C2CC(F)(CO)C2)=O)CC1 N1(C(c2ccn(C(C)C)c2)C(=O)NC(C(=O)OC)C)CCCC2CCC(C)CC12 N1(C(C2(CC)COC2)=O)CCCC(C(N2CCCCC2C(C)CO)=O)C1 CCC(C)(C)C(=O)C(=O)NCC(F)(C(=O)N1CC2C(CO)C2C1)C(C)C c1(C(=O)NCCN(C(=O)C(C)(O)C2CC2)C(C)C)cc([N+](=O)[O-])ccn1 C1(CNC(C(C)OCCC=C)=O)CN(C)CCN1C(=O)CNCc1cscn1 CC1(C)CC(NC(c2nc(Cl)cs2)=O)CCN(C(c2cncn2C2CC2)=O)C1 c1(NC2CC(F)(CNC(C3(C#C)CCCC3)=O)C2)ncnc2c1nnn2C c1(NCCC(C)=CC(=O)NC2CCC2CNC(=O)CNS(C)(=O)=O)ccccc1 C1(F)(CNC(C2C(C)(C)C2(C)C)=O)CCCN(C(C2CCCCC23CC3)=O)C1 C1(CNC(C2N(CC)CC2)=O)(NC(c2cccc(F)c2N)=O)CCC(C)(C)CC1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC2(CC1)OCCC2NC(=O)CSC(F)F S(=O)(=O)(c1cccs1)NCCC(=O)NC1CC2(C1)CC2NC(=O)C1=CCCC1 C(CC(C(=O)OCC1CCC1OC)NC(=O)OC(C)(C)C)=CC C1(C(N2CCC(C=C)C2)=O)CCN(C(=O)C2CCOCC2)O1 C1(CNC(CC)=O)CCN(C(C2CCCCC2(C)C)=O)C12CC2 C(c1ccccc1Cl)=C(C)C(=O)N1CC(NC(C2(C)CC2C)=O)C1 N1(C(Cc2n(C)cnn2)=O)CCCC(N(C(=O)C=Cc2cncs2)CCF)C1 Cc1ccc(C)n1CC(=O)OCc1cccnc1 c1(C(N(C(C)CNC(=O)CCc2nncs2)C)=O)ncc(C#N)cc1Cl C1(NC(C2(C)CC2C(F)(F)F)=O)CCC2CN(C(c3cc(O)cs3)=O)CC2C1 C1(C(C)NC(CC(=O)NCC)=O)CN(C(C2C=C2C)=O)CCO1 c1(OCC)cc(CC(=O)NC2CC(C(=O)Nc3cc(I)cnc3Cl)C2)cc(C)c1 C1(C)(NC(C=C2CCC(C)CC2)=O)CCCN(C(=O)CCc2nncn2C)C1 N1(C(CC(COC)NC(C2(C)CCCN2C)=O)=O)CC(C)C(C)C1C C1(NC(CSC(C)C)=O)CC(NC(=O)CCC(=O)N2CCC(O)CC2)CCO1 n1(CC(N2CC(NC(C(C)=CC)=O)C3C2C3)=O)ncc(C#N)c1N C1(C(=O)Nc2ncc(C)cc2Cl)CCCC12CCN(C(C1CC1F)=O)C2 C1(C)(CNC(C2N(S(C)(=O)=O)CCC2)=O)CC(F)(F)CN1C(c1cnnn1C)=O C1(C(=O)NCC(CC=C)NC(=O)CCc2ccncc2)CCCCN1CCC N1(C(C2CCN(C(=O)C3C(C)CCO3)O2)=O)CCc2nc[nH]c2C1 c1(C(N2CCC(NC(C=CC(N)=O)=O)C23CCC3)=O)ccc2c(c1)NC(=O)NC2 Cc1cc(C)c(C(=O)NC(C2CN(C(C3CN(C)C(=O)N3)=O)CCO2)C)[nH]1 c1(C(=O)NCC2C(C)CN(C(c3ccncc3)=O)CC2)ccc(O)c(F)c1F c1(C(C)NN2CCCC(C(C)(C)C)CC2)ccc(Cl)c(Cl)c1 C1(NC(C(CCC)C)=O)CCN(C(c2c(F)cc(Cl)cc2F)=O)CCC1(F)F Cn1cc(C(=O)NC(C)(C)C(=O)NCC(F)CNC(=O)C(F)=CCCF)cn1 c1(C(C(N2CCN(C(C(CC)OC)=O)CC2)=O)OC)cc(F)cc(F)c1 N1(C(CSC(C)C)=O)CC2ON=C(CNC(c3cc4occc4s3)=O)C2C1 C1(C)(CNC(CN(C2CCC2)C)=O)CN(C(=O)C(O)CC(F)(F)F)C(C)(C)C1 C(CCN=C(NCCC(C)(F)F)NC1Cc2ccccc21)SC C(=O)(C1=CCOCC1)NC(CSC)(C)C(=O)NCC(C)(O)C1CC1 Nc1ccnn1CC(=O)NC1CC(CNC(=O)Cc2csnn2)C1 CN1CC2(CCN(C(=O)C(c3ccccc3)NC(C3CS(=O)C3)=O)C2)C1 Cc1nc(C)n(O)c1C(=O)NCCC1CCN(C(=O)CCSc2nccn2C)C1 C(=O)(C1=CC2CC=CCC12)N1CCC(CNC(c2c(C)[nH]c(C)c2C)=O)CC1 N1(C(c2c(C)scc2)=O)CCC(CNC(C2(C(F)(F)F)CC2)=O)C(O)C1 N1(c2nn(CC)c(C3CC3)c2)CCC2(CCCC2C(N2CC(C)(C)C2)=O)CC1 N1(C(C(COC)OC)=O)CCC2(CC1)CC2C(=O)NCCNC(=O)CCOC N1(C(=O)C(F)C2CCC2)CC2CC2(C(=O)NC2CC(F)(CF)C2)C1 c1(SCC(=O)N(C2CC3CCC(C2)N3)CC2CC(C)C2)ccc2c(c1)OCO2 C1(C(=O)NCC2(C)CC2)CC(O)CN1C(=O)C(C)N1CCCC1 N1(C(CC(=O)NCC)=O)CC2C=CC1C(C(N1CC(S(C)(=O)=O)C1)=O)C2 c12cc(Br)cnc1CNC2=O.C1(CC)CCCCC1SCc1cscn1 c1(OC)ccc(I)c(C(=O)OCCCCCCn2cc(CCCC(C)=O)nn2)c1 CCC(C)CC(C(=O)NOCCCF)NC(=O)CCc1cccn1C N1(C(C(CCC)OC)=O)CC2CCC2(CC(=O)N(c2ccc(F)cc2)C)C1 N1(C(COCCOC)=O)CCN(C(C2CC23CC(O)C3)=O)C2(CCC2)C1 c1(CC)nc(N2CCC(NC(=O)CC(F)(F)CC)C(C)C2)c(F)c(Cl)n1 c1(CC(NOCC(=O)NC(C)=O)=O)cc(Cl)sc1Cl c1(N(CCNC(CCC2C(C)=NOC2=O)=O)CC2CC2)ncc(C#N)cc1Cl C1(C#CC(=O)OC(CC2CCCCC2)C(=O)OC)(CC)CC1 C(=O)(CCCCN(C)C(C1CN(C(C)=O)C1)=O)NCc1n(CC)ncc1 c1(CN2CC(n3cc(C(=O)Nc4csnc4C4CC4)nn3)C2)ccc(F)cc1 Cc1cc(NC(=O)NCC(c2c(F)cccc2F)N(C)C)cc([N+](=O)[O-])c1 C1(C)(C(=O)NCC2=CCCN(C(COCCCC)=O)C2)CCc2ccccc2C1 N1(C(Cc2cc(C)no2)=O)CCn2nc(CNC3CNC3)nc2C1 N1(C(CCC=CCC=C)=O)CC(C(=O)NCc2n[nH]c3c2CCC3)CCC1(C)C N1(C(C2C(=C)CC2)=O)CCCC(NC(C2(O)COC2)=O)C1C N1(C(c2c(C)nco2)=O)CC2CC(NC(c3ocnc3C(F)(F)F)=O)C(C2)C1 CC1CCOC(C(N2CCC(N3CCN(C(C4(CCO)CC4)=O)CC3)CC2)=O)C1 c1(CN(C(C2CCN(C(C3CC(C)OC3=O)=O)C2)=O)CC)ccccc1COC c1(C(NNC(=O)NCC)=O)cc(Br)cc(S(N)(=O)=O)c1C c1(C(N2CCC(C)N(C(C3CC3(Cl)Cl)=O)CC2)=O)cc(F)cc2nn[nH]c12 Cc1ncc(N)cc1C(=O)NC(C)CN(C(=O)C(c1c(C)noc1C)C)C CCCCC(C(=O)Nc1ccc(C2SCCCS2)cc1)NC(=O)COC Cc1cccc(F)c1CC(=O)NC1CCCC1CNC(c1[nH]c(O)nc1C)=O N#Cc1cccc(NC(=O)CCNC(=O)NC2CCC(F)C2)n1 c1(OCC(N2C(C)C(NC(C3CCCC(=O)N3)=O)CC2)=O)ccc(F)cc1Cl N1(C(C(CCOC)NC(=O)C=Cc2ccncn2)=O)CCC2(C=CCO2)CC1 C12CS(=O)(=O)CC1NC(=O)C(=O)N2.c1(C(=O)NCC2CC2)ccoc1C1CC1 CC(C)(C)CCC(F)C(=O)NCC(C(=O)NCC1C2CCCCCC12)C(C)(C)C C12(CNC(=O)C=CC3CC3)CC3CC(CC(C3)C1NC(C1(CCF)CC1)=O)C2 C(C(O)CN(C)C(C1(CO)COC1)=O)N(C(C=C(COC)C)=O)C Cc1nc(-c2cn(C(C)C(=O)NC(C(C)C)c3cnn[nH]3)nn2)sc1C Cc1nc(C(=O)NCC(F)CNC(=O)CCn2cccnc2=O)c2ccnc-2[nH]1 c1(C(N(C(CN(C(c2c(C)ncs2)=O)C)C)C)=O)cncc2sccc12 C(=O)(CC(C)CC(C)(C)C)N1C(CNC(c2c(OC)nc(Cl)cc2)=O)CC1 C(=O)(C1=CCCCCC1)N1C(C)CC(NC(c2ccc(C(F)F)cc2)=O)C1 c1(C(N2CCC3(CC2)OCCO3)=O)csc2c1CCN(Cc1sccc1Br)C2 Cc1ccccc1C1CCN(C(c2ccc(OCF)cn2)C(=O)NC2(C)CC2)C1 C1(C)(CC)CC(NC(c2csc(C)c2NC(N)=O)=O)CN1C(=O)CSC C(C)(C)(CCCNC(=O)Cc1ccn(C)n1)NC(C1CCC(C)C1)=O c1(CCN2CC(C(=O)NCc3cccc(C(C)=O)c3F)C2)nsc2ccccc12 C1(CC#C)(C(N2CCC(CO)(NC(=O)C(O)C3CC3)C2)=O)CCCCC1 c1(CCC(=O)NC(CN(C)C(C2CC3CCC2C3)=O)(C)C)ccccc1Cl CS(=O)c1ccc(CN2CCC(C(=O)O)CC23CC3)cc1 c1(C(=O)NCC2CCC(NC(=O)CC3CCSC3)C2)c(F)cc(O)cc1F c1(C(N(C)CC2CCN(C(c3c(C)ccs3)=O)C2)=O)ccc(OC(F)F)cc1 c1(C(=O)NCC2(O)CCN(C(=O)C=Cc3cc[nH]c3)C2)ccc(CO)cc1F.N c1(CC(N2CC(CCCCNC(C(C=C=C)C)=O)C2)=O)ccc(F)c(C)c1 c1(C(=O)NCC(CC(C)C)CO)n[nH]c2c1CN(C(=O)Cn1cccn1)C2 C(C)(C(C(=O)NCC(c1cnn(C)c1)O)NC(c1csc(Cl)c1)=O)OC C(=O)(C1=CCc2ccccc21)NC(CC)CNC(=O)C(c1cccc(C)c1)O C1(CC)CCCCC1C(=O)NCC(C1CCN(C(C2(O)CCCC2)=O)CC1)C CS(=O)C=CC(=O)NC1CCN(C(=O)CC2CN(C(=O)OC(C)(C)C)C2)CC1 Cn1cc(S(N)(=O)=O)c(C(=O)NCC2CCN(C(c3cnco3)=O)C2(C)C)n1 CCS(=O)(=O)CC(=O)N1CCCCC1CN(C(c1cn(C)[nH]c1=N)=O)CC C1(CC)CCC(C(=O)NC2CC(CNC(=O)C(C)Cc3ccncc3)C2)O1 c1(C(=O)NCC#CCNC(c2ncc[nH]c2=O)=O)[nH]cc2c1CCS2(=O)=O c1(NC(C2C(C)S(=O)(=O)CC2)=O)ccc(F)c2ccccc12 C#Cc1cc(NC(=O)CCOC2CN(C(=O)C=C(C)C(C)C)C2)cc(F)c1 N1(CC)CCCC1C(=O)NC(C1CN(C(c2ccc(Cl)o2)=O)C1)C c1(OCCC(=O)NCCCNC(C(C)CC2CCC2)=O)ccc(Cl)cc1 C(CC(F)F)(C(=O)NCC1Cc2nccn2C1)N(C(=O)CSC(F)F)C C1(c2n(C(CC)(C)C)nnn2)(Nc2cc(F)ccc2OC)CCCCC1N(C)C c1(C(C2CCOC2)CN(N2CCCOC2)CC(F)F)ccccc1C(F)(F)F c1(C(=O)NC2(C)CC(NC(=O)OC(C)(C)C)C2)csc(C(=O)NCC=CCF)c1 CN1C(=O)C(C)(C)c2cc(C(N3CCCC(O)C(F)C3)=O)ccc21 C1(O)(CNC(CCNC(COC(CC)(C)C)=O)=O)CCN(C)C1 c1(C(N2CC(CNC(C=CCCC)=O)C(C)C2)=O)cc(C)sc1S(N)(=O)=O N1(C(c2ccc(C)o2)=O)CCCCC1CC(=O)NCCc1[nH]cnc1C c1(OCC)ncccc1NC(=O)C(C)NC(=O)C(CC1CC1)OC N1(C(Cc2ccc(OC(C)C)cc2)=O)CC(NC(=O)CCF)CC12CCCOC2 c1(C(N2CCC(CNC(c3cocn3)=O)(CO)C2)=O)nnc2ccccc2n1 N1(C(C2(CC=C)CCOC2)=O)CC2(C1)CN(C(c1ccnc(F)c1N)=O)C2 C1(C(=O)OCC)OCCNCC1N(C(=O)CSc1ccsc1)CC(N)=O c1(C(N(C2CN(C(=O)C(C)(C)NS(C)(=O)=O)CC2F)C)=O)cc(C2CC2)ccn1 C1(C)(OC)CN(CC(=O)N(CCC)CCNC(c2cnsn2)=O)C1 c1(SC)cn(C)nc1C(=O)NCC(O)CNC(=O)C(O)CC1CC1 CCC(C)C(O)C(=O)NCC(C)(C1CC1)NC(=O)Cn1cc(C(F)F)cn1 C1(N(C(C2CC(Nc3nncs3)C2)=O)CC2CC2)CCCN(C(=O)CC)C1 CC1CN(C(=O)CC2CCC(=O)N2)C1C(=O)NCc1sccc1Cl c1(C(=O)NC(CNC(CCC(C)SC)=O)C(C)C)cccc2c1ccn2C C(CCCC#N)(c1n(CCOCC)nnn1)Nc1cccc(-n2cnnc2)c1 CCC(CC)C(F)C(=O)N1CC(C)N(C(C2SCCS2)=O)CC1C c1(OC)cc2ccccc2cc1NC(N1CCC(N)C2(CCC2)C1)=O Cc1c(C(=O)NCC2CN(C(=O)C(C)C)CCO2)[nH]c2c(C)cccc12 c1(-n2c(C(c3ocnc3Br)NC(C=C)(C)C)nnn2)cccc([N+](=O)[O-])c1 c1(C(N2CCN(C(c3cc(CC)ccc3C)=O)C(C)C2)=O)cccc2nc[nH]c12 C1(C(=O)NC(CC2CC2)C(=O)NCC(F)F)CC2(CCC2=O)C1 C1(CCC(=O)N(CCCCN(C(C(C)NC(CC)=O)=O)C)C)CCC(=O)C1 CC(C(=O)N(C)CCN(C)C(C1CCSC1)=O)n1ccnn1 c1(-n2c(-c3cnsc3)nc(-c3scc(C)n3)n2)cccc2cnccc12 Cc1csc2ncc(C(=O)NC3(CCCNC(c4cncn4C)=O)CC3)c(=O)n12 C12(C(C3CC3)CNC(=O)NC3(CO)C(C)C3)CCC(CC1)OC2 n1(CC(=O)NC2C(CC)CN(C(=O)CNS(C)(=O)=O)CC2)cc([N+](=O)[O-])cn1 C1(C(=O)NC2CC(F)(CNC(=O)CN3C(=O)CCC3=O)C2)CC2CCC1CC2 CC(C)C(C)C(C)CC(=O)NC(C)CN(C(=O)Cc1cnn2c1CCCC2)C Cc1c(C(N2CCCC(O)(CNC(c3cncs3)=O)C2)=O)nn2ccccc12 C(C(CNC(c1ncccc1O)=O)C(F)(F)F)NC(c1c(C(C)C)noc1)=O N1(C(c2nc(C)sc2C)=O)CC(NC(C23CC(F)(C2)C3)=O)C2CCCCC12 C1(CC=C)(NC(c2cncc(Cl)c2Cl)=O)CCN(C(=O)C(F)=C(C)C2CC2)CC1 c1(C(N(CC(O)CNC(=O)CC2CCCCCC2)C)=O)ccc2nsnc2c1 N1(C(=O)NC2CC(OC(C)C)C2(C)C)CCC(C)(C)C(CO)C1 C(C(=O)N1CCC(C(N2CCC23CCCCC3)=O)O1)C1C(OC)C1 C1(CC)CCCC1C(=O)N(C)CCN(C(=O)Cn1cc(C(C)O)nn1)C C=CC(CCC)CC(=O)N1CC(O)CCC1C(=O)NCC1(CC=CC)CCC1 C(CC1CCN(C(=O)CCOCCC(C)(C)C)C1)(C(=O)O)N(C)C c1(N(C)C)ccc(C(=O)NC2CCCC2CNC(C2CC(C)(C)C2)=O)cc1 C(=O)(C1CCc2nnc(C)n21)N(CC(CC)NC(c1ccc(F)c(F)c1)=O)CC CN1CCCCC(CNC(=O)C(c2ccco2)NC(=O)C2=CC(C)(C)C2)C1 C(C(C)(C)CC(=O)N(C)CC1(O)CCCN(C(=O)Cn2cnnc2O)C1)N(C)C N1(C(C2(CC)CC2)=O)CC2CC(NC(=O)CC3CCCC(C)C3)C2C1 C=C1CC(C(=O)NC(CC(N)=O)C2CC2)(CNC(=O)COCC(C)(C)C)C1 c1(CN(CC=C)Cc2ccc(N3CCCC3)nc2)cnc(OCC)nc1 N1(C(C(=O)NCCOC)=O)CCC(CNC(=O)CC(C)C)(OC)CC1 C#CC1CCCN(C(=O)CC2CCN(Cc3cc(N4CCCCC4)ccn3)C2)C1 C12(NC(c3cnc(OCC)s3)=O)CCC(CC1NC(C1C3CCCC13)=O)C2 c1(C(=O)NCCC2CCN(C(COCP(C)(C)=O)=O)C2)cccc(C=C(F)F)c1 C(C)(CN=c1[nH]c(C)nc(C)c1C)(C(C)C)NC(C(CC)NC(C)=O)=O C(=O)(C1CCC2(CCC(C)(C)CC2)OC1)N1C(CC)C(NC(=O)C=CBr)CC1 C1(CC=C)(NC(=O)C(N2CCSCC2)C)CCN(C(=O)C(C2CC2)C2CC2)C1 N1(C(CCC(C)(C)F)=O)CC2C=CC1C(C(N1CCC(C)(C#N)C1)=O)C2 c1(C(=O)NCC(CN(C(=O)CC2(N(C)C)CC2)CC)(C)C)cccc2scnc12 c1(N(C)CCC2CCCCC2)nc(N(C)CC2(CO)CCC2)c2c(n1)CCOC2 C1(NC(c2ccc(Cl)s2)=O)CCN(C(=O)CC(C2CC2)C2CC2)C(C2CC2)C1 C1(C(=O)NCCc2ccncc2F)(CC)CCCN1C(=O)Cc1sccc1C N1(C(c2cn(CCCOC)nc2)=O)CC2CC(C1)N(C(=O)CCC(C)N(C)C)C2 C1(NC(=O)OC(C)(C)C)CCCC1(C)CNC(c1ncncc1Br)=O CN1CCN(C(=O)CC2CCOC2(C)C)C(C(N2CC(N3CCNC3=O)C2)=O)C1 CCC(C(=O)NC(C1CCCCC1)CO)N(C)C(c1ccc(C)o1)=O N1(C(C2N(C(CCC#C)=O)CC(=C)C2)=O)CCC(C)(C#N)CC1 C1(C(N2CC3C(CNC(C=CCCC(C)C)=O)(C3)C2)=O)COC2(CO)CC1C2 O=C(CCC(F)(F)Cn1cc(C2CC(F)(F)C2)nn1)NCC1CC(O)C12CCC2 C(N=c1[nH]c2c(c(=NCC3(CO)CC=CC3)[nH]1)SCC2)C1C(C)(C)OCC1 Cc1cc2[nH]c(C(N3CC(NC(C4CCCO4)=O)C4(CC4)C3)=O)cc2s1 CCCCC(O)C(=O)NCC(C)(CC)NC(c1cccc(-c2nccs2)c1)=O c1(N(C(C(C2CCN(C(c3cccc(Cl)c3)=O)CC2)C)=O)C)ccccc1CO N1(C=O)CC2CC1CC2CC1CC(C(=O)NC(CSC)=O)C1 C(=O)(C(O)C(O)C(C)C)N(C1CCCCC1Oc1ccc(C(F)(F)F)cc1)CC c1(NC(C2CCCCC2)CC)ncccc1S(=O)(=O)N.C(C(C)C)CCN1CCCC1 C123CC1CC1CN(C2)C(=O)CC(CCC(=O)NC)C(=NC=CN=C1C)C(=O)N3 CN1CCC2(CCCN(C(=O)NC3COc4ccccc4C3O)C2)C1=O CC1CCC=C1C(=O)NCC1(O)CCN(C(=O)COc2ccc(F)cc2F)C1 C1(C2CCCCC2)(C(=O)NC2CC(C)(NC(c3c(C)nc(C(C)C)s3)=O)C2)CC1 CC1CCCN(Cc2cccc(NC(=O)Cc3cccc(-n4cncn4)c3)c2)C1 Cc1nn(CC(F)F)cc1C(N1CC(CNC(C2CCS(=O)(=O)N2)=O)C(O)C1)=O N1(C(c2nccc(CC)c2)=O)CCC(C)N(C(=O)C(c2cncnc2)C)CC1 CCC(C)(C(=O)N1C2CCC1CN(C(=O)C(F)=C1CCCC1)C2)C(F)F C1(NC(COCC)=O)CC(F)CN(C(=O)CNC(c2ccoc2)=O)C1 N1(CC=C)CCN2C(=O)N(CCNC(c3c(OC)ccc(F)c3F)=O)CC2C1 Cn1nccc1C(C)NC1CC(C(C(=O)NCC(F)(F)F)NC(=O)OC(C)(C)C)C1 C1(NC(C(CC)CO)=O)CCC2CCN(C(=O)C(c3ccc(F)cc3)=O)C1C2 N1(C(Cc2c(C)cco2)=O)CCN(C)C(CNC(=O)CC2CC3(CC3)C2)C1 C1(NC(=O)Cc2cc[nH]c2)CC2CC(NC(C3(CO)CC3(F)F)=O)CC2C1 CCC(C)(C)C(O)C(=O)N1CCC2(CC1)CC2C(=O)NC1CC2CCCC2C1 CC1Cc2cc(C(=O)NC3CC(F)CN(C(C4CN(S(C)(=O)=O)C4)=O)C3)ccc2O1 Cc1cnc(C(=O)NCC2CC2CNC(C2(CCO)CC2)=O)nc1 C(=O)(CCC(=O)NC)NCC1(F)CC(NC(C(c2cn(CC)nc2)(F)F)=O)C1 C1(C2N(C(C3(CC(=O)OC)CC3)=O)CCC2)CCN(C(C2CNC(=O)N2)=O)CC1 C(CC(C)C(=O)N1CCC(O)(C(=O)NC(c2ccsc2)C)C1)=CCC N1(C(C(C2CCC2)OC)=O)CCCC1C(=O)NC(C)CC(C)C CC(C)C1=NOC(C(=O)NC(CCN(C)C)C(=O)NC2COC(=O)C2)C1 C1(NC(C2CN(CCC)C(=O)C2)=O)CN(C(=O)C(F)=CC2CC2)CC12CCC2 S(=O)(=O)(c1c[nH]c(=NCCOC2CCC2)cc1C)NCC(CSC)OC N1(C(C2CN(C(=O)NC)C2)=O)CCC(NC(C2C(C)(C)C2(F)F)=O)CC1 C1(OCCNC(C2(CCOC)CCC2)=O)CCN(C(=O)CC2CC2(C)C)C1 C1(CC(=O)NC2C3CCN(C(C(COC)C)=O)CC32)CC(C)CC(C)(C)C1 N1(C(C2C(=C)CC2)=O)CC(C)OC2(CCN(C(C3CC(C)(C)C3)=O)CC2)C1 c1(CC)ccncc1NC(C1CC(O)(CNC(C2CCCN2C(N)=O)=O)C1)=O C1(CNC(C(CCOC)C)=O)CC2COCC2N1C(=O)C(C(C)C)n1cnnc1 C(=O)C(C)(F)C(C)(C)F.N1CCC2(CCC2)CC1.CC1CN2CCC1CC2C c1(CC)ncsc1C(=O)NCCC1(NC(=O)C(CC2CC2)OC)CCCC1 N#CC1(C(N2CC(F)CC2CNC(=O)Cc2csc(Cl)c2)=O)CCCO1 N1(C(C2C(CNC(C(C)C3CCC3)=O)C2(C)C)=O)CC=CC(O)C1 N1(C(CC2C=NN(C)C2=O)=O)CC(CO)C2(C1)CN(C(C1(CC#N)COC1)=O)C2 N1(C(=O)Cc2ccc(F)cn2)CC2OCCN(C(C3CC4CCC3C4)=O)C2C1 N1(C(CC(C)(C)O)=O)CC2CCOCC2(NC(C2C=CC=CC=C2)=O)C1 C#CCCCC(C)C(=O)NCCCNC(c1ccc(Br)s1)=O N1(C(C(CC)O)=O)CCC2CN(C(=O)COCCOC)CC2C1 CCC(O)CC(=O)N1CC(=O)CC1C(=O)Nc1cn(CCF)nc1C C1(CNC(C(C)(C)CO)=O)CN(C(=O)COCCO)CCC1(F)F N1(C(CCC(=O)N(C(C)C)C)=O)CCOC2(C1)CN(C(c1cnnn1C1CC1)=O)C2 C(CC1=CCN(C2CCCCC2)CC1)NC(=O)COC1CCCC1 C(=O)(N=c1nc(-c2ccccn2)[nH][nH]1)NC1C(CC(=O)OC)C(O)C1 c1(C(=O)NCC2CN(C(C3CCCC(F)C3)=O)CCO2)cnc2cccnn12 C(=O)(C1=CNC2=NCCC2=C1)N(C1CCN(C(C2CCCS2(=O)=O)=O)C1)C c1(C(C(N2CCC(N(C)CC)C2)=O)(F)F)cc(C(F)(F)F)cc(F)c1 C1(NC(c2cncc(COC)c2)=O)CC2CC(C1)N(C(=O)C(C)(C)C1CCC1)C2 N1(C(C#C)C)CCN(C(=O)CC2(NC(C3CCC(O)C3)=O)CC2)CC1 N1(C(=O)OC)CC2CC(N(C3CCC3)CC)C2C1.N(CCN(C)C)CC c1(C(N2CC(NC(c3c(COC)scc3)=O)C(C)(C)C2)=O)occ2c1CCCC2 c1(CC(C)C)nc(C(=O)NC23CC(NC(C4CCO4)=O)(C2)C3)cs1 c1(CN2CC(NCc3c(OC)ccc(Cl)c3)C(C)C2)ccc(S(=O)(=O)NC)cc1 C(c1ccccc1)=C(CC)C(=O)NCC(C1CC1)NC(c1ccncc1OC)=O CC12CCC(C(=O)NC3CCCCC3CC(=O)N(CCO)CC3CC3)(CO1)C2 N1(C(C(C=C)CC)=O)CCC2CCN(C(C3CCCN3N=O)=O)CC12 CCC(O)C(C)C(=O)N1CCC(C)(NC(C2CC3CCC(C2)C3)=O)C1 c1(C(=O)NC2CC(F)(CNC(C=CC=CCC)=O)C2)cccn2[nH]c(=N)nc12 Cc1c(C(=O)NCC(C2CC2)NC(=O)Cn2cnc(=N)[nH]2)cnn1C1CC1 CCCCC(O)CC(=O)NCC1CN(C(c2ccc(C3CC3)s2)=O)CC12CCC2 C(CCCC(=O)N1CC(CNC(=O)CCCN(C)C(C)=O)C(C)C1)OC c1(OCC=C)ccc(CC(=O)NC(C)(C)CN(C(=O)C2=CCSC2)C)cc1 C1(CCC)CN(C(=O)C(F)OC(F)(F)F)CCN1C(=O)CC1CCSCC1 CC#CCC(C(=O)NCc1cc(CCC)no1)NC(=O)C(CC)OCC Cc1cc(N2CC3CC(NC(=O)CC4CC5CC5C4)CC2C3)n2ncc(C)c2n1 N1(C(C2CCC(C)O2)=O)CCC(C(F)(F)F)C(N=c2nnn(C)[nH]2)C1 N1(C(C2(OCC)CCC2)=O)CC(NC(c2cc(Br)co2)=O)CC(C)(C)C1 c1(C(=O)NCC2COCCN2C(=O)C2=COCCO2)cc(Cl)c2ccccc2n1 C(=O)(CC(CN(C)C)C(F)F)NC1C(NC(c2cn(CCOC)nn2)=O)CCC1 O=CN1CCCC1C(N1CCCC1C1CCN(C(=O)COc2ccon2)C1)=O CC(C)(C)CC(=O)N1CC(F)(C(N2CC(n3cnnc3)C2)=O)C1 CC1(C)CCC(CNC(c2n[nH]c(C(C)(C)C)n2)=O)N(C(=O)CCC(N)=O)C1 c1(C(=O)NCCCCCN(C)Cc2onc(CCCCC)n2)sc(F)cc1C c1(CNc2cn(C)c(C(=O)Nc3c(F)cc(Cl)cc3F)c2)ccc(F)c(F)c1O CS(=O)(=O)c1cnn(CC(=O)NCC2CCC(NC(=O)OC(C)(C)C)CC2)c1 C(=O)(CCCCC(F)(F)F)N1CCN(C(=O)CC2CCOC2)CC1CF CC1CC(=O)NC(C(N2C3CCC2C(NC(=O)C2=CCCCO2)C3)=O)C1 C12(C(=O)NCCn3cc(CSC)nn3)COCC1C2(F)F C(=O)(C(C)S(=O)(=O)C(C)C)NCCCN(C(=O)CCC1(C)CCOC1)CC C(=O)(C(c1ccccc1)=CC(C)(C)C)NCC1C2N(C(C=C(C)Cl)=O)C(CC2)C1 c1(Cn2cc(C3N(C(C4(CO)CCCO4)=O)CCC3)nn2)ccc(F)cc1Br CN=c1ccc(C(=O)NC23CC(CNC(=O)Cc4ccsc4C)(C2)C3)c[nH]1 N1(C(Cn2nnc(C)n2)=O)CCCC(F)(CNC(=O)Cc2nc[nH]n2)C1 C(=O)(C(CNC(C1(CC)CCCO1)=O)CC1CCCC1)NCCC#CCC c1(C(C)=O)ncc(C(=O)NC(C)CCNC(c2cnc(C3CC3)[nH]2)=O)s1 O=C1NCC(C(=O)N2CC(NC(c3ccc(CO)nc3)=O)C2)c2ccccc21 N1(C(N=c2c(Br)cn(CC)[nH]2)=O)CCCc2cc(Br)c(Cl)cc21 c1(OC)cccc(OC)c1CCNC(C1(C#N)CCCO1)=O C1(C#N)(C(=O)NC(CNC(c2c(C)nc(C)s2)=O)CO)CC2(CC2)C1 N1(C(n2ccc(CC)n2)=O)CCC2CC12C(N1CCC1)=O Cc1c(C(=O)NCCN(C(C2CC(C)CCO2)=O)C(C)C)[nH]c2c(Cl)cccc12 c1(C(=O)NC2CC(NC(c3cocn3)=O)C2)cc2ccccc2c(=O)o1 C(C(=O)N(C1CCCCCC1)CCNC(=O)C(F)CC1CCC1)(C(C)C)SCC C1(C(=O)NCC2CC(C)N(C(=O)CN3CCOCC3=O)C2)COCCN1C=O Cc1cc(C(=O)NCC2(O)CCN(C(C3CC3C)=O)C2)c2c(C)nn(C)c2n1 Cc1ncc(F)c(C(N2CC(C(C)NC(=O)CSc3ccncc3)C2)=O)n1 C1(C(=O)NCC(c2ccncc2)C)CCN(C(=O)CSC2CC2)C(C)C1 Cc1cc(N)n(-c2cc(N3CCC(n4ccc(C(F)(F)F)n4)CC3)ncn2)n1 N1(C(C(F)OC)=O)CC(CNC(c2cc(C)oc2C)=O)C2CCCCC12 c1(NC(=O)NCC2CC(O)CC(CC=C)O2)cc(P(C)(C)=O)cs1 C1(C(=O)O)(NC(c2cncc(C(C)(F)F)c2)=O)CC2CCC1CC2 C1(NC(C(CCC)(C)CC)=O)Cc2ccccc2C1NC(=O)CCc1cc[nH]n1 c1(C(=O)NC2C=CCN(C(C(F)=CCC)=O)C2)cc2cc3c(cc2[nH]1)OCCO3 c1(C(N(C2CCN(C(=O)CC3COCCO3)C2)C)=O)csc(Br)c1Cl CCC1=C(C(=O)N2CCC2CNC(c2ccc(C3=CCCC3)s2)=O)CCCO1 c1(CNc2cn(C)nc2)ncn2c1CN(S(=O)(=O)Cc1cccc(C#N)c1)CC2 C1(C(=O)NCc2cncc(C(=O)NCC(CC)C)c2)CC2CC1CC2=O CCCC(C(=O)NCC1C2CC1N(C(C1CN(S(C)(=O)=O)C1)=O)C2)NC(N)=O N1(C(C(C=C=C)C)=O)C2CCCC1CC(NC(=O)COc1ccccc1)C2 c1(C(N2C(CCNC(C3CCN(C)C(=O)C3)=O)CCC2)=O)cc(F)c(N)cc1F C(=O)(CCCCCC(C)O)NCCC(C)NC(c1cnc(C2CC2)nc1)=O N1(C(C(C)SC)=O)CCC2(CC1)CN(C(C1CCN(S(C)(=O)=O)C1)=O)C2 c1(COC(C(c2ccccc2)NC(C(CC)O)=O)=O)cnc2ccoc2c1 N1(C(c2ncc(OC)cn2)=O)CCC(NC(c2ccc(C(F)F)s2)=O)C12CCC2 C1(CNC(C2CC(=O)NC2)=O)CCN(C(C2CC(CCO)C2)=O)CC1(F)F C1(CC(NOC)=O)CCCN(C(C2(OC)CCC2)=O)C1 c1(C(=O)NC2CC(N(C(CCN(CC)CC)=O)C)C2)ccc(Cn2ccnn2)o1 N1(C(C(C=C)(F)F)=O)CCC2(C=C(C(=O)NCc3nn[nH]c3C3CC3)C2)C1 n1(Cc2onc(C3C(C)C3)n2)c(=O)sc2ccc(-c3ccccc3)cc12 N1(C(c2c(-n3c(C)ncc3)nccc2)=O)CC2(C1)OC(=O)Nc1cc(Cl)ccc12 N1(C(C(c2ccccc2)OC)=O)CCCC2(C1)CN(C(=O)CCC1CCCO1)C2 c1(N(C)C)cnc(C(=O)NCC2CCCC2NC(=O)C(C)(C)O)cn1 N1(C(C2(C#C)CCC2)=O)CCC2(CCC2NC(=O)C(CC2CC2)OC)CC1 C1(CCC(=O)NCCCC(C)NC(c2ccnc(Cl)c2)=O)NC(=O)NC1=O C#Cc1cc(F)cnc1NC(C1CN(Cc2[nH]c(C)c(C(=O)O)c2C)CCS1)=O c1(C(N2CC(NC(C3CSC3)=O)C3(C2)CC3)=O)ccc2c(n1)COCC2 c1(NC(C(C)C)C)ccc(S(=O)(=O)NCC(O)C(C)C)cc1F Cc1ccc(C(=O)NC2CN(C(=O)COc3cc(Cl)ccc3Cl)C3CC23)nc1C CCCC(C(O)C(=O)NCCC(C)(C)N(C)C)NC(=O)C=CC1CCCC1 Fc1ccc(CNCc2cc(-c3cccc(Br)c3)no2)cc1N1CCCC1 N1(Cc2ccc(C)c(O)c2)CC2OCCN(C(c3ccccc3C(N)=O)=O)C2C1 Cc1nc(O)c2cc(NC(=O)C(=O)NCC3(C)CCCCC3)ccc2n1 c1(OCC)cc(CN(C)C(=O)Nc2ccc(F)nn2)cc(F)c1OC Cc1cc(=NCC(c2ccccc2F)NC(=O)CC2CCCCC2(C)C)[nH]cn1 c1(C(=O)NCC2C(CC)CCN2C(=O)C2=C(C)CC2)nc(C)ccc1C C1(NC(C(C)(F)F)=O)CN(C(c2ccccc2-c2cnco2)=O)CC1C#N C1(CCNC(C2CCC2CF)=O)CCCN(C(Cc2ccn(CC)n2)=O)C1 c1(CC)nc(C(=O)NCc2ccc(CC(C)NC(C3CC3F)=O)cc2)c(C)o1 C1(NC(CN(CCOC)C(c2ocnc2C2CC2)=O)=O)CCCC1C(N)=O Cc1ccc(NC(=O)CC(=O)NCCC(C)(C)NC(c2nc(Cl)sc2C)=O)cc1 N1(C(C(CCC)NC(N)=O)=O)CCC2(CC1)CC(NC(c1cn(C)cn1)=O)CO2 N1(C(C2(C=C)CCN(C(c3csc(CO)n3)=O)C2)=O)CCC(C)OC(C)C1 c1(C(=O)Nc2nc(-c3cc4ccccc4o3)cs2)ccc(Br)c(O)c1Br c1(OC)cnc(C(F)(F)F)cc1C(=O)NCCC(O)CNC(=O)C(C)CF CN1N=C(C(=O)NC2CCC(C)(CNC(=O)CCC=CC(=O)O)C2)CCC1=O CC(O)CC(C)CNC(C1OCCC1NC(=O)Cc1cnnn1C)=O c1(C(C)C(=O)NC2CN(C(C3CC4(CCC4)C3)=O)CC2O)ccc(S(N)(=O)=O)cc1 c1(N(CC(C)CO)C)ncc(S(=O)(=O)NCCC2C=CCC2)cc1Cl CC(CCC(=O)NC(C)CN(C(=O)CC(C)(C)F)C)N(C)C(=O)OC(C)(C)C N1(C(c2cnc(O)o2)=O)CCN(C(=O)CCn2ccnn2)C2CS(=O)(=O)CC12 CC12CC(NC(c3n[nH]cc3Cl)=O)(C1)C1(CN(C(=O)C(O)CN3CCCC3)C1)O2 c1(CC(=O)NC2(CNC(CCCCC#C)=O)CCOCC2)ncnc2sccc12 c1(C(=O)NCC2CC(NC(c3c(OC)n[nH]c3)=O)C2)cccc(S(C)(=O)=O)c1F N1(C(C(C)NC(=O)NC)=O)CC2CN(C(=O)CSc3ncccn3)CC2C1 N1(C(CC(=O)OCC)=O)CC2CCC(C1)C(NC(=O)C(C1CC1)N(C)C)C2 Cc1cc(C(=O)NC(C)(CNC(=O)CC2OCCC2(C)C)C2CC2)c(F)cc1N C1(NC(c2c(C(C)C)n[nH]c2)=O)CC(N(C)C)C1(C)C.C12CC(C1)C(=O)NCC2 c1(C(=O)NCC(CC)NC(C#CC2(CC)CC2)=O)ccc(C)c(Br)c1C N1(C(c2ccc(C)nc2O)=O)CCC2(CCCN2C(c2cc(O)ccn2)=O)C1 C(=O)(C1=CCCC(C)(C)C1)NC(C(C)C)(C)CNC(c1cc(C(C)(F)F)n[nH]1)=O C(=O)(C1CCCc2ncnn21)NC1CN(C(C=C2CCC(C)C2)=O)C(C)C1 C1(C)(C(=O)OC)CCN(C(=O)OCCNC(=O)NC(C)(C)C)CC1.C(CO)O CCCCCC(=O)NCC(=O)NCC1CCCN1C(c1ccccc1NC)=O N1(C(Cn2nc(C)c(Br)c2)=O)CCC2(CCCC2NC(=O)C2=CCC2)C1 c1(CC(=O)NCCCC2(NC(=O)C=C(Cl)Cl)CC2)sc(O)nc1O c1(C(N(C)CC2N(C(CC(C)SC)=O)CCCC2)=O)cnc(O)c(C)c1 c1(CC(N2CCC(NC(C(C(C)C)C#N)=O)C2)=O)cc2ccccc2cc1O C1(CNC(C2(C#C)CC(=O)C2)=O)CC(C(=O)NC2CC(C(N)=O)C2)=NO1 C(=O)(C1COc2ccccc21)NCCCCCCN(C)C(C1CCCCCC1)=O O=S(=O)(c1c[nH]ccc1=NCC1CCCCO1)NC(CO)C1CC1 CCCN(OC)C(=O)C(C1CCCO1)N(C(=O)Cn1ccc(C)c1)CC C=C(C)C1OCCCC1C(=O)NCC1CC(O)CN1C(c1ccc(Cl)c(N)c1)=O c1(OC)ccc(CCC(N2CCCC2C2(NC(C3(O)CCC3)=O)CC2)=O)cc1OC Cc1cc([N+](=O)[O-])c[nH]c1=NCCCN(C)C(C1(O)CC2CCC1C2)=O C1(CC(N2CC=CC(NC(C#CC(C)C)=O)C2)=O)CCOC(C)(C)C1 N1(C(c2c(-c3cnccc3)cc(C(F)(F)F)cc2)C2CC2)CC2CC3CC(C2)CC1C3 CC1CC2CN(C(=O)C(Cc3ccco3)NC(c3ccsc3C#N)=O)CCN2C1 c1(C(=O)NC(C)(C)CCCNC(=O)C2=COCCC2)ccc2ccccc2c1F C1(CNC(C(C)(C)C)=O)CCCC(NC(c2ccc(NS(C)(=O)=O)nc2)=O)C1 C1(O)(CNC(=O)NCCCNC(c2ccco2)=O)CCCNC1 c1(OCCNC(=O)NC2COCC2N2CCCC2)ccc(Cl)c(Cl)c1 C(=O)(C1=CCC(C)CC1)NC1C(NC(CC)=O)COC1 S(=O)(=O)(c1ccc(CBr)cc1)N1C(C(=O)Nc2ccccc2I)CCC1 N1(C(c2cccc(CC)n2)=O)CCN(C(C2CC2c2ccc(C)cc2)=O)C(C)C1 CC(F)(F)C(C(=O)NC1CC1NC(c1c(Cl)cccc1Cl)=O)c1ccccc1 c1(C(N2CC(C)C(NC(=O)CC(C)CN(C)C)C2)=O)cc2cn[nH]c2cn1 CC1CCN2N=C(C(=O)N3CCC(NC(c4cncs4)=O)CC3C)NC2=N1 C1(NC(c2c(C)scc2)=O)C(C)CCN(C(c2cc(N(C)C)ccc2N)=O)C1C N1(C(C2CC(C)C2)=O)CC2(C1)C(NC(c1noc3ccccc13)=O)CCS2(=O)=O C1(CN(C(c2cccc(C)c2)=O)C)CN(C(c2nc(C)nn2C)=O)CC12CC2 C1(NC)CC(C(=O)NOCC(=O)N)C1(C)C.c1(C)ncoc1C C#Cc1ccc(CSc2cn(C3CN(C(=O)C(O)CCCC)CC3C)nn2)c(F)c1Cl CONC(=O)CCCCC(C(=O)O)C1CCCCC1 c1(C(=O)OC)cncc(C(=O)NC2CS(=O)(=O)CC2NC(=O)CNC(C)=O)c1C C1(CNC(c2nc(C(C)=O)sc2)=O)CCCCN(C(C2(C)C=CCCC2)=O)C1 c1(C(=O)NCCC(CNC(CC(=C)C)=O)O)cc(F)cc(Cl)c1N C#CC1(C(=O)NC2CCOCC2)CCN(C(C2CCCO2)=O)C1 C1(NC(c2cc(C)c(Br)o2)=O)CN(C(=O)CNC(=O)C2CC2)CCC1C c1(OC)ccc(F)c(S(=O)(=O)NC(=O)NCC2CCCCN(C)C2)c1F c1(CC(=O)NCCC(C)NC(c2cc(C)[nH]n2)=O)c(F)cc(Br)cc1F C1(C(N(C)CC2CCCN(C(c3nn(C)c(Cl)c3Cl)=O)C2)=O)CC2CC2CC1C N1(C(C(C)c2cccs2)=O)CCC(n2cc(CNC(=O)Sc3nncs3)nn2)C1 Cn1nc2ccccc2c1C(N1CC(NC(=O)C(O)P(C)(C)=O)C2(CCC2)C1)=O CCC(O)C(F)(F)C(=O)N1CC2CC2(NC(C2(c3ccccc3Cl)CCC2)=O)C1 N1(C(Cc2scc(C)c2)=O)CC2CCC(NC(c3cnc(O)n3C)=O)CC2C1 C1(NC(CC(COC)(C)O)=O)CCC2(CC1)CC2NC(c1cc(C)[nH]n1)=O C1(CC)CC(C)CN1c1nnc(C2(CCO)CCCCC2)n1CCC#N C(=O)(CCCC(=O)NC1COCCC1NC(c1ccc(F)s1)=O)OCC c1(C(=O)NC2(CC=C)CN(C(C3CC34CCCC4)=O)C2)noc(C)c1[N+](=O)[O-] Nc1ccc(C(N2CC(O)CC2C(N2CCCC2CC2CC2)=O)=O)nc1 c1(NC(C(CC=C)=C)=O)nc2cc(F)cc(F)c2s1 Cc1cccc(C(=O)C(=O)NCC23CC2CN(C(C2CCC(C)CC2)=O)C3)c1 C1(NC(C2C(C)(C)C2)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C1C1CC1 C1(C(N(CC(C)(C2CC2)NC(=O)OC(C)(C)C)C)=O)Cc2nccnc2C1 C12(C(=O)NCC(CCNC(CCC(C)(F)F)=O)O)CC3CC(C1)CC(O)(C3)C2 c1(CCCC)ccc(OCC(=O)NC2CCCC2NC(=O)CCSC2CC2)cc1 CCC(C)(C)NC(=O)CNC(c1conc1CNC(=O)C(C1CCC1)OCC)=O c1(C(=O)NC2CCN(C(C(CC)O)=O)C23CCC3)[nH]c2ccccc2c1C S(=O)(=O)(c1cc(C(N2CCCCC(C(=O)O)C2)=O)ccc1OC)NC C(=O)(C(C)(O)CC(C)C)N1CC(CCNC(c2ccc(SC)s2)=O)C(C)C1 C(C1CN(C(C2CC=CC(O)C2)=O)CC1C(=O)N(C)OCC(F)(F)F)=CC CC(C)CS(=O)(=O)CCC(=O)N1CCN(C(C2CCC(F)(F)CC2)=O)C(C)C1C c1(C(=O)NCC2CCCCN(C(C(C)NC(CC)=O)=O)C2)cn(C)c(=O)nc1O c1(NS(=O)(=O)c2cccs2)ccc(CCNC(C)=O)cc1Br.C12(OC)CN(C1)C2 C1(CNC(=O)Cc2cc[nH]c2)CC2CCC1N(C(c1ccnc3ncnn13)=O)C2 N1(C(COC2CC(C(=O)OC)C2)=O)CCC(CCC2CCCCC2)CC1 CC1CCN(c2nnc(C(N)=O)s2)C(C)C1CNC(=O)Cc1sc(O)nc1O C1(C(=O)NC2CN(CC)CC2(C)C)CCOC2(CCCCC2)C1 C(C(CC(C)C)NC(c1cn(C)nc1O)=O)NC(C1C(OCC)CC1)=O C(=O)(C(F)(F)C(F)(F)F)N(CCNC(c1cc(-c2nc(C)sc2)nnc1C)=O)CC C1(COC)CN(C(=O)Cc2ccnn2C)CCN1C(c1onc(C)c1C)=O n1(CC(=O)N(C(C)CNC(=O)C(C)n2ccnc2)CC)ncn2cccc2c1=O CC(CC(F)(F)F)C(=O)NCCCNC(c1ccccc1)=O Cc1cc(N(C)C(C2CCC(n3cc(C4(C)COC4)nn3)CC2)=O)ccc1Cl CC12CN(C(c3cc[n+]([O-])cc3)=O)CC1CN(C(C1CCCO1)=O)C2 CC(C)(C)CCCCC(=O)NC1CC(NC(c2cnc3n2CCCC3)=O)C(O)C1 c1(N(CCCCC=C)C)nc(N(C(c2ccc(C)cc2)CC)C)nc2c1COC2 C1(CNC(C=C(CC)CC)=O)CC2(CO1)CN(c1ncc3c(n1)CCC3)C2 S(=O)(=O)(c1ccc(NC(c2nn(C)cc2OC)C)c(Br)c1)NC(CC)C1CC1 C(=O)(CC(C)(C)CC(F)F)N1CCCC(NC(c2cnc(OC)c(Cl)c2)=O)C1 N1(C(C(CCSC)NC(c2cccc(OC)n2)=O)=O)CC2(CCNC2=O)C1 Cc1nn(C)cc1CNC(c1csc(C#N)c1)c1nnnn1CCCF c1(C(N2C(CNC(c3cccc(C)c3O)=O)CCCC2)=O)cnn2cccc2c1 Cc1nccc(C(N2CC(NC(c3n[nH]c(C)c3C)=O)C(F)C2)=O)n1 C12CCN(CC1)C(=O)C(=O)N2.C1(C)(C(N(CC(F)F)CC#C)=O)CCC1 C(CC(C)(C)C)(C(=O)N1CC2C(C(N)=O)C2C1)NC(C1CCC(CC)O1)=O C(=O)(CCC(C)SC)NCCCN(C(C=CC)=O)CC N1(C(c2c(CNC(C3CCN(C)C3)=O)nccc2)=O)CCC2CCC(C1)N2C c1(C(=O)NCCC(C)(C)NC(=O)CCOc2ccccc2O)cccc(F)c1Cl c1(NC(C(CCC)C)c2nnnn2C2CC(F)(F)C2)ccc(C(N)=O)c(F)c1 c1(N2CC(=O)NCCC2)nc2cccnc2c(=NCC2CCc3cccnc32)[nH]1 CCCC(CCC)CC(=O)N1C2CCC1C1CC1(NC(c1sccc1Cl)=O)C2 CC1Cc2cc(C(C(=O)NC3CCCC3)N(C3CCC3OC(F)F)C)ccc2O1 C1(C(=O)NCCC2CN(C(C(C(CC)O)(F)F)=O)C2)CCc2ncccc2C1 c1(C(N(CC)CC2CCCN(C(=O)CC3(CO)CC3)C2)=O)cc(F)c(Cl)cc1F CC(C)C(C)C(C)CC(=O)N(C(C)CNC(c1c[nH]c2ncccc12)=O)C c1(C(C)C)noc(CCC(=O)C(=O)C)n1.C(CCNC(N)=O)NC1CC1 c1(CC(=O)N(CC(CC)NC(c2cc(C(C)C)[nH]n2)=O)C)ccccc1OC C(=O)(C1=C(C)OCC1)NCC(C1N(C(CCC(C)=O)=O)CCC1)(C)C C1(COC)(OC(C)(C)C)CCN(C(=O)NCc2ccc(C#N)o2)CC1 C(CCCCCO)NC(C1(CCNC(Cc2ccc(C)s2)=O)CCC1)=O C1(N(CCNC(C2CC=CCO2)=O)C(C2CCCS2)=O)CCCCCC1 CC1CCNCCC1N(C(=O)CCN(C)CCO)N1CCCC1 N1(C(C2N(C(c3c(C)[nH]cc3)=O)CC(O)C2)=O)CCCC(C)(C#N)C1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1F)N1CC(CC)C(O)C1 c1(C(=O)NCC2N(C(c3scc(C)c3Cl)=O)CCCC2C)cccc2sncc12 C(=O)(C(C(C)CCCC)N1CCN(C(c2ccc(F)cc2)C)CC1)NCCCC N1(CC(=O)NC2CC(c3ccccn3)C2)CCC(n2cccn2)CC1 c1(NC(C2(C)CCCN2Cc2ccc(F)cc2F)=O)cnc(Cl)c(Br)c1 C(=O)(C1CCc2nnc(C)n21)N1CC(F)(CNC(c2c(C)noc2)=O)C1 Cc1cc(-n2ncc(C(N3CC(N(c4cncc(Cl)n4)C)C3)=O)n2)cc(C)c1 C1(NC(C2CCC(C)C2)=O)CC2CCC(C1)N2C(=O)CC(C)C(F)(F)F C(CC(=O)NC(COC)CCOC)(CC(C)C)NC(C(CCC)C#N)=O C1(CN(C2CCN(CCC)C2)C(C2CCC3(CCC3)O2)=O)CCCS(=O)(=O)C1 C1(NC(C(C2CCN(C(C3(C(=O)NC)CCC3)=O)C2)F)=O)CCCN(C)C1=O c1(OC)c(Br)cc(F)c(F)c1NC(C12C=CC(CC1)C2)=O CC1=NOC(C(=O)N(C)CCN(C)C(c2c(-c3cccs3)noc2C)=O)C1C c1(OCC(=O)NCC(C)(C2CC2)NC(c2ccc(C)s2)=O)cc(Cl)ccc1Cl CCC(C)CC(C(=O)N1CC2CCC(CC2)C1)NC(=O)Cc1ccoc1 N1(Cc2cc(CC)c(Cl)cc2)CCc2ccnc(C(=O)O)c2C1 CCC(C)CCC(=O)N1CCCC(NC(=O)CCP(C)(C)=O)CC1 c1(CC(=O)NCC(CN)OC)ccnc(C)c1 C1(CNC(C)C)CC2CCC(C1)N2c1ccc([N+](=O)[O-])cn1.C1C(=O)N1 C1(O)(CN(C(C(C)C2CCCO2)=O)C)CCN(C(C2CC(C3CC3)=NO2)=O)CC1 N1(C(c2c(N)cncn2)=O)CC2CC1CCC2NC(=O)CCCC1CCCO1 N1(C(CN2C(C)CCC2)=O)CC2CC1(C(N1CCC3(CC3)C1)=O)C2 C1(CCC=C)(C(=O)Nc2c[nH]nc2OC)CN(C(=O)C(N2CCOCC2)C)C1 C(=O)(CCCC1(N(C)C)CCC1)N(C1CCN(C(=O)CC(C)NC=O)C1)CCC C12(NC(Cn3c(=N)nc[nH]3)=O)CCC1CN(C(c1sccc1Cl)=O)C2 c1(OC)cccc2c1C(NC(=O)N(C)Cc1csc(C)n1)CC(C)C2 C(CN=C(NCc1c(O)cccc1F)NCC1CCCO1)OCC=C C1(CNC(C2(CCC)CCC2)=O)CC(OC)CN1C(=O)C(C)SC(C)C C1(C(N2CCCC(N(C(=O)C(C)(C)N3CCCC3)C)C2)=O)CN(C)C(=O)CCO1 CC1=NN(C)C(=O)C1CC(=O)NC1CCCC(NC(=O)CN2CC(F)(F)C2)C1 CCC(C)C(C)C(=O)NCC1(C)CCCN1C(c1cc(C)cs1)=O C1(CNC(C(C=CC)O)=O)C2CN(C(C3(NC(C)=O)CCCCC3)=O)CC12 N(C1CCCn2cnnc21)C(CC(CC=C)NC(=O)CN1CC=CC1)=O C=CCC(F)(F)C(=O)N1CCC(CN(C)C(c2c(C)csc2C)=O)CC1 N1(C(C(C2CCCC2)NC(C(COC)(C)C)=O)=O)CCC(C2CCC2)C1 C(=O)(CC(C)O)NCC=CCNC(C(C)NC(=O)NC)=O.C(=O)(N(C)C)NCC c1(NC(CNC(C(C(C)C)NC(C)=O)=O)(C)C(C)C)nc2cccc(C)c2o1 c1(C(N(CCN(C(=O)C(=O)C(C)(C)C)C)C)=O)ccc2nn[nH]c2n1 N1(C(CCOCCOC)=O)CCC2C(NC(c3cc(CC4CC4)on3)=O)C12 C1(C(=O)NCCCCCC#C)CC2CCCC2N1C(c1cncc(OC)c1)=O c1(C(=O)NCC2CCN(C(CC)=O)C2(C)C)cc2nn[nH]c2cc1F C(C)(C)(CC(=O)NCC1CC2C=CC1O2)N(C(c1c(C(C)C)c[nH]c1)=O)C C#CC(CNC(=O)C(C)N(C)C(c1cscn1)=O)CC c1(CC(=O)NC2CC(N(C(c3cc(OC)n(C)n3)=O)C)C2)ccc(O)c(OC)c1 C(=O)(C(C)(C)CNC(C)=O)NC(CC=C)CNC(=O)C=CC1CCCC1 n1(CC(=O)NC(C2CCCN2C(=O)CCF)C)nnnc1C1CC1 c1(C(N(CC(N2CCC(OCc3cnn(CC)c3)C2)=O)CC)=O)nnc(S)n1C N1(C(C(CC)NC)=O)CCn2c(C(=O)NC(c3ccc(F)cc3)CO)cnc2C1 C1(C(=O)NC2(CCCCNC(CC(C)C)=O)CC2)CC2(CCO1)CC2 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CCN1C(=O)CCc1ncc(F)cn1 CCCCC(O)CC(=O)N1CCN(C(c2ccnc(O)c2)=O)CC1CCO N1(C(C2C(C)(C)N(C(C3CC4CC4C3)=O)CC2)=O)CCN2CCC1CC2 CC(CCCC(F)(F)F)(c1nnnn1C1CCC1)NCCCOC(F)(F)F C1(NC(c2c(COC)ccs2)=O)CC(NC(=O)C(C)O)C1(C)C Cc1nc(C(N2CC=CC2CNC(=O)CC(F)(F)F)=O)c(C)n1C C(CCCCCNC(=O)CN1CCCC(N(C)C)C1)NC(C(C)NC(=O)NC)=O C1(CN(C)C(=O)NC(C2C(Cl)(NC(=O)OC(C)(C)C)C2)=O)CC(C(=O)O)C1 CCC(CC(=O)N1CC(N(C)C(c2cncc(C(N)=O)c2)=O)C1)CC(F)(F)F C(CCCCSC(C)C(C)F)N(C(=O)OC)CCO C=CC(C)(O)CC(=O)N(CCCN(C(=O)C(CC)C(=O)OC)C)C C(=O)(CC(P(C)(C)=O)c1ccon1)NC(C)CCNC(C1(CC2CC2)CC1)=O C1(F)(CNC(C2(CCCC)CCC2)=O)CC(CNC(C2CNC(=O)C2)=O)C1 c1(OC)cc(N(C)C)ccc1C(N1CCC(NC(=O)C(F)CC2CC2)C1)=O c1(C(N(C2CCCN(C(CC(C)C(F)F)=O)C2)C)=O)cc2nccnc2cc1F CC1(C)CCC(C(=O)NC2CCC(CNC(=O)CC3CC4C=CC3CC4)C2)CO1 c1(OC)cc(S(=O)(=O)NC(c2ncc(C(F)(F)F)s2)C)sn1 C1(C(N(CCN(C(c2c(Cl)ncc(C)c2)=O)C)C)=O)CCC2CC(C)CN2C1 C1(CN(C(c2c(C(C)C)con2)=O)C)C2CN(C(c3cc(C#N)c[nH]3)=O)CC12 C(C(C)(O)CC(=O)N(C)CC1CN(C(c2c[nH]c(=O)cn2)=O)C1)OC c1(C(N2CC(CC)(NC(=O)C(C)OCC3CC3)C2)=O)cc(C)c(Cl)cc1OCC C(=O)(C1CCCc2c1ncn2C)NC(CN(C(Cc1c(C)cc(Cl)cc1)=O)C)C n1(CC)cc(NC(=O)NCCN(C)S(N)(=O)=O)c(C#N)n1 C12(C(=O)NC3CCN(C(c4c(CC)sc(=N)[nH]4)=O)CC3)CC(C)(CCO1)C2 N1(C(C=CC(C)C)=O)CCCC2CN(C(c3n[nH]cc3C(F)(F)F)=O)CCCC12 c1(C(=O)NC(CC)CNC(=O)CC2CCCCO2)c(-c2cccs2)noc1C Cc1cc(C(=O)N(C)CCN(C(=O)C(c2cccnc2)O)C)ccc1S(C)(=O)=O C1(N=[N+]=[N-])(C(=O)NCC2(C)C(C)CN(C(C=CC(C)(C)SC)=O)C2)CCOCC1 c1(CC)cncc(C(N2CCC(C(C)NC(C3(OC)CC(O)C3)=O)C2)=O)c1 Cc1coc(C)c1C(=O)NCC1C=CCN1C(=O)CC1CCC(C)CO1 C1(CNC(C(C(C)C)NC(=O)CCCN(C)C)=O)CCCC(C)(C)C1 C(=O)(CC(C)C(=O)NC1(CCCCNC(N)=O)CC1)NC(c1ccccc1)C CCCC(C)CC(=O)N(C1CN(C(=O)CC2CC3(CC3)C2)CCC1C)C C(CNC(c1cnncc1C)=O)(CC)(CC)NC(CC1C(CC)C1)=O N1(C(CC(C2CC2)NC(c2nc(C)oc2C)=O)=O)CCN(C)CC(O)C1 N1(C(CNC(=O)OC)=O)CC(O)CCC1C(N1CCC(OCC(F)F)C1)=O c1(OC)cccc(SCCC(=O)NC2CN(C(=O)C(C)=CC3CC3)C2)c1 C(=O)(CCCC(=O)N1CC2CC2(CNC(c2cncc(C(N)=O)c2)=O)C1)NCC c1(CNC(Cn2c(=N)scc2)=O)cccc(CNC(C2CCN(C3CC3)C2)=O)c1 CC1(C(=O)NC2(C(N3CCC(C4CC4)C3)=O)CCCCC2)CC2CCC1C2 C1(C(N(CC(C)(C)NC(CN(C(C(C)C)=O)C)=O)C)=O)CCCN1C c1(CNC(C=C(C)C(F)F)=O)cc2n(n1)CCN(C(=O)C(c1ccccc1)C)C2 N1(C(c2nc(COC)sc2)=O)CC(NC(c2cc(-c3ccco3)c[nH]2)=O)C(C)C1 C1(C(N(C(CC(C)C)C)C)=O)CCCCC1(C)NC(C1CCC1C(N)=O)=O C1(C)(c2n(CC)ncc2)CCN(C(=O)NCc2cccc(O)c2Cl)CC1 c1(NC(C2CCN(C)S2(=O)=O)=O)cccc2c1CCN(C(N)=O)C2 CC(CC#N)C(=O)N1CCC(NC(c2ocnc2C2CC2)=O)C1 C=C(F)C1(CC(N2CCOCC2CC(=O)N(C)CC2CCOC2)=O)CCC1 N1(C(C2CCN(C(CN(C(C(C)C)=O)C)=O)C2)=O)CC2CCN(C)C2C1 N1(c2nc(C(C)=O)c(C)s2)CC2CCCC1C2CNC(c1cncs1)=O C(=O)(CC(O)CCCC)NC(C(=O)NCCCCC(=O)NCC#C)CCCC C1(CNC(C(CC)SC)=O)CCC(NC(=O)Cc2coc(C(F)F)n2)CC1 N1(C(C(C)OCC=C)=O)CCN(C(c2nc(C)ncc2Br)=O)C(CC)C1 N#Cc1cc2c(nc1N1CC3CCCC(NC(=O)C4=NOCC4)C3C1)CCOC2 C1(NC(C2CC(=O)N(O)C2)=O)CCN(C(C2CC23CCOC3)=O)CCC1CO c1(C(N(C2CN(C(c3ccc(C(C)=O)[nH]3)=O)CC2F)C)=O)ccc2nncn2c1 C#Cc1cccc(C(=O)NC(C(=O)NCCCF)c2ccoc2)c1 C1(CNC(C2C(C=C)C2)=O)CN(C(c2cc(Br)c(C)cn2)=O)C2(CCC2)C1 N1(C(C=CC(CC)C)=O)CCCN(C(c2cnn(C(C)(C)C)c2)=O)C(CO)C1 CCC(C)CCC(=O)NC(C1CN(C(c2cnc(SC)[nH]2)=O)CCO1)C C#Cc1ccc(C(=O)N(C)CC2CN(C(C3CC(C#N)(OC)C3)=O)C2)c(F)c1 CC1=C(C)CN(Cc2cn(C3CCC3)nc2C)CC1 c1(C2(C(=O)NC(CC3CCOCC3)CO)CC(C)C2)ccc(F)cc1F N1(C(c2c(C)cno2)=O)CCC(O)(CNC(C2(N3CCSCC3)CCCC2)=O)C1 C1(CN(C)Cc2cnc(C)s2)CCCCN1C(C1CCC1C(C)(C)C)=O c1(CN(C)CC2CCCN(C(c3cncn3C)=O)C2)cc(C(F)(F)F)ncc1Br C12CC(=O)N(C1)CC(=O)NCCNC2=O.C1(CC(=O)NC)CCSCC1.C1CC1 Cc1ccc(C(=O)NC(C)C(C)NC(=O)CC2C=CCC2)cc1C#N c1(CNC(C2CCCCC2NC(c2ccnc(CO)c2)=O)=O)ccncc1CO C12(CNC(=O)CCC3CCCO3)CC(NC(c3ccccc3)=O)(CO1)C2 C1(CNC(C2CCN(C(=O)Cc3ccccc3Br)C2)=O)Cc2ccccc2O1 CCC(Cc1ccccc1)C(=O)N1CCCC1CNC(=O)C(C)(C)CF C(CN=C(NCC(c1cccs1)O)NCc1c[n+]([O-])ccc1Br)OCC C(=O)(C(CNC(=O)OC(C)(C)C)CC(C)C)Nc1c(C)ccc(Br)c1 C1(C(=O)NC(C(C)(C)OC)c2nnnn2C)(CO)CCN(C(=O)CC(C)(F)F)C1 N1(C(c2nc(C3CC3)cs2)=O)CC2CCCC(C1)N(C(=O)Cc1cn[nH]c1)C2 CC1CC(C)(C(=O)NC2CCN(C(c3cc(C(F)F)n(C)n3)=O)C2C)CC(C)O1 c1(SC)ccsc1C(=O)NCCc1cnn(-c2ccccc2)n1 c1(C(N(CCNC(=O)C(CO)N(C)C)CC)=O)cc(C)nc(N2CCCCC2)n1 C1(C)(C(=O)NCCOCCN(C)C(c2cnn(CC(F)F)n2)=O)CC1(F)Cl N1(C(C(CC)C#N)=O)CCC(C)C(CNC(c2cc(C#N)c[nH]2)=O)C1 C1(NC(C2CC(C)(C)N(C(c3cnccn3)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C(C)(F)F)=O)CCC2CC2(NC(C2CN(CP(C)(C)=O)C2)=O)CC1 c1(C(=O)NCCN(C(c2cnc3cccnn23)=O)CC)cc([N+](=O)[O-])oc1C N1(C(c2c(N)cc(F)c([N+](=O)[O-])c2)=O)CCCC(N=c2cc[nH]cc2)CC1 N1(c2nc(C)c(C)s2)CCCC(NC(c2cccnc2OC(C)C)=O)CC1 c1(C(=O)NCC(CNC(=O)CCc2ccc(C)cc2)OC)cc(C)cc(F)c1N C1(NCC2(C(C)C)CCC2)CN2CC(C)C1C2 C=CC1(C(=O)NCc2cnc(F)cc2C)CCN(C(=O)C(C2CC2)OC)CC1 C(CNC(=O)C(C)Oc1ccccc1F)(CC(C)C)NC(C1(COC)CCC1)=O C(=O)(CC1OB(O)c2ccccc21)NCC(CN(C(=O)CC(C)(O)C1CC1)C)O C(=O)(C(C)(C)C(=O)OC)NCc1c(C(=O)NC(C#CC)(C)C)n(C)nn1 N1(C(CC(=C)C)=O)CCC2C(C1)NC(=O)CN2C(=O)C(C)OC1CCCCCC1 C#CC1(C(=O)NCC(C2CC2)N(C(=O)CCc2ncc[nH]2)C)CCC1 n1(CC(C)(C)C)cc(CCC2CN(C(c3cn(CC(F)(F)F)cn3)=O)C2)nn1 N1(C(c2cc(OC)c(O)c(N)c2)=O)CC(NC(=O)C(C)CO)Cc2ccccc21 C1(NC(CCCc2ccc(C)s2)=O)CC2(C1)CN(C(=O)CC(C)(C)C1CC1)C2 c1(C(N(CC(CC)NC(=O)C=C(C)C)C)=O)cc2ccc(OC)nc2[nH]1 c1(C(=O)NCC(CCNC(c2cnn3ccncc23)=O)O)cc2c(nn1)CCC2 n1(CCC)cc(Cl)c(C(=O)NC2CCN(C(=O)C(C)Oc3ccccc3F)C2)n1 c1(CNC(CCC=CC)=O)ccc2c(c1)CCC2NC(=O)C(C)NC(=O)COC N1(C(C2(N(C(C3C4CCCOC34)=O)C3CC3)CCC2)=O)CC2CCOC2C1 C12(C(=O)NCC3CCN(C(COC(CC)C)=O)C3)CC(CCO1)C2 N1(C(C(=O)N(CCNC(C)=O)C(C)C)=O)CCN(C(C2CC2F)=O)CC1C C12(CNC(CCOCC)=O)CCCC1CCN2C(c1cccc(C(N)=O)c1F)=O N1(C(CC(C=C)C)=O)CCC2C(NC(=O)CNC(c3ccoc3C)=O)CC12 Cc1ccc(C(=O)NC2CN(C(C3C4COCC34)=O)CCC2(F)F)c(C)c1Br Cc1nc(CC(=O)NCC(C)CNC(=O)CNC(=O)CN(C)C)cs1 Cc1nn(C)c(C(=O)NCCC2CN(C(c3ccc(NC=O)cc3)=O)C2)c1Cl C(CN=c1[nH]c(=NCc2cnns2)c2sccc2[nH]1)c1n(C)cnn1 N1(C(C(N)Cc2cccnc2F)=O)CC(O)CC2CCCCC12 N1(C(C=CC)=O)CCCCCC(NC(c2cc(C3CC3)oc2C2CC2)=O)C1 N1(C(c2cc(C)nn2C(F)F)=O)CCC2(CC(C(=O)N3CCN(C)CC3CO)=NO2)C1 CC1CC(CNC(=O)C=Cc2cocn2)CN1C(=O)COc1ccccc1Br Cc1nc2cncc(C(=O)NC3COCCN(C(C4CN(C)C4)=O)C3)c2[nH]1 c1(C(N2C(CNC(=O)C3=CCCS3)CC(OC)C2)=O)noc2c1CCCC2 c1(C2(C(=O)NCCCCCCC)CCC2)cccc(C2=CCN(C)C2)c1 CC12CC(C(=O)NC3CC(F)(CNC(C4C5COCC45)=O)C3)(CCO1)C2 CC#CC1CCN(C(=O)CCN(CCO)C(c2c[nH]c(=NC)s2)=O)CC1 c1(C(=O)NCCC2CN(C(CCOC(C)=O)=O)CC2C)[nH]nc2c1COC2(C)C c1(OC)cc(C)c(C)cc1-c1ccnc(CC(=O)Nc2cccc(CF)c2)c1 N1(C(C2(COC)CC2)=O)CCCC(CCC(=O)NCCC2CC(C)(C)CO2)C1 C1(NC(N2CC(N(C(CCCN(c3n[nH]cc3C)C3CC3)=O)C)C2)=O)CCSCC1 Cc1onc(-c2ccncc2)c1C(=O)NCC(C)N(C)C(C1CCCC1(F)F)=O Cc1c(C(=O)NCc2ccoc2C(N2CC(O)CC2C)=O)ncn1C O=C(O)C(O)C(Cc1ccccc1)NC(c1ccc(N2CCC(O)CC2)cc1)=O C1(C(=O)NC(CNC(Cc2c(C)ocn2)=O)(C)C2CC2)Cc2cc(Cl)ccc2O1 N1(C(C(CC)n2cncn2)=O)C2CCC1CN(C(C1CCNC1=O)=O)CC2 C=CC1(C(=O)NCCCC(C)NC(C2C3CN(C)CC23)=O)CCCCC1 CC1(CNC(C23CC(C)(C2)C3)=O)CCCN(C(c2ncc(Cl)cc2F)=O)C1 C#CC1CC2(CC2)CN1C(=O)C(C)(C)NC(C1OCCC1C)=O O(NC(=O)C(C)N(C(=O)COCC(=O)OC)C)CCC1CC(=C)C1 c1(CC)cc(CC)nc(N2CC(CO)(NC(=O)Cc3ccc(F)c(Cl)c3)C2)n1 C1(NC(COCCC)=O)CCC(C)(C)CC1CNC(=O)CCCc1ccccn1 Cc1ccc(NC2(CNC(=O)C(C)(O)C(C)O)CCCC2)c(F)c1 O=C(C#CC1CCCC1)NC1(CNC(c2cccc(C3CCC3)c2)=O)CCOC1 C1(NC(c2cc(F)ccc2Nc2ccccc2)=O)CC2(CCN2)CC1 C1(C(=O)NCCN2CC(CO)C3(CC3)C2)C(C2CC2)CCN1C(=O)C(O)CC(F)(F)F C1(NC(C(C)NC(=O)NC)=O)CCN(C(=O)CC(C)n2cccn2)CC1O CC1C(NC(=O)C(=O)N(C)C)CCCN1C(c1ncc(Br)cn1)=O Cc1cc(CC(=O)NCCCC(C)NC(=O)C(C)Cc2cnn(C)c2)n[nH]1 C(C1=CCN(C2CCc3ccc(F)cc32)CC1)N1C(=O)c2ccccc2C1 N1(C(COCC(=O)OC)=O)CC2(CCCCN(C(=O)CSC(F)F)C2)C1 C1(C(=O)NCC2(C)CCN(C(=O)COC(F)F)CC2)CSc2ccccc2O1 N1(Cc2c(C)cccc2)CCC(F)(F)C(C(=O)Nc2ccnc(F)c2)C1 S(=O)(=O)(c1cc(C)c(Cl)cc1F)NC1C2CN(C(C(C)=O)=O)C(C2)C1 C1(CNC(c2c(CC)occ2)=O)N(C(c2ccc(F)cc2F)=O)CCCC1(C)C CC(C)(C)C(C#N)C(=O)N1CCN(C(C23CC2CNC3=O)=O)C(C2CCCC2)C1 CC(O)(CC(=O)NC1CCC(C(=O)NOCC(O)C(C)(C)C)C1)C1CC1 c1(C(C)C)[nH]nc(C(N2CCSCC2CC(=O)O)=O)c1Br c1(CC)nc(C)c(CNC(C2C(CC)CCN2C(=O)CN(C)CC)=O)o1 C12(CNC(c3ccc(C(C)C)o3)=O)CC(CO1)N(C(=O)CSCCC#N)C2 N1(C(C2N(CC)CC2)=O)CCCCC(NC(=O)COC(C)(C)C)CC1 C(=O)(CCC(=O)C(C)(C)C)NC1CC(CN=c2cc(C)nc[nH]2)(F)C1 C(=O)(C1CCCc2n[nH]cc21)OC1CCN(c2c(C)c(N)ncn2)CC1 c1(COC)noc(COC(=O)C(c2ccc(C)o2)N2CCOCC2)n1 N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)C(F)CC2CCOC2)C(CO)C1 N(C(=NCCc1nccs1)NOC(F)(F)F)C(c1ccccc1-n1cccn1)C CCC(C)(C)CC(=O)N(C(C)C(=O)N(CCCCCO)C)CC C1(NC2(c3n(CC(=C)C)nnn3)CCOCC2)CCc2nnc(C)n2C1 C=CCCCCCC(=O)NC1CC(F)(CNC(c2ccc(C)c(CC)c2)=O)C1 CC1(C(=O)NCC2(NC(=O)CCS(C)(=O)=O)CCOC2)OCCc2ccccc21 N1(C(C2N(C)CCC2)=O)CC(NC(C2CCCOC2)=O)Cc2ccccc21 C=CCC(C)(CNC(c1sccc1CNC(=O)COCC1CCOC1)=O)CO N1(C(C)=O)c2ccccc2CC1C(=O)NCC(C)NC(C1CCC2(CCC2)C1)=O C(CCC(C)C(=O)NCCCCCC(=O)NCCN(C(C)C)C1CC1)OC Cc1cccc(CN2CCC(CC(C)C)(C(=O)O)CC2)c1[N+](=O)[O-] c1(C(=O)NC2(CO)CN(C(C=CC3N(C)CCC3)=O)C2)csc2nccn12 CC1Cn2nccc2CN1C(C1OCCC1NC(C1(C#N)CCCOC1)=O)=O C1(NC(C(C)N(CC)CC)=O)CC12CCC(NC(=O)C(F)(F)C1CCCC1)CC2 C1(C(=O)NCCCC2CCCO2)CCCN(Cc2n[nH]cc2Br)C1 CCC(C)S(=O)(=O)c1cccc(C(N2CCC2CC(N)=O)=O)c1 C1(NC(C=CC)=O)CN(C(c2scc(Br)c2C)=O)CC1C1CC1 CN1CCC(C2CCCN(C(=O)CC3CCCCN3)C2)CC1 O=C(C#CC1CCCCO1)N1CC(N2CC(NC(C3CC(CF)C3)=O)CC2=O)C1 CC(C)C(CCC(=O)NC)NC(=O)C(C)N1CCCC1.C1(C(C)C)CN(C)CCO1 c1(C(=O)NCC(C)=CC(=O)N(C)CC2CN(C)CCO2)cnncc1O N1(C(c2c(C)cc[nH]2)=O)CCC(CCNC(=O)CC2CCCO2)C(F)(F)C1 C1(CC(=O)NCc2cn(C(C)C)nc2)CCC(NC(C2CC(F)C(=O)N2)=O)CC1 CC(O)(CC(=O)NCc1cccc(CNC(C2CCCCO2)=O)c1)C(F)(F)F CC1(CNC(c2cscc2C2CC2)=O)CCCN1C(C1OCC1(C)C)=O C(=O)(C(C)(C)CC(F)(F)F)NCC(C)(C(C)C)NC(C(CO)OC)=O C1(O)(CNC(=O)CCc2cnccn2)CCN(C(c2cc(Br)ccn2)=O)C1 C=CCC(C(=O)NC1(C)CCCC1C)NC(=O)C=Cc1ccncc1 C1(NC(C2CC(C)C2)=O)COCC1CNC(C1CC(n2ccnn2)C1)=O Cc1cc(=NC2CCN(C(c3cc(Cl)on3)=O)CC2C)[nH]cc1C#N c1(C(C)NC(c2n(CC)nnn2)c2csc(Cl)c2)ccc2c(c1)OCCCO2 c1(C(N2C(CNC(=O)CCc3cn[nH]c3)CC2)=O)cc(Cl)c(Br)cn1 N1(C(CCC2N(CC)CCC2)=O)CC=C(CNC(=O)C(O)COC)CC1 c1(OC)ccc(Cl)c(NC(C2CC2C(C)NC(=O)CN2CCN(CC)CC2)=O)c1 C1(NC(c2nc(C)[nH]n2)=O)CN(C(c2ccncc2C)=O)CC12CCOCC2 CC1CN(C(=O)C(c2ccccc2F)O)CC1NC(=O)CCc1cccnc1Cl C1(CNC(CC2C(CC)C2)=O)COCCN1C(C1CC(F)C(=O)N1)=O c1(CC)ccc(C(=O)NCC2CCCCCN2C(=O)CC(O)C(C)C)c(F)c1 C1(N(C(c2c(C)n(C)nc2)=O)C)CN(C(c2cnn(C(C)C)n2)=O)CC12CC2 C1(NC(C(c2cccnc2)OC)=O)CCC(C)(NC(=O)C(F)CC2CCC2)CC1 c1(OC)cc(C(=O)NCCN(C(=O)C(c2ccc(Cl)cc2)OC)C2CC2)n(C)n1 N1(C(C(C2CN(C(C(C=C)OC)=O)C2)OC)=O)CCC(O)CC(C)C1 C(c1c(F)cccc1F)=CC(=O)N(C1CN(C(C23CC(O)C2C3)=O)CC1O)C C1(C(=O)NCc2ccc(OC3CCOCC3)nc2)CCCCN1c1ncccn1 CCCCC(O)CCC(=O)N1CCCCC1CNC(c1ccc(COC)o1)=O Nc1cc(C(N2CC3(C2)CN(C(C2COC2)=O)C3)=O)cc(Cl)n1 C1(C(C)=O)C(C(=O)NC2CC(c3cn(CCF)nn3)C2)C1(C)C c1(C(N(CC(CC)NC(=O)C(c2cccc(C)c2)O)C)=O)cc(=O)cc(Cl)[nH]1 C1(NC(C2C(CCOC)C2)=O)CCN(C(c2cc(C)c[nH]2)=O)C1 Cc1nnc2n[nH]c(NC(C3(F)CCCOC3)=O)c2c1C c1(C(N2C(CCNC(c3csc(F)c3)=O)COCC2)=O)cc2cccn2c(O)n1 c1(CC)cnc(O)c(C(=O)NC(C)CN2CCN(C(=O)C(F)C(C)(F)F)CC2)c1 Cc1ccc(O)c(CNC(=O)C(F)C2CC(NC(c3cccc(CO)c3)=O)C2)n1 C(C(CCCC)NC(C12COCC(C1)C2)=O)NC(C(C)OCCCCCC)=O C1(C(=O)NCC(C2CCN(C(C(C)SCC)=O)CC2)C)(C(F)F)CCOCC1 C1(NC(c2c(C)scn2)=O)CCOC(CNC(=O)CCCc2cccs2)C1 N#Cc1ccc(N)c(C(N2CC=CC2CNC(C2CCCN2CC(F)(F)F)=O)=O)c1 CC1CN(C(=O)C(=O)NC2CCSC(C(F)(F)F)C2)C(C)(C)C1 Cc1cc(CC(=O)NCCNC(=O)C(C)Oc2cccc(Cl)c2)n(C)n1 c1(CC(=O)N(CCC(C)NC(=O)CN(C2CCSC2)C)C)nc([N+](=O)[O-])n[nH]1 N1(C(=O)NC(C(=O)O)C2CC2)CCC(N2CCCCC2)C1 C1(NC(C2CCN(C(CC)=O)C2)=O)CN(C(C2(N=[N+]=[N-])CC2)=O)CC1F Nc1nc(C(=O)NCCC2CN(C(=O)CN3CCCC3)C2)ccc1O c1(CCC)cc(C(=O)NCC2CC2NC(=O)C(CC)N(C)CC)n[nH]1 C1(CC(N2CC(C)N(C(c3cnc[nH]c3=N)=O)CC2)=O)CC2(CCC2)CCO1 c12ccc(c(F)c1)NC(=O)N2.Cc1cn(C)nc1CN1CCOCC1 c1(N(C)C)ccc(C(=O)OCCCC2CCOC2)cc1[N+](=O)[O-] C12(CNC(C3CC(SC)C3)=O)CCCC1N(C(c1cc(C3CC3)ns1)=O)CCC2 CC(O)C(C(=O)NCCC(C)(C)NC(=O)CO)NC(c1cccs1)=O n1(CC(=O)N(CC(CNC(c2cc(C)[nH]n2)=O)C)C)cc(Br)c(O)nc1=O c1(NC(CC=CCNC(C(C2CCC2)OCC)=O)=O)ccccc1O N1(C(CCNS(C)(=O)=O)=O)CCC2(NC(=O)Cn3cccc(N)c3=O)CC2C1 N1(C(c2c(C)snc2)=O)CCC2CCC(NC(c3cc[n+]([O-])cc3)=O)C1C2 C1(CNC(c2ccc(C)s2)=O)CN(C(=O)Cc2nnc(S)n2C)C2COCC2O1 C1(NC(CCNC(=O)NC)=O)CN(C(c2cc(F)cs2)=O)CC1N=[N+]=[N-] c1(C(=O)NC2CN(C(c3ccc(N)c(Cl)n3)=O)C3C2C3)cc2cccn2cn1 Cc1nc2ccc(C(=O)N(CC(C)NC(=O)C(C)(C)c3sccc3Cl)C)cc2s1 Cc1c(C(N2CCCC(CCNC(=O)CC(=O)N(C)C)C2)=O)cccc1CO C1(CC(N2C(C)CCCC2)=O)CCN(C(=O)CCc2nccs2)C1(C)C c1(OC)cncc(C(=O)NC23CC(C2)N(C(=O)CC2CCCCN2C(C)C)C3)n1 c1(C(=O)Nc2cccc(CNC(=O)Cc3ccno3)c2)ccc2c(n1)CCOC2 C1(CCNC(CC)CCCO)CCC2(CCOCC2)CO1 c1(CNS(CCC(CC)CC)(=O)=O)cc(C#N)cc(S(C)(=O)=O)c1 N1(C(C(CC)(C)O)=O)CCC2(CC1)CC2NC(C1(c2cccs2)CCCCC1)=O CC(C(=O)N1CCOCC1)C(=O)OCC1CN(C(C2(COC)CC2(F)F)=O)C1 c1(C(=O)NC2CCC(NC(C=Cc3ccc(C)s3)=O)C2)cccc2ccnn12 C12(NC(c3ccc(OC)cc3)=O)CCCC1N(c1cc(C)cc(C#N)n1)CCC2 C1(CNC(c2cc3occc3s2)=O)CCC2CN(C(=O)CSC(F)(F)F)CCC2C1 N1(C(c2c(C)cc(F)cc2)=O)CCC2(NC(=O)CNC(=O)C(F)(F)F)CCCC12 Cc1nc2ccc(C(=O)NCCC(O)CNC(C3CCC4CC4CC3)=O)cc2s1 Cc1cc(C(=O)NC2CC3(NC(C4CCNC(=O)C4)=O)COC2C3)c(Cl)cc1N c1(-n2cc(C(C)NC(C(C(C)C)SC)=O)nn2)ccnc2ccc(F)cc12 c1(NC(C)=O)ccc2cc(-c3noc(C4(C)CC(O)C4)n3)ccc2c1 C(C(C)C(=O)N1CC(CNC(C2COCCO2)=O)C1)SC C(=O)(CCCC(=O)N1CCC(F)(C(=O)NC2(c3ncccn3)CC2)C1)N(C)C N1(C(CCN(C(c2c(OC)ccs2)=O)C)=O)CC2(C1)CC(C)(F)C2 C(=O)(C1Cc2ccc(C)cc21)N1CCC(O)(CCNC(COC)=O)C1 C(=O)(C(CC(C)C)C(N)=O)N(CCCOCCNC(c1cccc(C)n1)=O)C S(=O)(=O)(c1cccc(Cl)c1)Nc1ccc(NC(COC(C)C)=O)cc1Cl Cc1c(C(=O)NC2CCN(C(=O)C(C)c3ccco3)CC2C)cc(O)cc1N Cc1cc(=O)n(CCC(=O)NC(C(C)NC(c2c(C)ccn2C)=O)C(C)C)cn1 C1(C(N2C(C)CC(NC(c3ccnn3C3CC3(F)F)=O)C2)=O)CC2(CC(=O)N2)C1 C1(CNC(c2ncccc2F)=O)CC(C(F)(F)F)CN1C(=O)C(F)C1CCC1 CN1N=C(C(=O)NC2CC(CCNC(C3CC(=O)N(C4CC4)C3)=O)C2)CCC1=O Cc1cc(C(=O)NC2CCN(C(c3ccnnc3)=O)CC2O)c(C)n1NC(N)=O C1(CNC(CCCC#CC)=O)CC2(CCC2)CN1C(c1ccoc1)=O C(=O)(C(C(C)CC)NC(=O)CC1C=CCC1)OCC Cc1nc2cc(N(C(=O)NCC(N)C3CC3)CC3CC3)ccc2o1 CCC(CC(=O)NCc1ncc(C(=O)NCC(C)C2CCC2)cn1)C1CCC1 c1(C(N2Cc3cccc(C)c3C2)C(=O)NCC=C)n[nH]c2ccc(Br)cc12 N1(C(c2cc(CNC(C(CC)NC(N)=O)=O)oc2)=O)CC2CCC1C(O)C2O CC1NC(=O)OC12CN(C(=O)CC1CC(O)CN1C(=O)Cc1cccnc1Cl)C2 Cc1occc1C(=O)NCC(=O)NC(C)CC1CN(C(c2cscc2CO)=O)C1 N1(C(c2n(C)nc(C)c2Cl)=O)CC2CCCN(C(C3CCC4(CCC4)C3)=O)C2C1 N1(C(CC(O)Cn2ccnn2)=O)CCN(C2CCCCC2)C(=O)C1 N1(C(C2CC(OC)C2)=O)CCCC(C(C)C(=O)NCCC2(C)N=N2)C1 c1(NCC(c2ccc(F)cc2Br)C)cccc(S(=O)(=O)N=c2cc[nH]cc2)c1 c1(OC)c(C(N2CCC(O)(CCNC(C3CC4C=CC3O4)=O)C2)=O)ncnc1C c1(OC)nn(C)cc1C(N1CCC(O)C1C(=O)NC1(C)CCC(C)C1)=O C1(NC(CC(C(N)=O)NC(C)=O)=O)CC2CCC1N(C(=O)CC(O)C(C)C)C2 N1(C(C2CC3CC3N2C(=O)Cc2ccnc(Br)c2)=O)CCC(O)C(F)C1 CCCC(CCC)CC(=O)N1CCCC1(C(=O)NCC1CNC(=O)C1)CC CCCC(O)(CCC)CC(=O)NC1C=CCN(C(C2(c3cc(C)no3)CC2)=O)C1 N1(Cc2c(CC)cccc2)C2CCC1CC(NC(C1Cc3ccncc3C1)=O)C2 N1(C(CSC)=O)CCOCC(C)(CNC(C2(C3CCCO3)CCC2)=O)C1 c1(C(=O)NCC(C)CN(C(=O)CN(C2CCC2)C)C)cc(F)cnc1Cl c1(C(=O)NCC(CC)NC(c2snnc2C(C)C)=O)ccc(C)s1 c1(C(C)(C)C#N)ccc(C(N2CC(CCNC(=O)CC3CC=CC3)C2)=O)cc1 C1(COC)CN(C2CC2)CCN1S(C)(=O)=O.c12ccccc1sc(=O)[nH]2 c1(OCCC)ccc(CN2CCC(CC(N3CCN(CC(C)C)CC3)=O)C2)cc1 N1(C(c2cn(C(C)C)nc2)=O)CC(CNC(c2cn(C)cn2)=O)C(F)(F)C1 C(=O)(C(C)CSc1ccccc1)NCC(CNC(CN(CC)CC)=O)O c1(CN2CCC(NC(Cc3c(C#N)cccc3)=O)C2)cnc2ccccc2c1Cl C(=O)(CC(C)C(C)(C)C)NC1C2CN(C(c3c(OCC)nccc3)=O)CC1C2 Cc1cnc(C(=O)NCC(C)(C)C(=O)N2CC(N3CCCCC3)C2)c(C)c1 O=C1CCC(C(=O)NC2CCC(NC(c3cc(Cl)c[nH]3)=O)C2)CCO1 N1(C(c2c(C)csc2C)=O)CCN(C(=O)C(c2cnn(C)c2)O)C2(CC2)C1 C1(CNC(C(C)OC(C)=O)=O)CCCN(C(=O)C(c2ccncc2C)C)C1 c1(C(N(C)CC2N(C(c3scc(C)c3)=O)CCC2)=O)cc2sccc2n1C C(=O)(C(C)C(C)COC)NC(CCC)C(=O)N1CC(OCC(N)=O)C1 C(CC(C)(C)C(=O)NC(c1ccsc1)C)NC(CC(C)CN(C)C)=O C1(C)(OC)CCN(C(C2(COC)C=CCN2C(c2coc(C)n2)=O)=O)C1 c1(OC)cn(C)c(C(N2CC(NC(=O)Cc3cnc[nH]3)C3(CC3)C2)=O)cc1=O CCCC(CNC(c1ccc(CC)o1)=O)C(=O)NC(c1ccccn1)C c1(C(=O)NC2CN(C(c3noc(CC)c3C)=O)CC2C)cnc(C)c(N)c1 C1(C(N2C(C)CN(C(=O)CC3(N(C)C)COC3)CC2)=O)CCc2nncn2CC1 C(C(C)(C)C(c1ccc(C)o1)NC(c1ccc(C(=O)OC)o1)c1nnnn1C)OC Cc1ccc2c(c1)CCC2(C)NC(=O)Nc1ccc(C2CC2)cc1 CCC(CCC(=O)OC)NC(=O)C(N)CN1CCCCC1 Cc1nc(C(N2CCC(SC(C)C)CC2)=O)sc1C.C1C(=O)NCCN1C CCC(C)CC(=O)NC1CCC(NC(=O)Cc2sc(C3CCC3)nc2C)C1 N1(C(C(=O)NC2CC(n3ccnc3)C2)=O)CCC(=Cc2cccnc2)CC1 CCCCCCCCCCC(=O)NC1CC(NC(=O)CC(=O)OCCCCC)C1 c1(C(=O)NCC(CN(C(COCCOC)=O)C)(C)C)cc(N)cc(OC)c1OC c1(NC(COC(C2C(CC(C)C)OCCC2)=O)=O)ccc(O)cc1F Cc1cc(F)c(CN2CCN(c3cc(N4CCCCC4)ncn3)CC2)c(F)c1 c1(C(N(C2CN(C(C3(C)CC(C)=C(C)CC3)=O)C2)C)=O)cc2c(=O)[nH]ccn2c1 C1(C(=O)NCC2(CC=C)CN(C(=O)CC3CCCOC3)C2)(OC)CCCOC1 C1(CNC(C2C(C=C)C2)=O)CCN(C(=O)C2=CCCCC2)C1(C)C c1(CC(N2CC(CNC(C(CO)OC)=O)C(N(C)C)C2)=O)cc(C)ccc1C CC1CN(C(=O)C(=Cc2cscn2)F)CC1CCNC(C1(NC(N)=O)CC1)=O c1(C(=O)NCC(CN(C)C(C2CC(n3cnnc3)C2)=O)O)ccc(N)cc1Cl c1(C(c2nnnn2Cc2ccco2)NCC2(SC)CC2)cc2ccccc2o1 C(=O)(CCCCc1cnn[nH]1)N1CCC(NC(c2cc(OC)n[nH]2)=O)C1 c1(C(=O)NC(CNC(CC2C(C)(C)COC2)=O)C2CC2)cc(F)cc(Br)c1 N1(C(c2c[nH]nc2C)C(=O)NCCOC)CCc2c(ccc(F)c2F)C1 C1(NC(C2CCN(CC)C2)=O)CN(C(c2cn(CC)nn2)=O)CC1F C(N=c1cc(Cl)nc[nH]1)C1CN(C(Cc2ncc(CC)[nH]2)=O)C(C)C1 N1(C(c2cn(CC=C)nn2)=O)CCCCC1CCN(C(=O)CN(C)S(N)(=O)=O)C C1(CC(=O)NCC(CCOC)NC(C2(C#N)CC2)=O)CCN(C(C)=O)CC1 c1(C(N2CC(CNC(c3c(C)occ3)=O)C(F)(F)C2)=O)cc([N+](=O)[O-])cnc1N c1(CNC2CN(C(c3cccc(C)c3)=O)CC23CC3)c[nH]c2ncccc12 C1(CC)C(C(=O)N(CC(C)(C)NC(=O)C=CBr)C)CCN1C CC1CN(C(=O)CCc2cccnc2)CC1C(N1CCOC(C2(C)CC2)C1)=O C1(NC(CCCOCC=C)=O)(COC)CCN(C(=O)C(C)(C)SC(F)(F)F)C1 Cc1csc(C(N2CCN(C(=O)CCC3CC3(F)F)CC2)=O)c1Br c1(C(N(C2CCC(CNC(=O)OC(C)(C)C)C2)C)=O)cnc(Cl)s1.C1(=O)CN1 c1(C(=O)NCC2C(C)(C)N(C(C3CCCC(F)C3)=O)CC2)cn2ccccc2n1 Cc1ccc(C(=O)OC(C2CCOC2)C#N)cc1Br c1(C(=O)NC2(C)CC(NC(C3CCCS3(=O)=O)=O)C2)cccc2c1OCCC2 C1(COC)(NC(c2cccnc2)CC2CCOC2)CCCCC1 CC(C)(C)CCCCNC(=O)C(F)CC1CN(C(c2cscc2Cl)=O)C1 CN1CCN(C(C2CC3CCCCC23)=O)C(CNC(C2(C)CCSCC2)=O)C1 c1(C(=O)NCC(CN(C(=O)C(C)N(C)C)CC)(C)C)cn2c(n1)SCC2 c1(NC(C2N(C(CC(C)O)=O)C3C(C2)C3)=O)cc(O)nc(Cl)n1 Cc1c(NC(=O)Cc2csc(NC(=O)CNc3cccnc3)n2)cccc1Cl N1(C(c2cnn(C)c2F)=O)CC2CCCN(C(c3cn(C4CC4)nn3)=O)C2C1 N1(C(C(C)NC(C=C)=O)=O)CCC2(CC1)CCN(C(c1cnco1)=O)CC2 C(CCC(C)C)(C(=O)NC1(C)CCC(C)(C)C1)NC(c1c(OC)cc(C)cn1)=O c1(C(N2C(CNC(CN(C)C(N)=O)=O)CCC2)=O)cc(F)c(F)cc1C(F)(F)F C1(CNC(C2CCN2C(=O)CCc2cccnc2Cl)=O)OCCOC12CCC2 N1(C(CC=CC)=O)CC23CCCC2(C1)CN(C(=O)C(=O)N=S(C)(C)=O)C3 C1(O)(CNC(c2cncnc2C2CC2)=O)CCN(C(c2coc(O)n2)=O)C1 N1(C(CNC(C=C)=O)=O)CCOC2(CCN(C(c3ccccc3N(C)C)=O)C2)C1 C=CC1CN(C(=O)C(n2nc(C)cc2C)C)CC1NC(=O)CN(C)CCC C1(N(C(=O)CCC=CC)CC#C)CCN(C(=O)C(O)C2CCCC2)CC1 c1(CC)cc(NC(C2CC(CNC(C3(F)CCOC3)=O)C2)=O)ccc1C C1(C)(C(=O)NCC2N(C(c3c(CC)scc3)=O)CCC2)CC2CCC1C2 N1(CC(=O)N(CC(C)NC(c2ccncn2)=O)CC)CCCNS1(=O)=O C1(CC(N2CCOC(CC3CC3)C2)=O)(NC(C(CN(C)C)O)=O)CCCCC1 c1(C(=O)NCC2C(NC(CCC(=C)C)=O)CC2)ccc(N)c(Cl)n1 S(=O)(=O)(c1cccc2cnc(Cl)cc12)NCC(C)Cc1ccc(F)c(F)c1 c1(C(N2CC(O)(C(C)NC(C(F)=C(C)C)=O)C2)=O)cc(C)c(C#N)c(C)c1 C1(NC(c2cc(CC)no2)=O)CCC(CNC(=O)C(C)(C)c2cc[nH]n2)CC1 C1(CCC)CN(C(=O)Cn2ncccc2=O)CC1NC(=O)C(C)(C)OC(C)C CC#CCCCC(=O)N(C)CC1CCCN1C(=O)CCCCCOCC C1(F)(C(=O)NCC2CC(NC(C(C(C)(C)C)SC)=O)C2)CCC(F)(F)CC1 CCCCCC(CC)C(=O)N(CC(CC)NC(c1csc2ccncc12)=O)CC C(=O)(C(CNC(C12CCCN1CCC2)=O)CC(C)C)NC(C(=O)NCC)C S(=O)(=O)(c1cccnc1Cl)NC1CCC(C(=O)NC(C(C)(C)O)C2CC2)CC1 C(C(O)C(=O)NCCOC1CCN(C(=O)Cc2ccn(C(F)F)n2)C1)=CC N1(C(C=C(C)C(C)C)=O)CCCCC1C1CN(C(c2cc(Cl)n(C)n2)=O)C1 C(=O)(C(F)CCCCC)NCC1C(C(=O)NC2(C=C)CCOCC2)CC1 CCC(CC(=O)N(C1CCCC1)CCCNC(C1CC=C(C)CC1)=O)CC(C)C C1(C(=O)NCC(=O)NCC(C)NC(c2n[nH]c(C(C)(C)C)n2)=O)CCOCC1 C1(NC(c2cnc(O)nc2O)=O)CC2CC1N(C(c1ccc(F)c(Cl)c1)=O)C2 N1(C(c2c(CNC(C3(C)CC(C)C3)=O)c[nH]n2)=O)CC2CC(C1)N(C)C2 Cc1nc(C(N2CC(CNC(=O)CSC(F)(F)F)C3CC23)=O)cc(O)n1 c1(CC)nnc(NC2(CNC(=O)C(F)CC3CC3)CC2)nc1CC N1(C(C(c2ccccc2)NC(C)=O)=O)CCC2(C1)CN(C(c1nn[nH]c1Cl)=O)C2 C1(NC(C2N(C(C(C(CC)C)O)=O)CCC2)=O)CCn2nnnc2C1 C12(CNC(C(N3CCC(C(C)C)C3)=O)=O)CCOCC1C2 c1(C(=O)NCC2C(NC(CC(CC)SC)=O)C2)c(C)ccc([N+](=O)[O-])c1C c1(C(=O)NC2(CC=C)CN(C(=O)C(C)C(C)O)C2)cc(Cl)nc(Cl)c1 C1(NC(C2(C)CC2Br)=O)CC1C1CCCN(C(=O)COC2CCCC2)C1 C(=O)(C(C)C(O)C(C)C)N1CC(C(C)NC(c2c(C)ccc(CC)c2)=O)C1 CCC(O)(CN(C)C(C1CC2CC2N1C(=O)COCc1nc[nH]n1)=O)CC C1(C(C(=O)NC2(CSC)CC2)C)CN(C(=O)CC(C)(C)C)CCO1 C1(C(N2C(CNC(C3CSCCS3)=O)CC(F)C2)=O)Cc2ccccc2N1 C1(CNC(=O)OC(C)(C)C)CC2(C1)CN(N1CCCC3(C1)N(C)C3)C2 C1(C(=O)NC2CN(C(C3CCCN(CC)C3)=O)CC2C)CCC(=O)N(C(C)C)C1 Cc1cccc(C(=O)NCc2ccoc2C(=O)NCC=C(Cl)Cl)c1O C(C(=O)N1CCN(C(C)CNC(C2(F)CC=CC2)=O)CC1)(C(C)C)OC C=CC(CCC)CC(=O)NC1(C)CC(NC(=O)CSc2nc3ccccc3s2)C1 c1(CC)nccnc1C(N1CCN(CC(=O)NCC2CCC(=O)O2)CC1)=O C1(C(=O)NC(CN(C(CCSC)=O)C)C)CCCCC(=O)N1 C(CC(C)(C)CO)NC(N(C)CC1CC1)=O C1(C(=O)NC(C2CC(NC(c3cc(OC)no3)=O)C2)C)CCCSC1C c1(C(c2n(CC)nnn2)NC(C)CCCOC)ccc([N+](=O)[O-])c(C)c1 C(=O)(C(CC)CC(C)C)NCCC1CCN(CC(c2ccccc2)OC)CC1 Cc1ncc(C#N)cc1NC(C1CCCN1C(=O)CNCc1ccc(O)cc1Cl)=O C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)CSCC(N)=O)C(C)C1 N1(C(CCc2ccc(OC)c(OC)c2)=O)CCC2(CC1)CC2C(=O)NCCN C(=O)(C(C)S(N)(=O)=O)N(CCNC(c1nc(C)c(C)s1)=O)C C1(CCNC(c2cnc(O)o2)=O)(C(=O)NCc2ccn(C3CCC3)n2)CCCC1 CCCCC(C)CCC(=O)NC1CCC1CNC(=O)CCCCCC#N C1(NC(CC=CC)=O)CC2CN(C(C3(c4ccc(N(C)C)cc4)CC3)=O)CC2C1 C=C(C)CC(C(=O)N(CCNC(C1CC1C(C)(F)F)=O)CCOCCO)OC c1(CC)ccc(C(=O)NC2CC2CNC(=O)Cn2nnc(=O)[nH]2)c(C)n1 N1(S(c2ccc(C)c3c2nsn3)(=O)=O)CCC2(CC1)COC(C)(C)OC2 CCCC(CNC(=O)CCc1cnco1)C(=O)NC1C2CCCCCC12 C1(C(=O)NCc2c(C(=O)NC(c3onc(C)n3)CO)[nH]cc2)C=CC=CC=C1 C(=O)(C#CC1CC1)NC(CC=C)CNC(C1CC1(c1ccc(F)cc1)C)=O C#CCCCCC(=O)N1CCC(NC(=O)Cc2ccccc2)C(C)C1 c1(C(=O)NC2C(CNC(C3CCC(=O)O3)=O)CC2)ccc2occc2n1 C1(N(C(=O)C(O)Cn2cncn2)C)CCC(NC(=O)C=Cc2nccs2)CC1 C(=O)(CCC(C)CC)N(C1CCCCC1)CCNC(CCC=C)=O O(N=C1CCCCCC1)CC.C1(=O)C(=O)N(CC)CCN1.C(=O)C1CC1 C1(NC(c2nc(OC)oc2)=O)CC(F)CN(C(=O)CC2CCCC(=O)N2)C1 C(=O)(C(C)(CC)NC(C)(C)C)N(CCCNC(=O)NC1C(C(=O)OC)CC1)C c1(C(N2CCC(COC)CC2)C(=O)Nc2ccccc2C)ccc2c(n1)CCC2 c1(OC)cccc(CNC(=O)NCCCN2CCCC2CO)c1 C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC1CCN(C(CSCC(=O)OC)=O)CC1O N1(C(c2ccc(C(C)=O)cc2F)=O)CC2(C1)SCCC2NC(=O)CCF c1(C(=O)NCC(C)CN(C)C(c2cn(C)nn2)=O)nn(C)c2c1CC(C)(C)CC2 C1(C2CCCO2)(C(N2CCC(C)(CNC(c3cnc(C)s3)=O)C2)=O)CCCO1 c1(C2N(C(=O)CC(C(F)(F)F)n3cccn3)CCC2)ncc2c(n1)CCNC2 C=CC1(C(=O)NCC(O)CCNC(=O)Cc2csc(COC)n2)CCOCC1 N1(C(C2CC(N(C)C)C2)=O)CCCCC(CNC(c2cc(C3CC3)on2)=O)C1 C=C=CCC(=O)NCC(C)NC(C1CC2(CC2)C1)=O C1(CNC(C2(CSC)CCC2)=O)CCN(C(C2CSC2)=O)CC1(F)F C1(NCCCNC(N2CCOC(C3(O)CC3)C2)=O)CCC(F)(F)CC1 C(=O)(C(F)C(=O)NCC12CC(NC(c3ccc(O)nc3)=O)(CO1)C2)OCC C(=O)(CC(C)(C)C(F)(F)F)NC1CCCC(CNC(C2(C(C)C)COC2)=O)C1 C(=O)(C1c2c[nH]nc2CCC1C)N1CCC(NC(c2c(C)ccc(Cl)c2)=O)C1C C12(C(=O)NC(C(C)NC(=O)C(C)(C)c3ccn(C)n3)CO)CCCN1CCC2 c1(N2CCC(OCC)(CO)CC2)nc(N2CCC3(C=CC3)CC2)c2c(n1)CCS2 CCC(CCC(=O)NC1N(C(=O)CCCN2CCOCC2)CCC1(C)C)OC C(CCC(O)C(=O)NCc1cnn(CCO)c1)NC(=O)CCCF CCCCCC(O)CC(=O)N(CCNC(c1cn2c(n1)CCC(C)C2)=O)C1CC1 c1(C(=O)NC(CC=C)CNC(=O)C(C)n2cccn2)cc2sc(C)nc2[nH]1 O=C(N=c1ccn(-c2ccc(F)cn2)[nH]1)N1CCOC(Cc2ccc(F)cc2F)C1 CCCC(CCC)CC(=O)NC(C)CN(C(=O)C=CC1CCCCC1)CC Cc1cc(Cl)cc(C)c1OCC(=O)NC1(CNC(=O)Cc2sc(S)nc2C)CC1 C1(CCC)(NC(=O)CCn2ccnn2)CCCN(C(c2cc(C)c(C)o2)=O)C1 C1(NC(C(C=CC)O)=O)CCN(C(=O)CCc2ccccc2F)CC(C)(C)C1 N1(C(C(N2Cc3ccccc3C2=O)C)=O)CCCc2c1ccc(Br)c2C c1(CC)ccc(C(C)=CC(=O)N(CC(O)CNC(=O)C=Cc2cncs2)C)cc1 O=C(C1=CSCCO1)N(C1CC1)CC1CCCN1C(=O)CCCc1cccnc1 N1(C(c2c(NC)ccc(Cl)c2)=O)CC2CC(CNC(C34CC(CO3)C4)=O)CC1C2 c1(NC(C2OCCN(Cc3c(OC)cccc3)C2)=O)ccc2ncnn2c1 N1(C(C2(CC(C)C)CC2)=O)CC2CC(C(=O)NCC3CCOC3)C(C2)C1 c1(C(N2CCC(CC=C)C2)C(=O)NCCCC)ccc(Cl)cc1Cl C1(C(=O)NC(CCCC)C)(CC)CCCN(C(=O)CCOCC(C)(C)C)C1 c1(OC)ccc(-c2nccn2-c2cnccc2C(=O)OC)cc1-c1ccno1 c1(C(=O)NCC(C)CN(C(=O)CC2C=CS(=O)(=O)C2)C)cncc(CCN(C)C)c1 c1(C(N(C(C)CNC(c2cc(Cl)cs2)=O)C)=O)ccc2c(c1)CCN(C)C2 N1(C(=O)NCC2CCC(OC)C2)CCC(O)(c2ccccc2C)CC1 CC(C)(C)C(C)(O)C(=O)NCCCOCCNC(c1ccccc1[N+](=O)[O-])=O C(C1CCCC1)=C(C)C(=O)N(CCCN(C)C(c1cc(-c2ccco2)cs1)=O)C C1(CNC(C2C(C)CCC2)=O)CC2(CO1)CN(C(=O)Cc1ccc(C#N)nc1)C2 c1(C(N2CCC(CNC(C3(CO)CCC3)=O)C2)=O)csc2cccnc12 C=C1CCN(C(=O)C(C)=C(C)C)C(C(=O)NCCC2CCCCCC2)C1 C1(NC(CC2C(OCC)COCC2)=O)CCCN(C(=O)Cn2cc(C)cn2)CC1 O(NC(=O)COC(F)F)CC(=O)N(C(CC)C)C Cc1cc(C)c(C(=O)NCCCOCCCNC(C2CN(C)C2)=O)c(C)n1 c1(C(=O)NC(CN(C(c2csc(S)n2)=O)CC)C)cc(Cl)ccc1C(F)F c1(C(=O)NC2(CC)CCCN(C(C(CC)C(C)C)=O)C2)c[nH]c2cccc(Cl)c12 c1(CCCC(=O)N(CC(C)(C)CNC(C2CC=CC2)=O)C)cccc(C(F)(F)F)c1 C1(C(=O)NC2(CC=C)CCN(C(=O)COCCOC)C2)CC2(CC(N)C2)C1 N1(C(CNC(C)=O)=O)CC2CC2C1C(=O)NC(C(C)(C)O)C1CC1 C1(C(=O)Nc2cn(C)nc2)CN(C(=O)Cc2ccccc2C#N)CCC1O N1(C(Cc2cccc(C)c2Cl)=O)CCCC2(NC(c3cccc(Cl)n3)=O)CC2C1 CCC(CC)(C(=O)NC1CN(C(c2[nH]c(O)nc2C)=O)CCC1C)OC c1(-c2c(OC)ccs2)nc(Cn2cc(Br)cn2)nn1CCc1cnn(C)c1 N1(C(C(COC)OC)=O)CC(C(=O)NCCCCCC2CC2)C(F)(F)C1 CCC(C)(C)C(O)C(=O)NC(C)CCNC(=O)CCC(=O)N(C)C(C)C Cc1ncnc(C)c1CC(=O)NC(C1CCCC1)CNC(=O)C=Cc1ncc[nH]1 c1(C(N(CC(C)NC(C2(F)CCCCC2)=O)CC)=O)ccc2[nH]c(C)c(C)c2c1 c1(OC)cc(N2C(C(N3CC(C)(O)C3)=O)CCC2C)ncn1 c1(C(N2CCC(CNC(c3c(C)ncnc3)=O)C2)=O)ncncc1C#N N1(C(C2N(C(c3ccc(C)c(O)n3)=O)CC=C2)=O)CCn2c(O)nnc2C1 c1(C(CC(=O)NCC(C(C)C)NC(c2cn(CC)nn2)=O)C)ccc(F)c(F)c1 N1(C(C2CN3CCC2CC3)=O)CC2CCCC2(NC(C2(C3CCCO3)CC2)=O)C1 C1(NC(c2cccnc2O)=O)CC2CCC(C1F)N2C(c1coc(Br)n1)=O CC1CCCC1CCN1CCC(CC(=O)N(C)CCc2ncon2)C1 C1(C(=O)NC2CCC2NC(c2cc(Cl)ccn2)=O)(OC)CS(=O)(=O)C1 Cc1ccc(CC(=O)NCC2CCCOC2(C)C)cc1Cl N1(C(c2c(C)n[nH]c2)=O)CCC2(CC(CC(=O)N3CCNC(C)C3)=NO2)C1 C1(C(N(CC)CC2CCCN2C(c2ncoc2C)=O)=O)CC(C)(C)CO1 c1(NC(=O)CC2CCC(NCc3cc(Cl)cc(Cl)c3)CC2)nc(Cl)c(Cl)cc1Cl Cc1cc(C(=O)NC2CCN(C(=O)C3=NOC(C)C3)CC2O)cc(F)c1 C12(C(=O)Nc3nc(CC)nc(C)c3)C3C4C1C1C2C3C41C(=O)N(CCN)CC C1(=CC(=O)NCCn2cc(C(CC(C)C)O)nn2)CN2CCC1CC2 N1(C(CCSCC)=O)CC2CC(NC(c3ccc(N(C)CC)cc3)=O)C2C1 C1(c2n(C)ccn2)CN(C(C2(C)CCCOC2)=O)CC1NC(=O)C(Cl)=CCl CC1CN(C(=O)CCC(=O)c2cccc(F)c2)CC1NC(C1CCNC(=O)C1)=O C(=O)(C(C)(C)CC(F)(F)F)NCC(CN(C(=O)C(c1cccn1C)=O)C)O C#CCCN=C(NCC(c1ccc(C)cc1)CC1CC1)N1CCC(NC(C)=O)C1 N1(C(C2N(C(C(CC(=C)C)OC)=O)CC2)=O)CC2CCCC(C1)N2C C1(NC(C(COC)O)=O)CCN(c2ncc3c(n2)CCCC3)CC(C)(C)C1 C1(CN(C)C(c2ccccc2NC(=O)OC(C)(C)C)=O)CCC=CCCC1 N1(C(c2ccn(C)c2)=O)CCC(NC(C2CCCO2)=O)C12CCCC2 C(=O)(CC(C)(O)C(F)(F)F)NCCN(C(c1c(C)cccc1Cl)=O)CC1CC1 C=CC(CCC)CC(=O)NCC1CN(C(c2ncoc2C)=O)CC(C)(C)C1 CCCCCCC(O)CCC(=O)NCC(C(C)C)NC(c1ccn(CC)c1C)=O C(=O)(C1=CCC(C(F)(F)F)OC1)NCCCC(C)(C)NC(=O)CC1CC2CC2C1 C1(NC(CCC)=O)CCC2CN(C(c3cn(CC)nc3C(C)C)=O)CCC2C1 C1(C(=O)NC2(CNC(=O)CC3COC(=O)N3)CCCC2)CCC(CO)CC1 C1(C(N2C(C(C)NC(=O)C3=COCC3)CCC2)=O)CCC(C2CC2)CC1 C1(CCNC(C(=O)NC(C)C)=O)CCCN(C(=O)CCN2CCC(F)C2)C1 C1(OCCOCC(=O)NCCCOC2CCOC2)CCN(C(=O)C(Cl)=CCl)CC1 N1(C(c2nc(C)oc2C)=O)CCC2(CC1)CCN(C(=O)COc1ccccn1)C2 N1(C(C(CC)F)=O)CCCC(N(C(=O)COCC(=O)NC)CC)C1 C=CCN=c1[nH]cc(C(N2CCCC2C2CCN(C(=O)C(O)C(C)CC)C2)=O)s1 C(CN=c1nc2n([nH]1)CC(N1CCN(c3cc(C)[nH]n3)CC1)CC2)OC C1(COC)(NC(c2[nH]nnc2C)=O)CCN(C(c2cc[nH]c2)=O)CC1 N1(C(c2c(O)ccc(OC)c2)=O)CC2OCCN(C(C3CC=CCO3)=O)C2C1 N1(C(c2n(CC)ccc2)=O)CCC(CNC(c2cc(C(C)C)n(C)n2)=O)C1(C)C N1(C(c2n(CC)ccc2)=O)CCCC(N(C)C(c2sc(C(C)C)nc2C)=O)C1 N1(C(COCCCCC)=O)CCC(NC(C2CC(O)(c3ccncc3)C2)=O)C1 Nc1cc(Cl)cc(Cl)c1C(N1CC(CNC(=O)Cc2cc(C3CC3)n[nH]2)C1)=O Cc1c(C(=O)NC2CN(C(C3CCCN3C3CC3)=O)CC2O)sc2ccccc12 C(=O)(CCCC(C)CC)NC(CC#C)CC(=O)N1CCCN(C)CC1 c1(C(=O)NCCCC2N(C(CN3CCC(C)C3)=O)CCC2)cc(=O)cc[nH]1 Cc1ccc(C(N2CCOCC(CNC(C3CCCC(C)(C)C3)=O)C2)=O)c(C)c1 c1(N2CCC(C)(NC(c3c(C)cccc3)=O)C2)cc(C(C)C)nc2ncnn12 C(F)(C(=O)Nn1cccn1)C12C(CN(C(=O)CCC3CCOCC3)C1)CC2 N1(C(C(c2c(C)cccc2Br)NC(C(C=C)CC)=O)=O)CCOCCC1C c1(NC(C2(COC)C=CCN2C(=O)C(O)C(F)(F)F)=O)cnc(C)c(C)c1 C1(C(=O)NC2CCC(CNC(C3(CO)CCCO3)=O)C2)(OCC)CCCCCC1 c1(OCC)noc(C(=O)NC(C)C(C)n2cncn2)c1Br S(=O)(=O)(c1cccc(C)n1)N1CCC(NC(c2ccc(OC)c(Cl)c2)=O)C1 C1(C(=O)NCC2(C(F)F)CCN(C(C3CC(O)C3)=O)C2)OCC2COCCC12 C1(N(CC#C)C(C2CCCC2C)=O)CCN(C(c2ccc(Cl)o2)=O)CC1 C1(CNC(C2(S(C)(=O)=O)CC2)=O)CCCCN(C(=O)CC2(O)CCCCC2)CC1 c1(C(N2CCCCC(CNC(CC3C(C)(C)C3)=O)C2)=O)c(F)ccc(N)c1F c1(NC2CC(F)(CNC(CCCN(CCC)CCC)=O)C2)ncc([N+](=O)[O-])cc1F N1(C(c2cnc(C)n2C)=O)CCC2(CCCC2NC(=O)COC2CCC2)C1 c1(C(=O)OCC(=O)N(CCC#C)CC2CC2)csc(C)c1CC c1(CC)cnn(CC(=O)NC2CCC2CNC(=O)CC2CCCOC2)c1 c1(C(=O)N(c2ccnc(Br)n2)CC2(O)CNC2)cc(Br)cc(F)c1F C1(C(=O)NC(C(=O)NCCC)CCN(C)C)(COC)CCCN1C(=O)CNC=O C12(C(N3CCC(OC)(CNC(=O)Cn4ccc(C)n4)C3)=O)CC1COC21CCC1 C1(C(=O)NC(CC(C)NC(C23CC(C)(C2)C3)=O)C)CC(=O)OC1(C)C c1(OC)csc(C(N2CCC(CC(=O)NCc3nc(C(C)C)no3)C2)=O)c1 c1(C(N2C(CC)CN(C(C3(SC)CC3)=O)CC2)=O)cc2c(=O)[nH]ccn2c1 Cc1ccc(-c2nnn(CC(=O)NC3CCC3NC(=O)CC#N)n2)cc1 c1(CC)nc(C(=O)NC2CCOCC2NC(=O)CCCOC)c(C)o1 Cc1ccc(C(=O)NCCC2CCCCN2C(=O)C(C)NC(N)=O)c(F)c1C N1(C(c2cnc(C#N)s2)=O)CCC(NC(C2CC(N(C)C)C2)=O)C(CO)C1 N1(C(C(C)SC)=O)CC(C)(C)CCC1CNC(c1ccc(C(F)(F)F)c(C)c1)=O C1(CNC(c2n[nH]c(C)c2O)=O)N(C(=O)CC2CC=CCN2C)CCCC1(C)C C1(CNC(C2(O)CCC(C)(C)CC2)=O)CCCCC1N=c1[nH]c2cc(Cl)ccc2s1 C1(C(N2CCCC(OCCOC)C2)=O)Cc2cccc(Cl)c2C(=O)O1 c1(NCC(=C)F)ccc(S(=O)(=O)NCC2COC(C)(C)CN2)cc1Br CCC(CC)CCC(=O)NC1(CCCNC(C2CCCSC2)=O)CC1 N1(C(Cn2c(=N)nc[nH]2)=O)CCSCC1C1CC1.C12CC(CO1)C(=O)NC2 C(C)(C)(CCCC(=O)NCCC1CCCC(C)C1)NC(Cc1cn(CC)nc1)=O C#CC1(C)CCN(C(C2CCC(O)CN2C(c2occ3c2CCC3)=O)=O)CC1 c1(C(N(c2nccc(SC)n2)C)=O)cc2c(s1)C1CCC2C1 CC1CCN(C(=O)CCCn2cncn2)CC1NC(=O)Cn1nnc(=O)[nH]1 CCCN=C(NC1CC(=O)N(C2CC2)C1)NC1CC1(c1ccccc1)F c1(NC=O)ccc(Br)cc1[N+](=O)[O-].c12cn(nn1)C(F)(F)C(=O)NC2 N1(CC2C(SC)CCC2)CCC(C)(Cn2cc(CCc3ccccc3)nn2)C1 C=C(C)CC(C(=O)N1CC(CCC(=O)N2CC(C3COCC3O)C2)C1)OC C1(CNC(CCC)=O)(NC(CN(C(c2ccc(CC)o2)=O)C2CC2)=O)CCCCC1 C(C1c2ccsc2CCN1C(C1COC(=O)C1)=O)NC(C(C1CC1)OC)=O N1(C(CCc2n(C)ccn2)=O)CCCC(C)(C)C1C(=O)NCCn1cccn1 C1(NC(CCN(CCCCOC)C)=O)CCN(C(c2c[nH]cc2C(F)(F)F)=O)C1 N1(C(CN(C)C(=O)C2CC2)=O)CC2CCCC1(CNC(c1ccoc1Cl)=O)C2 C=C(C)CCC(=O)NC(c1ccc(NC2CC2)nc1)=O.C12(O)CCN(C1)C2 c1(C(=O)NCC(F)(F)F)nc(Cl)c(Cl)s1.N12CCCC(C1)Cn1nnnc12 c1(OC)ccc(C(=O)NC(CNC(=O)CCC2CCCCO2)C(C)(C)C)nc1 c1(C(N2CC(NC(c3c(CC)onc3C)=O)C(CC)C2)=O)cc2cn[nH]c2cn1 C(CC1=CCN(C(=O)C=CC(c2ccon2)=O)CC1)NC(CCC1C(C)C1)=O C1(NC(C2C(OC)CC2)=O)CC2CC1N(C(c1cnc(C3(C)OCCO3)s1)=O)C2 C1(OC)CC(NC(=O)CSc2nc[nH]n2)CN(C(C23CC4CC2C3C4O)=O)C1 CCC(CC(=O)N(C)CC1(NC(=O)CSCC2CCCO2)CC1)C1CC1 N1(C(C(C)OCC=C)=O)CCC2(CCCC2N2Cc3ccccc3C2)CC1 c1(NC(C2(C)CCCN(C(CSCC=C)=O)C2)=O)cc(C)c(O)c(C)c1 c1(C(=O)NC(CNC(Cc2c(C)noc2)=O)C(C)C(C)C)ccc(Cl)c(C)c1O CC1OC2(CNC(=O)C=CSCc3ccco3)CC1(NC(=O)CC#N)C2 C(CC)(CC)(CCNC(C1CC(OC)C1)=O)NC(C(CC)=CCCC)=O N1(C(C=CC2(C)CCOCC2)=O)CCC2(CC1)CC(NC(C1COC1)=O)CCO2 c1(-c2nc(C(C)C3CC3)nn2CCCC(F)F)ccc2c(c1)OCO2 c1(NC(C(CC(F)F)N(C(c2cn(CCC)nn2)=O)C)=O)cc(C)c(F)cc1C N1(C(CCOCCOCC)=O)C2CCC(C(=O)NC3(C4CC4)CC3)C1CC2 C1(NC(C(=O)NCC(F)(F)F)=O)CCCCN1C(=O)C(F)(F)F c1(C(N(CC(C)CNC(c2cncn2C)=O)C)=O)ccccc1N1CCC(O)C1 Nc1cc(C(N2CC3(CNC(=O)COC4CC=CC4)CCC2C3)=O)c(F)cc1F N(C1CCCn2cnnc21)c1c(C)c(N2CCCC(C)CC2)ncn1 C(CS(=O)(=O)C1CC1)N(CC(F)(F)F)C(c1ccccn1)=O C(CC(=O)NCCc1cn[nH]c1)(C(C)(C)C)NC(C1C(CC)CCC1)=O C(C(C)(C)C#CC(=O)NCc1cnsc1)NC(C=CC1N(C)CCC1)=O C1(NC(c2cscc2C(F)(F)F)=O)C=CCN(C(=O)CC=C(Cl)Cl)C1 C1(C(=O)OCc2nc(C)c(Br)s2)C(C)(C)C(O)C1(C)C CCC(C)CC(=O)C(=O)NCC1(CN(C(=O)Cc2c[nH]nc2C)C)CC1 N1(CCN(C)C)CC2CCN(C(c3cn(CCC(C)(C)C)nn3)=O)C2C1 O(N1CCC(CC(=O)NCC2CN(C(=O)Cc3csc(C)c3)CCO2)CC1)CC c1(C(=O)NC2CC3CN(C(COC(CC)(C)C)=O)C2C3)[nH]c2ccccc2c1Cl C=CCCC(C(=O)NCCCC(=C)Cl)NC(C1CC(C(C)C)C1)=O C1(COC)(NC(=O)NCCCCCF)CCCN(C(=O)OC(C)(C)C)C1 c1(CNC(Cc2c(C)cc(O)cc2)=O)nc2c(s1)CCN(C(c1ccns1)=O)C2 CC(C(=O)N1CCC(OCC2CCN(C(C3CCSCC3)=O)CC2)C1)C(F)(F)F c1(NCCOCCCOC)cccc(C2(C)CCO2)c1 C1(C(=O)NC2CS(=O)C2)(NC(=O)CSC2CCCC(F)C2)CCOCC1 C12(C(N3CCCC(NC(c4nc(C(C)C)oc4)=O)C3)=O)CC1COC2(C)C O(NC(=O)C1=CCC(NC(C23CCN(CC2)CC3)=O)C1)CCCC=C N1(C(c2ccn(C(C)C)n2)=O)CC2CCN(S(=O)(=O)c3cnn(C)c3)C2C1 c1(C(=O)NCC2(OC)CN(C(C3CC(O)C(F)C3)=O)C2)n[nH]c2c1CCCCC2 C#Cc1ccc(C(=O)NC2CN(C(=O)CNC=O)CC2n2cccn2)c(F)c1 Cn1nc(CNC(=O)CNC(=O)CNC(=O)CN2CCNC2=O)oc1=O C(C)(C)(CCC(=O)NCC(C)(C)OCCNC(C1(C)CC1F)=O)OC N1(C(C(C)C#N)=O)CCC(C)(NC(=O)C(CO)c2ccccc2)CC1 C(C(C)(C)CC(=O)N(C1CCC(NC(=O)CC2(N(C)C)CC2)CC1)C)OC(C)=O CCCCC(C)(F)C(=O)N1CCCOC(CNC(c2ccn(C3CC3)c2C)=O)C1 c1(C(=O)NCC(CC)N(C)C(c2cnc(C)nc2)=O)cnc2[nH]ncc2c1 C(O)(CN=C(NC(C)C)NC1CCC(O)CC1)c1ccc(OC)cc1 C#Cc1ccc(OCC(=O)NCCCCCNC(=O)CCC(=C)Br)cc1 C1(NC(c2cnc(COC)s2)=O)C2CC1N(C(=O)CC(C)CF)C2 c1(CC(N2CC(Cn3cc(CN(C)C)nn3)C2)=O)cccc2ncccc12 C1(C(N)=O)C2CCC(C2)N1C(=O)CN1CCN(C(c2ccoc2Cl)=O)CC1 C(=O)(C1=NN(C)C(=O)CC1)NC(CCCC(=O)Nc1c(C)cc(F)nc1)C C1(CC(c2cccs2)=O)CCCCCN1C(C1CC2C(C1)C2(F)F)=O C1(C(=O)NC2(C(=O)NCC(C(C)C)O)CCC2)CCC(=O)N(C)C1 Cc1cc(C)n(CCC(=O)NCCN(C(c2cnc(CO)s2)=O)C(C)C)n1 c1(C(=O)NC(CC#C)C(=O)OC)ccc2c(n1)CN(C(=O)C(F)(F)C(C)O)CC2 c1(C(=O)NCC(CC)(CC)NC(=O)CS(=O)C(F)(F)F)ccc(C#N)c(C)n1 c1(C(N2CC(CNC(C(CCOC)C)=O)C(O)C2)=O)ccc2c(c1)CC(C)(C)O2 O=C(CS(=O)(=O)CCO)NC1COCCC1NC(C1(CC(F)F)CC1)=O c1(OC)ncc(C(C(=O)NC2CCOC2)N(C)Cc2nc(Cl)cs2)cc1C C1(C(C)(C)C)(C(C)C)CCN(C(=O)CC2CC2)C1.C1C(O)C(=O)N1 c1(C(=O)NCC(C)(CO)NC(c2cn[nH]c2)=O)ccc(SC(F)F)cc1 C=C(Br)CC(C)(C)C(=O)N1C2CCC1C(CNC(=O)Cc1ccc(C)o1)C2 C1(CNC(c2ccc(OC)c(C)c2)=O)CC(N=c2ccc(C#N)n[nH]2)C1 C1(NC(C(C)C)=O)CCN(CCC(c2ccccc2)O)CC1C C#CCC(C)(C(=O)N1CCCC(NC(N)=O)CC1)NC(c1cccc(O)c1)=O N#Cc1ccc(S(=O)(=O)NC2CCCC2O)cc1NC1CC(n2cccn2)C1 c1(C(=O)NCC#C)cc(Br)ccc1[N+](=O)[O-].C1CC(=O)N1 C1(NC(=O)Cc2ccc(-c3ccc(F)cc3)s2)CC2(C1)CN(C(C1CCOC1)=O)C2 C1(C(=O)NC(C(=O)NCc2cc(C)ncc2)CO)Cc2ccccc2C1 C1(NC(C(C)SCC)=O)CC(NC(C2(c3ccccc3Cl)CC2)=O)C(O)C1 c1(C2(C(N3CCCC(NC(C4C(OC)C4)=O)C3)=O)CCCC2)ccc(F)cc1F Cc1cc(CN(C(=O)C(CN(C)C)NC(=O)Cc2ccc[nH]2)C)no1 C(=O)(C(C)(C)C1=CCN(C(=O)CC(C)(C)COC(C)=O)C1)N(C(CC)CO)C c1(CC)nc(O)c(C(N2CC3CC(C2)C3NC(c2ccsc2C#N)=O)=O)cc1C N1(C(C(c2ccccc2F)CC)=O)CCC(C2CC2)C1CNC(=O)C(CC)CC C(C(N=[N+]=[N-])C(=O)N1CCCC(N(C(=O)Cc2cnn(CC)c2)CC)C1)OCC C(=O)(C(C)CC(F)(F)F)N1CCC(C(=O)NCC(C)(C)CO)(CC)C1 C(c1ccncn1)=CC(=O)NCCCCNC(=O)CC1(n2cccn2)CC1 c1(CC(N2CC3C(NC(CCCC(=C)C)=O)C3C2)=O)cccc2c1SCCC2 C(CN=C(NCC(c1ccc(O)cc1)(C)C)NC1CC1(F)F)SC C(CC(O)CC(=O)NOCc1cccc(C#N)c1)SC C(CO)(CCCNC(=O)C1=NOCC1)NC(CN(C(C)C)C)=O CC1CCCN(C(=O)CC2(O)CCCCC2)C1CNC(=O)Cc1ccc(F)cc1 C1(C(=O)NCCNC(c2c(CC)c[nH]n2)=O)CC(c2ccncc2)=NO1 C12(C(=O)NC3C(O)CCN(C(C(C)=C4CC4)=O)C3)CC3CC(C)(C1)CC(F)(C3)C2 Cc1c(F)ccc2[nH]c(C(N3CCN(Cc4ccc(C#N)s4)CC3C)=O)cc12 Cc1ccnc(C(N2CCCC(NC(=O)Cn3cnnc3O)CC2)=O)c1Br c1(C(=O)NCCCCNC(CN(C)CCO)=O)cc([N+](=O)[O-])c(F)cc1N c1(C(N2C(C)(CC(=O)NC3CCCC3C3CC3)CC2)=O)cccc2nccn12 C(=O)(C(C)C(F)(F)F)NC1C2CN(C(C3(C)CC(OC)(OC)C3)=O)C1C2 C1(C(=O)NCCC(=C)CNC(=O)COCCCC(C)C)CCC(C)NC1=O Cn1nnc(CNC(C2(F)CC=CCC2)=O)c1C(=O)NCC(O)CC1CCCC1 n1(CC)nc(C)c(CN2CCOC(C(=O)N(C3CC3)Cc3ccno3)C2)c1C C1(C)(C(N(CC#C)C)=O)CC(O)CN1C(c1ccc(NC)cc1)=O CC1=C(C(=O)N2CCN(C(=O)CCc3ccoc3)CC2C)CCCC1 C1(CC(=O)N(C2CCCN(C(c3ncncc3Cl)=O)C2)C)CCCC1(F)F c1(C(=O)NCC(CNC(COCCCCC)=O)F)c(F)ccc(C)c1F N1(C(CC2CCN(C(C(CC)CCOC)=O)C2)=O)CCC(C2(OC)CCC2)CC1 c1(C(N2C(CNC(c3c(C)csn3)=O)COCC2)=O)cccc(F)c1C#N C1(C2CN(C(=O)C=C3CCC3)C2)(NC(c2cccc(C)n2)=O)CC1 C1(CCNC(C(C)(C)N2CCOCC2)=O)CCCN(C(=O)Cc2ccsn2)C1 NS(=O)(=O)CC(=O)NC1COCC1NC(=O)C(C1CC(F)(F)C1)N1CCCC1 C1(CCN(C(C=C(C)C(F)F)=O)C)CCN(C(C23CC(C)(CO2)C3)=O)CC1 C1(n2cc(OC(CC)CC)nn2)CN(C(c2sncc2C(F)(F)F)=O)CC1SC C1(CNC(=O)CCc2ccc(F)c(F)c2)CCN(C(c2ccoc2)=O)C12CCC2 N1(C(CCS(C)=O)=O)CC2CC(NC(C34CCCCC3C4)=O)CC2C1 C(=O)(C(C)CC(C)(C)C)N1CCC(OCC(=O)N(C)Cc2c(C)ccs2)C1 CC(C)(CC(=O)NCCCCCCNC(C1OCCOC12CCC2)=O)C(F)(F)F N1(C(C2OCC(C)(C)OC2)=O)CCOC2C1CCN(C(=O)CCn1ccnc1)C2 c1(N2CCCC(C(C)NC(=O)CC(F)F)C2)nnc2c(c1C#N)CCCC2 C1(C(=O)NCC2CN(C(c3ccoc3)=O)CCO2)CCC2CCCCN12 C1(NC(CCCNC(=O)CN2CC3CC3C2)=O)CCC2(CC2)C1 c1(C(N2CCC(CNC(C3(C4CCC4)CC3)=O)C2)=O)cc2nc[nH]c2cn1 N1(N(C(C)C2CC2)C)CC2(NC=O)CCC1CC2.c1(C=O)cc[nH]c1C1CC1 C1(F)(C(=O)NCO)CC2(CCC2)C1.C12CCCN(CC1)C(=O)C1(CCCO1)CC2 C(=O)(NN1CCCC1C(=O)NCC1CCNC(=O)C1)c1nc(=N)[nH]cc1 CC1(C)CC(C(N2CC(CO)C(C)(C)C2)=O)CN(C(c2ccc(=N)[nH]c2)=O)C1 C(C)(CNC(c1conc1C(F)(F)F)=O)(C(C)C)NC(c1c(OC)csc1)=O Cc1nsc(NC2CCC(CNC(=O)CCn3cc(Cl)cn3)CC2)c1C#N CC1CCC(CNC(c2cccc(Cl)c2O)=O)N(C(c2ccc(C(F)F)s2)=O)C1 c1(CN2CCC(N(CC(=O)Nc3ccccc3)C)C2)ccc(C#N)[nH]1 C1(C(N2C(CC)CC2)=O)CN(C(=O)CCc2ccccn2)Cc2nccn2C1 CCC(CC)(CO)C(=O)N1CC2=C(C1)CN(C(=O)C=Cc1ncc[nH]1)C2 c1(SCC)nncn1CC.c1(C2C3CN(C3)C(=O)NC2)ccnn1C CC(C)(C)C(CN=c1[nH]cncc1I)NC(C1(C)CC(O)CN1C)=O N1(C(C2(COC)CCOC2)=O)CC2(C1)SCCC2NC(=O)Cc1ccsc1Cl C1(C(N(CC(CCC)C)C)=O)CC(C)(C)CCN1C(=O)CCC(C)SC c1(C(N(CCCN(C)C(c2scnc2C2CC2)=O)C)=O)cccc2cc[nH]c12 c1(CC(C(=O)NC2CN(C(c3ccc[nH]3)=O)CC2O)O)c(F)cccc1Cl C1(CN(C(COC2CN(C(C)=O)C2)=O)C)CCCN(C(C2CC(C)(C)CO2)=O)C1 N1(C(CC)=O)CCCC(C(=O)NCC(CO)NC(=O)CCN2CCCC2=O)C1 Cn1nc2c(c1NC(=O)NCC(c1ccc(S(C)(=O)=O)cc1)O)CCCC2 CC(=O)C(C)(C)CC(=O)N1CCCC(C)C1CNC(c1ccc(C)cc1)=O C1(C(=O)NCC(CC)NC(c2cncs2)=O)CN(C(C)C)CCO1 c1(OCCC)c(Cl)cc(CN2CC3CC2CC3(F)F)cc1Cl c1(-c2nc(CN3C(c4ccc(SC)s4)CCC3)on2)cc(C2CC2)ccn1 CC1(C)CC(NC(=O)C=CBr)CN(C(c2cc(C3(C)CC3)ccc2F)=O)C1 C1(C(N2CCCC(C=C)C2)=O)CCCN1NC(=O)c1cc(C)c(C)nn1 CC1CN(C(c2cnc(C3CC3)[nH]2)=O)CC1CNC(=O)C(C)N1CC(C)C1 N1(C(CCCSC)=O)CCc2ccc(CNC(=O)CC(O)C3CC3)cc2CC1 C(=O)(C(O)CCC(C)C)NC1CCN(C(c2c(C)ccc(SC)c2)=O)C1 C1(C(N(CCCNC(CCc2nc(C)sc2)=O)C(C)C)=O)CC2CCCC2C1 Cc1c(Br)ccc(C(=O)Nc2nc(CC(=O)Nc3nccnc3Cl)cs2)c1C c1(C(C)C)cccc(-c2cn(CC(C)NC(C3CCOC3C)=O)nn2)c1 c1(NS(C)(=O)=O)ccc(C(=O)NC2(CCNC(C3CCCSC3)=O)CC2)cc1 C(=O)(C(O)CC(C)(C)C)NCC(CNC(C(C)(C)OC(C)=O)=O)O N1(C(C(=O)NC(c2cccc(C3CC3)c2)C)=O)CCC2C(CCCN2C2CC2)C1 C(=O)(C(C)CC(C)C(C)=O)NCC(CNC(c1nc(CC)oc1C)=O)CO c1(C2C(C(=O)NCCC3CN(C(C(C=CC)O)=O)C3)C2)cc(F)ccc1F CCCC(CO)NC(C1CC(C)(NC(c2cnn(C3CC3)c2)=O)C1)=O N1(CCCCOCCOCCCC)CCCC(C(=O)OC)C1C N1(S(c2ccn(C)n2)(=O)=O)CC2CCN(C(c3c(F)ccc(Cl)c3Cl)=O)C2C1 C1(CN(C(CCn2cc(C(OC)OC)nn2)=O)C)CN(C(C)=O)CCCO1 N1(C(COc2cc(C)on2)=O)CCCC2(C1)CN(c1ncc(Br)cn1)CCO2 N1(C(CC2N(CC)C(=O)CC2)=O)CCC2(C1)CN(C(c1ccnc(C)n1)=O)C2 N1(C(C2N(S(CCC)(=O)=O)CCC2)=O)CCN(C(=O)C(=O)NCC)C(CF)C1 c1(C(=O)NC(CC)(C)CNC(=O)C(F)OC(F)(F)F)cc(F)cc(N)c1F N1(C(C2C(C)(C)COCC2)=O)CCCC12CCN(C(c1ncccc1Cl)=O)C2 n1(CC)ncc(C(=O)NC2CC(NC(=O)C(C)CCOC)C2)c1Br CC1(C#N)CN(C(=O)CN(CCS(C)(=N)=O)C(=O)OC(C)(C)C)C1.C(=O)C1CC1 N1(C(=O)Nc2c(C)n[nH]c2C)CCOCC(C(=O)N(C)Cc2cccs2)C1 c1(C(=O)NC(CNC(c2cc(C)c(O)nc2)=O)CO)ccc2nccn2c1 C(=O)(C(F)C(C)(C)O)NCc1cccc(C(=O)NC2C(N(C)C)CCCC2)c1 C1(C(c2n(C(CC)(C)C)nnn2)NC2CC(SC)C2)CC2(C1)OCCO2 C1(C(C)(C)NC(C=CSC)=O)CCN(C(c2coc(Br)n2)=O)CC1 CCCCC(C(=O)NCC(CC)(CC)NC(=O)Cc1cccs1)NC(N)=O C(CC(=O)Nc1ccc(F)c(C)c1)(C(C)C)NC(c1ncn(CC)n1)=O c1(C(N(CCCNC(c2cn(CC=C)nc2)=O)CCO)=O)ccc2c(c1)CC2 C1(C(N2CCN(C(C(C)=C3CCC3)=O)CC23CC3)=O)CCn2c(cnc2C)C1 c1(OC)cc(OC)c(CN2CC(NC(=O)Cc3ccsc3)C3(CC3)C2)c(C)c1 C1(C(N2CC(NC(C=C(CC)CC)=O)CC3(C2)CC3)=O)CCc2c(n[nH]c2C)C1 C(=O)(C1=CS(=O)CCC1)N1C(C(C)C)CN(C(=O)CCC(C)(F)F)CC1 c1(C(C)N(C)C)cccc(C(N2CCOC(NC(C3CCC4(C3)N=N4)=O)C2)=O)c1 C(CC(C)C(=O)NCCNC(C1CC(=O)C1C(C)(C)C)=O)OC c1(C(N2CC(CNC(CC)=O)C2)=O)cc(OC)c(O)c(OC)c1 c12ccc(cc1)[nH]c2=O.C(=O)(C(CN(C)C)N(C)C)N(CCCN(CC(C)C)C)C C1(C)(CNCC(C2CC(C)(C)C2)O)CCC2(CC1)OCCO2 N1(C(=O)CSc2ccc(F)cc2)CCC2C(CCN2C(c2cc(O)no2)=O)C1 c1(C(N2CCC(OC)C2)=O)ccc(OCC(c2ccco2)N2CCCC2)cc1 c1(C(=O)NC2CC(CCC(N3CCOCC3CCO)=O)C2)cccc2c1CCO2 c1(CC)cc(F)ccc1C(=O)N(C1CCC(NC(=O)C2=CC(C)(C)C2)CC1)C N1(C(C(F)=CCC)=O)CC(CNC(=O)CCC(=O)c2ccnc(OC)c2)C(C)C1 C1(C(N(C)Cc2cc(C)on2)=O)CCCCN(C(c2cnc[nH]c2=N)=O)C1 CCC(C(=O)N1CCCC1CC(=O)NOCC(O)CO)OC N1(C(COCCCC(C)C)=O)CC(NC(=O)CSc2ccccn2)C2CC12 C1(C(=O)NC2C(CNC(CCC#C)=O)C2)OCC2CCCC12 c1(C(C)C2CC2)nc(-c2cncc(F)c2)n(C2CCOC2(C)C)n1 c1(C(N2CC(C)C(NC(c3cnc(N)cn3)=O)C2)=O)cccc(F)c1C(F)(F)F Cc1nsc(C)c1C(=O)N(C)CC1(NC(c2ccnc(-n3ccnc3)c2)=O)CC1 c1(C(=O)NC2CCN(C(CCC3N(C)CCCC3)=O)C2)cnc2c(c1)CCCO2 C1(C(C)C)N(C(c2ccc(C#N)[nH]2)=O)CC12CCN(C(=O)C(F)(F)C1CC1)CC2 C(CCN=c1[nH]cnc2ccc(O)cc12)NC(c1cc2cnccc2[nH]1)=O c1(SC)ccc(C(=O)NCC2CN(C(=O)Cc3cc[nH]n3)CC2O)c(Cl)c1 C1(CNC(CCCC=C)=O)CCN(C(=O)Cc2conc2COC)CC1(F)F c1(OCC(=O)NCC2(CNC(CCC(=O)NC)=O)CC2)cc(C)ccc1CO C12(CC(=O)N(CC3N(C(CCCc4scc(C)n4)=O)CC3)CC)CCC(CC1)OC2 C1(NC(CC2(C)CC2)=O)CCN(C(C2CCC2c2ccc(F)cc2)=O)C12CCC2 CCC(C(=O)NCC(C)NC(c1coc(C)n1)=O)n1ccnc1 CC1(C)CCCOC1CCn1cc(C2CCN2C(C2CC(F)C(=O)N2)=O)nn1 CC(C)(C)CC(O)C(=O)NCC(CNC(=O)COc1ccccc1F)CO c1(C(N2C(CN(C(=O)C(N)=O)C)CCC2)=O)ccc2c(n1)OCCO2 CC(C)CCCC(=O)NCC1COCCN1C(=O)CCc1ccc(O)c(Cl)c1 CCC(CC(=O)N1CC(SC)C(C(N2CC(c3n[nH]c(C)n3)C2)=O)C1)SC CCC(CCN(C)C)C(=O)NC(C1(O)CCN(C(=O)CC2CC3(CC3)C2)CC1)C C1(C(=O)NCC2C(NC(C(C(C)C)O)=O)CC2)CC2(COC(=O)N2)C1 C1(N(CCC)C(c2ncn(C)n2)=O)CCN(C(=O)CCC2CCC(C)O2)CC1 CC1C(NC(=O)C(C)(C)c2cccs2)CCCN1C(c1csc(C2CC2)n1)=O c1(NC(c2c(CC)c(F)ccc2)=O)cnc2cccnc2c1 C1(C(N2CCC(N(C(c3c(C)ccnn3)=O)C)CC2)=O)CN2CCC1(C)C2 N1(C(C2(C)CCCCC2)=O)CC(NC(=O)COCC2CCC2)CC(O)C1 O=C1Cc2c(C(N3CCC3Cn3cc(-c4cncnc4)nn3)=O)ccnc2N1 N1(C(CN(C(C)=O)C)=O)CC(NC(c2c[nH]nc2-c2ccco2)=O)C(O)C1 c1(C(=O)Nc2cnn(C3CCCCC3)c2)cccc2ncnc(O)c12 C(=O)(CC(C)CC(F)(F)F)N1CCC(CCNC(C(C(C)C)F)=O)CC1 N1(C(c2c[nH]c(=NCC)s2)=O)CC2(COC(CNC(C3CCCOC3C)=O)C2)C1 C1(CCNC(CC)=O)CN(C(c2coc(C)n2)=O)CCS1(=O)=O C1(C(=O)NCCN2CC(NC(=O)CC3CCCC(O)C3)C2)CCCCCCC1 c1(N(C(CC=C)C)CC)ccc(S(=O)(=O)NC(C2CCN(C)C2)CC)cc1Cl c1(OC)cn(C)c(C(N2CC3(CCC3NC(C3CN(C)CCO3)=O)C2)=O)cc1=O CC1CN(C(C2CCN(c3nc(=N)[nH][nH]3)C2)=O)CCCN1C(=O)C(=O)N(C)C c1(N2CCC(OCC)CC2)ncnc(N2CCCC(C)(c3ccccc3)C2)c1C N1(C(C(COC)C)=O)CC2CN(C(c3cc(F)cc(F)c3O)=O)CCC12 O=C(CCCCCc1ccccc1)NCC12CC(CN1)C2 Cc1ncn2ccc(C(N3CCC(N(CCO)C(C4CCSC4)=O)CC3)=O)cc12 N1(C(C2(F)CCCN(C)C2)=O)CCC(C2CCN(C(c3cnn[nH]3)=O)C2)CC1 c1(C(N2C3CN(C(=O)CC4CCCC45CC5)C(C3)C2)=O)onc2ccccc12 c1(CC)ccc(C(F)(F)F)cc1C(=O)NCCCN(c1ccc(F)cc1)CC(C)O c1(C(=O)NCC(CN(C)C(c2cc(C3CC3)ccc2F)=O)O)cc(O)nc(O)c1 c1(N2CCN(C(C3C(C)OC(C)C3)=O)CC2C)cc(CO)c([N+](=O)[O-])cn1 CC1CCCCC1CC(=O)N(CCCCC(=O)N(C)Cc1cnnn1C)C c1(C(=O)NCC(C)(C)NC(C(C)=C2CC2)=O)cc(S(=O)(=O)CC#N)ccc1F C1(CC)CN(C(C2C3(CC3)C23CC3)=O)CCC1NC(c1cscc1Br)=O n1(CC(N2CC(F)(C(=O)NC(CC#C)CO)C2)=O)cccnc1=O C12(C(N3CC(C=C)C(NC(=O)C(CC)(CC)CC)C3)=O)CC1COC21CCC1 c1(C(=O)NCC(C(C)(C)C)NC(=O)C=Cc2cnc[nH]2)ccc(C#N)cc1[N+](=O)[O-] Cc1noc(C)c1C(N1CCC(CF)(NC(=O)CC(=O)NCC2CC2)C1)=O c1(C(=O)NCC2(C(N(C)CC3C=CCC3)=O)CCCC2)ccccc1F CC(C)C(C)C(CNCc1cc(Br)ccc1Cl)NC(=O)OC(C)(C)C CC1CC(C)OC1C(N1CC(C(C)NC(=O)CCC2(C)N=N2)C1)=O CCC(C)(COC)C(=O)N(C(C)C(=O)NCc1cc(C)c(C)o1)C c1(C(N(C)Cc2cocn2)=O)c(O)n[nH]c1-c1ccc(Br)cc1 C1(NC(C(C=C)C)=O)CC(F)CN(C(=O)C=C2CCN(C)CC2)C1 C(CCC(C)C)(C(=O)N1CC(CO)CC1CO)NC(CCC(CC)=O)=O c1(NC(CC(c2ccc(C)cc2)C(=O)N(C2CC2)C2CC2)=O)ncc2[nH]cc(I)c2n1 C1(NC(C2CCN(C(C)=O)C2)=O)CCCN(C(c2cccc(C3CC3)n2)=O)CC1 N1(C(C2CN(S(C)(=O)=O)C2)=O)CCN(C(=O)CCc2csc(=N)[nH]2)CC1.C1CC1 c1(C(N2CC(CNC(C3CC4C(C3)C4(F)F)=O)OCC2)=O)ccc2ncsc2c1 C12(CCCCO1)C(=O)NC2C.N1(CCC)CC(NC(=O)C(O)C2CCC2)C1 c1(C(N(C2CC3CCC(C2)N3C(=O)C2=CCCC2)C)=O)ccn2c(O)nnc2c1 Cc1nn(CC(N2CC(NC(c3occc3C(C)C)=O)CC2CO)=O)cc1Cl N1(C(C(C)SCC)=O)CC(NC(c2cc(N)ccc2Cl)=O)CC12CCCC2 N1(C(C(C)=CC2CC2)=O)CC(N=c2[nH]nc(C3CC3)s2)C(C)(C)C1 C1(NC(C2CCC(=C)CC2)=O)COCCN(C(=O)C=Cc2cnccc2C)C1 C(=O)(C1=CC2CCC(C1)C2)N1CCC(NC(c2cc(F)ccc2F)=O)(CF)C1 C1(NC(c2c(C)nc(CO)s2)=O)CCC2(CC1)CC2NC(=O)CS(N)(=O)=O CS(=O)(=NC(=O)CN1CC(O)C(O)C1)c1ccc(F)cc1 CCC(C)C(C)C(=O)NCC(C(C)C)NC(c1ccc(OCCC(C)C)cc1)=O C(=O)(C(C)(C)C(=O)NCC1C2CN(C(=O)C(C3CC3)N(C)C)CC12)NC N1(C(C(c2ccoc2)NC(=O)Cc2cc[nH]c2)=O)C2CCC1CC2 c1(CNC(C2OCCN(C(c3cc(CC)[nH]n3)=O)C2)=O)cccc(C#N)c1 C(=O)(CCCN=[N+]=[N-])NCC(Cc1c(C)cccc1)CO C(=O)(C1=CCCC(C)(C)C1)N1CC(CN(C(c2c(CC)scc2)=O)C)OCC1 C1(C(=O)NCCc2c(OC)c(Br)ccc2)CC(=O)N2CCCCC12 CCCCCCC(C)CC(=O)N1C2CCC1CC(NC(=O)C(C)OC)C2 N1(C(COC(C)C)=O)CCOC2(CCC(C(=O)Nc3nncn3C)CC2)C1 CC(C(=O)N1CCC(NC(=O)CC(C)(C)C2CC2)C(C(N)=O)C1)S(N)(=O)=O CC(CC(=O)NCc1cn(C2CN(C(=O)CCC3CC3C)C2)nn1)C(F)F C1(NC(c2c(C)cccc2F)=O)CN(C(c2sccc2Cl)=O)C2(CCCOC2)C1 CC(CC(=O)N1CC(=C(F)CNC(C2CCCCS2)=O)C1)c1cnn(C)c1 C#CCCCCC(=O)NCC1CC(C(F)(F)F)CCN1C(=O)C=NOC c1(C(C)=O)cc(C(=O)NCC2CC(NC(=O)Cc3ccc(C(F)(F)F)o3)C2)no1 C(=O)(C(C(C)C)NC(N)=O)N(CCC(=O)NCC(C)OCC=C)CC C1(NC(c2cccnc2)CCC)CC2CCCC2(CN)C1 C1(CNC(CC(C)n2ccnc2)=O)C2CN(C(=O)C=CCn3cncn3)CC12 C1(NC(CC(C=C)C)=O)CCN(C(c2cccc(OC(C)C)n2)=O)CC(C)(C)C1 C1(C)(C(N2CC(C)(COC)C2)=O)CN(C(c2cnncc2C)=O)CC1C C1(CNC(C=C(C)Cl)=O)COC(CNC(=O)CCSc2n[nH]c(C)n2)C1 C(=O)(C=CS(C)=O)NCCCCN(C(CCC)=O)C c1(C(N(C2CN(C(C3CCCCN3CC(F)F)=O)CC2O)C)=O)ccc(O)cc1 C(CC(C)C)(C(=O)NCC(C1CC1)N(C(=O)CSc1ccsc1[N+](=O)[O-])C)OC C(C(C)C)(C(O)C(=O)N1CC(O)CC1(C)C(=O)NC1(C)CCC(C)=C(C)C1)OC Cc1cc(Cl)c(CN2CCC(C(=O)Nc3cccc4[nH]ncc34)C(O)C2)c(Cl)c1 c1(CC)noc(C)c1C(=O)NCC1(NC(=O)CCc2cncnc2)CCOC1 c1(C(CNC(CC(=O)OCC)C2CCCC2)=O)ccc(O)cc1 CCCC(C(=O)NCc1ccc(CN(C(=O)C=Cc2ncc(C)[nH]2)C)cc1)OC C(C(=O)NCCC1CC(NC(c2cscc2C2CC2)=O)C1)(C(C)(C)C)SC C(CCCCCNC(c1cccn1C1CC1)=O)NC(c1cc(C(F)F)[nH]n1)=O N1(C(c2c(OC)scc2)=O)CC(NC(=O)CCC(C)(C)C)C(F)(F)C1 N1(C(c2c(C)ccc(C)n2)=O)CCN(C(=O)C(c2ccc(F)cc2)C)CCC1C C1(NC(=O)C(=O)OC(C)=O)COC2CC1C2.C(C1C(=O)N1)OC C1(C(N(C(Cn2ccc(C(=O)OC)n2)=O)CCSC)=O)CCC2(CC2)C1 c1(C(=O)NCC2CCN(C(=O)CN3CCSCC3)C2)cccn2c(O)nnc12 N1(C(CC=CCNC(C(NOC)=O)=O)=O)CCC(O)CC(C)C1 C(=O)(CCCCC(C)CC)N(CC1(CNC(c2ccc(CC)c(Cl)c2)=O)CC1)CC C1(CC)COCCN(C(=O)C(c2cccs2)NC(=O)C(O)CCN(C)C)C1 C(CCCCC(=O)N1CCCC1CCNC(C1CC(O)(C(F)F)C1)=O)N(C)C C1(C(=O)NCC(C(C)(C)C)NC(CCCC)=O)CCc2nnc(C)n2C1 n1(CC)cc([N+](=O)[O-])c(C(N2CCN(C(=O)CN3CC(C)(C)C3)C3(CC3)C2)=O)n1 C(=O)(C(O)C(F)(F)F)N1C(CNC(CCN2CCC(C(N)=O)CC2)=O)CCCC1 c1(C(=O)NCCC2(O)CN(C(C3C(OCC)C3C)=O)C2)cc(C#N)ccc1O C(=O)(C(C(C)(C)C)NC(c1cnc(CC)o1)=O)NCc1cn(CC=C)nn1 c1(NC(NCS(CC)(=O)=O)=O)c(C)ccc2cc(C)ccc12 c1(OC)c(C(=O)NCCNC(=O)CC(C)(C)F)sc(Cl)c1Cl N1(C(c2nnsc2CC2CC2)=O)CCC(c2ccc(Br)cn2)CC1 c1(C(N2CC(CNC(C3(C(F)(F)F)CC3)=O)C3CC23)=O)cc2cc(Cl)cnc2[nH]1 C1(NC(CCC)=O)CCN(C(=O)CCOC(C)C)CC1c1ccccc1 C1(CNC(C2C3CCN2CC3)=O)CC(F)CN1C(=O)CCC1CCCCO1 S(=O)(=O)(c1ccc(O)cc1)N1CC2N(C(c3cc(Br)ccc3Cl)=O)C2C1 c1(C(N2CC(C)C(NC(c3nc(Cl)ccc3Cl)=O)C2)=O)cc2n(n1)C(C)CCC2 C(C(CC(=O)N1CCN(C(=O)C=CC2CCC2)C(CF)C1)C(F)F)N(C)C C12(CC(=O)N(C3CCCC3)CCNC(CCNC(C)=O)=O)CCCCC1C2(F)F C1(C(=O)NCc2ccc(Cl)c(F)c2)CN(c2ncnc3c2CCC3)CCC1(F)F c1(CC(=O)NC23C(CN(C(C=CCOC)=O)C2)C3)ccc2sccc2c1 c1(C(=O)NC(c2c(OC)cc(O)nc2)=O)c[nH]c2ccccc12.CCO C(=O)(CC(C)CCC=C(C)C)NCC1C(NC(c2c(C#C)c[nH]n2)=O)C1 Cc1cc(Cl)ccc1C(=O)N(C)CC1CCCN1C(c1cnnn1C1CC1)=O C#CCC(CC(F)F)C(=O)N1CCCC(CC(N2CCCCC2C(=O)OC)=O)C1 N1(C(c2cccc(C#C)c2)C(=O)NCCCC)C2CCCC1CC(O)C2 C1(CNC(C(C)OCOC)=O)OCCC1C(=O)NCC1(CCOC)CC1 C12CC3(C1)CC3C(=O)N2.N1(C(CC=C)=O)CCCCC1COC c1(NOC(C2(Cl)CC2)=O)ccc(S(N)(=O)=O)cc1C(N1CCC(C(N)=O)C1)=O C1(CC)(OC(C2CN(CCOc3cccc(C)c3)CC23CC3)=O)CCCCCC1 C1(CNC(C(C)(C)OCC)=O)CC2CCCC2N1C(c1csc(C2CC2)n1)=O CON(CC1CSc2ccccc21)C(=O)c1cccc(S(C)=O)c1 C1(CC)CN(Cc2c(C)ncn2C)CC1c1cnn(C)c1 CCCCC(O)CCC(=O)NC(C1CCN(C(=O)C(c2ccccc2)C)CC1)C C(N=c1cc(Cl)nc(C2CCOCC2)[nH]1)C1CCN(C(COC(C)(C)C)=O)C1 C(CC(F)F)(C(=O)Nc1ccc(O)nc1)NC(c1c[nH]c(=S)cn1)=O N1(C(Cc2c(C)noc2Cl)=O)CCC(CNC(c2ccc(Cl)nc2O)=O)CC1C CCC1=C(C(=O)N2CCN(C)C(C(=O)NCC3CC(OC)C3)C2)CCCO1 c1(C(=O)NCC(CC)NC(C(C(CC)O)C)=O)c(F)cc(N)cc1F C1(NC(CCN(C(=O)CC2(O)CCC2)CC#C)=O)CC2(CCCC2)C1 O=C(C(F)C1=CCCCC1)NC1CCCN(C(=O)Cc2nnc3n2CCOC3)C1 c1(C(N(CC(CC)NC(c2ccnn2CC)=O)CC)=O)cnncc1OC N1(Cc2ccc(CC)cc2F)CC2CCC(C1)N2C(c1cc(=O)ccn1C)=O CCC(CC(=O)N1CC2C(CC(=O)NCCCc3nncs3)C2C1)OC C12(CCCCC1)CC(=O)N2.c1(C(C)(C)OC(C)=O)cn(CCC(F)(F)Cl)nn1 CC1(CCNC(C2COCC2n2ccnn2)=O)CCCC1 CC1CCC(CNC(C2CC3(CC3)C2)=O)N(C(c2nnc(C(C)(C)C)s2)=O)C1 Cc1ccc(C(=O)NC(C(=O)NCCn2ncnn2)C(C)C)cc1 CCCCCC(O)C(=O)NC1CCCC1NC(=O)CN1CCCC1CO C(C)(CC(C)C(F)F)NC(C1N(C(c2cc(C(C)C)on2)=O)CCSC1)=O CC(CS(=O)(=O)N(C)C)N=c1nc2sccc2c(NCc2cscc2Cl)[nH]1 C1(N(CCCO)C)CCCC12CCN(C(c1cc(F)ccc1I)=O)CC2 N(C1CCc2cccnc21)C(C1CCC(NCc2c(C)c(Br)cnc2)C1)=O C1(c2cn(CCNC(CCC=C)=O)nn2)CCCCC1=O C(CC(C)C)(C(=O)N1CC(c2ccon2)C1)N(C(Cc1c(C)nccc1)=O)C C(N=c1[nH]nc(CO)s1)C12OCC(NC(CCCSC)=O)(C1)C2 c1(NC(C(=O)N(C(CC)CC)CC)=O)cnn(CC(F)(F)F)c1 C1(NC(c2c(C(C)NC(COCC)=O)noc2)=O)CCn2ccnc2C1 C1(CNC(CC(C)SC)=O)CC2(CCC2)CN1C(c1nc(C(C)C)ncc1Cl)=O CC1C(C)N(C(c2cccc(Br)c2)C(=O)NC(c2ccco2)C2CC2)CCS1(=O)=O N1(C(C2(C(=O)NC)CCC2)=O)CC(CNC(C2CC=CCO2)=O)C(O)C1 C(C(C)(C)C(C)(C)C)NC(CC1(OCC)CN(C(=O)C(C)CO)C1)=O N1(C(C2N(CC)CCC2)=O)CC2OCC(NC(=O)CN3CCCCC3)C2C1 Cc1cccc2c(C(N3CCN(C(c4nc(=N)cc[nH]4)=O)C(C)C3C)=O)coc12 c1(NC(c2cn(Cc3cccnc3)nn2)=O)nnc(CCCF)s1 c1(C(=O)NC2CC(NC(=O)CC3C=CS(=O)(=O)C3)C2)ccc2c(c1)C(=O)NCC2 c1(C(=O)OC)ncnc2c1cnn2C1(OC2CC(F)C2)CCCC1 C1(CC=C)(NC(c2nc(C)ncc2Cl)=O)CCN(C(=O)CS(N)(=O)=O)CC1 c1(C(=O)NC2(C3(O)CN(C(=O)OC(C)(C)C)C3)CC2)cnc(-c2cccs2)nc1 CC1CCN(C(=O)C=CC2CCCC2)CC1NC(C1CCC(=O)N1C)=O CN1CCN(C(=O)CCN2CCOCC2)CC1CNC(C1(C)CCCO1)=O N1(Cc2c(OC)ncc(Br)c2)CCC2(CC1)CC2NC(c1ccc(C)c(I)c1)=O C1(C)(C(=O)NCCOCCCN(C(COCCC)=O)C)CC1F C1(CNC(CC(CC)CC)=O)CCCC2CN(C(c3ccnn3C)=O)CC12 c1(OCC(N2C(CN(C(C=CCC)=O)C)CCC2)=O)ccc(S(N)(=O)=O)cc1F N1(C(C(C=C)(C)C)=O)CCN(CCNC(=O)C(CCC)C(=O)OC)C2(CCC2)C1 c1(CNC(C2CC(C#N)C2)=O)nc2c(s1)CCN(C(C13CC(CO1)C3)=O)C2 c1(C(=O)NC2CC(OC)CN(C(=O)C(C)(C)C(C)O)C2)cc(C)cc([N+](=O)[O-])c1 CC(CC(=O)N1CC2C(NC(=O)C=Cc3ccccn3)C2C1)C(F)F C1(Nc2ccc(-c3nnc(C)o3)cc2)CC2CCCCC2C1 c1(CCNC(=NCCCC)NC2CC23CC3(F)F)cc(F)cc2c1OCOC2 c1(C(N2CC3=C(CN(C(C4CCCC(=O)O4)=O)C3)C2)=O)cc2ccc(O)nc2s1 C12(CC(=O)NC3C(CC=C)COC3)CC(S(C)(=O)=O)(C1)C2 C12(CNC(CCC(=C)Cl)=O)CCCCC1CN(C(=O)CC1CC(=C)C1)C2 C12COCC1n1cc(nn1)CN2C.C1(CSC)CC1(C(=O)O)C(=O)O N1(C(c2cc(C)c(C)[nH]2)=O)CC(C2CCCN(C(=O)CSc3nncs3)C2)C1 Cc1c(C(N2CCCC2CN(C(=O)C(C)C(F)(F)F)C)=O)sc2ccsc12 C1(F)(CNC(c2cnc(OC)s2)=O)CCCN(C(C2COCCN2C=O)=O)C1 N1(C(CC(CC)C)=O)CC2CC(NC(c3cnc4sccc4c3)=O)CC2C1 c1(C(N2CC(O)(CNC(C=CS(C)=O)=O)C2)=O)ccc(F)c(-c2ccccc2)n1 N1(C(C(CCC)NC(c2ncn(C(C)C)n2)=O)=O)CCC2(C=CCO2)CC1 CC12CCC(C(=O)NC3(CO)CN(C(=O)C(O)P(C)(C)=O)C3)(CC1)C(C)(C)O2 N1(C(C=COOC(F)F)=O)CCc2[nH]nc(-c3cccc(CC)c3)c2C1 c1(C(=O)NCCN(C(C(C)SCC)=O)C2CC2)cnc2c(C)cc(C)cc2c1O c1(C(=O)NCCC(C)N(C(CCCN(C(=O)OC)C)=O)C)[nH]ccc(=O)c1C C(CCC(=O)NC1CC(O)C1O)(C(C)C)NC(C1(CC#C)CCC1)=O CCC(CNC(c1ccc(F)cn1)=O)(CC)NC(C1CC2CC1CO2)=O C(=O)(C1CCc2cc(OC)ccc21)N(CCNC(c1cc(COC)no1)=O)C Cc1cc(C(c2ccccc2F)NS(=O)(=O)CCC2CC(F)C2)ccn1 CC1(C)C(NC(=O)Cc2nc(C3CC3)cs2)CC1CNC(=O)Cc1csnn1 N1(CC)CCOCC1C(N1C(C(=O)NC(Cc2ccco2)CO)CC2CC12)=O C1(C(=O)NC(CNC(c2nc(C)nn2C)=O)C2CCC2)CCn2ccnc2C1 C1(CNC(C(C)OCC=C)=O)CCCCCN1C(=O)CC(C1CCC1)C1CCC1 C1(F)(CNC(C(N2CCN(C)CC2)C)=O)CC(N=c2[nH]nc(C(C)(C)C)s2)C1 N1(C(C(C)(C)OC)=O)CCC(C(=O)Nc2ccccc2CC#N)CC1 Cc1ccnc(Cl)c1C(=O)NCC1CCCN1Cc1ccnc(Cl)c1Cl C#CC1(C(=O)OC)CN(C(=O)C(C)OCOC)C1 c1(C(N2CCC(NC(c3c(C)cccc3Cl)=O)C2)=O)cnc2c(Br)cccn12 N1(C(CN(CC)CC)=O)CCN(C(C2(C)CC(C(F)(F)F)C2)=O)CC(C)(F)C1 O=C(CCc1cn[nH]c1)NNc1ccc(-c2ccccc2)nc1 N1(C(c2ncc(OC)nc2)=O)CC(=O)NCC1C(=O)NC(C)Cn1cnnc1 C=CCCN=C(NCCC1CCC(C)O1)N1CCC(NC(=O)NC)C1 Cc1cc2cccc(NC(C3CCOC4(CCOCC4)C3)=O)c2cn1 C(=O)(CC(C)CC(C)C)N1CCC(CCC(C)(C)NC(C(C(CC)C)O)=O)CC1 C1(C(N2CC(N(C(=O)CN3CCS(=O)CC3)C)C2)=O)CCCc2ccccc2C1 N1(C(C2C(C)(C)CN(C(=O)CCC3CCC3)C2)=O)CC2C=CCC(C2)C1 C1(CC)CCCN(C(c2cnc(OC)s2)=O)C1C(=O)NC1CCC(C(N)=O)C1 c1(C(N2CCC(CNC(CCOC)=O)C2(C)C)=O)cc(Cl)cc(Cl)c1N C(=O)(C(F)C(F)(F)F)NC1CCC(CNC(=O)CC2CCCC2O)C1 O=C(CS(=O)(=O)C1CC1)NC1CCCC1NC(C1CCN1Cc1ccccc1)=O c1(CN(C)Cc2cn(-c3ccc(C(C)(C)C)nc3)nn2)ccc(C(=O)O)cc1 Cc1cc(F)ccc1Cn1cc(CCC(=O)NC(C2(O)CC2)C)nn1 C12(N(C(C(C)C)Cc3nn[nH]n3)C(c3ccccn3)=O)CCCC(CO1)C2 S(=O)(=O)(c1ccc(Cl)nc1C)N1C(C(=O)Nc2c(C)nc(Br)cn2)CC(F)C1 CCC(CC(=O)N1C(C(=O)NCCCOCCO)CC1C)CC(C)C CS(=O)(=O)c1ccccc1CC(=O)NC1CCC1CNC(=O)C(O)CF c1(C(N2CCC(OC)(CNC(C3(F)CCOC3)=O)C2)=O)cncc(Cl)c1Cl C1(C)(OCC(=O)NCC(C)OC)CN(C(c2coc(C(C)C)n2)=O)C1 N1(C(C2CCOC2C(=O)NOCCOCCF)=O)CCOC2COCC12 c1(CN2CC(C)(CNC(c3ccc(Cl)c(Br)c3)=O)C2)cc(Br)cc([N+](=O)[O-])c1O C1(NC(c2c(CC)nn[nH]2)=O)CN(C(=O)C(C)(O)C(C)C)CC(F)(F)C1 C(C)(N=c1[nH]c2c(c(=NCC3CCCC(F)(F)C3)[nH]1)COC2)C1(COC)CC1 c1(C(=O)NCC2CC(NC(C3(CS(C)(=O)=O)COC3)=O)C2)ccc(Cl)nc1O CCC(C)(C)C(=O)NCc1csc(C(=O)NC2(C(O)COC)CC2)c1 C1(C(N(CC(=O)OC)CCCOCCCNC(=O)NC2CCCC2)=O)CC1(F)Cl c1(C(=O)NCC2CN(C(C=NOC)=O)CC2(F)F)ccc2c(c1)ncn2C c1(C(=O)NC2CN(C(C=C(C)Cl)=O)CC2O)cc(C)cnc1C C1(CNC(c2c(OC)nc(C)cc2)=O)C(C2CC2)CCN1C(=O)CSC(C)(C)C C=CCCCC(=O)N1CCCC(NC(c2occc2-c2ccc(F)cc2)=O)C1 C1(NC(c2ccc(C)o2)=O)CCC2CC1CN2C(c1cc(=O)c(Br)c[nH]1)=O N1(C(CC=CCC)=O)CSCC1C(=O)N(C(C)C(C)SC)C c1(C(N2C(CNC(C(C(C)C)OC)=O)C=CC2)=O)oc2c(C)ccc(C)c2c1C CCCCCCCCC(=O)N1CC(O)CC1(C)C(N1CC(C#N)(COC)C1)=O N1(C(C(C)(C)c2cc[nH]n2)=O)CCC(SC)C(NC(=O)Cc2cccc(Cl)c2)C1 c1(OC)cc(OC)c(C(=O)NCC2(F)CN(C(C3CC=CCO3)=O)C2)c(OC)c1 CC1Cc2cc(C(N3CCC(NC(=O)C4=CCOCC4)CC(O)C3)=O)ccc2O1 C(=O)(CCCCC#N)N1CC(NC(CCN(c2ccc(Cl)cc2)C)=O)C2C1C2 C(=O)(C(F)C(F)(F)F)N1C(CNC(c2cc(C(N)=O)ncc2)=O)CC1 N1(C(C2CC(F)CN(C(c3ccnnc3)=O)C2)=O)CCc2c(F)cccc2C1 c1(C(CNC(c2cnn(C3CCC3)c2)=O)NC(CCSC)=O)cccc(C)c1 CCC(C)C(O)C(=O)NCCCCCCNC(c1ccc(F)cc1F)=O c1(-n2c(C(N(CCNC(CC3C(C)OCC3)=O)C)=O)cnc2)ccccc1F Cc1nn(C2CC2)cc1C(=O)NC(C1CCN(C(=O)CCCC2CCCC2)C1)C N1(C(CCC(C)OC)=O)CC2OCCN(C(c3ccc(C(C)C)nc3)=O)C2C1 N1(C(CC2CCN(C)C2)=O)CC=CC(NC(c2cn(CC(N)=O)nn2)=O)C1 N1(C(C(C=C)O)=O)CC2(C1)CN(C(c1ncccc1OC(F)F)=O)C2 c1(-c2cnc(C(=O)Nc3n(C)ncc3I)nc2)ccc2c(C3CC3)n[nH]c2c1 C(=O)(C1CCCc2ccccc21)NCCN(C(CC(C=C)CC)=O)CC1CC1 C1(CNC(C(CC)C(C)C)=O)CN(C(c2cc(N)c(C)cc2C)=O)CC(C)(C)O1 N1(C(C2(C)CC2(F)Cl)=O)CCOC(C(c2ccccc2)NC(=O)C=CC=C(Cl)Cl)C1 c1(C(N2CCCC(C(=O)Nc3cc(Cl)ccc3I)CC2)=O)n[nH]c2c1CCCC2 N#Cc1ccc(C(N2CC3(C2)SCCC3NC(=O)CCN2CCC2)=O)c(F)c1 CC1CC(N=c2[nH]nco2)CN1C(=O)C1CCCc2nncn21 Cc1cc(-n2nc(C3CCC3)nc2-c2cc(S(C)(=O)=O)co2)nc2ccccc12 CCS(=O)c1ccccc1C(=O)N(CCCCCNC(c1cc(F)c[nH]1)=O)C N1(CC(=O)NCCCNC(CC2(C)CCC2)=O)CCCC1=O C(c1cc(F)c(O)c(F)c1)=CC(=O)NC1C(OC)C2C1CCC2 c1(C(=O)NCc2c(C3CCN(C(C(C)=O)=O)CC3)cccc2)cc(C)cc(Cl)n1 N1(C(c2c(C(C)=O)c[nH]n2)=O)CCC(NC(C2(CC(C)C)COC2)=O)C(F)C1 c1(C(=O)NC2CCC(NC(C3CC(=C)C3)=O)C2)ccc2c(c1)nc(C)c(=O)n2C C1(NC(C2CC(SC)C2)=O)CN(C(c2ccccc2OCCF)=O)CC1(C)C N1(C(N(C2CCCC2)CCCC)=O)C(C)CC(C)CC1C.c12cccc(c1)N2 CC1(CN=c2[nH]nco2)CCCN(C(=O)C(c2cccc(Br)c2)O)C1 Cc1n[nH]c(C)c1CNC(c1cc(CCNC(=O)CC=CC(C)(C)C)on1)=O N1(C(C2(F)CCN(C)CC2)=O)CC2CCCC2(NC(=O)CCn2cccn2)C1 c1(N2CCCC(F)C2)nc(N2CCOc3ncccc3C2)c2c(n1)CSC2 C1(NC(=O)CN2CCCC2CO)CCCCN(C(=O)CC2=CCCCC2)CC1 CC(C(C)C(=O)NC1(CO)CCN(C(=O)C(C)CC(N)=O)CC1)S(C)(=O)=O c1(C(=O)NCC2(CCNC(c3cnc(OC)s3)=O)CC2)csc2c(O)ccnc12 CC1(C)CCC(C(=O)NC2CC(CF)C2)CN1C(C1(O)CCCC1)=O C1(CSC)CN(C(c2cnc(N)cn2)=O)C(C)(C)C1 C1(CNC(Cc2cn(C(C)C)nc2)=O)CCCCN(C(=O)CC=C(Cl)Cl)CC1 n1(CC)cc(NC(=O)C(O)CNC(=O)CC2CCN(C)CC2)ccc1=O c1(C(N2CCCC(C(N3CCN(C(=O)C4CC4)CC3)=O)C2)=O)cnnc(Cl)c1 N1(C(c2cnc(CCOC)s2)C(=O)NCCC)CCCC(O)C1.c1(C)ccccc1C N1(C(C(CC)(F)F)=O)CC2(CNC(=O)C(C)=CC(C)(C)C)CC2(C(F)(F)F)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1(CO)CCCN(C(C2C(C)C2)=O)C1 Cc1cc(C(=O)NC2CCN(C(=O)CC(=O)N(C)C)CC2O)c2ccccc2n1 c1(CN2CC(C(=O)NC3(CC)CC3)(CC)C2)cc(Cl)cc(Br)c1F C(=O)CCC(C)CN(C)C.C1(=O)COCC(=O)NCCN1CC.CN C(C(C)(C(=O)NC(C1CC(NC(c2cccnc2O)=O)C1)C)OC)OC C1(NC(C)=O)CCC(C(=O)NCC2(C)CCN(C(=O)C(C)C3CCOC3)C2)CC1 c1(CC(N2CCN(C(c3c(OC)cnc(F)c3)=O)CC2)=O)cnn2ccccc12 C(=O)(CCCCC#N)NCC(CC(=O)NCCN1CCC(OC)C1)C C12(C(N(CC(CNC(C=C(C)C(C)C)=O)O)C)=O)CC(C)C1C2 c1(NC(CC(C)N(C(C(C)S(C)(=O)=O)=O)C)=O)cnc2ccccc2c1 CC1CCN(Cc2c[nH]nc2-c2ccccc2Br)C(C(C)(C)C(=O)O)C1 N1(C(=O)OC(C)(C)C)CCCCC1C1CCCN1CC(C)CN(C1CCC1)C N1(C(CCNS(CC)(=O)=O)=O)CC(NC(C2CCCC23CC3)=O)C(F)C1 c1(CC(=O)NCCN(C(=O)COC2CCCOC2)CC)ccccc1C(F)(F)F C1(CCC)(NC(C2CC(C)N(C)C2)=O)CCCN(C(c2c(C)noc2N)=O)C1 c1(CC(=O)NCC2N(C(C3(OC)CCOC3)=O)CC2)c(C)nc2n1CCCC2 c1(CC)ccc(C(N2CC(F)CC2C(=O)N(CC)CC2CCCN2C)=O)c(C)c1 C1(CNC(c2cc(O)ccc2Br)=O)CCN(C(c2cnccc2Cl)=O)CC1(F)F C1(NC(=O)CN2CCCC2)CC2CCC1(CNC(c1ccc(F)cc1Cl)=O)C2 c1(CCC(N2CCN(c3nc(C)c(C)[nH]3)CC2)=O)c(F)ccc(Cl)c1F C1(CNC(c2nc(CC)oc2C)=O)CCCC2(CN(C(C3CC3CF)=O)C2)O1 N1(C(C(c2ccnn2C)C)=O)CCC2CN(C(c3nnc(O)cc3O)=O)CC2C1 C1C(N(C)C)C(=O)NC2(CCC2)C(=O)N1.C1(CSC)CCCSC1 C1(C(C)C)C(=O)N2C(=O)CCC2C(=O)N1.c1(CNCC(=O)OC)ccccc1Cl Cc1ncnc(N2CCOCC(CNC(C3(O)CC3)=O)C2)c1C#N C1(O)(C(=O)OC)CC2(CCCN(C3CCN(C(c4ccccc4)=O)C3=O)C2)C1 N1(C(CSCCCC)=O)CCN(C(=O)CCC2CCC(=O)C2)CCC1C Cc1ccc(C(=O)NCC2(C(=O)NCC3(C)CCN(C)C3)CC2)n1C C1(CNC(c2c(SC)cc(F)cc2)=O)C(C2CC2)CCN1C(c1csc(O)n1)=O Cc1cc(C(N2CC(NC(C3CN(C(C)C)C3)=O)CC(C)C2)=O)ncc1N N1(CC(C)NC(C2C(C)CCO2)=O)CCN(C(c2ccc[nH]2)=O)CC1 C12(CNC(c3c(C)con3)=O)CCC1CCN2C(=O)CCc1cccnc1Cl C1(NC(=O)CCCN2CCCCC2)CCOCC1NC(C1C2COCC12)=O C1(C(=O)NC(C#C)CC2CC2)CN(C(=O)COCC2CCCO2)CC1N(C)C CC1=NOC(C(=O)NCCN(CC(C)O)C(=O)CC2CCCC2)C1 C1(NC(c2ccc(C)n2C)=O)CCN(C(=O)C(C)(C)n2cc(Br)cn2)CC1CO C(=O)(C#CC1CCCCO1)N1CC(CNC(c2ccc(C)cc2F)=O)OCCC1 CCCCCCCCCC(=O)NCC(CNC(=O)Cc1ccns1)CO Cc1cc(C(N2CC(NC(c3cnn[nH]3)=O)CC2C)=O)c(C)c(C)c1 c1(NC(C2(NC(C3(C#C)CCCC3)=O)CCN(C)C2)=O)cc(CC)ccc1C CC1(C)CC(CNC(=O)Cn2cccc(N)c2=O)CN1C(=O)COC1CCCC1 n1(CC)ccc(C(=O)NC2CCCC(CN(C)C(c3cnsc3)=O)C2)cc1=O C12(NC(c3ccc(C)n3C)=O)CN(C(c3cn(C)c(O)n3)=O)CC1CS(=O)(=O)C2 n1(CC(=O)NCC(C(C)C)NC(C(COC)OC)=O)cc(C(F)(F)F)ccc1=O CCCC(C(=O)N1CCC(C)C1CNC(c1cn(C)nc1OC)=O)N(C)C C(=O)(C(O)CC(C)(C)C)N1C(CNC(C2(C(F)F)CC(=C)C2)=O)CC2(CC2)C1 C1(CC(=O)N(C)CC2(CNC(=O)CCn3cccn3)CC2)COC(C)(C)C1 c1(C(C)C)cc(C(=O)NCC(C2CC2)N(C(=O)COCCCF)C)no1 c1(C(N2CCC(C)(CCNC(Cc3scc(C)c3)=O)C2)=O)cn2cccnc2n1 N#CC1(c2ccccc2)CC2(CN(C(c3ncc(Br)cc3Cl)=O)C2)C1 CCCCC(C(=O)NCC1(NC(=O)CCC2CCCOC2)CC1)NC(N)=O S(=O)(=O)(CC(=O)OC)NCC(CC(=O)NC(c1ccccc1)CC)O N1(C(=O)CN2C(=O)CCC2=O)CCC2(CC1)CC(NC(=O)CC(O)C1CC1)CO2 C1(C(=O)NCC2(O)CN(C(C(n3c(C)ccn3)C)=O)C2)CC2(CC2)CO1 N1(CCN(C)C(C2(N(C(=O)CN3CCCC3=O)C3CC3)CCC2)=O)CCOC1=O c1(C(=O)Nc2ccc(C(N)=O)cc2)cc(Cl)ncc1Nc1cnc(O)nc1O C1(C(N(CC(C(C)C)C)C)=O)COCCC1NC(c1cn[nH]c1)=O c1(C(=O)NC(CCCC)CNC(=O)CC(=O)NCC2CC2)ncnc2c1CCC2 N1(C(C(CN(CC)CC)F)=O)CC(NC(=O)C=C2CCN(C)CC2)CC(O)C1 C1(C(N2CC(OC)C(F)C2)=O)(NC(=O)C(C(C)C)SC)CCC(C)(C)C1 c1(CC(=O)NC2C=CC(CNC(C3(C=C)CC3)=O)C2)ccc(N)c(OC)c1 c1(C(N(C)C)C2CC2)cn(CC2CCN(C(C(C)(C)C(F)F)=O)C2)nn1 Cc1ccc(O)cc1C(=O)NC1C2CCC1N(C(=O)CC1CN(C)C1)C2 C12(C(=O)NC(C)(C)CCCNC(=O)CC3(C(F)(F)F)CCC3)CCCC1C2(F)F N1(C(C23CC(CN(C(C4(Cl)C(C(C)=O)C4)=O)C2)C3)=O)CCC(F)(F)C(F)C1 N1(C(CCCC(C)(F)F)=O)CCC2CCN(C(c3cnc(S)[nH]3)=O)CC2C1 N1(c2n(CC3(C(=O)OC)CC=CCC3)nnn2)CCc2sc(Cl)cc2C1 N1(C(COCCCC#C)=O)CCOC2(CCN(C(c3cnc[nH]3)=O)CC2)C1 C=CCC(C)C(=O)NC1CC12CC(NC(c1ccc(OC(C)C)cn1)=O)C2 N1(C(C)C(=O)NC(=O)NC2CC2)CCCC2(CNC(=O)C2)C1 c1(OCC(=O)NCC2CC2NC(c2coc(Cl)n2)=O)ccc(F)c(Cl)c1 c1(NC(C)=O)cc(Cl)ccc1C(=O)NCC1CC(NC(C23CC4CC2C3C4)=O)C1 C1(C(=O)O)CN(C(=O)CCC2CC2)CC12CN(Cc1ccc(Br)c(F)c1O)C2 c1(NC(CCCC)c2nnnn2CCC(=O)OC)ccc(C(=O)OC)cc1C N1(C(C2C(c3cn(C)nc3)C2)=O)CCC(C2(NC(=O)CC3(C)CCCO3)CC2)C1 C(C(CCO)N=c1[nH]c(N2CCN(C)C(C(F)(F)F)C2)nc2ccccc12)OC C1(COC)CN(C(=O)Cc2ccc(OCC(F)(F)F)cc2)CCN1CC(C)C c1(CC(=O)NCC=CCNC(CCCOC)=O)csc2c(Cl)cccc12 N1(C(C(C)C2CC2)=O)CC2(COC(CNC(c3ccc(=O)oc3)=O)C2)C1 c1(C(=O)NC2(CC)CN(C(C3(C)CC4C=CC3C4)=O)C2)ncnc(O)c1F c1(OC)nc(C(=O)NC(C)C(C)(C)NC(c2cc(CCO)on2)=O)co1 C1(NC(COC(CC)C)=O)COCCC1NC(c1ccnc(C(C)C)n1)=O C(CC(=O)N1CCC(C)(C)C1CNC(=O)COC1CCCC1)(C(F)(F)F)OC c1(CC(=O)C(N2CC3C(NC(c4cc(C5CC5)[nH]n4)=O)C3C2)=O)ccccc1Cl Cc1ccc(F)cc1CN1CCN(C(c2cscc2F)=O)CC1 C1(CNC(c2ccn(C(C)C)n2)=O)CC2CCC1N2C(=O)CC1C=CS(=O)(=O)C1 C12(NC(=O)Cn3cc(Cl)cn3)CCN(C(=O)CCc3cc[nH]n3)CC1C2 CC1CC(NC(c2nn(C)cc2Br)=O)CN1C(=O)CCOCC1CC1 c1(C(=O)NCCCC(C)NC(=O)CC2CC3(CC3)CO2)cn2cccc(F)c2n1 C(C1C(C(N2CCCC(CNC(c3ccnc(CO)c3)=O)C2)=O)C1(C)C)=C(C)C N1(C(C2(CC#C)CCC2)=O)CC(C)OC2(CCN(C(C3CN(C(C)=O)C3)=O)C2)C1 N1(CC(N2C(CC(=O)NCC(C=C)O)CCC2)=O)CCOCC1=O N1(CC)C(C)CN(C(c2cccc(Br)n2)C(=O)NC2CC(F)(F)C2)CC1C c1(C(N2C3(CNC(c4ccn(C)c4)=O)CCC3CC2)=O)ccc2nnc(S)n2c1 c1(OC)cccc(C(=O)NCc2cn(C3CN(C(C4(SC)CC4)=O)C3)nn2)c1 Cc1cc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CCCC(=O)O3)=O)C2)cc1Cl c1(C(N2CCCC(NS(CC)(=O)=O)C2)C(=O)NC)cc(OC)c(OC)cc1Cl CCCC(F)(F)C(=O)NC(C1CN(C(c2oc(C(F)F)cc2C)=O)CCO1)C N1(C(CNC(=O)OCC=C)=O)CCC(N(C)C(c2[nH]cnc2CC)=O)C1 C12(NC(=O)NCc3onc(C(=O)OCC)n3)CC1CN(Cc1ccccc1)C2 c1(CC)nc(C(=O)N(CC(C)O)CCNC(=O)C(F)CC)c(C)o1 C12CC(=O)N(C1)CNC2=O.CCCC(CC)NC(c1c[nH]nc1C1CC1)=O C1(CNC(C(COC)C)=O)(CO)CCN(C(=O)COc2cccnc2C)CC1 C1(CNC(=O)CCc2nc3ncccn3n2)CCC2COCCC2C1 N1(C(c2cc(NC(=O)OC(C)(C)C)ncc2)=O)CC2CCCN2CC1C n1(CC(N2CC(NC(=O)CSC3CC3)C3C2C3)=O)ccc(O)nc1=O Cn1nc(CNC(=O)CCC2CC2)c2c1CCN(C(C1(C#N)CC13CCC3)=O)C2 CC1(C)CNCCC1CNC(=O)CNC1CCCC1Oc1ccccc1 c1(C(N2CCN(C(COCC)=O)C(C)C2C)=O)cc([N+](=O)[O-])cnc1C N1(C(C=C(C)C)=O)CCCC1C1(NC(=O)COCCc2ccc(Cl)s2)CC1 c1(C(N2CC(C(C(=O)NCC(C3CCC3)OC)O)C2)=O)ccc(F)cc1 C1(C(=O)NCCNC(C(C)C)=O)CCC(O)CN1C(c1ccc(=N)[nH]n1)=O Cc1ccc(C2(O)CCN(C(CC3CCC3)C(=O)NC3CCCC3)C2)cn1 N1(C(C(C2(O)CCC2)NC(c2c(C)c(=O)cc[nH]2)=O)=O)CCC2(CC(F)C2)C1 Cc1cc(C(=O)NC2CC(NC(=O)CCc3ccncn3)C23CCC3)ccc1F Cc1oc(C)c(C(N2CCN(C(c3ccc(F)o3)=O)CC2C)=O)c1C CC(C)CCC(=O)C(=O)NCC(N1CCC(C)(C#N)CC1)=O.N1CCCC1=O CCC(C)CC(C(=O)NCC(F)Br)NC(c1sc(O)nc1C)=O c1(C=O)cc(C)n(C(C)CC)n1.c1(C(C(=O)N(C2CCC2)CC)C)ccc(C)s1 c1(CC)cc(C)c(C(=O)NCC2C3CN(C(=O)CCc4nccn4C)CC23)o1 c1(C(N2CC(c3ccccc3)CC2(C)C)C(=O)NC)cc([N+](=O)[O-])c(C)cc1C c1(C(=O)NC(C2CCN(C(C(C)=C(C)C)=O)CC2)(C)C)cc2cccc(Cl)c2o1 C1(OC)CCC(C(=O)NCCC2(NC(c3ccoc3C(C)C)=O)CCC2)C1 C1(NC(CNC(=O)C(C)SC)(C)C(=O)OC)CC2COCC(C1)C2 N1(C(c2ncccc2Cl)=O)CCC2CN(C(=O)Cn3ccnn3)CCC2C1 c1(C(=O)NC(CCCC)CNC(=O)COCCF)cccc(C(F)F)c1OC Cc1ccc(C(=O)NC2CC(NC(c3cn[nH]c3)=O)C(O)C2)cc1 CCC(CCC(=O)N1CCOC(CC(C)C)C1)NC(=O)C(CN(C)C)C(C)C C(=O)(CC(C)CC(F)(F)F)N(C1CCN(C(C2CC2C2CC2)=O)CC1)CC N1(C(CN(CC(C)(C)C)C)=O)C2CC1CN(C(=O)CC1(O)CCCCC1)C2 CC(CC(=O)NCC1(F)CC(NC(C2CCCN2C(N)=O)=O)C1)c1ccccc1 CC1(C)CCC(N(C(c2ccc(Br)cc2-n2cncn2)=O)CC2CCC2)CC1 Cc1cc(O)ncc1C(=O)NCCC1CN(C(=O)C=CC(C)C)CC(C)O1 c1(N(C(CCNC(CNC(=O)OC)=O)C)C)nc(C(C)(C)C)ccc1C#N c1(NC(CC(C)O)C)ccc(NC(c2nnn(-c3ccccc3)c2CN)=O)cc1 N1(C(c2scnc2Cl)=O)CCN(C(=O)COCC2CCCO2)C(c2cn[nH]c2)C1 Cc1cccc2nc(C(N3CCCC3C(C)NC(c3cnc(O)s3)=O)=O)cn12 c1(C(N2CCCC(NC(C3(C)C=CCCC3)=O)C2)=O)cc(C(F)(F)F)cc(N)c1 CCC(C)(CCNC(c1ccnnc1)=O)NC(=O)Cc1ccn(C)n1 C12(CNC(C(C#C)(C)C)=O)CCC(CN(C(=O)CCCC(F)F)C1)C2 c1(-c2nc(CCC(=C)C)on2)ccc2cnccc2n1 Cc1cc(C(N2CCN(c3ccccc3OC(F)(F)F)CC2)=O)c(S(N)(=O)=O)s1 c1(C(N2C(C(C)(C)CNC(c3ccon3)=O)CCC2)=O)ccc2scnc2c1 C1(NC(CCC)(c2nnnn2C2(C)CC2)C2CC2)CCCCC1NS(=O)(=O)CC C(C(CC(F)(F)F)NC(C1(CC)CC1(F)F)=O)NC(CC(=O)NCC#C)=O C(=O)(CC(C)C(C)C)NC(CCSC)C(=O)NCCN1CC2CC2C1 Cc1nc(N2CC3(CCCC3NC(c3csc4nccn34)=O)C2)ccc1C#N c1(NC(C)COC(F)F)ccc(S(=O)(=O)NCc2nn(C)nc2Br)cc1Cl n1(C(C)C)cccc1C(=O)NC(c1ccccc1)C(=O)NCC1CSCCO1 CCCC(CNC(c1ccc(SCC)cc1)c1nnnn1C1CCC1)CCO CC1(C)CN(C(c2ccc(F)c(CO)c2)=O)CCC1NC(C1(C)CC2CC2C1)=O C1(C(F)F)(CNC(C2CC(F)(F)CS2)=O)CCN(C(=O)COC2CC2)C1 C1(CNC(C(C)(C)NC(=O)OC)=O)CN(C(=O)COC(C)=O)CCC12CCOC2 N1(C(c2cc(OCC)n[nH]2)=O)CCOC(C)C1C(=O)NOC(C)CC O=C(C1CCc2nccn21)N1CCC(C(N2CC3OCCC3C2)=O)C1 n1(CC(=O)NCCC2(C(=O)O)CCC2)ncc(O)nc1=O.[nH]1cc(Br)cn1 C1(C)(NC(c2cc(CNC(C(C)=C(C)C)=O)nn2C)=O)CCCCCC1 N1(C(C2(C#C)CCN(C(C3OC4CCC3C4)=O)C2)=O)CC(C)(C2CCC2)C1 N1(C(CN(C(=O)OC)C)=O)CCCC(C)C1CNC(C1CN2CCC1CC2)=O C1(NC(C(C)OCC=C)=O)CN(C(=O)CCc2nnc(C)n2C)CC(C)(C)C1 CS(=O)c1ccccc1CC(N1CC(OCCNC(C2(C)CCOC2)=O)C1)=O CC1C(NC(=O)Cn2ccsc2=N)CCN1C(=O)CCC1CCCN1C c1(N(C(=O)NCC(C(CC)CC)OC)C)cnc2ccccc2n1 c1(C(=O)NC(C2(O)CN(C(C(CC3CC3)OC)=O)C2)C)ccc(SC(F)F)cc1 c1(CC(=O)NC(C2CCN(CC(C)C)CC2)C)ccc2ncoc2c1 N1(CCCSc2nc(=N)[nH]c(Cl)c2N)CCc2ccccc2C1 N1(C(Cc2c(C)cccn2)=O)CCN(C(c2cnn3c2N(C)CC3)=O)CCC1C C1(NC(C2(CCC)CCC2)=O)CC(O)CN(C(c2cc[nH]c2C2CCCC2)=O)C1 c1(CC(=O)NC(C2N(C(c3ccc(CC)[nH]3)=O)CCCC2)C)cc(F)ccc1F C(CC(C)C)(C(=O)N1CCC(O)(C(C)NC(=O)CCc2cnoc2)C1)NC(C)=O c1(C(C)(C)C)[nH]cnc1C(N1CC(c2cn(Cc3cnns3)nn2)C1)=O c1(CCC(N2C(CNC(=O)CC3(O)CCCC3)CCC2)=O)ccnc(Cl)c1 c1(SC)cc(C)c(C(N2CCOC(CN(C)C(C3(CO)CC3)=O)C2)=O)o1 c1(NOC(c2ccc(Br)o2)c2nnnn2CCOCC2CC2)cnc2c(c1)CCC2 C1(NC(C2CC(C)C2)=O)CS(=O)(=O)C2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 CC1(C)CCC(CNC(=O)C(Cn2ccnn2)NC(c2ccc(C#N)o2)=O)OC1 c1(C(N2CC(C(C)NC(c3nc(OC)c(C)s3)=O)C2)=O)cc2n(c1)CCC2 Cc1cc(=NC(=O)C(=O)NCC2(F)CC(NC(C3OCC3(C)C)=O)C2)[nH]o1 CC1CCCCC1(CNC(=O)CCCC(N)=O)NC(=O)Cc1cnsc1 N1(C(C(C(C)C)c2ccc(F)cc2)=O)CCC(F)C(NC(c2ccoc2Cl)=O)C1 c1(C(=O)NC(C)C)cc2c(s1)CCCC2.n1(C(COC)COC)cc(C)nn1 c1(C(N(CCCNC(C2(F)C(C)C2)=O)C2CC2)=O)ccc2c(c1)CCC(C)(C)O2 CC(C)C(C)CC(=O)N1CCCCC1CN(C(=O)CN(C)C(=O)C1CC1)C C12(NC(Cc3ccc(OC)cc3Cl)=O)CCCC1N(C(c1cc(C)co1)=O)CC2 n1(CCNC(C23CC(F)C2C3)=O)cc(C(=O)O)nn1 C1(N(C(=O)CCNC(=O)C(=O)NC2CCOC2)C(C)C)CCCCC1 c1(C(C(=O)NCC(C)NC(=O)C=CC(C)(C)C)(C)C)cccc(OC(F)F)c1 C1(CC(=O)NCCN(C(=O)Cc2cc(C)[nH]n2)CC)CS(=O)(=O)C1 C1(C)(COC)CN(C(=O)N(C23CC4CC2C3C4O)C)CCO1 C1(CNC(C(N)=O)=O)C2CCCC1N(C(=O)Cc1cnccc1Cl)C2 N1(C(C2=NOC(C)C2C)=O)CCCCC2(CCN(C(C3(F)CCOCC3)=O)C2)C1 Cc1n[nH]c(C)c1C(C)NC(=O)CC=CCNC(c1csc(=N)[nH]1)=O c1(C(N(CC(C)O)CCNC(C2(CO)CCCC2)=O)=O)sccc1S(=O)(=O)C(F)F Cc1nc(CC(N2CCCC(N(C(=O)C(c3ccccc3Cl)O)C)C2)=O)[nH]c1C C(Cc1ccccc1)(C(F)(F)F)N(C)CCc1ccccc1N C12(CNC3(c4nnnn4-c4ccc(F)cc4)C(=O)NCC3)CCCCC1C2(F)F C1(C(N(CC#C)C(C)C)=O)CCn2cnnc2C1 C(=O)(C(C)CC(=O)OC)NC1(CC(=O)N(C(CO)CO)CC)CC1 C(C)(CCC(=O)N(C1CCOC1=O)C)NC(Cc1cc(C)[nH]n1)=O N1(C(C2C(C#N)C2)=O)CC2CCCC1C2CNC(c1conc1C(Cl)Cl)=O c1(C(=O)NCCC(C)NC(CS(=O)(=O)NCC)=O)nnc2ccccc2n1 c1(C(N2CC(CNC(C3(CC)COC3)=O)N(C)CC2)=O)cc2n(n1)CC(F)C2 N1(C(c2c(C)csc2)=O)CCCCC(C2CN(C3CCN(C4CCC4)C3=O)C2)C1 c1(CC2CC2)c(Cl)cccc1Cl.n1(CC(=C)C)c2nnc1N(C)CC1CCN2C1 c1(C(C(=O)NC2CCCC2)N(CCC)C2CC2)cc(C2CC2)cc(C)c1 c1(CC)nc(C)c(C(=O)NC2CC3CN(C(=O)C=CC(C)(C)C)CC3C2)c(C)n1 c1(C(c2ccccn2)CNC(N2CCN(CC)CC2)=O)ccc(C)cc1C C1(CNC(=O)CSc2cnc(O)nc2O)C2CCCCCC12 Cn1ncc(Cl)c1CC(=O)NCC(C)(C)CCNC(=O)C=Cc1cnc[nH]1 C(=O)(CC(F)(F)Cl)C(=O)CC1(O)CCCCC1.C1(N)CCNC1 N1(C(CN(c2cn(C)cn2)CC(=O)NCCCCNC(N)=O)=O)CCCC(C)C1.CO N1(C(CS(=O)(=O)NCC)=O)CCOc2ncc(-c3ncco3)c(C)c21 c1(N(CC(=O)NC)CC(=O)NC2CC3CC3C2)ncc(C(F)(F)F)cn1 C1(C(C2(C(F)(F)F)CC(C)(C)C2)N2CCC(C=O)CC2)C2CCCCCC12 N1(C(CC2=NNC(=O)C2)=O)CCC(C2CN(C(=O)CCN3CCCC3=O)C2)CC1 c1(C(=O)NCC(CC)NC(=O)C(C)(O)c2ccccn2)cc2n(n1)CCOC2 CCC(CCC(=O)NC(C)CCC(C)C)NC(C1CC(F)C1)=O c1(C(=O)NCC2N(C(C(C)OCCC=C)=O)CCCC2)ccc(F)c2[nH]ccc12 N1(C(C=C(C)Cl)=O)CCC2(CC1)COC(CNC(c1cc[n+]([O-])cc1)=O)C2 c1(C(N2CC(CNC(c3c(C)[nH]cc3)=O)C(C)(C)C2)=O)cc(F)cc2ccoc12 C(=O)(CCC(C)(C)NC(=O)CC1CC(=O)NC1=O)NCC1N(CC)CC1 N1(C(C2ON=C(CC)C2)=O)CCCC(C2CCN(c3ncc4c(n3)COC4)C2)C1 C(CCC[Si](C)(C)C)N(C)C(c1cc(-c2nc(C3CC3)no2)oc1Br)=O C1(CNC(N(C)Cc2nc(C#N)cs2)=O)NC(=O)CC1(C)C C(=O)(C1=CCCN(C(C23CC(C2)C3)=O)C1)Nc1c(C)ccc(I)c1C C12(C(N(C(CNC(COCCCCCC)=O)C)C)=O)CC3CC(C(=O)N1)C2C3 O=C1CNc2cc(C(N3CC(NC(=O)C=C(Cl)Cl)C4CCCCC34)=O)ccc2N1 N1(C(CCOC(CC(C)C)C)=O)C2CCC1CN(C(C13CC(CCO1)C3)=O)C2 N1(C(C(CC)n2cccn2)=O)CC(O)CC1CC(=O)NC(C)CN1CCCC1=O c1(SC)ccccc1C(=O)NCCC(C)CCNC(=O)CCc1cnn[nH]1 CCC(CC)CCCNC(C1CCN(C(C2CC3(CC3)CO2)=O)CC1O)=O c1(CCC(=O)N(CC(N2CCCC2)=O)C(C)C)cnccn1.C1CC1 N1(C(C(=O)Nc2scc(-c3nc(C)sc3)n2)=O)CCC(C)(C)CC(C)(C)C1 N1(C(c2ccc(CC)[nH]2)=O)CC2CCCC2(CNC(=O)Cc2nnc(C)o2)C1 C1(C)(C(=O)NCCCN(C(c2c(C)n(CCO)nc2)=O)C)CC(C)OC(C)C1 C1(C(N2CCC(C(C(=O)NC(c3ncccc3F)C)(C)C)C2)=O)CC(=O)CCO1 c1(SCC)cccc(C(=O)NCCCc2ncccn2)c1 C1(CN(C(=O)CC(C)(C)C)C)CCCN(C(=O)CN(C)Cc2ccc(F)cc2)C1 c1(N2CC(OCCOC)OCC2)cc(C)[nH]c(=NC(=O)OC(C)(C)C)n1 C(CC(F)=C(F)F)NC(C(C1CC=CCC1)NC(c1c(CC)c[nH]n1)=O)=O C(=O)(CCCN(C)N=O)N1CCN(C(C2N(C(C)=O)CCC2)=O)CC1CC1CC1 c1(C(=O)NCC2C(NC(C(F)=CC)=O)CCCC2)ccc(P(C)(C)=O)o1 C12(CC(=O)N(C(CNC(C(=O)NCCNC(C)=O)=O)(C)C)C3CC3)CCCC1C2 C(=O)(C(C)C1CCCO1)NC(C1CCC1C(=O)NCCCOCCO)C c1(OC)ncc(C(=O)NCCOC2CCN(C(=O)CN(C)C(C)=O)C2)nc1C Cc1cc(=O)c(C(=O)N(C)CCOCCN(C)CCC2CCCC2)c[nH]1 C(=O)(CC1=CCN(C)CC1)NC(C1CN(C(C2CCCN2C=O)=O)CCO1)C N1(C(C2CCN(C(c3n(CC)ccc3)=O)C2)=O)CCCC(OC2CC2)C1 CC(=O)CCCC(=O)N1CCC(NC(c2nc(C)ccc2F)=O)CC1C1CC1 CC1CCCN(C(=O)C(N2CC(C)(NC(c3cccc(N(C)C)n3)=O)C2)=O)C1 c1(C(=O)NCC#CCNC(C(c2n(C)ccn2)(F)F)=O)cc(F)ccc1N c1(C(=O)NC(C2CCN(C(CCOC)=O)C2)C)ccncc1C(F)(F)F CC1(C(=O)NCC2(CN=c3[nH]nc(C(C)(C)C)o3)CC23CCC3)CCCC1(F)F N1(C(c2cnc(C(C)(C)C)s2)=O)CCC(CNC(c2cnc[nH]2)=O)C(F)(F)CC1 C(=O)(N=c1ccn(CC(F)F)[nH]1)C1(C(=O)OC(C)(C)C)CC(C(C)(C)C)C1 c1(CC(=O)OCC23OCCC(OC)(C2)C3)ccc2c(c1)OCCO2 C1(C)(OC)CCN(C(C2CCCC(NC(c3c(F)cccc3F)=O)CC2)=O)CC1 c1(OC)ccc(Cl)cc1C(=O)NC1CCN(C(C2CCCS(=O)(=O)N2)=O)C1 CC(C)(C)CC(O)CC(=O)N1CCCC1C=CC(=O)NCC1CCc2nccn21 N1(C(C=Cc2c(C)n(C)nc2)=O)CC(C)CN(C(c2cn(C)nc2Cl)=O)CC1C CC(C)CC(O)C(=O)N1CCC(C)(NC(c2cnc(=N)[nH]c2)=O)C1 c1(C(N2C(CNC(C(N3C(CC)CCC3)=O)=O)CC(O)C2)=O)cc(C)c(F)cn1 N1(C(C2COCCN(C(c3ccnc(OC)n3)=O)C2)=O)CC2(CCOC(=O)N2)C1 C1(CNC(C(C)NC(=O)NC)=O)CN(C(C2CN3CCCN2CC3)=O)CCCO1 CN1CC(C(=O)NCC2CCCN(C(c3cc[n+]([O-])cc3)=O)CC2)OCCC1=O c1(C(N(CCC)CCNC(=O)C=C2CCOCC2)=O)ccnc2cc[nH]c12 C=CCC(CNC(c1csc(CO)n1)=O)NC(C1(Cl)CC1(C)C)=O N1(C(C2C(=O)NCC2)=O)CC2(C1)CN(C(=O)C(F)(F)C=Cc1ccccc1)C2 c1(OC)cc(CN2CCC(NC(c3c(Cl)cccc3Cl)=O)CC2)ccc1C(F)F N1(C(c2c(OC)scc2)=O)CCN(C(c2coc3c2COC3)=O)C(C)C1C Cc1cc(C(=O)NC(Cc2cc[nH]n2)C(=O)N(C)CC2CC2C)cc(C)c1 C1(NC(C(C)OC2COC2)=O)COC2(C1)CN(C(=O)CCCCCn1cnnn1)C2 C1(NCCn2c(N3CCCC(C)(CCC)C3)nnn2)CC(C)(C)CCC1O c1(C(N2CCCC(NC(C3(C)CCC(C)C3)=O)C2)=O)ccnc2ccsc12 c1(CC)ccnc(C(=O)N(C(C)CNC(=O)Cn2cc(C3CCOC3)cn2)C)c1 c1(CCC(=O)NC2CN(C(C(CC=C)CC)=O)CC2C)ccc2c(n1)NCCC2 C1(C(N2CCC(C(C)(C)NC(c3c(C)occ3)=O)C2)=O)OCC2COCCC12 C(C(CN=c1nnn(C)[nH]1)C(F)(F)F)N(C(C=C(C)CCc1ccccc1)=O)CC N1(C(CCOC(C)C)=O)CCCCC1C1CCCN1Cc1cc(Br)ccc1F N1(C(C)C)CCC(C(=O)NCc2ccc(N(C)C)nc2)CC1 C1(C(=O)NCC(C)C(F)F)CN(C(=O)C=Cc2ccccc2)CCO1 C(CC)(C(=O)NC1CC(CC(=O)N(C2CCC(C)C2)C)C1)=CCCC CN1CCC(C(N2CC3CCC3(CNC(=O)Cn3cnc(=N)[nH]3)C2)=O)S1(=O)=O CCC(C)C(CNC(=O)CC(C)(C)NC(=O)Cc1ccc(C)nc1)CO CN1CCC(C)(NC(N2CCCC2Cc2cc(F)ccc2F)=O)CC1 C(=O)(C1=CCCCO1)N(C1CC(NC(c2ccc(N)c(N)n2)=O)C1)C c1(OC)ccc(CN(C2CCCC2)C(C2CCC(n3ccnn3)C2)=O)c(OC)c1 n1(CC(=O)NC2CC(C(C(=O)NCC3(SC)CC3)F)C2)c(O)nnc1O C1(NC(c2ccn(CCO)c2)=O)CC2CC(C1)N(C(=O)CN(C1CCSC1)C)C2 C=CCCCCC(=O)N1CCC(C=CC(=O)NC(COC)C(C)C)CC1 C1(C(c2cn(C3CCCN(C(C)=O)CC3)nn2)OC(=N)O)Cc2nccn2C1 Cc1cnc(F)cc1C(c1nnnn1C)Nc1cccc(C(C)(F)F)c1C C1(NC2COC2)CC2(CC2)CN1C(=O)CN.CC(C)(C(F)(F)F)c1ccc(C(F)(F)F)cc1 c1(NC)cnc(C(N2CCC(C)(NC(=O)CN(c3ccccc3)C)C2)=O)cn1 C(N=c1cc[nH]cc1C#N)c1ccc(SCCNC(C2OCC(C)C2)=O)cc1 c1(C(CO)N(S(=O)(=O)CC2CC(n3ccnc3)C2)C)cc(Cl)cc(Cl)c1 CC1OCCN(C(C2CCCC3(CC3)C2)=O)C1C(=O)NCc1n[nH]cc1C1CC1 N1(C(CNS(N)(=O)=O)=O)CC2(NC(c3ccc(CCF)cc3)=O)CCCC2(F)C1 N1(CCC(=O)NCC(CO)NC(C(C)OCCCC)=O)CCNC(=O)C1 N1(CC)OCC(NC(=O)CCN(C(C2COCC(C)O2)=O)CC)C1=O N1(C(N2C(c3nc(C)c(C)s3)CCC2)=O)CC2CN(C(C)C)CC(C1)O2 C1(C(N(C2CN(C(CC(C)OC)=O)C2)C)=O)CC(=O)N(CCN(C)C)C1 C(CC(C(C)(C)C)NC(c1cn(C(F)F)c(C)n1)=O)N(C(CCOCCC)=O)C C1(C(=O)NCC2CN(C(c3ccoc3Cl)=O)C2)CC2CC(O)C(C1)C2 C(=O)(C(C)C(C)(C)C)N1CC=CC(NC(C(C(C)C)c2ccc(F)cc2)=O)C1 C1(CNC(C2CC2(F)F)=O)CC2(CCN(C(c3cc(=O)cc(Cl)[nH]3)=O)C2)CO1 CCC(CCCC(=O)NCC(C)(CC)C(N)=O)NC(c1nnsc1N)=O c1(NC)cc(C(=O)NC2CC(CNC(=O)C(F)C3CCOC3)C2)cc(Cl)n1 Cc1ncccc1C(N1CCC(C(C)(C)NC(=O)Cc2ccccc2C)CC1)=O Cn1nnc(C(N2CCC2C(=O)NCC23CCCCC2C3)=O)c1N CCC(O)C(C)C(=O)NCC(CC)(CC)NC(=O)CCc1nccn1C c1(CC)noc(C(=O)NC2CCN(CCNC(c3cnc[nH]3)=O)CC2)c1C c1(C(C(=O)NC(C)CC(C)NC(=O)CCc2ccon2)O)cc(F)cc(F)c1 C(=O)(CC(CC(N)=O)CC(C)C)NCC(CC)(C)NC(=O)CCOC1CCC1 C1(C2CCN(C(=O)C=CC(C)C)C2)(NC(CN2CCCCC(OC)C2=O)=O)CC1 c1(N2CC(C)CN(C)CC2)nc(NCC2(C)CCCC(F)(F)C2)c2ncsc2n1 CCC(C(=O)N1CCOC(CCNC(=O)CCOC(C)C)C1)C(C)(C)CC c1(C2CCC(OC(C)(C)C)C2)nc(-c2ccoc2)nn1Cc1cccc(Br)c1 C1(C(=O)NCCCN(C(C2C(C)=NOC2=O)=O)CCO)CC2(CCC2)CO1 N1(C(C(C)CCc2cccc(F)c2)=O)CC2CC(C1)C2c1nc(C(C)(C)C)no1 c1(C(=O)NCC2(F)CCN(C(c3cc(C)ns3)=O)CC2)c(C)sc(C)c1C#N CCC(CC(F)(F)F)NC(C1CN(C(=O)C=Cc2cc[nH]c2)CC1(F)F)=O N1(C(CC2COCC(C)(C)O2)=O)CC(O)(C2(CNC(C3(O)CC3(C)C)=O)CC2)C1 C(CC(=O)NC12CC(C1)N(C(c1ccnn1C1CCC1)=O)C2)(C(F)(F)F)OC c1(CCC)ccccc1S(=O)(=O)NC(C(C(C)C)C(C)C)c1nnnn1C C1(C2CC2)(C(N2CCC(C(C)NC(C3N(C(C)C)CCC3)=O)CC2)=O)CC=CC1 C1(O)(C(=O)NCCC2(CNC(C(n3cc(Cl)cn3)C)=O)CC2)CCCC(C)(C)C1 C(=O)(CC(C)N=c1cc(C)nc(N(C)Cc2ccc(Br)c(F)c2)[nH]1)NC C1(NC(C2CCC23CCC3)=O)CCCC12CN(C(c1cncnc1)=O)C2 c1(CC(=O)NC2C=CCN(C(C(n3cc(Cl)cn3)C)=O)C2)ccc2c(c1)CCO2 Cn1nccc1C1(NC(c2csc(Br)c2)=O)CC1 N1(C(C=CCC)=O)CCC2OCCN(C(=O)CCc3ccc(Cl)cc3F)C2C1 c1(N2CCC(NC(N(CC)Cc3cccc(Br)c3)=O)CC2)nc(C)ccc1C.C1CC1 c1(C(=O)NC(CNC(C(c2c(C)n[nH]c2C)C)=O)CO)cc2c(nn1)OCCS2 c1(OC)c(C(=O)NCCNC(=O)C(C)Cc2cnco2)cc(F)cc1F N1(C(c2c(C)nc(CO)s2)=O)CC(NC(C2(F)CC3(CCC3)C2)=O)CC2(CC2)C1 C1(COC(C(C)O)=O)CN(C(=O)CCCc2ccc(Br)cc2)C(=O)CO1 C(C(C)C(C)(F)F)NC(CC1C(NC(c2c(CC)cco2)=O)CCCC1)=O CN1CCC2(CC1)CN(CCCOC1CCCCC1)CCO2 c1(C(N2C(C(=O)Nc3scc(C)n3)CCCCC2)=O)c(Cl)cccc1[N+](=O)[O-] C(C(CC(=O)NC1COCC1O)OC)NC(c1c(OC)scc1)=O c1(C(C)C(=O)NCC2CCC2NC(=O)Cn2cc(Cl)cn2)c(F)cccc1F C(=O)(CC(COC)NC(C1CC(N(C)C)C1)=O)NC1CC(C=C)C1 C#CC1(O)CCN(C(C2CC3CC2CN(C(=O)CN2CC(C)(C)C2)C3)=O)CC1 Cc1ccnc(C)c1C(N1CCCC(N(C(=O)CCC(=O)C2CC2)C)CC1)=O C(=O)(C(C)(F)C(C)(C)F)NC1CCN(C(c2c(CCC)nco2)=O)C(C)C1 C1(C(N2CCN(C(CCCCC)=O)C(CO)C2)=O)CCc2cnn(CC)c2C1 C1(C(=O)NC(CC)CNC(=O)C(F)n2cccn2)CC2(CCC2)C1 CCC(CC(=O)N(CCNC(=O)C(COC)OC)CC1CC1)c1ccccc1 C(=O)(C1=NOC(C)(C)C1)NCC1N(C)CCN(C(=O)CCC2CC2(F)F)C1 c1(C(=O)OC)cccc(C(=O)NC2(CNC(=O)C(F)(F)c3ccnn3C)CC2)c1 c1(NC(C2N(C(C(c3cccc(Br)c3)(C)C)=O)CC=C2)=O)cc(O)c(Cl)cc1Cl N1(C(C(C(=O)OCC)F)=O)CCN(c2cccc(Cl)c2)CC1C c1(OC)cc(Br)c(C(=O)NC2CN(C(C34CCCN3CCC4)=O)C2)cc1F CC1(NC(C2CC(O)(CNC(=O)C(Cl)=CCl)C2)=O)CC(F)(F)C1 N1(C(CCC=CCCC)=O)CC=CC1(C)C S(=O)(=O)(c1cc(Br)ccc1Br)N1C(C(=O)Nc2ncc(Cl)nc2Br)CC(O)C1 c1(CC)ccc(F)c(C(=O)NC2CN(C(c3ccc(CO)o3)=O)C2)c1F c1(C(N(C2CCC(NC(=O)COc3cn[nH]c3)CC2)C)=O)nn(C)cc1S(N)(=O)=O C1(C(N(CCC(=O)NCC2(C)CC(O)C2)CC#C)=O)CNC(=O)CC1C N1(C(C2OCCN(C(Cc3nnc(C)s3)=O)C2)=O)CC2C(C1)C2(F)F Cn1nc(C(N2CCN(C(=O)CCc3cocn3)C(C3CC3)C2)=O)ccc1=O c1(OC)cc(NCC2CCC(NC(C3CCCC(C)C3)=O)CC2)ncn1 c1(C(N2CCCC(CCNC(C=C(CC)CC)=O)C2)=O)cc2ccccc2n1C CC(=O)C(C)(C)CC(=O)N1CC(=O)NCC1C(=O)NCc1cnc(N(C)C)nc1 CC1CCn2ncc(C(N3CCC(CCN(C(=O)C(C)(C)O)C)CC3)=O)c2C1 C1(C)(NC(CC(C=C)C)=O)CCN(C(=O)COc2ccc(Br)nc2)CC1 C1(O)(C(N2CC(CN(C(=O)COCP(C)(C)=O)C)OCC2)=O)CCCC(C)(C)C1 c1(C(N(CCOC)CCNC(=O)CC(C)c2cccnc2)=O)cc(C#N)c[nH]1 N1(C(C(CC)O)=O)CCC(O)(CCNC(c2cc(C)on2)=O)C1 C(CN=c1[nH]nc(C2CC2)s1)(C1CC1)NC(c1ccc([N+](=O)[O-])[nH]1)=O CC1CC2(CCC2)CN1C(=O)C(=O)NC1CCC(C)(C)CN1 N1(C(C(F)=CC)=O)CCN(CCCCCNC(c2ccc(COC)s2)=O)CC1 C(=O)(C(O)CCN1CCOCC1)NCC(C)N(C(CCCC)=O)CC CC1CN(C2CCCN(Cc3cn(-c4ccccc4)nn3)CC2)S(=O)(=O)C1 N1(C(CC2C(CC)C2)=O)CC2CC2(C(=O)N(CC(C)O)C2CC2)C1 C(=O)(C1=C(Cl)CCCC1)N1CCCC(C(C(=O)N(CC(F)F)CCC)C)C1 c1(CC(=O)NCCC(C)(C)NC(C#CC2(C)CC2)=O)c(F)c(F)cc(F)c1F c1(C(=O)NC(CC(C)NC(CS(CC)(=O)=O)=O)C)oc2c(Cl)cccc2c1C C(=O)(C(C)C(C)NC(=O)CC1CCCC1NC(c1cc(Cl)c[nH]1)=O)OC n1(CCCCOC)cc(COC(=O)Cc2ccn(C(C)C)n2)nn1.C1(C)CO1 C(=O)(C1=NOC2(CCC2)C1)NC(CC)CN(C(=O)C(C)(C(C)C)OC)C C12(C(N(CC(CC)NC(C3(CC)CCNC3=O)=O)C)=O)CC(C)(CO1)C2 c1(C(C(=O)NC(C)(C)CC)N(CC)CC2CC2)cccc2cnccc12 C1(C(=O)Nc2nc(C)c(Cl)cc2)CCCC12CCN(S(=O)(=O)c1cn[nH]c1)C2 c1(NC(C(CC(=C)Cl)NC(=O)C(=O)NCC)=O)c(C)cc(C)nc1O Cc1ccc(C(=O)NCCCN(C(=O)COC(C)=O)CCO)s1.CC(C)(C)C C(CC(C)C)(C(=O)N1CC(CCc2cn(CCc3[nH]cnc3C)nn2)C1)OC N1(C(c2c(CC)ncs2)=O)CCC(C(F)(F)F)C(NC(c2cscc2C#N)=O)C1 N1C(=NCCCCl)NCC1.c1(OC)ccccc1C(CF)N(C1(C)CC1)C C(=O)(CC(C)(O)COC(C)=O)N(CC)CC1CCCN(C(c2ccsc2)=O)C1 c1(C(=O)NC2CCN(C(Cc3ccc(C)cc3)=O)CC2)c(O)ncc2c1CCC2 c1(C(C(=O)NCCCC2(C)CC2)NC(C2CCOC2)=O)ccccc1 N1(C(CC2N(C(C3CC(=O)NC3)=O)CCC2)=O)CC2CCC(O)C(O)C12 N1(C(CSCCC)=O)CCCC(CCNC(c2[nH]ccc2CC)=O)CC1 N1(C(COC(C)(C)C)=O)CC2(CCC2)CC1CNC(C1CCCC1(F)F)=O N1(C(C2CCS(=O)(=O)N2)=O)CCC2CCN(C(=O)Cc3coc(C(F)F)n3)C2C1 C1(NC(CCOCC)=O)C2CCN(C(c3occ(C)c3C)=O)CCC12 Cc1nn(CC(N2CCC(C)(CNC(c3ccncn3)=O)C2)=O)c(C)c1[N+](=O)[O-] Cc1cc(F)ncc1N(c1nnc(C(C)(C)C)n1CC(=O)OC(C)(C)C)C N1(C(C2(CC#C)CCOCC2)=O)CCC2(CC1)CCN(C(C1CC(C)(C)O1)=O)C2 c1(NCC2(C)CCN(C(C3(CC)CC3)=O)C2)ncnc2c(F)c(F)ccc12 N1(CC=CC(=O)NC(C(C)NC(=O)CSCC(F)F)C)CCOCC1 CC(C(=O)N1CCC(CCCNC(=O)C(F)OC(F)(F)F)CC1)S(N)(=O)=O c1(C(N2CCCCC(N(C(C=NOC)=O)C)C2)=O)cc(C)c(Cl)cc1Cl C1(C(C)C)CN(C)CCN1C(c1nc(F)ccc1F)=O C1(NC(CCOCC(C)C)=O)CCCCN(C(=O)C=CC(C)C)CC1 c1(C(N(CCCN(C(C(C)C2CC2)=O)C)C)=O)cc(-c2cccs2)[nH]n1 c1(C(=O)NCC(C)(O)CNC(C2CCNC2=O)=O)ccc(O)c([N+](=O)[O-])c1 C1(NC(c2c(CN(C)C)cco2)=O)CCOCC1NC(c1ccccc1Cl)=O CC(C)(C)CC(O)C(=O)N1CCC(C(N2CC(N3CCC3)C2)=O)C12CCC2 C#CC1CN(C(=O)CC2CCCN(C(c3c(C)nsc3C)=O)CC2)CCO1 C=C=CC(C)C(=O)N(CC(C)(C)CNC(C1(C2(C)OCCO2)CC1)=O)C N1(C(c2cc[nH]c2)=O)CCCC2(CCCN2C(c2cnc(C3CC3)nc2O)=O)C1 C1(NC(C(C(C)C)O)=O)CCN(C(=O)CCOC2CCCC2)CCC1CO c1(OC)cc(OC)c(NC(c2ccc(OCC(F)F)cc2O)=O)cc1Cl c1(NC(C(CC)CCCCC)c2n(CC=C)nnn2)cccc2c1OCCO2 C1(C(=O)Nc2cc(COc3cnn(C)c3)on2)(CNC(C2C(=C)C2)=O)CCOC1 N1C(=NCC2CC2)NCC(=O)N1CC(F)F.Cc1ccc(C)o1.C(C)(C)(C)O C1CCCCC(=O)N1C1CC1.C1(C(=O)NCCCSC)Cc2nncn2C1.CCO C1(C(N(CC(=O)OC)Cc2ccc(Br)s2)=O)CC(O)C(F)C1 C=CC(C)CC(=O)NC(C)CCNC(=O)CC1CCC1 C(=O)(C1CCc2cccnc21)N1CC(NC(c2c(CC)non2)=O)C(N=[N+]=[N-])C1 n1(CC)nc(C(=O)NC2CCCC2C(=O)NCC2(C3CC3)CCC2)c(C)n1 c1(CC)c[nH]nc1C(=O)NCC(C(=O)NCC1CC(OC(C)C)C1)OC N1(C(C=CC(C)C)=O)CC2(CCC(CNC(C3(C)CNC(=O)C3)=O)O2)C1 c1(C(N2C(CC=C)(C(=O)NCC3CC3(Cl)Cl)CCC2)=O)cn(C)ccc1=O N1(C(CSC)=O)CC2CC(NC(C3(C(F)F)CCC3)=O)CC2C1 C(N=c1nc2sccc2c(NCCc2cncs2)[nH]1)c1scc(C(C)C)n1 N1(C(C(=O)NCc2c(C)cc(F)cc2)=O)CC2CC(N)CC1C2 C(=O)(C1=CS(=O)(=O)CCC1)NC(C)C(=O)NCCCc1ccccn1 C(=O)(CCCCCN(C)C)N(CCC(C)NC(=O)Cc1ccc(Cl)cn1)C c1(C(N(C(C)CNC(C2(O)CCC2)=O)C)=O)cc(Cl)nn1C CCCCC(O)CC(=O)NC1CC2C1CCN2C(=O)CC=C(C)C N1(C(CN(CC(=O)NC(C)C)C)=O)CC2CCCN(C(=O)CS(=O)(=O)NC)C2C1 C1(C)(C(N(CCC(=C)C)CC)=O)CN(C(=O)C(C#N)CC)C(C)(C)C1 C1(NC(C2CCC(=O)N2)=O)C2CCN(C(=O)CCc3ccc(C(N)=O)cc3)C12 c1(C(=O)NC(C2CCN(C(CCCC=C)=O)CC2)C)n[nH]c2ccc(OC)nc12 C1(NC(=O)Cn2cccn2)CN(C(c2ccccc2F)=O)CC1C(F)(F)F c1(OC)cc(C(=O)NC2CCCC2NC(=O)CCSC(F)(F)F)ccc1O N1(C(CC(C)CF)=O)CC2CN(C(=O)CC34CCCN3CCC4)CC2(C)C1 C1(S(C)(=O)=O)(C(=O)NCCCC(C)NC(=O)CC=CC(C)(C)C)CCC1 N(C(=NCCCF)NCC1(F)CC1)Cc1ccc(C2(C)CC2)o1 c1(C(=O)NCC2(F)CCC(CNC(c3occ(C)c3)=O)C2)ccc(C)c(Cl)c1N c1(C(=O)NCC2CN(C(c3cnc(C4CCOC4)s3)=O)C2)cccc2c[nH]nc12 CCCC(CC)CC(=O)N1CCN(C(C23CCC(F)(CC2)C3)=O)CC1C(C)C N1(C(CC2(C=C)CCC2)=O)CCC(NC(C2CC2c2cnn(C)c2)=O)C(C)C1 CCC(CCC(=O)NC(C)(CNC(C1CCCCNC1=O)=O)C(C)C)OC c1(C(=O)NCC2(C)CCCS2)ccncc1N1CCOCC1 CC(C)(C)C(=O)C(=O)NCCn1cc(C(=O)NCCN2CCC2)cn1 N1(C(C(C2CCCCCC2)OC)=O)CCOC2CN(C(=O)C(N)=O)CC12 Cc1nc(NCCCOC2CC2)cc(N2CCN(CC(F)(F)F)C(C)C2)n1 C1(C2CCCC2)(NC(CCCCCn2cc(CCSC)nn2)=O)CCNC1=O N1(C(C2CN(C(Cc3c(C)ncs3)=O)CC(C)C2)=O)CC2(CCC(O)CC2)C1 c1(C(CC)NCC(c2nnnn2CC)(C)OCCOC2CC2)c(F)cccc1F c1(OCC)c(OC)cc(CC(C)NC(c2n[nH]c(CO)n2)=O)cc1OCC C1(C)(C(N2CC3(CN(CC)C3)C2)=O)CN(C(C2CCCC2)=O)C(C)(C)C1 Cc1ccc(N)c(C(N2CCC(NC(=O)CCCCCF)C(C)C2)=O)c1F c1(CSC)cc(C)c(C(=O)NC(c2ccc(F)cc2)CNC(=O)C#CC2CC2)o1 N1(C(C2CC3(CC(=C)C3)C2)=O)CCC(C)(C)C(CNC(=O)CC(C)(C)O)C1 N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CC(NC(C2CC2[N+](=O)[O-])=O)CC2(CCC2)C1 C(=O)(C1=CC2(CCOC2)C1)NC1C2CN(C(Cc3c(C)ccc(C)c3)=O)CC21 c1(C2C(C(=O)NCC3CN(C(C4(CCC)CC4)=O)C3)C2)ccc(NC)cc1 C1(CNC(C(C)NC(CC)=O)=O)CCCCN(C(=O)CC2CC(=O)NC2=O)C1 C1(CC)COCCN(CCc2cn(C3CCOC3(C)C)nn2)C1 Cc1c(C(=O)N(CCCNC(C2(C)CC2)=O)C)nnn1C CN1N=C(C(=O)N2CC(O)(CNC(c3coc4c3COC4)=O)C2)CCC1=O CN=C(NCC(=O)Nc1cccs1)NC1CCN(C(c2ccccc2)C)C1 C(=O)(C1CCc2cc(Cl)ccc21)N(C)CCN(C(=O)C(O)CC(F)F)C c1(-c2cn(C(C)CN3CCC3C)nn2)cccc2ccncc12.c1(CC)cn(C)cn1 CON(CCC(=O)NCC=Cc1cccnc1)C(=O)CC(C)(C)n1ccnn1 C1(N(C(CC(C)=C(C)C)=O)C)CN(C(=O)COCCCC(C)C)CC1(C)C N1(C(C2CNC(=O)O2)=O)CCC2(CCOCC2)C(NC(=O)CC(O)C2CC2)C1 c1(C(N2CCCN(C(C(C=C)O)=O)CC2C)=O)cccc2cc(O)ccc12 N1(C(c2nc(CC(C)C)sc2)=O)CC2CC1CN2C(=O)CC1CCCN1C(C)C C1(CC(=O)NC2(CCOC)CCN(C(=O)C(O)CC(C)C)C2)CC(C)(C)CCO1 N1(C(C(C)CC(C)(C)C)=O)CC2(CCCCN2C(C2CC2CN(C)C)=O)C1 c1(CC(C(=O)O)NC(c2cccc(OCC=C)c2)=O)nccc2ccccc12 C1(NC(c2coc(C3CC3)c2)=O)CC2CCC1CN(C(=O)CC1(O)CCCC1)C2 CC1(C)CC(CNC(N2CCC(Cn3cccn3)C2)=O)OC(=O)N1 Cc1noc2nc(C(N3CC(N(C(=O)C(O)C4CCC4)C)C(C)(C)C3)=O)ccc12 CCC(C)(C)C(O)C(=O)N1CCN(C(=O)Cn2cnc(Br)c2)C(CF)C1 N1(C(c2occ(C)c2)=O)CC2CN(C(c3cccc(C(N)=O)c3)=O)C2C1 N1(C(C2CCC(CCCCC)CC2)=O)CCC(N=c2[nH]nc(C3CC3)o2)CC1C c1(C(=O)NCC2(OCC)CN(C(=O)C(C3CC3)OC)C2)ccnc(CC)c1 C1(COC)CCCN(C(=O)CSCCNC(=O)Cc2ncn(C)c2C)C1 CC1C(N(C)C)CCN1C(=O)CCc1cc(Br)c(Br)s1 C12(NC(C(C)NS(CCC)(=O)=O)=O)CCCC1CN(C(c1ccc(C)nn1)=O)C2 C1(NC(=O)CSC2CC2)CN(C(=O)CCC2CCCOC2)CCC1CO C(c1cc(Br)cs1)=CC(=O)NCC1(O)CC(CNC(C2CCCO2)=O)C1 c1(C(=O)NCCC2(NC(C(CCC)OC)=O)CCOCC2)cnc2cc[nH]c2c1 C1(CC#C)CN(C(c2ccc(COC)cc2)C(=O)NC(C)(C)C)CCO1 c1(SC)nc(Cl)c(C)c(=NC2CC(CNC(=O)C3=CCCC(C)(C)C3)C2)[nH]1 C1(C)(CNC(c2c(Cl)ccc(C)c2)=O)COCCN(C(=O)C(C)CC(F)(F)F)C1 C1(C(=O)NC(C)CCCCO)CCCN(C(=O)CCn2cccn2)C1C c1(CNC(c2nc(C(=O)NC(C)CCO)sc2)=O)c(F)cccc1F N1(C(CNC(=O)OC)=O)CCC2CCN(C(C3CCC34CCC4)=O)C2C1 N1(C(CNC(=O)OC)=O)CCC(C)C(CNC(=O)CC=Cc2ccccc2F)C1 N1(C(c2ccc(C)o2)=O)CC(CNC(=O)CCCOc2ccccc2)CC1(C)C c1(C(=O)NC(C(C)C)CO)cnn2cccc(-c3ccnnc3)c12 CC1(C)CC(C(=O)N2C3CCC2CN(C(C2CN(S(C)(=O)=O)C2)=O)C3)=NO1 N12CCCC(O)(C1)C2=O.C1(C(=O)NCC2(SCC)CC2)CCC(CC2CC2)CC1 CC(C)(C)C(CNC(C1CC(NC(=O)CCc2nc(=N)[nH][nH]2)C1)=O)CO C(=O)(C1=CC2(CCN(C(=O)CCCC(F)(F)F)C2)C1)NCCS(C)(=O)=O N1(C(CCCCCC)=O)CCN(C(c2cn(C(C)C)nc2C2CC2)=O)CC(O)C1 C1(CC(=O)NC(C)CN(C)C(=O)OC(C)(C)C)CCC(NS(N)(=O)=O)C1 C1(C(=O)NCCOCCCNC(C(c2ccn(C)n2)C)=O)CCC2CC2CC1 N1(C(c2c(COC)nn[nH]2)=O)CCN(C(C2CCCO2)=O)CC1C(F)F c1(C(C(=O)NCc2ccc(OCC#N)cc2)(C)O)ccc(Br)cc1F n1(C(C)C)ncc(C(N2CCCC2C2(NC(c3ccc(Cl)s3)=O)CC2)=O)c1Cl C(=O)(C1(C)CCCc2ccccc21)N1CCN(C(c2c(SC)ccs2)=O)C(C)C1 n1(CC)nc(Br)nc1C(N1CCCC(CC(N)=O)C1)C(=O)NC1CCOC1 O=C(C1=NOC2(CCNC2)C1)N1CCCC1c1cn2cccnc2n1 Cc1cc(N(CC(O)CN(C)C(c2c(C)noc2C)=O)C)c([N+](=O)[O-])c(C)n1 N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ccc(F)c(C(C)C)c2)=O)C(CO)C1 Cc1ccc2nc(C)c(C(=O)NCC3CCN3C(=O)CSCC(F)(F)F)cc2c1 c1(CC(=O)NC(C)C(CO)NC(c2cnn(CC3CC3)c2)=O)ccc(O)cc1 N1(C(C(C=C)(C)O)=O)CCN(C(=O)CN(C2CC2)CC)C(c2ccc(F)cc2)C1 C1(NC(C2CC(CCC)C2)=O)CN(C(=O)C(C)OCC(F)(F)F)CCC12CCC2 c1(C(=O)NC(C2(O)CN(C(c3cc(C4CC4)no3)=O)C2)C)cnc2sccn12 c1(C(N2CCC(O)(C(C)NC(=O)CCC(C)(C)C)C2)=O)ccc2nccnc2n1 Cc1oc2ccccc2c1CCNC(=O)NC1CCCN(CC2CC2)C1 C1(C2(O)CCC2)(CNC(C2N(C(C3N(C(C)=O)CCC3)=O)CC(F)C2)=O)CC1 C1(C2(C)CC2)CC(=O)CC12CCC2.C12CN(CC1(C)C)C2=O.C12CC3(C1)CN(C3)C2 C1(NC(C2CN(C(C)C)C2)=O)CC2CC1N(C(c1cc(C(F)F)n(C)n1)=O)C2 C1(NC(C(C)(CSC)NC(C(C(=O)OCC)F)=O)=O)COC2(CCCC2)C1 c1(OC)ccc2c(c1)CCN(C(=NCc1ccnn1C)NCC(C)OC(C)C)C2 C1(CC)CC2CCC(C1)N2C(=O)Cn1nc(Cl)ccc1=O c1(OCOC)ccc(F)c(F)c1C(N1CC(C)OCC1C)C(=O)NC1CCCC1 CC1CN(C(C2(F)CCCN(C(=O)C(O)CC3CCCC3)C2)=O)Cc2c[nH]nc21 C1(C(N(CC(C)CNC(=O)CCC2CCC(=O)N(C)C2)C)=O)COC2COCC12 C1(NC(c2ncc(N)nc2)=O)CC2CC(NC(=O)Cc3nc[nH]n3)CC12 c1(OCC(N2CC(CC)C(NC(c3ccoc3)=O)C2)=O)cccc(F)c1F Cc1cc(NC(=O)CC2CCCN(Cc3cc(I)ccc3O)C2)cc(Cl)c1 N1(C(c2n(CC)cnn2)=O)CC(NC(=O)Cc2ccsc2C)CC(C)C1 N1(C(CC(=O)NC(C)C)=O)CCCN(C(=O)COCCc2ccccn2)C(C)C1 c1(C(=O)NC2C(CNC(c3cc4sccc4s3)=O)CCC2)nnc2n1CCOC2 C(=O)(CCCS(C)(=O)=O)NC1CC(NC(c2c(CC)nn(C)c2Cl)=O)C1 CC1CN(C(=O)C(C2(O)CN(C(=O)CC3(C#N)CC3)C2)F)CCN1C C1(C(N(CCC)CC)=O)CCC(C)(C)N(C(=O)CN2CCC(OC)C2)C1 S(=O)(=O)(CCC(F)(F)F)NCC1(C)CCN(C(=O)CCc2ccc(O)c(O)c2)C1 c1(OC)cc(C)c(C(N2CC(N(C)C(c3cncc(CC(C)C)c3)=O)C2)=O)cn1 c1(C(=O)NCC2N(C(C(CC)NC(C)=O)=O)CC(O)C2)cc(F)cc(Cl)c1N C=CC1COCCN1C(c1cc(-c2ccncc2)[nH]n1)C(=O)NCC1CC1 c1(OC)c(Cl)cc(C(N2CCC2(C)C(N2CC3CCC2CO3)=O)=O)c(OC)c1Cl N1(C(C(CC)F)=O)CCC(OCCCCCOC(=O)CN(c2ccccc2)C)CC1 C1(NC(=O)Cc2cc(Cl)on2)COCCN(C(=O)CC2(O)CCCC2)C1 N1(C(C(CCCC)N(C)C)=O)CCCC2CN(C(=O)C(=O)NCC)CC12 C1(C(=O)NCC2C3CC2N(C(c2ccc(CO)cn2)=O)C3)CCCCC1C1CC1 CC(C(=O)NC1CC1C(N1CC(N(C)C)C1)=O)S(C)(=O)=O C#CC1(C(=O)NOCc2nc[nH]n2)CCN(C(=O)C(C)=C(C)CC)C1 C1(C(=O)NCC2N(C(=O)CC3(O)CCCC3)CC2)C(C(F)(F)F)C1[N+](=O)[O-] CCC(CNC(=O)CCN(CCCO)C(C1CCC2CC1CO2)=O)C(C)(F)F c1(C(N2CC(F)(CNC(COCCOCC#C)=O)C2)=O)cn(C)c(=O)n1C N1(C(CC(C(C)(C)C)NC(=O)CSC(F)(F)F)=O)CC2(CCOC(=O)N2)C1 Cc1ccc(Br)cc1C(=O)NCCC1C(C)CCCN1C(=O)C1=CCOC1 Cc1nn(C(C)C(=O)NC2CCN(C(=O)C(F)(F)CO)C2)c(C)c1[N+](=O)[O-] N1(C(c2c(OCC)scc2)=O)CCC(CO)C(NC(c2cc(O)nn2C)=O)C1 C(CC(CC)C(=O)NCC1CC(NC(=O)COC2CCCC2)C1)=CC c1(-n2cc(C3CCN(C(Cc4ccc(C)nc4)=O)CC3)nn2)cc(Br)ccc1Br C12(C(N3CC(O)(CCNC(C=CCOC)=O)C3)=O)CCCC1CC(F)(F)CC2 CC1CN2CCN1CC2C(=O)NCCC1CN(C(C2CC3C=CC2C3)=O)CCO1 C1(C(N2CCC(C#N)(NC(c3ccccc3)=O)C2)=O)CC2CCCC(C1)C2 C1(C(N2CC(CN(C(CC3(OCC)CC3)=O)C)C2)=O)CN2CCN1CC2C c1(CC(=O)N(C(CNC(CSCCC)=O)C)C)csc2ccc(C)cc12 Cc1cc(Cl)c(C(N2CCCN(C(c3cc4c(ccn4C)[nH]3)=O)CC2)=O)cc1F N1(CC#CC)CCN(C(=O)C(CCOC)NC(C2CCCSC2C)=O)CC1 Cc1ccc(C=CC(=O)N(C)CC2CCCN2C(=O)C=Cc2ccncn2)cc1 CC1ON=C(C(=O)NCC(O)CNC(c2ccc(C(C)(C)C)c(Cl)c2)=O)C1C C#Cc1cccc(OCC(N2CCC(F)C(NC(=O)CC(Cl)Cl)C2)=O)c1 c1(C(=O)NCC(CO)NC(C=COCC)=O)cc2ccccc2cc1F C(C(F)(C(=O)NCC1(n2nccn2)CC1)C(C)C)NC(C1(CC)CCOC1)=O.C1CC1 CC(N(C)N(C)CC1CCCc2ccccc21)C1CCCN(C(C)(C)C)C1 CC1CCN(C(c2c(C3CCC3)cnn2C)=O)CC1NC(c1ncc(Cl)s1)=O CN1Cc2ccc(C(N3CC4CCC3CN4C(=O)C(F)OC(F)(F)F)=O)cc2C1 N1(C(CSc2n(-c3ccc(OC)cc3)ccn2)=O)CC(C)N(C(C)=O)CC1C Cc1cc(C(=O)NCCCC(C)(C)NC(=O)CCS(C)=O)ncc1N Cc1ccncc1C(N1CCCC1CCNC(=O)CSc1cccs1)=O C(CCC(=O)NC(c1nocc1C(=O)N(CC(C(C)C)OC)C)C)OC C(=O)(C1CCc2cccc(Cl)c21)N1CC(NC(C=CC(C)C)=O)C1 N1(CC)CCOC(CNC(C2(CC)CCC2)=O)C1.C1(=O)C(C)=CCN1 c1(C(N2CCC(NC(c3cn[nH]c3)=O)C(CO)C2)=O)cc(F)cc2nc[nH]c12 c1(CNC(c2ccc(OCCOC)cc2)=O)ccc(C(=O)O)c(OC)c1 N1(CC)CC(C(N2CCCC(N(C(=O)CCc3cnco3)C3CC3)C2)=O)CC1=O CCC(C)CC(C(=O)NC1(CO)CC(O)C1)NC(=O)Cc1cnccc1C Cc1cc(N2CCC(C)(NC(c3cc(C4CC4)n(C)n3)=O)CC2)nc(C(C)C)n1 N1(C(c2n[nH]c(C)c2F)=O)CCCC2(C1)CN(C(=O)CCCCNC(N)=O)C2 C12(CCN3C4CC(NC(C(C)O)=O)CC3CC4)CC3CC(C)(C1)CC(F)(C3)C2 C=CCCC(C(=O)NCC1(C)CNC(=O)O1)NC(C1CCCOC1)=O C1(C2CCC2)(CNC(CN(C(=O)C(C)SC(C)C)CC)=O)CC1 C(CCCCC(=O)N(CCNC(C1CCCSC1C)=O)C(C)C)NC(C)=O N1(C(C(CO)OC)=O)CCOC(C2CN(C(=O)Cc3c(C)noc3C)C2)C1 N1(C(c2cc(OC)cc(CC)c2)=O)CC(C)N(C(C2CC(F)(F)CS2)=O)CC1C Cc1cc(N2CCC(C)(C)CC2)nc(=NCc2cnc(O)[nH]2)[nH]1 c1(C(=O)NC(CC=C)CNC(=O)CCSC)cc(C(F)F)ncn1 N1(C(=O)NCCS(=O)(=O)NC(C)C)CCCC(C2CC2(F)F)C1 C1(NC(=O)CC23CCCC2C3)CCN(C(c2cnoc2-c2ccoc2)=O)CC1F CC(C)C(F)C(=O)N1CC(N2CCN(C(C3(O)CCC3)=O)CC2)C1 CC1COCC(C(=O)NCC2(O)CC(C(=O)NCCNC(=O)C3CC3)C2)O1 C(=O)(CCC(F)(F)C(F)(F)F)NCC1=CCN(C(c2c(C)sc(O)n2)=O)CC1 c1(CNC(C(C)N(C(c2cc(O)cc(=O)o2)=O)C2CC2)=O)cc(F)cc(F)c1 CC1CCn2cc(C(=O)NCC3CC3NC(c3c(N)cccc3F)=O)nc2C1 c1(C(=O)NC(CNC(c2ccsc2C(F)F)=O)CO)ccnc2ncccc12 C(=O)(C1=NOC(C)C1)NC1C(C(=O)NC2(C(C)C)CC2)COCC1 C1(C(=O)NCCC2C(C)C2)CC(O)C(O)CC1CNC(C1CCC2CC12)=O CC1(C)C(CNC(=O)CCc2cnn[nH]2)CCN1C(c1ncn(C(C)(C)C)n1)=O c1(CC)cccc(C(=O)N(C)CC2CN(C(c3cccc(OC)n3)=O)C2)c1O c1(C(N2CC(c3cn(-c4cccc(N)c4)nn3)C2)=O)cccc2c1CCCCC2 N1(C(=O)NC(c2cccc(C#N)c2)C)CCN2CCC1C2 CCCC(CNC(=O)CNC1CCCC1CN(C)C)C(=O)Nc1nnnn1C C1(C(=O)NC(CC)C(=O)NCC(F)(F)F)CCN(c2cc(C)ncn2)CC1C N1(C(c2nc(C)oc2)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)C(CC2CC2)C1 c1(CC)cccc(CC)c1NC(=O)C(CO)NC(=O)C#CC1CC1 C(=O)(C(C)(C)CN1CCCC1)NC(c1ccncc1)C c1(CC)oc(C(N2CCC(CN(C(=O)CSS(C)(=O)=O)C)C2)=O)cc1C N1(C(C2(NC(C3C(C)(C)COC3)=O)CCC2)=O)CCOC(C#N)C1 c1(C(c2n(CCSC)nnn2)NCC(C)(C)CCC(C)O)ccc2c[nH]nc2c1 CCC(CC(C)C)C(=O)NCC(C)(O)CNC(=O)CCCN1CCCC1 N1(C(C(=O)NCCOCC(=C)C)=O)CCC2CCC1C2 O=C(CCCCc1cccc(O)c1)NC(CNC(c1cc(Cl)sc1Cl)=O)CO N1(C(C(OC)OC)=O)Cc2ccccc2C1CNC(=O)C1=NOC2COCC12 N1(C(C(C(C)(C)C)O)=O)C2CCCC1CC(NC(=O)C=CC1CCCO1)C2 C(=O)(C(CNC(C1C2CC3C(C2)C13)=O)CC(C)C)Nc1cccc(SC)c1 Cc1ccc2c(=NC3CC4CCC(C3)S4)[nH]c(=NC(C)c3ncc[nH]3)[nH]c2c1 C(=O)(C1=NN(C)C(=O)CC1)N1CC2(CC(NC(C3(COC)CC=CCC3)=O)C2)C1 CCCCCC(O)C(C)C(=O)NC1CCCCC1C(N1CCC(F)(F)C1)=O Cn1ncc2c1CC(C(=O)NCC1CC(NC(=O)Cc3ccsc3Cl)C1)CC2 c1(OC)c(CN2CCC(O)C2C(=O)Nc2cccc(F)c2OC)cc(F)cc1Cl C(=O)(CCCC(=O)NCC1CCC(NC(c2ncc(F)cc2C)=O)C1)OC N1(C(C(C=C)(C)C)=O)CCC(C)(CCNC(C2CCOC(C)(C)C2)=O)CC1 c1(N2C3C(CN)(CCCC3)CC2)ncc2c(n1)CCCCC2 c1(C(=O)NC2(C)CN(C(C3CC4CCCCN4C3)=O)C2)coc2ccc(F)cc12 c1(NC(=O)Nc2ccc(OCCC)c(C)c2)cnc(C#N)c(Cl)c1 C1(C(=O)NC2(C(N(C)CC3CCCCO3)=O)CC2(C)C)C2CC(=O)CC12 C1(C(=O)CN(C)C)(CNC(CC(C)NC(=O)OC(C)(C)C)=O)CCCCO1 C12(C(=O)NC3C(NC(c4cnn(CC)c4C)=O)CCC3)CC1COC2(C)C N1(CCC(=O)NCC2(CCNC(c3cnc(S)nc3)=O)CC2)CCC(O)CC1 n1(CC(=O)NC2C(CNC(c3ccc(C(C)F)cc3)=O)CC2)nc(Cl)ccc1=O c12cc(c(Cl)cn1)N2CC.N1(C(=O)OC(C)(C)C)C2CCC(C2)C1CO C=C1CC(C(=O)NCCCS(C)=O)(CNC(=O)C(O)C2CC2)C1 C1(OC)CN(C(c2conc2C)=O)CC1NC(c1c[nH]nc1OC)=O c1(CC)noc(CCNC(C2(C)CC(NC(=O)C(CO)OC)C2)=O)n1 C=CCCCC(C(=O)N1CC2CCC(CC2)C1)NC(c1cnc(O)o1)=O N1(C(CNS(NC)(=O)=O)=O)CCC(CNC(=O)Cc2c(C)n[nH]c2C)C(CO)C1 N1(C(c2c(CC)ncs2)=O)C2CCC1C(CNC(=O)C(C)(C)OCC(F)(F)F)C2 Cc1cnn(C)c1CN(C)C(C1CC=CCN1C(=O)CCC(C)N(C)C)=O CN1CCC(C#N)(C(=O)NCC23CCCC2CCN3C(c2cn[nH]c2)=O)CC1 C1(C(=O)NCCC(C)(C)CNC(C2(COC)CCNC2=O)=O)(OC)CCCCC1.CSC.Br.C.N C(=O)(C(C)(C)C(O)C(C)C)NCC1CCC(C(=O)NCc2nccc(OC)c2)C1 C1(C(N2CC(COC)(NC(=O)CSc3nc[nH]n3)C2)=O)CCc2nc[nH]c2C1 C1(C2CC2)(CNC(=O)NC(C)CCC2CCCO2)CCC1 c1(C(N(C2CCN(C(=O)C(C)(C)CF)C2)CC)=O)ccc2c(c1)N(C)CCO2 N1(C(C(c2cc(Cl)cc(Cl)c2)C)=O)CCC2(CCOC(C)C2)C1 Cn1[nH]c(C2CCC(C)CC2)nc1=NC(=O)C1(C)C(C)(C)C1(C)C c1(CC)ccc(CC(N2CCC(C(C)NC(c3cncc(Cl)n3)=O)CC2)=O)cc1 C1(C)(N(C)C)CCCC1NC(=O)C(C1CCN(C(=O)CCc2nccs2)C1)F C1(C(=O)NCCC(C)N(CCC)C)CCN(C(=O)Cc2cn(C)cn2)O1 O=C1CCN(CC2(Cc3ccccc3)CC3(CCC3)C2)C(=O)N1CC1CC1Cl N1(CCCC(=O)N(C(C)CN(C)C(C2CCS(=O)(=O)N2)=O)C)C(=O)CN(C)C1=O CC(F)(F)C(F)C(=O)NCCC1(C(N2CC(O)(C(F)F)C2)=O)CCC1 C(c1cccnc1)=CC(=O)NC1(CCCNC(=O)C=Cc2cc[nH]n2)CC1 N1(C(C2N(C(CCOCC(C)C)=O)CC=C2)=O)CCCC(CCF)C1 c1(C(N2CC3C(C2)C3(F)F)C(=O)Nc2c(C)cccc2)ccnc(Cl)c1Cl C1(NC(c2c(C)nc(C3CC3)s2)=O)CCN(C(c2ccn(C)c2C)=O)C12CCC2 c1(C(N2CCC3CN(C(=O)C(Cl)(Cl)Cl)CC23)=O)ccc2nc(Br)nn2c1 CC1CCC(CC(=O)NCC2CCCN(C(c3n[nH]cc3N)=O)CC2)CC1C C1(C(=O)NC2CCN(C(C=CC=CCC)=O)C2)CCC(NCCC)CC1 N1(C(CCOCC#C)=O)CC2(C1)CN(C(=O)CNC(N)=O)CC2CO c1(CC(=O)NCCC(CNC(CC(CN(C)C)O)=O)O)cccc(F)c1O c1(NC(C)=O)ccc(S(=O)(=O)NOCC2CC2CC(C)C)cc1 C1(NC(CNC(c2c(C)occ2)=O)=O)CCC(Nc2ncnc(=N)[nH]2)CC1 N1(C(c2n(CCC)ccc2)=O)CC(F)(F)CC1C(N1CCN(C)CC1CC)=O N12CCN(C)CC1CNC(=O)C1(CC1)C2=O.C1(C2CCC2)(C=O)CC1.CO c1(OC)ccccc1CCNC(=O)C(c1nc(Cl)cs1)N(c1nccs1)C(C)C N1(C(CC(C)C2(CC(F)(F)F)CC2)=O)CCN(CC(=O)NC2CC2)CC1C C1(C(=O)NC(CN(C)C)(C)C)CC2(CC(NC(=O)Cc3ccccn3)C2)C1 Cc1nc(Cl)cc(=NCCCC(C)NC(c2cccnc2-n2cccn2)=O)[nH]1 C1(NC(c2nc(C(C)C)sc2)=O)CCN(C(=O)C(N)=O)C(c2ccccc2)C1 Cc1cc(C(N2CCN(C(C3CC3C3CC3)=O)C3CC23)=O)c(F)c(F)c1 N1(CCC)CCCC1C(=O)N(C)CCN(C)C(c1ncc[nH]1)=O C1(NC(c2ccccc2F)=O)CC(NCc2ccc(F)nc2)C12CCC2 C(N=c1cccc(S(=O)(=O)N(C)Cc2cnn(CC(C)C)c2)[nH]1)c1nnc(C)s1 C1(NC(C2CCC(CC)O2)=O)CC2CCC(C1)N2C(=O)Cc1cccnc1N c1(C(N2CC(NC(C3(C(F)F)CCC3)=O)CC(F)C2)=O)n[nH]c2ccc(Br)cc12 C1(C(=O)NCc2cccc(OC)c2Cl)CC12CCN(C(=O)CC13CC(C1)C3)CC2 CCCC(C(=O)NC(C)CCNC(c1cnn[nH]1)=O)NC(N)=O C1(C(CO)NC(c2cnc(C(C)C)o2)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1 c1(C(=O)NC(c2nc(=O)o[nH]2)C)cncc(CNC(C2CC=CC2)=O)c1 c1(C(N2CCC(C(C)(C)NC(C(CC)F)=O)C2)=O)cc(Cl)c(O)c(Cl)c1 Nc1cc(Cl)nc(C(=O)NCC2CN(C(c3ccccc3Cl)=O)C2)c1Cl CCCCC(CC)CCC(=O)N1CCC(CCC(=O)NC23CCC(C2)OC3C)C1 c1(C(=O)NC2C(NC(CCOCC#C)=O)CC2)oc(C2CCC2)nc1C c1(C(=O)NCC(=O)N(CCCNC(C2CC3C=CC2C3)=O)CC)ccc(Cl)cc1Cl O(N=C1CCCCCC1)CC(=O)NCC1C(NC(C2(C)CC2)=O)CCCC1 c1(C(=O)NCCCCCNC(C2C3CCCC(=O)C32)=O)c[nH]c2cccc(F)c12 Nc1nccn2ncc(C(N3CCC(NC(=O)C=Cc4cscn4)C(F)C3)=O)c12 c1(C(N2CC(CC(=O)NC)N(C(C3CC3F)=O)CC2)=O)cc(F)c(C#N)c(F)c1 CC1CC2(CCO1)CC2C(=O)NCC1CC(NC(=O)COC2(C)CCCC2)C1 n1(CC(=O)NC2CCN(C(c3c(C(C)O)cccc3)=O)C2)ncc2ccccc12 C=CCN=c1[nH]cc(C(=O)NCC2(NC(=O)COCCOCCO)CCC2)s1 CCC(CNC(=O)NCc1c(C)cc(C)nc1O)(CC)C(F)(F)F C1(NC(c2cc(SC)c(N)cc2)=O)CN(C(=O)C(C)(O)C2CCC2)CC2(CC2)C1 C1(C2CN(C(=O)C=C3CCCC3)C2)(NC(c2n(CCC)nc(C)c2)=O)CC1 C12(C)CCN(C1)C2=O.C1(C#N)(C(=O)NCC(N2C(C)CCC2)=O)CC(=O)C1 N1(C(C(CC)(CC)CO)=O)CCN2C(=O)C(NC(c3cnco3)=O)CC2C1 c1(NC(CC)CC2CC2)ncccc1S(=O)(=O)NCCC1(CO)CC1 C(=O)(CCCCCNC(C1CC(C)CC(C)C1)=O)NCC(CC(=O)NC)C c1(C(=O)NCC(CC)NC(=O)C(CSC)OC)cnc(Cl)n1C n1(CC)cc(NC(C2COCCC2NC(=O)C(F)(F)COC)=O)c(C#N)n1 Cc1ncc(CC(=O)NCC(C2CCCC2)NC(=O)C(=O)N(C)C)s1 N1(C(Cc2cc(C)no2)=O)CC(NC(c2ccc(C3CC3)s2)=O)C(C(F)F)C1 c1(CCC(=O)N(CCNC(C(c2cccc(O)c2)C)=O)C)ccc(N(C)C)nc1 C1(CC(=O)NCC#CCNC(=O)Cc2ccsc2Cl)CCCCCO1 c1(OC)ccccc1C(C(N1CCC(C)(N)C1)=O)OC.C(=O)CCSCCOC CC(C)(C(=O)N1CC2CC(NC(C3CC34CCSCC4)=O)C1C2)C(N)=O C(CCCCC(=O)NC1CC(C(C)(C)C)C1)N(C(C1(CC=C)CC=CC1)=O)C c1(NC(C(F)(F)C2(OC)CCC2)=O)cc(C#N)cc(C)n1.C12CC(C1)CNC2=O C1(CN(CCNC(=O)CC2CC2Sc2ccc(F)cc2)CC)CCCCS1(=O)=O O=C(C1Cc2ccccc21)NCC1C2CC1N(C(c1cncc3c[nH]nc13)=O)C2 c1(NC(C2OCCN(C(C=Cc3ncn(C)c3)=O)C2)=O)cccc([N+](=O)[O-])c1 c1(C(N(C2CC(NC(c3cnns3)=O)C2)C)=O)ccnc(-n2cncn2)c1 c1(-c2scc(C)c2)c(C(N2CCn3ncnc3C2)=O)nn2ccccc12 C=CCCC(C(=O)NC1(C)CS(=O)(=O)C1)NC(C1C(C#N)C1(C)C)=O C(C(F)(F)CN=c1nc2sccc2c(NCC(F)F)[nH]1)(C1CC1)OC C(=O)(C(C)CCNC(=O)C(C)N(C(=O)COc1ccsc1)C1CC1)OC N1(C(C(C2CCC2)OC)=O)CC(CO)(NC(C23CCC2C3)=O)C1 CC1CCSCCN1C(C12CCC1CN(C(=O)C=C1CCC1)C2)=O CC1CCC(C)(C(=O)NCC2CN(c3nccnc3F)CCO2)C1 CCC(C)(C)CCCC(=O)NC(CC(C)(C)C)C(=O)NCc1ccoc1 c1(CC(=O)NCc2ccc(C(=O)O)o2)cc(O)ccc1C(=O)O Cc1cc(C(=O)NC2(CO)CCCN(C(=O)Cc3cnc(C)[nH]3)C2)cc(N)c1 n1(C2N(C(CC3N(C(=O)OC(C)(C)C)CC(O)C3)=O)CCC2)cc([N+](=O)[O-])cn1 N1(C(C2C(OC)C2)=O)CCC2CN(C(C3CC(C)(C)C3)=O)CCC12 Cc1ccc(COC2CCN(C(=O)CC(C)F)CC2)cc1 C(CCC(C)(C)C(=O)NC1CCN(C)CC1C#N)NC(C(CC=CC)C)=O N1(C(c2nnc(C)s2)=O)CCC2(CC1)CC(C(=O)NCCOc1cccnc1)CO2 C1(C(C)C)CC(CC(=O)NCCNC(C2CCCN2c2ccccc2)=O)CCO1 C(=O)(CC(C)C(C)(C)C)NCc1occ(C(=O)Nc2c(C)ccnc2)n1 CC1(C(=O)NCCC2CCC(NC(c3cn(CCF)nn3)=O)C2)CNC(=O)C1 C(=O)(CCCN(C)C)N(C1CCN(C(=O)Cc2cnnn2C)C1)CC c1(C(N2CCCN(CCNC(CCS(C)=O)=O)CC2)=O)ccc2sncc2c1 C(CC(=O)N1Cc2ccccc2CO1)N(CCC(=O)NOC(C)(C)CO)C c1(C(=O)Nc2[nH]c(C)c(C(N3CCC(C)(C)CC3)=O)c2C)cccc(Cl)c1C#N C#CCC(CC(=O)NCCCCCC=C)NC(=O)C(O)CCSC Cc1cc(C(F)F)n(CC(N2CC(NC(=O)CN(C)C(C)C)CC2CO)=O)n1 N(C1CCCc2ccoc21)C(C1COCCC1NC(C1CCNC(=O)C1)=O)=O C#Cc1ccc(OCC(=O)NC(CNC(=O)C(O)CCC)CC)cc1 c1(C(N2CC(NC(=O)CCCCC3CC3)(CO)C2)=O)cc2c(Cl)cccc2[nH]1 CC1(C)CC(NC(=O)COc2ccc(F)nc2)CN1C(=O)CC#N n1(CC)nc(-c2ncccc2C(F)(F)F)nc1CCCCC1CC1 C(=O)(C(F)C(F)(F)F)NCC(CNC(=O)CSCc1ccncc1)O C1(C(N2CC(CC(C)N(C)CC)C2)=O)CCN(C(=O)NC(C)C)C1.c1c(=O)n1 N1(C(c2cnc(SC)[nH]2)=O)CC2CN(C(=O)C3=CCSC3)CCC12 C1(COC(N(C)C(c2ccc(F)cc2)c2ccccc2)=O)CC2(COC2)C1 C1(NC(C2CCN(C(C(C)=C(CC)C)=O)C2)=O)CC(C)OC1=O c1(NC(=O)CC2CCN2C(=O)NS(=O)(=O)CC)ccc2c(O)nnc(O)c2c1 CCCC(CCCNC(=O)C=C1CCC(C)(C)CC1)NC(c1nc(O)sc1C)=O Cc1cc(C(=O)NC2(C(=O)NOC3CCOC3)CCN(C)C2)c(C)nn1 N1(C(c2c(C(C)C)cco2)=O)CC2C(CN(C(=O)CCF)C)C2C1 c1(CC(=O)NC2CN(C(c3csc(C)c3C)=O)CC2F)cnc2n1CCCC2C c1(C(=O)NC2C(F)CCN(C(CC(CC)C)=O)C2)cnc2c(c1)CCCC2 c1(C(=O)NCC2CN(C(COCCCC)=O)CC2C)cc(F)c(Cl)c(N)c1Cl C1(NC(c2c(OC)cc(C)cc2)=O)CCC2(CC1)CN(C(c1c[nH]cc1Br)=O)C2 O=C(CCCCC1CC1)N1CCC(N(CCO)C(c2cc(O)cs2)=O)CC1 N1(C(C(C(CC)O)C)=O)CC2CCN(C(=O)CSc3cccc(OC)c3)C(C2)C1 c1(C(=O)NC23C(CN(C(C(CC#C)C)=O)C2)CC3)cn(C)c2ccc(F)cc12 C=C1CCN(C(=O)CC2COCCOC2)C(C(N2CCC(OCC(C)C)C2)=O)C1 C(C1CN(C(C2OCCC2(C)C)=O)CC1C(N1CC(CS(C)=O)C1)=O)=CC c1(C(=O)Nc2cccc(NC(c3c(CC)non3)=O)c2)cc(C)c(F)cc1F S(=O)(=O)(c1cc(NC(c2ccc(-c3ccccc3C)o2)=O)ccc1O)NC C=C(C)CC(C(=O)N1CC(NC(c2ccnc(C3CCC3)c2)=O)C1)OC CC(C(=O)NC1CCC(C(=O)NCc2ccc(C(F)(F)F)cc2)CC1)C(C)(F)F C12(OC)CCCC(C(=O)OCc3cccc(Cl)c3C#N)(CC1)C2 C1(NC(n2nnc(C)n2)=O)CN(C(C2(C)CC2)=O)CC1C(F)(F)F C1(CNC(CC=C)=O)(OC)CCN(C(C2(CC=C)CCCC2)=O)C1 c1(OC)ccccc1C(C)(C)C(=O)N(C(CO)C(C)C)C C(=O)(C1=CCc2ccccc21)NCC1C(NC(C(C)(C)C(F)F)=O)CCC1 N1(C(CC2(NC(C(C)n3cncn3)=O)CC2)=O)C2CCC1CC2 N1(C(c2nc(C)sc2)=O)CCC(NC(=O)C(C)SC(C)C)CC1 C(=O)(CCCCOC)NC1CCC(CC(N2CCC(=CCC)C2)=O)C1 N1(C(c2nc(CC)sc2)=O)CC(CNC(=O)COC(C)=O)CC1C n1(CC(C)NC(=O)COC2CC2)cc(CNC(c2csc(C(F)F)n2)=O)nn1 C1(CNC(c2c(CC)[nH]cc2)=O)CC(F)CN1C(C1CC(=O)N(CCOC)C1)=O C(=O)(C(C)C(O)C(C)CC)NCC(CC)N(C)C(c1cnc2nccn2c1)=O c1(C(=O)OC)cn(C)nc1C(=O)NC(C(C)NC(c1sc(C)cc1Cl)=O)C(C)C c1(C(=O)NC2CC(NC(c3cc(OC)ns3)=O)C2)cccc2c(C)c(C)[nH]c12 Cc1noc2cc(C(=O)NC3CC3NC(c3ccc(F)c(Cl)c3)=O)ccc12 C1(CNC(C(=O)NC2CCC(C(=O)OC)CC2)=O)CCCN2CCCCC12 C1(NC(CN(c2ccccc2)C)=O)CCSC12CN(C(c1ncc(F)cn1)=O)C2 CC(C)C(C)(O)C(=O)NCCOC(C)(C)CNC(=O)CCC(F)(F)F C=CCC(CNC(c1ccc(Cl)s1)=O)C(=O)N1CCCC1CCN(C)C C1(CN(CC(C)(C)Cn2cc(CN3CCCC3C(=O)O)nn2)CC)CCCC1O C1(CC(=O)NCC(C)SC)CN(C(c2cn(C3CC3)cn2)=O)C(C)(C)C1 N1(C(c2ccoc2Br)=O)CCC2(CCCN(C(C3CCCOC3)=O)C2)C1 c1(C(N(CCCNC(C2C(F)(F)C23CC3)=O)CC)=O)cc2c(s1)CCCC2 Nc1ccc(-c2noc(-c3scnc3-c3ccccc3OC(F)(F)F)n2)cc1 C1(CN2CCN(c3nnc(-c4nc(O)sc4C)s3)CC2)CCCCC1=C(C)C c1(C(N2CC(C=C)(CC(=O)NCC(C)(C)n3cccn3)C2)=O)c[nH]c(C)cc1=O C1(NC(C2CC(F)C2)=O)CN(C(c2ccc(CCO)cc2)=O)Cc2nccn2C1 CC1CCC(CNC(c2cc(O)ncn2)=O)CN1C(=O)C1=CCCCO1 Brc1cc2nccc(N3CCN(Cc4ncn5ccccc45)CC3)n2n1 CC1CCN(C(=O)CC2CC(=O)NC(=O)C2)CC1CNC(=O)C=C1CCN(C)C1 c1(C(=O)NC2CC2CNC(C2(C(F)(F)F)CC2)=O)cccc(=O)o1 C1(C)(CNC(CCC#C)=O)CN(C(=O)Cc2occc2C)C(C)(C)C1 Cc1ccc(OCC(N2CC3CC(NC(=O)CSCC(C)C)C3C2)=O)c(F)c1 C1(CNC(c2cn(CC(=O)NC)nn2)=O)(NCc2nccs2)CCCCC1C C=CC1(CC(=O)NC2CC2NC(=O)CC2(C=C)CCCCC2)CCOCC1 C(C)(C)(CN(C)N1CCCC1c1ccccc1F)N(CC)CC Cc1cccc2oc(C(=O)NC3CN(C(=O)CCC(C)O)C3)cc12 N1(C(c2c(C)c[nH]c2CC(N)=O)=O)CC2CCCC(C1)N2C(c1cccnc1)=O n1(CC)ccnc1C(N1CCC(C(C)NC(=O)C(CN(C)C)N(C)C)C1)=O N1(C(c2cc(C(CC)CC)no2)=O)CC(N(C)C(c2cc(Cl)no2)=O)C2(CC2)C1 C=CC(COC)N=c1nc(N2CCCC(N3CCCC3)C2)c2ncccc2[nH]1 N1(C(CCOCCOC)=O)CC(C)(C)OCC1CNC(=O)CSC(F)(F)F c1(OC)ccc(C(=O)N(CCCNC(=O)C(C(C)C)c2cccnc2)C)cc1 Cc1cnc(C(=O)NCC(C(N2CCCCC23CC3)=O)N(C)C)cc1C c1(C(=O)NCC2C(C)(C)N(C(=O)Cc3ccoc3)CC2)ccc2[nH]c(=N)[nH]c2c1 c1(C(=O)NC2CCN(C(c3[nH]cc(CC(C)C)c3)=O)C2)nccc(C)c1O c1(C(=O)NC2CCN(C(C(F)OC)=O)C2C)cnc2ccccc2c1 C1(C(=O)NC(CC)C(=O)NCCCN2CCCC2=O)CCC2(CC2)C1 N1(NC(C(N=[N+]=[N-])CCC(N)=O)=O)CCc2oc3ccccc3c2C1 Cc1ccc(F)cc1-n1nc(-c2cnn(CCO)c2)nc1C1CCC2CC12 c1(CN2CC(NC(C3OCCN(C(C)=O)C3)=O)C(F)C2)c(I)ccnc1F N1(CC2=C(C(=O)OC(C)(C)C)C2(C)C)CCOC2CCOCC12 N1(C(Cn2c(C)ccn2)=O)CC(NC(c2cnn(C)c2N)=O)C(C)(C)C1 N1(C(C(C)C(F)(F)F)=O)CCOC2CN(C(=O)CCSCc3ccccn3)CC12 N1(C(CC)=O)CCN(C(C)C(=O)Nc2ccccc2C#CC)CC1(C)C CCC(C(=O)OC)C(=O)N1CC(C(=O)NC(CO)CCO)(CC)C1 N1(CC(CC=C)C)CC2CC2(C(=O)O)C1 C1(NC(C(CC)=CCCCC)=O)CC(NC(=O)CC2(COC)CC2)C12CCC2 C(C1CCCc2ccccc21)NC(CC1(C)CN(C(c2cccc(Cl)c2O)=O)C1)=O c1(N2CC(CNC(CCC(C)SC)=O)C(C)(C)CC2)ncc2c(n1)CCCC2 c1(C(=O)NC(C)C(C)NC(=O)C=C(Cl)Cl)cccc2c(Br)cccc12 C1(NC(CN2CC(C)(OC)C2)=O)CCCCCC1NC(c1[nH]c(O)nc1C)=O C1(CNC(C2(OC)CCCOC2)=O)CC(C)CN(C(=O)CC2COCCOC2)C1 N1(CCNC(c2c(CC)ncs2)=O)CCCN(C(=O)Cc2cncc(O)c2)CC1 CCCS(=O)(=O)CC(=O)NCC1(F)CC(NC(=O)C(c2ccc(F)cc2)OC)C1 Cc1ccc2c(c1)CCC(C(=O)NC1CC3(C1)CC3NC(=O)C(C)C)O2 NC1CN(C(=O)CC2COc3ccccc32)C2(CCCOC2)C1 N1(C(c2ccnc(CC(C)C)n2)=O)CCCC(C)C1CCNC(c1cnns1)=O N1(C(C(C(=C)C)(C)C)=O)CC2CC(NC(=O)C(c3c(C)noc3C)(C)C)CC1C2 C1(NC(C(c2cnn(C)c2)C)=O)CC12CCN(C(=O)Cn1cnc(C#N)n1)C2 CC(C)CCC(=O)C(=O)NCc1cn(CC(=O)N(CC(N2CCCC2)=O)C)nn1 C(=O)(C(C)(C)C(F)F)NCC1C(CNC(CNS(CCCOC)(=O)=O)=O)C1 C(=O)(C(C)CS(C)(=O)=O)N1CCC(N(C(C(CSC)C)=O)CC2CC2)CC1 C1(C(=O)NCC2(O)CCN(C(C3(C(C)(C)C)CCC3)=O)C2)COCC2(CCC2)O1 C1(CC)CCC(O)(C(N2CC(O)(CN(C)C(c3conc3C(C)(C)C)=O)C2)=O)C1 N1(C(c2cnc(OCC)nc2)=O)CC(CNC(=O)C(O)COC)C(F)(F)C1 C1(NC(C(C)OCC=C)=O)CCN(C(=O)C=C2CCCC2)C1C1CC1 Cc1oc(C(=O)NC(c2ccccc2)C2(NC(=O)C3CC3)CC2)cc1Br N(C(=NCC(F)F)N1CCC(N2CCCCC(O)C2=O)C1)C12CC(C)(OCC1)C2 CC(C)CC(C(=O)NCCCn1ccnn1)ONC(c1ccc(=O)n(C)n1)=O c1(C(=O)NC2(COC)CN(C(C3CC3C)=O)C2)cc(C)cnc1N c1(C(=O)NC(CC)CNC(c2ncoc2C)=O)cnc(O)nc1O C#CC(CC(C)C)NC(C1CC(F)CN1C(c1cn(C2CC2)cn1)=O)=O CCC(CO)CCNC(=O)C(c1cccs1)N(C(=O)CC1CCCS1)CC c1(CC)cccc(C(=O)N(CC(C)CNC(c2cccn(C)c2=O)=O)C)c1N N1(c2c(OC)cccc2)CCN(C(=O)NC2CC3(C2)CC3F)C(C)C1 C1(C)(CCNC(Cc2c(C)occ2)=O)CCN(C(C2CCCC(C)CC2)=O)CC1 N#Cc1cc(Br)cc(Br)c1NC(C1COCCN1S(=O)(=O)C(Cl)(Cl)Cl)=O N1(C(CC(C)C)=O)CC(N(C(=O)CCCNC(c2ccsc2)=O)C)C2(CC2)C1 c1(C(=O)NC2CCN(C(C3CCCC3C(F)F)=O)CC2F)ccc([N+](=O)[O-])cn1 c1(C(CC)NC(=O)CCC2(C)CNC2)ccccc1OC(F)F C(=O)(C(C)(C)CCNC(=O)C(C)n1cccc1)NC(c1n(CC)ncc1)C c1(C(N2CCC(C)(CNC(c3cc(F)cs3)=O)CC2)=O)c(F)ccc(F)c1O N1(C(c2scnc2Cl)C(=O)NCC2CCCO2)CCC2(CCSC2)C1 C(CC(CC)C(=O)NC(C(=O)NCc1cnc(CC)[nH]1)C(C)CC)=CC N1(C(CC(=O)NCC)=O)CCC(C)C(NC(C2C=CCC2)=O)C1 N1(C(c2ccon2)=O)CCCC2(CCN(C(c3cnc4c(F)cccn34)=O)C2)C1 CCC(CC)C(C(=O)NC1(CNC(=O)C(C)Oc2ccccc2F)CCC1)OC C1(F)(CNC(C(C)SC)=O)CCC(NC(c2ccc(-c3ccc(Cl)cc3)s2)=O)C1 C1(NC(=O)CCN2CCCC2=O)C2CCC1N(C(c1cnn(C3CC3)c1Cl)=O)C2 C(C(C)CN=C(NCc1cnc(N2CCCC2)s1)NCC(C)(C)C)OCC N1(C(C2(C)CCCC2)=O)CCn2ncc(-c3cccc(C4(C)OCCO4)c3)c2C1 C1(C(=O)NC2C(NC(=O)CCc3ncc[nH]3)CC2)Cc2cccc(F)c2O1 N1(C(CCC)=O)CC(C(=O)NCCOCC(C)(C)O)C(CC)C1 CCCC(CCC)CC(=O)NC1(CNC(C23CCCN(CCC2)C3)=O)CCC1 C(=O)N=c1c(F)c[nH]cc1Cl.C12(CNC(=O)OC(C)(C)C)CCCC1C2(F)F c1(N2CC(C)C(CNC(=O)C=C3CCN(C)C3)CC2)ncnc2ccc(Cl)cc12 C1(C(F)(F)C(=O)NC(C)C(C)NC(c2cc(C)[nH]n2)=O)(OC)CCCC1 C12(NC(=O)C=Cc3cn[nH]c3)CCCC1N(c1nc(Cl)nc3[nH]cnc13)CCC2 c1(C(N2CCCC(NC(C3CC(=C)C3)=O)C2)=O)cc(C(F)(F)F)cc(C)n1 C1(C(C)C)CCC(c2nc(C(=O)NCCC(C)NC(=O)COC(F)F)cs2)CC1 c1(OCCC(N2CCCC(C(C)NC(C(C)=C3CC3)=O)C2)=O)c(C)cccc1C n1(CC=C)cc(C(N2CC(C)(C(=O)NC(c3noc(C)n3)CC)C2)=O)nn1 C(=O)(CC(CC(C)C)NC(=O)CCNC(=O)OC)NC(C(=O)NC)CC C1(CC(=O)NC2CN(C(=O)CC3(O)CC3)CCC2CO)CC2(CCC2)CO1 C1(CCOC)CC(c2nnnn2C2CC(F)(F)C2)(NC2CNC(=O)C2)C1 C1(CC)CN(c2ccccc2)CCN1C(=O)NCCC(F)Cl C(CC(CC)C(=O)NCC1CC(NC(=O)CCCn2c(O)nnc2O)C1)=CC c1(SC)ncccc1NC(=O)CC1(NCCOc2ncccc2Cl)CCC1 c1(C(N2CC(C3(NC(=O)CC4CC(F)(F)C4)CC3)C2)=O)cc2c(=O)cc[nH]c2s1 c1(C(N(CC(CNC(c2ccc(OC)nc2)=O)C)C)=O)c[nH]c2cc(F)ccc12 c1(C(=O)NCC(C)N(C(C2C(CCC)CCC2)=O)C)cc(O)nc2ccccc12 CCCCCS(=O)(=O)CC(=O)NCC(CO)NC(=O)C(c1cccc(F)c1)O c1(OCC)ccc(C(=O)NC2CC3(C2)CC3NC(c2cc(C)oc2C)=O)cc1.O c1(CC(=O)NC2C(NC(C3CCC(=O)C3)=O)C2)ccc(F)c(Br)c1 C#CC1CCC(NC(=O)COC2CC(NC(c3cn(C)cn3)=O)C2)C1 N1(C(C(COCC)NC(=O)CNC(N)=O)=O)CCC(C(C2CCC2)O)CC1 C(=O)(C(C)CC(C)(F)F)NC1C(F)CCN(C(c2ncn(C(C)C)n2)=O)C1 C1(CCNC(C2CCN(CC)C2)=O)CC2CCC(C1)N2C(C1(C)COCCO1)=O c1(C(N2CC(C)(NC(CCc3cncc(C)c3)=O)C2)=O)ccc(C)c(C)c1F c1(C(C)C(=O)NCCCC(N2CCCCC2CO)=O)ccc(F)c(F)c1 C1(CC(=O)OC(=O)C(F)(F)F)CN(Cc2cccnn2)CC1C(=O)O C1(C)(CNC(Cc2c(C)nc(S)s2)=O)CN(C(c2cc(Cl)ccn2)=O)CCO1 C1(CC(=O)NCC(CNC(COCCOC)=O)CO)COCC1(C)C CCCCC(O)C(C)C(=O)NCCN(C)C(c1ccc(O)c(C)c1)=O N1(C(C(C)OCCCC)=O)CC(OC)CC1CNC(C1(CCCC)CC1)=O C1(CC)(NC(C2CC(N3CCCC3)C2)=O)CCCN(C(=O)C2=COCCC2)C1 C(=O)(C(CC(C)C)C(C)C)N1CCC(NC(c2ccc(C)c(Cl)c2)=O)CC1C C1(NC(C(C)O)=O)CCN(c2ncnc(Cl)c2CO)CC1F C1(C(=O)[N+]([O-])(Cc2cnns2)NCC2(N3CCCC3)CCC2)CCC(C(F)(F)F)C1 Cc1cc(C(N2CCN(C(=O)Cc3cncn3C)CC2CC2CC2)=O)ccc1Cl C(C(C)(C)C(=O)NCC(C)N(C(c1ccccc1F)=O)CC)OC c1(CNCCNC(C(C)C)=O)nccn1C(F)F C1(CNC(N(C)Cc2ccc(Cl)cc2)=O)CC2CC(=O)C1O2 C12(C(=O)NCC3(F)CC(NC(COCCC=C)=O)C3)CCCC1CC2 c1(OC)cc(C(=O)NC2CC2CNC(c2ncoc2C2CC2)=O)nn1C c1(C(=O)NCc2c(C(C)C)nn(C)c2)c2ccccc2nn1C C1(C2CC2)(CNC(C(C)CC2CCC2)=O)CCN(C(=O)CC2CC2)C1 N1(C(C=C(CCN(C)C)Cl)=O)CCOC(CCNC(=O)C=CC2CCCC2)C1 C(CN=C(NC(C)COCC1CC1)N1CCC(n2cncn2)C1)OCC=C CC(CC(=O)NC1(CCNC(c2nccn2C)=O)CCCC1)P(C)(C)=O c1(OC)ccccc1C=CC(=O)NCCCCN(C(=O)C(C1CCOCC1)F)C C1(C)(C(=O)NC(c2nccs2)CC)CN(C(=O)C(C)COC)CC1C C(C(C)(C)CCNC(=O)CC(C)(C)OCC(F)(F)F)OC c1(CCC)cc(C(N2CC(NC(=O)CCCn3ccnc3C)C3CC23)=O)ccn1 C12(C(=O)NCC(CNC(=O)CCN3CCOCC3=O)OC)CCC(CC1)C2 c1(SC)ccc(C)c(C(=O)NCC2CCN2C(=O)C(O)c2cnc[nH]2)c1 c1(NC(C(=O)N(CC=C)CC2CC2)=O)ccc(F)c(C(F)(F)F)c1 O=C(NNC(=O)c1coc(C(F)(F)F)c1)C(=O)Nc1ccc(F)cc1 N1(C(C2CCCN(C(c3c(OC)cc(F)cc3)=O)C2)=O)CCC2(CCCC2)CC1 CC1CN(C(=O)CN2CC=CC2)CC(C)C1NC(=O)CCSC(F)(F)F C1(C(N(CCCCCNC(=O)CC2CCCO2)C)=O)COCC1(C)C c1(C(N2CC(NC(C(N(C)C)C3CC3)=O)CC2(C)C)=O)ccc(S(C)(=O)=O)o1 C(=O)(C1=CCCCCC1)NC1CC2CC(NC(=O)Cc3ccns3)C2C1 CC(C)(CCl)C(=O)NC1CCC(C(=O)NCC2(C#N)CCC2)CC1 C(CC(C)(C)CC(=O)N1CC(CC(C)NC(C2Cc3ccccc3O2)=O)C1)OC Cc1nc(N)cnc1C(=O)NCCC1(O)CN(C(=O)Cn2ccccc2=O)C1 c1(C(=O)NC(CN(C(c2nc(C3CC3)cs2)=O)CC)C)cc(O)ccc1Cl c1(C(=O)OCc2ccc(C#C)nc2)occ2c1CCCC2 N1(C(C(c2cccnc2)C)=O)CCCCC1CCN(C)C CCCCC(C)(F)C(=O)NCC1(OC)CCN(c2nnc(C)o2)C1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(CCNC(C=CC(C)C)=O)C(C)C1 c1(C(=O)NC(C(C)(C)O)C(=O)N2CCC(C)(F)C2)ccc2occc2c1 c1(N2CCCC(NCC(C)C)C2)ncccc1S(=O)(=O)NCCCC#N N1(C(C=COCC)=O)CCCC1(C)CNC(C1CCCC(C2CC2)O1)=O N(C(=NCCC(C)(C)O)NCC1CCCCC1)Cc1c(C)nccn1 N1(C(C(CC)C)=O)CC(O)CC1CNCc1c[nH]ccc1=N N1(C(C(=O)Cc2ccccc2)=O)CC2(C1)CN(C(c1cnc(S)nc1)=O)C2 C1(CC)CN(C(=O)Cc2cnc(C)[nH]2)CCC1CNC(C1CCCCCC1)=O C1(CNC(c2ncc(C(F)(F)F)s2)=O)CC(F)(F)CN1C(C1CCCSC1)=O C(=O)(CC1c2ccccc2C(=O)N1C)N1CC2CN(C(CC)=O)CC2(C)C1 c1(OC)ccc2nccc(C(=O)NCC(O)CNC(=O)C(C)(C)CF)c2c1 c1(-c2c(C)nc(C)nc2O)cc2c(C(F)(F)F)cc(O)nc2o1 c1(OC)ncc(C)cc1C(N1CC2CC(C1)N2C(=O)C1=CCCCC1)=O O=C1CCC(CNC(=O)Cc2ccnc(O)c2)CN1 c1(N(C(=O)NCC(CC)NC(C)=O)C)cc(F)c(F)c(F)c1 C(C(=O)N=c1ccn(-c2cncnc2)[nH]1)C1(C)CN(C(=O)C=C2CCOCC2)C1 C12(CC(=O)N(C)CCN(C)C)CC3CC(CC(C3)C1)C2.C12CC(F)(C1)CCC(=O)N2 c1(CNC2CCCC(CCN)C2)ccc([N+](=O)[O-])cc1Cl Cc1ncsc1C=CC(=O)NCC1(NC(=O)CSC(C)(C)C)CCC1 N1(C(CCC2(NC(C(C3CC3)OC)=O)CCC2)=O)CCC(N(C)C)C1 c1(CCN(C)C(c2cncc(SCCC3CC4C=CC3C4)c2)=O)cccc(F)c1 c1(C(=O)NC2CN(C(C3CCOC3)=O)C2)cc2c(Br)[nH]nc2s1 C(=O)(C(C)CCCC(C)=O)N1CCC(C(N(CC(=O)OC)C)=O)C1(C)C C1(CC=C)(NC(c2ncccc2F)=O)CCN(C(=O)CCC(C)OC)CC1 Cc1nc(CC(=O)NOCC(=O)NCC2=NOCC2)c(C)o1 Cc1cn2nc(N3CCC(F)(F)C(CNC(c4cc(Cl)ccc4Cl)=O)C3)sc2n1 C1(CCC(=O)NCCCN(C(C=COCC)=O)C2CCCC2)CCCC(O)C1 c1(CC(=O)NC2COCCN(C(=O)Cc3ccsc3)C2)coc2cc(Cl)ccc12 Cc1ccc(C(=O)N(C2CCCN(C(c3cc(C)co3)=O)C2)CCF)nc1 c1(C(C)=O)ccc(C(=O)Nc2ccnn2CCN(C)C)c(F)c1 C(C(C(C)C(C)C)NC(c1cn(C)nc1C)=O)NC(CNC(C(CC)CC)=O)=O N1(C(C(CC)(C)CO)=O)CCCC2(CCN(C(c3nc(C4CC4)oc3C)=O)C2)C1 c1(CN2C(C(=O)NCc3ccnc(Br)c3)CCC2)ccc2cc(F)ccc2n1 N1(C(CN2CC(NS(CC)(=O)=O)OCC2)=O)CCN(C(C)=O)CC1C C1C(O)CC(=O)N1.C1(NC(CCNC(C)=O)=O)CCC(OCF)CC1 CC1OC2(C(=O)NCC(C)(C)NC(=O)C(c3ccc(C#N)cc3)C)CCC1CC2 c1(NC(C2CCCCN2C(c2ccc(Cl)o2)=O)=O)nc(Cl)cnc1Br C1(C(=O)NCC2(C(=O)NC(C)CN=[N+]=[N-])CC(=C)C2)CC(=O)NC(C)C1 N1(C(C(c2cnccn2)C)=O)CCC(C2CC2)C1CNC(=O)C(C)C(C)(C)C N1(C(CCCOCC=C)=O)CCC(NC(=O)Cn2c(C)csc2=O)C(F)(F)CC1 Cc1cnc(N2CCC=C(Cl)C2)c(S(=O)(=O)NCC2CCCN(C)C2)c1 N1(C(C(C=C=C)C)=O)CCC2(C1)CN(C(c1ncsc1Br)=O)CCO2 c1(C(=O)NCC(C2CC2)NC(C(CC)F)=O)ccnc(O)c1 c1(C(N2CCC(C(F)(F)F)CC2CNC(=O)C(F)F)=O)nnc(O)nc1O c1(OCC(C)C)cc(CCCNCC(=O)OCCC(F)F)ccc1O c1(-c2onc(C(C)NC(N)=O)n2)cnnc2ccccc12 c1(OCCCC(=O)N2CCC(CCNC(=O)CC3CC34CC4)C2)ccc(Cl)cc1 N1(C(c2ccc(C)cn2)C(=O)NC(C)(C)C)CCc2ccc(Cl)c(F)c2C1 Cc1ccc2c(c1)CC(C)N(C(c1ccc(Cl)c(Br)c1F)C(=O)NC1(C)CC1)C2 C1(C(N(CCNC(C2CCSC2)=O)Cc2ccccc2)=O)CCCC2C1C2(F)F C1(OCC)CN(C(c2cn(C)nc2C)=O)CC1CNC(c1cc(CC)ncn1)=O N1(C(c2c(OC)ccnc2)=O)C2CCCC1CN(C(c1cnn(C3CC3)c1)=O)C2 c1(C(N(CC(C)NC(C2CN(C(C)=O)C2)=O)C)=O)cccc(SCC#N)c1 C1(S(N)(=O)=O)(C(=O)NC(c2cccc(Cl)c2)C)CC1.N12CCC1SC1(CC1)C2=O C1(CNC(C(C)OCCCC)=O)CCCCN1C(c1occ(C)c1C)=O CC(C)(C)CCC(F)C(=O)N1CCC(C2CC2)C1C(=O)Nc1ccc(F)cc1O C1(CC(=O)NC(CNC(=O)CC2(O)CCC2)C(C)C)(CC=C)CCCC1 CC(C)(Cc1cnn[nH]1)C(=O)N1CC(CNC(=O)Cc2ncncc2Cl)C(O)C1 C1(NC(=O)Cc2cnoc2)CCC(F)(CNC(c2cccnc2S)=O)C1 c1(OCC)ccnc2sc(C(N3CCC(NC(=O)C(F)(F)CC)C(F)C3)=O)cc12 C1(OC)CN(C(c2cnc[nH]2)=O)CC1C(=O)NCC1(c2oncc2C)CC1 Cc1cc(Br)ccc1C(C)N(CC(=O)O)C CCCN=C(NCCC1CCCN(S(=O)(=O)CCC)C1)N1CCCC(C)(C#C)C1 C(C)(CCC#N)(c1nnnn1CSc1ccccc1)NCCOCC(=O)OC C(=O)(C1CCC(Nc2ccc([N+](=O)[O-])c(O)c2C)c2ccccc21)OC C1(C2CCCN(C(C3CC3C3CC3)=O)C2)(OC)CC1.C1C(=O)NCCS1 C1(CN(C(COCc2nnc(C)s2)=O)C)CCCN(C(C2CCCCN2C)=O)C1 C1(CC(=O)NCCNC(C(C(C)C)c2cccc(Cl)c2)=O)Cc2ccccc2O1 c1(-n2c(C(c3ccc(F)cc3)C3CC3)nc(-c3scc(C)n3)n2)cc(C)cc(C)c1 N1(C(CN(C(CC2CC(=C)C2)=O)CC(C)C)=O)Cc2nncn2C(C)C1 C1(C(N(C2CC3CC3C2)C)=O)CC1C1CN(C(=O)CCc2nccs2)C1 C=CCCCCCC(=O)N1CCCC(C)(C)C1CNC(c1cnncc1OC)=O C=CC(C)(O)CC(=O)N1CC=CC1CNC(C1CCC(F)(F)CC1)=O C1(CCC#C)CCCN(C(=O)CC2(C)CCN(C(c3ccc(CO)s3)=O)C2)C1 N1(C(CCC(=O)OC(C)(C)C)=O)CC2OCC(NC(=O)CCc3ccon3)C2C1 C(CCCCC(=O)NC(c1nocc1C(=O)NC(C)CC(C)(C)CO)C)=CC c1(C(=O)NCC2CN(C(C(COC)COC)=O)CC2C)n[nH]cc1[N+](=O)[O-] CC(CCNC(=O)C(C1CCCC1)NC(C1CCSCC1)=O)C(F)F N1(C(C2OCC(C)C2)=O)CCCC(C)C1CNC(=O)CC1OCCC1C C(CC(=O)NC1(C2(OC)CCC2)CC1)(C(F)F)NC(CCSC)=O c1(C(=O)NC(CN(C(COCC#C)=O)CC)C)cc2c(F)c(F)ccc2s1 CN1CCN(C(=O)CC2CCCOCC2)C(C(=O)NCc2cc(C(N)=O)no2)C1 N1(S(=O)(=O)Cc2csc(Cl)c2)CC2CC1CN2CC(F)F C(CC(F)F)(C(=O)NCC(CO)C(C)(C)C)N(C(CN(C)C)=O)C c1(N2CC(NC(CC(C(C)C)O)=O)C(C)C2)ncnn2c(Br)ccc12 c1(NC(C2CC(NC(C=C(C)C(C)C)=O)C2)C)nc(C)nc2sc3c(c12)CCC3 Cc1cccc(N)c1C(=O)NC(CC(=O)O)C(C)C c1(CCC)c(C(=O)NC2CCN(C(=O)C(=O)C(C)(C)C)C2)[nH]c(C)c1C(C)=O C(=O)(CCCC(F)F)N(CCCNC(C(n1cc(Cl)cn1)C)=O)C1CC1 C(CN=c1[nH]c(N2CCC3CCCC3CC2)nc2ccsc12)OCCOC N1(C(CC(CCC)(C)C)=O)CCCC2(C1)CN(C(=O)C(CC)N(C)C)C2 C12(CNC(C3=NOC(C)C3)=O)CCCC(CN(C(=O)CSCc3cccs3)C1)C2 C1(C)(NC(COC)=O)CCN(C(c2ccc(Cn3ccnn3)o2)=O)CC1 c1(C(=O)NCC2C(C(N3C(C#C)CC3)=O)C2)cccc(O)c1 CCCCCC(O)CC(=O)N(C)CC=CC(=O)NCCCF Cc1ccc2c(=NCc3ccncc3)[nH]c(CN3CCCS3(=O)=O)nc2c1 N1(C(Cc2cc(COC)on2)=O)CCOC(CNC(C2CCC2(C)C)=O)C1 CCCC(C)CC(=O)NCC1(NC(c2cnoc2)=O)CCOCC1 N1(C(Cn2ncc(CC)c2)=O)CCC(NC(=O)CCSC)C(F)C1 C(C(C)C(=O)NCc1cccnc1)N(C(c1cnccn1)C(=O)OC)CC S(=O)(=O)(c1ccc(NCC2OCc3ccccc32)cc1Cl)N(CCC(N)=O)CC N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(C)(C)C1CNC(C1CCSC1)=O C1(C(N2CCN(C(C3(C)COC(=O)N3)=O)CC2)=O)CC2(COC(=O)N2)C1 N1(CC)CC=C(COC(C2CC2(C)CC)=O)CC1 CC1(CNC(=O)CC2CCCCN2C(c2ccc3c(c2)CC3)=O)CCCCCC1 c1(NCc2ccc(CC(C)C)s2)cc(I)c(Cl)cn1 C(=O)(C(C)(C)CF)NC1(COC)CN(C(c2cc(C(C)(F)F)ccn2)=O)C1 C1(CNC(C(C)OCCC=C)=O)(CNC(=O)Cc2c[nH]ccc2=O)CCOCC1 N1(C(CCC(C)SC)=O)CCC(F)(CNC(c2csc(CO)n2)=O)CC1 C1(NC(CCCCNC(C)=O)=O)CN(C(c2ccnc(O)c2F)=O)CC(C)(C)C1 n1(C(C(=O)OCC)C)cc(C2(O)CN(C(c3occc3CN(C)CC)=O)C2)nn1 N1(C(c2sccc2I)C(=O)NCC(F)F)CCOC2CC12 c1(C(=O)OC)ccc(N)c(C(=O)NCC(CC(F)(F)F)NC(=O)NC(C)(C)C)c1 C1(C2CCN(C(c3cc(F)c[nH]3)=O)CC2)(NC(C2(C#N)CCC2)=O)CCC1 N1(C(c2c(C)ccc(C)c2)=O)CCC2CCN(C(c3sccc3CSC)=O)C2C1 CC1(C)CCCC(O)(C(N2CC3OCC(NC(=O)CCC4(C)CC4)C3C2)=O)CC1 n1(CC(=O)NCCN(C(CCn2c(C)ncc2)=O)CC(C)O)ccc([N+](=O)[O-])n1 CC(C(=O)N(C)CC1CCCN1c1nccc(-c2cnccn2)n1)S(N)(=O)=O c1(C(N2CC3(CCN(C(C4(CO)CCCO4)=O)C3)C2)=O)ncnc2cc[nH]c12 N1(C(CCOCCC)=O)CCC2(CC2)CC1C(=O)NCCc1nnc(C)s1 Cc1cc2[nH]c(C(=O)NCC(C3CC3)NC(C3CCN(C4CC4)C3=O)=O)cc2s1 CCC(C)(C(=O)N=c1c(Cl)c[nH]cc1Cl)c1c(F)cccc1Cl CC(C(=O)N(C)CC1CCCN(C(C23CC(C(C)(F)F)(C2)C3)=O)C1)C(F)(F)F c1(CC(=O)NC(C2CN(C(C3OC(C)CC3C)=O)C2)C)ccc(CO)cc1 N1(CC(COC)OC)CC2CCOC2(CNC(=O)OC)C1 S(=O)(=O)(c1ccc(S(=O)(=O)N2CCCCC(CO)C2)cc1)NC(CN(C)C)CO c1(C(=O)Nc2n(C)ncc2)ccc(-c2ccc(C3(C)OCCO3)cc2)cn1 C(C)(CC(=O)N1CC(C(O)C(=O)NCC(O)CCC2CC2)C1)OC c1(CNC(=O)CN2CCCC2CNC(C2CC2C2CCCO2)=O)ccc(Cl)cc1 N1(C(C2CCCCCC2)C(=O)NCCOC)CCC(S(=O)(=O)CC)C1 c1(OCC)ncc(S(=O)(=O)NCC2CCC2(F)F)s1 C(=O)(C(C)(C)C(O)C(C)C)NCC1C(C(=O)NCCc2cncc(C)n2)CCO1 CC(C)CC(C)C(=O)NC(C)(C)CNC(=O)CCc1nc(C2CCCC2)n[nH]1 N1(C(c2c(C)n(CCO)cc2)=O)CCCN(C(=O)C(C)c2cccs2)C(C)C1 N1(C(C2N(C(C)=O)CCOC2)=O)CCC2CCC(NC(c3cnns3)=O)C1C2 N1(C(C2(C(C)(F)F)CC2)=O)CCC2(CCCCN(C(C3CSCCS3)=O)C2)C1 c1(C(N2CC(NC(C(c3ccccn3)C)=O)C2)=O)cccc(Cl)c1O CCC(CC(=O)N1CCC(CN(C)C(C2CCSC(CC)C2)=O)C1)C1CC1 C(=O)(CC(F)(F)C(F)F)N1CCC2C(NC(=O)C=CC3CCOC3)C21 c1(C(=O)NCC2(COC)CN(C(=O)C(C)CCOC)C2)ncn2c1CCC2 C1(NC(C2CC(O)(CNC(c3ccn(C(C)(C)C)c3)=O)C2)=O)CCC2CC1CO2 c1(OC)nc(Cl)c(C(N2CCC(C(C)(C)NC(C3COCC3(C)C)=O)C2)=O)s1 C(C(=O)NCC(C)(C(C)C)NC(C12CC(F)(C1)C2)=O)(C(C)C)OC C1(C(F)(F)F)(SCC(n2cc(CC(O)C(=O)O)nn2)(C)C)CCCCC1 Cc1cc(C)c(C(=O)NC(C)CCNC(=O)CSCc2ccccn2)c(C)n1 C1(CO)(C(=O)NC23CC(CNC(=O)OC(C)(C)C)(C2)C3)CCc2c(F)cccc21 C1(CNC(CCC(C)OCC)=O)CN(C(c2ccc[n+]([O-])c2)=O)CC1(F)F CCCCCS(=O)(=O)CC(=O)NC(CNC(c1c(COC)nn(C)c1Cl)=O)CO N1(C(COC)=O)CC(NC(c2cccc(S(C)=O)c2)=O)C2(CCOCC2)C1 N1(CC)CCC(C(=O)NCC2CC2NC(C2CCC(=C3CCC3)CC2)=O)CC1 C1(NC(CC(=C)C)=O)C2CCCN(C(=O)Cc3[nH]cnc3C)C2C1(C)C CC(CS(C)=O)C(=O)N1CC(N(C(=O)C(C2CCC2)C2CCC2)C)C1 c1(C(=O)NC(C(=O)NCc2c(C)n[nH]c2)C2CCOC2)ccc(C)n1C C1(CNC(c2cncnc2-c2ccccc2)=O)CCCCC1O c1(CC)cc(C(N2CCC2(C)CCO)C(=O)NCC(F)F)on1 CC(CNC(=O)CN1CCOC1=O)CC(=O)NCCCc1cn[nH]c1 N1(C(C(C)OCC)=O)CCC(CC(=O)N(C)C(C)C)(CF)C1 Cc1cc([N+](=O)[O-])nn1C(C)C(=O)NCCCN(C(=O)C(F)C(F)(F)F)C C12(NC(CCN(S(C)(=O)=O)C)=O)CCCC1N(C(=O)CCN1CCCC1=O)CC2 N1(CC#C)CCN(C(=O)NC2CCCNC(=O)C2)CC1=O C1(C(=O)NC(C(=O)N(CC(C)C(C)(C)C)C)C2(C)CC2)CC2(C1)CC(O)C2 CC(C)CCCCCCNC(C1(CNC(c2nnc(O)nc2O)=O)CC=CC1)=O CCCCC(CNC(c1c[nH]c(=NC)s1)=O)NC(C1CCC(C)CC1)=O C1(CNC(C=Cc2scc(C)n2)=O)(NC(=O)C2=CCOCC2)CC2CCC1CC2 N1(C(C2CCN(C(C)=O)C2)=O)CC(C2(NC(=O)CCCCC#N)CC2)C1 C12CCN(CC1)C(=O)C2.Cc1occc1C(=O)NCC1CC1CNC(=O)C1CC1 C(=O)(CC(C)N(C)C)NCCC(C)NC(c1cnc(C2CC2)[nH]1)=O C(=O)(C(O)CCCNC(C1CN(C)CC1c1ccccc1)=O)OC c1(C(N2C(C)CCN(C(C3(C)CCCCC3)=O)CC2)=O)nn(C)c2c1CCCC2 N1(C(C(C)N(C)C)=O)CC(C(N2CC(S(C)(=O)=O)C2)=O)C2(CC2)C1 c12ccc(s1)C(NC(c1cccs1)=O)OC2=O.C1(CC2CC2)CC1.C1(C)CC1 C1(N(C)C(=O)C2CC2)CCN(C(c2cc(-c3ccccn3)no2)=O)CC12CC2 c1(-c2ccc(C#N)nc2)nc2c(s1)CN(C(=O)Cc1cc(F)c(F)cc1F)CC2 N1(C(N2CC(N(C)Cc3ccc(OC(C)C4CC4)cc3)C2)=O)CCCCC(F)(F)C1 C1(C(C(=O)NCCCSC)N(CC#C)C)CCS(=O)(=O)CC1 c1(C(C)=O)[nH]c2ccc(Br)cc2c1C(N1CC2C(=O)N(C)C(=O)C2C1)=O C1=CN=CN=C(N2CCCC2c2cccs2)c2n1ncc2 C1(CNC(c2cocn2)=O)CCN(C(c2ccc(Br)s2)=O)CC1(F)F C(=O)(C(C)(C)C#N)N1CCC(C(C(=O)NCc2onc(COC)n2)F)C1 c1(CC(C)NC(C(c2cccs2)NC(C2CC(SC)C2)=O)=O)cnccn1 C1(C(=O)O)CCN(C(C2N(C)CC(F)C2)=O)CC1n1cc(-c2cnccn2)nn1 C1(C(=O)NCC2C(C(=O)NCc3ncn(CC)n3)CCC2)CCS(=O)CC1 C1(C(=O)NCc2c(C)cco2)C2CCC(C2)C1NC(C1SCCS1)=O C=CC1CCCC(NC(C2CCCCC2CNC(c2ccc(CO)cc2)=O)=O)C1 N1(C(=O)Cn2cnnn2)CCCCC(C2CN(C(=O)Cc3nccs3)C2)C1 C1(CNC(c2[nH]cc(C)c2)=O)CCN(C(c2cnncc2C)=O)CC1O N1(CC(C(=O)C(C2CN(CCC(CC)N)C2)OC)=O)CCCNC1=O.OC CCCCCC(O)CC(=O)N(CC(C)N(C(=O)C(C1CCCC1)NC(C)=O)C)C N1(C(c2c(CC)nc(C)[nH]2)=O)CCCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 C12(NC(CN(C)CCO)=O)CC(NC(=O)CC3(N(C)C)CC3)(C1)C2 C#Cc1cccc(N(C(=O)CCC2CC(NC(C3(O)CCC(C)CC3)=O)C2)C)c1 N1(C(=O)CCn2cccn2)CCN(C(C23CCCC2C3(F)F)=O)C(C(F)F)C1 N1(C(C(C)Cc2ccccc2)=O)CCCC12CN(Cc1ccc(F)c(Cl)c1F)C2 C1(CC(=O)OCCCSCCC)Cc2ccccc2O1 c1(CNc2c(C(=O)Nc3c(OC)nc(Br)cn3)scc2)ccc2ncccc2c1 CN1CCc2cc(-c3nc(-c4cncc(Br)c4)nn3C3CCC3)sc2C1 C(=O)(CC(C(F)(F)F)OC)N(C1CCN(C(c2cc(O)cc(=O)o2)=O)C1)CCC CC1CC(C(=O)O)(NC(C2(C)CCCCC2)=O)CCO1 c1(C(=O)NC(C(C)NC(Cc2c(C)nc[nH]2)=O)C(C)C)ccc(F)cc1[N+](=O)[O-] CC1(C)CCN(C(=O)C(C2CCN(C(=O)CC3CC4C=CC3C4)C2)F)CC=C1 c1(CC(N2CC(F)(F)C2)=O)ccccc1-c1ncccn1 Cc1cc(C(=O)NC2CC(CO)N(C(c3cnn(C)c3N)=O)C2)sc1Br C(CC1=CCN(C(=O)CC2CC2(Cl)Cl)CC1)NC(c1cc(OCCC)ncc1)=O C(=O)(C1=NNC(=O)CC1)NCC(CCNC(C(c1c(OC)cccc1)=O)=O)O N(C1c2ccccc2CC1NC(C1CCCS1)=O)C(=O)Cc1ccsn1 Cc1nc(CN(C(=O)CCC2CCCN2C(=O)CC2(N(C)C)CC2)C)no1 c1(OC)cccc2c(C)c(C(=O)NC3CC3CNC(=O)C=Cc3cc[nH]c3)oc12 c1(CNC(C=C(C)C)=O)ccnc(N2CCN(C(=O)CCC3CC3(C)C)CC2)c1 CC1(C(=O)NCC2(NC(=O)CN3CC=CC3)CCCCC2)COc2ccccc21 C1(NC(C2OCCN(C(COCC)=O)C2)=O)CCN(OC)CC1 c1(C(N2CC(C(C)C)N(C(c3ccoc3)=O)CC2)=O)cccn2nnnc12 N1(C(c2c(CC)occ2)=O)CC(N=c2[nH]nco2)CC(C)(C)C1 N#CC1(C(N2CC(F)CC2COc2ccc(Cl)cc2)=O)CCCNC1 C1(CC(=O)NC2CC(=O)N(c3ccc(Cl)cc3)C2)CN2CCN1CC2 C1(CNC(CC(C)OC)=O)CC(OC)CN1C(c1ccc(-c2cnn(C)c2)o1)=O C1(NC(C)CCCCc2ccccc2)CCCC12CCCCO2 c1(CC)ccc(O)c(C(=O)NCC2CN(C(=O)C3=CCOCC3)CCN2C)c1 CCC(CC)CCC(=O)N1CC(NC(c2oncc2C)=O)CCC1C N1(C(C(C)CC(N)=O)=O)CCC2CN(C(C3CCCN3C3CC3)=O)CC2CC1 c1(C(=O)Nc2ccc(OC)c(C)n2)cc2ccccc2[nH]1 N1(C(C(CC)C2CCOCC2)=O)CCC2(CC1)CCN(C(=O)C(C)N(C)C)C2 C1(NC(C2(C=C)CCC2)=O)CC2CC(NC(C3(O)CCC3)=O)CC12 C1(C(=O)NCc2nc(C)[nH]n2)CCCCN1C(C1CCO1)=O C1(CC)CN(C(c2ccnc(CO)n2)=O)CCC1NC(c1cscc1OC)=O C=CCC(CNC(c1nccnc1CC)=O)C(=O)NCc1cccc(O)c1 S(=O)(=O)(c1ccc(NCC(c2cnn(C)c2)(C)C)cc1Br)NCCC C(=O)(CC(C)CC(C)(C)C)N1CCN(C(c2ccc(C)c(C)c2)=O)C(CC#N)C1 c1(C(=O)NCC(N(C(CCCCC#C)=O)C)C2CC2)ccc2c(c1)C=CS2(=O)=O N1(C(CCC(C)OC)=O)CCC2C(C(=O)NCC3(O)CC(CO)C3)C2C1 C1(C(=O)N(CC(N(C(=O)CNC=O)C)C2CC2)C2CC2)OCCCO1 C=CCC(CC)C(=O)NC1CCCC1NC(=O)CCOCC1CC1 CC1C(=O)N(C)CCN1C(C1CC2CC2N1Cc1cccc2c1OCC2)=O S(=O)(=O)(c1ccc(Cl)nc1C)N1C(COC)CN(C(c2scc(C)c2Cl)=O)CC1 CC1=C(C(=O)N2CCCC2C2(NC(=O)C(O)C3CC3)CC2)C(C)(C)CCC1 C1(C)(CNC(C2C(CC)C2)=O)CCCN(C(=O)C(CC(C)C)N(C)C)C1 c1(C(=O)NCCC(C)NC(C2CCN(C)C2)=O)cnc2occc2c1 C(=O)(C=CS(F)(F)(F)(F)F)NCC(C1CC1)NC(c1cccc(C)c1F)=O N1(C(C(C2CCN(C(C3(O)CC3)=O)CC2)C)=O)C2CCC1CCSC2 c1(OC)ccc(CCCC(=O)NC2CCCCC2CNC(=O)CCCSC)cc1 c1(C(=O)NCCC2CC(NC(C(COC)OC)=O)C2)nccc2cccnc12 Cc1ncc2n1CCC(C(=O)NCCC1CCCN1CC1CCCCO1)C2 CCC(CC)(CCNC(=O)CCCCSC)NC(=O)C=Cc1cocn1 CCC(CC)C(=O)N1CCC(N2CCN(C(=O)CCC(=O)OCC)CC2)C1 N1(C(c2nn(C)c(F)c2)=O)CC(NC(c2c(F)cc(F)cc2F)=O)C(C2CC2)C1 c1(C(N2C(COC)CN(C(=O)CC3OCCCO3)CC2)=O)ccc([N+](=O)[O-])cn1 n1(CC(N2CC(NC(C3CCC4(C3)N=N4)=O)C2)=O)nnc2c1CCCC2 C(=O)(C#CC1CCOCC1)NCC(C1CCOC1)NC(=O)CCc1cscn1 N1(C(CSCC(N)=O)=O)C2CCC1CN(C(=O)CC(F)(F)C(F)(F)F)C2 N1(C(CSC)=O)CC(F)(F)CC1(C)CNC(c1cc(-c2ccns2)on1)=O c1(OC)ncc(N(C)C(c2scnc2C(C)C)=O)cn1 C1(CNC(C(C)(C)N(C)C)=O)C(C2CC2)CCN1C(c1nccn2nccc12)=O c1(C(=O)NC2CCC(C(=O)NCc3ccc(C)o3)C2)ccc2ccoc2c1 C1(CC(=O)NCCC2(O)CN(C(C3(CCOC)CCC3)=O)C2)CCCCC1O C1(NC(c2cc[nH]n2)=O)(CNC(c2csc3cncn23)=O)CC2CCC1C2 c1(OC(C)=O)ccc(C(=O)NC2(CC(CC(=O)NC3CC3)C3CC3)CCC2)nc1 c1(OCCOC)ccc(NCCC2CC2(F)F)cc1 C(CCN(CCC(C)C)C(=O)Cc1nnc(C)o1)(C(C)C)NC(C(C=C)O)=O C=CCC(C)(C)CC(=O)NCC1(COC)CN(C(c2ccc[n+]([O-])c2)=O)C1 C(=O)(CC(C1CCC1)C1CCC1)NC(C1CC(OC)C1)C C(CCCCCNC(=O)C(N1CCOCC1=O)C)N(C(C1OCC(C)C1)=O)C N1(C(c2cn(C)nc2)=O)CCC2CCCC12C(=O)NCCC(C)(C)F c1(NC(C(C)NS(CC)(=O)=O)=O)c(NC)ncnc1Cl CC1CC(CCNC(=O)CC2(NC(=O)CC3CCCC3O)CCC2)CCO1 c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)CC2CC2)cc2oc(C)cc2[nH]1 c1(C(=O)NC(CCNC(CN(S(N(C)C)(=O)=O)C)=O)C)ccc(C#N)nc1C c1(NC(=O)C(N2CCN(C(=O)CCCCCl)CC2)=O)cc(F)ccc1F c1(C(=O)NCC2N(C(CCCC#C)=O)CC(OC)C2)ccc(C)c(CO)c1 CCC(C(c1nnnn1C(C)C)NCC1(C(F)(F)F)CC=CC1)=Cc1ccsc1 C(C)(C(C)(C)C(=O)NC1(C2CCC2)CC1)NC(C(C)OCCC=C)=O c1(CC)cc(N)ccn1.C1C(CO)NC(=O)C2CC2CC(=O)N1 c1(CC(=O)NC(C(=O)NC(C(C)(C)OC)C)CC2CC2)cccc(F)c1 N1(C(CC2(OC)CCCCC2)=O)CC(CNC(=O)CCCCCF)CCC1C C(=O)(CCCC(=O)C(C)(C)C)NC(CCCNC(C(CCCCC)O)=O)C c1(NC(=O)NC2C(C(=O)NC)CCCC2)ccc(Cl)cc1C(F)(F)F C1(CN(C(C2C(C=C)C2)=O)C)CCCN1C(c1conc1C)=O C(=O)(CC(N)C(F)(F)F)N(CC(C(=O)NC1(CCC)CCC1)(C)C)C Cc1cc(N(CC(O)CN(C(=O)Cn2cncn2)C)C)nc(CC2CC2)n1 N1(C(CC(C)(C)C)=O)CCC2(C1)CN(C(C1CN3CCCC3CO1)=O)C2 c1(C(=O)NC2CN(C(CNC(C)=O)=O)CC2C)ccc2c(c1)-c1ccccc1C2 c1(C(=O)NC(CN(C(=O)CNC(C)=O)CC)C)ccc(-n2nc(C)cc2C)cc1 C(=O)(CC(C(F)F)NC(C1CC1(F)F)=O)NCCC(=O)OCC N(C(=NCCC1(OC(C)=O)CCOCC1)NCC1CCC1)CC(C=C)C CCCC(CC)C(=O)N1CCC(CCNC(C2(F)CCN(C)CC2)=O)C1 c1(CC)cccc(C(=O)NC2CCCC2NC(=O)CC2CCC2OC)c1O CC(C)CC(C(=O)NC1CCN(C(C2C(C3CC3)C2(F)F)=O)C1)NC(N)=O c1(C(=O)NC2C(OC)CN(C(CNC(CC)=O)=O)C2)cc2sccc2s1 c1(OC)ncc(C(N2CC(O)C(O)C2CNC(=O)CCCC2CCC2)=O)c(C)n1 C=CCCCC(=O)N(CCC(=O)NC(CC)C(C)(F)F)CCO N1(C(CCNS(CC)(=O)=O)=O)CCC(NC(=O)C(C)(C)c2ccncc2)C(C)C1 Cn1cc(S(N)(=O)=O)c(C(N2CCC(O)(CNC(C3C4CCCC34)=O)CC2)=O)n1 C1(NC(CCC=CC(C)C)=O)CN(C(c2ccc(C#N)o2)=O)Cc2nccn2C1 C1(CN(C(C2C(C)(CC)C2)=O)C)CCN(C(c2ccc(CO)cn2)=O)CC1 C1(S(C)(=O)=O)(NC(=O)NCCCN2CCCC(C)C2)CCC1 NS(=O)(=O)N1CCC(C(=O)NCC2CN(C(C3CCN4CCCC4C3)=O)C2)CC1 C(=O)(CCCCC(C)(C)C)N1CCN(CC(=O)NCc2ncc(C)[nH]2)CC1 O=C(C#CC1CC1)NCc1ocnc1C(=O)NC1COCCOC1 N1(CC(O)COc2ccccc2)CCN(C(=O)OC)C(C)C1 N1(C(Cc2c(C)nccc2)=O)C2CCC1CN(C(=O)CCC(=O)c1cccs1)C2 N1(C(C(Cc2ccco2)NC(C(C)N=[N+]=[N-])=O)=O)CCCC(F)(C(N)=O)C1 N1(C(c2c(N)cc(Br)cc2)=O)C2CCC1CC(N)C2 C1(C(N2C(C(CNC(c3c(C)csc3)=O)(C)C)CCC2)=O)CCOC(C)(C)C1 c1(C(N2CCC(CCNC(c3nc(Cl)c(Cl)s3)=O)C2)=O)ccc2nonc2c1 C(C1CCCCC1)=CC(N1CCC(CNC(C2(C)CCCS2)=O)C1)=O FC1CCc2[nH]c(=NC3CC=CC3)[nH]c(=NCC3(c4ccccc4)CC3)c2C1 O=C1CCN(C(=O)C(c2ccccc2Cl)c2ccccc2)SC1 FCC(N=c1[nH]c(N2CC3CC3C2)nc2c1COC2)c1ccccc1F C(CN=c1[nH]c(Cl)nc(C2CC2)c1F)(C(C)(C)C)NC(C(C(C)C)NC=O)=O c1(C(=O)NCC2CN(C(C3(NC(C)=O)CC3)=O)C(C)C2)ccc(O)c(F)c1F CC1CN(C(=O)CC2CCC2C)CC1(C)CNC(C1C=CC=CC=C1)=O C(=O)(CCCC(F)(F)Br)NC1CCC(NC(C(CC)C)=O)C1 c1(C(=O)NCC2C(C)CN(C(=O)C=Cc3cn[nH]c3)C2)cc2cncn2c(O)n1 c1(C(C(=O)NC(C(C)NC(C2(CC#C)CCC2)=O)CO)C)cc(C)cc(F)c1 C1(C(=O)NCC(C)N(C)C)C=CCN(C(=O)CC2CCC(O)C2)C1