SMILES N1(C(Cc2cc(C)cc(F)c2)=O)CCC(C)N(C(C2CC3C(C2)C3(F)F)=O)CC1 c1(C(=O)NC2C(CNC(C3N(C)CCC3)=O)CCC2)ccc2c(c1)CCC2 c1(OC)ccnc(C(=O)NCC2CC(C)N(C(=O)Cn3cc(CO)nn3)C2)c1C C1(OC)CN(C(=O)CN2CCC(C)CC2)CC1NC(C1CCCN(C(C)C)C1)=O Cc1nn(C)nc1C(=O)NC1COCC1CNC(=O)CC(C)c1ccccc1 C1(O)(C(C(=O)NC(C)Cc2cn[nH]c2)NC(CCCOC(C)C)=O)CCCCC1 C(=O)(N=c1[nH]c(Cl)ncc1C)c1c(C(=O)Nc2ccc(CC)cn2)scc1 C(=O)(CCCCCSC)N1CC(N(C(=O)C=C(C)C(C)(C)C)CC)C(O)C1 C(=O)(C(C(C)O)NC(c1cnn(CCNC(c2ccncn2)=O)c1)=O)OC c1(C(N2CCC(CO)CC2)C(=O)NCCSC2CCCCC2O)ccc(O)nn1 c1(C(C)C)cc(C(=O)NC2CCCC(NC(=O)CN(CC(C)(C)C)C)C2)nn1C Cc1cc(C(=O)NCC2CC2CC(=O)NCC2CCCC2C)ncc1F Cn1cnnc1CCCNC(=O)C#CCNC(c1nccn1C)=O N1(C(CS(=O)(=O)NC)=O)CC(C(=O)NC2(CO)CCC(C)C2)CC(C)C1 c1(C(N2CCCCC(Nc3c(C#N)c(Cl)ncn3)C2)=O)cc2cccc(F)c2o1 Cc1cc(-c2cncc(C(=O)Nc3nc(C4CC4)c(Br)s3)n2)cc(C)c1 C1(C)(C(=O)NCC2N(C(c3cc(C)sn3)=O)CC2)CC(C)OC(C)C1 CCC(CN=c1[nH]c(=NCC2=CCCC2)[nH]c2ccc(Cl)cc12)n1cccn1 c1(OC)cc(Cl)ccc1CNC(C1(C)CCCN1Cc1cccnc1OC)=O C1(O)(C(=O)NC2CN(C(c3c(OC)c(C)cs3)=O)CC2O)CCC(C)(C)CC1 c1(CC(=O)NC2CCN(C(C3C(CC)CCC3)=O)C(C)C2)nnc2n1CCOC2 N1(C(CCC=C=C)=O)CCn2ncc(CNC(c3nnc(O)nc3O)=O)c2C1 C(=O)(CC(O)C(C)C)N1CCC(C(C(=O)NCCc2ccn(CC)n2)C)C1 c1(CC)ncc(C(=O)NC(C)(C)CNC(C2CC2CF)=O)s1 c1(C(=O)NC23CN(C(c4c(CC)c(C)ccc4)=O)C(C2)C3)cc2ccccn2n1 C1(NC(Cc2c(C)nn(CC)c2C)=O)CN(C(c2ccncc2)=O)CC12CCC2 c1(CC)cncc(C(=O)N(C2(CCCCO)CC2)C)c1.C12COCC1C(=O)N2 c1(C(=O)NCCCC2CCN(C(C(OC)OC)=O)CC2)cn2ncccc2n1 Cc1csc2c(N3CC(CC(C)NC(=O)Cc4ccco4)C3)ncnc12 N1(C(CCC)=O)CCC(NC(c2nccnc2Cl)=O)C(F)C1 N1(C(C(CC)SC)=O)CCC2(CCCC2N2CCC3(CC2)CC(C)=NO3)CC1 O=C(CCCC1CCC1)NCC1CCC1NC(=O)C(C1CCCCC1)O CC1(C)CC(NC2CCC2)CN(Cc2cc(N)n(-c3ccccc3)n2)C1 N1(C(C2=C(C)OCCC2)=O)CC2CCCCC2(NC(=O)C=C(Cl)Cl)C1 c1(OC)ncc(F)c(N2CC(CNC(c3ccc(F)c(C)c3)=O)(OC)C2)n1 C1(C(N2CCCC(CC(=O)NCC(c3ncon3)C)C2)=O)CCCC1C1CC1 N1(C(C2(CC)CC2(F)F)=O)CCCN(C(=O)C(C)(F)CC)CC1 CCC(C)(COC)C(=O)NCC1CCC1NC(c1cc2n(n1)CCC2)=O c1(NC(CCN(C(=O)C(F)CC2CCC2)C)=O)cnc2ccnn2c1 C1(C(N(C2CCC2O)C)=O)CCCN(C(c2cnnc(O)c2)=O)C1 CS(=O)(=O)c1cncc(C(=O)NC2CCCN(C(C34COCC3C4)=O)C2)c1 N1(C(COC(CC)C)=O)CCC2CCN(C(c3c(O)cc(F)cc3F)=O)CC2C1 N1(CC)CCC(N(C(c2ccc(COC)s2)=O)CC)C1 c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC1CN(C(=O)CC(C)C2CC2)C1 C1(CNC(C2C=C(C)CS2)=O)CN(C(c2cc(C)nn2C)=O)CCC12CCC2 C1(C(N2CC3C(CNC(c4cc(C)sc4)=O)(C3)C2)=O)CC2(C1)CC(C)C2 c1(CNCc2cn(-c3c(C)ccnc3)nn2)ccc2nnnn2c1 N1(C(C(=O)NC(C)C)=O)CCC(NC(c2scnc2C(C)(C)C)=O)C(F)C1 Nc1cc(C(=O)NCC2(NC(=O)CC3(O)CCC3)CC2)cc(F)c1 C1(CC(=O)NCC2(O)CN(C(c3cc(N4CCC4)ccn3)=O)C2)CC(=O)NC1=O N1(C(CNS(NC)(=O)=O)=O)CC(CNC(=O)Cc2nonc2C)N2CCC1C2 c1(OC)ccc(Cl)c(C(N2CC(NCc3nc(C(N)=O)co3)C3(CC3)C2)=O)n1 c1(OC(F)F)cc(C)cc(F)c1NC(c1ccnc(OC)c1)=O.CO CC1(C)C(NC2CCC23CCCC3)CC1O N1(C(C2(CCC)CC(=O)C2)=O)CC2(CC(CC(=O)NCC(C)C3CC3)C2)C1 C(C(CC(=O)NCC1C2CCCC12)NC(=O)CN1CC(=O)NC1=O)OC CC1=NOC(C(N2CCCC2CN(C(=O)C=CCN2CC3CC3C2)C)=O)C1 C1(C(=O)NCCCNC(CP(C)(C)=O)=O)CC1C1(C)COC1 N1(CC(=O)NC(C(C)C)CNC(C2CC(C)(F)C2)=O)CCNC(=O)C1 S(=O)(=O)(c1cnc2ccoc2c1)N1CC(C)N(S(C)(=O)=O)CC1 C1(C(=O)Nc2c(C(=O)OC)[nH]nn2)CCN(C(=O)OC(C)(C)C)CC1(C)C N1(C(CC)=O)CCCC(C(N2CCC3C(NC(c4ncn(CC)n4)=O)C23)=O)C1 c1(C(=O)NCC(CC)NC(C2CC(C(F)F)C2)=O)cnn(-c2ccncc2)c1C CC1CC(NC(C2(C)CCN(C)C2=O)=O)CCN1C(=O)Cc1cc(Cl)cc(Cl)c1 C(=O)(C(CCCCN)CC(F)(F)F)CC=CCNC(c1cn(C2CC(N)C2)nc1)=O C(C(N=c1[nH]c(=N)[nH]c(=NCc2cccc(C(N)=O)c2)[nH]1)C(C)C)OCC N1(C(c2nn(CC)nc2C)=O)CCCC2(CCN(C(=O)CCNC(C)=O)C2)C1 C1(NC(C(C)(N(C(c2nc(OCC)oc2)=O)C)C2CC2)=O)CC2COCC2C1 c1(C(=O)NCC2CCCN(C(C(C)SCC)=O)C2)c(OC)cc(Cl)cc1F C(CCN=C(NCc1ccc(SC)o1)N1CCC(C(F)(F)F)(SC)C1)OC Cc1ccc(N2CCCC2C(=O)NCC(N2CC(N3CCNCC3)C2)=O)cc1 N1(C(=O)OC(C)(C)C)CC2CC(C1)C(CO)C2Nc1[nH]c2cnccc2c1Cl C(=O)(C(C#N)C(C)(C)C)NC(C)(C)CCNC(=O)Cc1cncc(O)c1 N1(C(C(=O)NC(C)C)=O)CC(C)(C)OCC1CNC(C1(C#N)CC1)=O C(C1=CCN(C(C2CC(C3CC3)=NO2)=O)CC1)NC(c1ccc(=O)oc1)=O c1(C(=O)NCCC(=C)CNC(C2(C)CNC(=O)C2)=O)ccncc1Br CC1CCN(C(c2csc(CNC(C3(N4CCCC4)CC3)=O)c2)=O)CCO1 C1(C2CCN(C(=O)C(C)(C)C(C)O)CC2)(NC(C(CCC)N(C)C)=O)CC1 N1(C(CC(n2c(CC)ncc2)C)=O)CC2CCN(C(=O)CCN(C)C(C)=O)CC12 C1(NC(C=CC)=O)CCSC12CN(C(C1CCCN(c3nccs3)C1)=O)C2 N1(Cc2c(C)nn(C)c2C)CCN(C(c2ccc(C#N)cc2)=O)C2(CC2)C1 N#CC1CN(Cc2cnn(C3CC3(F)F)c2)CC1NC(=O)C(N)=O C1(NC(c2c(Cl)cn(CC)n2)=O)CC(CNC(C2SCCS2)=O)C12CCC2 C#Cc1cc(C(N2CCC(CCNC(=O)C(C)CCC)C2)=O)cc(N)c1 C(=O)(CC(C)(C)C(=O)NCC1(NC(=O)CS(N)(=O)=O)CCOCC1)OCC c1(OCC)cc(C(=O)NC2CCCN(C(=O)COC3CC3)C2)cc([N+](=O)[O-])c1O C1(CC=C)(NC(c2ncccc2CC)=O)CCCN(C(C2CCOC2=O)=O)C1 C1(C(N2CC(O)(CNC(CC3C(C)CCO3)=O)C2)=O)CC(=O)NC(=O)C1 C1(NC(C2C(C(C)NC(C(CC)CN(C)C)=O)C2)=O)CC2(CCCCO2)C1 CCC(C)CCCC(=O)NC(C1CCCN1C(c1cccc(C#N)c1C)=O)C Cc1ccc2c(CCNC(N3CCC(O)(Cc4ccccc4)C3)=O)cn(C)c2c1 C=Cc1cc(C(=O)NC(C)C(C)NC(c2cc(CSCC)on2)=O)cc(F)c1 CC1CCCC(C)N(C(c2conc2CNC(=O)C(C)n2cccc2)=O)C1 C1(C(=O)NCC(=C2CN(C(CC3(CSC)CC3)=O)C2)F)CCCCN1C(C)C c1(C(N2C(CNC(c3c(C)csc3)=O)C(C)(C)CC2)=O)cccc2c1C(=O)CC2 c1(C(=O)NC(CC2CN(CC(c3ccc(CC)o3)=O)C2)C)cc(O)nc(O)n1 CC(O)C(=O)N=c1ccn(CC(N2CC(F)C(F)C2)=O)c(O)n1 C1(NC(C2N(C(C=NOC)=O)CCOCC2)=O)CCOCC12CCC2 N1(C(C(C(C)CC)N(C(CC=CC)=O)C)=O)C2CCC1CC1(CC1)C2 c1(NC(c2c(Cl)cnn2C)c2n(CC=C)nnn2)sc(Br)c2c1OCCO2 C1(CC(=O)NC(CNC(C2(SCC)CC2)=O)C(C)C)CCCCCO1 C1(NC(CCc2nc(C)sc2)=O)C2COCC1CN(C(c1cnncc1C)=O)C2 C=CC1CN(C(C2C3CC4C(C3)C24)=O)CC1NC(=O)C(C)CC(N)=O CC1(C(=O)NCc2ccnc(Oc3ccc(F)cc3)c2)CC=CCO1.C1CN1 CC(C)=C=CC(=O)NCCCN(C(=O)CC(C)C)C1CC1 C1(C(=O)OC)CCC(NC(C2CC(n3cc(CNC)nn3)C2)=O)CC1 CCC(CC)(CO)C(=O)NCCC1CN(C(c2cc(Br)n(C)c2)=O)C1 CC(C)(C)C1=NOC(C(N2CC=CC(NC(c3ccnc(Cl)c3F)=O)C2)=O)C1 C1(NC(c2cc(C3(C)CC3)n[nH]2)=O)CC(NC(=O)C(=O)C(C)(C)C)C12CCC2 N1(C(Cc2cc(C)sc2C)=O)CCN(C(=O)CNC(c2ccco2)=O)C2CCC12 C(=O)(C(C)CCCCCC)N1CC(C(N2CC(C#C)(F)C2)=O)C(C)(C)C1 c1(CNC(c2n(CCOC)nnn2)CCCSC)ccnc(Cl)c1Cl C1(C(N(C(CCCC)C)C)=O)CN(C(=O)Cc2c(C)cnn2C)CCN1C c1(OC)c(Cl)cc(C(=O)NC23CCCC2CN(C(c2cnccn2)=O)C3)nc1Cl Cn1cnc(C(N2CC(O)(C(F)C(=O)NCC3CCCS3)C2)=O)c1 CCCC(CCCNC(c1cc(C(C)(F)F)ccn1)=O)NC(C1(N(C)C)CC1)=O N1(C(C)=O)CCCC1(C)C(=O)NCC1(O)CCN(C(=O)CCCC2CC2)C1 C#Cc1c[nH]nc1C(=O)NCC1CC(F)CN1C(c1ccoc1Cl)=O c1(C(=O)NC(CC=C)CNC(C2CC(C(C)C)C2)=O)ccc(C2CC2)cc1C c1(CC)ccc(C(=O)NC2CCC(C)N(C(c3cc[nH]n3)=O)C2)cc1CC N1(C(c2nc(C(=O)OC)oc2)=O)C2CCC1CC(NC(C1(C#N)CC1)=O)C2 c1(NC(C2(C)CCC3(CC2)CC3)=O)nc2c(F)cc(Cl)cc2s1 C(CC(CC)C(=O)NCC(O)CC(=O)NC(C)C(C)C(=O)OC)=CC C(=O)(CCCC(C)(C)C(=O)N1CC2(CNC(=O)C(C)SC)CCC1C2)OC n1(CCOC)cc(C(=O)NC23CC(C2)N(C(=O)CCc2nc(O)n[nH]2)C3)c(C)n1 c1(C(=O)N(c2cnc(C3CCNC3)s2)C(c2ccco2)=O)ncc(Cl)cn1 C1(N(C(c2cc(CCO)on2)=O)CC)CCCN(C(=O)Cn2ncc(Cl)c2C)C1 c1(C(=O)NCC2C(C)CCN(C(=O)C(C)(C)CO)C2)ccc(S(N)(=O)=O)nc1 C(=O)(C(C(C)(C)C)NC(N)=O)NCC1(NC(C=Cc2cnc(C)s2)=O)CC1 CCCC(CCCNC(C1CCC(O)CC1)=O)NC(=O)CCF CC1(C)CCN(C(c2csc(Cl)n2)=O)C1C(=O)NC1C(=O)OCC1CO CCC(CC)C(c1nnnn1Cc1ccco1)NC1CC1CC(C)C CC1CCC(NC(=O)CC2(O)CCCOC2)CN1C(=O)Cc1ccon1 CN1C(C(N)=O)CCC1C(N1CCOC(CNC(C2(C(C)(C)C)CCC2)=O)C1)=O C1(CNC(CC(C)(C)NC(=O)CCNC(=O)CO)=O)CC2(CCCO2)C1 c1(C(N2c3ccoc3C2=O)=O)cc(F)c(Cl)c(Cl)c1.N1(CCO)CCN(C2COC2)CC1 C1(CC(=O)NC2CC(C#N)C2)CCC(C(=O)O)CC1 c1(C(N2CCC(NC(CC3C(C)(C)OCC3)=O)(CF)C2)=O)cncc2ccccc12 CC1CN(C(c2c[nH]c(=S)cn2)=O)CCN1C(c1cocn1)=O c1(CN2CC(OC)C(NC(c3cc(C)cc(C)n3)=O)CC2)ccc(S(N)(=O)=O)o1 c1(CC)nc(C)oc1C(=O)NCCOCC(=O)NCC(O)CO C1(C(=O)NCC(CCNC(C=CCCC)=O)OC)CCc2c[nH]nc2C1 c1(CCC)ccc(CC(C)C)cc1.C12CCN(C1)CC(O)COC2 c1(OC(CC)C)ccc(CN2CC3C(CNC(c4cscc4C)=O)C3C2)cc1 c1(C(=O)NC2C(NC(=O)CSC3CCCO3)C2)cc(C(F)(F)F)ccc1F C12(C(N3CC(CNC(CC4(C)CC4(F)Cl)=O)C3)=O)CC3CC(C1)CC(F)(C3)C2 C(CCCC(=O)NC(C1CC1)C1CC1)NC(CC(C)C)=O N1(Cc2ccc(C(=O)OC)cc2)CC2CN(C(c3cc(O)ccc3Br)=O)CC12 C(C(=O)NC1CN(C(c2ccncc2O)=O)CC1C)(C(C)C)NC(C)=O c1(OCC)cc(F)ccc1C(=O)N(C)CCn1cc(-c2cncs2)nn1 c1(C(N2CC3OCC(NC(CC4C(C)(C)C4)=O)C3C2)=O)cncc2ccccc12 C(CC(N)=O)(C(=O)N1CCC(C)(C)CC1)NC(c1c(OC)scc1)=O C1(N(C2CCOCC2)C(C(N)=O)=O)C2CC(n3cc(-c4ccncc4)nn3)C1C2 c1(OC)ncc(C(=O)OCC(n2cc(-c3cncc(N)c3)nn2)C)cc1C C(=O)(CS(=O)(=O)C(C)C)NC(CNC(CC(=O)NCC)=O)CC Cc1ccc(Br)cc1CC(=O)NCC1CCCN1Cc1ccc(Br)cc1Br N1(C(C2(F)CCN(C(C3(CCN(C)C)CC3)=O)C2)=O)CC(C#N)C2(CCC2)C1 C(=O)(C#CC1(C)COC1)N1CCC(N2CCN(C(C3C(C)OC(=O)N3)=O)CC2)C1 C1(CNC(C(F)=CCC)=O)CC2(CCC2)CN1C(c1ncc(C#N)cc1C)=O c1(C(N2C(CNC(C(C3CC3)OC)=O)CC(O)C2)=O)[nH]c2ccc(C)cc2c1C N1(C(C2C(=C)C2)=O)CCCC(C)(C(=O)C2=CCCC2)C1 C(=O)(C#CC1CC(F)(F)C1)NC(CNC(CC(CCCC)C)=O)(C)C C1(CCC)(NC(=O)CCc2cc(C)[nH]n2)CCCN(C(=O)CS(=O)(=O)CC)C1 c1(C(=O)Nc2c(SCCC(=O)OC)cccc2)cc(F)c(O)c(Cl)c1 C1(C(=O)NCC(CC=C)(C)C)CC(C)(C)CN1C(c1ccnc(O)c1F)=O c1(CNC(CN(CC)CC)C(=O)OC)ccc(C(O)C(F)(F)F)cc1 C1(NC(C2CCCC2)=O)COC2(CCCN(C(=O)COc3cncc(Cl)n3)C2)C1 CCCC(C)CC(C)Nc1cccc(-c2c(C(CN3CCCCC3)NC)c[nH]n2)c1 c1(CC(N2CCC(C)C(NC(c3cc(Cl)ccn3)=O)C2)=O)cccc2ccoc12 CCCCC(CNC(c1ccc(SC)cc1)=O)NC(c1n[nH]cc1C1CCC1)=O C1(CC(=O)NCC(C)(O)C2CC2)C2CN(C(c3csc(Cl)c3)=O)CC12 CC(C)CC(O)C(C)C(=O)N1CCC(N=[N+]=[N-])(C(=O)NC2CC(N3CCCC3)C2)C1 N1(C(C)C)CCCC1C(=O)NC1CCC1CNC(=O)Cn1cnnc1 c1(C(N2CCOCC(NC(C(CC)(C)C)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 c1(OCCC(=O)N(C(CNC(CN(CC)CC)=O)C)C)ccccc1F N=c1[nH]cnc2c(C(N3CCCC(NC(=O)C=CC4CC4)CCC3)=O)cnn12 c1(OC)cc(Br)ccc1CCC(=O)NC1CN(C(=O)CNC(C)=O)CC1C Cc1c(C(=O)NC(C)(CO)C(=O)NC2CCN(CCF)C2)ccn1C c1(N2CCC(CCNC(=O)CCN3CCCS3(=O)=O)CC2)ncc2ccnc-2[nH]1 N1(C(C2C(C)OC(=O)N2)=O)CCC(F)(C(=O)NCC2CCSC2)CC1 C(=O)(CCN=C(NCCc1cnn(C)c1)NCC1CCCC1OC)NC C#Cc1ccc(NC(C2CCC(CNC(c3coc(SC)c3)=O)O2)=O)cc1 c1(C(CC(=O)NCCn2ccc(C)n2)NC(=O)C(C)C#N)ccccc1Br CC(C)(CC(=O)NCC1CCC1NC(c1cc(F)ccc1F)=O)CC(F)(F)F C(CC(C)C)(C(=O)N1CCC(OC)CC1)ONC(c1c(CC)n[nH]c1)=O N1(C(c2c(C)ncs2)=O)CC(NC(=O)C(C)CC(C)(C)C)CC(C)(C)C1 CC(C)(C#CC(=O)OC(C)(C)C)CNC(=O)Nc1nc(-c2ccccc2)ns1 CC1CN(C(=O)CC2(CS(C)(=O)=O)CC2)CCC1NC(=O)CN1CCNC(=O)C1 c1(OC)c(C(=O)NC2(C)CN(C(c3cc(N)ccc3O)=O)C2)ccc2c1CCC2 N1(C(c2n(CCC)ncc2)=O)CCCC(NC(c2cncc(C(C)(C)C)c2)=O)C1 C1(CC(N2CC(C)(NC(c3c(C)cc(F)nc3)=O)C2)=O)CC(C)CC(C)(C)C1 C12(CNC(C3N(CC)CCCC3)=O)CCC(CC1)CN2C(=O)C(C#N)C(C)C CC1(C)CCC(NC2CC3C(C(=O)NC(=O)CCc4ccc[nH]4)C3C2)C1 C#CCCN=C(NCC(C(C)CC)OC)N1CCc2cc(Br)ccc2C1 C1(C(C)C)CC(C(N2CC3CC2C3NC(=O)Cn2cccnc2=O)=O)CCO1 C1(CNC(C2C(CC)CCC2)=O)CC(O)CN1C(=O)CCCc1ccsc1 C1(CC(C)NCCc2ccc(OC(F)(F)F)s2)CC(C)(C)NC1=O CC(C)(CNC(C1(C)CC2CCC1O2)=O)CC(=O)NCCc1ccnc(O)c1 C12(NC(C(CCCC)C)=O)CC(C)(C1)OC21CN(C(=O)CC(C)C)C1 CC1=C(CNC2CC(NC(=O)OC(C)(C)C)C(O)C2n2cccn2)C(C)(C)CCC1 C1(NC(c2ccncc2O)=O)CCCCN(C(c2cc(Br)cnc2Br)=O)C1 C1(N(C(=O)CCC2CCCOC2)CC)CCCN(C(C2CN(CC(C)C)C2)=O)C1 N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CCN(C(=O)Cc2occc2C)C(CO)C1 CC1(C)COC(C(=O)NCC(C2CCC2)NC(=O)CCN2CCOC2=O)C1 N1(C(c2c(CSC)n(C)nc2)=O)CCN(C(=O)C(=O)NC2CC2)C2CC12 c1(C(=O)NC(C2CCCCC2C)C)cc2c(cc1F)NCCC2 S(=O)(=O)(c1ccc(N2CC3CC2C3)cc1Br)N(C1C(C)C1)CCO N1(C(=O)NC2CC(n3cc(C4CC45CC5)nn3)C2)CC2C(C1)C2(F)F C1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)O)CNC(=O)C(C)(C)C1 C(=O)(C(C(C)CC)N(C(=O)Cc1cc(CC)no1)C)NCC(C#C)CC CCC(C#N)C(=O)NCC1CCCN1C(=O)CCCSC(C)(C)C N1(C(C(c2ccccc2)NC(Cn2ncc(C#N)c2)=O)=O)CC2COCC(C2)C1 C1(Cn2cc(CCCCCCC)nn2)CC(C)(C)CCN1C(=O)CC(F)(F)CC N1(C(=O)C(F)(F)CN2CCCC2)CCN(C(=O)CCc2cncnc2)C(CO)C1 CCC(C)CC(C(=O)NC1CCCCCC1)NC(=O)CC1(N(C)C)CCC1 C1(NC(C2(CSC)CC2)=O)CCOCC1C(=O)NCc1ncnn1C N1(C(c2c(C(N)=O)ccs2)=O)CCCC2(CCCN2C(c2ccncn2)=O)C1 N1(C(c2cnc(CC)o2)=O)CCC2CN(C(c3ccccc3)=O)CCC12 c1(C(=O)NC2CN(C(C=CCCC)=O)CC(O)C2)cc(F)c(F)cc1OC C1(C(=O)NCC(C)(CO)NC(c2cnn(C)c2C#N)=O)(OC)CCCC(C)(C)C1 C(=O)(C1CCc2c[nH]nc21)N1CC2C(CN3C(C)CCCC(C)C3)(CCC2)C1 c1(OCC)ccccc1NC(=O)CN(CC1CC1)CC(C1CC2C=CC1C2)=O CC1CN(C(c2nscc2I)=O)CCCN1C(=O)CCC1CC1 n12cnc(c1)C(=O)NCC2.C(C)(CCCO)NC(CCC)=O c1(C(N2CC(C(C(=O)NCc3ccco3)OC)C2)=O)cncc(F)c1C C(=O)(C1CCc2nnc(C)n21)NC(CC)CNC(c1csc(C(C)C)n1)=O C(C(O)C(C)(C)C)N(C)C(C1(C)CC=CCC1)=O.C1=CCNC1=O c1(C(CNC(C)=O)NC(CC(=C)I)=O)ccccc1F CC1CN(C(=O)CC2(O)CC2)CCN1C(c1ccc(-n2cccc2)cc1)=O C12(C(=O)NCC(C)N(C(=O)CC3OCCO3)CC)CC3CC(C1)CC(F)(C3)C2 C(C(C)(C(=O)NCC(C)(Cn1cccn1)NC(C1CCCN(C)C1)=O)OC)OC c1(OC)ccccc1-n1ncc(C(=O)N(c2cccc(F)c2)C)c1C C(CC(C(=O)N(C)CCc1ccccc1)NC(=O)C(CC)OC)OCC C1(CN(C(C2C(C(=O)OC)C2)=O)C)COCCN1C(c1ccoc1C(C)C)=O C1(F)(C(N(CC(C)O)C2CC2)=O)CCN(C(=O)CC2(N(C)C)CC2)CC1 Cc1cc(F)cnc1C(=O)NCC1CC(CNC(c2ccccc2CO)=O)CO1 CC12CN(C(c3cccc(-c4ccccc4)n3)=O)CC1(C)CS(=N)(=O)C2 C1(c2cccc(Cl)c2)CCN(CCC(=O)N(C2COC2)NC(=O)OC(C)(C)C)CC1 C=CC(CCC)CC(=O)N1CCC2(C(=O)NCCC3C=CCC3)CCCC12 N1(C(C(C2CC2)OC)=O)CC2(NC(=O)Cc3csc(Br)c3)CCC1CC2 C1(CNC(C#CC(C)C)=O)CC2CCC(C1)N2C(=O)CCC(=O)c1ccc[nH]1 N1(C(C(CC=C)CC)=O)CCC2(CC1)CC2C(=O)NCC1C=CCOC1 C1(CCOC)(NC(=O)C=Cc2ccoc2)CCN(C(=O)Cc2nnc(C)o2)C1 C1(CC(=O)NCC2CCC(C)CN2C(C2(F)CCCC2)=O)CCCC2(CCC2)O1 c1(C(N2CC(C)(C)C(NC(c3ccc(O)cc3)=O)C2)=O)ccc(P(C)(C)=O)cn1 S(=O)(=O)(c1cnc2sccc2c1)NCC1CC(c2cccc(C)c2)C1 C12(CNC(c3c(CC)n[nH]c3)=O)CCC(CC1)N(C(C1(C)CCC13CCC3)=O)C2 c1(CC(=O)N(C2CN(C)C2)C)ncccc1NC(=O)OC(C)(C)C C(C(=O)NCC(C)(O)CNC(c1ncnn1CC)=O)(C(C)C)OCC CC(C)CC(C(=O)NCC1C=CCOC1)NC(c1cnc(S)nc1)=O C1(N(C(C23CC(C2)C3)=O)CC)CCCN(C(=O)CC(=O)N(C)C)C1 CC1CCn2cc(C(=O)NC3CCN(C(C4(C#N)CCOC4)=O)CC3F)nc2C1 CN1C(=O)CCC1(C)CNC(C1(CO)CCN(C(C2CCCC2C2CC2)=O)C1)=O c1(CCNC(N(C2CCCN(c3ccccn3)C2)C)=O)cccc(C(F)(F)F)c1 C(=O)(CCCS(C)(=O)=O)NCCC(C)CCNC(=O)CN(c1ccnc(Cl)n1)C CCC(CC)CCCC(=O)NCC1(C)CCCN1C(=O)Cc1c[nH]ccc1=O c1(CC)nc[nH]c1C(=O)NCC(C)(C1CC1)NC(=O)CCc1ccc(C)s1 C1(O)(NC(C(CN(CC(=O)NC)CC)O)=O)CCOCC1 C12(CNC(CC(CC)OC)=O)CCN(CC1)CC2.C1(CO)C(=O)N1 C=CCC(C(=O)N1CCCCC1CCCO)NC(=O)C(C)SCCCC C(=O)(C1(C)CCc2ccccc21)NCC(CC)NC(C1(F)CCC1)=O N(C1CCCOc2ccc(Br)cc21)C(=O)NC1CN(C)CC1c1ccccc1 C1(C(C(=O)NC2C3CCN(C(c4ccnnc4)=O)C23)O)CCS(=O)(=O)CC1 C1(NC(CCC(N)=O)=O)CC2CC(C1)N(C(=O)CCC(=O)OC(C)(C)C)C2 C1(C(=O)NC(C(=O)NC(C(CCC)O)CO)CCOCCO)CCC2(CCC2)O1 C1(CC(=O)NCC(CC)NC(c2cc(O)ccc2N)=O)CCCC(C)(C)O1 c1(C(C)C)ccc(C(N2CC(O)(CNC(c3ccc(-c4ccco4)s3)=O)C2)=O)o1 CN1CCN(C(c2cccc(C(=O)NCc3cccs3)c2)=O)C(C(C)(C)C)C1 c1(C(=O)NCC2(C)C(C)CN(C(=O)C(C)(C)C(C)O)C2)c[nH]c2ccc(F)cc12 c1(OC)cc2c(cc1OC)CC(C(N1CCN(C(C)=O)CC1)=O)C2 c1(CC)ccc(CCC(=O)NCC23CC(NC(C4CC(=O)C4)=O)(C2)C3)cc1 N1(C(C(c2ccccc2)=O)=O)CCN(CCc2cccc(Cl)c2Cl)C2CC12 C1(C(=O)NCC(CC(C)C)NC(c2cc(O)cnc2Cl)=O)(OC)CCC(C)CC1 C(CN=C(NCc1cn(C)c(=O)n1C)NCC(C)CCC)COCC c1(OCC)cc2ccccc2cc1C(=O)NC1CC2(CCC2)CN1C(C)=O c1(C(=O)NCC2CC(C)C2)ccc(S(=O)(=O)N2CCC(C(F)(F)F)C2C)c(Cl)c1 C(=O)(CCCCCn1cnnn1)NC1(CNC(C2C(C)C2)=O)CCOCC1 c1(OC)ccc(C(N2CCCC(CO)(NC(C3CC3F)=O)C2)=O)cc1S(C)(=O)=O N1(C(C(C)CC2CC2)=O)CCN(C)CC1CNC(C1CCOC1C(N)=O)=O N1(CC(=O)NC2C(C)CCCC2)CCCC(C)(NC(=O)CNC(=O)C(C)(C)C)C1 CCCCC(CC(=O)O)N(C(C1CCCN1Cc1ccccc1)=O)C(C)C C1(C(=O)NC2(CNC(c3nc(OCC)oc3)=O)CC2)OC2CCC1C2 C(=O)(C1CC(=O)OCC1)OC.O(N(C)C(=O)CCC)C(=O)OC(C)(C)C c1(C(N2C(CNC(C(CC)(C)OC)=O)C=CC2)=O)cccc(S(=O)(=O)C2CC2)c1 c1(CC(N2CC(C)OC(CC3CCC3)C2)=O)cccc2occc12 C12(C(=O)OC)CC(C(=O)NC3(CN(C(=O)C(C)n4cccc4)C)CC3)(C1)C2 C1(CN(CC(C)NC(=O)CCn2cccn2)C)CCC1C(F)(F)F C(C(F)(C(=O)N1CC2CCC2(C)C1)C(C)C)NC(c1c(C)cc(CC)o1)=O C(C(CC(=O)NC(C)(CO)C1CCCC1)C1CCC1)NC(C(CC)OCC)=O N1(Cc2nc(C)on2)CCN(C2CCSC2)CC1.N1(C)C(=O)N1 C(C(C(C)(C)C)NC(c1cccnc1C(F)F)=O)NC(CC(C)OC)=O C1(C(C(=O)N(CC)Cc2ccco2)C)CCCN(C(=O)CCC(C)C)C1 C1(CNC(C(CC=C)CC)=O)CC2CCC1N(C(=O)CC(O)C(C)CC)C2 C1(NC(c2c(CC)cco2)=O)C2CCC1N(C(=O)Cc1cnc[nH]1)C2 C1(OCC(=O)NC(C)(C)CCNC(=O)Cc2nc[nH]n2)CCCCCC1 N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CNC(=O)CCC(C)C Cc1[nH]nc(C(N2CC3(NC(=O)CNC(N4CCCC4)=O)CC2C3)=O)c1C N1(C(C2(C)CCC2)=O)CCC(C2(NC(c3sc(Cl)cc3Br)=O)CC2)C1 C1(CC)CCN(C(=O)CC2COCC2NC(=O)CCc2nncs2)C1 O=S(Cc1ccccc1)CCNc1ccnn1Cc1ccccn1 c1(C(=O)NC(C(CO)NC(c2c(F)ccc(OC)c2)=O)C)cc2c(s1)CCCC2 C1(OC)CCCC1C(N1CC(NC(=O)Cc2ncc(C)s2)C1)=O c1(OC)n[nH]c(C(=O)NCCOCCNC(C2CCC(O)CC2)=O)c1Br C1(C(N(C)CC2(O)CN(C(=O)CC3=NNC(=O)C3)C2)=O)CCCc2ccccc2C1 C1(NC(C2CN(C)C(=O)N2)=O)CCC2CN(C(=O)COCC3CCCO3)CC2C1 c1(C(=O)NC(CNC(=O)C=Cc2ccccc2Cl)CO)c[nH]c2cccnc12 C1(C(=O)OCC)CCC(NC(=O)C(=O)NCc2nc(C)c(C)s2)CC1 N#Cc1c(NC(C2CC23CCOCC3)=O)ncnc1Cl C(=O)(CC(C)(O)CC(=O)O)N1CCCC(C(=O)NCc2ccnc(C)n2)CC1 C(=O)(C(C(C)(C)C)C1CCC1)N1CC(N(C(c2cnc(CC(C)C)s2)=O)C)C1 c1(C(=O)NCC2C(OCC)CN(C(c3cc(Cl)no3)=O)C2)c(Cl)ccc(C)c1O N1(C(C(C(CC)C)NC(C2CSC2)=O)=O)CCCC(N=[N+]=[N-])C1 N1(CCc2cn(C(C)(C)C)nc2)CC=CC2COCC12 c1(CC)cc(C(=O)NC(C)CNC(c2ncccc2SC)=O)sc1C c1(CNC(=O)OC(C2(CC3CC(=C)C3)CC2C(=O)O)=O)ccnn(CC)c1=O CCC(CCCC(=O)N1CC2C3CCC(C3)C12)NC(=O)Cc1ccn(CC)n1 c1(C(=O)OC)cccc(CNC(C)(C)CCCF)c1Br N1(C(C)C)CCCC(C(=O)NC2CNC(=O)C2)C1.C12CC(C1)CNC(=O)N2 N1(C(C2C(C)OC(=O)N2)=O)CC2CCCC2(CNC(=O)C(C)CC2CCC2)C1 C1(NC(C(C)C2CCC2)=O)CC2(CCN(C(=O)CCc3cocn3)C2)C1 c1(C(=O)NC2CC(C(=O)OCC)CC2O)cc(S(=O)(=O)CC#N)ccc1F CC(CC(F)(F)F)C(=O)NCCCOCCNC(=O)C(O)C1CCC1 N1(C(Cc2cn(C)nc2)=O)CCC2CCC(NC(C3CC34CCOC4)=O)C1C2 C(=O)(CCCC(F)(F)F)NCC(C)(Cn1cccn1)NC(c1occ(C)c1C)=O N1(C(C(CC(F)F)NC(COCC=C)=O)=O)CC2(COC(=O)C2)C1 Cc1cc(Cl)c(C(=O)NC2CC2NC(c2ccnc(CO)c2)=O)cc1N C(C(=O)N(C)CC1CCCC1)(C(C)O)NC(C(C)CO)=O CC(N=[N+]=[N-])C(=O)NC1CCCCC1C(N1CC(N2CC(O)C2)C1)=O n1(C2N(C(=O)OC(C)(C)C)CCC2)cc(CC=Cc2ccccc2)c(Br)n1 C(=O)(C1CCCn2nccc21)NCCCCNC(c1ccc(OC)c(F)c1N)=O C(=O)(CS(=O)(=O)CC(=O)NC1CCCCC1NC(c1cnc[nH]1)=O)OC C=CCC(CC(=O)NCC1(C)CCCCO1)NC(C1CCCCCN1C)=O C1(NC(Cn2ncn(C)c2=O)=O)CC2CC(C1)N(C(C1COC(=O)C1)=O)C2 O=C(CCCC1CC1)NC1(C(=O)NCCCc2ncco2)CC(CO)C1 N(C(=NCCCn1ccnn1)NCCc1ccccc1Br)CC(C)C C(=O)(C(C)n1cncn1)NCC(C1CC1)NC(C1(CC)CC1)=O CC1CN(C(=O)C(=O)NCCOc2cccnc2)CCC1C c1(NC(C2C(NCc3ccc(OC)c(O)c3)C2)=O)ccc(C(C)C)c([N+](=O)[O-])c1 N1(CCC)CCCC1C(N1CCCC1C(C)NC(=O)Cc1ccc(C)s1)=O N1(C(C)C)CC(C(=O)N(C)CCN(C(=O)CC2CC(O)C2(C)C)C)CC1=O c1(CC(c2cn(CCCC(=O)N(C)C)nn2)O)ccc(F)cc1.C12(CC1)C(=O)NC2 C1(CC(=O)NC(c2cccnc2)C)CCC(NC(c2cnc(C)cn2)=O)CC1 CCC(CC(C)C)C(=O)N1CCC(CCNC(c2ncncc2F)=O)C1 N1(C(c2cn(CCC)nc2C)=O)CCN(C(c2csc(C)c2OC)=O)C2CC12 C(=O)(C1=NN2CCCN=C2N1)N1C(CNC(C(C)SC)=O)CCC(C)(C)C1 c1(C(N2C(CN(C(C3(COC)CCC3)=O)C)COCC2)=O)ccc(C#N)c(Cl)c1 Cc1cc2cc(NC(C3CCN(C(c4ccncc4Br)=O)CC3O)=O)ccc2[nH]1 C(C(CO)(CO)NC(=O)Cc1nocc1C)N(C(C(COC)NC(C)=O)=O)C C(CCCCCCC(=O)N1CC(CNC(c2ncc[nH]c2=O)=O)C(C)(C)C1)SC N1(C(c2c(C)nn[nH]2)=O)CC2(CCCC2NC(C2CC(=O)N(CC3CC3)C2)=O)C1 C1(C(=O)NC(CNC(CCc2onc(CC)n2)=O)C2CC2)CCC(N(C)C)CC1 C1(CNC(C(CC)SC)=O)CN(C(C2(CCF)CCC2)=O)CCC1(C)C c1(CN(C(C2CC2NC(c2nocc2Br)=O)=O)CC)ccc(OC)cc1 n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CN(C(=O)COC(C)=O)CCN2C)n1 C(=O)(CC(O)CC(C)(C)C)NCC1C(C(N2C(C(N(C)C)=O)C=CC2)=O)CCO1 c1(C(N2CCN(CCCN(C(CCC)=O)C3CC3)CC2)=O)c(C)cc(Br)cc1F c1(C(N2CCC(NC(C(CCC)CC)=O)C(F)C2)=O)ccc(O)c2c1CCCC2 S(=O)(=O)(c1cccnc1CN(S(C)(=O)=O)C)NC(c1ccc(C)o1)C C1(NC(CN(C(C)=O)C)=O)CCCN(C(c2cc(C3(Cl)CC3)n(C)n2)=O)C1C C1(O)(CC)CCCN(C(c2ccc(CNC(=O)C(C)=C3CCC3)nc2)=O)C1 c1(C(N(CCCCNC(C2CC2F)=O)C)=O)c(O)nnc2c1CCCC2 C12(C(N3CC4C(C(N)=O)C(C4)C3)=O)C3C4C1C1C2C3C41Cc1cccs1 C1(C(=O)NC2CC(NC(CCc3cc(C)no3)=O)C2)CCC2C1C2(F)F C1(NC(C2C(CC)C2)=O)CC2CC1N(C(C1(F)CCC1)=O)C2 c1(-c2cn(CCC3CN(C(C4C(C)CC=CC4)=O)C3)nn2)ccc2ncsc2c1 N1(C(c2ccnc(OC)n2)C(=O)NC2CCC2)CC(C)CCC12CC2 c1(N2CCC(CNC(C3C(C)=C3)=O)C2)nc2c(cc1C#N)CCC2(C)C c1(CC(=O)NCc2nc(CNC(c3cnc(C)s3)=O)sc2)cccnc1Cl c1(OC)cccc(CC(N2CCCC(NC(=O)C(C)(C)C(N)=O)C2C)=O)c1Cl c1(CC(=O)NCC2(C)CCCN2C(=O)Cc2cc[nH]c2)ccc(F)c(Cl)c1 C(=O)(C(C)(CSC)NC(c1cnc(=N)[nH]c1)=O)NCCN(C)CC C(CCC(=O)NCC1CNC(=O)O1)(C(C)C)NC(C1C(C(=C)C)OCC1)=O c1(C(=O)NC2CC(O)(CNC(c3c(CC)nc[nH]3)=O)C2)oc(COC)cc1C c1(C(N(C(C)CCNC(=O)CCC(F)(F)F)C)=O)cc2c(cc1N)CCC2 C1(C(=O)NCC(C(C)C)NC(C2(C)CC=CC2)=O)CCOC(C(F)(F)F)C1 c1(OC)ccc(OC)c(C(O)CNC2(CO)CC2)c1 N1(C(CCCOCC=C)=O)CC(C)(C)OCC1CNC(=O)C(O)CCCC NCS(=O)(=O)Cc1cnn(CCc2nnnn2Cc2cc(Br)cs2)c1 C1(CNC(CCC)=O)CCN(C(=O)COCc2nc[nH]n2)C1(C)C c1(NC(=O)NC(Cc2c(C)noc2C)C)cccc([N+](=O)[O-])c1F c1(N2C(C(CC)N(C(=O)C=CC3CCCC3)CC)CCC2)ncnc2c1CCC2 CC1(C)CC(C(=O)NC2CC3(C2)CC3NC(c2ccc(C3CC3)o2)=O)CNC1=O Cc1[nH]c2c(CN3CCC(C(=O)OC(C)(C)C)CC3)cccc2c1C N1(C(c2ncc(F)cc2F)=O)CCC2C(C1)CN2C(c1ccn2nccc2c1)=O C1(NC(C(C)CN(C)C)=O)(CO)CCCN(C(=O)C(C)(C)C2CC2)C1 CN1CCCC(C(C2CC2)Nc2ncccc2F)C1.C1(C(C)(C)C)COc2nnnn21 C1(CC(=O)NC(=O)CN(C2CC2)CC2CC(N(C)C)C2)COCCO1 Cc1cccc2cc(C(C)(C)NC(=O)Cc3nc4cc(Cl)ccc4n3C)cnc12 N1(C(c2c(CC)c[nH]n2)=O)CCOC2CN(C(C3(C)CC=CCC3)=O)CC12 N1(C(C(n2c(C)ccn2)C)=O)CC(OC)CC1CNC(C12CSCC1C2)=O c1(C(=O)NC2CCN(C(CCOC(C)C)=O)CC2CO)cc(Cl)c(N)cc1F Cc1sc(N)c(C(=O)NC2CCCC(NC(C3(C)CC(C)(C)C3)=O)CC2)c1C C(C(=O)NCC(=O)OCC)(C(C)C)OCC.C1(C=O)CSCCN1C(=O)COC N1(C(CC2C(C)(C)C(O)C2)=O)CC2(C=C(C(=O)NOCCCF)CO2)C1 Cc1nc(NCC(c2ccsc2Cl)C)cc(N(C)Cc2ccco2)n1 C1(C(N(CC(CN(C)C)O)C)=O)CC=CCN1C(=O)C=C(C1CC1)C1CC1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(C(C)(C)NC(CC(C)(F)F)=O)C12CC2 Cc1cc(C)nc(-c2cccc(C(=O)NCC(c3cccc(C#N)c3)O)c2)n1 c1(OCC(=O)N(CC(N2CCC(OC)C2)=O)CCOC)ccccc1C C1(CC(N2CC(SCC(=O)NCC(C)NC(=O)OC(C)(C)C)C2)=O)CCCCC1 N1(C(c2ccc(CC)s2)=O)CCC(CNC(c2cc(N)nc(Cl)c2)=O)CC1C Cn1ncc(C(=O)NCC(C)(C)CNC(C2CC3C=CC2C3)=O)c1C#N CC1(C)C2CN(C(c3sccc3NC(c3ccsc3Br)=O)=O)CC12 c1(OC)cc(C(=O)NCC2C=CCN2C(C2CCCOC2)=O)ccc1C(F)F C(=O)(CCC(=O)C1CCc2ccccc21)NC1C(c2cc(F)c(F)c(F)c2)(C)C1 CCC(CC(=O)N1CC(C2(NC(=O)CCNC(c3cccs3)=O)CC2)C1)C(C)C c1(C(=O)NCC2N(C(c3c(SC)nn(C)c3)=O)CC2)nn(C)c(C)c1Br C(C(C)(C)CNC(C1(F)CCOC1)=O)N(C(=O)C(C)c1ncco1)CC C1(CNC(C(c2cnccn2)C)=O)CCN(C(C2CC2C2(C)COC2)=O)CC1(F)F Cc1cccc(C(F)C(=O)NC(CN(C)C(c2cncc(F)c2)=O)(CO)CO)c1 C12CC(C)CN(C1)C2=O.C(=O)(CS(=O)(=O)N1CCCCC1)NCC(C)C c1(C(N(C2CCS(=O)(=O)C2)CC)=O)ccccc1C(N)=O C=C1CCC(C(N2CCCC(CCNC(C3CC(O)CN3C)=O)C2)=O)CC1 C1(NC(C(=O)NC(C)C)=O)CCN(C(=O)CNc2ccccn2)CC1C(C)C c1(CC)conc1C(=O)NCc1cc(C(=O)N(CCO)CC2CC2)cs1 c1(C(=O)NCCCCCCNC(c2cncc(C)c2)=O)ccc(C)c2c1CCC2 C1(NC(C(C)=C(CC)C)=O)CCCC12CN(C(=O)C(c1c(F)cccc1F)C)C2 c1(C(=O)NC(CNC(C2COC3CC2C3)=O)C2CC2)cc(C2CC2)nc(O)c1 c1(C(N(CCN(C(C(COC)N(C)C)=O)C)C)=O)cnc2cc(C)nn2c1 c1(SCCC(=O)NCC2(C)CCCN2C(C2CCC(=O)N2)=O)ccc(C#N)cc1 c1(CCNC(Cc2c(NS(CC(C)C)(=O)=O)cccc2)=O)ccc(Cl)cc1Cl c1(C(=O)NCC2C3CN(c4nccc(C(C)C)n4)CC32)nccc2ccn(C)c12 c1(C(=O)NC2C(C)CN(C(=O)CCc3ccsc3Cl)CC2)ccnc2c1CCC2 N1(C(c2ncc(Cl)s2)C(=O)NCCSCc2ccncc2)CCC(CO)CC1 c1(C(=O)NC2(C)CN(C(C(C3CCCO3)OC)=O)C2)[nH]cnc1C#N c1(OC)n[nH]c(C(N2CCCC2c2ncon2)=O)c1Cl N1(C(C(C)CC2CC2)C(=O)NC(C)(C)C)CCc2cc(F)cc(Br)c2C1 c1(CNC(C2CC(F)(F)C2)(C#C)C)ccc(Br)c(Cl)c1 N1(C(N(C)CCO)=O)CC(CF)OCC12CNC(=O)OC2 c1(C(=O)NC(C)CNC(C2CN3CCCC3CO2)=O)ccc2c(O)ncnc2c1 CC(C)C(CC(=O)N(CC(C)C(F)(F)F)C)NC(c1cscn1)=O N1(C(C(CC=C)C2CC2)=O)CCC(=C(F)F)CC1.C12C(=C)C1C(=O)NC2=O Cc1cnc(NC(CO)CCO)c(S(=O)(=O)N2CCC(CS(C)(=O)=O)C2)c1 N1(C(C(COC)N)=O)CCOCC(n2cc(CC(=O)O)nn2)C1 N1(CCC(C)F)CCC(CC(=O)Nc2ccccc2CN2CCN(C)CC2)CC1 c1(C(=O)NCCNC(=O)CC2OCCCO2)cccc(=O)o1 C1(C)(C(C)O)CCCN1CCc1cccc(-c2nn[nH]n2)c1 c1(C(C(=O)NCC2(F)CN(C(c3cnc(O)o3)=O)C2)O)cccc(OC(F)F)c1 C(C(COC)C(=O)NC(CN(C)C)C(=O)N1CC(CC(C)C)C1)OC C#CC(CNC(=O)NCC(c1ccc(F)c(F)c1)(F)F)CC(C)(C)C n1(CC(=O)NC2(C(C)NC(=O)COC3CCCC3)CCC2)ncccc1=O c1(C(N2CCC(S(=O)(=O)N3CCCC3)C2)C(=O)NCC=C)c2c(nn1C)CCC2 c1(C(N2CCC(CCNC(CNS(NC)(=O)=O)=O)C2)=O)ccc(O)c(CO)c1 c1(C(N2CC(C)(NC(C(CCC)C)=O)C2)=O)cc2cc(N)ccc2[nH]1 C(CNC(C1C(C)CCN1C(=O)Cc1ccn(C)n1)=O)(CC(C)C)OC C1(C(N(C(c2ccccc2Cl)C(=O)O)C)=O)CCC2(CCOCC2)C1 C(=O)(N=c1ccc(C2CCOCC2)n[nH]1)N(C(c1ccncc1Cl)C)C1CC1 C1(C(=O)NCC(C)CNC(=O)CCOCC(F)F)CCN(C2CC2)C1=O c1(C(=O)OCC2(Br)CCCC2)ccc(OC(F)(F)Cl)cc1 N1(C(CNC(=O)NC)=O)CCN(C2CCCN(C(C3CCN3C)=O)C2)CC1 c1(SCCC(=O)NCC(C(C)C)NC(C2CN(C(N)=O)C2)=O)c(F)cccc1Cl C1(CC(=O)NCC=CCNC(=O)C(c2ccc(Cl)cn2)(F)F)CCC2(CC1)CC2 c1(NCC(=O)Cc2ccsc2)cccc(Cl)c1OC(F)(F)F C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(C1(C2CCCO2)CCC1)=O c1(NC)nc(C(N2C3CCC2CN(C(=O)CCF)C3)=O)ccc1[N+](=O)[O-] c1(OC)cc(C(N2CC(NC(=O)C=C(C)C(C)(C)C)C(O)C2)=O)c(O)c(Cl)c1 c1(CC(N2CC(NC(C(C(CC)C)O)=O)C2)=O)c(Br)sc2ccccc12 N1(C(c2nc(C)oc2C)=O)C2CCC1CC(N(C(=O)CCCCO)C)C2 C1(C(=O)NC(=O)C(Cl)(Cl)Cl)COCCC12CN(C(c1cc(F)cc(Cl)c1)=O)C2 c1(C(=O)OC)sc(N2CCNCC2)nc1CC1CCOC1 C1(C)(NC(CC2CC(C)(C)C2)=O)CCN(C(c2ccccc2N2CCCC2)=O)C1 N1(C(C2(CC=C)CCN(C(C3CCCN3CCC)=O)C2)=O)CCN(C)C2(CC2)C1 N1(C(C2C(C=C)CC2)=O)CC(F)(F)CC1CNC(=O)CCOc1ccc(C)cc1 N1(C(C(C(C)C)SC)=O)CCC2(C)CN(C(C3CCC(C(C)(C)C)O3)=O)CC12 c1(OC)ccc2oc(C(N3CCC4CCC34CNC(C3(C)CC3)=O)=O)cc2c1 CC1CN(C(=O)CNC(C2CCC(C)(O)CC2)=O)CC(=O)N1 Cc1cn2c(n1)C(C(=O)N(CCCCNC(=O)CC1(O)CCCOC1)C)CCC2 c1(N2CC3CC(NC(c4cc(CCC)[nH]n4)=O)C3C2)cc(C)c(C#N)cn1 N1(C(C(C)=CC)=O)CCN(C(C2CCC(=O)N(C(C)C)C2)=O)C(CC(F)F)C1 c1(C(=O)NCC2N(C(C(COCC)(C)C)=O)CCC2)cc2cccnc2[nH]1 c1(C(N2CC3C(NC(C(C)CN(C)C)=O)(C3)C2)=O)cnc2n(c1=O)CCS2 c1(C(=O)NCC(C)(O)CN2CCOCC2)nc2nc(O)c3ccccc3n2n1 c1(C(N2CC(c3onc(C)n3)C(N)C2)=O)nc2ccccc2nc1O N1(C(c2cn(C)nc2N)=O)CCN(C(=O)CCS(C)=O)C(CS(C)(=O)=O)C1 Cc1cc(C(N2CC(NC(C3CC4CCC(C3)O4)=O)C(C)C2)=O)n2nccc2n1 C1(NC(CNC(=O)COc2ccccc2[N+](=O)[O-])=O)CCS(=O)(=O)C12CCC2 CCCCS(=O)(=O)CC(=O)NC12CCCC(NC(c3ccns3)=O)(C1)C2 C1(F)(C(N(CCC(=O)NC(C)CCC2CCCO2)C)=O)CCCC1 Cc1nc(C)c(C(=O)N(C)CC2COCCN2C(=O)CN(c2ncccn2)C)[nH]1 c1(NCCCC(C)NC(c2ccnn2-c2ccncc2)=O)ncc(C#N)cc1F c1(CN=[N+]=[N-])ccc(CSc2ccnc(Cl)c2)cc1[N+](=O)[O-] CCC(O)C(C)(C)C(=O)NCC1C=CC(NC(=O)CC2CC(C)C2)C1 C12(NC(c3n(CC)ncn3)=O)CC3CC(C1)CC(N(CC(=O)NC)C)(C3)C2 C1(C(=O)NC(C2CSC2)C)CCN(C(C2CCCC(C#N)C2)=O)CC1(C)C C1(NC(CC)=O)CN(C(c2ccc(-c3sccc3C)s2)=O)C2(CCCOC2)C1 C1(Cn2c(C(C3(C)CCOC3)Nc3ccccc3)nnn2)CCS(=O)(=O)CC1 Cc1cc(NC(C2CCCN(C(c3nc[nH]n3)=O)C2)=O)n(C(C)C)n1 C1(C(=O)NCCCN(C(C2(C=C)CCC2)=O)C)CNC(=O)CC1C N1(C(c2cc(C)ns2)=O)CCCC2(CC(NC(c3cnn(C)c3Cl)=O)CO2)C1 CCC(F)(C(=O)OC)C(=O)N1CC2C(N(C)C(c3cc(F)cnc3O)=O)C2C1 Cc1cnc(C(=O)NCCCCCCNC(C2(C(C)(F)F)CC2)=O)c(O)c1 C(c1ccc(F)cc1)=C(C)C(=O)NCC1CC1NC(=O)C=Cc1ccsc1 c1(CC)oc(C)cc1C(=O)NC(CO)C(C)NC(=O)C(C1CCC1)OC Cc1nc(C(N2CCSCC2C(=O)NC2CCOCC2F)=O)c(C)s1 c1(C(=O)NCC(N2CCN(C(=O)Cc3cnns3)CC2)=O)ccc(O)nn1 c1(C(N2CCC(c3n(C)ncc3)C2)C(=O)NCC2CCOC2)ccc(Cl)cc1Cl C1(CNC(Cc2cn(CC)nc2)=O)CN(C(=O)CC2COCC2O)CC(C)(C)C1 C1(CO)CCCCN(C(C2CC2CNC(=O)Cc2csc(Br)c2)=O)C1 N1(C(c2c(C)ccnc2)=O)CC2(C1)CN(C(C1(C)CC1Br)=O)CC2CO N1(CCCN2CCSC(C)(C)C2Br)CC2(C(=O)OC(C)(C)C)CC1CO2 C1(C(=O)NCC2CCC(CO)CC2)CCN(C(=O)C2CCCSC2)O1 Cc1ncnc(C(=O)NCCC2CCCN(C(=O)CC(C)F)CC2)c1C c1(C(=O)NCc2ncc(C)c(C)c2)nccc2c(Cl)cccc12 c1(C(=O)NCc2c(C3CCN(C(CC=CC=C)=O)C3)n[nH]c2)cccn(C)c1=O C1(O)(CCNC(CCOCCOC)=O)CCCN(C(c2cnn3c2SCC3)=O)C1 c1(C(N(CC(C)NC(c2c(C)cns2)=O)C)=O)nccnc1N C(c1ccoc1)=CC(=O)NCCN(CCC)C(C1CC1OCC)=O Cc1oc(C(F)(F)F)nc1C(=O)NCC1CC1NC(=O)CC1C=NN(C)C1=O N1(C(CC)=O)CCC2(CCN(C(c3cccc(N(C)C)c3)=O)C2)C1 C1(CC(N2C3CN(CC(c4c(CC)nccc4)=O)C(C3)C2)=O)CN2CCC1CC2 c1(N2CCC(OC)(CNC)CC2)ncnc2ccc(Oc3ccccc3F)cc12 Cc1sccc1C(N1CCC(CNC(=O)C(C2CCOCC2)O)C1)=O Cc1cnc(C(=O)N(C)CCNC(c2csc(-c3ccccc3)n2)=O)cc1Cl C(=O)(CC(C)C(F)F)N1CCC(NC(CC2(C=C)N=N2)=O)C1C(C)C c1(N(C2CCC3(CC2)OCCO3)C)cc(S(=O)(=O)Nc2ccccc2)ccn1 CCCC(CC(C)C)C(=O)N1CCC(CNC(=O)C(C(C)(C)C)OC)C(C)C1 C1(NC)CCN(CC2CC(O)C2(C)C)CC1 C(=O)(CCCCC(N)=O)NC(CC)CN(C(=O)C=CC(c1ccccc1)=O)C C12(C(=O)NCC(c3ccccc3)CNC(CCOCC)=O)CC(F)C1C2 CCCCCC(O)C(=O)NC1(COC)CCCN(C(c2ncccc2Cl)=O)C1 c1(OC)ccnc(-c2nc(C3CC3C(F)F)n(CCCO)n2)c1 c1(C(=O)NCC2C(CNC(C(C)S(N)(=O)=O)=O)C2)cnc2c(c1)CCCO2 C=CCC(C)(CC)C(=O)NC1(CNC(=O)CC2CC3(CC3)C2)CCCCC1 C1CCC(=O)NOC(CC(C)C)C(=O)N1.C(CC(O)CO)N(C(C)=O)C N1(C(C(=C(C)C2CC2)F)=O)CCCCC1CNC(=O)CNS(C)(=O)=O N1(C(CNC(=O)OC)=O)CCC(OCCNC(=O)C(C)(CO)N(C)C)CC1 CC1CCCN(C(=O)Nc2ccccc2F)C1c1noc(-c2ccccc2)n1 c1(C(=O)N)conc1C1CC1.CC1C(=O)NC(C)CCN1C.N(C)C Cc1ccc([N+](=O)[O-])c(C(N2CC(NC(C3(O)CC3(C)C)=O)C(O)C2)=O)c1 c1(C(=O)NCC(CNC(CN(C)C2CC2)=O)F)cc2cccc(Br)c2s1 C1(NC(c2[nH]cc(C)c2)=O)CC2CC(NC(=O)Cn3ncn(C)c3=O)CC12 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C1(O)CCN(C(c2ccnnc2O)=O)CC1)C c1(C(N(C(C)CNC(=O)CCCC(F)F)CC)=O)sc2nccc(C)c2c1C C=CC(O)C(C)(C)C(=O)N1CCC2(CC1)CC2C(N1CCC(OCCC)CC1)=O C1(C(=O)NCC(CN(C(C=CCOC)=O)C)O)CC2(CC2)CN1C N1(C(C(CCC=C)NC(=O)COC2(C)CCCC2)=O)CCC2(CCCC2)CC1 C1(N(C(=O)CC2CC2)C)CN(C(c2ccccc2OCC(F)(F)F)=O)CC1F C1(OC)CN(C(=O)CNC(c2ccccn2)=O)CC1NC(=O)C=Cc1cocn1 c1(OCC)nc(C(=O)NC(C)CNC(c2nc(O)sc2C)=O)cc2ccccc12 c1(NCC2(C)CC2Br)[nH]c(=NCCc2cnc3n2CCCC3)nc2scnc12 Cn1nc(C(N2CC3CC3(CNC(C3CCCC3(F)F)=O)C2)=O)cc1C(C)(C)C C1(C)(C(=O)NC2CC(CNC(CC(=C)Br)=O)C2)CC(OC)CN1C N1(C(CCN(CC)CC)=O)CC(NC(C2COCC2C(N)=O)=O)C(C)C1 c1(OC)cc(C(=O)NCCC2CCC(NC(=O)Cc3cccs3)C2)cc(Cl)c1O N1(C(Cn2cc(-c3c(C)ccnn3)nn2)=O)CC(OCc2cccs2)CC(C)C1 n1(CC(C)(O)C(N2CC(=O)N(C(C(=O)O)C3CC3)C2=O)=O)cnc2ccccc12 CC1CCCC(CC(N2CCC(C)(NC(C3(NC4CC4)CCCC3)=O)C2)=O)C1 C12(C(=O)NC3(CNC(C4C(C)CN(C)C4)=O)CCC3)C3C4C1C1C2C3C41C Cc1[nH]cc(C(=O)NCC2CCN2C(=O)C=CCF)c(=O)c1Br c1(C(N2C(CCNC(C3C(C)(C)C3)=O)CCC2)=O)cccc2c1COCCN2 CC1CN(C(=O)COCC(F)F)CC(C)N(C(c2cc3c(s2)CC(C)(C)C3)=O)C1 C1(c2nnnn2C)(NCCC2(C(=O)OCC)CCCC2)COCC1C N1(C(C(C)CF)=O)CC(NC(c2ccc(C3CCCO3)[nH]2)=O)C(O)C1 C1(CC=C)CCCN(C(=O)C(C)(C2CC2)N(C(=O)CN(C)CCC)C)C1 N1(C(CCC(C)C)=O)CCC2(CCCN(C(=O)CCCc3nccs3)C2)C1 n1(CC(=O)OC(C)(C)C)ccc(=O)n(C)c1=O.C1(OC)CC2N(C1)C(=O)NC2 c1(OC)cc(CC(=O)NCC(O)CCNC(C2OCCO2)=O)cc(Cl)c1 c1(C(N2CCn3c(C)cnc3C2)=O)ccnc2cc(Cl)ccc12 Cc1cc(C(=O)NCCN(C(=O)CC(C)c2ccccc2)C)nn1C N1(C(c2ccnc(Br)c2)=O)CCC(C2CN(C(c3cc(Br)cnc3F)=O)C2)CC1 N#CC1(CNC(=O)CCC2CCCN2C(=O)CC2CCCC(O)C2)CCCC1 N1(C(c2ccnc(O)c2)=O)CCC2CCN(C(=O)COC3CC(F)(F)C3)C2C1 c1(CNC(C=CC(C)(C)SC)=O)cnn(C)c1C(N1CC(CO)C1)=O C#Cc1ccc(C(=O)NC(CNC(c2cccc(OC)c2OC)=O)C2CC2)cn1 c1(CN(C)C)ccoc1C(N1CCCC1C1CCN(C(=O)CCC2(C)CC2)C1)=O C1(OC)CC2CC(C(=O)NCC3(C)CCN(C(c4sc(F)cc4C)=O)CC3)CC12 Cc1ccc(C(=O)N(C)CC2CN(C(=O)C(F)C3CCC3)CC23CC3)c(N)c1 N1(C(C=CCCC(C)C)=O)CCC(NC(c2cnn3occc23)=O)CC(C)(C)C1 C(CCC(C(=O)NCCN=[N+]=[N-])NC(c1cc(F)ccc1O)=O)OC C(C1CCCCc2ccccc21)c1c(O)nccc1.c12nc(ccc1Cl)CN2 C#CC1(O)CCN(C(=O)CC2C3CN(C(C45CSCC4C5)=O)CC23)CC1 N1(C(C(CC=C)CC)=O)CCN(C(c2csc(C(C)C)n2)=O)C2CCC12 c1(-n2cc(C(CC)N(C(=O)CC3(C)CCC3)CC)nn2)cccc(C(F)(F)F)c1 C(C#CC(=O)NCC(CO)(CO)NC(c1oc(CC)cc1C)=O)(OCC)OCC c1(C(NNC(=O)NC(c2ccc(OCC)c(Br)c2)C)=O)nc2ccc(C)cc2[nH]1 C(=O)(C(O)C(C)(C)C)NCC1(CN(C(=O)C(c2ccccc2)O)C)CC1 C1(CNC(c2ccn(CCN(C)C)n2)=O)C2CN(CC3CCCCO3)CC12 C1(NC(c2cc(C)n(C)c2)=O)CCN(C(=O)CCc2cnn(C)n2)CC1CO N1(C(C=CC2(C)COC2)=O)CC(NC(c2cnncc2O)=O)C(O)C1 Cn1cnc(N2CCC(CCNC(c3cccc(F)n3)=O)C2)c(Br)c1=O c1(C(=O)NCc2ccc(Cl)cc2F)c(Cl)cc(Cl)cc1Cl.C12(CC1)C(=O)N2 O=C(C1=CCOC1)NCCOCCNC(=O)Cc1csc(Br)n1 C1(CNC(C2CCCS2(=O)=O)=O)CC12CCN(C(C1CCC(F)(F)CC1)=O)CC2 c1(OC)c(C(=O)NCC2(O)CCN(C(=O)C(F)C3CCOC3)CC2)ccnc1F C1(NC(=O)Cc2ccccc2F)CCCC2CN(C(=O)CCc3nc[nH]n3)CC12 c1(NC(=O)CN(C)CCOC)ccc(C(=O)N(CC)Cc2ccc(Cl)s2)c(Cl)c1 C(=O)(C1=CCC(NC(=O)C(C)(C)n2cnnn2)C1)NCC(CC(=O)OC)C N1(C(C2(CC)CC2)=O)CC2CN(C(C3CCC=CCC3)=O)CC(C1)O2 C1(OC)CN(C(C2(C)CCC(C)(C)C2)=O)CCC1NC(=O)CC1CCOC1 N1(C(COc2cccc(C)c2)=O)CCCCC(CNC(=O)CC2CCCC2C)C1 N1(C(C2CC(C)(O)C2)=O)CC2CC(C1)N(C(=O)CCC1CC1CC1CC1)C2 CC1CN2CCN1CC2C(=O)N(CCCNC(C12CCC(CC1)OC2)=O)C1CC1 N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(c3cnc(Cl)s3)=O)CC2C1 c1(OC)c(C(=O)NCC(CNC(=O)C=Cc2ccncc2)OC)cc(F)cc1F C1(C(=O)NCC(C)(CO)NC(CN(S(C)(=O)=O)C)=O)CCS(=O)(=O)N1 c1(OC(C(=O)NC2(CCNC(C=C(C)C)=O)CC2)C)ccc(C)cc1C C#Cc1cccc(CC(N2CC3CC2C3NC(=O)C(N2CCSCC2)C)=O)c1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)NC(C)CN(C(c1cncc(C)c1)=O)C C(=O)(C1COc2ccccc21)N1CC2C(NC(CCSCCCC)=O)C2C1 N1(C(C2CCC(=C)CC2)=O)CC=C(CC(=O)NC2CSCC2C)CC1 c1(-c2nnc(NC(N3CCC(C(F)(F)F)(CO)C3)=O)s2)ccc(F)cc1Cl CC(C)CC(C)(C)C(=O)NCC1CC1NC(=O)COc1ccc(C#N)cc1 c1(C(N)=O)ccc(C(=O)NC2CCCC2NC(C2CC3CC3C2)=O)cc1 N1(C(C2C(CC)OCC2)=O)CC2=C(C1)CN(C(=O)C(c1ccc(F)cc1F)=O)C2 C(=O)(C1=CC2CCCCCCC12)N(C1CCN(C(c2cc(Cl)nc(Cl)c2)=O)C1)C C(=O)(C(C)CC(=O)NCC1(C(=O)NCCC(C)N2CCCC2)CC=CC1)OC O=C1NCCOc2ccc(CNCC3CCCN(Cc4ccccc4)C3)cc21 Cc1ccc(C(=O)NC2CC(O)CN(C(c3ccc(O)cc3)=O)C2)cc1C c1(NC(C(C)(C)C)C2CC(F)(F)C2)cc(Cl)cc(Br)c1 C1(N(C(=O)CC2CCCOC2)CC)CCN(C(C2(c3occc3C)CC2)=O)CC1 c1(OCC)nc(Cl)ccc1C(N1CCCC(CNC(C23C=CC(CC2)C3)=O)C1)=O c1(CNC(CC2N(C(C3(N(C)C)CCC3)=O)CC2)=O)ncccc1O N1(C(CCC)=O)CCC(C2CCCCN2C(=O)Cn2cc(C(C)O)nn2)CC1 Cc1cc(NC(c2ccc3c(c2)CCO3)=O)c2cc(-c3ccco3)ccc2n1 C(=O)(C(CCC(N)=O)N(C)C)N1CC(C(C)C)N(C(=O)CCC(C)(C)C)CC1 c1(NC(C(=O)Nc2cccc(-c3ccncc3)c2)=O)ccc2c(c1)CCNCC2 N1(C(COC(CC2ON=C(C)C2)=O)=O)CCN(C(C(C)(C)C)=O)CC1 N1(C(COCCC=C)=O)CC2CN(C(c3cnc(OC)c(Cl)c3)=O)CC2(C)C1 C(=O)(CC(C)C(C)(C)NC(c1sc(C)cc1C)=O)NC1CC(C#C)C1 C=CC1(O)CC(C(=O)NC2(CC(N3CCC(SC(=O)OC)C3)=O)CCCCC2)C1 Cc1ccc(C(=O)N(C2CCCC(N(C(=O)COCC(F)F)C)C2)C)nn1 c1(C(=O)NCCCN(C(=O)C(C)C2CCC2)CC)cc2ccncc2s1 N1(C(c2cc(C)c(C)s2)C(=O)NCCOC)CCCc2ccc(C)cc21 Cc1ncc(CCC(=O)NC2(CNC(c3csc(-c4ncccn4)n3)=O)CC2)o1 C1(CC(=O)OC)CCCN1C(C1C=CC(NC(C2CCC(=O)N2)=O)C1)=O Cc1noc(C2CC2)c1C(=O)NCC1(C)CCCN1C(=O)CC1(C)CCCCC1 c1(C(=O)OCc2c(C)sc(-c3ccco3)n2)sccc1S(=O)(=O)N1CCOCC1 N1(C(COC)=O)CCC(CON(C2C3CCC23)C)CC1 N(C(=NCc1ccc(F)cc1)N1CCC(F)C1)C(c1cccs1)C(c1cc[nH]n1)O C1(CC(=O)NC(C(C)C)CCN(C(=O)C=CCO)C)NC(=O)CNC1=O N1(C(C(C)n2cccc2)=O)CC=CC1CNC(c1ccsc1C(F)(F)F)=O c1(C(=O)NCCC2(CNC(C3CC4CCC4C3)=O)CC2)ccnc2ccsc12 CC1CCCn2cc(C(N3CC(O)(CNC(=O)C(c4ccccc4)F)C3)=O)nc21 C1(C(=O)NCC(C2CC2)NC(c2cc(OC)ns2)=O)CCC2(CC1)CNC(=O)C2 CC(C)(CS(C)(=O)=O)C(=O)N1CC2CCCC2(NC(c2cnc3n2CCC3)=O)C1 C1(NC(c2c(OC)ccs2)=O)CCCCN(C(c2cc3ccccc3[nH]2)=O)CC1 CC1CCC(C(N2CCN(C(=O)CCF)CC2)=O)CN1C(=O)Cc1ccnn1C N1(C(CCOCC(C)(C)C)=O)CCN(CCNC(C2(CCF)CC2)=O)CC1 c1(C(=O)NCCC2C(C)(C)CCO2)ccc2c(=O)[nH]ccc2c1 Cc1noc2cc(C(N3CC4CC(NC(=O)CC(C)(F)F)CC4C3)=O)ccc12 C1(OC)CN(C(c2cccc(C)n2)C(=O)NC2CCOC2)CC1O c1(C(=O)NC2C(C)N(Cc3c(Cl)cccc3Cl)CCC2)cnc2cnccc2c1 c1(C(=O)NC2C3OCC(NC(c4occ(C)c4)=O)(C3)C2)cccc(O)c1[N+](=O)[O-] N1(c2cc(C)nc(N3CCOC(c4cn[nH]c4)C3)n2)CC(C)C(C2CCC2)C1 N1(C(CN(S(CC)(=O)=O)C)=O)CCC(NC(=O)C=Cc2ccc(C)o2)C12CCC2 c1(C(=O)NCCN(C(C=C(CC)C)=O)C2CC2)nccc(Cl)c1C c1(SC)nnc2n1CCC2.C1(C2CC2)CN2CC1C2=O.c12cn(nn1)C2 C(=O)(C1=COCCO1)N1C(CNC(CC2CC(OCC)C2)=O)C=CC1 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CC(CO)N(C(C23CC(O)C2C3)=O)C1 C(=O)(C1=CNC2=NCCCC2=C1)NCCN(C1CCCCCC1)C(C(CC)C)=O C1(C(N(C(C)CC(N)=O)C)=O)CC2CCC(C1)N2C(C1CC1C1CC1)=O C(=O)(C1=CCCCC1)N1C(C(C)NC(c2csc(O)n2)=O)CCCC1 N1(C(C(n2ccc(C3CC3)n2)C)=O)CCC(C(C)(C)NC(C2CC23CC3)=O)CC1 c1(CNC(C(=O)NC(C2CC(C)C2)C)=O)cccc(CO)n1 C(CN=c1[nH]c(N2CCC(=CBr)CC2)nc2c1CCCC2)N1C(=O)NCC1 C1(NCc2c(N(C(C(CC)CCOC)=O)C)nc(C)cc2)CCCCN(C)C1=O C(=O)(C(CN(C)C)CC(C)C)N(CCNC(COCC)=O)Cc1ccccc1 N1(C(c2ccc(CCC)[nH]2)=O)CCCCC(NC(c2ncc(F)c(OC)n2)=O)C1 CC1(C)C2CCC1(C(=O)NC13CC(CN1C(=O)C(=O)NCCOCCO)C3)C2 CC1=C(F)CN(C(=O)C(C(C)(C)O)NC(=O)C=CC(=O)N(C)C)CC1 C1(CCCC)CN(C(=O)CC(C)(C)OC)CCN1C(C1CCCNC1=O)=O C1(CCC(=O)NC)CCN(C(C)C)C1.c1(CCCNC(=O)CS)ccncc1 Cn1cnc(CCNC(C(CCCO)c2ccccc2)=O)c1 C1(NC(C(C)O)=O)CCN(C(C2CC3CCC2CC3)=O)CC(C)(C)C1 Cn1cccc1C(N1CC(CNC(=O)CCc2cnc(C3CCC3)o2)C1)=O CON(CCO)C(=O)C1(N(CC(CC(=O)OC)C)C2CC2)CCC1 C(=O)(CC(C)C(=O)NC(C(=O)Nc1cnn(CCF)c1)C1(C)CC1)OC N1(C(C2OCC(C)C2)=O)CC2(CCC2)CC1CNC(C1CC2CCC(C1)N2C)=O c1(SC)cccc(C(N2CCCC2C2(O)CN(C(C3(OC)CCC(C)C3)=O)C2)=O)n1 CC(C)(C)CN=C(N(C)CC1C=CCCCC1)NC1CC(OC(=O)N(C)C)C1 c1(C(N2C(C)C(NC(=O)CCC3CCC3)CCC2)=O)ccnc2ccnn12 C(=O)(C(CC(C)(C)C)OC)N(C(CC(=O)NC1CC(CC)OCC1)(C)C)C CCC(C)(C)CCCC(=O)N(C(C)C(N1CCC12CCCSC2)=O)CC C1(C(N2C(C)(CC)CCC2)=O)CC2(CC(NC(c3c[nH]nc3C3CC3)=O)C2)C1 O=C(CCC(=O)c1ccc(F)cc1)NC(=O)Cc1cn(CC2CC2NCCl)nn1 Nc1cc(F)c(C(=O)NC(CNC(=O)CCC2CC2)CO)cc1F c1(C(=O)NC(C(C)NC(=O)C(C)C(C)O)C)cncc2nnn(C)c12 C1(N(C(c2ccc(=O)oc2)=O)CC)CCCN(C(C2(COC)CCOC2)=O)C1 c1(C(N2CCC(N(C(=O)CN3CSCC3=O)CC#C)CC2)=O)ncc(F)cc1F C1(NC2CC(c3ccccc3)(CC(=O)OCC)C2)CCC(S(C)=O)C1 C(CCN1CCCC1)(C(=O)N1CCCC1)NC(=O)NCc1c(CC)occ1 C1(NC(CC(C=C)CC)=O)CN(C(c2cc(CC)[nH]n2)=O)CCC12CCC2 C1(CNC(c2cc(CO)on2)=O)CN(C(=O)CCc2cnc(O)[nH]2)CC1O c1(N2CCCC(C=C)C2)nc2c(c(=NCC3(N(C)C)CCSC3)[nH]1)SCC2 C=CCC(CNC(c1sccc1F)=O)NC(=O)C(n1ccc(C(F)(F)F)n1)C N1(C(CCc2ccc(C)cc2)=O)CCC(F)C(NC(=O)Nc2ccccn2)C1 N1(C(C2CN(C(c3n(C=C)ncc3)=O)CC2C=CC)=O)CCC(C)CC(C)C1 CC1(C)CC(NC(=O)C=C2CCC2)CN(c2ncc(C#N)cc2F)C1 c1(C(=O)NCC23CC2CN(C(=O)CCn2ccnn2)C3)cncc2nc(O)[nH]c12 n1(CCCC)nccc1C(N1CCC(N(C(C2CCCC2C(F)F)=O)CC)C1)=O C(=O)(C1=CC2CCCCCC12)N1CC2CCC(NC(=O)CCCC(F)F)CC2C1 C(=O)C(C)(O)C(C)C.C1(CC)CCCN(C(CC)C(=O)NCc2cnc(SC)[nH]2)C1 c1(C(=O)NC(CCN(C(Cc2cn(CC)nc2)=O)C)C)ccncc1C(F)F c1(C(=O)NC2C(NC(Cc3c(CC)cccc3)=O)CC2)cccc(Cl)c1O N1(C(C(c2ccc(Cl)s2)C)=O)CCC2C1CCCN2C(=O)Cc1nncn1C N1(C(C(C)(C)C2CC2)=O)CCN(C(C2C=CCC2)=O)C(C2CC2)C1 c1(C(=O)NCCCN(C(C(CCCC#C)C)=O)C)ccc2ncc(Br)n2c1 c1(OC)ccc(CC(N2CC(CNC(=O)CC3CCC(CN(C)C)O3)C2)=O)nc1 Cc1ccc(OCC(=O)NCC2(C)CN(C(=O)CCCC(C)F)CC2C)cc1C c1(CC)cccc(C(=O)NCC2CCCCN(C(=O)CC3OCCCO3)C2)c1F N1(C(C2C(CNC(Cc3cc(CC)no3)=O)CCO2)=O)CCCC(CN(C)C)C1 C(=O)(CCC(=O)C1CC1)NCCCN(C1CCCC1)C(c1nc(CC)sc1)=O CC(c1ccccc1F)=CC(=O)NC(C)(C)C(C)NC(c1c[nH]cc1Br)=O c1(C(N2CC(NC(CCCC=C)=O)C(C=C)C2)=O)oc2ccccc2c1Cl C12(NC(Cc3c(CSCC)cccc3)=O)CCCC1N(C(c1cocn1)=O)CC2 c1(C(=O)NCC2C(NC(C=C(COC)C)=O)CCC2)c[nH]c2cccc(C#N)c12 C1(C(=O)NCC(C)(F)F)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C(=O)NCC(C)N(C(C(CCC)OC)=O)C)cccc(C2=CCOCC2)c1 c1(C(=O)NC(c2ccc(C#N)cc2F)C)cn2cc(C(F)(F)F)ccc2n1 C1(C(=O)NCC(c2ncc[nH]2)C)CC(C)(C)CCN1C(=O)CCC1CCOCC1 c1(C(=O)NC2(CNC(c3ccc(O)nc3Cl)=O)CCC2)ccnc2ncnn12 Cn1ncnc1CNC(c1cn(CCNC(C2CCCC2)=O)cn1)=O C1(C)(CNC(CC2(COC)CCC2)=O)CCCN1C(=O)CCc1ccc(C)nc1 CCC(C)(CC)C(=O)NCc1ccoc1C(=O)Nc1cnc(Cl)nc1C c1(C(C(=O)NCCOCCNC(=O)C=Cc2ncco2)O)ccc(F)c(F)c1 N(C(=NCCc1ccn(CC)n1)N1CCC(c2ccccc2F)C1)C(CC)C c1(C(=O)NCCC2COCCN2C(c2nc(Cl)cs2)=O)c[nH]nc1[N+](=O)[O-] c1(OCOC)cc(F)c(CN(C)Cc2ccoc2C)cc1Cl C=CCCC(C)(C)C(=O)N1CC(NC(c2c(Cl)cccc2Cl)=O)C2(CC2)C1 CCCCCCn1nnnc1C1(NCc2cnc(C(C)C)s2)CC1(C)C Cc1nc(C(=O)NCC(C)(CO)NC(c2cscc2Cl)=O)nn1-c1ccccc1 c1(OC)ccc(CC(O)C(=O)NC(CO)C(C)NC(=O)Cc2conc2C)cc1 C(N=c1[nH]cncc1Br)C1(CNC(C(C)(C)c2cncnc2)=O)CCCC1 N1(C(CN(C(C)C)C(c2ccnc(N(C)C)c2)=O)=O)CCCCC1CO N12C3CCC1CC(C3)C2=O.Cc1c(NC(=O)C(F)C(C)(F)F)cccc1F c1(C(C)C)ccc(CC(=O)NCC2(O)CC(NC(C3COC(=O)C3)=O)C2)cc1 N1(C(c2c(C)nc(C(C)C)o2)=O)CCN(C)CC1CNC(C1CC12CC2)=O C#Cc1ccc(F)cc1NCC1C(NC(=O)NC(C)(C)C)CCC1 N1(C(c2nc(C)[nH]n2)=O)CCCC(C(=O)NCCCNN2CCN(C)CC2)C1 c1(CC)cc(C(=O)NC(C(N2CC3CC2C3C(N)=O)=O)c2cccs2)c(C)o1 N1(C(C(C2CCCC2)OC)=O)CCCCC1CNC(C1(N2CCCC2)CC1)=O c1(CC(=O)NC(C(C)(C)C)CNC(c2cncc(F)n2)=O)ccc(C#N)cc1F C1(NC(=O)CC(O)c2ccccc2)(CNC(=O)C(O)C2CC2)CCCCC1 Cc1cc(C(N2CCCC2(C)C(N2CCn3ncnc3C2)=O)=O)cc(C)c1O CCC(CC)(CO)C(=O)N1CCCOC(CNC(c2cn(C)nc2C)=O)C1 C1(C(=O)NC2CC3(CC(OC)C3)C2)CC12CCN(c1ccc(C(C)=O)cn1)CC2 CC(C)CC(CNC(=O)C(CC1CC1)CC1CC1)NC(=O)Cc1ccccc1Cl c1(NC(C2C(C(=O)NC(C)CO)C2)=O)onc2ccccc12 N1(C(c2scc(C(N)=O)c2)=O)CCN(C(C2CC2CF)=O)C(c2ccccn2)C1 c1(CNC(C2C(C3C(C)C3)C2)=O)cccc2c1CCN(C1CCN(C)C1=O)C2 N1(C(C(C)S(N)(=O)=O)=O)CC(NC(C2CC3(C2)CC(F)C3)=O)CC(C)(C)C1 C1(NC(C(CC)OCC)=O)CC2CN(C(c3ncc(Br)cc3O)=O)CC12 Cn1cc(Cl)cc1C(=O)NCC1CCCCC1NC(c1cnccc1Cl)=O c1(C(N2CCC(=CCNC(C(CSC)O)=O)CC2)=O)cnc(O)cc1F C1(C(N(CC(CN(C)C(c2ccc(F)cc2)=O)O)C)=O)CCC2(CCC2)CO1 C1(C(N2C(CC)CC(O)C2)=O)CCC2(CC2)N1C(c1cc[nH]c1)=O n1(CCC)nnnc1C(C1CC1C1CC1)NCCNC(=O)C(C)C C12(C(=O)NC(CNC(C(C(=O)OC)C)=O)(C)C(C)C)CCC(CC1)OC2 C12(C(=O)NC3C(NC(C4(OC)CCC4)=O)CCCC3)CCCN(CC1)S2(=O)=O C1(C(=O)NCC2CN(C(C(CCNC(=O)C3CC3)O)=O)C2)CCc2ncnn2C1 C(C(F)(F)C(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)C(SC)C1)SC CCC(CC)C(F)C(=O)N1CCCC(F)(C(=O)NCC(n2cccn2)C)C1 C1(C2CC2)(CNC(c2n(CC=C)ccn2)=O)CCN(C(=O)C=CS(=O)(=O)CC)C1 C1(CNC(=O)NCC(c2ccsc2)C)CCCC1N(C)C C(=O)(CC(C)CC(=O)OCC)NC1(CC=C)CCCN(C(=O)C=CC(F)(F)F)C1 N1(C(C(C)OCC=C)=O)CC(=O)NC(=O)C1 N1(C(C=NOC)=O)CCC(C)N(C(=O)CCOc2ccc(Cl)cc2F)CC1 Cc1cc(C(=O)NC2CCC(C)N(C(c3cc(C#N)c[nH]3)=O)C2)cnc1C C1(NC(Cc2ccc(C)c(C)c2)=O)CCC2CC1CN2C(=O)CCC(F)F N1(C(c2n(C)nc(C(F)F)c2)=O)CC(NC(c2ccc(F)s2)=O)C2(CC2)C1 C(=O)(N=c1ccc(C(F)(F)C(F)(F)F)n[nH]1)N(C1(OC)CCC(C)C1)C(=O)C1CC1 CCCCC(C)(CO)NC(=O)CCCCCNC(c1cc(C)nc(C)c1)=O C1(C(=O)Nc2ccc(CC(=O)OC)cc2)CC2(CCOCC2)CO1 c1(OCC)ccc(CCC(=O)NC(CNC(C2CCN(C)CC2)=O)C2CC2)cc1 CCN=c1ccc(C(N2CCCCC(NC(=O)C(C)OCC3CC3)C2)=O)c[nH]1 N(C(=NC(C)c1nncn1C)NCC1(SC)CC1)C(CC)CC Cc1nn(C(C)C)cc1COC(c1ccc(CC(=O)N(C)C)cc1)=O c1(C(=O)NC2(CNC(CCC)=O)CCCC2)cnncc1C C(N=c1[nH]c(=NCCC#N)[nH]c2c1CCCC2)c1ccnc2[nH]cc(C)c21 c1(C(N2C(CCN(C(COCC=C)=O)C)CCCC2)=O)ccc(Br)c(O)n1 N1(C(C(=O)N(C)CC2(OC)CCCCCC2)=O)CCC(C)CC(C)C1 n1(-c2ncc(C(=O)NCC(=O)N(C3CCC3)CC#C)s2)c(C)ccc1C C(=O)(C1CCc2nccn21)NC(C)C(C)C(=O)NCC1CN(C(N)=O)C1 C1(C(C)C)CN(C(C(=O)NCC2CCOC2)C2CC2Cl)CCO1 Cc1nccnc1C(=O)NC(C)CCN(C(=O)Cc1cncs1)C C(C(C)(C)CNC(=O)CC1(CO)CC1)N(C(C(C)=CC1CC1)=O)C CC1CN(C(C2(C#N)CC3(CC3)C2)=O)CCC1NC(C1(C2CC2)CCC1)=O CC1(C(=O)NCC#CCN(C)C)CC12CCN(C(c1ccon1)=O)CC2.C(=O)OC c1(CC)c(C(N2CCCC2C2(C(=O)OC)CC2)=O)cnn1-c1ccccc1 N1(C(CCC(C)OC)=O)CC(N(C)C(c2ccnc(C(F)(F)F)n2)=O)C2(CC2)C1 c1(OC)cc(C(N2CCOC3CC23)=O)c(NC(c2cccc(O)c2F)=O)cn1 C1(C#N)(CC)CC2CCC1CC2(C#N)NCCCC1CC1(Cl)Cl N#Cc1c(Br)ccc(C(=O)NC2Cc3ccccc3C2O)c1F N1(C(=O)NC2CCC(C)C2)CCN2CCCC2C1 C1(CC)CN(C(=O)C(C)Cn2ccnc2)CCN1C(c1cc(Cl)cnn1)=O CCCC(CC1CCCC1)C(=O)NCC(C)(C)OCCNC(=O)Cc1ccsc1 c1(SC)cccc(NC(=O)Cc2ccc(C3CCNCC3)cc2)c1 Cc1ccoc1C(=O)NC1COCC1CNC(=O)C(C)c1ccco1 c1(C(N2C(C)(CNC(C3C(CC)OCC3)=O)CCC2)=O)cc(O)cc(O)c1 CN1C(=O)CCc2cc(NCC3CCCC3C(C)(C)C)ccc21 C1(C(=O)NC2N(C(C(COC)N(C)C)=O)CC=CC2)CC(C)(C)OC1=O Cc1csc(=O)n1CC(=O)NCCN1CCN(C(=O)CCCc2cnn[nH]2)CC1 c1(OC2CC(NC(C(C)SCc3cccs3)=O)C2)cccc(Br)c1 N1(C(c2c(C)cc[nH]2)=O)CCC(C(N2CCC(C)(CCO)C2)=O)C1C C(=O)(C(C)C(C)c1ccccc1Cl)NCCCN(C(c1c(CC)noc1)=O)C c1(CCN)nccc(C(=O)N(CC2CC2)CC2CCCO2)n1 C1(NC(CC(C)F)=O)Cc2ccccc2C1NC(c1ccc(Cl)c2occc12)=O N1(C(=O)C=CCn2cncn2)CCC(C(C)CCNC(C(C)O)=O)CC1 c1(OC)nc(C)c(C(=O)NCC(=O)Nc2nc(Cl)cs2)s1 C(N=c1[nH]c(Cl)nc2c1SCC2)C1CN(C(C(C)NC(C)=O)=O)CC12COC2 CC(C)CCC(F)C(=O)NCCOCCOCCCNC(=O)C(C)C#N C1(CC=C)(C(=O)NC(C2CCCN2C(=O)CCC2CC(F)(F)C2)C)CCOC1 c1(OC)ccc2c(CC(=O)NCC(C3CCC3)NC(c3cnco3)=O)coc2c1 c1(C(N2CC(C)C(C(N3CCC(O)(C(F)F)C3)=O)C2)=O)cn(C)c(=O)n1C C1(CC(=O)NCCC2CC(NC(Cc3cn(C)nn3)=O)C2)CCCCCC1(F)F C1(C)(C(N2CC(C(C)NC(c3c(COC)cco3)=O)C2)=O)CCC(=O)N(C)C1 C(=O)(CCS(=O)(=O)Cc1ccccn1)NCCN(C)C(C12CCCN1CCC2)=O C1(C(C)NC(=O)CCCC(N)=O)COC(C)(C)CN1C(c1cnc(O)c(F)c1)=O CC(C)C(N=[N+]=[N-])C(=O)NC(C(N1CC2(CCCN2C)C1)=O)C1CCCO1 c1(CNC(c2coc(C3CC3)n2)=O)n[nH]c2c1CN(C(=O)Cn1cccn1)CC2 CCCCCC(C)(CC)C(=O)N1C2CCC1CC(NC(=O)C#CC1CC1)C2 c1(C(=O)NC(C)CNC(C2CC2C2CC2)=O)cc2ccccc2n1C C1(F)(CNC(c2cnc(C)n2C)=O)CCC(CNC(=O)CCCC2CC2)CC1 c1(C(=O)NCC2(O)CN(C(c3n(CCC)ncc3)=O)C2)nn(C(C)C)cc1Br C1(CC(C)C)(C(=O)NC2CC(CCNC(=O)C(CO)N(C)C)C2)CCCC1 c1(NC(=O)NCC2C(OC)(OC)CC2)ncoc1-c1cc(C)no1 C(CC(=O)N(C)C(c1cc(C)on1)C)(C(F)F)Nc1c(C(=O)OC)cccc1 c1(OC)ccc2cc(C(N3CC4CC(NC(=O)C(F)C(C)C)C3C4)=O)n(C)c2c1 N1(C(c2c(C)cc(C)o2)=O)CCC2CCN(C(c3ccc(CN(C)C)[nH]3)=O)C2C1 C=CC1OCCC1C(=O)NC(C1(O)CN(C(=O)CC2(C(F)(F)F)CC2)C1)C C(=O)(C(C)NCCN(C)C)NC(CCN(C(C)C)NC(=O)OC(C)(C)C)C N1(C(C=C(CC)CC)=O)CCCCC1C1CCN(C(=O)C2=C(Cl)CC2)C1 C1(CC(=O)NCC(n2cccn2)C)CCN(C(c2ccc(F)c(F)c2)=O)C1(C)C c1(CN2CCC(O)(C(=O)Nc3cccnc3Cl)C2)ccc(Cl)c(I)c1 C1(NC(C=C(C)CNC(=O)CC2C=NN(C)C2=O)=O)COC2(CCC2)C1 Cc1nn(C2CCCN(CC3CCC(CCC(=O)N(C)C)C3)C2)c(C)c1Cl C12(C(=O)NCC(CN(C(c3ccc(CC)[nH]3)=O)C)(C)C)CCC(C1)OC2 c1(C(N2C(CNC(C(C(C)C)F)=O)C(C)CCC2)=O)nccc2ncccc12 CC1C(NC(=O)C(=O)Nc2sccc2F)CCCN1C(=O)OCC(C)(C)C C#CCC(CC#C)C(=O)N1CCCCC(NC(=O)CC(C)C(F)(F)F)C1 Cc1cccc(N)c1C(=O)NCC#CCNC(=O)C(C(C)C)c1ccccc1 Cc1ccc(NC(C2CCN(C(c3c[nH]ccc3=O)=O)C2C)=O)c(O)n1 N1(C(c2c(CC)noc2)=O)CC2(CC(NC(=O)C(N3CCCC(C)C3)=O)CO2)C1 Cc1[nH]c2ccccc2c1C(=O)NC1CCCC1C(=O)NC(C1CCOC1)C c1(N2CC(CC)C3(C2)CCC3)[nH]c(=NC2CC(N)C2)nc2c1cnn2C(C)C.SC N1(C(COCCC#C)=O)CCCC1C1CCN(C(=O)CSCCN(C)C)C1 C(=O)(C(F)C(C)(C)O)NCC1C(C)CCN1C(=O)C=Cc1ccccn1 N1(C(C(C)NC(N)=O)=O)CCC=C(C(=O)NCC2CCCCS2)C1 c1(C(CNC(c2cc(C)[nH]n2)=O)NC(=O)C(F)(F)c2cscn2)ccc(F)cc1 C1(CC)(NC(=O)C(O)C2CCOC2)CCN(C(=O)Cc2cccc(C)c2F)CC1 C1(C2(NC(=O)CSn3cncn3)CC2)CCCN1C(c1cccnn1)=O CCCCCC(=O)N1CCOC(CNC(=O)CN2CCNC(=O)C2)C1 C1(CNC(Cn2ccc(C)n2)=O)CN(C)CCN1C(c1ccc(C(C)C)cn1)=O c1(C(=O)NC2CC(N(C(=O)CSC(F)(F)F)C)C2)cccn2ccnc12 C1(C(=O)NC(CNC(c2c(CC)n(C)nn2)=O)C2CC2)C2CCCCCC12 N1(C(C(COC)OC)=O)CC(NC(c2ccoc2)=O)CCC(O)C1 C1(C(n2cc(C3COCCN3Cc3ccncc3Br)nn2)C)CC2CCC1CC2 c1(C(N2CC(C)(NC(C3C(=C)C3)=O)C2)=O)ccc(-n2cccc2)cc1O NS(=O)(=O)c1ccc(C(=O)NCC(O)CNC(=O)CN2CC3CC3C2)cc1 C1(NC(=O)CCc2cnco2)CCN(C(=O)CC2CC2)C(c2ccccc2)C1 C1(C(N2C(CCNC(C3(C)CC=CCC3)=O)CCC2)=O)CCC2C(C1)C2(F)F C12(C(N(CCCNC(=O)Cc3cc[nH]n3)CCO)=O)CCC(F)(CC1)CC2 N1(C(C2(O)CC(C)(C)C2)=O)CCC(NC(c2cc[nH]c2)=O)C(CO)C1 Cc1cc(C(N2CC(N3CCN(C(=O)Cn4cnnc4O)CC3)C2)=O)c(O)nn1 CC(CC(=O)NCC(C)CN(C)C(C1CC(C)(C)C1)=O)c1ccco1 N1(C(Cc2c(C)nc[nH]2)=O)CCC2CN(C(=O)C(O)CC[S+](C)C)CC2C1 C1(c2ccccc2)(C(=O)NCCCC(c2cccnc2)=O)CCCCO1 CN1CCN(CC(=O)NCC23CC2CN(C(=O)COc2ccccc2)C3)CC1 c1(NC(CC)(CNC(C2CCC(C)CC2)=O)CC)ccc(C#N)c(C)n1 c1(C(N2C(C(=O)Nc3cc(OC)cc(F)c3)CC2)=O)c[nH]c2ccc(F)cc12 C1(NC(CC2N(C)CCCC2)=O)CCCCCCC1NC(=O)CC=CC(C)(C)C CS(C)(=O)=NCC(=O)NC1CCN(C(=O)Cc2cccnc2Br)C12CC2 c1(OC)ccc(C(N2CCN(C(=O)Cn3cnnc3O)C3CC23)=O)cc1Cl C(CCCC(C)NC(=O)C(CC1CC1)CC1CC1)NC(CCCSC)=O C(=O)(CC(C)CC(C)(C)C)NC1CN(C(c2cnc(C)n2C)=O)CC1O CC1CC(NC(=O)C(=O)Cc2ccccc2)CCN1C(=O)Cc1cocn1 CCC(CC)C(=O)N(C(CC)CC(=O)NCCC1(COC)CCC1)C c1(C(=O)NCC(CC)NC(c2cnc(C)[nH]2)=O)c(C)oc(C)c1Br c1(C(C(C)C)NC(C2(c3ncon3)CC2)=O)ccccc1Cl C(=O)(CCCNC(=O)COC)N(CC(C)NC(=O)CCOC(C)CC(C)C)CC C(CCCNC(=O)CCC1CCCOC1)(c1ccccc1)NC(C=C(C)Cl)=O CCCC(C(=O)OC)C(=O)NC1CC1NC(c1sc(O)nc1C)=O c1(CCC(=O)NCCN2CCN(C(C3C(=C)CC3)=O)CC2)ccc2ncsc2c1 C1(C(=O)Nc2cn(CC#C)nc2)CCN(C(=O)C2=C(C)OCCCS2)O1 C1(CC)(NC(=O)C(C)CC(F)F)CCN(C(c2ccncc2)=O)CC1 c1(CC)sc(C(=O)NCC2CCN(C(=O)CCC3CCOCC3)C2)cc1C c1(N(CC=C)C)ccc(Br)c(S(=O)(=O)NCCc2c(F)cncc2F)n1 c1(CC(=O)NCC)ccccn1.C1(C(F)F)CC1 C1(C(=O)NC2(CC)CCOC2)CC2CCC(C1)N2C(c1cc(C(C)=O)[nH]n1)=O N1(C(c2c(NC)c(F)ccc2)=O)CC2CCCC(C1)N2C(C1(SC)CCC1)=O Cc1cccc2[nH]c(C(N3CCC4CCC(C3)N4C(=O)CNC(N)=O)=O)cc12 C1(C)(NC(c2ncn(CC)c2)=O)CCN(C(c2cc(-c3csc(C)n3)c[nH]2)=O)C1 C(CN=c1nc(C#N)[nH]cc1C)C1N(C(Cc2cnc(C)s2)=O)CCCC1 C12(NC(c3nn(CC)c(C)c3)=O)CCCC1CN(C(c1cc(C)oc1C)=O)C2 C(=O)(C(C)(C)CC(C)C)NCC1OCCC(NC(c2c(Cl)cnc(CC)n2)=O)C1 C1(C(=O)NCC(C)N(C)CC2CC23CCOC3)COCCN1C1CCCC1 Cc1cc(Br)c(Cl)cc1NC(C1CC1NC(c1cc(=O)cco1)=O)=O C1(C)(NC(C(C)CCN(C)C)=O)CCCN(C(=O)CC2CCC(C)C(C)C2)C1 C1(CNC(C(COC)C)=O)CC2CCCCC2N1C(=O)CCn1cccnc1=O N1(C(C(F)OC)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C(C)C)=O)C(C)C1 c1(C(=O)NC2CC3CN(C(C4ON=C(C)C4)=O)C2C3)c(C)[nH]c2ccccc12 Cc1ccc(C(=O)NC(C2CCN(C(=O)CC3COCCO3)CC2)(C)C)c(C)c1 c1(OC)ccc(C(=O)NCCCNC(C2CS(=O)(=O)CC23CC3)=O)c(OC)c1Cl C(=O)(C#CC1CCCCO1)NCCCN(C(c1c(Br)ccc(C)n1)=O)C1CC1 Cc1cccc2oc(C(N3CCCC4(C3)CN(C(C3(C)CC3(F)Cl)=O)C4)=O)cc12 c1(C(C)C(=O)NCC2(F)CN(C(=O)CCN3CCCC3)C2)nc(F)ccc1Cl N1(C(CC2CN(CCN(C)C)CC2N)=O)CCc2cc(C(F)(F)F)ccc21 N1(C(CCC)=O)C2CCC1CC(CNC(c1ccc(OC(F)F)cc1)=O)C2 c1(C(=O)NCC2CC(NC(C(C)N(CC(F)(F)F)C)=O)C2)ccc(N)cc1Cl C(=O)(C(CNC(c1ccn2nccc2c1)=O)CC(C)C)NCCN(C(=O)OC)C C1(C(N2CCCC(OCC)C2)=O)CC2(CCN(C(=O)C(c3cccn3C)=O)C2)C1 CN1CC(C)(C)CC1C(N1CCCC1c1cn(-c2c(F)cccc2Cl)nn1)=O Cc1cc(C(N2CCCCC(NC(c3ccc(Cl)nc3O)=O)C2)=O)nc(C)c1 C(=O)(C1=NOCC1)N(CC(CC)NC(=O)Cc1cccc(OC(F)F)n1)CC N1(C(=O)CS(=O)(=O)N2CCOCC2)CCC2CCN(C(=O)C(F)C3CC3)C2C1 CN1N=CC(CC(=O)NCC2CN(C(C3CCS(=O)(=O)C3)=O)C2)C1=O CCC(C#N)C(=O)NC1(C)CC(NC(c2cc(C(F)(F)F)on2)=O)C1 c1(C(=O)NCCN(C(CC(C)n2ccnc2)=O)C)ccc(C(=O)N(C)C)c(F)c1 c1(CNC2(c3n(C(C(=O)OC)C)nnn3)CC(F)(F)C2)ccc(C)c(Br)c1 C1(CC(=O)NC2(COC)CN(C(=O)C(CO)N(C)C)C2)CC2(CC2)CO1 C(=O)(C1=CCc2ccccc21)NCC1C(NC(c2cc(C3C(C)C3)on2)=O)CCC1 c1(C(=O)NCC2C(NC(C(CC(C)C)O)=O)CCC2)ccc2c(c1)CC(C)O2 Cc1nn(CC(F)F)cc1-c1nc(-c2occc2C)nn1CCCN(C)C c1(C(=O)NCC2C(NC(C3CN(CC)C(=O)C3)=O)C2)cncc(Cl)c1C N1(C(C(COC)(C)O)=O)CCN(C)C(CNC(=O)Cn2nc(C)cc2C)C1 c1(OC)cc(C(N2CCC(CNC(C3CNC(=O)C3)=O)CC2)=O)cnc1Cl C#CC1CC2(CC2)CN1C(=O)NCC(C(C)C)c1ccccc1 N1(C(C(C)OCCOC)=O)CCC2CCCC12C(=O)NCC1CCC(C)(CO)O1 C(=O)(CCCCCCC(=O)NC(CO)C(C)NC(=O)C(F)OC(F)(F)F)OC N1(C(C2CC(O)CN2S(=O)(=O)CCc2ccccc2)=O)CC2(CC2)CC1CN C(=O)(CC1=NN(C)C(=O)C1)N1CC(CC)C(NC(c2cc(Cl)c(Cl)[nH]2)=O)CC1 CN1CC2CC1CN(C(=O)CCC1CCCCN1C(=O)COc1ccsc1)C2 C1(NC(C2CCCC(C)CC2)=O)CC2CCC1N(C(=O)C=Cc1cccnc1)C2 C1(CNC(c2c(CNC(CCC#C)=O)ocn2)=O)CCC(=O)NC1C C1(CNC(C(C)CCN(C)C)=O)CC2(CCN(C(C3(C)CCCN3C)=O)CC2)C1 c1(C(C)C)ncc(Br)c(=NC(CNC(C2CCC(=O)N(C(C)C)C2)=O)CO)[nH]1 C1(C)(CNC(c2cc(CCC)[nH]n2)=O)COCCN(C(=O)C(C)c2ccsc2)C1 c1(N(C)Cc2cc(Br)cs2)nc(N2CCN(CS(C)(=O)=O)CC2)c2c(n1)CCS2 N1(C(C2(CC#C)CCCO2)=O)CC(C(N2CC(F)(CF)C2)=O)CCC1(C)C C(C1CCCC1)=C(C)C(=O)NCC1CN(C(C2(n3cc(C(C)C)nn3)CC2)=O)C1 N1(C(C(CSC)O)=O)CC(NC(=O)Cc2csc(C)c2)C(C2CC2)C1 CCC(C)(C(=O)NCCOCCCNC(=O)Cc1ccoc1)OC N#Cc1cnn2ccc(N3CCCCC(NC(=O)Nc4ccccc4F)C3)nc12 C(=O)(CCCCC(C)C)N1CCCC(O)(CCNC(CC(C=C)C)=O)C1 C(C(O)C(C)(C)C)NC(c1scc(CNC(CC2C(CC)C2)=O)c1)=O c1(C(N(C(CNC(=O)C(C)(F)C(F)(F)F)C2CC2)C)=O)cc([N+](=O)[O-])ccc1Cl CCC(C)(C)C(O)C(=O)N(CCC(=O)NC(C)(CO)C1CC1)C C#Cc1ccnc(C(N2CCN(C(c3cc(O)cc(=O)o3)=O)C3CC23)=O)c1 c1(C(C)NC(c2c(C(=O)NC(CC=C)=O)ccs2)C)[nH]c(C)nc1C c1(C(=O)NC(CCC)CCCNC(=O)CC(CC)C2CC2)cn2cccnc2n1 Cc1noc(C)c1CC(=O)N(C)CCC1CCCCN1C(C1CC1C(C)(F)F)=O C1(C2CCC2)(C(=O)NCC(CO)NC(C2(c3cccc(F)c3)CC2)=O)CC1(F)F C1(NC(c2cc(C)cc(F)c2N)=O)CCCC2CN(C(=O)C3=CCOCC3)CC12 C#CCC(CC(=O)NC(c1nnnn1C)C)NC(C1(C)CCOCC1)=O C(=O)(C1CCc2nccn21)N(C)CC1CCN(C(C2CCCS2(=O)=O)=O)CC1 C(=O)(C(CC(C)C)N(C)C)NC(CCN(C(CC(C)SC)=O)C)C c1(C(=O)OCC)cc(N(C2CCN(C(c3ncoc3CC)=O)C2)C)nc(C)n1 N1(C(C(C=C)O)=O)CCCCC1CCC(=O)N1CC(N(S(C)(=O)=O)C)C1 C1(CO)CCCC2(CCN(c3nnc(-c4csc(CO)n4)s3)CC2)O1 C1(O)(CNC(=O)C(c2ccccc2)O)CN(C(=O)CCCC2CC2)C1 C1(C)(CNC(CN(CCOC)C)=O)CCC(NC(=O)C(C)=CC(C)C)C1 c1(OS(C2C(NCCOC)CC2)(=O)=O)ccc(S(=O)(=O)C2CC2)cc1F c1(OC)c(Br)ccc(F)c1CNC(c1ccc(F)cc1F)C1CC1 C(C(CC(=O)NC1CN(C(=O)CC2(C)CC2)CC(C)(C)C1)C(F)F)N(C)C C(=O)(C(C)CC(F)(F)F)NC1C(CCC)CN(C(C2C=CC=CC=C2)=O)C1 c1(C(N(C2CCN(C(C34CCC3C4)=O)C2)C)=O)cccc(C#N)c1 c1(C(N2CC(CC=C)(NC(c3nc(C)sc3C)=O)C2)=O)cc(C#N)ccc1O C(=O)(CCC(F)F)N1C(C(C)(C)CNC(=O)CCCc2ccccc2)CCC1 N(C(=NCCCF)NCC(C(=O)OC(C)(C)C)Nc1ccccc1)CC(=C)C C1(F)(CNC(c2c(C)onc2)=O)CC2CCC(C1)N2C(=O)Cc1ccsn1 CC1CN(C(c2cccc(C#N)c2)=O)CCC1N(C(=O)C1=CCOCC1)C c1(C(N(C)CC2CN(C(=O)C=Cc3cncnc3O)C2)=O)cc2ncccc2s1 c1(OCC)cc(Cl)ccc1C(=O)NC1CN(C(C2CCCC2(F)F)=O)C1 c1(C(N2C(C)CCC(NC(C3CC34CCOC4)=O)C2)=O)cccc2c1OCCN2 c1(OC)ccc(CN2CC3CC2CN3C(=O)C(C)NC(=O)C(C)(C)C)cc1F C1(NC(c2n(C)nc(CNC(=O)CCCCCF)c2)=O)CC2(C1)CC(C#N)C2 N1(C(COCC)=O)CCN(C(c2scnc2CC)=O)CC1COC CCCCC(C(=O)N1CC(C(N2CC(CC)(OC)C2)=O)CC12CCC2)C(C)C C(CC1CC1)(CC(=O)N1CCOCC1CCO)NC(c1ccn(COC)n1)=O S(=O)(=O)(c1cc(C(=O)Oc2ccc(C(=O)O)cc2Cl)c(Cl)cc1Cl)NC CCC(CCC(=O)N(C(C)CN(C)C(c1ccc(C(=O)OC)s1)=O)C)OC C(=O)(C1=CC2CCCC12)NC1(CNC(CNC(C(C)(C)C)=O)=O)CC1 C1(CC(=O)NC2(CCC)CC2)CCCN(C(C2CC(F)C(=O)N2)=O)C1 C12(CNC(C3CC(C#N)C3)=O)CCC(NC(=O)Cc3cccc(Cl)c3)(CC1)CO2 CC1=C(C(=O)Nc2ccc(-c3ccc(OC(C)(C)C)cc3F)nc2C)CCO1 N#CC1CN(Cc2ccc(N3CCCC3)nc2)CC1NC(c1cc(Cl)ncc1Br)=O N1(C(C2(S(C)(=O)=O)CC2)=O)CC2CCCC2(CNC(=O)Cc2ccc(O)cc2)C1 c1(NCc2c(CNC(CN(C)CC)=O)cccc2)ncc2ncnc-2[nH]1 CC1CN(C(c2cnnn2C)=O)CC1NC(C1(C)C=CCC1)=O N1(C(C2N(C(c3c(CC)nn(C)c3)=O)CC(C)C2)=O)CC2CC2C2CC12 C1(NC(C2CCSCC2)=O)CCCC(C(=O)NCC2C3CCCC23)C1 C1(CC(=O)NC(c2ccccc2)CNC(c2c[nH]c(=N)o2)=O)CCCN1C=O CC1CCCCC1CC(N1CCC(CF)(NC(=O)CNc2ncccn2)C1)=O N1(C(c2c(C)cnnc2)=O)CC2CCCC(C1)N2C(C12CCC(C)(CC1)CC2)=O c1(CC)cnccc1C(=O)NCC1C(C)CCN1C(=O)Cc1cnccc1C c1(C(=O)NCC2CC(C)N(C(c3cnnc(Cl)c3)=O)C2)cc(Cl)cc(F)c1N c1(C(N2CCC(N(C(=O)C3=NOCC3)CCC)CC2)=O)cn2c(n1)CCC(C)C2 C1(NC(N=S(CC#C)(C)=O)=O)CCOC2(CCC2)C1 C(C(CC1CCCC1)C(=O)NCCCN1CCC1)NC(CSCC=C)=O CC(C)CC(CC(=O)N1CCC(CCN(C)C)C1)NC(=O)CCC(C)(F)F Cc1cnn(C)c1C(N1CC(NC(c2ccc(OCF)cc2)=O)C(O)C1)=O C(=O)(C1c2c[nH]nc2CN1C(=O)CSC(F)F)NCc1cc(OC)ncn1 N1(C(c2cc(OC)ns2)=O)CCC(NC(=O)C=Cc2cccc(F)c2)C(C)(C)C1 c1(C(=O)OC)cc(F)ccc1NC1(CC(=O)NCC2(SC)CCCC2)CCC1 C1(C(=O)NC2(CC)CCN(C(C3SCCCS3)=O)CC2)CCC2CC(C)CN2C1 O=C1NCC2(CCN(c3nnc(-c4cccs4)n3CCCOC(F)F)CC2)N1 CC1(F)CCN(C(C2(C)CN(C(=O)CCn3cccc3)CC2C)=O)CC1 Cn1ccc(C(N2C3CCC(C3)C2CNC(C2CC2c2cccs2)=O)=O)cc1=O Cc1ccn(CC(C)C(=O)NCC2(NC(C3CC(=C4CC4)C3)=O)CCOC2)n1 C1(CC(=O)N(C2CCCC2)CCCNC(c2c(C)n[nH]c2)=O)CC(C)(C)CO1 C1(O)(CC)CCN(C(=O)CC2CC2CNC(=O)C(C2CCCCC2)F)C1 Cc1n[nH]c(C)c1CCC(=O)NCCC1COCCN1C(=O)CN(C)C1CC1 C(=O)(CCC(=O)c1ccc(F)cc1)NC1C(CNC(C(C)(F)F)=O)CCC1 C1(CC)C(NC(=O)CCN2CCCC2)CCCN1C(c1ccc(F)c(F)c1)=O C1(Cn2cc(C(C)(C)SC)nn2)N(C(C23CCCC2C3)=O)CC1(C)C c1(C(N2C3(C#C)CC(C2)C3)C(=O)Nc2cccc(Cl)c2C)c(Cl)cc(Cl)cc1Cl c1(N2C(C)CC(NC(C3CNC(=O)CC3C)=O)C2)c(C#N)c(=O)n(C)c(=O)n1C N1(C(CCNC(=O)OC)=O)CCN(C)C(CNC(c2cc(C3CC3)[nH]n2)=O)C1 C1(NC(c2cnc(C)nc2)=O)CC2CC(NC(C3(CCF)CC3)=O)C2C1 c1(C(=O)OCC)ncc(Br)cc1NC(C1(c2cccs2)CC1C)=O C1(C)(C(N2CC(F)(CC)C2)=O)CCN(C(=O)C#CC2CC2)CC1 N1(C(c2c(S(C)=O)cccc2)=O)CCC(C2CCCN(c3nnns3)C2)CC1 CC1(C)C2CCC1(C(=O)NCC(N1CCN(C(=O)CCn3ccnn3)CC1)=O)CC2 c1(OC)c[nH]c(C(=O)NCCCCCCC(c2cncn2C)C(=O)NC)cc1=O Cc1cccc(C(N2CC(O)CC2C(=O)NCCC(C)C(C)(C)C)=O)c1C C1(c2ccccc2F)(C(=O)NC(C)C(CO)NC(=O)C(C)CO)CCCCC1 C1(NC(C(C)Oc2cccnc2)=O)CC(N=c2nn[nH]n2-c2ccccc2)C1 C1(NC(C(CC)NC(N)=O)=O)CCN(C(=O)C(Cl)=CCl)CCC1(F)F C1(O)(CNC(C2CC(OC)C2)=O)CCCN(C(=O)CCCc2nncn2C)C1 c1(C(C(C)C)NC(C(=O)OC)COC(C)(C)C)ccc2c(c1)OCCO2 CN1CC(C)(C(=O)NCCCNC(=O)Cn2cc(CO)nn2)CCC1=O N1(C(C(C(C)C)O)=O)CCOC2(CCCCC2NC(C2CNC(=O)C2)=O)C1 C1(NC(c2c(C(C)C)ncnc2)=O)CC2CN(C(C3(C#N)CC3)=O)CC2C1 c1(C2C(CNCc3nc(CC)on3)C2)ccc(Br)cc1 C1(C(F)(F)F)(NC(N2CCN(CCOCCO)CC2)=O)CC2CCC1CC2 c1(C(=O)NCC2N(C(CCCc3nnc(C)n3C)=O)CCC2)cccc(O)c1C CCCC(C)CN=c1ccc(S(=O)(=O)N(CC(C)N(C)C)C)c[nH]1 c1(C(=O)NCC(CC)NC(=O)CCC=CBr)cc(N)cc([N+](=O)[O-])c1 CCC(CCC(=O)NCC1(CO)CCN(C(=O)CCCn2ccnc2)C1)OC c1(C(=O)NC23C(CN(C(c4cc(=N)[nH]c(=N)[nH]4)=O)C2)CC3)cccn2cnnc12 C1(CC)CN(C(=O)C(CC2CC2)NC(C2CC(O)CN2C)=O)CCN1C C1(NC(=O)OC(C)(C)C)CCCCC1CNC(C1CN(C(=O)C(N)=O)CCO1)=O N1(C(C2CC(C)N2C(C2CC(O)CN2C)=O)=O)CC2COCC2(C)C1 C(=O)(C(CCCC)C(C)C)NCC(C(=O)NC(C1CCCCC1)C#C)CC1CC1 N1(C(c2cn(CC=C)nn2)=O)CCOC2(CCN(C(C3(CC)CC3)=O)C2)C1 C(=O)(C(C)(C)CF)N(C)CC1C(NC(C(CC)OC)=O)CCC1 c1(C(N2CCC(NC(CCCC)=O)CC2C)=O)ccc(Cl)c(F)c1F CCC(CN=c1ccc(S(=O)(=O)NCCC2CCCS2(=O)=O)c[nH]1)N1CCCC1=O Cc1cccc2[nH]c(=NC3CC(CNC(=O)C4=CCCCO4)C3)sc12 N1(C(=O)NCCn2nnc(C)n2)CCC(OC)C1(C)C C1(C(N2C(C)CC(CNC(c3ccncc3)=O)C2)=O)CC2C=CC1C21CC1 CC1CSCCCN1N1CCCC1.C1(C=O)CCN(CC(F)F)CC1 C1(C(=O)NCCn2cc(C(N3CC(OCC)C3)=O)nn2)OCCC1(C)C N1(C(c2c(CCC)nco2)=O)CCC(F)(F)C(CNC(c2sc(F)cc2C)=O)C1 C1(C(=O)NCC=CC)CCN(C(=O)Cc2cccnc2)C1C N1(C(C)=O)CCCc2cccc(N3CCCC3)c21.Cc1cc(C(=O)C)c(C)[nH]1 N1(C(C2(c3cn(C4CC(COC(C)=O)C4)nn3)CC2)=O)CCOC(C)C1CO CC(C)CC(C)CC(=O)N1CCC(F)C(NC(=O)C(C)(C)c2cscn2)C1 c1(C(=O)NC2C(OC)CN(C(=O)CC(C)N(C)C)C2)cccc(C)c1O N1(C2(C)CC2)N=C(C(=O)NCC2CCN2C(c2cc(C3CC3)[nH]n2)=O)CCC1=O N1(C(C2(SC)CC(C)(C)C2)=O)CC(C(=O)NCC2(O)CCN(C)C2)CC(C)C1 C1(C(=O)NC(CC)CN(C(=O)C=Cc2nccs2)C)CN(C)C(=O)CCO1 CC1C(C(=O)NC2C3CC2N(C(C2(C)CCCC2)=O)C3)CCN1C CCCC(O)(CCC)CC(=O)NCC(C)CN(C(=O)CS(=O)(=O)CC)C c1(SC(C)C)ccccc1C(=O)N(CC(C)NC(c1ccc(COC)cc1)=O)C c1(C(=O)NCC2CN(C(C(=O)NCC)=O)CC23CC3)ccc2nnn(C)c2c1 C1(CC(C)C)(C(=O)NC2CCC(CNC(C3(C#N)CC3)=O)C2)CCNC1=O c1(CN2C(CNC(c3ccc(=NC)[nH]c3)=O)CCC2)cn(C)c2c(Cl)nccc12 c1(C(=O)NC2CCC(NC(COC3(C#C)COC3)=O)C2)cnc(CN(C)C)nc1 N1(C(C2(C=C)CCN(C(=O)CCOC3CCC3)C2)=O)CC(C)OCCC1C N1(C(c2nc(C)sc2)=O)CC2CC(C1)C2C(=O)CC1CCCC1C c1(C2(C)CC2)ccc(C(=O)NCC2CC(F)(F)CN2C(c2cnsn2)=O)cc1F C1(C)(SCc2cnc(C(C)(C)C#N)s2)CC2CC2C1 C(=O)(C(C(C)NC(c1ncccc1Cl)=O)C(C)C)Nc1c(OC)cc(F)cc1 C12(CNC(c3ncn(C)c3)=O)CC1CN(C(=O)CCCC1CCOCC1)C2 C1(c2n(CCOC(C)C)nc(-c3ccccc3)n2)CN2CCC1CC2 C(=O)(CCCC(C)(C)C)N(C1CC1)C.CC1CCCc2n[nH]nc21 c1(C(=O)NCC2CN(C(CC(=O)OC)=O)C2)oc(C2CC2)nc1C(F)F.C1CC1 C=C(C)c1cccc(NC(=O)C(CCC)NC(=O)CC2CC(F)(F)C2)c1 c1(CC)nc(N2CC3C(NC(=O)CC(C)(O)COCC)C3C2)c(F)c(Cl)n1 CC1(C)CCC1C(=O)NCC1(CCNC(c2ccn(C3CC3(F)F)n2)=O)CC1 N1(C(C(CC)SC)=O)C(C)C2CC1C2NC(=O)CNC(c1cnoc1C)=O C1(NC(C2(CC#C)CCCCC2)=O)CC2CCC(C1)N2C(=O)C1=C(C)CCCC1 C1(NC(C2OCCN(C(c3cnn(CC)c3C)=O)C2)=O)=CN=C(O)CN=C1C c1(CC)cccc(C(N2CCOC(CNC(=O)CSCC(C)C)C2)=O)n1 N1(C(c2ncc(OCC)nc2)=O)CCCCC(CNC(C2(F)CC=CC2)=O)C1 C1(NC(C=CC(C)(C)SC)=O)CN(C(=O)C=C2CCN(C)CC2)CC1CN(C)C c1(C(C)(C)C)scnc1C(=O)N(CCNC(C1CCCN1C1CC1)=O)C1CC1 C1(C(=O)NCCCN(C(CC=C)=O)C)CC2(C1)CC(F)C2 C1(OC)CC(NC(c2cncnc2)=O)CN(C(=O)Cn2ncc(Br)n2)C1 C1(N(C(c2c(C)nc[nH]2)=O)C)CCN(C(=O)C(C)Oc2ccc(F)cc2)CC1 C1(=O)CCN=C(NC2CCS(=O)(=O)C2)NCCN1.C1(SC)CC(=O)N(C2CC2)C1 CCCCC#CC(C)(C)NC(C1CC(C)N1C(C1CCC(=O)NC1)=O)=O Cc1cc(=NC(=O)C(=O)N2CC(CNC(c3cncc(F)c3)=O)C(O)C2)[nH]o1 C(CC(O)C(=O)NCC(CC1CCCC1)C(=O)NCC(c1ccccc1)C)SC C1(c2onc(CN(C)C)n2)CN(CC2(C)CSCCO2)CCO1 N1(C(c2cc(C)[nH]c2C)=O)CCCC(CO)(NC(C2CCSC(C)C2)=O)C1 C1(c2n(C)nc(-c3cccc(OC(C)(C)C)c3)n2)CCCC1S(C)(=O)=O C(=O)(C(C(C)C)NC(N)=O)NC(CC(C)NC(C(C1CCCC1)OC)=O)C c1(CN2CC(O)(CNC(C(C(C)C)c3ccccc3)=O)C2)c(F)cccc1F C(=O)(C(O)CCCNC(C1CCOC(C)(C)C1)=O)NCC(C=C)(C)C N1(C(c2cc(C)on2)=O)CCCC(C2CN(C(=O)C(C3CC(F)(F)C3)O)C2)C1 c1(OCC(=O)N(CC(CC)NC(=O)Cc2cncn2C)C)cncc(Br)c1 C1(C(N2CC(c3ccccc3)(NC(C(F)OC)=O)C2)=O)CCN(C)C(C)C1 C1(C(=O)NC2(C)CN(C(C3(CC#C)CCCO3)=O)C2)CC(c2ccccc2)=NO1 C1(C(=O)NCC(C#C)CC)C(C)CCN1C(=O)C=Cc1cocn1 N1(C(=O)Nc2csc(-c3ccc(Cl)cc3)n2)c2ccc(Cl)cc2N2CCC1C2 c1(CC(N2CCC(N(C)Cc3ccc(Cl)nc3)C2)=O)ccnc(O)c1 Cc1cncc(C(=O)NC2CCCC(NC(c3ccccc3Cl)=O)C2)c1 N1(CC)CC(C(N2CCC(C)(NC(=O)C(F)=CCCF)C2)=O)NC1=O c1(OC)ccccc1CCOC(=O)CC1CCCC(C)C1 c1(C(=O)NC2(C)CN(C)C(=O)CC2)cc2n(c1)CCCNC2=O c1(CC(=O)NCC(CNC(C2(CC=C)CCC2)=O)C)ccc(F)c(Br)c1 CC1CC=C(C(=O)NC2CCCCC2NC(=O)COc2ccc(Cl)nc2)CC1 N1(C(c2ccc(N(C)C)cn2)=O)CCCCCC(Nc2ccccc2[N+](=O)[O-])C1 c1(C(C(=O)NC2(c3cn(-c4ccc(OC)cn4)nn3)CC2)=O)ccc(Br)c(F)c1F O=C(N=c1[nH][nH]c2c1CCCC2)C1CCN(C(c2cc(Br)ccn2)=O)CC1 N1(CC(=O)NC2(C)CCN(C(c3c(C)cco3)=O)C2)CCSC2CCCCC12 CCCC(C)(CCC)C(=O)NC1C2CC3C(C2)C13C(=O)N(CC(=O)N(C)C)C C(CCCCC(=O)NCC(CO)NC(=O)CCN1CCC(F)C1)=CC N1(C(C2N(C(c3cc(C)c(C)nn3)=O)CC(O)C2)=O)CC2(CCC1CO)CC2 N1(C(CSCC#C)=O)CCCC(C(C)C(=O)NCC2(CC)CCC2)C1 N1(C(CC2OCCC(C)(C)C2)=O)Cc2ccccc2C(NC(=O)CC2CCC2)C1 c1(C(=O)NCC(CC=C)NC(=O)CC(C)(C)COC(C)=O)ccc2[nH]ccc2c1 N1(C(c2c(C=C)cncc2)=O)CC=C(C(C)(C)C(=O)NCC(C)(O)CC)C1 c1(OC)cc(CNC(Cn2cncn2)C(=O)O)cc(C#N)c1 CC(C)CC(O)C(=O)N1CCOCC1CNC(=O)CCN1CCCCCC1 c1(C(=O)NCCC2CC(OC)CN2C(C2CCOC2)=O)c(F)cc(Cl)cc1F C1(CNC(C(CC=C)C)=O)CC2(CCOCC2)CN1C(=O)C(F)=C1CCCC1 c1(C(N2CCC(C(C)NC(=O)Cn3cc(Cl)cn3)C2)=O)ccc2nc(O)oc2c1 C1(CNC(c2scnc2C(F)(F)F)=O)COCCN1C(=O)CC1(O)CCC1 C1(NC(c2ccn(CC(C)C)n2)=O)CC2(C1)CC2NC(=O)Cc1cccc(Cl)c1 S(=O)(=O)(c1ccc(NC2CCCC3CC23)cc1Br)N1C(C(N)=O)CC(F)C1 c1(C(=O)NC2CC3CN(C(Cc4cc(C)no4)=O)C2C3)ccc(P(C)(C)=O)nc1 N1(C(=O)CC2CCCCO2)CCOCC1NC(CC1CC(NS(C)(=O)=O)C1)=O Cc1cc(Cl)c(Cl)cc1CC(N1CC(NC(c2c(C)cccc2C)=O)C(F)C1)=O C1(C(=O)NC2C(C(=O)NCCCCC(=O)OC)CCC2)OCCCC1(C)C C1(CCOC)CN(C(C2CCCCC(=O)N2)=O)CCN1C(=O)CN1CC(C)C1 c1(C(=O)NC2CC(C)N(C(c3cnc4sccn34)=O)C2)c[nH]c(=N)nc1O C1(N2C(N3CC(C)(C)OC3=O)CCCC2)CCC2(CCNCC2)CO1 c1(CC)noc(C(N2CCOCC2CN(C)C(C2(COC)CCCC2)=O)=O)c1C Cc1cc(C)c(C(=O)NC(C2CC2C(=O)NCc2nn[nH]c2C2CC2)C)s1 CCCCCC(CC)C(=O)NCC(=O)NCC(=O)NC12CC1COC2(C)C C(=O)(C#CC1(C)CC1)NCCC(C)(C)OCCOC(C)C(=O)Nc1ccccc1 CCC(CN(C)C)CC(=O)NCC(C)CNC(c1cnc(OC)c(C)c1)=O C(CCCCC(=O)NC(C)CCN(C)C(c1cn(C2CC2)nn1)=O)=CC CC(C)CC(CC(=O)NC1(CNC(=O)CCc2cc[nH]n2)CCOC1)CC(N)=O C(=O)(C(C)CS(C)(=O)=O)NC1(CNC(c2cn(CC)nc2C(C)C)=O)CCOC1 N1(C(C(C)C#N)=O)CCC(C2(NC(c3cc(C4(C)CC4)ccc3F)=O)CC2)C1 N1(C(CCOCCOCC)=O)CCC2(CCN(C(c3ccc(C#N)[nH]3)=O)C2)C1 N1(c2nnc(CC)o2)C(CNC(=O)C=Cc2cocn2)CC2COCC12 c1(OC(=O)CCN(C(C2CCCO2)=O)C2CC2)ccccc1Cl c1(C(N2CCC(CC=C)(NC(c3cc(C)sc3C)=O)C2)=O)cccc(F)c1F c1(CC)noc(C)c1C(=O)NCC1(F)CC(CNC(C2CC2F)=O)C1 N1(C(c2c(C)nc[nH]2)=O)CC(N(C)C(c2ccnc(C3CC3)c2)=O)C2(CC2)C1 Cc1nc2ccccc2n1CC(=O)NC1CN(C(C2CCSC2)=O)CC1O CC1(C)CC(N=c2[nH]nc(C(F)F)o2)CN(Cc2nc[nH]c3nccc2-3)C1 C(C)(C(=O)N1CC(c2ncccn2)C1)(C1CCC1)NC(COCCN(C)C)=O c1(CNC(N2CCOC(C(C)C)C2)=O)cc(F)cc2c1CCC2 c1(C(=O)NC(C)C(C)NC(=O)C=Cc2ccccc2)ncc(Cl)cc1Cl c1(OC)ncnc(OC)c1C(N1CC(CN(C)C(C2CCCCC2(C)C)=O)C1)=O CP(C)(=O)CC(=O)NCCOCCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O CC1(C=O)CC(c2cc(Cl)cc(Cl)c2)=NO1.C12CCCN(C1=O)CN2 c1(C(=O)NC2CCCC(CNC(c3ccc(C)n3C)=O)C2)cc(F)cc(Cl)c1N c1(CC)cc(C(=O)NCC2CC2C(=O)NC2CC(CC)(CC)C2)on1 C=Cc1ccc(C(=O)NCCC2CC(C(N3CC(OC(=O)N(C)C)C3)=O)C2)cc1 c1(C(N(CC(CN(C(C2C(OC)CC2)=O)C)O)C)=O)cccc(C)c1[N+](=O)[O-] c1(N(CCCC)C(c2csc(-c3ccc(C)cc3)n2)=O)ccc(F)cc1 c1(CNc2c(NC)ccc(F)c2)cc(=O)n2c(n1)CCCC2 c1(OC)cc(C(=O)NC(C2CCN(C(=O)CC#N)CC2)C)cc2c(C)c(C)[nH]c12 CC(C)(C)CCCCNC1(c2nnnn2-c2ccccc2)CCCCCC1 n1(CC(=O)N(C2CCCC2)CCC2CCC(NC(=O)CNC=O)C2)nnc(=O)[nH]1 c1(C(=O)NCCCCCCN(C(=O)CC2CCC(=O)N2)C)ccc([N+](=O)[O-])s1 CC1CC(CC(=O)NC2CCOC2(C)C)CN1C(=O)CC=C(Cl)Cl O=C(NNc1cccc(Br)c1F)c1ccc(SCC(F)(F)F)nn1 C1(CC(=O)NCCNC(C2C=CCCC2)=O)COCCO1 C1(F)(CNC(C(C)O)=O)CCC(CNC(=O)Cn2cc(CO)nn2)C1 C1(CCN(C(=O)CC2(C)CCCO2)C)CCCCN1C(=O)CCCN1CCCC1 C1(C(=O)NC2(C)CC(NC(=O)CC3(O)CCOCC3)C2)CC2C(C1)C2(C)C C1(COC)CCC(NC(=O)CC2CCCN2C(=O)CC2CC(SC)C2)CC1 c1(C(=O)NC)cccc(NC(=O)C(N2CCNC(C)C2)=O)c1Br C1(NC(c2c(C)nc[nH]2)=O)CCCCC1NC(C1CCN(c2ccncc2)C1)=O O=C(NNc1cc(F)c(Br)c(F)c1)NCCc1ncc(C(F)(F)F)cc1Cl C1(CNC(=O)C(O)C2CCC2)CC2CCCCC2N1C(=O)CCC1CCCOC1 c1(C(N2CCCSCC2)=O)cccn2ncnc12 C1(CC=C)(NC(c2cccc(NC3CC3)c2)=O)CCCN(C(=O)C(C)O)C1 N1(C(c2n(CC)nnc2)=O)CCC2CCN(C(c3nnc(C(C)(C)C)s3)=O)C2C1 C1(C2CN(C(C3CC(C)(C)O3)=O)C2)(NC(c2c(C)nc(CC(C)C)o2)=O)CC1 CCCCC(=O)NC1CC(C(F)C(=O)N2CC(C3CCCCO3)C2)C1 C1(NC(C2(COC)CC(=C)C2)=O)CCN(C(=O)CSc2nncs2)CC1CO C1(CNC(CCC2CCN(C)CC2)=O)COC(C)(C)CN1C(=O)CC1CCCO1 C12(CNC(C3CCC4(CC4)C3)=O)CC1CN(C(=O)C=CCO)C2 c1(CC(C(=O)NC(C)CCN(C(=O)CCc2nncn2C)C)O)ccc(Cl)cc1 c1(C(=O)NC2CN(C(C3CCC(C)NC3=O)=O)C2)cn2cc(Cl)cnc2n1 C(=O)(C1CCc2c[nH]nc21)NC(CCC=C)C(=O)Nc1cc(Cl)ccc1O C1(CNC(=O)C(N2CCC(C3CC3)C2)=O)CCC2(CCCCCC2)O1 N1(C(c2c(C)[nH]nc2Cl)=O)CCCC(C)C1CNC(C1CC(=O)NC(=O)C1)=O Cc1cc2c(cc1C)C(C(=O)NCCCCC(C)NC(C1CCCSS1)=O)CO2 C1(C(=O)OC)CCC1(C)C(=O)N(CCCNC(=O)C(C)CC)C1CC1 C1(C(c2nnnn2C2CCC2)NC(c2ncc(C(C)C)s2)C)CCC(C)CC1 C(=O)(C(C)CN(C(=O)C=C(C)C)C)N(C1CCCOC1)CC N1(C(C(C)(C)CO)=O)CCN(c2ncc([N+](=O)[O-])cn2)CC(O)C1 CCCN(C1CC1)N(C)Cc1cnc2ccccc2c1 CC(C)CCCC(C)C(=O)NC(C)CNC(c1cccc2c1OCC2)=O N1(Cc2n(CC)ncn2)CC2CCN(C(=O)CS(=O)(=O)C(C)(C)C)CCC2C1 c1(C(N2CCC(CC)CC2C(N2CCC(C3CC3)C2)=O)=O)cccc2ccccc12 c1(-c2cc(C(=O)NC3CN(C(C(CN(C)CC)O)=O)C3)no2)ccc(OC)cc1 N1(C(C(C=C)CC)=O)CCCC(C)C1CCNC(c1nc(Cl)ccc1N)=O N1(C(c2cccc(C(C)C)n2)=O)CCCC12CCN(C(c1cncs1)=O)CC2 N1(C(C(C(C)(C)C)NC(C)=O)=O)CC2CC(C1)N(C(=O)CCC1OCCO1)C2 Cc1cc(N2CCN(C(C)C(=O)N3CCCC3)CC2)cnc1O N1(C(c2ncn(C(C)(C)C)c2)=O)CCCOC(CNC(C2(C)CC2)=O)C1 N1(C(C(C)CC(F)F)=O)CC2COCCC2(NC(c2ccc(Cl)cc2Cl)=O)C1 C(c1ccsc1)=CC(=O)NCC(CC)NC(C1(N2CCNC2=O)CC1)=O C1(OC)COCCC1CC(=O)Nc1cccc(NC(C2(CO)CCCC2)=O)c1 c1(C(N2CCN(C(C(=O)NC(C)C)=O)C(C)C2C)=O)nnc(O)c2ccccc12 c1(NC(C2CC(O)CCN2Cc2c(F)cccc2F)=O)ncc([N+](=O)[O-])cc1Br C(CN=c1ccc(C(=O)NC2(C(C)C)CCCC2)c[nH]1)NC(=O)OC(C)(C)C C1(NC(COCP(C)(C)=O)=O)CCC2(CCN(C(=O)C3Cc4ccccc43)C2)C1 c1(NC(c2n(CCC)nnn2)c2scnc2Cl)cccc(OC(C)CC)c1 c1(NC(C(=O)NC2CC(F)(CNC(C(C3CC3)OC)=O)C2)=O)cccc(C)c1 c1(N(CCCCN(C(C(CC)NC(N)=O)=O)C)C)ccnc(C(F)(F)F)n1 c1(CC)cccc(F)c1C(N1CCOCC1CCNC(=O)C=Cc1ncc[nH]1)=O N1(C(C(C#C)(C)C)=O)CCCC(C(=O)NCC2(CO)CC3CC3C2)CC1 N1(C(C(CN(C)C)(C)C)=O)CC2(NC(=O)C(C3CCCCCC3)O)CCC1CC2 C(=O)(CCCCCN(C)C(c1nccn1C)=O)NCC(COC)OCC O=C(C(F)CC1CCCC1)NCC=CC(=O)NCC1CCCCS1 c1(C(N2C(CN(C)C(C3CC3c3ccsc3)=O)CC(F)C2)=O)cc2ccncc2[nH]1 Cc1cc(Br)cnc1C(=O)NCCC1CCN(C(C23CC(N(C)C)C2C3)=O)C1 C(CCC1CCC1)(C(=O)NCc1cnn[nH]1)NC(c1ccc(SC)o1)=O CC(C)(C)C1=NOC(C(=O)NC(c2ccccc2F)CNC(=O)C(C)(Cl)Cl)C1 Cc1cccnc1C=CC(N1CCC(NC(=O)CCc2cn(C)cn2)CC1C)=O N1(C(c2c(C)con2)=O)CCn2ncc(-c3cn(CCCCCO)nn3)c2C1 N1(C(c2cc(Cl)cc(Cl)n2)C(=O)NC(CC)(C)C)CCC(C2CCCC2(C)C)C1 CC(C)C(C(=O)NC1(C)CN(C(=O)C(C)(C)O)C1)NS(C)(=O)=O N1(C(C2C=CC(NC(CC3(N(C)C)CC3)=O)C2)=O)CCOCC(CO)C1 C(CCCCC(=O)NC1CCN(C(c2cnc(OC)c(Cl)c2)=O)CC1C)OCC C(=O)(C1=CC2(CCOC2)C1)N1C(C)CC(NC(=O)CC2CC(=O)C2)CC1 C1(C)(CC)C=C(C(=O)NC(C(=O)N(C)CC)C2CCC2)C1 CC1(C#CC(=O)NCC23CC2CN(C(=O)C(c2cc(Cl)cc(Cl)c2)=O)C3)CC1 C1(C(=O)NC(C2CN(C(C(C3C(C)C3C)OC)=O)C2)C)CCCCC1 C1(CC(=O)NCC2(F)CN(C(=O)COCCc3ccccc3)C2)CC=CCC1 C(=O)(CC(CC)C(C)C)NCC(CCCC)NC(c1ccsc1Br)=O N1(C(COC2(C)CCC2)=O)CC2(CC(C(=O)NC3(CN(C)C)CC3)CO2)C1 N1(C(C)=O)CCCC(C)C1CNC(=O)CCc1ncc[nH]1 c1(NC(c2ccc(-c3cc(C)c(O)cc3)c(C)n2)=O)ccc([N+](=O)[O-])c(Cl)c1Cl C1(C(=O)NC2C=CC(CNC(=O)CNC3CCOC3)C2)CC2OC1C1CC21 N12CC3CC1CN3C(=O)C(O)c1cccc(c1)C2=O.c1(CC)nccnc1OC C1(C)(C(N2CCCC(CN(C(C(C(=O)NC)(C)C)=O)C)C2)=O)CCC(C)C1(C)C N1(C(C2C(C=C)CC2)=O)CCN(C(c2ccc(CSCC)cc2)=O)C2(CC2)C1 Cc1ccc(S(=O)(=O)NCc2ncc(CSc3ccccc3)o2)c(C#N)c1 C1(C(N2CCC(C(=O)Nc3cccc(OCC)c3)CC2)=O)CCS(=O)(=O)C(C)C1 N1(C(C2CC(C(=O)OC)C2)=O)CCCC(NC(=O)Cn2ncn(C)c2=O)C1 Cc1cccc2c(=NCCC(C(F)(F)F)Nc3ccccc3)[nH]cnc12 Cc1cccnc1-n1cc(-c2ncccc2C)nn1 C1(CC)CCN(CCNC(c2cn(Cc3csnc3NC)nn2)=O)CC1 N1(C(CC(C)(C)O)=O)CCC2(CCC2)C(NC(C2CCC(=O)NC2)=O)C1 N1(C(=O)Nc2nc(-c3ccc(F)cn3)cs2)CC2CCC(C1)O2 c1(C(N(CC(CN(C(C(CC)F)=O)C)O)C)=O)cc(OC)ccc1F c1(CNC(Cc2cc(C)ns2)=O)cccc(CNC(C2CCS(=O)(=O)N2)=O)c1 c1(C(=O)NC2CN(C(c3c(CC)n(C)nc3)=O)C2)cc(OC)c2c(c1)CC(C)O2 c1(C(=O)NC2C(CNC(CSC)=O)C2)cccnc1C1CC1 C1(C(C(=O)NCC(CC)CO)(C)C)CCCN(C(c2cscc2C)=O)C1 N1(CC(=O)NCCC(=C)CNC(=O)C(C)C(=O)OC)CCc2sccc2C1 C1(C(=O)NCC(COC)(C)CO)CCOCCN1C(=O)Cn1ncnn1 c1(CC(N2C(CCNC(=O)Cc3ccsc3)CCC2)=O)ccccc1O.C(C=C)=CC C(c1ccncc1)=C(C(=O)N(CCN(C(C1(OC)CCOC1)=O)C)C(C)C)C CCCC(C)(O)CC(=O)NC(CC(=O)NCCc1cnc(C)cn1)C1CC1 c1(C(=O)NCC2N(C(C(CC=C)C)=O)CCCC2)c[nH]c2cccc(F)c12 C1(C)(CNC(c2c(C)nn(C)c2)=O)CCC(NC(C2CC2c2cnc[nH]2)=O)CC1 C1(NC(Cc2c(CC)con2)=O)CCS(=O)(=O)C12CN(C(=O)CCC(=O)OC)C2 c1(N2CC(C)C(C)C2)nc(N2CCC3(CCCC3)CC2)nc2c1CSC2 c1(C(CC(=O)O)NC(c2ncc(C(C)=O)s2)=O)ccc(Br)c(C)c1 C12(CNC(CC=C=C)=O)COCCN1C(=O)CN(C(c1cccc(Cl)c1F)=O)C2 N1(C(C2(C)CC=CCC2)=O)CCCC(C(=O)N(C2CC2)C2CC2)CC1 C(=O)(CC(C)(C)F)NCC1C(NC(c2cc(OC)ns2)=O)CCC1 C1(NC(c2csc(Br)c2)=O)CCN(Cc2cc(Br)c[nH]2)CC1F C(=O)(C1CCCc2nc(C)[nH]c21)NC1(C)CN(C(c2cc(C)nn2C2CC2)=O)C1 O=C(CCC1=CCCCC1)NCC1COCC1NC(C1CCCN1C1CC1)=O C1(CNC(N2CCC(n3cc(C(N)=O)nn3)CC2)=O)COC2COCC12 c1(OC)cc(F)cc2[nH]c(NC(N3CC4CN(C5CCC5)CC4C3)=O)cc12 c1(CC(=O)N(CC(CN(C(Cc2nnc(C)o2)=O)C)O)C)ccc(C)c(C)c1 C1(C(N2CCCN(C(c3ccc(C)nc3C)=O)CC2)=O)CC2CSCC(C1)C2 C(=O)(C(O)CC(C)(C)C)NCC(CC=C)NC(=O)CC1CCC2(CC1)CC2 N1(C(c2c(C)nsc2)=O)CC2(C)CN(c3nc4cc(F)ccc4o3)CC2(C)C1 N1(CCCC)CCC(N=c2[nH]c(CCN3CCCC3)nc3c2CCC3)C(F)C1 c1(OC)ccc(CCC(N2CC(C(F)(F)F)C(CNC(=O)CC3CC3)C2)=O)cc1 C(C(C)C(=O)NC1COCC1NC(c1c[nH]nc1C(C)C)=O)OC(C)=O c1(OC)ccc(C(=O)NCC2CN(C(=O)C=CSC)CC2C(F)(F)F)c(C)c1 C12(CNC(COCC)=O)CC1CN(C(C1CCCC1(C)OC)=O)C2 N1(C(CCOC(CC(C)C)C)=O)CC(NC(=O)C=Cc2cc[nH]c2)C2(CCC2)C1 N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)C(C)(COC)COC)CC1C N1(C(c2nc(C)c(C)[nH]2)C)CCC(O)(Cc2cn(C3COCC3O)nn2)CC1 CC1CCCN(C(=O)C=Cc2cnn(C)c2)C1CNC(=O)CCCC#N C(=O)(C(O)CCC(C)C)NC(C(=O)NC(CC=C)CO)CN=[N+]=[N-] C(C(C)(C(=O)NCC1CC(O)CN1C(=O)CC=C(Cl)Cl)OC)OC c1(N2CCC(C=C)CC2)[nH]c(=NCc2c[nH]nc2C2CCCCC2)nc2scnc12 n1(C(N2CC(CC)N(C(=O)CCn3cncn3)CC2)=O)ccc2c(C)cccc12 c1(NC(N(CC(O)C2CC2)C)=O)ccc(N2CCOCC2)nc1C C(=O)(CCCCCCCC1CC1)Nc1cn(CCN(CCCN(C)C2CC2)C)nn1 C1(C2CCN(C(=O)Cn3ccnn3)C2)(NC(C(C)C(C)(F)F)=O)CC1 C1(C(=O)NCC2N(C(CC(n3c(C)cc(C)n3)C)=O)CC2)CCCC1S(C)(=O)=O c1(CC)nn(C)c(CC)c1C(=O)NCC1CCCN1C(=O)CN(C)C(C)C C1(NC(CCOC(C)C)=O)COCC1CNC(=O)CN(C1CCC1)C C1(C(=O)NCc2c(COC)noc2)CN(C(=O)CC(C)(F)F)CC12CC2 C(=O)(C(C)CC(F)F)NCC(CCC)NC(C1(C)CC2(CC2)C1)=O c1(N2CC(NC(CCC(C)SC)=O)(CO)C2)ccnc2ncnn12 CCCCCCCC(=O)NCC1(F)CN(C(=O)CC2CC(F)(F)C2(F)F)C1 CCC(CC(=O)NC1(C)CCN(C(=O)CCn2ccnc2C)C1)C(C)(C)C N1(Cc2ccc(C)o2)CC2CCN(S(=O)(=O)c3ccc(O)cc3)CC2C1 c1(SC)ccc(O)c(C(=O)NCC(CC)N(C)C(c2cccc(C)c2F)=O)c1 Cc1ccc(OCC(N2CCN(C(=O)CC3CC3)C3CC23)=O)c(Br)c1 C1(CC)C(N)CCCN1Cc1ccc(N2CCCC2)o1 CC1CN(C(C2CC(=O)NC(=O)N2)=O)CCCN1C(=O)Cn1cccn1 Cc1n[nH]c(C)c1CCC(=O)NCC1CCCN1C(C1CC1c1cccnc1)=O c1(C(=O)NC2C(NC(COCC(C)(C)C)=O)C2)ccc(OC(F)(F)F)cc1 c1(CNC(=O)NC2CC(CO)C3CC23)nccc(Cl)c1O C(=O)(CS(=O)(=O)C(C)(C)C)NCC1(O)CCN(C(c2ccc(COC)[nH]2)=O)CC1 C1(CC(N2C(C)CC(CNC(C3(C)C(C)CCC3)=O)C2)=O)CN2CCC1CC2 Cc1c(C(=O)NC2CN(C(C3COCC3(C)C)=O)CC2O)cnc2ccccc12 CCC(CNC(=O)CCCCCF)CC(=O)NC(C)CCC(C)(C)C CCCC(C(F)(F)F)NC(C1CCC(C2CC2)N1C(=O)C=CC(=O)OCC)=O Cc1n[nH]c(C)c1C(C)CC(=O)NCC(F)CNC(=O)COCc1ccco1 Cc1ccc(C(=O)NCCC2CN(C(=O)CCCC(C)(F)F)C2)c(N)c1C C12(C(=O)NCC(C)CNC(=O)C(c3ccc(Cl)s3)C)CC3CC1C2C3 Cc1ccc(CC(N2CCN(C)CC2CNC(=O)COCC(F)F)=O)c(F)c1F C(=O)(C(CCSC)N1CCC(F)(c2ccccc2)C1)NCCSC N1(C(C=C(C)Cl)=O)CC2CCC(C1)N(C(c1cncc(F)c1C(F)(F)F)=O)C2 C#CCCCCCCC(=O)N(CC(N1CCC2(CC1)CC2C#N)=O)CC#C C1(NC(COC2CCCC(C)C2)=O)CN(C(=O)CS(N)(=O)=O)C(C)(C)C1 C12CCCN(C1)C(=O)C1N(CC1)C2=O.C(CCCN(C)C)N(CCO)CC CC1(C)CC(CCNC(=O)CN(C(=O)Cc2cccn2C)C(C)(C)C)CO1 c1(C(N2CC(CC)N(C(=O)CCCCCSC)CC2)=O)ncnc2c(C)csc12 CC12CC(NC(C3CC4CCC(C3F)N4C(=O)COC(F)F)=O)(C1)C1(CCC1)O2 c1(C)cn2cccnc2n1.Cn1cnnc1Cn1cc(-c2cnc(C(=O)N)s2)nn1 N1(C(C(COC)(C)O)=O)CC2CC(NC(c3ccc(OC)nc3Cl)=O)CC2C1 N12CCOC(C13CCC3)CNC2=O.C1(C(N)=O)CCCC(C(N)=O)CC1 c1(C(C)C(=O)NCCOCCNC(C2CC2C(F)F)=O)ccc(Br)s1 c1(C(N2C(C)CC(CNC(c3ncc(C)nc3)=O)C2)=O)cc(N)cc(N)c1 C=CCC(CNC(=O)C(c1ccccc1)OC)NC(=O)C(C)(C)C c1(CNC(C(C)OC(C)=O)=O)ccc(C(N2CCC2(C)C(C)C)=O)s1 c1(OC)cnc(C(N2CCCCC2C(C)NC(c2cc(C#N)cs2)=O)=O)nc1 N1(C(c2cncc(Br)c2)C(=O)NCCCSC)CCn2[nH]c(=N)nc2C1 C1(C)(CC)C=C(C(=O)NC2COCC2NC(c2ccc(F)cc2)=O)C1 C1(C(=O)NCC(CC=C)NC(=O)C=C2CCCC2)CCN(c2nncs2)CC1 C(CCC(C)C(=O)NC1CCCC(NC(=O)CCCNS(C)(=O)=O)C1)OC CCC(COC(c1cnn(-c2ccc(C)cc2C)n1)=O)CC(F)F C1(C(N2CC(NC(C(C3CCCC3)OC)=O)C(SC)C2)=O)CS(=O)(=O)CC(=O)N1 S1(=O)(=O)c2ccc(nc2)NCC(C)N1CC.C1(C(=O)NC)CCC(C)CC1 Cc1cc(C(=O)NCC2CC3CC3N2C(=O)CC2(OC(C)C)CC2)n(C)n1 C1(C(=O)NCCCCCCO)(CNC(c2c(CC)ncs2)=O)CC2(CC2)C1 Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(c2sccc2C(F)F)=O)cc(O)n1 C1(C(=O)NCC(C)(CNC(=O)C2=C(C)CC2)OC)CC(C)(C)C(C)(C)C1 Cc1cc(NC(C23CC2CN(Cc2ncccc2F)C3)=O)cc(Br)c1 c1(C(=O)NCC2CC(C)N(C(=O)CCc3cn[nH]c3)C2)csc(N=S(C)(C)=O)n1 c1(-c2nc3nn2CC2(CC2)C3)n[nH]c2ccccc12.N1(OC)CC2C(C1)C2(F)F CP(C)(=O)c1cnc(C(=O)Nc2cc(Br)cc3c2OCCC3=O)nc1 C(C(C)N=c1cccc(S(=O)(=O)NCC(c2ccccc2)(C)C)[nH]1)N(C(C)C)C N1(C(CC(C=C)C)=O)CC2(C1)SCCC2NC(c1cc(C)cnc1OC)=O N1(C(C(C)Oc2ccccc2)=O)CC2CCCC(CNC(=O)CSC(F)F)(C2)C1 N1(C(C2CC(OCC)C2)C(=O)NCCCC2CC2)Cc2ncsc2C1 C1(NC(C2(C)CS(=O)(=O)C2)=O)CCC2(CCCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 C#Cc1cncc(NC(=O)C(CCF)NC(=O)Cc2cn(C)cn2)c1 c1(C(N2CC(C(C)NC(=O)Cn3cnnn3)C2)=O)cccn2c(O)nnc12 CC(C)C(F)C(=O)NCCCC1CCN(C(c2cnn(C(C)(C)C)c2)=O)CC1 c1(C(N(C(C)C(=O)NC(C)CCSC)CCC)=O)nccnc1C C1(NC(C(c2cn(C)nc2)(F)F)=O)CCN(C(=O)C2=CCSC2)C1CC1CC1 C(=O)(CC(O)CC(C)(C)C)N(CCCNC(=O)Cc1cc(C)on1)CCOC C1(NC(c2n(C)ncc2)=O)CCC2CN(c3ccnc(C4CC4)n3)CC2C1 C1(CNC(c2scc(OC)c2)=O)CCCCN(C(=O)Cc2cc(C)cc(F)c2)C1 c1(CC(=O)NCCC2N(C(CC(CC)SC)=O)CCC2)ccc(C2CC2)cc1F c1(C(=O)NC2CCN(C(C(CC)C#N)=O)C2(C)C)cc2c(Cl)ccc(Cl)c2[nH]1 C1(CNC(=O)CCc2ccncn2)COCCN1C(=O)Cc1cnccn1 C(=O)(C1Cc2ccccc21)N(C1CCN(C(c2c[nH]nc2S(N)(=O)=O)=O)C1)C C(=O)(CCC(F)(F)F)NCCC1(C)CCN(C(c2c(C(C)C)ncnc2)=O)C1 C1(NC(CCSC)=O)COC2(C1)CN(C(=O)C(C(F)(F)F)=Cc1ccccc1)C2 N1(C(Cc2ccc(C)o2)=O)CCC(C)N(C(c2n[nH]c3c2COCC3)=O)CC1 c1(C(=O)NCC2(NC(C(C3CCC3)OC)=O)CCC2)ccc(Cl)cc1 Cc1nc2ncc(C(=O)N(C(C)CNC(=O)C(C)Cc3ccccn3)C)cc2o1 c1(C(N2CCC(NC(C3(C)CC3)=O)CC(F)C2)=O)ccc2[nH]nc(Cl)c2c1 N(C(=NCCC1COC(C)(C)OC1)NCC1CC1)CC1C(C(=C)C)CNC1 C1(NC(Cc2ncc(CC)[nH]2)=O)CCCCC1CNC(=O)Cc1cccc(F)c1 c1(NC(N2CCC2C2CCOC2)=O)ccc(F)c(F)c1 C1(C(C(=O)NC2(C(C)NC(c3occc3C3CC3)=O)CCC2)C)CCOCC1 c1(N2CCC3(C(C(=O)NCC4(F)CCC4)C3)CC2)ncc2ccccc2n1 N1(C(c2c(C)n[nH]c2C)=O)CCCC(C(=O)NCc2cccc(Cl)c2)CC1 C1(C2(C=O)CC2)CCCN1C(=O)CC1CCC(C(F)(F)F)O1.N(CCO)(CC)CC c1(C(=O)NCC2N(C(CNC(=O)NC)=O)CC=C2)snc(O)c1Cl C1(OCCNC(CCCOCC)=O)(CNC(=O)Cn2ncnn2)CCOCC1 CN=c1[nH]nc(CC(=O)NC2CC2NC(c2ccc(SC)cc2)=O)s1 C1(O)(CNC(c2c(C)cco2)=O)CCCN(C(C2CCCN(C)C2)=O)C1 C(=O)(C(F)CC(C)C)NC1CCC(NC(c2ocnc2COCCOC)=O)CC1 N1(C(=O)OC(C)(C)C)CCC2(CCOC2)C1.C12COCC1SC2 N1(C(CCC2(C#N)CCC2)=O)CC2CCC2(C(=O)NC2CC(CF)C2)C1 c1(C(=O)NC2(C3CN(C(C4C(C(C)C)C4)=O)C3)CC2)ncccc1N=[N+]=[N-] C1(C(N2C(C(C)Nc3ncccn3)CCC2)=O)CN(C(=O)CC(C)(C)O)CC1C C1(CCNC(C(C)S(N)(=O)=O)=O)CCN(C(=O)Cc2ccn(C)n2)CC1(F)F c1(C(N2CCC(C)(CNC(c3cc(F)c[nH]3)=O)C2)=O)ccc(O)c2c1CCCC2 c1(C(N(C2CCCN(C(CC)=O)C2)C)=O)cccn2c(O)nnc12 C1(C(=O)NCC2(OC)CN(C(C3CC(C)(C)CN3C)=O)C2)CCS(=O)(=O)C(C)C1 C1(C(N2CCCC2(C)CO)=O)(NC(CC(=O)OCC)=O)CC(F)(F)C1 Cc1nc(N2CCOCC2)sc1CC(=O)NC1(CC(F)F)CC1 c1(C(N2CCC(N(C)C(C3CC3C(F)F)=O)CC2)=O)ccn2ccccc12 c1(C(N(C2CCN(C(c3cc(CCC)n(C)n3)=O)C2)C)=O)[nH]cc2c1CCCC2 c1(CC)cc2c(NCC3CCCC3NC(C3(O)CC(C)(C)C3)=O)nc(C)nc2s1 Cc1ccc(F)cc1C(=O)NC(c1nocc1C(=O)NC1CCCCCCC1)C CCCCCCCCCc1nc(CC(N2CCCC(F)(F)CC2)=O)no1 N1(C(CCCn2cc(-c3ccn(CC)n3)nn2)=O)CCC(CO)C1(C)C S(=O)(=O)(c1cc(C#N)ccc1F)NC(CNC1CN(C(=O)OC)C(C(C)C)C1)=O C1(C(=O)NC2C(CNC(C=CCC)=O)CC2)CCOC1(C)C Cc1nc(O)nc(S)c1C(N1CCCC1(C)CNC(=O)Cn1cccc1)=O C1(C(=O)NCC2N(C(CC3CCC(C)NC3=O)=O)CCC2)CC2C=CC1C21CC1 n1(COC)ncc(C)c1C(C(=O)NCC1CCOC1)N(C)Cc1cccc(C)c1 C(=O)(C1=C(Cl)CCC1)NCC1N(C(C2(C#C)CCCC2)=O)CCC1 CCCCC(C)C(=O)NCC(CNC(c1ccc(Br)cc1Cl)=O)CO C12(C(=O)NCC(CNC(C(C(C)C)n3cccc3)=O)C)CC(C)(C1)OC21CCC1 CC1(C)COCC1C(=O)NCc1ccc(C(=O)NCCCCS(C)=O)cc1 c1(N(C(=O)NC(C2CCSCC2)C(=O)OC)Cc2cnn(C)c2)cc(O)ccc1F C1(NC(c2nc(CNC(CCC=CC)=O)oc2C)=O)CCn2cnnc2C1 Cc1cc(F)ccc1S(=O)(=O)C(=O)NCC(C1OCCCO1)(C)C c1(C(=O)NCC(C)NC(C=C(C)c2ccsc2)=O)cc2c(ccn2C)[nH]1 N1(C(CSCC=C)=O)CC2CC2(CNC(C2CC(CC)C2)=O)C1 N1(C(CC#C)=O)CC2CCC2(CCNC(c2ccsc2Cl)=O)C1 C(=O)(C(CO)C(F)(F)F)N(C)CC1CCN(C(c2cncnc2C2CC2)=O)C1 C1(CC(=O)NCC2(CNC(CCc3ccn(C)n3)=O)CCC2)CCOC(C)(C)C1 C1(N(C(C2C(C)C2)=O)C)CCN(C(=O)COCc2nc(C3CC3)no2)C1 c1(C(N(CCC(=O)NCCN(OC)C)C2CC2)=O)cccc(Cl)c1 CCCCC(C)(F)C(=O)N1CC(CCNC(C2CC23CCCC3)=O)(OC)C1 Nc1cc2c(cc1C(=O)NCCCCCNC(=O)CCc1cncnc1)OCO2 N1(C(C2(CC)CCN(C(C3CCN(C)CC3)=O)C2)=O)CCOC2COCC12 C(=O)(C(C)(C)C(=O)N1CCC(CC(=O)NCC2CC3(CC3)C2)C1)OCC c1(C(=O)NCC(CNC(=O)CCC2OCCO2)OC)cccc(C(F)(F)F)c1O N1(C(=O)NC(c2scc(C(=O)OC)n2)C)CCOC(c2cccc(O)c2)C1 N1(C(C(C)(C)OC(C)C)=O)CCCC(CCC(=O)NCC(C)CC2CCC2)C1 C1(NC(CCCNC(=O)C=CC2CCOC2)=O)CCn2ncnc2C1 C(CNC(=O)CCc1nccs1)(C(C)C(C)C)NC(c1ccn(COC)n1)=O Cc1nc(CC(=O)N(CCC(C)NC(C2CCCO2)=O)C)c(Cl)s1 c1(CC)ccnc(C(=O)NC2CC2CNC(C2(C(C)(C)C)CCCCC2)=O)c1 c1(C(=O)NCC(CCC)NC(c2c(C)n[nH]c2C)=O)cc2ccnc(Cl)c2[nH]1 c1(CC(N2CC(C(C)NC(=O)CC3CCC4CC34)C2)=O)c[nH]c2ncccc12 C1(C(=O)NCCC2(O)CCN(C(c3cccnc3O)=O)C2)CN2CCCN1CC2 S(=O)(=O)(c1c(OC)cccc1F)NC1CC(C(N(CCOC)C)=O)C1 CC1CCN(C(c2ccon2)=O)CC1NC(=O)Cn1cc(Br)ccc1=O CCCCCCC(=O)NC(c1ccnn1C)C(N1CC([N+](=O)[O-])C1)=O N1(C(C2C(OCC)CC2)=O)CC2(CCN(C(c3cnc(O)n(C)c3=O)=O)C2)C1 c1(-c2ccc(NCC3CCC(CCCC)O3)s2)ccc2c(OC)cc(=O)oc2c1 C1C(C(=O)OC)NC(=O)N1C1CC1.c1(CCC(=O)NCCCOCC)scnc1C C1(C(=O)NC(c2ccccc2)COCC)CC2CC2N1C(=O)CSC C(=O)(CC1=CCCC1)NC1CCC(NC(C(CC)(O)c2cccc(Cl)c2)=O)CC1 C(=O)(C#CC1(C)COC1)N1CCCC(C)(C(N2CC(C(CC)C)C2)=O)C1 C1(C(C)C)Cc2cc(F)ccc2N(C(c2cc(Cl)ccc2C(F)F)=O)C1 c1(C(N(c2nc(OC)c(C)cn2)C2CNCC2F)=O)cc(F)cc(F)c1OC N1(C(CCOC)=O)CC(CNC(c2cncnc2)=O)(OC)C1 c1(C(=O)NCCC2(C(N(C3CC(OC)C3)C)=O)CC2)cccnc1 C(c1sc(Cl)nc1Cl)=CC(=O)NCC1C2CN(C(C3CN(C(N)=O)C3)=O)CC21 c1(C(N(CCCCNC(=O)C(F)CC2CC2)C)=O)cnc(O)cc1C(F)(F)F c1(OC)cc(O)ccc1NC(c1oc(CNC(=O)C2=CCCC2C)cc1C)=O C(=O)(C1=Cc2ccccc2C1)NC1CC(C(=O)NC2CN(c3ccncc3)C2)C1 Cc1c(C(=O)NC2CCN(C(C3CCC(C)CC3)=O)C2)cnn1CCN(C)C C1(CCNC(c2ncn(C(C)C)c2)=O)COCCN1C(C1CC(C(C)(C)C)C1)=O C12(NC(C3C(C)C3C)=O)CCC1CN(C(=O)CCc1cc(Br)ccc1F)C2 CC1CN(C(=O)CC2CN(Cc3cccc(-n4cncn4)c3)CCO2)CC(=O)N1 C(=O)(C(CC=C(Cl)Cl)c1ccccc1)NC1(C)CCC(O)CC1 C(C)(CC(=O)N1CCC(CC(=O)NCc2ncc(CO)o2)C1)OC C1(C(N2C(CN(C(c3c(C)occ3)=O)C3CC3)CCC2)=O)CCC12CCC2 C(CCCC(=O)N(C1CCN(C(c2cnccc2Br)=O)C1)C)OCC C12(CNC(Cc3cc(COC)on3)=O)CC1CN(C(=O)CCNC(C)=O)C2 c1(C(N2C(CN(C(C(CCC)(C)O)=O)C)CCCC2)=O)ccc([N+](=O)[O-])cc1F n1(CC=C)nnnc1C(CCOC)(C(C)CC)NCc1noc(C2CC2)n1 CCCC(CNC(=O)C(CC)CCOC)C(=O)N1CCC(NC(N)=O)CC1 C(=O)(CCn1cccn1)NCC(C1CCC1)N(C(=O)CNC(c1cc[nH]n1)=O)C c1(NC(c2cncc(NCc3nc(C)c(Br)cc3)c2)=O)cccnc1[N+](=O)[O-] C1(NC(Cc2c(CC)cc(F)cc2)=O)CN(C(=O)C=C2CC2)C2(CCC2)C1 N1(C(CCCNC(=O)OC)=O)CC2CC2(C(N2CCCC2CNC(C)=O)=O)C1 Cc1nn(C)cc1C(=O)NC(c1cn(CC(F)(F)F)nn1)C(=O)NCC1(C)CC1 c1(CC)ncncc1C(=O)NCC12CC1CN(C(=O)C(=Cc1cccs1)C)C2 C(=O)(CCCC(N)=O)NC1(C)CCN(C(Cc2c(C)cco2)=O)C1 C(=O)(C(C(=O)N1CC(CCCCNC(=O)C(F)C(C)C)C1)OC)OCC CC1(NC(C2CC(O)CN2C(=O)COC2CN(C(N)=O)C2)=O)CCC(O)CC1 CCCC(CC)CC(=O)NCCC(F)Cn1cc(-c2ccc(F)cn2)nn1 c1(C(=O)NC2CC(CNC(CC(=C)C)=O)C2(C)C)ccc2cc(O)ccc2n1 N1(C(c2c(CC)ocn2)=O)CCC(F)C(NC(C2(C)CCN(C)CC2)=O)C1 C1(CC=C)(NC(=O)C=Cc2cc[nH]n2)CCCN(C(C2CCC3CC2CO3)=O)C1 N1(C(C2CCCO2)=O)CCCC2CN(Cc3nnc(-c4ccccc4F)s3)CC12 C=CC1CN(C(=O)C(c2cncn2C)O)CC1NC(=O)CN1CCCCC1=O N1(C(c2c(C)nc(C)o2)=O)CCCC(C)(CNC(=O)C(c2ccccc2)F)C1 C1(N(C(=O)CN2CC3CC3C2)C)CN(C(c2cc(C(F)(F)F)nn2C)=O)CC1F CC(C(=O)NCCCCn1cc(COC(F)(F)F)nn1)C(=O)N1CCOCC1 c1(NC(C)=O)ccccc1CC(=O)NC1CC1NC(C1C(C)(C)C1(C)C)=O CCC(C)C(C(=O)N1CC(OC(F)F)C1)NC(=O)Cc1cnsc1 c1(C(=O)N(C2CC2)CC2CCC3CC23)ncccc1NC(=O)CC(C1CC1)C1CC1 c1(COC)cnc(OC)c(C(=O)NC2COCC2NC(C2C=CCCC2)=O)c1 c1(C(C2CCN(C(C=COCC)=O)C2)=O)ccc(O)c(O)c1O CC(C)(C(=O)NC(C1CC2(C1)CC(O)C2)=O)C(=O)N1CCOCC1 C12(C(=O)OC)CC(CC(=O)OCC3CC(O)C3)(C1)C2.C1(C=O)(CO)CCOC1 N1(C(CONC(c2c(C)ocn2)=O)=O)CC=CC1(C)CO CC(c1cccc(Cl)c1)=CC(=O)NC1CN(C(C2CCN(C)C2=O)=O)CC1(C)C C1(NC(c2c(SC)ccs2)=O)CCC2CC1CN2C(=O)CC1(O)CCCOC1 C=CCC(CC=C)C(=O)NC1CCN(C(C2CCOCC2)=O)C12CCC2 C(N=c1nc2ncn(C)c2c(NCCC(C)O)[nH]1)c1cccc(C)c1F C1(C(=O)NC2CC23CC(O)C3)(COC)CCCN1C(=O)C(C)=NOCC#N c1(OC)ccc(C2CSCCN2C(=O)CCCn2cccn2)cc1 C(=O)(CC(C)C(=O)N1CC(C(C)NC(=O)CCc2nc(C3CC3)no2)C1)OCC c1(C(=O)NCC2CC(NC(c3occc3C3CC3)=O)C2)ccc2[nH]nc(O)c2c1 C1(NC(CC(CC)C2CC2)=O)CN(C(c2nnn3c2CSCC3)=O)CC(C)(C)C1 CC1CN(C(c2sccc2Cl)=O)CCC1NC(=O)Cc1cnn(C(F)F)c1 N1(C(C=C(CCC)CCC)=O)CCN(C(c2[nH]ccc2C2CC2)=O)CC12CC2 C1(C)(COC)C=CCN1C(=O)CCC1CCN(C(C2CC=CC(O)C2)=O)C1 CCCCC(C)CCC(=O)NCC1C=CC(NC(c2ccoc2Br)=O)C1 c1(OCCN(C)C)cccc(F)c1.C12COCC1C(=O)NC2 c1(C(=O)NC(C2CCCN(C(c3cscc3C(F)F)=O)C2)C)ccc(=O)n(C)c1 N1(C(C=CCN(CC#C)C)=O)CCC2(CC1)CN(C(=O)C1=CCCC1)CC(C)O2 c1(CNC(C(N2CC(C)SCC2)c2nncn2C)=O)ccc2c(c1)OCCO2 N12CCC(C1)N(CCO)CC(=O)N(CCC)C(C)CC2=O.C(C)(C(=O)NC)OC(C)=O Cn1nnc2cc(C(N3CCCC3(C)CNC(=O)CC3CC4CC4C3)=O)ccc12 c1(C(C)C)ccc(C(N2CCCC(NC(=O)CCC(C)CN(C)C)C2C)=O)c(O)n1 N1(C(C(CN(C)CC)F)=O)CC(Cn2cc(CCC3CCOC3)nn2)CC1CO c1(C(=O)NC2CC(CCNC(CC3CC(=C)C3)=O)C2)conc1C(F)(F)F c1(C(=O)NCCC(C)(C)CNC(C2CCOC2)=O)ccc2ncnn2c1 CC1(CCC(=O)NCC(=O)NCC(=O)NC(N)=O)CN(C(=O)CO)C1 C1(C(=O)NC(c2ccccc2)CNC(C(C)NC(CC)(C)C)=O)CC(C2CC2)C1 C#Cc1cc(C(=O)NC2CCC(C)N(C(=O)C=Cc3nnn(C)n3)C2)ccc1Cl CCC(CC(=O)NCC1(C)CN(C(c2ccc(C)cn2)=O)CCO1)C(F)F C1(C(N(CC(=O)NC(c2cncnc2)C)CC)=O)CCCC(C#N)C1 CC(C)CC(CNC(c1cn[nH]c1)=O)C(=O)NCC1(F)CCOCC1 CC(C(=O)OCC(C)(C)C)C(=O)NNc1nc(Cl)c(C#N)[nH]1 c1(C(=O)NC(CCCC)CNC(=O)CC)[nH]cc2c1CCC2 C(=O)(C(C)(CCC)CCC)N1CCC(N(C(CCC)=O)C)C(C)C1 N1(C(CCC(C)(C)C)=O)CC2CCCN(C(C3CC4C=CCC(C3)C4)=O)C2C1 c1(OC)cccc2c1CN(C(c1cnn(C)c1Cl)C(=O)NC1CCCCC1)C2 C1(CNCC2CC(C(F)F)OC2)CC12CCCCC2 C(c1cnn(C)c1)=C(C(=O)NC1CCC(CNC(c2c(CCC)[nH]cc2)=O)C1)C c1(CCC(C)N(CC(C)C#N)C(=O)NCC(=O)OCC)nc(C)cs1 C(CC1=CCN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC1)NC(C1(C)ON=C(C)C1)=O c1(C(N2CC(C)(C(=O)Nc3c(C)cc(Br)cc3F)C2)=O)cccc2c1cnn2C C1(C(=O)NC2CC(O)(CNC(c3cc(C)[nH]c3C)=O)C2)CCCCC1(C)C C1(CC)CN(C(c2ccccn2)=O)CCC1NC(c1ccc(OC)s1)=O C=C(F)CN=C(NCc1ccnn1C)NC1CCC(F)(F)CC1 NS(=O)(=O)c1c[nH]c(C(=O)OC2CCCC2C#N)c1 c1(N2CCC(C(C)NC(=O)NCC3(C=C)CCC3)C2)ccccc1C c1(OC)ccc(C(=O)N(C2CCCC(NC(=O)CC3CCSCC3)C2)C)c(C)c1 C(C(C)(C)CC(=O)NCC#CC(=O)NCC1CCC2(CC2)CO1)OC C(=O)(C1CCc2c[nH]nc21)NC(CCNC(C(=Cc1ccccc1)CC)=O)C C1(NC(C=C(CNC(CN2CCC(OC)C2)=O)C)=O)CCC(F)(F)CC1 N1(C(c2c(NC(C(C)OCC)=O)cccc2F)=O)CCC2(C(=O)O)CCCC12 CC1CC(NC(=O)C(F)=CC2CC2)CN1C(C12CC(c3ccccc3)(C1)C2)=O C(=O)(N=c1cc(C)n(CCO)[nH]1)C1CCN(C(COC)=O)C1.c1(N)cc(C2CC2)[nH]n1 N1(C(Cc2n(C)nnc2)=O)CC2CCC2(CC(=O)NC2(CC(N)=O)CC2)C1 CC(C(=O)N(C)CCN(C)C(C1CC(N2CCCC2)C1)=O)c1ncco1 c1(C(=O)NCC2(F)CN(C(CCCCNC(N)=O)=O)C2)cc2cc[nH]c2cn1 c1(NC(C)=O)cccc(C(=O)NC(C2CCCCN2C(=O)C(C)C)C)c1 N1(C(C2N(C(C)C)CCC2)=O)CCC2C(C1)CN2C(=O)COc1cnc(Cl)cn1 C(=O)(C1CCc2ccccc21)NCCC1(NC(Cc2cc(C)sc2)=O)CCC1 c1(C(CC(=O)NC2CC(C)(NC(CC(C)SC)=O)C2)C)c[nH]c2ccccc12 c1(C(N(C2CN(C(c3c(CC)n[nH]c3)=O)CC2F)C)=O)cc2cccnc2cn1 C(CCC(O)C(=O)NCC(C)(C)CC(F)F)NC(C(C)c1cccs1)=O c1(C(=O)OCC2CC(C)CC(C)C2)c(F)cc(F)cc1Br Nc1ccc(=NCCOc2cnc3ccccc3c2)[nH]c1 N1(C(Cc2c(C)n(C)cn2)=O)CCCC(C)C1CNC(=O)CCN1CCCC1 c1(C(N(CC(CC)NC(C(C(CC)C)O)=O)C)=O)c(F)cc(C)cc1Br c1(C(=O)OC)cc(C(N2CCC2CNC(C23CCCC2C3(F)F)=O)=O)cc(C)c1 C1(CC)CCCCN1C(C1C(C)CN1C(=O)C=CC(F)F)=O C1(C(=O)NC(CCN(C(CC(C)NC(N)=O)=O)C)(C)C)CCC2CC1C2(C)C c1(C(C(C)C)C(=O)OCc2cnn[nH]2)ccccc1C#N Cc1c(F)ccc(C(N2CC(C3CN(C(C4CC4[N+](=O)[O-])=O)C3)C2)=O)c1C C1(CC=C)(NC(=O)Cn2ccc(C)n2)CCCN(C(c2cnc(O)c(F)c2)=O)C1 CCC(CC(=O)N1CCN(C(c2cc(C)ncn2)=O)C(CS(C)(=O)=O)C1)C(C)C C(=O)(CCCCCCNC(c1cccc(-c2cc(OC)ccn2)c1)=O)OCCC CCC(O)CC(=O)NCc1csc(C(N2CC=CC2)=O)c1 CCC(CNC(=O)CC(C(C)C)NC(=O)CC(C)CCO)(CC)CO C1(C(=O)Nc2ccc(NC(C(CC(C)C)O)=O)cc2)CCn2cnnc2C1 C1(C(N2CC(C)=C(C)CC2)=O)CCN(C(C2(C)CCCOC2)=O)CC1(C)C C=CCC(C(=O)NCCN(C(=O)C(CC)SC)CC(C)O)c1ccccc1 N1(C(C(CC(C)C)C)=O)CCCC(C2(NC(c3ccc(F)cc3)=O)CC2)C1 c1(CCC)c(C(=O)NC23CC2CN(C(c2[nH]c(=N)sc2CC)=O)C3)cnn1CCO c1(CC(F)(F)F)nc(CS(=O)(=O)Cc2ccccc2)n(-c2ccccc2)n1 C(C(CC(=O)N(C)Cc1cn[nH]c1)NC(=O)CN1CCCC1C)OC CC1CCCn2cc(C(=O)NCC3CC(NC(=O)CCCCCF)C3)nc21 C1(F)(C(N(CC(C)NC(=O)C(c2ccc(Cl)cc2)(C)O)C)=O)C(C)(C)C1(C)C C(CCC)(C(=O)NC1(CNC(=O)CC(C)c2cnn(C)c2)CC1)=CCC N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3COCCO3)=O)CC2)C1 c1(C(=O)NC2CCN(C(CSCCCC)=O)C(C)C2)cccc2cccnc12 Cc1nc(C(=O)N(CCC#N)CC2CCCC2(C)C)nn1-c1nc[nH]n1 C1(C(=O)NC23CC(C)(C2)C3)(CC)CCCN(C(=O)CC2CCCOC2)C1 C(CN=C(NCC(C)C#N)NCc1cncnc1)c1ccc(OC(C)C)cc1 C(=O)(CCCCCc1cccc(OC)c1)NCC(CCNC(CCCC)=O)OC c1(C(=O)NC(CC)(C)CNC(C2CCCCO2)=O)cc2c(cc1C)OCO2 C(C)(C)(CCC(=O)NCCN(CC(F)F)C)OC.c12cc(C)c(o1)c(=O)[nH]2 C(=O)(CC(F)(F)C(F)F)N(CCCNC(=O)CCC(F)(F)F)CC c1(OC)cccc(C(=O)N(CC(C)C(=O)N(C)C(c2nc(C)no2)C)C)c1 C(=O)(C1=CC2(CCN(C(C(=O)NCC(C)CC(F)(F)F)C(C)C)C2)C1)OC c1(CCC(=O)NC2CN(C(CSCC#C)=O)CC(O)C2)c(C)nc(SC)nc1O C1(SCCC(=O)NC2(O)COC2)CCCN(C(=O)C=CCn2cncn2)C1 c1(CN(CCN(C(CC2ON=C(CC)C2)=O)C)C)ccnc2ccccc12 CCC(CC(=O)N1CCC(C(=O)NCC(F)C(C)(C)O)(CC)C1)CC(C)C c1(N(C(c2nc(CCCC)sc2)C(=O)NCCSC)C)cccc(Cl)c1 N1(C(C2(C#C)CN(C(=O)C(O)CCSC)C2)=O)CCC(CO)C(O)C1 Cc1sc(Cl)cc1C(C(=O)NCCCOCC1CC1)N(CC(C)C#N)C c1(CC)ccc(O)c(C(=O)N(C)CC2CCCN(C(=O)C(=O)NCC(F)F)C2)c1 c1(C(=O)OC)cc(-c2cncc(-c3nccn3CCCCCO)c2)ccc1O c1(C(=O)NC2(CC(=O)Nc3ccc(Cl)nc3Cl)CCC2)ccc(F)c(Br)c1 C1(OC)CCN(C(=O)CCC(C)(C)C)C(c2cn(C3CCCC3)nn2)C1 C(=O)(CCC(F)(F)C(F)(F)F)NCC1N(C(=O)C(O)CC2CC2)CCN(C)C1 N1(C(c2nnc(C)s2)=O)C2CCC1CC(CNC(C1CCSCC1)=O)C2 C1(CN(C(C(CC)N(C)C)=O)C)CCCN(C(=O)C(CO)N(C)C)C1 C=CCCC(C(=O)NC1CCOC1)NC(=O)CC1(C)CC1 N1(C(CSC(C)C)=O)CC(C)CN(C(c2ccc(F)cc2Cl)=O)C(C)C1 C1(C(N2CC(F)(CNC(c3cc(CCCO)on3)=O)C2)=O)CN2CCC1CC2 C(=O)(CCCCC(C)C)NC1CCN(C(c2ccc(C)cc2Cl)=O)C1C(C)C C1(CC=C)(NC(c2cnc(N(C)C)cn2)=O)CCCN(C(c2cnc[nH]2)=O)C1 CC(C)CC(C)(C)NC(=O)C=CC(C)NC(C1CCCCO1)=O Cc1ccncc1-n1cc(C2CCN(C(C3CCC(C(N)=O)CC3)=O)C2)nn1 C1(NC(C(C2CCN(C(=O)C3=CCCOC3)CC2)C)=O)CC2(CCCO2)C1 Cc1cccc2nc(C(=O)NCC3COC(CNC(=O)C4=NOCC4)C3)cn12 C1(OC)CC(C(=O)N(C)C(c2cnn(C)c2)C)N(C(=O)C(CO)NC(N)=O)C1 C1(O)(C(C(=O)NCc2c(C(C)C)noc2)NC(=O)C(C)OC2CC2)CCCCC1 c1(CN(C(C(C)OCC(F)(F)F)=O)C)ccccc1CNC(=O)CCNC(N)=O C1(CC)(NC(C2C(C(=O)OCC)C2)=O)CCCN(C(=O)CCCN(C)C(C)=O)C1 Cc1cc(C)c(C(N2CCC3CC23C(=O)NCc2nccn2C(C)C)=O)cn1 c1(C(N2C(COC)(CNC(=O)CNS(N)(=O)=O)CCC2)=O)ccc(F)c(O)c1 c1(NC(=O)NC2CC3(C(=O)OC(C)(C)C)C2C3)cc(O)nn1-c1ccccc1 C1(C#CC(=O)N2CCC(CO)C(NC(c3ccc(F)c(Cl)c3)=O)C2)(CC)COC1 c1(C(N2CCCN(C(C=C(COC)C)=O)C(CO)C2)=O)ccc2nc(O)[nH]c2c1 c1(C(=O)NC2CC(CNC(c3cccs3)=O)C2)c(F)c(F)cc(F)c1F N1(C(C(C)NC(c2ccccc2)=O)=O)CC2(CCCO2)C1 N1(C(CC2(C)CCC(=O)C2)=O)CCCC(O)(c2cn(C3CC3)nn2)CC1 Cc1cc(C(N2CCCC2C(=O)Nc2cccc(F)c2O)=O)ccc1F c1(C(N2CCC(O)(C(C)NC(=O)C(O)C3CCC3)CC2)=O)ccn2c1CSCC2 c1(CN(C(=O)NC(C2(n3ccnn3)CC2)C)C)ccncc1Cl C(CC(=O)N1CC(C(=O)NC2(CN(C)C)CCC2)C1)N(C)CCO n1(CC)nc(C)c(C(N2CCOC(C)C2c2nc(C)no2)=O)c1C(F)(F)Cl C1(C#N)(C(=O)NC(CC)CNC(c2cnc(C3CC3)o2)=O)CCOCC1 N(C(=NCCC1(CCO)CCOCC1)NC(C)C1CC1)C1C(C)C1C C1(C(=O)OC)CC(C)N1C(=O)CC1(NC(=O)Cc2cnn(CO)c2)CCC1 C1(=O)CCCCCn2cc(nn2)-c2cccnc2N1.c1(CCN)ccccc1 N1(C(C(c2ccsc2)CCNC=O)=O)CCCCC1CNC(=O)CCC1(C)CC1 C1(C(C)NC(=O)C2=CCC2)CN(C(c2cc(C3CC3)cs2)=O)CCO1 c1(C(=O)N(C(C2COCCN2CCO)=O)CCc2ccccc2)cc(I)ccc1Cl C(=O)(C(F)CC(C)(C)NC(c1cn(C)c(C)n1)=O)NC(CC=C)CC C(CC(C(=O)Nc1cccc(Cl)c1)NC(c1n[nH]c(C)c1Cl)=O)=CC c1(CN2C(C)(C(=O)Nc3ncc(Br)nc3I)CC2)c(F)cc([N+](=O)[O-])cc1F c1(C(=O)NCC2CN(C(C3(CC)CCC3)=O)C2)ccc2nc(O)oc2c1 c1(C2C(C)CCO2)c(Oc2cccc(Cl)c2)ccc2ccccc12 c1(C(N(C)CCN(c2nccc(CO)n2)C)=O)ccc(C(=O)OC)c(F)c1 c1(CCC)c(C(N2CCCC2C(C)(C)CNC(=O)CC2CCOC2)=O)nnn1C CCCC(C(=O)N1CCOCC1)NC(C1(CC2CC2)CCC1)=O C1(CNC(C2C(C)CCN2C(=O)CC2CC3(CCC3)C2)=O)CC(C2CC2)=NO1 Cc1cccc(C(=O)Nc2ccsc2C(N2CCOCC2C(C)C)=O)c1C Cc1ccc(Br)cc1C(N1CCCC(C(=O)NCCc2cscn2)C1)=O C(=O)(C#CC(C)(C)O)NC(C(C)NC(c1cn(C(C)C)nc1)=O)C(C)C c1(C(=O)NC2(CC=C)CCN(C(C3CCN3CC)=O)C2)coc2c1CCCC2 N1(C(Cn2ccc(C)n2)=O)CCC2(CC1)CCN(c1ncnn3ccc(Br)c13)C2 c1(C(C(=O)NC2CN(C(c3occ(C)c3)=O)CC2F)C)ccc(F)c(F)c1 CCC(CC)C(C)C(=O)N(C)CCNC(c1cc2c(s1)COCC2)=O N1(C(C(C)(CO)NC(C)=O)=O)CCN(C(C2CC(O)CN2C)=O)CC(C)(C)C1 C(=O)(C(COC)NC)NCCN1CCC(C(=O)OCC)C1 c1(C(N(CCN(C(CC(COC)C)=O)C(C)C)C)=O)cc(Br)ccc1OC N1(C(=O)OC(C)(C)C)CCC(F)(CNC(C2CC(CCO)C2)=O)C1 N1(C(C2(C)CCCNS2(=O)=O)=O)CCn2c(CNCC3CC(OC)C3)nnc2C1 c1(C(=O)NC(CCN(C(C(CC)OC)=O)C)C)ccc(C#CC2CC2)cc1 CC1CN(C(=O)CCOC2CC2)CC1CNC(c1csc(C(F)F)n1)=O n1(CC(=O)OCC)c(N2CCC(C)C2)nnc1-c1cc(Br)no1 N1(C(CN(C)CC)=O)CCC2(CC1)CC(C)N(C(C1CC3C=CC1CC3)=O)C2 C(=O)(CCC(C)CCCC)N1CC(NC(CCCOCC=C)=O)C(C(F)(F)F)C1 c1(C(=O)NC2C(C)N(C(c3ccc[n+]([O-])c3)=O)CC2)cncc2c(O)nccc12 CN1C(=O)CC(NC(=O)NC2CCC23CCCC3)C1c1ccc(F)c(F)c1 CC1(C)CN(C(C2CCC(C(F)(F)F)C2)=O)C(C)(C)C1O N1(C(c2ccc(OC(C)C)cc2)=O)CC2(CCC2NC(=O)C=C2CCCCC2)C1 c1(C(N2CC(CNC(CCC(C)SC)=O)C(N(C)C)C2)=O)ccc(CO)c(F)c1 C#CCCCC(C)C(=O)NC(CCC1CCC1)C(=O)NCC(C#N)CC c1(C(=O)NC(CCNC(C(C)=C2CC2)=O)Cc2ccccc2)c(Br)ncn1C CC(CC(=O)NC1CN2CCC1CC2)C(C)(C)NC(C1C=CC=CC=C1)=O Cc1cc(C(N2CC(CNC(C3(C(F)F)CCOCC3)=O)C3CC23)=O)c(C)n1C Cn1cc(C(N2C3CCC2CN(C(=O)CCn2cnnn2)C3)=O)cc1S(N)(=O)=O c1(C(N2C(CNC(CCn3c(C(C)C)ncc3)=O)CC2)=O)nn(C)cc1N N1(C(C2(CC)CNC(=O)C2)=O)CC2(CC(C(N3CC(=O)NC(C)C3)=O)CO2)C1 c1(NC(=O)OC(C)(C)C)ccc2c(c1)C(=O)CC(NC(c1cnco1)=O)C2 C1(NC(C(c2nc(C)sc2)=O)=O)CN(C(=O)C(C)(C)C)CC(C)(C)C1.C1(C(=O)N)CC1 c1(OCC2CCN(C(C3C(OC)CCC3)=O)CC2)cccc(F)c1[N+](=O)[O-] C1(CNC(C(CCCC)=O)=O)CN(C(c2cc3sccc3s2)=O)CCC1(F)F C1(CC)C(C(=O)NC2(CO)CC(O)C2)CCCN1C(=O)C(C)COC c1(OCCC)ccc(C(=O)NCC2CCC(C)CN2C(=O)CS(N)(=O)=O)cc1N C1(CNC(c2cnc(SC)[nH]2)=O)CCN(C(=O)C(F)(F)CO)CC1C C(=O)(C(C)(O)C(F)(F)F)N1CCC(OC)(CNC(C23CCCC2C3)=O)CC1 CC(C)CCCCC(=O)N(C)CC1CN(C(C2CCC3CCC2O3)=O)CCO1 C1(C)(C(=O)NC(CC)CN(C)C(c2csc(C(C)C)n2)=O)CC2(CCC2)C1 N1(C(c2cncc(SC)c2)=O)CCC2(CCC2NC(=O)Cn2nnc(C)n2)CC1 c1(N2CCCN(Cc3cc(O)c(Cl)cc3)CC2)ncnc2[nH]ccc12 C#CC1(C(=O)NC2CC(=O)N(C)C2=O)CCN(C(c2c[nH]c(C)c2)=O)C1 C(=O)(C(C(C)C)N(CC(C)NC(C1(C)CCCC1)=O)CC)NCC N1(C(C23CC(COC)(OC2)C3)=O)CCCN(C(c2cnns2)=O)C(C)C1 C(=O)(C(CC(C)C)n1ccnc1)N(CCNC(c1c(C)nc(Br)o1)=O)C1CC1 c1(C(N2CCC(CNC(c3c(COC)ncs3)=O)C2)=O)cc([N+](=O)[O-])ccc1C c1(C(N(CC(CNC(C2CC=C(C)CC2)=O)C)C)=O)coc2c1COC2 C12(C(N3C(C(=O)NCCN(CCC)C(C)=O)CCC3)=O)CCCC1CCC2 C1(NCc2ccccc2)C(C)CCCN1C(CSc1cccc(C)c1)=O N1(C(C(c2cn(C)nn2)NC(C=C(C)C(C)(C)C)=O)=O)CCC2(C1)CN(C)C2 C1(C2CCC2)(C(N2CC(O)(CNC(C(c3ccccc3)OC)=O)C2)=O)CC1(F)F c1(OC)ccc(Cl)c(CC(=O)NCC(C2CCC2)NC(C2CC2F)=O)c1 Cc1cccc(CN(CC(=O)NC(C)C(C)NC(=O)COC2CCCC2)C)c1 C(=O)(C1=NOC(C)C1C)N1C(CC)C(NC(c2ccnn2C(C)C)=O)CC1 c1(-c2cccc(C)c2)cnc(Cl)c(C(N2CC(O)C(O)C2c2ccccc2)=O)c1 C1(CC(=O)NC(C2(O)CCN(C(C3CSCCS3)=O)C2)C)CCC(C)(C)CC1 C#CC(C(C)(C)C)NC(=O)CC1(NC(=O)CCOCC2CC2)CCCCC1 c1(NCC2(OCC)CCOC2)cc(=NCCc2nc[nH]c2Br)[nH]c(CC)n1 C#CCC(O)C(=O)NC1CC1CNC(=O)Cc1csc(-c2ccc(Cl)cc2)n1 CCC1=C(C(=O)NC2CCC(CCC(=O)NCC3CC(C)(O)C3)C2)CCCO1 c1(CC)c(N2CC(CCOC)(OC)C2)ncnc1Cl.c12cccc(c1)CNC2=O C#Cc1cc(C(=O)NCC2(C)CCCN2C(c2ccc(=O)n(C)c2)=O)cc(F)c1 Nc1cccn(CC(=O)NC2CCCC(NC(=O)C=CSCc3ccco3)C2)c1=O C1(CNC(C(C)OCCOCC)=O)CCC(C(N2CCC(F)(CF)C2)=O)CC1 N1(C(CC2CC(=C)C2)=O)CCC=C(C(=O)N2CCCC(N(C)C)CC2)C1 c1(C(=O)NC(CNC(C(CC)(C)OC)=O)C)ccc(C(F)(F)F)c(F)c1 C1(C(N(C(CNC(=O)CCCCO)C2CC2)C)=O)CC(=O)NC1(C)C N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)CC2CC3CCC2O3)C2(CCC2)C1 C1(C(=O)NCC(N(C(=O)CC2CS(=O)(=O)C2)C)C2CC2)Cc2n[nH]cc2C(=O)N1 C1(CC)CCC(N=c2nc(O)c3c(ncn3C)[nH]2)C1 CC1CN(C(=O)C(F)C(C)(C)O)CCCN1C(c1cc(Cl)ncc1N)=O CCCC(C)CC(=O)NCC(C1CCCCC1)NC(C12CC(C1)C(C)O2)=O N1(C(CSC)=O)CC2(CCC2CNC(=O)CSc2cccs2)C1 c1(OC)cncc(C(N2CC=CC2CNC(=O)CCOCC(F)(F)F)=O)c1 S(=O)(=O)(c1cccc2c1OCCCO2)NC(c1ccc(=NC)[nH]c1)=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC1CC1C(=O)NCC(COC)CO Cn1cc(C(=O)NC(CNC(C2(S(C)(=O)=O)CCC2)=O)CO)n(C)c1=O c1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)cc(S(N)(=O)=O)co1 c1(C(N2C(COC)C=CC2)=O)n[nH]c2cccc(-c3cnoc3C)c12 N1(C(c2c(C3(C)CC3)cccc2)=O)CCN(C(C23CCCC(C2)OC3)=O)C(CO)C1 CC1=NOC2(C1)CC(C(N1CCC(NC(=O)Cc3cncc(C)c3)C1(C)C)=O)C2 c1(C(=O)NCC(CC)NC(=O)C(F)(F)C2(O)CCC2)ccc(COC)s1 C1(NC(CCOC)=O)CCCC1NC(=O)COCC1CCC1 Cc1cc(C)c(C(=O)NCC(C2CCCN2C(=O)COC(F)(F)F)(C)C)c(O)n1 c1(C(=O)NC2C(NC(CCc3cc(C)on3)=O)COC2)cnc2[nH]ncc2c1 CCC(COC)C(=O)NC1CCCC1CC(=O)NCC1CC(C(C)C)C1 CC(C)(CO)CC(O)CNC(c1ccccc1N1CCCCC1)CCO Cc1cc(C(=O)N(C2CCCN(C(=O)C(N3CCNC3=O)C)C2)CCF)n(C)n1 Cc1ncc(C(=O)NC2CC(C(N3CCC(CC(N)=O)C3)=O)C2)cn1 N1(C(c2c(CC)nc(C)s2)=O)CCN(C(=O)C(COC)N(C)C)CC(C)(C)C1 CC(C)C(C(=O)NCC(C)CNC(c1ccon1)=O)NS(N)(=O)=O N1(C(Cn2c(C)ncc2)=O)CC(C)N(C(c2ns[nH]c2=O)=O)CC1C N1(C(C=CCCC)=O)CCN(C(=O)CCN(C(=O)C(CCOC)OC)CC)CC1 c1(CN2CC(C(=O)NCCn3c(C)ncc3)SCC2)cc(F)ccc1Br CC1(CNC(=O)CCN2CCOCC2)CCN(C(c2cnc(C3CC3)s2)=O)C1 c1(C(=O)NC(CNC(=O)OCC)C)cccc(NC(C2CC=CCC2)=O)c1 C1(N(C(=O)Cn2cc(Cl)cn2)C)CN(C(C2CCCCC2(C)C)=O)CCC1O N1(C(Cn2c(C)ccn2)=O)CC(NC(c2ccc(C3(C)CC3)cc2)=O)CC1C C(N=c1nc(N(C)CCc2nccs2)c2sccc2[nH]1)c1c(OC)c(Cl)ccc1 C(CC(=O)NCC1(C)CCN(C(c2ccc(SC)cc2)=O)C1)(C(C)C)OCC C1(C(C)C)CN(C(=O)CC(C)c2ccccc2)CCN1C(=O)C1=COCCO1 N1(C(CCc2cc(C)on2)=O)CCC(C)(CNC(=O)Cc2ccc(Br)cn2)C1 n1(CCC)ncc(C(=O)NCC2CN(C(c3cc(F)cs3)=O)C2)c1C C(=O)(C1=NN(C)C(=O)CC1)N1C(CC)C(NC(c2cncn(C)c2=O)=O)CCC1 c1(C(=O)NCCCNC(c2[nH]cc(C(=O)OC)c2)=O)cnnc2ccccc12 c1(COC)ccc(NCc2ccccc2)c(C2(C)CC2N2CCCC(CN)C2)c1 N1(C(c2c(N)cnc(Cl)c2)=O)CC2CCCN(C(c3cnn[nH]3)=O)C2C1 C1(CC(=O)NCC2=C(C)CCC2)N(C(C2CCN(C)C2C)=O)CCC1(C)C C1(C(=O)NC2CCCC2C(=O)NC2CCN(CCO)CC2)CCS(=O)CC1 N1(C(=O)NCC2(c3ccc(C#N)c(Cl)c3)CCCCC2)CCN2CCCC2C1 CC(Cc1ccccc1)C(=O)NCCC(C)(C)NC(c1cc(C(N)=O)no1)=O c1(C(N2CCC(C(=O)Nc3c(C)ccc(O)c3)C2(C)C)=O)c[nH]c2cccnc12 CC(F)(F)C(C)(C)CNC(=O)C(=O)N(CCO)CC1CCC(=O)N1c1ccccc1 CCCC(CCC)=CC(=O)N(CCNC(=O)Cn1nccn1)C1CC1 CC1(C)CCCN(S(=O)(=O)N2CCC(F)(F)CC2c2ccccc2)C1 CC1CCC(CNC(c2nccnc2-n2ccnc2)=O)N(C(=O)COC(F)F)C1 C1(c2n(C3(C)CC3)nnn2)(NCC23COC(CF)(C2)C3)CCOC2(CC2)C1 O=C(C#CC1CCCO1)NCC1CN(C(=O)C2=CCCS2)CC12CCC2 C(CCCCC(=O)NC(C1(O)CCN(C(C2CC(SC)C2)=O)C1)C)SC C(=O)(C(CC1CCOCC1)NC(=O)CC1CC1CC)N(CC=C)CC1CCCC1 C(=O)(CC(C(F)(F)F)N(C)C(c1csc(O)n1)=O)NCC(COC)OC N1(C(c2cc(Cl)ncc2Cl)=O)CCCC2C1CCN2c1ncnc2cc(Br)sc12 C1(C(C)C)CN(C(=O)CC2(C)CC(F)(F)C2)CCN1C(C1CC(=O)NC1(C)C)=O C1(NC(CSCCCC)=O)CCC12CN(C(c1ccco1)=O)C2 c1(NC(C2C(C)(NC(=O)OC(C)(C)C)CCCC2)=O)ccc2c(c1)C(O)CC2 c1(NC(C(CCC#C)NC(=O)Cc2nc(=N)[nH][nH]2)=O)cccc2c1CCO2 N1(C(c2ccc(F)cc2Cl)c2nn[nH]n2)C2CCCC1CC(O)C2 c1(NC(C(N2C(CC(=O)OC)CC(F)(F)C2)=O)=O)cnc2ccccc2c1Br Cc1cc2ncn(CC(=O)NCC(C)N(C(=O)C=CCCC(C)C)C)c2cc1C N1(C(c2c(C(C)C)nns2)=O)CC2CCC1CN2C(c1cnc2ncccn12)=O C1(C(=O)NC(CC#C)CC#C)CCN(C(=O)C(CC(=C)C)OC)C12CCC2 N1(C(c2cc(CNC(CCC(=O)NCC)=O)no2)=O)CCC(CO)C(C)C1 N1(C(C=NOC)=O)CCC12CN(C(C1CCN(C3CC3)CC1)=O)C2.c1(C)ccccc1 C#CC1CCN(C(=O)C(F)C2CC(NC(C3(N(C)C)CC3)=O)C2)C1 C(=O)(C(CCF)NC(C1C=CCN(C(c2oc(C)cc2C)=O)C1)=O)OC C(=O)(CC(C)C(C)C(C)C)N1CCC(CNC(c2c(OC)scc2)=O)C(C)C1 c1(C(CN(C(N2C(Cn3ccc(C)n3)CCCC2)=O)CCO)=O)c(C)nn(C)c1F C1(CNC(CN(c2ccncc2)C)=O)CC(F)(CNC(C23CCC2C3)=O)C1 c1(OC)ccc(C)c(C(=O)N(C(CNC(c2cc(O)no2)=O)C2CC2)C)c1 C(=O)(C1=CNC2=NCCCN12)N1CC(CN(C(=O)C=CC(F)(F)F)C)OCC1 c1(C(=O)NC(CN(C(=O)C(C)CC(N)=O)CC)C)cc(Br)c2c(c1)CCO2 CCC(CCCC(=O)NCCCC(C)(C)C)NC(c1cnn(C)c1OC)=O C1(O)(CNC(C=CC(C)C)=O)CCN(C(C2CCN(CC(C)C)C2)=O)C1 C1(OC)CC(NC(=O)CCc2cc(C)on2)CN(C(C2CC(C)(O)C2)=O)C1 N1(C(C=C(C)C2CC2)=O)CCOC2(CCC(N=c3nc(C(C)C)[nH]s3)CC2)C1 C(C(C(C)(C)C)NC(=O)CC(C)O)NC(C1N(CC)CCC1)=O C1(C(=O)NCC(C)=CC(=O)NCC2CCC(=O)O2)CC12CCCC2 Cc1ccc2cc(C(=O)NC(C)(C)CN(C(=O)C=Cc3cn(C)nn3)C)[nH]c2c1 n1(CC(=O)NC(CNC(c2cnc(CC(C)C)[nH]2)=O)C)ccc(O)nc1=O c1(C(=O)NCC(CC(C)C)NC(C=C(COC)C)=O)ccc2c(c1)CCCS2 c1(C(N(c2ccoc2)CCNC(c2n(C(CC)C)ncc2)=O)=O)ccc(Cl)nc1 C1(c2n(C)nnn2)(NCCCSCCO)CC2(CCCOC2)C1 CCCCC(CC)C(=O)NCc1occc1C(=O)NCC(CC)n1cccn1 c1(CC(N2CC3C(CNC(c4c(C)ncnc4)=O)C3C2)=O)cccc2c1OCO2 N1(C(Cc2ccc(SC)cc2)=O)CCN(C(=O)C2=C(Cl)CCOC2)CC(O)C1 C(=O)(C1CCCn2c(Br)cnc21)NCCCN(C(C(C)O)=O)C1CC1 N#CC1CN(C(c2cncc(F)c2)=O)CCN1C(c1c(I)ccnc1Cl)=O C=C1c2ccccc2C(=O)N1C(C)C(N1CCC(C)S(=O)(=O)CC1)=O N1(C(C=CCN(C)C)=O)CCN(C2CCN(C(c3csnn3)=O)C2)CC1 CCCCCCC(C)C(=O)NCC1CCC1NC(C1(CC)CCC1)=O C(=O)(C(F)C(C)(F)F)NCC1(COC)CCCN1C(c1cccc(C(C)C)n1)=O O=C(CC(C1CCCCC1)c1ccon1)N(C1CC1)CC1CCC(=O)NC1 c1(SC(CC)C(=O)NC(c2ccc(C(C)C)cc2)CO)ccc(Br)cc1 C1(NC(C(CC=CC)NC(c2ccn(C(F)F)n2)=O)=O)CCC(=O)NC1C C1(NC(C2(C(C)C)CCCN2C(C2CCCOCC2)=O)=O)CC2(C1)CC(C#N)C2 c1(C(=O)NCCn2cc(C(c3ccccc3)(C)C)nn2)cnc2c(Cl)cccn12 C1(NC(CSc2ccc(OCC)cc2)=O)CCN(C(=O)CC(=O)OC)CC1F C1(COC)(NC(c2ccc(OC)s2)=O)CCCN(C(=O)C(C)SC)C1 C1(NC(C(=O)NCc2c(Br)cc(OC)c(F)c2)=O)CC(C)(C)NC(C)(C)C1 c12cccc(c1)C2=O.C1(CC(=O)NCC(N)=O)COCCO1 N1(C(CC(c2c(C)noc2C)C)=O)CCC(NC(C2CSC2)=O)C(C)(C)C1 N1(C(c2nc(CC)sc2)=O)CC(CNC(=O)C(=O)NCCC(N)=O)CC1C C1(NC(CNC(CCC)=O)=O)CC(C)CN(C(c2cc(CCCO)on2)=O)C1 N1(C(=O)OC(C)(C)C)CC(C(=O)NC2CC23CCCC3)CC(F)C1 C1(C(C)C)CN(C(c2ncn(C)n2)=O)CCN1C(c1cc(Br)n(C)n1)=O n1(CC)nc(C(=O)NCC2CC(C)N(C(=O)Cc3ncoc3C)C2)cc1C Cc1ccc2cc(C(=O)NC(C)Cn3cc(-c4cocn4)nn3)sc2c1 c1(SC)cn(C)nc1C(=O)NC1C=CC(CNC(C2CC=CCO2)=O)C1 C(CC)(C(=O)NC(C1CC1)CC)=CC.C12CCCN1C(=O)CN(C)C(=O)C21CCC1 C1(C(=O)NC(c2nc(C)no2)C)(CC)CCCN1C(=O)C(c1ccn(C)c1)C C1(C(N(CCNC(=O)CSc2cccc(Cl)c2)CC)=O)CCCCC12CCC2 N1(C(=O)OC(C)(C)C)C2CCC1CC(NC1(CCC#N)CCS(=O)(=O)C1)C2 c1(C(=O)NCC(C)N(C(C(C)OCc2ccc(C)cc2)=O)C)ccc(C)nc1N CC1=NOC(C(=O)NC(CNC(=O)CNC(c2cccc(F)c2)=O)C2CC2)C1C N1(C(c2ncc(C)[nH]2)=O)CC2(CCOCC2)C1c1cn(C2CC2)nn1 c1(C(=O)NCC(=O)NCC(C2CC2)SC2CC(O)C2)cnccn1 c1(C2N(C(=O)Nc3[nH]c(=N)sc3)CCC2)cc(C(F)(F)F)cc(F)c1 N1(C(c2c(C)ncnc2)=O)CC2CCCC(NC(c3cnoc3)=O)C2C1 N1(C(CCC2C(C)C2)=O)CCC2(CCC(N(C(=O)CC3CCC(=O)N3)C)CC2)C1 C1(NC(CNC(C2C(C)C2)=O)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1O CC1(C2(C(=O)NCCCCC3CC3)CC2)CC1 C1(C(=O)NCCC(C)NC(=O)C(C)(C)C2CCCO2)CCC(N(C)C)CC1 n1(CCC(=O)NCC(CN(C(Cc2cc(C)n(C)n2)=O)C)O)ccc(O)nc1=O c1(C(NNC(=O)Nc2cn(CC(=O)N(C)C)nn2)=O)cccc2ccoc12 c1(C(N2C(CNC(C3C(C)C3C)=O)C(O)C(O)C2)=O)cc(=O)c2ccccc2[nH]1 C1(NC(c2cc(C(C)C)on2)=O)CC(O)CN(C(C2OCCCC2(C)C)=O)C1 c1(C(N(C(C(=O)NC)CO)C2CC2)=O)nc(C(=O)OC)co1 C1(C(N2CC(O)(CCNC(c3nocc3Cl)=O)C2)=O)CCC2(CC1)CC(O)C2 C=CCC(C)(C)CC(=O)NC1COCC1NC(C1CCCN(C(=O)N(C)C)C1)=O Cc1nn(C)c(C)c1C(=O)NCc1cc(C(=O)O)ccc1C(F)(F)F N1(CC)CCCC(C(N)=O)C1.C1(=O)C(C)(C)n2cc(nn2)CC(C)C(=O)O1 N1(C(c2c(CC)nn(C)c2)=O)CC(C)N(C(c2ccc(COC)o2)=O)CC1C C(C(=O)N1CC(C)(O)CO1)N(C(=O)CC1=CCCC1)C(C)C C1(C2C(CC(=O)NC(CCC)c3ccco3)C2)CC(C#N)C1.C(=O)C(F)OC(F)(F)F C(=O)(CCC(=O)N(C)C)NC(C)CNC(=O)C(C)C1CCCC1 N1(C(C(CC#C)NC(c2cccc(CO)c2)=O)=O)CCCC(C)(C#N)C1 Cc1ncnc2c1CC(C(=O)N(CCC(C(C)C)NC(c1ccoc1)=O)C)CC2 N1(C(C(C)NC(N)=O)=O)CCCC(C2CCCN(C(C3OCCC3(C)C)=O)C2)C1 C1(CC(=O)NC2C=CC(CNC(C(C)O)=O)C2)C(C)(C)C1(C)C S(=O)(=O)(c1cccc2cnccc12)N(C(C(F)(F)F)C12CC(C1)C2)C1(C)CCC1 C(CCCC(=O)N(CC(C)(C)CNC(C1CCC1c1nc[nH]n1)=O)C)(OC)OC c1(C(N2CCCC(N(C(=O)CC3CCC3)CC)C2)=O)c2c(nn1C)CCCC2 c1(NC(C2(C)CCCC2)=O)cnc(Cl)cc1C(=O)NCc1ccccc1F CCCC(C)(O)CNc1cccc(-n2cc(C(C)(C)CC)nn2)c1 N1(C(CN2CCC(C)(C)C2)=O)CC2ON=C(CNC(=O)CC(=O)N(C)C)C2C1 CCCCC(O)C(=O)NC1(C)CC(C(=O)NC2(C)CCOCC2)C1 n1(CC(=O)N(C(C)CCNC(c2nc(C3CC3)cs2)=O)C)nc(O)ccc1=O C(CCS(C)(=O)=O)(N(C)C(=O)OC(C)(C)C)NC1CC2C=CCC12 Cc1nc(C)c(C(=O)NC2CCN(C(=O)CC3CCN(C)C3=O)CC2O)c(C)n1 N1(C(c2cc(C(C)=O)oc2)=O)CC(N(C)C(c2c(C)ncn2C)=O)C(F)C1 c1(C(=O)NC2CCC(NC(C(CCC)O)=O)CC2)ccc(C)nc1O c1(OC)cc(C(N2CC3(CCN(C(=O)C(C)C(C)(F)F)C3)C2)=O)c(N)c(C)c1 C(=O)(C1COc2ccc(Cl)cc21)N1C(CNC(=O)Cc2nc[nH]n2)CC(O)C1 c1(C(=O)NCCC(=O)NC(CNC(C2C(C)CCO2)=O)C)ncccc1O C12(C(N3CC(CNC(C4(C)CC4)=O)OCCC3)=O)CCCCN1CCC2 CC(C(=O)N1CCCOC(CNC(=O)Cn2cnnn2)C1)C(F)(F)F C(C(=O)N(CCC(=O)N1CC(O)(C(=O)OC)C1)OC)N1CC2N(CC)C(CC2)C1 C1(COC(=O)CCC(C)SCCCC)CN(C)C(=O)CCN(CC(C)(C)C)CC1 Cc1cc(C(=O)NC2CC(=O)N(C3CN(C(c4cnc(C)s4)=O)C3)C2)ccn1 N1(C(CCCCCC)=O)CC2=C(C1)CN(C(C1CC3CCC1C3)=O)C2 c1(C(C(=O)O)NC(N(C)CC2CCCN2C)=O)ccccc1Br C(=O)(C(C)(F)C(=O)N(CC(C)NC(=O)CN1CCCC1)C)OCC N1(C(C(N2CCOCC2)C)=O)CCCC1CC(=O)NCC1(CC2CC2)CC1 C12(C(N3CC(C)C(CC(=O)NCC4CNC(=O)C4)C3)=O)CCCC1OCC2 C#CCC(C)(CC)C(=O)N1CCCC(CNC(c2scnc2C)=O)C1 Cc1ccccc1COCC(=O)NC(C)C(C)NC(c1ncccc1O)=O N1(C(CCn2c(C)csc2=O)=O)CCN(C(c2cncc(CO)c2)=O)C(CO)C1 N1(C(c2c(CC)c[nH]c2)=O)CC(O)CC1CNC(c1csc(=NC)[nH]1)=O N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)C(F)(F)C(O)C3CC3)CC2CC1 C1(C(=O)Nc2cn(CCN3CCCCC3)nn2)CCCCC1C1CC1 Cc1ccc2cc(C(N3CCC(NC(C4CCC(C)CC4)=O)C(C)C3)=O)cn2c1 C1(C(=O)NC(C(C)C)C2CCC2)CN(C(=O)NC2CC2)CC1C(C)C c1(C(N2CCC(NC(CC(C)(C)SC)=O)C2)=O)cccc(S(N)(=O)=O)c1 c1(C(=O)NC2CC(C)(NC(C(CC)C)=O)C2)cccn(C2CCSC2)c1=O C1(C(=O)NC2C(C)(C)CCN(C(C=NOC)=O)C2)COc2ccc(O)cc2O1 c1(C(=O)NCCCNC(c2c(CC)scc2)=O)cc(C)c(F)o1 C1(C(=O)NCc2c(C(=O)NC3COC(C(F)F)C3)c[nH]n2)CC12CCCC2 c1(C(C)NC(c2c(C)nn[nH]2)=O)cccc(N2CCOC2=O)c1 c1(Cc2cn(CCCNC(C(CN(CC)CC)F)=O)nn2)cccc(S(C)(=O)=O)c1 c1(C(=O)NCC2CC3CC3N2C(=O)CC2CC=CC2)[nH]nc2ncnc(O)c12 C(=O)(C1CCc2scnc21)NCC(C1CCCCN1C(=O)CC1CCSC1)(C)C c1(CC(N2CCCCC(NC(C3(Cl)C(C(C)=O)C3)=O)C2)=O)cnc2cccnn12 C1(C(C(=O)NCC2C(NC(c3c[nH]cc3-c3ccc(Cl)s3)=O)C2)F)CCOCC1 c1(OCC(=O)N(C(C)CNC(c2ccc(C(C)O)cc2)=O)C)cc(F)cc(F)c1 C1(CNC(c2cc(C)on2)=O)CCN(C(C2(C)CCC(O)CC2)=O)CC1(F)F C1(F)(CNC(c2cccc(OCC)c2)=O)CCN(C(=O)C(C(=O)OC)OC)CC1 c1(C(N(CCOC)CCNC(C23CC(C)C2C3)=O)=O)cccc(C(C)C)n1 c1(C(=O)NCC(CCNC(C(C2CCCCC2)C)=O)O)ccn2nccc2c1 N1(C(C(CC)COC)=O)Cc2ccccc2C(NC(=O)C2=CCCC2)C1 C12(CNC(C(CO)NC(C3(C)CC(C)C3)=O)=O)CC(C)(CCO1)C2 Cc1cc(N)cnc1C(N1CCC(F)C(NC(=O)CC(C)C)C1)=O N1(C(CCC(C)NC(CSCCC)=O)=O)CCCC(C)C1CO C(=O)(CC1=CCCC1)N1CC(C)C(CNC(=O)CCNC(N)=O)C1 c1(C(N(C)CC2N(C(C3(CC(C)C)CCCC3)=O)CCC2)=O)cccnc1O c1(OC)ccc(C(N2CCC(OC(c3ccnnc3)=O)CC2)=O)c(OC)c1Cl c1(C(N(C2CCC(NC(c3ccnnc3O)=O)C2)C)=O)nccn2ccnc12 N1(C(C2=CC(C)(CC)C2)=O)CCC2CCN(C(c3sc(C)cc3Cl)=O)CC12 c1(OC)ccc(OC)c(C(=O)NC(CCN(C)C(C2CC(F)C2)=O)C(C)C)c1N c1(N2CCC(C)(NC(C3CCCCS3)=O)C2)ncc(C#N)cc1F CCCCCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C=CC=C(Cl)Cl)C1 C1(CC(=O)NC(c2cccc(C)c2)C)CCCN(C(=O)C=CC2(C)COC2)CC1 c1(C(=O)NC2(CNC(COC)=O)CCC2)cc2c([nH]1)CCOC2 C=CCC(CC)C(=O)NC1(c2cn(CCSCCO)nn2)CCOC1 N1(C(c2c(CC)c(F)ccc2)C(=O)NC(C)CC)C(C)CS(=O)(=O)CC1C CC1CCC(C(=O)N2CC(n3cc(CNC(=O)OC(C)(C)C)nn3)CO2)CC1C n1(C(CC)C)nc(C)cc1C(=O)NCC1CN(C(=O)C=CCn2cncn2)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(O)C(F)(F)F)ccc2cc[nH]c2c1F C1(N(c2nnnn2C2CC(F)(F)C2)C(c2cc(C(F)(F)F)cs2)=O)CCCC12CC2 C1(NC(COCCC(C)C)=O)COCC1C(=O)NCC1(O)CC(CO)C1 C1(C(C)NC(C2CC2C2CCCO2)=O)CCN(C(=O)C(c2ccnn2C)C)CC1 N1(C(c2c(C)nn[nH]2)=O)CCCOC(CNC(C2(C)CCCO2)=O)C1 CC12CCC(CNC(=O)NOCCCCC3CC3)(CC1)CO2 C1(C(N2CCC(CNC(C(CC=C)C)=O)C(C)C2)=O)C2CCC1(C)C2(C)C N1(C(CCC(C)OC)=O)CC2CC2CC(NC(c2c[nH]cc2Br)=O)CC1 C(=O)(CCCOC(C)(C)C)NCCN(C)C(c1cc(-c2ccccc2)ns1)=O N1(C(c2ccc(C)cc2C)=O)CCC(NC(=O)C2=C(C)CCOC2)CC(C)(C)C1 C=C(C)C(O)CC(=O)NCC1CCC1NC(c1cc(-c2csc(C)n2)c[nH]1)=O N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(C12CCCC1C2Br)=O C(=O)(C1=CCC(F)(F)CC1)NC1(CNC(C(C(C)OCC)O)=O)CCOCC1 C1(C(=O)NCc2ccc(CNC(c3cscn3)=O)cc2)CCc2c[nH]nc2C1 c1(C(C)C)cc(=NC2CC3CCC(C2)N3C(C2CC3(C2)CC3F)=O)[nH]c(Cl)n1 c1(NC(C2N(Cc3ccc(OC)cc3)CCC2)=O)ccc2c(c1)C(C)(C)C(=O)N2 c1(OC)cc(C(=O)NCc2ccc(CNC(=O)C(=O)N(C)C)cc2F)cc(C)c1 Cc1ccc(Cl)c(O)c1C(=O)N(C)CC1CCCC(NC(=O)C2=CC(C)(C)C2)C1 c1(C(N2CCC3CCCC23C(=O)O)=O)ccc2cnccc2n1 N1(C(C#C)=O)CCCC2(CCCCN2C(=O)CCc2ncc[nH]2)C1 C1(C#N)(C(N2CC(CNC(C=CC)=O)C(O)C2)=O)CC2(CC2)C1 CC1(C)CN(C(=O)C(C)(C)C2CCC2)CC(CNC(=O)CCNC(=O)C2CC2)O1 N1(C(Cc2ccc(C)cc2)=O)CCN(C(=O)C(C)n2ccnc2)C2CC12 Cn1cc(C(=O)NC(CNC(=O)C=C2CCSCC2)CO)c(C2CCC2)n1 C1(CN2CC(C3OCCN(C(C#CC(=O)N(C)C)=O)C3)C2)CCn2cnnc2C1 c1(C(=O)NCCC(C)NC(C2CCC(C)CC2)=O)cc(=O)c2ccncc2o1 C(C(F)(C(=O)N1CCCC(C)(C#N)C1)C(C)C)NC(C1CC(OCC)C1)=O N1(C(CCc2n(C)c(S)nn2)=O)CC2CCN(C(C3(F)CCCOC3)=O)CC2C1 Cc1cc(=NC(=O)CNC(c2cnc(C3CC3)nc2)c2nnnn2C2CC2)[nH]o1 c1(C(=O)NC2(CC=C)CCC2)ccoc1CNC(=O)C(C)(C)OC C(=O)(C(C)C(C)(C)C)NCC(CNC(=O)C=Cc1ncc[nH]1)OC N1(C(C(C)n2cccc2)=O)CCCC(O)(CNC(=O)CCC2CC(F)(F)C2)CC1 O=C(C1=CC2(CCN(C(=O)CC(F)(F)F)C2)C1)NCCC1CCCCC1O C1(C(N2CC(OC)C(NC(C3CC4CCC3O4)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 N1(C(C2(C#C)CC2)=O)CCC2CCN(C(=O)Cc3cccc([N+](=O)[O-])c3C)C2C1 C1(C(=O)NCC(C)(C2CC2)NC(c2c(CC)occ2)=O)CCN(C)C1C N1(C(C(CC(N)=O)NCc2cccc(C(=O)OCC)c2)=O)C2CCC1CN(C)C2 C1(C(=O)N(C(C)CC(N)=O)C)(CC)CN(C(=O)CCNC(=O)NC)C1 c1(C(=O)NCC(C2CC2)NC(CCSC)=O)cc(C#N)c(F)cc1F CCC(C(=O)NCCOC1CCN(C(=O)Cn2ncnn2)C1)N(C)C C1(NC(CSc2c(OC)cccc2)=O)C2CCC1N(C(c1sccc1SC)=O)C2 C1(NC(C2C(NC(C(C(C)C)=O)=O)CCC2)=O)CCCC2(CC1)CC2 CN1C2CCC1CC(=CC(=O)NC13CC1CN(C(c1ccc[nH]1)=O)C3)C2 c1(SCC)ccc(CN2CCC(NC(=O)C(c3nc(CSC)no3)C)C2=O)cc1 CC1CC(C(N2CCC2(C)CCO)=O)CCN1C(c1csc(F)c1)=O C1(CNC(c2occ(C(N)=O)c2)=O)CCCCN(c2ccc(C#N)nc2)C1 N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CC1)CCN(C(C1CC(C)(O)C1)=O)C2 C1(C(N(C2CCOC2)C)=O)C2CN(C(C3(C(F)(F)F)CCC3)=O)CC12 N1(C(C(C)NS(C)(=O)=O)=O)CCC(NC(C2(S(C)(=O)=O)CCCC2)=O)C12CCC2 C1(C(=O)NC(CC)C(F)(F)F)CN(C(=O)Cn2ccnc2C)CCC1(F)F c1(C(=O)NC(CC=C)CNC(C2CC(O)CN2C)=O)ncc([N+](=O)[O-])cc1C C1(C(=O)NCc2n(CC)cnn2)CCN(C(c2snnc2C)=O)C1C C(=O)(CCCN=[N+]=[N-])N1C(CC(=O)NC(C=C)C2CCC2)CC1 CC(C)CCC(=O)NCCCC(c1ccccc1)NC(=O)CC12CC(C1)C2 CC(O)C(C)C(=O)N1CC(O)(C(C)OC2CCC2)C1.c12cccc(c1)C(=O)OCC2.OC C1(CC#C)(C(N2CC(N=[N+]=[N-])C2)=O)CCN(C(c2cc[nH]c2C)=O)C1 N1(C(C(CC)N(C)CC)=O)CCN(CCNC(C2CC(n3cnnc3)C2)=O)CC1 C12(NC(c3scc(C(N)=O)c3)=O)CCCC1CN(C(C13CCC(CC1=O)C3)=O)C2 C(=O)(C#CC(C)(C)CNC(c1nc(O)sc1C)=O)N(C(C)C(=O)NC)CC C1(CC(=O)NCC(C)N(C(CCC)=O)CC)CCOC1=O CC(C)C(O)CC(=O)N1CC=CC(C(N2CCC(F)(CO)C2)=O)C1 C(=O)(C1CSc2ccccc21)N1CCC(O)(C(C)NC(CCC(=O)NC)=O)CC1 N1(C(C(C(C)C)C#N)=O)CCC(C2CC2)C1C(=O)Nc1ccc2nncn2c1 CC1CC2CCN(C(C3CCN(CC4CN(C)CCO4)CC3)=O)CC12 c1(C(=O)NC2C(NC(c3c(OC)cc(O)nc3)=O)CC2)cc2cccn2cn1 C1(C)(C(N2CCC(CNC(C(CC#C)O)=O)CC2)=O)CC(C(C)(C)C)=NO1 N1(C(C(F)OC)=O)CCC2(CC1)CN(C(C1CCCC(F)(F)C1)=O)C2 c1(C(=O)NCC(CC)NC(C2(C(=O)OC)CCC2)=O)coc(C(C)OC)n1 c1(C(=O)NCCOC2CN(C(=O)Cn3cc(Cl)cn3)C2)cc(O)ccc1F c1(OCOCC)cc(OCl)cc2ccccc12.c1ccccc1 N1(C(c2nn(CC)c(O)c2)=O)CC2(CC2)CC1CC(=O)NCCCS(C)=O C1(NC(C2C(OC)CN(C(COCCCC#C)=O)C2)=O)COCCN(C)C1 C1(CN(C(C(CC=CC)C)=O)C)CN(C(c2cccc(C#N)c2)=O)CC12CC2 CC(C)C(C)CC(=O)NC1(CCNC(C2(F)CCCOC2)=O)CC1 N(C1CCOc2cc(F)cc(F)c21)C(=O)NC(C)C(C)(C)c1ccccc1 c1(N2CC(CCO)(N(c3ccc(C)cc3)C(C)=O)C2)ncc2c(ncn2C)n1 c1(OC)cc(OC)nc(N(c2ncc(C)cn2)C(C2CCNCC2O)=O)n1 N1(C(C(CC=CCC)C)=O)CCC(CNC(c2nn[nH]c2Cl)=O)C12CC2 N1(C(CC(CNC(COCC(=O)OC)=O)O)=O)CC(=O)NCC1C(C)C c1(NC(C2N(c3ncc(C)c(C)n3)CCCC2)=O)cc(Br)c([N+](=O)[O-])cn1 C1(CC)CC(c2nnnn2C2CC(F)(F)C2)(NC2CSC2)CCO1 C1(NC(C)=O)CC2(C1)CN(C(c1cccc(C(F)F)c1F)=O)C2 N1(C(CSCCC)=O)CCC2CN(C(=O)C(C)Oc3ccc(F)cc3)C2C1 c1(C(C(=O)N(C2CN(C(C(CC)SC)=O)C2)C)O)ccc(Br)cc1 CC(C)C1=NOC(C(N2CCCC2C(C)NC(c2c(SC)cccc2F)=O)=O)C1 N1(C(C(C=C)O)=O)CC(NC(c2cnccc2C(F)(F)F)=O)CC2(CCC2)C1 N1(c2n(CC(=C)C)c(-c3cnn4cc[nH]c34)nn2)CCCC(C2CCC2)C1 C1(C(N2C(C)CN(C)CC2)=O)CCN(C(=O)C(O)O)CC1(C)C C(=O)(C1=CC2CC=CCC12)NCC1CC(NC(c2cc(C)c(Cl)c(N)c2)=O)C1 C1(N(CC(N2CCCC2=O)C)C2CC2NC(=O)OC(C)(C)C)CC2CC1CN2 C1(NC(c2nn(C)c(O)c2)=O)CCN(C(c2cnc(C3CC3)s2)=O)CC12CCC2 C1(NC(C(CC)F)=O)CN(C(=O)CN(C)Cc2ccc(Cl)cc2)CC1C c1(C(=O)NCC(C2CCCC2)NC(C(C)(C)N(C)C)=O)cccc2c1CCN2 Cn1cc(-c2cccs2)cc(NC(=O)CC(=O)NCC(F)(F)F)c1=O C=CCCCCC(=O)N1CCOC(CNC(C2CC(Oc3ccccc3)C2)=O)C1 CC(C)(CC(F)(F)F)C(=O)NC(=O)NCCN1CCC2CCCCC2C1 CC(CC(=O)NCC(C)(O)CNC(=O)C1=CCCSC1)C(F)(F)F CCC(CCOC)C(=O)NC1(CC)CCCN(C(=O)Cn2cc(Br)cn2)C1 C(=O)(CC(C)(C)C(F)(F)F)NCCCN(C(=O)C(c1cccc(F)c1)(C)O)CC CC1=C(C(=O)NC2CN(C(C3CC4C=CC3CC4)=O)CC2N(C)C)CCCO1 c1(C(=O)NCCCC2(NC(CCCCC)=O)CC2)cc2n(n1)CCNC2=O C1(C)(C(N2C(CN(C(=O)COCC3CCCC3)C)CCC2)=O)CCCNC1=O Cn1c(C(N2CCC3(NC(=O)OC(C)(C)C)CC3C2)=O)cc(=O)c2ccccc12 c1(C2C(C(N(CCCNC(C(CC)(C)O)=O)C)=O)C2)c(Cl)cccc1Cl C(CC(C)C)(C(=O)NCC(CC(F)(F)F)NC(c1coc(C(=O)OC)n1)=O)OC C1(O)(CNC(C2(CCOC)CCC2)=O)CCCN(C(=O)CCn2ccc(C)n2)C1 c1(C(N2CC=CC(C(N(C3CCNC3=O)CC)=O)C2)=O)cc2ccncc2[nH]1 Cc1nn(C)c2nc(O)cc(C(=O)NC(C)CC(C)NC(=O)CCC3(C)CC3)c12 N1(C(C(n2c(C)ccn2)C)=O)CC2(C(=O)NCC(O)CO)CC1CO2 N1(C(CC)=O)CCN(C(c2ccc(CC)nc2)=O)CC(O)C1 C(C(C)(COC)CC)NC(C(C=CC)O)=O.C1C(=O)N1CC(C)C C1(C(=O)NCCN(CCOC)C(C2(C(C)(C)C)CCC2)=O)CCC(=O)N1.S(C)(=O)(=O)N C(C1CCc2cc(F)ccc21)NC(c1ccc(N2CCCS2(=O)=O)cc1)=O C1(C(=O)NCC(=O)NCC2(C)CC2)CN2CCC1C2 N1(C(c2c(NC)cncc2)=O)CC(CNC(=O)C(C)c2ccco2)CC1(C)C N1(C(C(C=C=C)C)=O)CCN(C(=O)Cc2nnn(C(C)(C)C)n2)C(CO)C1 FC(F)(F)C(CN=c1[nH]cnc2ccc(I)cc12)N1CCCCCC1 N1(C(C2CC(O)(CC#C)C2)=O)CC=CC1(C)C(N1CC(N(C)CC)C1)=O C(c1ccncc1)=CC(=O)NC1CC(CNC(c2nnc(C(F)(F)F)s2)=O)C1 C1(CNC(C=CC(CC)=CC)=O)CCN(C(c2ccncc2NC)=O)C(C)C1 N1(C(C2C(C)C2)=O)CCC(CNC(=O)C(C)Cc2ccccc2F)C1(C)C N1(C(CC(CC2CC2)NC(C2ON=C(C)C2)=O)=O)CC2CC1CS2=O C12(NC(CCOCCOC)=O)CCCC1N(C(=O)COCCCC(C)C)CCC2 N1(C(C23N(C(c4ccc(Cl)o4)=O)CCC2C3)=O)CCC([N+](=O)[O-])CC1 N1(C(c2c(N)nccn2)=O)CCCC(NC(c2nn[nH]c2Cl)=O)C(F)C1 C1(C(N(C)CC2N(C(C(C)C)=O)CCOC2)=O)CCN(c2ccncc2)CC1 C#CC1CCCN(C(=O)C(=O)NCc2cc(-c3csc(C)n3)ccn2)C1 c1(-c2cn(CCCN(CCOCC(=O)NOCO)C)nn2)ccc(F)cn1 N1(C(=O)Cn2ncnn2)CCC2CN(C(C3(n4cncn4)CC3)=O)CC2C1 CCC(C)(F)C(=O)N1CCC(NC(=O)C(O)Cc2[nH]cnc2C)CC1 CCC(CC)(C(=O)NC1CC(C)N(C(=O)Cc2cnsc2)C1)OC N1(C(=O)C=CCNC(C2CCN2Cc2ccccc2)=O)CCC12CCCOC2 Cc1ncc(N)cc1C(N1CC(CNC(=O)C(c2cccc(F)c2)O)C1)=O C1(C(C(=O)N(C2CCN(CC)C2)C)C)CCN(C)CC1 N1(C(C(C(CC)CC)C)=O)CCC(C(=O)NC2CC3CCC2C(O)C3O)=C(F)C1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(c2cnn(C3CC3)c2Cl)=O)CC1(C)C C1(COC(C2OCCCO2)=O)CCCCC1.C12CN(C1)C(=O)O2 C1(NC(NC(C=C)C)=NCC2CCCS2)CCn2c(CCOC)nnc2C1 C#Cc1ccnc(C(N2CC(NC(=O)CCc3ccc(F)cc3)CC2C)=O)c1 c1(N(CC(C)(C)O)C(N(CCCCO)C)=O)cnc(C(F)(F)F)cc1 N1(CCSc2scc(C)n2)CCOC(C)(CNC(=O)C(C)(C)C(F)F)C1 C1(NC(C(CN(C)C)O)=O)CCOCC1NC(C1(CO)CCCC1)=O CN=c1c(C(=O)NC(C)C(C)NC(=O)Cn2cncc2C)c[nH]c2ccccc12 C1(C(=O)NCC(CCC)OCC)C(C)OCCN1C(=O)C(C)N(C)C N1(C(C(C)SC)=O)CCC2C(NC(=O)CCOC3CC3)CC12 c1(CC)ccc(C(C)C(=O)NC(C)(C)CNC(=O)C(C)(C)C2CCCCC2)cc1 c1(-c2c(Cl)occ2)nc(-c2ccco2)nn1-c1ccnc(F)c1 C(c1ccc(C)cc1C)=CC(N1CC(CNC(CSCC(=O)OC)=O)C(C)C1)=O C1(C(=O)NC(C)CC(C)NC(=O)CC2CCC2)(OC)CCOCC1 c1(C(=O)NC(C2CCCN(C(C3C4COCC34)=O)C2)C)ccnc2c1OCO2 N1(C(C(CCC=C)NC(=O)CC(C)n2cccc2)=O)CC2(C1)NC(=O)NC2=O N1(Cc2cncc(C)c2)CCC2(CCN(c3cc(C)ncn3)C2)C1 CC(C)C(C(=O)N1CC(C(=O)Nc2ccc(C(C)C)nc2)C(C)C1)C1CCC1 C1(NC(c2n(CC)ncc2)=O)C2CCC1CC(NC(c1cc(C)ccc1N)=O)C2 C1(C(=O)NC(C(C)NC(c2c(OCC)csc2)=O)(C)C)CCc2nc[nH]c2C1 c1(C(=O)NC(CC)CNC(=O)C(c2ccc(C)cc2)O)cc(C(N)=O)ccc1C N1(C(CC2C(C)=NN(C)C2=O)=O)CCC(C2CC2)C1CNC(=O)C=CCF C(=O)(C1=NNC(=O)C1)NCCN1CCN(C(c2cc(C(=O)OC)ncc2)=O)CC1 C#CCCCC(=O)N(C1CCN(C(=O)C=C2CCCO2)CC1)CCOC Cc1n[nH]c(C)c1CCC(=O)N(C1CN(C(=O)CC2CCC(=O)N2)CC1O)C c1(C(N2C(CCC)CN(C(=O)COC)CC2)=O)c(OC)ccc(C)c1OC c1(CNc2c(CNc3c(Cl)cc(C)c(Br)n3)nccc2)cccc2cnccc12 C1(NC(c2n(C)nc(CC)c2Cl)=O)CC2CCC1N(C(=O)CC(C)C(C)C)C2 S(=O)(=O)(c1cc(Br)c(F)cc1F)NCC1N(Cc2n(CC)ncc2)CCOC1 c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCC#C)=O)cccc([N+](=O)[O-])c1 N1(C(C(C)OCCOCC)=O)CCCN(C(=O)C=CC(C)(C)C)CC1C CCCCC(CC(=O)NC1CC(C(F)F)C1)NC(C12CCCN1CCC2)=O C(=O)(CCCCCNC(=O)Cc1cc[nH]n1)N1C(CC)(CC)CC1 CC1C(C)N(C(c2cc3ccncc3o2)C(=O)Nc2ccc(F)cc2)CCS1=O C(=O)(CS(=O)(=O)CCO)N1CCC(NC(c2cc(CC)n(C)n2)=O)C(F)C1 C1(C(=O)NC2(C(=O)NC(c3cn[nH]c3)C)CC2C)CC2CCC(C1)C2 N1(C(c2c(CC)nnc(C)c2)=O)CCCCC2(CCN(C(=O)C(C)(C)OC)C2)C1 C(=O)(C(F)CCC(C)C)N(C)CC1CCN(C(=O)C(F)(F)CCn2ccnn2)C1 c1(NC)cccc(C(N2CC=CC(NC(=O)C=C3CCC(C)CC3)C2)=O)n1 c1(N2CCC(C)C(NC(c3c(C)onc3)=O)C2C)ncc2ncn(C)c2n1 c1(C(N2CC(NC(C(N3CCOCC3)C)=O)C2)=O)ccc(C2CCC2(C)C)cc1 Cc1ncccc1NC(C1CSCCN1Cc1cncc(-c2ccccc2)c1)=O C1(NC(CC=CC(C)(C)C)=O)CCCC(C(=O)NC2(CC(C)(C)C)CC2)C1 c1(C(=O)NCC2C(NC(=O)CCCC3CCC3)CC2)cc(O)nc2cnccc12 c1(OCC(=O)NC2C(C(=O)NC3CN(C(C)=O)C3)CCC2)cncc(C)n1 C1(C2CCOCC2)(C(=O)NC(CNC(c2c(Cl)ccc(C)c2)=O)C)CC1(F)F C1(C(=O)NCCSCCC=C)CCC(O)CN1C(c1ccn(C)c(=O)c1)=O N(C1CCCc2ccc(Br)cc21)CC(C)(C)C N1(C(CCC(=C)Br)=O)CCC(CO)(NC(=O)CC2CCCNC(=O)C2)CC1 c1(C(=O)NCC2(O)CC(CNC(CC=CCC)=O)C2)cc(F)cc([N+](=O)[O-])c1 c1(CNC(=NCC=C)NC(CO)CCF)ccc2c(n1)CCCC2 CCC(C)C(O)C(=O)N1CCCC(C(N2CC(c3nc(=O)o[nH]3)C2)=O)C1C c1(C(C(F)(F)F)NC(=O)C(N2CCCC2CN2CCCC2)=O)ccc(Br)cn1 C1(NC(c2cc(OCC)n[nH]2)=O)CN(C(=O)CC(C)CN(C)C)C(CC)(CC)C1 CC1CN(C(C2CC2CNC(=O)C(F)CC2CCC2)=O)C(C)(C)C1 N1(C(C2(SC)CC2)=O)CCC2CN(C(=O)CC3CNC(=O)O3)CCC2C1 C1(OC)CCC(C)(c2nc(-c3ccncc3)nn2CC(=O)O)CC1 C(CC(=O)N(C1CCC(NC(=O)CCCN(C)C)C1)C)(C(F)(F)F)OC N1(C(CC(CC)(C)C)=O)CC2(CNC(C3(CCOC)CCC3)=O)CCC1CC2 C1(C(=O)NC2CCN(C(c3ccn(CC)n3)=O)C2C2CC2)CS(=O)(=O)CC12CC2 C1(NC(c2cnco2)=O)CC(C(=O)NCC2(CO)CC23CCC3)=CC1O C1(CC(N2CC(CNC(C3C(C)C3)=O)N(C)CC2)=O)CC(C)CC(C)(C)C1 c1(N2CCC(CNC(C(C)OCCCCCC)=O)C2)cc(C)ncc1C#N N1(C(Cc2nccc(OC)n2)=O)CC(C)CN(C(=O)C=CC(=O)N(C)C)C(C)C1 c1(C(=O)NC(C(C)C)CNC(=O)CC2CCN(C)CC2)cc(C#N)c(N)cc1O N=c1[nH]c(=NCCN2CCCC2=O)[nH]c(=NC(CC2CC2)c2ccccc2)[nH]1 Cc1cc(N)c(C(N2CCCCC2CCNC(C2(C)CCCO2)=O)=O)cc1C c1(C(=O)NCCCN(C(C(C=C)(C)O)=O)CC)cnc(O)c(Br)c1 CC1(C)CN(C(C2CC3(C2)CC(F)C3)=O)CC(CNC(=O)CC2CC2(Cl)Cl)O1 C1(CC(=O)NC2CCCN(C(C=C(Cn3c(C)nnn3)C)=O)C2)CCCCC1(C)C C1(CCNC(c2c(C)coc2)=O)CN(C(=O)C=CC2CCCC2)CCO1 C1(C)(CNC(C(CCOC)(C)C)=O)COCCN(C(C2CC(C)C2)=O)C1 N1(C(c2n[nH]c(C)c2Br)=O)CCOCC(NC(=O)C=CCN2CCCC2)C1 N1(C(C2CCC(=O)C2)=O)CCC(C2(NC(C3(Sc4ccccc4)CC3)=O)CC2)C1 C1(C(=O)NCC2(O)CN(C(c3nn(C)c(F)c3)=O)C2)CC2OC(=O)OC2C1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCC(CNC(C(C)(C)OCC)=O)C(C)C1 C1(C(=O)NCCSCC(=O)NC(C=C)(C)CC)CCCC12CC2 C=CC(CC)CC(=O)NC1CCCN(C(c2cnc(OC)cc2C(F)F)=O)C1 N1(C(CN(C(C)=O)C)=O)CCC2(C1)CN(C(c1cn(C3CC3)nn1)=O)CC(C)O2 C1(C2CCN(C(=O)CNC(=O)NC3CC3)C2)(NC(=O)CC2COC(=O)C2)CC1 c1(C(N(CC(C2CCCN2C(=O)C2=CCCCO2)(C)C)C)=O)cnn2ccccc12 C=CCC(C)(C(=O)N1CC(C)(C)CC1CNC(c1ccncn1)=O)N(C)C C1(=CC(=O)NCCC2COCCN2C(c2ncccc2F)=O)CN2CCC1CC2 c1(C(N2CCCC(CCNC(=O)CCC[N+](=O)[O-])C2)=O)ccc2scnc2c1 C(CC(C)C)(C(=O)NC(C)C(C(C)C)NC(C1CCCC1)=O)NC(C)=O c1(CC)c(C(=O)NOC(C)C)cnn1-c1ccc(OC)cc1 C(=O)(CCCCC(C)C)N1C(CCCNC(CCSCCC)=O)CCC1 C1(CNC(C(C)CO)=O)CCC2CN(C(c3coc(O)n3)=O)CCC2C1 N1(C(C2CC(N(C)C)C2)=O)CCC2(CCC(NC(C3CSCC(=O)N3)=O)C2)CC1 C(=O)(CCCS(N)(=O)=O)NC1CCN(C(C(c2ccc(C)nc2)(F)F)=O)CC1C N1(C(c2nnc(C)s2)C)CCC(C)(NC(=O)CC2CC=CC2)C1 Cc1cc(N(C(=O)C(C)(C)C2(O)CCOC2)C(=O)C(F)(F)F)cnc1Br N1(C(=O)Nc2nccc(-c3ccc(Cl)cc3)n2)CCCC2(CCNC2=O)C1 Cc1ccc2[nH]c(C(N3CCN(C(=O)C(O)C4CC4)CC3)=O)c(Cl)c2c1 Cc1cc(=O)oc2ccc(OCC(=O)NCC(O)CCNC(=O)CN(C)C)cc12 c1(C(=O)NCCCC2(NC(C(C)OC(C)(C)C)=O)CC2)csc(C(F)F)n1 Cc1cc(=NCc2nc3ccccn3c2Cl)[nH]c(NC2CCN(C)C(=O)C2)n1 C1(C(N(CCCNC(CCC=CC(C)C)=O)C2CC2)=O)CC1C1CCCC1 c1(CCNC(C2C(C)CNC2)=O)ccccc1Oc1ccncn1 c1(C(=O)NCCC(O)C(=O)N2CC(N3CCC3)C2)ccn2nccc2c1 N1(C(C(C2CCCC2)OC)=O)CCCC1C(=O)N(C1CCN(CC2CC2)C1)C c1(OC)c(C(N2CCCCC2c2cccs2)C(=O)NCCC2CC2)cccc1F N1(C(C=CC=CC)=O)CC(CO)C2(CCN(C(=O)C(C)(C)CC3CC3)CC2)C1 N1(C(CCc2ncn(C)c2)=O)CCC(NC(=O)CCSC(F)(F)F)C(O)C1 Cc1c(C(=O)NCC2N(C(c3ccc[nH]3)=O)CCC2(C)C)c[nH]c1C#N c1(C(=O)NC(C2CCN(C(C3(OC)CCSC3)=O)C2)(C)C)ccccc1Cl C1(C(=O)NCC(=O)OC(c2cccc(Cl)c2)C)CC1C1CCCC1 C1(N(C(CC(OCC)OCC)=O)C)CCCN(C(=O)C(C)(C)C)CC1 c1(NC(C2CC(C(=O)OC)C2)=O)cnn(C2CCCC2)c1C.C12(O)CN(C1)CC2 C1(OC)CN(C(c2ccns2)=O)CCC1NC(=O)CN1CC2CC2C1 S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CC(C(=O)Nc2cccc(C#N)c2)OCC1 n1(CC(=O)NCC2CN(C(c3cscc3C(F)(F)F)=O)C2)nnc(SC(F)F)n1 C1(C(=O)NC(C2CCCN2C(c2cc[nH]n2)=O)C)(COC)CCOCC1 c1(C(C(=O)NC(C)CC)N(CCOCC=C)C)cccc(C2CCCC2)c1 c1(NC2C3CN(C(C4CCC(CC)CC4)=O)CC32)cc(CO)nc(C(F)(F)F)n1 C1(C(N2C(CC(C)C)CC2)=O)N(C(C2CCC(=O)CC2)=O)CC12CCCC2 C1(C(=O)NC(c2ccc(F)cc2)CNC(CCCOC(C)=O)=O)CCCC1(C)C N1(C(C(COCC)NC(c2cncnc2C)=O)=O)CC(N(C)C)C2(CCC2)C1 CCCCC(CCC)NC(=O)CC(C)(C)NC(C1CC(F)C(=O)N1)=O C12(CNC(CC)=O)CCCCC1N(c1ncc(I)cn1)CC2 N1(C(=O)C=CCN2CCOCC2)CCC2CC(C1)CN(C(=O)C(O)C1CCCC1)C2 c1(C(=O)NCCN(CCOC)CC2CCCO2)c(C2CC2)cnn1C.C1(=O)CN1 C(C(C)(C)C(=O)N(C1CC(C(=O)Nc2cnc(SC)nc2)C1)C)SC N1(Cc2c(C)coc2)CCCC1(C)C.c1(NC(c2nc(C)c(C)s2)=O)ccc(F)cc1 CC1(C)CC(CC(=O)NCCC2CCCC23CC3)CN1C(=O)Cn1cnc(=N)[nH]1 c1(SC(C)C(N)=O)nc(CC(=O)N(C2CC2)CC2CC(C)CO2)cs1 Cc1cc(C(N2CCCC(O)(CN(C(=O)CN3CC=CC3)C)C2)=O)c(C)cn1 c1(C(=O)NCC2(OC)CN(C(CC(=C)C)=O)C2)ncc(C)cc1OC c1(C(=O)NCC2N(C(CC3(C)CCCO3)=O)CCC2)ccc(Br)cc1F C1(NC(C(c2cnn(C)c2)C)=O)CCCCCC1NC(c1cnc(O)n1C)=O C1(CNC(c2c(C)c[nH]n2)=O)CN(C(=O)Cn2cc(C#N)cn2)CCC1C Cc1c(CC(=O)NC2CC(CC(=O)NC34CCC(CC3)C4)C2(C)C)ncn1C C12(NC(=O)Cn3cc(C4CC4)cn3)CC1CN(C(c1ccc(C(F)F)cc1)=O)C2 Cc1cnc(NC(c2ccccc2)CF)c(S(=O)(=O)NCCc2cn(C)cn2)c1 c1(C(=O)NC2CCCN(C(=O)C(F)OC(F)(F)F)C2)ccc2ccccc2c1F C1(C(=O)NC(CCNC(CCOCCOC)=O)C(C)(C)C)CC1C1CCOCC1 Cc1nc2sccn2c1C(=O)N(C)CCC(=O)CO.c1(OCCN)cnn(C)c1 c1(C(N(C(c2cccc(OC)c2)C)C)=O)cc(S(=O)(=O)NC(C)C)ccc1Cl C1(C(=O)NC(C(C)F)C)CCC(C2CC2)N1C(c1cnns1)=O N1(C(C(OC)OC)=O)CCC(CNC(=O)C(=O)NC2CC2)C(C)C1 N1(C(C(=O)NCC=C)C2CC(C(=O)OCC)C2)CCCC1CC C1(N(CC(=O)Nc2ccsc2)C)CCCCCC1n1cccn1 c1(OC)c[nH]c(C(=O)N(CCC(C(C)C)NC(c2cccc(C)c2)=O)C)cc1=O C1(c2cn(CC3(O)CCN(C(C)(C)C)C3)nn2)CC2(C1)OCCO2 C(=O)(C1=NOCC1)N1CCC(CN(C(C(c2ccc(F)cc2)OC)=O)C2CC2)C1 c1(CNC(C(=O)NC)C)cc([N+](=O)[O-])c(O)cc1F.C12CC(O)CCN1C2=O C1(NC(c2c(C)n[nH]c2)=O)CCN(C(=O)CC(=O)OC(C)(C)C)CC1F c12ccc(cc1)-c1nnc(o1)SC(C)C2=O.C(C(=O)NCCNCC)=CC=CC Cc1onc(C(N2CCC23CN(C(C2CCC(=O)N2C)=O)C3)=O)c1[N+](=O)[O-] C1(CNC(CCCOC)=O)CN(C(c2ccc(C(=O)NC(C)C)[nH]2)=O)CCO1 c1(OC)cc(F)ccc1C(=O)NC1(CNC(=O)C(C)CC2CCC2)CC1 N1(C(C2(N(C(c3c(C)nco3)=O)C3CC3)CCC2)=O)CC(C)(C)OCC1C N1(C2CN(C(C(COC)O)=O)C2)CCN(C(=O)C=CC(C)(C)C)CC1 N1(C(COCCOCC)=O)C2CCC1CC(O)(CNC(c1cc(C)ns1)=O)C2 c1(CC)cn2c(n1)CCC(C(=O)NCC1CC(F)CN1C(C1CC1C)=O)C2 N1(C(C2CC2F)=O)CC2CCC(C1)N2Cc1ccc(Br)nc1Br c1(C(N2C(CCC)(C(=O)NC)CCC2)=O)cc2c(F)c(F)cc(F)c2[nH]1 c1(C(=O)NCC2OCC(CNC(=O)CC3CCC3)C2)ccc2ncnn2c1 c1(C(=O)NC2(C)CN(C(=O)C(Cl)=CCl)C2)cnc(S)n1-c1ccccc1 c1(CC(N2CCC(N(C(C(C(C)C)C)=O)C)CC2)=O)cc(Cl)cc2ccccc12 C1(CC)CCN(C(=O)CCOC(C)C)C1C(=O)NCc1cnn(CC)c1C c1(N(C2CCN(C(=O)Nc3ncc(CN)s3)CC2)C)ccccc1[N+](=O)[O-] c1(Oc2ccccc2)cccc(OCCCCCNC(C2C(C)C2C)=O)c1 C1(CC(N2CCN(C(C(Cc3ccc(C)cc3)C)=O)CC2)=O)CCC(C)(O)CC1 N1(CC=C)CCCN(C(=O)C(CO)NC(=O)CC2COCC(C)O2)CC1 c1(N2CCCC(CSC)C2)nc(N2CCCOC(CCO)C2)c2ccccc2n1 C1(N(C(=O)C(C)O)CC)CCN(C(c2[nH]ccc2Cc2cccnc2)=O)C1 C1(NC(c2c(C)nccn2)=O)CN(C(=O)Cn2nnnc2C(C)C)C2(CCC2)C1 C1(C(=O)NC2CN(C(c3c(NC)cncc3)=O)C(C)(C)C2)CC(C)(C)OC1(C)C c1(SC)cccc(C(=O)NC2CCOCC2NC(=O)C(C)(C)C(N)=O)c1[N+](=O)[O-] c1(C(=O)O)ccc(CNCc2c(I)ccnc2Cl)cc1Br N1(C(Cc2ccc(OC)nc2)=O)CCC2CCCC(C1)N2C(=O)C1=CC(C)(C)C1 N1(C(C(CC)N(C)C(C2CC2C#N)=O)=O)CCc2c(cnn2C)C1 N1(C(c2cc3c(nc2O)CCCC3)=O)CC2(CCOCC2)C2CCCC12 N#Cc1cc(C(N2CC3=C(C2)CN(C(=O)CCF)C3)=O)ccc1F C(CN=c1[nH]c2c(F)cccc2n1C)c1scc(CC)n1 CC1(C)CC(NC(=O)C2=CSCCO2)CCN(C(C2CCn3cnnc3C2)=O)C1 c1(SC(C)C)ccccc1C(=O)NCC1CN(C(=O)CC2(C3CC3)CC2)CC1C c1(C(=O)NCCC2(CNC(c3c(C)nc[nH]3)=O)CC2)cccc(=O)o1 N1(C(CCC(C)C)=O)C2CC1CN(C(=O)CNC(=O)COc1ccccc1)C2 N1(C(CC(CCC)O)=O)CCN(C(=O)Cc2ccon2)CC(O)C1 N1(C(C(C(C)C)n2cnnc2)=O)CCC(C)N(C(C2CC(C)(C(=O)O)C2)=O)CC1 CCCCC(C)C(=O)NCC(O)CN(C(=O)CC(F)(F)Br)C c1(NCC(CSC)OC)nc(N(C)CC2CCCCCC2)c2ncsc2n1 N1(C(C2C(CCOC)C2)=O)CCCC(C)(C)C1C(=O)Nc1ccc(C)nc1C C(=O)(C(C)SC(F)(F)F)NC(CN(C(C)=O)C(C)C)C1CCC1 N1(C(C2(C)CCNC2=O)=O)CCC2(CC1)CC2CNC(=O)C(F)(F)C(F)(F)F c1(C(=O)NCC2(CNC(CCN(C)CC)=O)CCCC2)cccc(CO)c1N O=C(C1CCCc2n[nH]cc21)NC1CN(C(c2coc(Br)n2)=O)C2CCCCC12 S(=O)(=O)(c1ccc(NCCCC2CCOC2)cc1Cl)N1CCC(CCC)(CO)C1 CC1(NC(c2ccccc2)=O)CCN(C(=O)CC2(O)COC(C)(C)C2)CC1 N1(C(c2c(F)cc(OC)cc2Cl)=O)CCc2[nH]nc(CNC(=O)C(C)(C)F)c2C1 C1(CNC(C=COCC)=O)CC2(CCOCC2)CN1C(c1cc(O)n(CC)n1)=O C(=O)(C(CC(C)C)ONC(C1CC(=O)NC1(C)C)=O)NC(CCC)CO c1(CC)nnc(C)cc1C(=O)NC(c1ccccc1)CNC(C1CC(C)(O)C1)=O c1(CC)ccc(O)c(C(=O)NCC2CN(C(C3CCCC3(F)F)=O)CC23CC3)c1 C1(CNC(CC(CC)(C)C)=O)CN(C(=O)C(O)CCC(C)C)CCC12CCC2 CCC(N)CCC(=O)Nc1cccc(Oc2cccnn2)c1 Cc1cc(C)c(C(=O)NCC(C)CNC(c2cn(C(C)(C)C)nc2C)=O)[nH]1 C(=O)(C(C)CC(F)(F)F)N1CCC(C#C)(C(=O)Nc2ccccc2OC)C1 C1(O)(CNC(C(C(C)SC)O)=O)CCN(C(=O)CC(=O)OC(C)(C)C)CC1 C1(CN(C(=O)CSCC(F)(F)F)C)CN(C(=O)CC2OCCCO2)CCO1 C(=O)(C1NCc2n[nH]cc21)NCC(CC(=O)OCC)c1ccccc1 C12(NC(c3ccnc(CO)c3)=O)CCCC1CN(C(c1ccc(F)c(F)c1)=O)C2 C1(C(=O)NC(CCC)C(=O)NCCOCCCO)CCCCC1(C)C CN1CCCC(C(C)(C)C(N2CCC(F)(CNC(c3cc(C(F)F)cs3)=O)C2)=O)C1 c1(OC)ccc(C)nc1C(=O)NC1(CO)CN(C(c2cc(C(F)F)[nH]n2)=O)C1 c1(NC(C2C(OC)CCCC2)=O)ccc(NC(=O)C(C(C)O)N(C)C)c(C)c1 Cc1nc(N)cnc1C(=O)NCC(C1CCCC1)NC(C1CC(=C2CC2)C1)=O C1(NC(c2cc[nH]c2)=O)CCCC2CN(C(C3(n4cnnn4)CC3)=O)CC12 C1(NC(c2nc(-c3cccnc3)cs2)=O)CCNCC1CO N1(C(CC(CC2CC2)NC(C2C3CCC(F)C23)=O)=O)CC2CC(O)CC1C2 c1(CNC(C2C3CN(c4c(OC)c(C)ncn4)CC32)=O)ccc2oc(C)nc2c1 CC(CC(=O)NCC1CCC(NC(=O)CCc2nc[nH]n2)CC1)C(F)(F)F N1(C(CC=CC)=O)CCC2(CO)CN(C(=O)CSc3ccc(O)cc3)CC2C1 c1(C(CNC(=NC)NCC2CCCC(C)(C)C2)(C)OC)ccc(F)c(F)c1 c1(C(N2CCCC(C)C2CCNC(C2(O)CCC2)=O)=O)noc2cc(F)ccc12 C1(C#N)(C(=O)NCC(CNC(CC(C)OC)=O)OC)CC(=O)C1 c1(N2C(CC#N)CN(C(=O)Cc3cc[nH]n3)CC2)ncc2cc(Br)cc(F)c2n1 C(=O)(C1=CC2CCCC12)NCC1(CNC(c2[nH]c(=NC)sc2)=O)CC1 Cc1ccc(C(=O)NC2(CF)CN(C(c3cc(C(F)F)nn3C)=O)C2)nc1C CCCC(C(O)C(=O)NCC(C)(C)CO)NC(C1(C)CCOCC1)=O N1(C(c2c(CC)nco2)=O)CCC(Cc2nc(C3CCCC3)no2)CC1 C(C(C)(C)CC(=O)O)NC(c1cnn(CC)c1-c1ccccc1)=O C12(NC(c3ccnnc3O)=O)CCCC1N(C(=O)C=CBr)CCC2 C(=O)(C1=CS(=O)CCC1)NCC(CN(C(c1c(NC(CC)=O)cccc1)=O)C)C N1(C(C(CCSC)O)=O)CCN(C(=O)C(C(C)C)Sc2cccs2)CC12CCC2 N1(C(C2N(CC)CC2)=O)CCC2(CCCC2NC(C2CCCC3CC23)=O)CC1 C1(CNC(CSCC#C)=O)N(C(C2CCC(=O)N2CCC)=O)CCC1(C)C C1(C(=O)NC2CCN(C(C=CC(C)(C)SC)=O)CC2)Cc2nccn2C1 CC(CNC(=O)CC1CC1(Cl)Cl)CN(C(=O)Cc1cnco1)C CN1C(=O)C(=O)N(CC(=O)NCc2ccnc(N3CCNCC3)n2)C1=O C1(C(N(C2CCSC2)C)=O)(CNC(C2CCC2)=O)CC2(CC2)C1 N1(C(CNC(c2cnc(CC)o2)=O)=O)C(C(N)=O)CCC1C c1(C(=O)NC(C2CCN(C(CS(CC)=O)=O)CC2)C)ccnc(F)c1F C(CCCCCNC(=O)CCc1cnn(C)c1)NC(C1C(CC)CCC1)=O c1(NC(C2C(NC(C(F)OC)=O)CCCCC2)=O)cccc2cccnc12 C1(CNC(CC(C)OC)=O)CC2(CO1)CN(C(=O)C(C)(F)c1ccccc1)C2 N#Cc1c(NC2CC3CN(C(C4CCC(N=[N+]=[N-])CC4)=O)CC23)ncnc1Cl N1(C(C2(C)CC2)=O)CCC2CCCN(C(c3c[nH]c(=O)c4ccnn34)=O)C2C1 N1(C(COCCCCC)=O)CCC(N(CCC)C(C2(C)CCOC2C)=O)CC1 c1(C(C(=O)N(CCC)CCNC(=O)CC2(OC)CCC2)C)c[nH]c2ccccc12 Cc1ccc(O)c(C(N2CCC(NC(=O)Cc3ccco3)CC2)=O)c1 C1(CN(C)C(C2CCCN2C(=O)Cc2cncs2)=O)CCCC2CC12 C(C(C)(C)Cc1ccccc1)SCCNC(CN(C(COCC)=O)C)=O N1(C(CC2C(CNC(C3CN(C(C)=O)C3)=O)C2)=O)CCOCC(C)(C)C1 C(C(C)(C)CNC(=O)CC1CC1(Cl)Cl)N(C(=O)Cn1ccc(C(F)F)n1)C N#Cc1ccc(Br)c(C(=O)NC2CCCC2NC(c2cnco2)=O)c1 c1(Cc2cn(-c3c4ccc(OC)cc4ncc3)nn2)nc2c(cc1C#N)COCC2 N1(C(c2cc(OC)nn2C)=O)CC(C2(NC(=O)Cn3cc(C(C)O)nn3)CC2)C1 c1(CC)c(C(=O)N(C)CC2CCCC2NC(C2CSCCS2)=O)ccn1C CC1CCC(CCNC(C2(CNC(=O)C(N)=O)CC3(CC3)C2)=O)CC1 N1(C(CC2(C)CCCO2)=O)CCC(C2(NC(=O)C(F)=CCCF)CC2)CC1 c1(OC)cc(OC)c(NC(=O)CCC(C2CCC2)NC(=O)C(=O)N)c(OC)c1 N#CC1(O)CC(C(=O)NCC2(N3CCNCC3)CCCC2)C1 C1(C(=O)NCCNC(C2CN(C(C3C(C)(CC)C3)=O)C2)=O)CC2(CC2)C1 CCCCC(CNC(C1CC1C#N)=O)NC(c1ccoc1CC(N)=O)=O Cc1c(C(=O)N(CC(C)(C)NC(=O)CC(C)C(F)F)C)cc(C(C)C)n1C c1(NCCC(C)(C)N(C)C)cc(=NCc2ccc(S(C)=O)cc2)[nH]cn1 N12CC(C1)NC(=O)C1(CC1)CNC2=O.C(C(F)F)OC(C)=O Cc1oncc1C(=O)N(CCCNC(=O)CN1CCC1)C(C)C N1(C(c2c(CC)cnn2C)C(=O)NCc2cccs2)CCCNC(=O)C1CC(C)C N1(CCOC)CC2CC1CN2C(=O)CNC(c1ccco1)=O C(C(=O)NC(C)CCO)(C1(O)CCC1)NC(C=CC(C)C)=O N#Cc1ccc(C(N2CC3CCC(NC(=O)CC(F)(F)F)(C3)C2)=O)c(O)n1 C(=O)(C#CC1CCCCO1)NCC1C(NC(c2ncc(C)cc2F)=O)CCC1 C(=O)(C(O)C(C)(C)C)N1C(CN(C)C(c2ncc(Br)cc2F)=O)CCCC1 CC(C)(O)C#CC(=O)NC(CNC(=O)C(C)(C)CC1CCOC1)CO N1(C(c2nc(C)n(C)c2)=O)CCCC(C)C1CNC(=O)C(F)OC(F)(F)F C1(CC=C)(NC(=O)Cn2ncnn2)CCN(C(=O)CSc2ccc(C)cc2)CC1 C12CC=CCC1C(=O)N2CC(C)(C)C.C(C(C)C(=O)OC(C)(C)C)OCC CC(C)C(C(=O)NOCC(F)(F)F)NC(=O)CCCCC1CC1 N1(C(C=NOC)=O)CCC2(CC1)CN(C(c1conc1C1CC1C)=O)CCO2 CC1(C)CN(C(=O)C2=CCCO2)CCC1NC(=O)C(C)(C)C1CCOC1 C1(NC(=O)NCC(C(=O)OC)OCCOCCCOC2CC2)CCCNS1(=O)=O N#Cc1cc(Br)ccc1C(=O)NC1CCN(C(C23CCCC2C3)=O)C1 C(=O)(CC(C)(C)CC(=O)N1CCC2C1CCCN2C(=O)Cn1ccnc1C)OC N1(C(CNC(N)=O)=O)CCC2CCN(C(=O)Cn3c(-c4cccs4)nnc3S)C2C1 n1(CC(=O)N(CCOCC=C)C)ncc(C#N)c1N C(N=c1[nH]c2c(c(=NC(C)C3CCOCC3)[nH]1)COCC2)C1(CC(C)C)CC1 c1(CC)nc(C)c(C(=O)N(CCCNC(c2ccncc2C)=O)C2CC2)s1 N1(C(C(C(C)C)O)=O)CC2CC1CN2Cc1cccc(-c2cncnc2)c1 C#CC(C)(C)C(=O)NCC(C1CC1)N(C(=O)C(C1CCOCC1)O)C C1(N(C)C(c2cnn[nH]2)=O)CCN(S(=O)(=O)Cc2ccccc2)CC1 CC(C)(C)C(C(=O)NCN)NC(c1ccncc1-n1cccn1)=O C(=O)(C(C)(F)C(C)(C)F)N1CCN(C(CCCCC)=O)C(CC(=O)NC)C1 C1(C(N2CCC(C)(NC(=O)C(=O)N=S(C)(C)=O)C2)=O)CCCN(S(N)(=O)=O)C1 c1(C(=O)NC(C)CCCNC(C2(c3cccnc3)CCC2)=O)ccncc1F O=C(O)C(CNc1ccccc1Cl)C(=O)N1CCCC1CC(F)F CC1CN(C(=O)CCCNC(C2CC=CCC2)=O)CC1NC(=O)C(C)CO n1(CCNC(=NCC)NCC2CCS(=O)(=O)C(C)(C)C2)c(=O)oc2ccccc12 C1(CC(=O)NC(C(CC)C)=O)CN(C(=O)CN(CCO)CCO)CCS1 C1(C(=O)NC(C)CCN(C)C(c2cncc(N)c2)=O)CCS(=O)(=O)C1(C)C c1(C(N(CC(C)NC(=O)C(C)(c2ccccc2)N(C)C)C)=O)cncn1C C(C)(CCCCNC(=O)Cc1cn(C)nc1C)NC(COCC#C)=O CC1C(NC(=O)C(C)(C)CC(F)F)C2CCN1CC2 N1(C(CN(CC)CC)=O)CC(CC(=O)N(C)CC2CN(C)C2)C(C)C1 C1(CNC(=O)C2=CCCCCC2)CN(c2ccncc2C#N)CCC12CCOC2 O=C(CC1C2CCCC2N1C(=O)CC1CCCNC1=O)N1Cc2ccccc2CO1 CC(C)C(C#N)C(=O)NC1C=CC(CNC(c2cnn(CCO)c2)=O)C1 C(=O)(C(C)C(C)COC)NCc1c(C(N(CC(=C)C)CC(=C)C)=O)cccn1 CCC(C)C(C)C(=O)N1CCC(C)(CNC(c2cc(Cl)ccc2N)=O)CC1 C1(N)CC2CC(C1)N(C(=O)C=CC=C(Cl)Cl)C2.CCCCCC=CCC=O c1(CN(C)C(=O)NCC2CCN(c3nc(Cl)ncc3F)C2)ccc(F)c(F)c1 CCC(CCC(C)C)NCC(O)COc1ccccc1Br Cc1ccc(CCC(=O)NC23CC2CN(C(=O)Cc2cccnc2O)C3)cc1 O=C(C1CCCc2nnnn21)NC1CCOC2(CCC2)C1 C(=O)(C(C(C)(C)C)NC(c1cc(OC)cc(F)c1)=O)N1C(C)(C(=O)OC)CCC1 C(CC(C)C(=O)N1CCCC1(C)CCC(=O)NCC1(C)CCCC1)=CC CN1C(=O)CCCC1C(=O)NC1CCCCN(C(=O)C(C)(C)c2ccno2)C1 c1(C(=O)NC(CC)CNC(c2cccnc2O)=O)ccc2c(c1)CC(C)O2 c1(NC(CCN(C)Cc2cccc(NC)n2)=O)ccc(C#N)c(Cl)c1 C1(C)(C(=O)NCCC(C)N(C(c2cnc(OC)nc2)=O)C)CCCNC1=O C(C(C(C)C)NC(=O)C(F)(F)c1ccccc1)NC(CSCC#C)=O C1(C(C)C)COCCN1C(C1(CN(C)C)CCCN1)=O C1(NC(c2c(C)cco2)=O)CCCCC1NC(=O)C(=O)N(C)C c1(CCNC(C(=O)Nc2cccc(-c3ccsc3)c2)=O)ncc(F)cc1F CC1(C)CC(CO)CN(CC(=O)Nc2cnc(Cl)c(F)c2)C1 C1(CNC(C(CSC)C)=O)CC2(CC2)CN1C(c1c[nH]c(C)cc1=O)=O CCC(CNC(c1ccsn1)=O)(CC)NC(C1CCN(C2CCCC2)CC1)=O C1(F)(CNC(C(c2ccccc2)OC)=O)CCN(C(=O)C(C)(F)F)CC1 CCC(CC(=O)N1CCC1Cn1cc(C2CC23CC3)nn1)C(F)F N1(C(CCC)=O)CCC(OCCNC(=O)C(OC)OC2CC2)C1 C1(C(N(CC(=O)NOC(COC)COC)CC#C)=O)CCOC(C)C1 C=CCC(C(=O)NC1CCC(NC(=O)C(CO)NC(=O)CCC)C1)C(C)C C(=O)(C#CC(C)(C)C)N1CC(C(C)NC(c2csc(-c3ccccc3)n2)=O)C1 Cc1cc(=NCC(C)NC(=O)C(=O)Cc2cccs2)[nH]c(C(C)(C)C)n1 C(C)(C)(C(=O)NCc1cn(CC(C)NC(=O)C(=O)N(C)C)nn1)OC(C)C c1(CNC(C(=O)Nc2ccc(C)c(Cl)c2F)=O)sc(Br)c2c1OCCO2 n1(CCC=C)cc(C2CCCN2CCC2CCC2)nn1 C1(OC)CC(CNC(=O)C(C(C)C)n2cnnn2)N(C(=O)CC2CCOCC2)C1 c1(NC(CCCCCCn2cc(C(C)OC)nn2)=O)ccc(S(C)(=O)=O)c(C)c1 c1(C(N2CC(C)C(NC(C3(O)CC3(C)C)=O)C2)=O)coc2c1N(C)C(=O)CCC2 N1(C(CCC)=O)CC(O)C(O)C1CNC(=O)CC1CCN(C)C1=O C1(C(N(C)CC2CCN(C)C2)=O)C2CC1N(C(=O)CC1CCCN1C)C2 C(=O)(C1=Cc2ccccc2C1O)NCC1(NC(C2=CCC(C)CC2)=O)CCCC1 N1(C(=O)C=CSc2cccs2)CCOCC(CNC(C2CC(OC3CC3)C2)=O)C1 CCC(CO)C(=O)NCCCCC(C)NC(c1scnc1C1CCCC1)=O C1(NC(c2cscc2Br)=O)CN(C(=O)CCn2cccn2)C2(CCC2)C1 C1(CCOC)CN(C(c2sc(=N)[nH]c2C)=O)CCN1C(c1ccn(C)n1)=O C(CCF)(C(=O)NCCNC(=O)C(C)C)NC(c1c(CC)c[nH]c1)=O N1(C(C)=O)CCC2(C1)CN(C(=O)CC1COc3ccccc31)C2.C=O N1(C(C2C(=C)C2)=O)CCCC(C2(NC(C3CC(O)C3)=O)CC2)C1 N1(C(c2nocc2C)C(=O)NCCCCCC)CCc2c(Cl)cccc21 N1(C(C2(C)C(C(=O)OC)C2)=O)CCC2(CC1)CC(NC(=O)CCCC(C)C)C2 C(=O)(CCCCC(F)F)N1CCC(CCNC(=O)CSCC2CCCCO2)C1 CCC(CC(F)(F)F)C(=O)N(C(C)CNC(=O)C(F)C(C)(C)O)C N1(C(C(CC)CCc2ccccc2)=O)CC2CCC1CN2C(=O)C1=CC(C)(C)C1 N1(C(c2n(C)c(O)nc2)=O)CC2CN(C(C3CC3C#N)=O)CCC2(CO)C1 C1(C#N)(C(N(CCNC(=O)C(c2cccc(OC)c2)(F)F)CC)=O)CCCCC1 C(=O)(CC(C=C)CC)NC1(CC=C)CCN(C(c2nccnc2Cl)=O)C1 c1(CN=C(NC(C=C)C)NC2CC2C2CC2)cc(OCC)c(O)cc1C O=C(C1=CC2(CCN(C(=O)CCNC(N)=O)C2)C1)N1CCC(C2CC2)C1 CN1CCc2cc(C(=O)NCC3CC(NC(=O)C4=CCCC4)C3(C)C)ccc21 C1(CC)CC(O)(CNC(C2(NC(=O)CCOCC(C)(C)C)CCC2)=O)C1 C(=O)(CC(CNC(c1ccc(F)c(F)c1C)=O)C(C)C)OC C(=O)(C#CC1CCOC1)NCCC(C)NC(c1c(C)oc(Br)c1)=O N1(C(CC(C=C)(C)O)=O)CCC(O)(C2(NC(c3cnccn3)=O)CC2)CC1 C12(CNC(CN3C(C)CC3)=O)CCC(CC1)CN2C(=O)C(O)CCn1cncn1 c1(C(N2CC3(C2)CN(C(c2csc(-c4ncc[nH]4)n2)=O)C3)=O)ncc(Cl)cc1Cl C1(CNC(c2c(CC)occ2)=O)CC(NC(c2c(Br)cnn2CC)=O)CC1O c1(C(N2CCCC(C)(CNC(C(C)C3CC3)=O)C2)=O)cc(C#N)ccc1F c1(C(=O)NCC2C(NC(CCN(C)CC)=O)CC2)noc2ccc(OC)cc12 c1(CC)ccc(O)c(C(=O)NCCN(C(C2CCSC(C)C2)=O)CC)c1 C(c1c(Cl)cccc1Cl)=CC(=O)NC1C(F)CCN(C(CCOCCOC)=O)C1 c1(C(N(C2CCN(C(=O)CSC(F)(F)F)C2)C)=O)cc(C(N)=O)ccn1 C(N=c1[nH]c(N2CCOC(C(C)C)C2)nc2cc[nH]c12)C1CC(NC)C1 C(=O)(C(C)C(CC)CC)N1CCC(N(C(c2nc(CC)oc2)=O)CC)C1 c1(C2N(C(=O)NCCc3cc(=N)[nH]o3)CCC2)ccc(Br)cn1 N1(C(NOC(C)(C)C)=O)CCCC(C(=O)NC2(C)C(NC(=O)C3CC3)CC2)C1 N1(C(CCOC)=O)C2CCC1C(CNC(=O)Cc1cccc(NC(C)=O)c1)C2 c1(C(=O)NCCN(CCOC)C(C2CCOC2)=O)ccc(Cn2cccn2)cc1 N1(C(C(C2CC2)OC)=O)CCCC1C=CC(=O)NC(CC)C(C)CN(C)C C(=O)(C1c2c[nH]nc2CN1C(c1cnc(=N)[nH]c1)=O)NCC(C(=O)NC)(C)C c1(COC)nc(OC)cc(N2CCC(F)(C(=O)OC(C)(C)C)C2)n1 C1(NC(C(C)=CC2CC2)=O)CCSC12CN(C(C13CCC(F)C1CC3)=O)C2 C(CN=c1[nH]n(C)cc1[N+](=O)[O-])(C(C)(C)C)NC(CCc1cnn(C)n1)=O c1(C(=O)NCCC(C)(C)NC(c2occ(C)c2)=O)cc2n(n1)CC(F)C2 n1(C(C(=O)NCC)C)cc(CN(C)C(C2(NC(=O)C(CC)OC)CC2)=O)nn1 c1(C(N(CC(C)N(C(=O)CC(=O)c2cnn(C)c2)C)C)=O)ccc(O)cn1 N1(C(c2cc(SC)oc2)=O)CCSCC1CCNC(=O)CC1CCCO1 CN1CC(NC(C2(NC(c3cc(=N)[nH][nH]3)=O)CC2(C)C)=O)C(=O)N1 C1(OC)(NC(=O)Cc2cccc3c2OCO3)COC(C)(C)OC1 C1(C(C)O)CCCCN1C(C1C2CN(C(=O)CC3CCNC3=O)CC12)=O Cc1cc(C(C)C(=O)NCC2CN(C)CCN2C(C2CCCCS2)=O)cc(F)c1 C1(NC(CCOCCCOC)=O)CCCCC1C(=O)NCCCCC1CC1C c1(C(=O)NC2CCC(CNC(C3CCCOCC3)=O)C2)cc2cccnc2[nH]1 Cc1cc(Cl)cc(C(=O)NCCN2CCN(C(c3cc(=O)n(C)o3)=O)CC2)c1O CC(=O)CCCC(=O)NC1CC(F)CN(C(=O)CCN2CCN(C)CC2)C1 N12CCC(O)(CC1)C(=O)N1CCC(CC1)C2=O.N1(CC)CCCC(C(F)(F)F)C1 CCC(CC)C(C)C(=O)N1CC(O)CC1CNC(=O)C(C)=CC1CC1 N1(C(C2N(C(C3CCN(OC)CC3)=O)CC2)=O)CC2CCCC2C12CC2 N1(C(CC=CCC)=O)C(C(=O)NCc2ccns2)CC1C C1(NC(CSCC#C)=O)CCC(CCNC(=O)C(C)SCOC)C1 N1(C(C(c2ccccc2)=O)=O)CC(NC(c2nn[nH]c2Cl)=O)CC2(CCOCC2)C1 C1(NC(C(c2ccoc2)NC(C(CO)OC)=O)=O)CC(=O)N(C(C)C)C1 CCC(N=c1nc(N2CCC(C(=O)NC)C2)c2sccc2[nH]1)c1ccncc1 c1(C(=O)NC2(CN(C(CC3(CSC)CC3)=O)C)CC2)nccc(C)c1N N1(C(C(C)S(C)(=O)=O)=O)CC2CCN(C(=O)C(C)(Cl)Cl)CC(C2)C1 C1(NC(CCC(CC)C)=O)CCCC12CN(C(c1cc(O)ncn1)=O)C2 N1(C(CCSCC)=O)CCC(C)(C)C(C(=O)NC(c2ccco2)CO)C1 N1(C(=O)NC(c2cc(Cl)ccc2Cl)C)CCNCC2(C)CCCC12 C1(CN(C(=O)COC2CCC2)C)CCCCN1C(=O)C(F)(F)c1ccsc1Cl C1(CNC(C(=Cc2ccncc2)C)=O)CCN(C(=O)C(C)OC(C)(C)C)C(C)C1 CCCCCC(O)C(=O)NC12CC(C(=O)NC3CCCC4(C3)N=N4)(C1)C2 CC(CCNC(=O)C(C)c1ccsn1)NC(=O)CCn1cccn1 C1(C)(COC)CN(CC(C2CCC(F)(F)CC2)C)CCO1 c1(C(=O)NCC(CNC(C(C)n2cccn2)=O)O)cc2c(o1)CCCNC2=O c1(NC(c2c(NC(C(c3ccc(F)c(F)c3)C)=O)c[nH]n2)=O)ccc(Br)cc1Cl n1(CC=C)cc(CNC(=O)COC(C)(C)CNC(c2csnc2Cl)=O)nn1 c1(C(=O)NCCN(C(C(CC)F)=O)CCOCCO)oc(C)nc1C Cc1cc(N)ccc1C(=O)NCC(C)(C)CN(C)C(C1CCN1C)=O c1(C(N2CC(CCNC(=O)C(O)Cn3cncn3)(OC)C2)=O)cncc(N)n1 C12(C(N3CC(C)N(C(=O)CC45CNC(=O)C(C4)C5)CC3)=O)CCCCC1C2(F)F C(=O)(C(C(C)(C)C)C(=O)N1CC(O)CO1)N1CCC(C)CC1 C(=O)(C(C)CC(C)(C)C)NCCC(C)(C)NC(CSc1ccc(C)cc1)=O N1(C(c2scc(-c3ccc(C)cn3)n2)=O)CCc2nc[nH]c2C1 CC(N=c1ccnc(NC(c2cc(F)c(F)c(F)c2)CO)[nH]1)c1ccc(O)nc1 Cc1nc2oc1NC(=O)N1CCCC2C1.C1(C(N)=O)CN(C2CC2)CC1C CC(CC(=O)NC(=O)C(F)(F)F)NC(C1CSCN1C(=O)C(C)(C)C)=O C1(CCNC(c2c(OC)nsc2)=O)CCCN(C(C2CC(C#N)(OC)C2)=O)C1 N1(C(c2ccn(C)n2)=O)CCC(CNC(=O)C(F)CC2CCC2)CC1 C1(C(N2C3CN(C(CCC(C)SC)=O)C(C3)C2)=O)Cc2ccccc2C1 CC1CCCC1C(N1CC(CCNC(c2cnc(O)o2)=O)C1)=O C1(n2cccc2)(C(=O)NCC2C(NC(=O)Cc3ccco3)CCC2)CCCC1 N1(C(C23CC(C2)C3)=O)CC2CN(c3nnc(CO)s3)CC2C1 N1(C(C)C)CCN(C(=O)NCC(C2CCOCC2)F)CC1C C1(CC(N2CC(C(=O)NCC)C2)=O)CCCCC1NC(c1cn(C)c(C)n1)=O N1(C(c2c[nH]c(=N)s2)=O)CC2(CCCCN(C(c3cc4ncccc4s3)=O)C2)C1 C(=O)(C(=O)N=c1nc(CS(C)(=O)=O)[nH]o1)OC(Cc1ccc(OC)cc1)C C1(NC(c2c(C)nc[nH]2)=O)CN(C(c2ncccc2C2CC2)=O)CC1(C)C Cc1cc(-n2cc(C3CCCCN3C(=O)CN3CCOC3=O)nn2)cc(C)c1Br S(=O)(=O)(c1cccc2nsnc12)NC1CCN(CCN(C)Cc2cccnc2)C1 c1(C(C2CCC2)N(C(=O)CCn2cc(C3CC3)nn2)C)cc(P(C)(C)=O)cs1 c1(CC(=O)NCC(CNC(C2CCN(CCC)CC2)=O)O)nsc2ccccc12 N1(C(CN(C2CCC2)C)=O)CCC2(CC1)CC2C(=O)NCCC(O)C(F)(F)F c1(CN=C(NC(C=C)CC)NC2CC(=O)N(CCC)C2)cc(Cl)ccc1N(C)C N(C(=NCCc1cc(OC)ccc1C)NC1CCCC(F)(F)C1)C(COC)C c1(C(=O)NCC2CCCCN2C(=O)CCCCCF)ccn2cncc2c1 c1(NC(c2cnn(C)n2)=O)cncc(CNC2COCCO2)c1 N1(C(COCC(C)C)=O)CCCCC(N(C)C(C2CN(C(C)C)C2)=O)C1 C1(NC(c2cnc(C3CCCC3)s2)=O)CCCCN(CCCC2CCOC2)C1 N1(C(C(CSC)OC)=O)CC(C2CCCCN(C(c3ccc(Cl)c(F)c3)=O)C2)C1 CN1CCCC1(C)C(=O)NCC(c1ccccc1OCc1ccccc1)N(C)C C1(CNC(C2CCCCO2)=O)CC12CCN(C(c1cc(F)n[nH]1)=O)CC2 c1(C(=O)NCC2N(C(C(CC)Oc3ccccc3)=O)CCC2)cnc(N)cn1 c1(C(N(C)CC2(CNC(c3c(C)cccn3)=O)CC2)=O)ccc2nncn2c1 Cc1nc(C)c(CC(=O)NC2C=CCN(C(=O)CC3(O)CCOC3)C2)s1 CC1(C)CN(C(C2(O)CCCCCC2)=O)CC(C)(C)S1(=O)=O S(=O)(=O)(c1ccc(F)c(Cl)c1)N1CC(F)CC(Nc2ncc(N(C)C)cn2)C1 C1(CC(C)NC(CC=C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1 c1(C(N(CCN(C(=O)COC(F)(F)F)CC)CC)=O)ccc(C)c(O)n1 c1(C(=O)NC2CCc3n(C)ncc3C2)cc2cc3c(cc2[nH]1)OC(F)(F)O3 C(=O)(CC1C(=O)Nc2c(F)cccc21)NC(CN(C(c1csc(C)n1)=O)CC)C c1(C(=O)NC(CNC(c2c(C)coc2)=O)CO)ccc(-c2nnc(O)o2)cc1 C1(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CC2CCC(C1)N2c1ncnn2cccc12 C12(CNC(CCCCC)=O)CCCCC1N(C(c1cccnc1F)=O)CC2 Cc1csc2c(CC(N3CCCC3C(=O)N(C)C3CC3)=O)cccc12 N1(C(C(C)OCCCC)=O)CCC2CN(C(c3cc(C#N)ccc3F)=O)C(C)C12 c1(CC)ccc(OCC(=O)NCC(C)N(C(=O)CC2CCC23CCC3)C)cc1 C(=O)(CCCCCF)N1CC(CNC(c2ccc(CCCC)cc2)=O)C(O)C1 Cc1ccncc1C(N1CC(NC(c2cccnc2O)=O)C(C)C1)=O C1(CNC(C=CC)=O)COCC1NC(=O)CSc1nncn1C(C)C Cc1cc(C(=O)NC2CCN(C(=O)CCn3cccn3)C(C)C2)ncc1Br C1(F)(CN2CC(C)(OC)C2)CCC(NC(=O)CC(=O)N(C(=O)CCS(C)=O)C2CC2)C1 C1(NC(CNC(=O)OC)=O)CCOC(C(=O)NCC2CC(N(C)C)C2)C1 CC1CN(C(=O)CN(C)C2CC2)CCN(C(=O)C(c2ccccc2)C)C1 N1(C(Cc2c(OC)nccc2)=O)CCC(NC(=O)Cc2csc(C)n2)C(F)C1 N1(C(CCCCC)=O)CCCOC(CNC(c2n[nH]cc2Br)=O)C1 N1(c2nc(C)nc3c2cc[nH]3)CCC2(CN(C(C3CCCC3O)=O)CC(C)O2)C1 C(CN=C(NCC1CC1)NC1CCC(C)(C(C)C)CC1)C1CCC(OC)CC1 C(=O)(C1Cc2ccc(F)cc21)NC1(C2N(C(C3C(C)C3C)=O)CCC2)CC1 C1(NC(CCCN(C)C)=O)CN(C(c2c(Cl)ccc(O)c2N)=O)CC2(CCC2)C1 c1(C(N2C(CNC(c3cnc(Br)s3)=O)CCC2)=O)nc2ncccn2n1 c1(C(=O)NC(CC=C)CNC(=O)C(C)CN(C)C)cc2nccnc2[nH]1 c1(C(=O)NCC(CC)(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)ccc(C)c(Cl)c1F N1(C(CC(C)NC(c2ccn(CCC)n2)=O)=O)CC(=O)NC(=O)C1C c1(OC)ccc([N+](=O)[O-])c(C(N2CC3C(NC(=O)CCC#N)C3C2)=O)c1 CC1(C(=O)NC(CNC(C2CCCN2N=O)=O)C2CCC2)CS(=O)(=O)C1 C1(C(C(=O)N(CC=C)C)C)CCCN(C(C2CN(C(C)=O)C2)=O)C1 c1(CN2CC(NC(C3Cc4ccccc4O3)=O)C(F)C2)c[nH]c2ncc(Br)cc12 CC1CCC(CNC(=O)C(C)(C)C(F)F)CN1C(c1coc(C#N)c1)=O C1(NC(CC2(C)CC2(F)F)=O)CCN(C(c2ccncc2N)=O)C1C1CC1 C(=O)(C(C)CCC(C)(C)C)NCC1(CNC(CSCC#C)=O)CCC1 CC1CC(NC(C2CCC3(CC2)CC3)=O)CCN1C(=O)COC1(C)CCCC1 C1(CC=C)(C(=O)NC2CCC2NC(C)=O)CN(C(=O)CCCOC(C)=O)C1 Cc1cccc(C)c1C(=O)NC1CC2(C1)CC2NC(=O)CC1(C)CC(F)(F)C1 C1(N(C(C2(COC)CCCC2)=O)CC)CCCN(C(c2cc(F)ccc2F)=O)CC1 c1(OC)ccc(C(=O)NCCOCCS(C)(=O)=O)c(Br)c1F c1(N2CCC(CC=C)(NC(=O)CC3COC(C)(C)C3)C2)cc(C)nc(COC)n1 C1(NC(C2C(C(=O)OC)C=C2)=O)CC2(CCC2)C1OC C1(CN2CCC(NC(c3c(C(=O)OC)c(C)[nH]n3)=O)C2)CCC(F)(F)CC1 CC1(C)OCc2c1n[nH]c2C(=O)NC1CC(NC(c2cnc(S)nc2)=O)C1 N1(C(CCC2CC(C)C2)=O)CCC(CC(=O)Nc2cc(CO)cc(F)c2)C1(C)C C1(OC(C(CC)Oc2ccccc2)=O)CCCCC1n1cc(C(=O)O)nn1 C#Cc1ccnc(C(=O)NCCN(C(=O)CCc2nncs2)CC(C)O)c1 N1(C(c2c(C)csc2Cl)=O)CCOCC(NC(=O)C(C)(C)C)C1 C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)CN2C(=O)CCC2=O)C1 c1(C(=O)NCCc2c(CNC(CC3C(C)OCC3)=O)nco2)c(F)ccc(F)c1Cl C1(CNC(CC(CC)C2CC2)=O)CCC2(CN(C(c3cc(CC(C)C)c[nH]3)=O)C2)O1 CC1(C)CC=C(C(=O)NC23CCC2CN(C(c2ocnc2C2CC2)=O)C3)CC1 C(CCCCN(C)C(C12CCC1CC2)=O)NC(CC=CCC)=O CC(C)(O)CC(=O)NC(Cc1ccco1)C(N1CC2CCC1C2)=O C1(F)(C(N2CCC(OCC(C)C)C2)=O)CCCN(C(=O)CC2COCC(C)O2)C1 N1(C(C(c2cccc(C)c2)C)=O)CC2(CNC(c3c[nH]nc3C)=O)CC(F)(C1)C2 c1(OC)cc(C)cnc1C(N1CCCC(CNC(=O)C(O)CSC)CC1)=O C1(NC(C(C)N(C(=O)Cc2ccns2)CC)=O)CCCC2(CC1)CC2 N1(C(C2CCCCN2Cc2cccnc2)=O)CCC(C2CCOC2)CC1 C(=O)(C1=NN(c2ccccc2)C(C(=O)NCc2coc(C)n2)C1)OC C(=O)(C(C)(F)C(C)(C)F)N1CCC(C2NCCCC2)C1.c1(CC)c(F)ccnc1F C(=O)(C(C)CCCC(C)C)NC(C(C)OC)CC(N1CCOCC(C)(O)C1)=O Cc1ccc(CNC(=O)COC2CN(C(c3ncccc3N)=O)C2)c(F)c1 CCC(C)(CNC(=O)CCOCCOC)C(=O)NCc1cc(C)nn1C CCCC(C)(CC)C(=O)N1CC(C)C(C)(CNC(=O)CCCc2ccccc2)C1 N1(C(C=CC(=O)N(C)C)=O)CC(F)(F)CC1CO.c12cc(no1)C(=O)NC2 c1(C(=O)NCC=C)ccc(C(N2CC(NC(c3ccc(C)o3)=O)C(C)C2)=O)cc1 CN1CC=CCC1CC(=O)NCCN(C(C1(CF)CC1(F)F)=O)C1CC1 c1(C(N2CCC(CNC(C(COC)OC)=O)CC2C)=O)ccc2ccccc2c1 C=CCC(CC=C)NC(C)(COCc1cccc(Br)c1)c1nnnn1C1CC1 CCCC(C)(O)CC(=O)NC12CCCC1N(C(c1cnc(C(C)C)s1)=O)CC2 C(=O)(C1=COCCO1)NCCCN(C(=O)CCc1c(F)cccc1F)C C1(C(N2CC(OC)(CNC(C3(C)CCCN3C)=O)C2)=O)CCCCCC(=O)C1 C1(C(N2C(C)CCN(C(c3c(C)cc[nH]c3=N)=O)CC2)=O)CC2CCC(C1)N2C Cc1nnc(CC(=O)NC(C)(CNC(=O)C(F)(F)c2cnn(C)c2)CO)o1 c1(C(C)C)ccc(C(=O)NCC2CC2CNC(C2CC(n3cnnc3)C2)=O)s1 N1(C(CSC)=O)CCN(C(=O)C(=O)N(C)C)C(c2ccccc2)C1 C(CC(C)C(=O)NC(C1CCN(C(=O)CCc2cccnc2F)C1)(C)C)OC c1(C(N2CC3(CC(NC(C4CCC5(CCC5)C4)=O)C3)C2)=O)cnc2n1CCOC2 Cc1cc(O)c(C(N2CC(N(C(=O)CN3C(=O)CCC3=O)C)C2)=O)nn1 C1(=O)N=C2N=CN(N2)CCC(=O)N(Cc2ccccc2)C(C)CN1C.N(C)C.N(C)C c1(C(N(CCNC(=O)COCCSC)CC)=O)ccc(-n2ccnn2)cc1 C1(NC(CC(CC)(C)C)=O)CN(C(c2cc(C(F)F)ncn2)=O)CC12CCC2 C1(C(=O)N(C)CCNC(=O)Cc2ccc(NC(C)=O)cc2)(COC)CCC(=O)N1 C=C1CCN(C(=O)C(C)C(F)F)C(C(=O)N(C)Cc2nccs2)C1 c1(C(=O)NCC2N(C(C=C3CCN(C)CC3)=O)CC=C2)csc2nccn12 c1(CCC)nc(C)c(C(N2CCCC2C2(NC(c3cnn(C)n3)=O)CC2)=O)o1 c1(C(=O)NCC(C)CN(C)C(c2ncc(F)cn2)=O)ccc(N)c(Br)n1 C1(CNC2(C)CCOCC2)CN(CCSc2ccccc2)CCCO1 C(N=c1nc2sccc2c(NCC23CCCN2CCC3)[nH]1)C1COCC(C)(C)O1 C1(C(C)C)C(=O)N1.c1(OC)cc(C(=O)NC(CC2CCC2)CO)on1 c1(C(=O)NC(C(C)NC(c2c(C)con2)=O)CO)cnn(-c2ccccn2)c1C C1(NC(C2N(C)C(=O)CCC2)=O)CCC2CCN(C(C3(n4ccnn4)CC3)=O)C12 C1(NC(C(=O)NC2(c3cccc(C)c3)CCCC2)=O)CCCNCCC1(F)F N1(C(c2cccc(-c3cnco3)c2)C(=O)NC(CC)C)CCC2(CCCOC2)C1 CC1(C)CC(CNC(C2C=CCCN2C(=O)CCc2csnn2)=O)CC1 c1(C(N2C3CN(C(CC(C)=C(C)C)=O)C(C3)C2)=O)cc2ccc(N(C)C)cc2[nH]1 c1(OC)ccc(N)c(C(=O)NC2C3CC2CN(C(C2CC4CC4C2)=O)C3)c1 N1(C(=O)NCCC2C(C)C(=O)CC2)CCCC2(C1)OCCCO2 C(=O)(C(F)CC(C)(C)C)NCc1cc(C(N2CCCC(C=C)C2)=O)sc1 Cc1cc2ncnc(N3CC4C(CNC(c5ccccc5COC)=O)C4C3)c2[nH]1 c1(C(=O)NCCN(CCOC)C(C2CCCCC2OC)=O)c(C)cncc1C N1(C(c2c(NC)cnc(Cl)c2)=O)CCC(NC(=O)C(CCC)N(C)C)C12CCC2 c1(OC)nccc(C(=O)NCCCCN(C)C(c2sccc2CC#N)=O)c1F N#Cc1c(F)cc(C(=O)NCC2(NC(c3cnc(O)o3)=O)CC2)cc1F C1(C(=O)NCC(CC(C)C)OC)CCCN(C(C2C3CCC(F)C23)=O)CC1 c1(C(=O)NCC(CC)(C)NC(C2CC(C(=O)OC)C2)=O)ccc(Cl)cn1 C(C1(C)CCOCC1)=CC(=O)NCC(C)CNc1ncc(Br)cn1 c1(N2CCCC(C(C)NC(Cc3c(CC)cccc3)=O)C2)nc(C)ncc1F CN(C)S(=O)(=O)NCC(N1CC=CC(NC(C2CC2c2ccccc2)=O)C1)=O CCCCC(CNC(c1cc(C2CC2)ncn1)=O)NC(c1cc(CC)c[nH]1)=O C(=O)(C1CCCc2ccccc21)N1C(C)CCC(NC(c2c(CC)cco2)=O)C1 C1(CC=C)(NC(=O)C=CC(C)(C)C)CCN(C(=O)CCS(N)(=O)=O)CC1 c1(N(C)Cc2cccc(F)c2F)nc(N2CCCCCCCC2)c2c(n1)COC2 C1(NC(COCC=C)=O)CCN(C(=O)CN2CC(=O)NC2=O)C(C2CC2)C1 c1(N(C)CC2CCCN2C(=O)C#CC2(C(F)(F)F)CC2)ncc(C#N)cc1F N1(C(C2(COC)CC2(F)F)=O)CCC(F)(CNC(c2cccnc2C)=O)CC1 C1(NC(C(C)(N(C(c2c(C)cns2)=O)C)C2CC2)=O)CCCCC1(F)F Cc1cc(C(N2CCCC(CN(C)C(C3CCCSS3)=O)C2)=O)cc(C)c1 Cc1c(C(N2CC3(CCC3NC(c3sccc3F)=O)C2)=O)cncc1Br N1(C(c2cnc(C)o2)=O)CCC(NC(=O)C(C)(O)c2ccccc2)C(F)C1 Cc1cc(C(=O)NCC(Cc2ccccc2)NC(=O)C=CCO)cn1C(C)C C12(CCSCC1)n1nnnc1C2NCC1(CC)CC1.c1(C2CC2)ccc(F)cn1 Cc1cc(O)ccc1CC(N1CC2CC2(NC(=O)CC(C)NC(=O)C2CC2)C1)=O C1(C(=O)NC2(CO)CC2)CC2(CC2)CN1C(=O)CC1CCCOC1 N1(C(Cc2cnc(C)[nH]2)=O)CC(CNC(c2ccc(Cl)c(N)c2)=O)C(C)(C)C1 CCCCCCCCC(=O)N1CC=C(CNC(C2CN3CCCC2CC3)=O)CC1 N1(C(C(C)CN(C)C)=O)CCCCCC(NC(=O)COCC2CCCC2)C1 C1(CC(=O)OC)CCCN(C(N2CCC3(CC2)CC3)=O)CC1 c1(C(N(C2CCN(C(=O)CSc3cccs3)C2)CCCC)=O)ncccc1SC c1(C(=O)NC2CCN(C(C(CC)COC)=O)CC2)ccc(SC)cc1OC CCC1=C(C(=O)NCC2CCN2C(=O)CC(C)OC)CCCO1 C(=O)(CCCCC(C)(C)C)NC1CCCN(C(CSCCCC)=O)CCC1 N1(C(C2C(OC)C2)=O)CCC(OCCNC(=O)CN(n2nccn2)C)CC1 C1(CNC(CCC=C)=O)CN(C(c2ccncc2-c2ccccc2)=O)CC1(F)F N#Cc1ccc(C(=O)NCC2CCN(C(c3ccnnc3C3CC3)=O)C2)o1 N1(C(C2CN3CCC2C3)=O)CCC2(C1)CN(C(C1CCCCO1)=O)C2 C1(C2CCN(C(=O)CNC=O)CC2)(C(=O)NCC(CCC)O)CCOCC1 C12(NC(=O)CCCc3nccs3)CCCC1(F)CN(C(=O)CCn1cncn1)C2 c1(C(=O)NC2CCCC(CNC(=O)C=C3CCCCC3)C2)c(F)ccc(F)c1O c1(NC(C(CC)NC(=O)Cc2cc(C)cs2)=O)cc(C)c(C)cc1C C(=O)(C1Cc2ccccc21)N1C(C(=O)NCC(C(CC)C)CO)CCC12CC2 Cc1cccn2c(C(=O)NCC3CN(C(C4(C(C)C)COC4)=O)CCO3)cnc12 C1(CNC(C2CC(OC)C2)=O)CN(C(c2cc3ccsc3s2)=O)CC(C)(C)O1 c1(-c2nc(-c3c(OC)n(C)nc3)on2)c[nH]c2nccc-2c1 C(=O)(CS(=O)(=O)C1CC1)N1CC2C(CNC(c3ccc(CC(C)(C)O)s3)=O)(C2)C1 N1(C(c2c(CC)c(Cl)ccc2)=O)CCC2CN(C(=O)Cn3cncn3)C2C1 c1(OC)cc(F)c(CN2CCC(C(=O)Nc3sc(C)cc3C#N)C2)c(F)c1 C1(C(=O)NC(C)Cc2cccc(Cl)c2)CCC(=O)CC1C C1(C)(CN(C(C=C(COC)C)=O)C)CCCC1NC(=O)C=CSc1nc[nH]n1 c1(C(N2CC(CSC)OCC2)C(=O)NCC2CC2)ccc2ccc(F)c(F)c2n1 N1(C(C2CC(NC(CCC3CCC(=O)C3)=O)C2)=O)CCCC(c2ncc[nH]2)C1 Cc1cnn2ccc(C(N3CCCC3C3(NC(C4CCCC4O)=O)CC3)=O)nc12 c1(C(=O)NCC(CNC(C2C(C)OCCC2)=O)C(F)(F)F)[nH]nc2ncccc12 c1(OC)nc(=NCC2CCCN2C(=O)C(C)O)nc(OC)[nH]1 CC1COCC1(C(F)(F)F)NC(c1nnnn1C1CC1)C1CCC1 C(=O)(C(C)C(O)CC(C)C)N1C(CNC(c2c(C)c(F)cnc2)=O)CC2(CC2)C1 C(C(N=[N+]=[N-])C(=O)N(C)CC1CN(C(c2cc(C)cnc2C)=O)C1)OCC c1(C(N2CCC(C(C)NC(C3(C#N)CCC3)=O)CC2)=O)cc(C(F)(F)F)ccc1O c1(-c2nn(CC(=O)NC(C)C)c(CCC(F)(F)Cl)n2)cc(F)c(N)c(F)c1 CC1CCC(C(F)(F)F)CN1C(c1ccc(Br)cc1F)=O C1(C(=O)NC2CCC(NC(C3CC3c3cccs3)=O)C2)(CO)CC(F)(F)C1 C1(CNC(c2c(C)ccnc2)=O)CN(C(=O)Cc2ccoc2)CCC12CCC2 C(CCOCCO)(C(=O)NCCc1ccn(C)n1)NC(C(CN(C)C)O)=O c1(C(N2CC(CNC(CCC=C=C)=O)C3(C2)CCC3)=O)nc2nc(C)ccn2n1 c1(CC)ccc(C(N2CCC(C)C2CNC(c2cccc(C3CC3)n2)=O)=O)cn1 Cc1cccnc1C=CC(=O)NC1CCN(C(=O)Cc2ccnn2C)CC1F N1(C(CCC2(C(N3CC(OC)C3)=O)CC(=C)C2)=O)CC(F)(F)CC1C C#Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(C)(O)COC)ccc1C C1(C(=O)NC2(CCNC(c3cncn(C)c3=O)=O)CC2)CCC2(C1)CC2(F)F N1(C(c2cc(C)ncc2Cl)=O)C2CCC1CN(C(=O)C(C)(C)C1=CCCC1)C2 C12(NC(CCCOCCOCC)=O)CCCN(C(=O)C3=CCCOCC3)CC1C2 c1(NCC(CN(C)C)OC)ccc(S(=O)(=O)NC(c2cncs2)C)c(Cl)c1 Cn1c(C(N2CCC(NC(c3cncc(CO)c3)=O)C(O)C2)=O)ccc1[N+](=O)[O-] c1(C(=O)NC2C(O)CCN(C(C(COC)OC)=O)C2)ccc(OC)c(OC)c1C C(CCCC(C)NC(=O)Cn1ccsc1=N)NC(C=C(C)Cl)=O c1(C(N(CC(C)NC(=O)CCNC2CC2)CC)=O)csc(Cl)c1Cl C1(NCC2CCN(C(=O)NCc3c(CC)cccc3)C2)CC2(CCCC2)CO1 c1(OCC=C)ccc(Cl)c(C(N2CCCC(O)(CNC(c3ccc[nH]3)=O)C2)=O)n1 C1(C2CC2)(CNC(c2cc(OC)c(C)nc2)=O)CCN(C(c2c[nH]nc2C)=O)C1 N=c1ccc(C(=O)NC2C=CC(CNC(c3cn(CC(F)F)cn3)=O)C2)n[nH]1 c1(NC(C2CS(=O)(=O)CC2N2CCOCC2)=O)nc2cccc([N+](=O)[O-])c2s1 c1(C(C)NC(C(=O)NCCCC)CC)ccc(OC)cc1 c1(C(=O)NC(CNC(C(C=C)(C)C)=O)(C)CO)cc(C)cc2c1NCCC2 Cc1cccc(N)c1C(=O)NC1CC(O)CN(C(=O)CC2CSCCS2)C1 C1(C(=O)NCC2C(C(F)(F)F)CCN(C(CSC)=O)C2)CCc2nn[nH]c2C1 Cc1cc(C)c(C(=O)NCC2(C(=O)NC3(Cc4cnn[nH]4)CCCCC3)CC2)s1 c1(OCC(=O)NC2C(CNC(Cc3c(C)ccnc3)=O)C2)ccc(Cl)c(F)c1 N1(C(c2c(C)ncn2C)=O)CC2CC(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 c1(C(=O)NC2(CF)CCN(C(C(CC(=C)C)C)=O)C2)ccc2c(Cl)nccc2c1 CC(C(=O)OCc1nccnc1O)C(C)NC(=O)OC(C)(C)C c1(CC(=O)NCC2CN(C(CCCOCC)=O)C3C2C3)c(C)nn(C)c1C C1(C(N2CC(CCNC(CCC(=C)Br)=O)OCC2)=O)CCC(C)(O)CC1 c1(CN2C(C(=O)NC3(C(=O)OCC)CCC3)CC(O)C2)cc(I)ccc1F c1(CCC(=O)NCC(C2CCOC2)NC(COCCCOC)=O)ccnn1C C(=O)(C(C)CCOC)NC1(CCCNC(C2C(=C)CC2)=O)CC1 Cn1c(=O)ccn(CC(=O)NC23CCCC2N(Cc2csnn2)CC3)c1=O CCCCCC(C(=O)NC1CCCC(CNC(=O)C=CC2CCCC2)C1)C(C)C c1(CC(=O)N(CCN(C(C2CC2C)=O)CC)CC)ccon1 Cn1cc(S(N)(=O)=O)cc1CC(=O)Nc1ccc(OCCO)cc1 CC1CN(C)CC1(c1nnnn1CCCF)NC1(CCF)CC2(CSC2)C1 C1(NC(C2C(CCC)C2)=O)(CNC(=O)C(O)CN2CCCC2)CCCCC1 C1(NC(CCCC#CC)=O)CCOC12CCN(C(=O)CC1NC(=O)NC1=O)CC2 C1(CC)(OCCNC(C(C)C2CCOC2)=O)CCOCC1.C1(CC(=O)N)CC(F)(F)C1 C1(N(C(c2c(C)snc2)=O)C)CC2CC1N(C(c1cccn1C)=O)C2 N1(C(c2ccc(C#N)o2)=O)CCN(C(C2CCCC2(F)F)=O)CC(CO)C1 CCC(C)C(C)C(=O)N(C)CC1(O)CN(C(c2ccc(SC(F)F)cc2)=O)C1 Cn1cccc(C(=O)NC2(C3CCCN3C(=O)C(F)CC3CC3)CC2)c1=O N1(Cc2cnc(SC)nc2Cl)CCC2CN(C(c3ncc(C)s3)=O)CC12 N1(C(CCOCCCNC(Cc2c(C)scc2)=O)=O)CC(CO)C1(C)C CSC1=C(C(=O)NCCC2(O)CCCN(C(=O)Cc3cnnn3C)C2)CCCC1 c1(C(=O)NCCC(C)N(C)C(c2cscn2)=O)n[nH]c2c1CC1CC21.C1(=O)CN1 c1(NC(NC2C(C)CCN(CCc3ccccc3)C2)=S)c2c(nn1C)CCC2 c1(C(N2CCC(NC(c3cccc(C)c3Cl)=O)C2)=O)n[nH]c2c1CC(C)(C)C2 C1(NC(c2ccc(Cl)s2)=O)COC2(CCN(C(c3cnc(Cl)s3)=O)CC2)C1 c1(CC(=O)N(C(CNC(CC(CC)OC)=O)C2CC2)C)ccc(Br)c(C)c1 N1(C(C(c2cccnc2)C)=O)CCCCC(NC(c2ccccc2C2CC2)=O)C1 N1(C(c2cc(Br)co2)=O)CC2CCC(C1CO)N2C(C1CC1[N+](=O)[O-])=O CC1CC(NC(=O)C(c2ccc(F)c(F)c2)=O)CN(C(c2cc[n+]([O-])cc2)=O)C1 CCC(CCCC(=O)NC1CCCC1(C)O)NC(c1ncccc1F)=O N1(C(C(CCNC(=O)OC(C)(C)C)(C)C)=O)CC2(CCCO2)C1OC(C)(C)C C1(NC(c2ccc(Cl)cn2)=O)CCN(C(c2csc(Cl)n2)=O)C12CC2 c1(CC(N2CC3CC2CN3C(c2cnc(O)cc2O)=O)=O)c(Cl)cc(Cl)cc1Cl c1(C(=O)NC(CNC(C=C(CC)C)=O)CO)cc2cc(C)ccc2[nH]1 C(=O)(CC(C)C(=O)NCCCC(=O)NCc1cnccc1Cl)OCC C1(O)(CCNC(C(C)N2CCC2)=O)CCCN(C(c2cc(=O)c(O)c[nH]2)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)CCCc1cnn[nH]1)N1CC(C)(COC)C1 N1(C(CCCOCC)=O)CC(NC(=O)C2=C(Cl)CC2)CC(O)C1 CC1(F)CN(C(=O)CN2CCOCC2)CCN(C(C2(C(F)(F)F)CCCC2)=O)C1 C1(C2(NC(C3CCN(C(=O)c4occc4C)O3)=O)CC2)(OC)CCC1 N1(C(c2c(C)ccs2)=O)CCC(C)(C)C1CC(N1CCC(C)(CCO)C1)=O N1(C(CC(CC)NC(CCCC#C)=O)=O)C2CCC1COC2 CC1=CCCN(C(C2(F)CN(C(=O)CC3CCCC(C)O3)C2)=O)C1 c1(OC)ccccc1CC(C)(C)C(=O)NCC(CNC(C1CC1(F)F)=O)CO c1(CNC2(c3n(C(C(=O)OC)C)nnn3)CC(C)C2)c(Cl)c(C)nn1C Cn1ncc(C(=O)NC(CC2CCC2)C(=O)N2CCCC2C(N)=O)n1 C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(c2ccnc(C)c2Cl)=O)C1 C(=O)(C(C(C)(C)C)C1CC1)NCc1cn(CC(=O)Nc2cccc(OC)c2)nn1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCN(C(=O)CC(=O)NC)CCC1C C1(OC)NC(C(=O)N(C2CCCCC2)Cc2ccc(F)cc2)CCC1Br C(CN(C)C)(C(=O)N1CC(n2cnnc2)C1)NC(C1C(C(C)(F)F)C1)=O C1(C(N(C(COC)COC)C)=O)C=CCCN1C(=O)CC1CCC(C)(C)C1 C1(C)(C(=O)NC(C)C(=O)NCCC(Cl)Cl)C=CCCC1 CC1CC(C)C1C(=O)NC1(CNC(=O)CSCc2cccs2)CCCC1 N1(C(C2CC(C(C)C)OCC2)=O)CC=C(CCNC(C2(C)CCCOC2)=O)CC1 C1(NC(CCCSC(C)C)=O)CN(C(=O)C(O)CC(=O)OC(C)(C)C)C(C)(C)C1 C1(CN(C(C2(COC)CCC2)=O)C)CCN(Cc2ccccc2)C1 C1(CNC(CCOC)=O)C(C2CC2)CCN1C(c1nc(Cl)cs1)=O C=C1Cn2c(C(N3CC4CCC4(NC(=O)CC4CCCO4)C3)=O)nnc2S1 c1(CCC(=O)NC2CC(NC(COC(CC)C)=O)C2)ccc(F)cc1Br C1(NC(c2cc(C)n(C(C)(C)C)n2)=O)CC(C)CN(C(c2ccc(O)nc2)=O)C1 Cc1cc(C(=O)NC(C)CNC(c2cnc3[nH]ncc3c2)=O)cc(C)c1O c1(OCC=C)ccccc1CC(N1CCC(N(C(=O)C(C)CCC)CC)CC1)=O c1(C(N(CCOCCC(=O)NCC(CC)O)C)=O)nccnc1CC c1(C2(C(N3CC(CC=C)(NC(=O)CCF)C3)=O)CCCC2)cccc(C)c1 CC(C)C(C#N)C(=O)NCC(C)CNC(c1ccc(Cl)cn1)=O N1(C(c2cc(C)oc2C(F)(F)F)=O)CCN(C(=O)CC2CC(F)C2)CC(O)C1 c1(C(=O)NC2C(C)(C)N(C(=O)Cc3ccsn3)CC2)noc2c(F)cccc12 CC(C)CCCC(=O)NCC1CN(C(=O)C2=CCCCO2)CC1O C(=O)(C1CCC(=O)c2cccn21)N1CCN(C(C(C(C)C)NC=O)=O)CC1C C(CN=C(NCC1CCc2ccccc2CC1)N1CCOC(CF)C1)SCC#C Cc1nocc1CNC(=O)C(C1(O)CCC1)NC(=O)C(C1CC1)C1CC1 Cc1c(C(=O)NC2CCN(C(=O)C(C)C(C)C)C2)cc([N+](=O)[O-])cc1Br C=C(CNC(=O)CC(C)C(C)(C)NC(=O)Cc1cnc(C)s1)c1ccccc1 N1(C(c2cnc(C)s2)=O)CCC(C(CO)NCC2(c3ccncc3)CC2)CC1 C12(C(=O)NC3(C)CCN(C(c4nc(C)n(C)c4)=O)C3)CCC(CC1F)C2 C1(NC(C(CCCC)C)=O)CCC2(CC1)CN(C(=O)CNC(c1ccco1)=O)C2 C1(NC(C2(COC)CCC2)=O)CCN(C(=O)Cc2ccc(CO)cc2)CC1 C1(C(=O)NCCS(=O)(=O)NC)N(C(=O)CCCC#N)CC12CCCC2 c1(C(C)NC(c2nscc2Br)=O)nnn(C)c1N C1(CC(=O)NCCCN(C(C2CCCCO2)=O)C(C)C)(OC)CCOCC1 N1(C(C(=O)NCC(=C)C)C(C)C)CCCN(S(=O)(=O)C(F)(F)F)CC1 C(=O)(C1=CS(=O)(=O)CCC1)NCC1C(NC(C=Cc2n(C)ncc2)=O)CCC1 CCCCC(C)C(=O)N1CCCOC(CCNC(c2c(C)ccnc2O)=O)C1 C(=O)(C(C)C(C)C)NCC1C(NC(c2nc(C(C)C)oc2)=O)COC1 c1(C(N2CCC(CCNC(C(C#N)C3CC3)=O)CC2)=O)cnc(O)c(Cl)c1 CC1CN(C(C2CN(C(c3cc(CCO)on3)=O)CC2(C)C)=O)CC1(C)CO N1(c2cc(C)nc(CO)n2)CCC2(COC(CNC(=O)C=C3CCCCC3)C2)C1 C1(NC(N(C(c2c(C)nn(C(F)(F)F)c2C)C)C)=O)CCn2ccnc2C1 Cc1cnc2n1CCC(C(=O)NC1(c3ncon3)CCOCC1)C2 Cc1ccc(O)c(C(=O)NCCCCCCNC(c2cc(C)[nH]n2)=O)c1 c1(COC)nn(C)cc1C(=O)NCC1C=CCN1C(=O)C(O)CN(C)C N1(C(c2on(C)c(=O)c2)=O)CC2(CCN(C(C3(c4cccs4)CCCC3)=O)C2)C1 c1(C(N(CC(C)(C)NC(C23CCCC2C3)=O)C)=O)n[nH]c2c1CCC2 Cc1cc(C(=O)NC2CCOC(CNC(=O)CCCC3CCOCC3)C2)[nH]c1C CCC(C)(C)C(=O)C(=O)N1C(C(=O)NOC)CC1C C(C(O)C(=O)NCC(C1CC1)NC(=O)CSC)=CCCC N1(C(c2ccc(C3CC3)o2)=O)CCN(c2ccc(CCO)cn2)C(CCO)C1 c1(OC)c(Cl)ncnc1NNC(=O)NC1CC1(F)F C(=O)(CCC(C)(F)F)N1CCC(N(C(c2nn(CC)c(C3CC3)c2)=O)CCO)C1 c1(C(=O)OCC)ccc(C(=O)NC(C)(CNC(C2C=C2C)=O)C(C)C)cc1 c1(-c2sc(NCc3c(C)cccn3)c(C)n2)cccc(O)c1C C1(CC=C)(C(N2CC(CC(C)NC(=O)CNC(=O)C(F)(F)F)C2)=O)CC=CC1 CCCC(C(=O)NCCCOCCNC(C1(NC(C)C)CCC1)=O)OC C1(CC)C(C(=O)NCC23CC(NCC4(C(=O)N(C)C)CC4)(C2)C3)CCN1C c1(SCC(=O)NC(C2CCCC2)CNC(=O)CSC(F)F)cccnc1 N1(C(C2CC(OC)C2)=O)CCC(C)(NC(=O)Cc2cc(C(F)(F)F)nn2C)C1 C1(CNC(c2ccc(NC)cc2)=O)CN(C(=O)C(O)CC(N)=O)C2(CCC2)C1 c1(C(C(C)C)NC(C(=O)N(CCn2c(C)ncc2)C)=O)cccc(C2CC2)c1 N1(C(c2n(CCC)ncc2)=O)CC(NC(=O)Cc2nocc2C(C)C)C(SC)C1 C1(NC(CCc2n(C)ncn2)=O)CN(C(=O)CSc2ccccc2)CCC1F c1(OCC=C)ccc(Cl)c(C(=O)NCC2CCN2C(c2cc(CCC)[nH]n2)=O)n1 C(=O)(C(C)(C(F)F)c1ccccc1)NC(C)CC(C)NC(=O)COCC1CCC1 c1(C(N2C(C)(C)C(CNC(=O)Cn3ccnn3)CC2)=O)ccc(N)c(F)c1F Cc1[nH]c2ncccc2c1C(=O)NCC1CN(C(=O)C(C)CS(C)=O)CCCO1 c1(N2CCC(CC=C)C2)nc2c(c(=NCCS(=O)(=O)C3CC3)[nH]1)SCC2 N1(C(C2N(C(C)C)C(=O)CC2)=O)CCCC(O)(CCNC(c2ccnnc2)=O)C1 C#CCCCC(C)C(=O)NCCCCCC(=O)NCC1CC12CCC2 C12(C(=O)NCC(=O)NCc3ccc(F)cc3Cl)CC3CC(C1)CC(O)(C3)C2 c1(CNC(C2CC(CCC)C2)=O)nc(C(=O)N(C2CCCC2C)C)c(C)o1 CCC(CC)C(=O)NCC(=O)NC(CC1CC1)C(=O)NC(C)(C)CC(N)=O N1(C(C2N(C(=O)OC)CC2)=O)CCc2cc(NC(=O)C(=O)N=S(C)(C)=O)ccc21 N12CCCC(C1)C2=O.O=C1CCC(C(=O)NCc2cccnc2)O1 c1(C(=O)NCCC(C)N(C(=O)CSc2n[nH]c(O)n2)C)cc2cccc(F)c2s1 C1(CC(=O)NC2C(NC(c3c(COC)noc3)=O)CCC2)CCOCC1OC c1(OCC)cncc(C(=O)N(C(CNC(c2ccnn2CCF)=O)C2CC2)C)c1 C1(C(=O)NC2(COC)CCCCC2)COCCN(C(C2(C)CC2C)=O)C1 N1(C(C2C(C(=O)OC)C=C2)=O)CCC(C)(C)C(C(=O)N(C2CCCC2(C)O)C)C1 N1(C(c2cc(C)n(C)n2)=O)CCC(C)(C)C1C(=O)NCC1COC(C)(C)C1 N1(c2nc(C)cc(OC)n2)CC2(CCOCC2)CC1CNC(C1CCCOC1)=O CC1(NC(C2CC2F)=O)CCCN(C(C2CC(O)C2)=O)C1 c1(C(=O)NCCNC(=O)NCc2csc(Br)c2)cccc(OC2CCCC2)c1 C1(C(=O)NCC(C)CC(=O)NC(CC2CCCC2)CO)(OC)CCC(C)(C)C1 n1(CC(=O)OCC)cc(C(=O)NCC(O)CN(C(=O)C(C)n2ccnc2)C)nn1 N1(C(N(CCF)CC)=O)CCCC(CC2CC2(F)F)C1 N1(C(C2(C)CCCCO2)=O)CCCC(C2CCN(C(=O)CSS(C)(=O)=O)CC2)C1 C(=O)(C1=NOC2(CCNCC2)C1)N(CCN(CCC1CCC(C)O1)C)C C(CCCC(=O)NCc1ncnn1C)N(C(c1c(C(C)C)onc1)=O)C Cc1c(NC(=O)C(F)=C2CNC2)cccc1-c1nn[nH]n1 C(CC(F)F)(C(=O)N1CCC1CC1CCCC1)N(C)C(c1cc(CO)on1)=O c1(C(N2CC(C)(CC(=O)NCC(N3CCCC3)=O)C2)=O)nnc2ccc(Cl)nn12 C#CCC(O)C(=O)N(C1CCN(C(=O)Cc2coc(-c3ccccc3)n2)C1)C CC1(C(N2CCC(CNC(c3cc(F)ccc3Cl)=O)C2)=O)CCC(F)(F)C1 CC1CCC(NC(C2CCC3(CC3)C2)=O)CN1C(=O)CC12CCC(CC1)C2 C1(C(=O)NCC2CCCO2)CC(F)CN(Cc2ccc(F)nc2)C1 C12(NC(C3N(CCC)CCC3)=O)COC(C1)C(NC(=O)CCC(=O)OC)C2 C(=O)(C(C(C)(C)C)NC(=O)CC(F)(F)CC)N1CCC(O)(CCC)C1 N1(C(C(C(C)C)OC)=O)CC2(CCN(c3cc(O)nc(=O)n3C)CC2)CC1C CC(C)(CC(=O)NC1CC(NC(=O)C(C)(F)F)C1)C(F)F CCCCC(F)C(=O)NC1CC1NC(=O)CS(C)(=O)=O C1(CNC(NC(C#C)C)=NCCCOC(C)C)Cc2cc(C)cc(Br)c2O1 c1(C(N2C(C3(NC(C4CCOCC4)=O)CC3)CCC2)=O)cc2ccccc2[nH]1 c1(CNC(C(=O)OCC)Cc2ccncc2)cc(C)c(Cl)c(C)c1 N1(C(C(CC)C)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)CC1c1cn[nH]c1 O=S(=O)(c1cccnc1NC12CCCC1C2)NCCn1ncc2ccccc12 c1(C(=O)NCC(C(=O)OC)CC2CCCC2)ccnc2[nH]c(C(F)F)nc12 C(=O)(C=CS(C)=O)NCCNC(C1CN(C(C2C(C)OCC2)=O)C1)=O c1(C(N2CC3CC(NC(c4ccc(CC)s4)=O)C3C2)=O)c(C)ccc(F)c1N Cc1cccc(C(=O)NC2CCC(C(=O)N(C3CCCC3O)C)C2)c1O N1(C(C=Cc2n(C)ncc2)=O)CCC(CNC(=O)C(F)=CCCF)C(O)C1 C(=O)(C1CCCc2nn[nH]c21)N1C(C)CC(CNC(c2c(F)ccnc2F)=O)C1 c1(CC)ccc(CCCC(=O)NCC(O)CNC(c2coc(OC)n2)=O)cc1 c1(C(=O)Nc2nccc(-c3cn(C)nc3)c2)cc(S(C)(=O)=O)ccc1O C(=O)(CC(C)(O)C1CC1)N(C(C(=O)NC1CCN(S(C)(=O)=O)C1)C1CC1)C C1(NC(C=CCOC)=O)CCN(C(C2(C(=O)C3CC3)CC2)=O)CC1F CC1OCCC1C(=O)CN(C(=O)CC1CCCC1O)CCO.C(=O)(CS)O C1(C(N(CCC(=O)NC(C2CCCC2)C#C)CC#C)=O)COCCN1CC C(C(C(=O)NC1CCN(C)CC1C)C(C)C)NC(C1(CCOC)CCC1)=O c1(CC(=O)NC2C(CNC(c3cc(OCC)no3)=O)CCC2)cc(F)ccc1F C(C)(CC1CCCCC1)(C(=O)NC(C)CN(C(=O)Cn1nnnc1C)C)OC c1(C(=O)NCC2(OC)CN(C(C3(C)CCCN3C)=O)C2)ccc(F)c(C(F)F)n1 c1(C(=O)NC(C2(CNC(c3cn(CC)nc3)=O)CC2)C)ccc2c(c1)CNC2=O CC(C)C(O)CC(=O)NC1CCC(NC(C2OCCC2C)=O)CC1 c1(C(=O)NC2CC(NC(C3(C)CCC(C)C3)=O)C2)n[nH]c2cccnc12 c1(C(=O)NCC2CCCCC2C(c2cnc[nH]2)=O)cccc(CC2CCOC2)c1 CCC(C(=O)NCCC(C)NC(c1coc(C(C)(C)C)n1)=O)OC n1(CC(N2CC(OC)C(OC)C2CSc2ccccc2)=O)cnc2c1CCCC2 c1(C(N(C2CCN(C(=O)CC(C)(C)OC)C2)CCC)=O)c(C)nn(C)c1OC C=C=CCCC(=O)N(C1CCCN(C(=O)C(C)SC(F)(F)F)C1)CC CN1CCC(C)(C(=O)NC2(C)CCCN(C(c3nscc3N)=O)C2)C1=O N1(C(C(C)CC2CC2)=O)CC(C(=O)NC(C)(C)CC2CC2)C(F)C1 CC(CC(=O)NCC(C)NC(c1cnn(-c2ccccc2F)c1)=O)C(F)F C1(CC=C)(NC(c2c(COC)cc[nH]2)=O)CCN(C(=O)Cn2nc(C)cc2C)C1 C(=O)(CCC(C)CN(C)C)NC1(CNC(c2ccc(OC)cn2)=O)CC(F)(F)C1 C(=O)(CCCC(C)CC)NC(CC#C)CC(=O)NCCCN1CCOCC1=O N1(C(CCC#C)=O)CCC2(CC2C(=O)NOCC2CCCC2)C1 N1(C(c2c(Br)sc(C)c2C)=O)CC2CCC(C1)C(NC(C1CC1C)=O)C2 Cc1ccc(C(N2CCC(C)C2CNC(=O)Cc2cc(Cl)ccc2F)=O)cc1Cl C(=O)(C(C)N=c1cc[nH]cc1)NCC1CCN(C(c2c(OC)scc2)=O)CC1C C1(COC)(NC(=O)Cc2ccsc2)CCN(C(c2cn(C3CC3)cn2)=O)C1 C#Cc1cccc(C(=O)NCC(C2(O)CN(C(=O)C=CC3CC3)C2)(C)C)c1C c1(C(N2CCC(CN(C(c3cc(COC)oc3C)=O)C)C2)=O)[nH]c(=N)ccc1C CC1(CNC(c2cc(C3CC3)cs2)=O)CCC(NC(=O)Cc2cc[nH]n2)C1 c1(N(C2CNC2)C)nc(Cl)ncc1Br.C(=O)CCCn1ccnc1 CC1(C)CCN(C(C2CCC3(CC3)C2)=O)C1C(=O)NCC1=CCCCCC1 CCCCCC(F)C(=O)NC(CCCC)C(=O)NCc1cc(C(C)C)no1 c1(C(=O)NCC2C(CNC(C3(C)CC=CCO3)=O)C2)n[nH]c2c1CCC2 C1(C(=O)NCC(C)C(=O)NCC(c2ccncc2)C)CCCCNC1=O N1(C(C(c2n(C)cnn2)(C)C)=O)CCN(C(C2(CF)CC2(F)F)=O)CC12CCC2 Cc1nc(C(=O)NC2CCC2NC(=O)COC2(C)CCCC2)c(C(F)(F)F)[nH]1 CC(C(C)(C)Nc1cnn(CC2CCC2)c1)NC(=O)OC(C)(C)C C1(C2CCCCC2)(NC(C2CC(C(=O)N3CC4CC4(CO)C3)=NO2)=O)CC1 N1(C(C2(C)C(C)C2)=O)CC2COCC(C1)N2C(c1cc2cnccc2[nH]1)=O N1(CC(c2cccc(F)c2)C)CCN(CCCn2nccn2)CC1C C1(CC(=O)NCC2N(C(c3cncn(C)c3=O)=O)CC2)CCC2(CC1)COC2 C#Cc1ccc(C(N2CCC(NC(c3c(C)csc3Cl)=O)C(O)C2)=O)cc1Cl c1(-c2c(C(=O)NCc3cc(OC)cc(F)c3)nccc2)ccccc1[N+](=O)[O-] C1(C(N(CC#C)C)=O)CCC2CCC1N2C(c1ncn(C)c1C)=O O=C1NC(C(=O)O)C2=C1C(c1cc3c(cn1)COC3)NC(=O)N2CCC1CC1 N1(Cc2c(OCC)cco2)CCC2(CC1)CC2C(=O)Nc1c[nH]nc1Cl C1(NC(COC)=O)COCC1C(=O)NCCC(N1CCCC1C1CCOC1)=O Cc1cc(-c2cn(C3CCN(C(c4c(C)ccn4C)=O)CC3)nn2)ccc1F c1(C(N(C)CCN(C)C(C2CCc3nccn3C2)=O)=O)cc(F)cc2nc[nH]c12 C1(CCC)CCc2nc(N(C(=O)C(CC(C)(C)C)OC(C)=O)CC)sc2C1 Cc1cccnc1-n1ccnc1-c1c[nH]c(-c2ccccc2)c1.c1nccnc1N C(=O)(C(C)(C)CC(C)(C)C)NCC12OCC(NC(C3N(CC)CC3)=O)C(C1)C2 C1(C(=O)NCCCC(=O)NC)CCN(C(=O)C=C(C)C(C)(C)C)C(C)(C)C1 C=CCC(C(=O)NCC1CCC(C(=O)NC(c2cn[nH]c2)C)C1)C(C)C n1(CC)cnc2[nH]c(=NCC3CC(O)C3)nc(N3CCOCC(C)(F)C3)c12 c1(C(N2C(C)(CCC)CC2)C(=O)NC2CC(F)(F)C2)cccc(C2CC2)c1F CC(C(=O)OC(C)(C)C)C(=O)N1CC2C(CN(C(=O)CCC=CC(C)C)C)C2C1 C=CC1OCCC1C(=O)NCC1CC1CNC(c1ccc(SC)o1)=O N1(C(=O)NCc2ccc(Cl)cc2C(F)F)CCCC1C1CCCO1 c1(C(C)=O)cc(NCCCNC(C2CCC(=O)N2)=O)ncn1 c1(CC(=O)NC(CCCNC(CC=C)=O)C)coc2cc(Cl)ccc12 c1(N(C(C2CN(C(C(=O)NC(C)C)=O)CC23CC3)=O)C)ccn2nccc2n1 c1(C(=O)OCCc2ccccn2)ccc(NC(c2ccon2)=O)cc1 c1(NC2CCN(C(C(n3ncc(C)c3)C)=O)C2)cc(O)nc(C)n1 c1(C(N(C2CC(NC(C3C(C=C)C3)=O)C2)C)=O)cnc(O)c2cncn12 Cc1cccc(CC(=O)NC2CC2NC(=O)COc2cnc(Cl)cn2)c1 c1(C(N2C(Cc3cn(CCC=C=C)nn3)CCC2)=O)nn(C)c2ncccc12 C(=O)(C(CC(C)C)C(N)=O)NCC(CN(C(Cc1cc(C)nn1C)=O)C)C N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(=O)C(N2CCSCC2)C)CC(F)C1 N1(C(CNS(NC)(=O)=O)=O)CC2CCC1CN2C(=O)C(F)C(F)(F)F c1(CNC(CC)Cn2cncn2)cc(OC)c(C)cc1F CC1CN(C(c2c[nH]c(Br)c2)=O)CC2(CCN(Cc3cc(Cl)ccc3Cl)C2)O1 N1(C(c2n[nH]c(C)c2C)=O)C(C)CN(C(c2cnccn2)=O)CC1C CN1Cc2ccccc2CC1C(N1CC(NC(C23CC(C2)C3)=O)C(F)C1)=O C1(=CC(N2CC(C(C)NC(CC3N(CC)C(=O)CC3)=O)C2)=O)CN2CCC1CC2 C(=O)(C(O)CCCNC(=O)C(C)CC(C)C)NCCC(=O)NCC#C c1(CC)cc(C(=O)OCC2CC2c2ccc(Br)cn2)c(Br)s1 N1(C(C2C(NC(C34CC(C3)C4)=O)CCC2)=O)CC2CCC1CO2 C1(N(C)C)CN(C(C2C=CCCC2)=O)CCC1CNC(C1CC=CCC1)=O Cc1ncn2ccc(C(=O)NC(C)(C)CN(C(=O)C3=CCCC3)C)cc12 N1(C(CC(=O)OCC)=O)CCCCC1CN(C(=O)C(C)(C)COC)C c1(C(=O)NC2(CC=C)CN(C(=O)C(C)C3CC3)C2)ccn2c(C)cnc2c1 C1(C(N(CC(C)(C)CNC(c2ccnc(CO)c2)=O)C)=O)OCC2CCCC12 C1(OCCC)CCCN(C(=O)CCCCNC(c2ccnnc2O)=O)C1 N1(C(C(COC)C)=O)CCN(C)C(CNC(=O)C=C(C)c2ccco2)C1 C1(C(N(CC(O)CN(C)C(c2n[nH]cc2[N+](=O)[O-])=O)C)=O)CCCCC(F)(F)C1 C1(C(=O)NCC2(F)COC2)COCCN(C(c2ccnnc2O)=O)C1 N1(C(C(C(C)C)O)=O)CCC(C2CC2)C1CNC(c1cccc2nsnc12)=O CCCC(CNC(=O)C1=CCCC1)C(=O)Nc1cccc(F)c1F C(C(C(=O)NC1(c2ncc(C)s2)CC1)C(C)(C)C)NC(CCCSC)=O C(CCCCC(=O)N(C1CCOC(C)C1)C)N(C(c1c(C)noc1C)=O)C C(=O)(C#CC(C)(C)C)NC(C1(O)CCN(C(=O)CCc2nc[nH]n2)C1)C C(c1ccccc1C)=CC(=O)NC1CCC(N(C(C2CC(CC)(CC)C2)=O)C)C1 C12(C(=O)NCC(CC(C)C)(C)NC(=O)C#CC3CCOC3)CCCN(CCC1)C2 C(=O)(C1=NOC(C)C1C)NC(C1C(C(N2C(C(=O)NC)C=CC2)=O)C1)C C(=O)(C(=O)C(C)(C)C)N1CC2C(C(N(C)CCC3CCC3)=O)(C2)C1 C(=O)(C(C)CC(F)(F)F)NCC1C(NC(c2c(C)n(C(C)(C)C(C)C)nc2)=O)C1 N1(C(CC2(OC)CCOCC2)=O)CCC(O)(C(C)NC(C2CCCC2O)=O)CC1 c1(C(N(CCOCCN(C(C(CC)OC)=O)C)C)=O)ncc(OC(C)=O)cc1F c1(C(N2C(C)C(C)N(C(c3cscn3)=O)CC2)=O)cnc2ncccc2c1 O=C(C(C1=NOCC1)N1CCCC1C1CC1(F)F)NCc1ccc(Cl)cc1 C(=O)(N1CCC(C(N2CCCC2CCC(C)C)=O)O1)c1nc(C)oc1 C(=O)(C(CNC(c1nc(C)oc1C)=O)CC(C)C)NC(c1nc[nH]n1)CC CCC(C)(C(=O)N1CCN(C(=O)CCc2ccnc(Cl)c2)C(C)C1)C(N)=O CC(C)C(C)(CNC(C1(CS(N)(=O)=O)COC1)=O)NC(=O)Cn1nccn1 c1(C(C)NC(C2OCCC2CNC(=O)C(CO)N(C)C)=O)cccnc1O c1(C(=O)NCC2COCCN2C(=O)CC(F)(F)F)ccnnc1O CCCC(C)(C)C(=O)NCCN(C(=O)CCC=Cc1ccccc1)CC1CC1 CCC(C)C(O)C(C)C(=O)NC(C(N1CCC2(CCCC2)C1)=O)C1CCOC1 C1(C(N2CCC(CN(C(=O)C(C)(C)n3ccnn3)C)C2)=O)CCCC(C)(C)CC1 C=CCCCCNC(=O)C(C)(C1CCC1)NC(=O)C(C)N(C)C(C)=O N1(C(=O)C=CCF)CCC2(CCCN2C(C2SCCCS2)=O)C1 c1(C(=O)NC(C(=O)NC(c2nnc(O)n2C)C)C2CCOC2)ccnnc1O c1(C2(F)CN(C(C3C(c4n(CC)ccn4)OCC3)=O)C2)ccccc1Br C12(CNC(C3(CC)CC3(F)F)=O)CC1CN(C(C1(CO)CCCCC1)=O)C2 C1(NC(CN(C)C(=O)C2CC2)=O)CCC(F)(CNC(c2cc(O)ncn2)=O)C1 c1(NCc2c(Cl)ccc(N(C)C)c2)sc2c(c1C(=O)NC1CC(O)C1)CCC2 C1(NC(c2cscn2)=O)CN(c2ncc(OC(F)F)cn2)CCC1(F)F c1(C(N(CC(CNC(c2nccc(C)n2)=O)C)C)=O)cc(N)c(C)cc1C N(C1CCCn2ccnc21)C(=O)CC1COCCN1C(=O)CC(C)(C)C#N.CNC n1(CCOC)cc(C(=O)NCCC2CCCN2C(C2CC(CF)C2)=O)nn1 N1(C(C2(N(C)C)CC2)=O)CCC(F)(F)C(CNC(c2nc(Cl)sc2Cl)=O)C1 N1(C(c2c(C)c[nH]n2)=O)CC(C)CCC1CNC(c1ccc(F)c(CO)c1)=O N1(C(C2C(C=C)C2)=O)CC2CCC1CN2C(C1(C#N)CCOC1)=O n1(CC(=O)N(C(CCNC(C2N(CCC)CCC2)=O)C)C)cc(C#N)cn1 C(=O)(C(C(C)(C)O)NC=O)N(CCCF)C.C1CC(C)(C)C1 Nc1cc(C(=O)NCCC2CCN(C(C3(C(F)F)CCCO3)=O)C2)cc(O)c1Cl CC1(C)CC(C(=O)O)N(C(=O)CNC(=O)CCCC2CC2)C1 C(c1c(C)coc1C)=CC(N1CCC(N(C(=O)C(C)C2CCC2)CC)C1)=O Cc1cc(C(C(=O)NCc2ccco2)N(C)CC2(O)CCOCC2)cc(F)c1 c1(C(=O)NC2C(CNC(=O)Cn3cccc3)CCC2)cc2sccc2[nH]1 C1(C(=O)NCCNC(=O)CCc2nnc(-c3ccccc3)o2)CCCS(=O)(=O)C1 C1(NC(c2nc(CC)oc2C)=O)CC2CC1CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 CN=S1(=O)CCN(C(=O)C(c2ccc3c(c2)OCO3)=O)CC1 N1(C(C(N2CCN(C)CC2)C)=O)CC2CCN(C(c3cccc(=O)o3)=O)CC2C1 CCCCC(C)CCC(=O)NCCCOCCCNC(=O)CCc1ccccc1 N1(CC(CC)S)C(=O)CN(CCS(N)(=O)=O)C1=O.c1(N)ccccc1Cl C1(C(=O)NC2CCCC(OC)C2)CCOCCN1C(=O)Cc1cccs1 c1(C(=O)NCc2nc(CC(=O)OCC)on2)cnn(CC)c1C1CCCC1 c1(NC(C(n2ncc(C)c2)C)=O)ccc(C(N)=O)cc1 C1(C(=O)OCC)(CC)CCCN1C(C12CC(CCO1)C2)=O CCCC(CNC(=O)Cc1ccsc1C)C(=O)NCCOCCO C(=O)(C(CCNC(=O)C(C)OCC1CC1)OC)NCCC(=O)OCC c1(C(=O)NC2C(NC(c3cccc(C(C)C)c3)=O)C2)cccc2c1CNC2=O N1(C(C(CC)C)=O)CCCOC(CNC(c2cnc(CO)nc2C)=O)C1 C1(CNC(c2nc(Cl)sc2Cl)=O)CC(F)(F)CN1C(c1cnnc(Cl)c1)=O N1(C(C(COCC)O)=O)CC(OCC)CC1CF C1(C(=O)NC(C2(OC)CCC2)C2CC2)OCCCC1c1ccccc1 c1(OC)cc(CN)cc(N)c1O.N1(CCC(=O)N2CC(CO)C2)CCN(C(C)C)CC1 C1(C(=O)NCC2CCN(C(c3cc(C)on3)=O)C2)CCc2n[nH]cc2C1C C1(NC(=O)NCC2CNC(=O)C2)CC2C=CCC(C1)C2 C1(NC(c2coc(C3CC3)n2)=O)CCCN(C(C23CC(C(F)F)(CO2)C3)=O)C1 Cc1ccncc1CC(N1CC(OCCNC(=O)CC2CC=CCC2)C1)=O C(CN=c1ccn2ncc(I)c2[nH]1)NC(C1(C(C)C)N=N1)=O c1(C(=O)NCCCC(C)(C)NC(COCCN(C)C)=O)ccc(O)c(=O)cc1 c1(NC(c2csc(CNC(c3cccnc3F)=O)n2)=O)ncccc1[N+](=O)[O-] Cc1nc(C(=O)N(C2CCCC(N(C(=O)CCC(C)C)C)C2)C)c(C)n1C Cc1ccnc(NC(C)(CCCO)c2nnnn2CC2CCCO2)n1 C1(C(C)NC2CC2)CCCCN1C(c1cn(C2CCOC2)nn1)=O c1(C(N2CCC(CNC(CN(C(COC)=O)C)=O)C2)=O)c(C)oc2ccccc12 Cc1[nH]nc2c1CCC(C(=O)N(C1CN(C(C3CCN(C4CC4)C3=O)=O)C1)C)C2 C1(C(=O)OCC)CC(C)N(Cc2ccc(Br)cc2OCC)C(C)C1 C1(CC)CN(C(=O)C(F)C(C)CNC(C2(C#N)CC2)=O)CCN1C C1(NC(C(c2cn(C)nc2)(C)C)=O)CCCC(NC(=O)COC2CCC2)CC1 C1(O)(CNC(C2C(C(=O)OC)C2)=O)CCCN(C(=O)CC2(OC)CCC2)C1 CC1CC(NC(=O)CC(C)n2cccn2)CN(C(c2cc[nH]c2)=O)C1 CC1CN(C(c2ccns2)=O)CC(CCNC(c2cc(C3CC3)ncn2)=O)O1 C1(C(C)NC(=O)Cc2ccns2)CCN(C(=O)CCC2CCC2)C1 N1(CCOC(CN2C(=O)CCC2)=O)CCN(C(=O)CN2CCSCC2)C(=O)C1 Cc1cc(CCC(=O)NCC(C)CNC(C2CCC2(C)C)=O)on1 C1(NC(C=C(C)C2CC2)=O)CC2CCC1CN(C(=O)CC1CCS(=O)(=O)CC1)C2 C1(CCNC(C(C)Cn2ccnc2)=O)CN(C(c2c[nH]c(=N)s2)=O)CCO1 c1(C(=O)NCCCNC(C(CC)n2cccn2)=O)cc(C(F)(F)F)cc(F)c1 c1(C(=O)NCC2(F)CC(NC(C3(C#C)CCC3)=O)C2)c(C)c(C)c(C)c(C)c1C C(=O)(C(CC(C)(C)C)NC(=O)OC(C)(C)C)N(C1CCOCC1)CCC c1(C(=O)NCC2CCC(CNC(C)=O)CC2)nnc(C)cc1NC1CCCS1 C(CC(O)CNC(=O)C(C1CCCCC1)O)NC(=O)COCCF c1(C(N(CC(C)N(C)C(C2CCCC2C(C)(C)C)=O)C)=O)ncccc1Cl C1(CCNC(C2C(C=C)C2)=O)CN(C(=O)COCc2ccnn2C)CCS1(=O)=O N1(C(c2cnn(C)c2Cl)=O)CC(NC(c2nncs2)=O)CC1(C)C N1(C(C(COC)C)=O)CCOC(CC2(C(=O)NC3CCCC3)CCCC2)C1 C1(CC(C)NC(C(CC)(C)O)=O)CC2CCC(C1)N2C(C1(CCF)CCC1)=O N1(Cc2c(C)ocn2)CCCC(NC(=O)C(C)Cn2cccn2)C1 c1(C(N(CCC2CCN(C(CCNC(C)=O)=O)CC2)C)=O)cccc(F)c1C(F)F CCC(C)C(O)CC(=O)N1CCN(CC(C)NC(c2ccc(F)cc2F)=O)CC1 N1(C(COCCC)=O)CCN(C(=O)Cc2cccc(Br)c2C)CC1CO N1(C(CC2C(C)CCN(C(Cc3ccn(CC)n3)=O)C2)=O)CC2(COC(=O)C2)C1 C(C(C)(O)CC(=O)NC1CCCC(C(=O)NC2CCC3(CC2)N=N3)C1)OC C(=O)(C#CC1CCC1)N1CC(CCNC(C2(C)CC(C(F)(F)F)C2)=O)C1 Cc1ccoc1C(N1CCCC1CNC(=O)CCNC(=O)CC1CCCCC1)=O N1(C(CCN(CC)CC)=O)CCC2(CC2)CC1C(=O)NC(c1cncn1C)CO c1(C(=O)NCC2CCCN(C(C(CC)COC)=O)C2)cc(F)c(Cl)cc1Cl C1(CC(N2CC(N(C(=O)CCn3ccccc3=O)C)C2)=O)COC(C)(C)CO1 CC1COCCN(C(=O)C(C)(C)C)C1.S1(=O)(=O)CCN1C C(=O)(CCC(=O)c1ccc(Br)cc1)NC(CNC(=O)C(F)=CCCF)CO C(C(=O)NC1CC(F)(F)C1)(C1=CCSC1(C)C)N(CC(N1CCCC1)=O)CC n1(CC)ncc(I)c1NC(=O)Nc1cccc(OC)c1.C1CO1 C1(C(N(C)CC2CCCCC2)=O)CCCCCC1NC(C1CCC(O)CN1C)=O C(=O)(C(C)C(O)C(C)C)N(C1CCN(C(c2cc(CC)[nH]n2)=O)C1)CC C(=O)(CCN=c1ccc(C)c[nH]1)N1C(CCNC(CCCCC)=O)CC(OC)C1 c1(C(=O)NCC(C)CN(C(=O)C(O)C2CCC2)C)cccc(C(C)(C)C)n1 c1(CC)ccccc1C(CNC(=O)CNC1CCCC1)NC(=O)C(C)N1CCCC1 C1(CNC(C2(SC)CCC2)=O)CC2(CC2)CN1C(C1CCCC(CF)C1)=O c1(C(=O)NC2CCCC(NC(COCCCCOC)=O)C2)c([N+](=O)[O-])cnn1C C1(C(=O)NCC2(CO)CCCC2)CC2CC2N1C(=O)Cc1cnns1 c1(C(=O)Nc2cccc(C(=O)NCC3(C)CC3)c2)cc(Br)cc(Br)c1 CCC(CN(C)C)C(=O)N(CCCN(C)C(c1cnn(CCC#N)c1C)=O)C c1(C(N2CC(C)(C(N3CCC(C(C)(C)O)C3)=O)C2)=O)cnn2cccc(F)c12 CN1CC2CN(C(C3C(c4ccccc4)C3F)=O)CCN2C1=O N1(C(c2cnn(CC3CCCCC3)c2)C(=O)NC(C)C)CCOCC(C(C)C)C1 C1(C)(CC(C)C)CCCN1C(=O)CC(c1ccccc1C)N c1(-c2c(C)ccc(CO)c2)cc(C(N2CC(NS(C)(=O)=O)C2)=O)c2cc[nH]c2c1 c1(C(C)NC(c2ccc(C)cc2OCC(F)F)=O)ccc2c(c1)NC(=O)C2 N=c1nc(C(=O)NC2(C(=O)NCC3CCOC3=O)CCCC2)cc[nH]1 C1(NC(C(c2cccnc2)NC(CC(=O)NCC)=O)=O)CC(C)OC(C)C1 C1(CC)CN(C(=O)Cc2ccsc2)CCC1NC(C1(OC)CCCSC1)=O C1(NC(=O)OC)CC2CCC(C1)N2C(c1c(NCc2ccccn2)c[nH]c1C)=O c1(Cn2cc(C(C)NC(c3csc(=N)[nH]3)=O)nn2)c(F)cccc1F CCN=c1[nH]c(C(N2CCOC(CCNC(=O)COC3CC(F)(F)C3)C2)=O)cs1 N1(C(C(C2CCOC2)OC)=O)CC23CCCC2(C1)CN(C(=O)CCP(C)(C)=O)C3 c1(CN2CC(NC(C(CCC)N3CCNCC3)=O)C(C)C2)ccnc(F)c1Cl c1(CNC(C(C#C)(C)C)=O)cc(C#N)ccc1Cl C(CCC(=O)NCc1nc(Cl)oc1C)(C(C)C)NC(C(CSC)OC)=O C1(C(=O)NC2C(CNC(=O)C=Cc3cncc(F)c3)CC2)CCn2nncc2C1 CC(CCCC(=O)N(c1ccc(O)cc1)C)NC(=O)C=CCO c1(CNC2(CC(=O)OC3CCN(C(C)=O)C3)CCC2)cccc(F)c1C c1(CCC(=O)N(C2CCN(C(C=CC)=O)C2)CCC)ccc(O)cc1 c1(N2CCC(O)(C(C)NC(C(C)=C3CCC3)=O)C2)nccc(C)c1[N+](=O)[O-] N1(C(C2CC3(CCN(C(C4C(C)(C)C4)=O)C3)C2)=O)CCC2C(=O)NCC2C1 c1(C(N2CC(CCCCOC)C2)=O)nc(C2CC2)oc1C C1(NC(C2(CNC(C3CCC(=O)O3)=O)CC2)=O)C(CC2CC2)CCC12CCC2 c1(C(N(CCCn2cc(CCCN)nn2)C)=O)nc(=N)cc[nH]1.n1(CCC)ccnc1 C1(C(N(CC(=O)NC(C)Cc2cnc[nH]2)C2CC2)=O)CC2(CC2)C1 c1(C(CN(CC(=O)OC)CC)C(=O)OC)ccc([N+](=O)[O-])cc1 Cc1nccc(F)c1C(N1CCC1C(=O)Nc1sc(-c2ccccc2)cc1Br)=O N1(C(CCC(=C)Cl)=O)CCN(C(c2cn3c(n2)SCC3)=O)CC1C Cc1oc(=O)oc1CS(=O)(=O)CCc1ccc(OC(F)(F)F)nc1 CC1SCCCC1C(=O)NCCC1CC(C(=O)NOCC2(C)CCC2)C1 c1(C(N2CC3C(CNC(=O)Cc4ccsc4)C3C2)=O)c(Cl)ccc(Cl)c1O C1(CC(N2CC(O)(CN(C)C(c3ccn(C4CCC4)n3)=O)C2)=O)CCOC1(C)C N1(C(CSc2cccc(C)c2)=O)CCN(C(c2sc(C)nc2C)=O)C2CC12 c1(C(N2C3C(NC(C(CCOC)OC)=O)CC(C3)C2)=O)ccc2ccccc2c1 N1(C(CN2CCC(C)CC2)=O)CC(C)(C)OC2(C1)CN(C(C1OCC1(C)C)=O)C2 c1(C(=O)NCC(C)Sc2ccccc2)csc(=NC2CC2)[nH]1 C1(C(=O)NCc2cc(C)[nH]n2)CC(C)CN(C(c2occ3c2CCC3)=O)C1 CN1CC2CCN(C(c3csc4ccccc34)C(=O)NCC3CC3)C2C1 N1(C(c2nccc(OC)c2)=O)CC(CC(=O)NC2CC(N(C)C)C2)C2(CC2)C1 N1(C(C2(OC)CCSCC2)=O)C2CCCC1CC(NC(=O)CN1CC=CC1)C2 S(=O)(=O)(c1ccc(NCC23CCSCC2C3)c(F)c1)N(CCC)CC N1(C(C(CC2CC2)OC)=O)CC2CC1(C(=O)NC1(CCCCO)CC1)C2 N(C1c2ccccc2CC1NC(=O)CCc1ccc(F)nc1)C(C1(OC)CC1)=O N1(C(CC2(NC(C)=O)CC2)=O)CC(CN(C)C(C2(O)CCSC2)=O)C2(CC2)C1 C(=O)(NN1CCCCC1C)c1cccc(N(CC(F)F)CC)n1 C1(C)(CNC(C(COC)C)=O)CCCN1C(c1cnn(C2CCCC2)c1)=O c1(NC(c2ccc(F)cc2)C)ncccc1S(=O)(=O)NCc1nocc1C1CC1 N1(C(c2c[nH]c(=N)o2)=O)CCC2C(C1)CN2C(C1CCS1(=O)=O)=O c1(C(C(=O)NCC2CCCO2)N(C2CCCC2)CCC)cc(C)c(Br)c(Cl)n1 C=C(C)CCCC(=O)N1CC(NC(C2CCCN2N=O)=O)CCC1C N1(C(COC(CC2N(C(=O)OC(C)(C)C)CC(F)C2)=O)=O)CC2CC(O)C2C1 c1(C(N(C)CC2(CNC(c3c(COC)ccs3)=O)CC2)=O)cnn2c1OCC2 c1(-n2cc(SC)nn2)ccc2[nH]c(C(=O)N(CC(C)(C)C)C(C)C(C)C)c(C)c2c1 CC(CN(C)C)CCC(=O)NCC1CC2CCC1N2C(c1ccc(Cl)nc1O)=O c1(C(=O)N=c2cc[nH]c(CCCO)c2)cnc2cccc(Br)c2c1 C1(NC(c2c(C(C)(C)C)nsc2N)=O)CC2CC1CN(C(c1ccc[nH]1)=O)C2 c1(C(=O)NC2CN(C(c3c(C)cn(C)c3)=O)C(C)CC2)cn(C)c2ncccc12 C(CCCCC(=O)N1CCC1CNC(=O)C(F)(F)CCn1ccnn1)OCC C1(C(=O)NC2C(C)CN(C(C3CCOCC3)=O)C2)CCn2ccnc2C1 Cc1ccc2cc(C(=O)NC3CC(CCNC(=O)C(C)CS(C)(=O)=O)C3)[nH]c2c1 C(=O)(CCN(C(C1CC1F)=O)CC)N(CC#C)CC C(=O)(C(F)C1=CCCCC1)NCC1CCN(C(C2CCCCN(C)C2=O)=O)C1 C1(C(N2C(C=C)CC2)=O)CC(O)CN1C(c1c[nH]c(C#N)c1)=O c1(C(=O)NCC2C(NC(COCCC=C)=O)COC2)cc(N)ccc1F C1(C(=O)NC2C(SC)CN(C(c3coc(SC)c3)=O)C2)COc2ccccc2C1 c1(C(=O)NCC2(O)CCN(C(c3cnc(Cl)[nH]3)=O)C2)nc[nH]c2nccc1-2 C(=O)(C1CCc2ccccc21)NC(CNC(C(C1CC1)OCC)=O)CC(C)C C(c1nc2ccccc2o1)=CC(=O)NCC(CO)NC(=O)COCC1CC1 N1(C(CSCC#C)=O)CCN(C(=O)CNS(=O)(=O)CCCOCC)CC(C)(C)C1 N1(C(C(CC)OC(C)=O)=O)CC(C)(C)CC1CNC(=O)CCOC1CCCCC1 C1(C(C)(C)NC(CSCC#C)=O)CCN(C(C2CCCCO2)=O)CC1 C1(C(N2C(C(=O)OCC)C=CC2)=O)CN(C(=O)CC(C)CN(C)C)CC1F C1(CCNC(C2CC2c2cccnc2)=O)CCCN(C(C2CC2C(=O)O)=O)C1 N=c1[nH]c2c(s1)CCCC2C(=O)N1CC(CNC(C2(CN)CCCC2)=O)C1 c1(OC)ccc(C(C(=O)NC(C)C)N(CC(C)(CO)CO)C)nc1OC c1(NC(N2CCOC(C)C2)=O)cncc(-n2ccnc2)n1.C1(O)CC(F)(F)C1 N1(C(COCCOCCOC)=O)CCN(C(C2CC23CC(O)C3)=O)CC1CF c1(C(=O)NCC(=C)CCNC(C2CC2C(C)(C)C)=O)ccc(-c2cc[nH]n2)cc1 N1(C(c2c(OC)cc(OC)cc2)=O)CC(NC(=O)C(C)CN)CC2(CCC2)C1 C1(NC(=O)Nc2c(F)cc(C)c(F)c2)CCOC2(CCSCC2)C1 N1(C(C(C)(F)F)=O)CCC2(CC1)COC(CNC(C1CC13CCC3)=O)C2 c1(SC)ccc([N+](=O)[O-])cc1C(N1CC2NCC1(C)C2)C(=O)OC c1(C(C)C(=O)NCC2(NC(c3ccc(F)cc3)=O)CCOC2)nc(F)ccc1Cl O(CP(C)(C)=O)CC(=O)NC(C1CCCCC1)CNC(C1C(CCC)C1)=O c1(C(N(CCNC(c2scc(C(C)=O)c2)=O)C)=O)n[nH]c2c1CCCC2 c1(CC(C(N)=O)NC(C2C(NC(c3c(C)scc3)=O)CCC2)=O)ccc(O)cc1 C(=O)(C1=C(Cl)CCC1)NC(C(C)NC(=O)CN1CCC(C(N)=O)CC1)CO N1(C(CCc2onc(CCC)n2)=O)CCC(NC(c2snnc2C)=O)C(F)C1 c1(SCC(=O)NCC2C(C(=O)NC(CSCC(=O)OC)=O)C2)nc(C)cc(C)n1 C(=O)(C(C(C)(C)C)NC(N)=O)N1CC(c2cn(Cc3nc(C)sc3)nn2)(F)C1 C1(C(=O)NCC(=CC(N2C(CCC)COCC2)=O)C)CC(C)(C)CN1C c1(C(=O)NCC(CNC(CC(C=C)CC)=O)O)cc(Cl)c(C)cc1Br C1(N(C(c2cn(CCCC)nn2)=O)C)CCCN(C(C2(SC)CC2)=O)CC1 c1(OC)cc(C(N2CC3CC2C3C(=O)NC(CO)C(C)C)=O)c([N+](=O)[O-])cc1O C12(C(=O)NC3CN(C(c4c(C)sc(C(F)(F)F)n4)=O)CC3C)CC1COC2(C)C c1(NC(c2c(OC)c(F)ncc2)=O)nn(C)cc1C#C[Si](C)(C)C C(C)(CC(=O)NCC1CCCN1CC(=O)N(C)C(c1nc(C)no1)C)OC N1(C(C2CCN(CC)CC2)=O)CCN(C(c2coc(Cl)n2)=O)CC(CO)C1 N1(CC)CCOC(C(=O)NC2CC(CNC(c3c(C)cnn3C)=O)C2)C1 N1(C(CC2(C=C)CCC2)=O)CCC(C)(NC(=O)C(c2ccccn2)C)C1 c1(SCC(=O)NC2CC(NC(C=C3CCC(C)C3)=O)C2)ccc(F)cc1Br C(=O)(C1=CC2CCC(C1)N2)NC(C(=O)N(C1CC(CC)C1(C)C)C)=O c1(C(=O)NC2(C)CN(C(c3ccn4nccc4n3)=O)C2)cc(O)c2ccoc2c1 N1(C(C2N(C)C(=O)OC2)=O)CCS(=O)(=O)C(CCNC(c2ccc(O)nc2)=O)C1 CC(C)C(F)(CNC(C1C=CCS1)=O)C(=O)NCC1(c2ccon2)CC1 C1(C(N2CCC(CC(C)NC(C(=O)NCC)=O)CC2)=O)CS(=O)(=O)CC(=O)N1 C(CC(C)C(=O)NCC1CC1NC(c1cnc(C2CC2)o1)=O)=CCC Cc1ccc(C(C)CC(=O)NCC2(C)CCN(C(=O)C(F)(F)C3CC3)C2)cc1 C1(NC(C2c3nnc(CC)n3CCC2)C)CCCC(C2CCC2)C1 c1(CCC)cc(C(N2CCC(CN(C(=O)C3=CCCC3)C)C2)=O)sc1C c1(C(=O)NCC2C(NC(C=C(CCC)C)=O)CC2)cc2c(C)ccc(Cl)c2[nH]1 c1(NC(c2c(NC(C3(O)CCOCC3)=O)ccs2)=O)cc(Cl)cc2[nH]ncc12 N1(C(C2(CC)CCCN2C(c2nc3ccccc3[nH]2)=O)=O)CCCC(C)(C)CC1 c1(CC(C(=O)NC(=O)N)C2CC2)ccc(O)cc1.c1(C(C2CCC2)N)ccccc1 C(=O)(CCS(C)(=O)=O)NC1CC(N(C)C(c2n[nH]cc2Cl)=O)C1 C(=O)(C1=CC2(CN(C(c3csc(Cl)c3)=O)C2)OC1)N1CC(C)(C(F)(F)F)C1 C=CCC(CNC(=O)CCCC(OC)OC)C(=O)N1CC(COC23CC(C2)C3)C1 O=C(CCN=c1[nH]c(=NCCCF)[nH]c2c1CCCCC2)Nc1ccccc1 N1(C(CC=CCC)=O)CCC(NC(c2coc(S(C)(=O)=O)c2)=O)C12CCC2 Cc1nc(F)ccc1CNC(=O)CC1CCCC1NC(C1CC(O)C1)=O C1(CNC(C(c2ccc(Cl)cc2)OC)=O)CCC(C)(C)CN1C(c1ccoc1)=O c1(N2CCCC(CC)C2)nc(C)cc(=NC2CN(C(=O)C(F)C(C)(C)O)C2)[nH]1 N1(C(c2c(SCC)nccn2)=O)CCC2C1CCCN2C(=O)CCC(C)(F)F N1(C(c2c(C)occ2)=O)CC(NC(=O)C=Cc2ccc[nH]2)C(C2CC2)C1 CC(C)(F)CCC(=O)NC12CC(C(N3CC(CF)OC(CF)C3)=O)(C1)C2 N(C1CCOc2ccc(Br)cc21)S(=O)(=O)c1cccc(N2CC3CSCC3C2)n1 n1(C(C)(C)C)nccc1C(N1CCC(OCCNC(=O)Cc2csnn2)C1)=O C1(CNC(Cc2cccc(OC)c2)=O)C(C)CCCN1C(c1coc(Br)n1)=O C1(NC(CCC(C)(F)F)=O)CN(C(=O)CC2CCCCC23CC3)C2(CCCC2)C1 C1(NC(c2cccc(N)c2O)=O)CCCCCN(C(=O)CCCC2CCCC2)C1 N1(C(CN2CCCC(CC)C2)=O)CC(NC(c2cn(C)nn2)=O)CC(C)(C)C1 c1(C(C(N2CCCC(NC(CC)COC3CC3)C2)=O)=O)cccc2c1OCC2 Cc1oc(Br)cc1C(N1CCCC1C1(NC(C2CC2F)=O)CC1)=O C(=O)(CC(F)(F)C(F)F)NCCC(C)N(C)C(C1C(F)(F)C12CC2)=O C1(NC(=O)OC(CC(C)C)C)CC2(C1)CN(C(=O)CN1CCCC1)C2 N1(C(C(C)C#N)=O)CCC(NC(C23CC2C3)=O)C(C)(C)C1 C(=O)C1=CCC2(COC2)OC1.Cc1nc(C(C)N(C)CCN(C(C)=O)C(C)C)n[nH]1 N1(CCN(C(C2(CC)COC2)=O)C)CCN(C(=O)COCC(C)C)CC1 N1(C(c2cc(C)c(Cl)cc2)=O)CC2OCCN(C(=O)CC3CCCN(C)C3)C2C1 C1(C(=O)NC2CCCCC2CNC(=O)COCCC(C)C)(OC)CCOCC1 CC(CN(C)C)CCC(=O)NCCCN(C(C1(F)CCN(C)CC1)=O)C1CC1 C(=O)(CCCSc1ccccc1)N1C(CNC(c2ccsn2)=O)CC1 c1(C(N2CCN(C(C3C(F)(F)C34CC4)=O)CC2)=O)nnn(C2CC2)c1C(F)F c1(NCC2C(O)CCC(C)(C)C2)[nH]c(=NCc2nc[nH]c2Br)nc2sccc12 C1(CNC(CCC(CC)C)=O)CN(C(=O)Cc2ccnnc2O)CCC1(F)F c1(OC)cc(CC(=O)NC(C)(C)C(C)NC(=O)CCc2ccsc2)c(F)cc1O CP(C)(=O)C1CCC(NC(=NCCCOc2ccc(C#N)cc2Cl)NCC2CC2)C1 C(CCC(c1ccccc1)NC(=O)Cc1cnco1)NC(CSCC=C)=O C(C(=O)NC1CC1)(C1CCSC1)N(C)CC1(C)CC1 C=CCC(C)(C)C(=O)NCC1CN(C(=O)C(F)(F)CO)CC1(F)F C1(C(C)C(=O)NCF)CCCN(C(=O)C(C)(C)N(C)C)C1 C(=O)(CCCC(=O)NCC)NCCCC1OCCN(C(C(COCC)C)=O)C1 Cc1cc(C(=O)NC(CNC(=O)C(C)O)C2CCC2)c2cccc(C)c2n1 C1(NC(c2cc(Cl)c(Br)c(Cl)c2)=O)CCc2nc(NC(=O)C(F)F)sc2C1 CC1(C)CN(C(=O)C(c2ccc(Cl)s2)=O)CC1NC(=O)C1=NNC(C(F)(F)F)C1 c1(C(C=C)NC(c2cnc(Br)s2)=O)cc(Br)ccc1C N1(CCCNC(=O)C(O)Cc2cnc[nH]2)CCN(C(=O)CCC2CC2(F)F)CC1 CCCCS(=O)(=O)NCC(N1CCOC(C(C)NC(=O)C(F)(F)CO)C1)=O C1(CNC(c2n(CC)ncn2)=O)CCC(C)N(C(c2cncnc2)=O)C1 C1(N(C(CC=CC)=O)C)CCCCN(C(C2CC=C(C)CC2)=O)C1 C1(CC)C(NC(=O)C=Cc2ncc[nH]2)CCN1C(C1CCS(=O)CC1)=O Cc1nc(=NCC(C)(C2CC2)NC(=O)CCc2ccc(OC(F)F)nc2)s[nH]1 N1(C(C(CCC)C#N)=O)CCC2(CC1)CC2CNC(=O)CCn1cc(C)cn1 N1(C(CC2CC(C)(C)C2)=O)CC(F)(F)CC1CCNC(C1CC1CF)=O N1(C(=O)CC2CCCC23CC3)CC2(C1)CN(C(c1cnc(Cl)s1)=O)C2 C1(C(N2C(C(N(CCCCCC)C)=O)C(O)CC2)=O)CCC2(CC1)CC2 Cc1ccc(C(F)(F)F)cc1CN1CCC(C)(C(N2CCC(O)C2)=O)C1 C1(N(C(=O)C(C)=CC(C)(C)C)CC)CCCN(C(c2ccc(N)c(N)n2)=O)CC1 C1(CNC(CC2CC(OC)CN2C(=O)C#CC(=O)N(C)C)=O)CCC(C)(C)CC1 C1(C2CN(C(C34CCCN3CCC4)=O)C2)(NC(C(CC)N2CCCC2=O)=O)CC1 C1(N2CCN(CC(c3ccsc3)=O)CC2)CCCC2(CC1)CC2 c1(C(=O)NC2CCCN(C(=O)C(F)F)C2)ccc2nc(-c3ccccc3)sc2c1 N1(C(C2(C#N)CC(C)C2)=O)CCC(NC(C2(C)CCCC2)=O)C(C)(C)C1 C1(C(N2CCC(CC(=O)NC34CC(CCC)(C3)C4)C2)=O)CC(=O)N(CCOC)C1 C1(NC(=O)OC(C)(C)C)CN(C(=O)NCCc2cc(Cl)cc(Cl)c2)CC1C1CC1 C(=O)(CC(C(C)CC)NC(c1cncc(OC)n1)=O)Nc1cccc(CC)c1F c1(C(N2CC(CN(C)CC3CCSCC3)C2)=O)ccc(-c2cnco2)cc1 c1(C(N2CCC(CNC(C(C(C)C)N(C)C)=O)CC2)=O)cnn2c(=O)cc[nH]c12 C(N=c1[nH]nc(C(N)=O)s1)C1C(NC(C2(C)CNC(=O)C2)=O)CCCC1 N1(C(=O)C2=CCCCC2)CCC(C2CCCN(C(C3COCCO3)=O)C2)CC1 Cc1ncnc2c1CC(C(=O)NC1(CCNC(=O)C(CO)N(C)C)CC1)CC2 C1(C(=O)NC(C2CC2C(N2CCC=C(C)C2)=O)C)CCCCC(=O)N1 C(=O)(N=c1ccn(CC(F)(F)F)[nH]1)N1CCC(C(C)C)C1 N1(C(=O)Nc2nn[nH]n2)CCC(N2CCCC2)(C(F)F)CC1 C1(O)(C(C)NC(CCCc2scc(C)n2)=O)CCN(C(=O)CSC(F)(F)F)CC1 c1(OC)ccc(-n2nnnc2C(C(C)OC)NC2CCSCC2)cc1 S(=O)(=O)(C1CCOC1)NC(c1cc(C(C)(C)C)nn1-c1ccccn1)=O C1(c2nn[nH]n2)(C(C)C)CCN(C(c2cc(O)no2)=O)CC1.C12CCCN(C1)C2=O c1(OC)ccc2cc(C(N3CC(CNC(=O)C(Cl)=CCl)CC(C)C3)=O)n(C)c2c1 C=CCCC(C(=O)OC)NC(c1cc(OC)c(-c2cc(F)ncc2F)cn1)=O c1(C(C(=O)NCCN(C(CC2N(CC)CCC2)=O)C2CC2)C)ccc(C#N)cc1 N1(C(c2cc(C)[nH]c2)=O)CC2(CC2)CC1C(=O)NCCc1ccon1 CC1CC(C(=O)NCC2CN3CCC2C3)N(C(=O)COc2ccccc2)C1 Cc1ccc2nc(-c3nc(CC4CC4)nn3C(C3CCOCC3)C)cn2c1 CC1CCC2(CCC2)CN1C(=O)CSc1ccc2c(c1)CCC2 c1(OC)ncc(C(=O)NCC2CCCCCN2C(=O)CCNC(=O)CO)cc1C C1(CNC(C2(S(N)(=O)=O)CC2)C)CC2(C1)CC(F)C2 C1(NC(C(CC)NC(C)=O)=O)CC2CC(NC(C3(F)CCCCC3)=O)CC2C1 CCC(C)C(CC(=O)NCCC(C(C)C)OC)NC(=O)C(O)CC(N)=O n1(CC(N2C3CN(C(C(CC(C)C)F)=O)C(C3)C2)=O)ccc2ccc(F)cc12 C1(CNC(c2c(C)snc2)=O)CN(C(c2ccccc2)=O)CCN1C.C1(N)CC1 c1(NC(C2CCC2)C)ncccc1S(=O)(=O)N1CCCC1C1CC1 N1(C(c2c(N)nccn2)=O)CCOC2CN(C(=O)CNc3ncccn3)CC12 c1(C(N2C(CNC(=O)Cc3csc(-c4ccsc4)n3)CC2)=O)cccc(F)c1F Cc1nc(CC(C)C)c(C(=O)NC(C)C(CO)NC(=O)CSC(F)(F)F)s1 N1(C(C(C)=CC)=O)CC2CCN(C(=O)C(c3ccccc3S(N)(=O)=O)C)CC12 n1(CC)ccnc1C(=O)NCCCCCN(C(=O)CC1CC1(Cl)Cl)C c1(C(=O)NC2C(NC(C(C)C(C)O)=O)COCC2)c[nH]c2ccncc2c1=O C1(CC(=O)NCCCN(C(=O)CC(C)N2CCCC2=O)CC)CCCC(C)(C)O1 C(CC1=CCN(C(C2(C(F)F)CCCC2)=O)CC1)NC(C1C(OC)CCCC1)=O C(=O)(CC(=O)NCC(CNC(=O)CC1CCCOC1)CO)OCC c1(OC)cccc(C(C)=CC(N2CCN(C(c3ccc(C)s3)=O)C(C)C2C)=O)c1 CN1CCC12CN(C(C13CC(CN1C(C1CCCCC1(C)C)=O)C3)=O)C2 N1(C(=O)C2CC2)CCNC(c2ccc(Br)cc2)C1.C12CCCCC1N2CC(F)(F)F N1(C(CC2CCC(C)(C)CC2)=O)CCCC12CCCN(C(C1CC(CF)C1)=O)C2 c1(CC(=O)NC(CC2CN(C(C(C=C)(F)F)=O)C2)C)ccc(Cl)c(OC)c1 N1(C(C(C)OCC)=O)CCC(NC(c2cnc(F)c(Cl)c2)=O)C(CC)C1 c1(C(=O)NCCC(C)NC(C2CCOC2C(F)(F)F)=O)ncc(C(F)F)s1 N1(C(CC=CC(=O)N(C)C)=O)C(CNC(C2CC2(C)C)=O)CC2CCCC12 CC1CN(C(=O)Cc2cc(Br)ccc2O)CCN1C(c1cc(F)nc(F)c1)=O C(CCS(C)=O)(C(=O)N1CC2(C1)CN(C(C1(c3ccncc3)CC1)=O)C2)N(C)C c1(OC)ccnc(C(=O)NC(C)(C)CN(C(=O)C(O)CC(C)C)C)c1OC N1(C(c2c(CC)onc2C)=O)CCN(C(=O)C(C)CF)C(c2ccccn2)C1 N1(C(C2(OC)CCOCC2)=O)CCC(C(F)(F)F)C(NC(c2[nH]cnc2C)=O)C1 C1(C)(COC)CN(CCCc2cn(CC3CCCC3)nn2)CCO1 C1(NC(c2c(F)cncc2Br)=O)CN(C(=O)CC2CCC2)CCC1F C(C(CNC(=O)CCc1nnc(S)n1C)C(F)(F)F)NC(C1(N(C)C)CC1)=O c1(C(=O)NC(C)CN(C)C(C2CCC(=O)N2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NC(C)CN(C)C(C2CN(C3CCC3)C2)=O)ccc(CO)s1 c1(C(=O)NCC(C)(CO)NC(CC2(COC)CC2)=O)cccc2nc(C)nn12 c1(C(=O)NCCC(C)NC(c2cccc(C(C)C)n2)=O)ccc2c(c1)COCO2 Cc1ccc(Br)c(F)c1CNC1CCC(=O)N(C)CC1 c1(C(=O)NCc2nc(CNC(CCC#C)=O)sc2)cnn(C(C)CC)c1C Cc1ccc(C)c(C(=O)NC2(CNC(=O)C3=CCSC3)CCC2)c1 c1(CC(=O)NCC(=O)NC(CN(C(N2CCCC2)=O)CC)C)cnc(C)o1 C(C(=O)N(C)OCC)NC(c1nc(OCC)oc1)=O.N12CCC(C1)C(C)C2=O N1(C(C=NOC)=O)CC2CC(NC(C3(C4CCOCC4)CC3)=O)CC2C1 C=CC(C(=O)N(C1CCN(C(c2csnc2C)=O)C1)CCO)c1ccccc1 C1(C(=O)NCC(CO)NC(CCNC(C=CC=CC)=O)=O)C(CN(C)C)C1(C)C N1(C(CCSCC)=O)C(C(=O)NCC2CCCSC2)CC2CCCC12 c1(C(N2CCC(N(CCC)C(c3cn(C)nc3CC)=O)C2)=O)c(C)cncc1C c1(C(N(CC(C)N(C(=O)C(N2CCOCC2)C)C)C)=O)csc(S)n1 C1(C)(C(=O)NCC(C(C)C)NC(C=C(C)Cl)=O)CC(C)(C)C1 Cc1ccc(CC(C)NCC2CC(C(=O)OC(C)(C)C)C23CCC3)nc1O CC(C)C1=CCC(C(=O)NCCC2CC(NC(C3(C)CCCOC3)=O)C2)CC1 c1(CC)oc(C)cc1C(=O)NCc1nnn(C)c1C(=O)NCC1CCCSC1 Cc1cn2ccc(C(=O)NC3COCC3NC(C3(OC(C)C)CCC3)=O)cc2n1 c1(C(=O)NC(C(C)NC(c2c[nH]cc2-c2ccccc2)=O)C)ccc(Cl)cc1O C(=O)(CCCC(=O)NC1CCCC1)NC1C(NC(Cc2n[nH]c(=NC)s2)=O)CC1 C(CCCN=[N+]=[N-])NC(C1N(C(CC2CCC(C)O2)=O)CC1C)=O O=C(C#CC1CCOCC1)NCC1(NC(C2CCCC3(CCC3)O2)=O)CC1 C#CCC(C)(C(=O)N1CCCC1CNC(C)=O)NC(=O)CC1CCOC1(C)C c1(C(=O)NC(CC=C)CNC(=O)COC2CCC2)ccc2cc(Cl)ccc2c1 C(=O)(C(C(C)C)NC(=O)CC(C)C)NC1(C(=O)NC2C(OC)C(O)C2)CCC1 c1(C(=O)NCCN(C(c2cc(Cl)no2)=O)CC)cc(C(F)(F)F)ncc1N N1(C(C(c2cccc(Cl)c2)C)=O)CCC(NC(=O)Cc2n[nH]cc2Br)C1C c1(CC(=O)NCC(O)CCNC(c2ccc(C(F)F)nc2)=O)cncnc1O N1(C(C2(OC(C)=O)CC2)=O)CCC(F)(C(=O)NC2(C3CCCO3)CC2)C1 c1(NC(NCCCN(C2(c3ccccc3)CC2(F)F)C)=S)ncccc1O c1(C(=O)NCCCCCNC(C(C)Cn2cccn2)=O)cnc2c(ccn2C)c1 c1(C(=O)NCC(CC(C)C)NC(C2(C)CC=CCC2)=O)c(F)ccnc1Cl C(=O)(C#CC(C)(C)CNC(C1CCC(C2CC2)C1)=O)N1CC(C)C(C(N)=O)C1 N1(C(CN(CCOC)C)=O)C2CCC1CC(CC(C)NC(=O)C(C1CC1)SC)C2 CC(=O)CCC(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cnsc1)C C1(c2n(CC)ccn2)OCCCC1C(=O)NCC1COCCN1C(=O)CC1CC1 c1(OC)cccc(C2CC(O)CN2C(=O)C(N)Cc2cn[nH]c2)c1 N1(C(c2ccc(C#N)cc2)=O)CCC(C2CCCN(C(c3ccoc3Cl)=O)C2)C1 N1(C(c2ccc(CC)o2)=O)CCC(NC(c2cnn(C(C)(C)C)c2Cl)=O)C1C C1(CN(C(=O)CSCCC#N)C)CCCN1C(=O)CCc1ccncc1 c1(NC(C2SCCN(Cc3c(C)cc(Br)cc3C)C2)=O)ccc(Cl)c(C#N)c1Cl C(CC1CCCCC1)(C(=O)NC(C)(CNC(c1coc(C(N)=O)c1)=O)CO)OC Cc1cc(C(=O)NCC2CN(C(=O)C(c3ccn(C)n3)C)CC2(F)F)cc(F)c1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NCC1(F)CCC(NC(C(C)N(C)C)=O)C1 N1(C(=O)C(c2cc(F)ccc2F)=O)CCC(C)C(CNC(C2(CC)CCOC2)=O)C1 C#CC1(C(=O)NC(C)COC)CCN(C(c2ccc(C(C)C)o2)=O)C1 C(C(C(=O)N(C)C(c1nccs1)C1OCCO1)n1cc(CO)nn1)OCC C=C(C)CCC(=O)NCC(C)(C1CC1)NC(=O)CN(C(=O)OC(C)(C)C)C1CC1 C1(C(N2CCC(=CCNC(CCCN(C)C)=O)CC2)=O)CCc2ccnn2C1 N1(C(c2c(NC(C)C)cccn2)=O)CCN(C(c2ccco2)=O)C2CC12 c1(-n2cc(C(c3cc(C(=O)OC)cc(C(O)SC)c3)=O)nn2)cnn2c1OCCC2 c1(CC(=O)NCC(CC)NC(=O)CC2CC3CC3C2)cnn2ccccc12 C1(NC(CCc2onc(C)n2)=O)CC2CN(C(c3nc(Cl)oc3C)=O)CC12 C=C(CNC(c1csc(C(C)C)n1)=O)CCNC(=O)C(C)C1CCOC1 C(C1=Cc2ccccc2OC1)=CC(=O)NC1CN(C(C2CCC(F)(F)CO2)=O)C1 C1(CC(N2CC(O)(CN(C)C(C34CCC(CO3)C4)=O)C2)=O)CCC(=O)NC1=O C1(CN=C(NCC2(OC)CCC2)NCC(F)F)CCOC2(CCOC2)C1 c1(CC(=O)NC2C3CCN(C(C(C)SC(F)(F)F)=O)C32)ccnc(Cl)c1F N1(C(C(N)CCSC(F)(F)F)=O)CCCC(c2ccncc2)CC1 N1(CCC)CCC(C(=O)NC2CN(C(=O)CN(C)C(C)C)C3CC23)CC1 c1(CC)oc2ccccc2c1C(N1CCOC2(C1)CN(C(=O)C(C)(F)CC)C2)=O C#Cc1ccc(C(=O)NCC(C)(O)CNC(=O)CN2CC(=O)N(C)C2=O)cc1C CCCC(C(=O)OC)C(=O)N(CC(O)CN(C(=O)COCCF)C)C N1(C(CC2CN(C(C)=O)C2)=O)CCC2(CC2C(=O)N(C2CCCCCC2O)C)C1 CCC(C)C(O)CC(=O)NCCCCC1CN(C(c2cc(CCCO)on2)=O)C1 c1(C(=O)Nc2cncc(C(N3CCC(N(C)C)C3)=O)c2)ccc(Br)c(F)c1 Cc1ocnc1CCNC(=O)C(c1ccnn1C)NC(=O)COC1CC=CC1 c1(CC(=O)NCC(CC)NC(c2nocc2Cl)=O)csc(C2CCOCC2)n1 C1(N(C(CNC(CC)=O)=O)C)CCCN(C(c2cc(Br)c[nH]2)=O)C1 Cc1cc(F)cnc1NC(c1nc(C(=O)Nc2cnc(C)c(F)c2)cs1)=O c1(C(=O)OCC(=O)NC(C(=O)NC)C)cc(C)nn1CC(F)(F)F CC1CN(C(=O)CCF)CCN1C(C1CCCN1C(c1ccccn1)C1CC1)=O C(C)(CCNC(C1(OC)CC1)=O)N(C(C=C(CC)C)=O)C N1(C(C(C)S(N)(=O)=O)=O)CCC2C1CCCN2C(c1nccc2n[nH]cc12)=O C1(CNC(c2cc(OCC)ns2)=O)N(C(C2CC(C)=NO2)=O)CCCC1(C)C C(=O)(C1CCc2c[nH]nc21)NC1(C)CCN(C(CSCC(=O)OC(C)(C)C)=O)C1 CC1CC2(CO1)CN(C(c1ccc(CNC(=O)C(C)(C)CCF)o1)=O)C2 O=C1CSC(C(N2CCC2C(N2CCC(n3ccnc3)C2)=O)=O)C1 Cc1cc(Cl)ncc1S(=O)(=O)N1CCC2CN(C(=O)NC(C)(C)C)CC2C1.C(C#N)O CCC(CC(=O)NCc1ncnn1C1CC1)NC(=O)CC1OCCO1 CCCCS(=O)(=O)CC(=O)N(C)CC1(O)CCN(C(c2ccccc2CO)=O)C1 CC1(C)CN(C(=O)Cc2ccccc2O)CC1NC(=O)C(O)Cc1ccccc1 CC(C(=O)NC1CCN(C(=O)Cc2nc(C3CC3)nn2C)C1C1CC1)C(C)(C)C Cc1ccc(C(N2CC(CC(=O)NC3CC(C)OC(C)C3)C3(CC3)C2)=O)c(O)c1 Cc1nc(C(N2CC3CC2CC3N2CCCC(C(C)(C)O)C2)=O)ccc1Br N1(C(C(CSC)C)=O)CC(NC(=O)C(C2CCCCC2)O)C(CC(C)(C)C)C1 c1(C(N2Cc3cccnc3C2)C(=O)NCCCC2CC2)nc(Br)c2ccccn12 c1(C(N(C(CCNC(c2cc(CC)[nH]n2)=O)C)C)=O)ccc(C(C)=O)cc1 C(CC(=O)N)OCCOCCCC(F)(F)F.C(CCN(C(=O)C)C)OCCOC N1(C(c2cccc(OCC)c2)=O)CCC(C)N(C(c2c[nH]ccc2=O)=O)CC1 c1(NC)cnncc1C(=O)NCC1CCC1NC(C1(F)CC1)=O c1(C(=O)NC2CCC(C)N(C(=O)COc3cn[nH]c3)C2)cncc2ncn(C)c12 c1(C(N(C(CC)CO)C)=O)c[nH]nc1C1CCN(C(=O)C(C)C)C1 c1(C(=O)NC2CN(C(CCOC)=O)CC(O)C2)nn(C)c(=O)c2ccccc12 C(=O)(C(CNC(c1ccc(F)cn1)=O)CC1CCCC1)N(CCCF)CC C1(C(=O)N(CCC(C)(C)NC(=O)CSC(F)F)C)(OC)CCSC1 c1(C(=O)NC2CCC2NC(C2CCS(=O)(=O)C2)=O)cnc2nccnc2c1 C1(CC(=O)NCCC(C)(C)NC(c2cc(OC)n[nH]2)=O)CCCCN1C c1(C(=O)NCCOCCCNC(c2c(CC)noc2)=O)[nH]cc2c1CCCC2 N1(C(c2cncc(OCC)c2)=O)CCCC2(CCC(NC(=O)CC(F)(F)Cl)C2)C1 CCC(CC(=O)NC(C)C(C)NC(=O)COC1CN(C(C)=O)C1)SC C1(C(=O)NCC(C)CNC(=O)CCc2cn[nH]c2)C2CCN(C)CC12 c1(OCC(N2C(CNC(C(C)OC)=O)C3CC3C2)=O)cccc(F)c1F c1(C(N)=O)ccccc1-n1ccc(-c2cnc(C3CC3)nc2)n1 N1(C(c2cc(SC)oc2C)=O)CCC=C(CNC(=O)CC(C)(C)CN(C)C)C1 c1(C(N)=O)cccc(C(=O)NC2CN(C(c3csc(F)c3)=O)CC2C(F)F)n1 C1(C(=O)NC(C)CNC(=O)CCc2cnco2)CCC(=O)N1 CC1(C)CC(NC(C23CSCC2C3)=O)CCO1.C12(CCCCC1)C(=O)NO2 C1(CCC)(NC(c2nn(C)nc2Br)=O)CCNC1=O N1(C(c2c(C3(C)CC3)c[nH]c2)=O)CC(C)(C)C(NC(=O)C(Cl)=CCl)C(C)(C)C1 C(=O)(C(CNC(=O)CC1CC1(C)C)CC1CCCC1)NCCSC N1(C(C2CC(SC)C2)=O)CCCC(C)(C)C1CNC(c1cncn1C1CC1)=O C1(CCNC(C2(CCNC(c3n(C)nnc3)=O)CC2)=O)CCC(C)(C)O1 CN=S(=O)(c1ccc(C(=O)OC)cc1)N(C)C.C12CCC3(CC(C3)C(=O)NC1)O2 Cc1cccc(F)c1C(=O)NC1CN(C(=O)Cc2ccc(F)cc2)CC1CO c1(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)C(F)(F)F)cccc2c1COC2 c1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)N(C)C)C2)n[nH]c2c1CC1CC21 O=S(=O)(c1cnc(NCc2sncc2Br)c(Cl)c1)N1CCCC2(C1)OCCO2 CC1CCN(C(c2ccc(CCC(=O)Nc3cnn(C)c3)[nH]2)=O)CC1(F)F Cc1ccc(C(N2CCC(C)(NC(c3cc4sc(C)nc4[nH]3)=O)C2)=O)c(F)c1F c1(C(=O)NCC2N(C(c3cn(C)nn3)=O)CCC2)cncc(N)n1 C1(CNC(C(CC#C)C2CC2)=O)CCN(C(=O)CCCCC)CCC1(F)F C(=O)(CCCCCCNC(C1CC(=O)CC(=O)N1)=O)NC(C(CC)C)C(=O)NC n1(CCOCC)nc(-c2cccc(CC)c2)nc1-c1cnc(-c2ccco2)s1 c1(C(N2CC3CC(O)CC2C3)=O)cc(Br)c2nccnc2c1 N1(CC(=O)N(CCNC(C(C(C)SC)O)=O)C(C)C)C(=O)CCCC1=O N1(C(C2C(CC)CCO2)=O)CCCCC1CCC(C)(C)NC(=O)Cc1cnoc1 CCC(C)C(C(=O)N1CCCC1CNC(C1OCCC1C)=O)N(C)C N1(C(c2cc3n(n2)CCC3)C(=O)NCCOC)Cc2ccc(OC)cc2CC1C c1(C(=O)NCCC(C)N(C(C(CC)OC)=O)C)cc2cc(F)cc(F)c2[nH]1 N1(C(c2cccc(C)n2)=O)C2CCC1CC(NC(C13CCC1C3)=O)C2 c1(C(N2C(CN(C)C(c3nnsc3N)=O)CCC2)=O)ccc(O)nn1 C1(NC(c2cccnn2)=O)CCCC12CN(C(c1cc3nc[nH]c3cn1)=O)C2 C1(CNC(c2c(C)cns2)=O)CCCC(NC(c2ncnn2C2CCOCC2)=O)C1 C1(C(=O)NCC2(O)CN(C(C3C(OC)CCCC3)=O)C2)CCC(N=[N+]=[N-])C1 C(c1nc2ccccc2[nH]1)=CC(N1C(CNC(C(C(C)C)(C)O)=O)CC(F)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(CCC=C)=O)CC(F)(F)F Cc1cn2c(C(C3CCCC3)NC3CN(C(=O)C(C)CC(N)=O)C3)cnc2s1 c1(C(=O)NCCC2CN(C(C(CCC)C)=O)C2)ccnc2cc[nH]c12 C1(C(NOCCOCC)=O)CN(C(=O)C(C)(C)CF)CC(C)O1 c1(C(=O)NC2C(NC(CCCC)=O)CCC2)ccc(C(C)C)cn1 c1(OC)cccc2ccc(C(=O)NCC(C)NC(c3cc(=O)n(C)cn3)=O)nc12 CC1CN(C(=O)CCc2nncs2)CC1(C)CNC(=O)C(c1cccn1C)=O C1(CCc2ccncc2)(NC(N2CCCC2)=O)CN(C(=O)COC2CCOC2)C1 C1(CNC(CC(C)OC)=O)CC2(CCOCC2)CN1C(c1ncccn1)=O N1(C(CC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)C1Cc2c(Cl)cccc21 O=S(=O)(c1cc(Cl)c(I)s1)N1CCCC1c1cc(F)c(F)c(F)c1 C(CC(CC)C(=O)N(CCCCN(C(=O)CC(C(F)F)n1ccnc1)C)C)=CC C1(C(=O)NC(C)CCO)CCCN(C(c2cc(Cl)c(Cl)s2)=O)C1 Cc1cc(C(=O)NC2(C)CCC(NC(c3ccon3)=O)CC2)cnc1O C1(C(N2C(C(=O)NC3CC(C)(CC)C3)C3CC3C2)=O)CC2OC1C1CC21 c1(C(N(CCCNC(c2cnn(C(F)F)c2)=O)CCO)=O)ccc2c(c1)CCO2 N1(C(Cc2c(C)n[nH]c2C)=O)CC2CCN(C(C3C4CC5C(C4)C35)=O)CC12 C(=O)(C(C)CC(C)(C)C)N1C(CN(C(=O)CC(C)(C)C(F)F)CC)CCC1 C(CCC(=O)N(C)C)NCCNC(C)=O.n1(C)cc(-c2c[nH]nc2C(=O)OC)nn1 CCCC(O)CC(=O)NCCC(C)N(C)C(c1scnc1COC)=O N1(C(C(Cc2cn(C)nn2)NC(=O)OC(C)(C)C)=O)CCCC(c2cccc(F)c2)C1 N1(C(C2CC(C)CN2C(=O)C=Cc2ccccc2)=O)CCC(O)C(C)(CO)C1 Cn1cc(C=CC(=O)NCCCCCC(=O)NOCC2(C)CC2)nn1 c1(C(=O)NCC2(NC(c3cnc(C(C)(C)C)o3)=O)CCC2)cc2cn[nH]c2cn1 C(=O)(C(CC(C)C)NC(c1sc(C)cc1C)=O)N(CCC#C)CC N1(C(c2n(C)ccc2)=O)CCCC2(CCCN2C(C2CCc3c[nH]nc3C2)=O)C1 c1(C(C)NC(CC(C)n2cccc2)=O)ccc(CNC(=O)COC2CC2)cc1 CC(C(=O)N1CCCCC(NC(c2ccsc2C#N)=O)C1)C(F)(F)C(F)F c1(C(=O)NCC2OCCC(NC(C3CCN(C)C3)=O)C2)cc2c(Cl)nccc2o1 C1(CC=C)(C(=O)NCCP(C)(C)=O)CCN(C(=O)C(C)O)C1 C1(NCc2c(OC)nc(Cl)cc2)CC2(C1)CC1(CCCC1)C2 CC1(C)CCN(C(c2cccc(F)c2F)=O)C1CNC(C1(C)CCCS1(=O)=O)=O c1(C(N2CCC(c3c(F)cccc3F)(C)C2)=O)cnc2ccccn2c1=O c1(CC)ccccc1C(CNC(c1ncncc1Cl)=O)NC(c1cc(F)n[nH]1)=O C(C1=CCN(C(=O)CCCSC)CC1)NC(CCc1onc(C(C)OC)n1)=O O=C1CC2CCC1C(C(=O)Nc1cncc(-c3ccc4c(c3)CCO4)c1)C2 C(=O)(CCCCC(=O)NCC1CC1NC(=O)COCCc1cccs1)OC c1(N(C)CC2CN(S(=O)(=O)Cc3ccc(Cl)c(Cl)c3)C2)cccc(C#N)c1[N+](=O)[O-] CON1CCC(C(=O)NCC2C=CCN2C(c2cc(C3(C)CC3)n[nH]2)=O)CC1 N1(C(C=COCC)=O)CCC2C(CCN2C(C2C3COCC23)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC(C)CN(C)C(C1CCCCN1S(C)(=O)=O)=O C1(NC(C(c2ccccc2F)C)=O)CCN(C(=O)CC2CCCC23CC3)CC1 N1(C(c2cc(Cl)ccn2)=O)CCN(C(C2CCS(=O)CC2)=O)C2CS(=O)(=O)CC12 Cc1cnc(N2CCOC(CN(C)C(c3cc(Cl)nn3C)=O)C2)nc1 c1(OC)ccc(C(=O)NCCC(C)CCNC(c2cc(SC)oc2C)=O)c(F)c1 C(C(C(=O)NCc1ncn(C)n1)n1cc(CN2CCNC2=O)nn1)OCC Cc1nc(Cl)ccc1CC(=O)NCC1CCCCC1NC(=O)C(C)n1cccn1 N1(C(CNC(CC)=O)=O)CC2CCC1C(CNC(=O)C(C)CNC(=O)C(C)=O)C2 C1(SCC(=O)NCCC(Cn2cc(C(C)(C)S(C)(=O)=O)nn2)F)CCC(=O)NC1 C1(CC)CN(C(C2CC(c3cc(OC)ccc3Cl)C2)=O)CC(=O)N1 C(=O)(CCC(CC)CC)N1CCC2(C(C(NOCC=C(C)C)=O)C2)C1 N1(C(c2cc(F)ccc2Cl)C(=O)NCCCSC)CCC(O)CC12CC2 C1(CN(C(C2CC(SC)C2)=O)C)CCCN1C(=O)C(C)=C1CCCC1 N1(C(C2CC(OCC)C2)=O)CC2(CCC2)CCC1C(=O)NCC1(C)CCCCC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCc1cccc(CNC(CCCCOC)=O)c1 c1(C(=O)NC23CN(C(C(COC)(C)OC)=O)C(CC2)C3)cc(F)c2[nH]nnc2c1 C(=O)(CCCCCF)NCCn1ccc(C(=O)NCC(COC)C(C)C)c1 c1(C(=O)NCC(CC)NC(c2cccc(N)n2)=O)ccccc1NCCO c1(C(=O)NCCCN(C(=O)CCN(C)CCO)C(C)C)ccc2nc(O)[nH]c2n1 c1(-c2c(C3(C(N4CCCC5(C4)OCCO5)=O)CC3)cccc2)cccc([N+](=O)[O-])c1 N1(Cc2c(OCC)cccc2)CCC(=O)N(CCc2cnoc2)C1=O C1(CC(=O)N(C(C=C)C)C)CC(C)(C)CN1C(=O)Cn1nccn1 c1(C(=O)NC(C(C)NC(CCCC)=O)C)c[nH]c2cc(C(=O)OC)ccc12 N1(C(C(C)N(C(C2(CC)CCCC2)=O)C)=O)CC(F)(C2CC2)C1 c1(OC)ccc(C(C)C(=O)NC2CCCC2NC(C2(O)CC3CC2C3)=O)cc1 N1(C(C(C)N(C(=O)C2CC2)C(CSCC=C)=O)=O)CCC(C)(C)C1 C1(NC(C(C)c2cccs2)=O)CC2C(NC(=O)CCCn3cncn3)C2C1 c1(-c2cn(CCN(C(CC(=O)OCC)=O)C)nn2)cccc(S(C)(=O)=O)c1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C(C)NC(=O)CC2COC(C)(C)C2)CC1 N1(C(C2C(=C)C2)=O)CC(C(=O)NC2CNC(=O)C23CC3)CC(C)(C)C1 c1(CC(C(=O)NCC(C(C)(C)C)NC(CCC(=C)Cl)=O)C)ccc(C#N)cc1 CC1(C)CN(C(C23CCNCC2CNC3)=O)Cc2ccccc21 c1(C(CC(=O)OCC)NC(c2ccc(NS(C)(=O)=O)cc2)=O)ccc(Cl)c(F)c1 Cc1nc2ccc(Br)cc2c(NC2CCCn3cnnc32)c1C c1(C(CC)NC(=O)NC(c2ccccc2)CC)ccc(C)cn1 N1(C(C2(CC=C)CCCC2)=O)CCN(C)C(CNC(C2CC2COC)=O)C1 c1(-c2cccc(N)n2)cc(N2CCCC2=O)ccc1F.Cc1cc(C=O)on1 c1(C(N(CCC(C)NC(c2ccc(C3CC3)o2)=O)C)=O)snnc1C(C)(C)C C(C(C(C)C(C)C)NC(=O)CNC(c1ccccc1)=O)NC(CC(CC)OC)=O C1(C(=O)NCCOCCOCCNC(c2cn(C)nc2)=O)CCS(=O)(=O)N1.C1CC1 c1(OC)c(Cl)ccc(C(N2CC(NC(=O)CCC3(C)CC3)CC2C)=O)c1F C1(CNC(C2(C)CC2(F)F)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CCC12CCC2 c1(C(=O)NC2CCOC2)ccccc1.C1(=O)CCOCC(=O)NC2CC(C2)N1 C12(C(=O)NCC(=O)NCC(C)C)CC1CCN2C(=O)CC=C(Cl)Cl C#CC(C)(C1CCOC1)NC(=O)C=CC(C)NC(=O)CC=CCC C1(NC(=O)NCC(C)OCC)CSC(C)(C)C1 C1(CNC(=O)COCC2CC2)CC12CCN(C(c1ccsc1Br)=O)CC2 c1(NC(c2cncc(NCc3ccc(C)c(Cl)c3)c2)=O)cc(F)c(C#N)cc1Cl N1(C(CSC)=O)CCCC(C)(C)C1CNC(C1CN(C(N)=O)C1)=O CC(CN=c1ccc([N+](=O)[O-])c[nH]1)NC(C1CC2(CC2)C1)=O c1(C(=O)NCC(CN(C)C(c2cnn(C)n2)=O)(C)C)ccnc(S(N)(=O)=O)c1 N1(C(C2(OC)CCC(C)C2)=O)CCCC(CCNC(=O)CC2(N(C)C)CC2)CC1 C1(C(NNC(=O)NCC2(C)CCCCC2)=O)COC2(CCC2)C1 c1(N(CCCNC(C2CC3(CC(=O)N3)C2)=O)C)nc2cc(F)cc(F)c2o1 C1(CC(N)=O)(C(C)NC2CC(n3cc(C(C)C)nn3)C2)CCCCC1 C(C)(C)(CC(=O)NC1(CCOC)CCN(C(=O)C(C)OC2CCCC2)C1)OC N1(C(c2ccc(C3CC3)o2)C(=O)Nc2c(C)cccc2C)CCCC2CCCC12 CC1=C(C)CC(C)(C(=O)NC(C)CCNC(c2cc(C#N)[nH]c2C)=O)CC1 c1(-c2c(NC(C)=O)cccc2)cccc2[nH]c(C(=O)NCC(O)C(F)(F)F)cc12 C1(C)(C(N(CCCCCC)C)=O)CCN(c2ccnc(N(C)C)n2)C1 CCC(CC)CCC(=O)N1CCCC(CC)C1C(=O)NCC1(CC(C)C)CC1 c1(OC)cc(O)c(C(=O)NC2CCC(Nc3cc(C(F)(F)F)ncn3)C2)cc1Br N1(C(Cc2nc(C)oc2)=O)CCN(C(c2nc(C(F)(F)F)ccc2F)=O)CC1C C(=O)(CCCc1ccccn1)NCC(C)N(C)C(C1CCC1C)=O CCC(C)C(CC)(c1nnnn1C(C)C)NC(C)CCC(=O)OC C1(C(=O)NCC2COCCN2C(C23CCCC2C3(F)F)=O)CN2CCCN1CC2 CC(C)CCC(O)C(=O)NC(C)CCCC(N1CCCNC(=O)CC1)=O C1(NC(=O)CC2CCC(=O)N2)CCN(C(=O)CC2(N3CCCC3)CC2)CC1O N1(C(C(C(C=C)C)C)=O)CC2CCC1C(CNC(c1c(C)cccc1Cl)=O)C2 N1(C(COC2(C)CCC2)=O)CC(C)(C(=O)NCC2(C)CC(O)C2)CC1(C)C CCS(=O)CC(=O)NC(c1ccccc1CO)CNC(=O)C(C)OC(C)(C)C CC(C)CCC(O)C(=O)N(C)CC1CCN(C(=O)Cn2cnc(C#N)n2)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC(C2CCCN(C(C3(C)C=CCC3)=O)C2)C1 n1(CC)c(C)cc(C(N2CCCC2CN(C(=O)C=Cc2cocn2)CC)=O)c1C FC1(F)CC1C1CCCN(c2nc(N3CCCCCC3)c3ncsc3n2)C1 C1(CNC(c2cccnc2Cl)=O)CCN(c2ncc(I)cn2)CC1(F)F C1(C2CN(C(=O)Nc3cn[nH]c3)C2)CCCCC1=O N1(C(C=CSC)=O)CCN(C2COCC2NC(=O)Cc2ccns2)CC1 N1(CC(N2C(N(C3CCC3)C)CCC2)=O)CCN(CCc2ccno2)CC1 C1(CC#N)CC12CCN(S(=O)(=O)CCCN=[N+]=[N-])CC2 c1(CN2CCC(C#N)(c3ccccc3)CC2)ccc2nn(C)cc2c1 N1(C(C(C)(C)C)=O)CCC2(CCC2NC(C23CC(F)(C2)C3)=O)CC1 C1(CNC(c2cn(CCO)nn2)=O)CCN(C(C23CSCC2C3)=O)C1 c1(NC(C2(OC)CCSC2)=O)ccc(NC(=O)C(C)CC(C)C)cc1C C1(C=O)C(C)C1(C)C.c1(C(C)CCO)nnc(O)o1.C12CC(C1)C(=O)NC(=O)C2 C12(C(=O)NC3(CC=C)CN(C(C4CCCN4CCC)=O)C3)CC1COC2(C)C C1(NC(c2c(C)coc2)=O)CCC2(CCN(C(c3sc(O)nc3C)=O)C2)C1 C1(C(N(C)CC2CCCN2C(=O)CCc2cnoc2)=O)CCS(=O)(=O)C1 c1(C(=O)NC2C(CNC(C(C)SC)=O)C2)ccc([N+](=O)[O-])cc1-n1cnnn1 c1(C(=O)NC2C(OC)CN(C(=O)C(C3CCOCC3)C)C2)cc(S(N)(=O)=O)co1 C1(N(C)C(c2cnn(CF)c2)=O)CCCCN(C(C2CC(=O)C2C(C)(C)C)=O)C1 c1(C(N2CC(C)C(C(=O)NCC3CCC(C)CC3)C2)=O)cncc(C#N)c1 Cc1ccc(SC(C)C(=O)NCCC2CCCN2C(=O)CCCF)cc1 Cn1cnc2ccc(CN3CCOCC3CCN)cc12 C1(C(N2CCN(C(C=CC)=O)CC2)=O)Cc2nn[nH]c2C(C)C1 Cc1cccc2c(C(N3CCCC(F)(CNC(=O)C(F)C(C)C)C3)=O)n[nH]c12 CCC(C)C(C(=O)N(CC(C)COC)C)NC(C1CCCC1CC)=O c1(CC(=O)N(CCNC(=O)CSc2nncn2C)CC)cnc2cccnn12 C1(NC(c2cnoc2)=O)CCCCC12CCN(C(c1ccns1)=O)CC2 C1(C(=O)NC2CN(C(c3coc(O)n3)=O)C2)CCc2nnc(O)n2C1 N1(C(CN2C(=O)CCC2)=O)CC2CCN(C(c3ccccn3)=O)C2C1 CCC(CC)(CCOC)C(=O)N(CC(O)CN(C)C(C1CC2(CC2)CN1C)=O)C N(C(=NCC(c1ccccc1)N1CCCC1)NC1CCCC1)C(C#C)COC C1(C(=O)NCC2CN(C(C3C(C)(Br)C3)=O)C2)Cc2cc(F)ccc2C(=O)O1 c1(COC)cc(C(=O)NC2CCCC2NC(=O)C=Cc2cc[nH]c2)n(C)c1 C1(OC)C(OC)CNC1NS(=O)(=O)Cc1nc(-c2ccccc2)ns1 c1(C(=O)NC2CCC(NC(C(C)CF)=O)C2)noc2c1COCC2 C1(n2cccn2)(CNC(C(CSC)O)=O)CCN(C(C2(CCF)CCC2)=O)CC1 N1(C(C2(C)COC(=O)C2)=O)CCOC(C)(CNC(=O)CCS(C)(=O)=O)C1 c1(-c2nccc(NCc3nc(C)sc3)c2)ccc2c(c1)C(C)C(C)O2 n1(C(C)C)cc([N+](=O)[O-])c(=NCC2CCCN(C(C3CC=CCC3)=O)C2)[nH]1 C(C(CC(C)C)C(=O)NCC(C(=O)OCC)OC)NC(CCOCC#C)=O N1(C(CCC(C)N(C)C)=O)CCC(CO)(NC(c2cc(C(F)F)[nH]n2)=O)CC1 C1(C(=O)NC2COCC2NC(c2ncsc2C)=O)(OC)CCC(C(F)F)CC1 N1(C(COc2c(OC)cccc2)=O)CC(NC(c2ccncc2O)=O)C(C)(C)C1 N1(C(Cc2ccc(C)cc2)=O)CC(C(=O)NC(C(N)=O)C2CC2)OC(C)C1 c1(C(=O)NC(CNC(C(F)=CC)=O)CCOC)sc2cccc(Cl)c2c1Cl c1(N(C(=O)CCN(CCO)C2CC2)C(C2CC(F)C2)C)cccc2occc12 N1(C(=O)OC(C)(C)C)CCC2(CCC(CNCc3ccnc(Cl)c3)C2)CC1 C12(C(=O)NCC(C=C)(C)C)CC(CO)(CN1C(=O)CCNC(=O)OC)C2 C1(CC)CC(O)CN1C(C1CCOC1CNC(=O)C(C)OC(C)=O)=O C(CCCC(=O)NCCCC(C)NC(=O)CC(c1ccccc1C(F)(F)F)C)OC C1(CNC(c2ncn(CC)c2)=O)CN(C(c2cc(SC)ccc2C)=O)CCN1C CCC(C)(COC)C(=O)N1CCCCC(C(=O)NCC(C2CCC2)OC)C1 N1(C(c2cccc(Cl)c2Br)C(=O)NCCSC)CC(C)CCC12CC2 c1(CC)cc(C(=O)NC(C)(C)CNC(C2CC(OCCOC)C2)=O)c(F)cc1C C12(C(=O)NCC(C3CCN(C(C45CC4C5)=O)CC3)(C)C)CCC(F)(CC1)CC2 CC1(CNC(c2ncc(C(F)(F)F)s2)=O)CCN(C(=O)CCCCO)C1 C1(C(N2CCC(N(C(CC3CCC(C)CC3)=O)C)CC2)=O)CC2(C1)CC(O)C2 C=C(Cl)C(C)(C)C(=O)NCC1CCCCN(C(C2CCN(CCF)CC2)=O)C1 c1(C(C(N2CCC(O)(C(C)NC(C(C)CO)=O)C2)=O)C)nc(F)ccc1Cl C1(C(N2CCCC(N(C)C(c3cnn[nH]3)=O)CC2)=O)CC(=O)C12CCCC2 c1(NC(C(C)CC2CCCO2)=O)ccc2ccn(CC(=O)N(C)C)c2c1 C1(C)(C(N(C)CC2(CC(C)C)CC2)=O)CCCN1C(=O)CC(C)n1cccn1 N1(C(C(C)CC(C)(C)C)=O)CCC2CCN(C(=O)CCc3cnn(C)c3)CC2C1 N1(C(=O)NCCN2CCCC(OC)C2)CCc2cc(Br)cc(F)c2C1 N1(C(c2nc(C(C)=O)sc2)=O)CCC(C(C)C)C1CNC(=O)Nc1ccco1 Cc1c(CCC(=O)NC(C)CCN(C(=O)C=CC(F)(F)F)C(C)C)cnn1C N1(C(C=Cc2ccn(C)c2)=O)CC(C)(C)CCC1CNC(c1cnco1)=O c1(C(=O)NCC(CC)NC(C2C(OC)C2)=O)c(C(C)=O)sc2ccccc12 CCC(C)CCC(=O)NCc1ccc(CN(C)C(C2(F)CC=CCC2)=O)cc1 CC1CN(C(=O)C(Cl)Cl)CC1(C)C(=O)NCC1(C(C)O)CC1 CC1(C(=O)NCCC(O)CNC(C2(Br)CC2)=O)CC(F)(F)C1 C(C(C)C(C)C(=O)N(C)CC1CCN(C(C2CC(OC)C2)=O)CC1)OC N(C1CC2(CN(C(c3ccc(F)s3)=O)C2)n2ccnc21)C(c1ccc(C)nn1)=O c1(CC(=O)NC2(C3CN(C(C4C(C)(C)C4)=O)C3)CC2)cccc2sccc12 N1(C(C(CC)(F)F)=O)CCN(C(c2cc(CCCO)on2)=O)C(CC(F)F)C1 c1(OCC)cccc(CNC(C2CC(C)(C)O2)=O)n1 C1(NC(c2cnc(OC)nc2)=O)CC2CC(NC(C3COC3)=O)CC2C1 C1(C(N(CC#C)CCF)=O)CCCCC1NC(=O)C(CO)NC(N)=O C1(NC(CCc2nc(C)c(C)[nH]2)=O)CC2CCC(C1)N2c1ncncc1Cl N1(C(c2scc(C)c2C)C(=O)NCCCSCC)CCC(O)C(C)(C)C1 c1(CCC(=O)NCC2(CNC(c3c(C)scc3)=O)CC2)ccc(Cl)cc1Cl N1(C(c2c(CC)csc2)=O)CC2(C(=O)NCC(c3nccs3)C)CCC1CC2 N1(C(C(C)(C)OCC(F)(F)F)=O)CC2(CCC(CNC(=O)CC34CC(C3)C4)O2)C1 Cc1ncc(NC(=O)C(CO)NC(c2csc(=N)[nH]2)=O)c(C)c1C N1(C(C(=O)N)=O)CCOC(C(=O)OC)C1.C1(C)(NC(=O)NC)C(=O)C1CC N1(C(c2occ(OC)c(=O)c2)=O)CCCC2(CCC2NC(=O)CC2CC2)C1 C(=O)(C(CC(C)C)C(C)C)NCC1C2CN(C(c3c(C)csc3)=O)C1C2 N1(C(c2nn(C)cc2Cl)C(=O)Nc2c(C)cc(F)cc2)CCC(C)C(O)CC1 C(=O)(C#CC1CCC1)NC1CC(C(C)NC(C2CC(=O)N(C(C)C)C2)=O)C1 c1(C(=O)NCC2N(C(CCc3cc(OC)no3)=O)CC2)ccc(Br)cn1 CCCCC(CNC(C1(C)COC1)=O)NC(C1CC(C)N(C)C1)=O CC(Cc1ccccn1)C(=O)N(CCCNC(=O)CSc1nnnn1C)C C(=O)(C(C)(F)C(C)(C)F)NCC(C(C)(C)C)NC(c1ccc(C#N)cn1)=O c1(C(N2CC(CCOC)C2)=O)cnn(CCNC(=O)C(C)C2CCCO2)c1 c1(OC)cccn2ncc(C(=O)NCC3(C)CCCN(CC(C)O)C3)c12 CN1CC(C)(C(=O)NCC2CCCN2C(c2cc(C(F)(F)F)ncn2)=O)CC1=O C(=O)(CC(C)(O)COC)NCC1(OC)CN(C(c2nnn(CCC)n2)=O)C1 N1(C(C2N(C)CCOC2)=O)CCC(F)(CNC(=O)CCCCn2ccnn2)CC1 Cc1c(C(N2CCCC(CNC(=O)CS(C)(=O)=O)CC2)=O)ccnc1Cl CCC(CC(=O)N1CC(CNC(c2ccc(-c3cccs3)cn2)=O)C(O)C1)OC c1(C(=O)NC2(CO)CN(C(c3ccn(C4CC4)n3)=O)C2)nc2c(s1)COCC2 CC1CC(C)N(C(=O)CSc2ccccc2)CCN1C(c1cc(O)nc(Cl)c1)=O C1(CC=C)(NC(c2cnc(C3CC3)nc2)=O)CCN(C(=O)C(C)n2cncn2)C1 c1(CNCC(c2ccc(OC)cc2)O)cnc2c(Br)cccc2c1 N1(C(=O)OC)CSCC1C(=O)NCC1(F)CC(C(C)(C)C)C1 N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCCN2C(C)=O)=O)C1 C1(C(=O)NC2CC(C(C)O)C2)CCC(O)CN1C(c1cccc(F)c1)=O c1(OC)cc2ccccc2cc1C(N1CC(NC(=O)CC2CCC(=O)N2)C1)=O N1(C(C(CCCC)F)=O)CCC2(CC1)CC2NC(=O)C=Cc1ccc(C(F)F)o1 c1(NC(C(C2CCN(C(c3ccncn3)=O)CC2)C)=O)nc(Cl)ccc1I N1(C(C(C=C=C)C)=O)CCCCCC(NC(c2cc(C)cc(C)c2C)=O)C1 Cc1cncc(C(=O)NC2CCC(NC(C3CCC(C(N)=O)O3)=O)CC2)c1C CC1(C)CC(CNC(c2cccc(N)c2)=O)CN1C(=O)C=Cc1ccccn1 c1(OC)cc(C(=O)NC2CN(C(=O)CCc3cnn[nH]3)CC2OC)ccc1Cl C12(NC(CNC(CC)=O)=O)CC(NC(c3cnoc3C3CC3)=O)(C1)C2 N1(C(C(C)C2CCCC2)=O)CC(C2(NC(=O)CCN3CCC3)CC2)C1 c1(C(=O)CC)cc(=NCC2(O)CC(CN=c3[nH]cc(CC)s3)(OC)C2)[nH]c(C)n1.OC Cc1nccn2ncc(C(N3CC4CC(NC(=O)C(O)C5CC5)C3C4)=O)c12 N1(C(C2N(C(C(CC)n3cncn3)=O)C3(CC2)CC3)=O)CC(O)C(O)C12CCC2 C1(C)(C(=O)NCC(C)(F)CNC(C2CC3CC3C2)=O)CCC2CC2C1 Cc1cc(C)n(CC(=O)NCC2CCC(NC(=O)C(C)OC3CCCC3)C2)n1 c1(CC2C(C)(C)C(CO)O2)ncnc2c1ncn2C.c1(C(=O)O)nc2ccccc2s1 CC1CN2CCN1CC2C(N(CC(C)(C)NC(c1csc(C(F)F)n1)=O)C)=O c1(C(=O)NCC2C3CN(C(C4CC(=C)C4)=O)CC32)cc(F)c(C)cc1F N1(C(c2c(C)nn(C)n2)=O)CC(O)(C2(CNC(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)C1 c1(OC)ccc2c(c1Br)C(NC1(c3ncccn3)CC1)CC2 C(=O)(CC(=O)N1C(C(=O)NC(c2ccncc2)(C)C)CC1C)NCC n1(CC(=O)NCC(C(=O)N(CCC#C)CCOC)OC)cccnc1=O N1(C(c2c(CS(N)(=O)=O)n[nH]c2)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 c1(CNC(C2(CC#C)CCC2)=O)c[nH]nc1C1CCN(C(c2cscn2)=O)C1 c1(NC(C2(C)CN(C(C(C)OC)=O)C2)=O)cnc(Cl)nc1C c1(C(N2CCCC(C)(NC(CNC(=O)NC)=O)C2)=O)cccc2nc(C)nn12 C1(CC(=O)NCC(N(C)C)C2CC2)CCC(NC(=O)C=Cc2ccco2)C1 C=Cn1nccc1C(N1CC(NC(c2sc(C)cc2OCC)=O)CC1CO)=O C1(NC(c2c(C)noc2)=O)CC(F)CN(C(=O)C(C)Oc2ccc(Cl)cc2Cl)C1 CC(CC(=O)NC1CCC(NC(=O)CNC=O)C1)C1CCCC1 N1(C(C=C(C)C(C)(C)C)=O)CCSCC1C(=O)NCCc1ccc(C)cc1 C1(CC(=O)NC(CC)(C)CNC(c2cscc2F)=O)CC=CCN1C CC1CCC(NC(=O)CNC(=O)C(F)(F)F)CN1C(c1ccnc(CO)c1)=O C1(C(=O)NCCCn2cnnn2)CCCCC1NC(C1CCSC1)=O C1(CNC(c2c(CC)noc2)=O)CC2CC(C1)N(C(=O)CSC)C2.N1(C=O)CCCC1 c1(C(N(CCN(C(C2SCCCS2)=O)CC)CC)=O)cnn2c1N(C)CC2 C(=O)(C(C)N(C(C1CN(c2ncco2)C1)=O)C1CC1)NCC N1(C(C2CCC(=O)N2)=O)CCC2(CC1)CC(C(=O)O)CCO2 C1(c2cccc(OCC#C)c2)NC(=O)N(CC2CSCCS2)C1=O C=CCCCCCC(=O)NCc1ccc(CNC(C2(C)CCC(F)(F)C2)=O)cc1 n1(CC(=O)NC(c2oc(C)nc2C)c2ccc(C)o2)cc(C(N)=O)c2ccccc12 N1(C(C2C(COC)C2)=O)CC2CC1CN(C(c1cc3occc3n1C)=O)C2 C1(NC(CC2(C(=C)F)CCC2)=O)CC2(CCN(C(c3cccc(N)n3)=O)C2)C1 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)NC(C)C(C)NC(C12CCC(CC1)C2)=O C1(NC(C=CCC)=O)CN(C(=O)Cc2ccsc2Br)C2CC12 CC1(C)NC(=O)CC1C(=O)NC(C)(C(=O)NCc1ccc(Cl)nc1)C1CC1 c1(NC(c2c(OC)cccc2)C(=O)OC)nc(C)ncc1C(=O)N(C)OC CCCC(CC)CC(=O)N1CCCC(CNC(c2ncc(C(N)=O)cc2Cl)=O)C1 Cc1cn2nc(N3CC=C(CCNC(=O)C(O)C4CC4)CC3)sc2n1 C1(NC(c2c(OC)ccs2)=O)CN(C(c2cc(O)nc(Cl)c2)=O)C2(CCOC2)C1 CCCC(CC)CCC(=O)NC1CCN(C(=O)CNC(=O)CC(C)(C)C)C1C CN1CC(NC(=O)CC(C)(C)CNC(=O)CC(=O)NC2CC2)CC1(C)C C1(C(=O)NC2C(NC(c3ccc(C(=O)OC)[nH]3)=O)COC2)(CO)CCCC1O c1(C(=O)NCC(CC)(CC)NC(=O)Cc2cncs2)nccc2n[nH]cc12 C(c1cn(C)cn1)=CC(=O)N(C(C)CCNC(=O)CCN1CCCC1)C N1(C(C(C(C)C)F)=O)CCC(C2(NC(=O)C(C3CCC3)C3CCC3)CCC2)CC1 C=C(Cl)CC(C(=O)NC)NC(=O)C(C(C)(C)C)NC(=O)CCC(C)(C)F NS(=O)(=O)c1cc(C(N2CC(C3(NC(=O)Cc4ccco4)CC3)C2)=O)c(Cl)o1 N1(C(C(C)CC(N)=O)=O)CCS(=O)(=O)C(CCNC(=O)CC(C)C(F)(F)F)C1 CC(C(=O)NC1CC2(C1)CC(NC(C1OCCN(C)C1=O)=O)C2)C(C)(C)C c1(C(N(CC(C)(C)NC(Cc2ccc(C)c(Cl)c2)=O)C)=O)cc(Cl)cc(F)c1F Cc1cc(C(N2CCCC(C(=O)NC3(C)CCOCC3)CC2)=O)nnc1C C(CC(=O)N(CC(O)CN(C)C(c1sc(COC)nc1C)=O)C)(C(C)C)OCC C1(NC(C2(c3ccc(OC)cc3)CC2)=O)CN(C(=O)CC2CSC2)CCC1CO N1(C(c2ccc(OC)cc2F)=O)CCC2(CC1)CN(C(=O)CC1CCSCC1)C2 C1(NC(c2cc(CCC)[nH]n2)=O)CC(O)CN(C(C2(CC)COC2)=O)C1 c1(C(c2nnnn2Cc2nnn(C)n2)NCC2C(C)C2)csc(Cl)c1Cl C(C)(CCCCC#N)(c1n(-c2c(CC)cccc2)nnn1)NCCC(C)O CCC(C)C(O)C(=O)NCC1(C)CCN(C(c2ccc(=O)n(CCO)c2)=O)C1 c1(NC(C2N(C(c3cn(CCC)nc3)=O)CCC2C)=O)ccc(O)c(=O)cc1 N(C1CCCc2ncccc21)C(=O)NCCCS(=O)CC(F)(F)F C1(O)(CNC(Cc2scc(C)c2)=O)CCN(C(C2CC(CN(C)C)C2)=O)C1 c1(C(=O)NCCCCC)ccc2c(c1)OC1(CCCCN1C(=O)COC)CC2 C1(C(N2CCC(NC(Cc3c(C)n[nH]c3)=O)C(O)C2)=O)CCc2c(ncn2C)C1 S(=O)(=O)(c1ccc(C)cc1)N(C(c1c(CC)noc1C)=O)CC1CCNC1 C1(NC(CC2C(C)(C)C2)=O)CC2(CCN(C(=O)CCNC(C3CCC3)=O)CC2)C1 N(C1CC(C)(C)Oc2c(Br)cccc21)OC(N1CC(NC(C)(C)C)C2(CC2)C1)=O Cc1nc(Nc2ccc(C(=O)N(C)C)c(Br)c2)cc(C(C)C)n1 c12ccc(cc1)SCCCC(=O)N2.c1(C(=O)OC)nnc(C(C)C)s1 CS(=O)c1ccc(C(=O)N(C2CCN(C(=O)C(F)C(C)(C)O)CC2)CCO)cc1 C(=O)(CCCC(C)(F)F)NCC1N(C(C2CC(C)OC(C)C2)=O)CC(F)C1 N1(C(C(CC=C)CC)=O)CCOCC(C)(CNC(=O)CCc2cc(Cl)cs2)C1 N1(C(c2c(C)nc(CCO)nc2)=O)CC2CCCC1C2CNC(=O)CSC(C)C c1(C(=O)NCC2CCN(C(c3ccco3)=O)CC2)cccc2c1CCO2 CCCC(C)(C)CC(=O)N1CCC2CC2(NC(c2cn3ccnc3s2)=O)CC1 c1(CC(=O)N(C(C)CCNC(C2CC2c2cn[nH]c2)=O)C)ccc(Br)s1 C(CCC(C(=O)NCCOC1CCOC1)NC(=O)CC(=O)N(C)C)OC Cc1cc(C)c(CC(=O)NC2CCN(C(c3cn(C)c(O)n3)=O)CC2)s1 Cc1cncc(C(=O)NCC2(CO)CN(C(c3ccc(OC(F)F)cn3)=O)C2)n1 C(C)(CN=c1[nH]c(C)cc(=NCc2nc(C)ccc2Cl)[nH]1)OC N1(C(C(C)NC(CC)=O)=O)CCC2(CCCCN(C(C3CC3C3CC3)=O)C2)C1 C1(COC)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CC1(C)CC1 N1(C(c2csc(-c3cnc[nH]3)n2)=O)CCN(Cc2ccc(O)c(F)c2)C2CC12 c1(C(N(CCCNC(Cc2scc(C)n2)=O)C(C)C)=O)ccc(O)cn1 C1(CN(C(C(C)OC)=O)C)CC(F)CN1C(=O)C(C)Cc1cnco1 c1(C(=O)NCC2(C)CCN(C(=O)CC3CC3)C2)ncc(P(C)(C)=O)cn1 c1(C(N(C2CCN(C(C3CC3(C)CC)=O)CC2)CC)=O)cc(OC)ncc1F CC(C(=O)NCC1(CNC(=O)CNC(=O)NC2CC2)CC1)C(C)(F)F C1(NC(C2N(C)CC2)=O)CCN(C(N)=O)CC1.C1(n2ccnn2)CCN(C)C1 N1(C(c2ccc(COC)[nH]2)=O)CCOC(CCCNC(=O)CC=CC(C)(C)C)C1 C(C)(C)(CCCC(=O)NCC1CCCC(OC)C1)NC(C(C)=CCC)=O c1(C(N2CC(CNc3nc(C)nc(Cl)c3)C(C)C2)=O)cc2c([nH]1)CCCC2 CC1(C)CCOC1CCC(N1CCC(NC(c2cocn2)=O)C1)=O N1(C(C(C)OCC2CC2)=O)CC2(CC(NC(=O)CC(C)c3cccnc3)CO2)C1 c1(NC(=O)CN(C2CCCC2)C)ccc(F)cc1.C=C1CNCC=CC(=O)NCC1 c1(C(=O)NCC2(F)CCN(C(COC(C)C)=O)CC2)cccc(C#CC2CC2)c1 Cc1cn2c(C(N3CC=CC3CNC(=O)COCC(C)C)=O)cnc2s1 C1(NC(C=CC(CC)C)=O)CN(C(c2ncccc2O)=O)CC2(CC2)C1 N1(C(COC(CNC(CCC#C)=O)(C)C)=O)CC(CC)C(O)C1 C1(C(C)C)CCOCCN1C(C1CC2CCC1CC2)C(=O)NC1COC1 c1(C2(C)CC2)ncc2c(n1)CCN(N1CCN(C(=O)NC3CCCO3)CC1)C2 Cc1cc(F)ccc1NC(C1CC(O)CN1C(c1ccncc1F)=O)=O CCCC(C(=O)NCC1CC1CO)NC(=O)C(Cl)Cl C1(NC(C2CCC(C)N(C(c3cscn3)=O)C2)=O)CCC2(CC1)CC2(F)F S(=O)(=O)(c1cn(C)c(=O)n(C)c1=O)NCc1ccc(CSC)o1 C1(C(=O)NC(C(C)(C)C)CO)C(C2CC2)CCN1C(=O)Cc1ncccc1F C(c1c(Cl)nc2sccn12)=CC(N1CCC(NC(=O)CC2(O)CCOC2)C1)=O C(CC(O)CNC(=O)C(C)OC(C)=O)NC(C=C(COC)C)=O C(=O)(C(C)(C)CC(F)F)N1CC(OCCNC(C(C(C)C)c2cnc(C)s2)=O)C1 C1(CNC(C(C=C)OC)=O)CCN(C(c2ccccc2)=O)C1(C)C c1(CCC(=O)NCC(CCOC)NC(c2nc(C)nn2C)=O)ccccc1C C1(CC)CCCN(C(=O)COC2CCN(C(c3sccc3C)=O)C2)C1 Cc1nn(C)c(C(=O)NCC2(NC(=O)C(C)(C)n3cnnn3)CC2)c1[N+](=O)[O-] C1(C(=O)NC23CC(C)(C2)C3)CC2CN(C(=O)C(O)C(F)(F)F)CC2C1 C1(CC)CCN(C(=O)CC2(OC)CN(C(=O)C(O)C(C)SC)C2)CC1 N1(C(C(CC)COC)=O)CC2(CC2)CC1CNC(=O)Cc1ccccc1C(N)=O N1(C(CS(CC)=O)=O)CC2(C1)C(NC(c1nc(C)c(C)nc1O)=O)CCS2(=O)=O C(C)(C(=O)OC(C)(C)C)(C(=O)N1C(C)CN(C(=O)C=CC(C)C)CC1C)OC C1(NC(c2cc(COCC)c(F)cc2)=O)CC2CN(c3ncc(Br)cn3)CC2C1 Cc1cc(C)c(SCC2(N(C)C(=O)OC(C)(C)C)COC2)c(O)c1 C1(NC(CCC2(CCC#C)N=N2)=O)CC2CCCC(C1)N2C(C1(Cl)CC1(F)F)=O N1(C(CCC(CC)NC(c2nnsc2C)=O)=O)CCC(O)C(F)(F)C1 c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC(O)C2)cc2nccnc2cc1F N(C1CCCCc2ccc(Br)cc21)C(=O)NCc1nc(C)c(C)n1C CC1CN(C(c2coc(C#N)c2)=O)CCN(C(=O)CCCCC2CCCCC2)C1 C#Cc1cccc(C(N2CCN(C)C(CNC(C3CCS(=O)(=O)C3)=O)C2)=O)c1 C(C(C(=O)N(C(C)CSC)C)NC(=O)CC1CC=CCC1)OC C(CC(C(=O)N1CCC(C)(O)C1)NC(C1CC2(CC2)CO1)=O)N(C)C C=CC(F)(F)C(=O)NC1CC(C)N(C(c2cccnc2NC)=O)C1 c1(C(=O)NCC2CC3(CN(C(C4C(C)CCO4)=O)C3)C2)n[nH]c2ccc(Cl)cc12 c1(C(N(CCNC(C2C(C)C3CCC2C3)=O)C)=O)c(F)ccc(N)c1F CC1(C)C2CCC(C2)C1(C)C(N1CC2CC1C2CNC(=O)Cc1ccccc1)=O CN1CC(C(N2CCCC(CNC(=O)Cc3ccc(C4CC4)cc3)C2)=O)NC1=O C1(NC(c2nc(CNC(C(C)=NOCC#N)=O)oc2)=O)CNC(=O)CC1C c1(CNC(C(C=CC)O)=O)ccc2c(c1)CN(C(c1ccc(F)c(F)c1C)=O)C2 CCCC(C)(O)CC(=O)NC(CC(=O)N1CC2C(C1)C2(F)F)C(C)OC C(=O)(C(COC)CC(C)C)N1CCCC(CCNC(C2(C=C)CCC2)=O)CC1 N1(C(c2cccc(C)c2F)C(=O)N(C(CC)(C)C)CC)CC2CCC(C1)C2(F)F c1(C(=O)NCC(CC)NC(=O)C=Cc2ncc[nH]2)cc(C2CCCC2)[nH]n1 C(=O)(C(C)C1=CCCC1)N1CCN(C(c2ncn(C(C)C)c2)=O)CC1CF N1(C(Cc2cc(C)on2)=O)CCC2(NC(=O)OC(C)(C)C)CCCCC12 N1(CC(N)=O)CCCC(C(=O)N(c2ccccc2)CCC(=O)C(N)=O)C1.O CCC(CC)CC(C(=O)NCC(=O)Nc1ccco1)N1CCC1C1CCC1 N1(C(C(N2CCCC(O)C2)C)=O)CCCC1(C)CNC(c1ccoc1Cl)=O C1(C(=O)NCc2n(CC)ccn2)CCC2CCC1N2C(=O)Cn1[nH]cnc1=N c1(-c2nc(C(C)O)nn2CCN2CCOCC2)ccnc(Cl)c1Cl C1(C(=O)NC)C=CCN1C(c1conc1CNC(C1CC1OC(C)(C)C)=O)=O N1(C(CC(=C=C)C)=O)CCN(C(c2scnc2Cl)=O)CC1CC(F)F c1(CN(C)CC2CNC(C)(C)C2)cccc(OCC(F)(F)F)n1 C1(C(=O)NCCC2CCSC2)CCCN(C(C2(Cl)CC2(F)F)=O)CC1 c1(C(=O)NCCN(C(c2c(C)[nH][nH]c2=N)=O)C)cc2cccc(F)c2o1 CC1(C)OCc2cc(NC(=O)Nc3cnn(-c4ccccc4F)c3N)ccc21 c1(C2(C(=O)NC3(CNC(c4c(C)nc[nH]4)=O)CCOC3)CCC2)ccccc1Cl c1(C(N2C(CC)C(NC(=O)CC3CCCCC3)CC2)=O)ccc2c[nH]nc2c1 O=C(C1CCc2c(Cl)cccc21)N1CC2(C1)CN(C(C1CCCC3(CC3)C1)=O)C2 C(=O)(C(C)(COC)CC)NCCCN(C(c1c(CC)occ1)=O)C C(=O)(CC(C)CC(=O)N1CC2(C1)CN(C(C1(COC)CC=CC1)=O)C2)OC N1(C(=O)NCC2(O)CC(C)(C)OC2)C2CCC1CC(CO)C2 c1(CC(=O)NCC#CCNC(c2cc(C(C)(C)C)n[nH]2)=O)cnn2c1CCCC2 C12(C(=O)NCC3N(C(c4n(CC)nnc4)=O)CCOC3)CC1COC21CCC1 c1(C(=O)NC2CCN(C3CCC(C)CC3)CC2)ccnc2ncccc12 C1(CC)C(NC(c2cc(-c3cccc(F)c3)no2)=O)CCN1C(=O)CC(O)CC Cc1ncccc1-c1cn(CC2CCCC2NC(C2CS(=O)C2)=O)nn1 c1(CC(=O)N(C2CCCN(C(=O)Cc3cccs3)C2)CC)cc(F)c(F)cc1F C1(CNC(C=C(C)C(C)C)=O)OCC2CCC1C2.C12C(C1(C)C)NC2=O CCC(C(=O)NCC1CC(F)(CNC(=O)Cn2nnc(=O)[nH]2)C1)C(F)(F)F c1(C(=O)NC2CCC(CN(C)C(C3CC34CC4(F)F)=O)CC2)c[nH]nc1[N+](=O)[O-] c1(OC)cccc(C(C(=O)NCc2ccc(F)cc2)N(C2(C)CC(C)(C)C2)C)c1 c1(CC(=O)NC(C)CN(C)C(C2(C#N)CCC2)=O)nn(C)c2ccccc12 C12(C(=O)NC3C(NC(c4nc(COC)sc4)=O)CCCC3)CC3CC(CC1C3)C2 c1(C(N2C(C)C(C(=O)NC3COC3)CC2)C(=O)N(C)C)cc(Cl)c(Cl)c(Cl)c1 C1(NC(c2n(C)ncc2)=O)CCN(C(=O)CC2CCCC(=O)N2)C1(C)C C12CC(N(C(c3cccc(C4CC4)c3)=O)C1)N2.Cn1cc(OC(=O)C2CC2)cn1 C=CCC(C(=O)NC(CCC)C(O)C(=O)NCCN1CCCC(O)C1)C(C)C c1(CC(=O)NCC=CCNC(C2(C)CC=CCC2)=O)cc(F)ccc1Cl c1(CCC(=O)NCC(CNC(CCC(=C)Br)=O)F)ccc(O)c(Cl)c1 C1(CNC(CCC2(NC(C=C(C)C(C)C)=O)CCCC2)=O)CC2(CC2)C(=O)O1 C12(CC(=O)NCC(N(C(=O)C=Cc3cscn3)C)C3CC3)CCC(CC1)C2 c1(C(=O)NCC(C)N(C)C(c2cn(C)nc2Cl)=O)cccc2c1CNC2=O N1(C(c2c(C)con2)=O)CCC2(CCCC2NC(C2(F)CCCCC2)=O)C1 O=S(=O)(c1ccnn1C1CC1(F)F)Nc1cnn(-c2ccccc2)n1 CC(O)C(C)C(=O)NCCC1CCN(C(=O)CSC(F)F)C1 C(=O)(C1=Cc2ccccc2C1C)NC(CC)(CNC(=O)C(F)(F)C(C)O)CC C1(c2n(CCCCCCC)nnn2)(NCC(C)(C)C2CCC2)CC2CCC1CC2 c1(C(=O)NC(CN(C(=O)C=NOC)CC)C)ccc(-c2ccc(Cl)cc2)cc1 C1(SCC(=O)NCC)CC(O)CN1C(c1ccccc1)=O.N12CCC(C1)NC2=O C(N=c1[nH]c(=NCCCc2ncc[nH]2)[nH]c2c1CSC2)c1nc(C(F)F)sc1 N1(C(c2c(C)nco2)=O)CC(NC(C2(C)CC(C)(C)C2)=O)CC12CCOCC2 C1(NC(c2cc(C)sc2)=O)CC2(CCN(C(C3CC(=O)CO3)=O)C2)C1 c1(C(=O)O)cnc(Cl)c(F)c1.c12ccccc1C1(CC1)CN2.c1(OC)nccc(C)n1 CCC(C)CC(=O)C(=O)N1CC2CC(C1)N(C(=O)C=CCF)C2 CCCCCCCCCC(C)CC(=O)N1CC2CCC(C1)N2C(C1SCCS1)=O C1(=CCNC(C(COC)O)=O)CCN(C(=O)C(C2CCCCC2)=O)CC1 C(C1c2ccsc2CCN1C(C1CCCCC1)=O)NC(CC1(C)CCC1)=O C1(C(=O)NC2(C)CN(C(c3cnc(OC)s3)=O)C2)CC2CCCCN2C1 N1(C(=O)OC(C)(C)C)CC2CCC2(C(=O)NC(c2nn[nH]n2)C2CC2)C1 C1(CCC(C)=CC(=O)NCC(C)(C)C)CCOCC1.C1(C(=O)N)CC1C(C)C Cc1ccc2c(c1)CCC(C(=O)NCC1CCCN1C(c1cnnc(O)c1)=O)O2 N1(C(C2N(C(c3ccc(C)cc3)=O)CC(F)C2)=O)CCC(C)(C#N)C1 c1(C(N2CCCC(NC(c3c(C)nn[nH]3)=O)CC2)=O)cc(F)cc([N+](=O)[O-])c1Br Cc1c(C(=O)N(C)CC2CCCN(C(=O)C(C)c3ncco3)C2)ccc(F)c1F C1(N(C(c2c(C)sc(Cl)n2)=O)C)CCCN(CC2CC(C)(C)C2)CC1 C1(NC(c2cc(CC)n(CCO)n2)=O)CCCN(C(c2coc(C#N)c2)=O)CC1 c1(CC(=O)NCC(CC)NC(c2cnc(C3CCCO3)s2)=O)cc(C)cs1 CC1CCN(C(=O)C=CCN(C)C)CCN1C(C1CCCCC1)=O Cc1nn(C)c(C)c1C(=O)NCC1(C)CCCN(Cc2ccccc2C(C)C)C1 N1(C(=O)C(Cl)=CCl)CC2(C1)CN(C(c1ccc([N+](=O)[O-])s1)=O)C2 CC1CN(C(=O)CCCN2CCOCC2)CC1CNC(c1cccs1)=O N1(C(c2cccc(CCC)c2)=O)CCC(C)C(NC(=O)CN(C)C(C)=O)C1 N1(C(C2CC=CCN2C(c2cc(CO)[nH]n2)=O)=O)CCC(CO)C(O)C1 C(=O)(CC(Cc1ccccc1)CC(C)C)OCc1onc(-c2ccc(CC)nc2)n1 Cc1ccc(F)c(CNC(C2CCN(C(=O)CC3CCC(=O)N3C)CC2O)=O)c1 C(=O)(C1=CC2C=CC1C2)NCCCN(C(C1CC(SC)C1)=O)C1CC1 Cn1ncc(C(=O)NCCC2CCCN2C(C2CCCCO2)=O)c1C(F)F C12(N3CC(CCNC(COC(CC)(C)C)=O)C3)CC3CC(C1)CC(C)(C3)C2 c1(N2CCC(OCCOC)C2)nc(C)cc(=NC(C)CN2CCOCC2)[nH]1 N1(c2nnn(C)n2)CCn2ncc(CNC(C3CC(C)(C)C3C(F)(F)F)=O)c2C1 C1(CC(=O)Nc2c(C)nc(Cl)nc2)CC2(CCN(C(c3cn[nH]c3)=O)CC2)C1 N1(C(C(=O)N(C(C)C)C)C)CC2CCC1CN2C(c1c(Cl)nn(C)c1Cl)=O CC(C)CC(C)C(=O)N(C1CCN(C(c2coc(C3CCCC3)n2)=O)C1)C c1(CC)[nH]nc(Cl)c1C(=O)NC(C1CCN(C(c2csnc2C)=O)C1)C c1(C(N2CCC2Cc2c(-c3cn(CCC)nn3)n(C)nc2)=O)c(C)cccc1Cl c1(N2CCC(OC)CC2)nc(=NCCC(CSC)(CC)CC)[nH]c2ccccc12 c1(C(N(c2nc(Br)c(Br)cc2O)C)=O)ccc2c(c1)CN(C(=O)OC(C)(C)C)C2 c1(C(C(=O)NC(CC)CNC(=O)C=CC(=O)N(C)C)F)c(F)cccc1F C1(NC(c2c(CNC(=O)CN3CCOC3=O)ocn2)=O)CC2(CCC2)C1O C1(CC(=O)NCC(C)(C)C(N)=O)CCCN(C(=O)CCc2cn[nH]c2)CC1 c1(C(=O)NCCC2CN(C(C(C3CCCO3)OC)=O)C2)cc(C)nc(Cl)c1N c1(C(=O)NCCNC(=O)Cc2ccc(F)cc2C(F)(F)F)cnc2n1CCCC2 CC(C)C(CO)C(=O)NCC1CCC(NC(=O)CC2CCC(C)(C)CC2)C1 N1(CC(c2ccc(NC3CCC3)cc2)=O)CCCC(S(=O)(=O)OC(F)F)CC1 Cc1ncc(C(=O)NCC2CCCC2NC(=O)Cn2cccnc2=O)n1C N1(C(c2c(C)coc2)=O)CCCC(N(C(=O)Cc2nc(=N)[nH][nH]2)CCO)C1 CC(C(=O)NC1CC(NC(C2C(C)(C)C2(F)F)=O)C1)S(=O)(=O)c1ccc(F)cc1 c1(SCC2CC(C(=O)NCC(=O)NC(c3ccccc3)C)C2)ccccc1 N1(C(C2CCC(=C)CC2)=O)CCC2C(CCCN2C(C2CCC(O)CN2C)=O)C1 Cc1ccc(CCNC(C2CCC(C)N2c2ncncc2F)=O)cn1 CC1(C)CCCCC1CN1CCC(=CC(=O)NC(c2ccccc2)C#N)CC1 c1(C(=O)NC2C(OC)CN(C(C(CC)F)=O)C2)cc2n(n1)CCNC2=O O=C1NC2(CO1)CC(C(=O)NCC1CCN1C(=O)C1=COCCC1)C2 C1(C2CCCCN2C(C2CC(F)C2)=O)(CNC(C23CC(F)(C2)C3)=O)CCOCC1 C1(C)(C(=O)NCC2C(NC(CCOCC(C)C)=O)C2)CC2(C1)CC(F)(F)C2 C1(OC)CN(C)C(C)(C(=O)NCC2(NC(C3CC(C)(C)C3)=O)CC2)C1 C1(C)(C(=O)NC2CC(CCNC(c3c(C)cn(C)n3)=O)C2)CCOC12CC2(F)F Cc1onc(C(N2CC(NC(=O)CCc3ccccn3)C3CC23)=O)c1Br N1(C(C2(COC)CC=CC2)=O)CC2(C1)CN(C(=O)CCc1ccsc1)CCO2 C1(=O)CC(C(F)(F)F)O1.C(=O)(C(CC)CCC)N1CCC1.O(CP(C)(C)=O)C(CC)CC C1(CNC(C(CC)C2CCOCC2)=O)CN(C(=O)CNC(=O)C2CC2)CCO1 c1(C(N2CCNC(=O)C2C)C(=O)NCC)cc2cc(Br)ccc2o1 N1(C(COCCCC)=O)CCC(NC(=O)CC2CC2C2CC2)C1C1CC1 C1(NC(C(C)C(C)C)c2n(CCOC)nnn2)(CC2CC2)CCCCC1 C(CC(C)(C)C(=O)N1CCC(C(=O)NC(CO)C2CC2)C1)SC CCCC(C)(C)C(=O)N1CCN(C(=O)CCc2nncs2)C(c2ccccn2)C1 C1(C(=O)NCC(CC)C#N)CC(NC(c2nc(C)oc2C)=O)C1(C)C C1(NC(c2cn(CCN(C)C)nn2)=O)C2CCCN(C(C3(C4CC4)CC3)=O)C12 N1(C(CCN(C(=O)CCc2nc[nH]n2)C(=O)OC)=O)CC2CC(CC)CC2C1 N1(C(c2ccn(C(C)C)n2)C(=O)NCC2CCCO2)CC(C)CC1C c1(CNC(N(C(C)CC(N)=O)C)=O)ccccc1OC1CCC1 C(C(C)(CC)C(=O)Nc1cnc(C)nc1)NC(C(F)=C(C)C)=O N1(C(=O)CN2CCCC2)CCOC2(C1)CN(Cc1cc(O)ccc1Br)C2 C1(CNC(c2cnc(N(C)C)s2)=O)CCCCC1NC(=O)CSc1ccccc1 c1(C(=O)NC(C(=O)NCC(CC)SC)C2CCCO2)ncncc1OC N1(C(C(COCC)C)=O)CCC(NC(=O)CCC2CCC2)CC(O)C1 c1(CC)ccc(C(C)C(=O)N(C)CCNC(=O)Cn2ccnn2)cc1 CC(C)C(C(=O)N1CCC(C(=O)N(C2(CO)CC2)C)C1C)C1CCC1 c1(C(=O)NCCCC2N(C(c3cc(C)no3)=O)CCC2)c[nH]c2cccnc12 c1(OCCC(=O)NC(C)C(C)NC(=O)C=Cc2cn[nH]c2)cc(Cl)cc(Cl)c1 c1(CNC(C2CC(O)CN2Cc2c(Br)cccc2Br)=O)ccc2ccccc2n1 C1(Cn2cc(COC(COC3CCCN(C)C3)=O)nn2)CC2(C1)OCCO2 c1(OCC(=O)NCC2CCCN(C(c3c(C)coc3C)=O)C2)ccc(F)c(F)c1 C1(C(N(CCOC)CCNC(C2(S(C)(=O)=O)CC2)=O)=O)CCn2cc(C)nc2C1 C(C(C(=O)NC(C)CC(C)C)NC(=O)C(c1cnn(C)c1)=O)OC C1(COC)(CNC(C2CCOC(C)(C)C2)=O)CCN(C(=O)Cc2ccco2)CC1 c1(C(N2CCN(C(CC3CC(C(=O)OC)C3)=O)C3C2C3)=O)cccc2nccn12 c1(-c2ccc(OC)cc2OC)nc2c(s1)CN(C(=O)COc1ccccc1)CC2 c1(OC)c(C(=O)NC(CNC(=O)CSc2ccccc2)CO)cccc1Cl C(=O)(C1CCOc2ccc(Cl)cc21)N1CCC(CNC(Cc2n(C)ncc2)=O)C1 Cc1cc(C(=O)N(C)CC2CCCC(NC(C3CC(OC4CC4)C3)=O)C2)sc1Cl N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC(O)(C(C)CNC(C2CNC(=O)N2)=O)C1 C=CC(F)(F)C(=O)N1CCOC(CCNC(c2cn(C(F)F)cn2)=O)C1 N1(C(CN(C2CC2)CC)=O)CCCN(C(c2cncc(O)c2Cl)=O)C(C)C1 Cc1conc1CC(=O)NCC1CC(CNC(=O)C(C)n2ccnn2)CO1 C1(NC(c2cc(OC)nn2C)=O)CC2CN(C(c3cc(CSC)on3)=O)CC2C1 CC1(C)C(CNC(=O)CCC2CC(NC(=O)CN3CCC(F)CC3)C2)C1(F)F C1(O)(C(=O)NC2CC(C)(NC(CN3CCC(C)C3)=O)C2)CCCCC1 C1(CS(=O)(=O)NC(c2c(C)c(Br)ccc2)=O)CCCC2(CCC2)O1 C1(NC(c2c(C)[nH]cc2)=O)CCCCCC1NC(c1cc(O)cc(Br)c1)=O C1(C)(NC(CCC(C)SC)=O)CCCCC1C(=O)N.N12CCC1C2=O.C(C)C C1(CN(C(CCN(C)CC)=O)C)CN(C(c2cnnc(C)c2)=O)CCO1 C1(CC)CC(C(N2CCC(OCCNC(C3(C(F)(F)F)CC3)=O)CC2)=O)CCO1 CCC(C)(C)CC(=O)NN1CCCC1C(=O)NCC(C)(C)CO Cc1cc(CC(=O)NCC(C)SCC(=O)NCCN(C)C)cs1 N1(C(=O)CC(F)(F)F)CCC2C(C1)CN2C(c1cnn(CC(F)(F)F)n1)=O C(=O)(C1CCc2ccc(OC)cc21)N(C)CC1N(C(CSCC)=O)CCC1 c1(OC)cc(C(N2CCC(N(C(=O)Cc3cnsc3)C)C2)=O)ccc1C#N C1(NC(C=Cc2n(CC)ncc2)=O)CN(C(=O)CCOC2COC2)CC12CC2 O=C(C1Cc2ccc(Cl)cc21)NCC12CC1CN(C(=O)CCC(F)F)C2 c1(OC)cccc2ccc(C(=O)NCC3(F)CC(NC(C)=O)C3)nc12 C1(C)CCCCN1N1CC(NC(=O)CCc2nc[nH]n2)C1.N1(C=O)CCCCCC1 N1(C(C(C)C(C)(F)F)=O)CC2CCCC(NC(c3cnc(Cl)[nH]3)=O)C2C1 C#CCC(C(=O)N1CCCCC1CF)NC(c1oc(C)nc1CC)=O C1(COCC(C)O)CCCN1C(=O)CCCC1CC1 C1(CC)CN(C(=O)C=CC2CCCN2C(=O)C(=O)C(C)(C)C)C(C)CO1 c1(SC)nc(C)c(CCC(N2CCC(C(=O)N(c3ccccc3)C)C2)=O)c(O)n1 c1(OCC(C)C)cccc(C(=O)N(CC(C)N(C(=O)C=C(Cl)Cl)C)C)c1 C(C(C)C)(C(O)C(=O)NC1(CCNC(C2CC2(C)C(F)F)=O)CCC1)OC C12(NC(=O)CSc3nncs3)CCC(CC1)N(C(C1CC(O)C1)=O)C2 C1(NC(C2CC(OCC)C2)=O)CN(C(c2ccc(O)nc2)=O)CC2(CCC2)C1 C1(C(=O)NCc2c(C)ccc(C)n2)CC2(CCCC2)CO1 CCC(C)CCCCC(=O)N(CCCCCC(=O)NC1(C)CC(F)C1)C N1(Cc2cn(-c3ccc(C)nc3)nn2)CCCN(C(=O)C(F)OC(F)(F)F)CC1 C#CCC(C(=O)NCCCC(C)CO)NC(=O)C=COC c1(CC)ccoc1C(=O)NC(C1CCN(C(C2(OC(C)C)CCOC2)=O)C1)(C)C C(=O)(CCCC(C)(C)C)NC1C(C)CN(C(c2sc(Cl)cc2Br)=O)C1 N1(C(c2cncc(N)n2)=O)CCN(C(C2CC(F)(CO)C2)=O)C2CCC12 C1(C(N2CCC(O)C2)=O)(C)CCCO1.CC(C)(C)OCC(=O)O CC1C(NC(c2cccc(F)n2)=O)CCN1C(=O)C(c1ccccc1Cl)(F)F CCC(C)(CC)C(=O)NCC1(CNC(c2ccc(C)cc2SC)=O)CCCCC1 CC1CC(CNC(c2cnc(N)c(Cl)c2)=O)CCN1C(=O)Cc1cnoc1 C1(COC)(NC(=O)C(O)CC2CC2)CCCN(C(=O)C#CC(C)(C)C)C1 C1(N(C(CN(C(=O)C(C)N2CCCC2)CC(C)C)=O)C)CCOCC1C Cc1cc(NC(C2CCN(C(=O)C(C)CC(F)F)CC2O)=O)cc(F)c1 c1(C(=O)NC2(CC(=O)NCCn3c(CC)nnc3)CCC2)ccc(C#N)[nH]1 C(=O)(N1CC2COCC2O1)C1(NC(=O)CN2CC(=O)NC2=O)C(C)C1 c1(-n2cc(C(C)NC(C)(C)COC(F)(F)F)nn2)c(C(F)(F)F)cccc1C c1(C(=O)NCCCCNC(c2cn(CCC=C)nn2)=O)[nH]c2c(c1C)CCCC2 N1(C(C(CC)NC(C)=O)=O)CC2CCC(NC(c3ccc(C)nc3SC)=O)C2C1 C1(C(C(=O)NCC(C2CCCC2)NC(C2(SCC)CC2)=O)C)CCOCC1 N#Cc1ccc(C2(C(=O)NC3CC3NC(C3(C4CC4)CC3)=O)CCC2)cc1 C(C)(CNC(=O)CCc1cnc[nH]1)(C(C)C)NC(c1c(CC)c[nH]n1)=O N1(C(c2ccnc(OC)n2)=O)CCC(O)(C(C)NC(=O)C(C)c2ccco2)CC1 C1(CCC)(NC(c2cc(COC)cs2)=O)CN(C(c2conc2CC)=O)C1 N(C1CCCn2ncnc21)C(C(CC#C)NC(c1c[nH]c(C#N)c1)=O)=O c1(CCN2CCC(NC(Cc3ccn(C(C)C)n3)=O)C2)cccc(F)c1 c1(OC)cccc(F)c1C(=O)NCC1CCN(C(c2cc(O)ccc2C)=O)CC1 O=C1NCC2(CN(C(=O)NC3(c4ccc(F)cc4F)CC3)C2)O1 CCC(C)C(C(=O)NCC1CC(O)CN1C(c1cscc1C)=O)NC(C)=O c1(NC(c2c(NC(C3C(C(=O)OC)C3)=O)cc(C)cc2)=O)c(C)ccnc1C#N c1(C(=O)NCC(c2ccccc2)NC(C(C)(CO)OC)=O)ccc([N+](=O)[O-])[nH]1 c1(C(N(CCCNC(CSCC)=O)C)=O)nc(N(C)C)nc(=N)[nH]1 c1(N2CCN(C)C(C3CC3)C2)ccc(S(=O)(=O)N2CCc3ccccc3C2)cn1 C(=O)(C(CC)C(=O)N1CCCC1NC(c1cc(C2(C)CC2)on1)=O)OCC c1(C(=O)NCCCN(C(C=NOC)=O)C2CC2)cn(C(C)(C)C)nc1C CC1COCCN1C(C1CCOC(C)C1)C(=O)Nc1ccccc1 C(=O)(C(Cc1cscn1)NC(C1CC(CCC(=O)O)CO1)=O)OCC CCCCCC(=O)NCC(=O)NCC=CCNC(=O)CC1CCCC1(F)F N1(C(C(C)OCC)=O)CCC(C(N2CC(C#N)C2)=O)C1CC N1(C(c2ccc(CC)cc2)=O)CCC2CN(C(C3C4CC5C(C4=O)C35)=O)C2C1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)C(C)SCCN(C)C)C(CCO)C1 N1(C(c2c(C)c(Br)cnc2)=O)CC2(C1)CN(C(=O)C#CC1CC1)CC2CO CC(C)CC(O)C(=O)NCC(CO)NC(c1ccn(C)n1)=O C1(CC(=O)NCC2C=CC(NC(CC=C)=O)C2)CCCC(F)(F)C1 c1(C(=O)NCCCN(C(c2c(C)nc(C3CC3)o2)=O)C)coc2ccc(Cl)cc12 N1(C(COCC)=O)CC(CNC(=O)Cc2conc2C)C(c2cncn2C)C1 C1(NC(CS(N)(=O)=O)=O)COCCN(C(=O)C(F)(F)c2ccncc2)C1 c1(C(=O)NCC2C=CC(NC(c3c(C)nco3)=O)C2)ccc(F)c2[nH]ccc12 C1(C(=O)NC2CCN(C(C3(N(C)C)CCCC3)=O)C2)CCOCC12CCCCC2 c1(OC)cc(Cl)cc(CN2CCC(O)CC2C(N2CC(F)C(F)C2)=O)c1O CCN=C(NCCOc1ccc(Cl)cn1)NCc1csc(C)n1 CCC(CC(=O)NCC(C)N(C(=O)CCc1cscn1)C)C1CCC1 N1(CC)CC(C(=O)NCC2C(C)CCN2C(c2n[nH]c(C)n2)=O)CC1=O c1(CSC)ccc(OCC(F)(F)F)cc1.C1(C)(C)C(=O)N2CCC(C2)C(=O)N1 C1(OCC)(CO)CCN(C(=O)C(CC)n2ccnc2)CC1.C(=O)C(C)n1ccnc1 Cc1ccc(Br)c(C(=O)NCC2COCCN2C(C2CC2(C)C)=O)c1F c1(NC(C(CC)NC(=O)CC2CSC2)=O)ccc(F)cc1F c1(N(C)C)cccnc1C(=O)NC1CC1CNC(c1cnc(CC(C)(C)C)o1)=O c1(C(N(CC(CNC(c2c(COC)cco2)=O)C)C)=O)c(O)cccc1Cl C1(C(C)C)COCCN(C(=O)C(O)Cc2cn(-c3ccc(Cl)cc3C(N)=O)nn2)C1 N12CCC3CC(C3C1)C2=O.c1(C(=O)NC)ccc(CN(c2nncn2C)C)cc1 c1(SCC(N2CC(C)C(NC(=O)COC3CC3)C2)=O)nc2ccccc2s1 c1(CC)ccc(O)c(C(=O)NC2CC3CC(NC(=O)Cc4ccoc4C)CC23)c1 C1(NC(c2cc(C)ncn2)=O)CC2CN(C(c3cscn3)=O)CC12 C(CC(=O)N1CCC(C#N)(CC)CC1)(CC(C)C)NC(C(C)NC(CC)=O)=O C1(O)(CNC(CCC(N)=O)=O)CCN(C(c2ccsc2)=O)CC1 C1(CC(=O)NC(CCNC(CC(=C=C)C)=O)C(C)C)Oc2ccccc2NC1=O Cc1ncc(C(N2CCOC(C3CN(C(c4cnc(S)nc4)=O)C3)C2)=O)c(=N)[nH]1 [N-]=[N+]=NCCCCC(=O)NC(CC1CCC1)C(=O)N1CC(NC(N)=O)C1 c1(CC(=O)NC2CCN(C(CSCC=C)=O)C2C(C)C)c(C)nn(C)c1C C1(CNC(C2CC2c2cccc(Br)c2)=O)CCCN(CCCC2CCOC2)C1 c1(OCC(=O)NCCC2CN(C(C3C(C)(COC)C3)=O)C2)c(C)occc1=O c1(Cc2nc(C(C)NCC3C(COC)C3)sc2)ccc(C)cc1 C(CCC(=O)NC(C)C(C)NC(c1cnc(C2CC2)s1)=O)NC(=O)OCC C1(O)(CCNC(C2(C)CNC(=O)C2)=O)CCN(C(C2CCCCC2)=O)CC1 c1(CC2CN(C(CCCN(C(C)=O)C)=O)C2)ccc(N)cc1 C1(C(N(CCCF)CC)=O)CC(NC(=O)CCc2ncccn2)C(O)C1 N1(C(C(C(C)(C)C)OC(C)(C)C)=O)CC(C2CN(C(=O)C(Cl)=CCl)C2)C1 Oc1ncnc2scc(-c3nc(C(n4cccn4)C4CC4)nn3-c3ccc(Cl)cc3)c12 N1(c2ncc(C)cc2[N+](=O)[O-])CCC(C2CCN(C(=O)C(C)N3CCC3)CC2)C1 C(=O)(CC(C)CC(F)(F)F)N1C2CC(NC(C3(COC)CCCC3)=O)CC1CC2 c1(C(=O)NC(C)C(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)cccc2ncn(C)c12 c1(NC(=O)CCNC(=O)Cc2cn[nH]c2)c[nH]nc1Cl CCC(C)(C)C(O)C(=O)N1CC2(C1)CN(C(c1nnn(C)c1C)=O)C2 C(C)(C)(CC(F)C(=O)NCC(C)(C)CO)NC(C(CN(C)C)O)=O C#CC1(O)CCN(C(=O)C(C)(C)NC(=O)C(F)C(CC)CC)C1 C(=O)(C1=CCN(C(=O)CC2CC3CC3C2)CC1)NCC1(O)CCC(C)C1 C1(NC(CC2ON=C(CC)C2)=O)CCN(C(c2c[nH]cc2COC)=O)CC1F C(=O)(CC1=CCOCC1)NCCCC(C(=O)N(C1CC=CC1)C)O c1(C(N2C(CN(C(=O)C(CO)C(C)(C)C)C)COCC2)=O)c(F)ccc(N)c1F c1(COC(C2(CNC(C)=O)CCOCC2)=O)ncc(C)cc1Br C1(C(N(C(C(C)SC)C)C)=O)C(C2CC2)CCN1C(C1Cc2ccccc2C1)=O c1(C(N2CC(CCNC(C(C(=C)Cl)(C)C)=O)C2)=O)ccc2c(c1)CC(=O)NC2 C1(C(N(C(CCNC(Cc2cccc(C)c2)=O)C)C)=O)CC1C1CCCC1 N1(C(C(F)OC)=O)CCCC2(CCCCC2NC(=O)Cc2nc(C3CC3)cs2)C1 C1(CCC(=O)NC2CC(CNC(CN(C3CCC3)C)=O)C2)CCC(=O)N1 c1(NCCC(CCC)C)cc(=NCc2cnc(C3CC3)nc2)[nH]cn1 Cc1nc(N(C)C(c2ccc(Cn3cc(CC4(O)COC4)nn3)o2)=O)ccc1F CCCCC(O)CC(=O)N1CCC(C)(C(=O)NCCN(CCO)CCO)CC1 N1(C(CCC)=O)CCC2C(C1)NC(=O)CN2C(C1CCCN1Cc1cccs1)=O c1(C=O)cnncc1C.c1(COC)ccoc1C(N1CC(C2NCCC2)(O)C1)=O c1(CC(CNC(=O)NC2CC(C(C)(C)C)C2)N(C)C)nn[nH]n1 c1(N(C(C(=O)NCC2CCCCC2)C2CC2(C)Br)CCCC)ccc(F)c(C)c1 c1(C(=O)NCC2C(NC(c3c(C)scc3)=O)CCC2)sccc1C#N C#CC1CCCN(C(=O)C(C2CC=CCC2)NC(C2CCC2C#N)=O)CC1 c1(OCCCOCC)cnc(C(=O)NCCNC(C2CCCC(O)C2)=O)c(Cl)c1 C1(CC)CN(C(=O)CCN(C(=O)Cc2cn(C)cn2)C)CCN1C C(=O)(CC(O)CC(C)(C)C)N(C(CC(N1C2CN(CC)C(C2)C1)=O)(C)C)C C1(CNC(CCCNC(=O)NCC#C)=O)CN(C(=O)CCCN=[N+]=[N-])CCC1C c1(OC(CCC=C)C)ccc(CNCC(C2CCC(C)CC2)(C)O)c(OC)c1 CC1CC(NC(c2cc(C#N)cs2)=O)CCN1C(=O)C=Cc1ccc(Cl)s1 CC1(CO)CCC(N=c2[nH]c(=NCc3cncs3)[nH]c3c2SCC3)CC1 c1(C(=O)NCC2N(C(Cc3c(C)noc3)=O)CCCC2)ccc(C#N)nc1O C(=O)(C(CC=C)NC(c1cocc1C)=O)NCCCC=C c1(C(=O)NCC(CC(C)C)NC(=O)C(F)F)cc(C(F)(F)F)cc(O)n1 C1(NC(CC2CC(=O)C2)=O)CCN(C(c2csc(Cl)n2)=O)CC12CCC2 C(CNC(=O)Cc1csnn1)(CC(F)(F)F)NC(C(N1CC(C)C1)C)=O C1(C(=O)NCC2(C(=O)NC(CC)C3CCC3)CCCC2)CCN(C)CC1 N1(C(C2(C(N(C)C)=O)CC2)=O)CCN(C(c2cc(S(N)(=O)=O)cs2)=O)CC(O)C1 C(C(=O)NC1(CCNC(C2(N(C)C)CC2)=O)CCOC1)(C(F)(F)F)OC(C)=O C12(C(=O)NC3CC(NC(=O)C=CBr)C3)CC(c3ccccc3)(C1)C2(F)F c1(CC2(CC(=O)N(CC(C)(C)NC(COCC(=C)C)=O)C)CC2)ccccc1 N1(C(CC(C)F)=O)CCC2CN(C(c3csc(-c4cnc[nH]4)n3)=O)CC12 C1(NC(C2(COC)CC(F)(F)C2)=O)CN(C(c2cn(C)cc2C)=O)C2(CCC2)C1 N1(C(=O)CC2CCCN(C(c3ccc(O)cc3)=O)CC2)CCC2(CCCC2)C1 Cc1cc(CC(N2CCC(C(C)NC(C3CC(O)C3)=O)C2)=O)ccc1Cl C(=O)(C#CC1CCCCC1)NCC(CCOC)NC(c1cn(CC)nc1C1CC1)=O CC1CCOC(C(=O)NCc2csc(C(=O)NCCC3CCC(C)(C)O3)c2)C1 c1(C(N2CCC3(NC(c4nn(C)c(O)c4)=O)C(C2)C3)=O)ccc(Cl)c(N)c1Cl CCCC(O)C(CO)NC(=O)CNC(=O)CCn1cnnn1 c1(C(=O)NC2(CO)CCN(C(C3(C)CCCC3)=O)C2)ccc(NC(N)=O)cc1 c1(C(C(=O)NC(CC)C)N(CCC(N)=O)C2CC2)cc(C)c(C)c([N+](=O)[O-])c1C C(=O)(C1=CCCC1(C)C)N1CCN(C(c2nn(C)c(F)c2)=O)CC1CCO C(CCCC(=O)NC(CNC(=O)CNC(c1ccccc1C)=O)CC(C)C)OC CCN=c1ccc(C(N2CC(NC(c3nocc3C(C)C)=O)CC2(C)C)=O)c[nH]1 C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NCCN(C)C(C1CN(C)CC1C)=O CN1CCC2CC(NC(=O)CCc3cnc(C4CC4)o3)CCC12 Cc1cc(C(N2CC(O)(CCNC(=O)Cc3cnnn3C)C2)=O)c(C)cn1 c1(C(N2CC(OC)(CNC(C3CCSC(C)C3)=O)C2)=O)cc2ccccn2n1 C(=O)(C1CCc2nccn21)N1CC2(CC(NC(C(C)Cn3cccn3)=O)C2)C1 C1(C2CCN(C(=O)CC3CCC(=O)NC3=O)C2)(NC(c2c(C)coc2)=O)CC1 C12(C(N3CCC(NC(C(C)(C)OC(C)C)=O)C(F)C3)=O)CCOC1CCOC2 C1(N(C2(C(N(C)C)=O)CC2)C(C2CC=CCC2)=O)CCN(C(=O)C=CCF)O1 N1(C(CCCCCC)=O)CC2CCCC2C1C(=O)N(CC(F)(F)CO)C C(=O)(C1CCCn2nccc21)NC1CC(C(C)NC(=O)CS(=O)(=O)N(C)C)C1 N1(C(CCCCC#C)=O)CC2CCCC(C1)N2CCC1CCCCCC1 c1(OC)c(C(N2CCC2CNC(c2ccnc3[nH]ncc23)=O)=O)cc(Cl)cc1Cl c1(CNC(NC(C)C2CC2)=NCc2cn(C)nc2C(F)(F)F)ccccc1C#N N1(C(CN(C)C)=O)CCCC(C)(C(=O)N(C(CO)C(=O)O)CC(N2CCOCC2)=O)C1 C(CCC(=O)NC(C1(C(=O)NCC2(S(C)=O)CC2)CC1)C)OCC c1(C(N(CC#C)C2CC2)=O)ccn(CCNC(=O)Cc2ccc[nH]2)c1 CCCCC(O)C(=O)N1CCC(CNC(=O)CC(C)F)C1(C)C C1(NC(C(C)NC(=O)NC)=O)C=CCCC1C(=O)NCCC1OCCC1(C)C C1(N(C(C(C2CN(C(C(C=C)C)=O)C2)OC)=O)C)CCOC(C)C1 c1(C(C(=O)N(C2CN(C(C3CC4CC4C3)=O)C2)C)CO)ccc(Cl)cc1 CC(C)S(=O)(=O)CC(=O)N1CCCC1CNC(=O)C=CC c1(-n2ncc(C(=O)NC3CCC(CNC(C(C)OCC)=O)C3)c2)ccc(Cl)cc1 N1(C(c2ncn(C)c2)=O)CCC2(CCCN2C(c2c(F)ccc(F)c2Cl)=O)C1 Cn1cc(S(C)(=O)=NC(=O)c2cnc3cc(C(=O)O)ccn23)cn1 C1(C(N(C)CC2(CNC(C3(C(C)C)CCC3)=O)CC2)=O)CC2C(C1)C2(C)C C(=O)(C#CC1CCC2(CC1)OCCO2)N1CCC(N(C(C(C)C(F)F)=O)C)CC1 c1(N2CC(NC(C3(C(C)C)CCC3)=O)CC(F)(F)C2)ncnc2c(Br)c[nH]c12 C(=O)(C1Cc2ccc(F)cc21)N(CC(C)(C)NC(C1CCc2nncn2C1)=O)C c1(C(=O)OC)ccc(S(=O)(=O)NCC2(F)CC(NC(=O)OC(C)(C)C)C2)c(Br)c1 c1(CNC(C(=O)OCC)Cc2cscn2)n[nH]c2c1CCOC2 Cc1ccccc1C=CC(N1CCC(NC(C2(C)CC=CCO2)=O)C1)=O C12(CC(=O)NCc3ncsn3)CCC1CN(C(=O)C(O)CC1CCCO1)C2 c1(C(=O)NCCCN(C(=O)C(c2cnn(C)c2)C)CCC)cnc(O)cc1O c1(N(C(C(=O)NCC)C(C)C2CCCCC2)CCC)ccc(F)c(F)c1 C1(C(=O)NCC2(OC)CCN(C(=O)CCc3cnco3)C2)CCCC(C)(C)CC1 c1(CC(=O)NCCCNC(COc2c(C)c(Cl)ccc2)=O)cnc2n1CCOC2 c1(C(=O)NC2CCC(C)N(C(=O)CC3CCSCC3)C2)cc2cc(F)ccc2s1 CC1(CNC(=O)CC2CC3(CCO2)CC3)CCCN(C(c2ccncc2)=O)C1 C1(C(=O)Nc2ccccc2NC(c2cc(C)cs2)=O)C2CCC1CN(CC)C2 C1(NCC(C)O)CCN(C(C2(C)CC(Oc3ccncc3)C2)=O)CC1 c1(N2CCC(CC=C)C2)ccc(S(=O)(=O)NC(c2ccccc2)C2CC2)cc1F c1(C(OC(C(N2CCN(CC)CC2)=O)=O)NC2CCCC3CC23)c(F)cccc1Cl c1(COC)nccc(N2CC3C(NC(c4cnon4)=O)C3C2)n1 N1(C(C2(CC)COC2)=O)CCOCC12CCN(Cc1c[nH]c3ncccc13)C2 N1(C(c2ccc(C(C)C)cc2)=O)CCCC(C)(C(N2CCCC2C#N)=O)C1 CC1CC(NC(C23CC2CCN3C(=O)CN(C)C)=O)CCN1C(N)=O N1(C(CC=CC=C)=O)CCC2(CCOCC2)C(CNC(=O)Cn2[nH]cnc2=N)C1 C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)(OC)CCC12CCC2 C(CC1=CCCCCC1)NC(CC1OCCCN(C(C2=C(C)OCC2)=O)C1)=O C1(CC(=O)NCC(CC=C)NC(c2cnc(N(C)C)nc2)=O)COC(C)(C)C1 c1(CCC(=O)NCC2(F)CC(NC(=O)CC3CCC(=O)N3)C2)ccc(Cl)nc1 C1(C(=O)OC)CCCC1C(=O)N(CCCCNC(c1cnc(CC(C)C)[nH]1)=O)C c1(CC)c(C(=O)NCC2CC(COC)CN2C(=O)CC)nnn1CC.C(C)=O c1(OC)cc(C(=O)NCC(CC(C)C)NC(c2cc(C(C)C)no2)=O)ccn1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CC(C(=O)NCCC(C)C(C)C)CC12CCC2 C(N=c1[nH]nc(Cl)s1)c1ccc(CNC(c2ccccc2)=O)cc1 c1(C(=O)OC2CCCN2CCl)cncc(N2CCCC2)n1.C1C(C2CC2)O1 C1(NC(c2ccc(C)nc2C)=O)CCN(C(=O)Cc2cccnc2O)CC(O)C1 Cc1cc(Br)ccc1S(=O)(=O)NC12CC(C(=O)N=c3cc(Cl)cn[nH]3)(C1)C2 N(C(=NCc1ccc(C(F)(F)F)cn1)N1CCC(CN(C)C)C1)C(=O)OC(C)C c1(C(=O)NC2N(Cc3c(Br)ccc(OC)c3)CC(F)(F)C2)ccc2nc[nH]c2c1 C1(C(=O)NC2(CC(=O)NC(C(CC)C)CN(C)C)CCC2)CCC(=O)N(C)C1 c1(C(N2C(CCCNC(C3CC34CC4)=O)CCC2)=O)cc([N+](=O)[O-])cc(Cl)c1Cl Cn1c(S)nc2cc(C(=O)NCCCNC(C3CCC3CF)=O)ccc2c1=O CN1CCN(Cc2ccccc2)C(NC(=O)C(F)(F)Oc2cc(F)cc(F)c2)C1 N1(C(c2ccc(C)s2)=O)CC(NC(C2CCCO2)=O)C2(CCOCC2)C1 c1(CC)c(C(=O)NC2C3CN(C(C4(O)CC4)=O)CC23)cnc2ncnn12 C1(NC(CN2CC(CC)C2)=O)CC2CCC(C1)N2C(c1oc(C2CC2)nc1C)=O c1(C(N(CC(C)NC(C2(CC=C)CC2)=O)CC)=O)nc(C)[nH]c2nccc1-2 N(C1CN(C(c2cocn2)=O)Cc2ccccc21)C(c1cc(C)c(C)[nH]1)=O C1(CNC(CC(=C=C)C)=O)CN(C)CCN1C(=O)CCNc1ncccn1 c1(CC(=O)NCC(C)(C)Cn2cc(C3CC=CCC3)nn2)ccc2ncoc2c1 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)COCC3CC3)C2)=O)cc1)NC CC1CC(=O)NCC1C(N1CCN(C(=O)CCc2ccn(C)n2)C(C)C1)=O c1(C(=O)NC2CN(C(=O)C3=CCSC3)CC23CC3)cc(Cl)c(F)cc1F C1(CC)CN(C(=O)CN2CCCS2(=O)=O)CCN1C(=O)Cc1nnc(C)o1 C1(C)(C(N(CCCNC(CN(CCC)C)=O)C)=O)Cc2ccccc2NC1=O C(=O)(C1=CCCCCC1)NCCCC1N(C(C(C)(Cl)Cl)=O)CCCC1 N1(C(c2ccc(C(C)=O)cn2)=O)CCN(C(c2ccc(C(C)C)o2)=O)C2CCC12 C1(C(=O)NCc2cncc(C(=O)NC(CO)C3CCC3)c2)CCC(=O)NC1 C12(C(=O)NC3(CSC)CC3)C(=O)C3CC1C2C3.c1(C(=O)NC)ccnc(COC)c1 C1(NC(c2nn(C)c(O)c2)=O)CCCCN(Cc2ccc(O)c(C(=O)O)c2)C1 N1(C(c2c(C)ccnc2O)=O)CCC2(CC1)CC2NC(c1ccc(O)nc1Cl)=O N1(CCn2c(C)csc2=O)CCC2(CCCN(C(C3CCCC4CCCN34)=O)C2)C1 c1(CNC(C2(C=C)CCC2)=O)cnn2c1CN(C(c1cc(C)on1)=O)CC2 C(=O)(CCCCC(=O)OC)N(CC(CC=C)C(=O)NC1CC(=O)N(C)C1)C c1(CNC(CC(=C)C)=O)nnc2n1CCN(C(c1cnc3sccn13)=O)C2 Cc1coc(C)c1C=CC(N1CC(CNC(C2CC2C#N)=O)C(O)C1)=O CC(C)CC(C(=O)NCC1CCOC1)N(C(=O)CC1CC2(CC2)C1)C C(=O)(CC(C)C(C)(C)NC(=O)C(CC)C(=O)OCC)N(CCC#C)CCO N1(CC(=O)NC(c2ccccc2)C)CCCC(CCNC(=O)C(C)(C)CO)C1 c1(C(=O)NCC2C(NC(CC3(C)CC3(Cl)Cl)=O)CC2)nc(O)nc(O)c1F C1(C(N2CC(O)(CNC(=O)CC3CCCSC3)C2)=O)CCC(=O)N1C1CC1 C=C(C)CC(C(=O)NCCN(CCOC)C(c1cc(OC)n(C)n1)=O)NC(C)=O c1(-c2cccc(C3(C(N4CC(O)C(F)C4)=O)CC3)c2)c(F)ccc2[nH]ccc12 C(=O)(C(CC(F)F)C1CCC1)NCC12CC(CNC(c3c(C)cco3)=O)(C1)C2 N1(C(c2ncn(CC)n2)=O)CCN(C(C23CC2COC3(C)C)=O)CC(C)(F)C1 N1(c2snc(C(=O)OC)n2)CCC(NC(c2ccc3ncsc3c2)=O)C12CCC2 Cc1ccc2cc(-c3c(C)noc3-c3ccc(C(N)=O)cc3)cnc2c1 c1(C(N2CCC(C)(NC(c3ccncc3)=O)C2)=O)cnc(Cl)c(N)c1 c1(C(=O)NC2CC(C)N(C(=O)CN(CC(C)(C)C)C)CC2)c(O)cc(F)cc1F N1(c2nnc(CCOC)s2)CC2(CCC(NC(=O)CC3CCCS3(=O)=O)CC2)C1 c1(-n2ncc(C(=O)NCC3N(C(COC4(C)CCCC4)=O)CC3)c2)ncc(Cl)cn1 Cn1cnn(CC(=O)NCC2CC2CNC(=O)CN2CSCC2=O)c1=O C=CC(C)(CCOCC)C(=O)NCCC(O)Cc1cnn(C)c1-c1nn[nH]n1 C1(C)(C(=O)NC2CC(CNC(C3(OC)CCOCC3)=O)C2)CCC(=O)CC1 C1(N(C(C2CCN(C(c3c(OC)nn(C)c3)=O)C2)=O)C2CC2)CC2CCC(C1)C2O CC(C)=C=CC(=O)NC(C(=O)NC(c1n[nH]c(CO)n1)C)C1CCOC1 C1(C(=O)NCc2c(CNC(C3(C)COCCO3)=O)cccc2)CC12CCOCC2 C1(C(=O)OC)CC2(C1)CC(C(N1CC(C)(CNC(C3C4CNC(=O)C34)=O)C1)=O)C2 N1(C(CC(C)(C(F)F)N(C)C)=O)CCC2(CCCCN(C(c3ccsc3)=O)C2)C1 c1(C(N2CC(F)C(F)C2)=O)cn2c(n1)CCC2 c1(C(=O)NC(c2ccncc2)CC=C)cc(Cl)nc(Cl)n1 N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)NCC2CCCN2CC)=C(F)C1 C(=O)(C1=CS(=O)CCC1)NCCN(C(C(C)CN(C)C)=O)C c1(NC)ccc(C(=O)NC2CC(N(C)C(C3CC(C(F)(F)F)C3)=O)C2)c(Cl)c1 CCS(=O)(=O)c1ccc(-c2noc(Cc3c(F)cc(C(F)(F)F)cc3Br)n2)cn1 C1(NC(C(c2ccc(C)cc2)F)=O)CC(O)CN(C(=O)CCCN2CCCC2)C1 c1(-c2nc(CC(CCCN(C)C(=O)OC(C)(C)C)CO)on2)c2c(nn1C)CCC2 N1(C(c2ncn(CC)n2)=O)CCC2C(CCN2C(=O)C(N2CCN(C)CC2)C)C1 c1(CC)nc(C)sc1C(=O)N(C)CCOCCN(C(=O)Cc1ccccc1F)C c1(C(=O)NC(C)(CNC(C2CCNC2=O)=O)C2CC2)nc(C2CC2)n2ccccc12 c1(C(N(C2CCCC2)C(CN(C(C)C)C)=O)C)ccccc1F c1(C(=O)NC2CC(CNC(CCC(C)OC)=O)C2)ccc(Br)cc1N C1(CC)(NC(=O)CC(=O)NCCCCl)CCCN(C(=O)CC2(C)CCCCC2)C1 O(P(=O)(CCC1CCCCO1)OCC)CC c1(OCC(=O)N(C(C)CNC(=O)COC2CCCCC2)C)cc(Cl)cc(Cl)c1F C(=O)(C(O)CCNC(c1cc(C(=O)NC)[nH]n1)=O)NC1(CC)CC1 c1(CC(=O)OC)ccc(NNC(=O)C(C)NS(=O)(=O)c2ccc(F)cc2)cc1 N1(C(C(CC(F)F)NC(c2cc(C)ncn2)=O)=O)CCCCCCCC1 C1(NC(C2(C#C)CCCC2)=O)CC2(CCN(C(c3cccc(C)c3)=O)C2)C1 n1(CCC)nc(C)c(C(=O)NCC2CC(NC(=O)C3=CCCCO3)C2)c1C CC1CN(C(=O)CCC(=O)NCC(F)F)CC1(C)CNC(=O)CSc1nncs1 C(=O)(CC(C)(C)SC)N(CC=CC(=O)N(CC(CC)O)CC)C c1(C(N(C(CC)C=C)C)=O)nc(C(F)(F)F)n2c1CCCC2 c1(C(N2C(CNC(Cc3c(C)nccc3)=O)CC2)=O)ccc(O)c(Cl)n1 C(=O)(C(CO)C(C)(C)C)N1CC(N(C(CSCC)=O)CCC)C(O)C1 N1(C(c2cnc(CC)s2)=O)CCOC(C)(CNC(=O)CC2(N(C)C)COC2)C1 CC(CCNCc1ccccc1OCC(F)(F)F)C(F)F CC1(C)CCCCCC1NC(C1C2CCCC2CN1C(C1CCSC1)=O)=O c1(C(=O)OCC)[nH]cc(C)c1C(=O)NC1CN(C(C2(C)CS(=O)(=O)C2)=O)CC1C CC1=C(C(=O)N2CCOC(CCNC(c3cncc(Cl)c3Cl)=O)C2)CCCO1 c1(SC)cc(C(N2CC3CC(NC(=O)COCC(F)F)C2C3)=O)ccc1N C1(CNC(c2onc(C)n2)=O)CCC(NC(=O)C(C)CF)CC1 C(N=C(NC)N1CCC(Oc2ccc(C#N)cn2)C1)c1c(CCC)onc1C.CC Cc1cccn2cc(C(N3CCCC(F)(CNC(=O)CCCN=[N+]=[N-])C3)=O)nc12 C1(CNC(COC2CCC(C)CC2)=O)CC2(CC2)CN1C(=O)C(C)N(C)C C1(C(NOCC(=O)NCc2ccsn2)=O)CCC(CO)CC1 c1(C(=O)NC2CCC(NC(CC3C(C)(C)OCCO3)=O)C2)cc(F)c(F)cc1Cl C1(C(N(CCNC(CCC#CC)=O)CC2CC2)=O)CCC(O)(C(F)(F)F)CC1 N1(C(c2c(C)n(C)cc2)=O)CCC(C)C(CC(=O)NCC(C)(C)C2(O)CCC2)C1 Cc1cccn2ncc(C(=O)NC(C)CCN(C(=O)C=C3CC3)C)c12 C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(C(CC#C)CC#C)=O)CC=C1 n1(CC(=O)NC2CC(N3CCNCC3)C2)ccc(C(=O)O)n1 N1(C(C2C(=C)C2)=O)CCC(CNC(c2cscc2C2CC2)=O)CC1C c1(C(N2CC(N(C(C3C(C(C)C)C3)=O)C)C2)=O)cc2ccc(Br)c(F)c2[nH]1 C1(NC(C(C)n2cnnn2)=O)CCCC2CN(C(=O)C(O)CC(C)(C)C)CC12 c1(C(N2C(CN(C)C(c3c(N)cccc3F)=O)CCC2)=O)cncc(N=[N+]=[N-])c1 C1(CNC(C(C2CCCC2)OC)=O)C2CN(C(=O)C(=O)Nc3ncc[nH]3)CC12 c1(CC)cc2cc(c1)Cc1ccc(cc1)NC2=O.c1(COC)ccc(Cl)cc1 N1(C(c2c(C)nsc2C)=O)C2CCC1C(CNC(=O)Cc1cc(F)cc(F)c1)C2 c1(CN(CC(CC)(C)COC)C2CC2)cc(I)ccc1Br c1(C(=O)OCC)ccc(C(N2CC3C(C(=O)NCc4cn[nH]c4)C3C2)=O)cc1 N1(C(CC(CC=C)NC(C2CCCCC2(C)C)=O)=O)CC2(CCC(=O)O2)C1 N1(C(CCC(CC)C)=O)CCC2CN(C(=O)CCN(CC)CC)C2C1 C1(OCCNC(C2CC(CCC)C2)=O)CCN(C(C2(C(N)=O)CCC2)=O)C1 c1(C(N2CC(C)C(CCNC(C3CC3CF)=O)C2)=O)csc2c1CCC(C)(C)C2 N1(C(Cn2cnc(=N)[nH]2)=O)CCN(C(c2cnn(CCC(F)(F)F)c2)=O)C2CC12 C1(NC(=O)NC(Cc2cccnc2)CO)COCC1C(=O)O c1(SC)cncc(C(N2CCC(CN(C(=O)C(=C3CCCCC3)F)C)C2)=O)c1 Cc1cc(=O)n(CC(N2CC3CC(CNC(c4ccon4)=O)C3C2)=O)cn1 C(c1ccc2c(c1)NC(=O)CO2)=CC(=O)NCC(CC)NC(CSCCC)=O c1(CC(=O)NC(CC)(C)CNC(c2ccsc2OC)=O)ccc2c(c1)CCCO2 CCCC(C(=O)NC1CC(O)C1)NC(=O)CCCn1ccnn1 c1(CNC(C=CC(C)NC(C(C)NC(C)=O)=O)=O)nc(C)c(C)[nH]1 N1(C(=O)CC2CCCOC2)CC2CCC1CN2C(c1cc2ncccc2o1)=O C1(NC(COCC=C)=O)(COC)CCCN(C(=O)C(C)P(C)(C)=O)C1 C1(C(=O)NCCCc2ccc(CNC(=O)OC(C)(C)C)cc2)CCCCC12CC2 c1(C(N(C2CC(NC(CCCC#C)=O)C2)C)=O)sccc1S(=O)(=O)N(C)C c1(C(=O)NCCOCCCNC(C=CC=CCC)=O)ccc(C)cc1 C1(C(N(CCCCNC(Cn2c(C)cc(C(F)F)n2)=O)C)=O)CC(C)(C)CN1C N1(C(=O)C2CC2)CCCCC1NCc1cnc(C(C)C)s1 Cc1cccc2ncnc(N3CC(NC(=O)C(c4cncn4C)O)CC3C)c12 C(CC(=O)O)(c1cccnc1)NCC(CO)NC(=O)OC(C)(C)C c1(C(=O)NCC(CN(C(=O)CN2CCCNC2=O)C)O)cnn(C2CC2)c1N c1(CC)cc(Br)ccc1C(N1CC(NC(c2cc(I)ccc2F)=O)C(O)C1)=O C(=O)(CC(F)(F)C(F)(F)F)N1CCC(N(C(C(=O)N(C)C)=O)C)C2(C1)CC2 C1(NC(c2c(C)nn(C)n2)=O)CCC2CCN(C(c3cnsn3)=O)C1C2 c1(C(=O)NCC(CC=C)NC(C2CCN(C)CC2)=O)cc2n(c1)CCCC2 N1(C(COC(C)(C)C)=O)C2CCC1CN(C(c1cncc(OC(F)F)c1)=O)C2 CC1(C)CN(C(=O)Nc2ccc(Cl)cc2)C1Cn1cc(CCC[Si](C)(C)C)nn1 N1(C(C2C(C)CCO2)=O)CCC(C2CC2)C1C(=O)NCc1ccncc1 CC1CN(C(C2(C)CC2(F)Cl)=O)CC(C)N(C(c2n[nH]c(C3CC3)n2)=O)C1 c1(C(=O)NCCNC(CCNS(NC)(=O)=O)=O)ccc(C)cc1.C1(=O)CCOCN1 N1(C(C(CSC)O)=O)CC(C2CN(C(=O)C(C(C)O)NC(C)=O)C2)C1 N1(C(C(CC)N2CCCC2=O)=O)CCC(CN2CCC(F)(F)C2)CC1 CC1Cc2cc(S(N)(=O)=O)ccc2C1NCCc1cc(F)ccc1Br C1(C)(CC)CC(C(=O)NC(C)CNC(c2ccc(NC(=O)NC)s2)=O)CCO1 CC1CCN(C(c2ccc(OC(F)F)cn2)=O)CC1CNC(=O)Cn1cnnc1 C(C(C)(C)CC(=O)NC(C)(CN(C)C)C(C)C)NC(CCC(C)SC)=O N1(CC)CCOCC1CC(=O)NC(C)CNC(=O)CCc1ccc(C)s1 c1(C(=O)NCC(CNC(=O)C(C)(C)O)OC)cn(C)nc1C1CCCC1.C(C)=O N1(C(C(=O)Nc2ccc(OC)c(OCC(N)=O)c2)=O)C2CCCC1COC2 C1(CCNC(C23CC(C(C)C)(C2)C3)=O)(OC)CN(C(c2cnc(C(C)C)[nH]2)=O)C1 c1(C(=O)NCC2(C)CCN(C(C3CCOC3=O)=O)C2)cnn2c1OCCC2 N1(C(CCC=C=C)=O)CCCCC(C2CN(C(=O)COC(C)C)C2)C1 C(=O)(C(O)CC(C)(C)C)N1CCCCC(NC(COc2ccc(CC)cc2)=O)C1 C#Cc1ccc(C(N2CCN(C(=O)CC3CC4CC4C3)CC2CCO)=O)cc1 c1(OC)ccc2nccc(C(=O)NCC3CCN3C(c3cc(C(C)=O)c[nH]3)=O)c2n1 CC1CCC(NC(c2cn(C3CC3)nn2)=O)CC1.C12CC1NC2=O N1(C(Cc2c(C)scc2)=O)CCOC(C)(CNC(c2c(Cl)c(C)nn2C)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2CC3CCC2O3)=O)cc(Cl)c(Br)[nH]1 c1(OC)c(C(=O)NCC(O)CN(C)C(C23CCC(CC2O)C3)=O)cc(Cl)cc1Cl S(=O)(=O)(c1cc(Cl)ccc1F)N1CCC2(C(C(=O)NC(CC)C(=O)NC)C2)CC1 C1(C)(NC(c2ccc(-c3ccc(F)cc3)o2)C)CCC(O)CC1 N1(CC(C)C)CCC(C(=O)NC(C2CN(C(C3(CF)CCOCC3)=O)C2)C)CC1 C1(CNC(=O)COCCF)CC2CCCCC2N1C(=O)CC1CCS(=O)(=O)C1 c1(OC)ccc(C(=O)NCC2CC(C)N(C(c3ccccc3C)=O)C2)c(OC)c1 N1(C(C(C)N(C)C)=O)CCN(C(=O)CC2CCN(C)CC2)CC(CO)C1 c1(C(C)C)ccc2c(c1)C(NC(N1CC3CC(O)CC3C1)=O)CCC2 c1(C(N2CCC(O)(C(CNC(CC(=C)Br)=O)C)C2)=O)c(C)ccc(C)c1N C(=O)(CC(C)(C)C(=O)N(CC(C)NC(c1cncc(Cl)n1)=O)C)OC C1(CNC(CC(CN(C)C)(C)C)=O)CC2CCCCC2N1C(C1CCC1)=O c1(C(C(CC)=O)=O)cncc(NC(C2(C)CC2)=O)c1.C1(CC(=O)N)(CN)CC1.OC c1(C(=O)NCC(CNC(c2cccc(C3CC3(F)F)c2)=O)O)cc(F)ccc1O c1(C(N2CC3CC(C(=O)NCCCC(C)(C)CO)(C2)C3)=O)cncc2[nH]ccc12 c1(NCc2ncc(OC)nc2)nccc(=NCc2cccnc2Br)[nH]1 C1(OC)CCCC(CNC(=O)CN(CC(C)C)C(c2nc(C)oc2OC)=O)C1 Cc1nn(C)c(C)c1C(=O)C(=O)NCC(C)N(CC(=O)NC(c1cccs1)C)C c1(C(N(C2CC(NC(C3(C(F)F)CC(F)(F)C3)=O)C2)C)=O)cnc2n1CCC2 C1(C)(C(=O)NCc2nnc(C)s2)CCCN1C(=O)C=Cc1cc[nH]n1 CS(=O)(=O)c1cc(C(=O)NC2CCC(NC(c3ccsc3CN(C)C)=O)C2)cs1 C(=O)(CCN=C(NCc1ccc(Br)c(F)c1)NC1CC12CC2)N(C1CC1)CC CC1CN(C(C2CCCOCC2)=O)CC2(CCN(C(c3cnc(O)n3C)=O)C2)O1 C1(C(=O)NCC2(N(c3cncnc3)C3CC3)CCCC2)CC(F)CN1CC C(=O)(C(O)C(CCC)NC(C1CCS1(=O)=O)=O)NC1(C#C)CC(F)(F)C1 C=CC1CCN(C(C2(NC(C3CCCOCC3)=O)CCOCC2)=O)C1 C1(CNC(C(C)(C)C)=O)CN(C(C2CCCCCC2)=O)CCC1C(F)(F)F N(C1CCc2cccnc21)C(C12C(NC(c3c(C)ncs3)=O)C3CC1C2C3)=O N1(C(C2(n3cc(Cc4cccc(C)c4)nn3)CC2)=O)CCCC2C(O)C(C)(C)C12 Cc1c(C(N2C(C(=O)NCC(F)CO)CC2C)=O)cccc1C#N C1(NC(C2CCCCC2)=O)CCCC12CCN(C(c1cc(Br)cs1)=O)C2 c1(C(=O)NC2(CNC(c3sccc3-n3cnnn3)=O)CC2)csc([N+](=O)[O-])c1 Cc1ccc(CCC(=O)NC2CCC(NC(C3SCCCS3)=O)C2)cn1 C1(C(=O)NC(C)CO)CCCN(C(c2cn(C)cn2)=O)C1 N1(CCNC(C(C)(C)F)=O)CCCN(C(C2C(c3ccncc3)C2(C)C)=O)CC1 C1(N(C(C(C(C)O)N(C)C)=O)C)CCCCN(C(c2ccc(O)cc2)=O)C1 Cc1cc(Br)c(NC(=O)NCC2CCOCC2C)cc1[N+](=O)[O-] CC12CCCCC1(C(N1CCC(CC(=O)NCCN3CCC(CO)C3)C1)=O)C2 N1(C(CCN(C(C)=O)C)=O)CCC(C(C)NC(=O)Cc2c(C)n[nH]c2C)CC1 c1(OC)cc(C=CC(=O)NCc2ccc(C3CC3)cc2C)cc(Cl)c1O N1(C(C2ON=C(CC)C2)=O)CCC2C(CCCN2C(=O)C(C)CC2CCCC2)C1 c1(NC)ccc(C(N2CCCC2CNC(=O)C(O)C2CCCC2)=O)c(C)c1 C1(C(C(=O)NCc2cccs2)N(C)Cc2cn(CC)nc2)CCC2(CC1)CC2 N1(C(C=Cc2cc(C)no2)=O)CCC2CC1CN2C(c1ccc2cnoc2c1)=O C1(C(N2CCC(NC(c3cn(C)nc3C3CCCC3)=O)C2)=O)CCC2(CCC2)O1 c1(C(c2nnnn2C2COC2)NC(C)CCCCO)cc(Br)cc2c1OCC2 C1(C(=O)NC(C)CN2CCN(C)CC2)CC12CCN(C(c1cnns1)=O)CC2 N1(C(C=CC)=O)CCC(C2(NC(c3cccn3CCC)=O)CC2)C1 Cc1cc(NC(=O)NC2CCN(C(=O)CC(C)(C)F)C2)ccc1NC(C)C C1(CNC(C2C(C)COCC2)=O)CC2(C1)CC(N)CCO2 c1(OCCOC)cccc(CC(=O)NC2CC(CO)N(C(=O)CC(F)F)C2)c1 N1(C(CCc2nc(C)sc2)=O)CCCN(C(=O)C(C)CC2CCCO2)CC1CO CC1CCC(NC(c2cncc(-n3cnnn3)c2)=O)CN1C(=O)CCC(C)(C)C C1(NC(CCNC(C)=O)=O)CCSC12CN(C(C1CCC1c1nncn1C)=O)C2 C1(NC(c2cncc(CC)c2)=O)CCCN(C(=O)Cc2ccnn2C)CC1 c1(C(=O)NCC(O)CCNC(C2(F)CCC2)=O)cnc2ccc(F)cn12 N1(C(C(c2cncnc2)C)=O)CC(CNC(c2ncc(F)cc2N)=O)C(C)(C)C1 N1(C(c2cc(CC)c(C)cc2)=O)CCC2(C1)CN(C(=O)CC1(O)CC1)CC(C)O2 N1(C(C(c2cc(C)oc2C)C)=O)C2CCC1C(CNC(c1cc(F)n(C)n1)=O)C2 C1(C(=O)NCC2(CCNC(=O)C(O)c3ccsc3)CC2)CC12CCOCC2 CC(C)(C)C(CNC(C1CC2(CCC2O)C1)=O)C(=O)NCCc1ccc(O)cn1 c1(NC(C2CCC(CN)CC2)=O)cnn2c1CCCC2 N1(C(c2c(COC)cco2)=O)CC2(CCCC(CNC(=O)C(C)C3CCC3)O2)C1 C(=O)(CC(C)CN(C)C)NCC(CC)NC(=O)CCc1ccc(CO)cc1 C1(CNC(c2ccc(OCC#C)cc2)=O)CN(C(C2CCCN2C)=O)CC12CC2 c1(C2(N(C(C(=O)NCC(n3cccn3)C)=O)C3CCCC3)CC2)ccccc1 C1(OC)CN(C(=O)CCCN(C(=O)C(C)(C)n2cncn2)C)CC12CC2 S(=O)(=O)(c1c[nH]ccc1=NCC1COCC(=O)N1C)N1CCCC(F)(CC)C1 c1(C(N(C2CCCN(C(C3(C)CC=CCO3)=O)C2)C)=O)cnc(O)c(F)c1 C1(OC)(CNC(=O)Cc2cncn2C)CCN(C(=O)C(c2ccc(F)cc2)=O)C1 Cc1csc2ncc(C(N3CC4CCN(C(=O)CC5CCCO5)C4C3)=O)c(=O)n12 C1(NC(=O)Cc2cncs2)CC2CCC1(C(=O)NCCCC(F)(F)F)C2 N1(C(c2ccc(C)c(Cl)c2Cl)=O)CC2COCC(C1)C2NC(=O)C(Cl)=CCl C(=O)(CC(C)CC(C)(C)C)N1CC(O)(C(C)NC(C=C(C)C(F)F)=O)C1 C=CCCC(C(=O)NCCCNC(=O)NC)NC(=O)C=CCCC c1(CC(=O)NCCOC2N(C(CC(CC)C)=O)CCCC2)cccc(C#N)c1 C1(C(=O)NC(CC)CNC(c2cc(Cl)c(Cl)s2)=O)CCc2nncn2C1 Cc1cnc(CN2CC(C(N3CCCCC(C)C3)=O)CC(F)C2)c(F)c1 c1(C(N2C(C)CC(NC(c3cc(CCC)[nH]n3)=O)C2)=O)coc2c(C)cccc12 CN1CCN(C(C2(F)CCN(c3ccc(CN)cn3)C2)=O)CC1 c1(C(=O)OCC)c(C)sc(CNC(CC2CCCN2C)C2CC2)c1Cl N1(C(C2CC2C2CCCC2)=O)CC2CCCC(C1)N2C(C1CCC2CC2CC1)=O c1(CC)cc(C(N2CC=CC2CNC(C2CC(N(C)CC)C2)=O)=O)ns1 Cc1cc(OCC(=O)NC2(CNC(c3cc(Cl)cn3C)=O)CCCC2)cc(C)c1 c1(CN2CCN(C3CN(C(C4C5COCC45)=O)C3)CC2)ccc(O)cc1O O=S(=O)(c1cccc(CNc2cc(Br)ncc2Oc2ccccc2)c1)N1CC1 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CCC1NC(C1CC=CC1)=O C1(CNC(c2c(OC)ccs2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC2(CCC2)O1 C1(C(=O)NCC2C(NC(C(c3nc(C)sc3)=O)=O)CCC2)CCCCCC1 N#Cc1c(N2CC3CC(C2)C3NC(=O)Cc2ccc3c(c2)COC3)cccc1F Cc1sc(C(=O)NCC2CC(C(F)F)CN2C(=O)CSC(C)(C)C)c(C)c1C c1(OCCOC)ccc(C(=O)OC(C)CC(=O)O)cc1 C1(CCNC(C(C=C)O)=O)CSCCN1C(c1cc(Br)nn1C)=O N1(CCNC(C2CC(OCC3(COC)CCOC3)C2)=O)CCCC(C)C1 c1(NC(=O)NC(c2ccc(C)nc2)C)ccc2c(c1)C(F)(F)C(=O)N2 C1(C(=O)NCCSCC(=O)Nc2c(COC)ncnc2)CC(C(C)C)=NO1 Cc1nc(C(N2CCN(C3CN(C(=O)C(F)F)C3)CC2)=O)c2ccccn12 Cn1c(C(=O)NC2CCC(CNC(c3cc(N)cc(N)c3)=O)C2)cc(Cl)c1Cl C1(NC(COC)=O)(CO)CN(C(=O)CCc2nnc(C(F)F)o2)C1 CC1C(NC(c2cnc(Cl)c(C3CC3)c2)=O)CCCN1C(C1CC2(CCC2)C1)=O C1(C(=O)NC(COC)C)C2CCCC1CN(Cc1c(Br)cc(Br)c(O)c1Br)C2 S(=O)(=O)(CCCOC)NC(C(COC)C)=O c1(C(=O)NCCNC(C(CC)OC)=O)cc2nc(Cl)ccc2o1 CC(C)C(C(=O)NCCc1ocnc1CO)C(C)NC(=O)CNC(N)=O CC1(C)CC(CNC(c2ccccc2)=O)CN(C(c2nnn3ccccc23)=O)C1 Cc1ccc(C)c(S(=O)(=O)NC2CN(C(c3nc(CO)cs3)=O)CC2O)c1 C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCN(C(=O)C=C2CCCC2)C1 N1(C(C(C2CCCC2)NC(CC2ON=C(C)C2)=O)=O)CC(O)CC1C(N)=O c1(C(=O)OC)ccc(C(=O)NCC2CCCCCN2C(c2cnco2)=O)cc1Cl C(=O)(CCCCCCNC1(CF)CCC1)NCC1(C)CCOC1 c1(OCCC)ccccc1C(=O)NCC(O)CNC(=O)C#CC(C)C c1(NC(CSS(=NC)(C)=O)=O)n[nH]c2c1CCN(C(=O)CCCC(CC)OC)C2 N1(C(CC#N)=O)CC(C2(NC(C3(C(=O)NCCc4ccccc4)CC3)=O)CC2)C1 C(c1ccc(Br)cc1)=CCCNC(c1c(C)nccc1)=O c1(C(N2CCCC(NC(c3c(CC)nn[nH]3)=O)(CO)C2)=O)cccc2c1COC2 C#Cc1cccc(C(=O)NCCNC(c2cc(O)nc(OC)n2)=O)c1F C(=O)(CC(C)CNC(=O)CCc1cncnc1)NCC(C#C)CC CC1CCC(C(=O)NCCCN(C)C)CN1C(=O)CCc1nc(=N)[nH][nH]1 C1(COC)CCN(C(=O)CNC(=O)COC2CC2)CC1.C12CCC1CNC2=O C12(C(=O)NCc3nccc(C)c3)CC(CO)(CN1C(C1CC3COCC3C1)=O)C2 C1(C(=O)N)(CO)CCCC1.C1(CC(=O)NC(C(=O)OC)C2CCCO2)OCCC1C c1(NC2CC(C)N(C(C3(CN(C)C)CC3)=O)C2)cc2nncn2cn1 c1(OC)cccc(Cl)c1CNC(N1CCC(C)C(NC(=O)OC(C)(C)C)C1)=O C(=O)(CC(C)CN=C(NCC1(O)CCN(C)CC1)NC1CCS(=O)(=O)C1)OC C1(NC(CNC(CN2CCC(C)C2)=O)=O)(CO)CCN(C)C1 C1(C(N(C2COCC2O)CC)=O)CC2CN(C(=O)CCCC(C)(C)C)CC2C1 C1(CNC(C2(SC)CCC2)=O)CC(C(=O)Nc2cc(C)ccc2O)=NO1 C1(CNC(CC(C)C(F)F)=O)CN(C(=O)CCn2ccnc2)C2(CCOCC2)C1 Cc1nc(C(=O)NCCC2CC(NC(C3C(C)C3(F)F)=O)C2)c(C)n1C1CC1 c1(SCC)cncc(C(N2CC(CNC(c3c(C)cnn3CC)=O)(OC)C2)=O)n1 Cc1cc(C(=O)NNC(=S)NC2CCS(=O)(=O)C2)c(C)n1C C#Cc1ccc(C(N2CCCC2CN=[N+]=[N-])=O)cc1C N1(C(c2cnc(SC)n2C)=O)CCC(NC(C2CC2C)=O)C(F)C1 C1(NC(COCCOCC)=O)CN(C(C2CCC(O)CC2)=O)CC1C C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC(CCNC(c2ccccc2)=O)CC1 Cn1ncc(Cl)c1CC(=O)NCCCN1CCN(C(C2CC23CCC3)=O)CC1 C1(NC(C2COCCC2(F)F)=O)C2CC1CN(C(c1ccccn1)=O)C2 CN=c1[nH]cc(C(=O)NCc2c[nH]nc2C(=O)NC(C)C(C)n2cccn2)s1 c1(NC(N2CCCC2)=O)nc(Cl)nc2[nH]cnc12.c1(O)cc(OC(F)(F)F)ccc1C c1(OCN2C3(CCC(N)C2)CCC3)cccc2[nH]c3ccccc3c12 c1(C(=O)NCC(C)NC(=O)C2=CCCC2)cc2ccnn2cn1 c1(C(N2CC(C(N3CCC(OCC)C3)=O)(SC)C2)=O)cnncc1O c1(OC)ccc(C(=O)NC2CC(CC(N3CC4C(C3)C4(C)C)=O)C2)c([N+](=O)[O-])c1 Cc1cc(C(=O)NCC23CC2CN(C(=O)C#CC2CC2)C3)ccc1F C1(CCC)(NC(=O)C(C)CCCOC)CCCN(C(c2c(C#N)cnn2C)=O)C1 C1(C)(CNC(CC2CCCC(C)O2)=O)CC(F)(F)CN1C(c1cnn[nH]1)=O CCC(C)C(O)CC(=O)NC1CCOC1C(=O)NCC(C)(C)C1=CCCC1 C1(F)(C(N2CCC(C(C)NC(c3cnccc3Cl)=O)CC2)=O)CCCC=C1F Cc1ccc(S(=O)(=O)NC2CCCC2NC(N2CCCSCC2)=O)c(F)c1 C1(C(=O)NCCN(CCC)CC)CC(O)CCN1C(=O)CNC(=O)NC CCCC(CC)C(=O)NC1CCCCC1CNC(c1ccc(F)s1)=O N1(C(Cc2c(C)cco2)=O)CCC(c2ccccc2)(NC(C2CC23CC3)=O)CC1 C(CN(C(C(C)(C)C)c1ccccc1)C)(C(C)C)OC.C1CO1 c1(OCC)cc(NCC2CC(NC(C3CC3F)=O)C2)nc(C)n1 Cc1nc(Br)ccc1C(N1CC2CCC2(CNC(=O)Cc2cc(Br)cs2)C1)=O N1(C(c2c(C)snn2)=O)CC(NC(c2cn(C)cc2C(F)(F)F)=O)CC(O)C1 c1(CC(=O)NC(CNC(C2N(CC)CCC2)=O)(C)C2CC2)nc2ccccc2s1 Cc1cc(NC(C(C)NC(c2cccc(F)n2)=O)C(C)C)nc(S(C)(=O)=O)n1 C1(C(N2CC(CNC(c3cncc(SC)c3)=O)C(C)C2)=O)CCN(C)C(=O)C1.C1CC1 c1(C(N2CCN(C(CC(CCC)C)=O)CC2CCO)=O)cc(F)c(C#N)c(F)c1 C1(NC(C(C)=CC2CC2)=O)COC2(C1)CN(C(C1CCCC3(CC3)C1)=O)C2 CC(C)CCC(F)C(=O)N(CCCNC(=O)C(C)C1CCOC1)C(C)C c1(C(=O)NCC(C)CN(C(=O)Cc2cncn2C2CC2)C)n[nH]c2c1CCOC2 N1(C(c2c(CC)ccs2)=O)C2CCC1CC(NC(C1C=C1C)=O)C2 Cc1cccc2cc(C(=O)NCCCOCCNC(C3COC(=O)C3)=O)oc12 CC(C)CC(C)(C)C(=O)NC1CCCC1NC(c1ccccc1CO)=O C1(NC(CC(C)F)=O)CCC(NC(c2nccnc2N)=O)CC1 C(=O)(C(C)CO)N(C(C(=O)N(CCCOCC)C)C1CC1)C N1(C(c2cc(OC)c(Br)nc2)=O)CCC(C)(C)C(NC(C2CCC2)=O)C1 CCCC(CC1CCCC1)C(=O)NCC1CN(C(=O)C(COC)N=[N+]=[N-])C1 C1(NC(C(CC=C)OC)=O)COC2(C1)CN(C(=O)CC1OCCO1)C2 c1(CC(=O)NCC2C(C(=O)Nc3cccc(OCC)c3)C2)cc(C)ccc1F N1(C(C2CCC(C)O2)=O)CC2CC(C1)CN(C(=O)CN1CCCCC1)C2 c1(C(N2CC(NC(C3C(CCC)CCC3)=O)(CO)C2)=O)cnc2c(c1)COCC2 c1(OC)ccccc1CN(C(=O)CN(CCN(C)C)C(C1CCC1)=O)C Cc1ccc(C(N2CCCC(N(C(=O)CC3CCC(C)CO3)C)C2)=O)cc1C C1(C(N2CCCC(C=C)C2)C(=O)NCC(=C)C)Cc2ccccc2C1 c1(C(N2CCC(O)C(C(N3CC4COCC4C3)=O)C2)=O)ccc(F)c(I)c1 C1(NC(C(CC2CCC2)OC)=O)CCC(C)(CNC(C2CCC(=O)O2)=O)C1 Cc1cc(Cl)c(Cl)cc1C(=O)NC1CN(C(=O)C(O)CC(F)F)C2(CCC2)C1 N(C1CCCc2occc21)C(CCCNC(=O)C=CC1CCOCC1)=O C1(C2CCCN(C(=O)CN(C)C)C2)(NC(CN(C)C(c2ccncc2)=O)=O)CC1 c1(CNC(=O)NCC2CC23CCC3)ncc(Cl)cc1Cl C1(NC(CC(C)N(C)C)=O)CC=CCC1C(N1CC(N(C)C)CC1C)=O C=C1CCN(C(C2COCOC2)=O)C(C(N2CCC(OCCO)C2)=O)C1 N1(C(c2c(SC)ccs2)=O)CC2(CCC2)CC1CNC(=O)CN(C1CCC1)C c1(C(=O)NC(CC=C)CNC(=O)Cc2ccn(CC)n2)cc2c(s1)CCC2 N1(C(c2c(C)cccc2N)=O)CC(C)(CNC(C23CCC2C3)=O)CC1(C)C c1(C(=O)NCCN(C(C(n2c(C)ccn2)C)=O)C(C)C)cnc(=NCCF)[nH]c1 C1(NC(C(CC)OC)=O)CCSC12CN(C(c1cc(O)ncc1Br)=O)C2 c1(C(=O)NCC(C2CC2)NC(C=C(C)c2cnn(C)c2)=O)ccc(S(C)(=O)=O)[nH]1 c1(C(N2C(CNC(C3CC=C(C)CC3)=O)C(C)CCC2)=O)c([N+](=O)[O-])cnn1C C(=O)(C1=CS(=O)CCC1)N1CC(C)C(CNC(C2(C)CNC(=O)C2)=O)C1 C1(NC(CCC=C)=O)COC2(CCN(c3ncc4[nH]ccc4n3)CC2)C1 C1(C(=O)NCC(CC2CC2)CO)(CNC(C=C(C)C(F)F)=O)CCCC1 N1(C(Cc2ccn(C)n2)=O)CCOC(C)(CNc2ccccc2)C1 CCC(C)(C)CC(=O)N1CCOCC(CNC(c2c(Cl)csc2Cl)=O)C1 CCCC(CNC(c1cc(C)nn1C)=O)C(=O)NC1CC12CC(OC)C2 C1(CC=C)(CNC(=O)Cc2cnoc2)CCCN1C(=O)C(O)CCN(C)C Cc1nc(C(=O)NCC2(F)CC(CNC(=O)Cc3cnn(C)c3)C2)c(C)s1 c1(C(N2CC(NC(C3N(C)CCC3)=O)C(F)C2)=O)cc2nnn(C)c2s1 CN1N=C(C(=O)N2CCC3CC23C(=O)NC2CCCC2C#N)CCC1=O c1(C(N2N=C(C=O)CC(C)C2)=O)cnc2ccc(Br)cc2c1 C(CC(=O)N1CC(O)CCO1)NC(C(c1ccccn1)C)=O c1(C(N(C(=O)NCCN(C2C(F)(F)C23CC3)C)C)O)ccccc1Cl c1(N(C)C)ccc(S(=O)(=O)NCC2COCO2)cc1 Cc1ncc(S(N)(=O)=O)cc1C(=O)NC1CC1NC(C1CCC(C)(C)O1)=O c1(OC)ncc(-c2scc(C)c2C)cc1C(=O)Nc1scc(C)c1C(N)=O C(CCC(C(=O)N(C)Cc1cocn1)NC(c1cc(CCO)on1)=O)OC C(=O)(C1=CCN(C(=O)Cn2cncn2)CC1)NC(C)C CC1CC2CC2CC1C(N1CCCC1CN(C(=O)CCc1cccnc1Cl)C)=O S(=O)(=O)(c1ccc(Br)cc1)NC1C(C)(C)NC(=O)CC1 c1(C(N2CCC(NC(C3CCC(C#N)CC3)=O)C2)=O)ccn2cccc2c1 N1(CC(=O)N(C2CCN(C(COCC(=C)C)=O)C2)CC)CCN(C)C(=O)C1 C12(C(=O)NCc3c(C)noc3)C(NC(c3ncc(F)cc3C)=O)C3CC1C2C3 CCCC(F)(F)C(=O)NC1CCOC(C(=O)NCc2cn(C)nc2OC)C1 C1(CC(=O)N(C2CCN(C(=O)C(C)C(=O)OC)C2)CCC)(COC)CCCCC1 c1(C(=O)NCC(C)NC(C=Cc2ccc(SC)s2)=O)ccc2nc(O)n(C)c2c1 c1(C(=O)NCC(C)N(C(=O)C(C)OCC(C)C)CC)cnsc1C C#Cc1cc(C(=O)NCC(C)(O)CNC(=O)C(C)(C)N(C)C)cc(F)c1 C(=O)(C(C)CC(=O)c1ccc(F)cc1)NCC#CCNC(C(C)SCCCC)=O C1(C(=O)NCCC(C)NC(c2c(C(=O)OCC)c[nH]c2)=O)CCN(C)C1C c1(CC(=O)NC2(CNC(C(CC)O)=O)CCOCC2)cc(F)c(F)cc1F CC(C(=O)NCC(C1CC1)N(C)C(C1CC(=O)C1)=O)S(C)(=O)=O C1(=O)CCCCCN1C.C1(C(=O)NCC2(C(=O)OC)CC2)C2CCC(C2)C1C c1(CC(=O)NC2CC(CNC(c3cncc(F)c3)=O)C(O)C2)n[nH]c2c1CCCC2 C1(CC(=O)NCc2cnc(C)s2)CC(NC(C23CC(F)(C2)C3)=O)C1(C)C c1(-n2cc(CC3N(C(=O)NC4CC4c4cccs4)CCC3)nn2)ccccc1F c1(C(=O)NCCC(C)NC(C2CC23CCC3)=O)cncc(S(C)(=O)=O)c1 Cc1cc(C(=O)NC2CCC(C)(N3CCOCC3)CC2)nnc1O c1(C(N(CCCNC(c2nccc(OC)c2F)=O)C)=O)nc2n(c1Cl)CCCC2 C1(CNC(C2C(c3cn(C)nc3)CCO2)=O)CN(C(c2csc(Cl)n2)=O)CCO1 N1(C(C(c2cncnc2)C)=O)CCCC(C)(C)C1C(=O)NC1C(C)CCC1C Cc1nsc(N)c1C(N1CCC(C(C)NC(=O)C#CC2CC2)CC1)=O C(=O)(C(C)(C)CCCO)NCC(C)(C1CC1)NC(C1CN(C)C(=O)CC1)=O Cc1ccc(Cl)c(F)c1C(=O)NC1CC(C(=O)O)C2CC12 c1(C(=O)OC)cc(C(=O)NCC2(CNC(c3nc(=O)n(C)[nH]3)=O)CC2)cn1C c1(C(=O)NCCC2CN(C(CN(C)C)=O)C2)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 C=CCCCC(C(=O)N1CCCC(C#N)C1)NC(=O)C(C)C(O)C(C)C Cc1nc(O)c2cc(C(=O)NCC3CC3NC(C3CC4CCC3O4)=O)ccc2n1 C(C(CC(F)(F)F)NC(C1CCC1(C)C)=O)NC(C1(CC#C)CCC1)=O N1(C(CC2CC(=O)NC2=O)=O)CC2CCC1C(NC(c1ncc(Cl)s1)=O)C2 c1(C(N(C2CCN(C(=O)Cn3nccn3)CC2)C)=O)cc(C(F)(F)F)cc(O)c1 CCCCCC(O)CC(=O)N(CCC(C(C)C)NC(c1ccc(N)c(F)n1)=O)C n1(CC(=O)NCC2(NC(C3CC=C(C)CC3)=O)CCC2)nc(C)c2c1CCCC2 CCCCC(CC)CC(=O)NCCN(CCOC)C(c1cc(Cl)nn1C)=O Cc1ncsc1COCC(=O)NCC(C)(C1CC1)NC(C1CCC(C)S1)=O C(=O)(C(F)(Cc1ccccc1)C(C)C)OC.C1(=O)C(CO)(CO)N1 c1(N2CCC(C(C)NC(C(CCCC)C(C)C)=O)C2)nc(Cl)nc2[nH]c(O)nc12 C(CCCCCCC(=O)NC(CNC(=O)C(C1CC1)C1CC1)CO)SC C1(N(C(=O)NC(c2ccc(C(F)(F)F)cc2)CC)CC(C)(C)C)CCCCC1O c1(-n2cc(-c3cnc(C)s3)nn2)ccncc1C(=O)NC1NC(=O)C2CC12 C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(=O)C(C)(C)CF)C2(CCOCC2)C1 C1(NC(c2ccc(F)cc2Cl)=O)CC(C2CCN(C(=O)C3=C(Cl)CCCC3)C2)C1 CCCC(CC(=O)NC(C)COCC)NC(=O)CC1CCC(=O)NC1 CCCC(CCCNC(C1CC(C)OC1C)=O)N=c1nc(C)[nH]s1 C(=O)(C1CCc2c[nH]nc21)NCC(CCOC)NC(c1ccc(F)c(C)c1)=O N1(C(=O)NC(C)Cc2ccncc2)CCC(F)(C(c2ccccc2)O)C1 CC(CS(C)=O)C(=O)N(C)CC1(NC(c2cccc(N3CCOC3=O)c2)=O)CC1 c1(CC(=O)N(C)C)cn2ccccc2n1.C12CCCN(C1)CC(=O)NC2 c1(C(=O)NCC2CCC(NC(c3c(C)ncs3)=O)C2)nc(O)c(C)s1 N1(C(CNC(CCCCC)=O)=O)CCC(NC(c2ccoc2)=O)C2(CCC2)C1 C1(C#N)(C(N(CC(=O)NC2CCN(CC)C2)CC)=O)CCCO1 C(CC(C)C)(C(=O)NCC(C)(C)NC(=O)CCc1cccc(OC(F)F)c1)OC n1(CC(C)N(C2CCCNC2)C2CC2)cc(Cl)cn1 Cn1[nH]c(C(=O)NCC2CC(CNC(C3(C(F)F)CCCC3)=O)CO2)nc1=O N1(C(c2c(C)nc(O)cc2)=O)CCC2(NC(=O)Cc3ccco3)CCCC12 C1(NC(CCN(C)CCO)=O)(CNC(=O)CC2OCCO2)CCSC1 C1(C(=O)NCC2(NC(CN(C(C)C)C)=O)CCC2)CCC2(CC2)C1 CC1(C)C=C(C(=O)NCC2CCCC2NC(=O)CC2CCC(C)(O)CC2)C1 N1(C(c2c(OC)csc2)=O)CCC(O)C(C(N2CCCCC2C)=O)C1 c1(C(=O)NCC(c2ccccc2)CN(C)C)ccc2[nH]c3c(c2c1)CN(C)CC3 c1(-n2cc(CCCC(C)=O)nn2)cc(C(=O)NCCCSC(F)F)c(=O)n(C)c1 C1(C)(NC(C2CCC(C)O2)=O)CCN(C(=O)CC(C)F)CC1 C1(NC(c2c(C)onc2-c2ccccc2Cl)=O)CCN(C(=O)C(C)C)CC1F N1(C(C(F)=CCC)=O)Cc2ccccc2CC1CNC(=O)CC1CNC(=O)C1 C(=O)(C(C)S(N)(=O)=O)NC(C1(C(N2C(CSC)CCC2)=O)CC1)(C)C n1(CC(=O)NCC(c2ccccc2)NC(C=CCCC)=O)c(C)ccc1C c1(COC)ccc(C(=O)N(C2CCN(C(=O)CO)CC2)C)cc1OC C(=O)(C1=CCCSC1)NC(C(C)O)C(=O)N(C1(CCO)CC1)C C=CC(C)CC(=O)NCC(C1CCCCC1)NC(c1cc(C(C)(F)F)on1)=O C1(CN(C(C2CCCC2F)=O)CC)CCCCN1C(=O)CCSCC(N)=O C(=O)(C1=CCCC1C)NCC(C)N(C)C(c1cn(C)nc1C1CCOCC1)=O CC(F)(F)CC(=O)NCC1(CNC(C2CCNC(=O)C2)=O)CC1 S(=O)(=O)(c1cccc(S(=O)(=O)NC(C)(C)C)c1)NCC(=C)CC c1(C(N(C)CC2N(C(C(C)SCC)=O)CCCC2)=O)cc(O)cc(=O)o1 N1(CCNC(=O)CC2CCCO2)CCN(C(=O)C(O)Cn2cncn2)CC1 c1(C(=O)NCC=CCNC(C2CC(OC(C)(C)C)C2)=O)ccc2ncsc2c1 N1(N2C(C=O)C(C(=O)C3=C(Cl)CCOC3)CC2)CC2(CNC(=O)N2C)C1.CC(=O)NC c1(NC(C2N(S(CCC)(=O)=O)CCNC2)=O)cc(F)ccc1[N+](=O)[O-] c1(CNC(C2CCCCN2C(=O)NCCC)=O)cc(F)c2cc[nH]c2c1 C1(C(=O)NCC2(C(C)N(C(=O)CC(C)n3cccn3)C3CC3)CC2)C2CC(=O)CC12 N1(C(c2nc(C(C)OC)oc2)=O)CCCC(O)(CCNC(c2cnns2)=O)C1 N1(C(C2(C#C)CCCC2)=O)CCN(C(=O)CCC(C(=O)OC)OC)CC(CO)C1 N1(C(C=CC)=O)CC2CCC1CC2NC(=O)CC(C)(C)O N1(C(c2nc(CC)oc2)=O)CC(NC(C2CCC(=O)N2)=O)CC2(CC2)C1 c1(C(=O)NCCCC(C)NC(C2CC3C=CC2C3)=O)cnn2cc(C#N)cnc12 N1(C(c2cn(C)nc2)=O)CC(CNC(=O)Cc2cccc(OCC(F)F)n2)C(O)C1 C1(C(N(CC(C)C#N)C)=O)CC2CC1CC2NC(=O)CCC(N)=O n1(CC(=O)NCC2C(CNC(c3c(N)cn(C)n3)=O)C2)cc([N+](=O)[O-])cn1 C=CC(CC)C(=O)NC(C1CCN(C(C2CC(OC(C)(C)C)C2)=O)CC1)C C1(C(=O)NCC(C(=O)NC2C=CCC2)N(C)C)(OC)CCOC1 c1(C(N2CCCC(CNC(C(C)c3ncco3)=O)C2)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NCC(C)CNC(c2ccnn2CC(F)F)=O)cccc(Br)c1 N1(C(C(CN(C(=O)CN(C2CCC2)C)C)(C)C)=O)CCCN(C)C(=O)C1 N1(C(c2cc(O)ccc2O)=O)CCN(C(c2cc(Cl)ncc2Cl)=O)C2(CCC2)C1 N1(C(C2(CC=C)CCOC2)=O)CCCC2(CCCN2C(c2cnn(C)c2C)=O)C1 C(C)(CCC(=O)NCC1CCN(C(c2csnc2Br)=O)CC1)SC Cc1cccc(C)c1C(c1nc(-c2nccs2)nn1CCc1ccc(Cl)cc1)C Cc1ccc(C(=O)NC2CC(C)CN(C(c3ccnc(C)c3C)=O)C2)cc1Cl C1(C(N(C2CCCOC2)CC)=O)COC(CNC(=O)CCCOC(C)=O)C1 C#Cc1c[nH]nc1C(=O)N(Cc1cncc(C(N)=O)c1)CC C(=O)(CS(=O)(=O)C(C)C)NCC1C(CNC(C2(OC)CCCCC2)=O)C1 c1(C(=O)NC2COC3CN(C(CCOC(C)C)=O)CC32)cnc(O)c2cncn12 CC(C)C(C)CC(=O)NCCC1CN(C(=O)C(O)CN(C)C)C1 n1(CCC)nc(C)c(C(=O)NC(CNC(c2n[nH]c(Cl)c2Cl)=O)CO)c1C C(=O)(C(CC(F)(F)F)NC(=O)Nc1cccnc1OC)OCCCC C(=O)(CC(F)(F)F)N(C(Cc1ccccc1Br)C(=O)NC1CC(CCF)C1)C n1(COC(c2ncnc3c2ncn3CCl)=O)c2ccccc2c(=O)c2ccccc12 C(CCN=c1ccnc(SC)[nH]1)NC(C(CC)F)=O c1(C(N2C3CC(NC(CCCC(C)=O)=O)(C3)C2)=O)cnc2c(F)cc(C)cc2c1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC2(CNC(c2csc(C)n2)=O)C1 C1CCS(=O)(=O)C(C)(C)C1.c1(C(C)C)nn(C)c(Cl)c1CNc1nnnn1C C1(C(N(CCOCCNC(c2c(CC)c[nH]n2)=O)C)=O)C(O)C(=O)N(C)C1C C12(C(N(C(C)C3CC3)C)=O)CC(NC(=O)CC3OCCO3)(C1)C2 c1(CC(=O)NCCN(C(=O)C2=NOCC2)CC)cc(C(F)(F)F)cc(Cl)n1 CCCCC(C)C(=O)N1CCC(O)C(NC(=O)CCC(=O)NC)C1 N1(C(C2(CC)CC2)=O)CC2(CCC(CNC(c3cc(C4CCC4)on3)=O)O2)C1 c1(C(C)NC(C(C2CCC2)OC)=O)cnccc1C n1(CC(=O)N(C(CC)CSc2ccccc2)C)cc(C=O)c(C)n1 CCC(CNC(=O)C(C)CN(C(=O)CSCC(N)=O)C)CC(C)C C(=O)(C1CCCc2nc[nH]c21)NCc1nc(O)cc(CNC(C(C=CC)O)=O)n1 Cc1nc2ncnn2c(C)c1C(=O)NCC1CN(C)CCN1C(c1ccon1)=O c1(CC(N2CCC(OCCNC(c3c[nH]nc3F)=O)C2)=O)ccc2c(c1)OCO2 C1(NC(c2ccnnc2)=O)CN(C(=O)Cc2ccc(Br)s2)CCC1CO C1(CCO)(NC(c2cnc(-c3ncccn3)s2)=O)CCNCC1 c12cccnc1N2.c1(C(N(CC(CN(C)C)O)C)=O)ccc(C(N)=O)cc1 C(c1ccc(F)cc1)=CC(N1CCC(N(C(CC=C(C)C)=O)CCO)C1)=O N1(C(C2C(=C)C2)=O)CC2(CC(NC(c3cn(C4CC4)nn3)=O)c3nccn32)C1 C(=O)(C(F)CC(CC)CC)NCC1C(CC)CN(C(=O)C=CC=C(C)C)CC1 c1(C(N2CC(C)N(C(=O)CCC3CCCCO3)CC2)=O)nncc2c1CCCC2 C(C(O)CC(=O)NC1COCC1CO)NC(Cc1n(C)nnc1)=O N1(C(c2ncc(C(C)C)cn2)=O)CCN2C(=O)C(C)CC2C1 S(=O)(=O)(c1ccc(NC2CCN3CCCC23)c(Br)c1)N(CC(OCC)OC)CC C(=O)(C1=CCC(NC(C2CC(C3CC3)C2)=O)C1)N(CC)CC1CCOCC1 c1(C(=O)NC(CC)CNC(=O)C(CO)NC(=O)C(F)(F)F)cc2sc(C)cc2s1 N1(C(C(CCC)NC(C2CNC(=O)C2)=O)=O)CCC(=O)N(C)CC1 N1(C2(C#N)CCN(C(=O)NCc3cccs3)C2)CCC2(CC1)CC2CCCO C(CC(=O)NOC1CCCC1)NC(C=CC(C)N(C)C)=O c1(CNC(C2COCCN(Cc3cc(O)ccc3Cl)C2)=O)ccc2c(c1)OCCO2 C(=O)(CS(=O)(=O)CC(=O)N1CCCC(NC(=O)CC2CCC2)CC1)OC N1(C(C2CC(CC)C2)=O)CCC(NC(=O)Cc2ccc(CO)cc2)C(O)C1 C(=O)(C1=CCSC1)N1C(C(=O)NCC(C)OCCO)CCC1 c1(C(C)C)cnn(C)c1C(=O)N(CC(O)CNC(=O)C(C)(C)CO)C C1(NC(C2CCOC2)=O)CCN(C(=O)C(F)C2CCC2)CC1C(N)=O c1(C(C)CC(=O)N(CCNC(C2COC2)=O)C2CC2)ccccc1Br C1(C(=O)OC)CCC(NC(=O)OC(C)(C)C)CN1C(=O)OCc1cn(C)nc1I N1(C(Cc2c(CC)con2)=O)CCC2(CC2NC(C2CCCC(F)C2)=O)C1 S(=O)(=O)(CC#Cc1ccccc1)NC(CCC1CC(C)OC1=O)=O C1(NC(Cc2ccn(C(C)C)n2)=O)CCC2CN(C(c3cc(Cl)cs3)=O)CC2C1 C1(C(=O)NC(C)(C)C)CC2CC2N1C(=O)N.C(CCC=O)OCCOCCOC N1(C(c2[nH]c(=NCC)sc2)=O)CCC2(CCCN(C(C3CCOC3(C)C)=O)C2)C1 CCN=C1NCCOCCN1.C(CCC)NOC n1(CC(=O)NC2CC(NC(Cc3cc(C)nn3C)=O)C(O)C2)nc(O)ccc1=O Cc1ccc(C)c(NCC(N2CCN(C(=O)CSC(F)(F)F)CC2CCO)=O)c1 C1(SCC(=O)NCC(O)CNC(C2(c3cnsc3)CC2)=O)CCCCO1 CN1CC2CCN(C(=O)CCN(C)C(c3ccc(C#N)o3)=O)C2C1 c1(C(N2CC(NC(C3(C#N)CC4CC4C3)=O)C2)=O)cc2c([nH]1)CCCC2 CC(O)(CC(=O)NC1C2CCC1N(C(c1[nH]nnc1C1CC1)=O)C2)C(F)(F)F c1(COC)ccoc1C(=O)NC(C)C(C)NC(=O)CCc1ncccn1 n1(CC)ncn(NC(=O)c2cc(C)n(CNC(=O)C=CCO)n2)c1=O Cc1nc(NC(C2(C)CN(C(c3cccc(O)c3)=O)C2)=O)c2sccc2n1 C(=O)(C1=CCCOC1)N1CC(C)C(CCNC(=O)CCc2cccs2)C1 N1(C(Cc2c(C)non2)=O)CCOCC1CNC(=O)CSc1cn[nH]c1 CCC(CC)(CC)C(c1ccccc1)N(S(=O)(=O)CC(=O)OC)C C1(NC(CCCOC(C)C)=O)CCN(C(=O)CCC2CC2(C)C)C1C N1(C(c2ccnnc2)=O)CCC2(CC1)CC(NCc1ccnc(O)c1)C2 N1(C(C(C)NC(=O)C(C)(C)C)=O)CCCC(NC(c2cnc(C#N)s2)=O)CC1 Cc1oc(Cl)nc1C(=O)NC1CCN(C(=O)CSC2CCOC2=O)C1C1CC1 Cc1cc(C#N)cnc1N1C2CCC1CC(CC(C)NC(=O)C=CBr)C2 C1(OC)CC(CCNC(=O)CC2CCC(=O)N2)N(C(=O)Cc2nc[nH]n2)C1 C(C)(CNC(=O)C(C1(O)CCCC1)F)(CC(C)C)NC(Cn1c(C)cc(C)n1)=O C12(C(N(CCC(=O)N(C)CC3(C#N)CC3)CCO)=O)CCC(CC1F)C2 C1(C(N(CC(C)C)C)=O)(NC(C23CC(C#N)(C2)C3)=O)CCCC1C C1(C(=O)NCC2CN(C(=O)CC(O)C3CCCC3)C2)C2CC3C(C2=O)C13 c1(C(N2CCN(C(CCC(C)C#N)=O)C(C(F)F)C2)=O)ccc2sncc2c1 C1(CC(=O)NC2CC(C)(CNC(c3cnc(C)[nH]3)=O)C2)CCCCC1O c1(C(=O)NCCN(C(C(C=CC)O)=O)CCOC)c(C)[nH]cc([N+](=O)[O-])c1=O C1(C(=O)NCC2CCC(NC(c3ccno3)=O)CC2)CN2CCN1CC2 C(=O)(CC(=O)NCC(C1CC1)NC(=O)Cc1cncn1C)OC N1(C(C2C(=C)CC2)=O)CCC2(CCCN(C(=O)CCc3cnc(OC)s3)C2)C1 Cc1ncccc1CCC(N1CC(F)CC1CNC(=O)CCc1cncs1)=O C(CC(C)(C)C)N(C(C(C)N(C)C(C1CCCOC1)=O)=O)CCN(C)C CC(C)CC(C(=O)NCc1cccs1)ONC(=O)C(C)(O)C1CCCC1 C1(CNC(C(CC)C)=O)CCOCC1C.C12(CC1)CC(=O)N2 C(=O)(N=c1cc(C)o[nH]1)NC(C(=O)Nc1cccc(C)c1)CC1CCCC1 N1(C(C(CCSC)NC(C2CC(F)(F)C2)=O)=O)CCn2nc(C)cc2C1 N1(C(c2nc(C)oc2C)=O)CCCC(C2CCN(C(=O)C(C)(C)CO)CC2)C1 CC(C)C(C)C(=O)NC1CCCCC1CNC(=O)C=CI c1(C(=O)NC(CC2OCCO2)CO)cncc2c1CCCC2 c1(NCC2(CNC(c3cc(C)c(C)s3)=O)CCC2)ncnc2cnn(C)c12 C1(NC(c2cnn(CCF)c2)=O)CN(C(c2cccc(F)c2)=O)CC12CC2 N1(C(c2cc(C)cc(OC)c2O)=O)CCCC2C1CCCN2C(C)=O C1N=C2NC3=C(C(=NCCOC14CCCC4)N2)COCC3.C(=O)(N(C)C)NCC C(=O)(C1CCCCc2ccccc21)N(CCCNC(C(CSC)(C)C)=O)C(C)C C1(NC(COC)=O)CC2(CCN(C(C3CCC4CCC34)=O)CC2)C1 c1(C(=O)NCC2CN(C(C(CC)C(C)C)=O)CC2O)cc2cccnn2c1 c1(NC(C(c2cccc(Cl)c2)CC)=O)ccc2c(c1)oc(=O)n2C C1(NC(CCCC#CC)=O)CN(C(c2cc(Cl)ccc2OC)=O)C2(CCC2)C1 Cc1ccc(C(=O)NCCNC(N2CCCC(Cc3ccc(O)cc3)C2)=O)cc1 C1(C(=O)OCCn2c(NC(C(=O)NC)=O)ccn2)CCC2COCCC2C1 c1(C(N2CC(CCC=C)(C(=O)NC(CC)C(C)(F)F)C2)=O)c[nH]c2cnccc12 N1(CC2CC3(CCC3O)C2)CCC2CN(C(=O)CC3(C#N)CCCCC3)C2C1 C(=O)(C(CC)CCOC)N1C(CCNC(C(CC)CC)=O)CCC1 C1(C(=O)NC2C(C#C)CCC2)CC2CC1CC2NC(c1ccn(C(C)C)n1)=O C1(CNC(=O)C=CC2CCCO2)COCCN(C(c2ccc(Cl)nc2)=O)C1 C1(NC(C2C3(CN(C(=O)OC(C)(C)C)C3)C2)=O)CCC2(CC1)CC2C#N c1(NC(C2(C)CCN2C(=O)Cn2cc([N+](=O)[O-])cn2)=O)cc(Cl)nnc1Cl C(=O)(C1CCOc2c(F)cccc21)N1CCCCC(NC(C(=O)NC2CC2)=O)C1 N1(C(C2CC(C)(CC)C2)=O)CC2CCCC(N(C(=O)CC(C)C(F)F)C)C2C1 N1(C(C2N(C)CCCC2)=O)CCC2(CC(NC(=O)C=CCF)C2)C1 C1(CCC)CC(C(=O)N(C)CC2CCCN2C(=O)C(CC)n2cncn2)CCO1 C1(CNC(C(CC)(C)CC)=O)CCN(C(=O)Cc2nncn2C)CC1(F)F C1(C(=O)NC2C(NC(c3ccn(C)c3)=O)COC2)CCOC1(C)C c1(OC)cc(CN(C2CCCN(C(C3CC(C)C3)=O)C2)CCO)nn1C C12(C(=O)NC3C4CC(NC(CC(C)SC)=O)CC43)CC1COC21CCC1 c1(C(N(C)CP(C)(C)=O)=O)coc2c1CN(C(=O)Cn1ncn(C)c1=O)C2 c1(COC)cc[nH]c1C(=O)NCCn1cc(C(=O)NCC2CC3(CC3)C2)nn1 C(=O)(C(O)CCCNC(c1c(OC)noc1C)=O)N(C(CC)C)CCO N1(CC)OCC(NC(=O)CC(F)(F)c2cscn2)C1=O.n12cc(nn1)COCC2 N1(C(CNC=O)=O)CCCCC1C1CCCN1C(C1CCC(=C(F)F)CC1)=O CCS(=O)(=O)c1cccc(C(=O)NC2CC(n3cc(C4(O)CCC4)nn3)C2)c1 C(CC(C(=O)NCCn1ncnn1)NC(=O)C(c1cnn(C)c1)=O)=CC CC1(C)CC1(C(=O)O)NC(=O)Cc1nc(-c2cccs2)cs1 c1(N(C2CCNC2)C(c2ccn(Cc3ccccc3)n2)=O)ccnc2ccnn12 N1(C(CCCCCSC)=O)CC2CCCC(C1)N2C(=O)C1CCCc2cncn21 c1(C(=O)NCC(CNC(c2ncccn2)=O)F)c(Cl)sc2nnsc12 C1(C2CCC2)(C(=O)NCC2(C)CCCN(C(C(C3CCC3)OC)=O)C2)CC1(F)F C1(CCC)CC(C(N2CCC(OCCNC(=O)COC(C)CC)CC2)=O)CCO1 c1(CC)conc1CC(=O)NC(CNC(=O)CCc1ncnn1C)C1CC1 c1(C(N2C3C(NC(c4ccn(C(C)C)n4)=O)CC(C3)C2)=O)cnn2c1NCCC2 [N-]=[N+]=NC1CN(C(=O)CCn2cc(Cl)cn2)CC1NC(=O)CNc1ccccn1 c1(C(=O)NC(C(=O)NC(Cc2cc(C)[nH]n2)C)C2(O)CCC2)cccn(C)c1=O CCCCC(CC)C(=O)NCC1(NC(=O)C(C(C)(C)C)C2CCCC2)CCCC1 C1(N(C(C(CN(CC)CC)F)=O)CC2CC2)CCN(C(=O)C(C)C(F)F)CC1 C(=O)(C(F)CCC(C)C)N1CCCC(C(C(=O)Nc2c(C)nn(C)c2)C)C1 C1(c2ccc(CN=c3c(C)cnn[nH]3)cc2)CC(C2CCC2)=NO1 c1(OC)ccc(C(=O)NCCNC(C2CCN(C)C(=O)C2)=O)c(Cl)c1 c1(C(=O)NC2CC(F)(CNC(C3CCS3(=O)=O)=O)C2)c[nH]c2cc(F)ccc12 N1(C(C(CCC)O)=O)CC(C2CCCCN(C(C3CCC(=O)N3CC)=O)C2)C1 C(CN=c1[nH]c(=NCc2ccc(CO)c(F)c2)[nH]c2c1COCC2)(C1CC1)OC C1(NC(C(C)NC(c2ccco2)=O)=O)CCC(NC(=O)C(C)(F)F)C1 c1(C(N2CC(NC(C3(C=C)CCC3)=O)C(OC)C2)=O)c(Cl)nc2cc(Cl)ccn12 N1(C(=O)CC2C=CCC2)CC2CCN(C(c3c[nH]cc(F)c3=O)=O)C2C1 N1(C(=O)NC2CCN(C3CCN(C)C(=O)C3)CC2)CCOCC12COCCN(C)C2 CC(C)CC(C)C(=O)N1CCCC(C)(CNC(c2cc(C(C)C)cc(O)c2)=O)C1 CCC(CC(=O)N1CCC2C(NC(c3cccc(OC)n3)=O)C12)SC C1(C)(CNC(C2CC(NC(C3C(COC)CC3)=O)C2)=O)CCCO1 C1(C(=O)NCC2CN(C(=O)C3=COCC3)CC2(F)F)(OC)CCCCCC1 c1(C(=O)NCc2ccc(CNC(C(C)CN(C)C)=O)cc2)sccc1S(C)(=O)=O c1(C(N2CCN(C(C(CCC)NC(C)=O)=O)C(CO)C2)=O)cnn2ccn(C)c12 Cc1cnc(N(CC(C)NC(=O)CC2C(C)(C)C2(C)C)C)nc1S(C)(=O)=O C(=O)(C(C)(C)C(C)O)N1CC(OC)C(NC(=O)Cc2ncccc2C)C1 c1(CNC(C(Cn2ccnn2)NC(C2CC(CCC)C2)=O)=O)ccncc1C C1(NC(=O)NC2C(CCC(=O)OC)CCC2)CC(=O)N(c2ccccc2OC)C1 CC1CNc2c(C(=O)NCCc3nc(-c4ccccc4)ns3)cnn2C1 N1(C(CC=CCC)=O)CC2(CCCC2NC(c2ncn(C)c2C)=O)C1 n1(CCOC)cc(C(=O)NC2CCC2NC(c2ncc(C(F)F)s2)=O)cn1 N1(CCNC(c2c(CC)scn2)=O)CCCN(C(=O)CCC2CCOC2)CC1 N1(C(C2C3CCN2CC3)=O)CCCC(C(C)NC(c2nc(COCC)sc2)=O)C1 c1(C(=O)NCc2c(F)cc(C)c(F)c2)c(F)cncc1C1=CCN(C)CC1 C1(CC(=O)N(C(CN(C(c2ncn(CC)c2)=O)C)C)C)CC(C)(C)CCO1 C=C=C(C)CC(=O)N1CCC(C2CCCN2)C1.C12CSCN1C1CN(C1)C2=O N1(C(C(COCC)C)=O)CC(NC(c2cc(C)sc2C)=O)C(O)C1 N1(C(CCCCC#N)=O)CCC2(CC1)CC2(CO)CNC(C1CCCC(O)C1)=O CCC(CCC(=O)N1CCN(C(=O)CCN(C2CC2)CC)C(CO)C1)OC C1(NC(C2(C)CC2)=O)CCC2(CCN(C(=O)CCc3ncc[nH]3)CC2)C1 c1(C(N2CC(CC(=O)NC(C(=O)NC(C)C)C)OCC2)=O)ncc(F)cc1F C(=O)(CC1=CCCCC1)N1C(c2nnc(C3(C)C(C)CCCC3)o2)CC(F)(F)C1 C1(C(=O)NC(CCC)C(F)(F)F)C(C2CC2)CCN1C(=O)CN1CCNC(=O)C1 C1(N(C)C)(CNC(=O)NCC(c2nccs2)OCC)CCc2ccccc2O1 c1(C(=O)NCCOCCNC(C(C(=O)OC)C)=O)c(OC(C)C)ccnc1F c1(NCc2ccc(CC)cc2)cccc(S(=O)(=O)N(C)C)c1.C(C)(=O)O N1(C(C(Cc2ccccc2)OC)=O)CCCC(CNC(c2cc(CF)on2)=O)C1 C1(CN(C(C(C(=O)OC)SC)=O)C)CN(C(=O)C=C(C)C(C)C)CC12CC2 C12(C(=O)OC)CC(C(=O)NCC3CN(C(=O)C(c4cnccn4)C)C3)(C1)C2 N1(C(=O)OC)CCC(C(C)C(N2CCN(C(C3CCC3)=O)CC2)=O)CC1.C1CN1 C(=O)(C(O)CC(C)(C)C)N1CC(c2c(CNC(CCCCCOC)=O)nco2)C1 Cc1cc(C(=O)NC(C2CN(C(c3cc(C)[nH]c3C)=O)C2)C)n(C)n1 CCC(C(=O)NCC(F)CNC(=O)C=CSC)OC1CCCC1 CCCC(CN(C(=O)COC(=O)CC(C(C)C)c1nc[nH]n1)C(=O)CO)CCO N1(C(C2C(C)C2)=O)CC(C2CC2)(C(=O)NCC2CC(C#N)C2)C1 C1(NC(CSC)=O)CCC2(CCCN2C(=O)C(C(C)C)c2ccc(Cl)cc2)CC1 CC(COCc1ccco1)N=c1ccnc(NC2CCCC(C)(C)C2)[nH]1 C#Cc1cccc(OCC(=O)NCC=CCNC(=O)C(N2CCCCCC2)C)c1 CCC(C(=O)N1CCC(C(C)(C)NC(=O)Cc2sc(C3CC3)nc2C)C1)C(C)C C1(NC(=O)CCSC(F)(F)F)COCCN(C(=O)CC2CC3CC3C2)C1 N1(C(C(c2ccc(F)cc2)C)=O)CCC(C)C(NC(=O)Cc2ccc(F)cn2)C1 C=CC(C)CCNC(c1occc1CNC(=O)C(c1cnn(C)c1)O)=O N1(C(CN2CC(C)(C)C2)=O)CC2(CCC(CNC(C3CC=CCO3)=O)O2)C1 c1(N2C(c3ccccc3)C3CC3C2)ccc2nncn2n1 N1(C(CC(C=C)C)=O)C2CCC1(CNC(=O)C(C)CCCOC)CC2 c1(C(COC(=O)C(O)CN2CCCC2)NC(C2CSC2)=O)cc(F)ccc1Cl C1(NC(c2c(C)nn[nH]2)=O)CC(NC(=O)CSCCC(F)(F)F)C1(C)C CN=c1ccc(C(N2CCCC2C(C)NC(=O)C(=O)NOC)=O)c[nH]1 C12(NC(C=NOC)=O)CCC(CNC(C3CC3COC)=O)(CC1)OC2 c1(OC(C(=O)NCC(CC)NC(=O)CSC)(F)F)cc(Cl)cc(Cl)c1 c1(C(N(CCCCN(C(C2N(CC)CC2)=O)C)C)=O)ccc(S(=O)CC#N)cc1 C(=O)(C1=NNC(=O)CC1)NCC1(CNC(c2cccc(NC)n2)=O)CC12CCC2 c1(CN(C(C(CC)C)=O)C)cccc(CNC(C2(c3cc[nH]n3)CC2)=O)c1 CC(C)C1C(=O)N1.c1(C(COCCNC(=O)OC(C)(C)C)O)ccccc1.C=O c1(CSC2CCC(CC)CC2)cc(C#N)c2c(n1)CCCC2 C=CC1CCCN(C(c2cnccc2Br)=O)C1.c1(C(=O)OCC)cc[nH]c1 N1(C(C2(CNC(C3CCC(CC)O3)=O)CCC2)=O)CC2(CCCC2)C1 n1(CCC(=O)OC)cc(CC2(O)CN(C(C3(CCS(N)(=O)=O)CCC3)=O)C2)nn1 N1(C(C2CCC(C)(CC)O2)=O)CC(C)N(C(=O)Cc2cnn(C)c2C)C(C)C1 n1(CC)nc(C(=O)Nc2ccc(N3CCCC3)c(Br)c2)c2c1CCOC2 C(=O)(CC(C)(C)C#N)NC(C)C=CC(=O)NCc1ncccn1 c1(CC)cc(Cl)ccc1C(=O)NCc1ccnc(C(=O)O)c1 C(=O)(CS(C)(=O)=O)NC(C(=O)N1CC(CC(=O)OC)C1)COC C1(C(=O)NCCC2(CNC(C(CC)(C)C)=O)CC2)Cc2cccnc2C1 Cc1nc2c(s1)CCCC2C(=O)NCC1CN(C(C2(CO)COC2)=O)CCCO1 CCCC(C)C(CC)(c1nnnn1C1CCCCC1)NC1CCC(C)CC1 C1(C)(CNC(c2cn(CCC)nn2)=O)CCN(C(=O)CC(=O)N(C)C)CC1 c1(COCCNC(C(c2ccc(Cl)s2)N(CCC(C)C)C2CC2)=O)ccccc1 C1(C)(C)CC(=O)OCc2cn1nn2.C1(NC(=O)OC(C)(C)C)CC(CCO)C1 C1(CC)CCN(C(=O)CSCCF)C1NC(=O)COC C1(NC(c2c(C)cccn2)=O)CN(C(C2Cc3nnc(C)n3C2)=O)CC(F)(F)C1 C1(CC)CC(O)CN1C(C1CC1C(C)NC(=O)Cn1[nH]cnc1=N)=O C(=O)(C1=CCN(C)C1)NCCC(C)NC(c1cnc(CC)o1)=O CC1=C(C(=O)N2CCCC(NC(=O)C=C3CCN(C)CC3)C(F)C2)CCCO1 CC1CN(C(c2nncn2C2CC2)=O)CC1CNC(=O)C(F)=CC1CC1 C1(N(C(C(C)Nc2ccccc2F)=O)C)CCCN(C(=O)C2=COCCO2)CC1 N1(C(C(COCC)NC(=O)CC(O)C2CCCC2)=O)CCC2C(=O)NCC2C1 N(C1CCCc2c(Cl)ccc(Cl)c21)C(N1CCC2CNC1C2)=O N1(C(C2C3CN(C)CC32)=O)CCC(NC(=O)Cc2cnc[nH]2)C(F)C1 N12CCN(CC1)C2=O.c1(C(C)NC2CNCC2F)ncccn1 C1(C(C(=O)OC2C(C(=O)NC)C2)OC(C)(C)C)CCCCC1 C=CCC(CC(C)C)C(=O)N1CCCC(CC)(NC(=O)C(O)CC2CCCC2)C1 n1(C(CC)CC)nc(C)cc1C(N1CCCC1CNC(=O)CN1CCCC1C)=O c1(N2Cc3c(-c4c(OC)c(C)ccc4)n[nH]c3CC2)nc(C)nc2cccc(Br)c12 c1(CC(N2C(CCNC(CCC3C(C)C3)=O)CCC2)=O)ccc2c(c1)CCCC2 c1(C(CNC(c2n[nH]cc2Br)=O)NC(CC=C=C)=O)ccccc1F N1(C(C2CC(=O)NC2)=O)CCCC2(C1)CN(C(c1cc(Cl)nc(Cl)c1)=O)CCO2 C(=O)(C1CC=Cc2ccccc21)N1CCCC(F)(CNC(=O)Cc2cnns2)C1 c1(C(=O)NCC2(CC(=O)NC3(c4nccs4)CC3)CC2)cccn2ccnc12 c1(CC)oc(C(=O)O)cc1S(=O)(=O)NC(C)C(=O)Nc1ccc(F)cc1 C1(CC(CNC(C2(C(=O)OCC)CNC2)=O)O)(C(F)(F)F)CCCCC1 C1(C(N2CCN(CCN(C)C(c3c[nH]c(=N)s3)=O)CC2)=O)(OC)CC2CCC1C2 CC(CC(=O)NC1(CF)CCN(C(=O)CN2CCCCC2=O)C1)C(F)(F)F c1(CC)ccsc1C(=O)NC(C)CN(C(=O)CCc1ncc[nH]1)CC C1(C(C)NC(C2C(C)C2C)=O)CN(C(c2sccc2Cl)=O)CCO1 c1(CCCN2C(C)(C(=O)O)CCC2)ccc(F)c(F)c1 CC(O)CC(C)N=c1ccnc(NCCC23CCCN2CCC3)[nH]1 N1(C(C2OCCN(C(c3cc(OC)c(Cl)nc3)=O)C2)=O)Cc2ccc(F)cc2C1 N1(C(C(C2CC2)OCC)=O)CCOC2(C1)CN(C(C1CC1C(C)(F)F)=O)C2.C1(C)CC1 N1(C(c2c(CC)ccs2)=O)CCCC(NC(C23CC(C2)C(C)(C)O3)=O)CC1 C12(C(N3CCC(O)(CC)C3)=O)CCC(CC1)N(C(C1(NC(N)=O)CC1)=O)C2 O=C(CC1NC(=O)c2ccccc21)NCC1(NC(C2CCC3C2C3(F)F)=O)CC1 C1(C(=O)NCCC(=O)NC)CCN(C(C2CC(C(C)C)C2)=O)CC1 C#CCC(CC(F)(F)F)C(=O)NCC1COC(C(F)(F)F)CN1 CC1(C)CC(CNC(c2cnccn2)=O)CN(C(=O)CCCS(N)(=O)=O)C1 Cc1cc(C(=O)NC2CC2NC(c2ccn(C)c2C)=O)cc(S(N)(=O)=O)c1C c1(C(NCP(C)(C)=O)C)cc(OCNC2CC2)n(C)n1 CCN=c1[nH]c(C)c(C(N2CCCC2C(C)NC(C2CCCCC2(C)C)=O)=O)s1 N1(C(C2N(CC)CCCC2)=O)CCc2c(CNC(=O)C3=CCC3)cccc2C1 c1(OC)ccc(C(C)C(=O)NC(CNC(c2cn(C)cn2)=O)CO)cc1OC Cc1ccc2c(cnn2C)c1-c1csc(NC(C2CC23CCOC3)=O)n1 c1(CN(C(c2ccc(F)cc2)C(=O)NC2CC(F)(F)C2)C)cc(O)cc(Br)c1 CC(C)CC(=O)NCC(CC1CCNCC1)CO C1(c2n(CC(F)F)ncc2)NC(=S)N(C2CC2)C2=C1C(=O)NC2c1ccccc1 Cc1cccnc1C=CC(N1CC(n2ccnn2)C(C)C1)=O C(=O)(C(C(C)NC(c1cc(C)ccc1C)=O)C(C)C)NCCN1CCC=C(C)C1 c1(CC(=O)N(C2C3CN(C(CC4CN(C)C4)=O)CC32)C)c[nH]c2cc(F)ccc12 c1(C(=O)NCC2N(C(C=CC=CC)=O)CCCCC2)cc2cccnc2o1 N1(C(C(N)=O)=O)CC=CC(NC(C2(O)CCC2)=O)C1 c1(-c2cc(OC)cc(COC)c2)ccc2nnc(C(N3CCOCC3C)=O)n2c1 c1(C(=O)NCC(C)(CO)NC(C2C(C)CC2)=O)cc(C(C)(C)C)n(C)n1 C(CO)(CCCCNC(=O)C(F)=C1CCCC1)NC(=O)CCC1CCC(O)CC1 C(CC(C)C)(C(=O)N(CC(O)CO)C)N(C(C(C)=CC(F)(F)F)=O)C c1(C(CNC(CS)=O)NC(c2cnn(C)c2)=O)ccc(C)cc1.C1(CSC)CC1 CC(C)CC(O)C(=O)NCC(C1CCC1)NC(=O)CC1(O)CCCN(C)C1 C1(C(=O)NC23CC(NC(c4cnc(C)s4)=O)(C2)C3)CCCN2CCCCC12 C(=O)(C(O)C1=CCCCC1)NCC(CNC(c1ccn(CC(C)C)n1)=O)CO C(=O)(CC(C(F)(F)F)NC(=O)C(C1CCCCC1)F)NC1(CC=C)CCCCC1 c1(OC)cccc(F)c1CNC(=O)CC1CN(Cc2ncccc2OC)C1 c1(C(=O)NCC2CC(OC)CN2C(C2OCCC2C(C)C)=O)cc2occc2[nH]1 C1(CC(=O)NCC(CC)(C)C)CN(C(=O)C(C(C)C)C2CCC2)C(C)(C)C1 c1(C(=O)NCC(CC=C)NC(c2c(Cl)cnn2C)=O)ccccc1CC C(=O)(C#CC(C)(C)CNC(c1cnc(N)cn1)=O)NCC(C(=O)OC)OC C1(NC(c2cccc(F)c2O)=O)CCC2CCN(C(=O)C(F)(F)CO)C1C2 C(=O)(CC(C)(C)CCC)NC(C1(O)CCN(C(C2(CC=C)CCOC2)=O)CC1)C CC(C)CC(O)C(C)C(=O)N1CC2(CCC2NC(=O)Cc2cc(Cl)ccc2Cl)C1 N1(C(c2c(CC)c[nH]n2)=O)CC(CNC(=O)C(C#N)C(C)(C)C)C2(CCC2)C1 C1(C)(CC(=O)NCCC=CCCC)CCN1C(c1cnc(C)o1)=O C1(OC(C2CCC2(F)F)=O)CC(=O)N(CCOC(=O)C2CC2)C1 N1(C(CCC2N(C(c3c(C)cc[nH]3)=O)CCCC2)=O)CCOCC(O)C1 C1(NC(CN(C)C)=O)CN(C(=O)CCC2CCOC2)CC1Cc1ccccc1 Cc1cc(CN=c2[nH]cc(CCNC(c3nccs3)=O)s2)cc(Br)c1 CC1(C)CC(NC(c2c(F)cccc2Cl)=O)CN(C(=O)C(C)(O)C2CCC2)C1 Cc1cc(-c2ccc(O)c(Cl)c2)c(O)c(C=O)c1 N1(C(C(N2C(CC)Cc3ccccc3C2)=O)=O)Cc2cc(F)ccc2CC1C c1(N(C)C)nc(Cl)c(C(N2CCOCC2CNC(=O)CCc2cnc(O)[nH]2)=O)s1 C=CCC(C)(C)CC(=O)NCC(C)CN(C)C(C12COC(CO)(C1)C2)=O N1(C(C(=O)NCC)=O)CCCC(CCNC(=O)CN(c2ccncc2)C)C1 N1(C(CC(CC(C)C)CN)=O)CCC(OCCO)S(=O)(=O)CC1 CC1CC(C(=O)NC2CCC(NC(c3cc(O)nn3C)=O)C2)CCN1C C1(CCNC(CSCC(C)C)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1(F)F c1(N(C(C)C)C)ccccc1C(N1CCC(N(C)Cc2scnc2Cl)C1)=O C1(C(=O)OC)(SC)CN(C(C2CN(C(C)=O)C2)=O)C1.C1(Cc2cc[nH]n2)C(=O)N1 CC1(C)C=C(C(=O)NC2CCN(C(=O)CCCCCc3cccs3)C23CC3)C1 C=CC1CCCN(C(=O)C(CC(N)=O)NC(=O)C(CC)=CC)C1 C12(C(=O)NCC(=C)CCNC(C3(CO)CCCCC3)=O)CCCN1CC(OC)C2 C1(CC)CN(C(c2cnc(Cl)c(C)c2)=O)CCN1C(c1cc(I)ccc1C)=O C1(C(=O)O)COCCN1C(C12CC1CN(C(=O)CCc1ncccc1F)C2)=O C1(CC)CCC(C(=O)N(C)CC2COCCN2C(C2CCOC2)=O)CC1 c1(C(N2C(C)(CNC(=O)CN3CCOCC3)CCC2)=O)cc2ccccc2s1 c1(CC(=O)NC2(CNC(c3c(CC)onc3)=O)CC2)cn2cc(F)ccc2n1 CCCCC(O)C(C)C(=O)NC1CC(CC(N2CCC2(C)C(=O)NC)=O)C1 c1(C(N2C(CNC(C(C)NC(=O)CC(C)(C)C)=O)CC2)=O)cnn2c1OCC2 C(c1c(Cl)cccc1Cl)=C(C)C(=O)N(CCCNC(=O)CCc1cn(C)nn1)C C1(C(=O)NCC2C(NC(c3cccc4c3COC4)=O)C2)CCc2ccccc2C1 c1(-c2cncc(OC)c2)ccc(F)c(COCc2n[nH]cc2C(F)(F)F)c1 c1(CNc2ccc(C(C(F)F)F)cn2)cccc2ncnn12 N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(=O)C=CCN2CCOCC2)C(C)(C)C1 N1(C(C2C(C(=O)OC)CC2)=O)C(C(N2CCC(O)(COC)C2)=O)CCC12CC2 c1(NC(CC(c2cn(C)nc2)NC(=O)C=CC(F)(F)F)=O)cccc(C#N)c1 c1(-n2cc(C(C)NC(c3c(C)nc(Br)s3)=O)nn2)cccc2ncccc12 c1(C(N(CCCN(C(CC2C(C)C2)=O)C)C)=O)cn2c(n1)COCC2 N1(C(C2CN(C(C)=O)C2)=O)CCOCC(C(=O)Nc2ccc(C)c(O)c2)C1 C1(C)(C(N2C(CNC(C(C)=NOCC#N)=O)CCCC2)=O)CCN(C)C1=O c1(CNC(C2(CNC(C(C)OC)=O)CC2)=O)ncn(C(C)C)n1 c1(C(=O)NC2C3CC(CNC(CC(=C)C)=O)(C3)OC2)ccc2c(c1)CC(C)O2 C1(CNC(C(CC(=O)OC)C)=O)CC2CCC1N(C(=O)CC1COCC(C)O1)C2 Cc1[nH]c2ccccc2c1C(=O)NCC(CNC(C1CCS(=O)(=O)C1)=O)CO C1(CNC(CSCC=C)=O)CN(C(=O)COCC2CCCCO2)CC2(CCC2)O1 c1(C(=O)NC2C(NC(C3CC(C)C3)=O)CCCC2)cc(C2CC2)nc2ccnn12 C1(C(N(CCCNC(c2ccc(C)cn2)=O)CCO)=O)CCOC(C)(C)C1 c1(C(=O)NCC(=CCCC)C)c(CCCC)nn2c1CCC2 c1(C(N2CCCC(C(C)(O)CNC(=O)C(N)=O)C2)=O)cc2ccc(F)cc2o1 C1(NC(C(C=C=C)C)=O)CN(C(c2cccnc2SC(F)F)=O)CC12CC2 c1(CCC(=O)NCCCN(C2CCCC2)C(C2(CSC)CCC2)=O)ccc(F)cc1 C1(CNC(C(F)=CCC)=O)CC(C)N(C(c2cncnc2C)=O)C1 C1(NC(=O)CC2CCC3CC23)CC2(C1)CN(C(=O)C=Cc1cncc(O)c1)C2 CN1CCC(CC(N2CCC(CNC(=O)CN3CC(C)(C)C3)C2)=O)C1 c1(C(=O)NCCOCCNC(C(CC)(C)CO)=O)n[nH]c2ccc(C)cc12 N1(C(C(C(C)C)F)=O)CCC2(CCCC2CNC(=O)C=C2CCCC2)CC1 C(=O)(CC(O)C(C)(C)C)N1CCC(COC)(NC(C2OCCN(C)C2=O)=O)C1 Cn1c(O)nc2c(S(=O)(=O)NC3CCCCC3C)cccc12 Cc1nnc(NC2CCCCN(C(=O)C(C)CC3CCC3)C2)c(C#N)c1C c1(C(C(=O)NCCSC)N(CC#CC)C)ccc(F)c2c1CCC2 C1(C(=O)NC(C)CCCNC(=O)COCC(C)(C)C)CC2(C1)NC(=O)NC2=O CCCCCCC(F)C(=O)NC1CC(CCNC(=O)Cc2nonc2C)C1 C(c1c(F)cccc1F)=CC(N1C2C(N(C)C(c3ccoc3)=O)CC(C2)C1)=O C1(CC(=O)NC(CCC)CO)CCCN(C(=O)CN2CCNC2=O)C1 O=C(CNC1CC12CCCCC2)NNC(=O)N1CCC(c2ccccc2)CC1 O=C(CCC(F)(F)F)NC(C1(O)CCCCC1)C(=O)NC1CCCSC1 Cc1cc(Br)cc(CN2CCC(N(C)C(c3cnc(O)cc3O)=O)C2)c1O C1(NC(=O)Nc2c(C)n(CCN(C)C)nc2)CC(C(=O)OC(C)(C)C)C12CCC2 C1(C(=O)NC2(CC=C)CN(C(=O)Cc3n[nH]c(=NC)s3)C2)CCN(C)C(=O)C1 C1(C(=O)NCC(CC)N2CCCC2)CCCCCN1C(=O)C(CC1CC1)OCOC c1(C(=O)NCCOC2CCN(C(CCC3C(C)C3)=O)C2)ccc(C)cn1.C(CF)O N1(C(C2C(C)OCC2)=O)CC2(C1)C(NC(=O)Cc1cccc(F)c1)CCS2(=O)=O N#CC1(C(=O)NC(c2ccc(C#N)cc2)CC2CCCCC2)CCCCCC1 C1(CC=C)(NC(C2CC2(C)C(C)C)=O)CCN(C(=O)CSc2nncn2C)C1 c1(CC)nn(C)cc1CNC(c1ccccc1)CCc1c(C)noc1C C=CC1(C(=O)NC23CC4CC(CC2C4)C3)CCN(C(=O)C#CC2CC2)CC1 c1(-c2nnc(N3C(C)COCC3)n2CC2CCOC2)nnc2n1CCNC2=O c1(C(=O)NC2CCN(C(C3(C)CC=CC3)=O)C2)ccc(-c2cc(O)ns2)cc1 c1(CC(N2CCC(N(C)C(C3CCN3S(C)(=O)=O)=O)C2)=O)cc(F)cc(Cl)c1 c1(C(N2C(CNC(C(CC)(C)OC)=O)CCCC2)=O)cc(C)c(C)cc1Cl c1(C(=O)NC2CC(C)N(C(=O)CCc3ccn(C)c3)CC2)cnn2ncccc12 C1(CNC(C(N2C(C(N)=O)CC(OCC)C2)=O)=O)CCC2(CCOCC2)CN1 Cc1ccc(C(=O)NC(C)CN(C(=O)CCC(=O)c2cccnc2)C)cc1CO C1(C(N2CCC(Nc3ncnc(O)c3Br)C2)=O)CC2(C1)CS(=O)(=O)C2 Cc1scc(C(N2CCC(CF)(NC(c3cccc(C(C)C)c3)=O)C2)=O)c1C C12(NC(COCC(C)C)=O)CC(CNC(=O)COCC(c3ccccc3)C)(C1)C2 C(=O)(CCCN(C)N=O)NCCCN(C(=O)Cc1cnn(C)c1)CCC N1(C(CCSC2(C)CCC2)=O)CC(NC(=O)Cn2ccnn2)CC12CCOCC2 Cc1ccc(CC(=O)NCC(C2CCN(C(=O)CSc3nncs3)CC2)F)cn1 C1(C(N(CC(C)C)CC)=O)CCN(C(=O)CCOCCN(C)C)C1C Cc1ccc(C=CC(=O)NC2CCCC2NC(c2cc(Br)no2)=O)cc1C c1(C(=O)NC2CCCC(CNC(C3(Br)CC3)=O)C2)coc2c1COC2 C1(CNC(C(C)SC)=O)N(C(c2cccc3oncc23)=O)CCCC1(C)C c1(N(CCN)CC)ccc(S(=O)(=O)N(C)C)cc1.C1(C(C(CC)=O)=O)CC(CSC)C1 N1(C(c2c(C)cncc2)=O)CCC2CCC(C1)N2C(=O)CN1CC2CC2C1 CCCC(F)(F)C(=O)NCC(O)CN(C)C.c12cc(on1)C(=O)N2 c1(CNC(C(c2ccccc2)OC(C)C)=O)nc(C2CC2)sc1Br c1(CN(C(Cn2ccc(C)n2)C=O)C(C)(C)C)ccc2c(c1)OCCO2 c1(C(N2CC(NC(C3CCCO3)=O)CC(C)(C)C2)=O)ccc2c(O)n[nH]c2c1 C1(=CCNC(C(C)OCCC=C)=O)CN(C(c2cnc[nH]2)C2CC2)CCS1(=O)=O C=CCC(C)(C)CC(=O)NC1CCN(C(c2ccc(CC3CC3)cc2)=O)CC1F Cc1ccc(C(=O)NCC2CCC2c2ccccc2)nc1C1CC1 c1(OC)ccc(C(=O)NC2CC2CNC(=O)CN2CCC(C)C2)cc1O c1(C(N2C(CNC(c3c(C)cn(C)n3)=O)CC3(CC3)C2)=O)ccc2cccnn12 c1(C(N2CC3C(CC(=O)OC)(CC3)C2)=O)cc(Cl)nc(Br)c1N CCC(CC)(CN=c1nc(C(C)C)[nH]s1)NC(=O)C(C)Oc1ccccc1 C1(NC(c2c(C)nc(CC)o2)=O)CN(C(c2ccc(C)cc2O)=O)C2(CCC2)C1 c1(C(=O)NCCN2CCCC(CO)C2)cc2ccccc2c(I)c1O Cc1cc(C(N2CCN(C(c3c(C)cnn3C)=O)CC2C)=O)c(O)c(C)c1 C(=O)(C1=CC2(CN(C(C3CCC(F)C3)=O)C2)OC1)NCCc1n(C)cnc1 C(=O)(CC(C)CC(C)C)NCCC1N(C(CCCc2nnc(C)n2C)=O)CCC1 C(C(CCC)C(=O)OC)c1c(NC(C(=C)C(=O)OCC)=O)cccc1 N1(C(c2c(OC)ccc(OC)c2)=O)CC(C)CN(C(=O)CSCCSC)CC1C c1(CC(=O)NC2(C)CC(NC(c3cnc(Cl)c(N)c3)=O)C2)ccc([N+](=O)[O-])cc1 C1(NC(c2c(N)non2)=O)CC2CCC(C1)N2C(C12CC(C(F)F)(C1)C2)=O N1(C(c2c(C)sc(O)n2)=O)CCCN(C(c2cc(N)cc(O)c2)=O)CC1 N1(C(C(C)CCN(C)C)=O)CCOCC1C1CCCO1 N1(C(C=CCC)=O)CCC(C(=O)OC)C1CCSC.C1(CCOC)(NC)CCC1 c1(C(=O)NCCN(C(C2CC2(c2ccccc2)F)=O)CC)cc(C(C)C)nn1C CC1=C(C(=O)NC2CCN(C(=O)Cc3ccc(F)cn3)C(C)C2)CCS1(=O)=O C1(S(C)(=O)=O)(C(=O)NC2CC3CN(C(Cc4n(C)ncc4)=O)CC3C2)CCCC1 c1(NC(C2C3(CN(C(Cc4ccc(C)nc4)=O)C3)C2)=O)c(F)cc(Br)cc1Br C(=O)(C1CCc2nnc(C)n21)N1C(CC)CN(C(C2(CN(C)C)CC2)=O)CC1 c1(NC(C)C)cncc(C(=O)NCC2(C)CCN(C(c3cc(CF)on3)=O)C2)c1 c1(C(=O)NCCCCCNC(COC(CC)C)=O)cncc(C(C)=O)c1 O=C(CC(C(F)(F)F)N1CCOCC1)OCC(c1cc2ncccc2[nH]1)=O c1(SC)ccccc1Cl.C12CCN(C1)C(=O)C(Cc1ccsc1)N(C)CC(=O)N2 C12(C(N3CC(C)(NC(C4(C(=O)OC(C)(C)C)CC4)=O)C3)=O)CC=CCN1CCC2 CC1(C)CCCC(C(=O)NC2CC(C(N3CC(F)(F)CC3C(N)=O)=O)C2)C1 C1(NC(C2CC(OC)C2)=O)CN(C(=O)CC(C)c2ccccc2)CC12CC2 Cc1cc(C(N2CCC(C(C)NC(=O)COCC3CC3)C2)=O)ccc1O C(=O)(C(O)C(C)(C)CC)NC(CN1CCN(C(C(CC=C)(F)F)=O)CC1)C N1(C(C)C)CCc2c(NC(=O)CC(F)(F)c3ccccc3)cccc2C1 c1(C(=O)NCC(C)NC(c2[nH]cc(C)c2)=O)cccc(C#N)c1Br C1(C(C)NC(C(COC)O)=O)CN(C(=O)Cn2cnnc2O)CCO1 c1(C(N2CC(COC)(CNC(=O)C(CO)N(C)C)C2)=O)cc2n(n1)CCCO2 CC1(C(=O)NCC2(CNC(c3cc(Cl)cs3)=O)CC(F)(F)C2)COC(=O)C1 CCC(CC(=O)NC(c1n[nH]c(C)n1)C(=O)NC1CC(O)C1OC)OC C=CC1OCCCC1C(=O)N(CCCN(C)C(C1CN(C)C(=O)N1)=O)C Cc1sc(C(=O)NCC2COCC2NC(c2cc(O)n(C)n2)=O)nc1O N#Cc1cccc(CNC(=O)NCC2CC2C2CCOCC2)c1Br CCCC(O)CCN=c1ccnc(NC(c2nccn2CC)C)[nH]1 N1(C(C(CN(C(c2c(CC)cncc2)=O)C2CC2)C)=O)CCC2(CC1)CC2 Cc1cc(=O)n(C)nc1C(N1CC(Oc2ccc(Cl)c(F)c2)C1)=O C12(C(=O)NCCOC(C)=O)CC(C)(CN1C(=O)CCCC1CC1)C2 C1(NC(CCc2cc(C)[nH]n2)=O)CN(C(C2CC3CCC2CC3)=O)CC12CCC2 c1(C(C)C)cc(C(N2CCN(C(=O)C(F)C(C)(C)O)CC2C)=O)cc(F)c1 O(NC(=O)C(Cc1ccco1)NC(c1[nH]ccc1COC)=O)CC(CC)C C1(C(N2C(CNC(=O)C=Cc3cc[nH]n3)CC(F)(F)C2)=O)CCc2nn[nH]c2C1 CCCC(CNC(c1ccnc(C)n1)=O)C(=O)N(C)CC1(OCC)CCC1 Nc1cc(C(=O)NC2CCCC(NC(c3cc(F)c[nH]3)=O)C2)cc(F)c1 C(=O)(C1CCCc2sccc21)NC(C(C)NC(C(C)C)=O)CO C=C(C)CCC(=O)N1CCN(CC2CCCN(C(C3CC3C(C)C)=O)C2)CC1 N1(C(CN(C(C(COC)OC)=O)CC2CC2)=O)CC2(CCC(=O)O2)C1 CC(C)P(=O)(CC(=O)NCCC1CN(C(=O)CC2CCCC2(F)F)C1)C(C)C N1(C(C(=Cc2ccc(F)cc2)C)=O)CCC2(C1)CN(C(=O)Cn1nnc(=O)[nH]1)C2 N1(C(C(C)n2cnnn2)=O)CCC(C(C)NC(=O)C(c2cccc(O)c2)C)CC1 c1(NC(C2CCN(C(C(COC)OC)=O)C2(C)C)=O)cccc2cccnc12 C=C1CON(C(=O)C(c2c(C)cccc2Br)NC(c2cc(C(C)=O)cs2)=O)C1 C1(C(C(=O)NC(C2(NC(C3CCCC3C)=O)CC2)C)=O)CCCCC1 C1(NC(CC)=O)(CC)CCCN(C(c2cnn(C3CCC3)n2)=O)C1.C1C(=O)N1 C12CN(CCC1(F)F)C2=O.c1(NC(C(CC)(C)O)=O)cc(C)c(OC)cc1Br c1(C(N2CC(C(N)=O)(CNC(c3cnsn3)=O)C2)=O)ccc2c(c1)C(=O)NC2 N1(C(C(CSC)C)=O)CCCC2(C1)CN(C(C1(C#N)CCCOC1)=O)C2 CC(C)C(C#N)C(=O)NCCOCCN(C)C(C1CNC(=O)N1)=O c1(OC)ccc(CC(=O)NCC2CCN2C(=O)CC2CCOC2(C)C)cc1 Cc1ncc(C(=O)NC2(CCCCNC(c3ccc(=O)n(C)n3)=O)CC2)c(=N)[nH]1 N1(CC(N2C(C(C)NC(CN(C(=O)OC)C)=O)CCC2)=O)CCN(C)CC1 Cc1cc(O)c(Cl)cc1CN1CCC(O)(C(=O)NC(CC(=O)O)C(C)C)CC1 CCC(C)(C(=O)Nc1ccc(NC(C2CC3(CCCC3)CO2)=O)c(C)c1)C(F)F c1(C(N2CC(O)(C(C)NC(C(C)C3CCCC3)=O)C2)=O)ccc([N+](=O)[O-])cn1 C1(CNC(c2scnc2C2CC2)=O)CC2CCCC(C1)N2C(=O)Cc1cnsc1 c1(OC)cc(C(N2CC(CN(C(=O)C3=C(C)OCC3)C)C2)=O)c(C)cc1O C12(C(=O)NCCCCN(C(=O)CCc3ncc[nH]3)C)CSCC1C2(F)F CCCCCC(O)C(=O)N1CCCC1C(N1CCCC(C)(CC)C1)=O Cc1cn2ccnc(C(=O)NCCC(C)N(C(=O)CN3CCC3C)C)c2n1 C(CC(=O)NCC1COCCOC12CCC2)(C(C)(C)C)NC(=O)OC(C)(C)C N1(C(=O)CN2CCCCC2c2cccnc2O)Cc2ccccc2CC1CO c1(C(N2CC(CNC(C(CCC)OCC)=O)C(C)C2)=O)cc(Cl)c(Cl)cc1N N1(C(c2c(C)cccn2)=O)CCC(NC(c2cccs2)=O)C(C(C)C)C1 C(=O)(CC(C(F)(F)F)NC(C12CC(CO)(C1)C2)=O)N(C1CCOC1=O)C C1(NC(c2c(F)ncc(OC)c2)=O)CCCC12CN(C(=O)CCCSC)C2 c1(C(=O)NC(C2CCOC2)CNC(C(C)(C)C)=O)cc2c(Cl)ccnc2s1 O=C(O)CC(CC1CC1)NC(C12CC(c3ccc(C(F)(F)F)cc3)(C1)C2F)=O C1(C(=O)NC2(CC)CCOC2)C2CC3C(C2NC(=O)COCC2CC2)C13 c1(OC)cc(NC(C2CCC3(CCC3)C2)=O)c(C)cc1C c1(CCNC2N(c3ccnc(N(C)C)n3)CCC2)ccc(C#N)cc1 N1(C(N)=O)CCCC1C(=O)NC1CC(CNC(=O)C(c2ccccc2)O)C1 C1(C(N(C2(CCC(NOCCCOC)=O)CC2)C)=O)OCCCC1(C)C N1(C(C(CC)C)=O)CCOC(CNC(=O)CC2CC3(COC3)C2)C1 C12(C(=O)NCCCCC3CN(C(C4CC(C)OC4)=O)C3)CCC(O)(CC1)CC2 c1(CC)ccc(C(=O)NCC(CC)NC(=O)Cc2cc(C)cs2)s1 N1(C(C2(CSC)CC2)=O)CCCC2(CCN(C(=O)C#CC3CCCOC3)C2)C1 c1(CC(=O)NCCN(C(=O)C(C)C(F)(F)F)CC(C)O)cc(O)nc(O)n1 CCCCCCCCNC(=O)C(N1CC2(C1)CN(C(C1(CO)CCC1)=O)C2)=O c1(C(C(=O)NCCCOC)N(CC(C)OC)CC#N)cc(C)cc2c1CCC2 N1(C(C2CC(F)CN2Cc2cc(C(F)(F)F)ccc2Br)=O)Cc2ccncc2C1 c1(SCC)ccc(Cl)c(C(=O)NC2CCC(C(=O)NCCCO)CC2)c1 C(=O)(CS(=O)(=O)CC1CCCO1)N1CC=CC(NC(c2c(NCC)scn2)=O)C1 c1(C(=O)NC2C3CC2CN(C(C2C=CCC2)=O)C3)ccc2c[nH]nc2c1 CS(=O)CCC(O)C(=O)NCC1CN(C(=O)CC2CC2)C1 c1(C(N(C)CC2OCCN(C(C(CCC)O)=O)C2)=O)nn(C)c(=O)cc1C CN1N=C(CC(=O)NC(c2ccnn2C)C(=O)NCC2(C)CCOCC2)CC1=O C(=O)(C#CC1CCOCC1)N1CC(NC(C(F)OC)=O)C2(C1)CC2 C1(C(=O)NC(C=C)(C)CC)CCC(NC(=O)CC2(C)CCCCC2)CC1 Cc1ccc2c(c1)CN(C(C1CCC(NC(C3(C#N)CC3)=O)C1)=O)C2 C1(CC)CN(C(=O)CCc2ccc(F)cc2F)CCC1NC(c1csc(O)n1)=O C1(C(=O)NC(C#C)(C)C2CCCC2)CCC(CCNC(=O)CCc2nc[nH]n2)C1 c1(C(O)Cn2cc(-c3ncoc3-c3ccccc3)nn2)c(F)cccc1F C1(CC(=O)N(C)CCNC(=O)CCCN2CCCCC2)(OCC)CCCC1.OCC c1(NC(C2CCC(CC)CC2)=O)cc(NC(C)(C)C)ccc1P(C)(C)=O C(=O)(C(C)S(=O)(=O)Cc1ccc(Br)cc1)N1CCC(N(C)CC)CC1 c1(C(=O)NCCN(C(=O)C(C)(C)F)CC)cc(-c2ccccc2)oc1C CC1(C)CN(C(c2ccc(F)cn2)=O)C(CNC(C2CCO2)=O)CO1 c1(C(=O)NC2CC(C)(NC(=O)Cn3cnnc3O)C2)c(F)cc(Cl)cc1F C(=O)(C(C)(F)C(C)(C)F)NCC(CC)(CC)NC(=O)Cc1cccc(C)c1C C(=O)(C(CC(=C)C)NC(C1CCC(=O)N(C)C1)=O)NCC(C#C)CC C1(C(C)NC(c2ccnc(N(C)C)c2)=O)CCN(C(=O)C=CCO)CC1 c1(OC)cncc(Cl)n1.C12(COC1)C(=O)NCCOC1CN(C1)C2=O.CC N1(C(CCc2scc(C)n2)=O)CCCC1C1CCCN1C(=O)CCOCC1CC1 c1(CC(=O)NCC(C)NC(c2cc(-c3ccncc3)ccn2)=O)nn(C)cc1Cl C1(NC(C(C=C)C)=O)CCC(CC(=O)Nc2cnc(SC)nc2)CC1 C12(C(=O)NC3(CNC(c4c(N)cccc4F)=O)CCC3)CCCCC1C2(F)F c1(C(=O)NCC2CCC2C(=O)NCC2CCCO2)cccs1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC2C(NC(=O)CC3(CO)CC3)(C2)C1 c1(NC(N(C(CC)C)C)=O)cnn(CCOC)c1 C1(C)(CNC(C2(C(=O)OCC)CCC2)=O)CN(C(=O)C(O)C(C)CC)CC1C Cn1ncc(C(c2nnnn2-c2ccccc2)NCC2CCCS2)c1Br N1(C(C(COC)(C)C)=O)C2CCC1(CNC(C1CCC(F)CC1)=O)CC2 C1(CN(C(C2(COC)C=CCC2)=O)C)CC(F)CN1C(c1cc(C)c(Cl)s1)=O Cc1nc(C(=O)NC2CCN(C(c3c(C)nn(C)c3C)=O)C2)c2ccnc-2[nH]1 c1(C(=O)NCCCN2CCN(c3cc(OC)ncn3)CC2)cccc2nccn12 C1(C)(CNC(Cc2c(C(C)C)con2)=O)CCCN(C(C2(C)COC(=O)C2)=O)C1 C1(CC=C)(CNC(=O)C(=O)Nc2ccnn2CC2CCOC2)CCOCC1 C1(NC(CCc2nc(C3C(C)C3)sc2)=O)CCC(N=[N+]=[N-])CC1 CCC(C#N)C(=O)NC1CC(C(C)NC(=O)C=Cc2cnccn2)C1 C1(CC(=O)OC)C2CN(C(C3(N)CCC4CC34)=O)CC12 c1(C(N2CC(COC)(NC(=O)C(C)=O)C2)=O)ccccc1OC c1(C(N2CC(CNC(c3cncc(C)n3)=O)C2)=O)nc2n(c1Cl)CCCC2 C(=O)(C1CCCc2sccc21)NC1C(C)(C)CN(C(c2ccoc2)=O)C1 N1(C(c2cccc(N(C)C)n2)=O)CC(NC(C2(CCF)CCC2)=O)C(C2CC2)C1 C1(C(=O)NC(CC=C)C)CCC=CC1NC(=O)CC=O.OC N1(C(CC2CC(OCC)C2)=O)CCCN(C(=O)CC2SC(=N)NC2=O)CC1 N1(C(C(CC2CC2)OCC)=O)CCCCC(NC(c2cc(COC)on2)=O)C1 C1(CN(C(=O)C(O)c2cnc[nH]2)Cc2cnns2)CCOC1=O CC1CCN(C(=O)C(F)OC(F)(F)F)C1C(=O)NC(c1ccoc1)C C(=O)(C1CCCc2sccc21)N1CC(C)(NC(c2onc(C)n2)=O)C1 CC1CC(CO)CN(C(C2CCCN(Cc3ccnn3C)C2)=O)C1 C(=O)(CC(O)CC(C)C)N1CCC(C)(C(=O)NC(CCC)C(F)(F)F)CC1 Cc1cc(CCC(=O)NC2CCCC2CNC(c2n[nH]cc2Cl)=O)nn1C C(=O)(C(O)C1=CCCCC1)NCCC(CC)(C)NC(C1CC12CCOC2)=O C1(C)(C(=O)NC(CNC(c2cc(C(C)C)[nH]n2)=O)C2CC2)CCC(=O)N1 c1(C(=O)NC(C2N(C(c3c(SC)ccs3)=O)CCCC2)C)cc2cccnc2[nH]1 Cc1ccc(C(=O)NCC(C)(CO)NC(c2cccc[n+]2[O-])=O)cc1C C1(CNC(C(CCCOC)C)=O)CC2(CCC2)CN1C(C1CCCN1C=O)=O c1(OC)cscc1C(=O)NC(c1ccccc1)CNC(CCC(C)(C)C)=O c1(C(=O)NC2CN(C(CSCCC)=O)CC2C(F)F)cn2ccnc2s1 C(=O)(N1CCC(C(=O)NCCC(C)(O)COC)O1)c1c(CCC)n[nH]c1 N1(C(c2c(N)non2)=O)CCC(C2CCN(C(=O)C(=O)NCC(F)F)C2)C1 C(=O)(CC(C)(C)C#N)NCC=CC(=O)N(C)Cc1nnc(CC)o1 c1(C(=O)NCC(CC=C)NC(=O)CCC(C)(F)F)cc2c(s1)CCS(=O)(=O)C2 N1(C(c2ccc(C)s2)=O)CCC(C)(CCNC(=O)CC23COC(CF)(C2)C3)C1 Cc1oc(C(C)(C)C)cc1C(N1CCC(CCNC(=O)C(C)c2ccsc2)C1)=O C(=O)(CCC(=O)NC(C(C)NC(=O)C(=Cc1cccs1)C)C(C)C)N(CC)CC Cc1noc(NC(C2CN(C(c3cccc(=O)n3C)=O)CCN2)=O)c1C#N S(=O)(=O)(C=Cc1ccccc1)NC1CCC(NC(c2ccsc2Br)=O)C1 N1(C(c2c(C)occ2)=O)CC2(CCC2)CC1CNC(c1ccc(CCO)cc1)=O N1(CC)CCC(C(N2CC=CC2(C)C(N2CCOC(CC)C2)=O)=O)CC1 CC(CC(=O)NCCC(N)=O)NC(=O)Nc1ccccc1 C(=O)(C1=C(C)Oc2ccccc2C1)NC(CCNC(CCSCCCC)=O)(C)C C(=O)(CC(CN(C)C)C(F)F)N(C1(NC(CN(C(C)C)C)=O)CC1)C C(CC(CC)C(=O)N1CC=CCC1C(=O)NCC1CCC(C)C1)=CC C(C(=O)NC(CNC(c1cccc(SC)c1)=O)C1CCC1)(C(C)(C)C)OC N1(C(=O)C2=C(Cl)CC2)CCCC(C2CN(C(=O)COCCO)C2)C1 c1(CC(=O)NCCN(C(c2cnc(C3CC3)[nH]2)=O)C2CC2)ccc(F)cc1 N1(CCC)C(=O)CCC1C(=O)N(C)CC1CCCCN1C(c1coc(CO)c1)=O C1(CC)CCN(C(c2cnn(CC)c2)=O)C1C(=O)N(CCc1cc(C)[nH]n1)CC N1(C(COCC#C)=O)CCC2CCN(C(=O)CCCCCCCSC)CC2C1 C1(NC(C(C)NC(N)=O)=O)C2CC3CN(C(c4cc5occc5s4)=O)C1C3C2 CC1CN(C(C2(CNC(C3CC(O)C(F)C3)=O)CC3(CC3)C2)=O)CC(CO)O1 c1(CCC)cc(C(N2CC(CNC(=O)CCc3nncn3C)CC2C)=O)n(C)n1 c1(C(=O)NCCCN(C)C(C2(CF)CCC2)=O)cncc(C(F)F)c1 C(CC(F)F)(C(=O)NC(C)CN1CCOCC1)NC(Cc1c(C)nccc1)=O C(C)(c1ccccc1C)=CC(N1CC(OCC)(CNC(c2c[nH]cc2Br)=O)C1)=O N1(C(COCCCOC)=O)CCN(C2CCN(C(C3CCC(=O)N3)=O)CC2)CC1 c1(C(N2CC(CC(C)NC(C(CC)(C)F)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl C1(C(N2CCCC(CCNC(C(C)=C(C)C)=O)CC2)=O)CC2CSCC(C1)C2 C(Cc1ccco1)(C(=O)N1CCC1Cc1ccco1)NC(C(C1CC1)OC)=O C=CCN=C(NCC(C(C)(C)C)OC)N1CCC(OC)CC1.C1CC(=O)N1C1CC1 c1(C(N2CCC(NC(c3cnc(OC)c(Cl)c3)=O)C2)=O)c(Cl)cccc1[N+](=O)[O-] C1(CNC(C(=CC2CCCC2)C)=O)CC2(C1)CN(C(C1CCCC1(F)F)=O)C2 N1(C(C(C)OC)=O)CCC2(CCCCC2NC(c2cc(C)no2)=O)C1 C(CCCCCN=[N+]=[N-])NC(C(C(C)NC(C1CCCCN1C)=O)(C)C)=O C1(O)(C(C)NC(=O)CCc2cn[nH]c2)CCN(C(=O)C(N2CCC(O)CC2)C)C1 CCC(O)C(C)(C)C(=O)N1CCC(CNC(c2sccc2F)=O)(OC)C1 c1(CC)ncc(Cl)c(C(=O)NCC2CN(C(=O)CC3(C4CC4)CC3)CCN2C)n1 C(=O)(C1=NOC(CC(=O)N(CC(CC(C)C)NC(C2(CO)CCC2)=O)C)C1)OC c1(OC)ccccc1CC(=O)NCCCOCCNC(=O)C=C1CCSCC1 C1(OC)CCN(C(C2C=CCCN2C(=O)CC2(O)CCC2)=O)C1(C)C O=C1Cc2cc(C(N3CC(NC(c4cc(Br)c[nH]4)=O)C(F)C3)=O)c(Cl)cc2N1 N1(C(c2c(C)ccs2)=O)CCCC(CNC(c2c(C)cnn2C(C)C)=O)CC1 CCC(CC(=O)NCc1c[nH]nc1C(=O)NC12CC(C)(C1)C2)C1CCC1 C12(C(=O)NCCN(C(=O)Cc3cn(CC)nn3)CCC)CC(OC)C1C2 CC1N(C(=O)C(C2CN(C(c3ccc(F)c(O)c3)=O)C2)N(C)C)CCCC1(C)C CC12CC(NC(=O)C(C3CCCCC3)O)(C1)C1(CN(C(c3ccc(F)s3)=O)C1)O2 c1(C(=O)NCC(C)N(C)C(c2ccc(F)o2)=O)c(Cl)cc(Cl)cc1Cl N1(C(C2(C(=O)OC)CC2)=O)CCC(C)(CC(N2CC3CC3C2)=O)CC1 C(CCOCCO)(C(=O)NC1CC(O)(CO)C1)NC(C1CCC(F)(F)C1)=O C1(NC(C=COCC)=O)CC2CCC1(CNC(c1cnc(C3CC3)o1)=O)C2 c1(COC)cccc(C(N2CC(NC(=O)C(Cl)=CCl)CC2CO)=O)c1C c1(CC(=O)NCC2N(C(CNC(=O)NC)=O)CCC2)ccc2nc[nH]c2c1 c1(OC)cc(OC)c(OC)cc1CN(C)CC1(O)CN(c2ncncc2F)C1 N1(C(CN(C)CC)=O)CCN(C(=O)CN2CC(=O)NC2=O)C2CC12 Cc1cccc(C(=O)NC2CC2C(N2CCC(O)C2)=O)c1 Cc1ncnc(C)c1CC(=O)N(CC(C)O)CCNC(=O)CSC1CC1 C1(C2CCCCN2)(C(N(CC(C)CO)C)=O)CCOCC1 CC1(C)CN(C(=O)Cn2ccc(=O)c(O)c2)CC(CNC(C23CC(C2)C3)=O)O1 N1(C(C(C)OCc2cccnc2)=O)CCC2CN(C(C3(CF)COC3)=O)CC12 CC(CCC(=O)NC1CC(NC(=O)CC2CN(C)C2)C(O)C1)N(C)C C1(NC(=O)C2CC2)Cc2ccccc2N(C(c2cn(Cc3cccs3)nn2)=O)C1 CCCCC(C)C(=O)N1CC2(C1)CN(C(c1ccc(N(C)C)cc1OC)=O)C2 C1(C(N2C(CC(=O)NC3CCC(N(C)C)C3)CC(O)C2)=O)CCCC12CCC2 N1(C(=O)CC2CCC2)CCCC2(C1)CN(c1ccnc3cc(Br)nn13)CCO2 Cc1cc(NC(c2cc(Cl)cn2C)c2nnnn2C(C)(C)C)cc(C(F)(F)F)c1 C1(C(N2CC(COC)(NC(=O)CCc3cccs3)C2)=O)(OC)CCSCC1 C(=O)(CC(F)(F)C(F)F)N1CCC(C#C)(C(=O)NCCC2CC(C)=NO2)C1 N1(C(CC(=O)NCC#C)=O)CC2COCCC2(NC(c2ccc(F)cc2C)=O)C1 N1(CCC(NC2c3n(C)ncc3CCC2)=O)CC2(CCOCC2)CC1CC(=O)NC Cc1cnn(CC(=O)NC2CCC(NC(c3cscn3)=O)C2)c1 c1(C(=O)NC2C(NC(C=C(C)C(F)F)=O)CC2)ncnc2c1CCC2 C1(C(=O)NC(c2ccccc2)CNC(C2(CO)CCC2)=O)CN2CCN1CC2 CCCCC(C)CC(=O)N1CCCC1C(C)(C)C(=O)NCC(=O)N(C)CC c1(NCCCN(C(c2n(CC)ncc2)=O)C)nc(O)n(C)c(=O)c1[N+](=O)[O-] n1(-c2ccc(-n3c(C)ncc3)s2)ccc(=NC(=O)C2CC2C(=O)OC(C)(C)C)[nH]1 C=CC(C)(CC)C(=O)NCC1(F)CCN(C(c2ccc(C)c(F)c2)=O)C1 C=CCCCCC(c1nnnn1CCCC(=O)OCC)Nc1cccc(F)c1 C(=O)(CCCCC(F)(F)F)NCCN(C(=O)C(C(C)C)C1CC1)CCOC C12(C(N(CCCCO)CC)=O)CCN(C(c3nc(O)sc3C)=O)CCC1C2 c1(C(N2CC(CC=C)(NC(=O)CNS(=O)(=O)N(C)C)C2)=O)cccc(Cl)c1C c1(C(N2CCC(F)(CNC(Cc3cc(C)on3)=O)C2)=O)cccc2cnn(C)c12 c1(-n2c(C(C(C(C)C)N3CCOCC3)NCCOCC)nnn2)ccc(OC)cc1 C(C1=NOC2CCCC12)NC(C(C1CN(C(CCC=C)=O)C1)O)=O C1(C(=O)NCC2C(CNC(COc3cccc(CC)c3)=O)C2)OCCOC1(C)C C(=O)(C(C)(C)CCF)N1CC2C(C(=O)NCCC(C)N3CCC3)(C2)C1 c1(CN(CCOCC)C(C2CCN2CC)=O)ccccc1Cl.C1CC(=O)N1 C1(C(=O)NC(c2nc(C(N3CCC3CC(C)(C)C)=O)co2)C)(CO)CC=CC1 c1(OC)ccccc1-c1ncc(C(=O)NC2CCC2CNC(=O)C(C)N(C)C)s1 CC(C)(C)C(CNC(C1CC12CCOC2)=O)NC(=O)CSc1ccc(O)cc1 N1(C(C(c2ccc(Cl)cc2)C)=O)CC2(C1)CN(C(=O)C(C)(C)S(C)(=O)=O)CCO2 C#CC1(C(=O)NC2CCOC2=O)CCN(C(=O)COC)C1 c1(NCc2cn(CCCCCCNC(C(C)(CO)OC)=O)nn2)cnc2ccnn2c1 N1(C(CSCc2nc(C)sc2)=O)CCC(C)C1CNC(=O)CCc1cc(Cl)no1 CCCC(O)C(=O)N(C1CCC(NC(=O)C(C)(F)F)CC1)C CC1CCCC2CCCN(C(c3c(F)cc(F)cc3[N+](=O)[O-])=O)C12 c1(OC)cnc(Cl)[nH]c1=NC(=O)C1(SC)CN(S(=O)(=O)C(Cl)(Cl)Cl)C1 c1(NCC(CC)C)cc(NC2CC2c2ccc(OC(C)C)cc2)nc(C)n1 C12(C(N3CC(CCNC(CCNC(=O)NC)=O)C3)=O)CCCCC1CCCC2 CCC(C)CC(C)C(=O)N1CCC(C(=O)O)C(F)(F)CC1 c1(CC)nn(C)c(C(=O)NCC2CCCCN(C(=O)CCc3cnoc3)C2)c1Cl CCC(CCC(=O)N(C(C)CC(=O)Nc1ccc(OC)c(O)c1)C)OC CCCN(OC)C(=O)CC(CCC)NC(=O)C(N)CCCC(C)C C(=O)(C(C)(C)C(C)C)NC(C=CC(=O)NCC1CCN(CCC)C1)C Cc1c(C(N2CC=CC2CNC(=O)C(F)C(F)(F)F)=O)oc2ccc(F)cc12 C1(CC#C)(C(=O)NCC(=C)CCNC(=O)CCC2CCCOC2)CCOC1 Cc1n[nH]cc1CN(C)C(c1ccoc1CNC(C12CSCC1C2)=O)=O C1(NC(c2nc(C(C)OC)sc2)=O)CCN(C(C2(CSC)CC2)=O)CC12CCC2 c1(C(N(C(CC)C(=O)NC2CC2)C)=O)ccnc(OC)n1 C(CC(CC)C(=O)N1CC(CC(F)C(N2CC3C(C(C)C)C3C2)=O)C1)=CC C1(NC(CS(=O)(=O)N(CC)CC)=O)CC2CN(C(c3c(Cl)n[nH]c3C)=O)CC2C1 Cc1nc(C(N2CC=CC(NC(=O)CCCCNC(N)=O)C2)=O)nn1C c1(CC(C(C(=O)Nc2cncc(OC)c2)F)C)c[nH]c2ccccc12 c1(CC)ncc(C(N2CCC(NC(c3csc(C#N)c3)=O)CC2C)=O)c(C)n1 CC1CN(C(=O)C(c2cnn(C)c2)NC(c2ccc(F)cc2)=O)CCN(C)C1 N1(C(CC(C)c2ccco2)=O)CCSCC1C(=O)NCCC1(C)CC1(F)F C(C(CO)(CO)NC(C1OCCC1(C)C)=O)N(C(C1(CC)CC1)=O)C c1(OC)ccc2c(c1)CCC2(O)CNC(=NC)N1CCN(c2ccccn2)CC1 c1(CC)nc2sc(C)cn2c1C(=O)NC1CCC(CNC(C2C3COCC23)=O)C1 C1(NC(CSC)=O)CN(C(c2cc(O)nc3c2CCCC3)=O)CC12CCOCC2 CC(CC(N)=O)C(=O)N1C(CNC(=O)CCc2nnc(C(F)F)o2)CC2CC12 C(C)(CCCCNC(c1cccc(C2CC2)n1)=O)NC(C=CC=CC)=O N1(C(CCSC)=O)CC2CC(CNC(C3(c4ccnc(Cl)c4)CCC3)=O)CC1C2 N1(C(C(COC)O)=O)CCN(C(c2ccn(C3CC3)n2)=O)C(C(F)F)C1 C(CO)(C(=O)N1CCCC1CN(C(=O)CN(C1CC1)CC)C1CC1)OC c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1c(Cl)cnn1C)=O N#CC1CCC(CC(=O)NCC2(NC(c3cc(C4CC4)n[nH]3)=O)CC2)C1 N1(C(c2cncc(OC)c2)=O)CC(C)CN(C(C2CC(F)(CO)C2)=O)CC1C N1(C2(C)CC2)CCN(CCC(=O)NC2CCN(C(c3nn[nH]c3Cl)=O)CC2)CC1 c1(C(=O)NC(CC(C)NC(c2cnc(C(N)=O)s2)=O)C)ccc(C2CC2)cc1 C(=O)(C1=CC2CCCC12)NCC1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 C1(CCOC)CN(C(=O)C2=NOC(C(C)(C)C)C2)CCN1C(=O)CS(N)(=O)=O C1(NC(CC(C2(O)CCCCCC2)(C)C)=O)CC2CCC(C1F)N2C(=O)C1CC1 N1(CCC(=O)NC(CNC(C(CC)F)=O)(C)C2CC2)CCN(C)CC1 c1(C(N(C2CCN(C(C3CC3F)=O)C2)CCC)=O)cc2c(nn1)OCCS2 c1(OC(C)C)nc(N2CC3C(C(=O)Nc4ccc(CO)nc4)C3C2)ncc1Br C=CCC(C)(C)CCN(C(=O)C(c1cccs1)NC(C)=O)C Cc1ccc(C(=O)NCC2CC=CCC2)nn1 C1(C(N2C(C)C(NC(=O)C(F)Cc3ccccc3)CC2)=O)CC2(CCCCC2)C1 Cn1c(C(=O)NC2CC(NC(C3(CO)CCCO3)=O)C2)cnc1S CC(O)C(C(=O)NC1CCC1)NC(C1CC1C(N)=O)=O c1(OC)c(Cl)cc(C(=O)NC2CC2NC(=O)CCOc2cccnc2)nc1Cl C1(CCNC(c2ccc(Cl)s2)=O)CSCCN1C(C1(c2cccnc2)CC1)=O c1(C(=O)NC2C(NC(c3c(CC)nn[nH]3)=O)CCC2)c[nH]c2cccc(Cl)c12 C(=O)(C1=CNS(=O)(=O)N=C1C)NCCN(C(C(C)OCC#C)=O)CC(C)O C1(C(N2C(CNC(C3C(C)(C)C3C#N)=O)CCC2)=O)CC(=O)CC(=O)C1 C1(NC(CCCc2n(C)cnn2)=O)CN(C(C2(c3ccnn3C)CC2)=O)CC1F Cc1ccc(CC(=O)NC2CCN(C(c3cc(O)nc(Cl)c3)=O)CC2F)c(C)c1 c1(C(=O)NC(CC(C)C)(C)CNC(C2CC=CCO2)=O)ccc2cncn2c1 O=C(CC1CCc2ccccc21)NC1CCN(C(C2C3CC4C(C3)C24)=O)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CC)CC1(CNC(=O)C(C1CC1)OC)C2 N1(C(CSCC(C)C)=O)CCCC(CN(C)C(c2cc(C(N)=O)cn2C)=O)C1 c1(C(=O)NCCCN(C(=O)CC2CCC(C#N)C2)C)cn(C)nc1Br Cc1cc(C(=O)NC2CC(O)CN(C(c3ccccc3C(C)C)=O)C2)cc(C)c1 N1(C(C(C)=C(CC)C)=O)CC2(COC(CNC(c3nccn4ccnc34)=O)C2)C1 C1(C(N2C(C(=O)Nc3ccc(OC)nc3C)CC3CC32)=O)CCc2ccccc2C1 C1(CNC(CCC=C(C)C)=O)CCCCN(C(C2(C#N)CCCO2)=O)C1 c1(CC(=O)NCC2CCN(C(c3ccc(C(N)=O)s3)=O)C2)nnc2n1CCCC2 c1(N2CCCC(CC)CC2)nc2ccsc2c(=NCC2(CO)CCCOC2)[nH]1 C1(CNC(=O)CN2CCOC2=O)CC2(C1)CN(C(=O)CO)C2 c1(OCC(N2CC(NC(c3nc(CC)oc3)=O)C(C)C2)=O)c(C)cc(C)cc1C c1(C(N2C(C(CNC(C(C)(C)F)=O)(C)C)CCC2)=O)cnc2cc[nH]c2c1 CCCC(O)CC(=O)NCC12CC(CNC(c3n[nH]c(C)c3Cl)=O)(CO1)C2 CCN=C(NCc1cnc(Cl)cc1C)N1CCC(O)C1 C(CCC(C)NC(c1cccnc1)=O)NC(C(c1ccccc1)C)=O c1(CN(C)C)cc(C(=O)NCC2CCN2C(=O)CC2CCCO2)ns1 C1(CNC(CC(CC)C2CC2)=O)N(C(=O)C=CCOCCO)CCCC1(C)C C=Cn1nncc1C(=O)NC(COCC)C(=O)NCCC1COCCO1 N#CC1CCCC(C(N2CC(CC(F)C(=O)NCC(C)(C)NC=O)C2)=O)C1 c1(CC)ccc(Cl)nc1NC(C)Cc1ccccc1C.C(CC)(CC)n1c(=O)c1=O c1(NC(c2ccncc2-c2ccccc2)=O)ccc2oc(Cl)cc2c1 Cc1cc(C(N2CCC(C(C)NC(=O)CC(c3cccs3)C3CC3)C2)=O)c(C)s1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCOC(C(C)NC(C2(C(C)(F)F)CC2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC(C1(O)CN(C(C(Cc2ccccc2)OC)=O)C1)C C(CNC(=O)CC=CC(C)(C)C)(CC(F)(F)F)NC(C(C1CC1)OC)=O c1(CNC(C(=O)OC)(C)c2cccnc2)cc(Br)sc1Br C1(NC(c2cscn2)=O)CC2CCC(C1F)N2C(c1sccc1OC(F)F)=O c1(CC(=O)N(CC(O)CN(C)C(C2CC(O)C2)=O)C)cncnc1O N1(C(CC2CC(=C)C2)=O)CCC(C2CC2)C1CNC(C1C2C3CCC(C3)C12)=O C1(C)(C(=O)NC2C(NC(C(c3c(C)cncc3)C)=O)CCC2)C(C)(C)C1(C)C c1(C(CC)C)nc(C)c(CC(=O)NC(C)CCCNC(=O)C(C)CO)c(C)n1 C1(CC(=O)NC(C2CCN(C(C3CC(=C)C3)=O)CC2)C(C)C)CC(O)C12CCC2 O=Cc1cccc(-c2cncc(CN3CCC(Br)CC3)c2)c1Br C1(C(N2C(C)(C(=O)NCCCN(C)C)C=CC2)=O)CC2(CCC2O)C1 CCCC(C(=O)OC)C(=O)NCC(C(C)C)NC(=O)COc1cnc(Cl)cn1 c1(OCC(=O)NC2CN(C(C(C)(C)Cc3ccccc3)=O)C2)nc(O)nc(O)n1 C1(NC(c2c(C)nccc2)=O)CN(C(=O)CCc2ccncc2)C2CCCCC12 CC(C)CC(C(=O)NCCC1CC(NC(C2(CF)CC2(F)F)=O)C1)C(C)C c1(C2(OC)CCN(C(c3n(CC)ccn3)=O)C2)cc(Br)ccc1F C(=O)(CC(O)C(C)C)N1CCC(OCC(=O)NCc2nc(C)c(C)s2)C1 N1(C(C2CC(C)=C(C)CC2)=O)CC2(CCCC2NC(=O)CCOC(C)C)C1 N1(C(c2c(C)oc(C#N)c2)=O)CCC2(CC1)CCN(C(=O)C=CI)C2 CCC(O)C(C)(C)C(=O)NC1CC(CNC(c2ccoc2C2CC2)=O)C1 c1(C(=O)NC2C(C(N3CCC(OC(C)=O)C3)=O)COC2)nccc(C)c1N CCC1(CNC(C2CN(c3ccc(Br)cc3)C(=O)O2)=O)OCCc2ccccc21 C=CCC(C(=O)NCC(C)N(C(=O)Cn1nccc1C)CC)NC(C)=O N1(C(C(CC)(CC)OC)=O)CC(NC(=O)CCCCCOC)C(C2CC2)C1 Cc1cccc(C(c2ccccc2)SCCCNC(=O)CCC2CCCN2C)c1 N1(C(c2c(C)noc2)=O)CC2CC1CN(C(=O)C(C(C)C)n1ccnc1)C2 C(CCC(=O)NCC1CCCN1C(C1CC2CC2C1)=O)N(C(C)=O)C CC(C)(CCCNC(c1sccc1F)=O)NC(=O)COc1ccccc1C(N)=O c1(CC)nsc(CNC(=O)C(C)CN(C(=O)Cc2cc(C)cs2)C)n1 N#Cc1ccc(C(N2CCC2CC(=O)Nc2ccc(C3CC3)cc2)=O)nc1 C(=O)(C1Cc2ccc(Cl)cc21)NCC(CC)NC(=O)C=Cc1ccccn1 CCCCC(CNCc1cccc(C#N)c1F)CCC c1(C(=O)NCC(CNC(c2ccccc2F)=O)OC)cc(S(N)(=O)=O)oc1C C(=O)(C(C)(C)C(=O)NCC1CC(C)(C)CN1C(=O)C(CC(C)C)N(C)C)NC CN1C(=O)C2CN(C(=O)C(=O)N(C3CNCCC34CCC4)C)CC2C1=O Cn1nnc2cc(C(=O)NCCCC)cc(Br)c12.C1(C(=O)N)CC(C)(C)CCO1 C1(COC)(NC(c2cc(Cl)cnn2)=O)CCN(C(=O)CCCc2ccccn2)C1 C(=O)(C(=O)CCC(C)C)NC1C(CC)CN(C(=O)COC2CCOCC2)CC1 C1(CC)CN(C(c2cc(C)ccc2I)=O)CCN1C(c1cc(C)on1)=O c1(C(N2CCC(O)(CN(C)C(C3CCCO3)=O)C2)=O)cccc2c1CCC2=O c1(C(CNC(CSC)=O)NC(=O)C(O)CF)ccc2ccccc2c1 C(CCN(C1CCCCCC1)N1CC(C(=O)OC)C(c2cncn2C)C1)OCC c1(OC)cc(Br)ccc1CN1CC2CC1CN2Cc1ccc(C(=O)N(C)C)nc1 C#Cc1ccc(OC)c(C(=O)NC2COCC2NC(c2conc2C2CC2)=O)c1 C1(CC(=O)NCC(=O)NC(CN(C(c2cncnc2)=O)CC)C)CCOCC1 C1(NC(CC2(OC)CCC2)=O)CCC12CCN(C(c1nsnc1OC)=O)CC2 C#CCCCCC(=O)NC(c1cn(C)nn1)C(N1CCC(C)(O)C1)=O C1(C(F)(F)C(=O)NC2CC(NC(=O)Cc3cnsc3)C2)(OC)CCOCC1 C1(NC(Cc2cc(C)[nH]n2)=O)CN(c2ncnc3scnc23)CC2(CC2)C1 C12(CNC(CC3C=NN(C)C3=O)=O)CC(NC(=O)CCOC(C)C)(C1)C(C)(C)O2 CN=c1[nH]c(=NCC(C)c2ccsc2)[nH]c(=NC2CCCCC2CC(C)C)[nH]1 Cc1cc(C(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)ncc1F c1(C(C(N2CC(OCC)(CNC(c3cc(F)c[nH]3)=O)C2)=O)(F)F)cccc(C)n1 c1(C(N2CC(NC(C3(O)CCOCC3)=O)CC(O)C2)=O)cccc2ccccc12 C(=O)(C(C)CC(=O)OC)NCC(CC)NC(c1ccc(OC)nc1C)=O Cc1nc(S)nc(C)c1CCC(=O)NCCC(C)N(C)C(c1ncccc1Cl)=O N(C1CN(C(C23CC(F)(C2)C3)=O)CCc2ccccc21)C(C(CC)OC)=O C1(C(=O)NCC=CCNC(C(C2CCCC2)OCC)=O)CC(CC)CO1 N(C1CN(C(=O)C(C)N(C)C)Cc2ccccc21)C(C1(C(C)C)CCCCC1)=O c1(NC(=O)NC2CC(SCCCOC)C2)c(C)nn(-c2ncccc2Br)c1C C(c1cnc(C)nc1O)=CC(=O)NC1CCN(C(c2cn(CC)nn2)=O)C12CC2 C(=O)(C(=O)N=S(C)(C)=O)NCC1CC(C)N(C(=O)CCC(C)(F)F)C1 c1(OC)ncc(F)cc1C(=O)NC(C)(C)CNC(=O)C(C)c1cc[nH]n1 CN1CCC(CO)(CNC(=O)C(CCC2CC2)NC(c2coc(C(N)=O)c2)=O)C1 c1(C(N(CCNC(=O)CCc2cccnc2Cl)CC)=O)c(C)cccc1C c1(C(C)C)ccc(C(=O)NCc2cc(C(N3CCCC3CO)=O)on2)s1 C1(NC(c2ncoc2C2CC2)=O)CCCC(CNC(C2CC(O)C2)=O)C1 c1(C(=O)NC(C(=O)NCC2OCC(C)(C)C2)C2(O)CCC2)cc2ccccc2o1 c1(C(=O)NC2C3CN(C(=O)C=CC4CCOC4)CC23)cc2c[nH]cnc-2n1 N1(C(CC2(C)CCC2)=O)CCC(O)(CCNC(c2cccc(F)c2)=O)C1 C1(NC(C2C(C)C2C)=O)CCOCC1C(=O)NC1(CN(C)C)CCCCC1 C(=O)(C1=C(C)OCC1)NC1CC(C)(C(N2CC(C)(OC)C2)=O)C1 CCCCC(=O)C(=O)N1CC(N(C(=O)Cc2ccc(OC)cc2)C)C(O)C1 CC1CC(CO)CN1C(=O)C#CCNC(=O)CCCC1CCCO1 Cc1nn(C)cc1C(=O)N(C1CC2CNC1C2)CCc1cnc[nH]1 c1(CCC=C)ccc(C(=O)NCC(C)(O)CNC(C2CCCOC2)=O)cc1 C1(NC(c2ccc(COC)s2)=O)C2CN(C(C3C4CCC3(OC(C)=O)C4)=O)CC12 CCC(C)(CO)C(=O)NCCC1CCN(C(c2csc(=N)[nH]2)=O)C1 C(CCO)N(S(C)(=O)=O)CCN(C(CCC)=O)C.N c1(C(=O)NCC(CCOC)Nc2ncc(C#N)cc2F)sc2nccn2c1C N1(C(C(CCOC)C)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 c1(CN(C)C(=O)NCC2(Cl)CC2(F)F)nc2c(s1)CCCC2 c1(COC(C(C2CCCOC2)OC)=O)cccn1C(c1ccncc1)C C(=O)(C(C#N)(CC)CC)NC1CC2(C(C(N3CC(C#C)OCC3)=O)C2)C1 Cn1nc(C(=O)NCC(C)(Cn2cccn2)NC(=O)CC2CC23CC3)cc1O CC1=NOC(=O)C1CC(=O)NCCC(C)NC(=O)Cc1nc(C2CC2)cs1 C(CC(N)=O)(C(=O)NCc1cn(C)nc1O)NC(CCC=C=C)=O c1(CC(=O)NC2CC2CNC(C2(c3cccs3)CC2)=O)ccc(O)nc1 O(NC(=O)CCCC(C)(C)NC(C1CC(OCc2ccncc2)(OC)C1)=O)CC c12cccc(c1)O2.c1(CC)ccc(C(=O)NC(C)CNC(=O)COCC(C)C)s1 c1(C(=O)NCC2N(C(CCC3CC(OC)C3)=O)CC2)ncccc1O c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CCOC2)cc(=N)[nH]c(Cl)n1 c1(C(N2C(CNC(C3ON=C(C)C3)=O)CN(C)CC2)=O)cnc2[nH]cc(C)c2c1 Cc1cc(CN(C(=O)C(N2CCC(c3nncs3)C2)=O)C)cs1 c1(COC)cc(C(N2CCCC2C2CCN(C(=O)CC3CCSC3)C2)=O)n[nH]1 c1(C(N2CC(NC(C3CCCN3C=O)=O)CC(OC)C2)=O)ccc(C#N)c(C)c1 Cc1c(C(=O)NC(C)CCCCNC(=O)CCC(C)N(C)C)cnn1CCN(C)C N1(C(C2C(CNC(C(C)n3ccnn3)=O)CC2)=O)CCN(C(C)(C)C)CC1 N1(C(CCSC)=O)CC2CCCC1C2CNC(=O)CC1CCCCCC1 c1(C(=O)NC(C2CCCN(C(c3cc(F)n[nH]3)=O)C2)C)ccc2nsnc2c1 C(=O)(CS(=O)CCC(F)(F)F)N(C1CN(C(c2cc3cccnc3s2)=O)C1)C C1(NC(CCC)=O)CCC2(CCCN2C(c2cccn(C)c2=O)=O)CC1 N1(C(c2c(CC)c[nH]n2)=O)CCCC2(C1)CN(C(=O)CN1OC(C)(C)CC1=O)C2 C#CC1(C(=O)N(C2CCC2C)C)CCN(C(=O)C(F)CCC)C1 N1(C(C(c2n(C)ccc2)=O)=O)CCOC2(CCN(C(C3CC(F)(F)C3)=O)C2)C1 c1(C(=O)OC)cc(NC(=O)C(=O)Nc2ccc(SCC(C)C)cc2)c(C)cc1F c1(C(=O)NC(CN(C(CC(c2ccc(F)cc2)C)=O)C)C)ccc2ncnn2c1 c1(C(N2C(NC(C(c3c(C)cncc3)C)=O)CC2)=O)cc(Br)cc(N)c1C Cc1ncc(NC(C2CCCCC2CNC(=O)C(C)CN(C)C)=O)c(C)n1 c1(N(C2C(C)CCNCC2)C(c2ccc(F)cn2)=O)cc(Cl)c(I)cc1[N+](=O)[O-] c1(C(=O)NC(C2(CNC(C(C)Cn3cccn3)=O)CC2)C)ccsc1C#N CC1C(NC(c2ccc([N+](=O)[O-])s2)=O)C(C)CCN1C(=O)Cn1cccc1 CC1(C)CN(c2cc(Cl)c(O)nn2)CC(CNC(=O)CN2CCC(F)CC2)O1 N1(C(C2(NC(CC3CCN(C)C3=O)=O)CC(F)(F)C2)=O)CCN2CCC1C2 C(=O)(CC(F)(F)C(C)C)NC1CCC(CCNC(C2(OC)CCSC2)=O)C1 C1(NC(C(CC)(F)F)=O)CCC2CC1CN2C(=O)C=Cc1ccccn1 CC1CN(C(=O)CCC2CCCN(C)C2)CCCN1C(=O)Cn1cccnc1=O C(CC1=CCN(Cc2cncs2)CC1)NC(C(c1c(C)noc1C)C)=O c1(C(=O)NC(C2CCCCN2C(=O)C=Cc2ccncc2)C)ncccc1Cl CC1(CNC(C2(CCO)CC2)=O)CCCN1C(c1cccc(C(F)(F)F)c1)=O C1(CC(=O)NC23CC(NC(CC4CC(=C)C4)=O)(C2)C3)C=CS(=O)(=O)C1 c1(SCCC)ccc(C(=O)NCC2(NC(=O)CC34CCCC3C4)CCC2)cc1 C1(NC(CN(C(C2(CC=C)CC2)=O)CCC)=O)CCn2ccnc2C1 C(=O)(C(C)(C)C)N1CC(c2cn(C3C(S(C)(=O)=O)CCC3)nn2)(O)C1.c1ccccc1 C1(CCNC(C2(C(CC)=O)CC2)=O)C(C)CCCN1C(c1coc(O)n1)=O c1(CNC(N2CC3(C(C)(C)CC3)C2)=O)c(Cl)cccc1[N+](=O)[O-] c1(CC(N2C(CNC(C(C)Cc3ccc(Cl)cc3)=O)CC2)=O)c(O)ncnc1O c1(C(N(C2CCCCC2)CCC(=O)OCC)=O)cc2n(c(=O)c1)CCS2 n1(CC(C)N(C(c2coc(C)n2)=O)C2CC2)cc(CNC(C2CC(=C)C2)=O)nn1 c1(NCC(C)(Cn2cccn2)NC(C2N(C)CCOC2)=O)ncnc2c1COC2 N1(C(C(CO)N(C)C)=O)CC(F)(F)CC1CCNC(c1cc2n(c1)CCC2)=O c1(C(=O)NC2(C)CC(NC(c3c(CC)c[nH]c3)=O)C2)cc2c(Br)cccc2[nH]1 N1(C(CC(C)OC)=O)CCCC2(CNC(c3cccc4occc34)=O)CCCC12 CC(N=c1cc2n([nH]1)CCOC2)c1nc(Cl)ccc1Br C1(C(=O)NCC#CCOC)C=CCN(C(c2ccc(SC)o2)=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)N(C)CC2CCCN(C(=O)CCN3CCC3)C2)n1 C1(NC(C(=O)NCC)C)COc2ccc(Cl)cc2C1=O C(C1=CCN(C(c2scnc2Cl)=O)CC1)NC(C1C(C)C1C)=O c1(C(=O)OC)c[nH]c2ncnc(N3CCOCC3C(=O)CC3CCCC3)c12 C12(NC(C(CC(C)C)O)=O)CCCCC1CN(C(c1nc3cnccc3s1)=O)C2 c1(C(=O)NC(C(C)NC(=O)Cn2nccn2)C)cnc2sccn2c1=O N1(C(C(CCC#C)O)=O)CCC2CN(C(=O)C=Cc3nccs3)CCC12 C1(NC(c2n(C)c(S)nn2)=O)CC2CCC1N(C(c1ncc(F)cc1F)=O)C2 C1(NC(C(C(C)(C)C)OC)=O)CCCCCN(C(=O)C=C(Cl)Cl)C1 N1(C(C(c2cccc(O)c2)C)=O)CC2CCC(C1)N2C(C1CCC2(CCC2)C1)=O c1(C(N2CCC(CN(C(=O)CSCCC#N)C)C2)=O)c(O)nnc2c1CCC2 Cc1c(C(=O)NC2CC(C)(CNC(=O)CCCCN(C)C)C2)cccc1O C#CCCCCCC(=O)NC1(C)CCC(C(=O)NOCC(C)O)CC1 C1(C)(C(N2CCC(CC=C)(NC(=O)CC(=O)NCC)C2)=O)CCNC(=O)C1 C1(SCC)CCCCN1C(=O)C(O)CCn1cc(-c2ccnn2C2CCC2)nn1 CC(C)(C)C(O)C(N)C(=O)N1CCCC(O)(c2cnn[nH]2)C1 C(CC(CC)C(=O)N1CC(C(=O)NOCC(C)(C)C)CC(C)C1)=CC N1(C(C2C(O)CCN2C(C2CC2c2ccc(F)cc2)=O)=O)CC2CCCCC2C1 C12(Nc3nc(CC)cc(CC)n3)CCCC1CN(C(C1(COC)CC1)=O)C2 c1(C(N2C(C(=O)O)C(c3ccccc3)CC2)=O)cc(Br)cc([N+](=O)[O-])c1 c1(NC(N2CC(F)(F)CC2c2ccc(C(F)(F)F)cc2)=O)c(O)ncnc1O C1(CCC2(OC)CC2)CC(C)N(C(=O)OC)C(NC(=O)OC(C)(C)C)C1 C1(NC(C2OCCN(C(CCCOCCC)=O)C2)=O)CCCCC1C#N c1(C(N2CC(CNC(=O)CCCc3nccs3)C3C2C3)=O)ccc(O)c(Cl)n1 C(CCSC)(C(=O)NC(C)CCC=C)NC(CCC#C)=O c1(C(N2C(C(=O)NC(CSCC)CO)CCCCC2)=O)cccn2ccnc12 C1(CNC(c2c(CC)c[nH]n2)=O)C2CN(C(=O)CC3CCC(=O)CC3)CC12 S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1C(C(=O)Nc2cnc(I)cn2)CC(F)(F)C1 CC(C)S(=O)(=O)CC(=O)N(C1CCN(C(C2CCc3cncn3C2)=O)C1)C CCC(Cc1cccc(C)c1)C(=O)NCC(C)CNC(=O)CCn1ccc(C)n1 N1(C(CN(C(C)=O)C)=O)CCCC(CNC(=O)CCN(c2ccccc2)C)C1 C1(CNC(CN(CCC#C)C)=O)CN(C(=O)C(C)(C)CSC)CC1O c1(C(=O)NCC(C)NC(=O)CCCCN2CCOCC2)cc([N+](=O)[O-])cc(=O)n1C C(=O)(C(F)(F)CC(C)C)N1CC(OC)(CNC(c2ccc(CO)cc2)=O)C1 N1(C(c2ccc(C#C)cc2)=O)CCCC1C1CCCN1C(c1cc[nH]c1)=O C1(C(=O)NCc2cncn2C2CC2)CCC(O)CN1C(c1cnc(S)nc1)=O C1(C)(C(=O)NCc2ccc(SC)o2)CCCN1C(c1ccsc1C#N)=O CC1CC(NC(=O)C2=CCCCO2)CN(C(c2cc(=N)[nH]c(=N)[nH]2)=O)C1 c1(CN2C(C(N3CCC(SC)CC3)=O)CC(O)C2)nc(C)c(C)cc1Br N1(CCCN(C)CCO)CC2CN(C(c3cnn(C4CCC4)c3)=O)CC2C1 N1(C(C2C(CC(=O)OC)C2)=O)CC(NC(=O)CCSCc2ccccc2)C(O)C1 C1(NC(CS(=O)(=O)NCC)=O)CC2(CCN(C(=O)C(CC)N(C)C)C2)C1 C(C(CC(=O)NC1CCN(C(c2ccc3oncc3c2)=O)C1)C(F)(F)F)N(C)C c1(CC)ccc(C(C(=O)NCCCOC)N(C)CC2CCCCC2)o1 C=CCC(C(=O)NC(C)C)NC.C1(=O)C(C)N1C.C(C)(C)(C)OC(=O)N(C)C C1(N(C)C(C2COCCO2)=O)CCC(NC(c2sccc2C#N)=O)CC1 N1(C(c2ccc(=O)oc2)=O)CCC2CCN(C(n3nnc4ccccc34)=O)C2C1 N1(C(c2cc(C(=O)NCC)no2)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 c1(CC(=O)NCC(c2cccc(C)c2)OC)c(F)cccc1Cl C1(C(=O)NC2C3(CC(NC(C(CN(C)C)(C)C)=O)C3)C2)CCC(N=[N+]=[N-])CC1 C1(CNC(C2(C(C)NC(c3cnsn3)=O)CC2)=O)(CO)CCCC1 Cc1nc(O)ccc1C(=O)NC(C)CN(C)C(C1CCN(S(C)(=O)=O)C1)=O C1(CC(N2CC(NC(c3nc(C)oc3)=O)C(C)C2)=O)OCCCC1(C)C O=S(=O)(NCC(C1CC1)C1CC1)N1CCC(F)(F)C1.c1(C(C2CC2)N)ccccc1 C1(CN(C)C(c2cc(CCCO)on2)=O)CCCN1C(c1ccc(C(N)=O)[nH]1)=O c1(NC(C23C(CN(C(C4(Br)CC4)=O)C2)C3)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C2C(C)(C)COC2)=O)CC2(C=C(C(=O)NCCC34CCCC3C4)CO2)C1 C(=O)(CCCC(=O)NC1CC(F)(CNC(C2CCC3(CCC3)C2)=O)C1)N(C)C N1(C(c2cnc(C3CC3)nc2)C(=O)NC(CC)C)CC(N(C)C)C(C)C1 c12cc(ccn1)NC2=O.C12(CNC(CC3(OCC)CCC3)=O)CCCCC1C2 C1(C)(C(N2CCCC(CN(C(c3cc(C)on3)=O)C)C2)=O)COC(C)(C)CO1 Cc1ccc2nc(SCC(N3CC(CNC(=O)CC4CCCCO4)C3)=O)[nH]c2c1 C1(CNC(c2ccc(Cl)s2)=O)CCCN(c2ccnc(N3CCCC3)n2)C1 Cc1ncn(C)c1C(C(=O)NC1CCC1)N(Cc1nccs1)CC1CCCO1 C=CC1(C(N2CC(OC)CC2CNC(C2COCCO2)=O)=O)CCCCC1 Cc1cnc(N(C2CCCNCC2)C(c2ccc(CO)o2)=O)nc1 CCCCC(O)CC(=O)NCCC1(O)CCN(C(c2ncc([N+](=O)[O-])n2C)=O)C1 c1(C(=O)NCCN(C(c2cnoc2C2CCC2)=O)CC)ccnc(CO)c1 NS(=O)(=O)c1ccc(C(N2CCOCC2CC(=O)Nc2sncc2C#N)=O)c(Cl)c1 c1(CCC)cc(C(=O)NC2COCC2CNC(=O)C(C)(C)c2cscn2)no1 N(C1CCCOc2ccc(F)cc21)C1(c2n(CC)nnn2)CC2COCC2C1 C1(NC(c2cc(OC)nc(C)c2)=O)CN(C(C2(C)CCCS2)=O)CCC12CCC2 c1(C(CC)NC(=O)CC2CCN(c3cc(C(C)=O)cnn3)C2)ccc2c(c1)OCO2 CC1CC(C)(NC(=O)C=CCN(C)C(C2CNC(=O)N2)=O)C1 c1(OC)ccc(Cl)cc1C(=O)NCCC1CC(NC(C2CC23CCCOC3)=O)C1 C1(C2CCN(C(c3c(C)nc(C)o3)=O)C2)(NC(C2CC3CCC2O3)=O)CC1 C1(CC(=O)NC(C2CCN(CC3(C)CC4CC4C3)C2)(C)C)CCCC1C1CC1 c1(C(N(CCCNC(=O)C(C)C2CCOC2)CC)=O)scnc1Br c1(C(=O)NCC2N(C(C3C(C=C)CC3)=O)CC(O)C2)cc(Br)ccc1OC Cc1ccccc1CNC(c1nnnn1-c1cccc(Br)c1)CC1CCCCC1 N1(C(C23CC(OC(C)=O)(C2)C3)=O)CC2(CCC2)CC1C(N1CCn2ncnc2C1)=O C(=O)(CCC(CF)CF)N(CC(=O)NCCC1CCOCC1)CC#C C(=O)(CCCC(F)(F)F)Nc1c(CN2CC(C)(CC(=O)OC)C2)nc(Cl)cc1 CC(CC(=O)N1CC(C(c2cn(Cc3nocc3Cl)nn2)C)C1)c1ccccc1 c1(-c2nc(Cc3nc(C(CC)(O)CC)on3)on2)cn2ccsc2n1 c1(CN(CCC)Cc2cnc(-c3ccccn3)s2)cccnc1 c1(C(N(CCCN(C)C(C2CC3(C)CC2CO3)=O)C)=O)onc2ccccc12 C(=O)(C1=CC2C=CC1C2)NCC1(O)CC(C(N2CC(C3CC3)(OC)C2)=O)C1 C#CC1CN(C(=O)CSCC(=O)OC)CCN1C(c1ccc(OC)nc1)=O c1(C(N2CCC(C)C(NC(=O)CSc3cn[nH]c3)C2)=O)ccc2nccn2c1 c1(C(N(C(C(=O)NCCC(C)SC)=O)C)C)cc2ccccc2o1.N1CCOCC1 CC(C(CO)NC(=O)CCSCC(N)=O)NC(=O)CCCOc1cccnc1 N1(C(CN2C(=O)NC(C(C)C)C2=O)=O)CC2(C1)CN(Cc1ccccc1)CCO2 C1(CNC(C2(F)CC2(F)F)=O)CCCCN1C(CCNC(N)=O)=O c1(C(N2CCC(O)(CNC(CSC)=O)C2)=O)nc(C)ccc1F N1(C(CCC(C)c2ccccc2)=O)CC2(C1)CN(C(=O)C1=CCCOC1)C2 c1(C(N2CC(=C)C2)=O)oc(CNC(c2ccc(CC)s2)=O)cc1C N1(C(Cc2nc(C)sc2)=O)CCC(F)(CNC(=O)C(C(C)C)N(C2CC2)C(C)C)C1 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)Cn2cc(C)cn2)C(C(C)(C)C)C1 c1(NCc2c(C)nc(-c3ccccc3Cl)s2)nccc(=NC(C)C2CCOC2)[nH]1 N1(C(C(=O)NC2CC(N(C(c3ncc(OC)cn3)=O)C)C2)C)CCP(C)(=O)CC1 C(c1ccc(N(C)C)cc1)=CC(N1CC(O)(CN(C(c2scc(C)c2)=O)C)C1)=O C1(C)(NC(C(COCC)C)=O)CCN(C(C2CCCS2)=O)CC1 N1(C(CCC(C)=O)=O)CC2(CC(NC(C3CCCCN(C)C3=O)=O)CO2)C1 C1(NC(c2cc(COC)no2)=O)CN(C(=O)CC2CC3(CCC3)C2)C2CCCC12 C1(NC(C(CC)NC(c2ccccc2)=O)=O)CC2CCC1CN2 C1(C(CNC(COC(C)C)=O)C)CCN(C(=O)C(C2(O)CCCC2)F)CC1 C1(C(N2C(CNC(C3C(OCC)C3C)=O)CC2)=O)C2Cc3ccccc3C12 c1(C(=O)NCC(=O)NCC(=O)N(C(C)CO)C)ccc(C#N)o1 N1(Cc2cncc(CCC)c2)CC2CN(C)CC2C1 C(C1c2ccccc2CCN1C(C1(OC)CC1)=O)NC(C1CCC(CC)O1)=O c1(C(=O)NC2CC(C)CN(C(=O)C(F)CC3CCCC3)C2)ccc(N=[N+]=[N-])cc1 C1(O)(CC(N2CC3CC(O)C2C3)=O)CCN(Cc2cc(-c3cccs3)[nH]n2)CC1 Cc1nc(O)ccc1C(=O)NCC1CCN1C(C1(CO)CC1(F)F)=O C1(C(N2CCC(OCCNC(C3CCC(=O)O3)=O)CC2)=O)CCN2CCOCC12 C1(C(N2C(CC)CCC2)=O)CN(C(=O)CC(=O)O)CC1(F)F NS(=O)(=O)c1cc(C(=O)NC2CCC2NC(=O)C=CC2CCCC2)c(Cl)o1 N1(C(C(C)C2CCCC2)=O)CC(CC(N2CCC(C(C)(C)C)CC2)=O)C2(CC2)C1 Cn1cc(C(N2CCN(C(=O)C(C)(F)F)C3CCC23)=O)c2cccc(Cl)c12 C1(NC(c2ccc(CC)s2)=O)CCCC(NC(=O)C(C)(C)CN2CCCC2)CC1 C1(=CC(=O)NC2(C)CCN(C(C(Br)=C(C)C)=O)C2)CCCCCC1(F)F C(C(C(C)C)NC(=O)CC1CCN(C(=O)Cc2cc[nH]c2)C1)NC(C)=O N1(C(CC(CCC)C)=O)CCOC2(C1)CN(C(=O)C1=C(C)OCCS1)C2 C(=O)(C1Cc2ccccc21)NCCCN(C(c1c(C)nc2sc(C)cn12)=O)CC CC(C)C(O)C(=O)NC(C(=O)N1CCC(CN(C)C)C1)C(C)C C(=O)(C(C)CC(F)(F)F)NCC1(NC(C=Cc2c(C)n[nH]c2)=O)CCCC1 C1(CNC(C=CCCC)=O)CCC(C)CN1C(=O)C(C)=C1CC1 C1(CN(C(C2CC(=C)C2)=O)C)CCCC(NC(=O)CCCc2ccc(Cl)cc2)C1 N1(C(CCC=CC(C)C)=O)CC(F)(F)CC1CCNC(=O)C(F)C(C)(C)O n1(CC(=O)NC2CN(C(C34CC3C4)=O)CC2C2CC2)cnc2c1CCCC2 CC(O)(C(=O)NC1COCC1C(=O)NC1CCN(S(C)(=O)=O)C1)C(F)(F)F c1(CC(C)(C)C)nc2cc(NCC3(C)COCCO3)ccc2o1 c1(CCC(=O)NCC2CCN(C(C3CC34CC(F)(F)C4)=O)C2)ccc(F)c(F)c1 C1(C)(NC(C(CCC)O)=O)CCCN(C(=O)CCCOc2ccc(C)cc2)C1 C(=O)(C1CCCc2ncccc21)NC(C)CNC(=O)CCC(C)(C)F C1(=C(C(=O)OC(C)(C)C)F)CCN(C(C2CCC(C)CO2)=O)CC1.CC(=O)O Cc1nc(C)n(CC(=O)NCCC2(O)CCN(C(C3(C#N)CCCO3)=O)C2)n1 C12(NC(C3CC(=C)C3)=O)CCN(C(=O)Cc3cccc(OCCCC)c3)CC1C2 N1(C(c2c(C#C)cn(C)n2)=O)CC2=C(C1)CN(C(c1cc(Cl)cc(Cl)c1)=O)C2 c1(C(N(C2CCN(C(=O)Cc3sccc3C)CC2)CC#C)=O)ccc(C)cc1Cl c1(C(=O)NC2(C)CCC(NC(C(C=C=C)C)=O)CC2)cccc2cnsc12 C1(CNC(C2C(C(=O)OC)C2)=O)CC2(CCN(C(c3cccn3C)=O)C2)CO1 Cc1ccc([N+](=O)[O-])cc1C(=O)NCC(CO)NC(=O)C(C)SC(F)(F)F C(=O)(CC(C)C(F)(F)C(F)(F)F)NC1(CNC(CCC(C)OC)=O)CC1 c1(-c2ccc(C)o2)nn(C)cc1C(C)Sn1cc(CSC2CCCC(C)C2)nn1 N1(C(c2nccc(OC)c2)=O)CCCC(F)(CNC(=O)CCC(C)(C)F)C1 c1(-c2cn(CCCCNC(=O)C(C3CCOCC3)F)nn2)ccc2ncsc2c1 CC(CCCC(=O)NCCCCC1CC1C)NC(=O)Cc1cc[nH]c1 c1(C(=O)NCC(COC)NC(C2C(C)C2(F)F)=O)ccc(C)cc1 c1(OC)ccc(C=CC(=O)NCC2C(C)CCCN2C(=O)CC(C)(C)F)cc1 Cn1cnc2c(-c3nnc(N4CCc5ccccc54)o3)nc(Cl)nc12 C1(C)(NC(=O)NCc2cccc(NC(c3c(C)cccc3)=O)c2)CCC12CCC2 c1(CCC(N2C3C(NC(C=C(C)C)=O)C(C3)C2)=O)cc(Br)ccc1C C(=O)(CCC(C)(C)F)N(C1CCN(C(=O)C(c2ccc(OC)cc2C)C)C1)CC C1(C(C(N2CCCC2C2CC2)C(=O)NCC)OC)CCC(F)(F)CC1 C1(CC(C)CNC(=O)NC2COC2)CCC(F)(F)CC1 C=CC(CC)C(=O)NC1CC(CNC(C2(CCC)CCC2)=O)CC1O C(=O)(C(CCC1CC1)NC(C1C=CCS1)=O)NC1(C)CC(O)C1 Cc1cncnc1C(=O)NC1CCC1C(=O)NCC(C)(C)C(N)=O c1(NC(C(COC)NC(C)=O)=O)cc(C)n(C2CN(C(=O)C(C)(C)C)C2)c1C C1(N(C(C(=O)N(C)Cc2onc(C)n2)=O)C)CCN(C2CCCCC2)CC1 CC(CCC(C)(C)C)C(=O)NCCCN(CC(c1ccc(F)cc1Cl)O)C1CC1 Cc1c(C(=O)NCCC2CCCN(C(c3c[nH]nc3C(F)F)=O)C2)cncc1Cl CC1=C(CNC(c2cccc(C)c2)C(F)(F)F)C(C)(C)CCC1 C1(NC(c2nccn2-c2cccc(-c3nc[nH]n3)c2)=O)CCC(F)(F)CC1 c1(C(=O)NCc2scc(C)c2)cc(CNC(=O)C(C)(C)C2CCCC2)nn1C c1(-c2c(F)ccc(OC(C)C)c2)cccc2c(C(=O)NC3CC3C3CC3)c[nH]c12 N1(C(C2C(C=C)C2)=O)CCOCC1CCNC(c1ccccc1C(C)(F)F)=O c1(C(N2CCC(O)(CNC(C(CC)SC)=O)C2)=O)ccc2ncc(=O)[nH]c2c1 C1(CNC(C2(CCC)CCNC2=O)=O)CN(C)CCN1C(=O)Cc1nc[nH]n1 N1(C(c2c(CNC(C=CC(=O)N(C)C)=O)nnn2C)=O)CCCC(N=[N+]=[N-])C1 c1(CC(=O)NC(C(CO)NC(CCC=CC)=O)C)ccnc(C(N)=O)c1 N1(C(C2CCC(=C)CC2)=O)C2CCC1CN(C(C1CC1C1CCOCC1)=O)C2 CC1SCCC1N=c1nc(N2CCN(C(=O)C(N)=O)CC2)c2ncccc2[nH]1 c1(C(=O)OC)cc(C(=O)NCC(F)CNC(=O)CC2(C)CC2)cc([N+](=O)[O-])c1 C(CC(C(C)(C)C)NC(c1ccccc1Cl)=O)N(C(CCOC)=O)C C1(NC(C2=C(C)CCC2)=O)CCOC2(CCN(C(c3cc(CO)[nH]n3)=O)CC2)C1 N1(Cc2c(C)nc(C)s2)CCS(=O)(=O)C(CCNC(c2cc(C)n(C)n2)=O)C1 c1(NC(=O)NC2(C(F)(F)F)CC2)nccc(NC(CC(=O)O)c2ccncc2)n1 C1(C(C(=O)NCC2(CO)CCCC2)F)CCN(C(c2ccoc2)=O)C1 CC1CCCC(C)N1CCCCSC.N12CCC1(CC)CC2 c1(OC)cc2nc(NC3CCCN(Cc4cccs4)C3)nc(O)c2cc1OC CCC(CC(F)(F)F)NC(=O)CC(CNC(=O)Cc1cnoc1)C1CCC1 c1(C(=O)NCCC2CN(C(C(CC=C)(C)C)=O)CC2C)ccc2oc(=N)[nH]c2c1 c1(C(=O)NC2CC(NC(c3n(CC)nnc3)=O)C2)c(F)ccc(C#N)c1F c1(C2(C)COC2)cn(CCCC(=O)NC(C2CCC2)C2CC2)nn1 c1(C(N2CC(O)(CNC(c3ccc(OC)s3)=O)C2)=O)cnnc(C)c1 C1(CN(C)C(c2cncc(CN(C)C)c2)=O)COCCN1C(C1COCCN1C)=O C1(CNC(CCc2c(C)noc2Cl)=O)CN(C(=O)C(C)N(C)C)CC1(C)C c1(C(C(=O)NC(C)C(CO)NC(=O)CSCCN(C)C)OC)ccc(Cl)cc1 N1(C(C2C(CC)CN(C(c3ccc4cncn4c3)=O)C2)=O)CC2C=CCC(C2)C1 N1(C(c2c(CC(=O)OC)scc2)=O)CC2CCN(C(=O)CCC(C)N(C)C)C2C1 CCC(CCOC)C(=O)N(CC(N1CC2(CC2)C1)=O)C1CCC1 Cc1ccc(C(=O)NCc2cn(CCN3CCOCC3)nn2)c(Cl)c1 C1(NC(CCc2ccc(CC)cc2)=O)CCN(C(C2CC23CC3)=O)CC1F C12(C(=O)NCC3(F)CCN(C(=O)COc4ccsn4)CC3)CCCCN1CCC2 Cc1oc(C2CC2)nc1C(=O)NC1(CCO)CN(C(C2(F)CCOC2)=O)C1 N1(C(C(n2cc(Cl)cn2)C)=O)CC2CCCC(C1)N2C(=O)C(C#N)CC1CC1 C1(CCNC(C2CC(=O)OC2)=O)CN(C(C2(CF)CCOCC2)=O)CCO1 C1(NC(C2(C)CCCC2)=O)CCN(C(=O)Cc2cccc(N)c2N)CC1F CCC(CC(C)C)C(=O)N1CC(C(=O)NCC2CCC2CO)C(F)(F)C1 CCC(C)(CC)C(=O)N1CCOC(CNC(C2(C#N)CC3(CC3)C2)=O)C1 C(C(O)CS(=O)(=O)c1cccs1)NCC(c1c(F)cccc1F)C CCCCC(=O)C(=O)NC(C(=O)NCc1c(F)cccc1F)C1CCOC1 CC1CCC(=CC(=O)NCC2(CNc3cn(CC(=O)N(C)C)nn3)CC2)C1 Cc1cc(C(=O)NC2CC(NC(=O)CCOC3CC3)C(O)C2)ccc1O c1(SC)cc(O)ccc1NC(=O)CC1CCCN1C(=O)Cc1ccccc1O C(C)(C(C)C(=O)N1CC(OCCO)C1)NC(c1cc(OC)n[nH]1)=O C1(N(C)C)CCCC(C(=O)OCN2CCCC2NC(=O)C(c2ccccc2)F)C1 CCCC(C)C(=O)N1CC2C(N(C(=O)CCOC3CCCCC3)C)C2C1 C1(NC(C(N2C(CSC)CCCCC2)=O)=O)CC2(CCC2)C12CCC2 Cc1nc(N2CCCC(CNC(c3ccno3)=O)CC2)c(C)c(Cl)n1 C=CCCCCCCCC(=O)NC1CN(C(=O)Cn2ncn(C)c2=O)C(C)(C)C1 N1(C(C(c2ccc(F)cc2)=O)=O)CCCC2(NC(C3CCCCCC3)=O)CC2C1 N1(C(C=CC(C)NC(=O)C2=C(Cl)CCOC2)=O)C2CCCC1CN(C)C2 c12ccc(cc1)-c1n[nH]c(n1)C1CC21.C(c1cccnc1)=CCNC c1(-n2c(C(C)(C)CC#N)nc(CN3CCC(O)CC3)n2)ccc(F)cc1C(F)(F)F C=CCN(OC)C(=O)C(F)CC(C)(C)NC(c1ncccc1Cl)=O CCC(C)(COC)CNC(=O)CCCCNC(=O)C(C)NC(=O)OC C1(F)(C(=O)NCC(O)CC2CCCC2)CCCN(C(c2cc3n(n2)CCC3)=O)C1 N1(C(CC(C=C)CC)=O)CC(C)CN(C(c2cnn(CC(C)C)c2)=O)CC1C Cc1ccc2ncc(C(=O)NCCC3CN(C(c4ccnnc4O)=O)C3)cc2c1 CCCC(CNC(C1(C#N)CCC1)=O)C(=O)NC(C(C)C)C(C)C Cc1nn(C(C)C)cc1C(=O)NC1CC1NC(C1CC1C)=O c1(C(=O)NCCCC(C)(C)NC(C2CCCN(C)C2)=O)cc(N)c(F)c(F)c1Cl CC1C(NC(=O)C2=CCC2)CCN1C(c1cc(C2CC2)cs1)=O C1(NC(CC(CCC)C)=O)CC(C(=O)N(c2ccccn2)CC(C)C)=CC1O c1(C(C)O)cc2ccccc2[nH]1.C12(C)CN(C1)C(=O)C1CCN1C(=O)CC2 N1(c2ncnc(C)c2Br)CCC2CCC(C1)N2C(c1cn2c(n1)CCC2)=O C1(NC(c2cc(F)n[nH]2)=O)CN(C(=O)C(F)n2cccn2)CC1O c1(C(=O)OC)ccc(C(N2CCC(N(C(=O)C(C(C)(C)C)SC)C)C2)=O)cc1F c1(NC(N(CC(C)NC(=O)OC(C)(C)C)C)=O)ncccc1Cl C1(c2cn(C)nc2)CN(C(c2ccoc2)=O)CCN1C(c1cc(C(N)=O)co1)=O N1(C(CN(C(C)=O)C)=O)CCC(C2CC2)(NC(=O)CN2CCN(C3CC3)C2=O)C1 n1(CCCC)nc(C(N2CC(NC(C3CC(C)=NO3)=O)C3CC3C2)=O)ccc1=O N1(C(=O)NC2C(C(C)(C)C)C2)CCC2CC(O)CCC2C1 c1(C(C(=O)NCC=C)N(C)Cc2ccc(NC(C)=O)cc2)ccc(Cl)cn1 O=C(O)C1=CCC(NC(c2ccn(C3CC3(F)F)n2)=O)C1 C1(C(=O)NC(C=C)(C)CC)C2CC(O)C(C2)N1C(C1CC2CCCC2C1)=O C1(NC(c2cc(CC)no2)=O)CC(NC(C2(COC)CC(F)(F)C2)=O)C12CCC2 CC(c1cccc(Cl)c1)=CC(=O)NC1(C)CCN(C(=O)CS(N)(=O)=O)C1 C1(C(=O)NCC2(COC)CCC2)CN(C(c2c[nH]nc2C)=O)CCO1 C(CN=c1[nH]ncs1)OCCNC(CS(=O)(=O)NC)=O Cc1ccc(NC(=O)CC2CCCN2Cc2cnn(C)c2C)c(F)c1 N12CCC3(CC1)CC(C3)NC2=O.c1(Oc2cnoc2)ccccc1[N+](=O)[O-] CCCC(C)(C)CC(=O)N1CC(NC(=O)C(C2CCC2)C2CCC2)CCC(O)C1 C1(C(=O)NC2(CN(C)C(c3ccc(C(N)=O)cn3)=O)CC2)OCC2CCCC12 CC1=C(C(=O)NC2(C(N(CCC(C)N(C)C)C)=O)CCCCC2)CCC1 C=CCCCC(C(=O)NCC(C1CCCCC1)O)NC(C1CC(=O)N(C)C1)=O N1(C(CC2(OC)CCC2)=O)CCN(C(c2cc(C3CC3)ccn2)=O)C(CCO)C1 C1(O)(CC)CCCN(C(C2(CC)CCCN2C(C2CCCCCC2)=O)=O)C1 C(=O)(CCC=CBr)N(CC(C)NC(=O)Cn1ccc(C(F)F)n1)CC c1(C(=O)NCC(CO)NC(CNC(C)=O)=O)cc2c(ccn2C)s1 C1(NC(=O)NC2CCN(CP(C)(C)=O)C2)Oc2ccccc2NC1=O C1(C#N)(N(C(CCCC#C)=O)C(C)(C)C)CCN(C(c2cc(F)ccc2C)=O)C1 C=CC1(C2(C(=O)NC(C3CCN(C(c4c(C)cnn4C)=O)C3)C)CCC2)CCC1 CCCC(CCC)=CC(=O)NC1(CO)CCN(C(=O)C(C)(C)C2CCO2)C1 c1(CCC(=O)NC2(CF)CCN(C(CCC(C)C)=O)C2)nc2ccccc2[nH]1 c1(C(N2CC(CNC(=O)CN3CSCCSC3)C2)=O)cccc2occc12 C1(NC(CCCN(C(=O)CCC(F)(F)F)C)=O)CC2(C1)CC2(F)F N1(C(C(C)SC)=O)CCOC(CNC(=O)CC(c2c(C)n[nH]c2C)C)C1 c1(-c2cn(CC3CN(C(CN(C)C(N)=O)=O)C3)nn2)ccn(C)c(=O)c1 c1cc2c(NC3C4CCCCCC34)[nH]c(=NCCn3cncn3)nc2s1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC2(CNC(C2(C(N)=O)CC2)=O)C1 C(CCCCCC(=O)NC(c1ccccn1)CO)NC(c1ccc(SC)o1)=O c1(C(=O)NCC2(F)CC(NC(CC(C)C)=O)C2)cccc(C(C)C)c1F C(=O)(C(C)(C)CCS(C)(=O)=O)N(CCCN(C(C(=C(C)C1CC1)F)=O)C)C c1(OC)ccc(C(C)=CC(=O)NC2CCC(C)(NC(c3cnsn3)=O)CC2)cc1 CN(CC(O)CN1CCCC1)N1CC2CN(CC(F)(F)F)C2C1 N(C1CCCc2occc21)C(C1(n2cnnn2)CCOCC1)=O C(=O)(C(F)(F)CCC1CCC1)NCCN(C(C(c1ccccc1)OC)=O)C1CC1 c1(C(N2C(C)C(C(=O)NCC(C)(O)CCO)CCC2)=O)ccc2ccoc2c1 n1(NC2CC(C)(COCC3N(CC)CCCC3)C2)ncc(O)nc1=O c1(C(C(=O)NC(CNC(C2(CC(=O)OC)CC2)=O)CO)C)ccc(Br)s1 c1(CC(N2CC(N(C(C(CC)N(C)C)=O)C)C2)=O)nnc(O)c2ccccc12 CC(=NOCC#N)C(=O)N1CC(CNC(C2NC(=O)OC2C)=O)CC1C C1(OC)(CNC(c2ccnc(C3CC3)c2)=O)CCN(C(c2cnc(Cl)s2)=O)C1 C1(CNC(=O)CC2(O)CCC2)CC2(CCN(C(c3csc([N+](=O)[O-])c3)=O)C2)CO1 C(=O)(C(C)(F)C(F)(F)F)NCC1(O)CCCN(C(c2c(CC)ccs2)=O)C1 C12(C(N3CC(NC(c4scc(C)n4)C)OCC3)=O)CCC(CC1F)C2 N1(C(c2cc(Br)ccc2C)C(=O)NCCOC)CCC(F)(F)CC1C C#CCC(CC(=O)NCCCCCCCOC)NC(c1ccsc1Cl)=O C(=O)(C#CC1CCCO1)N1CC(O)CC(NC(c2cc(=O)cc[nH]2)=O)C1 Cc1nc(O)ccc1C(=O)NCC(CNC(c1ccc(C(C)C)c(F)c1)=O)CO c1(C(=O)NCC2CC(C(N3CC(COC)OCC3)=O)C2)ccc(C)c(C)n1 C1(C)(C(=O)NCCCCC(C)NC(c2c(C)nccc2)=O)CCC(=O)NC1 C1(CN(C(c2c(OC)ccs2)=O)C)CCCC(NC(=O)CCc2cnco2)C1 C1(C(C)NC(c2nocc2Cl)=O)CCCCN1C(=O)C(=O)N(CCC(N)=O)C1CC1 CC1(C)CCC(CNC(=O)CC2CCCCN2C(=O)COC2CCOC2)CC1 c1(CC(C)C)n[nH]c(=NCCC2CCN(C(=O)CCc3cc(F)ccc3F)C2)s1 C1(NC(CCc2n(C)ncc2)=O)CCN(C(c2ccoc2Br)=O)C12CC2 C(CC(C)C(=O)NCC1CC(O)CN1C(c1[nH]c(O)nc1C)=O)=CC C(=O)(C(C)C(C)NC(=O)OC(C)(C)C)OCCC(=O)NCCO.C(CC(C)C)=CC c1(NCc2n(C)c(-c3nn[nH]n3)cc2)cc(Cl)ccc1OCC(F)F c1(CC(=O)N(CCCNC(C(CCC)O)=O)CCO)ccc(OC)cc1Br CC(C)(C)CC(O)CC(=O)NC1CC(C)(NC(=O)COCc2nccs2)C1 C12(NC(c3ccc(C)s3)=O)CCC(CN(C(c3csc(C)c3C)=O)C1)C2 CC1CN(C(=O)Cc2ccon2)CCC1NC(c1cc(Cl)ccc1C(F)(F)F)=O C1(OC)CCCC(CC(=O)NCC(C)CNC(c2ccc(C3CC3)cc2)=O)C1 N1(C(C(CCCC)NC(N)=O)=O)CC2=C(C1)CN(C(=O)C=CBr)C2 c1(C(=O)NC2C(NC(c3c(C)nsc3)=O)CC2)cccc(-c2nnco2)c1 C(C(C(=O)NCC1CC1[N+](=O)[O-])NC(=O)CCOCC1CC1)N(C)C C1(C(=O)NCC2N(C(c3ncc(C(=O)OC)nc3)=O)CCC2)C(F)(F)C12CCC2 C12(C(=O)NCc3c(CC)nns3)CCCC1CN(C(=O)C(C)(C)C#N)C2 c1(OC)cc(Br)ccc1CC(=O)NC1C=CC(C(=O)Nc2ccc(Cl)cc2O)C1 C1(F)(CNC(=O)C=CC(=O)NC2CC2)COCCN(C(C2COC(=O)C2)=O)C1 c1(CC)cncc(-c2nc(CCCSC)n[nH]2)n1.c1(C2CC2)ccccc1 C12(NC(CCCN(C)C)=O)CC(CNC(=O)C(F)OC(F)(F)F)(C1)OC2(C)C C1(CNC(=O)CC2COCCO2)CC2CCC1N(C(c1ncnc(O)c1Cl)=O)C2 C1(NC(C(C)(C)OCC)=O)CC(CN(C)C)CC1O.c12conc1C(=O)NC2 c1(C(=O)OC)ccc(OC(c2c(C)nn(CC(C)C)c2Cl)=O)c(Br)c1 Cc1coc(C(F)(F)F)c1C(=O)NCC(CC(C)C)NC(=O)CN1CCOCC1 Cc1nn(C)c(C)c1CC(=O)NCC1(C)CCC(NC(=O)C(O)C2CCC2)CC1 N1(C(C2C(CC(C)C)C2)=O)CC(NC(c2coc(CS(C)(=O)=O)n2)=O)CC(F)C1 c1(C(=O)NC(C2CCN(C(C3CCCC3O)=O)CC2)C)snc2ccccc12 C(C1=NOC2CN(C(c3nnc(O)nc3O)=O)CC12)NC(C1(SC)CC1)=O c1(COC(C2(c3ccc(Cl)cc3)CCCC2)=O)c(F)ccc(F)c1F Cc1c(NC(c2c[nH]nc2CCNC(=O)C(C(C)O)N(C)C)=O)cnn1C c1(CC(N2CCC(NC(C(CC)C3CCOCC3)=O)(CF)C2)=O)c(F)cccc1Cl C1(C(=O)OC(CCC)CC)CCC(F)(C(=O)OC(C)(C)C)C1 C1(CC(C)NC(=O)CC2CC2(C)C)CCN(C(C2CC(N(C)C)C2)=O)CC1 C1(C(=O)NC(C(=O)NC)C2CC2)COC2(C1)CN(C(=O)C1=CCCSC1)C2 c1(NCC2N(C(=O)C=CI)CCC2)ccnc2ncnn12 N1(C(COC2(C)CCC2)=O)CCC(CCNC(C2OCC2(C)C)=O)CC1 C1(NC(c2nncc(C)c2)=O)CCC2CN(C(=O)CCc3cnn[nH]3)CC2C1 C1(C(=O)NCC2(CNC(c3ccc(C#C)o3)=O)CCOCC2)CC(=O)NC1(C)C N1(C(CNS(C)(=O)=O)=O)CCC(N2CCC(NC(=O)CCC(F)F)CC2)CC1 N1(CC(=O)N(C2CCC(NC(C3(CC)CC3)=O)C2)C)CCC(=O)NC1=O C(=O)(C1=C(C)CCCC1(C)C)N(CC(C)NC(C1CCCCC1SCC)=O)CC C1(CNC(CC(C)(C)OC)=O)CN(C(c2ccc(C)nc2O)=O)C2CCN1C2 c1(C(N2CCC(NC(C#CC(C)C)=O)C(O)C2)=O)ccc2c(=O)n(C)cnc2c1 C1(CC(=O)OCC)CCC(NC(C)=O)C1.n12nnnc1C1(CCC1)NCC2 C1(C)(C(N(CC(C)NC(C(CC)(C)F)=O)C)=O)CC2CCC1CC21OCCO1 C1(C(=O)NCCCN(C(=O)Cc2ccoc2)C)CC(c2cccc(Cl)c2F)=NO1 C1(C)(CNC(COCC)=O)CC(F)(F)CN1C(C1CCc2n[nH]cc2C1)=O c1(C(=O)NC2(C)CCCN(C(CNC(CC)=O)=O)C2)ccc(S(=O)(=O)CC)cc1 c1(C(N2CCC(C)(C(=O)OCC)C2)C(=O)NC(C)(C)CC)cc(Br)ccc1C c1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)O3)=O)C2)cc2ccccc2cn1 Cc1cccn2cc(C(N3CCC(C(C)NC(=O)C(F)n4ccnc4)C3)=O)nc12 C(=O)(CC(C)(C)C#N)N1CCC(C(C)(C)CN(C(=O)C(F)OC(F)(F)F)CC)CC1 Cc1cc(C(=O)N(C2CC2)CC2CCCN2C(c2ccc(C(C)C)o2)=O)nc(C)n1 c1(C(=O)NC2C=CCN(C(=O)CC3CCSC3)C2)occ2c1CCC2 c1(N(C(c2ncsc2Br)C(=O)NC)C)ccc(NC(=O)OC(C)(C)C)cc1 c1(C(C(=O)N(C)CC2CN(C(=O)CC3CSCCS3)C2)O)cc(F)cc(F)c1 Cc1c(C(=O)NC2CN(C(=O)CC3C=CCC3)CC2C)ncn1C N1(C(C2N(CC)CC2)=O)CC(CNC(=O)CC2CCC(C)(C)O2)C(C)C1 CCC(C)C(O)C(=O)NCC(CNC(C1CC=CC1)=O)S(C)(=O)=O c1(NC(=O)CCc2cccnc2)cnc(SCC)nc1.CC1CCC1N(C(=O)C)C c1(C(=O)NC2CCC(CNC(c3cc(Cl)c(Cl)[nH]3)=O)CC2)ccc2cccnn12 CS(=O)c1cccc(C(N2CC=C(CNC(C3(Br)CC34CCC4)=O)CC2)=O)c1 C1(CC)CCN(C(=O)CC(C)C2CC2)C(C(=O)NC2CC(CCF)C2)C1 C1(CNC(c2ccn(CC)c2C)=O)CN(C(=O)CNC(=O)C(C)(C)C)CCC1C c1(CNC(CCCCC#C)=O)nnc2n1CCN(C(=O)C(O)CCCC)C2 C1(C(N(C2CCN(C(=O)CCc3nc(C)no3)C2)CCC)=O)CCCC1C(C)C c1(C(N(CCCCNC(C2CCCCC2(C)C)=O)C)=O)c(F)ccc(O)c1F N1(C(C(C)NC(C)(C)C)=O)CCN(C(c2ccn(CC(F)F)n2)=O)CC1CO c1(C(=O)NCCC2CCCN(C(C(C)CN(C)C)=O)C2)cn(C)c(=O)n(C)c1=O N1(C(=O)CCN(CCO)Cc2ccccc2Br)CC2CNCC2(CO)C1 C#Cc1cn(C)nc1C(=O)N(C1CCCC(NC(c2cncs2)=O)C1)C CC(C)(C)C(O)CONC(=O)COC1CCN(C(c2ncc(F)cn2)=O)C1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C(C)NC(c2ccccc2F)=O)OCC1 N1(C(CC(CC=C)NC(c2ncc(F)cc2N)=O)=O)CCOCCCC1C C1(NC(c2nnc(CC)s2)=O)CCCN(C(=O)CCc2cc(C)[nH]n2)CC1 C1(NC(CN(C2CCC2)C)=O)CCOCC1NC(=O)CCn1cnccc1=O c1(Cn2ncc(C(=O)OCC)c2)nc(C)c(C(N2CC(F)CC2C(F)(F)F)=O)s1 c1(OCC)ncccc1C(=O)NC1CCCC(C(=O)NOCCCF)C1 C1(N(C(CCOCCOC)=O)Cc2cccnc2)CC(C#N)C1.C1(=O)CN1 C1(C(N2C(C)(C(C)C)CC2)=O)CCCCN(C(=O)C(C)S(C)(=O)=O)C1 N1(C(C(CCC#C)O)=O)C2CCCC1CN(C(C1(Cc3ccccc3)CC1)=O)C2 c1(C(=O)NCC(CNC(c2cc(C)[nH]n2)=O)(C)C)ccc2c(n1)CCC(C)(C)C2 c1(C(=O)Nc2cc(-c3ccc(C(F)(F)F)cc3)cs2)cncc2cnccc12 c1(CC)ncccc1C(=O)NC1CCCC1C(=O)NC(C(N)=O)C1CCCC1 c1(CN(C(=O)CC2(C(N(C3CCOCC3)C)=O)CC2)C)cccc(CO)c1 N1(C(c2cn(CC=C)nn2)=O)CCC(O)(CCNC(C2C=CCCC2)=O)C1 C1(C2CCN(C(=O)C(O)C3CCC3)CC2)(NC(=O)CNc2ccccc2Cl)CC1 C=CCC(CC(=O)N1CC2CC2C2CC12)NC(=O)COC1CCCC1 C=CCC(C(=O)N1CC(NC(c2ccc(N(C)C)cc2C)=O)C(O)C1)C(C)(C)C c1(CN(CCC#N)C)ccccc1.C12CN(C1)OC(=O)C2 N1(C(C(CC=CCC)C)=O)CCC2CN(C(=O)C(=CC3CCCC3)C)CC2CC1 c1(C(=O)OC)cccc(CSCCC2CCOC2)c1O C(CCCCC(=O)NC1(C(=O)NCCc2csnn2)CC1(C)C)OCC Cc1nc(C2CC2)ccc1C(N1CCOCC1CN(C(=O)Cc1nc[nH]n1)C)=O c1(C(=O)NC(C(N2CC3COCC3C2)=O)C2(C)CC2)c[nH]c2nccc-2c1 CC1(C(N2CCC(C)(NC(=O)CC3COC(=O)C3)C2)=O)CNC(=O)C1 c1(NC(c2ccoc2)C)nccc(NC(CCO)c2nccs2)n1 C1(NC(c2nnn(C)c2N)=O)C2CC1CN(C(=O)Cc1cc(F)ccc1Br)C2 C1(NC(c2ccc(C)c(O)n2)=O)CC2CC(C1)N(C(C1C=CCS1)=O)C2 c1(N(CC(C)NC(c2coc(C(F)F)c2)=O)C)ncnc2c1ncn2CC1CC1 C1(CC)CN(C(=O)CNC(C2CCCN2C(C)=O)=O)CCN1C(=O)CCC(C)C c1(OC)ccccc1C1(C(=O)NC2CCC(NC(=O)CSC)CC2)CCCC1 Cc1cccc(C(=O)NC2CN(C(=O)CC3SC(=N)NC3=O)CC2O)c1Cl C(CN=c1[nH]c(=N)[nH]c(=NCC(C)c2nccs2)[nH]1)NC(=O)OCC Cn1cc(C(=O)NCCNC(C2CCCC3(C2)CC3(F)F)=O)c(=O)n(C)c1=O C1(C(=O)NC2(C)CCCN(C(=O)COCCF)C2)OCC2CCCC1C2 c1(C(=O)NC2CN(C(CCN(CCCCC)CCC)=O)C2)nc(O)nc(O)c1F CC1(C)CCCN(c2nnnn2C2(c3ccccc3Br)CCC2)C1C(N)=O C1(C(=O)NCCCN(C(=O)Cn2cnnc2O)C2CC2)CN2CC3CC2(CO1)C3 C(CC#CCO)NC(C(N(C(=O)C(C)(C)C1CC1)C)C1CC1)=O Cc1cc(C(=O)NC2CC3(C2)CC(NC(c2cccn(C)c2=O)=O)C3)cc(O)n1 N1(C(C2(CNC(=O)Cn3ccnn3)CC2)=O)CCCC2(COC2)C1 Cn1nc(C(=O)NCC2CC23CCN(C(=O)CNC(N)=O)CC3)c2c1CCC2 N1(C(C(C(C)C)NC(Cc2c(C)n[nH]c2C)=O)=O)CC2CCCCC2C1 S(=O)(=O)(c1ccc(F)cc1F)N(C)CCNC1CCC1(F)F c1(C(=O)NCCC2(NC(C(C3CCCCC3)OC)=O)CC2)ccc([N+](=O)[O-])cc1 N1(C(c2nnc(-c3cccc(F)c3F)o2)=O)CCCc2cncc(Cl)c21 N1(C(c2sc(C)c(O)n2)=O)CCCC2C(NC(=O)CCC(C)(C)F)C(C)(C)C12 CC1(C)CC1(C)C(=O)NCC1(CNC(c2cc(Br)n[nH]2)=O)CCC1 c12ccc(s1)S(=O)(=O)NC2.C1(NC(c2cccs2)C)CN2CCC1(F)CC2 N1(C(C(n2cc(Cc3ccccc3F)nn2)C)=O)CCC(C(=O)O)CC1(C)C C(=O)(C(O)C(C)(C)C)NCc1cn(CC(=O)NCC(C)CC2CC2)nn1 c1(OC)nccc(Br)c1C(=O)NC1(CO)CN(C(c2cncc(C3CC3)c2)=O)C1 C#CCC(C)(C(=O)NCCOCC(F)(F)F)N(C(=O)C(C)C1CC1)C1CC1 Cc1nn(C)c(C)c1COC(=O)C(O)Cn1cncn1 c1(Cn2c(C)cc(C)n2)c(Cl)cccc1Cl.c12cn(nn1)C(C)C(=O)N(C)C2 Nc1nc(Cl)ccc1C(N1CC2CC1C2NC(c1ccc(Br)o1)=O)=O Cc1ccc(C(=O)NC2CCCCC2NC2CN(c3ncncc3F)C2)nc1O C1(CNC(=O)C=C2CCC2)CC(C(F)(F)F)CCN1C(C1CC2(CCC2)CO1)=O CC1CN(C(=O)CC2CCCC2NC(c2ccncn2)=O)CC(C)(C)O1 c1(C(=O)NC(C2(O)CN(C(C(C)c3cc[nH]n3)=O)C2)C)cn2c(n1)COCC2 N1(C(C(C)OCCC=C)=O)CCCC1CNC(C1CCC(F)C1)=O C1(C(=O)NCCCN(C(=O)CSCC(C)C)CC)C2CCCOC12.CCOC C1(C(=O)Nc2c(C)cccn2)CN(C(c2cc(F)c(F)cc2I)=O)CCC1(F)F C(=O)(C1CCCc2sccc21)NCCN1CCN(C(C2C(C)C2C)=O)CC1 Cc1cc2c(o1)CC(C)(C)CC2NCCNS(=O)(=O)CC1(CC#N)CC1 CCCC(O)(CN1CCC(C(CO)CO)C1)C(F)(F)F CC(C)C(F)C(=O)N1CCC(NC(=O)C(c2ccc(F)cn2)(F)F)C1C n1(CC)nc(C(=O)NC2CCCCC2CC(=O)NCc2cc(C)nn2C)cc1O C1(NC(c2ncc(OC(C)C)nc2)=O)CCN(C(=O)CC#N)C(C2CC2)C1 C1(C(=O)NC(C)CN(c2cc(Cl)nc(C3(C)CC3)n2)C)CNC(=O)CC1C N1(CC(=O)NCC2CC(NC(C3(COC)CCC3)=O)C2)CCCNC1=O C1(NC(C2C(NC(Cn3c(C)nc(C)n3)=O)CCOC2)=O)CC2(C1)CN(C)C2 C(=O)(CC(C)C(F)(F)F)NCCC1CC(OC)CN1C(c1cnc(C)s1)=O CC(CC(F)(F)F)C(=O)NCCC(O)CNC(=O)C(F)(F)C(C)(C)O Cc1c(C(=O)NCC23CCC(CC2)N3C(=O)C(O)C2CC2)c(C(F)(F)F)nn1C Cc1nc(Cl)ccc1CCC(N1CCC(C(C)NC(C2(O)CC2)=O)CC1)=O c1(CC)cc(C(=O)NCc2csc(CNC(C3CCC(OC)C3)=O)n2)nn1C N1(C(c2c(CC)cco2)=O)CCC2(CC1)CC2NC(=O)CN1CC=CC1 C12CCN(CC1CC)C2=O.c1(NC(C(CC=CC)C)=O)c(CO)cccc1C N1(C(CC2(C)CC2(F)F)=O)CCCC(N(C(=O)CN2CCCCC2)CCO)CC1 c1(NC(C)(C)CC(=O)N2CCCCC2)ccc(S(C)(=O)=O)cn1 C(=O)(C1=CC(O)C(NC(=O)CNC(=O)CNC(C)=O)C1)NCCS(CC)=O C=CC1CCN(C(=O)C(C2(O)CCCCC2)NC(c2cc(C)oc2CC)=O)C1 c1(OC)ccc([N+](=O)[O-])c(C(N2CCC(NC(c3cnns3)=O)C(CO)C2)=O)c1 C12(C(N3CCC(CNC(CC(C=C)(C)C)=O)C3)=O)CCC(CC1)C2(C)C C(=O)(CC(C)CC(C)(C)C)NCCC(C)N(C(c1ccc(C#C)cc1)=O)C C1(NC(C2(CC(=O)OC)CC2)=O)(COC)CCN(C(C2(F)CCCCC2)=O)CC1 CCCCCC(CC)C(=O)N1CCCC(NC(C2CN3CCC2CC3)=O)CC1CC C12(CNC(c3ccncn3)=O)CCCCC1N(C(c1ccc(F)nc1)=O)CC2 C#CCCCC(C)C(=O)NC(C1CCCC1)CNC(=O)C=Cc1cncn1C C1(C(=O)NOC2CCOC2)CCN(C(=O)c2cnc(S)nc2)O1 c1(CNC(C(C)C)=O)nnc2n1CCN(C(=O)Cc1ccc(Br)cc1)C2 c1(C(=O)NCC2(NC(C3CCCN3C3CCCC3)=O)CC2)ccncc1Br c1(NC(C2CN(Cc3cc(B(O)O)co3)C2)=O)nc2cc(Cl)ccc2s1 C=CC(C)(O)CC(=O)N1CC(N(C(=O)CS(=O)(=O)N2CCCCC2)C)C(O)C1 Cc1cc(-c2cn(CCC(=O)NCC3OC(=O)NC3(C)C)nn2)cc(C)n1 C12(CC)CCC(C(N3CCC(CNC(c4ccncc4F)=O)(OC)C3)=O)(CO1)C2 C#Cc1ccc(NC(=O)Nc2n[nH]cc2C(=O)NC2CC2)cc1 C(=O)(C(F)(F)C(F)(F)F)NCC1CCCC(NC(c2ccc(N(C)C)cn2)=O)C1 c1(OCCC)ccccc1CN1CC2C(C1)N2C(C1CCC(F)(F)C1)=O C1(C(=O)NCC(C)(C)n2ccnc2)CC2(CC2)CN1C(C1CC2(CC2)C1)=O C(=O)(C(F)CCC(C)C)N1C(CN(C(c2cc(C)cc(C)c2)=O)C)CC(F)C1 c1(C(=O)NC(C)CN(C)C(C2(C#N)CC2)=O)ccc(Cl)c(Br)c1F C1(C(=O)NCC(CC)NC(c2cc(C)c(C)o2)=O)CCCN(S(N)(=O)=O)C1 CC1(CCNC(c2ccns2)=O)CCN(C(C2CCC(=O)N2C2CC2)=O)CC1 N1(C(C=CCC)=O)CCCCCC1CNC(c1c(Cl)cncc1Br)=O C1(NC(C)=O)COCCC1NC(c1ccc(-c2ccccn2)nc1)=O C1(NC(COCc2ccc(C)s2)=O)CCOCC1NC(=O)Cc1cncnc1O C1(N(C(CN(C)C)=O)CC2CC2)CCN(C(=O)C(COC(C)(C)C)N(C)C)C1 C#Cc1cccc(CCCC(=O)NCCNC(C2CC3(C)CC2CO3)=O)c1 N1(C(C=CCOC)=O)CCN(C(c2csc(Br)n2)=O)C(C(C)C)C1 Cc1cnc(Cl)cc1NC(C1(C)CCN(C(c2ccc(F)c(O)c2)=O)CC1)=O CC(CC(C)(C)O)N1CCC(CNC(C2(c3ccc(F)cc3)CCCC2)=O)C1 C(CCCC(=O)N1CCC(O)C1C(C)(C)C)NC(C(C)SC(C)C)=O C=CCCCCN=c1nc2ncn(CC)c2c(NCC(C)C(=O)N(C)C)[nH]1 Cc1cc(C(=O)NC2(CNC(=O)CNC(=O)CC(F)(F)F)CC2)nc(O)n1 c1(C(=O)NCC2(NC(C(CCOC)C)=O)CCC2)ccc2[nH]c(=N)oc2c1 N1(C(C2CCCC(C)CC2)=O)CCCN(C(c2ncccc2N)=O)CCC1 C(=O)(C1=CCCCCC1)NCC1N(C(C2CC(C)OC(C)C2)=O)CC=C1 N1(C(C2C(CNC(C(C(C)C)OC)=O)CCC2)=O)CCC2(CC1)CN(C)C2 C=CC(CCC)CC(=O)N1CCOC(CCNC(c2ccc3c(c2)COC3)=O)C1 c1(C(=O)NC2CC3CN(C(C(CC)C#N)=O)CC(C2)C3)cnc(O)c([N+](=O)[O-])c1 CC(F)CN=c1nc2c(cnn2C)c(NCC2CCCC2N2CCCS2(=O)=O)[nH]1 C1(CC)CN(C)CCCN1C(C1CC(O)CN1C(=O)C(Cl)Cl)=O C=CC1CCN(C(=O)CC2CC3(C2)CN(C(c2cc(C)ccc2OC)=O)C3)CC1 CCC(CNC(=O)C(n1nccc1C)C)(CC)NC(c1n[nH]c(C)c1Br)=O C1(OC)CCC(n2nc(-c3ccncc3)nc2C(C)OCc2ccccc2)CC1 C1(CNC(=O)NCCCc2[nH]nc(C(C)C)n2)CC12CCOc1ccccc12 C(C(=O)NC1CCC1NC(c1c[nH]cc1Br)=O)(C(C)C)SC c1(CC(C)NC(Cc2c(OC)ccnc2)=O)cc(C)ccc1C C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(=O)C(CO)OC)C12CCC2 CC(C)(C)C#CCCNC(=O)C(CNC(c1cc(F)c[nH]1)=O)CC1CC1 N1(C(C2C(NC(c3c(CC)onc3C)=O)CCOC2)=O)C2CCC1CC(OC)C2 c1(C(=O)NCC(N2CCN(C(C3CCCCS3)=O)CC2)C)cc(O)ccc1F C12(CNC(CCCCSC)=O)CCC(C1)N(C(=O)Cc1cc(F)ccc1F)C2 c1(C(N2CCC(C)C2CNC(c2nocc2Br)=O)=O)cc(F)ccc1O c1(C(=O)NC2CC(C)N(C(c3csc(=N)[nH]3)=O)C2)cccc([N+](=O)[O-])c1 c1(C(N(C(C)CO)C(C)C)=O)c[nH]c2ccc(-c3cccc(N(C)C)c3)cc12 n1(CC)nc(C)c([N+](=O)[O-])c1NC1CC(CCNC(=O)Cn2ncc(Cl)c2C)C1 c1(-c2cncc(CNC(CS(CC)(=O)=O)=O)c2)cc(F)c(C#N)c(F)c1 C1(n2cccn2)(C(=O)NC(C(=O)NCC)C)CCN(C(=O)CCCCCF)CC1 C(=O)(C=C1SCC(=O)N1C)N1CCCC(CCC)(NC(c2nc(Cl)oc2C)=O)C1 CC(C(=O)NCC1CN(C(=O)C(C)(C)n2cccn2)C1)C(F)(F)F c1(OC)c(CC(=O)NC2(O)CCCC(C)C2)cc(Cl)cc1Cl c1(C(=O)NC(C(CCC)C)C)coc2c1CN(C(=O)C(=O)NCC(F)F)C2 N1(C(c2c(C)cc(=O)n(C)n2)=O)CCCC2CN(C(=O)C=CC3CCC3)CCC12 c1(C(=O)Nc2cccc(CNC(CC(=C)C)=O)c2)cc2c(ncn2C)[nH]1 C1(C)(CNC(CCSC)=O)COCCN(C(c2c(C)noc2C2CC2)=O)C1 C(CC(F)(F)F)N(C(c1cn(CCO)nn1)=O)CC1CCCN1 c1(OC)cncc(-c2nc(CCOC(C)C)nn2CCn2cc(Br)cn2)n1 c1(OCC(=O)NCC2CC(NC(c3c(C)nsc3)=O)C2)cccc(Cl)c1 C1(NC(c2cc(C)nnc2O)=O)CCCCN(C(=O)C(C)(Cl)Cl)CC1 N1(C(CC2CCCN(C(C(C)CC3CCC3)=O)CC2)=O)CC2(CCCCC2)C1 C1(C(N2CC(C(N)=O)(CNC(C3(C)CCCCC3)=O)C2)=O)Cc2ccccc2O1 C1(NC(C2CCCN2C(=O)C2CC2)=O)CCOC12CCN(C(=O)CCC(F)F)CC2 c1(C(N(CCCCCNC(=O)CC2CCCO2)C)=O)nn(C)cc1Br c1(C(N(CCCN(C)C(C2(N(C)C)CC2)=O)C)=O)cc(O)cc(Cl)c1 CCCCC(CNC(c1occc1Cl)=O)NC(C1CCC(C)(C)C1)=O n1(CC)nc(C(=O)N(C)Cc2ccccc2CNC(=O)CS(=O)(=O)NC)c(C)n1 C(=O)(C(C1=CCC2CC2C1)NC(=O)N)OC.c1(C(C2CCC2)C)ccccc1Cl CCCC(CNC(=O)CCOC(C)C)NC(c1cc(=N)[nH][nH]1)=O CCC(CC(=O)N1CC(CC(C)NC(c2sccc2S(N)(=O)=O)=O)C1)C(F)F c1(OC)ccc(N)c(C(N2CC(C3(NC(c4ccc(Cl)[nH]4)=O)CC3)C2)=O)c1 c1(C(=O)OC)sccc1C(=O)NCC1(O)CN(C(C2(CN(C)C)CC2)=O)C1 C(C(C(=O)N1CCCC1CCCNC(c1cn(CCO)nn1)=O)NC(C)=O)OC N1(C(=O)NCC(C2CCC(F)(F)CC2)CO)CC2(CO)CC1CC2O C1(C(=O)NC2C(C)OCC2)CCC2CN(C(=O)C(C)(C)C)CC2O1 CC1(C)CN(C(=O)C(c2ccoc2)NC(c2ncc[nH]2)=O)C2CCCC12 Cc1cc(F)cnc1C(=O)NCCCCC(C)NC(C1CC2(CCC2O)C1)=O c1(C(N2CCCC(CNC(C(C3CCCC3)OCC)=O)C2)C)ccc(C#N)cc1 C1(N(C(=O)Cn2cc(CO)nn2)C)CCC(NC(c2cnc(OC)nc2)=O)CC1 c1(C(=O)NCC2CC(NC(CCC(C)(C)C)=O)C23CCC3)scc2c1CCCC2 CC1(C)CC(NC(C2CN(C(=O)CC3OCCCO3)CC2C2CC2)=O)C(C)(C)O1 C(=O)(C1CCCn2cncc21)NCC(CCCC)NC(=O)CCOC C1(C(=O)NCCCCC2CN(C(c3cc(C)no3)=O)C2)CCCCC12CCC2 N1(c2cc(C)[nH]n2)CCN(C(C2CCCC(NCc3ccoc3)C2)=O)CC1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CC2CC(C1)CN(C(C1CCC3CCC13)=O)C2 C1(CC(=O)NCC(CN(C(=O)C(C)(O)C2CC2)C)(C)C)CCCC(F)(F)C1 C1(CNC(=O)COc2ccccc2[N+](=O)[O-])CCC2(CCC2)C1NC(=O)C1CC1 Cc1cc(N2Cc3c[nH]nc3C2)nc(N2CCCC(n3ccnn3)CC2)n1 Cc1ccc(Cl)c(OCC(=O)NCC2(F)CC(NC(=O)C(=O)N(C)C)C2)c1 C12(CNC(C(C=CCCC)O)=O)CC1CN(C(c1cnn(CC)c1Cl)=O)C2 C1(C(=O)NCC2CC(NC(Cc3c(C)cco3)=O)C2)CC(C)(C)CO1 c1(NC(c2n(C(CC)C)nnn2)c2coc(C)n2)cccc(C#N)c1C c1(C(N(CC)CC2CCCN2C(=O)COC2CCCC2)=O)cc(=O)n(C)o1 C1(C#N)(CC(=O)N(C)CCOCCN(C)C(c2cccc(Cl)c2)=O)CCOCC1 CC1CC(C(=O)Nc2ccc(C(C)(C)C)nc2)N(Cc2ccc(F)nc2)C1 Cn1ncc(CNC(C2(C)C=CCCC2)=O)c1C(=O)NCC(c1cccnc1)O C(=O)(CCC(C)(F)F)N1CCN(CC(C)NC(c2c(CC)cncc2)=O)CC1 Cc1cc(Cl)ccc1-n1nc(CCn2ccccc2=O)nc1C1CCCN1C=O c1(C(=O)NC2CCN(C(c3ccc(CSC)o3)=O)C2)ccc2cnccc2n1 c1(C(N2CCC(OC)(CNC(c3ncccc3Cl)=O)C2)=O)ncc(C)cc1C CC(C)C(O)CC(=O)N(CCNC(c1csc(NC(N)=O)n1)=O)C(C)C N1(C(C(=O)NCC)=O)CCc2cc(NCC3CC3C)ccc21 c1(C(=O)NC(C(=O)NCCC)C)ccnc(CNC(=O)CN2CCCCC2)c1 N1(C(C2Cn3c(C)nnc3C2)=O)CCCn2nncc2C1 c1(C(N2CCC(NC(CCCCCN(C)C)=O)C(F)C2)=O)ccc2c(n1)CCO2 Cc1cccc(CNC(=O)CC2(C)CN(C(c3c(C)n[nH]c3C)=O)C2)c1 c1(CN2CCC(F)(C(N3CC(C)(C)C3)=O)C2)ccc(Cl)c(F)c1 CCS(=O)(=O)NCCC(=O)NC1(CNC(=O)CN(C)C(C)=O)CCC1 CN1CNC(=O)C12CCN(C(c1ccc3c(n1)COCC3)=O)CC2 N1(C(c2ccc(C(C)=O)cc2)=O)CCC2CCC12CNC(c1cc(F)c[nH]1)=O C=CCCCC(=O)NC1(C)CN(C(C2(c3ccccc3)CC(C)C2)=O)C1 N1(C(C)=O)CC=C(C(C)(C)C(=O)N2CCN(c3cc4cccnn4n3)CC2)C1 N1(C(C2C(C)=C2)=O)CCC(CF)(NC(c2ccc(C3CCOC3)s2)=O)C1 C1(F)(CNC(C(C)SCC)=O)CCN(C(c2cc(C3CCCCC3)n(C)n2)=O)C1 C(C)(C(O)C(C)C)NC(c1nc(CNC(c2c(C)snc2)=O)oc1)=O C1(=O)C(CC(F)F)c2ccc(cc2)C2C3CN1C2C3.Cc1cc(CC2CC2)c(C)s1 c1(C(=O)NCCN(CCCCCC)C(C2CC2CC)=O)nccc2ncccc12 CC1CC(NC(c2cc(O)cc(O)n2)=O)CN(C(C2(C)CC2Br)=O)C1 c1(OCC(=O)NC2C(NC(CC(CC)SC)=O)C2)c(F)cccc1F N1(S(CC#N)(=O)=O)CCC(O)C(NC(=O)Cc2ccnc(Br)c2)C1 Cc1cc(COC(=O)CCN2CCCC(OC(C)(C)C)C2)cc(C)n1 Cc1ccc(F)cc1C(N1CCC(C)C(C)C1)C(=O)NC1(C)CC1 c1(C(C)C)ccc(C(N2CC(F)(CNC(C3CCC3C)=O)C2)=O)c(F)c1 N1(C(c2n(C=C)nnc2)=O)CCC(C)C(CNC(c2cn(CC)cn2)=O)C1 c1(N2CC(=O)NCC2)ccc(NC(C2C(F)(F)C23CCC3)=O)cc1Cl N1(C(CCOCCOCC)=O)CC(NC(=O)CC2CSCCS2)CC(C)C1 C1(C(N2CCC(F)(C(N3CCOC4CC34)=O)C2)=O)CC2CCC1O2 C1(NC(C(CSC)OC)=O)CCCC(NC(c2cncc(C(F)F)c2)=O)C1 C1(C(N2CCC(N(C(=O)C(F)=C(C)C)CC)C2)=O)C(C)(C)C1(F)F C(=O)(C(C)CCC(C)(C)C)NC(C(C(=O)Nc1c(OC)cc(C)cc1)(C)C)C N1(C(C(CO)OC)=O)CC2CC1CN2C(=O)CC1(OC)CCOCC1 C1(CNC(c2ccc(OC)nn2)=O)CC2(CC2)CN1C(=O)C(C)(F)F c1(OC)ccc(OC)c(C(=O)NC2CC(CO)CN(C(c3cnn[nH]3)=O)C2)n1 N1(C(c2c(C)nco2)=O)CC2CN(C(=O)CCCC3CC3)CC2C(F)(F)C1 c1(OC)ccc(O)cc1NC(C1(F)CN(C(c2[nH]cc(C)c2C)=O)C1)=O c1(N(C(=O)NC(C)C)C)nnc(C2CCOC2)n1CC(C)SC(C)C C(c1cccc(F)c1)=CC(=O)NCCCCCCN(C(=O)CCCCC1CC1)C C=CC(CCC)CC(=O)NCc1cccc(NC(=O)C(=O)NCC2CC2)c1 c1(C(N(C(C(=O)OCC)C)C)=O)csc(CNC(C2(C#N)CC2)=O)c1 C1(NC(C(COC)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCCCCC1(F)F C(C(CN=c1[nH]n(C(C)C)cc1[N+](=O)[O-])C(F)(F)F)NC(c1c(C)ocn1)=O C1(O)(CC(=O)NC(C2CCCCC2)CNC(=O)C=CCN2CCCCC2)CCCC1 C1(C(=O)NCc2cncs2)CN(C(=O)CC2CCCC3CC23)CCO1 C1(O)(CNC(CCSc2n(C)ccn2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)C1 N1(C(CC=C=C)=O)CCCCCC1C(=O)NC1CCC(N(C)C)C1 CC1CN(C(=O)C=CC2CC2)CC(C)C1NC(c1ccc(Br)cn1)=O C1(C)(NC(C2(CCNC(c3cn(CC)nc3)=O)CC2)=O)CCC(=O)N(C)C1 c1(CN(C)Cc2n(CC)ccn2)nc(N2CCOCC2)[nH]c(=N)n1 N1(C(C(C#C)(C)C)=O)CCN(C(=O)Cc2cc[nH]n2)C2(CC2)C1 CC1CCC2(CCN(C(=O)CN(C(=O)CCc3ncccn3)C)C2)C1 C1(CNC(c2nccc(C)c2F)=O)CN(C(=O)CSc2cn[nH]c2)C2(CCC2)C1 C1(OCCC)CCC(NC(c2noc(C)n2)c2nnnn2C(C)(C)C)CC1 c1(N(C2CCOC2C)C(=O)NC(CC(=O)OCC)C2CC2)ccc(C)cc1C c1(C(N2CC(CN(C(C(Cc3ccc(C)cc3)C)=O)C)C2)=O)cnn(C)c1C#N C(=O)(C(CC(C)C)NC(c1ccc(F)c(C)c1)=O)N1CCC(SC)C1 c1(CN(C(C2CC2NC(=O)Cc2cc[nH]n2)=O)CC)ccc(Br)cc1 C1(NC(c2ccc(I)c(Cl)c2)=O)CC12CCN(C(C13CC(C1)C3)=O)CC2 C=C1CCN(C(C2CC(C)N(C)C2)=O)C(C(=O)NCc2[nH]ccc(=O)c2O)C1 N1(C2CCN(C(C(C)CF)=O)CC2)CCN(C(=O)C=CC2CC2)CC1=O c1(C(=O)NCC(C)N(C)C(c2nnc(S)n2C)=O)cc2cc(Cl)ccc2o1 N1(C(c2nc(O)cc(CC)n2)(C)C)COC2CCCCC2C1 N1(C(CC2(OC)CCOCC2)=O)CCCC(O)(CNC(c2nn[nH]c2Cl)=O)CC1 C(=O)(C(CC)CC(C)C)NC(CCCC(=O)N(CC)Cc1cnn(C)c1)C c1(C(=O)NCCC2CC(NC(CC(CN(C)C)O)=O)C2)ccn2cc(C)nc2c1 c1(OCC=C)ccc(CC(=O)NCC2(F)CC(NC(C3CCCC3C)=O)C2)cc1 N1(C(COC(C)(C)C)=O)CC2CCC1C1CN(C(=O)C=Cc3ncco3)CC21 CC1(C)CC(CNC(C2(C3CC3)CCC2)=O)N(C(=O)CCCn2ccnc2)C1 c1(CNC(C(COCC)NC(CC=CC=C)=O)=O)ccc(O)cn1 c1(NC(C(=O)NCCC(=O)OC)=O)ccc(NCc2cccc(I)c2)cc1 Cc1nncc(CN2CC(C)C2C(=O)NOCC(F)F)c1C c1(C(=O)NCC2(CCNC(c3ccc[nH]3)=O)CC2)nccc2c(F)cccc12 c1(C(C)(C)C(=O)NCC2CCN(C(=O)CS(=O)(=O)N(C)C)C2)ccc(F)c(F)c1 c1(C(=O)NC(C2CCN(C(c3c(CC)occ3C)=O)C2)C)cc(C)ccc1C C1(C(=O)NCC(CC)NC(c2sncc2Br)=O)COCCN1CC Cc1cc(O)c(Cl)cc1C(=O)NCC(C)CNC(c1ccc(Cl)[nH]1)=O N1(C(CCOCC)=O)CCC(F)(CNC(C2CC(O)(CC)C2)=O)C1 C1(C(=O)NCCCN(C(c2nc3cnccc3s2)=O)CC)CCc2nnnn2C1 CC1(C)CC(CNC(=O)Cc2cc[nH]c2)CN(C(=O)CC2COCC2(C)C)C1 C1(c2nn[nH]n2)(C(=O)NCC2(C(=O)NC)CC2)CCOCC1 C(=O)(C(C)(C)C(O)C(C)C)NCC(CC(=O)NCC(C(=O)OC)O)C1CCC1 C1(CC(N2C(C=C)CCC2)=O)CCCCN(C(=O)CCc2nc[nH]n2)C1 c1(NS(=O)(=O)C2CC2)csc(=NCC2C3CCOCC23)[nH]1 c1(CNC(C(=O)NC(c2nc3c(s2)CCC3)C)=O)cc2occc2n1C Cc1cc(C(=O)NC(C)CC(=O)NC2CCCC2)nn1-c1ccccc1 C1(NC(C(C)N(C)C)=O)CCN(C(c2cc(-n3cccn3)ccn2)=O)C1(C)C N1(C(CC2C(C(=O)NC3CC(CO)C3)CCCC2)=O)CC=CC(O)C1 C1(CC(=O)NC2CCCC2NC(C2CCC(=O)O2)=O)(COC)CCCC1 CCCCN=C(NCC1CCNC(=O)C1)N1CCN(CC(F)(F)C(F)F)CC1 C1(C(=O)NCC(C)CNC(C2(CO)CC2)=O)CC(=O)N(C(c2ccccn2)C)C1 c1(NC(C2CCCN(Cc3ccc(CCC)cc3)C2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(C(CO)OC)=O)CC(F)(F)CC1(C)CNC(=O)C(c1ccccc1)C c1(N2CC(C(C)NC(=O)C=Cc3cn[nH]c3)C2)nccc(-c2ccccc2F)n1 C(=O)(C1=CCCCCC1)NCC(C)CN(C(=O)CCc1cccc([N+](=O)[O-])c1)C CCCC(F)C(=O)N1CC(CC(C)NC(c2cnccn2)=O)C1 C1(NC(c2ccc(C)n2C)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC1(C)C C1(OCCCC)CC(NC(=O)N(CCC)Cc2ccco2)C1(C)C C1(CC=C)(NC(=O)C(O)C(C)C)CCN(C(c2cn(CC(F)(F)F)nn2)=O)CC1 C1(S(N)(=O)=O)(C(=O)NC2CCCN(C(C(F)OC)=O)C2)CCC1 c1(C(=O)NCCOCCNC(C2(CC(=O)OC)CCCC2)=O)nnc(O)cc1C N1(C(C(C)OCCN(C)C)=O)CCCC(CNC(=O)CC2C=CCCC2)CC1 C#Cc1cnn(C)c1C(=O)NC1CC2C(NC(=O)COCCCOC)C2C1 C1(C(N(C2CCN(C(C(C)OCCN(C)C)=O)CC2)C)=O)Cc2ccccc2S1 C1(CC)CN(C(=O)Cn2nccn2)CCC1CNC(c1c[nH]c(=N)o1)=O N1(C(c2c[nH]nc2[N+](=O)[O-])=O)CCC2(CCC2)C(NC(C23CC2C3)=O)C1 Cc1cc(C(=O)NC2CCC(CNC(=O)CC(C)(C)O)C2)nn1C N#CC1(C(=O)NS(=O)(=O)Cc2ccc(F)cc2Br)CCc2ccccc21 c1(C(=O)NC2CN(C(C(CC=CC)CC)=O)C(C)C2)cc(Br)c([N+](=O)[O-])[nH]1 N1(C(C)=O)CCC(CC(=O)NC2COCC2NCc2cnnn2C)CC1 C=CCCCC(C)NC(=O)C(COCC)NC(c1ccco1)=O C(=O)(C1=C(c2c(F)nnn2C)N(C)C(=O)N(C)C1c1cnn(C2CC2)c1)CC C1(C(N2CCC(COC)C2)=O)CC(CO)CCN1C(=O)Cc1n[nH]c(C)n1 Cc1cc(C(N2CC3C(NC(C4(Cl)CC45CCOCC5)=O)C3C2)=O)c(O)c(C)n1 C=CC(O)C(=O)N(C1CCC(NC(c2ccc(C(=O)OC)[nH]2)=O)C1)C C(=O)(C1=Cc2cc(F)ccc2OC1)NC1CCN(C(C=C2CCN(C)C2)=O)CC1 C1(C(=O)NCC2CCN(C(C3(CC=C)CCCCC3)=O)C2)CCCC2(CCC2)O1 c1(C(=O)NC2CC3(CC(C)C3)C2)nc(Cl)c(=O)[nH]c1N C1(C(=O)NCC=CC(=O)NCCC(CC)O)OCC2CCCC12 Cc1nccc(C(C(=O)NC2COC2)NC(C2CC(OC(C)(C)C)C2(C)C)=O)n1 C=C(C)C1OCCC1C(N1CC2(COC(CNC(=O)CCOC3COC3)C2)C1)=O N1(C(=O)N(C(CN(C(C)C)C)C)C2CC2)CCOCC1C1CCOCC1 Cc1cc(C(=O)N(C2CC(C#N)C2)CC(=O)NCCN2CCCC2=O)c(C)s1 C1(CCC)CN(C(C2CCCN2Cc2cn(Cc3csc(Br)n3)nn2)=O)CCO1 Cc1c(C(=O)NCCCCCCNC(c2cc(C(C)C)[nH]n2)=O)noc1C1CC1 Cc1nc2cc(C(N3CCN(C(=O)CCC(C)(C)C)CC3CF)=O)cc(O)c2o1 c1(CNC(C2C=CCC2)=O)c[nH]nc1C1CCN(C(c2cc(C3CC3)on2)=O)C1 C1(C(N2C(C)(CC)CC2)=O)CCCC(NC(=O)CC23CCCC2C3)C1 N1(C(CC(CCC)O)=O)CCC(C)N(C(=O)C(O)CN(C)C)CC1 CC1SCCCC1C(N1CC=CC1(C)C(=O)NC1CCC(C(N)=O)C1)=O c1(N(C)Cc2nnnn2C)[nH]c(=NCc2coc(CO)c2)nc2c1ncn2C C1(=O)C(C)(C)C(=O)O1.C1(c2nc(CC(=O)OC)no2)(C(=O)OCC)CCOCC1 C#CC1CCN(C(=O)C(c2ccnn2C)NC(c2scnc2Cl)=O)C1 C(=O)(CC1NC(=O)c2ccccc21)N1CC(NC(C(CSC)(C)C)=O)C(O)C1 Cc1nc2c([nH]1)C(C(=O)N1CC3CN(C(=O)C(=O)NC(C)C)CC3C1)CCC2 C(=O)(C(C#N)C(C)(C)C)NC1C(NC(CC2(OC)CCC2)=O)C1 C1(C(N2C(CNC(C3(COC)CC3(F)F)=O)CCC2)=O)CC(C)CCO1 C(CCC(C)NC(c1cnc(-c2ccncc2)s1)=O)NC(COC)=O C1(CNC(c2nc(CC)sc2)c2nnnn2CCCSC)CCCC(F)C1 Cc1nn(C)c(C)c1CC(N1CC2(CC2)CC1CNC(C1COCC1(C)C)=O)=O c1(C(=O)NC(CNC(CCCCCCC)=O)CO)cc2cccc(OC)c2o1 C(=O)(CS(=O)(=O)c1ccccc1C)NC1CCN(C(c2c(C)ccc(C)n2)=O)C1 C(N=c1nc(C2CC2)[nH]s1)C1C(CNC(=O)COCC2CCCC2)C1(F)F Cc1ccc(C)c(OCCC(=O)NC2CCCN(C(=O)CCF)CC2)c1 c1(C(=O)NC(C(CO)NC(c2oc(CC)c(C)c2)=O)C)coc2c1COC2 c1(CC(C)NC(CCN(C(CCN(CC)CC)=O)C2CC2)=O)cccnc1 N1(C(CCCc2onc(CCC)n2)=O)CCCN(C(c2cnc(S)[nH]2)=O)CCC1 C1(COC)CCCCN1C(=O)CC1COCCN1C(c1cc(C)ccn1)=O C=C=CC(C)C(=O)NCCC1CCCN1C(=O)C(C1CC(F)(F)C1)OC CC1CC(CC(=O)NCCCC2CCCCC2)CN1C(=O)Cc1cncn1C N1(C(=O)OC(C)(C)C)CCC(CF)(CNCC2CC2(F)F)C1 Cc1cc(C(F)(F)C(=O)NCC(O)CCNC(C2CCCN2N=O)=O)cnc1Cl C(=O)(CC(C)C(=O)OC)NCc1c(CC)n[nH]c1.c12cccnc1CNC2=O C(=O)(C1=NN(C)C(=O)CC1)N1CC(CCNC(=O)C=Cc2csc(C)n2)(OC)C1 CC(C)C(CCNC(C1CCCC1O)=O)NC(=O)CSCC1CCCO1 C1(c2ccc(C(=O)OC)cc2)CCCN(Cc2nnc(-c3ccccc3)o2)C1 N1(C(C(c2ccnn2C)NC(CCC=CC(C)C)=O)=O)CCCC2(C=CCO2)C1 C1(CNC(c2c(CCC)nsc2N)=O)CC2CCC1N(C(C1CC1(F)F)=O)C2 c1(C(N2CC(CNC(C3N(C)C(=O)CC3)=O)C2)=O)nnc2ccccn12 C1(CC(=O)NC2CCC(F)(CNC(c3c(C)ncn3O)=O)C2)(OC)CCOCC1 N1(C(C2N(C(CC3(OCC)CCC3)=O)CC=C2)=O)CCCC(C)(C)CC1 C1(OC)CC2(CCC(C(=O)NCCCNC(c3n[nH]cc3C(F)(F)F)=O)CC2)C1 N1(C(C2=CC(C)CC2)=O)CCCC2CN(C(=O)CCn3cc([N+](=O)[O-])cn3)CC12 Cc1occc1CC(=O)NCCOCCCNC(=O)C(c1ccccc1)O C12(CC(=O)NC3CCCOC3)CC1CN(Cc1cscc1Br)C2 c1(C(N2CCCN(C(CC(CC)C)=O)CCC2)=O)cc(O)c(OC)c(C#N)c1 Cc1ccsc1C(=O)NCC1CC(F)(CNC(C2CC2(c2ccccc2)C)=O)C1 N(C(=NCCCCl)N1CCN(C(c2ccco2)=O)CC1)CC(CC)C(C)C C(CN=C(NCCF)N1CCC2CCCOC2C1)N(C)C(=O)OCCSC.C(C)(C)(C)O C1(C(CC(=O)O)NC(=O)COC2CCCCC2)CCCC(=O)N1 CC1CCCN(C(=O)C(C2CC2)NC(=O)CS(C)(=O)=O)CC1 C1(NC(CC2CC(SC)C2)=O)C2CC(NC(c3ccc(Cl)cn3)=O)CC12 C(C1CCC(C)CC1)=C(C)C(=O)N1CC(NC(c2ccc(F)c(C(F)F)n2)=O)C1 C1(CCC=C)(C(=O)NCCOCCNC(=O)Cn2cc(Br)cn2)CCCC1 C1(NC(C(CC(C)C)F)=O)CN(C(c2cocn2)=O)C2(CCCCC2)C1 Cc1ccc(CCCNC(=O)CCn2cc(CNc3ccccn3)nn2)cc1 C#CCCC(=O)N(CC(C)C(=O)NCC1(C(C)C)CCCC1)C N1(CC(=O)NC(=O)CNC(N2Cc3ccccc3C2)=O)CCC2(COC(=O)N2)C1 c1(CNC(C2N(C(C(CC)n3cncn3)=O)CC2)=O)nnc(O)n1C CC1CC(NC(C2CCCCCC2)=O)CCN1C(c1cc(F)c[nH]1)=O Cn1nc(C(N2CCC(C3CCC3)(NC(=O)CC(=O)N(C)C)C2)=O)cc1Br c1(-c2scc(CNc3n(C(C)C)nc(Br)c3)n2)cc(F)ccc1F C1(C(N(CCOCCNC(C(CC)OC)=O)C)=O)CC(=O)c2ccccc2C1 c1(C(NNC(=O)NC(c2sccc2Cl)C)=O)cccc2ccccc12 S(=O)(=O)(CCC(F)(F)F)N1CCC(F)(C(=O)Nc2ncc(C)s2)C1 c1(OCC=C)cccc(CCC(F)F)c1.c1(C2C(=O)NN2C)csc(C(F)F)c1 C1(CCCOC)CCCCN1C(C1C2CN(c3cc(OC)ncn3)CC12)=O c1(C(N2CCN(c3nccc(OC)n3)CC2)=O)ccc(F)c2[nH]ccc12 N1(C(Cc2cc(C)sc2)=O)CC2CC(C1)CN(C(c1sc(N(C)C)nc1Cl)=O)C2 c1(C(=O)Nc2c(C)nsc2)nc2ccc(C(F)(F)F)cn2c1C1=CCC(C#N)CC1 C1(CNC(COCC#C)=O)OCCCC1(C)C.C12(CSC1)C(=O)N2 c1(NC(=O)NCCc2ccc(OCCCC)cc2)cnnc(O)c1Cl C1(C(=O)NCCN(C(Cc2cn(CC)nc2)=O)C)CCCCC1(F)F c1(N(C)C)nc2cccc(C(=O)NCCC3CN(C(C4CC45CC5)=O)C3)c2o1 C1(C)(NC(C(Br)=C(C)C)=O)CCN(C(=O)C(F)=CC2CC2)CC1 c1(C(=O)NCC(C2CC2)NC(C2COC2)=O)cc(Cl)c(Cl)s1 C1(c2ccn(C)n2)CCN(CC2CCN2C2CCNCC2)CC1 Cc1occ(-c2ccccc2)c1C(N1CCC(N(C(=O)CC2CC23CC3)C)C1)=O CC(C)(CNC(N1CCC(CCO)C1)=O)Cn1cc(CCCC#N)nn1 Cc1c(C(=O)N(C(C)CCNC(C2CCC2)=O)C)csc1Br N1(C(c2ccc(SC)s2)=O)CCC2CN(C(c3ccc(F)c(C)c3)=O)CCC12 c1(C(N2CCCCC2(C)C)C(=O)Nc2c(CC)cccc2)ccc(Br)cc1[N+](=O)[O-] CC1CC(C(=O)N2CCC(C)(CC(=O)NC3CCCCC3(C)C)C2)=NO1 C(C(=O)N=c1cc[nH]cc1N1CCOCC1)(C(C)C)c1c(O)ccc(C)c1 CC(O)(CNC(=O)CC1CCCC1NC(=O)C=CC(F)(F)F)CCO C(=O)(CCC(C)CN(C)C)NCCC(CCNC(c1nn(CC)c(C)c1)=O)C C(=O)(C(C#N)C(C)(C)C)N1C(C)CC(CNC(CC2(CSC)CC2)=O)C1 N1(C(C2OCC(C)C2)=O)CCC(CNC(=O)C(C)(C)N(C)C)C(F)(F)CC1 c1(C(=O)NCC2OCC(CNC(C(C)SC)=O)C2)oc2ccc(C)cc2c1C CC1CN(C(c2ccsc2)=O)CC1(C)CNC(=O)C(C)(C)Oc1ccccc1 N1(C(C2C(OC)CCCC2)=O)CCN(C(c2nn(C)cc2SC)=O)CC12CC2 c1(CNC(CC(C)SC)=O)cccc(NC(c2ccns2)=O)c1 N1(C(c2nc(C)[nH]n2)=O)CCCCC1CN(C)C(C1(c2ccncc2)CCC1)=O CC1OCC2(CCC(CNC(=O)C(=O)N(CC(F)(F)Cl)C)O2)C1C N1(C(CC2(COC)CC2)=O)CCC(NC(=O)CC23COC(C)(C2)C3)C(C)(C)C1 C1(C)(C(N(C)CC2(O)CN(C(C(c3cccc(F)c3)C)=O)C2)=O)CCSCC1 N1(CCOC)CCC(NC(=O)C=CC(C)(C)NC(=O)C=CC2CCOC2)C1 N1(C(C(COC)(C)OC)=O)CC2(CC(CNC(=O)CCc3ccn(C)n3)C2)C1 CCC(CC)C(=O)NCC(=O)NCC1CCCC1NC(=O)CSc1ccoc1 N1(C(C(C)OCCOC)=O)CC(O)(CNC(C2CC2F)=O)C1 c1(C(=O)NC(CNC(CC(CCCC)CC)=O)CO)ccc2c(c1)COC(=O)N2 N1(C(c2ccc(F)cc2)=O)CCC2CCCN(C(c3cc4[nH]ccc4s3)=O)C2C1 C1(OC)CCCCC1C(=O)NC12CC(C1)N(C(c1ccc(C(N)=O)nc1)=O)C2 n1(CC#C)cccc1C(=O)NC(C1CCCN1C(c1cnc(C2CC2)s1)=O)C N1(C(C2(CC)CC2)=O)CCC(C(=O)NC2(C(N)=O)CC2)CC1 C1(C(N(C(CCO)C(F)F)C)=O)C(C2CC2)CCN1C(=O)C(O)CN(C)C C(CCCCNC(=O)C(F)F)N(C)C(c1sccc1NS(C)(=O)=O)=O C1(OC)CC(CNC(c2[nH]c(C)cc2C)=O)N(C(=O)CCN(C)C(=O)OC)C1 C12(NC(C3CCC(OC)C3)=O)COC(CNC(=O)CCc3cccc(F)c3)(C1)C2 C1(CC(=O)NCC2(OC)CN(C(=O)C(F)=C(C)C)C2)CCCC(O)C1 N1(C(c2c(C)n(C)cn2)=O)CCC(NC(c2ccccc2F)=O)C(O)C1 C1(NC(=O)Nc2ccc(CC(=O)OC)cc2)C2Cc3c(Br)cccc3C12 C1(CCNC(c2n(C)nnn2)CC(C2CCCCC2)OC)CC(O)CCO1 c1(OC)cc(CN2CCC(NC(=O)Cn3ccnn3)C(F)C2)c(OC)cc1Br c1(C(N2CCC(NC(C3CCSCC3)=O)CC2)=O)ccc2cnnc(O)c2c1 S(=O)(=O)(c1cc(Cl)ccc1CS(C)(=O)=O)Nc1ccn(C2CN(C(C)=O)C2)n1 CC1(C(=O)NCC23CC2CN(C(=O)C=Cc2cccc(F)c2)C3)CC2(CCC2)C1 C(=O)(C(F)(CNC(=O)C=Cc1cn(C)nn1)C(C)C)N1CC(CCCCC)C1 Cc1cnc2cccc(C(N3CC(NC(=O)Cn4cncn4)CCC3C)=O)n12 c1(C(=O)NC(C2CCCN(C(CCC(=O)NC)=O)C2)C)ccc(F)c(F)c1F c1(NC(=O)N=c2ccn(C3CCCCC3)[nH]2)cccc(C#Cc2ccccn2)c1 N1(C(C(COC)O)=O)CCN(C(c2c(C)ccn2C)=O)CC1CF N1(C2C(NC(C(C=C)O)=O)CCC2)CCN(C(C2(C3CC3)CCC2)=O)CC1 N1(C(CN2CCN(CC)CC2)=O)CCC(C)(NC(c2ccc(C#N)s2)=O)CC1 c1(C(C)C(=O)NCCC2COCCN2C(=O)C2=C(Cl)CC2)c(Cl)cccc1Cl N1(C(Cc2cc(COC)on2)=O)CC(NC(C2CC(C)=NO2)=O)C(C(F)(F)F)C1 n1(CC)ccc(C(=O)NC2CCCCC2NC(=O)CC2(n3cccn3)CC2)c1C CC1=C(C)CC(C(=O)NC2CC(C)(C(=O)NCCC3CCSC3)C2)CC1 C1(C(=O)NCC2C(NC(c3cccc(C(=O)NC)c3)=O)C2)CCN(C)C(C)C1 c1(CC(=O)NCC(CC=C)NC(=O)Cc2cncs2)c(C)nc2ncnn2c1C CN1CCN(C(=O)CCOCC2CC2)C(NC(C2CC2c2ccccc2)=O)C1 C(=O)(CC(O)CC(C)(C)C)N1CC(OCCNC(C(CCC=C)(C)C)=O)C1 c1(-c2c(CC(=O)OC(C3CCCO3)C)ccnc2)cc(F)c(OC(C)C)cc1Cl NC(CC(=O)N1CCCC(CCC(=O)O)C1)C(F)F C(CC(C)(C)C)(C(=O)NCc1nc(=O)o[nH]1)NC(COCCCOC)=O N1(CC(=O)NC(C)CCCNC(C2CC(CC(C)(C)C)C2)=O)CCCCS1(=O)=O C1(CNC(CCC)=O)CC(NC(=O)C=C(C)c2ccco2)CCO1 C1(C(N(CCCNC(c2c[nH]nc2Br)=O)C(C)C)=O)CCC=CCCC1 Cc1ncnc(NC2CCN(C(=O)Cc3ccc(F)cc3)CC2)c1Br Cc1ccc(O)cc1C(=O)NC1CCC(CNC(=O)C#CC(C)C)CC1 Cc1csc(C=CC(=O)NCC(C(C)C)NC(=O)COc2ccon2)n1 c1(C(=O)NCC(CC)NC(=O)CCNC(C2CCC2)=O)cc(Br)n[nH]1 Cc1cc(C)c(C(N2CC(O)(CCNC(C3(C)CCCC3)=O)C2)=O)c(Cl)n1 c1(C(=O)NCCCN(C(C(C)=C2CC2)=O)CC2CCCC2)c(Cl)cc(Cl)nc1N C(C(F)(F)CNC(=O)C(CC1CC1)OC)OC.C1(=O)C(CO)N1 c1(C(=O)OCC)cc(C(=O)NCCC2CN(C(c3ccon3)=O)C2)no1 c1(C(=O)NC23CC(CNCc4ccc(Br)s4)(C2)C3)cccc2nc[nH]c12 C1(NC(c2noc(CC)c2C)=O)CCCC12CN(C(=O)CC1COC(=O)C1)C2 CON(CCC(=O)NCC1CC2(CC2)CO1)C(=O)CCC1CCCCO1 C1(c2cn(C(CNC(COCCCOC)=O)C)nn2)CN(C(C)=O)CC(C)(C)C1 C1(NC(COCCC#C)=O)CN(C(=O)CCCNC(N)=O)CC1O Cc1cc(F)cnc1C(=O)NCCCCCCNC(=O)CC(C)(C)O N1(C(c2ncc(C(C)C)s2)C(=O)NCCCF)CCCC2(CCCCC2O)C1 CC(C)CC(C(=O)NC(C)CNC(=O)Cc1coc(C(F)F)n1)N1CCCC1=O c1(NC2CC2)ncc(C(C)NC(C2(C(=O)NC3CCC(SC)C3)CC2)=O)cn1 c1(C(=O)NC2CCCCN(C(c3c(OCC)scc3)=O)C2)cnn2ccccc12 c1(C(=O)NC(CN2CCN(C(C=CC=CCC)=O)CC2)C)cc2cn[nH]c2cn1 c1(NC)cncc(C(=O)NCC2CC(F)CN2C(c2cc(COC)[nH]n2)=O)c1 N1(C(C(CCC)(C)CCC)=O)CCCC2(CCN(C(=O)C#CC(=O)N(C)C)C2)C1 c1(CC)nnc(N2CC3CC(NC(C4(CC)CCCO4)=O)C3C2)nc1CC C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)C(F)(F)c2ccncc2)C1 C1(NC(Cc2c(CC)cccc2)=O)CCC2CN(C(=O)CCOC(C)C)CC2C1 N1(C(C2CN(C(C)C)C2)=O)CCC(C(=O)N2CCC(C)C(C)C2)=C(F)C1 c1(OCC)ccc2cccnc2c1.N12CCCCCC1C(=O)NC1CC(C1)C2=O C1(C(=O)NC(c2ncc(C)[nH]2)CC)CCCN(C(C2CC3(CSC3)C2)=O)CC1 CCCC(C(=O)N1CCN(CCC)CC1)NC(c1cccc(C)n1)=O CC(CSC)CC(=O)NCC1CCN1C(C1(c2ncccc2F)CCC1)=O.C(N)(=O)N C1(NC(C(CC)(C)O)=O)CCCCN(C(=O)COc2c(C)nc(C)nc2O)CC1 c1(NCC2C(CCC)C2)ncccc1S(=O)(=O)N(C1CS(=O)(=O)C1)C c1(CCC(=O)NC(CNC(C(C)(CO)OC)=O)C)c[nH]c2cc(Cl)ccc12 S(=O)(=O)(c1cc(C)ccc1C)CN1CC(NC(CCSC)=O)C(C#N)C1 C1(C)(C(N2CCCC(N(C(C=CC(C)(C)C)=O)CCO)C2)=O)CCC(F)(F)C1 c1(NCC(=O)N(C)CCN(C)C(c2cc(Cl)nc(=N)[nH]2)=O)ccc(C#N)cc1F CCCCC(C)C(=O)NC1(COC)CN(C(=O)CC2CCC(C)O2)C1 c1(OCC(=O)OC)cccc(OC(=O)COCc2cn[nH]c2)c1 C(=O)(C(CC(N)=O)NC(C1CC12CCC2)=O)N1C(C)(CCO)CC1 C1(CC(=O)NCCOCCNC(C(C(CC)O)(F)F)=O)CCC2(CC1)OCCO2 C1(C(c2n(CC)nnn2)Nc2cccc3c2OCO3)CC(C)(C)OC(C)(C)C1 N1(C(Cn2ncc(CC)c2)=O)CCC(N(C(=O)CC2CC3(CCC3)C2)CC)CC1 N12CCC(C)(C)C(C1)NC(=O)c1c(cccc1F)OCC2=O.C12(CC)CC(C1)C2 CC1=C(C(=O)N2CCCC(NC(=O)C3=CCC3)CC2)Cn2nnnc2N1C c1(C(N2CCC(CC=C)C2)C(=O)NCC)ccc2nc(C)ccc2c1 CCC(C(=O)NC(c1cn(C2COC2)nn1)C)C(F)(F)F C#CCCCCC(=O)NCCN(CCCCCC)C(=O)C(c1ccsc1)N(C)C C1(NC(=O)C=CBr)COCCN(C(=O)CCc2cccc(F)c2Cl)C1 c1(C(=O)NC(CC)CN(C)C(c2cc(C)no2)=O)cncc(C(=O)OC)c1 c1(NC2CC(NC(C(c3c(C)noc3C)C)=O)C2)nccc(C#N)n1 c1(CC)ccc(C(=O)NCCC(O)C(=O)NCc2nn(C)cc2CO)cc1 C(=O)(C(CC)C(F)(F)F)NCC1(C#N)CN(C(C2CCC(C#C)CC2)=O)C1 C1(CC(=O)NC(c2nc(C(=O)NCC3CCCC(C)C3)co2)C)C(C)(C)C1(C)C c1(Cc2cn(C3CN(C(C(CC)CO)=O)C(C)C3)nn2)c(Cl)c(C)nn1C Cc1cc(C(C)C(=O)NC2CN(C(=O)C(C)CCO)C2)cc(C)c1 c1(CC)cncc(C(=O)NCC2CC2CNC(C2CC2C(F)F)=O)n1 C(C)(CC(=O)NCC1CCC(NC(=O)Cc2cccnc2)C1)OC C1(NC(CSc2n(C)cnn2)=O)CCOCC1C(=O)NCc1ccc(F)cn1 c1(C(N2C(C(C)NC(C3(CN(C)C)CC3)=O)CCC2)=O)cn2ccsc2n1 N1(C(C(C(C)C)F)=O)CCN(C(=O)CCCC2CCCC2)C(C(F)(F)F)C1 c1(C(=O)OC)c(Br)ccc(-c2ccc(-c3nc(C(F)(F)F)n[nH]3)cc2)c1F N1(CC(C)(C)NC(C2C(=C)C2)=O)CCN(C(=O)CC2OCCOC2C)CC1 c1(C(N(CC(C)NC(CCC=C)=O)CC)=O)ccc2c(Br)cnn2c1 C(=O)(C(C(C)C)N(C)C)NCCN(C(C(C)OCCOC)=O)CC C1(OC)CCCC1C(N1CCCC1CNC(=O)C=CC1CCCO1)=O N1(C(CCc2n(C)cnn2)=O)CCC2CC2(NC(=O)C(Cl)=CCl)CC1 c1(C(=O)NC(CCOC)CNC(=O)CCCc2nccs2)cccnc1Cl c1(C(=O)NC2C(NC(c3n(C)c(S)nn3)=O)C2)cnc(O)c2cccnc12 C1(n2cccc2)(CNC(C(C)CF)=O)CCN(C(c2sc(F)cc2Cl)=O)CC1 CC1(CNC(=O)Cc2cscn2)CCCN(C(=O)CCC2NC(=O)NC2=O)C1 c1(C(=O)NCC2C(C)(C)C(=O)N2)cccc(S(=O)(=O)N2CCSC23CCC3)c1 c1(C(N2C(CC)CN(C(C3(C(N)=O)CCC3)=O)CC2)=O)cc(=O)n2ccsc2n1 Cc1c(C(N2CC3(CCN3C(=O)CC3C=CCC3)C2)=O)sc2nnc(S)n12 C1(NC(Cn2ncc(C)c2)=O)C(C)CCN(C(c2cc(O)cc(N)c2Cl)=O)C1C c1(N(C(C(CC#C)O)=O)C2CC2N2CCOCC2=O)ccc(C)c(OCC)c1 Cc1ccc(C(=O)NC(C(=O)N(C2CCOC2)CCO)C2CC2)o1 C=CCC(CC)N=c1nc(N(C)Cc2nonc2C)c2cnn(C)c2[nH]1 c1(CCNC(c2n(CCSC)nnn2)c2ccoc2C2CC2)ccccc1Br c1(C(=O)NC(CNC(C=CCCC)=O)CO)cc2sc(C)c(C(=O)OC)c2[nH]1 c1(CC(=O)NC(CCOC)CNC(C)=O)sc(C2CCC2)nc1C Cc1cc(=NC(=O)C2CCCC23CCN(C(=O)CCc2ccsc2)C3)[nH][nH]1 N1(C(CC2N(C)CCCC2)=O)CC(CNC(c2cc(C(F)F)no2)=O)CC1(C)C C1(C)(C(=O)NCCn2cc(CNC(CC)=O)nn2)CCC(=O)C1 N1(C(CC2C(C)OC(C)C2)=O)CCCC(N(C)C(c2ccc([N+](=O)[O-])s2)=O)CC1 C1(NC(Cc2ncc(CC)[nH]2)=O)CN(C(c2cc(O)nc(O)n2)=O)CC(C)(C)C1 C12(CNC(C(C3CCOCC3)OC)=O)CC(CCO1)N(C(c1cc(C)cs1)=O)C2 c1(NC(C(N)=O)=O)cccc2c1C1CN(C(=O)COc3ccccc3)CC1O2 C1(OC)CC2CC(C(=O)NCCN(C)C(C3(C(=O)OC)CC3C)=O)CC12 C1(CNC(C(CCOC)C)=O)CC(NC(=O)C(=O)NC2CC2)C12CCC2 N1(C(c2cncc(OC)c2)=O)CCC(C2CC2)C1CNC(C1CCCC(F)C1)=O c1(OC)cnncc1C(=O)N(CCCNC(c1ccoc1)=O)C1CC1 CN1C(=O)CCCC1C(=O)NC1CC2CC(NC(=O)C(O)(C3CC3)C3CC3)C2C1 CCCC(C(=O)OC)C(=O)NCC1CC1CNC(=O)CC1CCC1 C1(C(=O)NCCC2(C)OCCO2)(CC)CCN(C(=O)C=C=C(C)C)C1 C1(N(C(c2cnsc2)=O)CC)CCCN(C(C2CC23CCSCC3)=O)CC1 c1(C(=O)NC2CC3CC(NC(CC(CN(C)C)O)=O)C2C3)ccc2nncn2c1 C(C(C)(CC)C(=O)NCCn1cccnc1=O)NC(CCC(=O)NCC)=O N1(C(c2cc(SC)oc2)=O)CCC(CF)(NC(=O)CCC(=O)OC(C)(C)C)C1 C(CCC(=O)NC(C)(CNC(=O)CCn1ccnc1)C1CC1)OCCOC c1(C(=O)NCC2(F)CCCN(C(c3nc(=N)[nH]cc3)=O)C2)ccnc2cc[nH]c12 N1(C(c2nc(COC)oc2)=O)CC(C)CN(C(c2cc(Cl)no2)=O)CC1C C1(C(=O)NCC(C)NC(=O)C(C)c2ccsn2)CC(F)(F)C1 c1(SCCC(N2C(CCCNC(C(CC)F)=O)CCC2)=O)ccccc1C C(=O)(C1CCCn2ncnc21)NCC1CN(C(C(C)C)=O)C1 C1(C(N2CCC(CCNC(c3cccc(OC(F)F)c3)=O)C2)=O)CC2CC1CO2 N1(C(c2cccc(Cl)c2OC)C(=O)NCCCCCC)CC2OC(=O)N(C)C2C1 N1(C(c2cnn(CCC)c2C)=O)CC(NC(c2cc(C)nnc2O)=O)CC(C)C1 N1(C(c2nc(COC)oc2)=O)C2CCC1CN(C(=O)CCC=CBr)C2 C12(CNC(C(=O)N(C)C)=O)CCC(CN1C(=O)C(C(C)(C)C)n1ccnn1)C2 C(=O)(C(C)(C)C(=O)N1CCCC1)N1CC(C(C)NC(CNS(NC)(=O)=O)=O)C1 C=CC(C)(CCOC)C(=O)N1CC2(CNC(C3(C)CC3C(=O)OC)=O)CC1CO2 C1(C(C)C)CCCN(C(C23CC2CN(C(=O)C(C)N2CCCC2)C3)=O)CC1 c1(C(=O)NC(C2CCCC2)CNC(C2C=CCC2)=O)ccc(C(F)(F)F)cc1 c1(C(=O)NC2CCCN(C(c3c(C#C)c[nH]n3)=O)C2)cnc(C)cc1Cl Cc1ccc(CC(=O)NC2CCC2CNC(C2CCCSC2)=O)cc1 C1(F)(CNC(C2CCCO2)=O)COCCN(C(=O)C=CCN2CCOCC2)C1 C1(COC)CC(CNC(C2CC23CC(O)C3)=O)N(C(c2ccoc2Cl)=O)C1 c1(NC(C(c2nc(C)sc2C)N(C(C)COC)CC=C)=O)ccc(OC)c(C)c1 Cc1ccc(CSCC(C)C)c(I)c1.C1(CC(C)C)C(=O)N1 C(CC(C(=O)N(C)Cc1nc(C)ns1)NC(c1nn(C)cc1C)=O)=CC c1(C(C(=O)N(CCNC(=O)CN(C)C(N)=O)CC)C)c(F)cccc1F N1(C(C(CC)C)=O)CC(NC(c2ccc3nncn3c2)=O)CC(F)(F)C1 C(=O)(C(C)CC=CC)N(CC(=O)NC(CC=C)CC)CCC O=C(CCCCSc1ccccc1)NCCC(O)CNC(=O)CCn1cccn1 CC(CC(C)(c1nnnn1C1CC(F)(F)C1)CC(=O)OC(C)(C)C)C(F)F CC1CCN(C(=O)Cc2ccnc(O)c2)CCN1C(=O)COc1ccsc1 c1(C(=O)NC(C)CNC(C2COC(=O)O2)=O)ccc(C(=O)N(C)C)cc1 c1(C(=O)NCC2C(NC(c3noc(CC)c3C)=O)CC2)cc(C)cc2ccoc12 Cc1cccc(C(O)C(=O)NCCCOCCCCCNC(=O)C=CC(C)C)c1 Cc1cc(C(N2CC3(CC(CNC(=O)CCC(C)N(C)C)C3)C2)=O)ccc1O N1(C(c2cccc(C)c2C)=O)CCC(C(=O)NCc2nn(C)c(=O)n2C)=C(F)C1 Cc1ccc(CN(CCCc2nnco2)C=O)c(OC2CCCCC2)c1 C1(C2CN(C(=O)C=C(C)Cl)C2)(NC(C2CC(C(F)(F)F)(OC)C2)=O)CC1 N(C1CCCCc2ccc(Br)cc21)CC12CN(C)C(CC1)CC2 c1(N2CCC(N(C)CC)CC2)nc2c(c(=NCC3CC(O)CCO3)[nH]1)CCC2 C=CCC(C)(O)C(=O)NC(CC1CCC1)C(=O)NCCC(O)C(F)F C1(C(N(CC(C)NC(c2coc(O)n2)=O)C)=O)COCOC1 CCC(C(=O)N1CCN(C(c2ccn3cccc3c2)=O)C(CO)C1)C(C)(C)CC C(CN1C(=O)COc2cc(Br)ccc21)NC(=O)NCc1cncc(C)c1 c1(N2CC(C(=O)NCC(CNC(C(CSC)OC)=O)F)C2)ccc(Cl)c(Cl)c1 CCC(CC)C(C(=O)N(C(CC)CC(N1CCC(O)C(CO)C1)=O)C)OC C12(C(=O)OC)CC(NC(N3CCCC3CN(C3CCNC3=O)C)=O)(C1)C2 Cc1c(C(N2CCC(NC(=O)C(Cl)(Cl)Cl)C(F)C2)=O)ccnc1Cl Cc1cc(F)cnc1C(=O)N(C1CCN(C(C2CC(C)(F)C2)=O)CC1)C C1(C(=O)NCCC2CCCCN2C(=O)C=Cc2cscn2)CCOCC12CCC2 Cc1cccn2nc(C(=O)N(C(c3ccccc3)CNC(C34CC3C4)=O)C)cc12 c1(NCC2C(CC)(NC(=O)COC(=O)OC)CC2)oc2ccccc2c1CCCO Cc1nc(N(C)CC23CCNCC2C3)cc(-c2ccco2)n1 N1(C(C2N(C(c3c(NC)cccc3)=O)CCCC2)=O)CCN2CCCCC2C1 c1(C(=O)NC(C2CCN(C(=O)C=CC3CCCC3)C2)C)ccc(Br)cc1O c1(OC)cc(C)c(C(=O)NC(CNC(=O)C2=CCCS2)C2CCC2)cc1OC CC(C)(CCCNC(=O)CSC1CC1)NC(=O)OC(C)(C)C.C12CCN(C1)C2=O C1(O)(C(C)NC(C(CC=C)C)=O)CCN(C(=O)COc2cncc(Cl)n2)CC1 c1(C(N2CCCC(CN(C(=O)CC3CCCO3)C)C2)=O)ccc(C2CC2)nc1O c1(C(N2CCC(C)C2CNC(c2coc(C(N)=O)c2)=O)=O)cc(O)cc(F)c1 C1(CNC(C(CC)c2cccnc2)=O)CCC(C)(C)CN1CCC1CCCCC1 c1(C(N2CC3=C(CN(C(C(CCSC)O)=O)C3)C2)=O)ccc(F)c(C)c1C#N S(=O)(=O)(c1ccc(NCCCF)cc1Br)N(C(Cc1cccc(C)c1)C)C CCC(CCC(=O)NC(C)(C)CCCOC)NC(c1cc(C)ns1)=O c1(C(=O)NCC(CC=C)NC(=O)Cc2ncc(C)o2)cc(C)c2[nH]cnc2c1 C12(C(N3CC(NC(C(C)OC)=O)(CO)C3)=O)CC(C)(C1)OC2C N1(C(c2c(C)ccs2)=O)CC(C(N2CCSCC2C2CC2)=O)C2(CCC2)C1 O=C(C1=CC2CCCCC12)NCCN(C(=O)COCCF)Cc1ccccc1 c1(C(=O)NCCC(CNC(=O)CC2CC(F)(F)C2)O)cc(Cl)ccn1 Cc1cc(C(N2CC(NC(c3ccc(C)s3)=O)CC(C)C2)=O)n2ncnc2n1 N1(Cc2cc(C(=O)OCC)no2)CCOC(CN(C)Cc2ccccc2)C1 C1(CNC(c2c(CC)scn2)=O)CN(C(=O)C(C)=C2CCC2)C2(CCOCC2)C1 C1(C(=O)NC2C(C)N(C(c3cc(F)c(F)cc3Cl)=O)CC2)CCC2CCCCN12 C(=O)(C1=CCN(C(C2CCCOCC2)=O)C1)NCC1CC(C(C)(C)C)C1 c1(N(CC(C)NC(=O)CN2CC3CC3C2)C)ccnc(C2CCCC2)n1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2cscn2)=O)ns1 CCCCC(C(=O)N(C)CCOCCNC(=O)Cc1cncn1C)C(C)C N1(C(C2(CC)COC2)=O)CCN(C(=O)CN2CCCC2)C(COC)C1 c1(C(=O)NCCN(CC(C)O)C(c2cc(C(C)C)nn2C)=O)cnn2c1OCC2 C1(CC(C)NC(=O)CC2(O)CCC2)CN(C(=O)COC2CCC2)C1 CC(C)C(C)(O)C(=O)NCCn1cc(CNC(=O)C=Cc2cc[nH]n2)nn1 N1(C(CCC(C)OCC)=O)C2CCC1CC(N(C(=O)C(=CC1CCCC1)C)C)C2 N(C(=NCc1ccccc1)NCC(c1cn(C)cn1)(C)C)CCOCC=C Cc1ncc(F)c(N2CC3CC3(NC(=O)Cc3ccc(F)c(F)c3)C2)n1 Cn1c(C(=O)NC2CC2NC(C2CC=CCC2)=O)nnc1S c1(CC(=O)NC2(C)CC(NC(CC(C)(C)O)=O)C2)c(F)cccc1F c1(N2CC(CNC(CC(C)n3cccn3)=O)OCC2)ncnc2[nH]ccc12 C(=O)(CCC(CF)CF)NC1C2CC(C(=O)NC(C)(CO)C3CC3)C(C2)C1 C#CCCCCCCC(=O)NC1C=CC(CNC(=O)CC(C)C(C)C)C1 C(C(O)CC(=O)NC1CCC(=O)NC1)NC(C=C(CC)CC)=O c1(C(N2CC(COC)(CNC(C3(O)CCSCC3)=O)C2)=O)cc(N)ccc1C C(N=c1[nH]c(=N)[nH]c(=NCC(F)(F)CC2CC2)[nH]1)C1N(C)CC(O)C1 c1(C(=O)NC(C2CCCCC2)C(C)NC(=O)C2CC2)nc2cncnc2nc1O CC(C)C(C)C(=O)NC1CCOC1C1CCN(C(C2(O)CC(F)(F)C2)=O)CC1 c1(C(=O)NCC2N(C(C=CC=CC)=O)CCOC2)ccc(F)c(Br)c1 C12(CNC(C3CC34CCOCC4)=O)CCCC1CN(C(c1sccc1Cl)=O)C2 S(=O)(=O)(c1ccc(F)cc1)N(C)CCNC1CN(C(=O)CC(F)(F)F)CCN1 N1(C(C(C)C2CCOC2)=O)CCOCC(NC(=O)CCOC2CCOCC2)C1 C1(c2n(COCC)nnn2)(NCC(c2ccc(F)cc2F)=O)COCC(C)(C)C1 Cc1cc(=NC(=O)C2c3ccccc3CN2C(=O)C(C)CCC(C)(C)C)[nH]n1C N1(C(c2cc(CCOC)on2)=O)CC(NC(=O)CC#N)CCC1C CCC(C)C(C(=O)NCC1(C(N2CC3C=CC3C2)=O)CCC1)N(C)C c1(C(=O)NC(C(C)NC(C2C(CC(C)C)C2)=O)CO)ccc(N2CCCC2)c(F)c1 c1(OCC#C)ccccc1CNCc1ccnnc1 N1(CCCC)CCCC1C(=O)NCC1(NC(=O)CN(C)C)CC(OC)C1 N1(C(C(F)OC)=O)CCN(C(=O)CCSC(F)(F)F)C(C(F)F)C1 C(=O)(C1=CCOCC1)N(C(C)CN(C(=O)Cn1nccn1)C)C Cc1ccc(NC(C2OCCC2CNC(c2ccccc2)=O)=O)cc1F Cc1ccc(C(=O)N(C)CC2CCCC(NC(c3nccnc3N)=O)C2)nc1O N1(C(CCC(=O)NC)=O)CC(CO)C2(C1)CN(C(=O)CCCCCl)C2 c1(C(=O)NC(CCSC)C(=O)NCCC(O)CO)cccc2cc[nH]c12 N#Cc1c(NC(C2CCN2C(=O)C(CO)c2ccccc2)=O)cccc1Cl C1(NC(C2C3CCCC23)=O)COC2(C1)CN(C(C1CN3CCN1CC3)=O)C2 C(C(F)C(=O)NC(C1CCCCC1)CNC(=O)C(C)CN(C)C)N(CC)CC CCCCC(CC)C(=O)N1CC(CCCCNC(c2ccc(F)o2)=O)C1 C(CC(=O)N1CC2CCC1CC2)(C(F)(F)F)NC(C(C(=O)OC)C)=O c1(OCC(=O)N(C2CCN(C(c3cc(CC)no3)=O)C2)C)ccc(Cl)cc1Cl N1(C(C2CC(C)OC2)=O)CC2(CCN(Cc3cnon3)CC2)C1 C1(C(=O)NCCC2OCCN(C(C3(C)CS(=O)(=O)C3)=O)C2)CCC2(CCC2)CO1 c1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCCC2C)ccc([N+](=O)[O-])cc1Cl C(=O)(C1=CS(=O)CCC1)NC1CCCN(C(C2C(C)CCO2)=O)CC1 Cc1ccc(NC(C2CN(C(C3CCCC34CCC4)=O)CC2F)=O)c(O)n1 c1(NC(CC(C)NC(c2cnc(O)n2C)=O)C)cc(C(F)(F)F)ncc1[N+](=O)[O-] c1(NS(=O)(=O)CCc2cn[nH]c2)cccc2c1OCCC2 C1(N(C(=O)CCNC(N)=O)CC)CCN(C(=O)C(N2CCOCC2)C)C1 N1(C(C=CC)=O)CCN(C(c2conc2Cc2ccccc2)=O)CCC1C N1(C(C2C(C)C2)=O)CCN(C(=O)CC2CN(C)C2)C(C2CCC2)C1 C12(CCNC(c3c(C)nc(CCC)o3)=O)CCC(C1)N(C(C1(SCC)CC1)=O)C2 C1(CC(=O)NC(c2ccc(C)s2)CO)CCn2cncc2C1 CCCCC(CCC)C(=O)NCCCOCC(=O)O CC1CN(C)CCC1NC(C1CCC(CNC(=O)CC(F)(F)F)O1)=O c1(OC)ccc(NC(=O)CN(C)CC23CC2CCN3)cc1NC(C)=O C1(NC(CC(=O)NCC)=O)COCCN(C(c2ccnc(OC)n2)=O)C1 N1(C(c2c(CC)nc[nH]2)=O)CCCC(N(C)C(C2(C)CCC(F)(F)C2)=O)CC1 CC(C)(C(=O)NCC1CCC(NC(C2CC3(CCOC3)C2)=O)CC1)S(C)(=O)=O C#CC1CCCN(C(C2(C)CCCN(C(c3cc(=O)cco3)=O)C2)=O)C1 C=C=C(C)CC(=O)N1CCC(N(C(C2(N3CC4CC4C3)CC2)=O)CC2CC2)CC1 Nc1cnc(C(=O)NC2C3CCC2N(C(=O)CC2(C(F)(F)F)CC2)C3)c(Cl)c1 C1(COC)CN(C(=O)C(C2CCOCC2)F)CCN1C(c1nc(Cl)cs1)=O C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC2=C(CN(C(c3c(C#N)csc3)=O)C2)C1 C1(C(N(CC(CN(C)C(c2[nH]nnc2C(F)F)=O)O)C)=O)CC2(CCO1)CC2 c1(OCCC(C)C)ccc(CNC(=O)NC2CCCC(F)C2)cc1 Cc1cc(=NCCc2ccc(C#N)cc2)[nH]cc1S(=O)(=O)NCC1CC12CCOC2 Cc1cc(C(N2CC(NC(=O)CCCc3ccc(Br)cc3)C(F)C2)=O)c(C)o1 CC1(C)CCC(CO)N(C(C2CN(C(=O)Cn3cnc(=N)[nH]3)CC2(C)C)=O)C1 C1(C(N(C)Cc2cc(C#N)ccn2)=O)CC12CCN(Cc1cccnc1)CC2 CC1(C)OCCC1CNC(c1ccc(Cc2cccc(O)c2)cc1)=O N1(C(C=C(C)CNC(c2cnn(C)c2C#N)=O)=O)CCN(C)C2CC12 N1(C(C(C)OCCC=C)=O)CCOCC(F)(CNC(c2cc(C(F)F)cs2)=O)C1 C1(CNC(=O)NC2CCN(C(C3(C#C)CCCC3)=O)C2)CC2(CC(OCC)C2)C1 C1(NC(C2(COC)CC(F)(F)C2)=O)CCN(C(c2sccc2F)=O)CC1O C(=O)(C(O)CCCc1ccccc1)N(CCCNC(C1N(CC)CC1)=O)C N1(C(C(CC=C)C)=O)CC2OCCN(C(c3scnc3C3CC3)=O)C2C1 C=CC(CC(=O)N1CC(NC(c2occc2Br)=O)C(O)C1)c1ccccc1 c1(C(=O)NCC(CNC(C2(C)CC2Br)=O)O)cccnc1OCCO C1(NC(C2CCCC23CC3)=O)CN(C(c2ccoc2Cl)=O)CC1O C#CCCCC(C)C(=O)N1CCCC1C(=O)NCCc1ncc(C)o1 c1(OC)ncc(Cl)cc1C(=O)NC1CC(CNC(=O)C(C)c2ccco2)CC1O c1(C2(C(N3C4C(NC(CCSC)=O)C(C4)C3)=O)CCC2)ccc([N+](=O)[O-])c(C)c1 O=C(CC1=CCOCC1)N1CC(O)CC1C(N1CCCC(CO)CC1)=O C1(NC(c2cc(SC)oc2C)=O)CCSC12CN(C(=O)C(c1ccccc1)F)C2 N1(C(CC(C)C)=O)CCN(C(=O)C(CC(C)C)N(c2ccccc2)C)C(CO)C1 C1(C(N2C(C)CCCC2)=O)CC(c2ccccn2)=NO1 N1(C(C=CC)=O)CCCC(C2CCN(C(=O)C(CC3CC3)CC3CC3)C2)C1 c1(C(=O)NC(CC(C)C)c2nc[nH]n2)ccc(OCC2CC2)c(F)c1 C1(CN(C(C2CCC2(F)F)=O)CC)CCN(C(c2ccc(C3CC3)o2)=O)C1 C(C(C(C)(C)C)NC(c1ncccc1Cl)=O)NC(C1C(OCC)C1)=O CCC(C(=O)N1CC2CCC2(NC(c2nnc(O)cc2O)=O)C1)C(C)C CC1OC2(C)CC1(C(N1CCC(CNC(c3ccnc(F)c3Cl)=O)C1(C)C)=O)C2 C1(NC(C(CC=C)OC)=O)CCN(C(c2ncn3c2CCC3)=O)C12CCC2 c1(C(N(CCC(C(C)C)NC(C(C2CC2)OCC)=O)C)=O)ccnc(F)c1OC c1(OC)ccc(C(N2CCC(C)C2CNC(c2nc(C)nn2C)=O)=O)cc1O c1(NCc2cccc(C(N3C(C(CC)O)CCC3)=O)c2)ccc(S(C)(=O)=O)cn1 c1(CC)nc(O)c(C(=O)NCC(CC)(CC)NC(=O)C#CC2CCC2)cc1C N1(C(CCCSC)=O)CCC(NC(c2cnccc2C(C)(C)C)=O)C(F)C1 C1(CNC(C(C)SC)=O)CCN(C(=O)CCNC(=O)CO)CCC1(F)F C(C(O)CC(=O)N1CC(F)CC1CNC(c1cc(C(F)F)cs1)=O)N(C)C C1(NC(=O)CC(F)F)CC2(CCN(C(C3C(F)(F)C34CC4)=O)C2)C1 N1(Cc2cn(CC)nc2)CCN(C(c2cc(Cl)ccc2OC)=O)CC1C(C)C C1(C(=O)NCC(CN(C)C)(C)O)CCCC(NC(=O)C=Cc2ccncc2)CC1 c1(CC)cc(C(N2CC(NC(c3cc(F)c[nH]3)=O)C(F)C2)=O)cc(C)c1 c1(C(=O)NC2C(NC(c3nc(C(C)C)sc3)=O)COC2)ccnc2ccccc12 O=C(C(F)C(F)(F)F)Nc1cn(-c2ccc(CC3CCCOC3=O)cc2)nn1 N1(C(C(C)C(C)(C)C)=O)CC(NC(=O)Cc2ccccc2[N+](=O)[O-])CC(C)(C)C1 c1(CCC(=O)NCC(CC=C)NC(c2conc2C(C)C)=O)nnc(C)n1C c1(OC)c(Cl)ccc(C(N2CCCN(C(=O)CC3C=CCC3)C(CO)C2)=O)c1F C1(NC(C(C)OC)=O)CC2C(NC(=O)CNC(c3cc(C)oc3C)=O)C2C1 c1(C(=O)NC2CC(NC(C(CC)n3cccn3)=O)C2)nn(C(C)C)cc1Br c1(CC)cccc(C)c1C(=O)Nc1ccc(Cl)nc1NS(=O)(=O)C(C)C C(=O)(CCCCCC(C)O)NCC1CC(O)(CNC(c2cc(CC)nn2C)=O)C1 C1(C(=O)NCC(CCOC)NC(=O)Cc2n[nH]c(=N)s2)CNC(=O)N1 C1(F)(C(=O)NCC2C(C)(C)C2CO)CCCN(C(=O)CC2CCC(=O)N2)C1 c1(C(=O)NC2CCN(C(CCC(CC)C)=O)C2)ccc2nnc(C)c(C)c2c1 c1(C(=O)NCC(C)NC(=O)CCN2CCC2)ccc(-n2ccnc2)nc1 c1(C(C)(C)C)ccccc1C(=O)NC1CN(C(C2CC2c2nnsc2Cl)=O)C1 N1(C(=O)OC(C)(C)C)CCCC(C(=O)NCC#CCN(C(=O)C=CS(C)=O)CC)C1 CCC1=C(C(=O)NCC2(O)CC(NC(=O)C(C)(C)CC#N)C2)CCCO1 C1(C)(NC(C2(COC)CN(C(=O)C(C)N=[N+]=[N-])C2)=O)CCC(=O)N(C)C1 C(=O)(C(CN(C)C)C(C)C)NC(C(N1C(CC)(CC)CC1)=O)Cc1ccco1 c1(C(c2nnnn2CC2CC2)NCC(CC)Oc2ccncc2)c(Cl)ncn1C c1(C(N2CC3CCN(C(C4C(OC)C4)=O)CC32)=O)cccc2cccc(OC)c12 N1(C(c2c(CC)nco2)=O)CCOC(C(C)NC(c2ccccc2C2CC2)=O)C1 CC#CC1CCN(C(=O)CCN(C(c2cc(C#N)cn2C)=O)CC2CC2)C1 c1(C(=O)NC(CNC(c2cnn(CCC)c2Cl)=O)(C)CO)ncnc2c1CCC2 C1(C)(C(=O)NCCC(=C)C)CCN(C(=O)C=C(C)c2ccccc2)CC1 CC1OC2(C(N3CC4CC(NC(c5cnnc(O)c5)=O)C3C4)=O)CCC1CC2 C(c1nc2ccccc2o1)=CC(=O)NC1CCN(C(C=C(CC)C)=O)CC1CO c1(SCC(CC)N(C)C)nnc(-c2ccc(OC)cc2)n1CCC#N N1(C(c2c(SC)scc2)=O)C2CCC1C(CNC(=O)C(C)CC(F)F)C2 Cc1ccc(C23CC(C(=O)NCCc4cc(C)n(C)n4)(C2)C3F)cc1 n1(C(C)C)ncc(F)c1C(N1CCOC(C(C)NC(=O)C=Cc2ccco2)C1)=O c1(C(N2C(CNC(C3CCCO3)=O)CC(C)(C)C2)=O)cc(Br)c2c(c1)OCO2 C12(C(=O)NCC3N(C(CCC(C)(F)F)=O)CC3)CCOC1CCOC2 N1(C(CCOCCCOC)=O)CC2CCC(C1)N2Cc1ccc(C)cc1F N1(C(c2cnc(C(C)O)s2)=O)CCC(C)(NC(c2n[nH]cc2CC2CCC2)=O)C1 N1(C(CCC(C)OC)=O)CCN(C(c2ccc(C)cc2N)=O)CC1C1CC1 c1(CNC(C(C(C)SC)O)=O)c(C)nn2c1CN(C(=O)CCCSC)CC2 c1(C(=O)NCC2CCC(NC(Cc3cc(C)[nH]n3)=O)C2)c(Cl)ccc(F)c1C N1(C(C=C(C)Cl)=O)CCC(CNC(=O)C(C(C)C)OCC(C)C)C12CCC2 N1(C(c2c(C)nccn2)=O)CCCC12CCCN(C(=O)Cc1ccc(Cl)cc1)C2 C1(CC)(NC(=O)CCOCC(F)F)CCN(C(c2occc2C)=O)CC1 CCC(C(=O)N(C1CCN(C(C2(C)CCCCC2)=O)C1)CCO)C(C)(F)F C1(CC(=O)NC(CC#C)C)CC(C)N(C(=O)CSCCCC)C1 C1(C(N(CCNC(C2C(C=C)C2)=O)C(C)C)=O)CC(F)C(=O)N1C C1(CC)CCCN(CC(=O)N(C)CC2CCCN(C(c3cn(C)c(O)n3)=O)C2)C1 C12(NC(c3nc(CNC(C)=O)sc3)=O)CC1CN(C(=O)CC(O)CN(C)C)C2 C1(F)(C(=O)NC2(CC)CCOCC2)CCCN(C(c2cc(C)c(C)o2)=O)C1 CC(C)CN=C(NCc1ccccc1CS(C)(=O)=O)NC1CCCC1(F)F C=Cn1nccc1C(=O)NC1CC(OCC)CN1C(=O)COCCCC C1(O)(c2cn(CCNC(C(CCC)F)=O)nn2)CCC(C)(C)CC1 C1(C(N2CCCC(CC)C2)=O)CN(C(c2cc(O)cc(=O)o2)=O)CCN1C C1(C(N(CC(c2ccccc2)N(C)C)C)=O)CCCC2(CC2)C1.N12CC(O)(C1)C2 C1(NC(Cc2cc(C)on2)=O)CCN(C(=O)CC2CCC=CCC2)CCC1CO c1(CC(=O)NC2(CN(C)C(C3CCCC(F)(F)C3)=O)CC2)cc(Cl)cc(Cl)c1 c1(C(=O)NCC2CC(NC(=O)CCF)C(O)C2)cccc2c1COC2 C1(C(C)(O)CNC(=O)CCc2ccc[nH]2)CCCN(C(=O)CP(C)(C)=O)C1 c1(NC(CC2N(C(c3ccc(OC)s3)=O)CCOC2)=O)c(C)ccc2c[nH]nc12 CC1CCC(NC(=O)CCC2CC(C)(C)CO2)CN1C(=O)CCn1cncn1 c1(C(=O)NC(CNC(c2c(C)occ2)=O)C2CCC2)ccc(F)c(C)c1N C1(NC(Cc2cn(C)nc2)=O)CC2(C1)CC2C(=O)NC1CN(CC(F)F)C1 N1(C(C(CSC)O)=O)CC(NC(c2csc(C(F)F)n2)=O)C(O)C1 CC(C)CC(CNC(=O)C(C1(O)CCCC1)F)NC(c1cc(Br)cs1)=O c1(OC)ccc(O)cc1C(=O)NC1(C)CCCCC1O C1(C2CC2)(CNC(C(CCCC)N(C)C)=O)CCN(C(c2cc(C)c(C)[nH]2)=O)C1 OC1CC2(CC(NC(c3sccc3Br)c3nnnn3C3COC3)C2)C1 N1(C(C2(C)CCC(=O)N2)=O)CC23CCCCC2(C1)CN(C(=O)CCCF)C3 c1(SC)ccc(Cc2cc(-c3ccccc3)cs2)cc1.N12CC(F)CC1C2=O c1(NC2C(NC(c3c(CC)nc[nH]3)=O)CS(=O)(=O)C2)cc(C#N)nc(C)n1 CC(CCCNC(c1cc(Cl)cs1)=O)NC(=O)Cc1nc(C(F)(F)F)n[nH]1 C1(NC(CC(CCC)CC)=O)CC2CCCC(C1)N2C(C1CCS(=O)(=O)N1)=O C(c1ccccc1C)=CC(=O)NC(C1CCCC1)CNC(c1c(C)cn(C)c1)=O C1(NC(CCOCC#C)=O)CCC(C)(NC(=O)C(F)Cc2ccccc2)CC1 N1(C(CCC2CCN(C(C(CC(=O)OCC)C)=O)C2)=O)CCc2ncn(C)c2C1 CCCC(C)(CC)C(=O)N1CC2CC1(CNC(c1cccnc1)=O)C2 C=C1Cn2c(C(N3CCN(C(c4c(C)ccn4C)=O)CC3CC)=O)nnc2S1 c1(CC(N2CCCC(C)(NC(C(C)NS(C)(=O)=O)=O)C2)=O)ccc2nsnc2c1 C1(CNC(=O)CCCCCCn2cc(CO)nn2)CCCC2(CCOCC2)O1 c1(CC(=O)NC(CCNC(C(CN(C)C)N(C)C)=O)C)ccc2c(c1)COC2 C12(C(=O)NCc3ccc[nH]3)CC(c3cccc(C(F)F)c3)(C1)C2F C1(NC(C(C)=C(C)C)=O)CC2(CCN(C(c3cccc(C4(C)CCO4)c3)=O)C2)C1 C1(C(=O)NC(c2c(C)n[nH]c2C)C)CN(C(c2cocn2)=O)CC(C)O1 C1(C(N2C(CN(C(c3snc(C)c3N)=O)CC)CCC2)=O)C2CN(C)CC12 C12(CNC(Cc3ccc(OC)cc3)=O)CC(C1)C(NC(c1cnc[nH]1)=O)CO2 c1(CC(=O)NCC=CC(=O)NCC(C)(C)O)cccnc1O C1(C(C)C)CN(C(c2nc(Cl)cs2)=O)CCCN1C(c1cc(C(C)(C)C)c[nH]1)=O N1(C(CC2(N(C)C)CCCC2)=O)CCC(CCCNC(C2CCOC2)=O)CC1 c1(C(=O)NC2CC(C)NC2)ccc(S(=O)(=O)NC(C2CCCCN2C)C)cc1 C1(c2onc(C)n2)CC(F)CN1C(C1COC(C)C1)C(=O)NCC(F)F Cc1nnc2n1CC(C(=O)NC(C)CCNC(=O)CNC(c1ccoc1)=O)C2 c1(C(C)NC(=O)C(=O)NCC2CS(=O)(=O)CCO2)nc2ccccc2[nH]1 CC1CCOC(C(=O)NC(C)(C(=O)NCC(c2cnc[nH]2)C)C2CCC2)C1 C1(CC=C)(C(=O)N(CC(O)COC)C)CCN(C(=O)CCOCC)C1 n1(CC)cc2ccc(C(=O)NCC=CCNC(c3ccc(F)o3)=O)cc2n1 c1(CNC(=O)NCC)ccc(S(=O)(=O)NCC2(CC(F)(F)F)CC2)cc1 C1(CC(=O)NCC(CCC)C)CN(C(c2cccc(CC#N)c2)=O)CC12CC2 CC(C)C(O)C(C)(C)C(=O)NC1CCC(C(=O)NCc2cncc(Cl)c2)C1 Cc1cc(-n2ccc(C(=O)NCCC(C)(C)O)n2)ccc1Cl CC1(C)CCC=C1C(=O)N1CC2CCN(C(=O)CC=C(Cl)Cl)C2C1 N1(C(C(C2CCOCC2)OC)=O)CCN(C(=O)CCCN=[N+]=[N-])C(C2CCC2)C1 C(=O)(C1CS(=O)(=O)c2ccccc21)N(C1CCCC1)CCNC(c1csnn1)=O C12(CN(C(C=CCN(C)C)=O)CC3CC3)CN(C(=O)C3=CCC3)CC1CS(=O)(=O)C2 CN1CC(O)CC1C(N1CCC(N2CCN(C(=O)CC(F)(F)F)CC2)C1)=O.c12cccn1c2=O c1(C(=O)NC(CC)CNC(=O)C(C)CC2CC2)noc2cc(F)ccc12 c1(C(=O)NCC2(OC)CN(C(C(CC)F)=O)C2)cccc(Cl)c1O N1(C(C(C)OCc2ccccc2Cl)=O)CC2CCCC(C1)N2C(C1(CF)CC1)=O CCCC(C(=O)NC(Cn1ccnn1)C(=O)NCCCCS(C)=O)OC c1(NCC(=O)NC(c2ccc(F)cc2)C)cn2c(n1)CCCC2C(=O)O N1(C(C(CC)SC)=O)CCc2c(ncn2C)C12CCN(C1CCCNC1=O)C2 N1(C(c2occ(C)c2)=O)CCN(C(=O)CCC2OCCO2)CC1CC(F)F C1(NC(CCCC(C)O)=O)CC2CN(C(c3ccc(NC=O)cc3)=O)CC2C1 C(=O)(CC(C)CC(C)(C)C)NCC12OCC(NC(C(C)OCC(C)C)=O)(C1)C2 C#CCC(CC(=O)NC(C1CSC1)C)NC(=O)CC1(COC)CC1 c1(C(=O)NC2CC(N(C(C(C(C)C)F)=O)C)C2)c[nH]c2ncc(Br)cc12 Cn1nc2c(c1C=CCSc1ccccc1)CCC2 N1(C(C(C)O)=O)CC(F)(F)CC1CCNC(c1scnc1C(C)(C)C)=O c1(CC(=O)NCC2(NC(C3CC3F)=O)CCC2)ccccc1Br c1(OC)cc(C(=O)NC2CN(C(C3CCCC3)=O)C2)cc(Br)c1OC(C)C c1(C(N(CCCNC(C2(C)CCCN2C)=O)C)=O)cnc(S(C)(=O)=O)s1 c1(C(=O)NC(CNC(C(C)N2CCCC2)=O)(C)C2CC2)cc(C(N)=O)co1 c1(C(=O)NCC2CC(CNC(c3c(C)cnn3C)=O)OC2)cc(Cl)cnc1C C1(CNC(c2cc(C(C)C)no2)=O)CC(NC(c2cn[nH]c2)=O)C1(C)C C(=O)(C1Cc2ccc(F)cc21)N1CCN(C(CN(C)CC)=O)CC12CCC2 C1(C#CC(=O)N(C(C)CNC(=O)CCc2c(F)cccc2Cl)C)(CC)CC1 C1(CNC(C(=O)NC2(CCC)CC2)=O)CC(C)(C)CN1 C1(OC)CC2CC(C(c3nnnn3C3(C)CC3)NCCCCF)CC12 c1(C(N2CC(O)(CNC(Cc3scc(C)n3)=O)C2)=O)cc2c(F)ccc(F)c2[nH]1 C1(NC(CCOc2ccc(C)cc2)=O)CCN(C(c2ncc(F)cn2)=O)CC1C C1(CC)CCC(C(=O)N(CCCCCNC(=O)CCCc2csc(=N)[nH]2)C)O1 C(=O)(C1CCc2c[nH]nc21)NC(CC=CC)C(=O)O C1(NC(=O)CC2CC=CCC2)CC(F)CN(C(c2cc(Cl)ccc2O)=O)C1 N1(C(C(CC2CN(C(C=C(CC)CC)=O)C2)F)=O)CC(O)CC(C)(C)C1 c1(C(N(CC(CC)NC(c2n[nH]c(C)c2Cl)=O)C)=O)cnc(C)c(C)c1 N1(C(C(=O)N(CC(C)NC(C=C(CC)CC)=O)C)C)CCCCC1=O c1(C(=O)NCC2N(C(c3ccc(OCC)c(OC)c3)=O)CC2)n[nH]c(C)c1[N+](=O)[O-] Cc1ccnc2c(NC3COc4ccccc43)ccnc12 c1(OC)cc(CN2CCC2Cc2cc(Cl)ccn2)ncn1 CC1CCC(CNC(=O)C=C2CCC2)N(C(=O)CN(c2ccncc2)C)C1 c1(C(=O)NC(CC(C)C)C(F)F)c2ccccc2nn1C CCCC(C(=O)OC)C(=O)N1CC(NC(c2cc(C(C)C)[nH]n2)=O)C(N=[N+]=[N-])C1 N1(C(C2ON=C(CC)C2)=O)CC(N(C(=O)C(c2ccccc2)=O)C)C2(CC2)C1 CN1CCOC(C(=O)N(CCCNC(C2CNC(=O)N2)=O)CC2CCCC2)C1 c1(C2(NCc3nc(-c4ccc(OC)cc4)oc3C)CC2)cc(Br)cc(Cl)c1F CC(C)C(CNC(=O)CCn1ccnc1)C(=O)N1CCC(N(C)C)(CF)C1 N1(C(CNS(C)(=O)=O)=O)CCC2CCN(C(=O)CSc3ccc(Cl)cc3)CC12 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)(CNC(c2cscc2Cl)=O)C1 C(c1ccc(C(N)=O)o1)=CC(=O)N(CCN(C(C1C(C=C)C1)=O)C(C)C)C N1(C(COC2(CCCC)CC2)=O)CCC(n2cc(-c3csc(C)n3)nn2)C1 C(CCC(C(=O)NCC(C)CO)N(CC(=O)OC)CC)OCC C1(c2nc(CC3(N(C)C)CCCC3)[nH]n2)CCN(CC2CCCS2(=O)=O)CC1 CCC(C(=O)NCCCC(C)NC(C1(C(N)=O)CC1)=O)C(C)C O=C(C=CSc1nc[nH]n1)NC(c1cc(C(F)(F)F)on1)C1CCCN1 N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(c2cc(C)ns2)=O)C1 C1(NC(C)=O)CC2CN(C(=O)C(C)(C)Oc3ccc(F)c(F)c3)CCN2C1=O c1(C(=O)NCCCCN(C(CS(=O)(=O)NC)=O)C)cc(F)ccc1C(F)F c1(C(=O)NCC(C2CCCC2)NC(=O)CCc2ncco2)cc(Cl)ccn1 c1(C(N(CC(CNC(C(F)OC)=O)O)C)=O)cnc(C2CCC2)cc1C C1(NC(=O)NC(C)C(C)(C)F)CCN(c2ccccc2C(F)(F)F)C1=O c1(OC)ccc2cnn(CC(N3CCC(C4(C(=O)O)CC4)CC3)=O)c(=O)c2c1 N1(C(C(CCC)OC)=O)CC(NC(c2c(OC)ncnc2C)=O)CC2(CCC2)C1 C(=O)(C(O)CCC(C)C)NCC(CC(=O)N(CC)CC1CCOC1)C1CC1 c1(C(N2CCC(NC(C(C)n3cnnn3)=O)C2C)=O)cccc2c1CCCCC2 c1(CC(=O)NC(C)C(N2CCOCC2CC2CCCC2)=O)ccc(Br)cc1 C1(NC(C2(C=C)CCC2)=O)CCCCC1NC(=O)CCN(C(CC)CC)C C1(C)(C(=O)NCCC2OCCN(C(CC(C)(C)OC)=O)C2)COCC1(F)F C(N=c1nc2[nH][nH]cc-2c(O)n1)C12CC(NC(Cn3c(C)ccn3)=O)(C1)C2 N(C1CCc2cc(CNC(C3(C#N)CC(=O)C3)=O)ccc21)C(C1(C)CC1(Cl)Cl)=O C=CC1(C(=O)NCCC2(O)CN(C(c3ccc(CCC)[nH]3)=O)C2)CCC1 N1(C(CC=CC)=O)C2CCC1CC(NC(c1cn(CC(=O)N(C)C)nn1)=O)C2 N1(C(C2CCCS2(=O)=O)=O)CCCC2(CCCCN2C(C2CCC(O)CC2)=O)C1 c1(C(=O)NC2CN(C(c3[nH]cc(CC)c3)=O)CC2C(F)F)cccc2[nH]ccc12 C1(CC)C(=O)N(C)CCN1C(C1CN(C(c2ccc[nH]2)=O)CCC1O)=O CCCCC(C)CCC(=O)N1CCC2C(C1)CN2C(=O)CCn1ccnc1 N1(C(c2ncn(C)c2)=O)CCCC(Nc2cnncn2)C1 c1(C(=O)NCC(CNC(C2(CC=C)CC2)=O)F)cc(Cl)ccc1Cl C1(NC(C23CC(C)(C2)OC3C)=O)CC2CCC2C1.N1(C(=O)NC)CC(NC=O)C1 C#CCC(CC(=O)NCC1CC2(CC2)C(=O)O1)NC(c1cc(Cl)c[nH]1)=O CCC(C)(C#N)C(=O)NC(CC(=O)N(CC(C)C(C)C)C)C(C)OC N1(C(C=Cc2cnc(-n3cc(CCN(C)OC)nn3)o2)=O)CCN(C(C)C)CC1 c1(C(N2C(C)(CNC(C3C(C)(C)C3)=O)CCC2)=O)cc(Br)cnc1N c1(CC)[nH]nc(C(=O)NC2CC3CC2CN(C(=O)C(CSC)OC)C3)c1[N+](=O)[O-] c1(COCc2cn(C3CN(C(C(C(=O)OC)OC)=O)C3)nn2)cc(C)cc(F)c1 C1(NC(CCCCOCC)=O)CC=C(C(=O)NC2(C)CCC(C)(C)C2)C1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(CCNC(=O)Cc2cccs2)CC1 C1(NC(C2CCCCO2)=O)CCN(C(C2CCCCC2(F)F)=O)C12CCCC2 Cc1cc(=NCCCCC#N)[nH]c(=NCCOCCS(N)(=O)=O)[nH]1 c1(C(=O)NC2(CO)CN(C(COCc3cc(C)no3)=O)C2)cc(Cl)c(C)cn1 C1(C(=O)NC2CCN(C(CCCC(C)O)=O)CC2F)CS(=O)(=O)CC(=O)N1 C(=O)(C1=CCc2ccccc21)NCCCC(C)NC(C(CC(C)C)NC(C)=O)=O C(=O)(C(CO)C(C)(C)C)NC1(C(N2CCC(C(C)(C)O)C2)=O)CCCC1 Nc1nccnc1C(=O)NOCc1cn(C2CCCCC2)nn1 N1(C(CNCCC)=O)CC(NC(=O)C=CC(=O)OC(C)(C)C)C(C(F)(F)F)C1 C1(C)(CN(CCN2CCN(C(=O)OCC)CC2)CC)CNCCC1(F)F Cc1cc(N(C(C)CNC(=O)COCc2cc(C)on2)C)n2nc(C)cc2n1 N1(C(CN(C(C(CC)C)=O)C)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 CC1CC=C(C(=O)N2CCC2CNC(=O)Cn2ccc(Br)n2)CC1 C1(NC(=O)COC2CC2)CCN(C(c2cccc(Br)c2Cl)=O)CC1O C(C)(C)(CC(F)C(=O)N1CCCC(N2CCC2)C1)NC(C(C(C)C)SCC)=O C1(C(=O)NCCC(C)(C)NC(CCc2ccn(C)n2)=O)CC2CCC1O2 c1(OC)ccc(CC(=O)NCC2CC(NC(=O)CC=C(C)C)C2(C)C)c(F)c1 C12(CN(C(CN(C(CN(C3CC3)CC)=O)C)=O)C)CCC(CC1)CC2 Cc1cc(C(C)C(=O)NCCCCN(C)C(C2C3CCC(F)(F)C23)=O)cc(F)c1 c1(CC(=O)NC2CCN(C(C=CC)=O)CC2O)nnc(O)c2ccccc12 Cc1cc(CN2CC3CC3(C(=O)NCc3cccc(C4CC4)c3)C2)cc(C)c1Br C1(CNC(C(COC)C)=O)CCCC2(CN(C(c3cc(N)c(Cl)c(O)c3)=O)C2)O1 N1(C(C(CC)COC)=O)CCCC(C)(C)C1C(=O)NC1CCC2CCC12 C12(C(N3CCC(N(C)C(C4C(C)(C)OC4(C)C)=O)C3)=O)CC=CCN1CCC2 N1(Cc2ccc(OC)c(SC)c2)CCC2(CCC(O)C2)C1 CCCCC(O)C(=O)N(CCC(C(C)C)NC(=O)C(C)Sc1ncccn1)C C1(NC(C(C(C)C)O)=O)CCCCN(Cc2ccc(Cl)cc2Cl)C1 C(=O)(C(CCCOC)NC(c1c[nH]nc1C(C)C)=O)NCC1CN(C(C)=O)C1 c1(C(N(C2CCN(C(=O)CCC(C)(C)O)CC2)CC)=O)ccc2c(c1)OCCO2 Cc1ccnn1C(C)C(=O)NC1CC(CNC(c2csc(C(C)(C)C)n2)=O)C1 Cc1cc(C(N2CC3CC2CN3C(=O)C(C)NC=O)=O)nc2nccn12 O=C(CCCCCn1cc(-c2ccc(Cl)cn2)nn1)NC1(C(=O)O)CCS(=O)(=O)C1 C1(NC(CC2CN(C(C=CCN(CC)CC)=O)C2)=O)CCCN(C)C1C c1(C(N2CCC(CNC(CCC(=O)NC)=O)C2)=O)sc(C#N)cc1Cl C(CCCCCC(C)C)n1cc(C2N(C(CC(C)(C)OCC)=O)CCCC2)nn1 N1(C(Cn2ncc(C)c2)=O)CC2CCN(C(C3COCC3C(F)F)=O)CCC2C1 c1(C(N(CC(CC)NC(C(CCCC#C)C)=O)C)=O)cc([N+](=O)[O-])c(C)cc1Cl c1(C(=O)NC2CC3CC2N(C(C2CC2F)=O)C3)cc2c(nc1O)CCCCC2 C1(NC(Cn2nc(C)c(C)c2C)=O)CC12CCC(NC(c1cccnn1)=O)CC2 n1(CC(N2CC(CC(C)NC(=O)Cc3cnoc3)C2)=O)nnc(C2CC2)n1 C=CC(C)(CCOC)C(=O)NC(C)C(=O)NC(C)CCC1CC1 C(=O)(CC(C)(C(F)F)N(C)C)N1CCC(C)(NC(C(CCOC)(C)C)=O)C1 C1(NC(C(C)OC2CCCC2)=O)CN(C(=O)Cc2c(F)cncc2Cl)CCC1F c1(C(N2CCC(CCC(=O)N(CCC)C3CC3)C2)=O)ccccc1C1CC1 N1(C(N2CC(C)N(c3ccccc3)CC2)=O)CC(CCO)C2CCCC12 c1(-c2nn(CC)c(C(F)(F)F)c2)ccc(N(C)C)cc1F C(c1ccc(C)cc1)=C(C(=O)NC(CN(C(c1ccc(CC)nc1)=O)CC)C)C CCCC(C)(O)C(=O)NCCCCN(C)C(C1(C)CCN(C(C)=O)C1)=O c1(OCC)ccc(C(=O)NC2CCC(C(=O)Nc3cnc(OC)cn3)C2)nc1 C1(NC(=O)Nc2c(OCCOCC)cccc2)CCOC2(CCS(=O)(=O)CC2)C1 C1(OC)CN(C(=O)C(C)(O)C2CCC2)CCC1NC(c1cc(Cl)cs1)=O C(=O)(CC(C(C)(C)C)NC(=O)CC1(N(C)C)CC1)NC1(CC)CC(C)(C)C1 CCN=c1[nH]c(C)c(C(=O)NCC(O)CN(C(=O)C(S(C)(=O)=O)C2CC2)C)s1 Cc1ncc(C(=O)NCC2CCN(C)C2)c(Cl)c1Br c1(C(=O)NCCOCCCNC(C(CCSC)O)=O)ccc(S(C)=O)cc1 C1(C)(NC(c2n(CCN(C)C)ncc2)=O)CCN(C(=O)CCC2CC(F)(F)C2)C1 N1(C(Cc2c(C)noc2)=O)CC(NC(=O)C=Cc2cscn2)C(O)C1 c1(-c2nc(CC(C)C)nn2-c2ccnc3ccsc23)ccc(F)c(S(C)(=O)=O)c1 CC1CC(NC(c2cnc(C3CC3)o2)=O)CCN1C(=O)CSc1nnc(S)s1 N1(C(C2(CCC)CC(=O)C2)=O)CCCC(CNC(C2CC(=O)NC2=O)=O)CC1 CC1(C(=O)NCC2(O)CC(NC(=O)CN3CCCC3CO)C2)CC=CCC1 c1(C(=O)NCCC(C)N(C(=O)CCc2ccoc2)C)ccn2ccccc12 c1(OC)ccc(CN2C(C(=O)Nc3cc(C4CCC4)no3)CC3CC23)cc1F c1(C(=O)NCC(C2CC2)NC(C#CC2(C)CC2)=O)ncn2cc(Cl)ccc12 c1(-c2ccc(C(N3CC(C(=O)OC)N(C)CC3)=O)cc2)nccn2nccc12 C1(CCS(=O)(=O)NC)NC(=O)CCN(CC(c2cccc(C)c2)(F)F)C1=O c1(OC)ccc(F)c(C(N2CCCC(C(=O)Nc3ccnc(Br)c3)C2)=O)c1 C1(CN(C)C)CCCN1C(=O)C(C1(O)CN(C(C2(Br)CC2(C)C)=O)C1)F C1(C(N2CC(NC(CC(C)C3CCCC3)=O)(CF)C2)=O)CC(F)(F)CS1 CCC(C(=O)N1CCOCC1CNC(c1c[nH]nc1C(C)(F)F)=O)C(C)C N1(C(c2cc(OC)no2)=O)CC(C(N2CCC3C(C(N)=O)C3C2)=O)C2(CC2)C1 c1(NCC(=O)NC)nccc(=NC(C)c2nc(O)n[nH]2)[nH]1 N1(C(C(=Cc2cnc[nH]2)C)=O)CCC2CN(C(=O)CCCN3CCCCC3)C2C1 N1(C(c2c(Cl)cc(C)c(C)c2)=O)Cc2ccccc2CC1CNC(=O)CC(C)F Cc1c(O)ccc(C(=O)NCC2CCN(C(c3ccc(Cl)nc3)=O)C2)c1C C1(CNC(C(C(C)C)OC)=O)CC2CCC1N(C(=O)CN1CCCC1=O)C2 N1(C(c2c(CNC(CC(C(C)C)C)=O)cc[nH]2)=O)CCC(O)CC(C)(C)C1 CP(C)(=O)C(CC(=O)NC12CCCCCC1N(C(=O)CCC#N)CC2)C(F)(F)F N1(C(CCCCC)=O)CCCCC(C(=O)NCC2CC2OC(C)=O)C1.OCC C(CC(=O)N1C2CCC1CC2)(C(F)F)NC(C1CCC(OC)CC1)=O C1(C(CC)NC(=O)NCCOCC(C)(C)OC)CN(C)CCO1 C1(C(=O)NC2CCC(CNC(C(CC)(F)F)=O)CC2)CCc2nccn2CC1 Cc1cc(C(=O)N(C)CCOCCCN(C(=O)C(F)n2cccn2)C)ccn1 c1(SC)ccc(OCCOC(=O)NC2C=CCC2)cc1 C1(NC(C2CC(CCC)C2)=O)CCC(NC(C2CC3C=CC2O3)=O)CC1 C1(NC(COCCN(C)C)=O)CS(=O)(=O)CC1NC(=O)C=CC1(C)CCOCC1 N1(C(CC2ON=C(C)C2)=O)CC(C)CC1C(=O)NC(c1cccnc1O)C CN1CCC(C(=O)NCCCn2cccn2)(NC(=O)C(F)=CC2CC2)C1 C1(CCOC)CN(C(=O)CSCCN(C)C)CCN1C(C1CC12CC(O)C2)=O C1(N(C2CCOCC2N(C)C)C(C2C3CN(C(C)=O)CC32)=O)CCCCC1(C)C N1(C(C2(C)C=CCC2)=O)CCC(C(F)CNC(c2cc(Cl)no2)=O)CC1 C(=O)(CCC(=O)NCc1cc(C(N2CCC(OCC(N)=O)C2)=O)n[nH]1)NC c1(OC)cc(Br)ccc1CNCCCCCN N1(C(C(C=C)O)=O)CCCC2CN(C(c3[nH]nnc3COC)=O)CCC12 C1(NC(CCN(CC)CC)=O)CC(OC)CN(C(C2CCC(C(C)C)CC2)=O)C1 c1(NC(C2C(NC(c3c(C)n[nH]c3)=O)C2)=O)ccc(I)c(C(F)(F)F)c1 C1(C(N)=O)CC1C(=O)NCCSCC(=O)NCCCOCF Cc1oc(C2CC2)nc1C(=O)NC1(C2CCCCN2c2nnc(C(F)F)s2)CC1 c1(COCC)cn(CC(C)(C)CNC(C2(CSC3CC3c3nccs3)CC2)=O)nn1 c1(C(=O)NC2C(CNC(c3cn(C)nn3)=O)C2)ccnc(-n2cncn2)c1 C1(C(=O)NC2C(C(=O)NCCCCC#N)CCC2)CCNC(=O)C1 c1(C(=O)OC)nc(NC2CCN(C(=O)CC3CC4(CC4)C3)CC2C)ncc1Cl N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2C(CCN2Cc2ncc[nH]2)C1 C1(C(=O)NC2CN(C(c3c(OC)nn(C)c3)=O)CC2C)CCn2c(cnc2C)C1 CC1(C)Cc2cccc(CNC34CCCC(CC3CO)C4)c2O1 N1(C(C)=O)CCC(C)(NC(=O)C(O)CN2CCCC2)C1.N12CCC(C1)C2=O c1(C(N2CC(NC(c3n(CCCC)ncc3)=O)C(C)C2)=O)cc(F)cc(C)c1N CCCCC(CC(=O)NCC(c1cccnc1)O)NC(C1CC1C(F)(F)F)=O C1(N(C(c2c(C)scn2)=O)C)CCCC(N(C(=O)Cn2cc(C(F)F)cn2)C)C1 c1(C)ccc(F)cc1.C1(C)(C(=O)OCC)CC1C(=O)N.C1C(=O)N(CC)CCCO1 CC1CCN(C(C23CC(C)(CO2)C3)=O)CC1NC(c1cccc(=S)n1O)=O C1(CNC(C(C)=CC)=O)CC2COCC2N1C(=O)C(O)Cc1ccccc1 N1(C(C2C(C)C2)=O)CCN(C(=O)C(c2cc(Cl)ccc2Cl)(C)C)CC1CCO N(C1CN(c2ncnc(Cl)c2F)CCc2ccccc21)C(C1C(=O)NCCC1)=O c1(CC)cccnc1C(=O)NCC(C1CCCN1C(=O)CN1CCCC1=O)(C)C Cc1cn2c(C(=O)NCC3(NC(C4C5CCN4CC5)=O)CCCC3)c(C)nc2s1 CCS(=O)(=O)CC(=O)NCCCCCN(C(=O)C(C)(C)C1CCCO1)C c1(C(=O)NC2(C(N(OC)CCO)=O)CCC(C)(C)C2)cccc2cncn12 CC1=NOC2(C1)CC(C(N1CCC(C)(C)C(NC(=O)CSCCN(C)C)C1)=O)C2 c1(-c2nnc(N3C(c4n(C)cnn4)CCCCC3)o2)nccc(Br)c1Br CC1CN2CCN1C(C(=O)NCC1CCN(C(=O)CCCC(N)=O)C1)C2 N1CCC2(CCCC2Nc2ncc(C#N)cc2F)CC1.c1(C=O)coc(Br)n1 c1(C(=O)NC2CN(C(C3C(C(C)C)CCO3)=O)CC(C)C2)c(F)cc(F)cc1F C1(NC(=O)NCc2c(NCCC)cccc2)CCN2CCCC12 C1(CNC(C(CCC)NC(C)=O)=O)(CO)CC12CCN(C(=O)C(C)NC=O)CC2 C1(NC(c2cc(C)ncn2)=O)CC2CCC1(NC(=O)CC1(N(C)C)CCC1)C2 C1(C(N2CC(CN(C(CC3(OC)CCC3)=O)C)C2)=O)CCCC2CC12 N1(C(Cc2cc(C)sc2)=O)CCN(C(C2CC3CCCC3C2)=O)CC1C1CC1.C1CC1 CCCC(C)C(=O)NCC1(CNC(=O)C(F)CN(CC)CC)CCOCC1 C1(C(=O)NC(C(=O)O)C2CC2)CN(C(c2ccc(-c3nccs3)cc2)=O)CCO1 O=C(N=c1ccn(C2CCSCC2)[nH]1)Nc1ccc(O)c(Cl)c1 C1(CC)CN(C)CCCN1C(C1CCN(C(=O)C(C)(C)O)CC1)=O Cc1cc(C)c(C(=O)NCC2(NC(=O)C=Cc3cc[nH]n3)CC2)c(S)n1 C#CC1CCC(C(=O)NC2COCCC2NC(c2[nH]nnc2C)=O)CC1 N1(C(CN(CC#C)C(c2ccn3ccccc23)=O)=O)CCC2CCC(C2)C1 CC(C)(C)CCC(F)C(=O)NC(CC1CCC1)C(N1Cc2cc(F)ccc2C1)=O N1(C(C(=O)Nc2ncc[nH]2)=O)CC(CNC(c2ccccc2F)=O)N2CCC1C2 C1(C(=O)NCC#CCC)CCCCCCN1C(c1ncc2ccccn12)=O c1(C(C(=O)NC2CCCN(C(c3cnc(C)[nH]3)=O)C2)C(C)C)ccc(C#N)cc1 c1(C(C)C)nc(NCC2CCCS2)cc(N2CCC(c3cc[nH]n3)CC2)n1 N1(C(C(N2CC(C)OCC2)=O)=O)CCCC2CCC(C)CC12 c1(C(=O)NC2CN(C(c3nc(C)c(C)s3)=O)CC2C)cc2oc(Br)cc2[nH]1 c1(C(=O)NC(CCN(C)C(C2CC2F)=O)C(C)(C)C)cc2ccc(F)cc2s1 c1(C(N2CCCCC(NC(CC(COC)(C)O)=O)C2)=O)ccc2c(c1)C(=O)OC2 C1(NC(CC(CCSC)O)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC1(C)C Cc1ncncc1C(=O)NC1CC2(C1)CC2NC(c1n[nH]cc1F)=O C1(CN2CCC(C(=O)NCCc3cn(C)nc3)C2)COC(C)(C)O1 c1(CNc2ccc(NC(c3ccccc3)CNC(C)=O)nc2)ccc(Cl)c(F)c1 CCC(C)(C)C(O)C(=O)N1CCC(C)C(NC(c2cc(C(C)C)oc2C)=O)C1C Cc1cn2cc(CC(=O)NCCC3CCCN3C(=O)CN3CCNC3=O)nc2s1 C(C(C)(C)C(=O)NCCCN1CCOCC1)N(C)C(c1cc[n+]([O-])cc1)=O c1(CC)ccc(S(=O)(=O)NC2CN(Cc3cccc(OC)c3)CC2(F)F)cc1 CC1CCCN(C(=O)C(=O)N(CCCCNC(C2CCCN2N=O)=O)C)C1 N1(C(C2(C)CC2(F)Cl)=O)CCC(NC(c2c[nH]cc2Br)=O)C(CO)CC1 C1(CNC(c2cc(CCC)oc2C)=O)CCCN(C(=O)C(C(C)C)OC)CC1 C(=O)(CC(C)CC(C)C)N1CCC(NC(c2n(COC)ncc2)=O)C(CO)C1 C12(CNC(CC(C=C)C)=O)CCCC(CN1C(=O)COc1cccc(C)c1C)C2 c1(C(C)C)ccc(CC(=O)NCC2CN(C(=O)CCCC3CCC3)CC2O)cc1 C(=O)(C1Cc2ccc(F)cc21)NC(CC=C)CNC(c1ccc(C)nc1C)=O c1(C(=O)NC2CN(C(C3(C#C)CCCC3)=O)CC2C)ccc(S(N)(=O)=O)cc1 c1(C(=O)Nc2n(C)nnc2)ncn2cc(-c3ccc(-c4cccnc4)cc3)sc12 Cc1ncc(Br)cc1NC(=O)C(O)C(F)F C(=O)(C(=O)N=S(C)(C)=O)NCC1CCCC(NC(c2c(CC)nc(C)nc2)=O)C1 CCCCC(C)C(=O)N1CCC(COC)(NC(c2c(C)cnn2C)=O)C1 C1(CNC(C2C(OCC)C2)=O)CC2(C1)CN(C(c1ccsc1C(F)(F)F)=O)C2 Cc1c[nH]c(CC(N)=O)c1C(=O)NCC(C)NC(=O)C(C)Cc1ccc(F)cc1 c1(OC)nc(NC(C2CN(C(C3CCCCN3C)=O)CCN2)=O)c(Br)cc1Br C1(CCN(C)C(C2CCCNC2=O)=O)CCCCN1C(=O)C(C)(F)F c1(NC(=O)COc2ccc(SC(F)(F)F)cc2)ccc2c(c1)OCO2 C1(C(=O)NCC(CC)(CC)NC(CC)=O)CCCC1C1CC1 c1(CC(=O)NCCN(CC(C)O)C(c2cnns2)=O)nccn1C CCS(=O)CC(=O)NC1CN(C(=O)Cc2c[nH]nc2O)CC1C C(N=c1[nH]c(N2CCC(c3nncs3)C2)nc2c1SCC2)c1cccc(CC)n1 C(C(C)(C(C)C)NC(C1CCN(C(C)=O)C1)=O)NC(C(C)(C)OC)=O C(=O)(C(C)(C)c1cscn1)N(C(CNC(c1cnc(C(F)F)s1)=O)C1CC1)C C1(NC(c2c(C#C)c[nH]n2)=O)CC1C1CCN(C(=O)CCOCCCOC)CC1 Cn1nc(C(N2CCC(CCC(=O)N3CC(n4cccn4)C3)C2)=O)cc1O C(=O)(C#CC1(C)CCCO1)NCC(CC(=O)NCCn1c(C)cc(C)n1)C C1(c2nnnn2CC2CCOC2)(NCCC=CC=C)CC1CCCC c1(N2C(CNC(C(C)=C(C)C)=O)C(C)CC2)ccc2c(n1)CC(C)(C)CC2=O N1(C(CCCCOCC)=O)CCC(NC(=O)CCSCC(N)=O)C(F)C1 C1(NC(CSCCCC)=O)COCCN(C(=O)CCC2COC(C)(C)O2)C1 N1(C(CC(=O)OC)=O)CCC(NC(c2ccc(C)c(C3CC3)c2)=O)C(F)C1 c1(NC2(C)CC(NC(C3CC(F)(F)C3)=O)C2)nc(C2CC2)nc2[nH]ccc12 C=CCC(CC)C(=O)NC(C1(O)CN(C(c2ccc(C(F)(F)CF)cc2)=O)C1)C N1(C(C(CC)C)=O)CC(CNC(c2cn(CCC3CC3)nn2)=O)C(O)C1 C1(CNC(c2cc(C)ns2)=O)CC(C)(C)CN1C(c1nn(C)c(Cl)c1Cl)=O C1(C(=O)NCC(C(N)=O)O)CCC=CC1NC(=O)CCCn1ccnn1 CC1CN(C(=O)CC(c2ccc(F)cc2)C)CC1CCNC(=O)C(C)(C)CF Cn1cc(Br)c(CS(N2CC(C(=O)O)C(C(F)(F)F)C2)(=O)=O)n1 CC1CCCC(C(N2CCCC2CC(=O)NCCOc2cccnc2)=O)C1 CN1CCn2cc(C(N3CCOC(CNC(=O)CCP(C)(C)=O)C3)=O)nc2C1=O N1(CC)C(=O)CCC1CC(=O)NCCC1(NC(c2n[nH]cc2C(F)(F)F)=O)CC1 c1(-c2n(C)nc(CCC(C)(C)C)n2)cc2ccccc2n1C(F)F c1(N2CCC(CC)(CO)C2)nc(NCC(C2CC2)OC)c2ccsc2n1 N1(C(c2c(CCC)n[nH]c2)=O)CCOC(C(=O)Nc2ccccc2)CC1 Cn1cc(C(=O)NCC(CNC(C2(n3nccn3)CC2)=O)CO)n(C)c1=O C1(C(=O)N(C2CCN(CC(C)C)C2)C)(COC)CCCN1C(=O)C(Cl)=CCl C1(NC(C(C2CCN(C(c3c(OC)n[nH]c3)=O)C2)C)=O)CCc2ncnn2C1 n1(CC(=O)NC2(CN(C(C(CC)(C)O)=O)C)CC2)c(C(N)=O)nc2ccccc12 CCCS(=O)(=O)C(C)C(=O)NCCN(C(=O)C1=C(C)OCCS1)C(C)C c1(C(N2CC(C)(CNC(CSCC#C)=O)OCC2)=O)cn2c(Cl)cccc2n1 N1(C(C(C)(C)C)=O)CCC(NC(=O)C(F)(F)Oc2ccc(F)cc2)CC1C1CC1 C1(C(=O)NCC(C)(C)NC(C=C(CC)CC)=O)CCc2c(cnn2C)C1 Cc1cc(C(=O)NCC2(F)CCN(C(=O)CC3NC(=O)NC3=O)CC2)nc(C)n1 c1(C(=O)NCC(Cn2cc(C(CC)O)nn2)(C)C)cc2c(C)n[nH]c2cn1 C12(CNC(Cc3cc(C)no3)=O)CN(C(C3CCCCS3)=O)CC1CCO2 N1(C(Cc2ccc(OCC)cc2)=O)CC2(CCCCN2C(=O)C(C)CF)C1 N1(C(C(C)(C)F)=O)CC(CC(=O)NC2COCC2CO)C2(CC2)C1 Cc1cccc(SCC(=O)NCC2CCN(C(C3CCCCS3)=O)C2)c1 C(C(CC(C)C)C(=O)NCC1CCCN1C)NC(c1cncc(C)n1)=O C1(CNC(CCOC)=O)CCC2(CCC2)C1NC(c1cccc(O)c1C)=O CCCC(O)C(=O)N1CCC1C(=O)NCCC(F)(F)CO C=CCC(C)(CC)C(=O)NCC(CO)NC(=O)CSC C1(CNC(C(CC)OC)=O)CCN(C(C2C=CCS2)=O)C12CC2 C1(C(=O)NCC(CC(=O)OC)C)CCC2CCC1N2C(=O)C(F)(F)C1CC1 C1(C(N2CCC(C3CCCCN3C(=O)CCF)CC2)=O)CC2CCC2C1 Cc1c(C(N2CCCC(CC(=O)NOCC(F)F)C2)=O)cccc1Cl c1(N2CC3C(C(=O)Nc4cn(CCOC)nc4C)(C3)C2)ncc2[nH]ncc2n1 C(C(C)(O)CC(=O)N1CCC(CNC(=O)C(C)(C)c2ccccn2)C1(C)C)OC N1(C(CCNC(=O)CO)=O)CCCC12CCN(C(c1ccoc1Cl)=O)C2 C1(C(=O)NCC2CN(CC)C(=O)O2)CC2CCC(C1)N2C(=O)CC(C)(C)C CC(CC(=O)NCC(=O)NCc1nncn1C1CC1)c1ccco1 NC(=O)CC(N=c1[nH]c2c(c(=NCC34CCC(CC3)O4)[nH]1)SCC2)C1CCCC1 CC1C(NC(=O)C=CCN(C)C)CC2CCC1N2C(=O)C(N)=O CC(C)CC(CC(C)C)(c1nnnn1C1(C)CC1)NC(c1cccc(Cl)c1F)C c1(C(N2C(C(N)=O)CCC2C(=O)O)=O)cccc2[nH]ccc12 Cc1ccc2c(=NC(C)c3ccc(Br)cn3)[nH]c(=NCC(C)CO)[nH]c2c1 CC1CN(C)C(=O)CN1C(=O)CCC(C)NC(c1cncc(F)c1)=O N1(C(CCN(C(C2CC(C)(O)C2)=O)C2CC2)=O)CC2(COC(=O)C2)C1 C=CC(C)CC(=O)NC1CCC(N2CCN(C(C3COC3)=O)CC2)CC1 c1(-c2c(OC)cccc2)nc(=NCC2CCCN2C(c2cscc2C)=O)s[nH]1 C1(C(N(C(C)C2CC2)CC)=O)CC(NC(=O)C(C)NC(C2CCC2)=O)C1 c1(OC)cccc(C(=O)NCCN(C(C2CC(Cl)(Cl)C2)=O)C(C)C)c1C C1(CC)(NC(=O)CC(F)(F)F)CCCN(C(=O)Nc2ccccc2C(C)(C)C)C1 C(CC)(CCC(=O)N(CC(O)CF)C)NC(c1[nH]cc(C(C)=O)c1)=O C1(C(N2CC(O)(CCNC(=O)C(CC3CCC3)OC)C2)=O)(SC)CC(=O)C1 N1(C(C2(C)CCNC2=O)=O)CC2(C1)CN(C(=O)C=Cc1cn[nH]c1)CCO2 c1(C(N2CCN(C(C3CCCCC3)=O)C3CC23)=O)ccc2c(O)nnc(O)c2c1 c1(C(=O)NCCC(CCC)C)ccnc2c1nnn2C CC(C)CC(O)CC(=O)NCc1ccc(C(=O)NC2CC3C=CC2C3)c(F)c1 C1(C(N2C(CC(=O)N(CCn3c(C)ncc3)C)CCC2)=O)CC2C=CC1C2 C1(NC(c2cc(SCC)ncc2)=O)CC2(CCCN(C(c3occc3Br)=O)C2)C1 Cc1cc(C(=O)NC(CNC(C2CCCC2O)=O)C(C)(C)C)nn1CCO CC1CCN(C(c2c(Cl)nsc2Cl)=O)CC1NC(c1occ2c1CCC2)=O n1(CCC(=O)NC2CN(C(C=CCC)=O)CC2(C)C)c(C)nc2ccccc12 c1(C(N(C2CC(=O)N(CCNC(c3ccccc3)=O)C2)C)=O)ccc(C(=O)O)nc1 CC(C)(Cc1ccc(Br)cc1)C(=O)NC1CC1NC(C1CC(C)(C)CO1)=O C1(C2CN(C(=O)CCCC3CCCO3)C2)(NC(Cc2c(C)cc(C)s2)=O)CC1 N1(C(c2c(CC)noc2)=O)CC(NC(=O)C(CC(N)=O)NC(C)=O)C(C)(C)C1 c1(C(=O)NC(CNC(Cc2cc(C)sc2)=O)C(C)(C)C)cnc2ncnn2c1C C12(NC(CC3(NC(C)=O)CC3)=O)CC(C1)N(C(c1scc(C)c1C)=O)C2 c1(C(N2CC3CC(C2)N(C(=O)CSCC(F)F)C3)=O)ccc2cncn2c1 C1(C(=O)NCCCC(C)NC(=O)CO)CC2(CCC2)C1 C(=O)(CC(C)C(=O)NCC(C)(F)CNC(C1CN(C)CCO1)=O)OC C1(COC(C2CC(C(=O)OC)C2)=O)CCCOC1.C1CC(=O)NC(=O)N1 N1(C(CC=CC)=O)CCCC1C1CCCN1C(=O)COc1cccc(Cl)c1C C1(OC)CN2CCCC2(C(=O)NC(c2cc(Cl)ccc2C)C)C1 C(c1ccc(Cl)cc1)=CC(N1CCC(CCNC(C2(Cl)C(C)(C)C2)=O)C1)=O c1(C(N(CCCCN(C)C(C2C3CCC(=O)C23)=O)C)=O)n[nH]cc1[N+](=O)[O-] C#CC1(C(N2CC3CC3(CO)C2)=O)CCN(C(c2cc(OC(C)=O)ccn2)=O)C1 C1(C(N2CC(COC)OCC2)=O)CC2CCC1N(C(=O)CCCN=[N+]=[N-])C2 C1(CCNC(=O)Cn2nccn2)CCCCN1C(c1ncncc1Cl)=O C(CCCCC(=O)N1C2CCC(C2)C1C(N1CCC(n2ccnc2)C1)=O)N(C)C C(CNC(C1CCCCO1)=O)(CC(=O)N1CC(F)(CO)C1)OC c1(C(=O)NC(CC)CN(C)C(C2CCCN(C)C2)=O)cc2cc(OC)ccc2o1 c1(C(=O)NC(CNC(C2(CCOC)CCC2)=O)(C)CC)ccc(F)cc1[N+](=O)[O-] C1(NC(=O)C=Cc2ncc[nH]2)C=CCN(C(C2CCC(=O)N2)=O)C1 c1(C(COC(C2C(C)(C(C)C)C2)=O)=O)ccc2ccccc2c1 c1(C(=O)NCCN(CCC)C(C2(F)CCOC2C)=O)cc(C)nn1C(C)(C)C c1(CCNC(C2(C)CSC2)=O)ccc(CNC(=O)CC2CCC(=O)N2)cc1 C1(C(=O)NC2CC3(C(NC(C4(C)COC4)=O)C3)C2)CC(F)(F)CCC1(C)C c1(C(N2CC(C)N(C(=O)Cn3ncnn3)CCC2)=O)cnc2sccn2c1=O CC(C)=C=CC(=O)N(CCNC(C1CCC(C)(C)C1)=O)CCOCCO C(=O)(CCN=c1ccc(C)c[nH]1)NC1C(NC(c2nn(CC)nc2C)=O)COC1 C1(C(=O)NCCN(C)C(C2CC3(CCC3)CO2)=O)CC(C)(C)CCO1 C1(CC(=O)NCC(CCNC(=O)CSc2ccncc2)O)CC2(CCC2)CO1 C=CCC(C(=O)N1CCC(CC)C1C(N1CCC1(CC)CC)=O)NC(C)=O C(=O)(CC(O)CC1CC1)N1CCC(OCC)C1 N1(C(CN(CC)CC)=O)CCC(NC(c2c(SC)cccc2F)=O)C1(C)C c1(C(N(CC(CNC(C(C)(CO)OC)=O)C)C)=O)cnc2cc(Br)ccn12 C(C(C)(O)CC(=O)NC1(C)CC(NC(=O)Cc2ccc(SC3CC3)cc2)C1)OC c1(-c2cn(CCN(C(C34COCC3C4(F)F)=O)CC)nn2)ccccc1[N+](=O)[O-] CC1(C)CCCC(C(C)(O)CNC(C2CC3CCC(C2)S3)=O)C1 c1(C(=O)NC2C(CNC(C(C=C)(C)CC)=O)CC2)c[nH]c2c(Br)cccc12 c1(OC)c(Br)cc(C(N2CCC(C)(c3ccccc3Br)C2)=O)cc1Br C1(C(N(CCCCCO)C)=O)CC12CN(C(C1CC(O)CN1)=O)C2 CC1C(C)N(C(=O)OC(=O)Cc2ccco2)CCN1C(=O)CN(C1CCC1)C C1(C)(CNC(CCOC)=O)CCN(C(=O)C(C)Cc2ccc(N)cc2)C1 c1(C(N2CCC(N(C)C(c3coc(O)n3)=O)C2)=O)cccc(C2CC2(F)F)c1 C1(CCOC)(NC(C2CCC3(CC3)C2)=O)CCN(C(=O)CCOCC2CC2)C1 C1(OC)CC(NC(c2cscn2)=O)CN(C(=O)C(C)(O)c2ccccc2)C1 c1(OC)cccc(-n2cc(CC3CCCN3CC3CC3)nn2)n1 C1(CC)CC(C(=O)NCC2C=CCN2C(=O)CCc2csc(C)n2)CC(=O)N1 C1(NC(C(C)CN2CCCCC2)=O)CCN(CCF)C12CCC2 Cc1ncc(C(=O)NC(C2CCCN(C(C3(S(C)(=O)=O)CC3)=O)C2)C)cc1N CC1(C)CCC=C(C(=O)NC2CCCC2Cn2cc(C3CCCCC3)nn2)C1 C12(CNC(C=Cc3nc(C)c(C)[nH]3)=O)CCCC(CN1C(=O)CC(C)C(C)C)C2 C1(CN(C2C(C)(C)CO2)CCO)CCN(C(=O)C(c2ccccc2F)O)CC1 C1(C(=O)NCC(C2CCN(C(CC3(C=C)CC3)=O)CC2)C)CN2CCC1CC2 C(CC(C(=O)NC(c1ccco1)C)NC(c1cc(Br)cs1)=O)SC N1(C(CCC#CC)=O)CC2(CC(CNC(c3ccc(OC(C)CC)cc3)=O)C2)C1 C1(c2n(CC)nnn2)(Nc2cc(COC)cc(C#N)c2)CCC2C3C=CC(C3)C12 C1(C(=O)OCc2cccc(OCC(=O)OCC=C)c2)CC2(CCO1)CC(F)(F)C2 C(CC1=CCOCC1)NC(C(CCC)NC(=O)CCOC(C)C)=O C(CC(C)(Cc1ccccc1)NC(C12CC3CC1C2C3)=O)NC(CC(=C)C)=O C(CCCCCNC(C1C2CCCC12)=O)N(C)C(C1CC(=O)N(C)C1)=O c1(CNC2C(C(=O)NCCc3ccccc3O)C2)cc2ccccc2cc1O C1(CCC(=O)N(C2(CCO)CC2)C)CCCCN(C(=O)CCCF)C1 C12(C(=O)NC3(CNC(C4CSC4)=O)CCCCC3)CCCC1CC(F)(F)CC2 C#Cc1cc(C(N2CCC(NC(=O)COCCCF)C(C)C2)=O)cc(Br)c1 Cc1cc2c(cc1Br)N(Cc1cc(C(=O)O)c(O)c(I)c1)CCO2 c1(C(=O)NC(C(C)NC(=O)CC(F)(F)Cl)C)cc(C(F)(F)F)cc(N)c1 c1(C(N(C2CN(C(c3ccc(Cl)[nH]3)=O)C2)C)=O)ccn2cccc2c1 CC1CC2(CC(C(=O)NCCCCC(=O)N3CCOCC3)C2)C1 C(=O)(CCC(C)(F)F)N1C2(C(=O)NCCOCC=C)CC2CC1 CC(C)CCC(O)C(=O)N1CCCC(CCC(=O)NCCN=S(C)(C)=O)C1 c1(N2CCC(CN(c3cncc(F)c3C)CC)CC2)ncc(C(F)(F)F)cc1Cl N1(C(CC)=O)CCC(CNC(=O)CCNC(c2ccccc2OC)=O)(OC)C1 CC1(C)CN(Cc2cc(C(=O)O)cs2)C(C)(C)C1O N1(C(C2C(C)(C)CC2)=O)CCn2c(CNC(C3(C)C=CCCC3)=O)nnc2C1 c1(OC)ccc(CN2CCC(O)(C(=O)NCc3cnn(C)c3)C2)c2ccccc12 c1(N(CCCS(C)=O)C)cc(S(=O)(=O)N2CCCCC2CCCO)ccc1C#N C1(C(=O)NC2CC(CNC(CN(CCC#C)C)=O)C2)CN2CCN1C(C)C2 N1(C(c2nn(CC)c(C)c2)=O)CCC12CN(C(c1cc(C(F)(F)F)n[nH]1)=O)C2 C1(COC)CN(C(c2cc(-c3ccn(C)n3)on2)=O)CCN1C(=O)CP(C)(C)=O c1(OCC)oc(C)nc1C(N1CC(CNC(=O)C=CC2(C)COC2)C(O)C1)=O C1(NC(C(C2(O)CCC2)NC(C=C(CC)CC)=O)=O)CN(C)C2(CCC2)C1 c1(CC(CNC(=O)NCCC2CC3C=CC2C3)CO)ccccc1F c1(C(N2CC(C(C)NC(C(C#C)(C)C)=O)OCC2)=O)cc(F)c(Br)cc1N C#CCCC(C(=O)N(C(C)C(=O)OC)C)NC(C1CN(C)C(=O)N1)=O c1(C(N2C(CCCC)CN(C(=O)C(C)O)CC2)=O)ccc(Cl)c(Cl)c1OC c1(OCC)cccc(NC(=O)C(C)N(C(c2cc(C)sc2N)=O)CC)c1 c1(CC)cscc1C(=O)NC1(CNC(c2cnsc2C)=O)CCOC1 CC(C)CCC(F)C(=O)N1CC(NC(C2CCNC(=O)C2)=O)CC(C)C1 C(C)(CNC(=O)CSc1nncn1C(C)(C)C)(C(C)C)NC(C(CC)F)=O C(CC(=O)NCCC(C(C)C)NC(C1CCC1)=O)(C(N)=O)NC(C)=O c1(OC)cccc(NC(N2CCN(c3cncc(OC)n3)CC2)=O)c1C#N O=C1CC(CNC2CCC(CCO)C2)CN1CCO O=C(NOC1CCCC1)C1(F)CCCC2(C1)OCCO2 C=CC1(CC(=O)NC2CC(NC(=O)C(C)c3ccco3)C2)CCOCC1 Cc1ccccc1C(=O)NC1CCC(CC(=O)NOCCOCCF)C1 Cc1ccc(C(N2CC(C(C)NC(C3C=CC=CC=C3)=O)C2)=O)cn1 C1(C(N2CCC(N(C(=O)Cc3csc(NC=O)n3)C)C2)=O)CC2CC1CO2 C(c1ccccc1OC)=CC(N1C(CNC(c2ccc(OC)s2)=O)CCC1)=O Cc1c(O)c(=O)ccn1CC(=O)NC1CCN(C(=O)CN2CCCCS2(=O)=O)C1 C1(N(C(=O)C(C)CC(N)=O)C(=O)OC(C)(C)C)CC2C(C1)C2(F)F c1(C(=O)OC)ccn2c1CN(S(=O)(=O)N1CCC1C(=O)OC)CC2 c1(NC2CCN(C(Cn3ccc(C)n3)=O)C(C)C2)ncnc2c1nnn2C(C)C c1(CNC(c2scc(CNC(=O)CC3CC(=O)NC3=O)c2)=O)cccc(C#N)n1 CCCCCC(C)(C)C(=O)NC(C)CNC(=O)CCc1cccnc1F Cc1ccnc(Cl)c1NC(N1CC2CC(NCC(c3ccccc3Br)F)C1C2)=O C1(NC(C)=O)CCN(C(=O)CC2CCC2C)CC1.C1(=O)CN1C c1(C(N(C)CC2CCCN2C(=O)CCF)=O)cc2cccc(Br)c2[nH]1 CCC(CC(=O)N1CC(NC(c2nnsc2C(F)F)=O)C(C)C1)c1ccccc1 N1(C(C2C(C)=C2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)C2(CCC2)C1 Cc1ccc(NCCC(N2CC(NC(c3cnncc3O)=O)CC2C)=O)cc1 c1(N2CCC(NC(C(CCC)N(C)C)=O)C(F)C2)ncc([N+](=O)[O-])cc1C N1(C(c2cc(CNC(C=CCCC)=O)sn2)=O)CC(C2CC2)C1C1CC1 C(C(N)=O)(C(F)(F)F)NC(C1N(C(c2c(C)cnnc2)=O)C(C)C1)=O c1(OCCOCC(=O)N(CC(CC)NC(=O)CC2C=CCC2)C)cccc(C)c1 C1(NC(C2C3CCC2(c2ccco2)C3)=O)CCCCN(C(C2C3CCCC23)=O)C1 C1(NC(CC23CC(C)(OC2)C3)=O)CCC2CCN(C(C3CC3(F)F)=O)C1C2 S(=O)(=O)(c1ccc(C)cc1C)NC(CC)C(=O)NC1CCCCC12CCNCC2 c1(CCC(=O)NCC2C3CC2N(C(=O)C=Cc2ccoc2)C3)ccc(F)cc1F N1(C(c2cnc(N3CCOCC3)nc2)C(=O)NC)CC(CCN)CC1(C)C c1(NC(CNC(CCNC)C)=O)cc(Br)c2c(c1)OCCO2 c1(OCCOC)ccccc1NC(N1CCC(c2ccn(C)n2)CC1)=O C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(CCC(=C)Cl)=O)(CC)CC1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCO3)=O)C2)ccccc1O N1(C(c2ccc(C(C)=O)nn2)=O)CCC(NC(c2cnc(C)nc2)=O)C(F)C1 C1(OCC(=O)NC2(CC#C)CC2)CC(NC(C2CC2(C)CC)=O)C1 c1(N2CCCC(CCC)CC2)nc2c(c(=NC(C)C3CC3)[nH]1)SCC2 C1(CNC(C(C(C)C)N(C)C)=O)CC2CN(C(c3cc(O)cc(Cl)c3)=O)CC12 c1(C(=O)NC(CNC(c2cccc(SCC)c2)=O)C)ccc(C(F)(F)F)cc1N c1(CNC(C2C(C=C)OCC2)=O)ccc2c(c1)CCOC2.C12CCCCN1C2=O c1(C(N2C(CCNC(C(C)C3(O)CCC3)=O)CCC2)=O)coc2c1CS(=O)(=O)C2 n1(C(C)C)cc(Br)c(=NC(=O)c2cnn(C)c2)[nH]1 N1(C(C(C)n2cccn2)=O)CCCC(CC(=O)Nc2ccccc2Br)C1 C1(NC(c2cc(OCC)n[nH]2)=O)CC2CCC1N2C(=O)CC1CCCC1(F)F N1(C(C(CC)N2CCCC2=O)=O)CC2(CCC(NC(=O)C=CC(F)(F)F)CC2)C1 C(C)(CCCCCO)NC(C1(C2N(C(c3nc(C)oc3C)=O)CCC2)CC1)=O C(CN=c1[nH]c(=N)[nH]c(=NCCCC2(C)CC2)[nH]1)c1nc(C)nc(O)c1 C1(OC)CC(C(N2CCSCC2)=O)N(C(c2cc(-c3ccnn3C)cs2)=O)C1 c1(C(N)=O)cccc(C(=O)NC2CC(NC(C3OC4CCC3C4)=O)C2)c1F c1(C(=O)NC2C(CNC(CC=C)=O)C2)nn(C(C)C)nc1Br CCC(C#N)(CC)C(=O)N1CCCCC(CNC(=O)Cn2nc(C)n(C)c2=O)C1 c1(SC)cccc(F)c1C(N1CC(NC(C2CCCCN2C)=O)C(O)C1)=O N1(C(Cc2ccn(CC)n2)=O)C2CCCC1CN(C(c1cc(C)cc(F)c1)=O)C2 Clc1nsc(NCCn2ccc(Br)n2)n1 N1(CC(CN(c2ccc(OCC(C)N)cc2)C)O)CCN(C)CC1.C(=O)O c1(NC2C(C)CCC2)cc(C(F)(F)F)nc2c(Br)cccc12 C1(NC(C2(C)CC=CC2)=O)CCCCN(C(=O)CN2CCCC2=O)CC1 C(=O)(CCC(=O)N(C)C)NC(C1CCCN(C(=O)C(C2CC(F)(F)C2)O)C1)C CCC(CNC(C1CCN(C)C1)=O)(CC)NC(c1ccc(C(N)=O)nc1)=O N1(C(CN(C(=O)C(C2CCOCC2)F)C)=O)CCC(C2CC2)(NC(N)=O)C1 c1(C(=O)NC(C)CNC(=O)Cc2nc(C(F)(F)F)n[nH]2)cnn(C)c1N CCC(CC)C(C(=O)N1CC2CC2(NC(=O)C(C)c2cc[nH]n2)C1)OC C=CC1CCCCN1C(c1c(Cl)ncn1C)C(=O)NCC(C)C C1(CNC(c2cc(CC(C)C)[nH]n2)=O)(NC(=O)CC(C)(F)F)CC(F)(F)C1 c1(CSCC(=O)Nc2ncc(-c3ccccc3F)o2)ccccc1Br CCS(=O)(=O)CCn1c(N(C2CCCC2)Cc2nccs2)nnc1CC(C)C C(CCCCN(C(=O)C(C1CCCC1)C1CCCC1)C)NC(CN(C)CC)=O Cc1cc(C(=O)NCC2N(C(=O)CS(N)(=O)=O)CCCC2(C)C)c(N)c(Cl)n1 c1(OC)cc(C(=O)NC2CC(C)N(C(C3CCC(C)CC3)=O)C2)cc(N)c1N C1(NC(C2CC(OC)C2)=O)CCN(C(=O)CCSC2CCCC2)C(C)C1 C#Cc1ccc(C(N2CC(CNC(=O)C(F)(F)C(F)(F)F)OC(C)C2)=O)cc1C C12(NC(CC)=O)CC(C)(C1)OC21CN(C(c2ccc3nc(=N)[nH]n3c2)=O)C1 n1(CC(=O)NC2C(C)(C)CN(C(=O)C3=COCCC3)C2)ncn2cccc2c1=O O=C1CCc2cccc(C(=O)NC34CC(C3)N(C(=O)CNS(N)(=O)=O)C4)c2N1 C1(NC(C2ON=C(C)C2)=O)CCN(C(c2ccccc2C)=O)CC1 CN1CCN(C(=O)CCc2cncnc2)CC1NC(=O)COCC(C)(C)C c1(C(=O)NC2COCC2CNC(C2CC23CCCC3)=O)sc2ncccc2c1Cl N1(C(CC(CC)C)=O)CCC2(CC1)CN(C(C1CCN(c3nncs3)CC1)=O)C2 C1(c2ccc(C(c3ccccc3)=O)c(F)c2)CN(N2CC3CCCCCC3C2)C1 CC(C)C(O)C(=O)NC(C1CCCCN1S(C)(=O)=O)=O.C1CN(C2CC2)N1.NC c1(C(N(C(CN(C(c2c(CC)nco2)=O)C)C)C)=O)cc2nc(C)[nH]c2cc1F N1(C(C(=O)N(C2CCCNC2)CC(C)C)=O)CCC(CCCF)CC1 c1(C(c2n(C(CC)Nc3cccnc3)nnn2)(C)C)cc(Br)cc(C)c1F C1(COC)CCN(C(=NCCc2ccc(F)cc2)NCC(c2nc(C)cs2)C)C1 C(=O)(C(CN=[N+]=[N-])NC(=O)C(C(=O)OC)OC)Nc1cnc(CC)nc1 c1(C(=O)NC2CCCN(C(=O)Cn3nccn3)C2C)cnc(OC)c(N)c1.COCBr c1(OC)ccc(CC(=O)N(CC(CO)(CO)NC(=O)C(C)CSC)C)c(C)c1 N1(C(c2cnn(C)c2C#N)=O)CC2CC(NC(C3CC34CCOC4)=O)CC1C2 C1(OCC)CC2CN(Cc3cc(C(=O)O)ccc3OCC)CC12 C(CCC(=O)O)(C(N)=O)NCC1CCN(C(=O)OC(C)(C)C)C12CC2 n1(CC)cc2ccc(NC(=O)NC3(C4CCC4)CCCC3)cc2n1 N1(C(C2CC(NC(COCC(=O)NCC)=O)C2)=O)CC(O)(c2ccccc2)C1 O=S(=O)(c1ccc(Br)s1)N1CCCC(Oc2ccccc2OC(F)(F)F)C1 c1(C(=O)NC(CC)CNC(c2cnccc2C)=O)ccc2c(C)cc(Cl)nc2c1 C1(C(=O)NC2(C(N(CC)CC)=O)CC2)COC(=O)C1 c1(CC(=O)NCC(CN(C)C(C2CC2c2ccco2)=O)O)nc2c([nH]1)CCCC2 C1(C(N2CC(O)(CC=C)C2)=O)CNC(=O)CN1C(=O)CSCC(N)=O C1(CC(=O)N(CC(CC)NC(c2cnc(C(N)=O)cn2)=O)C)CCCCC(=O)N1 n1(CC)ncc(C(=O)N(CCCn2cc(COCCN(C)C)nn2)C)n1 c1(C(=O)OC)cnc(C(=O)N(C(C2CC2NC(=O)C2CC2)C)C)o1 c1(C(C2CCC2)NC(c2n(CC)nnn2)c2coc(C)n2)ccc(F)cc1 Cc1ccc(Cl)c(NC(N2CCCN(CC(=O)Nc3ccccc3)CC2)=O)c1 CCC(C)(C)C(O)C(=O)NC(c1ccccc1)CNC(c1cccc(OC)n1)=O C(=O)(NNC(=O)C(C)(C)CCCCNC(c1cnc(CC)[nH]1)=O)C1CSC(C)=N1 Cc1ncnc(C(N2CCN(C(c3cc(C4CC4)[nH]n3)=O)C(C(F)F)C2)=O)c1C c1(NC(C2CN(C(C3(F)CCC3)=O)CCO2)=O)ccc(I)c(Br)c1 C(=O)(C1Cc2ccccc21)NCCCCCNC(C(CNC(C)=O)(C)C)=O C(C1=CCN(C(c2ccc(C(F)F)cc2)=O)CC1)NC(C1CC12CC(O)C2)=O Cc1ccc(F)c2[nH]c(C(=O)NCCN(C(c3ccnc(S)c3)=O)C3CC3)cc12 c1(C(=O)NCCn2cc(C(N3CC=CC3)=O)nn2)ccc(O)cc1 C=CC(C)C(=O)NC1CC(CNC(=O)CN(C)CCOC)C1 c1(C(N2CCCC(NC(C(CC)(C)OC)=O)CC2)=O)cc(C)c(C)c(F)c1 C12(NC(C3CC(N(C)C)C3)=O)CCCC1CN(C(=O)CC1CCCCC(=O)N1)C2 c1(NC2CN(C)C2)[nH]c(=NCc2c(Br)cccc2Br)nc2scnc12 C#CCCN=C(NCC(C1CC1)Sc1ccc(Br)cc1)N1CCC(NC(C)=O)C1 N1(C(C2(NC(=O)CC(=O)N(C)C)C(C)CCC2)=O)CC2CCC(C1)C(=O)O2 c1(CC)cccc(C(=O)NC(C2CCN(C(c3[nH]ccc3C)=O)C2)C)c1 C1(C(N2CC(OCC(=O)NCc3n(CCC)ccn3)C2)=O)CC2(CC(=O)C2)C1 c1(CC(=O)NCCCNC(c2cc3cc[nH]c3cn2)=O)ccc2c(c1)CCOC2 N(C)(C(=NCc1ccccc1)NC1CCC(c2cc(F)cc(Cl)c2)C1)CC.CC=O c1(N2CCC(CCNC(C(CC)N(C)C)=O)C2)ncnc2cc(Br)ccc12 Cc1cc(=N)[nH]cc1C(=O)NCC(C)(C1CCC1)NC(c1cccs1)=O c1(C(=O)NC2CC3(C(NC(C(CC(C)(C)C)O)=O)C3)C2)cc2ccoc2cc1F N1(C(C2(C(C)NC(=O)CCCF)CC2)=O)CC(=O)NC2(CC2)C1 CCC(CO)CCNCc1cc(C(F)F)nn1C C1(C(N2C3CC(=C)C(C3)C2)=O)C(C2CC2)CCN1C(=O)CCC=C(C)C Cc1cc(S(N)(=O)=O)ccc1CNC(=O)NCCc1cnnn1C c1(C(N2CCC(NC(c3nnn(CC)c3C)=O)C2)=O)cncc2ccc(F)cc12 Cc1cc(Br)cc(C(N2CC(NC(C3OCCN(C)C3=O)=O)C2)=O)c1F C1(CNC(C(CC)O)=O)C(CC)CCN1C(=O)C=NOC C1(C(N(C2CCN(C(c3cc(C)c(C)nn3)=O)C2)CC)=O)CCC(F)(F)CC1 c1(C(N2CC(CC(C(=O)N3CC(C=C)C3)F)C2)=O)ccc(C)nc1C C(CN=C(NCC1(F)CCCCC1)NC1CC1)=C(C)C1CC1 N1(C(CC(CN(C)C)O)=O)CCc2[nH]nc(CNC(C3(C)CC=CCO3)=O)c2C1 CC(C)CCCCC(=O)N1CCCC(CNC(=O)C(C)CCn2cccn2)CC1 CCC(O)C(C)C(=O)NCC1C2CC1N(C(c1cc(F)ccc1C(F)(F)F)=O)C2 C1(N=[N+]=[N-])(C(=O)NCc2nc(C)c(C)o2)CCN(C(C2CN3CCC2C3)=O)C1 C12(NC(C3CC4(C3)CC(F)C4)=O)CCCC1N(C(c1ccc(O)cc1)=O)CC2 c1(C(CNC(=O)CC2CCNC2=O)NC(=O)CCCC2CC2)ccc(Br)cc1 Cc1cncc(CC(=O)NC(C)(CNC(C2CC2(C)C)=O)CO)c1 N1(CCC(C(C)C)N)CCC(O)(C2CCC2)CC1 C1(C2CC2)(NC(Cc2n(C)ccn2)=O)CCN(C(=O)COc2cccnc2)C1 N1(C(C(COC)O)=O)CC2CC(NC(c3occ4c3CCC4)=O)C(C2)C1 C12(NC(=O)CCn3cnccc3=O)CCCC1N(C(C1CSC1)=O)CC2 c1(C(=O)NC2(C)CC(NC(CSCC(C)C)=O)C2)ccc(F)c(C(F)(F)F)n1 CC(C)C(O)CC(=O)NC1CN(C(=O)C(O)C(C)C)CC1O N1(C(CCC=C(C)C)=O)CCCCC2(C1)CN(C(c1cncn1C)=O)C2 c1(C(=O)NC(COC)C(=O)NCc2ncco2)ccnc2cc[nH]c12 C=C(C)CC(C)C(=O)NCC(C)(CO)NC(=O)CC1(O)CCOCC1 c1(C(=O)NCCCN(CCO)C(C2C3CCCOC23)=O)cn2ccnc2cn1 C1(N(CC(=O)NCC(C2CC=CCC2)NC(CSC)=O)C)CCCC1O c1(CN2CC(c3n(C)ccn3)C3(C2)COC3)cc(CN)cc2c1CCC2(C)C N=c1cc(C(N2CCC(NC(=O)C(Cl)=CCl)C23CC3)=O)c(Br)c[nH]1 C(=O)(C(C)(C)CC(F)F)N(CC(CNC(CC1CCC(C)C1)=O)C)C CC1CC(N=c2ccc3c([nH]2)CCCC3=O)c2ncnn21.C12(CCC1)C(=O)N2 C1(C(N)=O)CCC(NC(C2CCCCC2c2ccccc2)=O)CC1 Cc1[nH]c2ccccc2c1CC(=O)NC1COCCN(C(=O)CCS(N)(=O)=O)C1 C1(NC(C2(CCNC(=O)CCn3cccc3)CC2)=O)CC(C2CCCC2)C1 C1(NC(Cc2c(C)ncs2)=O)CCC(S(C)=O)C1 c1(C(N2CCCC(N(C(c3ocnc3C)=O)CC)C2)=O)ccc(N)c(N)c1 N1(C(C(C)n2ccnc2)=O)CCC2C1CCCN2C(c1cc(Cl)cc(F)c1Cl)=O c1(C(=O)NC2C3(CC(NC(COCC=C)=O)C3)C2)ccc(N)cc1C Cn1ccc(=O)c(CC(=O)NCc2nc(C3CCC3)no2)c1 CCCC(C)(CCC)C(=O)N1CC2CCC2(CNC(c2cnccc2OC)=O)C1 C1(C(=O)NCc2cncc(CC)c2)CN(C(c2cc(F)n(C)n2)=O)CC12CCC2 CC1CN(C(c2c(F)cccc2Cl)=O)CCCN1C(C1CCCC1(F)F)=O CCCCCC(C)(C)C(=O)N1CCC(N(C(=O)CCCN(C)C)C)C1 c1(-c2cc(C)[nH]n2)ccc2ncc(C(N3CCC(CF)CC3)=O)c(Cl)c2c1 C1(CNC(c2nc(C(C)=O)sc2)=O)CC(C)(C)CCC1NC(c1ccc(C)s1)=O C12(C(N(CC(N3CCCC(CC=C)C3)=O)CCC)=O)CCC(CC1)CC2 C(C(=O)NOC(CC(C)C)C(=O)NCC(c1ccccc1)O)(C(C)C)SC N1(C(C(CCC)NC(=O)CC2CC2C2CC2)=O)CC(C)OCC1C N=c1[nH]cncc1C(N1CC(C)(OCC(N2CCOC(C(N)=O)C2)=O)C1)=O C12(CNC(c3c(C(N)=O)csc3)=O)CCC1CCN2C(c1ccsc1)=O C(=O)(C(C)(CC)C(=O)NCC1(O)CN(C(=O)COc2ncc(F)cn2)C1)OCC c1(CC(CCOC)NC(CC)CC2CCOCC2)ccc(F)cc1F CC1(C)CCCCC1C(N1CCC(=CC(N2CC3CC2CO3)=O)CC1)=O c1(CCC(=O)N(C(C)CCNC(C2COC2)=O)C)ccccc1Cl n1(CC)nc(C(=O)N(C)CCNC(=O)C=Cc2nccs2)cc1C C1(CNC(C2(COC)CC2)=O)CCC2(CN(C(c3nnc(O)nc3O)=O)C2)O1 c1(C(N2Cc3c(C(=O)OCC)ncn3CC2)=O)cc(F)cc2cc[nH]c12 N1(C(c2ccc(CN(C)C)o2)=O)CCN(C(C2(C)CCCCC2)=O)CC(C)(C)C1 C(=O)(CCCCCS(N)(=O)=O)NCC(CN(C(=O)CCn1cnnn1)C)O Cc1cccc2c1OC(C(=O)NCCCN(C)C(C1C(C)(C)OC1(C)C)=O)C2 c1(CC)ccccc1OCC(N1CC(NC(=O)CC2CCC(=O)N2C)C(C)C1)=O Cc1nc(O)ccc1C(=O)N1CCC(C(=O)NC2CC3(CCCC3)C2)O1 c1(CC(=O)NC2(CO)CCN(C(c3cc(OC)ns3)=O)C2)cccc(Cl)c1F CC1CC(C(=O)NCC2CN(C(c3snc(Cl)c3Cl)=O)C2)Cc2nn[nH]c21 N1(C(COCCC=C)=O)CCC(C)(CNC(=O)C(c2ccc(C)o2)C)CC1 N1(C(CC(=C=C)C)=O)CC(NC(=O)C=Cc2nccs2)CC2(CC2)C1 Cc1c(Cl)ccnc1C(=O)NCC1(CNC(=O)CC2CCN(C)C2)CCCC1 C(=O)(CCC[N+](=O)[O-])N(CC(CNC(C(c1ccncc1)C)=O)C)C C1(CO)CCCCCC1OCCn1cc(C2(COCCO)CCC2)nn1 C1(N=c2[nH]c(=NCC3CCCO3)c3c(F)cccc3[nH]2)(CCOC)CCC1 N1(C(c2cncc(C)c2Cl)=O)CCC2CN(C(=O)CC3CCCC34CC4)C2C1 C1(S(N)(=O)=O)(C(=O)NC2C(CNC(c3n(CCC)ncc3)=O)CCCC2)CCC1 CN1CCN(C(C2CC3CCC3C2)=O)C(C(N2CC(C3CCCO3)C2)=O)C1 c1(C(=O)NCC2CCCN2C(=O)CCc2cccc(CO)c2)ccc([N+](=O)[O-])o1 C12(SCCNC(CC(CCC)O)=O)CC3CCC(C1C2)N3C(=O)OC(C)(C)C N1(C(C(CCC)N(C)C)=O)CCC(NC(=O)CC(C)(C)O)CC(C)(C)C1 c1(OC(C)C)cncc(=NC(=O)C(=O)NC2CCC(=O)N(C)C2)[nH]1 C1(C(N2C(C)(COC)CC2)=O)CCCCCC1NC(c1sccc1C)=O c1(C(N2C(C)C(C)N(C(c3cscn3)=O)CC2)=O)cnn2c1OCC(C)(C)C2 S(=O)(=O)(c1ccc(NCCOC2CC2)nc1)NC1CC(C)SCC1 C1(C(C)NC(=O)CC2CC(C(F)F)C2)CN(C(c2nccnc2N)=O)CCO1 C(=O)(C(C)C(O)CC(C)C)NCC1CCCN(CC(=O)OCC)C1 C(CC(CNC(c1cnoc1-c1ccoc1)=O)NC(C12CC(F)(C1)C2)=O)OC C1(CC)CCN(C(C2CNC(=O)N2)=O)C1C(=O)NC(C(C)C)c1ncc[nH]1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nccn2)cncc(P(C)(C)=O)c1 C=C1CC2CC1CN2C(c1ccc(C(F)F)o1)C(=O)NCCCF C(C)(C)(C(C)NC(=O)Cc1ccc(Cl)s1)NC(CCC1C(C)C1)=O Cc1cccc2sc(NC(C3CCN3Cc3ccc(O)c([N+](=O)[O-])c3)=O)nc12 c1(CC(=O)NC(CN(C)C(C2CCCC(C)(C)C2)=O)(C)C)cc(F)c(F)cc1F Cc1c(C(=O)N(C(C)(C)CC(=O)NCCC2CCC(C)O2)C)cncc1F N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(C2CCCCC2)=O)C(C)C1 Cc1nn(C)c2c(NCC3C4CCCC34)nc(=NCc3cscn3)[nH]c12 N1(C(C(c2ccc(C)cn2)(F)F)=O)CC2CCCC(C1)N2C(=O)CC1CC1C n1(CC(=O)NCCC2CC(NC(c3c(C)noc3)=O)C2)ccc(=O)c([N+](=O)[O-])c1 Cc1cc(C(F)(F)F)c(C#N)c(=NCCSCCc2ncnc3ccccc23)[nH]1 C(=O)(CC(CC)c1ccccc1)N1CCC(N(C(=O)Cc2cnoc2)CCC)C1 c1(C(C)C)ncncc1C(N1CC(CNC(=O)CC2(O)CCOC2)CC1C)=O C1(CC(C)NC(C2(C(=O)C3CC3)CC2)=O)CCN(C(=O)CCS(C)=O)CC1 c1(C(N2CCC(C(C)NC(=O)CCCN3CCCCC3)C2)=O)cncc(F)c1Cl c1(C(=O)NCCN(C(Cc2c(CC)con2)=O)CC(C)O)cccc(OC)c1F c1(CC(=O)NC23CCN(C(c4ccnc(O)c4)=O)CC2C3)ccc(Cl)cc1F C1(CC)(NC(c2ccc(O)c(N)n2)=O)CCN(C(c2[nH]c(O)nc2C)=O)CC1 Cc1ncc(C)c(=NCCC2CCN(C(c3cnn(CC(F)(F)F)c3)=O)C2)[nH]1 C1(CNC(CC2(C)CC2(Cl)Cl)=O)CCCN(C(c2cccc(Cl)c2N)=O)CC1 c1(C(N2CC(NCc3ncn(C)c3)C2)=O)ccccc1S(=O)(=O)N1CCCCC1 c1(CCCc2cc(C)[nH]n2)nc(-c2ccco2)nn1C1CCOC1 Cc1cc(O)cc(O)c1CNC1CC(C(N2C3COCC2C3)=O)C1 c1(C(=O)NCCC2CCCCN2CCC(C=C)C)ccc(Br)cc1N1CCOCC1 C(=O)(C(C)(CCC)CCC)NC1C2CN(C(C3(CC=C)CCOCC3)=O)C1CC2 C1(C(=O)NC2(CCCCNC(CCOCC(C)C)=O)CC2)CC(O)C(F)C1 C1(C(N2C(C3CCN(C(CNC(N)=O)=O)CC3)CCC2)=O)Cc2cccnc2C1 N1(C(C2(C(=O)OC)CCCC2)=O)CC2CN(C(=O)CC3CC(C)(C)C3)CC2C1 C(=O)(C(F)(F)C(C)(C)O)NCC1C2N(c3cc(C(=O)OC)nc(Cl)n3)C(CC2)C1 C1(NC(CCCCCCCC)=O)CCOC12CCN(C(C1(OC)CC1)=O)CC2 C1(NC(c2c(C)ccnc2)=O)CCCC(NC(c2ccc(C#N)s2)=O)CC1 C1(CC)(NC(=O)Cn2cc(CN3CCC(O)CC3)nn2)CCSCC1 c1(C(=O)NC2(c3ccccc3)CCN(C(C)=O)C2)ccc2c(c1)B(O)OC2 C1(CCNC(=O)CC2CCC(=O)O2)CCCCN1C(c1cc(C2CCC2)no1)=O C=CCC(C)(C)CC(=O)NC1CN(C(c2cncc3n[nH]cc23)=O)CC1O N1(C(C(COCC)c2ccccc2)=O)CCC(c2ccc(C)cc2)CC1C c1(CC(=O)NCCn2cc(C(=O)NC3(C#C)CC3)nc2)ncccc1C c1(C(=O)OC)c[nH]c(=NCC2CCCCN2C(=O)C(=O)NC2CC2)s1 C(C(C)(C)CNC(=O)CC1(O)CCOC1)N(C(=O)COC(F)F)C N1(C(Cn2c(C)nnn2)=O)CC(C(N2CCN3CCCC3C2)=O)C2(CCC2)C1 Cc1ccc(C(=O)C(N2CC(NC(=O)CN3CCSCC3)CC2C)=O)cc1 N1(C(C2(C)C(CC)CCC2)=O)C(CNC(=O)CCC=CC(C)C)CC2CCCC12 CC(C(=O)N1CCC(n2cc(C3CC3)nn2)C1)S(N)(=O)=O CC(C)(C(=O)N1CCC(C)(NC(c2ccc(N)cc2Cl)=O)C1)C1=CCSCC1 c1(C(=O)NC2CC(C)N(C(C3CC(=O)CCO3)=O)CC2)cn2cccnc2n1 c1(OCC)ccc(C)c(F)c1-c1ccc(C(=O)NCC2(O)COC2)nn1 N1(C(C2CCC(C)O2)=O)CCCC12CCN(C(c1cc(C3(C)CC3)on1)=O)C2 c1(CCC(=O)NCC(O)CNC(=O)C(=O)Nc2ncc[nH]2)ccncn1 c1(OC)c(C(=O)NC2COCCN(C(=O)C(C)c3ccco3)C2)c(C)nn1C CCC(C)(C)C(=O)N(C)Cc1ccc(CNC(C2(n3nccn3)CC2)=O)cc1 C(=O)(C(CCF)NC(=O)CCCn1cncn1)N(CC(=O)NC(C)C)C C1(NC(c2cccc(NC(C)=O)n2)=O)CCN(C(=O)Cn2cccc2)CC12CC2 c1(C(N2CCC2C(N2CCC(c3ccc(Cl)cc3)C2)=O)=O)n[nH]c2cccc(F)c12 C(C(C)(CC(C)C)NC(=O)C#CC1CC1)NC(c1c(CC)nco1)=O c1(NC(=O)NCCC)cccc(NC(=O)CCNC(c2nn(C)cc2Br)C)c1 C(=O)(C1=NOC(C)(C)C1)NCCC(C(C)C)NC(c1cc(C)c(Cl)s1)=O CC1CN(C(c2cc(Cl)sc2Cl)=O)CC2(CCN(C(C3CCC(=O)NC3)=O)C2)O1 C1(CCC(=O)NC(C)C(CO)NC(c2cnc(S)n2C)=O)CCC(=O)NC1 CC(C)CCN=C(NCc1ccc(Br)s1)NC1CC1c1c(Cl)cccc1Cl c1(C(=O)NCC(CC)NC(C2(F)CCCC2)=O)ccccc1CCn1ccnn1 CCCCC(CNC(c1ccc(C(F)F)nc1)=O)NC(C1CCCOC1)=O c1(NC(C2C(NC(C(CC)COC)=O)CC=CC2)=O)c(C)nc(C)nc1C Cc1cc(C)c(O)c(C(N2CC(S(C)(=O)=O)C2)=O)n1 C12(C(=O)NCCCCNC(c3cnc(OCC)s3)=O)CC3CC1C2C3 C#CCC(C)C(=O)NCC1CCC1NC(C1CCCC1C(C)C)=O c1(Oc2ccc(-n3c(C)nc(C)n3)cn2)c(C)cc(Br)cc1C N#Cc1ccc(S(=O)(=O)N2CCCc3n[nH]cc3C2)cc1F C1(C(N(C(CCNC(c2ccc(NC)cc2)=O)C)C)=O)CN2CCN1CC2 C(=O)(C(CC(C)C)C(N)=O)NCC#CC(N1C2CC(CC)CC1CC2)=O C1(CNC(c2nc(C(=O)OC)sc2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC12CC2 CCC(C)(C)C(O)C(=O)NC(C)CCC(=O)NCC(c1ccsc1)C c1(C(=O)NC(C(C)C)C(=O)NCc2nccn2C(C)C)cc2n(n1)CCC2 C1(C(=O)NC2CC(C(N(CC(C)C)C(C)C)=O)C2)CCCCCN1C N1(C(c2cnc(S(C)(=O)=O)s2)=O)CCCC12CCN(C(=O)Cc1cscn1)CC2 Cc1cccc(C(N2CCCCCC2CNC(c2cn(C)c(=O)cn2)=O)=O)c1N C(=O)(CCCC(F)(F)F)NCC12C(CN(C(c3c(OC)ncc(Cl)c3)=O)C1)C2 N1(C(c2cc(Cl)cc(Cl)n2)C(=O)NCC=C)CCC2(C1)NC(=O)NC2=O N1(C(c2nc(CC)on2)C)CCC(CC)CC1.c12nc(cs1)CCNC2=O c1(OCC)ccc(C(=O)NC(C)C(C)NC(c2cc(C3CC3)no2)=O)cc1 c1(C(=O)NCC(C)NC(c2ccc(OC)cc2Cl)=O)nn(C)cc1[N+](=O)[O-] C1(NC(C(c2c(C)n[nH]c2C)C)=O)CCN(C(c2ccc(C#N)cn2)=O)CC1F c1(C(N(C2CCCN(C(=O)CC(C)C)CC2)CCC)=O)cnc2cc(Cl)ccn12 C(CC(=O)NC1CCN(C(c2coc(C(N)=O)c2)=O)CC1O)(C(N)=O)NC(C)=O N#Cc1cccc(CN2CCOCC(C(=O)Nc3cc(Cl)ccc3O)C2)n1 C(CCCCCC(=O)N1CC(C2CC2(F)F)C1)NC(C1(CC)CCCC1)=O N1(C(C2C(C)N(C)CC2)=O)CC2CN(C(c3ccccc3Cl)=O)CC2(C)C1 c1(C(N2CC(C)(C)C2COC)C(=O)NCCCCCC)nc(C)n(C)n1 C#CCC(C(=O)Nc1cnc(CCC)nc1)NC(C1CC1Cl)=O CCCC(CC)C(=O)NC1CCCCC1CNC(=O)Cc1c(C)noc1Cl N1(C(C(n2c(C)ccn2)C)=O)CCN(C(=O)C=C(Cl)Cl)C(CC2CC2)C1 C1(CCNC(c2cc(Br)no2)=O)(NC(C2C(=C)CC2)=O)CCCC1 c1(OC)cc[n+]([O-])c(C(=O)NCCC2CC(NC(c3cc(Cl)c(C)cn3)=O)C2)c1 c1(CC(=O)N(CC(CC)(C)NC(c2cnc(OC)cn2)=O)CC)nc(C)c(C)s1 C1(CNC(c2cc(CC)n(C)n2)=O)CCC2CN(C(=O)C(O)CSC)CC12 C#Cc1cnn(C)c1C(=O)NCC1CCCCN1C(=O)C(COC)N(C)C c1(CC(=O)N(CC2CCN(C(CC3C(CC)C3)=O)CC2)CC)ccc(F)c(Cl)c1 c1(C(N)=O)ccc(CNC(=O)NCC2(N3CCCC3)CCOC2)o1 c1(OCC)c(C)cc(C(=O)NC2CC(NCc3ccccc3F)C2)cc1C C1(CNC(CCc2cncc(OC)c2)=O)CC(NC(=O)C(=O)N(C)C)C12CCC2 CCCC(C#N)C(=O)N1CCCC(C(C)C(=O)NCC2CC3(CCC3)C2)C1 CC1(C)CCCC1(O)CNC(=O)Cn1cc(CNC(C2CCNC2=O)=O)nn1 N1(CCCC(C)C)CCC(CC(C)NC(=O)C(F)CN(CCO)CCOC)CC1 CC(C)CCC(C(=O)NCC(C)CC1CCC1)NC(C12CCC(C1)C2(C)C)=O c1(C(=O)NCCN(C2CCCC2)C(COC(CC)(C)C)=O)cc(Cl)c(Cl)n1C C=CC(C(F)(F)F)NC(C1CCCN(C(=O)C(C)C(=O)OC)C1)=O C(=O)(CCS(=O)(=O)C1CCCC1)NCC1CC(OC)CN1C(C1CCCN1C)=O c1(C(=O)NCCC(C)N(c2ncnc(C(C)(C)C)n2)C)ccc(O)nc1 C(C(C(C)C(C)C)NC(c1cn(CCO)nn1)=O)NC(CCN(C)CC)=O C1(O)(C(C)NC(=O)COCC(C)(C)C)CCN(C(=O)CC2CC3CC3C2)C1 C1(C(=O)NCC2(C)CC2)CCN(C(=O)C2C3CC(=O)CC23)O1 C(CCN=c1cc[nH]c(=NCCCCc2ncc[nH]2)[nH]1)c1cccc(C)n1 C1(NC(c2c(C)n(CCO)cc2)=O)CCN(C(=O)CC(C)(F)F)CC1C(C)C C1(NC(c2ccccc2O)=O)(CNC(C2(CN(C)C)CC2)=O)CC2CCC1CC2 C(=O)(C(C)(C)C1=CCSCC1)NC1CCN(C(CCC(CCC)CC)=O)CC1F N1(C(CCC(CC)C)=O)CC2CN(C(=O)CCc3ccc(Cl)c(F)c3)CC2C1 C1(C)(CNC(C(CC)C(C)C)=O)COCCN(C(c2ccnc(OC)n2)=O)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CC2CCCC2(NC(c2ccn(C)c2C)=O)C1 N1(CC)CCC(n2nc(COC)nc2-c2cnn(CC3CCOCC3)c2)CC1 c1(C(=O)NC2(COC)CN(C(CC3CC(CC)C3)=O)C2)cnc2ccncc2c1 C(=O)(C1c2c[nH]nc2CN1C(=O)C1=C(Cl)CCCC1)Nc1cncc(C(N)=O)c1 CC1(C)OCCOC1c1nnc(N2CCCCC2)n1CC1CC12CCCCC2 C1(CNC(C2CCCN(C(C(CC)CC)=O)C2)=O)CC(=O)NC(C)C1 c1(NC(=O)OC)cccc(CC(=O)NCCS(=O)C(F)F)c1 c1(C(N2CCC(n3cccc3)C2)=O)csc(-c2ccoc2)n1 C(CCC(C(=O)NCC(=O)NCCOC)N(c1ccccc1OC)C)OC c1(C(N(CC(=O)OCCNC(=O)COC2CC2)C)=O)cc2c(nn1)CCC2 N1(C(=O)OC(C(C)(C)C)=O)CC2CC2(N(C(=O)CC=C(Cl)Cl)CCO)C1 Nc1ccc(Cl)cc1C(=O)NC1COCC1CNC(C1CCNC1=O)=O C1(C(=O)NCCC(C)(C)NC(c2c(CCC)n(C)nn2)=O)C2CCC(F)(F)C12 c1(C(N2CC(CCNC(CC=CC)=O)C(C)C2)=O)[nH]c2ccccc2c1Cl c1(CC)nccnc1C(=O)NCCC(O)C(=O)NC1CCCC(CO)C1 C(=O)(C(CCc1ccncc1)NC(=O)C(C#N)C=Cc1ccccc1)OCC C1(NC(C(C)n2cncn2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)O)C2 Cn1nc2cc(Br)ccc2c1C(N1CCC(NC(=O)CN=S(C)(C)=O)C1)=O c1(NC(=O)NC(Cc2ccoc2)CO)csc2c1CCCC2 Cc1ccc2c(=NC(C)c3nccn3C(C)C)[nH]c(N3CCC4(CC4)C3)nc2c1 Cc1cc(C(C)(C)NC(=O)CN(C(=O)CNC(=O)C(C)CF)C)cc(C)c1 C(=O)(CC(C(C)CC)NC(C1CC(CC)C1)=O)NC(CCC=C)C1CC1 c1(CC)nocc1CN(C)CC1CCC(=O)N1 c1(CCC)ccc(C(N2CCC(O)(CCNC(=O)C3CC3)C2)=O)cc1[N+](=O)[O-] C=CC(C)(C)C(=O)N(C)CC1CCCN(C(=O)CCCN2C(=O)CNC2=O)C1 O=C(C1COc2ccccc21)NC1(C2CCN(C(C3CC34CCOC4)=O)C2)CC1 c1(C(N(CCC)CCNC(C2CCC(C)(C)CO2)=O)=O)ccnc(S(N)(=O)=O)c1 c1(N(CCCC)C)nnc(-c2ccco2)n1CC(n1cccn1)C CC1CCCC1(C)C(=O)NCc1cn(CCN(CCCF)C)nn1 C1(CCCC)CN(C(=O)CNC(=O)CNC(c2ccoc2C)=O)CCN1C(C)=O C1(CC(=O)NCc2c(C)cns2)CN(C(=O)Cc2ccccn2)CCC1C n1(CC(=O)NCC(CC=C)NC(c2cncnc2)=O)cc(C)c(O)nc1=O N1(C(CNS(CC)(=O)=O)=O)CC2CC(CNC(=O)CC3OCCCO3)C2C1 c1(C(N2CC(O)(CCNC(C3CC=C(C)CC3)=O)C2)=O)cc(N)c(C)c(N)c1 N1(C(C=NOC)=O)CCC(CCNC(c2scc3c2CCCC3)=O)C(F)(F)CC1 C(=O)(C1SCCc2sccc21)N1CC(N(C(=O)CCc2cnoc2)C)C1 C1(CNC(c2cnc3ncccn23)=O)CCN(C(=O)C(F)F)CC1(F)F C1(C(=O)NC2C(NC(c3c(N)c(Cl)ccc3)=O)CC2)CCOCC12CCC2 c1(C(N2CC(NC(c3ccc(C(C)N)cc3)=O)C(F)C2)=O)cc(O)cc(O)c1 C1(C(=O)NCCN(C2CC2)CC)C(C)OCCN1C(=O)CC1CCC(C)CO1 N1(C(CC=CC=C)=O)CCN(C(=O)Cc2cc(OC)cc(C(F)(F)F)c2)C2CC12 Cc1ccc(C(C)C(N2CCC(CF)(NC(C3CC(C)(C)C3)=O)C2)=O)cc1 Clc1ccc(C2(NCCC3CC=CC3)CCCC2)cc1Cl c1(N2CC(CNC(C(CC)NC(C)=O)=O)C(C)(C)CC2)nc2cc(C)ccc2o1 CCC(CC(=O)NCCC1(O)CN(C(c2nc(=N)cc[nH]2)=O)C1)C(F)F CC(N=c1cc[nH]cc1S(=O)(=O)NC1(C)CCCC(C)(C)C1)C12CCCC1C2 N1(CCc2cn(C)nc2)CCC(NC(c2cc(=O)cc[nH]2)=O)C(O)C1 C(=O)(C1=CCCCCC1)NCC1CN(C(=O)CC2COCC2O)CCC1CO Cc1ccccc1-n1cc(C(N2CCN(C(C3(CF)CC3)=O)CC2)C)nn1 C1(C(=O)NC2CC(CCNC(=O)Cn3ccnn3)C2)CC(c2ccccc2)=NO1 C1(CC(N2CCCC(C)C2)=O)N(C(c2ccn(C3CC3)n2)=O)CCC1(C)C C(CC1CCC1)(C(=O)NOCCC1(C)N=N1)NC(c1cccc(CC)n1)=O C(C(=O)NC1C=CC(C(=O)NCc2scnc2C)C1)(C(C)C)SC C(=O)(C1CCCc2nnn(C)c21)NC1CN(C(c2c(CC)n[nH]c2)=O)CC(F)C1 C1(C(N2C(CC)CCC2)=O)Cc2c(C)cccc2O1 c1(C(=O)NC(CNC(C(C#N)C2CC2)=O)C2CCC2)ccc(-n2cccn2)cc1 Cc1c(Cl)ccnc1C(=O)NC(C1CCCCN1C(=O)CCCSC(C)(C)C)C N1(C(c2scc(C)c2C)=O)CCN(C(C2CC2[N+](=O)[O-])=O)CC12CCC2 C(=O)(C1=Cc2ccccc2C1O)NCCN(C)C(c1cccc2nc(O)oc12)=O C=CC1(CO)CCN(C(C2C=CCCN2C(c2cc(Cl)ns2)=O)=O)CC1 N1(C(C(C)OCCOC)=O)CCC2(C1)CN(C(=O)CCNC(C1CCCO1)=O)C2 Cc1nc(CO)ncc1C(=O)NCC(C1CCC1)NC(=O)C(Cl)=CCl c1(C2(C)CC2)cccc(C(=O)NC2(CNC(C3CCCS3)=O)CCCCC2)c1 N1(C(C=C(C)C(F)F)=O)CC2C(CN(C(=O)CC(C)N(C)C)C)C2C1 C1(C(=O)NCC(C)(C(C)C)NC(C=C(CCC)C)=O)CCN(C)S1(=O)=O C(CCCCF)NC(CCN(C)CCn1cc(CCO)nn1)=O N1(C(C(CCC)CCC)=O)CC2CCCCC2(NC(C2COC(=O)N2C)=O)C1 C1(NC(C(CO)N(C)C)=O)CN(C(c2cnc(C(N)=O)s2)=O)CCC1CO Cc1n[nH]c(=NC(=O)c2ncnc3c2cnn3-c2ccc(Cl)c(F)c2)n1C C1(CNC(C(C)OCCCC)=O)CCN(C(c2ccnnc2)=O)C12CC2 CCN=C(NCCC1CCCCC1)NC(C)CCN1OC(C)CC1 CC1OC2(CN(C(N3CCOC(c4cccc(F)c4)C3)=O)C3CC3)CCC1C2 c1(C(N2CCCC(N(C(C=COCC)=O)CC)C2)=O)cn2ccn(C)c(=O)c2n1 N1(C(c2ccc(CC)o2)C(=O)NCC2CC2)C2C=CCC1CCC2 c1(C(=O)NCCCCC(C)NC(C2CCS(=O)(=O)C2)=O)c(N)nn2ccccc12 CN=c1ccc(C(N2CCSC3CCC23)=O)c[nH]1 C1(NC(C2(C)CC3CC3C2)=O)CN(C(=O)Cc2ccsc2)C2(CCCC2)C1 c1(NC)cncc(C(=O)NCc2cc(C(N3CCC(N(C)C)C3)=O)n(C)n2)c1 C1(O)(CNC(C=CC=CCCCCC)=O)CCN(C(=O)CC2CNC(=O)C2)C1 C1(NC(C2(C3CCC3)CC2)=O)CC2CN(C(c3ccc(C)nc3)=O)CC12 C1(C(C)OC)CCN(C(=O)C=CC2CCCN2C(c2n[nH]c(=N)[nH]2)=O)CC1 N1(C(c2ccc(C#C)o2)=O)CCC(C2CC2)C1C(N1CCCOC(C)C1)=O C1(C(=O)OC)(C(N2CC3C(CNC(=O)OC(C)(C)C)C3C2)=O)CCS(=O)(=O)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(NC(c2nn(C)c(O)c2)=O)C(C(N)=O)C1 N1(C(C2N(C(COCCC#C)=O)CC=C2)=O)CCC(F)(C#N)C1 C1(c2cc(CNC(c3c(CC)non3)=O)on2)CCN(C(=O)C2=CCC2)CC1 C=C1CC(C(F)(F)F)(C(N2CC(O)(CNC(C3CCCCS3)=O)C2)=O)C1 C1(O)(C(=O)NCc2c(CC)ocn2)CC2(CCCN(C(=O)OC(C)(C)C)C2)C1 c1(CN(C(C2(CC)CN(C(c3ccsc3C)=O)C2)=O)C)cccc(C)c1 c1(C(N(CC(C)NC(C2(c3nccs3)CC2)=O)C)=O)cnccc1N(C)C Cc1ccc(C)c(C(N2CCN(C(c3cn(CCO)nn3)=O)C3CC23)=O)n1 N1(C(CC=CC)=O)CCC(c2ccccc2)(NC(=O)C(CC)OCC)C1 C1(CC#C)CCN(C(=O)C(CCC)NC(=O)Cc2cc(C)cs2)CC1 c1(C(=O)NC(CCNC(CN(C)CC)=O)C(C)C)c(F)ccnc1Cl Cc1nn(C)c(C)c1C(=O)NC1CCCCC1C(N1CCCC(C(F)(F)F)C1)=O C(=O)(C(F)CCC(C)C)NCC1CCN(C(C2CC(CC)OCC2)=O)CC1 O=C1CC(C(=O)N2CC3(C2)CN(C(c2cc4c[nH]nc4s2)=O)C3)c2ccccc21 Cc1nc(N2CCC(NC(c3cc[n+]([O-])cc3)=O)C23CCC3)ccc1C#N Cc1ccc2c(CCC(N3CC(F)(CNC(C4CC4(C)CF)=O)C3)=O)c[nH]c2c1 CC(O)C(C)C(=O)N(CC(C)(C)CNC(c1csnc1C1CC1)=O)C CC#CCC(C(=O)NCC1CC2CCCC2C1)NC(c1ccccn1)=O C1(C(C)(C)C)CC(CNC(C2(F)CCCC2)=O)CN(C(=O)Cc2ccsn2)C1 C(=O)(CCC1=CCCCC1)NC(CC(=O)NCC1(C)ON=C(C)C1)C C1(NC(C(CO)OC)=O)COC2CN(C(=O)CC3CCSC3)CC12 C1(CNC(C2(SCC)CC2)=O)CCCCCN1C(=O)CCc1cn(C)cn1 N1(CC(COCC(C)C)O)CCC(C)(NC(c2cnc(Cl)c(Cl)c2)=O)CC1 C1(C(=O)NCCC2(NC(C(=O)NCCOC)=O)CC2)CS(=O)(=O)CC12CC2 CC(N=c1[nH]c2cc(Cl)ccc2s1)C1CCCCN1C(=O)C1=COCC1 Cc1ccc(C(N2CC(NC(c3c[nH]c(=N)o3)=O)C3(CC3)C2)=O)c(C)c1 CC1CCN(C(=O)CCc2ncccn2)CC1NC(c1cscn1)=O CCC(C)(C)CCCC(=O)N1CC(C)N(C(=O)C(C)OC2CCCCC2)CC1C CC1CCC(OC(c2c(O)ncc(Br)c2C)=O)C=C1C(N)=O Cc1ccc(C)c(C(N2CCCCC(N(C)C(C3CCCCC3C)=O)C2)=O)c1C N1(C(CC=C(C)C)=O)CCN(C(c2ccnc(C3CCC3)c2)=O)C(C2CCC2)C1 C1(O)(C(=O)NCCOCCN(C(C2CCC(C)S2)=O)C)CC(C)(C)C1 c1(C(C)NC(c2c(C)n(CC(F)(F)F)nc2)=O)ccc2c(c1)CC(=O)N2C c1(COC)ncc(C(N2CCCC(CN(C)C(C3CCOC3C)=O)C2)=O)c(O)n1 c1(NC(C2CCCCN2S(=O)(=O)C(Cl)(Cl)Cl)=O)cc(O)c(Br)c(O)c1 CC1CN(C(=O)C(F)CC2CCOC2)CC1NC(C1CCNC(=O)C1)=O Cc1nc(C=CC(N2CCCC2(C)CNC(c2ccncc2)=O)=O)cs1 C(=O)(CC(C)n1ccc(C)n1)NC1(CCCNC(COCCCCC)=O)CC1 c1(C(=O)NCC2OCCCN(C(C3C(C)CCO3)=O)C2)cccn2[nH]c(=N)nc12 c1(NC2CC(NCCC(F)(F)F)C2)cc2cccc(Br)c2nc1Cl C1(C(N2CC(C)(NC(C(C)OC(C)(C)C)=O)C2)=O)(N(C)C)CCOCC1 C=C(C)CCCC(=O)NCCOCCNC(=O)C(C)(C1CCOCC1)OC Cc1cnc(NC(c2cccc(Cl)c2)C)c(S(=O)(=O)N2CCC(CCO)CC2)c1 c1(C(=O)NC2CCN(C(C3(C(=O)OC)C=CCC3)=O)C2)cccc2ncsc12 C(=O)(C(F)(F)CC(C)C)N1CC2C(NC(Cc3c(CC)cccc3)=O)(C2)C1 N1(C(C2C(C)=C2)=O)CCC2(CC1)CCN(C(C1(CC3CC3)CC1)=O)CC2 N1(C(Cc2c(C)snc2)=O)CCc2cc(-c3cn(C4(C)CC4)nn3)ccc21 c1(COCC)n[nH]c(=NC(CO)C(C)C(O)c2nc(CC)no2)o1 C(CCC(C(=O)NOC(C)CC)NC(=O)C1CC1)OCC C1(C)(C(=O)NC(CC)CN(C(=O)C(F)=C2CCCC2)C)CS(=O)(=O)C1 C1(NC(C2CCN(CC#C)CC2)=O)COCCN(C(C2CC3CCC2O3)=O)C1 c1(C(C(=O)NCC=C)N(C2CCS(=O)(=O)C2)C)cc(C(F)(F)F)cc(Br)n1 c1(CC)noc(C(=O)NCCCC2CCCN2C(=O)CC(=O)OC)n1 C(=O)(CC1NC(=O)c2ccccc21)N1CCC(NC(CNS(NC)(=O)=O)=O)CC1 Nc1ccc(C(N2CCCC2CCNC(C2CCCC(C(N)=O)C2)=O)=O)cc1O N1(C(C(CCC=C)NC(=O)CCSCC)=O)CC2CC(C1)N(C)C2 c1(C(N2C(C(C)NC(=O)CC3CCC34CCC4)CCC2)=O)cnn2ncccc12 CC1C(=O)OCC(C)(C)N1C(c1ccc(C#N)n1C)=O N1(CC)CCC(NC(c2ncoc2CNC(=O)C(C)(O)C2CCC2)=O)C1 N1(C(C2CN(C(=O)Cn3ccnn3)CCO2)=O)CC(F)(F)CC1CO CCC(C)C(O)C(=O)NC1CCC(NC(c2ccco2)=O)C1 CCC(C)(C)CC(=O)NC1CCC1NC(=O)C(C)CCCC CCC(C)C(C(=O)NC1CCC(CNC(C2(CC(C)C)CCCC2)=O)CC1)OC c1(OC)cc(C(=O)N(CC(O)CN(C(=O)C2=CSCS2)C)C)n(C)n1 C1(C(N2CCCC2c2ccco2)=O)CN(Cc2cnccc2C(F)(F)F)CCO1 C(C)(C(C)(C)C(=O)N1CCCC(OC)C1C)NC(c1n(CC)nnc1)=O c1(C(=O)Nc2scc(CC)n2)cc(Br)ccc1CC(=O)N(C)CCN(C)C N1(C(COC(C)=O)=O)CCC(NC(c2cc3c(cn2)CCCC3)=O)C12CCCC2 C1NCCCC12CCC2.c1(C2C(C)(C)CCNC2)c(N)cc(Cl)cc1F Cn1nc(C(=O)NCCC2CCCN2C(=O)CC2(C)CC2(F)F)cc1C(F)(F)F c1(C(=O)NC2CCC(N(C(=O)CCc3ccsc3)C)C2)ccc(Cl)c(F)c1O c1(C(=O)NCC(C2(O)CCN(C(c3nn(C)cc3N)=O)C2)C)ccc[n+]([O-])c1 C1(NC(C2C(=C)C2)=O)CN(C(=O)CCOc2ccccc2C(=O)OC)CC1C1CC1 C(CO)(C(=O)NCC1CCC1C(=O)NCC1CCCO1)N(C)C C=CC(C)(C)CC(=O)N1CCC(NC(C2CC23CCSCC3)=O)CC1C N#Cc1ccc(C(=O)NC2CCCCC2NC(C2CCOCC2)=O)nc1 C1(C(=O)NCC(CNC(C(C)(F)F)=O)(C)O)CC2(CC2)CN1 c1(C(N2CC(CNC(C3(OC)CCC3)=O)OCC2)=O)cccc(C(C)(C)C)c1N Cc1nc2cccc(C(=O)N(CC(C)NC(=O)C=Cc3cncnc3O)C)c2[nH]1 N1(C(c2c(C)oc(Cl)n2)=O)CCCOC(CCNC(C2CCCN2C=O)=O)C1 C1(C(N2CC(=C(CNC(c3cc(C(F)(F)F)cs3)=O)F)C2)=O)C(F)(F)C12CC2 C1(CC)CCCN(C(=O)CC2CN(C(=O)C=CC=C(C)C)CC2C)C1 Cc1c(C=CC(=O)NC2(CCCNC(C3COC(C)C3)=O)CC2)cnn1C C1(CNC(CCN(CCCCC)CC)=O)CCN(C(=O)CS(C)(=O)=O)C1(C)C c1(C(=O)NCC=CCNC(Cc2cncc(C#N)c2)=O)cc2c(nc1O)CCOC2 CCC(C)CCC(=O)N1CCN(C(=O)CCCC(=O)NC)C(C(C)C)C1 N1(C(c2cnc(O)[nH]2)=O)CCc2ccc(-c3ccc4c(O)ncnc4c3)cc2C1 C#CC1CCCN(C(C2CCC=CC2NC(C2CC(=O)C2(C)C)=O)=O)CC1 C(CCF)(C(=O)NCCCNC(=O)OC)NC(C(CC)=CCCC)=O N1(C(CCc2cccc(OC)c2)=O)CC2(C1)CN(S(=O)(=O)c1cccs1)C2 C1(C2CC2)(CNC(C(C=C)C)=O)CCN(C(c2cc(CC)nnc2C)=O)C1 C(=O)(C(C(C)C)C(C)C)NC12CC(CNC(CCCCOCC)=O)(OC1)C2 CC(C(=O)N1CCC(CNC(c2ccnn2CCF)=O)C1)P(C)(C)=O C1(NC(CC(C=C)C)=O)CN(C(=O)CC2CCC=CCC2)C2CCCCC12 C1(C(N(C2CCN(C(=O)C3=CCCCC3)CC2)C)=O)CC2CCCC2C1 N1(C(c2cnc(OC)nc2C)=O)CC(NC(=O)CCCCCF)C(C2CC2)C1 c1(CCC)cc(C(N2CCCC(N(C)C(C3CC4CC4C3)=O)C2)=O)cc(O)n1 c1(C(=O)NCCNC(c2sc(Br)cc2F)=O)cc2c(cn1)COCC2 C1(C(N2CCC(C(C)C)C2)=O)CCCN(C(=O)CC2C=NN(C)C2=O)CC1 C1(C(N2C(CN(C(CNC(CC)=O)=O)C)CCC2)=O)CCCN1N=O c1(CC(C)(C)C)noc2ncc(C(N3CCN(C(=O)C(N)=O)C(CO)C3)=O)cc12 C1(C(N2CCC3(CCC3)C2)=O)CCN(C(=O)C2(Cl)CCC2)O1 C1(C(N2CCC(N(C)CC)C2)=O)CC(NC(C2CCCC2O)=O)C(O)C1 c1(OC)cccc(C(N2CCC3(CC3C(=O)NC3CS(=O)(=O)C3)C2)=O)c1OC c1(C(N(CCC(C)NC(c2cn(CCC)nc2)=O)C)=O)sc2ccsc2c1C CC(C)(CN=c1[nH]ncs1)NC(=O)C(CCc1ccsc1)Nc1ccccc1Cl N1(C(C2(C)CC(F)C2)=O)CCCCC(CNC(c2ccc(SC(F)(F)F)o2)=O)C1 N1(C(CCC#CC)=O)CCC(C)(C(=O)NCC(C)COCC)CC1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(CCc2cn(C(C)C)nn2)OCC1 C1(OC(C)C)CCC(c2ccccc2)CC1.C12CCCN1C2=O C1(C(N2CC(C)C(C)(C)CC2)=O)CCCN1NC(=O)C=Cc1ccn(C)c1 C1(NC(COC(CC)C)=O)CC(O)CN(C(C2(OC(C)=O)CC2C)=O)C1 c1(OC(C)(C)C)ccnc(CNCC23CC(CCO2)C3)c1 c1(C(=O)Nc2ccc(-n3ccnn3)cc2)ccc2c(c1)CNCCN2 C1(CC)CCCCC1C(=O)N(C1CCN(c2nnc(C(=O)OC)o2)CC1)C C(=O)(CCCNC(=O)OC)N(C1CCN(C(=O)C(Br)=C(C)C)C1)CC C(CC(C)C(=O)NC(CNC(C1(c2ccn(C)n2)CC1)=O)CC)=CC N1(C(C(c2c(F)cccc2F)C)=O)CC(O)(C2CCN(C(C3CCC3)=O)CC2)C1 c1(C(=O)NCCN(C(=O)CCOCCCOC)C)ncccc1O C1(C(=O)NN2CCN(C(C(C)O)=O)CC2)CC2COCC(C1)C2.c12cn(nn1)C2 CC1CCN(C(=O)CCC2CC2)C1CNC(C1CCCC1O)=O c1(OC)ccc(S(=O)(=O)N2CCC3(CC2)CC3(C)C(=O)NC(C)CO)c([N+](=O)[O-])c1 C=CC(C)CC(=O)N1CC(C(=O)NCc2cccc(Cl)c2)C(C)C1 N1(C(CCCCOCC)=O)CC2(CC1CNC(c1ccncn1)=O)CC2(F)F CC(C(=O)NC1CC(O)CN(C(=O)Cc2cnccc2Cl)C1)S(N)(=O)=O c12cccc3nc([nH]c13)C1C(CC)(C1)CNC2=O.c1(SC(C)(C)C)ccccc1 S(=O)(=O)(c1cccc(Br)n1)N1C(C(=O)Nc2nc(Br)cs2)C=CC1 C1(C(=O)OCC)CCN(C(=O)C(Cc2ccc(C)cc2)NC(C)=O)C1C N#Cc1cnn2cc(C(=O)NC3CCCN(C(c4ccccn4)=O)C3)cnc12 C1(C2CC2)(C(N2C(C)(C(=O)NC)CC2)=O)CN(C(=O)CNC(=O)OC)C1 c1(C(=O)NC(CNC(C23OC(C)(C)C(C2)C3)=O)(C)C2CC2)cnn2ncccc12 N1(C(C(CC)OC)=O)CCOC2(C1)CN(CCN=c1cc(C)nc[nH]1)C2 CC(C)CC(CNC=O)CC(=O)N1CC2C(CNC(c3cnncc3O)=O)C2C1 C(=O)(CCCCC(C)=O)N1CC(C)(COC)C1 C1(NC(CC(C=C)CC)=O)CN(C(=O)CCC2CCCC2)CCC12CCOCC2 CC(O)(CC(=O)N1CC(NC(c2cccc(OC(F)F)c2)=O)C1)C1CC1 c1(NC(N(C)C)=O)ccnc2ccc(C(N3CCCCC3C(O)C(F)(F)F)=O)cc12 c1(C(=O)NCC(C2CCCOC2)OC)c(O)cc(=O)n2c1CCCC2 C=CCC(CNC(=O)C(F)CCCC)C(=O)NC(c1cc(C)no1)(C)C CC(C)C(F)(CNC(C1C=CCS1)=O)C(=O)N1CC(C)(O)C1 CC(C)(CCC(=O)NCC1CC2CCCC2N1C(c1cc(CO)[nH]n1)=O)[N+](=O)[O-] c1(C(C(=O)NC2CC(NC(c3ccc(OC)nn3)=O)C2)O)cc(F)c(F)c(F)c1 CC1(C)CN(C(=O)COC2CCC2)CC(C)(C)C1NC(C1CN2CCC1CC2)=O c1(OCCC(=O)N(C)CC2CCCN(C(C(CC#C)C)=O)C2)ccc(F)cc1Cl C(=O)(C1OCCc2ccccc21)N1CC=CC(NC(C(C)(C)n2cccn2)=O)C1 C1(O)(CCNC(C=CCN(C)CC)=O)CCCN(C(=O)C(C)C2(O)CCC2)C1 C1(C(CC)C(=O)N2CC(CO)(NC(=O)Cc3nncs3)C2)CCC(C)CC1 C=CCCCCCCC(=O)NCCCCNC(C1(c2ccnc(OC)c2)CC1)=O CC1(C)CC(C(=O)CC2C(F)(F)C23CC3)CC(C)(C)C1.C12CCCN(C1)C2=O C(C(C)(C)C(=O)NCC1(CO)CCN(C(C2CC=CCO2)=O)C1)OC CCC(C)CCC(=O)NCCn1cnc(C(N2CC(O)(COC)C2)=O)c1 N1(C(CC(=O)NC)=O)CCC(C2CCCN2C(=O)C(C2CCOC2)OC)CC1 N1(C(COCC)=O)CCC2(CCCC2C(N2CCC(C)(C)C2)=O)C1 C1(NC(=O)COCC2CCCCO2)CC2CC(C1)N(C(=O)Cn1ncnn1)C2 C1(Cc2cn(CC(=O)NCCCS(C)=O)nn2)CCC(C)(C)CC1 c1(C(N(C2CCCCC2NC(=O)Cn2cc(Br)cn2)C)=O)cnncc1O N1(C(CC)=O)CCCC1C(=O)NC1CC(N(C(=O)C(C)C2CCOC2)C)C1 N1(CCC)C(=S)NC(c2c(Br)n[nH]c2Br)C(C(=O)OC)=C1c1cnn(C)c1 C(=O)(C(C(C)NC(C1CC2C=CC1O2)=O)C(C)C)NCc1c(C)ccs1 C1(NC(CCCCC(CC)C)=O)CCOC12CCN(C(=O)CC(C)C(F)F)CC2 C(=O)(CS(=O)(=O)C1CC1)N1CC(CNC(c2ccc(C)nc2N)=O)CC1(C)C C1(C)(CNC(c2cc(OC)ncc2)=O)CCCN(C(C2CC(=O)C2(C)C)=O)C1 N1(C(C2N(C(c3ccnc(C)c3N)=O)CCC2(C)C)=O)CCOC2COCC2C1 N1(C(c2ccc(C)n2C)=O)CCC(NC(=O)CC2CCOC2)C(F)(F)CC1 N1(C(C(C)(c2ccccc2)OC)=O)CC2CCCC(CNc3nccc(C)n3)C2C1 N1(C(C2(C)CC(F)C2)=O)CCCC(CO)(NC(=O)C(F)(F)c2cscn2)C1 C(=O)(CCCCCN(C(=O)CC(C)(C)C)C)N(C)CC1CC1c1ccco1 CC(C)CC(C(=O)N1CCC(CN2CCCCC2)CC1)NC(c1nn(C)cc1Br)=O C1(NC(COC(CC)C)=O)CCCCN(CCc2ccccc2)C1 N1(C(CC2C(C)C2)=O)CC(O)(CN(C)C(c2csc(-c3cnc[nH]3)n2)=O)C1 Cc1c(C(N2CC(NC(c3n[nH]cc3Br)=O)C(O)C2)=O)ccn1C(C)C Cc1nn(C)c2c(NCC3(Br)CC3(F)F)nc(NCc3cc(Cl)ccc3Cl)nc12 N1(C(c2n(CCC)ncc2)=O)C2CCC1CN(C(C1CCOCC1)=O)CC2 C(=O)(C(C)CCCCCC)NC(CC#C)C(=O)NCC=CCl N1(C(c2ncn(CC)n2)=O)C2CCC1C(F)C(NC(c1coc(C(C)C)n1)=O)C2 Cc1cc(=NC(=O)C(CN(C)C)NC(c2ccc(=O)n(C)n2)=O)[nH]n1C(C)C C(C(C)(C(=O)N1CC2C(NC(c3coc(Br)c3)=O)C2C1)OC)OC c1(C2C(C(N(CCN(C)C)CC)=O)C3CCC2O3)cccc2c1CCCC2=O Cc1cccc2c1CCC2NC(c1ccc(OC(F)(F)F)cc1Cl)=O c1(CN2CCN(C(c3cc(F)ccc3Br)=O)C(CO)C2)c[nH]c2c(F)cccc12 N1(C(C)=O)CCC(N(C(=O)C(C)CC2CC2)C(=O)CC2(CN(C)C)CCC2)C1 C1(NC(CNC(=O)OCC=C)=O)CCN(C(C2CCN(C)C2C)=O)CC1 c1(C(=O)NCC2C(NC(c3ccc(CSCCOC)o3)=O)C2)nc(O)c(C)s1 C1(C)(CC(=O)NC(C(C)C)CNC(C2CCOC2)=O)CC(F)(F)C1 Cc1cc(C(N2CCC(c3nc(C)ns3)CC2)=O)nc(C(F)F)n1 C(CCC(=O)NC1CCCC1CNC(C1CC1C(N)=O)=O)=CC c1(C(N(CC(C)NC(=O)CCc2ncccn2)CC)=O)cccc([N+](=O)[O-])c1Cl C1(CNC(=O)C(F)n2ccnc2)C2CC1N(C(c1cccc(C(F)(F)F)c1)=O)C2 c1(N2CCC(N(C(=O)CN3CCOCC3=O)C)C2)c(C)cncc1[N+](=O)[O-].CN c1(C(=O)NCC(C)CNC(C2(F)CC2C)=O)ccc(CC(C)(C)C)cc1 c1(C(C)NCC(c2cccnc2)OC)ccc(Br)c(Cl)c1 c1(CN(C)C(c2conc2CNC(=O)CCC2(C)CC2)=O)ncccn1 c1(N2CCCC(CNC(c3cn4c(n3)CCC4)=O)CC2)nc2ccccc2s1 Cc1cc(C(N2CCN(C(=O)C(C)C(C)(C)C)C3CC23)=O)n2nc(C)c(C)c2n1 c1(C(=O)NCC(CC)NC(c2cc(C)ncc2C)=O)ccn2c1CSCC2 N1(C(C(CCC)=CCC)=O)CCC2(NC(=O)C(Cl)=CCl)CCCC12 C1(C)(C(=O)NCCCCN(C)C(c2ccc(N3CCCC3)cc2)=O)CCCOC1 N1(C(c2cc(Cl)cc(C)c2N)=O)CCN(C(c2nccnc2C)=O)CC(C)(C)C1 C1(C(CC)=O)CCC(C(=O)N(C2CC2)Cc2cn(Cc3cnnn3C)nn2)CC1 c1(C(=O)NC(C2CCN(C(c3cncc(SC)c3)=O)C2)(C)C)cnc(C)cc1C Nc1cccc(C2CCN(Cc3cn(C4CC(C5COCCO5)C4)nn3)C2)c1N CCCCCCCCCC(=O)NC1C2CCN(C(=O)C(=O)C(C)(C)C)C12 C1(NC(Cc2ccc(C(C)C)cc2)=O)CC2CC1N(C(C1CCCN(C)C1)=O)C2 C1(CNC(COCCCN=[N+]=[N-])=O)CCC(NC(=O)C2=CCCS2)CC1 C1(CNC(=O)CCOc2cccc(Cl)c2)CN(C(=O)C=Cc2ccoc2)CCCO1 c1(COC)nc(Cl)cc(=NC2CN(C(C3CCCN3C=O)=O)CC3(CCC3)C2)[nH]1 O=C(C1=CCCN(C(C2C3CCC(F)C23)=O)C1)NC(CCC1CC1)C1CC1 N#Cc1cc(S(=O)(=O)NC2CCOCC2)ccc1NCC(C1CCCC1)O Cc1[nH]c(=N)nc(O)c1CC(=O)NCC(C)CNC(=O)CC1CCC(F)(F)CC1 C1(C(C(=O)N(CC=C)CCOC)C)CCN(C(c2n[nH]cc2Cl)=O)CC1 c1(CSC)ccc(C)cc1OCCc1cccc(NC(=O)NCC(=O)N(C)C)c1 c1(C(=O)NC2C(C=C)CN(C(C3(C)CCCO3)=O)C2)nccn2cc(C)nc12 C1(C(=O)NC(CCC)C2CCCC2)CCN(C(=O)C(C)CC#N)C(C)(C)C1 CCCC(CC)CC(=O)NC1CN(C(=O)Cc2coc3ccccc23)CCC1O C#CCC(CC(F)F)NC(=O)CCN(C(=O)Cc1ccc(O)cc1)C1CC1 c1(N2CC(C(=O)OC)C(OC)C2)ncnc(N(CC)CC)c1N.C1CC1 c1(C2(C(C)NC(N3CC4C(C3)C4(C)C)=O)CC2)cccc(F)c1F c1(C(N2CCN(C(=O)CCCn3ccnn3)C3C2C3)=O)cncc2nc[nH]c12 c1(C(N(CC)CC2CCCN2C(=O)CCSC2CCCOC2)=O)cc(C)nn1C c1(CNC(c2c(C)scn2)c2nnnn2C2CC2)cccc(N(C)C)c1 C1(OC)CC(NC(=O)CCc2cc(C)[nH]n2)CN(C(C2(n3nccn3)CC2)=O)C1 N1(C(C(n2c(C)ccn2)C)=O)CCOC(CN(C)C(C2(F)CC=CCC2)=O)C1 C1(CNC(=O)NCC2CCC(C)(C)O2)CCCC(F)(F)C(=O)N1 c1(NC(C2CC(NCc3c(C)cc(O)cc3)C2)=O)cc(F)c(F)c(Br)c1 C(C)(CCC(=O)N1CCOC(CCNC(c2cnn(C3CCC3)c2)=O)C1)SC c1(CCNC(c2n(CCOC)nnn2)c2cc(C3CC3)[nH]n2)cncc(C)n1 c1(C(=O)NCCOCCCNC(C(C)c2cccs2)=O)ccc2c(n1)OCCO2 c1(N(C)CC2CC(=C)C2)cc(NCCC2CCCCC2C)ncn1 N1(C(C2(COC)CC2)=O)CCCC(CN(C2CC(=O)N(c3cnn(C)c3)C2)C)C1 c1(CC)ccc(C(=O)NCC2(C(=O)NC3CCOCC3)CCC2)[nH]1 N1(C(C(c2ccccc2O)OC)=O)C2CCC1C(NC(=O)CN(C)C(C)C)C2 C1(C(N(CC(=O)NCc2occ(C)n2)C2CC2)=O)COCC(C)O1 N1(C(C(=O)Nc2cc(C3C(C)C3)oc2)=O)CCCN(CC(F)F)CC1 C(=O)(C(CC(C)C)N(C)C(C1OCCCO1)=O)N(C)Cc1ccc(C)cc1 CC1(C(=O)NCCC2CCCCN2C(c2ncc(Cl)s2)=O)CNC(=O)C1 Cc1cc(=NC(CCO)C2CC2)[nH]c(C)c1C#N CCC(C)C(=O)NC(c1ccccc1)C(=O)NCCC1(C)CCOC1 c1(N2CC(CC=C)(NC(C3CCCCC3O)=O)C2)nc2c(cc1C#N)CCC2 C#CCCCCC(=O)NCC1C2CN(C(C3CCC3c3nnc(S)n3C)=O)CC12 C=C(C)C1CN(C(C2CC3(CCN(C(c4nnn(CC)c4C)=O)C3)C2)=O)CCO1 C1(C)(C(N2CC(CSC)C2)=O)CN(C(C2(SC)CCC2)=O)C1 N1(C(C(C)N(C(C)=O)C)=O)CC2(CC2)CC1CC(N1CCCC(CN=[N+]=[N-])C1)=O Cc1ccc(C)c(NC(C2(NC(c3cc(C)c(C)[nH]3)=O)CC(CO)C2)=O)c1 C(=O)(NNc1cc(C)nc(F)c1)N1CCC2(CCC(CC(=O)OC)C2)C1 C1(OCC#C)CCN(C(=O)CN(C(=O)CCC=C(C)C)C2CCC2)C1 N1(C(c2c(C)nc[nH]2)=O)CCCCC1CCC(C)(C)NC(C1CC(C)CCO1)=O C12(NC(CC)=O)CCC(CC1)N2C(=O)C(=O)NCC(=O)Nc1ccc(C)cc1 C1(C)(CC(=O)NCC(C(C)(C)C)NC(=O)CCc2csc(=N)[nH]2)CCS(=O)(=O)N1 C=C(Cl)CCC(=O)NC1CCCN(C(=O)C(O)CN(C)C)C1 C1(C(=O)NC2CC(CCNC(CCOCC(C)C)=O)C2)CCc2nncn2C1 N1(C(C(C2CC(F)(F)C2)OC)=O)CCCN(C(c2c(C)noc2C)=O)CC1C Cc1cn(CC(N2CCC2(C)C(N2CCOC3CC23)=O)=O)c(=O)nc1O Cc1nc(C(=O)NC2C3CN(C(c4cc(C)c(Br)s4)=O)CC23)c(C)o1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC(CNC(C(CC)CC)=O)C(O)C1 CN1C(=O)Cc2cc(S(=O)(=O)N3CCCC3CCC(=O)N3CCC3)ccc21 CCC(C)CC(=O)NCc1cc(C(=O)NC(C)Cc2cn[nH]c2)co1 c1(NC(=O)NC2CC(C(F)(F)F)CN(C(=O)CO)C2)cccc2c1CNC2=O c1(NC)nc(C)ccc1C(=O)NCC1CCCN(C(=O)CCOCC(F)F)C1 C1(C(N(C(CC(=O)OC)C)C)=O)CCN(C(C23CCC(C2)C3)=O)C12CC2 c1(C(=O)NC(CNC(C2(C#C)CCCC2)=O)(C)CO)cncc2[nH]ccc12 N1(C(CC(C)C)=O)CC2CCCC2(CNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(=O)Nc2cccc(OC)n2)[nH]c2ccccc2c1-c1ccnc2[nH]ccc12 C1(C(=O)NC(C)(C)C)C2CC(CC2F)N1C(C1CC1C1(C2CCCCO2)CC1)=O C1(C(=O)NC2CC(C)(NC(CCc3cn(C)nc3)=O)C2)CCC(C)(C)OC1 N1(C(C(c2ccccc2)C)=O)CC2N(C(c3ncsc3C(C)C)=O)CCC2(C)C1 Cc1cccc(C(N2CCC(NC(=O)CC3CC(C(F)F)C3)C(F)C2)=O)c1Cl c1(SCC(N2CCCC(NC(C3CC4CC4C3)=O)C2)=O)ccc(F)cc1 C(CC)(CCCC(=O)Nc1ccc(F)nc1C)NC(C=CCCC)=O N1(C(C(C(C)C(=O)NC)C)=O)CCC2(COCC(CC(=O)OC)O2)C1 Cc1cc2c(C(N3CCCN(C(c4oc(C)cc4C)=O)CC3C)=O)nccn2n1 c1(C(N(C2CCN(C(c3csc(C(=O)OC)n3)=O)C2)CC#C)=O)coc(C2CC2)n1 N1(C(C(C)S)=O)Cc2ccccc2CC1C(=O)Nc1ccc(OC(F)F)nc1 N1(C(CCSCCCC)=O)C2CCCC1CC(NC(=O)CC1CCC3CC3C1)C2 S(=O)(=O)(c1c(C(F)(F)F)cccc1Cl)NC(C#C)C(C)(C)C c1(CC(=O)NC2C3CN(C(C4(C#N)CCCC4)=O)C(C3)C2)ccc2c[nH]nc2c1 C(=O)(CCCC(=O)OC(C)(C)C)NCC1CC(NC(CC(C)N(C)C)=O)C1 C1(C(=O)NC(C2CCCN2C(c2ccc(CCC#N)cc2)=O)C)CCCCNC1=O C1(O)(NC(CNC2C(NC(C(C3CCOCC3)OC)=O)C2)=O)CCOC1C c1(C(c2nnnn2CC(F)F)NC(c2ccnn2C)C)cc(Br)ccc1Cl c1(OCC(C)N(C(=O)C=Cc2ccco2)CC)ccccc1F c1(C(N(C2CCN(C(=O)C=CC(C)C)CC2)CC(C)C)=O)nnn2c1CCCC2 c1(C(N2CC(C)C(NC(c3nc(O)nc(O)c3F)=O)C2)=O)cc(Cl)cc(Cl)c1O N1CCCN(C(=O)C=C(Cl)Cl)C(C)C1.Cc1nc[nH]c1-c1cn(CCCC=O)nn1 CC(F)CC(=O)NCC(C)CN(C)C(C1(C(=O)OC(C)(C)C)CC1)=O c1(OC)ccc(Cl)cc1C(=O)NCCN(C(=O)C(Cc1ccsc1)NC=O)C(C)C C1(NC(C2C(C)C2)=O)CCCC12CN(c1cc(Cl)nc(CS(C)(=O)=O)n1)C2 c1(C(N2CCC(C(=O)OC)(CO)C2)=O)cc([N+](=O)[O-])n[nH]1 Cc1cc([N+](=O)[O-])cnc1NC1CCCC(CNC(c2cncn(C)c2=O)=O)C1 C1(OC)CCCC(OCCC(c2nccn2C)Oc2nc(-c3ccccc3)ns2)C1 c1(CSCC(C)C)ccccc1OC1(C)CC1.C1CC(=O)NN1CCCN(C)C CCCC(CC)C(=O)NCC(C)(CC(C)C)NC(=O)Cc1ccc2c(c1)CC2 c1(C(N(C)CCNC(c2cn(-c3ncccn3)cn2)=O)=O)ccnc(C2CC2)n1 c1(C(C(=O)NCC(CN(C(C=CC)=O)C)O)C)ccc(C(F)F)cc1 c1(C(=O)NC23CC(NC(C(C)NC(C)=O)=O)(C2)C3)ncnc2[nH]c(C(F)(F)F)nc12 c1(OCC)cc(OC(=O)N(C)Cc2c(Cl)cccc2Cl)ccc1Br N1(C(c2cnc(CC)s2)=O)CCOCC1CNC(=O)C(C1CC1)C1CC1 C1(C(=O)NC(C)CCN(C(=O)CCc2cncc(O)c2)C)CCC2(CCC2)O1 C(c1c(F)cccc1F)=CC(=O)NCC(CN(C(=O)CC1CCOC1)C)O N1(C(CN2CCC(C)C2)=O)C2CC=C(C(=O)NCCc3cscn3)C1CC2 CC1CON(C(=O)c2cccc(C3SCCS3)c2)C1 C1(C(C)C)(C(=O)NC(CNC(=O)C(C)(C)OC(C)(C)C)C2CC2)CCCO1 Cc1ccc(C(C)(C)C(=O)NCCC2(NC(C3CCC4CCC34)=O)CCC2)cc1 C12(C(=O)NCCC(C)NC(C3CCCN3CC(C)C)=O)CCC(N=[N+]=[N-])(CC1)C2 Cn1c(C(=O)NC(CNC(C2CCCC(O)C2)=O)CO)cc2sccc12 c1(C(=O)NCC(CO)NC(C(=O)NCCOC)=O)cnc(O)n1C N1(C(C=CC=CC)=O)CC2(CNC(c3occc3-c3ccccc3)=O)CCC1C2 c1(OCCCNC(c2c(SC(CC)C)ccnc2)=O)cc(C)cc(C)c1 CC(N=c1[nH]c2ccc(O)cc2s1)c1ccc(N2CCCC(C)C2)cc1 C#CCC(CC(=O)Nc1cc(CO)cc(F)c1)NC(c1ncoc1CC)=O C(=O)(CCCC(C)(C)C)NC1CCN(C(c2ccc(CC)c(C)c2)=O)C(C)C1 C(=O)(C(CNC(=O)Cc1cc(C)on1)CC1CCCC1)NCC(CC)C c1(C(N2CC(F)(CNC(C3(C)C(CC)CCC3)=O)C2)=O)cc(C)nnc1O C(CC(=O)N1CCC(CNC(CCOC)=O)(OC)C1)(C(C)(C)C)OC C=C1Cn2c(C(N3CCN(C(=O)C(C)CSC)C(C4CCCC4)C3)=O)nnc2S1 c1(CC(=O)NCC(CNC(C23CCCC2C3(F)F)=O)OC)ccc(C)c(Cl)c1 N1(C(CSCCC#N)=O)CCC(CF)(NC(C2CCCOC2)=O)C1 N#CC1CCCC(C(=O)NCCCOCCC(=O)NCC2CCS(=O)(=O)C2)C1 CCCCC(C)C(=O)NC1CN(C(c2cccc(C3CC3)n2)=O)CC1C CC(CCNC(=O)CC1CCCOC1)CCNC(c1cc(=O)n(C)o1)=O c1(C(=O)NCC2(C)CCCN2C(=O)CCF)ccc2c(Br)cccc2n1 c1(C(C(N2CCC(CN3C(=O)CCC3)C2)=O)=O)c(F)ccnc1F Cc1nn(C)c(C)c1CC(C)C(=O)NC(C)CC(C)NC(C1(C)C=CCCC1)=O Cc1nc(C)c(C(C)NC(=O)COC2CC(NC(=O)CCC3CCC(C)O3)C2)[nH]1 C(=O)(N=c1[nH]nc(-c2ccc(C)o2)s1)N(CC1CC(=C)C1)CC N1(C(c2ccc(OC)s2)=O)CCC(O)(CCNC(c2sc(C)cc2Cl)=O)CC1 c1(C(N2C(CNC(CCC(=O)N(C)C)=O)CC2)=O)cc2c(F)cc(F)cc2[nH]1 C1(CNC(CN(C)C(c2cccs2)=O)=O)CCC(NC(=O)CC2(C)OCCO2)C1 c1(C(=O)NC(C(C#C)(C)C)C)cccc(S(=O)(=O)N(CC)CC)c1 N1(C(C(NOC)=O)=O)CCN(C(C23COCC2C3)=O)CC(C)C1 C1(n2cc(C(C=C)(C)O)nn2)CCCN(C(=O)COCCN(C)C)CC1 CCCC(C)(O)CC(=O)N1CCC(CNC(C2CN3CCN2CC3)=O)C(O)C1 Cc1cccc([N+](=O)[O-])c1NC1CC(CNC(=O)CC2CC3(CCC3)C2)C1 c1(OC)nc(N2CC3CC2CN3Cc2nc(Br)cs2)ncc1F C1(CCC(=O)NCC2CCC2NC(=O)Cc2ccccc2)CCCC(=O)N1 c1(CC)cc(C(=O)NCCOCCNC(=O)CCC(C)c2ccccc2)ccn1 c1(C(=O)NC2CC2NC(=O)C(O)Cc2ccc(F)cc2)cccc2ncccc12 c1(N2CCC3(CC(NC(C(C)OCCC=C)=O)C3)C2)nc(C)cc(C)c1C#N C(CC(C)N=c1nc(N2CCC3(CC2)CC3C#N)c2ncccc2[nH]1)OC C1(C)(CNC(C2C(C=C)OCC2)=O)CCN(C(c2nocc2CC)=O)CC1 CN1CC(C(=O)NCC2CCCC(NC(c3cc(F)c[nH]3)=O)C2)CCC1=O C1(Cc2cn(CCCCCC)nn2)CCCN(C(=O)Cn2nc(C)nc2C)C1 C(=O)(CCCCCNC(=O)CC12CCCC1C2)NCC(C)(C)N(C)C C#Cc1ccc(OCC(=O)NC2CC(F)(CNC(=O)CCC3CC3=C)C2)cc1.CC c1(CC(=O)NCC(C)NC(CC2C(C)CCC2)=O)cccc(F)c1F C1(NC(CC2N(CC)CCC2)=O)COC2(CCN(C(=O)CNC(C)=O)C2)C1 c1(C(N2CCC(CNC(c3ccc(F)cc3)=O)C23CC3)=O)ccc2c(n1)CCO2 c1(C(N2CC(NC(C3CC(C)(C)C3)=O)C2)=O)cc(C(=O)CBr)ccc1O C1(C(CNC(c2c(C)ocn2)=O)F)CCN(C(c2c[nH]ccc2=O)=O)CC1 Cc1cc(C(=O)NC2CCN(C(=O)C(=O)NC3CC3)CC2C)c2c(O)n[nH]c2n1 N1(CC)CC(C(=O)NCC2(OC)CN(C(=O)C(C)(C)CC3CC3)C2)CCC1=O Cc1nsc(C)c1C(=O)NCC1CCN1C(=O)CC1CSCCS1 C1(CC(=O)NC(CC)CC(=O)NC2(C3CCCCO3)CC2)CCC2(CC2)CO1 c1(C(N2C(CNC(C(C)OC)=O)CC2)=O)nn(C(F)F)cc1Cl N1(C(c2ccc(C)nc2)=O)CCCOC(CCNC(C2C3CCCCCC23)=O)C1 c1(CNC(C2CCC(NC(c3csc(C)c3C)=O)C2)=O)nnc2n1CCC2 C(=O)(C(F)C(C)(F)F)NCC(C)(CO)OC.C12CC13CC(C3)NC2=O N12CCC3(CCN(C3)N(C)CC1=O)C2.c1(CN)cccc(Cl)c1.n1(CC)cccn1 [N-]=[N+]=Nc1ccnc(NC(C2CCN2C2CCCC2)=O)c1 c1(C(CNC(C2CNCC2O)=O)N(C)C)ccccc1Cl C1(C(=O)NCC(C2CCC2)NC(c2cncc(C)n2)=O)CCC(F)(F)CC1 N1(C(C(c2ccc(C)cc2)C2CC2)=O)CC2CC1CN2C(C1SCCS1)=O C1(CNC(c2c(C(=O)OC)scc2)=O)CCN(C(=O)CC(C)F)CC1C C1(C(=O)NC(CNC(C=NOC)=O)(C)CO)CC(C)(C)CCO1 Cc1cc(C2CC2)ccc1C(=O)NCC1CC(C)CCN1C(C1CCS1(=O)=O)=O C(CCCN=c1[nH]c2ccc(C(=O)OC)cc2s1)NC(C=CC=CCC)=O c1(CC)ccc(C(=O)NCCCCCCNC(C2CC2(F)Cl)=O)cc1Br Cc1cc(C)c(OCC(=O)NCC(CO)NC(C2(C)CCNC2=O)=O)c(C)c1 C1(COC)CC(CNC(=O)CCc2cc[nH]n2)N(C(c2cc(C(F)F)[nH]n2)=O)C1 Cc1csnc1C(=O)NCC(CO)NC(c1ccn(C2CC2)n1)=O C1(C(=O)NC(C=C)C2CCC2)CC=CCN1C(=O)C(C(C)OC)N(C)C C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)C(=O)N(C)C)C2(CCCOC2)C1 C(C(C)C)(C(O)C(=O)NCC(C)(C)CNC(c1cc(Cl)ccc1O)=O)OC c1(C(=O)NC2CC(CCNC(CNC(C3C(C)C3)=O)=O)C2)ncc(N)cc1Cl c1(C(=O)NCC(C)NC(CCNC(CC(C)C)=O)=O)cnc(Cl)c(F)c1N N1(C(C2N(C(Cc3c(C)n(C)nc3)=O)CC(=O)C2)=O)CC2CC1CS2=O C1(F)(C(=O)NCC(C=C)O)CCN(C(=O)CC(C)n2cccn2)CC1 C1(NC(c2n(CCOCC)nnn2)c2nocc2Br)CCOCC1OCC O=C(C1CCCc2nccn21)NC1CC12CCN(C(=O)CCOCC(F)F)CC2 c1(C(=O)NCCCCC(C)NC(=O)CC2COCCO2)ccc(Cl)c(Cl)c1N c1(OC)ccc(-c2nc(-c3nccn3N3CCOC3=O)c(C)o2)cc1OC C1(CNC(c2cc(C(F)(F)F)ccc2C(F)(F)F)C)CC(C)NC(=S)N1 Cc1csc(=NCC(=O)NCC(C)(C)CNC(c2cc[nH]n2)=O)[nH]1 C(C1=NOC2COCC12)CNC(COC1CCN(C(C(CCCC)O)=O)C1)=O C1(NC(C2N(C(=O)COCC3CCCC3)CC=C2)=O)CCCCC12CCC2 c1(CC)ccc(F)cc1C(=O)NC1CN(C(=O)C(C)C(C)CC)CC1CO C(=O)(C1CCCCc2ccccc21)NCC1(O)CN(C(Cc2cc(C)no2)=O)C1 c1(C(=O)NCC2CCN(C(C(c3ccc(F)cc3)CC)=O)C2)cccc(N)c1C C1(C(N2CC(N(C(c3cn(CC=C)nn3)=O)C)C2)=O)CN2CCN1C(C)C2 N1(C(C2C(=C)CC2)=O)CC2CC2(CNC(c2cncc(C(F)F)c2)=O)C1 c1(OC)ccc(CNC2CC2C(=O)NCc2cc(Br)ccc2F)c(F)c1F Cc1cc2ccc(C(=O)NC(CO)CCCCNC(=O)CCC3CC3C)cn2c1 c1(CC)oc(C(=O)NC2CC(CCNC(=O)C(c3ccccc3)C)C2)cc1C c1(C(N(C2(CC(=O)NC3CCNC3=O)CC2)C)=O)cc(O)ncn1 C(CCCC(=O)NC1CCC1NC(c1ccn(C(C)C)c1C)=O)SC c1(NC)cc(C(N2CCC(NC(c3nc(C)cs3)=O)C(C)C2)=O)cc(Cl)n1 C(C(CNC(C1(NC(=O)CCc2ccccn2)CC1(C)C)=O)C(C)C)OC c1(C(=O)NCC(C#C)CC)cccc2ccc(O)nc12 C1(NC(COC(CC)C)=O)CCC(CNC(c2nc(C(C)(F)F)cs2)=O)C1 C(CCC(=O)NC(C)CCNC(C)=O)N(C(=O)OC)C.C1(CCC(=O)N)CC(F)(F)C1 N1(C(C(C)NC=O)=O)CCC(C2(C(=O)N(CC(N)=O)C3CC3)CCOCC2)CC1 N(C(=NCCC(C)=O)NCc1cc(F)c(F)c(F)c1)C1CC(C)(CC)C1 C1(NC(C(C)n2cnnn2)=O)CCC(O)CN(C(=O)C=CC(F)(F)F)C1 N1(C(c2cc(C)nc(O)n2)=O)CC2CC1CCC2NC(c1cc(Cl)cc(Cl)c1)=O CC(C)C(C(=O)NCC(C)(C)CN(C(=O)C(O)C1CCC1)C)N(C)C c1(SC)cncc(C(=O)NC2COCC2NC(c2c[nH]c(=N)o2)=O)c1 N1(C(C(C)OC2CCOC2)=O)CCC(NC(=O)C2=CC(C)(C)C2)C2(CCC2)C1 C(=O)(CN(CSc1ccc(Br)cc1)N(C)Cc1ccco1)OC N1(C(C(n2ncc(C)c2)C)=O)CC2CC(O)C1C2NC(c1cccc(Cl)c1O)=O c1(CC(=O)NC(CC=C)CNC(=O)C(n2cc(Cl)cn2)C)n[nH]c2ccccc12 N1(C(C2C3COCC23)=O)Cc2ccc(F)cc2C1.CC12CCCN(C1)C2=O c1(C(=O)NC2C(CNC(c3c(OC)scc3)=O)CCC2)ccccc1C(N)=O c1(C(=O)NCC(CC)NC(C2CCCCC2(F)F)=O)cc(Br)c2occc2c1 c1(C(N2CCC(CC(C)NC(C(CC)OC)=O)CC2)=O)cc(N)c(Cl)cn1 c1(C(C(=O)NC)N(c2ccc(C(F)(F)F)c(C)c2)CC)ccc2nonc2c1 N1(C(C(CC(C)C)OC)=O)C2CCC1CC(CNC(c1cc(C(F)F)no1)=O)C2 C(=O)(C(CCOC)NC(=O)OC)NC(CC)CN(C)C CC1CN(C(C2CCS(=O)(=O)CC2)=O)CCN1C(=O)CN1CSCC1=O N1(C(Cc2c(C)occ2)=O)CCC(NC(=O)C=C2CCOCC2)C1(C)C CC(C)C1=NOC(C(=O)NCCCCC2CN(C(C3CC4C=CC3C4)=O)C2)C1 c1(OC(C(=O)N(c2c(OC)ccc(F)c2)C)C)ccc2c(c1)CCC2 C1(C(CO)NC(c2cccc(Cl)n2)=O)CCN(C(C2CC(O)C2)=O)CC1 C1(C(=O)NCC)CCC2CCCCN12.C123CC(C1)(C2)C1(CCC1)OC3=O CC(C)CC(C)CC(=O)NCC(C)(C)CCNC(=O)C=CC(C)(C)SC C1(C(N(C(CCNC(c2cnn(CCOC)c2C)=O)C)C)=O)CCC(C)(C)CO1 CC(C(=O)N1CCCC1CNC(c1cncc(O)c1)=O)P(C)(C)=O C1(NC(c2ccc(C)cc2O)=O)CC2CC1CN(C(=O)CS(=O)(=O)CC1CC1)C2 CCC(CC(=O)NCC1CN(C(c2ccsc2C#N)=O)C(C)(C)C1)C(F)F N1(C(=O)CCCc2ccc(O)cc2)CCC2C(CCCN2c2ccncn2)C1 C(c1cccc2ccccc12)=CC(=O)NC1CN(C(c2c(C)occ2)=O)C2C1C2 c1(NC(C(C)NCc2cn(CCOC)nc2)=O)ccc(Cl)nc1 N1(C(C(CCC)OC)=O)CCCC(NC(c2cnn(CCN(C)C)c2C)=O)C1C C1(NC(C(Cc2c(C)noc2C)C)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 S(=O)(=O)(CCC(=O)NC(CNC(=O)CN1CC=CC1)C1CC1)NC CS(=O)(=O)CC(=O)NC1CC(F)(CNC(=O)CC(c2cccs2)NC(N)=O)C1 Cc1nnc2n1CC(C(=O)NC1(CNC(c3cc[nH]c(=N)n3)=O)CCC1)C2 n1(CC=C)c(N(C(C)CCOC)Cc2csc(C)n2)nnc1COC c1(C(N2CC(F)(CNC(C(CC)=CCCC)=O)C2)=O)ccnc(Br)c1N C1(NC(C(c2ccc(Cl)s2)C)=O)CCC(C)(CNC(=O)C=Cc2ccoc2)C1 CCC(C(=O)N1CC(O)(C2CCCN2C(=O)COCc2ccncc2)C1)SC c1(OC)cc(C#N)ccc1-c1noc(-c2cc3scnc3[nH]2)n1 C1(C(N(CC)CC2CCCO2)=O)CCC(CNC(C2OCCC2C)=O)O1 C(C)(C)(CC(=O)NC(C1CCCN1C(=O)CC1(N2CCCC2=O)CC1)(C)C)OC N1(C(c2n(CC)nc(C)c2)=O)CCC2(CCC(NC(=O)CCCN(C)C)CC2)C1 N1(C(C2(SC)CCC2)=O)CCN(C(c2nn(C)cc2N)=O)C(C)C1 CC(C)C(CCNC(=O)C(C1CC1)N(C)C)NC(=O)CN1CC=CC1 C=Cc1ccc(NC(C2CCN(C(c3cc(C(C)C)n[nH]3)=O)C2C(C)C)=O)cc1 C(C(C)(C)C(=O)N(C(C)CC(N1CCCC(CC(C)(C)C)C1)=O)C)OCC CCCCC(CNC(=O)CCc1cccnc1C)NC(C1(C)CSC1)=O CC(CC(=O)NC1CCNC(=O)C1)C(C)(C)NC(c1cccc2cncn12)=O c1(-n2ccc(CC(=O)NC(C)C(CO)N(C)C)n2)ccc(F)c(F)c1 C1(O)(CC(=O)N(C(CNC(c2cncc(C)n2)=O)C)C)CCCN(C)C1 c1(NC2CCC(N(C)C(=O)Nc3ccc(Cl)cc3)C2)cc(F)ccc1N1CCCC1 C1(C#CC(=O)N2CCC(N(C(=O)CC(C)F)CC3CC3)CC2)(CC)CC1 c1(CN(C)C(C2CCCCCC2)=O)cccc(CNC(c2cc(Cl)on2)=O)c1 Cc1ccc(C=CC(N2CCN(C(=O)CCc3cn(C)cn3)CC2CO)=O)cn1 c1(OC)ccc(C(=O)NOCC(CCNC(C(=O)O)C(=O)O)OC)cn1 c1(C(=O)NC(c2ccc(CNC(C(CC)COC)=O)cc2)C)ccc(Cl)c(C)c1 C(=O)(C(=O)N=c1ccn(CCC(C)C)[nH]1)NC(c1nc(CC)[nH]n1)C C(CN=c1ncc(F)c[nH]1)C1(CO)CCN(C(=O)C(F)OC(F)(F)F)CC1 c1(NC(c2ccccc2)COC)[nH]c(=NC2CCCCCCC2)nc2scnc12 N1(C(c2c(CC)oc(C)c2)=O)CCC(OC)C(C)(C)C1.C1=CC=CCNC1=O c1(C(=O)NC(CNC(C2CCCN2C2CC2)=O)CO)cc(F)cc2ccncc12 C(=O)(CC1=CCOCC1)NCC1(F)CCC(NC(C(C(C)(C)C)OC)=O)C1 n1(CCC(=O)NC2CC(C)(NC(=O)CCC3CC3)C2)cc(C#N)c(O)nc1=O C(CC1=CCN(C(C2(CC3CC3)CCCO2)=O)CC1)NC(C=C1CCN(C)C1)=O C1(OC)CC2CC(NC(=O)C(CO)NC(=O)CCc3nncn3C)CC12 C1(CCN(C(C(F)=CCC)=O)C)CCCCN1C(=O)CC1CCC(=O)N1C c1(C(N2CC(NC(C3(C(F)(F)F)CCCCC3)=O)C(F)C2)=O)cc[n+]([O-])cc1 C1(NC(CC2CC(C)(C)N(C(C3C4CC(=O)CC34)=O)C2)=O)CCCCC12CCC2 c1(C(N(CC(C)NC(C2CCS(=O)(=O)N2)=O)CC)=O)noc2c1CCCC2 C1(NC(CC2CC(NC(C(C)SC)=O)C2)=O)CCc2n[nH]cc2C1 C1(C(N2CC(CNC(COC(CC)(C)C)=O)C2)=O)CCCCN1CC1CCCC1 C1(C(=O)NC(C(N)=O)CO)(NC(c2ncncc2Cl)=O)CC(F)(F)C1 CCCCS(=O)(=O)CC(=O)N1CC2CC1CN2C(c1[nH]nc([N+](=O)[O-])c1Cl)=O Cc1cccnc1C=CC(=O)NCC1CCN(C(=O)C=Cc2ncco2)C1 c1(CCC(=O)NCC(CC)NC(COC(CC)CC)=O)nc(C)c(C)[nH]1 N1(CC(=O)OC)CCN(C(C)=O)C(C)C1.c1(C(N2CC2)=O)ccc(C)cc1F c1(CC(=O)NCCCNC(CC2CCC(C)(C)CO2)=O)ncn2c1COCC2 C1(C2CCOCC2)(C(N2CC(c3cn(Cc4nc(C)sc4)nn3)C2)=O)CC1(F)F C(=O)(C1CCc2ccccc21)N1C(C=CC(NOCC2(C)CC2)=O)CCC1 C1(NC(=O)CC2CCCSC2)CCC2(CC1)CN(C(C1CN3CCN1CC3)=O)C2 c1(CC(=O)NC(CC=C)CNC(=O)C(C)O)cc(OC)ccc1OC Cn1nc(Br)cc1CC(=O)NC12CC(CNC(=O)COCC(F)F)(C1)C2 c1(NC(CN(CCNC(C2(O)CC2)=O)CC)=O)c(C)nc2ccc(F)cn12 CC1CCC(C)(C(N2CC(CN(C(=O)CCCC#N)C)C2)=O)C1 C1(C)(CC)CN(C(C(=O)Nc2ccccc2OC)C2CCOC2)CCO1 c1(SC(C)(C)C)ncc(C(=O)O)cn1.C123CC(C1)(C2)CNC3=O N1(C(c2cc(CCC)c(C)s2)=O)CC(NC(C2CC=CCO2)=O)C(C)(C)C1 N1(C(C(CC=C)N(C)C)=O)CCC2(CC1)CC2N(C(=O)C=C1CCC(C)C1)CC CC(C)C(F)C(=O)NCCC1CC(NC(c2csc(Br)c2Cl)=O)C1 N1(C(CC)C(N)=O)CCN(C(=O)CCC=CC(=O)N(C)C(C)C)CC1 C1(CNC(CCSCC)=O)(NC(=O)CN2CCCCC2C)CCCCC1 c1(C(N(C2CCN(C(C3C(C)C3C)=O)C2)CC)=O)cc(F)c(C)cc1Cl N1(C(c2ccc(OC)o2)=O)CC(NC(=O)CCc2ccc(C)nc2)CCC1C C1(C(N(C2CN(C(CC3(OC)CCC3)=O)C2)C)=O)CC(=O)CO1 c1(OC(C)C)nc(C(N2CC(CCNC(=O)COCP(C)(C)=O)C2)=O)cc(O)n1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)CC2C)csc2c(F)cccc12 C1(C#CC(=O)NC2CC(O)(CNC(=O)C3=CCCCC3)C2)(CC)CC1 N1(C(c2cc(C)n(C)c2)=O)CC2CCC(C1)N2C(=O)CSC1CCS(=O)(=O)C1 c1(C(N2CCN(C(c3cnsc3)=O)C(CC(F)(F)F)C2)=O)cc(Cl)c(F)cc1F N1(C(C=Cc2c(C)cccc2)=O)CCC2CN(C(c3cc4c(s3)COCC4)=O)C2C1 c1(NC(C2CCCC(N3CCCS3(=O)=O)C2)=O)ccc(CCN2CCCC2)cc1 c1(C(=O)NCC(CNC(c2n(CC)ccn2)=O)CO)ccc2ccsc2c1 C(=O)(C(CC)C(=O)N1CCCC1CNC(=O)C(C(C)C)N1CCCCC1)OCC C=C1CC(C(N2CCC2)=O)(CNC(=O)CNC(=O)OC(C)(C)C)C1.C1(Cl)(C)CCC1 C1(C(=O)NCC2(C(F)F)CCN(C(COCCC)=O)C2)CC2CCC(C1)O2 Cc1cnc(NC(c2cc(Cl)sc2Cl)C)c(S(=O)(=O)NCCN2CCCCC2)c1 c1(-c2n(CCC#C)c(N(C)Cc3ncc(C)s3)nn2)ccc(OCC=C)c(C)c1 n1(C(C)C)ccc2cc(C(=O)NC3CCN(CC4CC4(F)F)CC3)ccc12 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC(NC(C2CC3(CCC3)C2)=O)C(O)C1 Cc1cccc(-c2cc(C(=O)NCC(C)(C)CNC(=O)C(C3CC3)N(C)C)on2)c1 C12(C(=O)NCCCCCNC(C(C)O)=O)CC3(F)CC(F)(C1)CC(F)(C2)C3 c1(CC)cscc1C(=O)NCCC(C)N(C)C(c1cnc(-c2ccsc2)s1)=O CC1(C)OCCOC1C(=O)NCC1CCCCN1C(=O)C(c1ccc(Cl)cc1)=O C1(NC(C(C)=C2CCCC2)=O)C=CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(=O)NC(C2CCN(C(c3nc(COCC)sc3)=O)C2)C)c[nH]ccc1=N c1(C(N(C(C)CNC(C2(C(F)F)CC2)=O)CC)=O)ccc(Cl)cc1Cl C(C(C)CC(=O)NNC(=O)C(C)(C)CCCCNC(c1cc(C)n(C)n1)=O)OC c1(C(N2CC(CCNC(=O)Cc3ccsn3)OCC2)=O)ccc2n[nH]cc2c1Cl c1(OC)ccccc1NC(=O)C(C)N(C1CCN(CC2CC(O)C2)CC1)C C1(CC(=O)N(CCN(C(C)C)C(c2cnn(CCF)c2)=O)C)CN2CCN1CC2 N1(C(C2(OC)CCN(C(CC(CCC)C)=O)C2)=O)CCCCCCC1C C(C)(CCCN=c1cc[nH]cc1[N+](=O)[O-])NC(C1CC(CCC)OCC1)=O C1(C(N2CC(CCNC(=O)C(C)n3ccnc3)(OC)C2)=O)(CO)CCCCO1 C1(OC)CC(C(=O)NCc2ncsc2C)N(C(=O)C(C)COC(C)C)C1 c1(OC)ccccc1CCC(=O)NCC1CC(NC(C2CC(OC)C2)=O)CC1O Cc1c(C(=O)NCCN(C2CCC(CCC(=O)N(CCCO)C)C2)C)nnn1C N1(C(c2c[nH]c(=NC)o2)=O)CCC(NC(C2CN(C(=O)NC)C2)=O)CC(O)C1 C1(C(=O)OC)CCOC1C(=O)NC12CC(NC(c3cc(C4CC4)[nH]n3)=O)(C1)C2 c1(NC(CCNC)c2cccs2)cc(NCCc2cnn(C)c2)ncn1 CC1CCCCC1CC(=O)N(CC(O)CN(C(=O)CN(C1CCSC1)C)C)C CC1CCNCCN1C(c1cncc(O)c1Cl)=O.C(c1ccsc1)=CC=O c1(C(N(C2CCN(C(C=CCCC)=O)C2)CCC)=O)ccc(=O)n(O)c1 N1(C(CCC#C)=O)CCC2(CC2NC(=O)CN(C)CCO)C1 N1(C(c2c(N(C)C)nccc2)=O)CC2=C(C1)CN(C(=O)CCC1CCOC1)C2 C1(CC#C)(C(=O)NCCC2CN(C(=O)C(C)(C)N3CCCC3)C2)CCCO1 C1(CNC(c2n(CC)ncc2)=O)CN(C(C2(OC)CCC(C)(C)C2)=O)CCCO1 c1(OC)c(Cl)cc(C(=O)NC2CCCN(C(=O)CN3CC=CC3)C2)nc1Cl C1(NC(C(C)OCC)=O)(CF)CN(C(=O)COCC2CCC2)C1 c1(CC(=O)NCCNC(C2(C)CC=CCO2)=O)ccc([N+](=O)[O-])cc1Cl C1(CNC(COCCCC)=O)C(C2CC2)CCN1C(c1cc(Cl)ccc1C)=O c1(C(=O)NC(CC=C)CNC(C2CCCCS2)=O)cccc(N2CCOCC2)n1 C#CCCCC(C(=O)NC(C)(C)CC)N1CCC(OCCN(C)C)C1 c1(NC(C(=O)NC(CC)Cc2ccc(Br)cc2)=O)ccc2c(c1)CCCN2C N1(C(=O)CCc2ccc[nH]2)CC2CCCC2(C(N2CC(F)(C3CC3)C2)=O)C1 Cc1nc(NC2CCCc3n[nH]cc32)c(Cl)cc1C#N.C(=O)(C(F)(F)F)NCCC(=O)O N(C1CCc2cccnc21)C(C(CC(C)(C)C)NC(=O)CC1CC(F)C1)=O C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(c2cocn2)=O)C1 c1(C(CNC(c2c(CC)ncs2)=O)NC2(CO)CCCC2)cccc(OC)c1.OC C1(O)(C(=O)NCCOCCNC(Cc2nc(C)oc2)=O)CCC(C)CC1 N1(C(c2cc(C)sc2C)=O)CC(C2CC2)(C(=O)NCCc2ccncc2)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C)CCN(C(C(COC)C)=O)C1 CC1(CC(=O)NCCC2CCCCC2)CCN(C(C2CCCO2)=O)CC1 C(=O)(C(CCC1CC=CCC1)N1CCN(c2ccc(OC)nn2)CC1)NCC=C C1(NC(C(C2CCC2)OC)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC1 c1(CC(=O)NC2C(CNC(CCSCCCC)=O)CC2)c[nH]c2ccc(F)cc12 C=CC(CC)CC(=O)NCc1nc(CNC(C23CC(OC)C2C3)=O)cc(O)n1 C1(N(C(=O)CCNC(=O)CO)C)COCCN(C(C2CC(=O)NC2(C)C)=O)C1 C1(NC(COCCC#C)=O)CC2CC(C1)N(C(=O)C=CC(c1ccccc1)=O)C2 c1(C(=O)NC2CN(C(C=CC(=O)OCC)=O)CC2O)cc2scc(Cl)c2[nH]1 c1(C(=O)NCC(CO)NC(c2c(C(C)(C)C)con2)=O)ccc(F)c(Cl)c1F C1(C(=O)NC(CN(C(c2c(OC)ccc(C)n2)=O)C)(C)C)CCC2(C1)CC2(F)F c1(C2N(c3nnc(CCC)n3CC)CCC2)cccc(F)c1 C1(NC(C2(OC)CCSCC2)=O)CCN(C(=O)CC2CCC3CC23)CC1(C)C CC(C)S(=O)(=O)CC(=O)N1CCC1c1cn(-c2cncc(OC(C)(C)C)c2)nn1 CN(C1CCc2c(F)cccc21)C(C1CC(=O)N(C2CCCC2)C1)=O C1(CNC(CNC(CC)=O)=O)CC(C)(C)CCC1NC(=O)CN(CC)CC C=C(C)CC(C(=O)NC1COCC1C(=O)NC1CCC1(C)C)OC CC(C)C(F)(CNC(C1C2CC(=O)CC12)=O)C(=O)NCc1cccnc1O c1(C(N2CC(C)(C)C(NC(C3CCOC3)=O)C2)=O)cc2cc(Br)cn2cn1 C1(NC(C(C)SC)=O)CN(C(c2c(C)nc(C)n2O)=O)CC2(CCC2)C1 C1(C(=O)NC(C)CCCNC(=O)Cc2cc[nH]c2)CCCN(CCC2CC2)C1 C(=O)(C1=CCSC1)ONC(C1(C)CC(NC(c2ccccc2)C)C1)=O N1(C(c2cnc(-c3c(F)cccc3F)s2)=O)CCc2cc(O)ccc2C1 C1(O)(CCNC(C2CC(=O)NC2)=O)CCCN(C(c2cncc(O)c2)=O)C1 CCC(CC(=O)NCC1(C(=O)NCC(=C2CCCCC2)F)CCCO1)OC(C)=O C1(C(N(C)CC2CCC2)=O)CCC(n2cc(Cc3cnc(C(C)(F)F)s3)nn2)C1 C1(NC(CC(C)(C)C)=O)CCC(C)(NC(=O)Cn2ccnn2)CC1 CCCC(CCC)CC(=O)N1CCC(NC(=O)CCN2CCCS2(=O)=O)C1 c1(OC)cc(C(=O)Nc2cnc(Cl)c(CO)c2)c(-c2cncn2C)cn1 N1(C(c2cnn(CC)n2)=O)CC(NC(c2cncn2C(C)C)=O)CC(F)C1 C1(C(=O)NCCC2CCN(C(C(CSC)(C)C)=O)C2)CCCC1C1CC1 N#Cc1ccc(F)c(NC(C2CCCC2NC(=O)CCc2ncc[nH]2)=O)c1 N1(C(C(CCOCCO)NC(C(CSC)(C)C)=O)=O)CCCN(C)CC1C c1(C(=O)NC2CN(C(CC3C(C)(C)C(O)C3)=O)C2)nncc2c1CCCC2 C1(CNC(C(C)SC)=O)CCCN(C(=O)C=Cc2ccsc2C(F)(F)F)C1 C(=O)(CCCC(O)c1ccccc1)NC(C1CCCN1CC1CCOC(=O)N1)C C(=O)(CC(C)(C)C(F)F)N1CCC(N(C)C(C2C(=O)NCC2(C)C)=O)CC1 C(C(C)CC(=O)N1CCC(C(=O)NCCc2n[nH]cc2C(=O)OC)C1)OC c1(NC(CCN(C)Cc2ccncc2)=O)cc(C#N)ccc1F c1(CCC=C)ccc(C(=O)NCC=CCNC(C2CN(C)CC2C)=O)cc1 c1(C(=O)NCc2cc(C(N3CCC(O)(CC)C3)=O)sc2)ccc(C)c(O)n1 C(=O)(C1CCCn2c(C)nnc21)N1CCC(C)(NC(c2nn(CC)c(O)c2)=O)C1 CC12CN(C(=O)CN3CCOC3=O)C(C(=O)NC3(C(=O)C4CC4)CC3)(C1)C2 c1(C(=O)NC(C)CC(=O)NCCC2CCCC2)cc([N+](=O)[O-])c[nH]1 N1(c2nc(N3CC(C)C(N(C)C)C3)nc3c2ncs3)CCC(C)(O)C(C)(O)C1 N1(C(C(CSC)O)=O)CCCCC1C1(NC(c2cccc(F)n2)=O)CC1 Cc1ccc(Br)c(C(=O)NCCCC(C)NC(=O)COCCC(C)C)c1 N1(C(c2cnnc(Cl)c2)=O)CCCC(C2CCN(C(c3cc(Cl)on3)=O)C2)C1 C1(NC(c2ccnc3cc[nH]c23)=O)CN(C(=O)CC2=CCOCC2)CC2(CC2)C1 C(=O)(C(C)(C)C(C)(F)F)NCCC(C)N(C(C(C)OCCC=C)=O)C C1(NC(c2cc(C)c(Br)o2)=O)C2CC1CN(C(C1CCSCC1)=O)C2 c1(C(=O)OC)csc(C(N2CC(C)C(F)C2)C(=O)NCCCSC)c1Cl Cc1ccccc1CC(C)C(=O)NCC#CCNC(C1(C(=O)NC2CC2)CC1)=O C1(NC(C(C(C)C)NC(C)=O)=O)CCN(C(=O)Cc2cc(C)cc(C)c2)C(C)C1 C1(NC(c2nc(COC)sc2)=O)CC2CN(C(=O)C(F)(F)C3(O)CCCC3)CC12 CCCC(CNC(=O)CCc1csnn1)NC(C1CCN1C)=O Cc1ncc(CNC(=O)C(C)CN(C(=O)C(=C2CCCCC2)F)C)o1 N1(C(CC2CCCC(NC(C=CC(CC)C)=O)C2)=O)CCCC2(CCC2)C1 C1(CNC(C2C(C)=C2)=O)(NC(=O)Cc2cnco2)CCC1 C1(NC(c2ccc(OC)s2)=O)CC(NC(=O)C=CSC)C12CCC2 Nc1c(C(N2CC(CNC(=O)Cn3cnc4ccccc34)C2)=O)cc(F)cc1Cl C12(N(C(C3CN(C(C4C(C)(C(C)C)C4)=O)C3)=O)Cc3ccccc3)CC(F)(C1)C2 c1(C(N2CC(CC)N(C(c3ncnc(O)c3Cl)=O)CC2)=O)ccc2snnc2c1 CCC(C)CCCCC(=O)NCC1CCC2(CN(C(c3c(Cl)cnn3C)=O)C2)O1 C=CC1CCN(C(=O)CC2CC(F)CN2C(=O)C(C)NC(=O)NC)C1 C=CCCCCC(=O)N(CC(CC)NC(=O)COc1ccccc1C(C)C)C C1(C(N(CCSC)C)=O)CSCCN1S(=O)(=O)Cc1cccc(C)c1 C1(C(=O)NCC2(F)CC(NC(c3c[nH]c(=N)o3)=O)C2)CS(=O)(=O)CC(=O)N1 C1(C(N(C2CN(C(c3cccc(OCC(F)(F)F)c3)=O)C2)C)=O)CCC(C)(C)C1 CC(C)CC(C(=O)N(C(C)C(=O)NOC1CCOC1)C)C(N)=O n1(C(C)C)ncc(Br)c1CC1CC1.[nH]1nnn(C2CCCC(CC3CC3)C2)c1=O C#Cc1ccc(Br)c(C(=O)NCC(C)NC(C2CCN(C)S2(=O)=O)=O)c1 C1(CC)(NC(=O)CC(C)(C)C)CCCN(C(C2CC2c2sccc2C)=O)C1 C(=O)(N=c1cc[nH]cc1F)C1CCCC(NC(c2cccc(O)c2O)=O)C1 N1(C(CC(C)C(F)F)=O)CC(CNC(c2cn3c(n2)CCC3)=O)CC12CCC2 N1(C(C(C)=CC)=O)CC2CCOCC2(NC(=O)CCCc2ccsc2)C1 CCCC(C)(O)CNC(C1(CCNC(=O)Cc2coc(C)n2)CCC1)=O c1(N2CC(c3c(NCC4CC(OC)C4(C)C)nco3)C2)ncc(C#N)cc1Cl c1(C(N2CC(C(C)NC(C3CS(=O)(=O)C3)=O)OCC2)=O)ccc2nc[nH]c2n1 N1(C(CC2(C)CCCC2)=O)CCCC(C)(CNC(C2CC23CCCC3)=O)C1 c1(C(N2CC(NC(CC(C)n3cccc3)=O)CC2(C)C)=O)ccc2occc2c1 c1(C(=O)NC2CC(CNC(C3(COC)CC=CCC3)=O)C2)c(N)ccc(C)c1F NC(=O)CCCCC(=O)NC1CCC(C(=O)NCCCNC(=O)C2CC2)CC1 N1(C(C(CC2CC2)OC)=O)CCC2C(NC(c3cc(C(C)C)no3)=O)C2C1 S(=O)(=O)(c1c[nH]ccc1=NCCC1CCCC1(F)F)NCCN=S(C)(C)=O Cc1cnc(C(N2CC(C(=O)NCC(F)Cl)C(C)C2)=O)c[n+]1[O-] c1(CNC(CC2OCCN(C(c3c(CC)cns3)=O)C2)=O)cnc2n1CCC2 C(=O)(C#CC1CCOC1)Nc1c(C)cc(NC(C2C3CC4C(C3=O)C24)=O)cc1 C1(C)(N(C(CC(C)n2cccn2)=O)CC(=O)OCCC2(O)CCCC2)CCSCC1 CN1CCCC12CCN(C(=O)CCC(C)(C)NC(=O)COC1CC1)C2 C(=O)(C1=NOC(C)(C)C1)NCC1CC(C)N(C(c2ccsc2Cl)=O)C1 n1(CC(=O)NC2C(NC(C3(C)CCC3)=O)CCC2)cc([N+](=O)[O-])cn1 N1(C(c2cn(C)nc2)=O)CCC(NC(=O)CCc2nc(O)n[nH]2)C12CCCC2 c1(C(=O)NCCN(C(=O)CC2CC(C)(C)OC2=O)C(C)C)ccc2cnoc2c1 C(=O)(CCCCCS(N)(=O)=O)N1CC2(CN(C(c3c(C)c(N)ccn3)=O)C2)C1 CC(C)CCCC(=O)N1CCCC1CC(=O)N(CCO)CC1CC1 C=C(F)C1(CC(=O)NCC2CCC(N(C(=O)C(F)=CCCF)C)CC2)CCC1 CC(c1cnn(C)c1)=CC(=O)NCC1CC2(CC2)CN1C(C1CCCS1(=O)=O)=O N1(C(C(C(=C)C)(C)C)=O)CCCC2(C1)C(NC(=O)Cc1occc1C)CCN2C C1(C(=O)NC(C=C)COC)CCCN(S(=O)(=O)CC2CC2)C1 C1(NC(C2CCC(C)O2)=O)COC2(C1)CN(C(c1cc(Cl)on1)=O)C2 C1(NC(C2(F)CCN(C(C3(C#N)CCCO3)=O)C2)=O)CC12CCOCC2 c1(C(=O)NC2(CC=C)CCN(C(=O)COCC(C)C)C2)cncc2cccnc12 CC(C)(C)CC(O)C(=O)NCC1(F)CC(NC(=O)CC2CCCC2(F)F)C1 C1(=O)C(CC(C)C)NC(=O)CC2CCN12.c1(CC)onc(C)c1CC CC1CN(C(=O)CN(C)CCO)CC(C)C1NC(c1cc2sccc2s1)=O Nc1ccc(-c2noc(-c3cnc(-c4cccs4)o3)n2)c(Br)c1F c1(C(N2C3CC(CNC(c4c(C)ccs4)=O)(OC3)C2)=O)cnn2c1OCC(C)C2 CCC(C)(C)CCCC(=O)OCC(N=[N+]=[N-])C(=O)OC(C)(C)C N1(C(=O)NCCCc2ccc(F)cc2)CC2CC(O)CC(C2)C1 C=CC1(CC(=O)NCC2(F)CC(NC(=O)CNC(=O)CNC(=O)OC)C2)CCC1 C(=O)(CCC(CF)CF)N1CCCCC(C(N(C)Cc2cncs2)=O)C1 c1(C(N2CCC(O)C(CO)C2)C(=O)NCCCC)ccc2cccnc2c1 C1(NC(C2(NC(C(C(C)C)C3CCC3)=O)CC(F)C2)=O)CCC(C2CC2)C1 C(N(C)N1CCN(S(C)(=O)=O)C2(CCCC2)C1)c1ccc(SC)cc1 C(CC(C)C)(C(C(=O)NC1CCOC1)N(c1ccco1)Cc1nc(C)no1)OC CCCC(C(O)C(=O)NCCN(C(C)C)C(C)C)NC(=O)C(F)OC(F)(F)F C=CCC(C)(C)C(=O)NCCC1(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1 c1(C(CC2(OC)CCC2)=O)ccc(S(=O)(=O)Nc2ccn3nccc3n2)cn1 c1(C(=O)NC(C2(O)CN(C(c3c(C)nsc3N)=O)C2)C)csc2cc(Cl)cnc12 C1(N(c2cnn(C)c2)CC)CCCN(C(=O)C(N)=O)CC1 c1(C(N2C(CNC(=O)Cc3ccc(F)cc3C(F)F)CC2)=O)n[nH]c2c1COCC2 C1(C(=O)OC)CC2(CCCC2)CN1C(c1cc(Cl)cc([N+](=O)[O-])c1)=O C12(CNC(c3ccc[nH]3)=O)CC(C1)C(NC(C1CCCC(F)(F)C1)=O)CO2 CCC(N=c1cc(C)c(C#N)c(C)[nH]1)C1CCOC1.c12ccccc1NS(=O)(=O)C2 CN1CCC(=CC(=O)NCCC(O)CNC(c2ccccc2C(F)(F)F)=O)CC1 c1(C(=O)NCCC(C)(C)NC(c2cccnn2)=O)ccc2sncc2c1 N1(C(C2(OC(C)C)CCC2)=O)CC(NC(c2scnc2Cl)=O)CC(O)C1 c1ccc(F)cc1[N+](=O)[O-].N1(c2nc(=N)s[nH]2)CCNC(CC(F)(F)F)C1 CC1S(=O)(=O)CC1C(N1CCC(N(C(=O)CCc2cnc[nH]2)CCO)CC1)=O C1(NC(COCC)=O)CCC(N(C)C(c2c[nH]c(C(=O)OC)c2)=O)C1 C1(CNC(=O)CSC(F)F)CC(C(=O)NCCCc2cnccn2)=NO1 C(CC(C)C)(C(=O)NC(C)C(=O)NCC(C)(C)C(N)=O)OC C1(C(=O)OC)CN(C(C2CCCCC(c3ccccc3)C2)=O)CC(C)O1 c1(N2CCCC(NC(c3cscc3Cl)=O)CC2)ncnc2cccc(F)c12 N#Cc1ccc(CC(=O)NCC2CCN(C(=O)C3=CCCC3)CC2)c(F)c1 c1(N2CC(N(C(C=C(C)c3cccs3)=O)C)C2)cc(C)nc(CC2CC2)n1 CC(=O)n1cc(CN2CCSC(C(=O)Nc3nnc(C)o3)C2)c2cccnc12 n1(CCCC)nc(C(=O)NC2CC2CSc2ccccc2)c2ccccc2c1=O N1(C(CN2CCC(OC)C2)=O)CCOC(C)(CNC(c2ncc(C)cc2F)=O)C1 Cc1ccnc(C(=O)N(C2CCC(NC(=O)COCC3CCCC3)C2)C)n1 c1(C(=O)NC(C(=O)NCC(=C)CC)COC)cncc(F)c1C CC1(C)C(CNC(C23CCC(C2)C3)=O)CCN1C(c1cc(O)cc(F)c1)=O C(=O)(CC(C)(C)CC(=O)N1CCN(C(=O)CCCCCF)CC1CCO)OCC C1(C(=O)NCCCN(C(=O)CC2COCC(C)O2)C(C)C)C2(CC2)C12CC2 Cc1ncnc(O)c1C(=O)NCC1CC(C)(C)CN1C(c1ccoc1)=O C1(NC(=O)Nc2cc(C(C)C)no2)CC(=O)N(C(c2ccccc2)C)C1 N12CC(C)(C1)OCC2=O.C1(CC(=O)N(C2C(N(C)C)CC2)C)COCC1O N1(C(C(C)C)=O)CC(NC(=O)C(C)CC2CC2)C(C)C1 C1(NC(C2CNCCN2Cc2ccc(F)c(Cl)c2)=O)CCc2ccccc2C1 O=C(C1=C(Cl)CCCC1)NCC1(CNC(=O)C2CC2)CCCCC1 CCC(CC)CC(=O)NCCCOCCNC(=O)C(C)C(C)c1ccc(Cl)cc1 C(=O)(CC(F)(F)CC)N1C(C(=O)NCCOCC=C)CSCC1 N1(C(C2CN(C(N(C)C)=O)C2)=O)CC2CC1CCC2NC(c1ncc[nH]c1=O)=O CC(CCC(=O)N(C)CCN(C(=O)Cn1cnnc1O)C)N(C)C CC(CS(C)=O)C(=O)N(C)CCNC(C1(CCF)CCOCC1)=O Cc1c[nH]cc([N+](=O)[O-])c1=NC1CCN(C(c2cnn(CC(F)(F)F)c2)=O)C1 N1(C(C=CC)=O)CC=C(C(C)(C)C(=O)N2CC(CSC)C2)C1 CC12CCC(n3cc(CNC4(N)CC4)nn3)(CO1)C2 C(CN=c1cc(Cl)nc(CS(C)(=O)=O)[nH]1)(N(C(C1C(C)OCC1)=O)C)C1CC1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC(C1)C2NC(=O)C(C(C)C)n1cnnn1 c1(C(=O)OC)ccc(S(=O)(=O)NC(C)Cc2ccccc2Cl)c([N+](=O)[O-])c1 c1(OC)cc(C(=O)NC(C)CCNC(=O)C(C2CCCCC2)O)cc(N)c1O N1(C(c2scc(COC)c2)=O)CCC(NC(=O)CCCSC)C(F)(F)CC1 N1(C(CC2C(C)C2(F)F)=O)C2CCC1CC(CNC(c1nnc(S)n1C)=O)C2 C1(C(=O)NC2COCCN(C(C(C(CC)C)OC)=O)C2)CN2CCN1C(C)C2 C1(C(CCC)NC(=O)C(O)Cc2[nH]cnc2C)CCN(C(=O)COC(C)=O)CC1 C1(NC(C(CC)SC)=O)CCCC1(C)NC(=O)CCn1nc(C)nc1C c1(-c2nc(NCC(=O)Nc3nnc(CCCC)s3)sc2)ccccc1F n1(CC(N2CC=CC(NC(CCC(C)OC)=O)C2)=O)cc([N+](=O)[O-])nc1C C1(NC(CSCCC)=O)C(C)(C)CN(C(c2cn3ccccc3n2)=O)CC1(C)C C1(C(C)C)CC(C(=O)N(C2CN(C(=O)CC(O)Cc3ccccc3)C2)C)CCO1 N1(C(C=Cc2ccc(C)s2)=O)CC2CCN(C(C3CC3c3ccnn3C)=O)CC12 N1(C(c2cc(C)n(CCO)n2)=O)CCN(C(c2ccsc2)=O)CC1CS(C)(=O)=O C1(F)(C(=O)NCc2cnc(CNC(=O)OC(C)(C)C)s2)CCCOC1 Cc1nn(C)cc1CCC(=O)NCC1C2CN(C(C3CCCN3C(C)C)=O)CC12 N1(C(CC2(C=C)CC2)=O)CC(C)CN(C(c2ccc(C)nc2OC)=O)CC1C CCCCC(C)C(=O)N1CC(C(=O)N(CC(C)C)CCOC)C2(CC2)C1 N12CCC(CC1)N(C(N)=O)C1(CC1)C2=O.C1(CC2CC2)CCN(C2CC2)C1.CC=O CC1CN(C(=O)C(O)C(C)(C)C)CCCN1C(C1CCN(C2CC2)CC1)=O Cn1cc(NC(=O)CC2(CNC(c3cccc4c[nH]nc34)=O)CC2)c(O)nc1=O C(=O)(C(CCC(C)C)NC(=O)C(F)C1CCC1)NCc1cccc(CC)c1 C1(O)(CCNC(=O)COc2ccccc2)CCCN(C(c2cccc(=O)o2)=O)C1 N1(C(C2(CC)CCCC2)=O)CCCC(CCNC(=O)C(c2cnn(C)c2)OC)C1 C1(C)(CN(C2(C3CCCO3)CCC2)C(C)=O)COCCN(C(C2CCOCC2)=O)C1 C1(CNC(C=CSC)=O)CCCC2(CN(C(c3n[nH]c4c(C)cccc34)=O)C2)O1 N1(C(CC(CC)C)=O)CCC2(CCC2NC(c2ccc3n[nH]cc3c2Cl)=O)CC1 c1(C(N2C3C(NC(CCCc4c(C)ccs4)=O)C(C3)C2)=O)cc(C)c(N)cn1 CC1(CNC(c2cccc(C3(O)COC3)c2)=O)CCCN1C(=O)Cc1ccsc1 c1(NC(C2N(C(c3c(CC)ncs3)=O)CCC2O)=O)ccc(Br)cc1I c1(C(=O)NCC(CNC(c2nc(C)oc2)=O)(C)C)cc(S(=O)(=O)N(C)C)c[nH]1 N1(C(Cc2c(C)cccc2)=O)CCCCC(NC(c2c(O)cccc2Cl)=O)C1 c1(C(=O)NC2CC(CC)NC2)cc(-c2cccc(F)c2)n(C)n1 CCC(C)(CC)C(=O)N(C)CC1CCCN1C(c1ccc(O)c(C(C)C)c1)=O N1(C(c2c(CC)scc2)=O)CCCC2(NC(c3cn(C4CC4)nn3)=O)CC2C1 C1(C)(C(=O)NC(CCC)CO)C=CCN1C(c1cccnc1C)=O c1(CNC(=O)C=CC2CC2)ccc2c(c1)CCC2NC(=O)C1CCc2c[nH]nc21 c1(OC)ccccc1-c1ncsc1C(=O)Nc1nc(-c2ccoc2)nn1C C1CCCCCN1C(C1(N(C)C)CCC1)=O.C1(CC(=O)OC)(N(C)C)COC1 N1(C(CCC(C)OC)=O)CCC(C)(C)C(C(=O)NC(C)(CO)CO)C1 c1(C(=O)NCC(N2CC(COC)C2(C)C)=O)ncnc(O)c1F c1(C(=O)NC)cccc(C(N2CC=CC(NC(=O)C3=COCC3)C2)=O)c1 C1(CC(N2CC(C)C(NC(C3(O)CCOC3)=O)C2)=O)CCC2(CC1)CC2 N1(C(C(CCC)C)=O)CCC(CNC(C2CC2C(F)(F)F)=O)C12CCC2 N1(CCNC(C)=O)CCC2(CN(C(=O)Cc3ccnn3C)CC(C)O2)C1 CC(C)C(F)C(=O)N1CCOCC1CC(=O)NCCCC(C)(F)F Cc1cc(Br)cc2cc(CN3CCC(C)(C(=O)O)C3C)oc12 C1(C(=O)OC2CCN(C(=O)OC(C)(C)C)CC2)(OC)CC2(CN(C(C)=O)C2)C1 Cc1ncn(C)c(=O)c1C(=O)NCCC(C)CCNC(c1cc(O)cs1)=O N1(C(c2c(C)nco2)=O)CCC(O)(CCNC(=O)CCC2CCCN(C)C2)C1 C1(CN(C(COCC(=C)C)=O)C)CCCN(C(=O)COC2CCN(C)CC2)C1 N1(C(C(CC)C#N)=O)CC2CCN(C(C34CC(C(F)F)(CO3)C4)=O)CCC2C1 c1(-c2scc(CC(=O)NC(C3CN(C(C=CSC)=O)C3)C)n2)ccc(F)c(F)c1 C1(CNC(C(F)OC)=O)CCC2CN(C(=O)Cc3cnn(C)n3)CCC2C1 n1(CC(=O)N(C2CCN(C(=O)Cc3c[nH]nc3C)C2)CCC)cc(F)ccc1=O N1(C(c2[nH]c(C)cc2C)C(=O)NCc2ccc(OC)cc2)CCN(C)C(=O)C1 C1(C(N2CCN(S(C)(=O)=O)CC2)=O)CN(C(=O)Nc2ccncc2)CC(F)(F)C1 c1(N(C)C)ncccc1CNC(N1CCCC1c1ccc(Cl)cc1)=O CC(C)CC(Cc1ccccc1)C(=O)NCCCC(c1nnnn1C)NC1CC1 c1(C(N2C(CCNC(=O)CCc3cccc(F)c3)CCC2)=O)ccnc(CO)c1 C12(C(N3CC(CNC(c4ccc(-c5ccc(C)s5)s4)=O)C3)=O)CC3CC1C2C3 C1(NC(c2cnn(C)c2N)=O)CC2(C1)CN(C(C1CCC1C(C)(C)C)=O)C2 C1(O)(CC(=O)N(CC(CC)NC(=O)CSCCCN(C)C)C)CCCN(C)C1 CCCCC(C(=O)NC1CCCC(O)C1)NC(=O)COCCC1CC1 C1(C(N(C2CC(NC(C3(CO)COC3)=O)C2)C)=O)CN(S(=O)(=O)N(C)C)CCO1 C1(CNC(c2cncc(C(F)F)c2)=O)C2CN(C(=O)COC3CCCOC3)CC12 C(=O)(CC(C)(C)CC)Nc1ccc(CC)nc1.C12CCOCC1Cc1cn2nn1 N1(C(c2c(C)nc[nH]2)=O)CC(C)CCC1CNC(C1(C2(O)CCC2)CC1)=O CCCC(C)(C)C(=O)NCC1CN(C(C2C3CCC23)=O)CC1C C1(NC(CN2C(=O)C(F)(F)C23CCC3)=O)CCCC1SC.C(c1ccco1)=CC CCCC(F)C(=O)NCC(F)CC(=O)N(C(C)CO)C C(C)(CNC(C1CCOC1C(C)C)=O)(CC(C)C)NC(c1c(CC)csc1)=O C(CCNC(c1cccc(=O)o1)=O)(C(=O)NCC1COCCO1)OC c1(C(=O)NCC(CNC(c2ccc(CC)s2)=O)F)cc(C)nc2c1CCCC2 C=CCCC(C)(C)C(=O)NCc1nc(C(=O)NC(CN2CCCC2)CC)co1 C(=O)(C(F)C(=O)NCCCC1CCCCN1C(c1c[nH]c(Br)c1)=O)OCC C(C(=O)N)(C(C)CC(C)(C)C)N(CC(=O)C(C)=O)C.C(C)(C(=O)OC)CN c1(C(N(CCNC(C(COC)O)=O)C(C)C)=O)cnn(-c2ccc(F)cc2)c1C c1(C(N2CCN(C(c3cc(C)c(C)[nH]3)=O)C(C)C2)=O)nn2cccnc2c1Cl c1(C(C(=O)NC2(CN(C)C(C3CC34CC4)=O)CC2)C)ccc(Cl)c(Cl)c1 c1(N2CCCC(CCNC(c3cc(F)cnc3O)=O)CC2)ncnc2c1COC2 N(C1CCCn2ccnc21)C(C(CC=C)CNC(=O)C(C(C)C)NC(C)=O)=O N1(CCC(N2CCC(C(=O)NCCCO)CC2)=O)CCCS1(=O)=O c1(C(=O)NCC(CC)(CC)NC(=O)CC2CC2(Cl)Cl)ccc(NC)c(F)c1 CC(C(=O)NC(CC1CC1)C(=O)N(CC(C)(C)C)C)S(C)(=O)=O Cc1c(C(=O)NC(CNC(=O)CCC2CCOC2)C2CC2)ccc(Br)c1F C(C(=O)N1CC(NC(=O)CCCN(C)C(=O)OC)C1)(C(C)C)OC c1(CCNC(C(CSCC)NC(c2cnccn2)=O)=O)ccc(F)cc1 CCCCC(C(=O)NCC1(CNC(=O)C(n2cc(C)cn2)C)CCC1)C(C)C c1(C(N2CC(C=C)C(NC(=O)C(C)(C)C(F)F)C2)=O)ccc(S(N)(=O)=O)c(C)c1 c1(NC(C2C(NCc3c(OC)ccc(Br)c3)C2)=O)ccc2c(c1)COC2=O c1(OC)ccc(C=CC(=O)NCCOCCNC(C2C3CC4C(C3)C24)=O)cc1 c1(N2CC(CO)CC(CC)C2)nc2cccnc2c(=NC2CC(=O)N(C)C2)[nH]1 c1(C(=O)NCCN(C(=O)C2=CC(O)CCC2)CCC)cc(Cl)c(Cl)c(Cl)c1 N1(C(C=COCC)=O)CCN(C(C2CN(C3(C(F)F)CCOCC3)C2)=O)CC1 CC1(C)CC(N=c2nc(N3CC=CCC3)c3cc(F)ccc3[nH]2)CCS1(=O)=O c1(C(CO)NC(=O)NC(C)C(C)F)ccccc1Cl N1(C(CC2(COC)CC2)=O)CCC2(CC1)CN(C(c1sc(COC)nc1C)=O)C2 C(CC(=O)NCC(C)C(C)(F)F)(C(F)(F)F)NC(c1c(OC)ccnc1)=O c1(CNC(C2CC(NC(Cc3cccc(OCC)n3)=O)C2)=O)ccc(F)c(C)c1 c1(N2C(C(N(C3CCCC4CC34)C(C)=O)=O)CCC2)ncc([N+](=O)[O-])c(C)n1 C=CC(C)(O)CC(=O)NCCC1(OC)CN(C(=O)CC2CC3CCC2C3)C1 C1(C(N(C(C)CNC(=O)Cc2ccc(C(N)=O)cc2)C)=O)CC(C2CC2)=NO1 c1(CCC)ccc(S(=O)(=O)N2CC3(CC3C(=O)Nc3cccc(O)c3C)C2)cc1 C(CCC(=O)NC(CCO)C(F)(F)F)(C(C)C)NC(c1cc(SC)oc1)=O C12(NC(CS(C)(=O)=O)=O)CCN(C(=O)Cc3cnccn3)CC1C2 C1(C(=O)NC2CN(C(C(N3CCNC3=O)C)=O)C2)CCc2nc[nH]c2C1 N1(C(C(C)=C2CCC2)=O)CC2(C1)CN(C(=O)CC1CSC1)CC2CO N1(c2n(CC(C)C)c(-c3oc(O)nc3Br)nn2)CCC(O)C(F)C1 N1(C(c2cc(C)nc(O)c2)=O)CCN(C(c2oc(CO)nc2C)=O)C2CCCC12 c1(C(N2C3CC(NC(Cc4n(C)ncc4)=O)C(C3)C2)=O)cnn2cccc(Cl)c12 c1(-c2cn(CCN(C(=O)CN(c3ccncc3)C)C)nn2)cc(F)cc(F)c1 N1(C(CCN(C(=O)C(C2CC2)OC)CC)=O)CCC(O)CC1 C1(CCNC(c2ccsc2)=O)COCCN1C(C1CCOC1C1CC1)=O C(=O)(C(C)(C)C(C)(C)C)NCC(C(C)C)NC(c1cc(F)cnc1O)=O Cc1cc(C(=O)NC(C(=O)NCCC(F)F)C2CCCO2)oc1C Cc1cc(CNC2(C)CCC(C(N3CCC(O)C(F)C3)=O)C2)cc(C)n1 CN(C)S(=N)(=O)N1CCCC1C(=O)NCC1C2CN(C(=O)Cc3nc[nH]n3)CC12 C1(C(N2C(CNC(C(C)SC(C)C)=O)CC(F)C2)=O)CC2(C1)CC(F)C2 c1(C(N2CCOCC(CNCCCC3CC4(CCC4)C3)C2)=O)cnc(O)cc1O c1(C(N2C3CCCC2COC3)=O)ccc(=NCc2cccc([N+](=O)[O-])c2)[nH]c1 c1(C(C2CCN(C(c3cnc[nH]3)C)CC2)=O)cccc2cnccc12 c1(OC)ccccc1OCCC(=O)NCC=CCNC(=O)CCC1CC1C1CC1 C(CCN=c1nccc[nH]1)N(C(=O)CC1CCCC(O)C1)C COn1cnc(C)c1C(=O)NCC1CN(C(=O)C(C2CCOCC2)C)CCN1C N1(C(C2CCCN2C(c2c[nH]c(=S)cn2)=O)=O)CCC2(CCOC2=O)C1 C1(C(N(C)CC2CC(F)CN2C(=O)CCc2c[nH]c(=N)[nH]2)=O)CCCC2(CC2)C1 c1(CC(=O)N(C(c2ccccc2)CSC)CC)ccc2nc(Cl)sc2c1 C1CCN=C2NC(=NC=C2Br)O1.C#CCCC(=O)NCCOCCN C1(NC(C2C(C)(C)C2)=O)CC2(NC(=O)C=C3CCSCC3)COC1C2 CC1CN(C(C(=O)NC2COC2)C(C2CC2)C2CC2)Cc2c[nH]nc21 c1(C(=O)NCC2(NC(C3CC(CC)OCC3)=O)CC2)c2c(c[nH]c1=N)CCC2 c1(NC(N2CCC(O)(C(F)(F)F)C2)=O)ccc(C(O)C(F)F)cc1 C1(CC)(NC(=O)C(C)SC)CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1 N1(C(C=Cc2ccc(C)o2)=O)CCC(C)N(C(=O)CCc2ccn(C)n2)CC1 Cc1cc(OCC(=O)NC2C3CN(C(C4CNC(=O)CC4C)=O)CC23)ccc1Cl C1(C(=O)NCC2OCCN(C(C)=O)C2)CC2CC(CN2)O1 C(=O)(C(O)C1=CCCCC1)N1CC(C)(CNC(C2(OC)CCCC2)=O)CC1(C)C c1(C(CC(=O)NCCN(C(=O)Cc2ccns2)C)C)c[nH]c2ccccc12 N1(C(c2cc(C)sn2)=O)CCC(C(C)(C)CNC(C2(O)CCCC2)=O)CC1 Cc1cc(O)ncc1C(N1C2CC1CN(C(=O)Cn1cnc(=N)[nH]1)C2)=O C1(C(=O)NC(C)C(=O)N(C)C)CC2(CC(NC(=O)C(C)C3(O)CCC3)C2)C1 c1(NC(C2CC(C(N)=O)C2)=O)ccccc1CNCc1ccncc1 CCC(CC(=O)NC1CN(C(c2ns[nH]c2=O)=O)CC1N=[N+]=[N-])C(F)F C1(NC(=O)C(c2ccccc2)O)CCN(C(C2CC=CCO2)=O)CC1F c1(CC(=O)NC2CCN(C(=O)Cc3cscn3)CC2F)cc(Cl)c2c(c1)OCO2 N1(C(C(C(C)C)OCC)=O)CC2(CCNC(=O)Cn3nc(C)cc3C)CCC1C2 Cc1cn(C)nc1C(=O)NCC1CC1NC(=O)C(C)CN(C)C C1(S(N)(=O)=O)(C(N(CCC)CCNC(=O)CCOc2ccccc2O)=O)CCC1 C1(C(=O)NC2(c3ccc(F)cc3)COC2)CC2CC2N1C(=O)Cc1cc(Br)cs1 c1(C(N2CC(O)CC(NC(COCCC#C)=O)C2)=O)cnc2ccccc2n1 Cn1nnnc1C(C)(CCC1CCCC1)NCCCOc1nncs1 C(=O)(C1c2c[nH]nc2CN1C(=O)Nc1nc(-c2ccc(C)cc2)c(C)s1)NC CC(C)(C)C(CC(=O)N1CCC(CCCNC(=O)Cc2cc[nH]n2)CC1)C(F)F c1(C(N(CCNC(C(C)OCC#C)=O)CC2CC2)=O)cncc2nc(C)[nH]c12 N1(C(CCSC)=O)CCCC(c2nc(-c3ccncc3)nn2-c2nccn2C)C1 Fc1ccc(CN2CCN(Cc3ccsc3)CC2)cc1Cl N1(C(c2cc(C(C)=O)sc2)=O)CCC(NC(=O)CC2CCN(C)C2)C(F)C1 N1(C(c2ccn(CC)n2)=O)CC(OC)CC(NC(c2cnn(CC(C)C)c2)=O)C1 c1(CCC(=O)NC(CNC(c2cn(C)nc2)=O)C2CCC2)ccc(N(C)C)cc1 C(=O)(CC(F)(F)F)N(CC(C)N(C(=O)C(C1CCOCC1)O)C)C C=C=CCC(=O)NCCN(CCCN(C)C)C(c1cc(-c2ccn(C)n2)on1)=O C#CCC(CC#C)C(=O)NCC1CC(CNC(c2cc(N)cc(F)c2)=O)C1 c1(CCCCC=C=C)cccc(F)c1.C1(c2nnnn2C(C)(C)C)CCCN1 c1(C(=O)NC(c2ccc(Cl)cc2)C)ccc(CNC(=O)C(N)=O)cn1 CN1Cc2ccc(C(N3CCOCC(CNC(=O)Cc4cccs4)C3)=O)cc2C1 CC(CCNC(C1CC1c1ccncc1)=O)CCNC(C1CC(F)(CO)C1)=O c1(OC)cccc2c1CC(C(N1CCC(N3CCCNC3=O)CC1)=O)N2 N1(C(C(=O)N(C)CC2CC(F)C(C#N)C2)=O)CCC2(CCCO2)CC1 n1(C(C(=O)NC(CNC(C=C(CC)C2CC2)=O)CC)C)ccnc1C CC(CS(C)(=O)=O)C(=O)NCC1CCN(C(=O)CCCCCF)C1 C1(CC(=O)NCCSCC#C)CCCC1NC(c1sccc1COC)=O N1(C(C(C)SCC)=O)CCN(C(c2cn(CC)nn2)=O)C2CCCC12 Nc1c(C(=O)NCC2(NC(=O)COC3CCOC3)CCC2)cccc1F c1(CC2CCC(C(=O)NC(=O)NCC3OCCN(C)C3)OC2)ccc([N+](=O)[O-])cc1 C(=O)(C1=CCCOC1)NC1C(C)CN(C(=O)COCCF)C1 C=CCCC(C)(C)C(=O)N(C)CCN(CC(=O)O)C CC(C)CC(C)(C)C(=O)NC(C)C(C)NC(C1(CCN(C)C)CC1)=O C(=O)(CCC(=O)Nc1nccs1)NCC(C1CCC1)NC(c1ccc(CC)s1)=O CS(=O)(=O)CCC(=O)N1CC2CCC2(CNC(C2(F)CCC=CCC2)=O)C1 N1(C(C)=O)CSCC1CNC1(CNC(=O)Cc2ncc(C)s2)CC1 N1(C(C2(C=C)CCC2)=O)CC(N(C)C(c2cc(C)cc(F)c2)=O)C(C)(C)C1 CC1(C)CC(CNC(=O)Cc2cccs2)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 C1(F)(CNC(COC(C)=O)=O)CCN(C(c2cnncc2C)=O)CC1 C1(CC#C)(C(=O)N(C2CSC2)C)CCN(C(c2ccncc2Cl)=O)C1 N1(CCC(=O)NCC(C2N(C(C=CC=CC)=O)CCC2)(C)C)CCN(C)CC1 c1(C(=O)NCc2ccn(CC(C)C)n2)ncc(C(F)(F)F)cc1Cl N1(C(CCOCC#C)=O)CCCC(CCNC(=O)C2=CCCO2)C1 CCC(CC)(CC)C(=O)NCC(C(=O)NC(c1csnn1)C)N(C)C C1(C(N(CCCO)C)=O)CCCN1C(C1CC1C(=O)C1CC1)=O Cc1cccc(CCNC(=O)C(C)NC(c2c(C)nsc2C)=O)c1 CCC(F)(F)CC(=O)NCCCCN(CCCNC(=O)Cn1ccc(C)n1)C c1(CC(=O)NC2CC2C(=O)Nc2nc(Cl)ccc2I)c(F)cccc1F CC(C)CC(C)CC(=O)NC(C)(C)CN1CCN(C(c2cnc(Cl)s2)=O)CC1 O(NC(=O)CN(C)CCOCCNC(=O)C(C)CN(C)C)CC(=C)C C1(C(=O)NCCC(C)NC(c2c[nH]c(C#N)c2)=O)CCCC1P(C)(C)=O C1(NC(c2cncnc2C2CC2)=O)C2CN(C(c3csc(C(F)(F)F)n3)=O)CC12 c1(NC(C2(F)CCN(C3CCCC3)C2)=O)cc(NCCN2CCC(O)CC2)ncn1 Cc1ncc2n1CCN(C(=O)CCNC(C1CC(=O)CCO1)=O)C2 C1(C(N2CCCC(NC(=O)Cn3cnnn3)CC2)=O)CCc2nc(O)[nH]c2C1 CCCC(F)C(=O)N1CCCC1CNC(C1(OCC)CCCCC1)=O N1(C(C(C=C)(C)CC)=O)CCC2C(C1)NC(=O)CN2C(=O)CCc1cccs1 N1(C(C(CC)COC)=O)CCC(CNC(=O)CCCC2CCC2)C(F)(F)C1 CC(C)(CCSc1c(F)cccc1Br)CC(=O)NC(C)(C)C N1(C(CC(C=C)(C)O)=O)CC(CNC(c2ccoc2C2CC2)=O)OC2COCC12 c1(N2CC(CCNC(C(CC)C)=O)C2)ncnc2ccc(OC(C)C)cc12 C1(NC(c2c(OC)nccc2)=O)CC2CCC1N2C(=O)Cc1csc(C)n1 N1(C(CNC(C)=O)=O)CC2CC(NC(c3cc(C(F)(F)F)ccc3Cl)=O)C1C2 C(CCN=c1ccnc(NCCNCCCN2CCOCC2)[nH]1)OC C1(CNC(CCOCCN(C)C)=O)CCC(C)(C)CN1C(C1CCNC1=O)=O Cc1cc(Br)cc(C(=O)NC(CNC(=O)CC(C)c2cnn(C)c2)CO)c1N c1(SCC(=O)N(C2CN(C(=O)CC3CCCCO3)CC2F)C)cccc(F)c1 N1(C(C(C2CC2)OCC)=O)CCC2(C1)CN(C(=O)C#CC1(C)COC1)CCO2 C1(C(N(C(C(=O)N(CCF)CC)C)CC)=O)CC(C)CC(=O)N1 Cc1nc2ccccc2c(C)c1C(=O)OCC(C12CC(c3ccccc3)(C1)C2)=O c1(C(=O)NCC(CC(C)C)(C)NC(=O)COCCCF)occ2c1CCOC2 CC1CC(C(=O)NCC2=CCN(C(=O)COCC3CCOCC3)CC2)CC(C)C1 C1(O)(C(=O)NCCC2(CNC(CNS(N)(=O)=O)=O)CC2)CCSCC1 C1(NC(C(CCF)NC(COCCCCC)=O)=O)CCC(C2CC2)C1 c1(CC)conc1CC(=O)NC1(CNC(=O)C(C)Cc2cnco2)CCOC1 c1(NC(C2C(C(=O)OC)C2)=O)cc(=NC(=O)c2cc3c(C)cccc3[nH]2)[nH][nH]1 N1(C(CCCSC)=O)CCN(C(c2c(C)nc(C3CC3)nc2O)=O)CC1C#N CN1CCC(O)(NCC2(F)CCN(C(=O)OC(C)(C)C)C2)C1 CC(C)(C)C(CO)C(=O)NC1CCCC1NC(c1c(Br)cnn1C1CC1)=O c1(NC(N(C(C2CCCO2)CC2CCCC2)C)=O)c(CCC(N)=O)c[nH]c1C C1(NC(CCOCCCOC)=O)CCN(C(c2csnc2OC)=O)C1C(C)C CC12CC(CCNc3nccc(N4CCC(C)(C(F)(F)F)C4)n3)(CO1)C2 c1(OC)cc(C(=O)NCC2CCCC2NC(c2cc(C)ns2)=O)sn1 C1(NC(C2N(C(C)=O)CCC2)=O)CC(F)CN(C(c2cnn(C(C)C)n2)=O)C1 C1(C(=O)NC(CC#C)C(=O)NCCC)CC2C=CC1CC2.C1CCCC1N(C)C C=C1CCC(C(=O)NC(C(=O)NCc2cccc(Cl)c2)C2CC2)CC1 c1(CC)ncncc1C(N1CC2CC2(CNC(=O)Cc2csnn2)C1)=O C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(C(CC)CC(F)F)=O)C(O)C(O)C1 C(=O)(C(S(N)(=O)=O)c1ccccc1)NCCCCN(C(c1sc(C)c(O)n1)=O)C CCC(CC)CCCNC(C1(COC)C=CCN1C(C1CC2C=CC1O2)=O)=O N1(C(CC2(N(C)C)CC2)=O)CCCC1C=CC(N1CCOCC1C(C)(C)C)=O c1(OC)cc(OC)c(C(=O)NC2CCC(NC(C3CNC(=O)C3)=O)CC2)c(N)c1 C1(C(=O)NC(CC)CNC(=O)Cc2cnn(C(C)C)c2)CN2CCCCC2CO1 c1(C(=O)NCC(CN(C(C2=C(C)OCC2)=O)C)(C)C)cc2c(C)c(Cl)ccc2[nH]1 c1(CN(C)C(=O)NC2CCN(c3ccncn3)CC2)ccc(F)cc1Br C1(C(=O)NC(CC(C)NC(C(CC)=CCCC)=O)C)CCCOC1C c1(C(N2C(CNC(=O)CC3CCC3)(CSC)CCC2)=O)ccc(OC)c(Cl)c1F c1(CC)nc(=N)[nH]cc1C(N1CC(NC(c2ccncc2F)=O)C2CC12)=O C(C)(CC(=O)N(NC(=O)OC(C)(C)C)C(C)C)c1c(C)ncs1 c1(C2(CNC(c3cnc(C4(C)CC4)[nH]3)=O)CCCO2)ccc(Br)cc1 Cc1cc(C(=O)NCC2CCN2C(c2ccnc(N(C)C)c2)=O)ncc1Cl Cc1ccc(C(CN2CCCCC2)Nc2ccc(-n3cnnn3)cc2)cc1 Cc1cc(CC(N2CC(N(C)C(c3cnc(N(C)C)o3)=O)C(F)C2)=O)ccn1 O(S(=O)(=O)c1ccccc1F)C1C(c2nc3cccc(CCC(=O)OC)c3s2)C1 c1(OC)cc(CN=c2[nH]c(CN3CCC(CO)C(O)C3)cs2)cc(O)c1O C1(NC(c2c(C(=O)OC)scc2)=O)CCCC2CN(C(c3ccn(C)n3)=O)CC12 N1(C(CC2C(C)CCO2)=O)CCC(CO)(CNC(c2csc([N+](=O)[O-])c2)=O)CC1 c1(NC(C2CC(CC(=O)NCC3(OCCO)CCC3)C2)=O)ccc(Br)nc1 C(=O)(C(C)(C)C1CCCCC1)N(CCNC(=O)CC1CCCO1)CC c1(C(N(CCOC)CCNC(=O)C2=NOC(C)C2)=O)cc2c(s1)CCCCC2 c1(C(=O)NCCN(C(C(CCSCC)NC(N)=O)=O)C)ccc(S(N)(=O)=O)o1 CC1(C)CN(Cc2nn[nH]c2Cl)CC1NC(C1CCN(c2nncs2)CC1)=O C1(NC(CN(CCC#C)C)=O)CC2(CCCN(C(=O)CCCc3ncco3)C2)C1 c1(C(=O)NC2CC(C)(NC(C(CCCCC)O)=O)C2)cccc2nc(C)[nH]c12 c1(OC)ccc(C(=O)C(=O)NCc2ccc(Cl)cc2)cc1F C=CCCCCC(=O)N1C2CCC1C(CNC(=O)CS(=O)(=O)N1CCCCC1)C2 c1(C(=O)NC(CNC(C2CS(=O)(=O)C2)=O)CO)c(C(F)(F)F)cccc1Cl CC1(C)CCCN(C(C2(C#N)CCC2)=O)C1CNC(c1cccnc1O)=O N(C(=NCCCN(C)C(C)C)NCc1c(F)cccc1Br)C(CC)C c1(C(N2CCC(O)(CN(C(=O)C=C3CCC3)C)C2)=O)cnn2ccc(O)nc12 C1(CC)C(NC(=O)COC2CCOC2)CCCN1C(=O)CCCCOC CC1(CNC(C2(CC(F)(F)F)CC2)=O)CCN(C(=O)C=CC(F)(F)F)C1 CC1CN(C(=O)Cc2cc[nH]c2)CC(C(=O)NCCN(CCCF)C)O1 Cc1ccc(C=CC(=O)NC2(C3CCCCN3C(C3CCC3(C)C)=O)CC2)o1 Cc1cc(O)c(F)cc1NC(C1CCN(C(c2ccc3cc[nH]c3c2)=O)O1)=O C(=O)(C(C#N)C(C)C)NC(C(=O)N(C1CC(OCC)C1)C)CCF N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(C)(C)C(CNC(C2CCN(C)CC2)=O)C1 c1(C(N2C(CCC(=O)N(CC(N)=O)C)CCC2)=O)ccnc(Br)c1F CCC(CC)C(F)C(=O)NCc1c[nH]nc1C(=O)NC1CCC([N+](=O)[O-])CC1 N#Cc1cc(CNC(=O)CC2CC3(C2)CN(Cc2cc(C#N)cs2)C3)ccc1F N1(C(C2C(=C)C2C(=O)OC)=O)CCC(CCNc2ncc(CC)s2)C1 Cc1cc(Br)c(NC(C2CN(Cc3ccc(O)c(F)c3F)CCC2O)=O)nc1C C(C(C)(C)C(=O)N(C1CCOC1)C)NC(C(CC)SC)=O c1(C(=O)NCC(C2CC2)NC(C=Cc2c(C)cccc2)=O)ncc(C#N)cc1Cl C(=O)(CC1OC(=O)c2ccccc21)N(CCC(C)NC(c1scnc1Cl)=O)C N1(C(c2cn[nH]c2)=O)CCC2(CCCC2NC(=O)C(O)(C2CC2)C2CC2)CC1 CCCCCCC(C)C(=O)NCCC1(CNC(=O)CC2CC(=O)NC2=O)CC1 N1(C(c2c(CC)nns2)=O)CCCN(C(C2CC3CCC(C2)C3=O)=O)CC1C c1(C(=O)NCCCC(CCC)NC(c2ccco2)=O)cnn2ccc(OC)cc12 CCC(C)CCCC(=O)NCCCN(C(=O)C(C(C)O)N(C)C)CC c1(C(N2CCCC2CSC2CC2)C(=O)NCCCOC)ccc(C#N)c(C)c1 c1(CC(C)C)ccccc1C(=O)NC(C12CCC(CC1)C2)C c1(N2CCC(NC(CC(CCC)C)=O)C(F)C2)ccc2c(n1)CCC2=O C#Cc1ccc(F)cc1C(=O)NC1(C)CC(NC(=O)CCc2cccn2C)C1 c1(NC(c2c[nH]n3c2nc(=O)c2ccccc32)=O)nc2ccc(Cl)c(Cl)c2s1 c1(CC(C)(CSC)NC(=O)CS)ccc(C(F)(F)F)cc1.CCC(O)C=O c1(C(=O)NC(CO)C2CCC2)ccc(F)c(O)c1 N1(C2CCCN(C(C3C(C(N)=O)C3)=O)C2)CCN(C(=O)C(O)C2CCC2)CC1=O c1(N2CCC(CC=C)(NC(=O)C(c3ccccc3Cl)C)C2)ccncc1[N+](=O)[O-] Cc1nn(-c2ccc(F)cc2)cc1C(=O)NCCNC(c1cnc(C2CC2)s1)=O CCCC(O)C(=O)NCC(c1ccccc1)CNC(=O)C=CC(C)(C)SC CC1(C)CC(CNC(C2NC(=O)OC2(C)C)=O)N(C(C2C(C)(C)C2(C)C)=O)C1 c1(CC(=O)NC2(C)CCN(C(c3ccccc3)=O)C2)c(F)cccc1Cl CC(C)CC(C(=O)NCC1CC(C)C1)ONC(c1cc(Cl)cn1C)=O N1(C(C)C)CCOC(C(=O)NC(C2CCN(C(=O)COc3ccsc3)CC2)C)C1 c1(OC)ccc(Br)c(CC(=O)NC2CCCC2NC(C2CCOC2)=O)c1 C1(C=C)(C(=O)NCCC2(OC)CN(c3nc(C)ncc3F)C2)CCOCC1 c1(OC)ccc(CO)cc1C(=O)NCCC1CCN(C(=O)Cc2ccsc2C)C1 C1(O)(C(C)NC(C(=O)NCC)=O)CCCN(C(C2(CC)CCCC2)=O)C1 C12(C(N3C(CNC(C4N(CCC)CCC4)=O)CC3)=O)CC3CC(C1)CC(O)(C3)C2 CC1CC(C(=O)NC2(C)CC(C(=O)NCCc3cccnc3F)C2)CCS1 N1(C(Cn2cc(C)c(O)nc2=O)=O)CC2CN(C(=O)CC3CC34CC4)CCC12 c1(C(=O)NC2C(CCC)CN(C(c3cc(CC)oc3C)=O)C2)ccc(O)c(F)c1 c1(NC(=O)CC2CCCCCN2C(C2CC=CCO2)=O)cccc2[nH]ccc12 C1(NC(c2cccc(Br)c2F)=O)CN(C(C2CC23CCC3)=O)CC2CC12 N1(C(CCCCN(C)C)=O)CCN(C(=O)C(=O)C2CCCC2)CC1CO C1(OCCNC(CCCSC)=O)CCN(C(=O)CCN2CCOCC2)CC1.C=O C1(N(C(=O)Cc2csc(S)n2)C)CCCN(C(=O)CN2CSCC2=O)CC1 c1(C(=O)NC2(CC(=O)N(C(C)C3CC3)CC)CCC2)cc2ccccc2[nH]1 N1(C(=O)CC2COCCN2C(C2CC3C=CC2C3)=O)CCN2CCOCC2C1 CCC(C(O)C(C)C)NC(C1(CC)CCN(C(=O)CCCC(C)=O)CC1)=O C=CCC(C(=O)N1CCC(CF)(NC(C2CC2C2CCCO2)=O)C1)c1ccccc1 C1(C(=O)OC)CC(OC)CN(C(=O)NCc2nc[nH]c2C2CC2)C1 N1(C(CC)=O)CC2CC(C(=O)NCCS(C)(=N)=O)(C2)C1 O(C=C(C#N)C(=O)NC1C2CCC(C2)C1NC(=O)COC)CC C#CC1CCCC(C(=O)NC2(C3CCCN3C(c3ccc(F)cc3C)=O)CC2)C1 C(=O)(C(F)CC(C)(C)C)NC1CC=C(C(=O)NCC(c2ncn(C)c2)O)C1 Cc1ccn2cnc(C(=O)N(C)CCN(C)C(c3cncnc3C3CC3)=O)c2c1 C(=O)(CCCCCNC(c1cc(CO)n(C)n1)=O)NCC(CC(C)C)N(C)C CC(C)CCC(C(=O)NCC(F)C(C)(C)O)NC(C1(C)CC(C)C1)=O C1(C(=O)NC(C(=O)NCC2C(=C)C2)CCOCCO)CC2(C1)CC(C)C2 c1(C(=O)NC2CC(CCNC(CC(C=C)(C)C)=O)C2)c[nH]c2cc(Cl)ccc12 C(=O)(CCS(C)(=O)=O)N(CCNC(c1nc(COCC)sc1)=O)C C1(C(=O)NCC(C)(CO)NC(c2c(OC)nsc2)=O)CC(C)OC(C)C1 C1(CNC(c2cccc(NC(C)=O)n2)=O)CC2(CO1)CN(C(c1cnoc1)=O)C2 CC1(C)C2CN(C(C3CN(Cc4cccc(C(C)(C)C)c4)CCS3)=O)CC12 Cc1cnc(C(=O)N(C2CCN(C(=O)COc3cccnc3Cl)C2)C)cn1 c1(C(N2C(CCNC(c3n(C)nnc3)=O)CCCC2)=O)ccc2c(c1)NCC2 c1(N(C)Cc2nnc3n2CCOC3)nc(=NCC2SCCS2)[nH]c2ccsc12 C1(N2N3C(CC(O)C3)C2=O)COCCC1(F)F.C(CCC)N(CC=C)CC=C.C=O N1(C(c2ncc(OC)cn2)=O)CC(N(C)C(C2NC(=O)OC2C)=O)C(C)(C)C1 N1(C(c2ccc(C)[nH]2)=O)CCCC12CCN(C(=O)C(F)CC1CC1)C2 C(C(C)(O)CC(=O)NC(CNC(=O)CN(c1ccc(Cl)nn1)C)C(C)C)OC N1(C(c2c(C#C)cn(C)n2)=O)CC2(C)CN(C(C3CC(CC)=NO3)=O)CC2(C)C1 C1(C(=O)NC2C(NC(CN(c3ccncc3)C)=O)CCCC2)CCCC12CCC2 Cc1nn2c(C(=O)N(CC(O)CNC(c3ccc(N)cc3C)=O)C)c(C)nc2s1 CCC(CNC(=O)C(CC1CCC1)NC(c1c[n+]([O-])c(C)cn1)=O)C(C)(F)F N1(C=O)CC(=O)N(C)C1C(C)C.C1(N2CCCC(C)C2)(CCC=C)CCNCC1 C1(CN(C(c2cnc(C(C)C)[nH]2)=O)C)CCCN(C(=O)C(=O)NCC(F)F)C1 N1(C(c2cc(C)no2)=O)CC2(CCC2)CC1C(=O)NC(c1cnn(C)c1)CO C1(N(C(CCCC#C)=O)C)CCN(C(=O)CCCC(C)C)CC12CC2 C1(NC(C(COC)CC(C)C)=O)CCN(C(c2n[nH]cc2Cl)=O)CCC1(F)F Cc1c(C(=O)NC(CNC(=O)C(C)(C)C2CCCO2)C2CCC2)cnn1CCO N1(C(CCCC(CC)CC)=O)CCC2(C=C(C(=O)NC(C)Cn3cnnc3)C2)C1 N1(C(Cc2c(C)ocn2)=O)CCOC(C(N2CCN(CCO)CC2C)=O)CC1 c1(C(=O)NCCC2N(C(CC(C)C(F)F)=O)CCSC2)cccc2nn[nH]c12 N1(C(c2ccnc3cc[nH]c23)=O)CCC2CN(C(C3CC3(F)Cl)=O)CC2CC1 C1(NC(C2CCN(C(=O)OC)CC2)=O)CN(C(=O)CCC(C)(C)OC)CC12CC2 c1(C(=O)NCC(CCCC)NC(=O)Cc2cccc(C)c2F)cccc(O)c1F Cc1ccc(Br)c(C(N2CC(CNC(c3nnn(C)c3N)=O)C(C)(C)C2)=O)c1 S(=O)(=O)(c1ccc(N2CCCCC2)nc1)N.CC1OCCC1C(N1CCCC1)=O C(c1ccc(O)cc1)=CC(N1C(CCNC(c2c(C)csc2)=O)CCCC1)=O c1(CC(=O)NC2C(NC(C3N(C)CCC3)=O)CCOC2)ccc2ncsc2c1 c1(OC)ncc(C)c(C(=O)NC(C)C(C)NC(=O)Cc2ccc(F)c(F)c2)c1Cl c1(C(=O)NC2CC3(C2)CC3C(=O)NCC2CCCC23CC3)occ2c1CCC2 c1(C(N2CCN(C(C(C=CC)O)=O)CC(O)C2)=O)ccc2nc(C)[nH]c2c1 C1(C(=O)NCC(NOC)=O)C(C)CCN1C(c1nonc1C)=O CC(C#N)CCC(=O)N1CCOC(C)(CNC(c2ncc[nH]c2=N)=O)C1 CCCCC(O)C(=O)N1C(CC(N2CCCCC2CCOC)=O)C2CCCC12 CN1C(=O)C(NC(=O)NC2OC3CCC2CC3)c2cc(Br)ccc21 C=CCC(CC)C(=O)NCCC(C(C)C)NC(C1(OC)CCOC1)=O c1(C(N(CC(C)NC(C=CC(C)(C)SC)=O)C)=O)cnn2c1CN(C)CC2 C1(N(C)Cc2ccc(C(=O)OC)[nH]2)Cc2ccccc2C1OC C1(CCNC(=O)C(F)CC2CC2)CCN(C(C2(Cl)CCC2)=O)CC1 C=CCCC(F)(F)C(=O)N1CC2CC1C2CNC(C12CC(CO1)C2)=O C(CC(O)C(=O)N(CCNC(C1CC12CC(O)C2)=O)CCc1ccccc1)SC C12(C)CCCN(C1)C2=O.C12(CN(CCN(C)C)C)CC(c3ccccc3)(C1)C2 C1(NC(CN(C(c2cnccc2C)C(=O)NC)CC(C)C)=O)CCS(=O)(=O)C1 C12(NC(C(C)(F)F)=O)CCN(C(c3ccc(OCC(F)(F)F)o3)=O)CC1C2 c1(CCBr)cc(F)c(F)c(F)c1.c12ccc(cc1)NC(=O)C(=O)N1CCCC21 O=C1Nc2ccc(C(=O)NC3COCC3NC(=O)CCOCC3CC3)cc2C1=O c1(C(N2CCC(O)(c3cn(CC(=O)OCC)nn3)C2)=O)cc(F)cc2c1CCC2 C(C)(CCC(C)(C)C)NC(CSCCNC(CCCCOC)=O)=O Cc1nc(CSC(CNC(=O)OC(C)(C)C)CO)c(C)c(O)n1 c1(C(c2ccccc2)NC(C2C(C)=C2)=O)nc(C)ccc1F C1(C(=O)NC)C2CN(C(=O)NC3CCN(C4CCCCC4)C3)CC12 C1(NC(CSCCC)=O)CC(C(=O)N(CC(C)C)CC2CC2)C1 C(CNC(=O)CN1CC2CC2C1)(C(=O)NC1CC2(CC2)C1)N(C)C(N)=O C1(c2ccccc2)(C(=O)NC2C(CNC(C(n3cc(Cl)cn3)C)=O)C2)CCCC1 C=CC(CC)CC(=O)N1CCC(N=[N+]=[N-])(C(=O)NC(C)CN(CCCC)C)C1 N1(C(CCCC#N)=O)CCCC(CC(=O)NCC2CC3(CCC3)C2)CC1 c1(C(=O)Nc2ncn(C)c2)csc(=NCc2c(I)ccnc2F)[nH]1 C(=O)(C(C)CC(C)CC)NCC1(OCC)CN(C(=O)C2=COCC2)C1 c1(C(=O)NC2CC(F)(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)ccc2cccnn12 c1(OC)cc(C#N)ccc1NC(=O)Cc1cc(F)c(C)cc1F C1(NC(C(c2c[nH]c3ccccc23)C)=O)CC2CCC1N(C(=O)CC1CC1)C2 c1(C(N2CCC(C(C)NC(Cc3cc(C)sc3)=O)C2)=O)cc([N+](=O)[O-])cnc1C c1(N2CCC(OCCOC)CC2)nc(=NCC2CCCC2OC)[nH]c2c1COC2 Cc1oc(Cl)nc1C(=O)N(CC(N1CCCC(C)C1)=O)CC(C)C N(C1CCOc2ccccc21)C(c1cccnn1)C(=O)NC1CCOC1 c1(C(=O)NCCCCCN(C(=O)CCCC(N)=O)C)ncc(C#N)cc1Cl Cc1ccc(-n2nnnc2C(C2CC2)Nc2nc(C)c(C)[nH]2)cc1 C1(NC(CC2C(C)CCC2)=O)CC2CC(C1)N(C(=O)CCS(=O)(=O)N(C)C)C2 C(=O)(C(C)S(=O)(=O)C1CCOCC1)N(CC(C)N(C(CCCCCOC)=O)C)C C(c1cncc(OC)c1)=CC(=O)NC(CNC(CNC(=O)OC)=O)(C)C1CC1 C1(NC(CC=CC(C)(C)C)=O)CC(F)CN(C(C2CC3C=CC2C3)=O)C1 c1(C(N2CCCC(CN(C(C(CC(=C)C)C)=O)C)C2)=O)cc2c(nn1)CCOC2 c1(CC(=O)NCCN(C(=O)C(c2cc(Br)co2)=O)C)cnn(C(C)(C)C)c1 N1(C(C2CCN(c3ccc(OC)cc3)C2)=O)CC2C=C(Br)C2C1 c1(OC)ccc(NC(=O)C(C2CCCCC2)NC(c2ccco2)=O)nc1 Cc1nc(S(=O)(=O)NC(C)C(c2ccc(Cl)cc2)C)c(-c2ccccc2)o1 C(=O)(C1CNC(=O)c2ccnn21)NC1CC(NC(c2c(OC)ccc(C)n2)=O)C1 c1(CC)c(C(=O)NC(CNC(=O)CCC2CC2C)CCOC)[nH]c(C)c1C(N)=O C1(CNC(NC(COC)C)=NCCc2cccs2)COc2ccccc2C1 Cc1c(C=CC(N2CCC(CNC(c3sccc3Br)=O)C2(C)C)=O)cnn1C C1(C)(C(=O)NC(CNC(C2(C(=O)OCC)CCC2)=O)CO)CC=CCC1 C(=O)(CS(=O)(=O)c1ccccc1C)N(CC(CNC(C(CC)(CC)CO)=O)C)C c1(C(N2C(CCNC(c3ccc(CO)o3)=O)CCCC2)=O)cc2sccc2s1 CC1=NOC(C)(C(=O)NCC2(C(N)=O)CN(C(C3(C(F)F)CCCO3)=O)C2)C1 C1(F)(CNC(C2(CCC)CC2)=O)CCCN(C(=O)C2=C(Cl)CCC2)C1 Cc1cccc(C(F)C(N2CCSCC2CCNC(=O)C=CBr)=O)c1 Cc1[nH]nc(C(C)C)c1C(N1CCC(N(C(=O)C(C)n2ccnn2)CCO)C1)=O OCCC(N=c1nc2sccc2c(N2CC3COCC3C2)[nH]1)C1CCC1 Nc1ccc(Br)cc1C(=O)NCC1CCCC(NC(=O)Cc2cccnc2)C1 c1(CNC(c2cnn(C3CC3)c2)=O)ncccc1O.C1CC(=O)N1 N1(C(CC(COC)C)=O)CCOCC(CNC(=O)C=C(C)c2ccco2)C1 N1(C(CC(C)(C)n2cc(-c3ccncc3F)nn2)=O)CC(F)(F)C(F)(F)C1.CCO C1(CNC(C2CCc3c[nH]nc3C2)=O)CN(C(=O)C2=CCCC2)CCC12CCC2 N(C(=NCCC)NCCC(O)(C(F)(F)F)c1ncco1)CCCCCCC#C CC1(CNC(=O)CN2CCCOC2=O)CCCN1C(=O)C=C1CCC1 C1(NC(=O)CCCN2CCCC2)CC2(CCCCN2C(c2ccc(Cl)nc2)=O)C1 CCC(O)C(C)C(=O)NC12CC(NC(c3cccc(OCCOC)c3)=O)(C1)C2 CC(C)C(C(=O)N1CCCN(C)C(=O)C1)C(C)NC(=O)CN1CCC(C)C1 CC(C)C(C)(O)C(=O)NCc1nc(C(=O)NCC(C)(C)n2ccnc2)co1 Cc1cc(C(C)NCC2(O)CCC(O)CC2)ccc1C#N C(=O)(CS(=O)(=O)CC(C)C)NCC(CC=C)C(=O)N1CCOCC1 N1(C(CSCC#C)=O)CC(F)CC1CN(C(=O)CC(N1CCCCC1=O)C)C Cc1cc(C#N)ccc1NC(C1CCC(NCc2cnc(Cl)s2)CO1)=O c1(CC(=O)NCC2(CNC(CN(S(C)(=O)=O)C)=O)CCCC2)cccc(C)c1 CN1C(=O)CCC1C(=O)NCC(O)CNC(=O)Cc1cccc(C(F)F)c1 Cc1ccc(O)cc1NC(C1(CNC(=O)C=CC(F)(F)F)CCCC1)=O c1(C(N2CCC(c3ccc(C)s3)CC2)C(=O)NCCC#N)ccc2c(c1)CCC2 Cc1ccc(C)n1CCC(=O)NCCC1CCN(C(C2CCCCCC2)=O)CC1 C(=O)(C(F)(F)CCC1CC1)N(CCCNC(c1scc(C)c1C)=O)CC C(=O)(C1=NOC(C)C1C)NCC(C(=O)NC(CC)(C)C)O C1(C(=O)NCCCC(=O)N(C)CC2(OC)CCCC2)(OC)CCCCC1 C1(C(N2C3C(NC(c4ccc(CN(C)C)[nH]4)=O)C(C3)C2)=O)CC2(C1)CC1(CC1)C2 c1(SC)ccc(Cl)c(C(=O)NC2CC(F)(CNC(=O)CC3CCCS3(=O)=O)C2)c1 CCC(C)C(O)C(=O)NC(C)CN(C)C(c1conc1C1CCC1)=O N1(C(C(F)OC)=O)CC=CC1CNC(=O)C(O)CC1CCCCC1 C(C(=O)Nc1ccc(Cl)cc1F)(C1=NOCC1)N1CC(C)OC(C)C1 c1(CCC(C)NC2CC(=O)N(CC3C(O)C(O)CN3C)C2)cc(Br)ccc1F C1(NC(c2cnc(C)s2)=O)CCN(C(c2cc(C#N)co2)=O)C1(C)C CN1CC(C(=O)NCC(CO)NC(c2cc(O)cc(O)n2)=O)CCC1=O CCCCCC(O)C(=O)NC(C)(C)C(=O)NC1CCN(S(C)(=O)=O)C1 CCC(CC)(C(=O)N1CC2CCC(C(=O)NC3(C)CCSC3)(C2)C1)C(C)C C(=O)(C1=CC2CC(C1)CC2O)N1C2(CNC(C(CCC)CC)=O)CCC1CC2 C1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)CCC(F)(F)CO1 N1(C(=O)OC(C)(C)C)CCC(CC(=O)Nc2ccc(F)c(F)c2)C(F)(F)CC1 c1(SC)cccc(NNC(=O)Nc2cncc(NC(=O)OC(C)(C)C)c2)c1 CC(C)C(C)(O)C(=O)NC1CCN(C(C2CCCN2C2CCOCC2)=O)CC1 CCCCC(F)C(=O)N1C(C(=O)NC)CC1C.C12(CC1)C(=O)NC2 CCC(CC(=O)N1CC2(CCN(C(C3COC4(C)CC3C4)=O)C2)C1)C(C)C C1(O)(C(C(=O)NCCOCCCNC(=O)C)F)CCCC1.n1(CF)cc(C2CC2)cn1 C(=O)(C1CCc2c(Cl)cccc21)NC1CC2(C(NC(C3CC4CCC3O4)=O)C2)C1 N1(C(c2cnn(-c3cccc(Cl)c3)c2)C(=O)NCC(=C)C)CCS(=O)C(C)C1C C12(C(=O)OCC)CC(CN(CC3CCCS3(=O)=O)C1)C2 N1(C(C23CC(C)C2C3)=O)C2CCC1CN(C(=O)Cc1sccc1Cl)CC2 C(=O)(C(=O)CCC(C)C)N1C(CNC(C2=CC(C)(CC)C2)=O)C(C)(C)CC1 C(=O)(C(CC)CCCC)N1CCC(C(N(CCCSC)C)=O)(C(C)C)C1 N#Cc1ccc2c(C(=O)NC3CN(C(c4coc5c4CSC5)=O)C3)c[nH]c2c1 C(=O)(C(C)S(N)(=O)=O)NCCC1CN(C(c2n(CC=C)ccc2)=O)CC1C CN1CCN(C2CCCC2NC(=O)Nc2cnn(CCF)c2)CC1 Cc1nc2c(N3CC(CC(C)NC(C4CCSC4)=O)C3)ncnc2s1 C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(O)(CNC(COC(CC)(C)C)=O)C1 C1(NC(C(c2cnn(C)c2)OC)=O)CCC(NC(=O)CCc2ccccc2)CC1 c1(OC)csc(C(=O)NC2CCC(CNC(=O)CCn3cc(Cl)cn3)C2)c1 c1(OC)cc(Cl)c(C(N2CCCC2C(=O)Nc2nccc(OC)n2)=O)cn1 CC(C)C#CC(=O)NC1(C)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)C1 S(=O)(=O)(c1c(Cl)cccc1Cl)NC1CN(C(c2ccc(F)c3ccoc23)=O)C1 c1(OC)cccc(COC(C)C(=O)N(CC(C)NC(c2cnccc2Cl)=O)C)c1 c1(C(CC)(C)C)ccc(C(=O)NC2CN(C(c3cnsn3)=O)CC2F)cc1 C1(C(=O)NC2CCC(N(C(=O)CNC=O)C)CC2)OCC2COCCC12 CN1N=C(CC(=O)N2CC(CNC(=O)CC3(O)CCOC3)CC(C)(C)C2)CC1=O N1(C(C2CN(C(C)(C)C)C(=O)C2)=O)CCCC(C)(CNC(C2CCS2(=O)=O)=O)C1 C1(C(=O)NCC2C(NC(CCc3scc(C)n3)=O)C2)CC2C=CC1C21CC1 c1(C(=O)NC2CN(C(C(n3cnc(C#N)n3)C)=O)C2)ccc(F)c(C(C)(C)F)c1 N1(C(C(C)N2CCCC2)=O)CCC(O)(Cc2ccc(Br)o2)CC1 C(=O)(C(CC(C)C)N(C)C(c1cc(C(N)=O)co1)=O)NCC(C#C)C(C)C Cc1ccn(CC(=O)N(C)CC2CCN(C(C3C4COCC34)=O)CC2)c(=O)c1 N1(CC(c2ccccn2)(C)C)CCC2(CC(=O)NC2=O)C1 C(=O)(CCCC(C)(F)F)N1C(CCCNC(Cc2c(C)ncs2)=O)CCCC1 N1(C(c2nccc(C)n2)=O)CCCC(NC(=O)CN(C)C(=O)C2CC2)C1C C1(NC(c2ccc(N(C)C)nn2)=O)COCCN(C(C2(C)CCOC(=O)N2)=O)C1 N#Cc1ccc(=NCC(=O)NCCCCCNC(=O)CCCS(N)(=O)=O)[nH]c1 C=CCCCCCCCC(=O)NC(C)C(C(C)C)NC(c1ccc(C)c(N)c1)=O C1(NC(CSCCCC)=O)(CCSCC(=O)NC(c2ccco2)=O)CCC1 c1(N2C(C)CC(CNC(C3(COCC)CCC3)=O)C2)ncnc(Cl)c1[N+](=O)[O-] C(c1cnc[nH]1)=C(C)C(=O)NC(C1CCOC1)CNC(c1occc1Br)=O N1(C(CC(CC)O)=O)CC(C)(C)OC2(C1)CN(C(c1csc(COC)c1)=O)C2 c1(NCC2(C)CCCN(C(=O)COc3cccnc3)C2)ccnc2[nH]cnc12 Cc1ccc(C(=O)NCc2ccoc2C(=O)NCC2CCC3CC23)c(F)c1 CC1CN(C(=O)CC2CCCC2O)CC1CC(=O)N(C)Cc1cn[nH]c1 c1(NC(C2CCN(C(=O)C=CC3CCOC3)C2)=O)cnccc1CO C1(C2CN(C(c3cccc(C)c3N)=O)C2)(NC(C2CC(CC)C2)=O)CC1 C(CCCCC(=O)N1CC2CC(NC(c3cnn(C4CC4)c3Cl)=O)C1C2)OC CC1=C(C(=O)NCCC2(NC(=O)COc3c(C)cccc3Cl)CCC2)CCO1 C1(CC)CC(NC(=O)C(=O)N(C(C)COc2ccc(OC)cc2)C)CCN1 C1(OC)CCCN(C(c2cccc(COc3nc(C)cs3)c2)=O)C1C C(=O)(C1=C(Cl)CCC(C)C1)NCC1N(C(CCCC#C)=O)CC(C)(C)C1 C1(NC(=O)Nc2ncc(CCO)s2)CC2CC1(c1ccnn1C1CC1(F)F)C2 c1(CNC(C(=O)OCC)CO)cc2c(Cl)cccc2s1 C1(NC(C2(C#N)CCCC2)=O)CN(C(c2ccnnc2)=O)CC2(CCC2)C1 C#CCC(C)(C(=O)NCC1(CC)CCOC1)NC(C)=O Cc1ccc(F)c(C(=O)NCCC2(CNC(c3ccc(C)c(O)c3)=O)CC2)c1 c1(OC)cc(C(N2CCCN(C(c3cc(Br)oc3C)=O)CC2)=O)cc(C)n1 N1(C(C(C)(C)CO)=O)CCN(C(c2ccc(O)nc2Cl)=O)C2CCCCC2C1 C(=O)(CCCC(=O)NC(C)CCCNC(=O)CCN(C1CCCCC1)C)OC Cc1cc(N2CCCC2CN(C(=O)C(C)Oc2ccccc2)C)nc(C)n1 c1(OC)nccnc1C(N1CC(O)CC1C(=O)Nc1ccno1)=O N1(CCC)CCCC1C(N1CC(CN(C(=O)C(F)=C2CCCC2)C2CC2)C1)=O C1(CNC(COCC(=O)OC)=O)CCCCC1NC(=O)COCc1nc(C)no1 C(CC(=O)NCC1CN(C(c2cc(C)n(C(C)C)c2C)=O)C1)(C(N)=O)NC(C)=O C(CC(=O)NC1CC(N(C(=O)CC2C=CCC2)C)C1)N(CCC)C N1(C(C(C)(C)NC(C(C)Nc2ccc(C)cc2)=O)=O)CCOCC(C)(C)C1 CCN=c1cc(C(=O)NCCC2CCC(NC(=O)C3=NNC(=O)CC3)C2)cc[nH]1 c1(NCCNC(C(c2cccc(F)c2)C)=O)ccc(C(C2CC(CF)C2)=O)cn1 C1(C(NOC(N2CCCC(Nc3ncccn3)C2)=O)=O)CCC2(CC2)C1 N1(C(c2c(OC)ccc(C)c2)=O)CCOCC(F)(CNC(=O)C(C)C(C)(C)C)C1 N1(C(c2c(C)ccnc2)=O)CC(CC(=O)NCC(C)C(C)(F)F)CC1(C)C c1(CCC)nc(C(=O)N(CCC(C)NC(C2CCCOC2)=O)C)cs1 N1(C(c2cc(Cl)sc2C)C(=O)N(C(CC)(C)C)C(C)(C)C)CC(C)SC(C)C1 C12(CCCC(C)(C)C1)c1nnnn1CCCN2.c1(CC=CCCC)ccc(F)cc1 N1(C(CCC(=C)Br)=O)CCCN(C(c2cccc(C(=O)OC)c2)=O)C(C)C1 C(=O)(CC(C)P(C)(C)=O)NCCC1(O)CCN(C(c2c(NC)cnc(Cl)c2)=O)C1 C#CCCCC(=O)NC(CNC(c1ccnc(Nc2ccccc2)n1)=O)CC=C N1(C(Cn2c(=O)ccc(C)n2)=O)CC(NC(=O)C(C)C(F)F)C2(CCC2)C1 C1(NC(c2c(C)csc2)=O)CCC2(CC1)CN(C(c1cnnn1C)=O)C2 N1(C(C(CC=C)N)=O)CC=C(c2cccc(Cl)c2)CC1 Cc1ccc(CC(=O)NCCC(C)N(C)C(c2ccc(CO)c(F)c2)=O)cc1Cl N1(C(C=CSC)=O)C2CCCC1CC(NC(C1CCCC3(CC3)C1)=O)C2 C1(CCOC)(NC(=O)C(C)c2ncco2)CCN(C(=O)CCCN(C)C(C)=O)C1 C1(C)(C(=O)NC2CN(C(C(CCC)(C)O)=O)CC2F)Cc2ccccc2C1 c1(OCC(N2CC(C)C(NC(=O)CC3CNC(=O)C3)C2)=O)cc(Cl)cc(Cl)c1 c1(C(N2CCC(O)(C(C)NC(C3CCC3)=O)C2)=O)nnn2ccccc12 C1(C(=O)NCCC2(NC(=O)C3=CCCCO3)CCC2)CCn2c(O)nnc2C1 C#CC1(C(=O)N(C2CC(C)CC(C)C2)C)CCN(C(=O)Cc2ccccn2)CC1 c1(CCC(=O)N(C2CCN(C(c3ccco3)=O)C2)CCO)ccc2c(c1)CCO2 N1(C(C2(CC=C)CC=CC2)=O)CCC2(NC(c3cc(O)nc(OC)n3)=O)CC2C1 C1(C(N)=O)(OCC2OCCC2C(=O)NCCOCC(=O)NC)CC(C)(C)C1 c1(C(=O)NC2(C(=O)NCC)CC2)cnn2c(C)cc(C)nc12 N1(C(CCC(C)(C)C)=O)CC2CC(O)C1C2NC(c1cnc2[nH]cncc1-2)=O CC1(C(=O)NC2CCC3COCCC3C2)CC2CCC1CC21OCCO1 C(=O)(C(CCC(C)C)NC(C)=O)NCCC1(OC)CN(C(c2cnco2)=O)C1 c1(OC)cccc(C2(C(=O)NCC(C)(C(C)C)NC(C3CC3OC)=O)CC2)c1 c1(NC(C)=O)cccc(C(=O)NC2CN(C(=O)C(C)C3CC3)CCC2F)c1C c1(C(=O)NCC(c2ccccc2)NC(CC=C=C)=O)ncc(F)c2ccccc12 c1(C(=O)NC2C(CNC(C(=O)NCCC(N)=O)=O)C2)n[nH]c2c1CCCCC2 CC1C(=O)CCC(C(N2CC(CO)(NC(c3nccnc3Cl)=O)C2)=O)C1(C)C C1(N(C(C2(NC(c3nc(C)sc3)=O)CC(CO)C2)=O)C)CCCC1(C)O C1(CNC(c2cnc(NC(C3(COC)CC(=C)C3)=O)s2)=O)CCCC1(C)O N1(C(c2cn(CC=C)nn2)=O)CCC(F)(C(=O)NCC(CO)OC)CC1 C(=O)(C1CCc2scnc21)NC1CCC(NC(C(C=C)O)=O)C1 CCC(C)CC(C)C(=O)N(CCCNC(c1ccc([N+](=O)[O-])cc1)=O)C N1(C(COCC(C)(C)C)=O)CC(=O)NCC1C(N1CCSC2(CC2)C1)=O C1(NC(c2cc(C)[nH]c2)=O)CN(C(=O)C(C)OCCC(C)C)C2(CCC2)C1 c1(C(N(C2CCN(C(=O)CCC(=O)N3CCOCC3)C2)CC)=O)c(C)nsc1N c1(C(=O)NC2CN(C(CC(CCOC)(C)C)=O)CC2F)cccc(C#CCO)c1 N1(C(c2cn(C(C)C)nc2)=O)CCC2(CNC(c3ccoc3)=O)CCCCC12 c1(C(N2CCC(C)C2C(=O)NC2CCCC(O)C2)=O)cc(=O)n(C)cn1 CCC(O)C(C)(C)C(=O)N1CC2(CC(NC(=O)CC(C)(C)COC)C2)C1 Cc1cc(C(N2CC(C(C)NC(C3(CO)CCOCC3)=O)C2)=O)cnc1CC#N C1(F)(CNC(C2(C(=O)NC)CC2)=O)CCCN(C(=O)CCCCCC#N)CC1 C(=O)(C#CC1CCCC1)N1CC(C=C)(CC(=O)N(CC(F)Cl)C)C1 C1(C(=O)NC2C(CNC(C(C(=C)C)(C)C)=O)CCC2)CC2(CCOCC2)C1 c1(C(N2CCC(c3ccon3)C2)C(=O)NC)ccc(-n2cccn2)c(F)c1 C1(CC=C)(NC(c2cc(C3(C)COC3)no2)=O)CCN(C(=O)C(F)C2CCC2)C1 c1(C(=O)NCC2OCCCN(C(C(CC(=C)C)C)=O)C2)cc(C#N)ccc1O CC(C)(C)CC(O)CC(=O)NCCNC(c1ccc([N+](=O)[O-])c(C(N)=O)c1)=O FC(F)(Br)CN=c1[nH]c(=NCC2CC3CCCC(C2)C3(F)F)[nH]c2c(F)cccc12 Cc1cn(CC(=O)NCC2CC(O)(CNC(=O)C(Cl)=CCl)C2)c2ccccc12 S(=O)(=O)(c1ccc(NC2CN(C)C2)c(Br)c1)N1CC(CC)OCC1C N1(C(CC(C)NC(C2CC(O)C2)=O)=O)CC2(C)CC1CCO2 c1(C(C)NCC2(NC(C)=O)C(C#C)C2)cc(OC)cc(OCC)c1 C(=O)(C1=CCCOC1)N(CC(=O)NCC1CC(C)CO1)CCOC N1(C(c2ccc(OCC=C)cc2)=O)CC(NC(c2coc(OC)n2)=O)CC1(C)C CC(O)(CNC(c1cn(CCO)nn1)=O)CNC(c1cn(C2CC2)cn1)=O C1(C)(NC(CCN2CCN(C)CC2)=O)CCN(C(C2COCCO2)=O)CC1 n1(CC(=O)NCC2CN(C(c3c(C)c[nH]n3)=O)CC23CC3)nc2c(n1)CCCC2 CC1(C)CC(CNC(=O)C(O)C2CCC2)CN(C(=O)C(c2ccc(F)cc2)=O)C1 c1(-c2cn(C(C)CNC(N)=O)nn2)ccc(C(F)(F)F)cc1 C1(C(=O)Nc2ccc(C)nc2O)C2C(CN1C(c1cc(O)cc(O)c1)=O)C2(C)C c1(CNC(CSCC)=O)ccc([N+](=O)[O-])cc1C#N CC1CCCC1(C(N1CCC1(C)C)=O)NC(c1ccsc1C#N)=O C(C(C)(CO)NC(=O)Cc1cn[nH]c1)NC(C=C(COC)C)=O c1(CC(=O)NC2CC(N(C(c3ccn(CCOC)n3)=O)C)C2)nnc(S)n1C CCC(CC)CCCC(=O)NC12CC(C(=O)NC(C)C(C)(C)CN(C)C)(C1)C2 c1(C(=O)NCC(CC)(CC)NC(CSCC=C)=O)ccc2nc(C)n(C)c2c1 c1(C(=O)NCC(CC=C)NC(C2(C)CC2C)=O)cc(OC)cc(Br)c1O N1(C(C(CC)CCOC)=O)CCCCC2(CCN(C(C3CCOC3)=O)C2)C1 CC1(C)CCN(C(c2cccc(Br)c2F)C(=O)Nc2ccc(Cl)cc2)CCS1 c1(N2CCC(C(=O)NCCN)C2)cc(=O)c(O)co1 Cc1ccc(CONC(=O)CC2CN(C(C3CCC4CC34)=O)CC2C)cc1 c1(C(=O)NC(C)CNC(=O)CCOCC(F)F)cc(C(C)(F)F)n[nH]1 C=C(Cl)CCC(=O)N(CCC(C(C)C)NC(=O)C(c1cscc1Br)=O)C C1(NC(CCOCC)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CC2(CC2)C1 C1(C)(CC)CCC(C(N2CC=CC2C(=O)NC2COCC2N(C)C)=O)O1 c1(C(N2CCCC(NC(CC(=C)Br)=O)CC2)=O)ccc2c(c1O)CCC2 N1(C(C2COCC3(CCC3)O2)=O)CCOCC12CCC2 N1(C(CC(C=C)C)=O)CCCC(N(C)C(c2ccc(CCO)cc2)=O)CC1 c1(C(N2CC(CC=C)(NC(C3CC4C=CC3O4)=O)C2)=O)ccc(Br)c(C)c1 N1(C(C=Cc2nnc(C(C)C)o2)=O)CC2CCN(C(C3OCCC3C)=O)C2C1 C(CCN=c1[nH]c(=NC(C)C(C)C)[nH]c2cccc(F)c12)c1c(C)n[nH]c1 C(C1CCCCC1)=CC(=O)NCCCN(C(=O)Cc1cocn1)C(C)C N1(C(C(CC(C)C)C)=O)CC23CCCC2(C1)CN(C(c1occc1Br)=O)C3 C1(NC(C2OCCC(=O)C2)=O)CN(C(=O)CCc2ccoc2)C2CCCC12 N1(C(c2cn(C)c(O)n2)=O)CC2CCN(C(=O)CCCCCF)CC12 c1(C(N2CCC(NC(C3(CCC)CC3)=O)C(C)C2)=O)n[nH]c2c1CCSC2 C(=O)(C=CS(=O)(=O)CC)NC1(C2OCC2(C)C)CC1.C12CCCCN1C(=O)CC2 N1(C(C2(CNC(c3ccc(CO)o3)=O)CCCO2)=O)CCOC(CCF)C1 Cn1cc(CC(=O)NCC2CCCC2NC(=O)Cn2cnnn2)cn1 N1(C(CCCNC(=O)C2CC2)=O)CC2CCN(C(=O)CC34CCCC3C4)C(C2)C1 CC1ON=C(C(=O)N2CC(NC(c3c(F)ccc(O)c3F)=O)C3CC3C2)C1C CCCC(CCC)C(=O)NC1CCN(CCCOc2ccc(F)cc2)CC1 N1(C(Cc2c(C)con2)=O)CCC2CCN(C(=O)C3=CCSC3)C2C1 c1(CCc2ccc(C)o2)nc(-c2ccc(Cl)cn2)nn1-c1nc(Br)nn1C N1(C(c2cc(C(=O)OC)on2)=O)CC2CC(NC(C3CCOC(C)C3)=O)CC1C2 Cc1ccc(Cl)c(C(N2CCC(C(C)(C)CNC(C3COC(C)C3)=O)CC2)=O)c1 N1(C(c2n(CCC)ccc2)=O)CC(NC(C2CCCCCS2(=O)=O)=O)C2(CC2)C1 Cc1cccc2c1CN(C(=O)Cc1ccccc1NCc1c(F)cccc1Br)C2 c1(C(=O)NCC2(NC(=O)CN3CCc4ccccc43)CC2)n[nH]c2ccc(F)cc12 c1(C(=O)NCC2N(C(CC=C(C)C)=O)CCCC2C)cc2ncccc2[nH]1 N1(C(C2(C(=O)NC)CCC2)=O)CCOCCC1C(=O)NC1CCC=CCC1 N1(C(C(F)=CCC)=O)CCCC(C2CN(C(c3ccn(CC4CC4)c3C)=O)C2)C1 c1(OC)cccc(C(N2CCN(C(c3ccc(C)c(F)c3)=O)CC2CF)=O)c1N Cc1ccc(F)c(C(=O)NCC#CCNC(=O)CC2=CCCC2)c1O c1(C(N2CC(C#N)C(NC(C3CCCO3)=O)C2)=O)cccc2nc[nH]c12 c1(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)ccn2nccc2c1 c12c(C)nc(nc1O)SC2.c1(CC(COC)C(C)C)ccc(F)c(F)c1 C1(NC(C2OCC(C)C2)=O)CC2CCC1(N=c1[nH]nc(C3CC3)o1)C2 C1(C(N2CCC(N(C(c3cccc(C)c3O)=O)C)CC2)=O)CC2CCCCC2O1 C1(NC(C(CCC)C)=O)CC(O)CN(C(=O)CCc2cccnc2F)C1 C1(NC(c2cn(CC)nc2C)=O)CCN(Cc2cccc(F)c2F)CC1(C)C C(C)(N=c1[nH]c2cc(C)cnc2s1)c1cc(O)cc(OC)c1.N1(CC)CCCCC1 C1(N(C(CCNS(C)(=O)=O)=O)CC2CC2)CCN(C(=O)C(C)(C)C#N)CC1 C(=O)(C(O)C(C)(C)CC)N1C(C(=O)NC2(C=C)CCCC2)(C(C)C)CCC1 C1(C(=O)NCC2CCN(C(c3n(C(C)C)ncc3)=O)C2)CCS(=O)(=O)C1(C)C CC1C(NC(=O)Cn2nccn2)CC2CCC1N2C(=O)CN1CC(=O)N(C)C1=O CC1(C)CCCC(C(=O)NC2CC(C)(NC(=O)CNS(=O)(=O)C3CC3)C2)O1 C1(C(CNC(=O)C(F)=CC2CC2)F)CCN(C(C2CC3C=CC2C3)=O)CC1 c1(C(N2CC(C(C)NC(COC)=O)OCC2)=O)cc2nc(=O)ccn2[nH]1 N1(C(C2(SCC)CC2)=O)CCN(C(c2cc(CC)ccn2)=O)CC1CC CCC1(CNC(=NCC(C)CC)NCc2cccs2)OCCc2ccccc21 C1(CC(=O)NCCC(C(C)C)CC(=O)NC(C2CCOC2)=O)CCC(C)(C)CO1 Cc1cc(=NCC2(F)COCCOC2)[nH]c(N2CCN(C3CCOCC3)C(=O)C2)n1 Cc1cccc(CNC(C2CCC(n3cc(CCOC(=N)O)nn3)C2)=O)c1F CCCCCCCCCCCC(=O)N(C1(C(=O)N(CCO)CCO)CC1)C C(C(=O)NCC=CCNC(c1ccsc1C#N)=O)(C(C)C)SC N1(C(C(C(CC)O)C)=O)CCC2CN(C(c3cc4nc(C)sc4[nH]3)=O)CC2CC1 c1(C(N(C(C)C(N2CCC(OCCN(C)C)C2)=O)C)=O)cc2ccccc2cn1 CCC(CCCC(=O)Nc1cnccc1C)NC(C1(C)CCCCC1)=O CCC(CC(F)(F)F)C(=O)N1CC(CNC(c2c[nH]nc2C2CCC2)=O)C(C)C1 C(=O)(C(CNC(C1CCC(=O)N(C)C1)=O)C(C)C)NC(C(CC)C)CO c1(C(C)NC(N)=O)cn(CC(N2CCCC2CNC(=O)CC2(O)CCC2)=O)nn1 c1(OC)ccc(F)c(C(N2CCCCC23CC3)C(=O)Nc2ccccc2Cl)c1OC N1(C(c2c(OC)ccnc2)=O)CCC(CC(=O)NCC(O)C(N)=O)C1(C)C c1(CC(N2CC(O)(CCc3cn(CCC(C)C)nn3)C2)=O)ccc(Cl)nc1 C1(C(N(C(C)CCNC(=O)CCc2c[nH]c(=N)[nH]2)C)=O)CC2C=CC1C2 CCC(C)C(C(=O)N1CC2(C)CC1(C(=O)N(C)Cc1ccoc1C)C2)OC CCCCCC(CC)C(=O)N1CCC(C)(NC(c2ccc(OC)nc2F)=O)C1 N1(C(CC2CCC(=O)C2)=O)CC2(C=C(C(=O)NC3CCC(O)C(O)C3)CO2)C1 C(=O)(C(F)C(C)C)NCC1(C(N)=O)CN(C(c2n(COC)ncc2)=O)C1 C(=O)(C1CCCn2cnnc21)N1C(CC)CN(C(=O)CCN(CC)CC)CC1 C(CCCCCC(=O)N1CC(C(=O)O)C2(COC2)C1)S.N(C)CC C(=O)(C(=O)C(C)(C)C)N.C1(CN(CC)CC)CCCCN1C(=O)C(F)n1cccn1 C12(C(=O)NCC3CC(NC(CN(c4ccccc4)CC)=O)C3)CC=CC(C1)OC2 C1(C(N2CCC(N3CCC(CN4CCOCC4)C3)C2)C)OC(=O)CC12CNC2 C12(NC(C3CN(C)c4c3cccc4)=O)CN(C(=O)CCC3CC3)CC1CS(=O)(=O)C2 N1(C(CN2C(C)CC2)=O)CC2CC2(NC(c2ccc(CNC(N)=O)cc2)=O)C1 C(C)(c1ccccc1C)=NC1(CC2CC(COC)CN2C=O)C(C(=O)OC)C1.C1(C)CC1 C1(NC(C2CCC(CNC(c3c(C)nns3)=O)O2)=O)CC(=O)N(C(C)C)C1 c1(-c2[nH]nc(C(C)Nc3cn(C(c4ccccc4)C)nn3)n2)ccc(F)cc1F CCCCCCC(C)C(=O)NCC1=CCCN(C(=O)CN(C)C)C1 Cc1cnn(C(C)C(=O)NCC2(O)CN(C(=O)C(C)(C)c3cnco3)C2)c1 c1(NC(C2(O)CCN(C(C(C=CC)O)=O)C2)=O)cc(OC)ccc1C C1(C(N2CC(C)N(C(=O)CC3NC(=O)NC3=O)CC2)=O)CCc2nc(O)[nH]c2C1 N1(C(c2cnc(COC)s2)=O)CC2CC1CN2C(=O)C=Cc1cc(F)c[nH]1 N1(C(C2CC(N(C)CC)C2)=O)CCCOC(CNC(=O)C(C2CCCCC2)O)C1 C1(CC(=O)N(C2CN(C(=O)Cn3cc(Cl)cn3)C2)C)C=CCCC1 N1(C(Cc2cc(COC)on2)=O)CC(NC(c2csc(O)n2)=O)C(SC)C1 c1(SCC)cccc(CC(N2CCN(C(=O)C(C)C(=O)OC(C)(C)C)CC2)=O)c1 CP(C)(=O)c1ccc(C(=O)NC2CCN(C(C3OCCCO3)=O)C2)cc1 C(=O)(C1CCc2c(Cl)cccc21)NC1(C2CN(C(CC(=O)OC)=O)C2)CC1 CC(C)(C)S(=O)CCCN=C(NCC1CCCCO1)NCC1C=CCC1 c1(OC)c(C(=O)NC23CC(C2)N(C(=O)CC2(CO)CC2)C3)cccc1F N1(C(CC(C=C)c2ccccc2)=O)CC2(CCN(C(C3(C#N)CC(C)C3)=O)C2)C1 C(CCC(C)C)(C(=O)NCC1C(=O)NCCC1C)NC(C)=O C1(NC(C2CCN(C(c3cc(=N)[nH][nH]3)=O)C23CC3)=O)CCc2nn[nH]c2C1 C(CC(CC)C(=O)N1CC(O)(CNC(=O)COc2cn[nH]c2)C1)=CC c1(OC)cc(C(C(=O)NCC(CO)NC(c2occc2C)=O)SC)c(F)cc1O Cc1cc(C)c(C(=O)NC2CCN(c3ccccc3F)CC2)c(O)c1 C=CC1(C(=O)NC2CCCC2)CCN(C(C2CCOC(C)(C)C2)=O)C1 c1(C(C)NC(CCCOC)c2nnnn2CC(F)F)ccc(OC)c(C)c1 N1(C(C(CC)SC)=O)CCCC(F)(CNC(=O)C=NOC)C1 N1(C(CC2CC(C)C2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 c1(C(=O)NCC(C)(CC)NC(C(COCC)C)=O)cncc(C(=O)OC)c1C C1(C(=O)NCC2CCN(C(Cc3nnc(C)o3)=O)CC2)CCCNS1(=O)=O C(=O)(C(C)(F)C(C)(C)F)N1CC(CNC(=O)CCC(C)(C)F)CC(C)C1 C1(C(=O)NCC(CNC(C(C)NC(CC)(C)C)=O)C)CCS(=O)(=O)CC1 C1(CNC2(C)CN(CC(=O)OC(C)(C)C)C2)CCC(c2ccccc2)CC1 Cc1nccnc1C(=O)NCC1CCCN1CC(=O)NC1CCCC1 C12(CNC(c3ncn(C(C)C)n3)=O)CC(CO1)N(C(c1cccc(=S)n1O)=O)C2 c1(N2C(C(=O)Nc3ncc(C)nc3Br)CC3(CC3)C2)nc(Cl)c2c(ccn2C)n1 CC1(C)OCC2CC12C(=O)NCC(C1CC1)NC(C1C2CCCCC12)=O CC(CC(=O)N1CCCC1CNC(c1ccnn1CC#N)=O)CC(C)(C)C C1(CNC(c2cnc(C(C)C)[nH]2)=O)CN(C(=O)C(c2ccccc2)F)CC1(F)F C(=O)(C(C(C)C)c1ccc(Cl)cc1)N1CC(CC(=O)OC)(C(F)(F)F)C1 Cc1c(C(N2CCC(OCCNC(C3CCCN3C(C)C)=O)C2)=O)ccn1C Cc1cnc2c(C(=O)NCC(C)(C)CNC(=O)CSC(F)(F)F)cccn12 CCC(CC(F)F)C(=O)NCCCN1CCN(c2nsc(NC(C)=O)n2)CC1 C(=O)(C(C)(C)C(C)(C)O)NC1CC(CCNC(C(C)OCC)=O)C1 c1(SC)ccnc(N2C3CN(C(c4cc(I)c[nH]4)=O)CC23)n1 c1(NC(C(N2CC3C(C)C3C2)C2C(CC)C2)=O)ccccc1C c1(OCC)cccc(C(=O)N)c1.c1(C(=O)N)n[nH]c(C)n1.C1CCOCCOCC1 C(C)(C)(CCCNC(c1cc(-n2cccc2)ccn1)=O)NC(COCC)=O C=CC(C)(CCOC)C(=O)NC1CCC(CCC(N2CCC(C(N)=O)C2)=O)C1 c1(C(C(=O)OCC)OC(c2c[nH]nc2CC)=O)ccccc1Cl C(=O)(C1=C(Cl)CCC(C)C1)NC1COCCN(C(c2c(NC)cncc2)=O)C1 c1(N2CCN(C(COC)COC)CC2)nccc2oc(Br)cc12 c1(C(C)(C)C)cnn(C)c1C(=O)NC1CC(CNC(=O)C=Cc2ccc(Cl)s2)C1 C1(C(N(CC(C)(C)CNC(=O)CC2CCCO2)C)=O)CCCC2(CCC2)O1 c1(CC(=O)N(CCCNC(=O)Cc2cc(Cl)ccc2O)C)nc2ncccn2n1 CCC(CC)C(C)C(=O)NCC1(CN(C)C(c2ccnn2C2CC2)=O)CC1 N1(C(C(C)C(C)(C)C)=O)CCC(C2(NC(=O)COCC3CCCO3)CC2)CC1 c1(CC(=O)NCCCN(C(c2ocnc2C)=O)CC)cccc2c1OC(C)(C)C2 S(=O)(=O)(c1cc(C)ccc1C)NCC(=O)NC(C(F)=CC)=O.C12CCC(CC1)C2 N1(CCc2c(OC)cccc2)CCC(NC(C2CCC(=O)N2)=O)CC(C)(C)C1 C1(OC)CN(C)C(C)(C(=O)NC2CN(C(=O)CCc3cncs3)C2)C1 CCCC(C)(O)CC(=O)NC1CCN(C(=O)C(=O)NC2CC2)C1 C(=O)(C1CCCc2ncnn21)N(CC(=O)N(C1CCCCC1S(C)(=O)=O)CCO)C C=CCC(CC(C)C)C(=O)Nc1cccc(NC(C2CCCNC2=O)=O)c1 Cc1cc(OCC(N2CCC(CN(C)C(c3cc(C(C)(C)C)no3)=O)C2)=O)no1 C(=O)(C(O)C(F)(F)F)NC1C(CNC(=O)CCCNc2ccccc2)CCCC1 N1(C(C(CC(CC)C)NC(c2ccc(C(C)C)o2)=O)=O)CCCC(C2(C)CC2)C1 N(C(=NCCNS(C)(=O)=O)NCc1cc(Br)cc(I)c1)C(C=C)C C1(C(N(CC(F)Cl)C)=O)CN(C(=O)C(C)(C)C2CCOC2)CC12CC2 C(CCC(F)(F)F)N(C(=O)CCCN(C)C(C1CCCOC1)=O)C C1(C(N2CCC3(C2)CN(C(C2(C4(O)CCC4)CC2)=O)C3)=O)CCC2(CCOC2)O1 C1(OC)CC(NC(=O)CC2CCSC2)CN(C(C2(C)CC2C)=O)C1 c1(C(N(C2CCN(C(C34CC(C)C3C4)=O)C2)C)=O)cccc2c1CCC2=O C1(C(NOCC(C(C)C)O)=O)CCC2CCC1N2C(=O)CCc1cnco1 CC1CCCn2ncc(C(=O)NCC3CC(NC(C4C(C)C4C)=O)C3)c21 CC1Oc2cc(C(N3CC(NC(=O)C(N)=O)C(C(F)F)C3)=O)ccc2NC1=O C(CN=c1[nH]c(=N)[nH]c(=NCC(C)Cn2ccnc2)[nH]1)c1c(OC)cccc1C C1(CN)CN(C(=O)Cn2cn[nH]c2=N)CC1C.Cc1occc1CC(=O)N1CCC1 C1(CC=C)(NC(C2CC23CCCC3)=O)CCN(C(=O)CS(=O)(=O)NC)CC1 C1(NC(C2(C#N)CCC2)=O)CN(C(c2ccc3c(c2)OCC3)=O)C2(CCOC2)C1 C1(NC(CC(C)(C)N(C)C(C2CCCC(C#N)C2)=O)=O)CCOC12CCCC2 c1(SCC)ccc(C(=O)NC2CCCN(C(C)=O)C2)c(F)c1 C1(C)(C(=O)NC2(C)CC(NC(c3ccn(CC(C)C)n3)=O)C2)CC2CC2C1 c1(-c2ccc(CCCC)s2)ccc(C(N2C(C(=O)O)CC2C(C)C)=O)cc1 C1(NC(CC(C)(C)O)=O)CC(C2CCN(C(=O)Cc3cc(F)ccc3Cl)C2)C1 CC(C)CCCCC(=O)NCCN(C(=O)CCC1CC1(F)F)C1CCCC1 C1(CCNC(=O)CSc2cncs2)COCCN1C(=O)C(F)=C1CCCC1 N1(C(C(CSC)O)=O)CCCCC1CCC(N1CC(F)(F)C1C1CC1)=O CC1CCN(C(=O)CN2CC3CC3C2)CC1NC(c1ccc(Cl)cc1N)=O C(=O)(CC1NC(=O)c2ccccc21)NCCNC(=O)NCCON CCC(CC(=O)NCCN(C(=O)CC1CC(F)(F)C1)CC1CC1)C1CC1 c1(C(N(CC(C)N(C(CCSCCCC)=O)C)C)=O)[nH]c2ccc(C)cc2c1C c1(C(=O)NC2C(NC(C3(CC#C)CCCC3)=O)CCC2)cncnc1C1CC1 C1(C(N(C(C)CNC(c2cnc(SC)s2)=O)CC)=O)CC(C)=NO1 c1(-c2n(C(COC)C)nc(C(C)C)n2)cc(Br)c2cccnn12 CC(C(=O)NCC1CC1C(=O)NCCN1CCC1)C(C)(C)C CC1CN(C(C2CC3(CCO2)CC3)=O)CCC1NC(c1cnc[nH]1)=O c1(C(N2CCC(N(C)C(C3CC4CC4C3)=O)C2)=O)ccc2c(c1)COC2 N1(CCNC(CCN(CC#C)C(C2CC2Cl)=O)=O)CCCC1=O C1(NC(C2(C=C)CC2)=O)C2CCC(C2)C1NC(=O)Nc1c(C)cccc1C N1(C(CC2(C)CCOC2)=O)CC2(CCN(C(=O)CCn3ccnc3)CC2)C1 CC(C)(C)CC(C(=O)NCC1CCCCO1)NC(c1cccn2ccnc12)=O c1(C(C(=O)NCCCOC)N(C2CCOC2C)CC)cc(F)ccc1C c1(C(N(C)CCC2CCCCN2C(=O)COC2CCCC2)=O)nnc(O)nc1O C1(C(=O)NC(c2cc(C)on2)C)CC2CCCC2N1C(=O)C=CC1CCCC1 Cc1ncccc1CC(=O)NCC1(NC(C2CCCN2N=O)=O)CC1 C(CN=c1[nH]c(N2CCn3cnnc3C2)nc2cccc(F)c12)OC(C)C CC1CN(C(Cn2cc(Sc3ccncc3)nn2)=O)CC(C)O1 CCCCCC(C)CC(=O)N1CC2(CCC2NC(c2cnn(C)c2SC)=O)C1 C=CCCCC(=O)N1CCCC1(CC=C)C(=O)Nc1cncc(C)c1 C1(C(N)=O)(NC(CC2C(NC(CC(C)O)=O)CC2)=O)CCCCC1 C(=O)(C(C)C(CC)CC)N1C(C(=O)NC(C#C)C2CC2)CCCCC1.C1(C)CCCC1 C(C(C)(C)CC(=O)NC1CN(C(=O)CSC)CCC1F)SC C1(N(C)C(C2CC2c2cnn(C)c2)=O)CCCN(C(C2(C)CC(F)(F)C2)=O)CC1 N1(C(CCC=C)=O)CC2(CC(NC(=O)COc3cnn(C)c3)CO2)C1 N1(C(CCOCCNC(c2c(COCC)nn(C)c2)=O)=O)CC(O)CC1(C)C c1(C(C(=O)NC2C3CN(C(C(C(C)C)SC)=O)C2C3)C)cc(C)cc(C)c1 c1(C2(C(C=C)N(C(C)CCC(=O)OCC)C3CC3)CC2)ccc(Cl)cc1 C1(NC(C2C(C)N(C)CC2)=O)CN(C(C2CC(N(C)C)C2)=O)Cc2ccnn2C1 N1(CCn2cc(CCCNC(CCc3n(CC)ccn3)=O)nn2)CCC(F)(F)CC1 c1(NC(C(C)C2CCOC2)=O)cnc(O)c(F)c1 N1(C(C2N(C)CCOC2)=O)CCC(C2(O)CN(C(C3CC4(C3)CC4F)=O)C2)CC1 c1(-c2cccc(NC(CC(CCC)NC(C)=O)=O)c2)ccc2cnoc2c1 CON1CCC(C(=O)NCCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CCO2)CC1 N1(C(C(COC(C)C)(C)C)=O)CC2CC(NC(c3ccc(C(N)=O)nc3)=O)C1C2 N1(C(CCSCC(C)C)=O)CCC(CNC(C2(N(C)C)CCCCC2)=O)CC1C C1(CC(N2CC(CC(C)CNC(C(N3CC(C)C3)C)=O)C2)=O)CCC(=O)C1 c1(C(=O)NCC23C(CN(C(c4scc(COC)c4)=O)C2)C3)cnc(Cl)c(N)c1 c1(C(=O)NCC#C)cc(OCC)nc(C)n1.C1CC(=O)NC2C(CC2)N1 C(=O)(C1=C(Cl)CCCC1)NCC(CCC)NC(c1ccn(CC)c(=O)c1)=O c1(OC)cc(OCc2ccccc2N2C(=O)C(C)C(C)C2=O)c2c(n1)CCCC2 N1(C(=O)Cc2cccc3c2OCO3)CC2CN(C(c3coc(CO)c3)=O)CC2C1 N1(C(C2CC2F)=O)CC2CN(Cc3ccc(C(F)(F)F)cc3Cl)CC2C1 C1(CC)CCC(C(=O)NCC(C)(C)NC(c2cc(C)ns2)=O)C1 C(CCCC(CO)NC(=O)CSc1n[nH]c(=N)s1)NC(C(CSC)C)=O C(CN=c1cc[nH]c(=NCCCC2(NS(N)(=O)=O)CCC2)[nH]1)N1S(=O)(=O)CCC1 c1(C(=O)OC)cc(N2CCC(C)(NC(c3ccc(Cl)s3)=O)C2)nc(C)n1 c1(C(N2CC(O)CC2C(=O)OC)=O)cc2ncccc2[nH]1.C12CC3(CC13)C(=O)N2 CC1CC(C(=O)N(CC(=O)N(C)C)C)N1C(=O)COc1cn[nH]c1 c1(N(CC(=O)NCC)CC)nnc(CC2COCCO2)n1CC N1(C(c2n(C)cnc2)=O)CCN(C(c2ccc(C(C)(C)C)s2)=O)C2CCC12 C12C=CCCN1C(=O)CC=CCNC2=O.n1(C(C)C)cnnc1C(C)C N1(C(CNS(C)(=O)=O)=O)CCC2(CCOC2)C(CNC(c2csnn2)=O)C1 c1(C(C(=O)NCCCC2CC2)NC(C(C)N(C)CC)=O)ccc(CO)o1 C1(C2CC2)(COC)CN(C(=O)C(C(C)C)NC(C2(O)CC2)=O)C1 C1(NC(C2(CC#C)CCN(C(=O)CC3CC(=O)C3)C2)=O)CCCCC1N=[N+]=[N-] N1(C(c2ccc(OCOC)cc2)=O)CCCC12CCS(=N)(=O)CC2 c1(C(=O)NC(CNC(C(C)(C)SC)=O)CO)cnc(C(F)F)nc1 Cc1nn(C)c(C)c1C(N1CCCC(CNC(=O)CN2CCC(C)(C)C2)C1)=O N1(CCCCC)CCOC2(CCN(C(=O)Cn3nc(C)c(C)c3C)CC2)C1 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CC(NC(C34CCCC(CCC3)C4)=O)CC1C2 N1(C(C(C)CC2CCCCC2)=O)CCC2(CCC2CNC(c2ccns2)=O)CC1 C1(C(N(CCC)CC)=O)CC(=O)CN1C(c1cc(CC)sn1)=O C1(C(N2CC(C(C)NC(C3CCC(=C)CC3)=O)C2)=O)CCOC2(CCOCC2)C1 c1(C(=O)NC2CN(Cc3c(F)cccc3F)CC2O)c(F)cc(F)cc1Cl Cc1nnc(O)c(C(=O)NCC2CN(c3nnc(C(F)F)o3)CC2C)c1C N=c1[nH][nH]c2ccc(C(N3CCC(O)C3C(=O)NC3CSC3)=O)cc12 C1(O)(C(N(C)CC2CCCN2C(C2CC3CCC2C3)=O)=O)CCCCCC1 S(=O)(=O)(c1c[nH]ccc1=NCC(CO)C1CCC1)N(CCC(O)C(C)(C)C)C C#CC1(C)CCCN(C(c2csc(C(=O)OC)c2)C(=O)Nc2ccccc2Cl)C1 CC1(C#N)CN(C(=O)C(Cc2ccoc2)NC(c2cnn[nH]2)=O)C1 Nc1[nH]c(=O)c(Cl)nc1C(=O)NCC1CCCCC1NC(c1cnns1)=O c1(C(=O)NCCCOCCNC(C2(C(=O)NC)CCC2)=O)c(Cl)ccc(C)c1O N1(c2cc(C)nc(NC3CC(C)C4=CCC3C4)n2)CCc2cc(F)cc(F)c2C1 n1(C(C)(C)C(=O)NC2CCC(CNC(C3CC(C#N)C3)=O)C2)cc([N+](=O)[O-])cn1 C(C)(CC(C)NC(=O)C(F)(F)C1CCCC1)NC(C1(CCCC)CC1)=O C1(NC(CSCC(=O)NCCCOC2CCC2)=O)C2CCC(=O)C12 N1(C(CC(C=C)c2ccccc2)=O)CC2(CNC(=O)CC(C)(C)C)CC1CO2 c1(CC(N2C(CNC(C3N(C)CCOC3)=O)CC2)=O)cccc(C(F)(F)F)c1Cl c1(C(=O)NC2C(C(=O)NCCC(=O)Nc3ccc(Cl)cc3)C2)cc(F)ccc1Cl C1(NC(c2ncc(Cl)cc2Br)c2n(CC)nnn2)CCOC2(CCCC2)C1 C1(NC(CCNC(C)=O)=O)CCCN(C(=O)Cc2ccccc2C)CC1F c1(C(=O)OC(C)CNC(c2cnn(C)c2)C(=O)OC(C)(C)C)ncc(F)cc1F C1(CC(=O)NCC(C)NC(C2(c3ccc(F)cc3)CC2)=O)CCOC(C)(C)C1 C(=O)(CC(C(N)=O)NCCCOCCC(C)C)OCC c1(OC)cc(N)ccc1C(=O)N(C)CCNC(=O)C(Cc1ccccc1)N(C)C N1C2CCc3c(cccc32)OC(C=C)(C)c2nnc1n2CCOC.C1(OC)CCCC1 C=CC(C)CC(=O)N(C)CCN(C)C(C1C(c2ccncc2)C1(C)C)=O C1(O)(CNC(c2n(C)c(S)nc2)=O)CCCN(C(C2CN3CCN2CC3)=O)C1 C1(O)(C(C(=O)NCC2C(CN(C)C)C2)F)CN(C(=O)Cc2cncs2)C1 C(CCC(=O)N1C(=O)CCCn2ccnc21)n1cc(CC(C(C)(C)O)O)nn1 N1(C(CSCC(=O)OC)=O)CCCCC1CCC(N1CCCC1C(C)(C)OC)=O C(=O)(C(C)CC(F)(F)F)NC1CN(C(C2CC(C(C)C)C2)=O)C(CO)C1 c1(C(N(CC(CNC(C(c2ccc(Cl)s2)C)=O)O)C)=O)ccnnc1S CC(C)(C#N)CC(=O)N1CCC(O)(CCNC(=O)CS(=O)(=O)NC2CC2)CC1 C1(ONC(C2(NC(C=CC(=O)N(C)C)=O)CCC2)=O)CCCC1C n1(CC)c(C(=O)NCC(C)(CO)NC(=O)CCCn2cccn2)cnc1O c1(CC(=O)N(C2CCN(C(C3(O)CC3(C)C)=O)CC2)C)ccc2c(c1)CCC2 C12(C(=O)OC)CCC(C(=O)NCCC3(O)CN(C(C4CCCO4)=O)C3)(C1)C2 c1(CCC(N2CCC(CNC(=O)CC3CC3)C2)=O)ccc(Br)c(F)c1 c1(C(=O)NCCC2CN(C(C3COCC(C)O3)=O)C2)ccc(F)c(Cl)c1F C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCOC(C)C1C(=O)O Cc1cc(C(=O)OCCOC2CC(OC(=O)OC(C)(C)C)C2)nc(Br)c1 N1(C(CC2(OCC)CCC2)=O)CCC(C)CC1C(=O)Nc1cccc(C(C)C)c1 N1(Cc2n(C)nc(-c3ccsc3)n2)Cc2ccc(F)cc2C1 c1(OC)cccc(C(F)(F)C(=O)NC2CCCC2NC(=O)Cn2nnnc2C)n1 C1(NC(CCOCCC)=O)CN(C(C2CCC(C)(C)O2)=O)CC2CCCC12 N1(C(C2C(C)C2)=O)CC(CNC(=O)CC2=NNC(=O)C2)C2(CCOCC2)C1 N1(CCN2CCOCC2)CCCc2cc(C(c3ccc(OC)nc3)O)ccc2C1 c1(OCC)ccc(F)cc1COC(=O)C(N1CCCC(c2nc(C)nn2C)C1)=O C#CCC(CC(F)F)C(=O)N1CCC(CCOC)(NC(C2CN3CCC2C3)=O)C1 N12CC(C(CS(C)(=O)=O)C1)C2=O.c1(NC(COC(C)=O)=O)cccc(F)n1 c1(COC)ccc(C(=O)NCC(O)CNC(=O)Cc2cccnc2OC)cc1C c1(C(N(CCNC(C(CO)N(C)C)=O)CC2CC2)=O)cc(O)nc(N(C)C)n1 Cc1c(CCC(N2CCC(C)(NC(=O)CC3C=CCCC3)C2)=O)cnn1C CC1CN(C(C2(CCF)CCC2)=O)CC1(C)CNC(c1cc(Br)sn1)=O N1(C(C2C(C(C)C)C2)=O)CC(NC(c2cccc(OCC3CC3)c2)=O)C(F)C1 C#CC1(CNC(=O)CCC2CN(C(=O)Cc3ccccc3O)CCO2)CCOCC1 N(C(=NCCCCCCSC)NCC1COC1)CC1C(OC)CCC1 C(=O)(CCCCCC(C)O)NCC(C(C)(C)C)NC(c1c(CC)[nH]c(=N)s1)=O C1(NC(C=CC)=O)CN(C(=O)CSc2ccc(C)c(C)c2)Cc2nccn2C1 N1(C(C2(COC)C=CCN2C(=O)Cc2ccsc2C)=O)CC=C(CO)CC1 CCCCCCCCC(=O)N(CC(C)CNC(c1nc(O)c(C)s1)=O)C C1(C(N(CC)CC2CCCCO2)=O)CCC(NC(=O)Cn2cnnn2)CC1 C1N=C(NC2CC=CCC2)NCC2CCCC12.N1(S(C)(=O)=O)CCCC1 C1(C)(CNC(C2CC(C)OCC2)=O)CCCN(C(C2(F)CC2)=O)C1 C=CCC(CC)C(=O)NCC1CC(OC)CN1C(c1cc(Br)sn1)=O c1(NC(N2CCCC(NC(=O)CN3CCOC3=O)CC2)=O)ccc(Cl)c(F)c1F CC1CC(NC(C2(C(F)(F)F)CCC2)=O)CCN1C(=O)CCC1CC1 C(=O)(C(CC(=C)Cl)NC(C1CCC(F)C1)=O)NC(C#C)(C)C O=C1OC2CC(C(N3CCCN(C(C4CC(CCO)C4)=O)CC3)=O)CC2O1 c1(OC)ccnc(F)c1C(N1CCCC(C(C)NC(c2cc(CF)on2)=O)C1)=O CN1CC(O)CC1(C)C(=O)NCc1cc(C(=O)NC2(CCF)CCC2)on1 C1(N(C(CC(C)OCC2CCCCO2)=O)c2ccccc2)C2CN(C3CC3)CC12 N1(C(CC2(NC(C(n3ncc(C)c3)C)=O)CC2)=O)CCCC2(CCOC2)C1 C1(C(=O)NC(CNC(c2c(C)nn(C(C)(C)C)c2)=O)C2CC2)CC(C)(C)CN1C c1(C(N(CC(CNC(C(c2ccnn2C)C)=O)O)C)=O)cc2c(nn1)CCCC2 C1(C(=O)NC(CCCC=C)C2CC2)CC12CCN(C(=O)C1=CCSC1)C2 C1(C(=O)NCCCNC(C(C2CCCCC2)N(C)C)=O)C(C#N)C1(C)C c1(C(N2CCCC(N(C(COCCCC)=O)CCF)C2)=O)cnn2ncccc12 CC1CN(C)C(C)CC1NC(C1C(CNC(C2(C)C=CCCC2)=O)C1(C)C)=O Cc1ccc(Br)cc1CC(=O)NC12CC1CN(C(=O)C(C)Cc1ccco1)C2 N1(C(CC2(OCC)CC2)=O)CC(NC(c2ccn(C)c2)=O)CC(O)C1 C=CCCC(CC(C)C)C(=O)N1CC(CNC(c2ccnc3nccnc23)=O)C1 c1(CC(=O)NCC(CC)NC(=O)CCc2nc(SCC)no2)cccc(C)c1C C1(C(N(CCCO)CC)=O)CCOC1CNC(=O)CCCc1cnn[nH]1 c1(C(C)C)nnc2cc(N3CC(NC(C4CCC4(C)C)=O)CC4(CC4)C3)ncn12 N1(C(C(CCC)OC)=O)CCN(C(C2CCCC2OC)=O)CC1C1CCCC1 C=Cc1ccc(C(=O)NC2COCC2NC(=O)C(CC(C)C)NC(N)=O)cc1 CC(C(=O)NCC1(C)CCN(C(C2(c3cc[nH]n3)CC2)=O)CC1)C(C)(F)F c1(N2CC(CNC(CNC(CCC(C)C)=O)=O)C2)ncnc2sc([N+](=O)[O-])cc12 C1(C2CC2)(C(N2CCC(COC)C2)=O)CN(C(=O)C(C)N=[N+]=[N-])C1 CCCCS(=O)(=O)NCC(=O)N(C)CCN(C(=O)C(c1cnn(C)c1)OC)C c1(C(N2CCC(CNC(C(CC)(CC)CC)=O)C2)=O)cnc2ccc(C)cc2c1 C(c1ccccc1C)=CC(N1CCC(N(C(CSC)=O)CC(C)C)CC1)=O N#Cc1cc([N+](=O)[O-])ccc1C1CCCN1C(=O)NCCCc1cccnc1 c1(C(=O)NC2C3C(C)N(C(=O)CO)C2C3)cc2c(cc1Br)OCCO2 c1(N(CC(C)CNC(=O)C(C)(C)C(F)F)C)nc2ccccc2cc1[N+](=O)[O-] C1(N(C(COC(CC)C)=O)CC)C2CN(C(c3cnoc3C3CCC3)=O)CC12 Cc1ccc2c(C(=O)NCC3CCN(C(C4(F)C(C)(C)C4(C)C)=O)C3)onc2c1 c1(OC)ccc(Br)cn1.c1(C2C(=O)OC2COC(C)(C)C)cnn(C2CC2)c1 CC1CN(C(=O)COCCCF)CC1C(N1CCC(C(C)(C)C)CC1)=O N1(C(C=C(C)C(F)F)=O)CCC(N(C(=O)CC2CCC(C(F)(F)F)O2)CCO)C1 c1(C(=O)NCC2CC(c3cc(Cl)cc(Cl)c3)C2)[nH]cc2c1CCCC2 C(=O)(C1=CC2(CCOC2)C1)NC(CC(C)NC(c1c(C)nc(CC)nc1C)=O)C C1(C(N2CCCCC(NC(CS(N)(=O)=O)=O)C2)=O)CCc2[nH]nc(O)c2C1 c1(C(N2CCC(N(C(c3c(SC)n(C)nc3)=O)C)C2)=O)cccc2ncnn12 CCCCC(C)C(=O)NCC1CC(O)(CNC(c2cnc(C(C)C)nc2C)=O)C1 N1(C(c2cc(COC)sc2)=O)CCCCC(NC(=O)C(C)(C)c2cccnc2)C1 c1(C(=O)NC2C(NC(C(C)SC)=O)CC2)ccc(O)cc1[N+](=O)[O-] CCCC(CNC(C1CC(=O)C1(C)C)=O)C(=O)NCc1cn(C(C)C)nn1 C1(NC(C2C(C)(C)C2c2ccccc2)=O)CCCN(S(N)(=O)=O)C1 C(CC1CC1)(C(=O)NC1CCSC1)NC(=O)CCC1CC1 C1(CC)CN(C(c2ccc(CNC(=O)C(=O)NC(C)C)o2)=O)C(CC)CO1 N1(C(CCCC(C)C)=O)CCCN(C(=O)COCC(C)(C)C)C(C)C1 C1(CC(=O)NCC(C)(C2CC2)NC(CC(C)c2ccncc2)=O)CC(C)(C)CO1 C(CC(CNC(=O)CCN(C)C(C)=O)NC(=O)C(CO)c1ccccc1)OC C(CCCOC)(C(=O)N(CCO)CCOC)NC(C(C=C)CC)=O C12(NC(=O)Nc3cc(Cl)ccc3Cl)CCC(CC1)N(C(=O)CCC(F)(F)F)C2 Cc1c(C(=O)NCCC(C)NC(c2sccc2F)=O)nn2c1CCCC2 C(CC1C(=O)N1)N(C)C(C1CC2(CSC2)C1)=O.c1(CN)cccc(C)n1.CO c1(C(N2CCC(CC(=O)NC(C34CCC(CC3)C4)C)C2)=O)ccc(O)nn1 CC(C)CC(CC(=O)NCc1nncn1C1CC1)NC(=O)C(C)(O)CC(C)C N1(C(C2(C3CCCCO3)CCC2)C)C(=O)CCN(Cc2csc(C(F)(F)F)c2)C1=O C1(CC(=O)N(C(CC)CO)C)CCCN(C(C2CCN(C)C2C)=O)CC1 N1(C(COC(CC)CC)=O)CC=CC(C(=O)NCC2(O)CC2)C1 C=CCCC(=O)NCC(CNC(c1cn(C2CCCC2O)nn1)=O)CO C=CCCC(O)Cc1ccc(NC(N2CC(C(=O)NC)C2)=O)cc1 c1(C(=O)NC)c(NC(C2CC3CC3N2Cc2cncc(CC)c2)=O)cccc1Br Cc1ccc(CC(=O)NCCC2(C(=O)NCC3CCN(C)C3)CCCC2)o1 C1(C(=O)N(O)Cc2cn(CC3CCOCC3)nn2)NCCC12CCC2 c1(CNC(n2ccc3ccccc23)CC)cccc([N+](=O)[O-])c1 c1(C(N(C2CCN(C(c3cn(CC(C)C)nc3)=O)C2)C)=O)cc[n+]([O-])cc1 C1(NC(C(CC#C)O)=O)CCCCN(C(=O)CC2CSCCO2)C1 C1(NC(CCCOC)=O)CCN(c2cc(-c3ccco3)nc(C3CC3)n2)C1(C)C C(=O)(CC(C(F)F)NC(c1ccnnc1O)=O)N1C(CC)CC(C)C1 C1(O)(CC=O)COC(C)(C)C1.C1(SCC)CCC(NC(C2CCN(CC)C2)=O)CC1 CC1CN(C(=O)CCCC2CCC2)CC(C)N(C(c2cc(N)cc(F)c2)=O)C1 N1(C(C(C2CCOC2)OC)=O)CC2(CCN(CC3CCCCCC3)CC2)C1 c1(C(=O)NC(C(=O)NCC(CO)NC(C)=O)C2CCCO2)cc(CO)oc1C C1(N)CCN(C(=O)CC(C)(C)N(C(=O)CCC2CC(OC)C2)CC)CCO1 C(C)(C)(CC(=O)N1CCOC(C2CN(C(=O)C(C)SC(C)C)C2)C1)SC C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NCC1C(NC(COC(C)=O)=O)CCCC1 C(=O)(CCC(F)(F)C(F)F)N1CC(NC(C(C(=O)OC)(C)F)=O)C1 N1(C(C(CCC)OC)=O)CC2CCC(C(=O)NCC3C(C)(C)C3(C)C)(C2)C1 C1(C(=O)NCC(CN(C)C(c2cnccc2Br)=O)O)C(F)(F)C12CC2 C1(C)(C(N(CCOC)CCNC(=O)Cc2nocc2C)=O)CC=CCC1 C1(NC(C(C)(C)OCC)=O)CC2CC(NC(c3ccccc3SC(F)F)=O)CC12 CN1CCN(C(=O)C2=CCSC2)CC1C(=O)NCC12CCC(CC1)CC2 C(=O)(C1=NOC2(CCOC2)C1)NCC12C(CN(C(CNC=O)=O)C1)C2 C1(C(=O)NOC2CCCC2)C2CN(C(=O)CC3CC4CC4C3)CC12 CCC(C)(CC)C(=O)NC12CC(CNC(c3cnn(C)c3N)=O)(C1)OC2C CCC(C(=O)NC(C)CC1CN(C(=O)CNC(=O)CCC(C)C)C1)C(C)C N1(C(c2sccc2Br)C(=O)Nc2ccc(OC)cc2)CC2CCC1C(O)C2O N1(C(CCC(C)SC)=O)CC(C)CN(C(=O)Cc2c[nH]c(=N)nc2O)CC1C C1(NC(C=CCNC(c2cnn(CC)c2C)=O)=O)CCC2(CCC2)C1 N1(C(CCCOC(C)C)=O)CCC2(CC1)CCN(C(C1CCCN1C)=O)CC2 C1(C)(CC(=O)N(CCOCCN(C(=O)C(C2CC2)C2CC2)C)C)CCCO1 CCCCC(C)(F)C(=O)N1CCC1Cn1cc(CN2CCS(=O)CC2)nn1 CCC(C(=O)NC1CC(NC(c2cc(O)nn2C)=O)C1)C(C)(F)F N1(C(CC(C)C)=O)CCC(CNC(C2CC2c2ccsc2)=O)C1(C)C c1(C(N2CCC(NC(Cn3nnc(C)n3)=O)C2(C)C)=O)nn2cccnc2c1Cl c1(C(=O)OCC(=O)Nc2ccc(F)cn2)ccccc1-c1nc(C2CC2)no1 S(=O)(=O)(c1ccc(Br)c(C(=O)OC)c1)N1CC=C(CNC)CC1 C1(C)(NC(c2c(C)cco2)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 C12(CNC(Cc3cccc(SC)c3)=O)CCCOC1CCN(C(=O)C(C)S)C2 N(C(=NCCF)N1CCC(c2cccnc2)C1)Cc1nc(COC)on1 Cc1cc(C(=O)NC2CCCN(C(C3(CO)CCCO3)=O)C2)c(Br)cn1 c1(NC)cc(C(=O)NCC=CCNC(c2occc(=O)c2OC)=O)cc(Cl)n1 C1(NC(=O)NC23C(C)(C)OCC2C3)CCc2c[nH]nc2C1 c1(C(C(=O)NC2COC2)N(C)Cc2ccncc2)cc(F)nc(F)c1F c1(C(N2CC=CC(NC(Cc3ccc(C)nc3)=O)C2)=O)c(C)oc(C)c1C c1(C(=O)NCCC(C)(C)NC(Cc2c(C)ncs2)=O)[nH]cc2c1CCCC2 N1(C(c2cc(C(C)(C)C)on2)=O)CCC2CN(C(N3CCC(O)CC3)=O)CCC12 c1(C2(NC(=O)NC3C(SCC)COC3)CC2)ccccc1F Cn1ccc2cc(C(=O)NCC3CN(C(C4CC4CN(C)C)=O)C3)cnc12 c1(C(C(=O)N(CC(C)C)CC(=O)NCC2SCCS2)=O)cccn1C C1(NC(C2C(C)C2)=O)CC2CC1N(C(C1(c3ccc(F)cc3)CCCCC1)=O)C2 c1(CC(=O)OCC(=O)N(CCC#N)CC)ccc(F)cc1CC c1(NC(C2(CNC(CC(C=C)c3ccccc3)=O)CCC2)=O)ccc(N)c(O)c1 c1(C(N(C2CN(C(C3CCC(C)(CC)O3)=O)C2)C)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(C(COCC)C)=O)Cc2[nH]nc(C(N3CC(CC)OC(C)C3)=O)c2C1 CC1(CNC(=O)Cc2ccc(CO)cc2)CCCN1C(c1ccsc1Cl)=O Cc1cc(C(=O)NCC(C)NC(=O)CC(C)(C)C#N)cc(C)c1F C1(CCN(c2ncc(Br)s2)C)CC2CC1C1CCCC21 c1(C(=O)NCC2C(NC(c3c(CCC)nco3)=O)CC2)cc2cccc(C)c2[nH]1 C1(NCC(=O)NC(C(=O)N(c2cccnc2)CC)c2ccoc2)CCC(C)C1 C1(NC(=O)NCCSC)COCCC12CN(C(=O)OC(C)(C)C)C2 N1(C(CCC=CC(C)C)=O)CCC(C(=O)NCCc2ocnc2CO)C1C CC(C)(C)CCCCC(=O)N1CC=C(CCNC(C2CN3CCC2C3)=O)CC1 C1(CNC(CNC(C)=O)=O)CC(NC(=O)CSc2ccc(Cl)cc2)C1(C)C c1(C(N2CC(C(C(=O)NCC#CCCO)OC)C2)=O)ccc(C#N)n1C c1(N2C(C)(C)CC(C(=O)O)CCC2)ncnc2c([N+](=O)[O-])cccc12 c1(OC)cccc2sc(NC(CN(C)C)CC(C)C)nc12 C1(NC(C)=O)CCN(c2cc(C)nc(CC3(O)CCCC3)n2)C12CCCC2 C(=O)(C(C)CCCCCC)NCCC1CC(C(=O)NC(CC(=C)Cl)CO)C1 c1(C(=O)NCCC(C)(CC)NC(C(CC)OC)=O)cnc(OC)nc1C(F)F c1(OC)ccc(-c2ccc3c(c2NC(=O)CCS(C)(=O)=O)OCO3)c2cn[nH]c12 N1(C(c2ccc(CC)cc2)C(=O)NC(C)C)CCCN(c2ccccc2C)CC1 Cc1[nH]nc(C(=O)NC2CCC2CNC(c2ccc(CO)c(Cl)c2)=O)c1[N+](=O)[O-] C1(NS(CC)(=O)=O)CC2(C1)CN(C(c1ccnc(Oc3cccc(Cl)c3)c1)=O)C2 CCCCCCCCC(=O)N1CCN(C(C2CC3(C2)CC(CO)C3)=O)CC(C)C1 c1(OC)n[nH]cc1C(=O)N(CCCNC(C1CCC1C(C)(C)C)=O)C N1(C(c2onc(COC)n2)=O)CC2(C1)SCCC2NC(c1csc(O)n1)=O N1(CC(CCC(=O)OCC)CC)CCn2c(C(F)(F)Cl)nnc2C1 n1(CC)cc(CNC(=O)NC(C(F)(F)F)c2ccccc2)c(C)n1 C=Cc1cncc(C(=O)NC(C2CCN(C(C3CCC(C)(C)CO3)=O)CC2)C)c1 c1(CC(=O)N(CC(C)NC(c2ccnc(F)c2F)=O)C)cc(F)cc(F)c1 S(=O)(=O)(c1nc(NC2CCc3c(n[nH]c3C)C2)ccc1Br)NC(C(CC)CC)C C1(C(=O)NCCCCCNC(c2c(C(=O)OC)n[nH]c2)=O)CCCN(C(C)=O)C1 c1(C(=O)NC2C(C)(C)C(CNC(=O)Cc3cnccc3Cl)C2)cc2sccc2[nH]1 c1(C(=O)NCC(CCNC(Cc2cc(C)sc2)=O)O)cc2c(Cl)cccn2n1 C(=O)(CCCCCC#N)NC(c1cccnc1)C(=O)NCc1ccc(OC)nc1 C1(O)(CCNC(C2COCCO2)=O)CN(C(C2CC2c2ccc(Cl)s2)=O)C1 CC(C)CC(O)C(=O)NCC1CC2CC2N1C(c1cc(C(C)C)nn1C)=O C1(CNC(=O)NC(COC)C)CCC=CN1C(=O)OC(=O)CN(C)C N1(C(c2cn(C)nc2)=O)CCCCC(NC(=O)CNC(C2CCC2)=O)CC1 C1(CC)CN(C(C2(c3c(C)cccc3Cl)CC2)=O)CCN1C(=O)C(C)CC(N)=O C(CNC(c1cc(Cl)nnc1O)=O)(CC(F)(F)F)NC(C1(CC#C)CC1)=O C1(C(C(=O)OC)F)CCN(C(c2cnn(CCN)c2)=O)C1 C(=O)(C(F)(F)C(C)(C)O)N1CC(CCC)N(C(=O)CSCc2cccnc2)CC1 C1(C(=O)NC(C)C(C)(C)CO)CCCCCN1C(=O)CCCN(C)C C1(NC(c2n(CC)ncc2)=O)COCCN(C(=O)C(C)S)C1 c1(C2C(C(=O)NC(=O)C(=O)NC3CN(CC(F)F)C3)C2)ccc(Br)c(Cl)c1 N1(CCC(=O)NC(CCN(C(C2N(CCC)CCC2)=O)C)C)CCNC(=O)C1 C1(C(=O)NC2CC(=O)N(C)C2=O)COc2ccc(F)cc2C1 N1(C(c2c(C)nc(C3CC3)o2)=O)CCCC(C2CC2NC(c2ccn(C)c2)=O)C1 Cc1c[nH]c(C(=O)NCCC2(C(=O)NCC(C)(C)CO)CC2)c1C C(=O)(C1=CC(O)C(NC(=O)CC2CC(C)(C)CO2)C1)N(C(C)CO)CC C1(C(=O)NC2CCCC2CNC(c2cnc(Cl)s2)=O)(COC)CC1(F)F c1(N(C2CCC(C)(C)CC2)C)nc(=N)[nH]c(=NC(CF)c2ccccc2)[nH]1 C1(NC(C2C(CCC)CN(C(=O)C=CCF)C2)=O)(CO)CCN(C)CC1 Cc1nc2ncnn2cc1C(N1CC(CCCCNC(c2cscc2Cl)=O)C1)=O Cc1oc2cc(C(=O)N=S(C)(=O)CCC3(C)CNC3)[nH]c2c1C N1(C(Cc2ccc(C)s2)=O)CC(N=c2[nH]cnc3cnn(C)c23)CC2(CCC2)C1 C(=O)(CC(C(C)=O)OC(c1cccc(-c2nnc(C)o2)c1)=O)OCC C1(C(N(CC(CC)C)C)=O)(CCOC)CCN(C(c2ncc(C)cc2C)=O)CC1 C1(NC(c2c(CC)n[nH]c2)=O)CCCCC1NC(c1cnn(C)c1CC)=O c1(NC(C(N2CCC(NC(=O)OC(C)C)CC2)=O)=O)cc(Cl)c2nncn2c1 CCC(C)(COC)C(=O)N1CCC(CNC(=O)C(C2CC2)N(C)C)C1 C(CC1CCCC1)(C(=O)N=c1ccn(CCO)[nH]1)NC(c1cc(CC2CC2)on1)=O C1(NC(c2c(C)nc(C)[nH]2)=O)CCCC(NC(=O)CC2CC=CC2)CC1 C1(C(=O)NC(C(C)C)C(C)NC(=O)C=Cc2ccnn2C)CCC2(CC1)CC2 CCN=c1[nH]c(C(N2CCCC(C)(CNC(C3CC3CCOC)=O)C2)=O)cs1 N1(C(C(CC)CC)=O)CCC2C(CCCN2C(c2c[nH]c3cc(Cl)ccc23)=O)C1 C(=O)(CCC(N)CO)Nc1cc(C(=O)NC)ncc1 Cn1ncc2ncc(-c3nc(CCN(C)C)nn3Cc3ccccc3F)cc12 C(=O)(C(C)(C)CC(C)C)N1CC(CC(C(=O)NCCC(C(C)C)OC)F)C1 C(c1ccc(C(F)F)o1)=CC(=O)NC(C1CCN(C(C2CCCC2)=O)C1)C C1(C(=O)NCc2cn(C3CCN(C(CN(C)C)=O)CC3)nn2)CCC2(CCC2)C1 c1(CC(N2CCCC(N(C(Cc3ccc(C)s3)=O)CCO)C2)=O)cc(Cl)ccc1O c1(C(C(=O)NCC(C)CN(C(=O)Cc2cscn2)C)C)cncnc1 C1(C(=O)NCc2c(CC)nco2)CN(C(=O)CC2CN(C(C)=O)C2)CCC1(C)C c1(NC(=O)Nc2ccccc2)c(C#N)nc(Cl)c(Cl)c1Cl.C12CC1CN(C)C2=O C1(CNC(=O)Cn2cc(CC3(O)CCOCC3)nn2)CCC2(CCC2)CO1 C(=O)(C(CCc1ccsc1)NC(c1c[nH]cc1CC#N)=O)OC c1(C(N(CCOC)CCNC(c2c(C)ccn2C)=O)=O)cc(C)nc(O)n1 C1(CNC(c2cc(C)no2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1C c1(C(=O)NC2C3(CCN(C(CCCCC#C)=O)C3)C2)sc2[nH]cnc(=O)c2c1C Oc1ncnc2c1CCN(N1CCCC(c3ccc(O)cc3)C1)C2 N1(C(CCC(C)C)=O)CCN(C(C2(c3cccs3)CC2C)=O)CC2(CC2)C1 Cc1cc(CC(=O)NC2CC2NC(=O)Nc2ccccc2C(F)(F)F)ccn1 c1(C(N(C2CCCN(C(=O)CC3CCCCO3)C2)CC)=O)cnn2c(C)cccc12 n1(CC)ncc(Cl)c1C(=O)NC1CCC(N2CCN(C(=O)C3=CCC3)CC2)CC1 C(=O)(C(CC)C(=O)NC1CCCN(C(=O)CSCc2cccs2)C1)OCC C(C(C)(C)C(=O)Nc1cccc(C(=O)NC2COCC2COC)c1)SC CCCC(CC)C(=O)NN(C(C1(NC2(F)CCCC2)CC(CO)C1)=O)C C#CCC(C(=O)NCCC1CCCN(C(c2nnccc2C)=O)C1)C1CC1 C1(C(=O)NC(CC#C)C(=O)NC)C2CC3C(C2NC(C2CCS2(=O)=O)=O)C13 N1(C(C(=O)NCCCC)C2CC2Cl)CCOc2c(C(=O)OC)cccc2C1 N1(C(C2N(C(C)=O)CCC2)=O)CCC(NC(c2nnccc2C)=O)C2(CCC2)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CCCC2CN(C(c3sccc3F)=O)CCC12 c1(C2(C(=O)NC3C(OC(CC)C(=O)OC)CCCC3)CC2)ccc(N=S(C)(C)=O)s1 c1(CNC(C(N2CCCC(C(=O)OCC)C2)=O)=O)oc2ccccc2c1Cl CCCCC(CC(=O)NC(C1(O)CCCC1)(C)C)NC(c1cc(Cl)no1)=O c1(C(=O)NCC2N(C(C34CC(OC)C3C4)=O)CC2)ccc(O)c2c1CCCC2 C1(CC(=O)NC2CCN(C(c3c(CCC)n[nH]c3)=O)C2)(OC)CCCCC1 c1(C2(C(=O)OC)CC2)cccc(NC(=O)Nc2nc(-c3cccc(Cl)n3)cs2)c1 C(C(CCCC)NC(C1CN(C2CCOCC2)C1)=O)N(CC=C)C(C)C C12(OC)CCC(C(N3CCC(C(C)NC(=O)CC4CC(=O)NC4=O)C3)=O)(CC1)C2 c1(C(N2C(CC(=O)Nc3cc(N(C)C)ncn3)COCC2)=O)cc(Cl)ccc1Br C1(NC(c2cc(-c3ccc(Cl)cc3)ns2)=O)C2CN(C(=O)CC3CCCO3)CC12 N1(C(COCC)=O)CCCC(C2CN(C(=O)C=C(C)c3cccs3)C2)C1 C(=O)(C(O)CC(C)(C)C)N1CC(CCCC)N(C(=O)Cn2ncnn2)CC1 N1(C(=O)CC2CCC2)CC(C2CN(C(C3CC34CC(F)(F)C4)=O)C2)C1 N1(CC(=O)N(CC(CC)NC(C2CCS2(=O)=O)=O)CC)CCC(=O)NC1=O C1(Cc2cn(CCC=C=C)nn2)CN(C(c2cnc(C)cn2)=O)CCO1 N1(C(CCCN(C(C)=O)C)=O)CCCCC1CCN(C)C(C1CC1CN(C)C)=O N1(C(C2(C#N)CC3CC3C2)=O)CC2COCC(C1)C2NC(=O)C(F)=C1CCCC1 C(=O)(C(CCC)CCC(=O)OC)NCC(CNC(CCCCCSC)=O)(C)OC c1(C(=O)NC(CNC(C(C)C2CC2)=O)C2CCC2)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NCCN(C(c2cccc(O)c2)=O)CC)csc(N=S(C)(C)=O)n1 N1(C(C(C)O)=O)CCCC(C(=O)NCCc2cnn(C)c2)CC1 C1(C(N2CCCCC2CO)=O)CSc2ccccc2O1 CC1CCCN(C(=O)CC2CN(C(C3CCO3)=O)C(C)(C)C2)CC1 Cc1nc2c([nH]1)CC(C(=O)NCCC1CCCN1C(=O)C(C)OCC(C)C)CC2 CCC(O)C(F)(F)C(=O)NCC1CN(C(=O)CC(COC)COC)CC1(C)C C1(C(N(C)CC2CCN(C(c3coc4c3COC4)=O)C2)=O)OCC2COCCC12 c1(C(=O)NCCC(=C)CNC(C2CC2CC(C)C)=O)ccc2nonc2c1 c1(C(N(CC(C)CNC(=O)C(=O)NCC2CC2)C)=O)cn2c(n1)CCC2 c1(C(=O)NC2CC(C(C)NC(Cn3ncc(CC)c3)=O)C2)n[nH]cc1[N+](=O)[O-] c1(C(N(CC(C)N(C)C(c2ccc(N)cn2)=O)C)=O)cccn2nnnc12 C1(CNC(C2(CC=C)CC=CC2)=O)CN(C(=O)CSCC)C2CCN1C2 c1(C(N(CCCNC(C2C3CC4C(C3=O)C24)=O)C)=O)ccc2cnnn2c1 N1(C(=O)Cc2ccccc2)CC2(C1)CN(C(C1(Cc3cccc(F)c3)CC1)=O)C2 c1(CCC(=O)N(C)CC2(O)CN(C(C3C4CNC(=O)C34)=O)C2)cc(F)cc(F)c1 Cc1nn(C)cc1-c1ccc(C(N2CCN(C(C)(C)CO)CC2)=O)cc1 Cc1cc(C)c(C(=O)NC2CC(CNC(=O)CCn3ncn(C)c3=O)C2)cc1C C1(C(=O)NCC=O)CC12CN(C(=O)NC)C2.c1(C2CC2)ccn(C2CCCCO2)n1 N1(C(CCN(CCCCC)C)=O)CCC(C2(NC(=O)CCCNC(C)=O)CC2)C1 Cc1cc(C(=O)NCC2CCC2NC(c2ccnn2CCF)=O)ncc1N C1(CCCC)CN(C(C2CC2C2CC2)=O)CCN1C(=O)Cc1csc(Cl)n1 C1(C(=O)NC(C(CO)NC(c2nc(C)sc2)=O)C)CCC(C)(C)OC1 c1(C(N2CCCC2c2cc(C)nn2C)C(=O)NCCC)sc2ccccc2c1C N1(C(CN(C(=O)CN2CCC(OC)C2)CC#C)=O)CCC2(CCOC2)CC1 Cn1ncc2c1CC(C(=O)NCC(C1CCC1)NC(C1C3COCC13)=O)CC2 N1(C(c2c(C)n(C)nn2)=O)CCN(C(=O)CCOCc2ccccc2)C(C)C1 c1(C(=O)NC(C(C)NC(c2ccc(CC)[nH]2)=O)C)ccccc1CC#N c1(C(=O)NC2C(NC(c3cccc(SCC#N)c3)=O)C2)cc(O)cc(=O)o1 Cc1ccc(C=CC(=O)NC2CC2NC(C2CCC(OC(C)C)CC2)=O)c(C)c1 CC1(C)CC(C(=O)NC2CCN(CC3CC=CCC3)CC2)N(c2ncccn2)C1 CCC(CN1CCC1C(=O)NCCn1cc(C2CCN(C)C2)nn1)CC N1(C(C=NOC)=O)CCN(C(c2cc3c(s2)CCC3)=O)C(C(F)F)C1 Cc1nc2ccccn2c1C(N1CCNC(CO)C1)=O N1(C(c2cnn(C)c2F)=O)CCN(C(C2CCN(CCF)CC2)=O)C2CC12 N1(C(C(CC=C)C(C)C)=O)CC=C(C(C)(C)C(=O)N2CC3CC(C2)C3(C)C)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CCCN(C(=O)Cn2cncn2)CC1 c1(CNC(C2CCC(n3cc(CC4CCC(=O)C4)nn3)C2)=O)cc(F)ccc1Cl C(=O)(CC(C(C)C)NC(=O)CCc1ccco1)NCC(C=C)O CCC(CCC(=O)NCC1CC(NC(=O)Cc2cccc(O)c2F)C1)OC c1(C(=O)NCC2CC(F)(CNC(C3CCN(C)C3=O)=O)C2)cccc2sncc12 C1(CNC(CS(CC)(=O)=O)=O)CC2OCCC2N1C(c1ccc(C)c(C)c1)=O N1(C(CS(C)(=O)=O)=O)CC(NC(=O)CCCCc2ccccc2)C(C2CC2)C1 CCCC(O)C(=O)N(C)CC1CCN(C(C2(C)CCSCC2)=O)C1 c1(C(=O)OC)nc(=NCC2(C)CCCN(C(=O)C3=C(Cl)CC3)C2)c2c([nH]1)CCC2 C12(CCNC(C(C)(C)NC(C)=O)=O)CCC1CN(C(c1c[nH]c(=N)nc1C)=O)C2 N1(C(CC2CCC(C)C2)=O)CCC2(CC1)C(NC(=O)CC1CN(C)C1)CS2(=O)=O Cn1c(CCC(=O)NC(CC2CC2)C(=O)NC(c2ccccc2)CF)nnc1S c1(C(C)=O)cn(C)nc1C(=O)NCC1CC1CNC(=O)C=Cc1cocn1 C1(C(C)(C)O)CCN(S(=O)(=O)N2CCC(CC3(O)CCOCC3)C2)CC1 c1(C(=O)NCC2CC(NC(CC3C(C)OCC3)=O)C2)ccc2oncc2c1 C(=O)(CCN(CCO)C(C1CN(C2COC2)C1)=O)N(CCOC)C c1(CN2C(C(=O)Nc3cccc(C(=O)OC)c3C)C=CC2)c(O)ccc(Br)c1O C1(CNC(CCc2cc(C)[nH]n2)=O)CC(NC(=O)C=Cc2scnc2C)C1(C)C c1(OCC)ccccc1C(=O)NC(C)(C)CCCNC(=O)C(CC)OC c1(C(=O)NC23CCC(NC(CCCC#C)=O)(CC2)C3)ccc(F)c(S(C)(=O)=O)c1 c1(C(=O)NCCCCNC(c2cnncc2C(F)(F)F)=O)ccc(O)c(Cl)c1 C1(O)(CNC(=O)C=C2CCCC2)CC(CNC(c2ocnc2C(F)(F)F)=O)C1 N1(C(C2C(CC(C)(C)C)C2)=O)CCCCCC(NC(=O)CC2CCC(=O)O2)C1 C#CCC(CC#C)C(=O)NC1CN(C(C2(SC)CCC2)=O)CC1N1CCCC1 C(C(COC)CC(=O)NC1CC(O)CN(C(=O)CCCc2cnccn2)C1)OC c1(C(=O)NC2CN(C(c3ccnc(C)c3O)=O)CC(O)C2)ccnc2c1CCC2 c1(CNC(c2cc3cc(Cl)ccc3o2)C)c(Cl)c[nH]c2nccc1-2 C(=O)(C1=C(Cl)CCOC1)NCC12N(C(CCOCCN(C)C)=O)C(CC1)CC2 N1(CC)CCC(N(C(=O)CCCn2cc(C(=O)OC)nn2)C)C(C)C1 c1(C(N2CCN(C(c3ccn(C(C)(C)C)n3)=O)CC2)=O)cc2[nH]ccc2s1 C(=O)(C(F)(F)CC1CC1)N(C1CCN(C(C2CCCCC2C)=O)CC1)CC C#CCCCCC(=O)NC(C)CNC(C1(OC)CS(=O)(=O)C1)=O C1(CC(=O)NCCCC2CCC(NC(C3(CC#C)CC3)=O)C2)CCC(C)(C)CO1 c1(NC(C2N(C(C)=O)CCC2)=O)ccc(F)c(NC(C2OCCOC2(C)C)=O)c1 C1(CNC(C=CCOC)=O)(NC(=O)C(c2ccccc2F)C)CCCCC1C CC1CN(C(=O)CCc2cncs2)CC(C)N1C(=O)CC1CCCCCCC1 S(=O)(=O)(c1cnc(NCCOC(F)F)c(Cl)c1)NCC1CCCC(C)C1 N1(C(COC(C)C)=O)CCOCC(CNC(=O)CCc2ccc(Cl)c(F)c2)C1 Cc1ccc(CS(=O)(=O)NC(=O)Cc2cccc(N3CCCC3=O)c2)c(C)c1 C12(NC(c3cn(CCNC(CC4CC(OCC)C4)=O)nn3)=O)CCC(SC)C1C2 c1(SCC=C)ccccc1C(N1CC(NC(c2cnccc2NC)=O)C(O)C1)=O Cc1oc(CCC(C)C)nc1C(N1CCOC(CNC(=O)C=CC2CCC2)C1)=O N1(C(CC(C)C2CCCO2)=O)CC(C)(C)OC2(C1)CN(C(c1cc[nH]c1)=O)C2 CCC(C)CC(C)N=c1[nH]c(N2CCC3(CCC3)C2)nc2c1CCCCC2 C1(CC(=O)NCC(c2nccs2)C)CCCN(C(C2(C)CCOCC2)=O)C1 c1(C(=O)NC(CN(C(C(CC)N(C)C)=O)CC)C)sc(C)nc1C(F)(F)F Cn1cncc1C(=O)NC1CC(CNC(=O)Cc2csc(N3CCCC3=O)n2)C1 Cc1noc(C)c1-c1cn(CC2COCCN2C(C2(C)CC(C#N)C2)=O)nn1 Cn1ncc(C(=O)NC2CN(C(C3(O)CCC3)=O)CC3(CC3)C2)c1S(C)(=O)=O c1(C(N2CCCC(NC(COCCCCOC)=O)C2C)=O)ccn2nccc2n1 C1(NC(Cc2c(C)ocn2)=O)C(C)(C)C(NC(=O)C(O)CC2CCCC2)C1(C)C c1(OCCCOC)ccc(C(=O)NC(C)CCNC(=O)CCC=C(C)C)cn1 C(C1=CCN(C(=O)CCc2nc(C)c(C)o2)CC1)NC(c1c(SC)cccc1)=O C1(NC(C(CCC)O)=O)COC2C(NC(=O)C=CSc3nc[nH]n3)COC12 C(c1ccccc1C(F)(F)F)=CC(=O)NC(CSCC)C(=O)NC C1(NC(C(CC#C)NC(c2nn(C)cc2C)=O)=O)CC(C)N(C)CC1C C(=O)(C1Cc2ccc(Cl)cc21)NC(C(C)NC(=O)CCCCc1cnn[nH]1)CO C#CC1(C(=O)NC2CCC(C3CC3)C2)CCN(C(c2cnc(N(C)C)nc2)=O)C1 Cc1cc(C(=O)NCC(CNC(c2cscc2Cl)=O)CO)nc(O)n1 C1(NC(C(C)OCC2CC2)=O)CN(C(c2cc(F)cc(F)c2O)=O)CC(F)(F)C1 C(=O)(C(O)P(C)(C)=O)NCC(C)(C1CC1)NC(CCC(C)C)=O C1(NC(C(C)C2CC2)=O)Cc2ccccc2C1NC(c1cnsn1)=O C(=O)(CCC(C(=O)OC)NC(=O)CSCCn1cc(C)cn1)OCC c1(C(=O)NCCCNC(CCC2(C(C)(C)C)CCCO2)=O)cccc(CCO)c1 n1(C(C)C)cnc(C(=O)NC2CC(CNC(=O)OC(C)(C)C)C2)n1 c1(OC)cc(-n2nc(CO)nc2C2CCCN(CC(F)(F)F)C2)ccc1F C1(CC(N2CCC(CF)C2)=O)(NC(=O)C(O)CC2CCCC2)CCCCC1 C(=O)(CC1=NNC(=O)C1)NCC1CN(C(c2nc(CC)sc2)=O)C(C)CC1 C=CC1(C(=O)NC2(CCCC(=O)NC3CCC(F)C3)CCC2)CCC1 c1(C(=O)NC2C(CNC(c3ccc(C(N)=O)[nH]3)=O)CC2)[nH]cc2c1CCCC2 c1(OC)ccc2oc(C(=O)O)cc2c1.C1(COCC2CC2)CC12CCOC2 N1(C(c2scc(C)c2C)=O)CCC=C(C(=O)N(C)OC2CCCC2)C1 CC(C)(C)CC(O)CC(=O)NCCCN(C(=O)CC(F)(F)F)Cc1ccccc1 C1(C(=O)NC(C)CN(C(=O)CSC(F)(F)F)C)CN2CCCCC2CO1 C1(C(=O)NC2(C(C)C)CCC2)C2CCC(C2)N1C(=O)CC(C)F c1(C(=O)NC2C(CNC(C(C(=C)Cl)(C)C)=O)C2)ccc(S(=O)CC#N)cc1 C(=O)(C#CC1CCCCC1)N1CCC(CC(=O)NCC(N2CCCC2)=O)C1 C1(C(=O)NCC23CC(NC(c4scc(OC)c4OC)=O)(C2)C3)CC2CC2CC1C C12(NC(CSCC(C)C)=O)CCN(C(c3ccccc3C#N)=O)CC1C2 N1(C(COCC#C)=O)CCC(C2CCN(C(=O)CCC(C)(C)C)C2)C1 N(C1CCCn2nccc21)C(Cn1c(C(C)OCC)ncc1)=O CC(O)CCCC(=O)NC(C)CCNC(=O)C1=NNC(=O)C1 C(=O)(CC(=O)NC1COCC1CN(C)C)NCCC1C(C(=O)OC)C1 Cn1cc(CC(=O)NC2(CCCNC(C3(C)CC=CC3)=O)CC2)nn1 Cc1cc(N2CCC(C(C)NC(=O)CC(C)C(F)(F)F)C2)ccc1[N+](=O)[O-] c1(NC(C2CCN2C(=O)CSc2ccc(Br)cn2)=O)nc2ccccc2s1 C=C(Cl)CC(C(=O)NCCN=[N+]=[N-])NC(=O)CCNC(N)=O c1(OCC)ncc(NC(C2CC(OC)CN2C(c2c[nH]c(=N)s2)=O)=O)cc1C Cn1ncc2c(N3CC4(CC4)CC3CNC(C3(C(F)F)CC3)=O)ncnc12 c1(OC)cc(C(=O)N(C)CCOCCNC(c2sccc2OC2CC2)=O)ccn1 c1(C(=O)NCc2cccc(NC(C3C(C)COCC3)=O)c2)ccc(F)c(N)c1 c1(CN(CCNC(C2CC2c2ccccc2)=O)CC)nc2cnccc2s1 N1(C(C(c2ccccc2Cl)C)=O)CCC(C(C2CC2)NC(=O)C=CC2CCC2)CC1 N1(C(CC2N(CC)CCOC2)=O)CC(O)(C2(CNC(=O)CNC(C)=O)CC2)C1 C1(NC(C(COC)COC)=O)CN(C(=O)COc2ccn(C)n2)C(C)(COC)C1 N1(C(c2cc(OC)ns2)C(=O)NCCCSC)CCS(=O)(=O)C2(CCCCC2)C1 O=C(CCCS(=O)(=O)N1CCCC1)NCC=CCNC(=O)CC1CCOC1 n1(C(CC)C)nc(C(N2CCC(CNC(=O)CC(C)(O)C3CC3)CC2)=O)cc1C CC1CN(C(C2CCC2C)=O)CCCN1C(c1ccc(-n2ccnn2)cc1)=O O=C(CC1=CCOCC1)NCC1CN(C(=O)CCc2ccncc2)CCO1 CC1CCCn2ncc(C(=O)NC3CCCCN(C(=O)CCc4ccco4)C3)c21 N1(C(c2c(C)cccc2)=O)CCC2(CC(C(=O)NCCCCCO)=NO2)C1 C(=O)(C(C)(C)Cn1cc(-c2nccnc2CO)nn1)NC(CC)COC N1(C(Cc2ncn(C)c2)=O)CCCCC1CCNC(=O)CCC1CCCOC1 Cn1ncc(CNC(=O)Cn2ccnn2)c1C(=O)NCc1cn[nH]c1 Cc1ccc(CCNc2ncccn2)c(Br)c1 c1(CNC(=O)NCC2(C(F)(F)F)CCC2)cccc(F)c1Sc1ccccc1 N1(C(CCOCC)=O)CCC(NC(c2cc(C(=O)OC(C)(C)C)c(C)o2)=O)CC1 C1(C(N2CCC(=C)CC2)=O)CC2OCCC2N(C(C2CCC(F)(F)C2)=O)C1 Cc1ccc(C(=O)NC(C)CCCNC(C2CC2c2cnc[nH]2)=O)c(N)c1 Cc1onc(C(=O)NCC(C2CCC2)NC(=O)CC(F)(F)F)c1[N+](=O)[O-] C1(N(C(C(C)OCC)=O)CC)CCCN(C(c2ccnn(C)c2=O)=O)CC1 N1(C(N2C(C)(CC)COCC2)=O)CCc2nnnn2CC1 C(CC(=O)NC(C(=O)N(CC(O)COC)C)c1cccs1)OCC C(CC(F)F)(C(=O)N1CCC2(CCO2)C1)NC(C1CC(CC2CC2)C1)=O C1(C(=O)NC(CN(C(c2cnn(C3CCC3)c2)=O)CC)C)CCCN1C c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)Cc2ccco2)cc2ccccc2o1 O(NC(=O)CS(=O)CC)CC(=O)NC1CN(CC)CC1C c1(CC(=O)NCCC2CN(C(CC3C(C)OCC3)=O)C2)ccn2cncc2c1 c1(C(=O)NCCC2(O)CCN(C(CC=C(C)C)=O)CC2)cc(O)ccc1[N+](=O)[O-] n1(C(C)C(=O)NC(C)(CNC(=O)Cn2cccn2)C2CC2)cnc(C#N)n1 C1(O)(C(C)NC(c2ccc(SC)s2)=O)CCN(C(=O)C=CC(C)(C)SC)CC1 c1(C(=O)NC(C2CCCN2C(=O)C=C(Cl)Cl)(C)C)cccn(C2CCSC2)c1=O N1(C(C2CN(C(=O)NC)C2)=O)CC2CC(N3CCCC(C)(O)C3)C1C2 c1(OC)ccc(CCC(N2CCCCC2C(=O)NCC#N)=O)cn1 c1(C(=O)NC(CNC(C(CC)(C)CO)=O)C)ccc(NC(=O)OC)c(C#N)c1 CCCCCC(O)C(=O)N1CCCC(C)(C(=O)NCC2CCS(=O)(=O)CC2)C1 C1(C(=O)NC2C(NC(=O)COCc3ccncc3)CCC2)Cc2cscc2C1 C1(NC(c2c(OC)scc2)=O)C2CCN(C(=O)C=Cc3nc(C)cs3)CC12 C1(C(=O)NCC(C)(O)CNC(=O)CCCN2CCCC2)CCOC2(CCCC2)C1 c1(-c2cc(NC(c3cnc(OC)c(C)c3)=O)ncc2)cccc(C#N)c1F c1(NC(Cc2ccc(OC)cc2C(F)(F)F)=O)cc([N+](=O)[O-])c(N(C)C)cc1F C1(C2CCC2)(C(=O)NC2CN(C(C(c3cn(CC)nc3)=O)=O)C(C)C2)CC1(F)F c1(C(=O)NC(C)CC2CN(C(c3c[nH]c(C(C)(C)C)n3)=O)C2)ccc(Cl)nn1 C1(NC(=O)C(c2cc(Br)c(Cl)s2)N2CCCC2Cc2ccsc2)CCC(F)(F)CC1 N1(C(CSCCC(C)C)=O)CC(C(=O)N(CC2=CCCOC2)C)C(CO)C1 c1(NCC(N(C(c2c(C)scn2)=O)C)C2CC2)nc2c(cc1C#N)CCCC2 CC1CCN(C(=O)CN(C)S(N)(=O)=O)C1CNC(=O)CCC=CBr Cc1nnc2n1CC(C(N1CC(CNC(=O)C3=C(C#N)CCC3)C(C)C1)=O)CC2 C1(C(N(CCC(N2CCC(C)(N(C)CC)C2)=O)C(C)C)=O)CC2(CCO1)CC2 Cc1ccc(C(=O)NCC2CCCC(NC(c3coc(C4CC4)n3)=O)C2)nc1 C1(C(=O)NC(CC)CN2CCCC2)CN(C(C2(CC)CCCCO2)=O)CC1(F)F C1(CC(=O)N(CCCOC)C)CN(C(C2CCC2)=O)C(C)(C)C1 C(CC(=O)NC1C(C)(C)C(NC(C2(C)COC2)=O)C1(C)C)(C(F)(F)F)OC C1(c2ccno2)(C(=O)NCC(C)N(C(C(CC)SC)=O)CC)CCOCC1 c1(NC(C2C(CC)CCN2C(=O)C(C)OCCOC)=O)ccc(O)c(Cl)c1 C(=O)(C(C)C1=CCCC1)NCC(F)(F)F.c12c[nH]nc1NC(=O)C1CC(C1)C2C c1(C(N2CCC(C(=O)NCCCc3ccccc3Cl)C2)=O)n[nH]c2c1CCC2 C(CCC(=O)NCC1CC1CNC(=O)CCc1cnn[nH]1)SC c1(OC)cc(C=CC(=O)NC(C)CNC(c2cncc(C(F)(F)F)n2)=O)ccc1O c1(C(=O)NCC=CCNC(CC2ON=C(C)C2)=O)ncc(Br)cn1 N1(C(C(CC)C)=O)CC2CCCC2(CNC(C2(CO)CCC2)=O)C1 CC1CCCCC1(CO)NC(C12CC(CN1C(=O)CN1CCC(F)CC1)C2)=O Cc1nc2ncccn2c1C(=O)NCC1CN(C(c2ccc(Br)c(O)c2)=O)C1 n1(CC)nnc(C)c1CN1CCC1CNC(=O)Nc1cnn(C(C)(C)C)c1 C1(CNC(c2cccc(C(N)=O)c2)=O)CN(Cc2ccc(F)cn2)CCCO1 c1(SC)cc2ccc1N1CC2C1.c1(C(=O)Nc2ncsc2Br)nnnn1C1(C)CC1 c1(C(=O)NCC(CNC(c2cc(C)sc2)=O)C)ccc(Cn2cncn2)cc1 C(=O)(CS(=O)(=O)C1CCCC1)NCC1N(C(CC(CC)CN(C)C)=O)CCC1 C(=O)(C1CCc2nccn21)NCC1(F)CCN(C(CC(=C=C)C)=O)C1 C#Cc1cccc(C(=O)NC2(CNC(c3ccsn3)=O)CCC(C)(C)CC2)c1F c1(C(=O)NC2(C)CN(C(c3cnn4c3OCCC4)=O)C2)cc2sc(F)cc2[nH]1 CC(F)(C(=O)N1CCC(CNC(=O)C=CCO)C1)C(F)(F)F N1(C(c2cc(OCC)n[nH]2)=O)CC(NC(C2CC2F)=O)C(CC)C1 C(=O)(C(C#N)C(C)(C)C)NCc1occ(C(N2CCC(CC=C)C2)=O)c1 Cc1cccc(C(=O)NC2CCCN(C(=O)COc3ccc(F)c(Cl)c3)C2)c1F C=CC1CN(C(=O)CNC(=O)CC2CCCC2)CC1NC(=O)CCC(C)OCC C1(C(N2C(C)CS(=O)CC2)=O)CC2(CCC2)CN1C(C1CC(=O)N(C)C1)=O N#CCCCC(=O)N1CCOCC1CCNC(C1(c2ccno2)CC1)=O c1(C(=O)NC(CN2CCN(C(C(C)C3CC3)=O)CC2)C)nccn2nccc12 C#CC1CC(NC(=O)C(C2CCC2)NC(=O)CSCCC)C1 Cc1ccc(C#N)cc1C(=O)NCC(C)C(=O)NCCCC(=O)NC1CC1 C(=O)(CN=c1ccc(Cl)n[nH]1)N1C(CNC(c2n3c(nn2)SC(=C)C3)=O)CCC1 C1(NC(CC(C)(C)C)=O)C2CCC(C2)C1C(=O)N(C1CS(=O)(=O)C1(C)C)C CCC(CC)(CC)C(C(=O)OC)NC(c1nc2ccccc2n1CCOC)=O c1(C(=O)NC(CNC(c2ccc(C(=O)OC)[nH]2)=O)C)cccc(C(C)(F)F)c1 N1(C(COC)=O)CCC(C(=O)Nc2cc(C)ccc2OC)C(C)(C)C1 N1(C(C(CCC=C)(C)C)=O)CCOC2(CCN(C(C34CCC3C4)=O)C2)C1 N1(C(C=CCN(C)CC)=O)CCSCC1CCNC(=O)C(=Cc1ccccc1)C c1(C(=O)NC(C2CCCN2C(c2ns[nH]c2=O)=O)C)ccc(C(F)(F)CF)cc1 CCCCCC(=O)NCC(C)N(C(=O)C(CCSC)NC(N)=O)CC C(=O)(C1CCCc2ccccc21)N1C(CC)CN(C(=O)CCC(F)F)CC1 c1(C(=O)OC)ncc[nH]c1=NC1CC(NC(=O)CC2C=CCCC2)C1 c1(C(N(C(CNC(C(CC=C)C)=O)C)C)=O)c(F)cccc1[N+](=O)[O-] C(=O)(CC(C(F)F)n1ccnc1)N(CCCN(C)C(c1ccc(Cl)cn1)=O)C c1(C(N2CCC(C)(C(=O)NOC3CCNC3=O)C2)=O)nccc2cc[nH]c12 CC1CC2(CCN(C(C3CC3(Cl)Cl)=O)CC2)CN1C(C1CCCSC1)=O CC1(C)CC(NC(C2CCC(=C(F)F)CC2)=O)CN(C(C2CCCC23CC3)=O)C1 N1(C(c2c(C)nsc2)=O)CCCCC1CNC(c1ccc(Cn2cccc2)cc1)=O c1(CC)ccc(-c2nc(Cc3ccccc3F)nn2CCOc2nncs2)cc1 C1(C(=O)NCc2ccc(N(C)C)c(F)c2)CCOCC12CCCC2 C1(C(=O)NC2(CF)CCN(C(C(C(C)C)F)=O)C2)CC2CCCC(C1)C2 C1(C=O)(C(F)F)CCCC1.c1(N2CC(C(N3CCC3C)=O)C2)nnc(O)s1 CC12CCC(=O)N1CCCN2C(=O)C(c1cccnc1)O C(C(CO)C(C)(C)C)NC(c1c(C)cc(CNC(c2ccnc(CO)c2)=O)o1)=O c1(CN=C(NC(C(COC)C)C)NC(C)C)ccc(C#N)c(F)c1 C1(CCC(=O)NCC=CCNC(Cc2c(C)noc2)=O)CC(C)(C)CO1 N1(C(c2cc(C(=O)OCC)[nH]c2)=O)CC2CCCC2(C(C)NC(=O)C(C)OC)C1 C1(NC(c2c(C)cccc2C)=O)CN(C(c2cn(CCO)nn2)=O)CC(F)(F)C1 c1(C(=O)NC2C(NC(C3(SC)CCC3)=O)C2)c(O)nnc2c1CCCC2 Cc1cc([N+](=O)[O-])nn1CC(=O)NCC#CCNC(C1CCN(C)C1C)=O c1(CN(C(C2CCN(CCC)C2)=O)C)nn(C)cc1Br c1(OC)ncc(Br)cc1CC(=O)NCCCCC1(N)CC1.c1(=O)c(=O)[nH]1 C1(SC)CN(C(c2cc(F)n(C)n2)=O)CC1NC(C1(CO)CCOC1)=O C(CNC(C1CC1C1CCCC1)=O)(CC(=O)NOC1CCOCC1)OC C1(CNC(C2(C=C)CCC2)=O)CCCCC1NC(=O)C(c1ccc(OC)cc1)C c1(C(=O)OC)ccccc1C(=O)N(C1CCN(C(=O)CC(F)(F)F)C1)C c1(OC)cc(NC(C2C(O)CCN2C(c2sccc2Br)=O)=O)nc(Cl)c1 c1(CN(C)CC2CN(C(=O)C(=O)NC3CCCC3)CCO2)cc(Br)ccc1I c1(CCCC)ccc(C(C)C(=O)NCC(c2ccccc2)O)cc1 N1(C(COCCC#C)=O)CC(F)(F)CC1CCNC(c1ocnc1C(F)(F)F)=O CC(CCC(C)(C)C)NC(=NCc1ccccc1Br)NCc1ccnn1C c1(C(N2CC3C(CNC(=O)CC4CC4C(F)(F)F)C3C2)=O)n[nH]c2c1CCCC2 C12(NC(CC3CC(OC)C3)=O)CCCC1N(C(C1CC3CCC1C31CC1)=O)CC2 N1(C(c2cc(C)sc2)C(=O)NC2CCC2)CCS(=O)(=O)CC1C1CC1 CC(CC(=O)N1CC2CC1C2C(N1CCc2nn(C)cc2C1)=O)CC(C)(C)C CC1(C(=O)NC2CCC(C(N)=O)C2)CN(Cc2c[nH]c(C(N)=O)c2)C1 N1(C(C(C)(C)CO)=O)CCC2C(CCCN2C(c2csc3cncn23)=O)C1 c1(CN(C(=O)NCC2CCN(CC)C2)C2CC2)ccc(C)cc1 c1(C(=O)OC)cc2cccnc2nc1NC(N1CCOC2(CCSC2)CC1)=O C(C(CC(C)C)NC(=O)C(C)CCc1ccc(F)cc1)NC(C)=O.c1(=O)c(=O)[nH]1 c1(C2C(C(=O)NC3CCN(C(c4ccsn4)=O)C3)C2)ccc2oc(O)nc2c1 C1(CNC(CCC2(C)CC2)=O)C2CCCC1N(C(=O)CC1C=CS(=O)(=O)C1)C2 C1(CC=C)CCCN(C(=O)CC(COC)NC(=O)C(C)C2(O)CCC2)C1 N1(C(CN(CC)CC)=O)CC2C3CCC(C2C1)N(C(c1cccc(CO)c1)=O)C3.CC c1(CN2CC(CNC(c3ccc(C)s3)=O)OCC2)c[nH]c2cnccc12 c1(C(=O)OC(C(C)=O)C2CC2)ccn2ncc(Cl)c2n1 CCCCC(=O)C(=O)N(CC(C)(C)CNC(C1CCOC(CCC)C1)=O)C N1(C(c2cn(CC)nn2)=O)CCC2(CCCCN(C(=O)Cc3nncs3)C2)C1 C1(NC(C2(CC#C)CCCO2)=O)CN(c2nnc(CO)s2)C2(CCOCC2)C1 c1(OC)cc(-n2nc(C3CCCC3)nc2Cn2c(C)csc2=O)ccc1Cl Cc1cccc(F)c1CC(N1CCC(F)C(NC(=O)CC2CCSCC2)C1)=O c1(COC)nc(NCc2cc(Br)ccc2C)cc(=NCCC2CCCN(C)C2)[nH]1 c1(C(=O)NC(CN(C(c2ccc(OC(C)C)cc2)=O)C)C)cccc(S(C)=O)c1 N1(C(C(=O)NCC(C=C)C)=O)CCN(C)C(Cc2ccc(OC)nc2)C1 N1(C(C=C(CC)CC)=O)CC2CC(CNC(c3ccc4occc4c3)=O)CC1C2 N1(C(C2C(=C)C2)=O)CC(C)(C)C(NC(=O)CCSCCCC)C(C)(C)C1 S(=O)(=O)(c1cccc(C(=O)O)n1)NC1C(OC)C2(C1)CCC2 Cc1ccc2[nH]c(C(=O)NCC(C)CNC(C34COC(CCO3)C4)=O)cc2c1 c1(C(C(C)C)O)cn(CC2CCC(C(=O)O)C2)nn1 CCCC(C)C(=O)N(C1CCC(NC(c2ccc(C(C)C)o2)=O)CC1)C C1(CC(N2CCCC(CCNC(c3n(CC)ccn3)=O)C2)=O)CCCS(=O)(=O)C1 C12(C(=O)NC3C4(CC(NC(C5C(C)(C)OC(=O)C5)=O)C4)C3)CCC(CC1)C2(C)C CC(C)CC(=O)NC(C)CC(C)NC(c1csc(C(F)F)c1)=O c1(C(C(=O)NC(C2CN(C(=O)CC=CC(C)(C)C)CCO2)C)(C)O)ccc(F)cc1 C1(CNC(C(COCC)C)=O)CC2(CO1)CN(C(=O)CCCCNC(N)=O)C2 N1(C(C2C(C)OCCO2)=O)CCCC12CCCN(C(C1(C)CCN(C)CC1)=O)C2 C1(NC(C2CCCN(C(C)=O)C2)=O)CC1C1CCCC1.c1(CC(C)O)cn(CO)nn1 CC1COC2(C1)CN(C(=O)C(CCN(C)C)NC(=O)CN1CCCNC1=O)C2 n1(CC(=O)CCC2N(C(C3(C)CC3)=O)CCC2)nnn(-c2cccs2)c1=O N1(C(CCNC(C(=CC2CCCC2)C)=O)=O)CCCC(C)C1C(=O)O C1(NC(C(C2CC2)OCC)=O)CN(C(=O)CN(C)CCO)CCC1F C12(C(=O)NC(C(=O)OC)C3CC3)C(NC(=O)C(C)N3CCCC3)C3CC1C2C3 N1(CC(C2(OC)CCCC2)=O)CCC(C(C)C)CC1C(C)(C)O C1(CN(c2nnc(CC)o2)CC)CCCN(C(=O)CSc2cnn(C)c2)C1 C1(NC(c2c(C)cco2)=O)CCCC(NC(c2ccc(F)c(N)c2)=O)CC1 N(C(=NCCOC)NC1CCOc2ccccc21)CC(c1ccco1)OCC C(CCCCC(=O)N1CC(N(C)C)C1)N(C(c1cccc(NC)n1)=O)C c1(CC)nc(C(=O)NC(C)(CNC(=O)C(C)c2cncs2)C2CC2)co1 C12(C(N(CC(C)CO)C)=O)CC1CN(C(c1ccc(F)cc1)=O)C2 c1(-n2ccc(C(=O)NCCC(C)NC(c3cncnc3)=O)n2)ccc(Cl)c(F)c1 Cc1cnc(Cl)c(NC(C2CSCCN2C(c2noc(C)c2C)=O)=O)c1 CC1C(NC(=O)CC2CCC(=O)NC2)CCCN1C(c1ccc(C(N)=O)cn1)=O c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(c2c(C)ncn2O)=O)CC1C C1(NC(CNC(C2C(C)C2)=O)=O)CCOCC1C(N1CCC(C(C)C)(CO)C1)=O C(=O)(C(C(C)C)C1CCC1)NC(C(=O)NC1C(C(=O)NC)CCC1)C1CCCC1 CCCC(O)CC(=O)N1CC(=C(F)CNC(c2nncn2C)=O)C1 c1(C(=O)NC2C(CNC(C(C3CCCCC3)C)=O)C2)cn(C)nc1C(F)F C(=O)(CCCCCCC(=O)N1CCC1NC(c1c(C)nc2sccn12)=O)OC c1(C(=O)Nc2c(C)ccc(Br)n2)nc(-c2cccc3ncnn23)c2ccccn12 C1(NC(C(CSC)OC)=O)(CNC(c2csc(C)c2)=O)CC2CCC1CC2 CCC(CC)C(O)CNC(=O)C1=CCC(NC(C2CC(O)C2)=O)C1 N1(C(CN(C)CC)=O)CC2CN(C(c3nc(Cl)sc3C)=O)CC2C1 c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cn(C3CCOC3)cn2)=O)C1)=O Cc1cc(C(=O)NC(C2CCCN(C(=O)Cc3cn[nH]c3)C2)C)cc(C)c1F N1(C(C=CCCC)=O)CCC2(C=C(C(=O)NCC3CCCC34CCC4)C2)C1 c1(C(N2CC3C(CN=c4[nH]ccnc4F)C3C2)=O)cc2ccccc2s1 C1(C(N(C2CCCC2)CCNC(C2(C)CC2(Cl)Cl)=O)=O)CCn2cncc2C1 S(=O)(=O)(c1ccccn1)N(c1nc(OC)c(Br)cn1)C1CCCNCC1 c1(NC(C23C(CN(C(c4ccc(Br)s4)=O)C2)C3)=O)cccc2cccnc12 c1(OC)ccc(Cl)c(CC(=O)NC2CC(F)CN2C(=O)CNCC(C)(C)C)c1F N1(C(CSCC#C)=O)CCC2(NC(=O)C(=O)N(C)C)CC12 c1(CC(=O)NC2(CNC(=O)CC34CC(C3)C4)CCC2)ccc2ccccc2c1 C#CC1CCN(C(=O)C(CNC(=O)C(C)SCCCC)CC2CCCC2)C1 C(=O)(CCCC(F)(F)CO)N1C2C(CNC(C3(F)C(C)OCC3)=O)C(C2)C1 C(=O)(CC1COc2ccccc21)N1CC(OCCNC(c2cn(C)nc2)=O)C1 C12(C(=O)OC)CC3CC(CC(C3)C1NC(c1cc(C)nc(C)c1O)=O)C2 N1(C(C(C)c2cccs2)=O)CC2CCC1CC2NC(=O)CCC(N)=O C1(CNC(C2C3CC4C(C3=O)C24)=O)C2CCCC1N(C(c1c[nH]cc1Br)=O)C2 S(=O)(=O)(c1ccc(Cl)cc1F)NCC(=O)NCC(C)NC(=O)C1=NOC(C)(C)C1 C12(NC(C(CC)SC)=O)CN(C(c3cnccc3Cl)=O)CC1CS(=O)(=O)C2 c1(C(c2n(CCCC)nnn2)NCc2ccoc2C)cnc(C(F)(F)F)nc1 CC1CN(C(C23CC(C#N)(C2)C3)=O)CC1(C)CNC(C1COCCO1)=O CN(S(=O)(=O)N1CC(O)C1)Cc1cc(F)cc(Br)c1 C(C1CCCc2nc[nH]c21)NC(=O)C(c1ccc(Cl)cc1F)O C(=O)(C1CCc2nccn21)NC(C)(CNC(c1cnn[nH]1)=O)C1CCC1 Cc1cccn(CC(N2CC3(CC3)CC2CNC(=O)CN2CC=CC2)=O)c1=O CS(=O)(=O)c1cc(C(=O)NCC2CCC2NC(=O)Cc2ccccc2)ccc1F C1(OC)CN(C(=O)Cn2nccn2)C(C)(CNC(=O)CSCCN(C)C)C1 N1(C(C(CC)SC)=O)CCC2(CC1)CCN(c1cc(-n3ccnc3)ncn1)CC2 C12(CNC(c3nc(CC(C)C)sc3)=O)CC1CN(C(=O)CCCc1ccsc1)C2 C12CCCN(C1)C(=O)c1cnccc1N(C)C2=O.n1(CC)ccc(CN(C)C)n1.NC Cc1cccc(C(n2cc(-c3cccs3)nn2)C)n1 CCCCCC(O)C(=O)NC1(C(N2CC3(CCC(=O)N3)C2)=O)CC(O)C1 C(C(C(=O)N(CC(O)CNC(c1ccc(Cl)cn1)=O)C)C(C)(C)C)OCC=C C1(C(N2C3CN(C(c4c(CC)non4)=O)C(CC3)C2)=O)COc2ccccc2C1 C1(C(=O)NCC(CO)NC(CCC)=O)(COC)CCCCCC1 CC(CN(C)N1CCOCC2(CCOCC2)C1)c1cccc(Cl)c1 C1(C(=O)NCC(O)CNC(C2CCC(C(=O)OC)O2)=O)(COCC)CC=CC1 c1(C2(C(=O)NCC#CCNC(Cc3cn(C)nc3)=O)CC2)ccc(Cl)cc1Cl C(=O)(C(C)CC(F)(F)F)NC1C(O)CCN(C(CCc2scc(C)c2)=O)C1 N#Cc1ccc(OCC(=O)Nc2cc(N3CCCC3)nc(Cl)c2)nc1 C1(c2n(C)ncc2)CCCCC1NCc1ccc(O)nn1 C1(NC(c2cc(C)n(C)n2)=O)CCCC2CN(C(c3nncs3)=O)CC12 N1(C(c2c(C)c(N)ccc2)=O)CCC2CC(NC(c3ccncc3)=O)CCC2C1 c1(N(C)C)cc(C(=O)NCC2OC3(C)CC2(O)C3)c2ccccc2n1 C(=O)(C1=C(Cl)CCC(C)C1)NCCCN(C(CCN1CCC(C)CC1)=O)C c1(C(N2C(C)(c3cn(CC(N)=O)nn3)COCC2)=O)cc2ccncc2cc1F N1(C(C(C2CCC(=O)N2)C)=O)CC(NC(=O)C(=O)NC2CC2)C(CO)C1 C1(C(CO)NC(C(C=C)C)=O)CCN(C(=O)CCCC2CCCO2)CC1 C1(NC(c2ccccc2)=O)CCC12CCN(C(=O)CCN1CCCCC1)CC2 c1(C(N2C(CCNC(c3cc(C4CC4)no3)=O)COCC2)=O)cc(F)ccc1O c1(C(=O)NC(C2CCN(C(c3cnccc3C#N)=O)C2)C)ncc2cc(Cl)ccn12 C1(C(N2CC(NC(c3ccc(C)c(Cl)c3)=O)C(F)C2)=O)CCC2C(C1)C2(F)F N1(C(CC2CCCC(=O)C2)=O)CC(=O)NCC1C(=O)NCCCc1cncnc1 CCCC(C(O)C(=O)NOC(C)C)NC(=O)Cn1ccnc1CC C1(O)(C(=O)NCC(c2ccccc2-c2ccccc2F)=O)CC2(CCNC2)C1 c1(C(=O)NCC(C)(C)NC(C(C)c2ncco2)=O)cc(Cl)cc2cccnc12 c1(N(C)CC)ccc(C(=O)NCCN(CC(C)O)C(c2scnc2C)=O)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC(C1CCCCC1)(C)C C1(C(N(CCC(C)NC(c2scc(OC)c2OC)=O)C)=O)CCCNS1(=O)=O C1(NC(CCCOCC)=O)CC(CNC(=O)C(c2ccccc2)C)CC1O C(C(O)CC(F)(F)F)NC(CC1N(C(C2CCN(C)CC2)=O)CCCC1)=O N1(C(C=CC(C)(C)SC)=O)CC(NC(=O)Cn2ccc(=O)cc2)C2CCCC12 c1(OC(C)C(N2CCC(N(C)C(c3ns[nH]c3=O)=O)C2)=O)ccc(Cl)cc1 N1(C(CC(CN(C)C)O)=O)CCC(NC(c2ccnc(C(C)C)n2)=O)C12CCC2 Cc1cc(F)ccc1NC(=O)C(c1nocc1Br)N(C(C)C)C1CC1 c1(C(N2CCC(C)(NC(C3CC4(F)CC3C4)=O)C2)=O)cccc2occc12 CC1CCc2ncc(C(N3CC4C(CNC(c5ccc(Br)o5)=O)C4C3)=O)n2C1 C(CC(C)C(=O)NC1(C)CN(C(C2(C)CC2(Br)Br)=O)C1)OC CCC(O)CC(=O)N1CC(O)CC1c1cn(-c2ccc(Br)nc2)nn1 N1(C(CCCC#C)=O)CC(=O)NCC1C(=O)NCC(C)(C)CC(C)C N1(C(C=C)=O)CCCC(CN(C(=O)C(CC)c2ccccc2)CC)C1 N1(C(C(c2cccs2)SC)=O)CCC(C2CC2)(NC(c2cc(C)cs2)=O)C1 C(CC(C)(C)C(=O)NCC1CCOC1C(=O)NCCC(C)(C)N(C)C)SC c1(NCCC(C)OC)[nH]c(=NCc2cc(C)nn2C)nc2c1ncn2C(C)C c1(C(N=c2[nH]n(C)c(C(=O)OC(C)(C)C)c2)=O)ccc2ncccc2c1Cl c1(C(N2CCC(CC=C)C2)C(=O)NCCSC(=O)CC)cc([N+](=O)[O-])sn1 CCC(c1ccccc1)=CC(N1CCCC1c1ccc(Br)c(F)c1)=O c1(SCC2(CN(C(C)C)C3CC3)CC2)ccc(C(=O)N(C)C)s1 C1(NC(C(CCSC)O)=O)CN(C(=O)CC2(C)CCN2C(C)=O)CCC1O c1(CC(N2C(C)(CC)CC(NC(C3CSC3)=O)C2)=O)c[nH]c2c(C)cccc12 C=CC1(COC)CCN(Cc2nnnn2C)CC1 C12(C(N(CC(CC)NC(C34CCC(C3)C4)=O)CC)=O)CC3CC1C2C3 C1(S(C)(=O)=O)(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2F)CCCC1 C=C=CCCC(=O)NC(c1nocc1C(=O)N(C1CCN(C)C1)CC)C C12(C(N3CCC(C)(NC(c4c[nH]cc(F)c4=O)=O)CC3)=O)CCCCC1C2(F)F C#CC1(N(C)C)CN(C(C2CCCC2CNC(c2ccc(OC)o2)=O)=O)C1 C1(C(=O)NCC2(CC)CCCCO2)CC(O)C(O)CC1CNC(=O)C(C)C1CC1 C1(C(N2CCCC(CCNC(C(CC)CC)=O)CC2)=O)CC2(CCC2)CCO1 c1(C(N2C(C(=O)NC(N3CCCCC3)CC)CC2)=O)cc(C)nc(C)n1 c1(C(=O)NC(C2CC2C(N2CC(O)C(O)C2CO)=O)C)ccc([N+](=O)[O-])o1 c1(OC)ccc2c(n1)N(C)CCN2C(=O)CN1CCC(C(N)=O)CC1 S(=O)(=O)(c1cccnc1NCC1CC(O)CN1C)NCc1n(CC)c(C)nc1 C=CCC(C(=O)NCC1(CNC(=O)C=Cc2cnn(C)c2)CC12CCC2)C(C)C C(=O)(C1CCCc2nncn21)Nc1c(CNC(=O)C2=CC(O)CCC2)cccc1 N1(C(C(C)NC(=O)OC)=O)CCC(OCCNC(=O)CC2CCC2)CC1 N1(C(c2cc(C(C)=O)oc2)=O)CC(CNC(C2(N(C)C)CC2)=O)CC(C)(C)C1 CCCC(C#N)C(=O)NC1CCCC(NC(c2cc(O)nc(Br)c2)=O)C1 CCCCC(CC)C(=O)N1CCC(COC)(NC(C2CN3CCN2CC3C)=O)C1 N1(C(c2cn(C)nc2C2CCC2)=O)CC(NC(c2ccon2)=O)CC2(CCC2)C1 c1(OC)ccc(Cl)c(Cl)c1C(N1CC2CCC1C(NC(=O)C(F)=C1CCC1)C2)=O CCCCCCCCC(=O)N1CC2CCN(C(c3cc(C(N)=O)co3)=O)CC12 N1(C(C(COC)N(C)C)=O)CC(C)N(C(=O)C(n2ccnc2C)C)C(C)C1 n1(CCNC(C2C(C)(C)C2)=O)cc(C(=O)NCCCC2CCCCC2)cn1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(NC(C(C)Cc2cccc(F)c2)=O)C1 N1(C(CC2CCC(=O)O2)=O)CCC(CNC(C23CC(F)(C2)C3)=O)C(F)(F)C1 C1(C(=O)NCCCCNC(C2C(C)C2C)=O)CCCCN1Cc1cccc(F)c1 Cc1ccnc(C)c1C(=O)NC1CCOCC1C(=O)NCc1ncsc1C c1(-c2ncc(N(C)CC3C(C(=O)OC)CN(C)C3)cn2)ccc(C(=O)O)c(F)c1 C1(C(=O)NCCCN(C(c2cnc(N(C)C)o2)=O)CC)Cc2c[nH]cc2S1(=O)=O Cc1nc(NC(c2nc(C(=O)NC(CO)C3CC3)cs2)=O)nc(Cl)c1Br Cc1cc(C(F)(F)F)nn1CC(=O)N(CCCNC(=O)C=C1CCC1)C1CC1 c1(OC)ccc(C(=O)NC2CCN2S(C)(=O)=O)c(NC(c2ccncc2Br)=O)c1 S(=O)(=O)(c1cccc(N2Cc3cnc(Cl)cc3C2)n1)N1C(C)C(O)CCC1 C(=O)(C1=CCC(C)(C)CC1)NC(CNC(C1CN(C(=O)NC)C1)=O)(C)C1CC1 C#CC1CCC(C(N2CCC(C(C)NC(=O)COc3ccccc3C)C2)=O)CC1 c1(NC(C2CCC(CNC(CC=CCCCCC)=O)C2)=O)cc(Cl)nc(C)n1 C1(C(=O)NCC(F)C(C)(C)O)(CC)CCCN1C(=O)C(CN(C)C)CC CC1(C)CC(=O)NCC1C(=O)NC1CCN(C(c2ccsc2)=O)CC1 Cc1ccc(C(=O)C(=O)NCC2CCN2C(=O)Cc2nc[nH]n2)s1 CC(C)(C)CC(C)(C)C(=O)NCC1(C)COCCN(C(C2(F)CC=CCC2)=O)C1 c1(N)ccc2cc(Br)cnc2c1.n12nnnc1C(CC1CC1)C(=O)C1CC2C1.CO C(C(CC(C)C)C(=O)NCC1(CCNC(c2nn(C)c(N)c2C)=O)CC1)OC C1(CNC(C(CNC(C2CN(C)C(=O)N2)=O)(C)C)=O)CC12CCOCC2 C(=O)(CCC1=CCCCC1)N1C(C(=O)NC(C(=O)OC)C2CCC2)CN(C)CC1 Cc1nc(O)[nH]c1C(=O)NCC(C1CCC1)NC(C1(c2cc[nH]n2)CCC1)=O C(CCCC(=O)N1CCC(C)(CO)C1)N(C(C(C)=CCC)=O)C c1(OC)c(NC(=O)CSC(c2ccc(F)c(Cl)c2)C)cccc1F c1(C(N2CCC(C)(C(=O)NCCc3ccsc3)C2)=O)ccc2cc(O)ccc2n1 N1(C(C=C2C(C)(C)CCCC2)=O)CC2CC(NC(c3cncc(F)c3)=O)CC2C1 N1(C(c2c(C)con2)=O)CCC(C(C)(C)C)(CNC(=O)CC2COCCO2)C1 C1(C(=O)Nc2ccc(OCC)nc2)CCCCN(C(c2ncccc2Br)=O)C1 CC1=C(C(=O)NC2CN(C(c3snc(Cl)c3Cl)=O)CC2F)SCCO1 c1(NC(C2CCOCC2)COC)ncccc1S(=O)(=O)N1CCC2(CCCC2)C1 c1(NC(c2n(CC=C)nnn2)C2(SC)CC2)ccc(-n2nccc2C)cc1 C1(OC)(OC)CCC1C(=O)NC(CNC(c1ccc(SC)o1)=O)CO C1(NC(=O)Cc2csnn2)CCC2CCN(C(c3cnns3)=O)C12 N1(C(C(COC)NC(C)=O)=O)CC(NC(=O)C(C)C(F)F)CCC1C CC1CNC(=O)C1.c1(C(C)C(=O)OC(C)(C)C)nc(-c2ccccn2)cs1 C1(NC(c2cc(C)nn2C(C)(C)C)=O)CN(C(=O)Cn2cnnn2)CC2CC12 C1(C(=O)NCCOC(CNC(C=CC)=O)(C)C)CC2C=CCC(C1)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCCC2(C1)CN(C(C1CC3CC3C1)=O)CCO2 Cc1cccc(C(O)C(=O)NCC(C2CCC2)NC(c2cc(C#N)on2)=O)c1 C1(OC)CC(CCNC(C2CCSC(C)C2)=O)N(C(C2(OC)CCC2)=O)C1 CC1CCN(CCC(=O)NCC2(C(N)=O)CN(C(=O)CC(F)(F)F)C2)CC1 N1(C(CCn2ncc(C)c2)=O)CCC(CNC(c2nnc(O)cc2C)=O)C(C)C1 CN1C(=O)OCC1C(=O)NCC1CCN(C(c2c[nH]nc2C(F)F)=O)CC1 CCCCCCCC(=O)N1CC2CCC2(C(=O)Nc2nccc(Cl)c2I)C1 c1(C(N2CCC(C)(CNC(=O)C(F)(F)CO)C2)=O)c[nH]c2ccccc2c1=O N1(C(CCCOCCC)=O)CC(O)CCC1C(=O)Nc1cccc(OCF)c1 c1(C(=O)NCC(CO)NC(C(C)CC2CC2)=O)ccccc1OCC(N)=O C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CCCC(NC(C2(C)CCCCCC2)=O)C1 C(C(C(=O)N1CC2COCC2O1)C(C)C)NC(c1n(CC)nnc1)=O N1(C(C2(CC#C)CCCO2)=O)CC(OC)CC(NC(c2ccc([N+](=O)[O-])o2)=O)C1 C#Cc1cc(C(=O)N(C)CC2CCN(C(=O)CC3(CC)CCC3)C2)ccc1C CC1CC(=O)NC1C(=O)NCc1cccc(NC(=O)CCC2CCCCC2)c1 C(C(C)(C)CC(=O)N1CCCC(C(C)(C)C)C1)N(C)CC1(C(=O)OC)CCC1 C=C(F)C1(CC(N2CC3(CCC3)CC2CNC(=O)CC(C)F)=O)CCOCC1 Cc1ccnc(NC(C2CCN(C(=O)CC3(O)CCCOC3)C2)C)n1 N1(C(C=C(CC)C)=O)CCC(N(C)C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CC(N2CCCC(C)(NC(=O)CCc3nccs3)C2)=O)CCCC2(CCC2)O1 c1(C(C(=O)NC(C)C)N(CCC(C)C)C(N)=O)cccc(NC2CCOC2)c1 C=C(C)CCCC(=O)NC1CC(O)(CNC(=O)C(c2cc(F)ccc2F)OC)C1 C1(CNC(Cn2cc(C)c3c2cccc3)=O)CC2CCC(C1)N2C(C1CC1C)=O Cc1cc([N+](=O)[O-])cnc1N1C2CCC1C(CNC(C1(O)CCOCC1)=O)C2 n1(CC(=O)N(C2CCC(NC(=O)C3CC3)C2)C)nc2n(c1=O)CCOC2 C(C(=O)NCC(c1ccsc1)C)(C1CCCC1)NC(C=CCOC)=O C(CN=c1[nH]c(=NC)[nH]c(=NC2CCC(CC3CCCN3C)CC2)[nH]1)SCC Cc1nc2cc(NC(C34CC3CN(Cc3ccccc3)C4)=O)ccc2o1 c1(N2CCCC(CCCNC(=O)C(=O)OC)(OC)C2)nc2c(C)c(C)ccc2s1 c1(OC)ccc(CC(=O)NCC2(NC(=O)Cc3cncnc3)CC2)nn1 Cc1c(C(=O)NC(C(=O)NCC(C)F)C2(C)CC2)ccn1C c1(C(=O)OCC)cnc(Cl)cc1NC(C1CC12CCN(C(=O)CC(=O)OC)C2)=O c1(CC(=O)NC2CCCN(CCCCCOC)C2C)cc2ccccc2nc1O N1(C(C(C2CCCOC2)OC)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC1C N1(C(C(CCOC)NC(C2CCC(C)CC2)=O)=O)Cc2cccc(C)c2CC1 CCS(=O)CC(=O)N1CCC(NC(=O)C=Cc2ccc(C3CC3C)o2)C1 C#CCC(CC(=O)N(CCNC(c1ccnc(C)c1)=O)C(C)C)c1ccccc1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CC(NC(=O)CC3CCCC3O)C1C2 n1(CC)c(C(=O)NCC2(C)CC(NC(=O)C3=NOC(C)C3)C2)cc2ccccc12 C(=O)(C(C)P(C)(C)=O)N(C1CCN(C(C(CCC)c2cccc(Cl)c2)=O)CC1)C Cc1cc(C(=O)NCC2(O)CCN(C(=O)C(C)CC3CC3)C2)c(Br)c(C)c1 C(=O)(C(CNC(c1cc(C2CC2)no1)=O)C(C)(C)C)NCCC(C(C)C)OC c1(C(=O)NCC(CNC(C(C2CC2)SC)=O)O)ccc(CS(N)(=O)=O)cc1 N1(C(C(C2CN(C(C3CCOC3)=O)C2)OC)=O)CC(=O)NCC1C(C)C C(C)(CNC(=O)C=CC(C)(C)C)(CO)NC(C1C(C(=O)OC)CC1)=O c1(OC)cc(N(C)CCNC(=O)C(C(C)O)N(C)C)ccc1NC(C)=O n1(CC(=O)NC2CCC(NC(c3csnn3)=O)C2)cc(Br)ccc1=O C1(NCC)CCCCN(CCc2nccs2)C1.C1(C2CCCC2)C(=O)O1 N1(C(c2c(CC)ncs2)=O)CCC2(C1)CN(C(c1cc(C(C)=O)on1)=O)CCO2 Cc1cc(OCCC(=O)N(C)CC2CCN(C(=O)C(C)CC(C)C)C2)cc(C)c1 C=CC(C)CC(=O)N1CC(C)(CC(=O)NCCC(C)(O)C2CC2)C1 c1(C(N2CC(C)C(CNC(C3SCCS3)=O)CC2)=O)ccc(F)c(S(N)(=O)=O)c1 N1(C(C(C=CC)O)=O)CC2CCCC2C1C(N1C2CCC1CC(CCO)C2)=O Cc1cccc(CC(=O)NCC2CCC2CNC(=O)CC2CCCOC2)c1Cl c1(NCC(c2cccc(Br)c2)C(=O)OC)cc(Br)ncc1[N+](=O)[O-] C(=O)(C(C)CCCC(C)C)N(CCN(C(c1nc(C(C)OC)oc1)=O)C)C(C)C S(=O)(=O)(c1cccc(C(N2CC(CO)CC(C)C2)=O)c1)N(CC)CC1CCOCC1 C1(CC(=O)NCCN(C)C(C2CCC(=C3CCC3)CC2)=O)CC(O)C12CCC2 N1(C(C2(COC)CCCC2)=O)CCCCC(NC(=O)C(c2ccc(Cl)cc2)O)C1 C1(C)(NC(CN(C)Cc2ccccc2)=O)CCN(Cc2cc[nH]n2)C1 n1(CCN(C(C2N(C)CC2)=O)C)cc(-c2csc(NC(C)(C)C)c2)nn1 N1(C(C=CCOCCOC)=O)CCC(NC(=O)Cc2ccccc2O)C(O)C1 c1(C(C)C)nc(NC2C3CC2CN(C(=O)CCC2CCCCO2)C3)cc(Cl)n1 c1(OC)ccc(CC(N2CCC(NC(C3C(C)C3C)=O)C2C(C)C)=O)c(OC)c1 c1(CC)cccc(C)c1C(N1CCC(CN(CCCNC(C)=O)C(C)C)C1)=O c1(CCC(=O)N(CC(C)NC(C2(C)ON=C(C)C2)=O)C)cccc([N+](=O)[O-])c1 N1(Cc2ccn(CC)n2)CCC2(CC1)CN(C(C1CCCCC1OC)=O)C2 C1(O)(CN(C)C(C2CC(F)C2)=O)CCN(C(=O)CSc2cn[nH]c2)C1 n1(CCOC)nc(C(=O)NCC2C=CCN2C(=O)Cc2cnn(C)c2)ccc1=O N1(C(CC(CC)C(F)F)=O)CCCC2(CCN(C(=O)C=CC3CCCC3)C2)C1 C1(F)(CNC(c2cncc(C)n2)=O)CCCN(C(=O)C2=CCCCC2)C1 C1(NC(=O)NCC2CCC(C)(CC)O2)CCOC2(CCSCC2)C1 C1(NC(c2cn(C)c(=O)cn2)=O)CC2CCC(C1)N2C(C1C2CCCCCC12)=O C1(CNC(C2CCC2c2ccncn2)=O)CCCCN1C(C1(F)CC=CC1)=O C(=O)(C(F)Cc1ccccc1)N1CC(CC(=O)NC2CCN2C2CCCC2)C1 C(=O)(C1=COCCC1)NCC(C)C(=O)NC1CC(CN(C)C)C1 c1(OC)c[nH]nc1C(=O)NC1(C)CC(NC(=O)C(c2ccccc2)C)C1 C12(C(N3CCCC(CCC(=O)NCc4nc(C)c(C)[nH]4)C3)=O)CCCC1OCC2 N1(C(c2cc(C)[nH]c2C)=O)CCC(CN)CC1C.C1(C)(C=O)CCN(C)C1 N1(C(CCN(CC(C(C)C)C)C)=O)CC(NC(c2nsnc2O)=O)C(N=[N+]=[N-])C1 C1(C(N2CC(CC)N(C(=O)CCc3nccn3C)CC2)=O)OCCOC12CCC2 n1(C2(C(=O)NCC3C(CNC(CCCSC)=O)C3)CC2)cnc2ccccc12 C1(CNC(C2(OC)CC2)=O)CCN(C(=O)CC2CCCCC2(F)F)C12CC2 C(CN=C(NCc1cnc(-c2ccccc2)o1)NC(CC)C1CCC1)OCC c1(C(N2CC(C)(CNC(C3CN(C(C)=O)C3)=O)OCC2)=O)ccc(C#N)c(C)n1 N1(C(c2ccc(=O)oc2)=O)CCC(NC2CC(C(=O)OCC=C)OCC2)CC1 Cc1nccnc1C(=O)NC1CC(NC(c2ccnc(OC3CCOC3)c2)=O)C1 CC(CC(=O)NCCC1CC(NC(=O)Cn2cnc([N+](=O)[O-])n2)C1)C(F)F N1(C(c2ccc(OC)s2)=O)CCCC(C(=O)Nc2ccnc(Cl)c2)C1 c1(CC(N2CCC3C2CCN3C(c2ccc(Br)nc2)=O)=O)ccc2nonc2c1 C1(NC(Cn2cc(-c3ccc(OC)nc3)nn2)=O)CCCC(C(C)(C)C)CC1 N1(CC2(NC(C34CC(C(C)C)(C3)C4)=O)CC2)CCN(C(=O)CN2CCCC2)CC1 c1(C(=O)NC2CC(NC(C3CCC(C)C(C)C3)=O)C2)cnc2ccc(C#N)cn12 N1(C(C(C#N)CC2CC2)=O)CCCC(CNC(=O)C=Cc2cnccn2)CC1 CC(CCCc1ccccc1)C(=O)NC1(c2nc[nH]n2)CCCC1 C1(C(N2C(C)(CC(=O)NCCCC#C)CC2)=O)(C(N)=O)CCCCC1 N1(C(c2c(OC)ccnc2)=O)CCOCC(NC(=O)C(C(C)C)C2CCC2)C1 C(CC(C(C)(C)C)NC(c1ccc(C#N)o1)=O)N(C)C(c1cccc(F)c1Cl)=O N1(C(C(C(CC)O)C)=O)CCCC2(CCN(C(c3nc(=O)n(C)[nH]3)=O)C2)C1 N1(C(c2c(C(C)C)occ2)=O)CCC(C(C)NC(=O)CC2CCC(C)O2)CC1 CC1COCCN(C(C23COC(C2)C(NC(C2CC2Cl)=O)C3)=O)C1 Cc1ccc(C(F)C(=O)NCCCN(C(=O)Cc2cnccn2)C(C)C)cc1 c1(C(N2C(C)CN(C(=O)Cc3c[nH]ccc3=O)CC2)=O)cc(F)c(Cl)cc1F N1(C(c2cn(C)nc2O)=O)CC2CN(C(c3cc(C#N)ccc3N)=O)CC2C1 CC(C(=O)NCC(C)(O)CNC(C1CCC(O)CC1)=O)C(C)(C)C C1(CNC(C(C2CCCCC2)NC(=O)CCCC2CCCO2)=O)C2CCCCC12 c1(Cn2cc(CC(C=C)O)nn2)cccc(CNC(C2C3COCC23)=O)c1OC Cc1cnc(C(=O)NC(CC(F)F)C(=O)NCC(F)C(C)(C)O)c(F)c1 CCCCC(C)(F)C(=O)NCc1ccc(C(=O)NC(C(=O)OC)C2CC2)s1 Cc1cc(Cl)c2c(c1)CCN(C(c1cccc(N3CCCNC3=O)c1)=O)C2 CCC(CO)(C(=O)NC1(CCCC(=O)N(C)CCC2CCCO2)CCC1)OC C1(C(N2CC(C(C)(C)O)(CNC(=O)Cc3ccsn3)C2)=O)CC(=O)C1(C)C c1(C(N(CCN(C(=O)CC=Cc2ccccc2)C(C)C)C)=O)cc2cscc2s1 CC1CN(C(c2cncc3cccnc23)=O)CC(C)N(C(C2COCCO2)=O)C1 N1(C(c2cc(C)c(O)cc2)=O)CC2CCC1CN2C(c1ccc2snnc2c1)=O C12(C(=O)NC3C(C)(C)OCC3)CCCC1CN(C(c1cnc(=N)[nH]c1)=O)C2 CCC(C)CC(=O)N1CC(NC(c2ccc(C3CC3)s2)=O)C(CC)C1 Cc1cc(C(=O)NCCCN(C2CCCC2)C(c2csc(C#N)c2)=O)c(C)cn1 N1(C(C(C)OCC)=O)CC(NC(c2nc3cccnc3s2)=O)C2(CCC2)C1 C1(C(N2CC(NC(c3c(C)cns3)=O)C(C)(C)C2)=O)CCCC2(CCC2)C1 C1(NC(=O)CC2CC2)CN(CCc2cn(-c3cccc(F)c3)nn2)C2CCCC12 N1(C(c2cccc(C)c2Br)=O)CCC(C)(C(=O)NCC2CN(C(C)=O)C2)CC1 N1(C(c2cc[nH]c2)=O)CCN(C(=O)C(O)Cc2cccc(Cl)c2)C2CCC12 c1(CC)ccc(C(N2CC3CC2C3NC(C2(C3CC3)CC2)=O)=O)cc1Br C1(NC(=O)Oc2cc(COC)oc2-c2ccccc2)Cc2cc(OC)ccc2O1 C1(CNC(c2c(C)ncnc2O)=O)C2CCCC1N(C(C1CC(C)OC1C)=O)C2 C(=O)(CC(CC)C(C)(C)C)NC1CCCC1.CCCCN(CCO)C(=O)C1CC1 C1(n2c(-c3cnn(CCO)c3)nc(C(C)C)n2)CCC(F)(F)CC1 C1(C)(C(N2CCN(CC3CN(C(CCC#CC)=O)C3)CC2)=O)COC(=O)OC1 C1(F)(C(=O)NC2CC(C)(NC(=O)CCN3CCOC3=O)C2)C2CCCCC12 c1(C(=O)OC)cc(O)cc(S(=O)(=O)N2CCC(C)C(c3ccccc3)C2)c1 c1(C(=O)OCC2CCCO2)ccccc1.C1CO1 c1(C(=O)N(c2ccccn2)O)ccc(SCCCNC(c2cn[nH]c2)=O)cc1 C1(C2CC2)(CNC(c2cc(CC(C)C)on2)=O)CCN(C(C2CNC(=O)C2)=O)C1 c1(C(C)=O)cc(C(=O)NC2CCCCC2n2cc(COC(C)C)nn2)cc(F)c1 Cc1cc(Cl)cc(Cl)c1OCC(=O)NC(C)CNC(=O)Cc1cccn1C C1(N(C)C)(CC)CCN(C(C2C3CC2N(C(=O)C(C)=C2CCCC2)C3)=O)C1 CC1(C)CCCC(O)(C(=O)NC2CCC2NC(c2cccc3nccn23)=O)CC1 CC1CN(C(c2cc[n+]([O-])cc2)=O)CCN1C(=O)CCc1cnccn1 c1(C(N2CCC(CNC(C3(OC)CCC3)=O)C23CC3)=O)cc2occc2n1C c1(C(=O)NC2CC(CCNC(C(C)(C)SC)=O)C2)n[nH]c(C)c1Br C1(NC(c2c(C)csc2)=O)CCN(C(c2cc(Cl)ns2)=O)CCC1CO C(C(=O)NCC1C=CCN1C(c1cc(C(N)=O)no1)=O)(C(C)(C)C)SC c1(OC)ccc2c(c1)CC(C(=O)NC(C1CCCCC1)C(C)NC(=O)CC#N)O2 c1(C(=O)NCCNC(C23OCCCC2C3(F)F)=O)c(O)nc2ccccc2c1Cl c1(CC)ccc(F)cc1C(=O)NC1CC1NC(c1c[nH]nc1Br)=O Cc1noc(C)c1CC(=O)N(C1CC1)CC1CN(C(=O)CO)C1.C1(=O)CCN1 N1(C(Cc2ncc(C)s2)=O)CC2C3CCC(C2C1)N(CC1CCOC(C)C1)C3 Cc1ccc(C(C(=O)NCCCC2CC2)N(CC(=O)N(C)C)C)c2ccccc12 c1(C(N2CC(CNC(C3(OC)CCC3)=O)(OC)C2)=O)cn(C(C)(C)C)nc1C Nc1ccc(C(N2CC3CC2C3NC(c2cnn(CC3CCC3)c2)=O)=O)c(Cl)c1 N1(c2nc(=N)nc(N(C)Cc3cccnc3)[nH]2)CCC(C2CCN(C)C2)CC1 C1(CC(=O)NC(C#C)C2CCC2)CCN(C(=O)C(O)C=CCCC)CC1 C12(C(N3CCC(N(C(=O)Cc4cscc4C#N)C)C3)=O)CCC(CO)(CC1)CC2 Cc1cc(=O)ccn1CC(=O)NCC1(O)CCN(C(=O)CCc2cn(C)cn2)C1 c1(N2CCC(NC(C(C)NS(CC)(=O)=O)=O)C23CCC3)ncnc2c1nnn2C C1(C#N)(C(=O)NC(CCOC)CNC(C2CC(C)=NO2)=O)CCCCC1 N1(C(C=CC(C)NC(c2ccc(C(C)C)o2)=O)=O)CCN2C(=O)OCC2C1 C(C(C)(C)CC(=O)NCc1cc(C(C)C)n[nH]1)NC(C1C(C)OCCO1)=O C1(NC(c2ccc(C)nc2O)=O)CN(C(=O)C(C)(C)CF)Cc2nccn2C1 NC(=O)C(O)CCCNC(C1CC(O)CN1C(=O)Cc1ncccc1F)=O N1(C(C2CCCN(c3cc(C)nn3C)C2)=O)CC(C)(C)CC1CO c1(CNC(C)C(=O)OC)ccc(C2N=N2)cc1.S(S(C)(=O)=O)CC(=O)NC(C)(C)C N1(C(c2c(CC)nn[nH]2)=O)CC(NC(=O)Cc2csc(S)n2)C(SC)C1 c1(CNC(=O)NCC2(O)C3(c4ccn(C)n4)CCC2C3)c[nH]c2ccc(Br)cc12 N1(N2CCC2)CCN(C(=O)C=CC(=O)OC(C)(C)C)CC1.C(=O)(C(Cl)=CCl)OC.CC Cc1ccnc(Oc2ccc(NC(c3cnc(C)[nH]3)=O)cn2)c1 c1(CC(=O)NCC2(O)CN(C(=O)NC3(O)CCC3)C2)ccc(C2CC2)o1 c1(C(c2cn(C3CCN(C(=O)Cc4cocn4)C3)nn2)(C)C)cccc(Cl)c1 C[S+](C)CCC(O)C(=O)NCC1CCN(C(C2(C)CCC3(CC2)CC3)=O)C1 C1(C(N2CC(NC(c3c(C(=O)OC)cccn3)=O)C2)=O)CCC2C1C2(F)F n1(CC(=O)NCC2CC(NC(c3cnoc3-c3cccs3)=O)C2)cc(C2CC2)cn1 C=CC1OCCC1C(C)(C)NCc1nc(C)cs1 CC(C)CC(O)C(=O)NC1CC(NC(=O)C(C(C)C)c2ccccc2)C1 c1(C(=O)NC2C(C(N(C(CC)C)C)=O)OCC2)ncccc1Cl CCCC(C#N)C(=O)N1CC(CNC(c2cnc(C3CC3)nc2)=O)C(O)C1 CCC(CC)C(C)C(=O)N(C(C)C(=O)N(C)CC1CCCCC1O)C CC1(C)CCCOC1C(N1CC(CNC(c2cc(C#N)c[nH]2)=O)CC1(C)C)=O c1(N2CCC(F)(C(=O)Nc3c(C)cc(Cl)nc3)C2)ccn2ncc(I)c2n1 c1(C(=O)NCC(C(=O)OCC)CC)cc2cc(C)cc(C)c2[nH]1 CC1CC=C(C(=O)N2CCCC2CC(=O)NCC(O)CC(C)C)CC1 C1(C2CCC2)(CNC(CN2C(C)CC2)=O)CCN(C(=O)Cc2nc[nH]n2)CC1 N1(C(CCC)=O)CCCC(C(N2CCC(N(C)C(c3cc(Cl)n(C)n3)=O)C2)=O)C1 CC(C)C(C(=O)NC1CC(CCNC(=O)Cc2ccc(Cl)cn2)C1)N(C)C N1(C(c2ccc(C(F)(F)CF)cn2)=O)CC2CC1CN2Cc1ccccc1 c1(CN(C)CC2CCCCCCN2)cc2ccccc2nc1O N1(C(CC(C)N(C(CSCC)=O)C)=O)CC(C)C(C)C1C Cc1cc2c(C(=O)NCC(C)N(C)C(C3CCC4(CCC4)C3)=O)cccc2o1 c1(C(=O)NCC(C)NC(=O)C(C)Cc2ccccc2)ccc(F)c2cnccc12 c1(C(=O)NCC2CN(C(c3c(C)onc3)=O)C2)cccnc1CC(C)C c1(CC#N)cccc(S(=O)(=O)N2CCCC3(CCOC3)C2)c1 C1(F)(CNC(c2cccc(F)c2F)=O)CCCN(C(=O)CCC2CCCOC2)C1 C(=O)(CC(C(C)(C)C)NC(C1CCC2CC1CO2)=O)Nc1cccc(CC)c1 C12(NC(c3ccc(O)nn3)=O)CCC(C1)N(C(=O)Cc1nc(C3CC3)cs1)C2 c1(C(CC)(C)C)ccc(CCCNC23CC4CC2C3C4)cc1 c1(C(N2CC(CNC(C=CS(C)=O)=O)C(C)(C)C2)=O)cnc2ccccc2c1 c1(C(N2CC(O)CCC(NC(C(C)(C)C(F)F)=O)C2)=O)cn2cccc(Cl)c2n1 C1(NC(C2CCSC2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC2(CC2)C1 C1(C)(C(=O)NC(CCC)CCCNC(c2ccc(C)o2)=O)CCS(=O)(=O)CC1 C1(NC(CN(CCCCCC)C)=O)CC2(C1)CN(C(C1CCOC1C)=O)C2 c1(C(N2C3CN(C(=O)CC4CC4(Cl)Cl)CC2CC3)=O)ccc2c(c1)OC(F)(F)O2 CCC(CCOC)NC(=O)CCCC1(NC(c2c[nH]nc2OC)=O)CCC1 C1(C(=O)NCC2C(NC(Cn3nnc(C)n3)=O)C2)CCc2ccccc2O1 N1(C(C(CC)N(C(=O)C2CC2)C)=O)CC(NCc2ncnn2C)CC(C)C1 c1(C(=O)NCC2CN(C(C=CS(C)=O)=O)CC2O)cc(F)c(Br)cc1F c1(C(=O)NC2CCC(N(C(CCC=C)=O)C)C2)c(C)ccnc1C C(=O)(C1CCCc2n[nH]cc21)NCC1C(C)CCN1C(=O)CCc1cnoc1 c1(C(=O)NC2(CNC(=O)C=CC3CCCCCC3)CC2)cc2cc(O)ccc2[nH]1 c1(C(=O)NCCCN(C)C(C2CCC(=O)N2C2CC2)=O)cc2cnccc2o1 CC1(C#CC(=O)NC(CCCC=C(C)C)=O)CCCO1.c1(C)cnc2n1CCC2 CC1CC2CCC(C(=O)NCC3=CCN(C(=O)C(=O)C(C)(C)C)CC3)CN2C1 c1(C(=O)NCC2CCCN2C(=O)CCCc2ccncc2)ccc(O)nc1 c1(C(N2C(C(N(C)Cc3ccc(Br)cc3)=O)CC(F)C2)=O)c(Br)ccc(F)c1F c1(NCCNC(=NCCCC2(OC)CCC2)NC(C)CC)ncnc2[nH]cnc12 N1(C(c2c(C)onc2)=O)C2CCC1C(CNC(=O)Cc1csc(Cl)c1)C2 Nc1cc(C(=O)NCC(CNC(=O)C(O)C2CCCC2)S(C)(=O)=O)cnc1Cl CCCCCCC(C)C(=O)NC1COCC1CNC(=O)CC1(SC)CCC1 c1(C(=O)NCCCN(C(CC(CC)OC)=O)C)cn2cccc(Br)c2n1 c1(-c2n(-c3c(C(C)C)cccc3)nc(-c3ccc(N)cc3)n2)ncc(F)cc1N c1(C(N2C(CNC(=O)CC3CC3C3CC3)C=CC2)=O)ccccc1C(F)F CC1CCC(CNC(=O)CCc2ccc(F)cc2)N(C(=O)COCCF)C1 C1(CCCC)CN(C(C2NC(=O)C3CC23)=O)CCN1C(=O)C1=CCCC1 CCCC(CC)CC(=O)N1CCC(OC2CN(C(c3cnn(C)c3N)=O)C2)CC1 c1(SC)ccccc1C(=O)NC1(C)CCN(C(=O)CC2CC(C(C)(C)C)C2)C1 c1(COC)cc(C(=O)NCCCCC2CC2)no1.N12CC(C1)CNC2=O c1(C(=O)NC23CC(C(=O)NC(c4ncc[nH]4)CC)(C2)C3)ncc(F)cc1F C1(NC(CSCCNC(CCc2cc(C)[nH]n2)=O)=O)CC(O)CC1O Cc1cnccc1C(C)C(=O)NC1CCCCC1N(C)C(c1cccs1)=O C1(C(N2C(CNC(c3c(N)csn3)=O)CC3CCCC32)=O)CCOC2(CCC2)C1 c1(CC)cc(NC(c2ccc(Oc3ccc(C)nn3)cc2)=O)cnc1C n1(CCC(=O)NC(CC=C)CNC(c2c[nH]nc2C(C)C)=O)cnc(C)cc1=O C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(NC(=O)CC(C)(C)CN(C)C)CC(C)C1 c1(CNC2CCCC(CC(=O)O)(C(F)(F)F)C2)c(OC(F)F)ccc2ccccc12 C12(C(=O)NC(C(=O)OCC)CCc3ccccc3)CCC(CC)(C1)OC2 Cc1cc(C#N)nc(NC23CCCC2CN(C(=O)C(C)N(C)C)C3)n1 c1(CC(N2CC(NC(C(C)(C)SC)=O)C(C)(C)C2)=O)ccc(S(=O)(=O)N(C)C)o1 c1(C(C)OCC)cn(CCOCCNC(=O)CCn2ccnn2)nn1 c1(C(=O)NC2C(CC(=O)O)CC2)cncc(-n2cc(C3CC3)nn2)c1 c1(CC)ccc(C(=O)NCCCC(C)(C)NC(c2ccc(C)c(F)c2)=O)c(C)n1 c1(OC)ccc2c(c1)C(CCN(CC(F)(F)F)Cc1cccc(C)c1)=CC2 N1(C(CN(c2ccccn2)C)=O)CCC(O)(CCNC(=O)C(C)(C)N(C)C)C1 CCCN=C(NCC1CC1Cl)N1CCC(F)(c2cc(OC)cc(OC)c2)CC1 c1(C(=O)NCCOCCOCCNC(C2CC2Cl)=O)ccc2c(c1)CCN2 C#CCC(O)C(=O)NC1CC(NC(=O)C(F)(F)c2ccsc2Cl)C1 N1(C(c2cc(OC)n(C)n2)=O)CCOCCC1C(=O)NC1C(C)C1C C(=O)(C#CC1CCC1)NC1C(CNC(c2c(COC)cccc2)=O)CCCC1 C1(C(N2CC3C(NC(C=C(COC)C)=O)(C3)C2)=O)CC2(CC(C)=NO2)C1 N1(Cc2ccc(C)o2)CC2CCC1CN(c1ncc(I)cn1)C2 O=C(C(C1=CCCSC1)N1CCSCC1CCSc1ccccc1Br)NCCO N1(CC(N2CC(CNC(C(COC)OC)=O)C2)=O)C(=O)c2ccccc2S1(=O)=O c1(OC)c(C(N2CC=CC(NC(=O)CSC(F)(F)F)C2)=O)[nH]c2ccccc12 [N-]=[N+]=NC1CN(C(=O)CC2OCCO2)CC1NC(C1CNC(=O)N1)=O c1(C(=O)NCC2C3CN(C(c4ccc(OC)cn4)=O)CC32)cc2ccsc2cn1 c1(CCNC(Cc2c(I)ccc(C)c2)=O)cc(Br)c2c(c1)CCO2 c1(OC)ccc(CN2CCNCC2C(=O)NCc2ccc(Br)cc2)c(Br)n1 N1(C(CC=CCC)=O)CC2CCC(C1)N2C(=O)Cc1nnc(S)n1C c1(CC)c(C(N2CC(CC(C)NC(=O)COC)C2)=O)oc2ccccc12 N1(C(Cc2ccn(CC)n2)=O)CCCN(C(C2CC3CCC3C2)=O)CCC1 N(C(=NCCCF)NCC(=C1CCSCC1)F)Cc1ccc(C(C)C)c(F)c1 C12(CCNC(COC(C)=O)=O)CCC(C1)N(C(=O)CCOC1CCCCCC1)C2 C1(C(=O)NC2CCN(CCC)CC2)C2CC(O)C(C2)N1C(=O)C=CCO c1(OCCCC(=O)N2CC(N(C(=O)C(C3CC3)OC)CC)C2)cccc(C)c1C c1(NC(c2ccnc(C)n2)=O)ccc(NC(c2scnc2C)=O)c(F)c1 c1(SC)cc(NC(c2cc(-c3ccn(C(C)C)n3)ccn2)=O)ccn1 C(CC(C(C)(C)C)NC(=O)C1=C(Cl)CC1)N(C(CCCN(C(C)C)C)=O)C C1(CNC(C(C)NC(CC)=O)=O)CN(C(=O)C(O)C(C)C)CCC1C(F)(F)F C1(CC(F)F)(C(=O)NCCCC(C)NC(C2CCC(C)(C)O2)=O)CCOCC1 C1(C)(CNC(c2cc(CC)nn2C)=O)CCN(C(C2CC2(F)Cl)=O)CC1 N1(C(C=CC=CC)=O)CCCCC1C1CCN(C(=O)C(C)n2cnnn2)CC1 N1(C(C(C2CCCC2)OC)=O)CCN(C(=O)C=CSCc2ccco2)CC(C)(F)C1 C#CC1(CNC(=O)C(CC(N)=O)NC(=O)CCSCCC)CCOCC1 c1(N2CCN(CC3(C#N)C(C)(C)C3)CC2)cc2occc2[nH]1 C1(CNC(CC2CC(CN(C)C)C2)=O)CN(C(=O)C(C)(C)CC2CCC2)CCO1 C1(CNC(=O)COC(F)(F)C(F)(F)F)CCCCC1NC(=O)CN1CCOCC1 Cc1cc(C(N2CC3(NC(c4cc(C(C)C)[nH]n4)=O)CCC2C3)=O)cc(C)c1N C1(CNC(c2c(CC)ccs2)=O)CCC2(CN(C(c3[nH]ncc3C#N)=O)C2)O1 C1(NC(C=CC(=O)N(C)C)=O)(CF)CCN(C(C2COC(=O)O2)=O)C1 CN1CC(O)CCC1C(=O)NC1CC(Cn2cc(COc3ncccn3)nn2)C1 N1(C(C(C)OC)=O)CCCCCC1CNC(c1ccc(Br)nc1O)=O N1(C(c2cc(C)sc2)=O)CCC(F)C(NC(c2nc(C)oc2C)=O)C1 c1(C(C(=O)NCC(C2CCCC2)NC(C2(C)CC2(F)F)=O)(C)O)ccccc1F c1(C(=O)NC(CN(C(=O)CC(C)SC)CC)C)nnn(C)c1N Cc1ccc(CNC(C23COCC2C3(F)F)c2nnnn2C)nc1C C(=O)(CCCNC(=O)NC1CC1)N(C(CO)C1C(Cc2cscn2)C1)C C(=O)(C1COc2ccccc21)N1CCCN(C(c2c(O)cccc2Cl)=O)CC1 C(CCCCNC(c1cnc(C(C)OC)s1)=O)NC(C1C(=C)CC1)=O CCC(S(=O)(=O)NCC1CCC(N)CC1)c1ccccc1 C1(C(=O)NC2C(CC=C)CCCC2)CN(C(C2(C)CCCO2)=O)CC1(F)F C(=O)(C1=C(C)CCCC1)N(CC)CC1CCCCN1C(=O)CCc1cc[nH]n1 C1(CCNC(CS)=O)(C)CC1(F)F.C1(c2cc[nH]n2)(NC(CC(C)=O)=O)CCC1 N1(C(c2n(CC)ccn2)=O)C2CCCC1CC(N=c1[nH]c(Cl)ncc1C1CC1)C2 N1(C(CC2CN(C)C2)=O)CC2CCCN(C(C34COC(CF)(C3)C4)=O)C2C1 N1(Cc2cnc(N3CC4CC4C3)s2)CCOC2(CCCNC2)C1 c12ccc(O)c(c1)C(=O)NCC(=O)OC2.N1(C(C)=O)CCOC(CNC(C)=O)C1 c1(SCc2cn(CCCNC(CNC(CC)=O)=O)nn2)cc(C)cc(F)c1 c1(NC(C2CCN(C(=O)CNCCC(F)(F)F)C2)=O)cccc2c(O)nccc12 c1(CN2C(C)(C(=O)NCc3cc(OC)ncc3)CC2)cccc(OC)c1OC N1(C(C2=CCN(C)C2)=O)CCC2(CCN(C(=O)Cc3ccc(F)cc3)C2)C1 CC(CCNC(=O)CSc1ccccc1)CCNC(=O)CC(C)c1cnn(C)c1 C1(CN(C(c2cnccc2Cl)=O)CC)CCN(C(=O)Cc2ccc(F)cn2)CC1 N1(C(CC(CC)O)=O)CCCC2(CCCN(c3ncnc4[nH]cc(I)c34)C2)C1 N1(c2nc(COC)nc(C)c2)CC2CCC1C1CN(C(C3CC3(C)Br)=O)CC21 C1(C)(CNC(C2CCN(C)CC2)=O)CCCN(C(=O)CCCNC(=O)C=CCl)C1 N1(C(CC(CNC(c2c(C)ccnc2)=O)O)=O)CCC(C)(C)C1CO C1(NC(C=CC(CC)C)=O)CCN(C(=O)Cn2nc(C(F)(F)F)cc2C)CC1O CC(C)(CCNC(=O)CSc1nncs1)C(=O)NCC1CCC(CO)O1 C12(NC(C(CCSC)O)=O)CCCC(NC(=O)CCc3ccc(N)cn3)(C1)C2 c1(C(N2C(C)CC(CNC(CN(C)CC)=O)C2)=O)cc(Br)cc2c1OCO2 C(=O)(C1=CCCCC1C)N(CCOC)CCNC(=O)Cc1ccc(OC)cc1 C(Cc1ccccc1)(Cc1ccccc1)(c1nnnn1C)N(C1CCCO1)C N1(C(COCC=C)=O)CCC(C)C(CNC(=O)Cn2cccn2)C1 CC(=Cn1ccnn1)C(=O)N(CC(C)N(C(=O)CC1C=CS(=O)(=O)C1)C)C C(=O)(C(CC1CCCC1)NC(=O)C1CC1)N(C1CCCCC1)CC(=O)OC CC1(C)C(=O)CC1(P(C)(C)=O)C(=O)NC1CCN(C(=O)Cc2csnn2)CC1 C(=O)(C#CC1CCOC1)N(CCCCCNC(C1CCCCN1S(C)(=O)=O)=O)C c1(OC)ccc(=NC(=O)Cc2cc(-c3c(OC)cccc3F)cs2)[nH]n1 N1(N2CCC(CN3CCN(Cc4ccc(SC)o4)CC3)C2)CCOC2COCC12 c1(C(=O)NC2C(OC)CN(C(C3N(CC)C(=O)CC3)=O)C2)cnc2[nH]ccc2n1 C=C(C)CC(C)C(=O)NCC(CC(C)C)NC(c1ccc(OC)c(N)c1)=O CCS(=O)(=O)c1cccc(S(=O)(=O)N2CCCC(CO)CC2)c1 N1(C(Cc2nc(NC=O)sc2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C2CC12 c1(C(N(C)CC2CCN(C(C3(C#N)CCC3)=O)C2)=O)csc2ccncc12 c1(C(=O)NC(C)CCCNC(C2CC23CCCC3)=O)ccc2nnc(S)n2c1 Cc1cc(=NC(=O)C(C)OC(=O)CCc2ccc(Cl)cc2Cl)[nH]o1 C(C(C)CC(=O)N1CCCCC1C(=O)N(CCS(C)(=O)=O)C)OC N1(C(C(CC)CN(C)C)=O)CCC(NC(c2cc(C(N)=O)[nH]n2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc(NC(C2CCN(C)C2)C)cc1Br)NCc1nnc(COC)s1 C1(N(C(C2C(=C)C2)=O)CC)CCCN(C(c2cc(OC)cc(C)c2)=O)CC1 CC(C)(CCN=c1ncc2ccccc2[nH]1)NC(C1(c2ccc(F)cc2)CC1)=O CCC1=C(C)CC(COC)N1Cc1cnn(C(C)(C)C)c1C1CC1 N1(C(CCCC(=O)NCC)=O)C2CCC1CN(C(=O)C(C)C(O)CC)C2 C1(C(=O)NCc2cc(C)no2)C(C)OCCN1C(=O)C(C)CC(N)=O N1(CC)OCC(NC(=O)CC2(C)CCN(C(C3SCC=C3C)=O)C2)C1=O CC1COCC(CC(=O)NC(C(=O)NCCC2CC=CC2)C(C)O)O1 N1(C(CC(=O)NCC)=O)CCC(C)C(NC(=O)CCNC(C)C)C1 c1(C(=O)NCC(=O)NC2CC(CNC(=O)CC3CSCCS3)C2)cccc(O)c1 c1(C(N(C2CN(C(C(C)OCC#C)=O)CC2(C)C)C)=O)cccc2nn(C)nc12 CC(C)(CCC#N)C(=O)NC1CCC(NC(c2ccc([N+](=O)[O-])cn2)=O)CC1 c1(C(=O)NCC2(C)N(C(C(C=C)O)=O)CC(F)(F)C2)ccc2cnc(C)n2c1 c1(CC)onc(C(=O)NCCCCCn2cc(C3(O)CCCC3)nn2)c1C C1(NC(CC(CCC)C)=O)CN(C(=O)CCc2cc(C)[nH]n2)Cc2ccnn2C1 C(=O)(C(C)(C)CC(=O)NC(C)(C)CNC(=O)CCN1CCC(F)C1)OC N1(C(C2(F)CC(C(=O)OCC)C2)=O)CCC(NC(=O)CS(N)(=O)=O)C12CCC2 C(CC(C)CCS(=O)(=O)N1C(NC(=O)OC(C)(C)C)CC2OCCC12)OC S(=O)(=O)(c1cnc(Cl)c(Cl)c1)NC1(C#C)CCC(C(C)(C)C)CC1 C1(CNC(C(N2CCSCC2)C)=O)CCCN(C(c2ccc(F)cn2)=O)CC1 c1(CNC(C2CN(C(=O)OC(C)(C)C)C2)C(=O)NCC(=O)O)cncc2c1CCC2 c1(C(N2CC(CNC(c3cc(CCC)nn3C)=O)(OC)C2)=O)cc(C)c(O)nn1 C1(NC(c2[nH]cc(C)c2)=O)CCOC12CCN(C(C1CCCC13CC3)=O)CC2 c1(CNC2(CNC(c3c(C)ccc(Cl)c3)=O)COC2)ccc2cc(F)ccc2n1 C1(C(=O)O)CCCCC1C1CCN(CC(N2CCCCCCCCC2)=O)CC1 Cc1ccc2c(c1)CCC(C(=O)OCc1cn(C(c3ccccc3)(C)C)nn1)O2 N1(C(C(CC#C)C2CC2)=O)CCOC2(C1)CN(C(C1CC3CC3C1)=O)C2 N1(C(C23CC(OC)C2C3)=O)CCC(N(C)C(c2cc(C(C)(C)C)n[nH]2)=O)CC1 CCC(C)CC(=O)NCC1(c2ccccc2)CC(NC(=O)CCN2CCC2)C1 C(=O)(C1Cc2ccccc21)NC1CCCN(C(c2ccnc(C)n2)=O)C1 c1(C(=O)NCCCC(C)NC(=O)Cc2ccon2)cccc(C2(F)CC2(F)F)c1 c1(OC)cc(CC(N2CCC(O)C(NC(C3CCCN3C=O)=O)C2)=O)ccc1C Nc1cc(Br)ccc1C(N1CCCC1CCCNC(=O)C(O)C(F)F)=O C1(NC(c2ccc(Br)cc2)=O)CN(C(=O)Cc2cncs2)CCC12CCC2 N1(C(CC(=C)Br)=O)CC(CNC(c2ccc(OC)nn2)=O)CC12CCC2 C(CN=c1nc(N2CCC(CN(C)C)C2)c2ncccc2[nH]1)c1ccc(C)cn1 C1(C(N(c2cccnc2)C(C)C)=O)CCN(c2ccnc(C3CC3)n2)CC1 C1(C2C(NC(C=CC(=O)N(C)C)=O)CCO2)CCN(C(=O)CC2CCSC2)CC1 C(=O)(C1SCc2cccnc21)NCC1C(NC(C2(CC)CCC2)=O)CC1 c1(OC)cc(CC(=O)NC(C(C)NC(C23CC(F)(C2)C3)=O)C(C)C)ccc1Cl N1(CCC)CCCCC1C(N1CCC(F)(CNC(c2coc(C)n2)=O)C1)=O C(=O)(CCC(=O)NC1(COC)CN(C(C2CCCN(C)C2)=O)C1)NC c1(C(N2CC3C(CNC(CC=CC)=O)C3C2)=O)c(C)oc(C)c1Br C12(C(N(CC(CC)(O)CC)C)=O)COCC1CN(C(C1CCCC(C#N)C1)=O)C2 C(=O)(C(C(C)CC)NC(C12CCCC1CCC2)=O)NC N1(C(C(C)OCC#C)=O)CCN(CC(=O)NC(C2(OC)CCC2)CC)CC1 C1(C(C)NC(C(CC)Nc2ccccc2)=O)CCN(C(=O)C(C)(C)COC)CC1 Cc1cc(Cl)ccc1C(=O)Nc1cc(-c2ccccc2NS(C)(=O)=O)ccn1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nccn2)cc(F)ccc1Cl C(=O)(C(F)C(C)(C)O)N(C1CCN(C(C(CC)O)=O)CC1)CC C1(C(C)(C)C)(CNC(C2(CC#C)CC2)=O)CCN(C(c2ccc(F)cn2)=O)C1 c1(NC(C2CCC(C(C)C)N2C(=O)C=CCF)=O)cc(F)c(O)cc1C n1(CC(=O)NC2C(NC(CC3(C)CCCCC3)=O)C2)ccc(O)nc1=O Fc1ccc2c(c1)C(c1nc(-c3cccs3)nn1C13CC(C1)C3)CO2 n1(CCC(=O)NCC2(F)CC(CNC(C(C=C)O)=O)C2)cc(Br)ccc1=O c1(C(=O)NCC(CC)NC(C2CC2c2ccccc2)=O)ncccc1O C(=O)(C(C(C)(C)C)NC(N)=O)NCC(CNC(C(C)CC1CCCC1)=O)C C(=O)(C1CCCc2cncn21)N1CCCC2(CN(C(C3C(=C)C3)=O)C2)C1 N1(C(CC2(C=C)CCOCC2)=O)CC(NC(C2OCCO2)=O)C(C2CC2)C1 c1(C(N2CCCN(C(C3CCCN3C3CC3)=O)CCC2)=O)ncc2ccccn12 O=C1CCN(C(c2cncnc2C2CC2)=O)CCCN1 c1(CC(=O)C(=O)OC)ccc(O)c(C)c1.C12CCN(CC1)C2.C1(SC)CC1C(C)C c1(C(=O)NC2C(NC(c3cc(C)c(O)cc3)=O)CC2)cc(P(C)(C)=O)cs1 C1(C(C(=O)NC2(CC(N)=O)CCC2)NC(c2cn[nH]c2)=O)CCCCC1 c1(NC(=O)NC(c2n(CC)cnn2)C)ccccc1OC(c1ccccc1)C c1(CC)ccccc1C1CN(C(c2sc(C3(C)OCCO3)cc2Br)=O)CCO1 O=C(CCCCCF)NCC1C2CCC(C2)N1C(C1CCCOCC1)=O N1(C(=O)CCC2CCCN2C(=O)CCC2CCCO2)CCCC2(CC(O)C2)C1 c1(NC(C2CN(C(C3CC3c3ccccc3)=O)CCN2)=O)nc(F)c(Br)cc1Br Cc1cccc2c(C(=O)NC3CN(C(=O)CC(C)(C)C#N)CC3N=[N+]=[N-])c[nH]c12 c1(C(=O)NCCN(C(c2ccc(F)cn2)=O)CC)cccc(C)c1[N+](=O)[O-] c1(CN(C(=O)CNC(=O)CC2CC2)CC)cccnc1 C1(NC(CCC2(NC(CSC)=O)CCCC2)=O)CCN2CCC1C2 Cc1c[nH]c2ncc(C(=O)NCC3C4CN(C(=O)CCCN(C)C)CC34)cc12 C1(NC(c2cnc(OC)nc2)=O)CCN(C(c2sc(C)cc2C)=O)CC(C)(C)C1 Cc1ccc(OCCC(=O)N(CC(C)NC(C2CC(N(C)C)C2)=O)C)c(C)c1 C#CCCC(=O)NCc1ncoc1CCNC(=O)CSCc1csc(=N)[nH]1 C1(SC)CCC(N=c2nc(N3CCC4(CCNC4=O)CC3)c3sccc3[nH]2)C1 C1(NC(COC(C)=O)=O)CCC(N(C)C(c2sc(Cl)cc2Cl)=O)CC1 c1(OC)cc(N(C)C)ccc1C(=O)NCCC(O)CNC(=O)C#CC1(C)CC1 Cc1cccc2c(=O)c(C(=O)NCC3CN(C(=O)C(C)CC(C)(C)C)C3)c[nH]c12 Cc1ccc(Cl)c(C(=O)NC(C2(O)CCN(C(=O)C(C)C3CCOC3)C2)C)c1 c1(C(=O)NC)cc([N+](=O)[O-])ccc1N1CC2(CN(C(=O)CC(C)SC)C2)C1 C1(NC(C(C(C)C)CN(C)C)=O)C2CCC1CN(C(c1cc[nH]c(=N)n1)=O)C2 N1(C(CCC#C)=O)CCC(NC(=O)CCN(C)Cc2ccccc2)CC1C1CC1 N1(c2n(CCC#C)c(-c3ccc(Br)c(C)c3)nn2)CCc2c(I)n[nH]c2C1 C1(NC(C2(NC(=O)OC)CC2)=O)C2CCC(C2)C1C(=O)NC1CCCC1N=[N+]=[N-] C1(CC#C)(C(N2CC(OCCNC(=O)CCc3cccnc3)C2)=O)CCCCO1 c1(CC(=O)NC2N(C3CCN(C(C(N)=O)=O)C3)CCCC2)nsc2ccccc12 C(=O)(C#CC1CCOC1)N1CCC(C)(NC(c2c(C)ccc(SC)c2)=O)CC1 c1(CCCC(=O)N(CC(C)(C)NC(C(C)C(C)(C)C)=O)C)nc2ccccc2[nH]1 C1(O)(C(C)NC(=O)Cn2cnnc2O)CCN(C(=O)CNC(=O)C(F)(F)F)C1 CCCC(CC(=O)NC(C)C(N)=O)NC(C1C=CCC1)=O N1(C(c2cc(C)[nH]n2)=O)CCC(C)(C)C1CNC(=O)CCN1CCCC1 Cc1cc(Br)ccc1CNc1c[nH]nc1C(=O)NCc1ccco1 CC1=CC(C)CN(C(=O)C(C)CNC(c2cccnc2N(C)C)=O)C1 c1(OC)cc(C(N2CCOCC(CNC(c3nnc(S)n3C)=O)C2)=O)cc(F)c1 N1(C(C=COCC)=O)CCN(C2CCN(C(C34CCC3CC4)=O)CC2)CC1 C(=O)(C(C)(C)C#C)N1CCC(CC(=O)N(CC#C)CC=C)C1.C1(=O)CN1C1CCC1 C1(N(C(C(CCC)NC(C)=O)=O)CCC)CCCN(C(=O)CCF)CC1 N1(C(CC=C)=O)C2CCC1CN(C(=O)C(C1CCOC1)NC(C)=O)C2 C12CC(C)N(C1)CN(C(=O)OC(C)(C)C)C2.C(C(=O)C1CCC1)(N(C)C)CC CC1CCCCC1(C)C(N1CCC(C(=O)Nc2ccccc2)C(C)C1)=O C1(C(N2CCC(C)C2CN(C(=O)C(C)CF)C2CC2)=O)CCc2cnn(C)c2C1 c1(C(N(CC(CC)NC(C2CN3CCN2CC3)=O)C)=O)ccc2c(c1)ncn2C C(=O)(CCCCC#N)N(CCCOCCN(C(CN1C(C)CCC1)=O)C)C c1(CC)nc(N(C2CCCN2C(=O)Cc2ncccc2C)CCOC)[nH]c(=N)n1 C12(NC(C3C(NC(Cc4cccc(C)c4)=O)CCOC3)=O)CC3CC(CC1C3)C2 C1(NC(N(CC(CCC)C)C)=O)CC(=O)N(C(=O)OC)C1c1ccccc1 C(=O)(N=c1cnn(C2CCOC2)[nH]1)N(CCC#N)CC C(=O)(C(O)CC[S+](C)C)NCC(CC1CN(C(CC(C(C)C)O)=O)C1)(C)C c1(NC(C2CCCC2c2ccccc2)CC)ccc(O)c(C)c1 C1(C(=O)NCC(C(=O)OCC)C)CCN(C(=O)C(CO)C(C)(C)C)O1 Cc1nccc(C(=O)NCC2CCC(NC(c3ccnnc3Cl)=O)C2)n1 N1(C(CCC(C)OC)=O)CC2CCC(C1)C2CNC(c1ccc(N)c(SC)c1)=O C(CCCCC(=O)NCC1CC1CNC(c1cccc(F)c1N)=O)OC c1(C(=O)NC(C)C(C)(C)NC(=O)CC2C=CS(=O)(=O)C2)ccc2nn[nH]c2c1 c1(C(=O)NCC(C2CCCCC2)NC(CC(C(C)C)O)=O)cc(F)cc(Cl)c1N CC(C)CC(C(=O)OCc1ccc(C(C)C(F)(F)F)cc1)C(C)C C1(C(N2CC(NC(=O)CC(=O)N(C)C)CC(C)(C)C2)=O)CC2OC(C)(C)OC2C1 c1(C(c2n(CCCC)nnn2)NCCn2ccc(Br)n2)cnc(N(C)C)cn1 C1(NC(CC2CC(C)N(C(C3CC=CC(O)C3)=O)C2)=O)CCOC2(CCC2)C1 N1(C(COCC)=O)CCC(=C(c2ccco2)C(C)C)C1 Cc1c(C(=O)NCC(C2CCCC2)NC(=O)CCC2NC(=O)NC2=O)ccn1C c1(C(N(CCCNC(C(C)C(F)F)=O)C2CC2)=O)n[nH]c2c1CC(F)(F)CC2 N1(C(Cn2nc(C)oc2=O)=O)CC2(CCN2C(=O)C(c2ccc(Cl)cc2)CO)C1 c1(CC(=O)NC2CCC(NC(c3c(C)ccc(N)c3)=O)C2)ccc([N+](=O)[O-])cc1 N1(C(c2cc(C)oc2)=O)CCCN(C(C2CCN(CCO)C(=O)C2)=O)CC1CO C1(C(=O)NCCN(C(=O)CC2=CCN(C)CC2)C(C)C)CCCN1S(=N)(=O)N(C)C c1(C(=O)NCC(CC=C)NC(=O)CC(C)(CC)CO)cc2ccncc2cc1F C1(NC(C(CO)OC)=O)CN(C(=O)C(c2ccccc2F)F)C2CCCC12 CCC(CNCC1(c2cccc(F)c2F)CCCC1)(CC)CO Cc1ccc(C)c(CC(=O)NCCNC(=O)C(c2cccc(Br)c2)C)c1 C12(C(=O)NCC3C(NC(c4c(CC)occ4C)=O)C3)CCC(CC1)C(C)(C)O2 C1(C)(CNC(C2N(CCC)C(=O)CC2)=O)CCN(C(C2(CC)CC2)=O)CC1 C(=O)(C1=C(CC)OCCS1)NCC(CC)(CC)NC(=O)CC(C)(F)F N1(C(c2cc(C(C)C)on2)=O)CC2CCC(C(N3CCC(F)(C(N)=O)C3)=O)(C2)C1 n1(CC)nc(C)c(C(=O)NC2CC(CC(N3CCCC(C)CC3)=O)C2)c1C C(=O)(CCCCCNC(=O)C(C)(C)C)N1CCC(C(C)O)C1 C12(CNC3(c4nnnn4CCOCCO)CCCC(C)C3)CCC(CC1(F)F)C2 c1(CNC(C2(NC(Cc3ncn(C)c3)=O)CCC2)=O)cc(F)ccc1O CCCC(C(=O)NCCCOCCCNC(c1ccoc1Cl)=O)c1ccccc1 CC1Oc2ccccc2N(CCC(=O)Nc2cn(C)nc2Cl)C1=O C=CCC(CNC(=O)CCn1cccc1)NC(c1ccc(C2CCOC2)s1)=O c1(C(=O)NC(C)CNC(=O)Cn2ncc(Br)n2)cc2c(Cl)cccn2n1 c1(C(N2CCCC(N(C)C(C3CCC(F)(F)CO3)=O)C2)=O)ccn2ccccc12 N1(C(C2(OC)CCSC2)=O)CC2(CCCC(CNC(=O)CCCOC(C)C)O2)C1 N1(C(c2scc(OC)c2)=O)CC(C)(C)CC1CNC(c1cc(C)sc1C)=O c1(C(N2CCN(C(C(CCC)C(C)C)=O)C(C)CC2)=O)cccc2c1C(=O)CC2 N1(C(C(C2CC(NC(C(CCC)C#N)=O)C2)F)=O)CCN(C)C(C)(C)C1 CC1(C)CC(=O)NC1CNC(c1nnnn1C1CC1)CCC1CCCC(=O)N1 CC(C)CC(O)C(C)C(=O)NCCOCCNC(c1ccc2cncnc2c1)=O C1(CCNC(C2CC2F)=O)CC(F)(F)CN1C(c1ccc(F)s1)=O N1(C(CC(C)C)=O)CCN(C(C2CCC(CC(F)(F)F)CC2)=O)CC(C)(C)C1 C(=O)(C#CC1CCOCC1)NC(CNC(C(c1cccc(C(F)(F)F)c1)CC)=O)C c1(C(N2C(C(=O)NC3CCCN(C)CC3)CC3CC32)=O)ncc2ccccn12 C1(CNC(C(C)CF)=O)CCC(NC(=O)CC2(NS(C)(=O)=O)CCCCC2)CC1 c1(-n2cc(C(=O)CCSCCOC3CCC3)nn2)cccc(C(C)(C)OC)c1 N1(C(CCc2cc(C)no2)=O)CCC2CCC(C1)N2C(=O)C=CCF N1(C2(C(=O)NC3C(CNC(=O)CSCC4CCCO4)C3)CC2)CCNC1=O C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1C)N2C(=O)CC(C)n1ccnc1 c1(C(=O)NC2CCN(C(C3C(C)CC3)=O)CC2)ccc(F)cc1O C(C(=O)NCc1cc(OC)ns1)(C(C)O)NC(c1cnc(OC)s1)=O c1(C(=O)NCCC(CC)(C)NC(c2ccc(OC)cc2F)=O)cc(C)ccc1C C(=O)(C1CCCc2nn[nH]c21)N(C1(CNC(=O)CN2CC3CC3C2)CCCC1)C Cc1scc(CNC(=O)COC2CN(C(C3(C#N)CC=CC3)=O)C2)c1C C1(OC)CN(C(=O)C(=Cc2cn[nH]c2)C)CC1C(=O)NC1CCC(=O)NC1 C1(NC(=O)Cc2c(CN(CC)CC)csc2)CC(NC2(C3CCC3)CC2)CCO1 C(=O)(CS(=O)(=O)CC(F)(F)F)NC(CN(C(C(c1c(C)nn(C)c1)O)=O)C)C CC(C)CCCC(C)C(=O)NC(C)CNC(=O)Cc1ccc(F)cn1 C1(CNC(c2nc(C3CC3)cs2)=O)CN(C(c2cnoc2)=O)CCO1 C1(C)(NC(c2c(C)occ2)=O)CCCN(C(=O)CC2CCCOC2)C1 C(CN=c1cccc(S(=O)(=O)NCCn2ccnn2)[nH]1)NC(COC)=O Cc1nc(C(N2CCCC(CN3CCOCC3)C2)C(=O)N(C)C)nn1C CC(CNC(=O)CCC1CCOCC1)CN=c1[nH]cc(C#N)c2ccsc12 C(=O)(CC(O)C(Cl)(Cl)Cl)NCCN1CCCN(C(CC)=O)CC1 N1(C(COCCCC#C)=O)CCCC(CCCCNC(C2CCN(C)C2)=O)C1 CCCCC(CC)CCC(=O)NCCC(C)(C)NC(C1CC(=O)NC(=O)N1)=O N1(C(C(c2ccnn2C)NC(Cc2cn(CC)nn2)=O)=O)CC(CO)CC1CO c1(C(=O)NC2CN(C(C(C3CCCCC3)C)=O)CC2F)cc([N+](=O)[O-])ccc1Cl C(N=c1[nH]c2cc(Cl)ccc2s1)C1(CNC(c2n[nH]c(O)n2)=O)CC12CCC2 C1(C(N(CCNC(Cc2ccn(CC)n2)=O)C2CC2)=O)CC=C(C)CC1 C1(CCNC(CC2(C)CCN2C(c2cc(Cl)c[nH]2)=O)=O)CCCC2CC12 C1(CC(=O)N(C2CCN(C(=O)Cc3cc(F)ccc3O)C2)C)CC(C)(C)CCO1 N1(C(C2N(C(C(C)NC(N)=O)=O)CCCCC2)=O)CCn2cnnc2C1 Cc1cn2ccc(C(=O)NC(C)CCNC(c3cc(C)n(C)c3C)=O)cc2n1 C(=O)(CC1=CCN(C)CC1)NC(CCOC)CNC(=O)C(F)(F)c1ccccc1 c1(C(=O)NC(CNC(C2C(COC)C2)=O)C(C)(C)C)nc2ccc(C)cn2c1N Cc1nccc(C(=O)NCC(C)(C(C)C)NC(c2cccc(OCF)c2)=O)c1C C1(NC(C(C)N(CC(F)(F)F)C)=O)CCCCCN(C(c2cnc(O)n2C)=O)C1 C(C(=O)NCC(C)CNC(c1ncn(C)n1)=O)(C(C)C)NC(=O)OCC C1(C(=O)NCC(C)NC(c2c(C(F)(F)F)cnn2C)=O)CC12CC(C)(C)C2 C=CCC(CC)C(=O)NCC1CN(C)CCN1C(c1cnc(C2CC2)s1)=O C=CC(C)(CC)C(=O)N1CC2CC(NC(=O)C(C)Cc3cccc(F)c3)C2C1 C(=O)(C(CN(C(=O)Cn1ccnc1)C1CC1)C(C)C)N(CC(N)=O)CC C1(CNS(CC(N2C(c3c(C)cccc3)C(O)CC2)=O)(=O)=O)COCC(C)(C)O1 CN1C(=O)CCCC1C(=O)NC1CCN(C(=O)C(=O)NCC(F)F)CC1CO N1(C(c2c(C)n[nH]c2C)=O)C(C)CC2CN(C(c3ccc4ccnn4c3)=O)CC12 C=CCC(CNC(=O)COCC1CCC1)C(=O)N1CCC12CC(O)C2 c1(C(N(CC(=O)NCCCCSc2nc[nH]n2)C2CC2)=O)cscc1F c1(C(=O)NC(CNC(C2(CC)CCC2)=O)C2CC2)cccc(C2CC2)n1 c1(NC(Cc2cccc(NC(Cc3ccc(C)nc3)=O)c2)=O)cnc(Cl)c(C)c1 N1(C(C2C(=C)C2)=O)CCOC2(CCN(C(=O)Cc3cccc(OCC)c3)C2)C1 Cc1cc(C(N2CC(C(C(=O)NCCN3CCOCC3)N(C)C)C2)=O)c(C)nn1 C1(NC(C(CCF)NC(c2cn(CC)nc2C)=O)=O)CCC(=O)N(C)C1=O CC1(C)CN(C(c2cc(C(N)=O)no2)=O)CC1NC(=O)Cn1cnccc1=O c1(C(N2CC3C(NC(CC(c4c(C)noc4C)C)=O)(C3)C2)=O)cc2n(c1)CCC2 N1(C(c2c(CC)nc[nH]2)=O)CC(NC(c2cc3scnc3[nH]2)=O)CC2(CC2)C1 C(=O)(CC(C(F)(F)F)N(C)C)N(CC1(F)CC(C)C(N(CC)CC)C(=O)NC1)C C(C(CC(=O)N1CCC(C)(N(C)C)C1)NC(C1CC(F)(F)C1)=O)OC c1(CC(N2CCC(C(C)NC(c3c(SC)nn(C)c3)=O)C2)=O)cc(Cl)ccc1Cl C=CC(CC)CC(=O)NC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)C1C(CC)C1 Cc1nc(Br)cnc1NC(=O)CC1CCN(Cc2cc(CO)ccc2O)CC1 C1(NC(CCN(C)CC)=O)CN(C(c2cc(Cl)cnn2)=O)C2(CCCOC2)C1 C1(C(=O)OC)CCN(C(=O)CNc2cccc(OC(C)(C)C)n2)C2COCC12 c1(C(=O)NCC(CCNC(C=C(C)C)=O)O)cc(Cl)ccc1OC(F)(F)F c1(SC)cc(C)c(C(=O)NC(C2CCN(C(=O)Cc3cn[nH]c3)C2)C)o1 c1(C(=O)NCC2(CCNC(C(C)SCCCC)=O)CC2)ncc(F)cc1C N1(C(C(F)=C(C)C)=O)CC(F)(F)CC1CCNC(c1ncoc1C1CC1)=O Cc1ccc(NC(c2ccn(C(F)F)n2)c2nnnn2CC(F)F)c(F)c1 C1(O)(CNC(C2(NC(N)=O)CC2)=O)CCCN(C(c2ccon2)=O)C1 Cc1nc(C(=O)NC2CC(F)CN(C(C3CCC(O)CC3)=O)C2)c2n1CCCC2 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(OC)C(NC(c2cc(Cl)n(C)n2)=O)CC1 c1(N(C)C)nc(F)ccc1CNC1CC(CC(N2CCCC2CC#N)=O)C1 c1(NC(C2CCC(C)N2C(c2c(O)ccc(Br)c2O)=O)=O)cc(Cl)c(Br)cc1Cl N1(C(c2ccc(C(F)(F)F)cc2Cl)=O)CCC2(CCN(C(C3CCSC3)=O)C2)C1 C#CC1(NC(C2(CNC(=O)C(O)CCSC)CC3(CC3)C2)=O)CCC(C)CC1 N1(C(c2c(OC)n[nH]c2)=O)CCOCC1C(=O)NCC(C)C(C)(C)C c1(C(=O)NCCN(c2nnc(CO)s2)CC)c(C)oc(C)c1C C1(NC(CCN(C)CC)=O)CC2CC(NC(=O)C(C)Cc3ccccc3F)CC12 c1(C(=O)NCC(C)CNC(=O)CC2CC2)nc(C(F)(F)F)oc1Br c1(C(=O)NCC(C(C)C)NC(=O)CCc2ccc[nH]2)cccc2occ(Br)c12 C1(CC(=O)NCC2CCN(C(CC3CCC(C)C3)=O)C2)NC(=O)NC1=O C1(NC(C2CC(=O)C2)=O)CC(O)CN(NC(C2CC(Cc3ccccc3)C2)=O)C1 N1(C(C(c2c(C)noc2C)C)=O)CC2CC(NC(c3cn[nH]c3)=O)C1C2 Cc1ccccc1C=CC(=O)NC1CCOC1C(=O)Nc1cncnc1O CC1CC(CNC(C2(c3cccc(F)c3)CCCCC2)=O)CN1C(=O)CN(C)C n1(CCC(=O)NCC(CNC(=O)C(O)CSC)OC)ncn(C)c1=O C1(C)(C(=O)NCC(CN(C(=O)CNc2ccccn2)C)O)CC1(F)F C1(CNC(=O)C=C2CC2)COC(CNC(=O)CCc2ccon2)C1 c1(C(N2CC(O)(CNC(C(n3cncn3)OC)=O)C2)=O)nccnc1C(F)(F)F Cc1ncc(C=CC(=O)NC2(CNC(c3cnc[nH]3)=O)CCCC2)c(O)n1 N1(C(=O)N(CC2(C)CCC2)C2CC2)CCCCC1c1cccc(O)c1 CC(C)CS(=O)(=O)NC1CC2(CCO2)C1 C1(CC(N2CCC(C(C)(C)NC(=O)Cc3cnco3)C2)=O)CCCC(F)(F)C1 Cn1cnc(C=CC(=O)NC2CC23CC(NC(C2(C(N)=O)CCC2)=O)C3)c1 Cn1nc(CN2CCC(C)(C)C2)cc1C(C1CCCCO1)=O.C1(=O)CO1 C=C(C)CC(C(=O)NC1CC2CC(NCc3ccc(=O)n(C)c3)C2C1)NC(C)=O N1(c2n(CCC#C)c(C3CC3c3ccccc3Br)nn2)CC2(C1)CC(C)(O)C2 C1(C(N2CCC(C(=O)NC)C2)C(=O)NCC)CCC2COCCC2C1 C1(c2n(C)ncc2)COCCN1.c1(Cc2ncon2)cn(C)nc1Br C(CNc1ccc(N2CCC(C)CC2)c(Cl)c1)(CCS(C)(=O)=O)OC CC1CN(C(c2ccnc(C(C)(F)F)c2)=O)CCC1NC(=O)CCN(C)CCO C1(OC)CC2(C1)CC(C(=O)NC(C)CCNC(=O)CC(CC)OC)C2 C1(F)(CNC(C(c2cccs2)SC)=O)CC(NC(c2cnccn2)=O)C1 C1(C(C)C)CN(C(C2CCCCS2)=O)CCN1C(=O)CC1CCC(C)CC1 c1(-c2cc(C(=O)NC(C)CNC(C3CCCS3)=O)sn2)ccc(Cl)cc1 C1(Nc2cc(OCC)ncn2)CC2(CCN(C(c3cc(Cl)ccc3C)=O)C2)C1 c1(CC(=O)NC23CC2CN(C(=O)C=Cc2cnccn2)C3)ccccc1C(F)(F)F c1(C(C)C)nc(Cl)sc1C(=O)NC(CNC(c1ccncc1F)=O)C1CC1 C=C(Cl)C(C)(C)C(=O)NCC(CC(C)C)NC(c1ccc(OCCOC)nc1)=O C1(O)(c2n(CC)c(N(Cc3ccccc3)CC3CCC3)nn2)CCC(C)(C)CC1 CN1CCCC(C(N2CCCC2C(C)(C)C(=O)NCCC2CCCOC2)=O)C1 C1(NC(=O)CC(F)(F)F)CN(C(=O)C=Cc2cccc(Cl)c2)CC2CCCC12 c1(SCC)ccc(C(N2CC(OC)CC2CNC(C2CCC(C)O2)=O)=O)cn1 c1(CCC)n[nH]cc1C(=O)NCC(CC)NC(=O)CC(C)N(C)C C1(C(=O)NCC(C)(C)NC(=O)C(F)=C2CCC2)CCCN1C=O c1(OC)ncc(C(=O)NCC2CC(OC)CN2C(=O)Cc2cccc(C)c2)cn1 C1(CNC(C(C)OC(C)(C)C)=O)CCCC2CN(C(=O)CC3CC3(F)F)CC12 C1(C)(CC)CN(C(=O)C(C)(O)CN(C)C)CCO1 c1(C(N(CC(CN(C(COCCC(C)C)=O)C)O)C)=O)n[nH]c2ccc(Cl)cc12 C(=O)(C(CC(F)F)NC(C1CC(C)(C)C1)=O)NC1(C)CS(=O)(=O)C1 C1(NC(CC2C(C)C(=O)CC2)=O)CN(C(c2snc(O)c2Cl)=O)CC12CC2 C1(CNC(C(=O)NCC)=O)CC2CC1CN2C(c1cc(C)nn1C(C)(C)C)=O C1(N(C(=O)C=C2CC2)CC)CCCN(C(=O)C(C)OC)C1 C1(C(N2CCC(=C)CC2)=O)CN(C(=O)C(CO)N(C)C)CC(C)(C)C1 N1(C(CC(=C)Br)=O)CC(CNC(=O)COC2CCOC2)C2(CCC2)C1 c1(C(=O)OC)cnccc1N1CC2C(CNC(c3nccnc3C)=O)C2C1 N1(C(=O)CCOCC(F)F)CC2CC1CN2C(c1nccc(Br)c1O)=O N1(C(C2C(NC(c3nc(C)sc3)=O)CC2)=O)CCCC2NC(=O)CC12 c1(C(C)N(C(=O)CCc2cnn(C)c2)CCNC(=O)CC2(O)CC2)ccc(Cl)nc1 N1(C(C(C(C)C)(C)O)=O)CC2C3CCC(C2C1)N(C(c1cccc(F)c1O)=O)C3 C1(CCNC(C2C(C)C2C)=O)CN(C(c2n[nH]cc2Cl)=O)CCS1(=O)=O C(c1ccc(C(N)=O)o1)=CC(=O)N(C1CC(NC(CC(C)F)=O)C1)C C1(CNC(c2cc(=O)n(Cc3ccccc3)[nH]2)=O)CC(F)CN1C(CNC)=O.CO CCC(C)(C)CC(=O)NC(C)C(C)NC(c1ncoc1-c1cnn(C)c1)=O C1(NC(c2ccc(SCC3CC3)cc2)=O)CCCCN(C(=O)CCCC2CC2)C1 N1(C(C(C)N(C(c2ccc(C(C)C)o2)=O)CC)=O)CCCC(C(C)C)CC1 c1(C(N2CC3CN(C(C(C)(C)F)=O)CC(C2)O3)=O)cc2c(nc1O)CCCCC2 N1(C(c2c(C)ncs2)=O)CCOC(CC(=O)NC(C)CC(=O)NC(C)C)C1 C1(NC(CN(CC)CC)=O)CCCN(C(=O)CCCOC(C)(C)C)C1C N1(C(=O)Cn2nnc(C3CC3)n2)CC(NC(C23CC(F)(C2)C3)=O)CC(O)C1 N1(C(CC(=C)C)=O)CCC2(CCN(C(=O)C(C)C(F)F)CC2)C1 C#CC1CCN(C(=O)OCC)C1.c12nc(C)c(s1)C(C)N2C N1(C(c2c(OC)cccc2OC)=O)CC2(C1)SCCC2NC(=O)CSC1CC1 Cc1ccc(O)c(C(N2CCCCC2c2nc[nH]n2)=O)n1 c1(C(=O)NC(C2CCN(C(C(C)=C3CC3)=O)C2)(C)C)ccc(C(C)=O)cn1 Cc1oc2ccccc2c1C(C)N(C)C.C12(S(=O)(=O)Oc3cnn(c3)CCS1)CC2 N1(C(C2CC=C(C)CC2)=O)CCC(C2CC2)(CNC(=O)Cc2ccoc2)C1 c1(N2CCC(NC(c3cc4ccc(Br)cc4s3)=O)C2)ncc2cccc(O)c2n1 C1(C(=O)NC2CC(CNC(=O)C3=CCCOC3)C2)CCn2c(O)nnc2C1 N1(C(C2(C)N(C(c3nc(C)sc3C)=O)CC=C2)=O)CCC2(CC(CO)C2)C1 c1(OC)ccc(-c2cnc(CNC(c3ccc(N(C)C)nc3)=O)nc2)c(C)n1 N1(C(C2C(C)(C(F)F)C2)=O)CC(CNC(c2cnoc2C2CC2)=O)C2(CCC2)C1 O=S(=O)(c1cc(OC(F)F)cc(F)c1)NCC1(O)CCCCCC1 N1(C(c2ccc(C(N)=S)cc2)=O)CCC(C2(O)CCC2)CC1 c1(C(N2CC(c3cn(CCOC)nn3)OCC2)=O)cc(N)cnc1Br CC1CCC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)C(C)CO)C1 c1(C(=O)NC2C(CNC(C3(C)CC3(F)Cl)=O)CCCC2)c(F)cccc1[N+](=O)[O-] C1(CNC(CNC(=O)OCC)=O)C(C)CCCN1C(=O)Cc1sccc1C C1(C(N(C2CCN(C(CC(=C)Br)=O)C2)C)=O)CC2OC(=O)OC2C1 CCCCCC(=O)NCC1C(C)CCN1C(=O)Cc1nocc1C(C)C c1(N2C3CC(=C)CC2CC3)nc(=NCSC2(OCC)CCC2)[nH]c2c(F)cccc12 CC1COC(C)(C)CN1C(Cc1ccccc1)C(=O)NCCC#N Cn1ccc(C(N2CC(NC(c3cn(C4CC4)cn3)=O)CC3(CC3)C2)=O)c(O)c1=O c1(NC(C2(CSC)CN(C(=O)C(O)C(F)(F)F)C2)=O)ccc(F)c(Cl)c1 Cc1[nH][nH]c(=NC(=O)C2CN(C(c3ccc4n[nH]cc4c3)=O)C2)c1Br C1(CNC(c2cccc(SC)c2)=O)C(C)CCCN1C(=O)CCC1CCC1 N1(CC(=O)NC2CC(F)(CNC(C3(CC4CC4)CCC3)=O)C2)CCC(CO)CC1 C1(C(NOCCC(C)C)=O)CN(C(=O)CCc2cccnc2)CCC1(C)C C1(CCOC)(C(=O)NCC2CC2Cl)CCN(C(C2CCCCN2C)=O)CC1 S(=O)(=O)(c1ccc(NC2CC(CF)C2)cc1Br)NC(CC#CC)C C1(NC(C(C(C)O)(F)F)=O)CC2(CCCCN2C(c2cnncc2O)=O)C1 c1(OC)ncccc1CC(N1CCC(NC(c2cccc(C(C)(F)F)n2)=O)C1)=O c1(C(=O)NCCCN(C)C(C2OCCC2c2cnn(C)c2)=O)ccccc1Cl c1(NC(=O)NC(c2cc(OCC)c(OC(F)F)cc2)C)ccc(S(C)=O)cc1 Cc1nccc(C(=O)NC2(C(=O)N(C(C)CN(C)C)C)CCN(C)C2)c1C N1(C(C2N(C(C)=O)CSC2)=O)CCCCC1CCCNC(=O)CC1COCCO1 C1(COC)CN(C(c2cccc(SC)c2)=O)CCN1C(=O)C(C)C(F)F c1(N(C(=O)C(CC)C2CCC(=O)N2)CCC)cccc(N(C)C)c1 c1(CN(c2cccs2)CCOC)ccc(OC)c(-c2cccc(C)c2C)c1 C1(=O)CCO1.C(C(=O)OCC)OCCOCC N1(C(C=C(C)CN2CCOCC2)=O)C2CCC1C(NC(=O)COCCCF)C2 C(=O)(C1=CCCN(C(=O)CSCC=C)C1)NCCC(CC#C)C C(C)(C)(CCCCC(=O)NC1C2CN(C(c3nnc4ccccn34)=O)CC12)OC c1(Cn2c(N3C(C)CC(C4CC4)C3)nnc2-c2ccc[nH]2)occ2c1CCOC2 N1(C(C2CCCC(=O)N2)=O)CC2(CCC2NC(=O)C(=C2CCCCC2)F)C1 N1(C(CC(CC)(F)F)=O)CCOCC12COCCN(C(=O)CCC(C)O)C2 C1(NC(C(CC)C#N)=O)CCN(C(C2CN(CP(C)(C)=O)C2)=O)CCC1(F)F c1(C(N(CCNC(c2nnn(COCC)c2N)=O)C)=O)ccc2c(c1)CN(C)C2 CN1CCCCC1COC(C1CCCN1C(c1cc(Br)cn1C)=O)=O N1(C(CCCC#CC)=O)CCC2(CC1)CC2CNC(C1CC1OCC)=O O=C(N1OC2C=CC1CC2)C1CCN1C(C1(F)CC=CCC1)=O N1(C(=O)CSCCN2CCOC2=O)CCC(CO)C1c1ccccc1 Cc1ncc(Cl)cc1CC(N1CCC(NC(=O)CC2CNC(=O)C2)C(O)C1)=O c1(NC(C(CN(C)C)NC(c2n(CC)c(O)nc2)=O)=O)c(C)cc(C)cc1C c1(CC(=O)NC(C2CN(C(=O)C=Cc3cn[nH]c3)CCO2)C)cc(F)ccc1O c1(C(N2CCCC(c3c(C(=O)OCC)con3)C2)=O)cnc2c(Br)cccc2c1 Cc1cc(C(=O)NCCC2(NC(=O)CCC3CCC(=O)N3)CCC2)c(C)cc1Cl c1(N2CC3C(C)C3C2)ccc(Br)c(S(=O)(=O)N2CCOCC2C2CCCO2)n1 C1(CC(N2CC(NC(C(C)CSCc3ccccc3)=O)C2)=O)CCCS1(=O)=O CC1(C(=O)NCC2(CCNC(c3cncnc3)=O)CC2)CCC(=O)NC1 C1(C(=O)NC2CCCC2NC(=O)CCS(C)=O)(NC(C)=O)CCCCC1 C(=O)(C1=CCCOCC1)NCC12CN(C1)C2.c1(OOC)c[nH]c2nccc-2c1 N12CCCN(CC1)C(=O)c1cc2ncn1.C1(OC)CC(c2ccccc2)CO1 CC1CC(N=c2[nH]c(-c3ccccc3)nc(=NCC3CC3)[nH]2)CN1C1CC1 c1(C(=O)NCC2N(C(C=CC=CC)=O)CC2)ccc(N)cc1Cl Cc1ccc2c(c1CO)CCCN2CC(c1cccc(C#N)c1)O c1(N2CCC(NC(C3CC3C(=O)OC)=O)C23CCC3)nc2ccc(N)cc2s1 c1(C(=O)NCCCNC(c2cc(-c3cccnc3)on2)=O)sccc1F C1(C(=O)NC(CN(CC)CC)C)CC2CC1CC2NC(c1ncnc(C)c1C)=O c1(CC)nccnc1NC(C1(SC)CN(C(=O)CC2CCC3CC23)C1)=O C1(NC(C(CC)(C)OC)=O)CC2CC(NC(c3[nH]ccc3C3CC3)=O)C2C1 N1(C(CC(C)N2CCCC2=O)=O)CCN(C(=O)COCC(F)(F)F)CC12CC2 c1(C(=O)NCC(C)CN(C)C(C2CCS(=O)(=O)C(C)C2)=O)ccc2nn[nH]c2c1 c1(CN(CCNCc2ccnc(-c3ccccn3)c2)CC)cnc(Cl)c(F)c1 N1(C(C(CC(C)C)ONC(=O)C2CC=CC2)=O)CCC2(CCOC2)C1 C1(NC(c2n(CC)ccn2)=O)CCC(N(C)C(c2cocc2C(N)=O)=O)CC1 c1(OCCNC(c2ncc(C(N3CC(NC(C)=O)C3)=O)o2)=O)ccc(F)nc1 N1(C(C=CCC)=O)CC2CC(NC(c3cc(Br)n(C)c3)=O)C(C2)C1 O=C(C#CC1CCCOC1)NCCC1CN(c2ncnc(Cl)c2F)C1 CC1CCCCCC1NC(=O)CCOCCCNC(=O)CC1OC(C)(C)OC1=O C1(CCOC)CN(C(c2cc(O)nc(C)n2)=O)CCN1C(C1CC(C)(F)C1)=O c1(C(C)C)n[nH]c(=NCC2CC(NC(c3ccc(NC(N)=O)cc3)=O)C2)o1 C1(C(=O)NCC=C(C(=O)N(C(CC)C)CCO)C)CC=CCC1C C1(CC(=O)NCC(C)CNC(=O)C=Cc2ccc[nH]2)COC2CC1C2 c1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)cc(C)ccc1N N1(C(C2C(C)C2)=O)CC2CN(C(=O)C(C)(C)C(F)(F)F)CCC12 N1(C(N2CCCC2c2cc[nH]n2)=O)CCOCC1CCc1ccccn1 N1(C(C(CC)C)=O)CCN(C(=O)CCc2nc(C(C)C)no2)C(COC)C1 C(=O)(C1=NOC2(CCC2)C1)N(CCCCNC(=O)Cc1cc(F)ccc1F)C c1(C(=O)O)nn(-c2ccccc2)cc1C(N1CC(C(=O)O)CC1C(F)(F)F)=O Cc1cc(=O)ccn1CC(=O)NCCC1CN(C(=O)CC2(O)CCC2)CCO1 O=C(CCCCCNC(C1(O)CCSC1)=O)NC1CC(CSC)C1 c1(C(=O)NC2CC(CO)N(C(=O)Cc3cc(Cl)ccc3Cl)C2)csc2nnsc12 C1(CC(N2CC(CNC(C3(CC)CC(C)(C)C3)=O)C2)=O)CCCCC1(F)F C1(C(N2CC(C(C)NC(c3c(C(C)C)noc3)=O)C2)=O)CC12CCC(F)(F)CC2 CCCC(C(=O)N(C)CC1CC1(C)C)NC(=O)C(C)OC(C)=O C(C1=CCN(C(=O)C(C2CCCN(C)C2)(C)C)CC1)NC(Cc1c(C)noc1Cl)=O c1(C(=O)NC2(C)CC(NC(C3COCCC3(F)F)=O)C2)ccc(=N)[nH]c1Cl N#Cc1ccc(C(=O)NCC#CCNC(c2cc3c(s2)CCC3)=O)c(F)c1 C(=O)(CCS(C)(=O)=O)NCC(=O)NC1CCC(NC(C(CCC)C)=O)C1 C1(C(=O)NCc2c(C(=O)NOCc3ccccc3)cccn2)CCCC(F)C1 C1(CNC(CC(=C)Br)=O)CCN(C(c2nc(CC3CC3)cs2)=O)CC1C N1(C(C(CO)NC(C2C(C)N(C)CC2)=O)=O)CC(CO)C(C2CC2)C1 N1(C(C(C)SCC)=O)CC2(C)CC1(C(=O)NC(CC)CC(F)(F)F)C2 Cc1oc(CO)cc1C(=O)NC1(CC(=O)NC2CCN(CCCO)C2)CC1 N1(C(C=C(C)Cl)=O)CCCCC(NC(c2cc(Cl)c(Cl)cc2O)=O)CC1 C1(CNC(N2C(C)CC(C(=O)OC)C2)=O)CCCCCC1C1CC1 c1(C(N(C(C)CNC(c2cn(C)nn2)=O)CC)=O)cc(Cl)ccc1C c1(C(N2CC(NCc3ccncc3Br)C3(CC3)C2)=O)ccc2ccccc2c1Br N1(C(C(CCSC)O)=O)C2CCC1C(CNC(c1oc(C)nc1C(F)(F)F)=O)C2 c1(OC)cncc(C(=O)NC2COCC2NC(=O)CSc2c(C)n[nH]c2C)c1C C1(NC(C2CC(C)NC(=O)C2)=O)CN(C(=O)C(C)(C)c2ncco2)CC12CCC2 C1(NC(CCNC(=O)NC)=O)CC2CC(NC(C3CC34CC(C)(C)C4)=O)CC2C1 c1(C(=O)NCC2C3CN(C(C4CC(C)OC4)=O)CC32)c(Cl)nc2ccccn12 CCC(C(=O)NC1CCCC(NC(=O)Cc2ccc(F)c(F)c2)C1)C(C)(C)CC C1(C2CCCN(C(=O)Cn3cnnc3)C2)(NC(c2cnn(C)n2)=O)CC1 Cc1cc(NC(c2nn(C)c(C)c2Cl)=O)ccc1NC(c1[nH]nnc1C)=O C1(CNC(c2c(SC)snn2)=O)CC12CCN(C(=O)C(=Cc1cccs1)C)CC2 N1(C(c2ccc(OC)c(Cl)n2)=O)CCC2(C1)CN(C(c1ocnc1C)=O)C2 C1(CCC)(CNC(C2(C(C)(F)F)CCC2)=O)CCCN1C(=O)C(CCOC)OC n1(CC(=O)N(CCCN(C(CC(COC)(C)O)=O)C)C)ccc2ccc(F)cc12 C1(NC(C(C)NC(=O)C(N2CCOCC2)C)=O)C2CCCC1COC2 C(CC(C)CC(C)(C)C)NC(c1c(CNC(c2ccc(C)c(C)c2)=O)n[nH]c1)=O c1(CCCC)nc(C)c(CC(N2CCC2CNC(=O)C(C)=C(C)C)=O)s1 c1(C(=O)NC2CN(C(c3n(C)ncc3)=O)CC2F)nccn2ccnc12 N1(C(C2CC(SC)C2)=O)CCCC2(C1)CN(Cc1ccsc1)CCO2 C=C(C)C(C)(C)C(=O)NC1C2CC(NC(C3CCC(F)C3)=O)CC12 c1(CC)cc(C(N2CCC(C)C2CNC(c2ncoc2C)=O)=O)c(C)nn1 CCC(C(=O)NC12CCCC1N(C(c1ccc3nncn3c1)=O)CC2)C(C)(F)F c1(C(=O)NCCCCNC(c2cnn(C)c2N)=O)cc(Br)cnc1O N1(C(C(SC)SC)=O)Cc2occ(C(N3CCC(C(C)(C)C)C3)=O)c2C1 c1(C(=O)NC(CN(C(CNC(=O)NC)=O)CC)C)cncc2ccccc12 CC(C)CC(C)C(=O)N(CC(C)(C)C(=O)N(C(C)C(C)C)C1CC1)C N1(C(C#CC)=O)CCN(C(=O)C(c2cncc(C)n2)N2CCOCC2)C(CC)C1 c1(CNC(C2(CNC(=O)CCn3ccc(C)n3)CC(=C)C2)=O)c(C)cnn1C c1(OC)cc(C(=O)NCC2CC2NC(C23CC2COC3(C)C)=O)cc(C)n1 c1(N(CC(C)NC(C2CS(=O)(=O)CC(=O)N2)=O)C)ncc([N+](=O)[O-])cc1Cl C1(C(=O)NC2CC(CC3CC3)C2)CCCN(CC2CC2)C1.c12nnnn1C2 c1(C(=O)NCc2ccc(C(=O)N(CCCl)C3CC3)cc2)cc([N+](=O)[O-])c(O)cc1F Cc1cc(F)cc(NC(C2CC(CNC(=O)CC3CC4(CCC4)C3)CO2)=O)c1O C1(F)(C(=O)NCC=CC(=O)NC(C2CCCO2)CO)CCCCC1 CC(F)(F)CCC(=O)NCC1CCCC1NC(=O)C(O)CC1CCCC1 C(CCC(C)C(=O)NCC=CCC(N1CC(=O)NCC1C)=O)OC c1(C(=O)NC(CCCC)CNC(C2CCC(C)(C)C2)=O)ccc(C2CC2)c(F)c1 CCC(CC)C(C(=O)NC1CC(O)(CNC(=O)CC2C(C)(C)C2(C)C)C1)OC CC1=C(C(=O)NC2CCN(C(=O)C=CC3CCCO3)C2(C)C)CCC1 c1(C(C)C(=O)NC(C2CCN(C(C3CN(C)C3)=O)CC2)C)noc2ccccc12 Cc1cn(CC(=O)NC2CC2CNC(c2nnsc2C2CC2)=O)c2ccccc12 C1(NC(CCCOCCC)=O)CCCN(C(c2ccc(C)c(C)c2)=O)C1C c1(CC)oc(C)cc1C(=O)NC1CCC(CNC(=O)C(CCO)N(C)C)C1 CC1SCCN(C(=O)CC2(NC(c3cc(C4CC4)nn3C)=O)CCC2)C1C C1(NC(C(CC)C)=O)CC1C1CCN(C(c2cc(NC(C)=O)ccc2F)=O)CC1 C(=O)(C(C)(C)CSC)NCC(CC=C)NC(C1C(CCC)C1)=O Cc1nccc(C(N2CCN(C(=O)C(O)CC3CCCC3)C3CC23)=O)c1O O=C(CCCCCCCO)NCCc1nc(-c2cc3cc(Cl)ccc3o2)no1 C1(C)(CNC(c2cc(SC)oc2)=O)CCN(C(=O)CCC2CCCCO2)C1 C(=O)(C(C)CC(C)CC)N(c1cccc(C(NOCCOCC)=O)c1)CC C(CC(C)C)(C(=O)NCc1ncccc1C(=O)N(C)CC1(O)CCC1)OC C=CCC(CC(C)C)C(=O)N(CC)CC1CCCN(C(c2cnncc2C)=O)C1 c1(CN2CCC(O)(C(=O)Nc3cccc(OC)c3Br)C2)ccc2cc[nH]c2c1 C(C(=O)Nc1cccc(Cl)c1C)(C(C)C(C)(C)C)N1CCC(CC(C)O)CC1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CCCC1CF c1(NC(C)=O)ccc(CNC(C2(c3ccc(C)cc3Br)CC2)=O)cc1O C(=O)(C1=C(Cl)CCC1)N1C(C(N2CCCC(N3CCC3)C2)=O)(COC)C=CC1 C1(CNC(=O)C=Cc2nccs2)CN(C(c2ccn(CCF)n2)=O)CCCO1 c1(C(N2CCN(C(C(CC(C)C)F)=O)CC2)=O)ccc2c(c1)N(C)CCO2 CC(C)CC(C)CN1CCC(NC(=O)C(C(C)C)NC(=O)Cn2cccn2)CC1 N1(C(C(CCC)=CCC)=O)CCN(C(=O)CC(O)CC(C)C)CC(O)C1 c1(CC(=O)Nc2nc(C(=O)OCC)c(C(F)(F)F)s2)ccc2ccc(O)nc2c1 Cc1cccc(Cl)c1C(=O)NCCOCCN(C)C(c1nscc1N)=O Cc1[nH]nc(C(=O)NCc2csc(CNC(C3CCCC(=O)O3)=O)n2)c1C N1(C(C2(CC#C)CCCO2)=O)CCCC(N(C(=O)C=CC=C(Cl)Cl)CCO)C1 c1(C(N2CC3C(CNC(c4cccc(SC)c4)=O)(C3)C2)=O)cnn2c1N(C)CC2 C(CN=c1[nH]nc(-c2ccon2)s1)NC(C(N1CC(C)OC(C)C1)(C)C)=O C1(C(=O)OC)CN(C(=O)CNC(=O)CSCC#N)CC1C N1(C(c2n(CC=C)ccc2)=O)CCCN(C(c2cc(OC)nc(F)c2)=O)CC1C C1(CNC(C=C(C)C2CCC2)=O)CCN(C(=O)CC2CCOC2)CCC1(F)F C1(C(=O)NCCOCCN(C)C(c2nsnc2O)=O)CCC(C)(C)C1 CC1c2c[nH]nc2CCC1C(N1CC(CNC(c2ccc(C#N)nc2O)=O)C1)=O N1(C(CSC(C)C)=O)CC2(CC2)CC1CC(=O)NC1CCOC1C Cc1noc(C(=O)NCCCCCNC(=O)C(F)(F)c2csc(C)c2)n1 C(=O)(C#CC1(CC)COC1)NC(C1(C(=O)NC(CCC)C2CCC2)CC1)C C=CCC(CNC(C1CC(C)N(C)C1)=O)C(=O)N1CCC(O)(C(C)C#N)C1 C1(C(=O)NC2CC(O)(c3ccccc3)C2)CCCC2(CC2)C1 C1(C(N2ON=C(C(C)NC(CSCCCC)=O)C2)=O)CCC(N=[N+]=[N-])C1 C1(NC(c2ccn(COC)n2)=O)CN(C(c2ccc[nH]2)=O)CC1n1ccnn1 C(C(C)(O)CO)N(C(CC)CNC(C(=O)O)=O)C.C(C)(C)(C)O CC1CCN(C(=O)N(CCS(C)(=N)=O)C(C)C)C1c1cn(-c2ccc(C(=O)O)o2)nn1 c1(CC(=O)NCC(=O)NCC(COC)C)ccn(C)c1 C1(F)(CNC(C2CCCO2)=O)CCN(C(c2cccc(-c3ccoc3)c2)=O)C1 C1(CN(C(=O)CCS(C)=O)C)CCCCN1C(c1ccc(C(F)(F)F)cc1)=O C1(CO)CCN(C(C2(CNC(=O)CN3CCCC3C(F)(F)F)CCOC2)=O)CC1 CC1=NNC(=O)C1CN(C)C.N12CCOC(CO)(C1)Cc1cccc(c1)C2=O Cc1cc(Cl)c(C(N2CCS(=O)(=O)C(CCNC(=O)CC=CC(C)C)C2)=O)cc1C CN1CCOC(C(=O)NCCCOCCCNC(c2cnn(C)c(=O)c2)=O)C1=O C(C(=O)N1C(CO)CC1CO)(C(C)(C)C)NC(c1c(CC)noc1)=O c1(C(N2CC3(CN(C(CC(C)OC)=O)C3)C2)=O)cc(Br)cc2c1CCN2 CC(C)CCCCCC(=O)N1CC2CCC2(CNC(c2ncc(Cl)cc2F)=O)C1 N1(C(CC(C)SC)=O)CC(F)CC1CC(=O)NCC1CCCCCC1 c1(C(N2CCC(CNC(C3(C)CC(=C)C3)=O)C2)C)ccccc1Br C1(NC(c2ccc(C(C)C)nc2)=O)CCC2(C1)CN(C(C1(C)CC1C)=O)C2 c1(CN(CC)Cc2coc(COCC)n2)cccc(C(F)(F)F)c1F c1(C(N2CC=C(CN(C)C)CC2)C(=O)NC(C(=O)OCC)C)ccnc(F)c1F C=CCC(F)(F)C(=O)N1CC(C(C)(C)O)(COC)C1.C12(CCC1)C(=O)N2 C(=O)(C(C)(F)C(C)(C)F)N1CCN(CCCNC(C(C)c2cccs2)=O)CC1 N1(C(c2scc(C)c2)=O)CC2CCOC2(CNC(=O)C(C)(C)c2cscn2)C1 S(=O)(=O)(c1ccc(NC(CF)CF)c(Cl)c1)NCCc1cc(C)no1 CCC(CC(=O)NC1(C)CCN(C(=O)COc2cc(F)cc(F)c2)CC1)C(F)F CC1CN(C(C2(C)CC2(F)F)=O)CCCN1C(=O)Cc1csnn1 C(CCCOC(N(CCOCCOC(C)(C)C)C)=O)NC(=O)O.C=CC C1(N(C(c2c(C)cno2)=O)C)CC2CCC(C1)N2C(=O)CCS(C)=O Cc1[nH]c2ccc(C(N3CC(NC(=O)C4CC4)C4CC34)=O)cc2c1C C1(NC(COCC)=O)CCCC12CN(C(=O)CCn1ccnc1)C2 C1(NC(c2cn(C)nn2)=O)CC2CC(C1)N(C(c1ccccn1)=O)C2 C(=O)(C1=Cc2ccccc2C1)N1C(C(=O)Nc2cnn3c2CCC3)CC=CC1 c1(OC)ccc(OCCC(C)(C)CC(=O)N(CC(c2nn[nH]n2)C)C)cc1 C(=O)(CCCCC1CC1)N1CC(CC)(NC(C2(CCOC)CCCC2)=O)C1 N1(C(C2(NC(C3CC4CCC3O4)=O)CCCC2)=O)CC2CC(O)CC1C2 c1(C(N2CC3(C(NC(CC(C(C)C)O)=O)CCC3)C2)=O)c[nH]c(=O)c2ccnn12 c1(C(=O)NC2(C)CCCN(C(C(C(=O)OCC)CC)=O)C2)cn(C)c(=O)nc1O Nc1ccc(F)c(C(N2CCN(C(=O)CN3CCS(=O)(=O)CC3)C3CC23)=O)c1 C(=O)(CCCN(C(=O)C(n1ccnc1C)C)C)NCC(=CCCC)C C1(C)(CNC(CCCCC=C)=O)CN(C(C2CSCCS2)=O)C(C)(C)C1 c1(OCOC)cc(-c2cnn(C)c2C(F)F)cc(OC)c1OC Cc1cc(C(=O)NCCCN(C(=O)CCc2csc(Br)c2)C)nc(O)c1 c1(OC)cc(OC)nc(C(=O)NCC2(C)CCN(C(C3NC(=O)CC3C)=O)C2)n1 Cc1ccc(Cl)c(OC(C)C(N2CCC(CNC(c3cc(C#N)cs3)=O)C2)=O)c1 c1(C(=O)NCCC2(O)CCCN(C(=O)CC(F)(F)F)C2)cnnc2ccccc12 c1(C(=O)NCC2N(C(c3c(C)nc(Br)o3)=O)CC2)ccc2c(c1)C=CCC2 c1(C(=O)NCC2CCN(C(c3scnc3C3CC3)=O)C2)cc(Cl)cc(Cl)c1O c1(CC)ncc(Cl)c(C(=O)NCC2CCCN2C(=O)C2=CC(C)CC2)n1 N1(C(=O)C(F)F)CCOC2(CCCN(c3ncc4c(Br)cccc4n3)C2)C1 c1(C(=O)NC(C(=O)NC2CCC(=O)NC2=O)CO)ccn2ccnc2c1 C1(CNC(C=CCCC(C)C)=O)CN(C(C2(F)CCC2)=O)CCC1C(F)(F)F CC1(C)CC(Nc2cc(F)ncn2)CN(C(=O)CC2CC(=O)NC2=O)C1 C(=O)(C(CC)CCc1ccccc1)NCCC1(NC(CS(=O)(=O)NC)=O)CCC1 N1(C(c2c(CC)ccs2)=O)CC(C(=O)NOCc2ccc(F)cc2)C(C)C1 CC1(C)CC(C(N2CCC(C(=O)NCC3CCCC(=O)N3)CC2)=O)CCO1 N1(C(C(C)SCC)=O)CC(C(N2CCCC(F)(F)C2)=O)C2(CC2)C1 C(CC(=O)Nc1cncc(C)c1)(CC(C)C)NC(C12CCC(OC)C1C2)=O C(c1cccc2ccccc12)=CC(N1CCCCC(NC(=O)C=CC2CC2)C1)=O N1(CC(=O)N(C(c2cn(C3C(OC)CCC3)nn2)(C)C)C)CCNC(=O)C1 CC(C)C1=NOC(C)(C(N2CC3CCC2C3NC(c2cnn[nH]2)=O)=O)C1 O=C1CCC(C(=O)NCC(C(F)(F)F)N2CCN(C(=O)C#CC3CC3)CC2)CN1 N1(C(CCCC(=O)N(C)C)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 c1(CNC2CCCC(C(=O)NCc3cn[nH]c3)C2)cc(Cl)cnc1F O=C1NC2(C(=O)NC3CC(NC(C4(n5ccnn5)CC4)=O)C3)CC3CC1C2C3 C(=O)(C1(C)CCOc2ccccc21)N(C)CCNC(C1CC2C=CC1O2)=O c1(CC)nn(C)c(CC)c1C(=O)NCC(C)(O)CNC(=O)CC1=CCCC1 C(=O)(CCCCN1CCCC1)N(C1CCN(C(C2(F)CCCCC2)=O)C1)CC#C CCC(CC(=O)N1CCC(C(=O)NCC(C)(C)CSC)C(C)(C)C1)C(F)F C123CC(C)(CN1C(=O)N2)C3.CC(C)(C)CN.CNC c1(C2C(=O)N2)ccnc(Cl)c1Cl.C1(C(C#N)N(CCCSC)C)CCC(C)CC1 Cc1ccc2c(CN3CCCC3CCC(=O)Nc3ccc(I)nc3)c[nH]c2c1 C(=O)(C(COC)CC(C)C)NCCCC(=O)N(C(=O)CC(C)O)C.CN N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(c2ccsc2Cl)=O)C(C)(C)C1 C1(OC)CCn2cc(C(=O)NCC3C(C)CCN3C(=O)CN3CC=CC3)nc2C1 C(CC(C(=O)NCC1CCN(C(=O)C(C)N(C)C)C1)NC(C)=O)SC N1(C(C(CSC)C)=O)CC(N(C)C(c2cncc(C#N)c2)=O)C2(CC2)C1 c1(C(N(C(CN(C(C(CC(C)C)O)=O)C)C)C)=O)cc2ccsc2n1C Cc1cc(C(N2CCC(CNC(c3csc(Br)c3Cl)=O)C2)=O)nn1C N1(C(c2c(COC)cccc2)=O)CC2(C1)CN(C(C1CC(C(C)=O)C1(C)C)=O)C2 CC(CCO)CCN=c1nc(N(C)Cc2ccno2)c2cc(Cl)ccc2[nH]1 C(=O)(C(O)C(C)(C)SCC)NCCN(C(C(C)(C)NC(=O)NCCC)=O)CC CC1CCCN(C(N2CCCC(Cc3csc(Nc4ccnnc4O)n3)C2)=O)C1 Cc1cc(F)c(C(=O)NC2CCN(C(c3cccc(F)c3Br)=O)CC2O)cc1F c1(NC(=O)OCC)cc(-c2cccc(NC(=O)CCc3cnn[nH]3)c2)ccc1Cl C1(C(C)C)CCC(C(=O)NC2CCCC2NC(C2(c3ccno3)CCC2)=O)CC1 N1(C(CCCC(=C)C)=O)CCC2(C1)CN(C(c1cnsc1C)=O)CC(C)O2 C(=O)(C(CCCCO)NC(=O)CC1CC=CCN1C)NCC1CC(COC)C1 c1(CC)ccc(C(N2CCC(CCNC(c3cc(CO)[nH]n3)=O)C2)=O)c(OC)c1 c1(C(=O)NC2CN(Cc3c(O)cccc3Br)CC2O)c(F)ccc(O)c1F c1(CC(=O)NCC(CC)NC(=O)Cc2cc(C3(C)CC3)on2)cnn(C(C)C)c1 C(CC(=O)N1CCN(C)C2(CC2)C1)(C(C)(C)C)NC(C(C)=C1CC1)=O N1(C(c2nc(C)c(Br)cc2)=O)C2CCCC1CC(n1ccnn1)C2 c1(NC)ccccc1C(=O)NCCC(O)CNC(=O)C=CC1CC1 N1(C(CC2ON=C(C)C2)=O)C(C(=O)NC2(CO)CC(O)C2)CCC1C1CC1 C#CCCCCCC(=O)NCC1C(OC)C(OC)CN1C(c1nncs1)=O c1(CC(=O)NCCCn2cc(-c3c(OC)nccc3)nn2)cnc(O)nc1O C1(NC(c2scc(C)c2)=O)C2CCN(C(=O)CCn3cnnn3)CCC12 c1(C(=O)NC(CC)(CC)CCNC(C2CC2Cl)=O)ccc2ccccc2c1 C1(NCc2c(OCCOC)ccc(Cl)c2)CCC12CCCCC2 c1(C(=O)NCCNC(C23CCCCC2C3Br)=O)sc([N+](=O)[O-])cc1Cl C(N=c1[nH]c2cc(Cl)ccc2s1)CC1(CCNC(C2CC(C)(C)OC2)=O)CC1 c1(C(N2CC(NC(c3cc(C)sc3C)=O)C2)=O)ccnc2ccc(F)nc12 C12(C(=O)OC)C3C4C1C1C2C3C41NC(=O)N(C)CC1CCCCN1 C(=O)(C(Cc1cn(-c2ccncc2)nn1)NC(C1CCN1S(C)(=O)=O)=O)OC C1(C(N2CCCC(CCC)(NC(c3csnn3)=O)C2)=O)Cc2cc(F)ccc2O1 c1(C(N(CC(CC)NC(=O)CC2CCC(=O)O2)C)=O)cc([N+](=O)[O-])ccc1C NS(=O)(=O)c1ccc(S(=O)(=O)NC2CCc3ccccc32)cc1 N#Cc1ccc(Br)c(F)c1NC(C1CC2CC2N1C(C1CCN(CCO)CC1)=O)=O C1(CC)(NC(=O)CCn2c(C)csc2=O)CCCN(C(C2(C#N)CC=CC2)=O)C1 CCCCC(C)C(C(=O)NCCO)N1CCc2cc(C(C)(C)C)ccc21 CCC(c1ccc(C)cc1)=CC(=O)NCCCN(C)C(C1CCC12CCCO2)=O C1(CCNC(CN(CC)CC)=O)CCCN(C(c2c(C)oc(C)c2C)=O)CC1 c1(OCC)ccc(CN2CCC(CC(=O)NCc3c(F)cccc3Br)C2)cc1Br N1(c2c(C#N)cnc(N3C(C)(C(N4CCCC4)=O)CC3)n2)CCc2sc(Br)cc2C1 Cc1ccc(C(=O)NCC(=O)NCCC(C)NC(=O)CC(C)N2CCCC2=O)s1 C12(NC(CONC(=O)C(CO)OC(F)(F)F)=O)CCC(C1)N(C(=O)C(F)(F)F)C2 N1(C(C2(OCC)CCC2)=O)CCC2(CC1)CCN(C(=O)C(C#N)CC)C2 C1(NC(c2cccs2)=O)CC2CC1N(C(c1cc(Br)c[nH]1)=O)C2 N1(C(CC=CCC)=O)CCC(OCC(=O)OCC)C1 Cc1cc(C)c(C(N2CCC(N(C)C(C3CC(C(F)F)C3)=O)C2)=O)cc1C CCC(CC)C(F)C(=O)N1CC(C)CCC1CNC(c1cc2n(n1)CCCN2)=O N1(CC(=O)NC(Cn2cc(-c3cnc(C(C)C)o3)nn2)C)CCOCC1=O C1(C(=O)NC(C(C)C)(C)CO)CN(C(C2CCC(C(N)=O)C2)=O)CC1(F)F C1(C(=O)Nc2nc(C)c(C)s2)C2CCC(C2)C1NC(c1cnnc(Cl)c1)=O CCCC(C(=O)N(CC(C)CNC(=O)CCc1cc(Cl)no1)C)C1CCC1 c1(SCC(=O)NCCC(C)(C)NC(CCC=C=C)=O)cc(=O)n2ccsc2n1 C1(CC(=O)N(C)CCC2CCCC2)CC(F)CN1C(c1ccc[nH]1)=O C(C)(C(=O)NCCC1(O)CN(C(=O)CCCSC)C1)(C1(C)CC1)OC C(=O)(C(O)CC(F)(F)F)N(CC(C)(C)NC(c1ccc(N2CCOCC2)nc1)=O)C N1(C(=O)Nc2cc(C(F)(F)F)cc(Cl)c2)CCN(C)CC1Cc1ccc(C)cc1 c1(C(C(=O)NC(CNC(C2CC(OCC)C2)=O)C)(F)F)ccc(Cl)cc1 Cc1cccc(O)c1C(N1CC2CN(C(c3ccc(I)c(F)c3)=O)C2C1)=O CCCC(C)(C)C(=O)NCC(O)CCNC(C1CC(C(F)(F)F)(OC)C1)=O c1(C(=O)NC(C)(C)CCNC(C2CC23CC3(F)F)=O)nccc2cccnc12 C(=O)(CC(C)C(=O)NC(C)(C(=O)NC1CC(C)OC1=O)C1CCC1)OC(C)=O N1(C(C(C)(C)NC(=O)OC)=O)C2CCC1C(F)C(NC(=O)CC(F)(F)C(F)F)C2 c1(CN(C(c2cc(C(C)C)on2)C(=O)NC2COC2)CC)ccccc1F N1(C(C(n2ncc(C)c2)C)=O)CCC(O)C(NC(c2ccon2)=O)C1 CS(=O)(=O)c1ccnc(NC2CN(C(=O)Cc3ccc(Br)cc3Cl)CC2C#N)n1 Cn1cc(C(=O)C(N2CCC(NC(=O)CC(O)c3ccccc3)C2)=O)cn1 c1(NCC2(C)CCCN(C(C(C=C)(C)CC)=O)C2)cc(C#N)nc(C)n1 C1(CC(=O)NC(CC)CN(C(=O)CCc2nc(C)cs2)CCOC)OCCC1(C)C C1(C)(C(=O)Nc2cc(OCC)ncn2)CCCN(C(=O)C(O)C(C)C)C1 CC(C)CCCC(=O)N1CCCCC1C1(NC(=O)COCCF)CC1 C12CCC(CC1)N2.N1(CC)CCC(CCC2CCCNC2)C1 C1(C(=O)NC(C23CCC(CC2)C3)CNC(C(=O)NCCOC)=O)OCCC1(C)C c1(C(N2CC(C)(C(=O)NC(CCC)c3ccco3)C2)=O)[nH]cc(C)c1C Cc1cc(C=CC(=O)NCC2CCN2C(=O)C(c2cnn(C)c2)C)ccc1F c1(C(N2CC(NC(Cc3n(C)ncc3Br)=O)C2)=O)cc2ccccc2cn1 NS(=O)(=O)CCCC(=O)N1CC(O)C(O)C1CNC(C1CC2CC2C1)=O c1(CN(C)C(C2CC2c2cc(Br)cc(Br)c2)=O)noc2c1CCCCC2 C1(NCCNC(C2C(CC)C2)=O)(C)CCOCC1.c1(N)nc(C)cs1.C1(=O)C(C)N1 c1(C(=O)NC2CC(CNC(C3(CC=C)CCCC3)=O)C2)ccc(S(N)(=O)=O)nc1 N1(C(CNC(=O)NC)=O)CCC2(CC1)CC2(CO)CNC(c1ncccc1C)=O C1(C(=O)NCCC(C)NC(c2ccc(C(C)C)o2)=O)COC(C)(C)O1 C#CCCCCCCCNC(c1ccc(C)nc1O)=O.C1=CC(=O)N2CC1C2 c1(C(=O)NC2(C(=O)NC3CCN(C(=O)NC)C3)CCSC2)cnc(N)cn1 C1(c2n(CCCSCC)nnn2)(NC(C2CCC2)C)CCCC(OC)C1.OC C1(C(=O)NCC2(C#N)CCC2)(COC)CN(C(c2ccc(C)o2)=O)C1 CCC(C)(C)CCCC(=O)NC(C)(C)CNC(c1cc([N+](=O)[O-])ccc1OC)=O N1(C(C2(OCC)CC2)=O)CCC2(COCC(C(=O)NC3(NC(N)=O)CCC3)O2)C1 c1(OCC)nc(C)ccc1C(=O)NC1CCC1NC(=O)C=Cc1cscn1 Cc1ccc2scc(C(N3CCOCC3CNC(C3CC(F)C3)=O)=O)c2c1 c1(C2(CN(C(C(N3CCC(CC)C3)=O)=O)CCCO)CC2)ccc(Cl)c(Cl)c1 Cc1cc(F)cc(C)c1C(=O)NCC#CCNC(C1(C(C)C)CCC1)=O C1(NC(C2C(c3cc(C)sc3)C2)=O)CC2CCC(C1)N2C(=O)C(N1CCSCC1)C C#CC1CN(C(=O)CC2C(=O)N(C)N=C2C)CCN1C(=O)COc1cc(C)on1 CC1CCCC=C1C(=O)NCCCCCNC(=O)Cn1ccc([N+](=O)[O-])n1 Cc1ccc(C#N)cc1S(=O)(=O)N1CCC2C(CCN2Cc2cc(C)nn2C)C1 C12(C(N3CC4C(NC(C(C(CC)CC)C)=O)C4C3)=O)CC3CC(C1)CC(F)(C3)C2 c1(COC)nnc2ccc(=NCC3CCC(C(F)(F)F)O3)[nH]n12 C1(CNC(C2OCCN(C(C(C#C)(C)C)=O)C2)=O)CCC2(CCC2)O1 C#CC1(F)CCN(C(=O)C(c2ccoc2)NC(=O)C(C)=C(C)CC)CC1 CCCCC(C)(F)C(=O)NC(CC(=O)N(C)CCc1ccccc1)C(F)(F)F C1(C(N2C(C3(NC(C(C4CCC(=O)N4)C)=O)CC3)CCCC2)=O)CN2CCN1CC2 S(=O)(=O)(c1ccc2[nH]c(=NCC(CO)OC)sc2c1)N(CCCC(=O)NC)C N1(C(c2ccc(CC)nc2)=O)CCOC(C(=O)NCC(c2ccccn2)O)CC1 C1(C(N2C(C(C)C)CN(C(=O)CCSC(F)(F)F)CC2)=O)CCc2ccnn2C1 c1(C(=O)NC2C(NC(CC3(OC)CCC3)=O)COC2)ccc(C2CC2)c(F)c1 CCC(CCC(=O)N1CCC(NC(=O)CSc2ccc(Cl)cc2O)C1(C)C)OC CCC(C)C(C(=O)NC(c1ncc(C)cn1)C)N(C(=O)C=C(C)C(C)C)C C#CC1(NC(C2CN(C(c3c[nH]nc3OC)=O)C(C)(C)C2)=O)CCC(C)(C)C1 c1(COC)ccc(O)cn1.C12C=CCN1C(=O)CONC2=O C1(NC(Cc2ncc(C)s2)=O)CC2CC1N(C(c1cc(Cl)cnn1)=O)C2 c1(CC)noc(CN(C(C2CCN(C3CNC3)C2)=O)C(C)C)n1 C1(C(N2CC(SC)C2)=O)COCCN(C(=O)CC(N)CO)C1 n1(C(C(=O)NCC2(F)CC(NC(C3(C#C)CC3)=O)C2)C)nc(C)c([N+](=O)[O-])c1C N1(CCC(N2CCN(c3ccc(Cl)cc3)CC2)=O)CCC(F)C(O)C1 C1(NC(c2ccc(CN=[N+]=[N-])s2)=O)C2CN(C(c3cccs3)=O)CC12 Cc1ncc(C(=O)N(CCCNC(=O)Cc2ccc(C(F)(F)F)nc2)CCO)n1C c1(NC(c2c(Cl)n[nH]c2C)c2n(CC)nnn2)ccc2c(c1)CN(C)C2 CC(C)CC(C)(C)C(=O)N1CC(O)CC1Cn1cc(C2(C(=O)OC)CCC2)nn1.N(C)C c1(NC2C(CC)CN(C(C3CCCCS3(=O)=O)=O)CC2)ncccc1[N+](=O)[O-] c1(C(=O)NCC2(CCNC(C34CCC(C3)C4)=O)CC2)coc2c1COC2 c1(C(=O)NCC(C)NC(C(c2cccc(C)c2F)O)=O)cc2n(c1)CCOC2 c1(SC)cc(C(=O)N(C(C)CNC(=O)C=Cc2ccc(C)s2)C)cc(Cl)c1 n1(CCC(=O)NCC2(OC)CN(C(c3cc(C)c(C)o3)=O)C2)cc[nH]c(=O)c1=O c1(OC)cc(CO)ccc1C(=O)NC1CCN(C(=O)Cc2cccnc2)C(C)C1 N1(Cc2ccc(C)cc2)C2CCCC1CC(NC(c1cc(O)ccc1Br)=O)C2 C(=O)(CCCCCC(C)O)NCCCN(C(C(CC)c1cccnc1)=O)CC c1(NC(C(=O)NCc2n(CCC)ccn2)=O)ncc(C)cc1F C(=O)(CC(C)C(C)(C)C)NC1C(CC(=O)N(CC(C)OC)C)C(O)C1 N1(C(c2c(C)c[nH]n2)=O)CCC2(CC1)CN(C(C1C3CCC(=O)C13)=O)C2 c1(CSC)cc(C(N2CC3(CCC3NC(=O)C(F)C(C)(C)O)C2)=O)ccc1F N1(C(c2c(C)nn3c2NCCC3)=O)CCc2cc(Br)cc(F)c21 c1(NC(C2CN(c3ncnc4cc[nH]c34)CCS2)=O)cc2[nH]ccc2cc1Cl CCCC(C(=O)N1CCCC1C1(O)CN(C(c2ncn(C)c2C)=O)C1)OCC N1(C(CC(=O)NC)=O)C(CNC(c2c(F)cc(C)cc2F)=O)CC2COCC12 Cc1cnc(C(N2CC(CNC(=O)CCn3cc(C)cn3)C2)=O)c(F)c1 N1(CC(N2CCN(C(C3CCN(C)CC3)=O)CC2)=O)CC(=O)Nc2ccccc21 N1(C(C=COCC)=O)Cc2occ(C(N3CCC(O)C(C)(CO)C3)=O)c2C1 C(=O)(C(C)(C)C(C)NC(C1CC1(F)Cl)=O)NCCC(C)F C=CCC(CNC(=O)C1CC1c1ccccc1)NC(=O)C(C)=C(C)CC O=C(CS(=O)(=O)CCO)NCC1CCCCN1C(C1CC(OC(F)(F)F)C1)=O N1(C(C(N2CCCCC2)C)=O)CC(C2CC2C(N2CC(S(C)(=N)=O)C2)=O)C1 c1(C(N)=O)ccccc1C(=O)NCC1CC1CC(N1CC(F)CC1CO)=O N1(C(c2c(C)snn2)=O)CCCC(CCNC(=O)C(N2CCN(C)CC2)C)C1 c1(C(=O)NC2(C)CCN(C(c3c(C)cnn3C)=O)CC2)cnc2c(c1)NCC2 C1(c2n(C(C)(C)N(C(=O)CC(C)C)C(C)(C)C)nnn2)(OC)CN(CCCl)CC1C C(C(=O)NCC12CCCC1OCC2)(C(C)(C)C)NC(c1n(CCC)ccc1)=O C1(O)(N(C(C(F)OC)=O)C)CCN(C(C2(c3cccs3)CCCC2)=O)CC1 C1(C(=O)NC2CN(C(CNc3nccc(OC)n3)=O)C(CO)C2)CC2C(C1)C2(F)F CC(C)CCCC(C)C(=O)NC(C1(O)CCN(C(C2CCCC2(C)C)=O)CC1)C Cc1nc2ccc(NC(=O)NCc3cncc(Cl)c3Cl)cc2nc1C N1(C(CSCC)=O)CCOCC1C(=O)NC(Cc1cccc(Br)c1)CC(=O)NC c1(C(=O)NC2C(CNC(CCC=C)=O)C2)ccc2nccc(Br)c2c1 S(=O)(=O)(c1cccc(=NC(C)CCO)[nH]1)NCC(N1CCC(C)CC1)C C1(C(=O)NCC(C)(C)NC(=O)CSc2nc[nH]n2)CCCCC1C1CC1 C(=O)(CCCS(N)(=O)=O)N1CCC(N(CCC)C(c2cc(F)cc(F)c2)=O)CC1 C12(C(=O)NC(C)CS(C)=O)CC(c3ccccc3F)(C1)C2(F)F N1(c2nccc(OC)n2)CC2C3CCC(C2C1)N(C(=O)CCN1CCOC1=O)C3 N1(C(C(c2ccc(C)s2)C)=O)CCOC(CCCNC(=O)Cc2cncn2C)C1 N1(C(c2n(C)ncc2)=O)CC2CC1CN(C(=O)Cc1cc(O)cc(Br)c1)C2 C12(NC(C(C)C3CCC3)=O)CC(C1)N(C(=O)COCc1cccnc1)C2 Cc1cc(F)cc(C)c1C(N1CC(CC(C)NC(c2nnn3c2CCC3)=O)C1)=O C(CC1=CCN(C(=O)CC2CCC2OC)CC1)NC(CC1(OC)CCOCC1)=O N1(C(C(C(C)O)(F)F)=O)CC(C2CN(C(c3ccc(C4CC4)cc3Cl)=O)C2)C1 C1(F)(C(=O)NCC(C)N(C)C)CCN(C(C2CCC(C)(C)C2)=O)CC1 C(=O)(C(C)CCOC)NCC(=O)NCC(=O)N(C(CC)C1CC1)C C1(C(N2CC(NC(=O)Cc3cncn3C3CC3)(CO)C2)=O)OCC2CCCC12 C(=O)(C(=O)CC(C)C)NCC(C1CCCC1)NC(c1cc(C)no1)=O N1(C(c2cc(CC)nn2C)=O)C(CNC(c2sc(C)nc2C)=O)CC2CCCC12 C(c1ccc(C(N)=O)cc1)=CC(=O)NC1CC(NC(c2nc(C)sc2)=O)C1 N1(C(C(CCC)F)=O)CCC(C)C(CC(=O)Nc2cn(C)nc2C2CC2)C1 N1(C(C2CN(C)C(=O)CC2)=O)CC2CCC1C(NC(C1CN(C)C1)=O)C2 c1(OC)cc(CCC(C)NC2CCCC(n3cccn3)C2)cc(F)c1 n1(CN2C(c3ccccc3)C3CC3C2)nc(C)c(N2CCN(c3ccc(F)cc3F)CC2)c1C C#CCC(C)(C(=O)NCc1nc(C)sc1C)NC(=O)C(O)C(F)(F)F C(C(CC(C)C)C(=O)N1CC(C)C(C)(CNC(=O)C(C)(CO)OC)C1)OC Cc1cc(C(=O)NC2CC(CNC(=O)C(C)C3CC3)C2)c(Br)cc1F C1(NC(C2(CC=C)CCC2)=O)CS(=O)(=O)CC1NC(=O)CN1C(=O)CNC1=O Cc1cccc2[nH]c(C(N3CCN(C(c4ccc(F)cc4N)=O)C4CC34)=O)cc12 CC(O)CCCNC(c1coc(C(C)NC(=O)CCC2CC2(F)F)n1)=O C1(NC(CC(C)SC)=O)CCC2CN(C(=O)C=Cc3ncc[nH]3)CC2C1 c1(SCCNC(N2CC(=O)NC(C(F)(F)F)C2)=O)cnc2n1CCOC2 C1(C(=O)NC(C(C)C)CNC(=O)C(C)CC2CCCC2)CCc2cnnn2C1 c1(C(N(CC(C)CNC(c2coc(C(N)=O)c2)=O)C)=O)ccc(F)c2occc12 c1(CCN(C(CSC(C)(C)C)=O)C(c2sc(Br)cc2F)=O)nc2ccccc2s1 c1(C(CCC(=O)N(C(CCNC(C(C(C)C)O)=O)C)C)=O)ccc2c(c1)CCC2 C1(COC)CN(Cc2csc(C3CC3)n2)CC(C)(C)O1 N1(C(=O)Cc2cccs2)CC2CN(C(c3cc4scnc4[nH]3)=O)CCC2(CO)C1 CC1(C)CCCN(c2nnc(C(F)F)o2)C1CNC(=O)CCc1nc[nH]n1 Cc1[nH]c(=NC2CCN(C(c3ncc(Cl)nc3Cl)=O)C2)ccc1C#N C1(C(=O)NC2C(NC(c3cc(OC)ncn3)=O)C2)CCN(C)C(=O)C1 Cc1ccc(COCCNC(=O)CSCCC)cc1F.C1C(=O)CO1.C1(N)CC1 c1(OCC)nc(NC(c2ccccc2)CC2CCCCN2)ncc1C c1(C(=O)Nc2ncc(OCC)nc2)ccc2ncc(-c3cc(O)ccc3F)n2c1 C1(C(=O)NC2(C)CCN(C(c3cc(OC)n(C)n3)=O)C2)CCC2(CC1)CC(O)C2 c1(C(C(=O)NC(C(=O)OC)(C)C2CCC2)=O)cc(O)cc(F)c1 N1(C(Cn2c(C)cc(C)n2)=O)CC(C)CCC1CNC(C1(CO)CCOCC1)=O c1(C(N2CCC(C(C)NC(C3CC(O)C3)=O)C2)=O)cc(N)cc([N+](=O)[O-])c1 N1(C(CCC=CC)=O)CC(C)(C)OCC1CNC(C1CCC(=O)N(C(C)C)C1)=O N1(C(C=CC(CC)C)=O)CCOC2(C1)CN(C(c1cc3ncccc3s1)=O)C2 c1(C(C)=O)cc(C(=O)NC2(CCNC(=O)C(F)C3CCCC3)CCCC2)oc1C c1(C)nc2ccccc2o1.c1(C(=O)OO)c(F)cc(F)cc1Br CN=c1[nH]c(C(=O)NC2CCCN(C(c3cccc(Cl)c3)=O)C2)cs1 N1(C(CS(CCOC)(=O)=O)=O)CCC(C2(NC(=O)CN(C)C(=O)C3CC3)CC2)C1 C(CCN=c1nc(N2CCC(CC3CC3)CC2)c2sccc2[nH]1)c1nnc(C)s1 CC1OC(C)CC1CC(=O)NCCOCCN(C)C(C1(CO)CC(F)(F)C1)=O N(C1CCCn2nccc21)C(CCN(C(c1c(NC)cnnc1)=O)C)=O CCC(CCCC(=O)NC1CCN(C)CC1C)NC(C1(n2cccn2)CC1)=O C(CNC(c1c(C)nsc1NC)=O)(C(C)(C)C)NC(COCCOC)=O c1(C(=O)NC2(CF)CCN(C(CC(C=C)C)=O)C2)cc(OC)cc(Br)c1 c1(OC)cccc(C(CF)NC(=O)C(C2CCCCO2)OC)c1 C(=O)(C1=CS(=O)CCC1)N1CCC(=CCNC(C2ON=C(C)C2)=O)CC1 N1(C(CNC(=N)N)=O)CCOC2(C1)CN(C(c1ccc(SC3CC3)cc1)=O)C2 c1(C(N2CC(N(C(C(CCC)c3ccccc3)=O)C)C2)=O)cc(C)c(F)cc1N C(CC(=O)NC1(c2nc[nH]n2)CC1)(C(F)(F)F)NC(C(CC)(C)NC(C)=O)=O C12CCN(CC1O)C2=O.c1(C(=O)NC)cccc(NC(C2(O)CCCOC2)=O)c1 C(=O)(CC(C)(C)C(=O)N1CC(CCCCNC(=O)C(C)CSC)C1)OCC CCCCC(C(=O)N1CC(S(C)(=N)=O)C1)NC(=O)CN1C(=O)CCCC1=O c1(CCn2c(N3CCC(c4cncc(C)c4)CC3)nnn2)ccc(Cl)cc1F N1(C(CC2CCCN(C(CC(C)O)=O)CC2)=O)CC2CCCN2CC1C c1(CNC(C2(C)CC(C)OCC2)=O)nc2c(s1)CN(C(=O)C(C)(F)F)CC2 n1(C(CC)C)cc(Cn2nccc2C(N2CC(COC(C)=O)C2)=O)nn1 CC(C)(F)CCC(=O)NC12CCOC(CNC(C3CS(=O)(=O)CCO3)=O)(C1)C2 CC(CC(=O)NCCNC(=O)CN(C)C(=O)C1CC1)n1ccnc1 CC1=C(C(=O)Nc2nccc3c(Br)nccc23)C(C)(C)CCC1 Cc1nn(C)c2ccc(C(=O)NC3CC(NC(C4CCC(F)(F)C4)=O)C3)cc12 C1(C(N(C(CC)C)CCOC)=O)C(C)OCCN1C(=O)CN(C1CCC1)C N1(C(c2ccc(SC(C)C)cc2)=O)CC(NC(C2CCC(=O)C2)=O)CC12CCC2 C1(CNC(C(C(C)OC)N(C)C)=O)(NC(=O)C(O)CCN(C)C)CCCCC1 C1(CNC(C(c2ccnn2C)C)=O)CCC(NC(C2(F)CC2)=O)CC1 C1(C2CCCO2)(C(=O)NC(c2nc(C)c(Br)s2)CC)CCN(C)C1 c1(NC(=O)NC2CC(C)CN(CC3CC3)C2)c2c(nn1-c1ccccc1)CCCC2 n1(CC(=O)NC(CC)(C)CNC(=O)C2=C(Cl)CC2)cc([N+](=O)[O-])cn1 C1(C(N2CCC(O)(Cc3cn(CCC=C)nn3)C2)=O)CC12CCOC(C)C2 N1(C(C(CC)C(C)C)=O)CCCC2(C1)CN(C(c1ccc(C)c(F)c1F)=O)C2 C(=O)(CCCCC(C)=O)N(CCn1cc(Cc2c(CC)cncc2)nn1)C C1(NC(CCSCCCC)=O)CCCC12CN(C(c1cc[nH]c3nccc1-3)=O)C2 C1CN=C2N=c3ncn(C)c3=C(N2)N1.N1(C(COCCOC)(C)C)CCCC1=O Cc1ccc(C(=O)NCC2CC(NC(C3(C)C=CCC3)=O)C2)cc1F N1(C(CN(C)CC)=O)CCC(C(N2CCCC(Nc3nccnc3C)C2)=O)CC1 c1(CC)cc(C(=O)NC2CC(NC(C3CC34CCCC4)=O)C2)nn1C c1(C(=O)NC(CN(C(CCC)=O)CC)C)ccc(Oc2ccccc2)cn1 C(=O)(CC(CC1CC1)NC(=O)COCCCN=[N+]=[N-])N(C(CO)CO)C C12(C(=O)NCCN(C(c3cn(C)[nH]c3=N)=O)C3CC3)CCN(CC1)CC2 C(C)(CCC(=O)N1CC(C)CC1C(N1CCC(C)(C(N)=O)C1)=O)OCC c1(NC(=O)CCC2CCOC2)cc(CC(=O)NCc2cnsc2)no1 N1(C(c2c(C)cccc2)=O)CCCN(C(c2coc(Br)c2)=O)C(CO)C1 CCCC(C(=O)OC)C(=O)NC(c1ccccc1)C(N1CCC(C(=O)OC)C1)=O C12(CNC(C(C)(N(C(C3C(C)CCO3)=O)C)C3CC3)=O)CCC(CO1)C2 C1(CNC(CSC(C)C2CC2)=O)CN(C(c2cc(CC3CCC3)c[nH]2)=O)CCO1 C1(CC(C)C)CCN(C(=O)CSCCNC(=O)Cc2ccc[nH]2)C1 Cc1c(C(=O)NC(C)(CNC(c2sc(F)cc2Cl)=O)CO)ccn1CC1CC1 CC(C)C(CCNC(C1CC1Cl)=O)NC(C12CC3CC1C2C3)=O C1(NC(C(C=CC)O)=O)CCC2CN(C(=O)Cn3cnnn3)CC2C1 C1(COC)(SC2COC(C)(C)C2)CCS(=O)(=O)CC1 C1(C(=O)NC(C(C)C)C(C)(C)O)CN(C(c2ccccn2)=O)CCN1C Cn1cc(C(N2C3CCC2C(C(=O)NC2CCN(CCF)C2)C3)=O)ncc1=O CC(C)C(C)C(C)CC(=O)NCCCCN(C(=O)C(C)(C)c1ccnn1C)C c1(C(=O)NCC2(CNC(C(C)(C)N(C)C)=O)CCOCC2)cc2n(n1)CCCC2=O c1(C(C(=O)NC2(CNC(=O)OC(C)(C)C)CC(COC)C2)=O)cc(F)cc(Br)c1 C1(C)(C(=O)NCc2c(C(N(C(CCSC)C)C)=O)c[nH]n2)COC(=O)N1 N1(C(C2(O)CCC2)=O)CCCC(F)(C(N2C3CSCC2C3)=O)C1 C(=O)(CCCc1nc(C2CC2)no1)N(C(C)CNC(C1CC1C(C)C)=O)CC CN1CC(C)(C)CC1C(N1CCC(F)CC1C(N1C2CCC(C2)C1COC)=O)=O Cc1nc(=NC(=O)c2ccc(-c3cn(Cc4ccccc4)nn3)s2)o[nH]1 CC1=C(C(=O)N2CC(C)N(C(=O)CCCc3cnn[nH]3)CC2C)CCCC1 c1(C(=O)NC(CC(C)Nc2cc(CC)nc(CC)n2)C)nccc2ccccc12 C12(NC(c3ncc(OC)cn3)=O)CCC(C1)N(C(C1(n3cccn3)CC1)=O)C2 c1(-c2ccc(C3C(C(=O)OC)=C(CC)NC(=S)N3)cc2)ccc2oc(O)nc2c1 N1(CC2CCC(c3ccccc3)CC2)CC(c2c(C(=O)OC)cc[nH]2)C(C)(C)C1 c1(C(=O)NC2(CC=C)CN(C(c3snc(C)c3N)=O)C2)cc(F)c(F)c(Cl)c1F N1(C(c2c(CCC)nns2)=O)CCCN(C(=O)CNS(N)(=O)=O)C(CO)C1 N1(C(c2cn(CCC)nn2)=O)C(C(N2CCNC(=O)C2C)=O)CCC12CC2 C12(CNC(CCOCCC)=O)CN(C(=O)C(O)C3CC3)CC1(C(F)(F)F)C2 N1(CC(=O)NCC2N(C(C(CCC#C)O)=O)CCC2)C(=O)c2cccnc2C1=O C1(NC(C2C(CCC)C2)=O)COC2(CCN(C(c3cccs3)=O)CC2)C1 c1(CC)ocnc1C(=O)NCC1(F)CC(NC(=O)C(C)OCCC(C)C)C1 c1(OC)ncc(-c2cn(CC(=O)NCC3CCCCC3(F)F)nn2)cc1C N1(C(c2cn(C)nc2)=O)CCC=C(C(=O)Nc2cc(F)c(F)c(F)c2)C1 N1(C(C23C(CN(C(C(C)N(C)C)=O)C2)COC3)=O)CCC2(CCCOC2)C1 CCC(CCCC(=O)NC1CCC(C)(C)CC1)NC(=O)C(CC)CC C(=O)(C(C#N)(CC)CC)N1CC2(CN(C(c3c(CCCCC)cc(Cl)s3)=O)C2)C1 C1(NC(=O)CCc2ncc[nH]2)CN(C(c2ccon2)=O)CCC1C(F)(F)F C1(C(=O)NC(C=C)CO)(CC=C)CN(C(C2CCCO2)=O)C1 N1(C(C(COC)C)=O)CC(C)(C)CC1CC(=O)NCC(F)Cl C1(CC(=O)OCC)CN(c2ncccc2C(F)(F)F)CC(C)O1 c1(C(=O)NCCC(C)NC(c2nnc(O)nc2O)=O)ccc(CO)c(F)c1 C1(CNC(CC=CC=C)=O)CCCC(NC(c2nncn2C(C)C)=O)C1 CCC(CC)C(C)C(=O)NCCOCCCNC(=O)CCc1nc(C)cs1 C12(COC)CN(C(c3cnc(C(C)C)nc3)=O)C(CNC(=O)CC(C)SC)(C1)C2 CC(C)C(CO)C(=O)NC(C1CCCCC1)CNC(c1cnc(F)c(Cl)c1)=O CCCC(O)CC(=O)NC(CO)C(C)NC(=O)CCCc1cncs1 C1(CC(=O)NCCC2(NC(C3CC(=O)NC3=O)=O)CC2)C2CC3CC(C2)CC1C3 C(=O)(C1CCCc2n[nH]cc21)NC(CNC(c1cc(C)nc(C)c1O)=O)(C)C c1(CC(C(=O)OC)NCc2cn(CC(CC)C)nn2)cccc(F)c1 C=C1CCC(C(N2CC(OC)CC2CNC(=O)CNC(=O)CC)=O)CC1 c1(-c2n(CC=C)nc(C3CC3C)n2)ccc2nc(O)n(C3CCCC3)c2c1 c1(CC)ccc(NC(=O)CCC(C)NC(C2CCN(OC)CC2)=O)cc1C c1(C(=O)NC(C)CN(C(=O)C=CCN(C)C)C)cn(CCO)nn1 C=CC1CCN1C(=O)CCNC(c1cc(C2CC2)[nH]n1)=O C1(C(N2CCCC(NC(CCCC#CC)=O)(CO)C2)=O)CCC2(CC1)CC2(F)F C1(CC(N2CC(CN(C(=O)CCC(F)F)C)OCC2)=O)CCCCC1(C)C C1(C2CCN(C(=O)CC(c3cccs3)N(C)C)C2)(NC(CCC(=C)C)=O)CC1 C=CC(C)(C)CC(=O)N1CCC(=C)CC1C(=O)NC(C(C)(C)O)C1CC1 N1(C(CCOC)=O)CCC2CCC(C1)N2C(C1CCCCCCN1C)=O C1(C(N(CC(C)N(C)C(c2cocn2)=O)C)=O)CCc2n[nH]c(C)c2C1 N1(C(c2cc(C(N)=O)[nH]n2)=O)CC(CNC(=O)C(F)=CC2CC2)OC2CCCC12 Cc1ccccc1C=NOCc1sc(C2CC2(F)F)nc1C C(=O)(CCCCC(F)(F)F)NCC1CCC(C)(C)CN1C(C1CC12CCC2)=O Cc1cccc2c1CC(C(=O)NC(CNC(=O)CCCC1CCCC1)C(C)C)O2 C(=O)(C(F)CCC(C)(C)C)NCC1CC(NC(C(C)=C(CC)C)=O)C1 c1(CC)ccc(C=CC(=O)NC2CN(C(=O)CCn3ccccc3=O)C3CC23)o1 C1(N(C(=O)CN2CCSCC2)C)CC2CC1N(C(=O)C=Cc1cn(C)nn1)C2 C1(N(C(CCN(C(C)=O)C)=O)C)CCN(C(=O)C(C)OC2CCCC2)C1 N1(c2cccc(C(C)O)c2)CCCc2ccc(P(C)(C)=O)cc21 CC(C)C(C)C(=O)NCC(C(=O)NCc1ccc(OCCO)nc1)N(C)C N1(C(CCC2CC(OC)C2)=O)CC(NC(c2conc2C)=O)C2CCCC2C1 N1(C(C(C)O)=O)CC2CC1CCN2C(=O)CCc1cc(Cl)no1 C(CC(=O)NCC1(C)CCOCC1)(C(F)(F)F)NC(Cc1c(C)cnn1C)=O c1(C(N2CCC(C3N(C(C=CC=CC)=O)CCCC3)C2)=O)cc(F)c(Cl)cc1Cl N1(C(C(Cc2ccco2)NC(c2cc(CC)[nH]n2)=O)=O)C2CCCC1COC2 c1(C(N2C(C(=O)NCCN3CCN(CC)CC3)CSCC2)=O)c[nH]nc1[N+](=O)[O-] c1(-c2c(F)cccc2)nccc(=NCC2Cc3ccccc3O2)[nH]1 Cc1cc(O)c(Cl)cc1C(=O)NCC1CCN1C(C12CC1COC2(C)C)=O C1(C(=O)OC)CCC(C2CCCC2)CN1C(c1cc2occ(Br)c2[nH]1)=O C1(C(=O)NC(CN(CCCC)C)C)CN(C(c2cnns2)=O)C(C)(C)C1 N1(C(CSCC)=O)CC2CCN(CN(C)C)CC2C1.C12(CC1)N(C(C)C)C2=O N1(C(Cn2c(=O)ccc(C)n2)=O)CCC2(CCN(C(C3NC(=O)OC3C)=O)C2)C1 N1(C(c2scc(C(=O)OC)c2)=O)CC(C2CN(C(=O)C(C)CC(N)=O)C2)C1 C#Cc1ccc(CCCC(=O)Nc2cnn(CCN3CCNC3=O)c2)cc1 C#CC1CCCCN1C(c1ccc(CNC(=O)C(O)C(C)C)nc1)=O Clc1cc(CCCn2cc(CCC3CCOCC3)nn2)on1 C(=O)(C(O)CCC(C)C)N1C(CNC(Cc2nc(CC)sc2)=O)CCCCC1 C1(NC(c2c(C)nco2)=O)CCCC12CCN(c1ccncn1)C2 C(=O)(CCS(=O)(=O)NC)N1CC(CCC)C(NC(=O)C(C)CN(C)C)C1 c1(C(N(CCNC(c2cnnc(C3CC3)c2)=O)CC)=O)cc2cccnc2cc1F n1(CC)nc(C(=O)NCC(C2CCCC2)NC(=O)C(C)CN(C)C)ccc1=O CCCC(C(=O)N(C)CCC1CCN(C(=O)C(C)(O)C(C)C)CC1)S(N)(=O)=O C(CCN=c1[nH]c(=NCCC(OC)OC)[nH]c2c1COC2)n1c(CCC)ncc1 Cc1ccc(NC(C2(C)CCCN2C(c2cc(F)ccc2Br)=O)=O)c(C(N)=O)c1 c1(SC)cc(C(N2C(C(c3ccccc3)=O)CC2C(=O)OC)=O)c(C)o1 c1(C(N2C(CNC(C(C3CCCC3)OCC)=O)CCC2)=O)ccc(C(F)F)cc1 CN1CCN(C(=O)CCCNC(C23CCCN2CCC3)=O)CC1(C)C C(=O)(CC(C)C(C)(C)C)NC1C(NC(Cc2nc(C(C)C)sc2)=O)C1 Cc1cccc(CCC(=O)N(C(C)CCNC(C2CCC2)=O)C)c1Cl c1(CNC(=O)N(CCc2cccs2)CC2CC2)nnc2n1CCCC2C(F)(F)F C1(CN(C(C(CC)O)=O)C)CN(C(=O)CCn2ccnn2)CC12CC2 N1(C(C2CC(C)(F)C2)=O)CCC2C(CCCN2C(=O)C=CSCc2ccco2)C1 C=CC1(C(=O)NC2CN(C(c3ccnnc3O)=O)CCC2CO)CCCCC1 C1(NC(=O)CC2CCCOC2)CC2CN(C(c3ccc4cncn4c3)=O)CC2C1 N1(C(c2scc(CC)n2)=O)CCC(O)C(C(=O)Nc2cc(Cl)cnc2OC)C1 CN1C2(CCN(CC3CCCCC3)CC2)C(NC(c2ncccn2)=O)CS1(=O)=O N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)CCCCCC(C)O)C2CCCC12 CCC(C)CCC(=O)N1CCN(C(C2COCCOC2)=O)C(C(C)C)C1 N#Cc1ccc(C(=O)NC2C3CN(C(c4coc(Cl)n4)=O)CC23)c(O)n1 Cc1cc([N+](=O)[O-])cnc1N1CC2(CN(C(c3ccc4c(c3)OCC4)=O)C2)C1 c1(C(N2C3C(NC(c4ccccn4)=O)CC(C3)C2)=O)cc2cn[nH]c2cn1 C1(C(N(CCNC(CCCNC(C)=O)=O)C)=O)COCCN1C=O N1(C(C2N(C)C(=O)NC2)=O)CCC(C2CCN(C(=O)C(C)(C)CCC#N)CC2)C1 c1(C(=O)NC2(C3CN(C(Cc4ncc(C)s4)=O)C3)CC2)noc2c(F)cccc12 C1(C(N(C)Cc2nc(C)sc2)=O)CN(C(=O)C=CC2CC2)C2(CCC2)C1 c1(NC(=O)NCCN(C)C(=O)OC(C)(C)C)ccc(Br)cc1-n1cncn1 c1(C(=O)NCCN(C(CCOC)=O)CC(C)O)ccc2n[nH]c(C)c2c1 C(CCCCC(=O)NC1CCN(C(c2cc(C)c(C(F)F)cn2)=O)C1(C)C)=CC CCCCCS(=O)(=O)CC(=O)Nc1ccc2c(c1)N2C.c1(NC)ccc(F)cc1 c1(SC)ccc(Cl)c(C(=O)Nc2ncc(CN3CC(C(=O)OC)C(O)CC3)nc2)c1 C1(CC(=O)NCC2(C)CCC2)C2CCCC2N1C(C1(N)CCC1)=O.C(N)=O Cc1onc(Cl)c1C(=O)NC(C)CCCNC(=O)CCCOc1ccc(F)cc1 C(CCC(=O)NCC1CCCC1C(=O)NCc1cnns1)OCC C1(C(=O)NCC(C(C)C)NC(CCc2onc(CCC)n2)=O)CCCCC1(F)F C12(C(=O)NCC3N(C(C(C(=O)OC)OC)=O)CCCC3)CCCC(C1)OC2 C=CC1(NC(C2CC(CCNC(=O)C=C3CCOCC3)C2)=O)CCOCC1 C1(C(=O)NC2C3CC2CN(C(=O)CNS(=O)(=O)C2CC2)C3)CCCN2CCCC12 C=C(CNC(=O)Cc1ccccc1)CCNC(C1(C=C)CC1)=O c1(OC)ccc(CNC(C2CC2NC(=O)C2CC2)=O)c(C)c1 c1(NC(c2ccc(Cl)nc2F)=O)ccc(NC(C2COCCO2)=O)cc1F c1(C(=O)NCC(C)CNC(=O)CN(C)C(c2cccs2)=O)cc2sccc2n1C C1(CC)C(C(=O)N(CC(O)CN(C)C(c2cc(Br)ccn2)=O)C)CCN1C C(=O)(CC1OCc2cc(Cl)ccc21)NC1CN(C(CNS(C)(=O)=O)=O)C(CO)C1 c1(C(=O)NCC2(F)CC(NC(C(C)O)=O)C2)c(Cl)cc(Cl)nc1N C(N=c1[nH]c2ccc(Cl)cc2s1)C1CCCC(NC(C2CC(C)OC2)=O)C1 c1(C(=O)NC(CNC(C(CC)OC)=O)CO)ccc(OCC(N)=O)cc1 C1(CC(=O)N(C2CCCC2)CC#C)C2CCCC2N1C(C1CC(CC2CC2)C1)=O N1(C(CC(C)(C)C(F)(F)F)=O)CCC2CC(NC(=O)CS(N)(=O)=O)CCC2C1 C(CC1=CCCCC1)NC(C1C(NC(C(CCSC)O)=O)CC=CC1)=O c1(CC(C)(C)C)nc(-c2cc(CO)[nH]n2)n(C2(C)CCCCC2)n1 Cc1cccc(C)c1C(O)C(=O)NCC(C)(C)NC(c1cc(Br)n[nH]1)=O C1(C)(C(=O)OC)CC(NC(=O)C(C)N(C(=O)COCC(C)SC)C)C1.N1CCCC1 N1(C(CC)=O)CCCCC1C(N1CC(CCNC(=O)CCC2CCCN2C)C1)=O C1(CNC(C(C)CO)=O)CCCC2CN(C(=O)CC3(N(C)C)CCCC3)CC12 CCCCCC(C(=O)N(C)CC1CN(C(=O)CCCOCCOC)CCO1)C(C)C C12(CNC(C(CC#C)C)=O)CCC1CN(C(c1ccc(Br)cc1O)=O)C2 C1(C(=O)NC2(C)CC(NC(COCC)=O)C2)Cc2cc(C)ccc2S1(=O)=O c1(C2CN(Cc3c(OC)cc(F)cc3F)C2)nnc2ccc(SC)nn12 c1(C(=O)NCC23C(CN(C(C(CCC)OCC)=O)C2)C3)cc(F)ccc1C C1(NC(=O)NCc2cc(C(=O)OC)cc(F)c2)CCC2=NN=NN(C2)C1 C1(CNC(=O)CCn2cnnn2)CCC2(CO1)CC(NC(c1csc(Cl)n1)=O)C2 c1(C(=O)NC(c2n(C)ncc2)C(N2CCCC(CC3CC3)C2)=O)ccc(O)cc1 C1(c2nnnn2C2CC2)(Nc2cncc(NC(C)=O)c2)CCN(C)C(C)C1 N1(C(C(C2CCC2)OC)=O)CCCCC(CNC(c2cc3n(n2)CCO3)=O)C1 CCC1C(=O)Nc2ccc(C(=O)N(CCCOCCNC(C3CC3F)=O)C)cc21 C(C(C(C)C(C)C)NC(C1(CCF)CCC1)=O)NC(CCNC(C)=O)=O c1(C(=O)OC)sc(NC(c2ccc(NC(c3cn(C)cn3)=O)cn2)=O)nc1C N1(C(C=COCC)=O)CCC(CNC(c2cn(C)c(=O)nc2O)=O)C12CCC2 C1(C(N2C(CNC(=O)Cc3ccon3)CCCCC2)=O)CC1C1CCCCC1 CCCCCCCC(F)C(=O)NCCC1CN(C(=O)C=NOC)C1 Cc1ccc(O)c(CC(N2CC(NC(C3(C)CCCCCC3)=O)CC2(C)C)=O)c1 Cc1nc(CNC(C2CC3CCC2C3)=O)oc1C(=O)N(C)Cc1cnnn1C c1(OC)ccc(C(=O)NCC(C2CCC2)NC(=O)C(=Cc2cnn(C)c2)C)nc1 C12(C(c3n(CCCC)nnn3)NCC3(CC4CC4)CCC3)CCCC1C2(F)F c1(N2CC(CNC(C(COC)O)=O)N(C)CC2)cc2c(cn1)C(=O)CCC2 c1(CCC(=O)N(C(C)C)CC2CN(C(=O)COCCF)C2)ccccc1[N+](=O)[O-] C(=O)(C1SCCc2sccc21)N(C)CC1CN(C(C2CC(O)C2)=O)CCO1 C1(CC(=O)N(CCC(=O)N(CC(C)C#N)CC)CC)COCC(C)O1 C(=O)(CC(F)(F)Br)N(C)CC1N(C(c2cc(C)ns2)=O)CCC1 c1(CNC(C2N(CC)CCOC2)=O)ccc(CNC(C2CC2F)=O)c(F)c1 CC1CN(C(C2CC3C(C2)C3(F)F)=O)CCN1C(=O)Cc1ccc(Cl)s1 C1(N(C(CNC(C(CC)C)=O)=O)C)C2CN(C(c3csc(COC)c3)=O)CC12 C(=O)(C(C)C(O)CC(C)C)N1CCC(COC)(CNC(C2CC(C#N)C2)=O)CC1 CC(C)CC(C)CC(=O)N1CC2(CCCC2)C1C(=O)NCC1CCCCO1 c1(C(=O)NCC(C)N(C)CC2CCC3CC3C2)ccc2sccc2c1 N1(C(C#CCNC(Cn2c(C)nnn2)=O)=O)CC(C#N)(N(C)C)C1 C(=O)(CCCC(CC)NC(C1Cc2nccn2C1)=O)Nc1ccc(CC)nc1 C(CCN=c1nc2scnc2c(N2CCC(S(C)(=O)=O)C2)[nH]1)C1(C)CC1 N1(C(C(C(C)NC(c2c(C)non2)=O)C)=O)CC2OC(=O)N(C)C2C1 N1(C(C(C2CCOC2)NC(CC(CC)C(C)C)=O)=O)CC2CCOC(=O)C2C1 c1(OC)ccc(F)c(C(=O)NCC(O)COCC(C)C)c1F Cn1ncc(C(N)=O)c1C(=O)N(C1CCCCC1NC(C1(C)CC1(F)F)=O)C C1(NC(c2n(CC=C)nnn2)c2occc2Br)CCOC(c2cccc(Cl)c2)C1 CC1(C)OC(C)(C)C1C(=O)NCC1CCCCC1NC(=O)CCn1cnnn1 C(=O)(C1=NOC2COCC12)N1C2CCC(NC(C3CCC(CC)CC3)=O)C(C2)C1 C1(C(c2cn(CCCC(=O)O)nn2)NC(c2cc(OCC)n[nH]2)=O)CCCCCC1 CCCC(C)(O)CC(=O)NCC(C)=CC(=O)NCC(N1CCCC1)=O C(=O)(C(C)(C)CCC(=O)NCC1CCCC2(CN(C(=O)CCCF)C2)O1)OC N1(C(c2cn(CC=C)nc2)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)CC1CF C1(C(=O)Nc2ncn(C)n2)CN(Cc2c(Br)cncc2Br)CCC1O N1(C(C2(C#N)C(C)(C)C2)=O)CC2(C1)CN(C(C1C3CC4C(C3=O)C14)=O)C2 C(N=c1[nH]cnc(Cl)c1C(=O)OC)C1CC(NC(C=COCC)=O)C1 c1(C(N(C2CCCN(C(=O)C(C)CO)C2)CC)=O)cc(C(F)(F)F)cc(F)c1 N1(CC(=O)NC(=O)C2CC2)CCC2C(CCCN2C(c2sccc2Cl)=O)C1 N1(C(CCC2CCN(C(C(C=C)O)=O)C2)=O)C2CCCC1CC(=C)C2 C(=O)(CC(C)C(=O)OC)NC1CCN(CCNC(C=COCC)=O)CC1 c1(C(N(CCN(C(C2CCC(CCC)CC2)=O)C)C)=O)ccc2nn[nH]c2c1O N1(C(C2CSCCN2Cc2cscc2F)=O)CC(c2ccccc2)C2(COC2)C1 c1(C(=O)NC(C2CCCC2)CNC(C2(C)C(C)C2)=O)cc2n(n1)CCCO2 N1(C(C2N(C(C3CC(OC)(OC)C3)=O)C(C)C2)=O)CCC(F)C(F)C1 c1(-n2c(C(C3(CCl)CCC3)NC(CCC=C)(C)C)nnn2)ccc2c(c1)CCC2 CN1C(=O)NCC1C(=O)NC1CC(CNC(=O)CC2(O)CCCCC2)C(O)C1 C1(CCN(C)C)CCOCC1.c1(C2CN2)ccccc1 N1(C(c2c(C)con2)=O)CC2CC(C1)CN(C(c1cc3ccnn3cn1)=O)C2 N1(C(C23C(C)OC(C)(C2)C3)=O)CCC(C2CC2)(CNC(c2ccc[nH]2)=O)C1 N1(C(c2ccc(SC)o2)=O)CCC2(CCN(C(=O)C(C)C3CCC3)C2)C1 N1(C(CC(CC)C)=O)CC2C3CCC(C2C1)N(C(C1CCC2(CCOC2)O1)=O)C3 C1(C(=O)NCC2CCN2C(=O)CCc2ccccc2F)CC12CCSCC2 S(=O)(=O)(c1ccc(Br)c(F)c1)N1CC(C(=O)Nc2nccnc2Br)C(O)CC1 N1(C(CC=CCC)=O)CCOC(CCNC(C2(C#N)CCOC2)=O)C1 C12(C(=O)NC3CCC(NS(CC(=O)OCC)(=O)=O)CC3)COCC(C1)OC2 CCCC(C(=O)N(C)CCOCCOC)NC(=O)C(N1CCSCC1)C c1(C(=O)NCC(C)NC(=O)C(c2ncc(Cl)n2C)(F)F)cc2cc(Cl)ccc2o1 N1(C(CC2C(NC(CNC(=O)OCC=C)=O)CCC2)=O)CCCC(N=[N+]=[N-])C1 c1(CC)cc(CNC(=O)CN(C2CCC2)C(c2scnc2Cl)=O)n[nH]1 C1(CS(Cc2c(CC)occ2)=O)CCS(=O)(=O)C1.c1(C2C(=O)N2)ccccc1 c1(OC)cc(NC(C2CC(F)CN(C(c3c[nH]cc3C)=O)C2)=O)nc(Br)c1 c1(C(N(CCCNC(CC(C)OC)=O)C(C)C)=O)cc(C2CC2)cc(F)c1 C12(C(=O)NCC(=C)CCNC(c3cncc(C)c3)=O)CCCC1NC(=O)C2 C1(C(=O)NCCCCNC(CC)=O)CCC(=O)N(CC)C1 c12n[nH]cc1C(=O)N2.C(C(=O)NCCCC1(C)CC1)SCCC CCCC(C)CC(=O)N(CC(CO)(CO)NC(c1cnc(C2CC2)[nH]1)=O)C N1(C(c2c(C(C)NC(c3cnc(O)o3)=O)noc2)=O)Cc2ncsc2C1 N1(C(C(CC)COC)=O)CCc2ccc(C(=O)NC3CC3C3CC3C)nc2C1 c1(CNC(=O)C=C2CCCCC2)ccc(CCNC(C2CC23CCOC3)=O)cc1 C=CCCCC(C(=O)NCCCO)NC(=O)Cc1ccc(C#N)cc1 N1(C(C(COC)O)=O)CC2CN(C(c3ccnc(OCCO)c3)=O)CC2C1 C1(F)(C(N2CC3C(CNC(COCCCC#C)=O)C3C2)=O)C(C)(C)C1(C)C C1(NC(CCC2CC(OC)C2)=O)CN(C(C2(C#N)CC3(CC3)C2)=O)CCC1CO c1(Cc2n(CC)c(CN(C3CCC(C)C3)C)nn2)c(F)cccc1F c1(C(=O)NC2C(CC)CN(C(c3csc(O)n3)=O)CC2)noc2cc(F)ccc12 C1(CNC(CCC(=O)OC)=O)(NC(=O)CCC2NC(=O)NC2=O)CCCCC1C N1(CC(=O)NC2C(C)(C)CCC2)CCN(C(C2(N)CCC2)=O)CC1=O Cc1nc(NC(C)(CNC(=O)C(C)C(C)O)Cn2cccn2)ccc1[N+](=O)[O-] c1(CNC(=O)NC2CCNC2)ccc(-c2ccc(C(F)(F)F)c(F)c2)cc1F c1(NC(Cn2cc(CNC(C3C(C)CCC3)=O)nn2)=O)ccc(O)c(F)c1 C1(NC(c2c(C(C)=O)ccs2)=O)CCOCC1NC(c1ccc(C(F)F)cn1)=O c1(OC)ncc(C)cc1C(N1CC2(NC(=O)C(C)N(C)C)CC1C2)=O CC1OC(C)C(C)N(C(=O)NC(c2nccn2C)C)C1C c1(C(=O)NCC2CC(C)N(C(C3CC3(Cl)Cl)=O)C2)cnc2[nH]nnc2c1 c1(C(N2CCC(CCCNC(CC3C(C)C3)=O)CC2)=O)ccnc(Cl)c1N c1(N(C(C(=O)Nc2c(C)cccc2)CC2CC2)C)ccc(SC(F)(F)F)cc1Cl c1(OC)ccnc(O)c1C(N1CC=CC(NC(c2nccc(C)n2)=O)C1)=O C1(N(C(C(C2CCC2)OCC)=O)C)CCCN(C(=O)Cn2ncc(Cl)c2C)C1 N1(C(c2c(C)nns2)=O)CCC(C)(CCNC(c2cn(CCCC#N)nn2)=O)C1 c1(C(=O)NC(C)C(C2CCCC2)NC(=O)C(C2CCOCC2)=O)ccc(CO)nc1 c1(N(CCN(C(=O)Cc2nn(C)cc2Br)C)C(=O)C2CC2)cc2occc2[nH]1 N1(C(C2CCCC23CC3)=O)CC2CCCC(C1)N2C(c1c(F)ccc(F)c1O)=O C1(CNC(C2C(CC)CCC2)=O)CCCC12CCN(C(C1C=C1C)=O)CC2 c1(C(=O)OC)nccnc1C(=O)NC(C)CC(C)NC(=O)C(c1cnn(C)c1)O c1(C(C)=O)ccc2c(c1)CN(Cc1ccc(-c3ccc(N)cc3Br)o1)CC2 Cc1nnc2n1CC(C(N1CCC1CNC(=O)CCc1ccc(C(F)F)o1)=O)C2 N1(C(C2C(=C)C2)=O)CCN(c2ncnc(Cl)c2CO)C(C)C1 C1(C(C)C(=O)NCC=CBr)CCN(C(=O)CCc2cccn2C)C1 c1(C(c2nnnn2CCCF)NC(c2ccc(C)o2)CC)ccc(OC)nc1 c1(C(=O)NCC2(OC)CCN(C(C(CC)SC)=O)C2)cc2ccc(OC)nc2[nH]1 c1(C(=O)N)c[nH]c2ncccc12.C1(OC)CC(CO)(NC(c2ccc(C(N)=O)o2)=O)C1 C1(=CCNC(C(C)=CC)=O)CCN(C(=O)Cc2ccc(-c3ccsc3)cc2)CC1 c1(CC)cc(C(N2CCCCC2c2cn(Cc3cnn(C)c3)nn2)=O)c(C)o1 CC1COC2(C1)CN(C(=O)C#CCNC(c1csnc1Cl)=O)C2 C1(C(=O)NCC(=O)OCC=C)CSCN1C(C1CC(OC2CC2)C1)=O CC1(CCNC(c2csnn2)=O)CCN(C(C2CC3CC(=O)C2O3)=O)CC1 N#CC1(C(=O)NC2COCCC2NC(C2(C3CCC3)CC2)=O)CCCC1 CCCCC(C(=O)NCCN(C)CC)NC(c1cc(C)cc(O)n1)=O N1(C(c2n(C(C)C)ncc2)=O)CC2ON=C(CNC(c3ccsc3)=O)C2C1 c1(CC)cc(C(N2CC(CC(C)NC(=O)C=CBr)C2)=O)ccc1F c1(C2(C)CC2)cc(C(=O)NC2COCC2NC(=O)CC2CCOCC2)no1 c1(CNC(c2ccccc2OC)C(=O)OCC)nc2c(s1)CCCC2 C1(C(=O)NCC(CO)NC(c2cnc(N(C)C)s2)=O)CCOC(=O)N1 C(=O)(C(C)CCCC(C)C)NC1CC2CN(C(c3ncc(C)nc3)=O)C(C1)C2 CC1CN(C(C2CCCC(F)C2)=O)CCC1CNC(c1c(O)cccc1Cl)=O N1(C(c2c(OC)c(C)cs2)=O)CC(NC(=O)C(C)=C2CCCC2)C(C)(C)C1 C(=O)(C1=CCCCO1)NC1CCC(CCNC(=O)Cc2nc[nH]n2)C1 C1(CC(=O)NCC(N(OC)C)=O)CCN(C(=O)C(C)CC#N)C1(C)C c1(CN2CC(CC(=O)N(C)CC3CCC(=O)N3)OCC2)ccc2occc2c1 c1(C(=O)NC2(COC)CCC2)n[nH]c2c1CN(C(C1(C)CCN(C)C1)=O)C2 Cc1cc([N+](=O)[O-])cc(Cl)c1NC(=O)CC1CN(Cc2cc(C#N)ccc2Cl)C1 Cc1cncc(C)c1C(=O)NCCCCC(=O)NC(c1ccccc1O)C C1(CC(N2CC(C)(OCC(=O)N(CCCOC)CCO)C2)=O)CCCC(C)O1 C1(C(=O)NCC2(CO)CC2)(CNC(c2c(C)noc2)=O)CC12CCC2 c1(OC)cccc(C(C)C(=O)NC(C)C(C)NC(=O)CSC)c1 C(=O)(C1CCCc2nn[nH]c21)N(CCOCCCNC(C1C(C)C1C)=O)C N1(C(c2c(CC)cc(Cl)cc2)=O)CC2(CC(NC(=O)C(C)(Cl)Cl)CO2)C1 N(C(=NCCC1CC1)NCc1cncnc1)CCC1CCCC(C)C1 C1(C(=O)NCC(C)NC(c2cocn2)=O)CCCCC1P(C)(C)=O C(CCCCC(=O)N1CC(O)CC1(C)C)N(C(C1C(CC)CCO1)=O)C c1(OC)ccc(C2CC2C(=O)NC2(C)CCCN(c3cc(C)nc(Cl)n3)C2)c(C)c1 C(=O)(C(C(C)C)NS(C)(=O)=O)NC(C1CCCCC1)CNC(c1c(C)occ1)=O N1(C(COCCC)=O)CC(O)C(O)C1CNC(=O)CC1OC(C)(C)OC1=O c1(CNC(=O)NC2(C3CC3)CC2)cc(Cl)ccc1[N+](=O)[O-] S(=O)(=O)(c1ccccc1Br)N1CCC(CN(C(C(C)(C)C)=O)O)CC1 C(CC(C)C)(C(=O)N(C1CC=CC1)C)ONC(c1ccc(N(C)C)cn1)=O C1(C(N(CC(C)NC(CN(S(CC)(=O)=O)C)=O)C)=O)(OC)CCSCC1 C1(C(=O)OC)Cc2ccsc2CN1C(=O)C(=O)NCCc1ccc(C)cc1[N+](=O)[O-] C1(NC(COCC(=C)C)=O)CCN(C(C23CCCC2C3(F)F)=O)C12CCC2 c1(C(=O)NCC2CCN(C(C(CN(CC)CC)F)=O)C2)c(F)cc(F)cc1Cl c1(CCC(=O)N(CCN(C)CC2CCN(CC)C2)C)ccc(O)nc1 c1(C2(C(=O)NC3CC(CCNC(=O)Cn4ccnn4)C3)CC2)ccc(Cl)c(F)c1 N1(C(C(C=C)OC)=O)CC(C(=O)NC2(COC)CCC2)C(C2CC2)C1 N1(C(C(C(C)C)NC(N)=O)=O)CCCOC(CNC(C2COCCO2)=O)C1 CC1CCCC=C1C(=O)NC1CC(C(C)NC(c2c(F)cc(F)cc2F)=O)C1 CCC(C)C(O)CC(=O)NC(C(=O)NCCC(F)(F)CO)c1ccoc1 N1(C(C(CC=C)C)=O)CC2CCCC(C1)N2C(C1CCN(CC(F)(F)F)CC1)=O C1(C(C)C)C(=O)NCCN1C(C1CCN(C(c2n[nH]c(C(F)(F)F)c2F)=O)C1)=O N1(C(C(CC)=CC)=O)CC(CNC(c2cc(-c3ccccc3)ns2)=O)CC1C C=CCC(C)C(=O)NC(C)C(C1CCCCC1)NC(=O)CCCNC(=O)C1CC1 N1(C(c2c(C)ccs2)=O)CCC2(C1)CN(C(=O)CCc1ccc(C(C)C)cc1)C2 N1(C(CN(CC(=O)NC(C)C)C)=O)CCN(C(C2(C)C=CCC2)=O)CC(C)(F)C1 CC#CCC(CO)NC(C1(NC(=O)CCc2ncccn2)CCCC1)=O C1(NC(c2ccc(CC)nc2)=O)CCC12CN(C(=O)C=CC(=O)NC1CC1)C2 c1(C(=O)OC)cccc(C2CC2)c1.C1C(C2(C)CC2)N(C)C(=O)N1.C1(C)CC1 c1(C(=O)NC2CC(NC(=O)COCc3nc[nH]n3)C2)cc(C2CC2)cc(F)c1 c1(CNC(C(c2ccsn2)N(C2CC(F)(F)C2)CC=C)=O)cccc([N+](=O)[O-])c1 C(CCCC(C)NC(=O)CCCOc1ccc(C)cc1)NC(CC(=O)OCC)=O C1(C(N2CCCN(CC(N3CCOCC3)=O)CC2)=O)CC2(CCC2)CCO1 O=C(N=c1c(Br)c[nH]cc1I)C1CCN(S(=O)(=O)C2CCCCC2)C1 c1(C(=O)NC2CCC3CC2CN3C(C2CC=CC2)=O)coc2ccc(F)cc12 C1(NC(C2(CC)CC2)=O)CN(C(=O)C(c2cccc(Br)n2)C)C(C)(C)C1 c1(CNCCCCCC(C)(C)C)cccc(S(=O)(=O)NC2CC2)c1 C12(CNC(COCCOCC)=O)CC1CN(C(=O)COc1nc(C)no1)C2 N1(C(C(C)(C)SCCC)=O)CC2CN(C(=O)C3CC3)CC2C1.C1(=O)CCCCN1 Cc1nc(N(C)C)sc1C(=O)N(CCCCN(C)C(C1CCCC1C)=O)C Cc1ccc(F)c(C(=O)N(C(CC(C)C)C(=O)NC2CCN(C(C)(C)C)C2)C)c1 C=C(C)CC(C(=O)NCCc1cnn(C)c1C)NC(=O)CNc1ccccn1 c1(C(=O)NCC(CNC(CCC#C)=O)F)cc(F)ccc1-n1ccnc1 c1(C(=O)NC(CNC(CC(CC)C)=O)(C)CC)ccc(C)c(N)c1 CC1(C)CCCCC1NC(=O)CC1C2CC1N(C(C1CN3CCC1CC3)=O)C2 C(CCCC(=O)N1CCC(CCNC(=O)CCc2cncs2)CC1)NC(N)=O N1(C(CC(=O)NCC#C)=O)CC2(CC(CC(=O)NC3(CC=C)CCOC3)C2)C1 C1(F)(CNC(C(=Cc2cn[nH]c2)C)=O)CCC(NC(=O)CC2CC2(Cl)Cl)C1 CC(O)C(F)(F)C(=O)NCC(C)(C1CCC1)NC(=O)CN1CCCCC1=O N1(C(C2C(C)CCC2)=O)CCC(C)(CCNC(C23CCC(C2)C3)=O)C1 C1(NC(C)=O)CCCN(Cc2cnn(C)c2CCO)C1 c1(C(N2CC(NC(C3CCCC3)=O)CC(C)(C)C2)=O)cc(F)c(C#N)c(F)c1 C1(N)(C(=O)NC(C(=O)OCC)CSC)CCOCC1(C)C C#Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(C)(C)C2)=O)ccc1C Cc1ccc(C(N2CCC(C(F)(F)F)C2C)=O)cc1S(=O)(=O)N(C)C C12(C(=O)NCc3c(C)non3)CC(C)(CN1C(c1sccc1C#N)=O)C2 c1(CC)cc(C(c2nnnn2C(C)C)NCCO)ccc1NC1NC(=O)NC1=O N1(CC(=O)NC(=O)NC(C(=O)NC)Cc2ccncc2)CCC(C(=O)OC)CC1 CC(C)C(C(=O)NC1CCN(C(C2(C)CCC2)=O)CC1F)C(C)C C(=O)(C1COc2ccccc21)N1CC2CCN(C(c3n(C=C)nnc3)=O)C2CC1 C1(CNC(CC(C=C)CC)=O)CN(C(C2CC(CC(F)F)C2)=O)CCC12CCC2 N1(CC)CCCC(C(=O)NC2CC(O)(CNC(c3csc(C(F)(F)F)n3)=O)C2)C1 C(=O)(C1CCc2nccn21)N1CCCC(C(=O)NCCn2cncn2)C1 N1(C(CSCCSC)=O)CCC(C(CO)NC(=O)CCc2ccon2)CC1 CS(=O)(=NC(=O)CCn1cc(Br)cn1)c1ccccc1Cl CC1CC(CNC(=O)NC2(C(F)(F)F)CC=CC2)CC(C)O1 c1(NC(C=CC(C)NC(c2ccc(CO)nc2)=O)=O)ccc(O)cc1Cl CC1COCC(C(=O)NC2CC(O)(CNC(c3ccnn3C3CCC3)=O)C2)O1 C1(C(C)(C)C)CCN(C(C2CCCOCC2)=O)C(CNC(c2cc[nH]n2)=O)C1 N1(C(C(CCO)N(C)C)=O)CC2CS(=O)(=O)CC2(CNC(c2cnco2)=O)C1 Nc1ncc(C(=O)NCCOC2CCN(C(=O)C=CC3CCC3)C2)cc1Br c1(NC)cnccc1C(=O)N(CC(N1CC(N2CCOCC2)C1)=O)C1CCC1 CC(Cc1cnn(C)c1)C(=O)NC1CN(C(=O)COc2ccsn2)C1 N1(C(CNC(C(C)(C)OC(C)C)=O)=O)CCC(O)C(C)(C)C1 C1(O)(C(=O)NC2C3(CC(NC(c4scc(C)c4)=O)C3)C2)CCCC(C)(C)C1 N1(CC(=O)NC2CC(CNC(=O)CC3CCC4CC34)C2)CCCS1(=O)=O C1(CCNC(c2ncn(CC)c2)=O)C(C)CCCN1C(=O)C1=COCCC1 c1(NC(=O)NC2CC(Nc3ccccn3)C2)ccccc1CC1CCOCC1 c1(C(=O)NC(C2CCCCC2)CO)cncc(NC(c2ccc(Br)cc2)=O)c1 c1(C(N2CCCC3(C2)CN(C(C2CC=CC2)=O)C3)=O)ccc2cc[nH]c2c1F c1(N2CCN(CC(C)(C)NC(=O)C(N)=O)CC2)nc(Cl)nc2c1CCOC2 C1(NC(C(CC=C)CC=C)=O)CN(C(=O)Cc2[nH]cnc2C)CCC12CCC2 N(C1CCc2c(Br)cccc21)C(=O)NC1C(c2c(C)cccc2)(C)C1 C(=O)(CC(F)(F)C(F)F)N1CC(CC=C)(NC(c2nonc2CC)=O)C1 C1(CNC(CC=CCNC(CCCOC)=O)=O)COCC(C)O1 Cc1cc(CC(=O)NC(C)CNC(=O)C(F)CC2CCCCC2)on1 C1(NC(CN(CC)CC)=O)CCC(CN(C(=O)CNS(N)(=O)=O)C)CC1 O(N=C1CCCCCC1)CC(N1CC(OC)(CNC(=O)C(O)CN(C)C)C1)=O C1(C(N2C(C(N(C)Cc3cnc[nH]3)=O)CC(O)C2)=O)CCCC2(CC2)C1 C1(C(=O)OC)CN(C(=O)C(=O)NCC(c2c(Cl)cccc2Cl)(C)C)CCN1C N1(C(C(C)Oc2ccccn2)=O)CCc2[nH]nc(CNC(c3cnco3)=O)c2C1 N1(C(c2c(C)c[nH]n2)=O)CC(NC(=O)Cn2nnc(=N)[nH]2)C2(CCC2)C1 N1(C(C=Cc2ncn(C)c2)=O)CC2CC(C1)N2C(c1nocc1C1CC1)=O N1(C(c2c(OC)csc2)=O)CC(NC(C2(O)CCSC2)=O)CC(O)C1 C(=O)(C(=O)C(F)(F)F)NCC1CCCC(NC(c2c(CC#N)ccs2)=O)C1 c1(NC(C2(NC(C(C)CCN(C)C)=O)CC(F)C2)=O)cnc2[nH]ncc2c1 C12(NC(C(c3ccc(CC)s3)=O)=O)CC1CN(C(C1CCC(C)CC1)=O)C2 C1(CC2(C(=O)N)CC2)COCC1NC(C1CN(C2CCOC2)C1)=O.CO Cc1nc2ccc(C(=O)NC3CC4CC3N(C(=O)CC35CCCC3C5)C4)cc2o1 c1(CCC)nc(NC2CCCN(C(=O)CC)C2)c(C)c(Cl)n1 N1(C(C(C(CC)C)c2ccccc2)=O)CCC(C#N)(C(C)(C)O)CC1 N1(C(c2c(C(C)N)noc2)=O)CC(=O)N2CCCCC2C1 c1(C(N(C(CN(C(C(C)SCC)=O)C)C)C)=O)cc2c(cn1)OCCO2 Cc1c(C(=O)CNC(=O)C(c2ccc(Cl)cc2)C2CC2)sc2ccccc12 N1(C(C2N(CC)CCC2)=O)CCN(C)C(C(=O)NOC(CO)CO)C1 c1(NC(N2CCC(N(c3ccccc3)C)C2)=O)ncnc2c1ncn2C c1(C(=O)NC(CCOC)CNC(=O)CC(F)(F)Cl)ccc(N=[N+]=[N-])cn1 CC(CS(C)(=O)=O)C(=O)N1CC2(CCCN2C(=O)CC(Cl)Cl)C1 Cc1ccc(C(=O)NCC2(C(=O)NCCC3NC(=O)NC3=O)CCCC2)nc1 Cc1nncc(C(=O)NCC23CC(C2)C(NC(=O)C(O)C2CC2)CO3)c1C N1(C(C(=O)NCCCCc2ccccc2)=O)CCn2c(cc3c(Cl)cccc23)C1 c1(OC)ccc(C(=O)NCC2C(C)CCN2C(c2coc(C(C)(C)C)n2)=O)nn1 C1(C(N2CC(CC(=O)NCC3CC(OCC)C3)(OC)C2)=O)CC12CCCC2 c1(S)cccc(O)c1.C1(C(N2CC(n3cc(C(=O)OC)nn3)C2)=O)CCC(C#N)C1 Cc1nc(C(F)(F)F)ccc1C(=O)NC1CN(C(=O)Cc2cscn2)CCC1F c1(C(C(=O)NCCC(=C)CNC(C2C3CCC23)=O)(F)F)ccc(C)cc1 N1(C(C(=O)NCCOc2cc(O)nc(O)n2)=O)CCS(=O)(=O)CC1CCO C1(C(N2CCCC(NC(CSCC#C)=O)C2)=O)CCCC2(C1)CC2(F)F c1(OCC)cccc(NCCC(C(C)C)NC(c2cnc[nH]2)=O)c1[N+](=O)[O-] N1(C(C(C)(C)C#N)=O)CC2CC1CC2NC(=O)CNC(c1cccs1)C1CC1 c1(C(=O)NC(CC=C)CNC(c2cc(OC)n[nH]2)=O)cc(O)ccc1OC(F)F C(C(F)(F)C(C)(C)O)NC(C1(CNC(CCC2N(C)CCC2)=O)CC12CCC2)=O c1(CN2CCC(O)(C(=O)Nc3c(C(=O)O)cc[nH]3)C2)cccc(F)c1Br C1(C(=O)OCC)CC(C)(C)CN1C(c1nccc(Cl)c1C)C(=O)NC1(C)CC1 N1(C(c2sccc2Cl)=O)CC(CO)C2(C1)CN(C(c1csc(O)n1)=O)C2 C(=O)(C(CCC)S(N)(=O)=O)N1CC(OC)CC(NC(C=CC=CC)=O)C1 Cc1ccccc1C(=O)NCC(N1CCN(C(=O)CC23CCC(CC2)C3)CC1)=O CC1CN(C(c2cc[nH]c(=N)c2)=O)CCC1NC(c1nccnc1Cl)=O Cc1csc2ncc(C(=O)NCCC3CCCN3C(=O)Cc3cccc(N)c3)n12 C12(NC(CSCC)=O)COCCC1CN(C(c1cnoc1C1CCC1)=O)C2 c1(C(C(=O)N(CC(C)O)CCNC(CC(=O)OC)=O)C)cc2ccccc2o1 N1(C(C2(NC(c3ccn(CC)n3)=O)CC2)=O)CC(CNC(=O)COC(C)=O)CC1C c1(C(N2CCCN(C(C(C)C3CC3)=O)C(C)C2)=O)cc2c(n1C)CCOC2 C1(CC(=O)NCC2CC(NC(=O)CCn3cccn3)C2)CCCCCO1 C(=O)(C1=C(C#N)CCC1)NC(C(=O)N(C)Cc1ccoc1)CCF N1(C(c2c(C)noc2N)=O)C2CCC1CC(NC(C1CCC3(CCC3)CC1)=O)C2 N#CC1(C(N2CCC(F)(CNC(c3cncn3C3CC3)=O)C2)=O)CC2(CC2)C1 Cc1cc(NC(=O)CCC2CCN(C(C3CC3C#N)=O)C2)cc(C)c1C Nc1ccnc(C(N2C3CCC2C(NC(=O)Cn2nccn2)C3)=O)c1Cl Cc1nc2c(C(=O)NC3CC3CNC(c3ccc(C)c(C#N)c3)=O)ccnc2[nH]1 CC1=NOC(=O)C1CC(=O)NC1CCC1NC(c1ccncc1OCC(F)(F)F)=O c1(C(=O)NC(CCN(C)C(C2CCC3CC23)=O)C(C)(C)C)cc(Cl)ccc1CO N1(C(c2cnc(CC)nc2)=O)CCC2(CCCN2C(C2OCCC2(C)C)=O)C1 CC(C)C(O)C(=O)NCC12CC1CN(C(c1ccc(CO)cn1)=O)C2 C1(C(=O)NCC2CCCN(C(=O)Cn3cncn3)CC2)Cc2cccc(F)c2O1 C1(CCNC(CC=CCC)=O)CC(F)(F)CN1C(C1CC2OC1C1CC21)=O CC(C(O)C(F)F)NC(=O)CC1CCN(C(=O)C#CC2CC2)C1 N1(C(CN(C2CCC2)C)=O)CCCCCCC1C(N1CC=CC1CF)=O c1(C(N2CC(NC(C(CC)(C)CO)=O)C(O)CC2)=O)c[nH]c2cc(F)c(F)cc12 C12(C(N3CC(=C(CNC(C(n4ncc(C)c4)C)=O)F)C3)=O)CCCC(CO1)C2 Cc1ccn(CC(=O)NC2(CCCCNC(C3CCOC3C(F)(F)F)=O)CC2)n1 CCC(CC(=O)N(CCN(C)C(C1(O)CC(F)(F)C1)=O)C(C)C)C(C)(C)C c1(C(=O)NCC(CC)NC(C(C2CCC2)OCC)=O)oc(Br)cc1C CC1(CNC(=O)C(CC#N)NC(N)=O)CCCN(C(=O)CC23COCC(C2)C3)C1 C1(O)(C(N2CC(F)(CNC(CNS(NC)(=O)=O)=O)C2)=O)CN2CCC1CC2 c1(C(COC(c2cc(NC)n(C)n2)=O)=O)cccc(F)c1Br c1(OCC(=O)NC2CCC(CNC(CCSCCC)=O)C2)ccc(F)nc1 C(C)(C)(CC(=O)NCC(C)(O)CSC)NC(C(CC)SC)=O C1(NC(c2ncc(CC)s2)=O)CCC(C)N(C(=O)CN2CCCS2(=O)=O)C1 C1(CNC(CC(=C)C)=O)CC2(CO1)CN(C(=O)CC1CCC13CCC3)C2 C1(CNC(C(Cc2cc[nH]n2)NC(=O)C=CC(F)(F)F)=O)C2CCCCC12 c1(N2CCC(NCC(C(C)C)NC(=O)C3=CCOC3)C2)ncccc1C(F)(F)F N1(C(COCCCOC)=O)CCCC12CCCN(C(c1cc(C)oc1C)=O)C2 c1(OCC)nc(NC(C)(CNC(C2C(C)OC(C)C2C)=O)C2CC2)ncc1C N1(C(C2(COCC)CC(=C)C2)=O)CCCCC1c1nn[nH]n1 c1(C(=O)NCCOC2CCN(C(CC=CCC)=O)C2)cc2ncccc2cc1Cl N1(C(C(c2ccco2)NC(CCC2(C#N)CCC2)=O)=O)CCC2CCCC12 Cn1cc(C(F)(F)C(=O)NC2CCC2NC(=O)CC2CC=CC2)cn1 C#CCC(CC#C)C(=O)NC1CN(C(=O)C(n2ccc(C)n2)C)CC1C1CC1 C1(C(=O)NCC(C)NC(c2c(C)noc2C(C)C)=O)CC(c2ccncc2)=NO1 c1(C(N2C(C3CCN(C(CCc4cc(C)no4)=O)C3)CCC2)=O)c[nH]c(=O)cn1 C1(CNC(C(=O)NCCCC(C)=O)=O)CCC(F)(F)CO1 Cc1cc(N)c(C(N2CCN(C(=O)Cn3cnnc3O)CC2C(F)F)=O)cc1C C1(NC(c2ccc(SC)o2)=O)CC(F)CN(C(=O)CC2CC2(Cl)Cl)C1 C1(NCCn2cc(C(=O)NCC3CC(C(C)C)C3)nc2)CC(=O)N(C)C1 C(CC1CCC1)(C(=O)NC1CCC2CC12)NC(C(C)=C1CCC1)=O c1(OC)ccc(-c2nc(-c3ccccc3CCCC)no2)cc1.N1(C(c2ccc(Cl)cc2)=O)CCN(c2ccccc2)CC1 n1(CC)ccnc1C(=O)N(CCC(=O)NCC(Cl)C(C)(F)F)C1CC1 C1(C(CC)NCc2cncn2C(C)C)Cc2ccccc2C1 C1(NC(c2c(C)cc(F)c(Cl)c2)=O)CC1C1CCN(C(=O)Cc2cnc[nH]2)CC1 C(=O)(C#CC1CCCOC1)NC1(CO)CCN(C(c2nn(C)c(Cl)c2)=O)CC1 N1(C(C2CC(OC)C2)=O)CCN(C(=O)C(C)C(=O)N2CCCC2)C(C)C1 N1(C(=O)C=Cc2cccs2)CC2CCN(C(C3COC4(CO)CC3C4)=O)C2C1 C1(C(=O)NCC(CC)O)C2CCCC2CN1C(C1CCC1C)=O CC(C)C(C)CC(=O)NCC(C)C(=O)N1CCCC1 C1(CC(=O)N(CCC)CCNC(c2ccc(CN(C)C)o2)=O)CCOCC1 C1(C(N2C(CC#C)CCCC2)=O)CN(C(=O)CC2CCOC2(C)C)CCC1(C)C N1(C(c2oc(C)c(CO)c2)=O)CCN(C(C2OCCC2C(F)(F)F)=O)CC1C CCC(CC(=O)N(C1CCN(C(c2ccn3nnnc3c2)=O)C1)CC)C(F)F c1(C(N(CCCCNC(Cn2c(C)cc(C(F)F)n2)=O)C)=O)ccc(Cl)cc1N Cc1cc(C(C)C)nc(=NCC(CC(C)C)NC(=O)CN2CCCCCC2)[nH]1 c1(OC)ccccc1OCC(=O)NC1CCN(C(c2ccnnc2Cl)=O)C1 c1(CCC(=O)N(c2cccnc2)C2CCCC2)nc2cnccc2[nH]1 N1(c2nccc(OC)n2)CCCC(C2(NC(C3CCCC4(CC4)C3)=O)CC2)C1 C1(CNC(C2(NC(C3C=C(C)CS3)=O)CC2C)=O)CC12CCOCC2 Cn1cc(-c2cc(C(=O)NCC3CCCC3NC(=O)CSC(F)F)on2)cn1 N1(C(=O)CCc2ccccn2)CCOC2(CCN(C(=O)Cn3ccnn3)C2)C1 C1(NC(c2c(CC)nc(=N)[nH]c2)=O)COC2(C1)CN(C(=O)C1=C(Cl)CCCC1)C2 CCCC(C)C(=O)NC1(C)CN(C(C23CCC2C3)=O)C1 N1(C(C(C)n2cccn2)=O)CCC=CC1C(=O)Nc1cnc(N(C)C)nc1 N1(C(c2cn(CCC=C)nn2)=O)CCC2(CC1)CC(C)N(C(=O)CO)C2 Cc1cccnc1C(=O)NCCC(C(C)C)NC(c1ncnn1C)=O CC1CC(C)N(C(c2cnc(O)n(C)c2=O)=O)CCN1C(c1c[nH]c(=N)o1)=O C(CC(C)C)(CS(=O)(=O)N1CCOCC1CC1CCCO1)OC CCCCCCCN(C)C(C1(CNC(=O)CC2CC3(CC3)CO2)CC2(CC2)C1)=O c1(OC)ccc(C(N2CC(N(C(=O)CCC3CCCO3)C)C2)=O)c(F)c1 N1(C(CC(C)C)=O)CCCC(NC(c2cccc3ccsc23)=O)CCC1 c1(C(N2CCOC(c3nc(C(=O)OC)cs3)C2)C(=O)NCC)cccc(CC)c1 c1(C(N2CCC(N(C(C(CCCCC)O)=O)C)C2)=O)cnc2ccccc2c1 N1(C(C2CC23CCC3)=O)CC(CO)C2(C1)CN(C(c1ccccc1CCBr)=O)C2 C1(CC)CCN(C(c2ccc(Cl)s2)=O)C(C(=O)NCCOCCN=[N+]=[N-])C1 Cc1cnn(CC(=O)NCC2CN(C(c3cnc(C(F)(F)F)s3)=O)C2)c1 c1(C(N2C(CN(C(=O)Cc3ccoc3)C)CCC2)=O)cnccc1Br C1(CCC(=O)NCC2(C)C(C)(C)C2)CCCCN(C(=O)Cc2cccs2)C1 N1(C(C=NOC)=O)CCC(C)(C)C(NC(=O)C(C)Oc2ccc(Br)cc2)C1 N1(C(C2(COC)CC2)=O)CCC(C2CCCN(C(=O)Cc3sccc3C)C2)C1 C1(CNC(C(F)=C(C)C)=O)CCN(C(=O)CCn2ccc(C)n2)CC1CO c1(CC(=O)NCC2(F)CCCN(C(c3c(C)c[nH]c3)=O)C2)ccc2ncsc2c1 n1(CC(=O)NCC(N(C(=O)CC2CC2)C)C2CC2)ncnn1 CN1N=C(CC(=O)N2CCCC(NC(C3(n4nccn4)CC3)=O)C(F)C2)CC1=O C1(CC(=O)NC(C(=O)OC)C2CCC2)CN(C(=O)CC2CCCN2C)CCO1 c1(OC)ccc(CN=C(NCC2(C)COC(=O)N2)NC2CC(C)(CC)C2)cc1 N1(C(=O)NC2CC3CC(Cc4ccccc4)C2C3)CCC2(CCCNC2=O)CC1 C(CN=C(NCc1ccc(C)n1C)NC1CCCC(F)(F)C1)SC Cc1nn(-c2ccccc2)cc1CNC1CCOC1C c1(C(N2CCC3(C(NC(C4CC(=C)C4)=O)C3)CC2)=O)ccc(N)c2ccncc12 c1(C(=O)NC2C(C)CCN(C(=O)C(C)(C)C)C2)cc(F)cc2c1C(=O)CC2 N1(C(C2CCC(CC)O2)=O)CCC(C2CCN(C(=O)CC(C)(C)O)CC2)C1 CCC(CC)C(F)C(=O)NCC1CC(COC)CN1C(=O)Cc1cccnc1O C(CC1=CCN(C(C2CN(C)CC2C)=O)CC1)NC(C(C)(C)OC)=O CC1C(NC(c2cn(CC(F)F)cn2)=O)CCN1C(C1CCOCC1)=O N1(C(C(CC)(F)F)=O)CCC2(CC1)CN(C(C1CCCC(C(C)(C)C)CC1)=O)C2 c1(C(N(C(CC(=O)N(CC#C)CCF)CC)C2CC2)=O)c[nH]c2cnccc12 S(=O)(=O)(c1ccc(N2CCN(C)CCC(C)C2)c(Br)c1)NC1CCC(CC)CC1 C1(O)(CC(N2CC=CC2CNC(=O)C(N2CCCC2)C2CCCC2)=O)CCCC1 Nc1c(C(N2CCC(CNC(C3(C(N)=O)CC3)=O)C2)=O)sc2ccccc12 C1(C(N(CC(CC)NC(=O)Cc2c(C)cnn2C)C)=O)CC(C)CC(=O)N1 C1(N(C(=O)COc2ccn(C)n2)C)CCCCC1NC(c1nc(C2CC2)cs1)=O c1(C(=O)NC(C(=O)NC2CC(OC)C2)Cc2ccccc2)cc(F)ccc1O N1(C(C(=O)NCC2C(C)CCS2)=O)CCn2ncnc2C1 c1(C(=O)NC(C2CN(C(=O)CN3CCCC3=O)C2)C)cc(-c2ccccc2)cs1 O=C1CCC(CNC(=O)CCNC(=O)CN(C2CCCC2)C)CN1 c1(CC)cccc(C(N2CCCC2COc2ncccc2Cl)=O)n1 C1(NC(=O)CCSC(F)(F)F)CC12CC(NC(c1c[nH]nc1F)=O)C2 N1(C(c2ccn(C)n2)=O)CC2C3CCC(C2C1)N(C(c1ccc(S)cc1)=O)C3 C1(C(=O)NCC2C(CNC(C(OCC)OCC)=O)C2)(CF)CC(F)(F)C1 [N-]=[N+]=Nc1cc(NC(N2CCS(=O)(=O)C(CO)C2)=O)ccn1 N1(C(COCCOCC)=O)CCN(C(=O)C(c2cnn(C)c2)C)C(CC)C1 C1(CC(=O)NC(C)CNC(=O)Cc2nc(=N)[nH][nH]2)CCCCC1F c1(C(CNC(=O)CC#N)N(C)C(C2(CF)CCC2)=O)ccc2ccccc2c1 C(=O)(CCCS(C)(=O)=O)NCC(C)(CNC(C1CCCCS1)=O)OC O=C1CCc2nc(N3CC4CCC3C(NC(C3CCCC5(CC5)C3)=O)C4)ccc21 C(C(C)C(=O)NCC1CCC(=O)O1)N(C(C1CC(C(=O)OC)C1)=O)C C=CCCC(CC(C)C)C(=O)NC1(CCNC(C2CCN(CC(C)C)C2)=O)CC1 C12(C(=O)NCCCOC(N(C)C)=O)CCCC1NCC2 C(=O)(C1CNC(=O)c2ccnn21)N1CCC(CNC(=O)Cc2ccsn2)CC1 Cc1ncc(Cl)cc1C(=O)NCC(F)CNC(c1cnn(-c2ccncc2)c1)=O N1(CCNC(C(n2ccc(C)n2)C)=O)CCN(C(C2(n3cncn3)CC2)=O)CC1 c1(C(=O)NC(C2(O)CN(C(C3CCCC(C)C3)=O)C2)C)cnc2c(c1)CCCO2 C1(C#N)(C(=O)NCc2ccc(C)cc2)CC12CCCC2 c1(OC)cccc(SCC(N2CCOCC2CN(C)C(C2CCCOC2)=O)=O)c1 c1(C(=O)NC2(COC)CCN(C(=O)CCOC(C)C)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NC2(C)CCN(C(CC=CC=C)=O)C2)cc2c(Br)cccn2n1 c1(CSc2cccc(Cl)c2)cccc(I)c1.n12cc(nn1)CN(C)C(=O)C2 c1(OC(C(=O)N(CCN(C(C=CC(CC)=CC)=O)C)C)C)ccc(Cl)c(C)c1 CCC(CC)(CCOC)C(=O)N1CCC1CNC(c1ncc2[nH]ncc2n1)=O N1(C(=O)Cc2ccoc2)CC(NC(C2(C(F)(F)F)CCCC2)=O)C2CCCCC12 CC1=C(C(=O)NC2CC2NC(C2(CC3CC3)CCCC2)=O)C(C)(C)CCC1 C1(CC(N2CCC(N(C(=O)Cc3nnc(C)o3)CC)C2)=O)OCCOC1(C)C CCCC(C)CC(=O)N1CC2CC2C1CNC(=O)Cc1ccccc1OCC c1(C(=O)NC(CCCC)CNC(=O)C#CC2CC2)cnc(OCC(F)F)c(Cl)c1 c1(NC(C2N(C(c3n(C)ncc3Br)=O)CC(F)C2)=O)nc(Br)cn2ccnc12 N1(C(c2c(C)[nH]cc2)=O)CCc2ccccc2C(NC(=O)C2=CC3CCC2C3)C1 Nc1[nH]c(=NCCn2ccnc2-c2ccccc2)[nH]c2ncnc1-2 C1(CNC(NC(CC)CC)=NCC2CCC3(CCC3)OC2)CC2(CO1)CC(F)(F)C2 C1(CNC(C2CC(SC)C2)=O)CC2CCCCC2N1C(C1CNC(=O)C1)=O C(CN=c1nc(C)c([N+](=O)[O-])c[nH]1)NC(C1(C)C(CC)CCC1)=O c1(C(N2CCCCC(CO)C2)=O)cn2ccccc2n1 c1(C(c2n(CC)nnn2)NCCc2cc(C)no2)cncc(C(F)(F)F)c1 c1(OC)cc(C(=O)NCC(CO)NC(C2(C)CCCNC2=O)=O)cc(Cl)c1 CN1CCN(C(c2cccnc2N)=O)CC1CNC(=O)C#CC1(C)CC1 CCCC(C)(C)C(=O)N1CCCCC(CNC(=O)CC2CCCN2C)C1 c1(OC)nc(N2CCOC(CNC(c3sccc3CC(C)(C)O)=O)C2)cc(C)n1 CCCC(CCCO)C(=O)N1CCC2(NC(C3CCC(C)O3)=O)CCCC12 n1(CC(=O)N(CC(C)C)CC(=O)N(C)CCN(C)C)ncnn1 c1(NC(C2CN(C(c3cc(Br)ccc3F)=O)CCS2)=O)c[nH]c2ncc(Br)cc12 c1(NC(CN(C2CCCN(C(=O)C(C)(C)C)C2)C)=O)ccc(N(C)S(N)(=O)=O)cc1 N1(C(c2cnc(Cl)s2)=O)CC2CC(C1)N2C(c1cnn2ccsc12)=O c1(C(=O)NCCC2CCC(NC(C(CSC)(C)C)=O)C2)n[nH]c2c(C)cccc12 C1(C(=O)OC(C)(C)C)CC(C)(C)CCN1C(C1CC(S(N)(=O)=O)C1)=O N1(C(C2CN(C)C(=O)N2)=O)CCC2(CCN(C(C3CC(Cl)(Cl)C3)=O)C2)C1 C1(C(=O)NC2C(NC(CSCC#C)=O)CCC2)CCCCN(C)C1=O CN1CCC(C)(C(N2CC(CCCCNC(=O)C(F)CC3CC3)C2)=O)C1=O N1(C(C2CC(C)(NC(C3CC4C=CC3O4)=O)C2)=O)CCCN2CCCC2C1 C(CCC1CCC1)(C(=O)NCCCSC)N(c1cccc(C)n1)C(C#C)C Cc1ccc(S(=O)(=O)N(c2ccc(O)cc2)C(C2CCCC2)=O)cc1C Cc1[nH]c(C#N)cc1C(=O)NC(C)CCC(=O)NCCCc1cc[nH]n1 CCC(C)CC(=O)NC1CC(C)CN1CC(=O)Nc1nnc(-c2ccccc2)o1 N1(C(C=CC(CC)C)=O)CCCC(O)(CNC(c2ccsc2)=O)CC1 c1(C(N2CCC(F)(CNC(c3c(C)cco3)=O)CC2)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(CCS(=O)(=O)c1ccccc1)NC1(CNC(C2(C)CC(C#N)C2)=O)CCC1 C=C(C)C1OCCCC1C(=O)NCC1CN(C(c2cnsc2C)=O)CCC1(C)C Cc1oncc1C(=O)NCC(=O)NC1CC1CNC(C1CCNC1=O)=O c1(C(=O)NCCCCCN(C(c2c(C)coc2C)=O)C)ccn2cnnc2c1 C1(CC(=O)NCCOC)CCCN1C(c1ccsc1Cl)=O c1(C(N2CCC(N(C)C)(CC)C2)C(=O)NC(CC)C)cc(Cl)ncc1Cl c1(CN(C(=O)CCn2cc(-c3ccsc3)nn2)C)cccnc1Cl Cc1cc(Br)cc2cc(C(N3CCCC3CNC(C3(N(C)C)CC3)=O)=O)oc12 CCN=c1[nH]cc(C(=O)N(C)CC2CCN(C(C3CC3F)=O)C2)s1 Cc1coc(C)c1C(N1CCN(CCCNC(c2ccc(C(F)F)o2)=O)CC1)=O C(C(C)(O)CNC(c1csnc1C(F)F)=O)NC(C(c1ccccc1)C)=O CCC(F)(F)CC(=O)NCCCNC(C1COCC1C(F)(F)F)=O C1(CNC(=NCC)NCCN2CCOCC2)CCC2(CCC2)C1O N1(CCc2cn(CC(N3CCC(c4nc[nH]n4)C3)=O)nn2)CCC(F)(F)CC1 Cc1cc(Cl)c(C(N2CC(NC(c3coc(C(F)F)n3)=O)CC2C)=O)cn1 c1(OC)ccc(C=CC(=O)NC2CN(C(=O)C(C)CC3CCC3)CC2O)cc1F c1(C(N(C)CC2CCN(C(C3(C)C(C(=O)OC)C3)=O)C2)=O)scc2c1CCCC2 C1(CNC(c2n[nH]c(C)c2O)=O)CC2(C1)CN(C(=O)CCCc1ccccn1)C2 c1(CNC(=O)CONC(=O)c2ccsc2)nccc2[nH]ccc12 OCCC(N=c1nc2scnc2c(N2CC3CCC3C2)[nH]1)c1cccnc1 c1(OC)ccc(CN2CC3C(C(N4CC(C)CCC4C)=O)C3C2)c(Cl)n1 Cc1nnccc1C(=O)NCC(C(=O)NC1COC(C)(C)C1)N(C)C C1(NC(c2ccc(F)c(F)c2)=O)CC2CC1CN(C(=O)C(F)(F)CO)C2 C#CCC(CC(=O)N1CCCCC1CCCO)NC(=O)CCc1ccsc1 N1(C(c2c(C)ocn2)=O)CC2CCC2(NC(=O)Cc2ccc(OCC#N)cc2)C1 CC1NC(=O)CCC1CNC(=O)C(N1CCC(Cc2nccs2)C1)=O c1(C(=O)NCC(CN(C(C(CC)C#N)=O)C)C)ncn2cc(Br)sc12 c1(C(N2CCC(C)(NC(C(C)CSC(F)(F)F)=O)C2)=O)cccc2c1ccn2C N1(C(c2c(CC)cno2)=O)CCC2(CCN(C(C3CCCC(O)C3)=O)CC2)C1 C1(C(=O)NC(C)C(C)NC(=O)Cc2csc(CCn3cncn3)n2)CC=CCO1 C(CCCCCNC(=O)C=CCCC(C)C)NC(Cc1c(C)ocn1)=O CC1COCC(C(=O)NCCn2cc(CNC(=O)CCN(C)C)nn2)O1 c1(N(CCNC(=O)C2CC2)CC)cc(Cl)nc(C(C)(C)C)n1 c1(C(CC(=O)NC2(C)CN(C(Cc3ccc(C)s3)=O)C2)C)c(C)noc1C Cc1n[nH]c2cc(C(=O)NCC3CN(C(C4CCCCO4)=O)CCN3C)ncc12 N1(C(c2c(C(C)(C)C)cccc2)=O)CCC(NC(C2CC3CCC2O3)=O)C12CC2 c1(C(=O)NC(CCOC)CNC(C23CC(C#N)(C2)C3)=O)ccc(F)c(O)c1 C1(N(C)C(=O)OC(C)(C)C)CC2CC1N(NC(C1CCC(C(F)F)CC1)=O)C2 N1(C(C(=O)NC2(C)CCCO2)=O)CCn2ncc(S(C)(=O)=O)c2C1 C1(CCC2N(C(=O)OCC)CCC2)CCCCC1CC c1(OC)ccc(-c2nc(CCNC(=O)C(N3CCCCCC3)=O)cs2)cc1 C1(CNC(CCc2ncc(C)[nH]2)=O)CN(C(c2cnc(CC3CC3)s2)=O)CC12CC2 C1(CC(N2CCCC(OCC#C)C2)=O)CC(C)(C)CN1C(=O)CCc1cnco1 N1(C(c2cccc(-n3cccn3)n2)=O)CC2CCC1CN2CCn1ccnn1 CC1OC2(C(=O)NCC3CC(NC(=O)Cc4csc(NC=O)n4)CCO3)CC1C2 C(=O)(C(C(C)C)C(C)C)N1CCC(C(C)NC(CCc2cc(C)nn2C)=O)CC1 N1(C(c2c(OC)scc2)=O)CCCC(NC(=O)CCC(=O)NC2CCCC2)C1C c1(C(N2CCC(N(C(=O)Cc3nc[nH]n3)CC)C2)=O)ccc(S(=O)(=O)CC#N)cc1 c1(C(=O)OCC)cc(Br)c(C)cc1NC(C1CC(=O)N(CCOC)C1)=O C1(CC(=O)NC)CN(C(C2CCC(F)C2)=O)CCN1C(=O)CCS(C)(=O)=O C1(CNC(C(C)OCC)=O)CCCC2(CN(C(=O)CCc3cncs3)C2)O1 C1(CNC(=O)C(O)C(F)F)CN(C(=O)C=C(Cl)Cl)CCC12CCOCC2 C1(CC)CN(CC)CC1C.C1CC(=O)NC(C2CC2)C(=O)N1CC C=C1CC(C(=O)NCc2cscn2)(CNC(c2cnn(C(C)C)c2)=O)C1 c1(CC(=O)NCC(CN(C(=O)C2=C(C)CCC2)CC)(C)C)cnn2c1CCCC2 S(=O)(=O)(c1cc(C(=O)NCC2CCN2C(C2(C)CC=CC2)=O)ccc1OC)NC Cc1cnc2c(C(N3CCN(C(C4CC=CCO4)=O)CC3CF)=O)cnn2c1 Cc1nc2cc(C(=O)NCC(C3CCC(F)(F)CC3)C)cnc2[nH]1 CC1(C)C2CCC1(C(=O)O)C(NC(c1c[nH]nc1Cl)=O)C2 CC1CCOC(C(=O)NCC=CC(=O)N(C2CC2)Cc2nc[nH]n2)C1 C1(NC(c2c(C)nns2)=O)CC12CCN(C(=O)CC(=O)N(C)C)C2 CC(C(=O)NC(C)CC1CN(C(c2cccc(CF)c2)=O)C1)C(C)O c1(C(=O)OCCC(N2CCC(CCOCC)C2)=O)ccc(F)cc1 Cc1ncccc1CC(=O)NCCCC1CCCN1C(=O)C(C)C1(O)CCC1 C1(NC(C=CC=CC)=O)CN(C(c2ccc(Br)c(F)c2)=O)C2(CCOC2)C1 C=CC1(CC(=O)NCC(C)(CC)OC)CN(C(=O)C=CC2CCOC2)C1 O=C(C1=NOC2(CCN(c3ncncc3I)C2)C1)Nc1cc(Br)c(F)cc1[N+](=O)[O-] n1(CC)nnc(C)c1CNC(=O)C(C)(C1CC1)N(C(=O)CC1CC1(C)C)C Cc1noc(C)c1S(=O)(=O)N1CCCC1.C1(N)CC2CN(C(=O)CCCF)CC2C1 C(=O)(C#CC1(CC)COC1)N1CCC(NC(c2c(Cl)cn(CCC)n2)=O)C1 c1(C(N2CC(NC(C=CC(=O)OCC)=O)C3C(C2)C3)=O)csc(S(N)(=O)=O)c1 Cc1cccc2c1OC(C(=O)NCC(O)CNC(C1CCC(N=[N+]=[N-])C1)=O)C2 Fc1ccc(-n2ccnc2-c2cc(Br)cc(Cl)c2)cc1-c1ccc(F)cc1F N1(C(=O)CN2CCC2)CC2(C1)CN(C(c1cc(O)ccc1[N+](=O)[O-])=O)CC2CO Cc1ccc(CCC(=O)NC2CC2CNC(C2(F)CC2)=O)o1 C1(CN(c2ccccc2F)C(=O)C(C2CCOCC2)F)COC2(CCNCC2)C1 c1(COC)cccc(CC(=O)N(CCCNC(C2CC2C(C)(C)C)=O)C)c1 N1(C(c2c(OCC)ccc(C)n2)=O)CCC2CC2(NC(=O)Cn2cccn2)CC1 C1(CNC(c2cnc(OC)s2)=O)CCN(C(C2(C)CNC(=O)N2)=O)CC1O C1(CC)(NC(=O)C(C)S(N)(=O)=O)CCN(C(=O)CCc2nc(C)cs2)CC1 c1(OC)ccc(CCC(N2CCOC(C(C)NC(=O)COCCCF)C2)=O)cc1 c1(C(=O)NCCC(C(=O)N(CC(O)CO)C)OC)ccc(O)c(F)c1 C(C(C)C)(C(C(=O)Nc1cccc(Cl)c1C)N1CCCC1C(C)(C)OC)OC c1(-c2scc(C(C)NC(=O)NC3CCC(C4CCNCC4)N3)n2)ccc(Cl)cc1 CCCCC(C(=O)N1CCC1C(C)O)NC(c1cccc(F)c1O)=O C(=O)(C(C)(O)CCC)NC1CN(C(C(C(=O)OCC)F)=O)C(CO)C1 C(CC(=O)N1CCSCC1C1CC1)(C(F)F)NC(=O)COC1CCC1 C(C1CCOCC1)=CC(=O)NCCC(F)(F)Cn1cc(C(C2CC2)C2CC2)nn1 c1(C(CNC(NC(c2ccc(Cl)cc2)CF)=NCC2CCC2)F)cccc(F)c1 CN1CCN(C(=O)CCc2cscn2)C(C(=O)NC2CN3CCCC2C3)C1 C(=O)(C(O)C(C)CC)NCCCN(C(c1c(OCC#C)nccc1)=O)CCO Cn1cncc1C(=O)C(=O)NCCCCCNC(=O)CC1(C2CC2)CC1 c1(OC)cncc(C=CC(=O)NC2CC2(C)C(C)C)c1 CC1(CNC(C2SC3C=CC2CC3)=O)CCN(C(C2CCOCC2)=O)CC1 Nc1c(F)ccc(Cl)c1C(=O)NC1CCN(C(=O)Cn2cnnc2O)CC1 CCCC(C(=O)NCC1CCCN1C(=O)C(c1ccc(F)cc1)F)NC(N)=O c1(COC)cccnc1C(N1CCCC1CN(C)C(c1cn(C2CC2)nn1)=O)=O C1(NC(c2c(COC)cc[nH]2)=O)CN(C(c2cc(C)c(C)nn2)=O)C(C)(C)C1 N1(C(c2c(C)cccc2Br)=O)CCN(C(C2CC(C)C2)=O)C2(CCC2)C1 C1(CC=C)(NC(=O)Cc2cc(C)no2)CCN(C(C2CNC(=O)N2C)=O)CC1 c1(C(N(C2CCN(C(CCCCSC)=O)CC2)CCO)=O)cc(C#N)c(O)nc1N CC1CC(NC(c2cnncc2O)=O)CN1C(=O)CC1CCC2CC12 c1(C(=O)O)cc2ncc(CN3CC4CC4C3CO)cc2[nH]1 C1(NC(Cc2n(C)ccc2)=O)CCC2(CCN(C(C3(C)C=CCCC3)=O)C2)C1 c1(OC)nc(Br)ccc1S(=O)(=O)NC1CCCc2c1cnn2C(C)(C)C c1(-c2ccc(CNCc3c(OC)csc3)cn2)ccc(Br)c(C)c1 C=CC1(CC(=O)NC2CCCN(C(=O)CCC=CC)C2C)CCOCC1 C(=O)(C(CCC(N)=O)N(C)C)NCCC(C)CCNC(C1CC1c1cccs1)=O C(=O)(C(C)CC(N)=O)N1CC(c2oc(C)c(NC(C3CCC(N(C)C)C3)=O)n2)C1 c1(C(N2CC(CNC(C(CC(C)C)O)=O)OCC2)=O)cc(O)nc2ncn(C)c12 c1(-c2cccc(OC)c2C)cccc2c(C(=O)NCc3noc(CO)n3)n[nH]c12 C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C(CN(CC(C)(C)C)C)=O)C(CO)C1 C#Cc1cccc(CC(N2CCOC(C3CC3)C2)=O)c1.C1(CC(C)C)C(=O)N1C c1(OC)cc(CN2CCOCC2C(C)N=c2ccnc[nH]2)c(OC)cc1C c1(C(C)C)ccc(C(=O)N(C)CC2CN(C(C3COC(=O)C3)=O)CCO2)c(F)c1 c1(C(=O)NC2C(C(N3CCC(C(=O)NC)C3)=O)CC2)cccc2c1CCC2 N1(C(Cc2n(C)nnc2)=O)CCC(C)(C)CC1C(N1CC(CC(N)=O)C1)=O CC(C)(O)C(F)C(=O)NCC1(F)CC(NC(C2CC3CCC(C2)O3)=O)C1 C(=O)(C(C#N)C1CC1)NC(C1CCCN1C(=O)CSS(C)(=O)=O)C C#Cc1cc(C(=O)NC2(C)CCN(C(=O)COCc3nc[nH]n3)CC2)cc(F)c1 C1(C(=O)NCCc2ccc(CC)cc2)CCCCN(C(C2CCCN(C)C2)=O)C1 N1(C(C(CCOC)(C)C)=O)CCC2(CC1)COC(CNC(=O)C(F)(F)CSC)C2 Cc1nc(C2CC2)sc1CC(=O)NCCCC(C)(C)NC(C1CC2(CSC2)C1)=O c1(C(N2CC(CCCNC(C=CC)=O)OCC2)=O)ccc2oc(C)nc2c1 c1(NC(C2CC2C(=O)Nc2ccnn2-c2ccccc2)=O)ncccc1OC(F)F C1(CCNC(CCCOCCC)=O)CCCN(C(=O)CCC2CC(F)(F)C2)CC1 C1(NC(c2c(C)snc2)=O)CCC2(CC1)CN(C(c1ccc(CF)cc1)=O)C2 N1(C(c2cccc(OC)c2)C(=O)NC(CC)C)CC(C)(C)OCC1CC(=O)OC CC(O)(CC(=O)N1CCC(NC(=O)CCn2ccnc2)CC(O)C1)C(F)(F)F Cn1nc(CC(N2CCCC2C2(C(=O)NC3C(O)CC3O)CC2)=O)cc1Cl C1(C(C)NC(c2cc(CN(CCC)C)on2)=O)CN(C(=O)C=C(C)C)CCO1 C1(O)(CNC(c2c(CCCC)ocn2)=O)CCN(C(=O)C=CC2(C)COC2)CC1 C(C(C)(C(=O)NC1C=CCN(C(C2C=CCS2)=O)C1)OC)OC C(CN=c1[nH]cncc1I)(CC(C)C)NC(c1c2ccc(OC)cn2nc1)=O c1(C(=O)NC(C)(C)C(N2CC3(CCNC3=O)C2)=O)cc2ccccn2c1 c1(OCC)oc(C)nc1C(=O)NC1CCCC1NC(c1ccon1)=O c1(OC)cc(C)c(C(c2nnnn2CCC2(C)CC2)Nc2cn[nH]c2)cn1 N1(C(CC(COC)C)=O)CC2(C(=O)NCc3nc(CO)n[nH]3)CC1CCO2 C(=O)(C1CCOc2ccccc21)NCC1(C)CC(NC(c2cc(C)c(C)s2)=O)C1 c1(OC)cncnc1C(=O)NCCC(=O)NCc1cn[nH]c1 C(=O)(CC(C)(C1CCC1)N(C)C)NC(C)CC(C)NC(=O)C(N1CCOCC1)C Cc1ccc2c(NC(C3CC3NC(c3cc(C)c(Br)cc3C)=O)=O)cccc2n1 N(C1c2ccccc2CCC1C)C(=O)Nc1c(C)n(C(C)C(C)(C)O)nc1 C1(C)(NC(C=C2CCC(C)C2)=O)CCCN(C(=O)C2=COCCC2)C1 Cn1nc2ccccc2c1-c1nc(C2CCC(O)C2)n(C2CC2)n1 CCC(C)(C)C(C(=O)NC1CC(CCNC(c2ccc(F)c(C)c2N)=O)C1)OC C(CC(=O)NCCC(=O)NCCC1(C(=O)NC)CC1)SCC#C c1(CN2C(C(N(C)CCO)=O)CSCC2)cc(Cl)cnc1Br C1(C)(CNC(=O)NC(C(C)c2ccccc2)C#N)CC=CCO1 CCC(CC(=O)N1CC(C)(C)CC1CNC(C1(C)CC1)=O)C(C)(C)C C1(C(=O)OC)CCC(C)(C)N(C(=O)CCc2cn(C(C)CO)nn2)C1 O=C(C1=CCCN(C(C2CC3CC(=O)C2O3)=O)C1)NCCN1CC2CC2C1 N1(C(CC(CCC)C)=O)CC(NC(=O)Cc2c(Cl)c(CC)nn2C)CC2(CC2)C1 Cc1ncc(C(=O)NCC(C(C)(C)C)NC(=O)CN2CC3CC3C2)n1C c1(CNC(=O)C(=O)NCc2ncco2)ccc(C2CCOCC2)cc1 CN1CCC(CN(C(=O)C(CC2CCOCC2)NC(=O)CCC2CCOC2)C)C1 c1(CNC(CC(COC)NC(=O)Cc2cnnn2C)=O)ccc(F)nc1F C(=O)(C1=NN(c2ccc(C)cc2C)C(=O)C1)N(C(=O)CNC)CCC c1(C(c2nnnn2C)NCc2occ(C)c2)cccc(C(C)C)c1 N1(CCC)CCN(C(=O)CCC2CCCN(C(C3CCCS3)=O)C2)CC1 c1(C(=O)NC(CN(C(C(C)=CC)=O)CC)C)c[nH]c2cc([N+](=O)[O-])ccc12 c12ccc3c(c1)CN(C3)C2=O.C1(N(C(C)(C)C)C)CCN(Cc2cccnc2)C1 C(=O)(C(CC(C)(C)C)NC(=O)CCCNC(C)=O)N1C(C(=O)OC)C=CCC1 c1(CN(C(C)C)C)cn(C(C)C(=O)NC2CC(CCO)C2)nn1 c1(N2CCC(C(N(CC=C)OC)=O)CC2)ncnc2c1ncn2CCS N1(C(c2ccc(CC(C)C)nc2)=O)CC(N(C(=O)C=CBr)CCO)C(C)(C)C1 C1(N(C(C(C=C)O)=O)C)CCN(C(c2cc(Cl)cc(Cl)c2F)=O)CC12CC2 N1(C(c2cnc(O)c(F)c2)=O)CC(NC(C2CC(F)C2)=O)CC2(CC2)C1 C(=O)(CS(=O)CCC(F)(F)F)NC1(C2CCN(C(c3ccn(CC)n3)=O)C2)CC1 N1(C(c2c(CC)onc2C)=O)C(CNC(C2CC2(F)F)=O)CC2COCC12 N1(C(c2c(C)ccs2)=O)CC(=O)CC1C(=O)NCC1CCCOCC1 C#CCCCCCC(=O)N1CCCCC1C(C)NC(c1c(C)ncn(C)c1=O)=O C(=O)(C(F)(F)C(O)C(C)C)N1CCC(NC(c2[nH]cc(S(=O)(=O)NC)c2)=O)C1 Cc1c[nH]nc1C(N1CCC1CC(=O)NCC1(N(C)C)CCSC1)=O CCC(CC1CCCC1)C(=O)NCCCOCCCNC(C1CNC(=O)N1C)=O c1(NC(C2N(C(c3n(CC)ccc3)=O)CCC2(C)C)=O)ccc2occc2c1 c1(OCC)cccc(C(C)(C)C(=O)N2CCC(N(C)Cc3ncc(CC)o3)C2)c1 c1(C(=O)OC)ccc(C(=O)OC)c(NCCN2CCOC3(CCSC3)C2)c1Cl CC1(O)CCC(CC(N2CCC(CF)(NC(c3cc4n(n3)CCO4)=O)C2)=O)CC1 c1(C(=O)NC(C2CCN(c3nnc(C(F)F)s3)C2)C)cnc2c(c1)CCCO2 C1(NC2(c3cc(F)cc(F)c3)C(=C)CC2)CC1C1CCN(C(=O)OC(C)(C)C)CC1 N1(C(CCc2c(C)noc2)=O)CCCCC(C(=O)NCCCCN=[N+]=[N-])C1 Cn1nccc1C(C)(C)C(=O)NCCSCc1cn(CC2CCCO2)nn1 N1(C(C2(CC=C)CC2)=O)CCCCC(C(N2CCCC(OCC)C2)=O)C1 C(=O)(C1=COCCC1)NCC(CC(=O)NC1(C)CC(O)C1)OC C(=O)(C(CO)C(C)(C)C)NCCCNC(CC(c1cccs1)NC(C)=O)=O N1(C(c2cc(C)c(Cl)cc2)=O)CCCC2CN(C(=O)C#CC3CC3)CC12 c1(C(=O)O)ccc(CN2CC(C(=O)O)CCC2CO)c(Cl)c1 C1(CNC(=NCC(C)C2CCOCC2)NCCF)CCCOC1(C)C N1(C(CCOC)=O)C(C(=O)NCCn2cc(CO)nn2)CC1C c1(C(N(CCCNC(C2C3CCCC23)=O)C)=O)cccc(S(=O)(=O)C2CC2)c1 c1(C(N2CCC(CN(C(C(CCOC)C)=O)C)C2)=O)ncc2ccccc2c1O CC1(C(N2CCC2CNC(=O)C2=CCCSC2)=O)COC(=O)OC1 N1(C(CCCOCC)=O)CCOC2(CCCN(C(=O)C3=C(CC)OCCS3)C2)C1 C=C1CCN2C(C1)c1nnc2n1CC(N1CCN(C)CC1)CC.C(C)(=O)OC C#CCC(C)(C(=O)N(C)CC1CCCN1CC)NC(C1CCC(=O)N1)=O C1(CNC(C2CC(=O)N(O)C2)=O)CN(C(=O)CCN2CCCC2)CC1(F)F C1(C)(C(N2CCCC(N(C(CCOCCOC)=O)C)C2)=O)CCCCC1(F)F c1(CC(N2C(CNC(=O)CCC3CCOC3)C=CC2)=O)ccc2c[nH]nc2c1 C1(C(c2cn(CCN3CCSCC3)nn2)C(=O)Nc2cccnc2)CCCCO1 N1(C(c2c(C)snn2)=O)CCOC2(CCN(C(C3(C)CCC(F)(F)C3)=O)CC2)C1 N1(CCCCCC#C)CCCc2occc2C1 Cc1ccc(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C2)c([N+](=O)[O-])c1 c1(OC(C2N(C)C(NC(=O)OC(C)(C)C)CC2)=O)cc2oc(O)nc2cc1F C(N=c1[nH]c2c(c(=NC3COC4(CCC4)C3)[nH]1)CSC2)C1(C(C)C)CCOCC1 N1(C(C2C(NCc3ccc(OC)c(I)c3)C2)=O)CC2OCCOC2C1 c1(C(C)=O)cnc2n1CCN(C(c1ccn(C3CC3)c1C)=O)C2 N1(C(CN(C(=O)OCC)C)=O)CCC2(CC2NC(c2cccnc2CC)=O)C1 c1(C(N2CCCCC(N(C(C(CC)C)=O)C)C2)=O)ncc([N+](=O)[O-])n1C Cc1cc(C(N2CC(O)(C3CCCCN3)C2)=O)c(N)s1 c1(CN2CC(NC(c3cnc(C)[nH]3)=O)C(F)C2)cc(Cl)c(C)cc1O N1(C(C#CC2(C)COC2)=O)CCC2(CNC(=O)COC3CCCC3)CCCCC12 c1(C(N(CCNC(=O)C(C)(O)CC(C)C)CC)=O)nccc2ncccc12 N1(C(c2ccc(CC)[nH]2)=O)CCC(O)(C(C)NC(=O)Cn2ccnn2)C1 c1(CC(C)C(=O)NCC(F)CNC(=O)C2=CCSC2)ccccc1Br c1(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CC2)cc(O)c(O)c(O)c1 c1(C(=O)NCC(CC)N(C(c2c(CC)nns2)=O)C)ccc2nc(O)cn2c1 C1(CNC(C2(CCCC)CCCC2)=O)CCN(C(=O)Cn2cnnc2)C12CC2 Cc1coc(C)c1C=CC(=O)NC1CC1NC(=O)Cn1cnc([N+](=O)[O-])c1 C1(CC(=O)OC)CCC2(CCN(C(=O)CC3(CC4CC4c4ccccc4)CC3)C2)C1 N1(C(Cn2c(C)cc(C(F)F)n2)=O)CCCC2(C1)CN(c1nnnn1C)CCO2 Cc1coc(C(N2CCCC2CCNC(=O)CCc2c(C)noc2Cl)=O)c1C c1(C(N2C(CNC(CC(C)C)=O)COC(C)(C)C2)=O)cc2cc(F)c(F)cc2[nH]1 N1(C(c2cnn(CC)c2Cl)=O)CC(NC(=O)COCC(C)C)C2(CCC2)C1 C(=O)CS(=O)(=O)CC(C)C.N1CCC(C)C1Cc1cn(C2C(OC)COC2)nn1 N1(C(C2CCCC23CC3)=O)CC2CC(C1)N(C(C1CCCCS1)=O)C2 CN=c1nc(C(=O)NC2CC(CNC(=O)C(C)(F)F)C23CCC3)cc(C)[nH]1 N1(C(C(Cc2ccco2)NC(c2c(C)c(O)ccc2)=O)=O)CCC(F)(F)C(O)C1 c1(CCC(=O)O)ccc(CNC2CCCCC2n2ccnc2)nc1 C1(CCNC(C2CCCC2O)=O)CC2CCC(C1)N2C(c1cc(CCO)on1)=O c1(C(=O)NC(CNC(Cn2cc(C(=O)NC)nn2)=O)(C)C)cc(C)c(C)s1 c1(C(N(CCN(C(c2cc(C)sc2)=O)C(C)C)C)=O)[nH]ncc1C#N N1(C(CCN(CC)CC)=O)CC(C(N2CC3CCC3(C)C2)=O)CC(C)C1 N1(C(c2c(C)cnnc2)=O)CC(=O)NCC1C(N1CCCC(CC(N)=O)C1)=O C1(C(=O)NCC(=C)CCNC(c2ccc(SC(F)F)cc2)=O)CCC(C)(C)CC1 C(CC1=CCN(C(C2CCN(C)C(=O)C2)=O)CC1)NC(C1(CC)CCNC1=O)=O N1(C(CN(C)C(N)=O)=O)CCC(F)(CNC(c2ncccc2N(C)C)=O)CC1 c1(C(N2CC(CCNC(c3c(C)nsc3)=O)OCC2)=O)cc(C)c(C#N)c(C)c1 C(C)(CCC(=O)NC1(NS(C)(=O)=O)CC=CC1)NC(CC=CC=C)=O C1(CN(C(c2c(C)onc2)=O)C)CCCN(C(c2cccnc2C(F)F)=O)C1 C1(CN(C(C=CCC)=O)C)CCCN(C(=O)C=Cc2cncn2C)C1 N1(C(c2ccc(Cn3cc(CCC(=O)CCO)nn3)o2)=O)CCC2(CCCOC2)C1 N1(C(c2cccc(C)n2)=O)CCC2(CC1)CCN2C(=O)CSC1CCCCO1 Cc1cnn(C)c1S(=O)(=O)NC(CCC(=O)N(C)C)c1ccccc1 N1(C(C(CC)C)=O)CC2OCCN(Cc3cccc(OC4COCCO4)c3)C2C1 CC1C(C(=O)N2CCC3(CCCN3C(=O)C#CC3(C)CC3)C2)=Cc2ccccc21 N1(C(CC(C=C)CC)=O)CCCC2(CCN(C(=O)CCOC)CC2)C1 CC(=O)CC(C)(C)CC(=O)NCC1CC(NC(c2cnoc2)=O)C1 c1(CCN2CCC(CN3C(CC)CCCC3)CC2)oc2ccc(Cl)cc2c1C N12CC3CC(C1)N3C(=O)C1C(CCCC1)OC2=O.CC(C)(C)C(=O)CNC=O O=C(CC(F)(F)Cl)NCCNC(c1ccc(-c2nc[nH]n2)nc1)=O c1(C(=O)NC(C(N2C(CC)CC(O)C2)=O)C2CCCO2)ncn2c1CCC2 CC(C)(CCC#N)C(=O)NCC1CCC(NC(c2ccc(CF)cc2)=O)C1 c1(C(=O)NC(CC)CN(C)C(c2ncccc2OC)=O)cnc(OC)c(Cl)c1 CON(C)C1CN(C(c2nc(CNC(=O)Cc3ccccn3)oc2C)=O)C1 c1(C(N2CCC(CNC(c3cnoc3-c3ccco3)=O)C2)=O)csc2cncn12 C1(CNC(C=CCC)=O)CCN(C(=O)CCc2cncn2C)C12CC2 C1(NC(c2sccc2C(F)F)=O)CN(C(=O)CN2CCOCC2)C2CCCCC12 c1(C(=O)NCC2C(CNC(c3cn(CCC)nn3)=O)C2)ccc(O)c(C(N)=O)c1 N1(C(C=CC(C)NC(C2(C)CCCC2)=O)=O)CCC2(CCCCO2)C1 CC(C)CC(C)CC(=O)NC1(C(=O)NC2CC3CCCC3C2)CCCC1 Cc1ccc(-c2cn(C(C)C(=O)O)nn2)c(Cl)c1.C1=C(C(=O)O)CONC(=O)C1 C1(COC)CCN(C(C2CC(NC(C3CC=CCC3)=O)C(O)C2)=O)C1(C)C C1(CC(C)C)CC(C(N2CCC23CN(C(=O)C2=COCC2)C3)=O)CC(=O)N1 CCCC(C(=O)NCc1c[nH]nc1C(=O)NC1CNC(=O)C1)OCC C1(CN(C(c2n(CC)ncn2)=O)C)CCN(C(=O)C(N2C(=O)CCC2=O)C)CC1 N1(C(C(CCOC)C)=O)CCCCC2(CCN(C(=O)C(=O)NCC(F)F)C2)C1 C#CCCCCCC(=O)NCCC1CC(C(=O)NCC2CCN(C(N)=O)C2)C1 C1(NC(=O)Cc2ccccc2O)CN(C(c2[nH]ccc2C2CC2)=O)C2(CCC2)C1 n1(CC)nnc(-c2nc(-c3ccc(OC)cn3)nn2-c2cnnn2C)c1C CCCC(CCC)C(=O)NC12CCC(NC(C3(C#N)CCCCC3)=O)(CC1)C2 c1(OC)ccn2cc(C(=O)NCCCN(C(c3csc(C)c3)=O)C(C)C)nc2c1 c1(C(=O)NC2CN(C(c3c(COC)cco3)=O)C2)ccc(C(C)(C)OC)cc1 CC1(C#N)CCCN(C(=O)C(=O)NCc2ccc3c(c2)OCC3)C1 c1(NC(=O)NCc2nccc(OC)n2)cc(C)ccc1Br N1(C(CC2CCCC(C)O2)=O)CC2(CCN(C(=O)CN(S(C)(=O)=O)C)CC2)C1 C(=O)(C(C(C)C)NC(c1ncc(F)cn1)=O)NC(C(=O)OCC)C C=CCC(C)(CC=C)NC(=O)C1=CCC(NC(=O)CC(CC)C2CCC2)C1 CC(C)C(CCN(C(=O)CCc1cn[nH]c1)C)NC(c1cn(C)nc1Cl)=O N1(C(C(CC)OCC2CC2)=O)CCOC(C(=O)NOCC(O)C(C)C)C1 c1(C(N2CCC(NC(C3C(C(=O)OC)C3)=O)C(C)C2)=O)cnn2c1NCCC2 c1(CC(=O)NC(CNC(C(C=C=C)C)=O)C(C)C)ccc(OC)cc1Cl C=CCCCC(=O)N1CCC1(C)CC(N1CCCC1C1CCOC1)=O C1(C(N(CC#CC)CC#C)=O)CCCCCCN1C(=O)C(C)OCC=C N1(C(c2scc(C)c2)=O)CCCCC(C(=O)NCC2OC(=O)CC2(C)C)C1 c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)ccc(N2CCCCCC2)cc1 C(=O)(C(C(=O)N1CC(CNC(C2(C)CCN(C)CC2)=O)(OC)C1)C(C)C)OCC C(CCC(C(=O)N1CCC(c2nc[nH]n2)C1)NC(=O)CCC(F)(F)F)OC c1(N2CCCCC(NC(c3c(C(C)C)nn(C)c3)=O)C2)ccncc1[N+](=O)[O-] c1(C(=O)NCC(CCCC)NC(c2cocc2C)=O)cnc2c(cnn2C)c1 c1(-c2c(C)c[nH]n2)nc(-c2ccsc2)nn1-c1ccn(C)n1 CCCCCC(=O)NCC1CN(C(=O)CCOCCCC)C2CC12 c1(C(N(CC(C)(C)NC(=O)CCc2nccn2C)C)=O)c(F)ccc2c1OCC2 C#CCC(C)(CC)C(=O)NC1CN(C(=O)Cc2nc(C3CC3)nn2C)CC1SC O(NC(=O)C(CNC(C1(C)CCCC1O)=O)CC1CC1)CC(=C)Cl c1(NC(C2CCN(C(C3=NOC(C)C3)=O)C2C2CC2)=O)ccc2ccncc2c1 c1(C(N2CCC(OC3CCCCC3)CC2)C(=O)NCC(=C)C)cc(Cl)sc1C N1(C(C2CCCN(Cc3cn(CC(C)(C)C)nn3)C2)=O)CCCC(B(O)O)C1 CC1=C(C)CN(c2nccc(N(C)Cc3nccn3C(C)C)n2)CC1 c1(C(N2CCC(N(C(COCC(=O)NC)=O)C)C2)=O)cc(OC)cc(Cl)c1 C1(N(C(=O)CCn2cnnn2)C)CCC(NC(c2cnc(S)[nH]2)=O)C1 C(C)(C(=O)N1CC(O)CO1)N(C(C(COC)OC)=O)C1CC1 N1(C(C(COCC)C)=O)CCCC(N(C(=O)C=Cc2ccncc2)C)C1 c1(CNCC2N(C(c3nc(CCCCC)sc3)=O)CCC2)cncc(C)c1 C1(CNC(=O)CSCC(F)F)(NC(C2CC(=C3CC3)C2)=O)CCCCCC1 O=C(C(Cn1cccn1)NC(=O)Cc1ccon1)NC(c1ccncc1)C1CC1 N1(C(=O)NC2CCCC(C(N)=O)C2)CC2CCC1C(O)C2O Cc1nc2ccc3cc(C(=O)NC4CCN(CCC5CCCC5)C4)ccc3n2n1 c1(CC)cc(F)ccc1CC(=O)N(C1CCCN(C(C2(Cl)CC2(C)C)=O)C1)C c1(NC(C2(CC#C)CCCO2)=O)cccn(-c2ccccn2)c1=O Cc1nc(C(=O)NCC(C)(C)NC(c2nc(=N)cc[nH]2)=O)c(C)o1 c1(C(=O)NC2C=CCN(C(=O)Cc3ccccc3CO)C2)cn2cnnc2cn1 CCCCC(C(=O)NC1CCN(C(c2ccc(CC)nc2)=O)C1)ON=C(C)C N(C(=NCc1ccccc1)N(C)CC1CCC1)C1CCC(CC)CC1.S(C)(=O)(=O)N C1(CNC(C2CCN(CCCC)C2)=O)(CNC(=O)C(C)(C)SCC)CC12CCC2 c1(C(N(CCCN(C(C(C(C)C)O)=O)C)C)=O)cc(C(F)(F)F)cnc1N Cn1cc(C(N2CC3CC3(CO)C2)=O)c(CNC(C2(CC3CC3)CCCO2)=O)n1 N#CC1(C(=O)NC2CC(NC(C3CCCCC3)=O)C23CCC3)CC2CCC1CC2 c1(C(=O)NC2N(Cc3c(COC)cccc3)CC(O)C2)ccc(CC#N)c(F)c1 N1(C(C=C(C)C)=O)CC(NC(=O)CCCc2ccsc2)CC(C)C1 c1(C(=O)NC2CC(C)CN(C(C3(O)CC3)=O)C2)cc(Br)cn2ncnc12 C(=O)(CCCC(F)(F)C(F)(F)F)N1CC(SC)C(NC(=O)COC(C)(C)C)C1 c1(CC#N)ccc(C(=O)NC2(CCNC(c3cn(C4COC4)nn3)=O)CC2)cc1 c1(C(=O)OC)nc(C)c(C(N2CCC(C(=O)NC3(C)CCCC3C)C2)=O)s1 c1(C(N2CCCC(O)C2O)=O)cc(F)ccc1OC(F)(F)F CC1(C)CCOC(C(=O)NCC#CC(=O)NC(c2ccccc2)(C)C)C1 C1(C(=O)NCC2CCN(C(=O)Cn3cnc(Br)c3)C2)CCCS(=O)(=O)C1 c1(C(=O)NCC2(NC(C=CCC)=O)CC2)cccn2ncnc12 c1(COC)ccccc1C(=O)N(C1CCCC(C(=O)OC(=O)C2CC2)C1)C c1(C(=O)NCC2(NC(c3nc(CCC)sc3)=O)CCC2)nc(OC)ccc1Cl C#Cc1ccc(F)c(C(=O)NCC2CC2NC(C2(Cl)CC2(C)C)=O)c1 c1(C(N2CC(CNC(c3c(C)noc3C)=O)N(C)CC2)=O)cc(F)c(F)cc1O C1(CNC(c2ccn(C(C)C)n2)=O)CC2COCC2N1C(=O)CSc1nncs1 C1(CC)CCOCCN1C(C1CCCN(CCOCc2ccc(Cl)cc2)C1)=O C1(CNC(=O)NC2(C(=O)OC)CC(O)C2)CC(OC)(OC)CO1 CC1C(NC(=O)Cc2cc(Cl)ccc2Cl)CCCN1C(=O)Cn1cccnc1=O Cc1ccc2c(c1)CCC2Nc1conc1C1CCNCC1 C1(CNC(C(C(COC)C)C)=O)C(C2CC2)CCN1C(=O)C(CCOC)OC C(=O)(N=S(C)(=O)C1CCNCC1)C1(NC(N)=O)C(C)(C)NC1 C1(CC(N2CCC(CC)CC2)=O)CCC2CN(C(=O)C(C(CC)CC)OC)CC12 C(C(=O)NC1CC(CCNC(=O)C=Cc2ccccc2)C1)(C(C)C)OCC CCS(=O)(=O)C=CC(=O)N1CCC(C)C(NC(=O)CCOCc2ccccc2)C1 c1(SCC(=O)N(C2CCC(NC(c3cnn[nH]3)=O)C2)C)ccc(F)cc1 N1(C(C(=O)NCC(C(C)C)c2ccnn2C)=O)CCCC(O)(C2CC2)C1 c1(NC(C(CC)SC)=O)cc(CCO)ccc1C c1(COC)ccoc1C(=O)NCc1cc(C(=O)NC2COC(C(C)C)C2)on1 CC(=NO)C1CC(C(=O)NCC2(NC(=O)CCCCO)CCC2)C1(C)C S(=O)(=O)(c1ccnc(NC(=O)Cc2ccc3c(c2)CN(C)C3)c1)NC N1(C(C=C(COC)C)=O)CC2C(NC(=O)Cn3cc(-c4ccccc4)nn3)C2C1 C1(NC(c2cc(C)ncn2)=O)CCSC12CN(C(c1cccnc1C1CC1)=O)C2 C1(CCC)(NC(C)=O)CCCN(C(c2cnn(C3CCOCC3)c2)=O)C1 N1(C(C2OCCN(C(C3(CC=C)CCOC3)=O)CC2)=O)CCC(O)C12CCCC2 C(C(C)C(=O)N1CCC2CC12)NC(COCC#C)=O N1(C(C=NOC)=O)CCN(C(C2(n3cccc(O)c3=O)CC2)=O)C2CCCCC12 N1(C(CC2CC(CC)C2)=O)CCC(C)(CN(C)C)C1.C12(CCC1)C(=O)NC2 c1(SC)nc(C)c(C(=O)NCC2C3CN(C(c4c(C)nsc4C)=O)CC23)s1 c1(-c2c(CC)ncnc2)cc(NC2(CC)CC=CCC2)c(O)c(C(N)=O)c1 c1(-n2c(CC3CC3)nc(-c3c(OC)nccn3)n2)cccn(C(F)F)c1=O N1(C(C2CCN(C)CC2)=O)CCCCC2(CCN(C(=O)CC3(C4CC4)CC3)C2)C1 c1(C(N(CCCCNC(C2(C)CCCO2)=O)C)=O)c(Cl)cccc1[N+](=O)[O-] C(=O)(CCN=c1ccc(C)c[nH]1)NCCC1OCCN(C(C(CC)(C)CO)=O)C1 CCCCCCC(=O)NC(CC(=O)NC1CCOC(CC)C1)C(F)F C12(C(=O)NCC3(CC(=O)NC4COCC4CO)CC3)CCN(CC1)CC2 N1(C(c2c(OC)c(C)sc2)=O)CC2CC(NC(c3c(C)nn(C)c3Cl)=O)CC1C2 C1(CC=C)(NC(=O)CC(C)O)CCN(C(=O)NCc2ccccc2)CC1 C=CC(C)CC(=O)NC(C(=O)NCCC(C)(C)F)C1CC1 c1(C(=O)NCC(C)(C2CC2)NC(C2N(CC)CCOC2)=O)cc(C)cc(Cl)n1 N1(C(COC(C)C)=O)CCN(CCCCCNC(c2scnc2C2CC2)=O)CC1 N1(C(c2c(C)c(Br)cs2)=O)CC(C)(C)CC1CNC(=O)C(C)CO c1(C(C(=O)CSCC=CCN)=O)csc2cnccc12.c1(NC=O)ccc(Cl)s1 CC1(C(=O)NC2CC(NC(=O)CCC3(c4ccccc4)CC3)C2)CCCO1 N1(C(CN(C)CC)=O)CCC2(CCC2CNC(c2ccc(C(C)C)cn2)=O)CC1 C1(NC(C2(COC)CC=CC2)=O)COC2C(NC(=O)CSC3CC3)COC12 c1(CNC(c2cc[nH]c2)=O)ccsc1C(N1CCC(c2cnco2)C1)=O C12(CNCc3cccc(OC)c3N(C)C)CC3CC(CC(C3)C1N)C2 C12(NC(C3CN(C)C(=O)C3)=O)CCC(NCc3ccc(CC(=O)O)cc3)(CC1)C2 N1(CC)CCN(C(=O)C(C)N(C(c2cn3c(n2)CCC3)=O)CC)CC1C N1(C(C2CCCC3(CCOCC3)O2)=O)CCOC2(CCCN(C(=O)CCF)C2)C1 c1(OC(C)C)ncncc1C(=O)Nc1ccsc1CO c1(C(Cn2cc(-c3c(OC)ccc(C#N)c3)nn2)=O)cccc2c1S(=O)(=O)CC2 N1(C(c2cc(NC)oc2)=O)CCC2(CC1)CN(C(=O)CC13CC(C1)C3)CC(C)O2 Cc1cccnc1CNC(=O)C(C)N(C(c1c[nH]c(C)c1)=O)C1CC1 CC(CC(F)(F)F)C(=O)N(CCCN(C)C(C1CC2(CCCC2)CO1)=O)C CC1CCCC=C1C(=O)N1CCOCC(CNC(c2cccc3c[nH]nc23)=O)C1 CS(=O)(=O)c1cnc2cc(C(=O)NC(c3cc(F)ccc3F)C(=O)O)sc2c1 c1(OC)ccc(C)c(C(=O)NCCC23CCC(C2)N(C(=O)CNC(C)=O)C3)c1 c1(C(N(CC(CC)NC(C(CCC)OC)=O)CC)=O)cc2cc(C)ccc2o1 C1(C(=O)NC2(C(O)CO)CC2)CC(O)CCN1C(C1CCC2CC1CO2)=O Nc1ccc(C(=O)NCC2CCCCC2NC(C2(F)CCCCC2)=O)cc1 C1(N(C)C(c2cncs2)=O)CC2CC1N(C(=O)C(c1ccccc1F)(C)F)C2 CC(C)(C(=O)NC(CNC(=O)Cn1cc(C(C)=O)nn1)C1CC1)c1cnsc1 N1(C(C2(C#N)CCC2)=O)CCOC2(CCN(C(=O)CCCc3cnn[nH]3)CC2)C1 c1(C(N2C(CCNC(C(C(C)C)O)=O)CC(F)(F)C2)=O)cccc2ccoc12 N1(CCCCNC(C(CSC)C)=O)CCCN(C(c2ccc(=N)[nH]c2Cl)=O)CC1 N1(C(C(C)N(C)C)=O)CCC(CCN(C)C(C2CC=CCC2)=O)CC1 c1(OC(COC)C(=O)NCC(C)(C)NC(=O)CN(C)CCO)cc(C)ccc1Cl C1(CNC(C2CCN(C)CC2)=O)CCN(C(C2CCCC2F)=O)CC1O CN=c1nc(C(=O)NC2CN(C(C3CCCN3C=O)=O)CC2C)cc(C)[nH]1 N1(C(C2(c3cc(F)c(Cl)cc3Cl)CC2)=O)CCCC(O)(c2ccccc2)CC1 C1(CNC(CCOC(C)=O)=O)CCCCN1C(=O)C=CC1CC1 C1(NC(c2c(CCC)n(C)nc2)=O)CCC2(CCN(C(c3cn(C)cn3)=O)C2)C1 c1(OC)cccc2cc(C(=O)NC3CCC3CNC(=O)Cc3cc(C)cs3)[nH]c12 N1(C(Cc2n(C)cnn2)=O)CCCCC(NC(=O)CCn2ncn(C)c2=O)C1 C(=O)(C1=CNC2=NCCC2=C1)N1C(C)C(NC(=O)CC2CC2(Cl)Cl)CCC1 CC(N=c1[nH]c(=NCC2CC(F)C2)c2c(F)cccc2[nH]1)c1cc(Br)ccc1F N1(C(c2c(CC)ncs2)=O)Cc2n[nH]cc2C1C(=O)N1CCC(CCN(C)C)C1 C(C(F)C(C)(C)O)NC(C1CC(C)(NC(CC(C)F)=O)C1)=O CC1(C)CN(C(c2cnc[nH]2)=O)CCN(C(c2ncoc2Br)=O)C1 c1(C(N2C(CC(=O)NCCC(C)F)CC(O)C2)=O)ccc2cccnc2n1 c1(NC(CC2(OC)CN(C(C3CCCN3C(N)=O)=O)C2)=O)ccc(F)cc1O c1(C(N2CCC(CN(C(CC=CCC)=O)C)C2)=O)ccc(C(F)(F)F)nc1 C(CCN=C(NCC1CC2(CCOCC2)O1)N1CCCC(CC(F)(F)CF)C1)OC N1(C(C2CCCC2NC(C23CCCC2C3)=O)=O)CCc2ncccc2C1 C1(NC(c2n(CC(C)C)ncc2)=O)CCCCN(C(=O)CC2COC(C)(C)C2)C1 Cn1cc(C(N2CCC(CCNC(c3ccc(O)cn3)=O)CC2)=O)c(O)nc1=O N1(C(C(CCC)OCC2CCCCC2)C)CC2C(C1)C2(F)F C1(NC(c2ccc(SCC)cc2)=O)CCN(C(c2cnc(C)[nH]c2=N)=O)C1(C)C c1(COC)cccc(C(N2CCCC2C(N2CC[Si](C)(C)C2)=O)=O)c1 c1(CCC(=O)NCCC(C)N(C(=O)C2=NNC(=O)CC2)C)ccc(C#N)cc1F CC1CCC(Cl)=C(C(=O)NCC(O)CCNC(=O)COc2cccc(F)c2)C1 CCC(C(=O)OC)C(=O)NCC1CCCCN1C(c1cc(Cl)ccc1F)=O c1(S)ccc(F)cc1.C1(C(CNC(C=C(CC)C)=O)(C)O)CCN(C(=O)CCF)CC1 N12CC3C(CS(=O)(=O)C3C1)C2=O.CC1CC(C)(CSC(C)(C)C)C1 c1(C(C)NC(C(=O)N(C)Cc2nnc(C(=O)OCC)s2)=O)ccc(C)cc1F c1(CC(=O)NCC(C)CNC(C2(C3CC3)CCOCC2)=O)cccc2sccc12 Cc1noc(C)c1C(=O)Nc1ccccc1NC(C1CC1Cl)=O Cc1ccsc1NC(=O)NC1(c2ncccn2)CCOC1 C#Cc1ccc(C(=O)NCC2CN(C(=O)Cc3ccnc(Br)c3)C2)cc1Cl c1(CN(CC)Cc2cccc(O)c2)ccc(-c2ccc(C(=O)N(C)C)nc2)cc1 c1(C(=O)NCC(CC)NC(=O)CC2CC(C)=NO2)c(C)nn(C)c1N C1(CNC(C(C)(F)F)=O)COC(C(F)(F)F)CN1C(C1CCCC1)=O c1(C(C)NC(=O)NC2C(C(CC)(C)C)CCC2)ccc2c(c1)CC(C)O2 N1(c2nnc(C3CCC(CO)O3)n2CC2CC2)CCOC2(CCCC2)C1 c1(C(N(C2CCN(C(c3cccc(NC(C)=O)c3)=O)C2)C)=O)nc(C)ccc1C c1(-c2cn(CCCCCCNC(CC3C=NN(C)C3=O)=O)nn2)cc(Cl)ccc1F C(CCN=C(NCc1nnn(C)n1)NCC(O)Cc1ccccc1)OC(C)C N1(C(C2CCC(C)(CC)O2)=O)CC2(CC(CNC(c3cnc(C)[nH]3)=O)C2)C1 Cn1c(C(N2CCCCC2CCNC(C2CC(=O)NC2(C)C)=O)=O)cccc1=O C1(NC(C2(C)C(C)CCC2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 C1(C(N2CCCC(CNC(CCCOC(C)=O)=O)C2)=O)Cc2nn(C)cc2C(=O)N1 Cc1cccn2ncc(C(N3CCC4C(C3)CN4C(=O)C(=O)NCC3CC3)=O)c12 c1(C(=O)OC(C2(O)CN(C(=O)OC(C)(C)C)C2)C)cc(C(C)(F)F)ccc1C C(=O)(C1CO1)N(CCCC)CCCC.c1(C(=O)OCC)ccccc1 C1(c2ccccc2)(C(=O)NC(CN(C(COCC)=O)CC)C)CCOC1 C(=O)(CCCCCNC(=O)CC1CCSC1)N1CC(C)(C(N)=O)C1 N1(C(c2cn(CC)nc2C)=O)CC2CC1CN2C(=O)CCC1CCOC1 C(=O)(C(C)(C)C(F)F)N(CCCCNC(c1cc(OC)no1)=O)C C(CCCN=C(NCc1ccccc1)NCC1CC12CCSCC2)OC(C)C C1(CNC(=O)CC2(C(F)(F)F)CCC2)CCCCN(C(C2C=CC=CC=C2)=O)C1 c1(C(N(C2CC2)CC2CCCN(C(C=CSC)=O)C2)=O)cc(C)ccc1O CC1=CC(C)=NS(=O)(=O)N1CC(=O)NC1CCN(C(=O)Cn2cccc2)CC1C C1(C(=O)OC)(CCNC2CCC2N(C)C)CCN(C(=O)CCc2csnn2)CC1 C1(CCC)CCCC1C(=O)NCCC1(CNC(=O)Cc2csc(=N)[nH]2)CC1 c1(OC)cc(OC)nc(C(N2CCC(C(C)NC(=O)CC(C)C3CC3)CC2)=O)n1 c1(OC)cc(CC(=O)OCC(=O)C2(C(F)(F)F)CC2)ccc1C C1(C(=O)NCCNc2c(C)ccnc2)CCC(C)C(C)C1 C12(C(=O)NCC(CC)(C)C)CCC(CC1)N(C(=O)C(C)C1CCC1)C2 C1(NC(CC2CCCN(C)C2)=O)CCS(=O)(=O)C12CN(C(C1(CO)CC1)=O)C2 Cc1nn(C)c(Cl)c1CC(=O)NC1CCCCC1CNC(=O)CCC1CCOC1 c1(OC)cc(C(N2C(C)CN(C(=O)C(O)CSC)CC2C)=O)c2occc2c1 C12(CNC(C3CCS3(=O)=O)=O)CCCC1N(C(=O)CSCCC(F)(F)F)CCC2 c1(C(=O)OCC)nccc(C)c1NC(C1(C)CC1(Cl)Cl)=O C1(CN(C(=O)C(CO)c2ccccc2)C)C2CN(C(c3ncn(C)n3)=O)CC12 Cc1cc(N2CCC(C(F)(F)F)(CO)C2)nc(=NCC(C)CC2CCC2)[nH]1 N1(C(c2cnoc2C2CC2)=O)CCN(C(=O)CCc2cocn2)C(c2cccs2)C1 N1(C(C2(C)CC=CCO2)=O)CCN(C(C2COC(=O)N2)=O)CC2(CC2)C1 c1(CCCOC)ccc(-c2nc(-c3cc(Cl)ccn3)nn2C(C)C(C)(C)C)cc1 c1(C(=O)NCC(C(=O)N(C(C)C(N)=O)C)CC2CC2)cc2n(n1)CCO2 c1(C(N2CC(CNC(CCCOC)=O)C(C(F)(F)F)C2)=O)c(F)ccc(F)c1F C(=O)(CC(C)C(C)(C)NC(c1ncoc1CC)=O)NC(C=C)C1CCC1 c1(CCCC)nc(CN2CC(NS(C)(=O)=O)C2)c(Cl)[nH]1.N12CC(F)CC1C2=O Cc1nc2cncc(CC(=O)NCC(C(C)C)NC(=O)C(=O)N(C)C)c2[nH]1 c1(C(N2CCC(CN(C(C(C)S(C)(=O)=O)=O)C)C2)=O)c2ccccc2nn1C c1(C(=O)NC2(CC=C)CN(C(=O)CSCC3CCCCO3)C2)cc(C)sc1C O=C1CCC(C(=O)N(c2ncnc3occc23)C2CC3(C2)CC(N)C3)=NN1 C12(C(N3CC(NC(C45CCCCC4C5(F)F)=O)C3)=O)CCCN(CCC1)C2 C1(NC(=O)C(F)OC(F)(F)F)CC(O)(C(N(C(CC#C)C)C)=O)C1 C(CCCCC(=O)N1CCCC1C(C)NC(C1(N(C)C)CC1)=O)OC c1(C(=O)NC(C2OCCN(C(c3cc(COC)no3)=O)C2)C)cc(O)ccc1Cl c1(C(C(=O)NCC=C)N(C(C)C(=O)OC)CC(C)C)nn(CC)cc1Br Cn1nccc1C(F)=CC(=O)NCC1CC(NC(c2cccc(C(F)F)c2)=O)C1 N1(C(C=C2CCC(C)C2)=O)CCC(C(N2CC3C=CC3C2)=O)C1C(C)C C=C1CCC(C(=O)NCCCCN(C)C(C2(C(F)F)CCCO2)=O)CC1 C(=O)(CCCC(C)(C)C)NCCC1CN(C(C2(CC)CC(C)(C)C2)=O)C1 c1(COCC(=O)N(C2CCN(C(=O)C(F)=CC3CC3)C2)C)cccc(C(N)=O)c1 Cn1ncc(C(=O)NC2CC3C(NC(C4CCC(CC#N)CC4)=O)C3C2)c1Cl C1(C(N)=O)CCCC(SCC(=O)Nc2ncccc2F)C1 C(c1ccc(Cl)cc1)=CC(=O)NCC(C1CC1)NC(CCNC(C1C(C)C1)=O)=O C12(CCNC(=O)NC(c3ccc(NS(C)(=O)=O)cc3)C)COC(C)(C1)C2 C1(C(=O)NC(CNC(=O)C=Cc2ncc[nH]2)C2CCC2)CCc2nnnn2C1 C1(C(=O)NCC(CC)NC(c2cc(OCC)n[nH]2)=O)CCCNC1=O C1(=O)C(O)COCC(=O)N1.c1(N(C(C)C)C(c2ccccc2)F)ccccc1 N1(C(C2(CC=C)CC2)=O)CC2CC(C1)N(C(=O)C(C)CC(C)(C)C)C2 C(=O)(CCC(C)C)N(CC(=O)N(C)CCC1CCCN1C)CCOC C1(CN(C(CNS(CC)(=O)=O)=O)C)CCCN(C(c2cnn(C3CC3)c2Cl)=O)C1 N1(C(c2c(CC)cc(N)cc2)=O)CCN(C(C2CC(CF)C2)=O)CCC1C C1(CC(N2CC(CC=C)(NC(=O)Cc3cc(C)cs3)C2)=O)CCN(OC)CC1 CCC(CC)C(C)C(=O)NCC1(C2CC2)CCN(C(C2CCOC2)=O)C1 C(C(C)(C)C#CC(=O)N1CCC(CO)C(O)C1)NC(COC(CC)(C)C)=O C(=O)(C1=CCCCCC1)N1CCCC(NC(=O)CCn2ccnc2)C1 c1(CC)nc2c(C(=O)Nc3cc4c(cn3)C(=O)CCC4)ccnc2[nH]1 C1(CC)C(NC(c2ccc(SC)s2)=O)CCCN1C(=O)C=CC1CCOC1 C(=O)(CCCCCCSC)NC(C(=O)NC(CC=C)C(=O)OC)CO C1(C(C)C)(C(N2CC(O)(c3cnn[nH]3)C2)=O)CCCN1C(=O)C=C1CCOCC1 N1(C(c2c(OC)nccn2)=O)CC2(C1)CN(c1ncc(C)cn1)C2 N1(CC#C)CC2CN(C(c3c(Br)cncc3Br)=O)CC2C1 c1(CC(=O)NCC2N(C(C(C)SC)=O)CC2)ccnn1C C1(C2CC2)(CNC(c2c(C(C)C)n[nH]c2)=O)CCN(C(=O)C(=O)C(C)(C)C)C1 N1(C(c2nccc(CNC(C(C)CC3CC3)=O)c2)=O)CCOC(C)CC1 c1(OC)cccc(O)c1NC(C1CC1C(C)NC(=O)C(O)CC(C)C)=O C(=O)(CCC(C(C)C)NC(=O)CC1CC=CCN1C)NCC(CCC)CCC C#CCC(C)(C)C(=O)N(CCN(C(C1C2CCC1CC2)=O)CC)CC CC1(NC(=O)C2CC2)CCN(C(C23CCC(CO2)C3)=O)CC1 c1(C(N2CCC(COCCO)C2)C(=O)NCC=C)nc(Cl)cc(Cl)c1C c1(C(N2CCC(O)(C(C)NC(c3cc(C)[nH]n3)=O)C2)=O)cccc2sncc12 C1(CCN(C2CCCC2)C(CN(C)CC2CCCCN2)=O)CCS(=O)(=O)C1 CCC(O)(CC)CCNC(C1CC(C)(NC(C2OCCCO2)=O)C1)=O C1(C2CCOCC2)(NC(C(COC)C)=O)CC1.c1(C2C(=O)N2)cnn(C)c1 c1(C(N(C)CCN(C)C(C2(O)CCSCC2)=O)=O)c(F)ccc2cnn(C)c12 CCC(CNC(=O)CC=CC(C)(C)C)(CC)NC(c1cc(CSC)n(C)n1)=O C(C(C(C)C)NC(c1conc1C1CCCO1)=O)NC(C1(COC)CC1)=O C1(NC(c2nnnn2C(C)(C)C)C2(SC)CCC2)C2CCCOC12 C1(NC(C2CCC(=C)CC2)=O)CN(C(c2ccsc2C#N)=O)CC1N=[N+]=[N-] C(=O)(CCCS(N)(=O)=O)NCC(C1CCN(C(C(C(C)C)F)=O)CC1)(C)C n1(C2CN(C(c3cc(C)on3)=O)C2)cnc(=N)[nH]1.C(CS(C)(=N)=O)NC(=O)C c1(C(N2CC3(CN(C(C=C(C)C(C)C)=O)C3)C2)=O)cc(C)c(C)c2ncccc12 C1(C(=O)OC(C)(C)C)(COC)CCCN(N2CC(OC)C3(CC3)C2)C1 N1(C(COC)=O)CCC(CNC(c2cc(C)sc2S(N)(=O)=O)=O)C(C)(C)C1 C#CCC(C(=O)NCc1cncn1C(C)C)NC(=O)Cc1ccc(C)o1 C#CC1(O)CC(C(=O)NCCC(C)(C)CNC(=O)CNC(c2ccncc2)=O)C1 c1(C(=O)NC(C(C(C)C)NC(COCCC)=O)C)ccn2ncnc2c1 c1(C(N(CC(CNC(COC)=O)C)C)=O)c(C(F)(F)Cl)n[nH]c1C C1(NC(C(C2CC2)SC)=O)C2CC1N(C(=O)CCCc1nc(C)no1)C2C c1(C(=O)NCC2CC(OCC)C2)cc(Br)c2[nH]c(C)nc2c1 C1(C(C(=O)NC2CC2)OCCOCCCC#C)CCN(C(=O)CC(C)(C)C)C1 C1(CNC(c2cnc(S)nc2)=O)CC2(CCC2)CN1C(c1cc(F)ccc1Cl)=O C12(C(N3CC(O)(C(C)NC(=O)CN4C(=O)CCC4=O)C3)=O)CCCC1CCN2 n1(CCC)cc(CNC(=O)Cc2ocnc2CNC(=O)CC(=O)OC)nn1 Cn1cc(C=CC(=O)NC(Cn2cncn2)C(=O)NCCc2ncccn2)nn1 C1(CNC(c2c(C)sc(O)n2)=O)(NC(c2nc(=N)cc[nH]2)=O)CC2CCC1CC2 c1(C(=O)NCC(CC)NC(=O)C(C)(C)COCC(F)F)cnc(SC)n1C CC1(C)CC=C(C(=O)N2CCOC(C(=O)NCc3ccnc(F)c3F)CC2)CC1 C(=O)(CC(C)(C)C(C)(F)F)N1CCC(CNC(CCc2c(C)ncs2)=O)C(C)C1 N1(C(C2(C#C)CC2)=O)CC2(C1)CN(C(C1CCN(C)C1)=O)CC(C)(C)O2 C1(OC)CC(C(=O)NC2CCN(C(c3cnnc(C)c3)=O)CC2)N(C(C)=O)C1 C1(=CCNC(C(c2cccnc2)C)=O)CCN(C(C23CC(C#N)(C2)C3)=O)CC1 C1(Cc2ccc(F)cc2)(OCCO)CCSCC1.C12CCCC1NC(=O)NC2 C1(OCc2ccc(Oc3cccc(SCC)c3)cc2)CCC2(CCOCC2)C1=O C1(NC(C2(C=C)CCC2)=O)CN(C(c2ccnc(SCC)c2)=O)CCC1CO Cc1ccc(C(=O)Nc2ccccc2-c2ccc(O)c(F)c2)c(O)c1 C(CCCCCNC(C1SCCC1C)=O)NC(c1c(CC)scn1)=O N1(C(C(CC)N(C)C)=O)CC2(CNC(=O)C=Cc3scnc3C)CCC1CC2 N1(c2cccc(S(=O)(=O)N3C(C)SCCC3)n2)CCc2c(C)cc(Br)cc2C1 C(CC(C)(C)C(=O)NC1CCCN(C(c2ccc(F)c(O)c2)=O)CC1)OC C1(C(N2C(CC)CC2)=O)CC(C)N1Cc1coc(C(N)=O)c1 Cc1cc(NCCCN(C(=O)C(C)CSc2ccccc2)CCO)nn1C N1(C(C(CC)SC)=O)CCOC(CCNC(=O)CC2(O)CC2)C1 N1(CC(C)C)CCCC1C(=O)NCC1(CNC(=O)C=Cc2cscn2)CC1(F)F C12(CNC(C3CC(=C)C3)=O)CCCCC1N(C(=O)C(C)CCOC)CCC2 C(=O)(N=c1[nH]nc2[nH]ccnc1-2)C12C(CN(C(CCc3c(C)nccc3)=O)C1)C2 C1(C)(C(=O)NC(C2CCN(C(Cc3ncn(C)c3)=O)C2)(C)C)CNC(=O)C1 CC#CC1CN(C(=O)C(C)N(C(=O)C=CC(=O)N(C)C)C2CC2)C1 C(c1cccc(Cl)c1Cl)=CC(=O)NCCCNC(C1CC2C=CC1O2)=O N1(C(=O)C=Cc2cccnc2)CCC2(CCN(Cc3cccc4nc[nH]c34)C2)C1 C12(NC(C3C4CCCCCCC34)=O)CCCC1N(c1cc(C3CC3)ncn1)CC2 Cc1cnc(N2CCCN(C)C(=O)C2)c(S(=O)(=O)NC2(C)CC(C)OC(C)C2)c1 C1(C(=O)NC(c2cccc(C)c2)CNC(CCC=C(C)C)=O)CCC12CCCO2 c1(C(N2CC3CC(NC(=O)Cn4ncnn4)CC3C2)=O)cc2ccc(Cl)cc2o1 Cc1cccc2oc(N(C)CC3CCCN(C(=O)C4=C(Cl)CCOC4)C3)nc12 C(Cc1ccccc1)(C(=O)NCCN(CC(C)O)C(=O)CC1OCCCO1)OC C(=O)(C(C)(C)C(F)(F)F)NC(CNC(c1cn(CC(CC)O)nn1)=O)CO C1(C(=O)NCC2(OC)CC2)CCC(CNC(=O)CNC(=O)C2CC2)CC1 C1(NC(c2ccc(C(C)C)nc2)=O)CCC(O)CN(C(=O)CCn2cccn2)C1 N1(C(CC2(C)CCCC2)=O)CC(NC(C2CCCC(O)C2)=O)CC2(CC2)C1 c1(CCC(N2C(C)(CNC(CN(C3CC3)CC)=O)CCC2)=O)c(F)cccc1Cl c1(C(=O)NCC2C(NC(C3CCC(=C)CC3)=O)C2)ccc(F)cc1C(F)(F)F N1(C(=O)CC2CC3CC3C2)CCCC(CNC(C2(Cl)CC2)=O)C1 c1(C(=O)NC2CCN(C(C3CCCC3)=O)C2)cc(C(F)(F)F)ccn1 c1(N2C(CCCNC(c3cnn(CC4CCCC4)c3)=O)CCC2)ncc(I)cn1 N#Cc1cc(C(=O)Oc2cccc(C(=O)NC34CCCC(C3)OC4)c2)cc(O)c1 CC(C)(C#N)CCCC(=O)NCC1CCCC(NC(c2ccc[nH]2)=O)C1 N1(C(C2CC(CC)C2)=O)CCC2CCN(C(=O)C=C(C)c3ccccc3Cl)C2C1 Cc1nn(C2CCCC2)c(Cl)c1C(N1CCC(CO)(NC(=O)NC(C)(C)C)C1)=O C(C1=CCN(C(C2CN(C3CCC3)C2)=O)CC1)NC(CC1C(=O)NC(=O)N1)=O C#Cc1cccc(C(=O)NC(CN2CCN(C(=O)CN(C)C(N)=O)CC2)C)c1 N1(C(C(CC)O)=O)CCn2nc(C)c(CNC(c3cc(=O)n(C)o3)=O)c2C1 C12(CNC(COC3(C)CCC3)=O)CCC(CNC(c3ccnnc3O)=O)(CC1)CO2 N1(C(C=NOC)=O)CCC2CCC(NC(c3cc4c(C)cccn4n3)=O)C1C2 CC(C)CC(C(=O)NCC(O)CN(C)C(C1CC(C(N)=O)(CO)C1)=O)C(N)=O Cc1nc(NCC(C)(F)F)cc(=NCc2cc(F)cc3c2CCC3)[nH]1 N1(C(C2OCCN(C(CCCC#C)=O)C2)=O)CC2(CCC2)OCC1C CC1CN(C(=O)C(O)C(C)c2ccccc2F)CCN1C(c1cc(CF)on1)=O Cc1cc(CC(N2CCC(C)(NC(C3CC4(C3)OCCO4)=O)CC2)=O)ccc1F C1(NC(c2cnc(C)[nH]2)=O)CN(C(=O)CCc2cn(C)nn2)CCC1(C)C c1(C(=O)NCCCN(C(CSCCC#N)=O)C2CC2)cc2[nH]ccc2cc1Cl C1(NC(=O)CNC(=O)C2CC2)CCN(C(c2occ3c2CCC3)=O)CC1CO N1(C(CC2CC(CC)OCC2)=O)CC2CC(C1)N2C(=O)C(C)(C)CN(C)C Cc1cc(C(=O)NC(c2cn(C3CCN(C)C3=O)nn2)C)c2n[nH]cc2c1 N1CCC(C=O)C12CCC2.C1(COCCNC(=O)OC(C)(C)C)CCCO1 C=C1CC(C)(C(=O)NC2COCC2C(=O)NC2(c3nc[nH]n3)CC2)C1 C1(C2CCN(C(=O)CCc3nncs3)C2)(NC(=O)CCCc2cnn[nH]2)CC1 c1(OC)ccc(CC(N2CCC(C(F)C(N3CCNCC3)=O)CC2)=O)c(Br)c1 C(=O)(C1=CCCC1(C)C)NCC1(F)CC(NC(C2CN(C(C)C)C(=O)C2)=O)C1 Cc1scnc1C(=O)N(C(C)(C(=O)N1CCC1C1CCCC1)C1CC1)C c1(C(=O)NC2CN(C(c3c(C)c(=O)cc[nH]3)=O)C(C)(C)C2)cc2nnn(C)c2s1 C1(CNC(C2(C)CC(=C)C2)=O)CC(O)CN1C(c1ccc(C(=O)N(C)C)cc1)=O C(CC(C(=O)NC(c1cccc(Cl)c1)CNC(=O)CCC1CCC1)N(C)C)SC C1(CCC)CN(C(c2cccc(C3CCCOC3)c2)=O)CCN1C(=O)C1CC1 C1(C(N(C(CCNC(CN(C(C)C)C)=O)C)C)=O)CCc2cc(F)ccc2O1 N1(C(CC(CNC(=O)CC(COC)COC)OC)=O)CCn2c(C)nnc2C1 O=C1CC(C(=O)NC2COCC2NC(C2(CCF)CC2)=O)c2cccnc2N1 C(C(CC(F)(F)F)NC(=O)C(=O)N(C)C)NC1CN(CCCC)C(=O)C1 O=C1NC(=O)C2(CCC(C(=O)Nc3ccc(OC4CCCCC4)cc3)CC2)N1 C(CC(=O)NC1(C)CSC1)(C(F)(F)F)NC(C(C)CC(F)F)=O CC1CN(C(C2C3CN(C(=O)CCc4cccc(O)c4)CC23)=O)CCC1=O N1(C(CNC(CC)=O)=O)CCC2(CC1)C(OC)CC2NC(c1ncn(C)c1C)=O Clc1ccccc1-c1ccc(-c2ccc(NC3CC3)s2)cn1 Cc1ccc2occ(CC(=O)NC(C3CN(C(=O)CSC(F)(F)F)C3)C)c2c1 C(CN=c1nc(C#N)[nH]cc1C)=CCNC(C(CC)C(C)O)=O c1(C(=O)NC(C2CN(C(C3COC(=O)N3)=O)CCO2)C)ccn2cccc2c1 c1(N2CC(COC)N(c3ncc(C(F)(F)F)cn3)CC2)ncnc2n[nH]c(Br)c12 N1(C(COc2ccc(OC)cc2)=O)CCC(CNC(=O)C(C)C(C)C)C12CC2 N#Cc1ccccc1CNC(C12CCN(C(=O)CC34CCCC3C4)CC1C2)=O c12cccc(c1Br)C(=O)N2.c1(N(C(C)=O)C)ccc(-c2ccccn2)s1 C1(C(=O)N(C2CC(O)C2(C)C)CC)CCC2(CC1)CC2.c1(CC)ncccc1C=O CN1C(=O)CC2CN(C(C3CCCN3C(C3CCCC3)=O)=O)CCC12 CCCCC(O)C(=O)N1CC(NC(=O)C(F)F)C(C(F)F)C1 C#CCC(C)(C(=O)Nc1ccc(F)c(CC)c1)NC(C1CCOC1(C)C)=O C1(C#N)(CC)CCN(C(C2(C)CCC(C)C2(C)C)=O)CC1 N1(C(C2C(CC)CN(C(=O)CC3(C)CCCCC3)C2)=O)CCC(C2CCCC2)C1 Cc1ccc2cc(CC(=O)NCC=C3CCN(C(=O)C(C)N(C)C)CC3)ccc2n1 c1(C(N2CC(O)(CNC(CC3C(C)C3)=O)C2)=O)ccc2ncsc2c1 C(=O)(CCCC(=O)NC1(C(C)NC(C2CCOC2C(C)C)=O)CC1)NCC Cc1cc(CC(N2CC(CN(C)C(c3ccn(C4CCOCC4)n3)=O)C2)=O)no1 Cc1cc2[nH]c(C(N3CCC(n4cc(-c5cc[nH]n5)nn4)C3)=O)cc2o1 c1(C(=O)NCCNC(CC(C)C2CCCO2)=O)cc(Cl)cc(Br)c1 C1(NC)CCCC1C(=O)NCCCF.C1(C)(C)C=CC(=O)NCCOC1 c1(OCCn2cc(-c3nc[nH]n3)nn2)cnn2c1OCCCC2 C1(CNC(C(C)(C)OC(C)=O)=O)CCCC(CNC(c2ccns2)=O)C1 CCCC(C)(CCC)C(=O)N(CCCCCCNC(=O)C(C)(O)C(F)(F)F)C C=C(C)CCCC(=O)NC1CC(C(=O)NCC(CC(C)C)OC)CC1O C(=O)(C1=CC2(CCOCC2)C1)NC1CC(NC(C(C)OCCC#C)=O)C1 CCC(C)C(C)CNC(C1(C)CN(C(C2(n3cccn3)CC2)=O)C1)=O C1(O)(CNC(=O)NCCC(C)(C)c2ccccc2)CCCC1(C)C N1(C(c2c(C)nc(C)s2)=O)CC(=O)NCC1C(N1CC=CC(O)C1)=O C12(CNC(CCNC(=O)OC)=O)CCC(CN1C(c1ccc(OC)nc1)=O)C2 N1(C(c2cccc(SC)c2)=O)CCC(NC(C2CC(CCO)C2)=O)CC1C N1(C(=O)OC)CC(C(=O)NC(C)CNC(=O)CN(C(C)=O)C2CC2)S(=O)(=O)CC1 C(=O)(C(F)C(C)CNC(c1sccc1F)=O)NCc1cc(OC)ncn1 N1(C(COCC#C)=O)CC(NC(=O)C(F)C(F)(F)F)CC12CCC2 CN1CCCCC1C(=O)NCCC1CCN(C(C2(C(=O)NC3CC3)CC2)=O)CC1 C1(NC(CCNC(=O)NC)=O)CCN(C(=O)COC)C12CC2 c1(-c2n(CCOC)c(N3CCC(F)(c4ccccc4Cl)C3)nn2)ncc(C)cc1Br c1(C(=O)NCC2(CN(C(C3(CC=C)CCOC3)=O)C)CC2)cc(N)c(F)cc1F N1(C(N2C(CC)CN(C(=O)CC3CCCC(C)O3)CC2)=O)C(=O)NC(C)(C)C1=O CC1CCOC1C(N1CCCC1CCCNC(=O)C=CSCc1ccco1)=O c1(C(=O)NC2(CNC(=O)CCC3CCCN3C)CC(OC)C2)cccc(C)c1C C1(C(=O)NC(C#C)CC2CCC2)(CNC(=O)CCC2CCCO2)CC12CCC2 C1(N(C)C)CCCN(C(=O)C(C)(C)C2CCCC2)C1.C1(CNC(C)=O)CCN1 C1(CN(C(=O)Cc2ccncc2)C)CCCN(C(=O)CC2CCCC(=O)N2)C1 N1(C(C(CC)N(C(=O)C(C)CC2CCC2)C)=O)CC(C2=NOC(C)C2)C1 c1(C(=O)NC(C)CC2CN(C(=O)COC3CCCOC3)C2)ccnc2[nH]nnc12 C1(COC)CN(C(=O)CSCC(=O)OC)CCN1C(=O)CC1CCS(=O)(=O)C1 N1(CC)CC(C(=O)NCc2cc(C(N3CC(CCO)C3)=O)cs2)CC1=O c1(CC)ncc(CNC(=O)C(C2(C)CC2)NC(C2CC(C)=NO2)=O)[nH]1 c1(-c2onc(C(N(CCOC)CCOC)C)n2)coc2ccc(OC)cc12 N1(C(C(C)CO)=O)CCOC(C(C)NC(c2ccccc2C2CCCC2)=O)C1 C(N=c1[nH]cnc2c(OC)cccc12)C1(C)CCCN(C(C(OC)OC)=O)C1 N1(C(C2(C)CC(=C)C2)=O)CC(N(C)C)C(CNC(=O)C(C)c2ccsc2)C1 C12(C(=O)NC3CN(C(=O)CCCn4cccn4)CC3O)CCCCC1CCCC2 C1(N(C)C)(CSC)CC2CCC1CC2.C1(=O)CCC(=O)NCC2CCC(C2)N1 C1(C)(COC)CC(NC(c2cn[nH]c2)=O)CN1C(C1CC(F)(CF)C1)=O N1(C(CCCOCCOC)=O)CCN(C)C(CNC(=O)C(O)CC(N)=O)C1 C1(CNC(C(CC#C)C)=O)CCN(C(=O)CCSCc2ccccc2)CC1(F)F C12(NC(c3csc(-c4ccccc4)c3)=O)CC1CN(C(C1(CO)COC1)=O)C2 C1(C(C)C)(C(=O)N(C)CC=CC(=O)N(C)CCN2CCCC2)COC1 c1(CNC(C2C(NC(C=Cc3cc(C)no3)=O)CCO2)=O)ccc(C)c(C)n1 C(CCCC(=O)NCC=Cc1cccnc1)N(C)C(c1ccnnc1O)=O c1(C(=O)OC)ccccc1CC(=O)NCCCN(C(=O)CCC(F)F)CCO C1(C(N2C(C)(C(=O)NC)CC2)=O)C2CCCC2CN1C(=O)CC1C=CCCC1 C1(C(N2C(C(=O)NCC)CCC2)=O)(NC(=O)C2=C(Cl)CC2)CCCCC1 Cn1c(NCC2(C)CCCN(C(=O)CC3CCC(=O)N3)C2)cc(O)nc1=O c1(C(=O)NCC(CN(C(=O)C(C)(C)n2cncn2)C)O)n[nH]cc1C1CC1 N1(C(C)=O)CCC(C)(C(=O)NCC2CCCN2C(c2cnoc2)=O)CC1 C(=O)(C1=CCOCC1)NCCC1CCC(NC(C=C2CCN(C)CC2)=O)C1 C1(C(N(C2(C)CN(C(=O)CCn3ccnc3)C2)C)=O)CCCC1C1CC1 C1(C(N(C2CN(C(=O)CCCc3ccncc3)C2)C)=O)CCS(=O)(=O)N1 C(N=c1[nH]c(N(C)Cc2ccccc2Br)nc2c1CCCC2)c1ncc(C)cn1 N1(c2ncc(C)c(SC(C)C)n2)CC2CC1CCC2NC(c1ccncc1)=O N1(C(c2c(OC)ccc(C)n2)=O)CC2CCCN(C(C3CC3C)=O)C2C1 CC1CCC(C(=O)NC(c2cccc(O)c2)C(N2CCCC2(CO)CO)=O)CC1 Clc1ccc2c(c1)OCC2NC(=S)NCC(F)(F)F CN=c1[nH]cc(C(=O)NC(C)CNC(C2CC2(c2ccccc2)C)=O)o1 C1(NC(=O)NCCC2N(CC(=O)N(CC)CC)CCC2)CN(C)CCO1 C1(C(=O)Nc2cnc(Cl)c(Cl)c2)CCc2nc(-c3cccc(O)n3)sc2C1 C12(C(N(CC(C)(C)NC(C3CCCNC3=O)=O)C)=O)CCCC1CC(=O)C2 N1(C(c2cccc3ccccc23)C(=O)OC)Cc2ccc([N+](=O)[O-])cc2C1 C(C)(C)(CC(C)(C)C)NC(C1C(C(C)C)OCC1)=O.C12CCC(CC1)CC(=O)N2 c1(C(=O)NCC2CN(C(C3CC(CC)C3)=O)CC2C)cc(=O)c2ccncc2o1 c1(COC)cccc(C)c1N(C)CCC1CCSC1 C1(CNC(CCN2C(C)CCCC2C)=O)CN(CCC2CCCC2)CCC1(F)F C(CC1=CCN(C(C2CC2C)=O)CC1)NC(C1N(C(C)=O)CC(O)C1)=O C(C(O)C(=O)N(C(C)CN(C(=O)C1CN1)C)C)SC.N1(C(C)C)CCCC1.C(C)(=O)N C(CC(CC)C(=O)NC(C)C(CO)NC(c1ccccc1SCC)=O)=CC C1(C(=O)Nc2nc(O)cc(C(=O)OC)n2)CCCC2CCCCC12 C(=O)(CCCC(=O)NC1CS(=O)(=O)CC1NC(=O)C(F)(F)c1cnccn1)NC C1(C(N2C(CC)CN(C(=O)Cc3cccn3C)CC2)=O)CCc2nnnn2CC1 CC1CCN(C(=O)CCc2cccc(Cl)c2)C1CNC(=O)Cc1cc(Cl)n(C)n1 O=C(C#CC1CCC1)NCC12CC1CN(C(=O)CCC1CCC(C(F)(F)F)O1)C2 N1(C(c2cccc(CCC)c2)=O)CC2(CNC(=O)C(C)(C)CF)CC1CO2 c1(C(NOCCCC)=O)occc1CNC(=O)C(C1CCCC1)OCC C(=O)(C(N=[N+]=[N-])C(C)C)NC12C(CN(C(C(COC)OC)=O)C1)C2 C1(OCC)CC2(C1)CC2C(=O)NCC1CC(O)CN1C(=O)C(C1CCCCC1)C N1(C(C(=O)NCCCC2CC2)C2C(CC)C2)CCC2CC12 N1(C(C2C(=C)C2)=O)CCC2C(C1)CN2C(=O)C(=O)N=S(C)(C)=O C1(CNC(C=COCC)=O)CCCC(CNC(c2cnn(C3CCC3)c2)=O)C1 CC1(NC(C2CC3CC3C2)=O)CC(NC(c2ccsc2-n2cnnn2)=O)C1 Cc1nc2c(C)cc(C(N3CCOC(CN(C(=O)C(C)CO)C)C3)=O)cn2n1 N1(C(CCCC2(C)N=N2)=O)CCC(C2CC2)C1CNC(=O)CN1CC(=O)NC1=O CC(C)S(=O)(=O)CC(=O)N(C)CC1(CNC(C2CCC(=O)O2)=O)CC1 CCCC(CCC)CN=c1cc(C)[nH]c(=NCc2ccnc(C)c2)[nH]1 C1(NC(c2scc(C)c2)=O)CCCC12CN(C(=O)CC1CCC(C)(C)O1)C2 Cc1ccc(C(=O)NC(C2CCOC2)CNC(CCNC(=O)N)=O)c(C)c1.C1(NC)CC1 c1(C(N(CCNC(C(CC=C)Cc2ccccc2)=O)CC)=O)ccc(N)c(Cl)c1O N1(C(C=Cc2ncn(C)c2)=O)CCN(C(c2n[nH]cc2Br)=O)C2CC12 C(=O)(C1=CCC(C)CC1)NCC#CCNC(c1ccc(C(C)=O)cc1F)=O c1(CC)ccc(C(N2CCC3C(CCN3C(=O)CNC=O)C2)=O)c2ccccc12 C(=O)(C1=C(C)CCC1)N1C(CNC(C2CC(O)CN2OC)=O)(CO)CCC1.C(N)=O CCC(=O)NNC(=O)C(C)(C)CCCCNC(C1CCCCC1(F)F)=O C1(C(C(=O)NCCOC)N(C)Cc2ncnn2C)CCCOC1 c1(C(=O)NCCCNC(c2cncc(N3CCCC3)n2)=O)ccn2c1CCCC2 Cc1nnn(CC(=O)N(CCC(C)NC(C2(CO)COC2)=O)C)n1 c1(CC(=O)NCC(C)N(C(c2cc(C3CC3)nn2C)=O)CC)sc(O)nc1O C1(CC(=O)NCC(O)CNC(=O)CC(F)(F)F)NC(=O)CNC1=O c1(OC(C)C(N2CC3CCN(C(=O)COC4CC4)C3C2)=O)c(F)cccc1F N1(C(CCSCCC)=O)CC(CNC(C2(OC)CCC2)=O)C(C)C1 S(=O)(=O)(c1ccc2oc(=O)ccc2c1)N(C)CC1(F)CCOC1 C1(C(=O)NCC2(NC(C34CC(COC)(OC3)C4)=O)CCOC2)CCN(C)C(=O)C1 C1(NC(c2nc(C)nn2C)=O)CCC2(CC1)CN(C(C1CC1F)=O)CCO2 C1(NC(N2CCC(C(C)C)C2)=O)CCC(C)(C)CC1c1ccccc1 Cc1cc(C)c(CC(=O)NCC(C(C)(C)C)NC(C2CCCC23CC3)=O)s1 C1(C(N(C(CC)CO)CC)=O)CC2CN(C(c3ncc[nH]3)=O)CC2C1 n1(-c2c(C)cc(Cl)cc2)nc(-c2ccsc2)nc1C1=NOCC1 N1(C(CNC(C)=O)=O)CCCC(NC(=O)CC2CCCCC23CC3)CC1 N1(CC)CCN(C(=O)C(C)(CNC(C2CC2C2CCCC2)=O)CC)CC1=O c1(C(N2CCCC(N(C(=O)CN(C)C(C)=O)CC)CC2)=O)cc2ccncc2s1 c1(OC)ncc(C(=O)NCC2CN(C(=O)CNC(=O)N(C)C)CCO2)cn1 N1(C(c2cc(-c3ccc(C(F)(F)F)cc3)no2)=O)CCC(N2CC(F)(F)C2)CC1 C=C(C)c1cn(CC(C2CN(C(=O)CCNC(=O)NC3CC3)C2)F)nn1 CCCS(=O)(=O)C1CCCC1C(c1nnnn1C1CCC2(CC1)CNC(=O)C2)NCC N1(c2nc(N3CCC(c4cccc(C)c4)C3)nc(C)c2)CCC2(CCCOC2)C1 c1(C(N(CC(C)N(C(c2c(C)cc(SC)o2)=O)C)C)=O)cc(C)cc(C)c1 C1(CNC(CC=CC=C)=O)(NC(=O)C(C2CCCOC2)OC)CCC(F)(F)CC1 CCC(F)(F)CC(=O)NC1(CNC(=O)Cc2cc(F)cc(Cl)c2)CC2CCC1C2 C(CCF)(C(=O)NC(C)CCO)NC(c1c(COC)cc[nH]1)=O N1(C(C(CSC)OC)=O)CC2COCC2(C(=O)NCc2cccc(F)n2)C1 c1(CC)c(N2CC3CCC2C(NC(=O)C(CSC)OC)C3)nc(C)nc1Cl c1(OC)cc(C(N2CCC(NC(=O)C3=CCOCC3)C(O)C2)=O)c(Cl)cn1 N1(C(C2(C(=O)OCC)CC2)=O)CC2CN(Cc3ccc(C(F)F)cc3)C2C1 CC(CCN(C)C(C1CN(C)C1)=O)NC(=O)OC(C)(C)C CC1(C)CN(C(C2CCC2)=O)CC(CNC(C23CCCCC2C3)=O)O1 C(C(C(=O)NCC1CN(CC)C(=O)O1)C(C)C)NC(CC=CCC)=O N1(C(C(=O)NCC2C(COC(=O)NC)CCC2)=O)CCC(OC(C)(C)C)CC1 n1(CC)nc(C(C)C)cc1C(=O)NCC(O)CN(C)C(C1(c2cccs2)CC1)=O c1(CN2C(c3cc(CC)c(C)o3)CCC2)cc(Cl)cc(Br)c1F C(=O)(C1(C)CCn2c(C)nnc21)NCC1C(NC(CCc2c(C)cccn2)=O)C1 C1C(C2CCC2)CC(=O)N1C1CC1.C(C(C)(C)C)NC(C1(OCC)CC1)=O C(=O)(CS(=O)(=O)C1CC1)N1CC(CC)N(C(=O)Cn2nc(O)ccc2=O)CC1 c1(C(=O)NCC(CN(C(=O)CC2COCCO2)CC)O)csc(CC(F)(F)F)n1 c1(OC)n[nH]c(=NC(C)C2CC2)cc1-c1ccc(C(F)(F)F)c(Cl)c1 CCCC(C(=O)NC)NC(=O)CCCCNC(C1(CC(=O)OC)CC1)=O N1(Cc2nc(C)oc2)C2CCCC1CN(C(=O)C(c1cnn(C)c1)C)C2 N1(C(C)=O)CC(C2CCCN(C(c3cncc(-c4c(OC)ccc(C)c4)c3)=O)C2)C1 C1(OC)CN(C(c2ccnc(CN(C)C)c2)=O)CC1NC(=O)Cc1cccs1 N1(CC#C)CCC(C(=O)NC2(CNC(=O)C(=C3CCCCC3)F)CCOC2)CC1 CC1(CNC(=O)COCC(F)(F)F)COCCN(C(C2(C)CCCCOC2)=O)C1 N1(C(C(C)C)=O)CCN(C)CC1n1cccn1.N12CCC(CC1)NC2=O c1(OC)ncc(F)cc1C(=O)NC1CC1CNC(=O)CCc1ccc(C)cc1 N1(C(C(C2CCC2)OCC)=O)CCC(C)(CNC(c2c[nH]nc2C(F)(F)F)=O)C1 N1(C(C(CC)CCOC)=O)CC23CCCC2(C1)CN(C(=O)Cc1scnc1C)C3 N1(CCC)CCCC(C(N2CCC(O)(CNC(c3ccoc3C(C)C)=O)C2)=O)C1 N1(C(CCC(=C)Cl)=O)CC(C(N2CCC(OCC)C2(C)C)=O)CCC1(C)C C1(CCC)(NC(=O)CNC(=O)NC)CCCN(C(c2cc(OC)ccc2Cl)=O)C1 C12(C(=O)NCC(C)NC(=O)CC3CC(C)(C)CO3)CCC(C)(CC1)OC2(C)C Cc1[nH]nc(C(=O)NCC(C)(C2CC2)NC(C2CCCC2C(C)C)=O)c1C CCC(C)CCC(=O)N1CC(NC(=O)CCC2(C)CC2(F)F)C(O)C1 C(CCC(C)C)(C(=O)NCCCC1CCOCC1)NC(CC1(C(=C)F)CCC1)=O N1(C(c2c(OC)cnc(F)c2)=O)CCC2(CC1)CC2CNC(c1cc(F)n[nH]1)=O CC1(C)CCCC1C(=O)NC1CCCC1NC(c1ccon1)=O C1(CC)CCCCCC1(c1nnnn1CCCF)NCC(c1cn(C)nn1)(C)C Cc1ncc(C(=O)NC2CN(C(c3cn(C)nn3)=O)CC2C)n1-c1ccccc1 C1(NC(C(C)NC(C=C(C)C(C)C)=O)=O)CCCCN1C(C)C.C1C(C)(C)NS1 C1(C(=O)NCC2CCC(NC(c3ncn(C(C)(C)C)n3)=O)C2)CC(S(N)(=O)=O)C1 N1(C(C=CSC)=O)CC2(CC2)CC1CNC(=O)Cc1sccc1Cl C(C(C)(C)CC(=O)NCCCNC(C1CC1(C)C(F)F)=O)OC(C)=O N1(C(C(C)OCCC=C)=O)CCC(C2CC2)(CNC(=O)COc2ccn(C)n2)C1 c1(CN)sc(C(C)NC(C(=O)NCc2c(C(=O)OC)non2)=O)cc1C C(=O)(CCCC(=O)C(C)(C)C)NCC1CCN(C(C(C)CCC(C)(C)C)=O)CC1 C(C(C)(O)CC(=O)N1CCC(Cn2cc(-c3ccc(Cl)cc3)nn2)C1)SC C1(C)(CNC(CC=CC=C)=O)CCCC1NC(=O)Cc1cccnc1F C=CCCCCCCCC(=O)N1CCCN(Cc2cn(CCOCC)nn2)CC1 CC1=CCC(C(=O)NCC2(C)CCCN2C(=O)C=Cc2cc(C)no2)CC1 c1(CC)nc(NC(CCN(C(=O)C2=CCS(=O)(=O)C2)C)C(C)C)c(C#N)cc1C N1(C(C=CC(CC)C)=O)CCC2(CC(C(N3CCCC(F)C3)=O)C2)C1 c1(C(N(C(C(N2CCCC2C2CCCC2)=O)C2CC2)C)=O)nnc(O)nc1O C1(OC)CC(CNC(=O)CC2CCCC23CC3)N(C(=O)C#CC2CC2)C1 C#CCC(C(=O)N1CCC(NC(c2cncc(C)n2)=O)C1C1CC1)C1CC1 N1(C(c2nc(CC)oc2)=O)CC=C(CCNC(c2cc(Cl)ncc2OC)=O)CC1 N1(C(CCCOCC)C(=O)NCCC2(C)CC2)CCC(C(=O)OC)C2(CCC2)C1 C(C)(C)(CC(C)(N=c1ccn(CCOC(C)C)[nH]1)c1nnnn1C)SC C1(N2CCC(C)CC2)(CNC(C)(C(=O)OCC)c2ccccc2)CCCCC1C C#CCC(C)(CC)C(=O)NCCC1CCCN1C(=O)CCc1cc[nH]n1 C=CC(CC)CC(=O)NCC=C1CCN(C(=O)CC2CC(C)(C)CO2)CC1 CN(C)S(=N)(=O)N1CCCC1C(=O)NC1CN(C(=O)C=Cc2cnc[nH]2)CC1O c1(C(=O)NC2CC(C)N(C(=O)Cc3cn[nH]c3)C2)cc(O)c2sccc2c1 Cc1ccc(Cl)c(C(N2CC(NC(c3n[nH]cc3C3CCC3)=O)CC2(C)C)=O)c1 C1(C(N(C2CCN(C(=O)COCC(=O)OC)C2)CCC)=O)OCCN(C)C1=O C1(C(=O)NCC2CC(NC(C(c3ccccc3)OC)=O)C2)CCC([N+](=O)[O-])CC1 C1(C)(CC)CCCN(C(=O)C(C)(CO)NC(C2CCCC(=O)CC2)=O)C1 N1(C(C2N(C(c3c(OC)ccc(I)c3)=O)CCOC2)=O)CCNCC12CCC2 CC(C(=O)NCC1(CC(=O)NCCOC(=N)O)CC1)n1cncn1 CC(CC(=O)N1C(C(=O)NCCOCF)CCC1C1CC1)C(C)(C)C C1(C(N(CC(C)NC(=O)C2=COCCO2)C)=O)CCCCC(=O)C1 N1(C(C)=O)CCN(C(c2cncc([N+](=O)[O-])c2)=O)CC12CCCC2 c1(CCC(=O)NC2CCCC2NC(c2ccc(Br)o2)=O)nnc(O)nc1O c1(C(N(C2CN(C(c3cn(C(F)F)cn3)=O)C2)C)=O)ccn(C)c1 c1(C(C(=O)N(CCCNC(=O)C(C)Cc2ccncc2)CC)C)ccc(C)cc1 C1(CNC(C23CC(F)(C2)C3)=O)CC2CC2N1C(C1(F)CCCCC1)=O Cc1ncc(CC(=O)NC(C2CN(C(c3ccncc3F)=O)CCO2)C)c(O)n1 C(C(O)CC(=O)N1CC(O)(c2cc[nH]n2)C1)C(=O)Cc1ccsc1 C#CCC(CC(F)F)C(=O)N1CCOCC(C(=O)NC(C)CC(C)(C)C)C1 CC1(C)C(=O)CC1C(=O)NC(C)(C)C=CC(=O)NCC1(C)CCCS1 C1(CNCC(C2CCC(F)(F)CC2)C)C(=O)Nc2ccccc2S1(=O)=O CC(CN(C)C)CCC(=O)N1CCC2C(C(=O)NCCC(=O)NC3CC3)C2C1 C1(NC(C=CCOC)=O)CCOC(C(=O)NCc2nonc2C)C1 Cc1[nH]c(C)c(C(N2CC(CNC(C3CCCOC3c3cn[nH]c3)=O)C2)=O)c1C CN=S(C)(=O)c1cccc(C(=O)NCCNC(=O)CC2OCCCC2(C)C)c1 c1(OC)ccc(CC(=O)NC2CCC2NC(c2cn(C)nc2C(C)C)=O)c(Cl)c1 N1(C(C2ON=C(C)C2)=O)CCCC(NC(C2(S(N)(=O)=O)CC2)=O)C1C C#Cc1cccc(C(=O)NCC2CC(C(=O)N(C3(CO)CC3)C)CO2)c1C C(CC(C(C)C)NC(=O)CS(=O)(=O)CC)N(C(COCC(=O)OC)=O)C C1(C(N(C)CC2CC2(C)C)=O)CC=CCN1C(c1cccnc1)=O C1(CC=CC)CCCN(C(=O)C(C2CCN(C(=O)C(C)c3ccsc3)CC2)C)C1 c1(C(C(=O)NCC=C)NC)cc(C)cc(C)c1O.C1CCCC(N2CCCC2)C1 C1(CNC(CC2(CC)CCCC2)=O)CN(C(c2nc(Cl)sc2C)=O)CCC1(F)F C1(C(=O)NC(C(=O)NC)CC2CCC2)CCC2(CC2)N1C(=O)C(C)CSC N#Cc1ncc(C(F)(F)F)cc1NC(C12CC1CN(C(=O)Cc1cc(Br)cs1)C2)=O c1(CC)cc(C(=O)NCCN(C2CCCC2)C(c2nnn(C)c2C)=O)c(C)o1 C(=O)(C(O)C1=CCCCC1)NCCCC(C(=O)NCCCc1n(C)ncc1)(C)C c1(NC(CNC(C2COCCO2)=O)C2CC2)ccn2ccnc2n1 c1(C(c2n(C)nnn2)NCC2CNCC(C)(C)O2)cc2ccc(Cl)cc2o1 C1(CC(=O)N(CCNC(=O)C(c2ccccc2)C2CC2)CC)COCC(C)(C)O1 C(C(N=[N+]=[N-])C(=O)NC1CCC(NC(c2ccnn2CC(F)F)=O)CC1)OCC c1(N(CCCC)C)ccc(C(=O)NC(CO)C(C)NC(=O)CCOCCC)cc1 c1(CC)nc(C)c(C(N2CCCC2CN(C)C(c2cc(CF)on2)=O)=O)s1 CCC(O)C(=O)NCC1CC(CNC(=O)C(C)Cc2cccnc2)C1 Cc1nc(NCC(C2CC2)N(C)C(C2CC3CCCC23)=O)cc2nncn12 C1(C2CCCCC2)(C(N(C2CC(NC(=O)CCNC(C3CCC3)=O)C2)C)=O)CC1 C1(OC)CN(C(=O)Cn2ncn(C)c2=O)CC1NC(c1ccc(Cl)o1)=O C1(n2cccn2)(NC(CCOCC)=O)CCN(C(=O)C(CCSC)OC)CC1 c1(CC)onc(C)c1SCC.C1CCC(C(F)(F)F)O1 C(C)(CCCCCO)NC(CC(CNC(c1cccc(CO)n1)=O)OC)=O c1(SCC(=O)NCCC(CNC(=O)CC2CCOC2C)OC)ccc(C)cc1C N1(C(C(C)N2CCCC2)=O)CCC(C(O)CNC(=O)CCCNC(N)=O)CC1 C12(C(=O)NCCC3N(C(c4cc(C(C)=O)oc4)=O)CCSC3)COC(CCO1)C2 c1(C(N(C(CCNC(CC(C)C)=O)C)C)=O)cncc(-n2cccn2)n1 C(C)(C)(C(=O)N1CC(c2ocnc2CNC(C2CCC(=O)N2)=O)C1)NC(=O)OC N1(C(c2c(C)cco2)=O)CCN(C(=O)C2CC2)C(c2cn[nH]c2)C1 C1(C(=O)NCc2n(C)ncc2)CCC2CCC1N2C(=O)Cn1ccccc1=O c1(C(=O)NCC(CNC(C(C)OCC#C)=O)(C)C)cnc(S)n1C C1(C)(C(=O)NCCSCC)CCCN(C(=O)CNC(=O)C(C)(C)C)C1 C(C)(CN=c1[nH]cnc(Cl)c1Br)N(C(C(C)CCN(C)C)=O)C N1(C(C2C(CC)OCC2)=O)CCN(C(c2ccc(COC)s2)=O)CC12CCC2 N1(C(C2(OC)CCC2)=O)CCC(CCNC(=O)C(F)=C(C)C2CC2)C1 C1(C(=O)NCc2n(C(C)C)ccn2)CCCC(NC(=O)C(C)c2cc[nH]n2)C1 c1(NC(C2CCNC23CCC3)=O)cccc(S(=O)(=O)NCC(F)(F)F)c1 c1(C(N2CCC3(NC(c4conc4C4CC4)=O)C(C2)C3)=O)cnc2ccccn12 S(=O)(=O)(C1CCN(C(c2cc(C)ncn2)C(=O)NCC2CC2)C1)NC C(C(CC(=O)N(CC(C)(C)O)C)NC(c1csc(F)c1)=O)OC c1(N2CCC(C)(OCC)C2)nc(N2CCC(N(C)CC)C2)c2ccc(C)cc2n1 Cc1sc(O)nc1C(=O)NC(C(=O)NCCc1cc[nH]n1)c1ccoc1 N1(C(C23CC(CN(C(C(CC4CC4)OC)=O)C2)C3)=O)CCC2(CCCCO2)C1 C(=O)(C1SCCc2ccccc21)N(CCn1cc(-c2nccc(OC)c2)nn1)C c1(OC)cc(F)ccc1N1CCN(C(=O)NC(c2cccnc2)CN(C)C)CC1 c1(OC)ncnc(C(=O)NCC(F)CNC(c2cn(CCO)nc2C)=O)c1F c1(C(=O)NCC(CC)NC(c2conc2C2CC2)=O)cnc2c(cnn2CC)c1 N1(C(C(C)Oc2cccc(C)c2)=O)CCC(NC(=O)C#CC2CC2)CC(O)C1 C12(C(=O)NC(CCC(C)C)C)CC(CO1)N(C(=O)CC(=O)N(C)C)C2 C1(C)(CNC(C2CN(C(C)C)C2)=O)CCN(C(c2c[nH]nc2-n2cnnn2)=O)C1 Cc1ccc(CN2CC(C(=O)Nc3csc(Br)c3)CC(F)C2)c(F)c1 Cn1cc(S(=O)(=O)NCC2(F)CCCN(C(=O)Nc3ccc(F)c(F)c3)C2)cn1 C1(C(N2CC(C)(CNC(c3cccnc3O)=O)OCC2)=O)CN2CCCN1CC2 C(=O)(C(C)OC1CCCC1)NCC1(CN(C(COC(C)C)=O)C)CC1 C12(CNC(c3c(C)nc[nH]3)=O)CN(C(C3(C)CCCCC3)=O)CC1CCO2 C(=O)(C(O)CC(F)(F)F)NCCOCCNC(C1CCCOCC1)=O c1(C(N(C(CNC(=O)CCC2CC(F)(F)C2)C2CC2)C)=O)ccc(O)c(F)c1F c1(C(N2C(CNC(C3CCNC(=O)C3)=O)CC(OC)C2)=O)ccc2c(c1)CCN2 Cc1ncc(CC(C)C)cc1-c1nc(C2(C)CC2)nn1CCCC(C)C Cc1ccc(=N)[nH]c1C(N1CCC(C)(CNC(C2(C)CC(C)C2)=O)C1)=O c1(CN(CC(C)(C)O)C(=O)NCCN2CCCCC2)ccc(F)cc1F C=C(C)C(CC(=O)NC1CCC(N(C)C(C2CCC(F)(F)CC2)=O)CC1)OCC N1(C(c2n(C=C)nnc2)=O)CCC2CN(C(C3(C)CC(C)(C)C3)=O)CCC2C1 CC(C)(C)C(CNC(c1cn[nH]c1)=O)C(=O)NCC1CCCC12CC2 C1(C(N2CC(N(C(C3CC(OCC)C3)=O)C)C2)=O)COCCO1 C1(C(C)C)CN(C(c2ccc(-c3cn[nH]c3)cn2)=O)CCN1C(=O)C(C)C1CC1 C1(C(N2CCC(CNC(=O)Cn3cccnc3=O)CC2)=O)(OC)CCCOC1 Cn1c(C(N2CCC(C)(O)C(C(=O)O)C2)=O)nc2cc(Br)ccc12 N1(C(C=Cc2ccc(C)cn2)=O)CCC2(NC(=O)CS(N)(=O)=O)CCCCCC12 n1(C(C)C)ncc(CNC(C2CN(C(=O)OC(C)(C)C)CC2CO)=O)c1F c1(C(N2CCC(C)(CNC(C3CC(=O)C3)=O)C2)=O)c(Cl)oc2ccccc12 CC1(NC(=O)CCc2nnc(C(F)F)o2)CCCN(C(C2CC2F)=O)C1 C1(OC)CC(CNC(=O)C(C)(C)c2ccn(C)n2)N(C(c2cnc(C#N)s2)=O)C1 N1(C(C(C2CC=CCC2)NC(CN2C(C)CCC2)=O)=O)CC2CCCC2C1 N1(C(C(=O)OC)=O)CCn2ncc(CNC(c3csc(C)c3)=O)c2C1 N1(C(c2c(SC)ccc(N)c2)=O)CC2CC(NC(c3c[nH]nc3C)=O)CC1C2 N(C(=NCCc1ccccn1)NCC1CCOC1)C(CC)C C=CC(CCC)CC(=O)NCC1(CNC(C2Cc3ccccc3O2)=O)CC1 c1(C(C)C)conc1C(c1nnnn1C)NCCn1cnnn1 N1(C(C2C(C(C)C)CCC2)=O)CCN(C(C23CC=CCN2CCC3)=O)CCC1C C1(O)(CNC(C2(C)CC2(F)F)=O)CCCN(C(c2cncn2C2CC2)=O)CC1 N1(C(C2N(C)CC2)=O)CCCC1CC(N1CCC(CC2CC2)C1)=O C(=O)(C(=O)N=S(C)(C)=O)N(CC(C)NC(=O)C(c1ccc(F)c(F)c1)O)C C(C)(CC(=O)NCCC1CCN(C(c2cnc(S)n2C)=O)C1)(C(F)F)N(C)C C1(NC(c2cnc(O)s2)=O)CC2(C1)CC(NC(C1(CC3CC3)CC1)=O)C2 C1(C2CCCCC2)(C(C)(C)C)CC1.c12ccnc(n1)NC(=O)NCCO2 c1(C(=O)NCC2C(OCC)CN(C(c3n[nH]cc3CC)=O)C2)cc(C#N)cn1C c1(C(N(C2COCC2CNC(C2CCC(C)(F)CC2)=O)C)=O)ccc(F)cc1F c1(OC)ccc2[nH]cc(C(=O)NC3CN(C(=O)Cc4coc(C)n4)C4CC34)c2c1 c1(OC)ccc(Br)cc1C1(C(=O)NCC(C)NC(=O)C2=CCSC2)CC1 c1(C(N2CCOC2)COC)ccc(Br)nc1[N+](=O)[O-] N1(C(C(C(C)C)C2(C)CC2)=O)CCCCC2(C1)CN(C(c1cnc(O)n1C)=O)C2 S(=O)(=O)(c1nccs1)NCC1CCC(C(=O)NCCc2ccc(Br)s2)CC1 N1(C(C(C)=CC=C)=O)C(C(=O)NC2(C(C)C)CCC2)CCC1C(C)C c1(C(=O)OC)ccc(NCC2CCC(OC)CC2)c(C#N)c1 CN1CCc2[nH]nc(C(N3CC(CNC(c4ccc[nH]4)=O)C4CC34)=O)c2C1 c1(CC(=O)NC2CC3C(NC(C(C=CC)O)=O)C3C2)ccc(F)c(F)c1 C(=O)(C(=O)C(C)(C)CC)N1CC(CC=C)(NC(C2CC(N=[N+]=[N-])C2)=O)C1 N1(CC2CCC(C(=O)OC)C2)C(=O)NC(C)(c2ccc(F)cc2)C1=O N1(C(CC)=O)CC(C2CCCN(C(=O)C=CCN(C)C)C2)C1 N(C(=NCCCF)NCCC=C=CC)C(c1cccc(Cl)c1)C#C c1(C(C)NC(=O)NCC2(c3ccccc3Cl)CC2)ccc2c(c1)CC(C)O2 C1(C(N(CC(=O)OCC)C)=O)CCN(C(=O)CCOCC(F)F)C(C)(C)C1 c1(CNC(C2(O)CCN(C(c3ccc(OC)nc3)=O)C2)=O)ccc(F)cc1Cl Cc1nccc(N2CC3CC2C3C(N2CCC2c2ccccc2)=O)n1 CC1(NC(C2(CF)CC2)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)C1 C1(NC(C(C)OCC=C)=O)C2COCC1CN(C(C1CC3CC(=O)C1C3)=O)C2 c1(OC)ccc(NC(=O)C(=O)NCc2ccc(Cl)cc2)c(C)c1 c1(OC)ccc2ccc(NC(C3CC(C4CC4)=NO3)=O)cc2n1 C1(NC(c2c(SCC)cc(Br)cc2)=O)CC2(CCC(C)(C)CC2)C1 C(=O)(C1CNC(=O)c2ccccc21)NCC1CCC(NC(C2C(=C)CC2)=O)CC1 CCC(CNC(=O)C(C(C)C)NC(=O)Cn1ccnn1)C(C)(F)F c1(OC)ccc(Cl)c(C)c1C(=O)NC1CC(N(C(=O)CN(C)C2CC2)C)C1 c1(C(=O)NCC2C(C)CN(C(c3cscn3)=O)CC2)ccc(C#CC2CC2)cc1 C1(NC(CC(=O)NCC2CC2)=O)CCOC12CCN(C(=O)C=CBr)CC2 c1(C(=O)NC2CCC(C)(NC(C(CC)O)=O)CC2)cn2cccc(F)c2n1 C1(CNC(C=CSC)=O)CCN(C(=O)CC23CCCC2C3)C12CC2 C1(CNC(C2(O)CCN(C(=O)CC(F)(F)F)CC2)=O)CC1C1CCCCC1 N1(C(C(C)C(F)F)=O)CCCCC2(C1)CN(C(=O)Cc1sccc1Cl)C2 C1(NC(CC(=O)NCC#C)=O)CCCN(Cc2nc(CCC(C)C)no2)C1C c1(CNC(N2C(CN(C)C)C(C)(C)C2)=O)ccnc2c1ncn2C C1(NC(c2c(CC)[nH]nc2Cl)=O)CCCCCN(C(C2CC(C)(CC)C2)=O)C1 C1(N(C(=O)COCC(F)(F)F)C)CCC2(CC1)CCN(C(=O)CC1C=CCC1)C2 C(=O)(C1=CCC(C(F)(F)F)OC1)NCCN(C(c1n(CC)ccc1)=O)C1CC1 C(CCC(=O)NC(c1cnn(C)c1)C(=O)NC(c1nc[nH]n1)C)OC(C)C c1(C(=O)NC2CCCC(CNC(CN(C)C)=O)C2)cncc2c1CCC2 Cc1c(C(=O)NC2CCN(C(c3cnncc3O)=O)C(C3CC3)C2)cncc1Cl C1(CNC(CC=C)=O)CC2(CO1)CN(C(=O)CCCC(OC)c1ccccc1)C2 c1(C(n2cc(CN(CCO)C(C3CCCN3C)=O)nn2)C)ncccn1 c1(C(C(=O)NCC2(NC(=O)CCCc3cncs3)CCC2)SC)cccc(Cl)c1 Cc1cc(C(C(F)(F)F)OC(c2ccc(N3N=CCC3=O)cc2)=O)cc(C)c1 C(CCCCCNC(C1C2CCCCC12)=O)N(C(C1OCC(C)C1)=O)C C1(C(=O)NC2(CNC(C3CC(C)(O)C3)=O)CC(OC)C2)CC2CCC1C2 C1(C(=O)OC)CCC2C(=O)N(c3c(CCC(=O)N(C)C)ncn3C)C(=O)N2C1 CC(C)C(C(C)NC(C1CC(N(C)C)C1)=O)NC(c1cncc(O)c1)=O c1(C(=O)NCC(CCOC)NC(=O)C(C)(F)C(=O)OC)c(F)ccc(C)c1Cl C#CC1CN(C(C2CCCN2C=O)=O)CCN1C(=O)C=CCOCCOC c1(C(N2CCN(C(C=C3CCC(C)(C)CC3)=O)CC2)=O)noc2c1CCCCC2 c1(C(=O)NC2C3CN(C(C(CC)(F)F)=O)CC32)cnc(CC(C)C)nc1O C(=O)(C(CO)C(C)(C)C)NC1C(C)(CN(C(CC(=C=C)C)=O)C)CCC1 C1(OC)CCCC1N=c1cc(C)[nH]c(=NCc2c(N)cccc2F)[nH]1 c1(CC(=O)NCC(CC(C)C)NC(=O)C(C)CC(C)(F)F)cc2ccccc2o1 N1(C(C2C(C)(C)C2(F)F)=O)CCC(C2CN(C(c3ccnc(O)c3)=O)C2)CC1 C(CC(C(C)(C)C)NC(c1cnc(O)o1)=O)N(C(=O)CC1(O)CCCCC1)C c1(C(=O)NC2CN(C(=O)C(=O)Nc3ncc[nH]3)C3CC23)coc2c1CCCC2 c1(CC(=O)Nc2c(C(=O)OC)cc(F)c(F)c2)cccc(F)c1[N+](=O)[O-] C12(NC(C(CC)OC3CCCCC3)=O)CC(CNC(C3(C#N)CC3)=O)(C1)OC2C C(C)(CCCCO)NC(C1CC(C)(NC(CCNC(COC)=O)=O)C1)=O S(=O)(=O)(c1cncc(C(F)(F)F)c1)NCC1CCC(NS(C)(=O)=O)CC1 c1(SCCC(=O)N(C2CCN(C(=O)C(C)Cn3ccnc3)C2)C)ccccn1 c1(C(C(=O)NCCNC(C(CC)=CCCC)=O)C)ccc(Cl)nc1 N1(C(=O)NCC)CCN(Cc2ccc(-c3onc(-c4scc(C)c4)n3)cc2)C2CC12 C1(C(=O)NCC2C(C)(C)CCCO2)CCCN1NC(=O)C(=O)NC1CC1 N1(C(C(C(CC)C)O)=O)CC(C)OC2(CCN(C(=O)CC3CC4CC4C3)C2)C1 N1(CC(C)NC(=O)C(O)CNC(=O)CC2CCN(C3CC3)C2)CCCC1=O c1(C(=O)NC(C)CCCNC(=O)C(O)CC(F)(F)F)ccc2ccccc2c1 c1(C(=O)NCCCCCN(C(=O)CC(C)(C)C(F)F)C)ccc2c(n1)CCOC2 c1(CCC)ccc(C(C(=O)NCC)N(C2CC(F)(F)C2)C)s1 Cc1c(C(N2CC(NC(C34CC(F)(C3)C4)=O)C2)=O)cc(S(N)(=O)=O)cc1[N+](=O)[O-] c1(OC)ccc(C=CC(=O)NC(C)CNC(C2(F)CCC2)=O)cc1Cl CCC(CNC(=O)C(O)Cn1cncn1)(CC)C(=O)NCc1nccn1C(C)C N1(C(Cn2ccc(C)n2)=O)CCC(C(=O)NC(=O)CSc2cn[nH]c2)C1C CC1CN(C)C(C)CN1.c1(C(=O)C(F)(F)F)csc(=NCc2cc(Br)cnc2F)[nH]1 c1(C(N2CC(CNC(c3cc(C)[nH]n3)=O)C(C)CC2)=O)ccc(C)c2c1CCC2 C1(C(=O)OC)(CN2C(CN(C(=O)Cc3n[nH]c(C)n3)CC)CCC2)CCCCC1 N1(C(C(=O)NCCCC)CCC2CCOCC2)CC(C2(O)CCC2)C12CCC2 CC1(C(N2CC(C(N)=O)(CNC(c3cccnc3)=O)C2)=O)CCCS1 c1(OC)cnc(C(=O)NC2CN(C(=O)CCCc3cccs3)CCC2O)c(F)c1 N1(C(CC)CC)CC(C(=O)NC23CC(C2)N(C(c2cc(=O)n(C)o2)=O)C3)CC1=O c1(N(C)CC2CC=C(C)CC2)ncc(C)cc1S(=O)(=O)N1CCC1 C1(CNC(CC(CCC)C)=O)CN(C(=O)CC2CC=CCC2)CC(C)(C)O1 c1(N2CC(CN(C)C(C3CC34CC(O)C4)=O)OCC2)ncnc(Cl)c1C(C)=O C1(CNC(CCC(=C)C)=O)(NC(=O)C(C)CC(C)C)CCC(F)(F)CC1 C1(NC(C(CNC(C)=O)(C)C)=O)CCCN(C(=O)CC2C=CCC2)CC1 n1(CCC)ncnc1CNC(=O)C=CC(C)NC(C1CC2CC2C1)=O c1(C(=O)NC2CC(OC)CN(C(CCC(C)OC)=O)C2)ccc2c(c1)CCCO2 CCCCCCC(C)C(=O)N1CCC2CCC(C1)N2C(=O)C(C)CCO C1(CN(C(C=CC(CC)=CC)=O)C)CCCN1C(c1cc(C)[nH]n1)=O CC1CCS(=O)CCN1C(=O)Cc1cccc(C(F)F)c1 N1(C(C2(OC)CCN(C(CCCCCC)=O)C2)=O)CCC2(COC(=O)N2)C1 C(=O)(C#CC(C)(C)C)N1CCC(c2c(CNC(C3(CCC)CC3)=O)c[nH]n2)C1 C1(NC(c2c(Cl)cc(C)nc2)=O)CCN(C(c2ncc(Cl)s2)=O)C12CCCC2 CCC(C)CC(CO)NC(=O)CCC1(NC(c2cnsc2)=O)CCCC1 C1(N(C(C2CN(C)C(=O)N2)=O)C)CN(C(=O)COc2cccc(O)c2)CC12CC2 c1(CC(=O)NC2CC(CCNC(CC(CC)C3CCC3)=O)C2)ccc(F)cc1F c1(CC(=O)NC(C)CNC(=O)C(C)(C)Cc2cnn[nH]2)ccc(-n2cccc2)cc1 N1(C(c2occ(C)c2)=O)CCC(F)(CNC(C2CCCCN2C(N)=O)=O)CC1 C(=O)(C(O)C(C)(C)C)N(CCCNCC(=O)NC(C(CC)C#N)=O)C1CC1 c1(OC(C)(C)C)ccc(OCC(=O)NCCNC(C2(C)CC2(F)Cl)=O)cc1 C(c1ccc2c(c1)CCO2)=CC(=O)NC1C(OC)CC(F)(F)C1 N1(C(C(CC=C=C)NC(=O)CN(C)C(=O)OCCOC)=O)CCC(O)C(F)(F)C1 C12(C(=O)NCCC3CC(NC(=O)C(O)CC(F)(F)F)C3)C3CCC(CC13)C2(F)F C(=O)(CCC(CC)OC)N1CC(CCC)C(NC(C(Cn2cncn2)CC)=O)C1 CC1(C)CCC=C(C(=O)NC23CC(CNC(=O)C#CC4(C)CCCO4)(C2)C3)C1 c1(C(=O)NC(CNC(CC2C(C)CCC2)=O)C)c(F)c(F)cc(F)c1F c1(NCC(C)S(N)(=O)=O)cc(S(=O)(=O)NCC2(N(C)C)CCCC2)ccc1C#N C(c1cc(F)c(F)c(F)c1)=CC(=O)N(c1ccc(NC(=O)OC(C)(C)C)cc1)C1CC1 c1(C(=O)OCC)ccc(C(=O)NCCCCC(C)NC(=O)CN(C)CC)nc1 C#CCCC(O)C(=O)N1CCOC(CCNC(=O)CCNC(=O)C(C)(C)C)C1 C#CC1(C(N2CCC(CCN(C)Cc3cn(C)nc3CC)CC2)=O)CCCC1 C(=O)(C(C)CC(C)C)N(C(C(NOC(COC)COC)=O)C)C c1(CNC(C2CC(=O)NC2)=O)cccc(CNC(c2ncc(Cl)s2)=O)c1 c1(NC2(C)CC(NC(CCCN(CCC)C(C)C)=O)C2)ncc2c(ncn2C)n1 N1(C(C(C(C)(C)C)O)=O)C2CCC1CN(C(=O)CC1OCCCO1)CC2 C1(CNC(=O)COc2cn[nH]c2)CC2(CCC2)CN1C(C1C=CCCC1)=O Cc1cnn(CCC(=O)NC2CC(NC(C3CC34CCC4)=O)C2)c1 N1(C(CC(C=C)(C)C)=O)CCC2CCN(C(c3cc4c(cn3)OCCC4)=O)CC12 C12(NC(CCC(=O)N(C(C)C)C)=O)CC(CNC(C3(C)CC3(Cl)Cl)=O)(C1)OC2C c1(C(N2CCC(CN(C(C(C)c3ccco3)=O)C)CC2)=O)cc2n(n1)CCCN2 Cn1ncc2ncnc(N3CC(F)CC3C(=O)Nc3ccc(F)cc3[N+](=O)[O-])c12 CCCC(CCNC(=O)C(CC1CCCC1)NC(=O)C(C)N1CC(C)C1)CCC C1(CCCC(=O)NC(C)CC2CN(C(=O)C(=O)N(C)C)C2)CCCC(=O)N1 C1(O)(C(=O)NC(C=CC(=O)N(C2(C#C)CC2)C)C)CCCC1 n1(CCC(=O)NC(CC)CN(C)C(C2COC2)=O)sc2ccccc2c1=O C1(N(C(=O)CC2CC2C2CC2)CC)CCN(C(=O)C=CC(=O)OC(C)(C)C)CC1 c1(CCSC)nc(-c2cncc(-n3cccc3)c2)n(-c2cccnc2)n1 N1(C(c2cc(C)sc2C)=O)CCCCCC1CNC(=O)CCc1cn(C)nc1C c1(CC)cccc2sc(NC(=O)NC(c3ncc(-c4ccc(F)cc4)o3)C)nc12 C1(NC(Cc2c(C)noc2)=O)CCN(C(=O)COc2ccc(Cl)nc2)CC(O)C1 CC(C(F)(F)C(F)(F)F)=CC(=O)NCCCOCCNC(=O)CSC(F)F C1(C(=O)NCC(CNC(CC(C)OC)=O)(C)C)CCS(=O)(=O)N1C N1(C(C=CCC(C)(C)NC(C(C)OCC=C)=O)=O)CCN(C)CC1CCO N1(C(C(C2CCCCC2)OC)=O)CCN(C(=O)CC2(O)CCC2)C(COC)C1 N1(C(CN(c2ccccc2)C)=O)CCC2CCC(C1)N2C(=O)CCCC1CC1 C1(CNC(c2cc(C(=O)OC)sc2)=O)CC(C)N(C(c2cc(C(N)=O)no2)=O)C1 Cc1nc(N(C)C)sc1C(N1CC(C)(NC(=O)CC2CC(N(C)C)C2)C1)=O Cc1ccc(N)c(C(N2CCC(NC(=O)C(C)(C)C)C2c2ccccc2)=O)c1 c1(C(=O)NC2C(NC(CCC(N)=O)=O)CCOC2)cncc2cccnc12 N1(C(CCc2c(C)noc2Cl)=O)CC2=C(C1)CN(C(=O)C(C)C(O)C(C)C)C2 c1(NC(C2(CN)CCO2)=O)ccc(-c2cnco2)cc1 c1(C(=O)NCCCNC(Cc2cncc(C)c2)=O)ccc2cnccc2c1 c1(C(=O)NCCCCNC(COc2ccc(C)cc2)=O)nn(C)c2c1CCC2 C=CC1(C(=O)NCC2CC(NC(=O)C(CC(C)C)OC)C2)CCCCC1 c1(CC)nc(C)[nH]c1C(N1CCC(F)(CNC(=O)COCC2CCC2)C1)=O C=C(C)C1OCCC1C(N1CCC(F)(C(=O)N(CC)Cc2ccccn2)CC1)=O c1(OC)ncc(Cl)cc1C(N1CCC(CCNC(=O)CC2CCCCN2C)C1)=O c1(OCC(=O)NCC(C)N(C)C(c2csc(CC3CC3)n2)=O)ccc(O)cc1 C1(C(=O)NCC(C)(CO)NC(=O)Cc2n[nH]c(C)n2)(CC)CNC(=O)C1 c1(OCC)cc(C(N2CCCN(C(=O)CN3CCS(=O)CC3)CC2)=O)oc(=O)c1 c1(C(N2CC(C)C(CNC(C3COC(=O)O3)=O)CC2)=O)n[nH]c2c1CCSC2 CCC(C(=O)OC)C(=O)NCCCN1CCN(C(C2CNC(=O)O2)=O)CC1 N1(C(C=CC=CC)=O)CCCC(NC(C2CCCC2(C)C)=O)C1C N1(C(C2(COC)CCCO2)=O)CCOC2CN(C(C3(C#N)CCCC3)=O)CC12 Cn1cnc2[nH]c(C(N3C4CCC3CC(NC(=O)CCC(F)(F)F)C4)=O)cc12 C(=O)(CC(C)C(F)F)NCCN(CC(C)O)C(c1nc(C2CC2)ncc1Cl)=O S(=O)(=O)(c1ccc2nc(N3CCS(=O)C(C)(C)C3)cnc2c1)NCC(CCC)C C(CCC(C)(C)NC(c1cnc(OC)s1)=O)NC(CC=C)=O C1(C(=O)NCC2(C(=O)NC(C)Cc3ccnn3C)CC2)(N)CCCC1.C1CC1 C1(C(=O)NCCCCn2cc(C3CC=CCC3)nn2)CC2CCC(C1)O2 C1(C(=O)OC)C2CN(C(c3cnn(-c4ccc(F)cn4)c3)=O)CC12 CCCCC(C(=O)NC)NC(C1COCCN1C(=O)C(c1ccn(C)c1)C)=O c1(C(N2C(CNC(c3ccc(C)cc3)=O)C3CC3C2)=O)cc2sccc2n1C c1(C(=O)NCC2CC(NC(C(C)=C(CC)C)=O)C(O)C2)ccc([N+](=O)[O-])[nH]1 c1(CNC(=O)NC(C(c2ccccc2Br)OC)C)ccc(C)nc1O c1(NC(C2(C)CCN2C(=O)CCCCCBr)=O)cccc2c1CC(=O)N2 C1(NC(c2cc(CC)oc2C)=O)CCN(C(C2CCN2CC)=O)C(C)C1 N1(Cc2cn(CC(C)O)nn2)CCCC(NC(C2(C)CC2(Cl)Cl)=O)C1 CC1(C)CCC(CNC(c2cccnn2)=O)N(C(c2cnns2)=O)C1 c1(C(=O)NCC2CCCN2C(C2(c3cccnc3)CC2)=O)ccc2cc[nH]c2c1 Cc1ccc(C(N2CCC(N(C(=O)C#CC(C)(C)C)CCO)C2)=O)c(=O)n1C C1(CNC(C2(C)CC2(Br)Br)=O)CC(NC(=O)CNC=O)CC1O C1(C(=O)NC2(CC=C)CC2)CC(O)CN1C(=O)CC(C)SCC C1(C)(C(=O)NCC(CCOC)NC(=O)Cc2ccc(C)cc2C)CC2CCC1O2 c1(C(C)C2CC2)ncc2c(n1)CC1CCC2N1S(=O)(=O)C1CCN(C2CC2)C1 Cc1ccc(C(CNC(C2(F)CC=CC2)=O)NC(C2COCCO2)=O)cc1 Cc1nc(O)[nH]c1C(=O)NC1(C2CCCCN2C(=O)CC2C(C)(C)C2(C)C)CC1 C=CC(CC)C(=O)N1CCC(CN(C(=O)Cn2c(C)ccc2C)CC)CC1 C(=O)(C1=CCC2(COC2)OC1)N1CCOCC(CNC(CCCNC(C)=O)=O)C1 CC1CCCCC1C(=O)N(C1CCN(C(=O)CC(=O)Nc2nccs2)CC1)CC N1(C(c2c(C)n[nH]c2)=O)CC(NC(c2cccc(C(F)(F)F)c2C)=O)C(C)(C)C1 c1(C(=O)NCC(CNC(C2CCSC2)=O)C(F)(F)F)cnnc2ccccc12 c1(C(c2nc(-c3ccccc3)no2)N(C(COC2(C=C)COC2)=O)C)ccc(F)cc1 N1(C(C(c2cn(C)nc2)O)=O)CCN(CCNC(c2coc(CO)c2)=O)CC1 c1(NC(CC2(C)CC2)=O)cccc(SCC2CC2CNC(=O)COC(F)F)c1 c1(C(=O)NCCCNC(c2cnc(Cl)[nH]2)=O)cnnc(-c2ccccc2)c1 c1(C(N(C(c2ccccc2OC)C(=O)OCC)C)=O)ccc(SC)c([N+](=O)[O-])c1 C1(CC)(NC(=O)Cc2occc2C)CCN(C(C2(C(F)F)CCOCC2)=O)CC1 C=C(C)CCCNC(C1CCN(C(C2CC2NC(C)=O)=O)C1)=O N1(C(C2(OC)CC2)=O)CCCC(C2CCN(c3c(C#N)ccc(C)c3[N+](=O)[O-])C2)C1 c1cccc(C2COC2)c1.c1(C2(C(N3CC(CN(C)C)C3)=O)CC2)cn(C)nn1 C1(NC(c2c(C)ccn2C)=O)CN(C(=O)C2=COCCO2)CC1N=[N+]=[N-] c1(C(C(C)C)N(C(c2cc(CO)[nH]n2)C(=O)NCC2CCC2)C)cccc(Cl)c1 N1(C(=O)NCc2cc3n(c2)CCCC3)CC2CC3CC(C2)CC1C3 c1(CC)onc(C(=O)NCCc2cn(CCCCC(=O)O)nn2)c1C N1(C(C(C)(C)C(F)(F)F)=O)CCCC(C2CC2NC(=O)C2=CCCCO2)C1 c1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CC2)nc2sc(C)cn2c1C Cc1cncc(C(N2CCN(CCNc3ccc(C)[nH]3)CC2)=O)c1 c1(NC(C2(C)N(C(Cc3cccc(C)n3)=O)CC2)=O)ccc2c(Br)nn(C)c2c1 Cc1ccc(N)c(C(=O)N(CCCCNC(c2cnn3ncccc23)=O)C)c1F N(C1CCOc2ccccc21)C(C(C)OCCN=c1[nH]cc(C#N)o1)=O c1(C(N2CC3C(N(c4nccc(C(=O)OC)n4)C)C3C2)=O)ccc2ccnn2c1 C=C1CC2CC1CN2C(C12CN(C1)C2=O)=O.C1(C)(COC)CC(F)(F)C1 C12(CNC(c3ccn(CC)c3C)=O)CC(NC(=O)C3=CCSC3)(C1)C(C)O2 c1(C(=O)NCC(CN(C(CC(CCC)O)=O)C)O)c(F)ccc(Br)c1C Cc1ccc(C(CNC(=O)C(C)O)NC(=O)C(C)(C)c2ccno2)cc1 CCC(C)C(CC(=O)NCCc1ccnc(O)c1)NC(C1CC(=O)CS1)=O c1(C2C(=O)N2)ccc(Br)c(OC)c1.C(=O)(C(C)N(C1CCCC1)C)OC c1(C(=O)NC2(CO)CCN(C(CC(CC)C)=O)C2)ncc(C#N)cc1Cl C1(C(=O)NC(CC)C)C=CCN(C(c2cc(Cl)cn2C)=O)C1 Cc1ccc2c(c1)CCC(C(=O)NC(C)CNC(C13CC(F)(C1)C3)=O)O2 N1(C(C(C)(O)C2CC2)=O)CCN(C(=O)Cc2cccc(F)c2F)CC1CF C(C(CC(C)C)C(=O)O)NC(=O)NCc1c(OC)cc(F)cc1 N1(C(c2c(C)n(CC(C)C)nc2)=O)CCCCC12CN(C(=O)COCCCF)C2 C1(C(=O)NCCC2CN(C(c3cncc(C)n3)=O)C2)Cc2nccn2C1 C(CCCCCC(=O)NC(C)(C)CCF)NC(c1cc(C(C)C)[nH]n1)=O CC1(C(=O)NCC2CC2)CS(=O)(=O)C1.C12COCCN1C1CCCC1CNC2=O c1(-c2ccc(C(=O)NCC(C)N(C(C(CC)N(C)C)=O)CC)o2)ccccc1F C(=O)(C1=CC2CCCCCC12)N1CCC(CCNC(c2cccnn2)=O)CC1 C1(O)(C(=O)NC2CCC(NC(C3(CO)CC3)=O)CC2)CCCCCC1 CN1CCC(CN(C(=O)C(c2cnn(C)c2)NC(c2cc(CCO)on2)=O)C)C1 Cc1ncc(CC(=O)NCC2C(C)CCN2C(=O)CC2(C)CC(F)(F)C2)c(O)n1 C1(C#N)(C(=O)NCC(CC(C)C)NC(=O)C(C)C(C)O)CCCOC1 CC1CN(C(C2CCN(C)CC2)=O)CC1CNC(c1ccc(-c2cccs2)o1)=O N1(C(c2c(C)[nH][nH]c2=N)=O)CCC2(C1)CN(C(c1ncsc1C1CC1)=O)C2 N1(C(C(CC(=C)C)C)=O)CCC2(CCC2NC(=O)CC2=CCCCC2)CC1 S(=O)(=O)(c1ccc(NCC(C)OC(C)(C)C)c(C#N)c1)N1CC(C)SC1 c1(C(=O)NCCOC2CN(C(CCC(C)OC)=O)C2)cc(C)cc2ccncc12 c1(C(=O)NC2CC(CNC(C3(C)CCCC3(F)F)=O)C2)ccc2c(c1)CNC2=O S(=O)(=O)(c1ccccn1)N1CC(CNC(c2cc(OC)c(O)cc2)=O)OCC1 Cc1cc(C)c(CN(C=O)C(c2ccc3nnnn3c2)=O)c(C)c1 CCC(C)(C)COC.N12CCC1C2NC(C1CN(C(=O)OC(C)(C)C)C1)=O c1(C(N(CC(C)NC(C)=O)C)=O)c(Cl)ccc(Cl)c1O C1(O)(CNC(CSCCC)=O)CCN(C(=O)C(n2ccc(C3CC3)n2)C)C1 c1(CCC)ccc(NC(=O)C(c2ccco2)NC(C2CC3CC3C2)=O)cc1 c1(CC(=O)NC(CNC(c2c(OCC)ccc(C)c2)=O)C)cn2c(C)csc2n1 C1(CC(=O)NCCC2CCN(C(=O)Cc3cc[nH]n3)CC2)CCCC2(CCC2)O1 c1(NC(CN(CCCNC(C2CC(OC)(OC)C2)=O)C)=O)ccccc1CO C1(NC(C(CCNC(c2ccn(C(C)C)n2)=O)OC)=O)CN(C)CCN(C)C1 CC#CCC(C(=O)NCC1CC[Si](C)(C)C1)NC(=O)C=Cc1cc[nH]n1 C1(C(N2CC(COC)C2)=O)C2CC3C(C2NC(C2(C(C)(F)F)CC2)=O)C13 C1(CC(N2CC(C)(CC(=O)NCC(C(C)C)O)C2)=O)CCCOCC1 Cc1cc(Cl)c(Cl)cc1C(N1CCN(C(=O)Cc2ccc(F)c(Br)c2)C2CC12)=O Cn1nc(C(=O)NCCC(O)CNC(C2(F)CCCOC2)=O)cc1Cl N=c1nc(O)cc(C2CCN(C(C3CC3C(=O)Nn3cccn3)=O)CC2)[nH]1 N1(C(c2occ(C)c2C)=O)C(CNC(c2coc(Cl)n2)=O)CC2CCCC12 N1(C(Cn2nc(C)c(Cl)c2)=O)CC23CCCCC2(C1)CN(C(C1CC12CC2)=O)C3 N#Cc1cccc(CCNCC(c2ccccc2Cl)O)n1 c1(CNC(CCNC(CCCC#N)=O)=O)ccc([N+](=O)[O-])o1 C1(C(=O)NCC2N(C(CC3CCC(OC)CC3)=O)CC2)Cc2cscc2C1 C1(NC(C(C)OCCC#C)=O)CC(C)(CNC(c2ccccn2)=O)C1 C1(C(C)C)CN(C(c2ccoc2C2CC2)=O)CCC1NC(=O)C(=O)C(F)(F)F Cn1c(C(=O)NC2CCC2NC(=O)C(F)n2ccnc2)ccc1C#N C=CCCC(C(=O)N1CCN(C(C)=O)CC1)NC(C1CC(F)(F)C1)=O C1(CCN(C)C)CN(Cc2nnc(-c3cccc(-n4cccn4)c3)o2)CCCO1 C1(CCC)CN(C(=O)CCC2CC2(F)F)CCN1C(=O)Cc1nnc(C)o1 CC(C(=O)NC1CN(C(c2cc(-c3cccnc3)n(C)n2)=O)CC1O)C(F)F Cc1nn(C)c(Cl)c1C=CC(=O)NCC1CCN(C(c2ccccn2)=O)C1(C)C c1(C(N(C2CN(C(C(C)OCCC=C)=O)CC2(C)C)C)=O)ccnc2[nH]nnc12 N1(C(=O)CC2CCN(C(C3CCCC(C4CC4)O3)=O)C2)CCOC2(CC2)C1 N1(C(C(C)NC(=O)NC)=O)CCCC(NC(=O)CC2CCOCC2)CC1 c1(NCc2ccc(C(=O)O)cc2F)cnc2cccnn12.N12CC3CC3(C1)C2=O N1(C(CC2CCN(C)CC2)=O)CCCC2(CCCCN2C(C2CCN(C)C2)=O)C1 C1(C(=O)OC)CCCCN1CCNC(C(C)(C)NC(=O)OC(C)(C)C)=O N1(C(C(C)N(C(C(CCC)OCC)=O)CCC)=O)CCC(C)(CSC)CC1 Cc1cccc(C)c1CN(CC(C)C#N)C(c1cccc(I)c1)=O C1(NCCN2CCC(C(=O)NC(c3ccccc3Cl)C)C2)CC(=O)N(CCN)C1 c1(C(=O)OCC)cc(CNCCCN2CCCCC2C2CC2)nn1C C1(C(=O)OC)CC(F)(F)CC1C(=O)N(C1CCCN(C(=O)C=C2CCCC2)C1)C CC(CN(C)C(c1coc(C(C)NC(c2ccnnc2)=O)n1)=O)C(C)(C)C C=Cn1ncc(C(N2C(C(=O)OC)CC2C)=O)c1N.C12(CC1)CC(=O)NC2 Cc1ccc(CC(=O)NC(C)C(C)NC(=O)C(C(C)C)N2CCCC2=O)c(C)c1 c1(C(=O)NCCCC)cc(-c2csc(NC(=O)CC3CCCC3C)c2)ccc1F C1(S(C)(=O)=O)(C(=O)NC(CCCNC(CC(C)C)=O)C)CCCCC1 C12(NC(c3[nH]cc(C(C)=O)c3)=O)CCCC1CN(C(=O)CC1CNC(=O)O1)C2 C1(O)(C(C)NC(=O)CSc2n[nH]c(O)n2)CCN(C(=O)CC2COC(=O)C2)C1 C1(NC(C2C(NC(c3c(NCC)scn3)=O)C2)=O)CCCC(F)(F)C1 C1(C(C)C)CCN(C(=O)CN(C)C)C(CNC(=O)CCc2ccc(F)nc2)C1 c1(NC(C2OCCN(Cc3scc(C)c3)C2)=O)ccc(C(N)=O)c(F)c1 N1(C(C(COC)(F)F)=O)CCC(CO)(CNC(=O)CCc2nncs2)CC1 c1(-n2c(C(F)Cc3ccccc3)nc(C(CC)O)n2)ccc(S(N)(=O)=O)cc1 c1(CC)cc(CC)nc(NC2(CNC(=O)C(CC)OC)CCCCC2)n1 N#CC1(C(=O)NCc2cc(C(=O)NCc3ccsc3)co2)CC(=O)C1 C1(OC)CN(C(c2cncs2)=O)C(C)(CNC(=O)CC#N)C1 CN1CCC2(CN(C(c3cnn(CC(F)F)c3)C(=O)NC3CC3)CCO2)C1 C1(O)(C(C)C)CCC(NC(c2cnn(C3CC3)c2Cl)=O)C1 C(C(=O)N1CCCC(CNC(=O)Cn2ccccc2=O)C1)(C(C)C)OC C1(NC(C(C2CC(N=[N+]=[N-])C2)N2C(C(C)(C)C(C)CCl)CCC2)=O)CN2CCC1(C)CC2 C1(CC)CN(C(=O)Cc2c(Cl)cnn2C)CCN1C(=O)C(CO)c1ccccc1 N1(C(C2(C)CC2(F)F)=O)CCC(NC(=O)Cc2cc[nH]n2)C(O)C1 C(=O)(C#CC1CCOC1)NCc1c(C2CN(C(C3(SC)CC3)=O)C2)ocn1 C(=O)(C(C)(C)C1CCC1)NS(CC)(=O)=O.C(=O)(CC1(CO)CC1)NCCN C1(NC(C2CCN(CC#C)CC2)=O)CC(O)CN(C(=O)C(COC)NC(C)=O)C1 C1(C(N2CCC(N(C(c3nnc(O)cc3C)=O)CC)C2)=O)CN2CCCC2CO1 CCC(CC)C(F)C(=O)N1CCC(F)(C(N2CC(CO)CC(C)(C)C2)=O)CC1 c1(CCC(=O)NCCCCCCNC(C=C(C)C(C)C)=O)ccc2[nH]ccc2c1 C=CC1COCCN1C(=O)CC1CCCC1NC(C1CCCC1)=O CCC(C)C(O)C(=O)NCc1ccc(C(=O)N(C)CCC2CCCN2C)o1 Cc1cc(C(N2CC(CNC(c3cncnc3)=O)C2)=O)c(Br)cc1F c1(C(C)(C)CSC2CCCC2NCCn2cc(C34CC(C3)C4)nn2)ccccc1F Cc1cnc(C=CC(=O)NC2CC(N(C(=O)CCN3CCC3)C)C2)[nH]1 N1(C(c2ccon2)=O)CC(F)(F)CC1CNC(C1(c2ccccc2)CCOC1)=O C1(NC(c2ccc(OC)nc2)=O)CC2CC(CN3CCCCC3)CC12 C(CCC(C(=O)N(c1csnc1OCC)C)NC(c1cnn(C2CC2)c1)=O)OC CCC(CC(=O)NC(C12CCC(CC1)C2)CNC(=O)CN(C)C)NC(=O)CSC N1(C(c2cc(CC)no2)=O)CC(CNC(=O)CCc2cnc(O)[nH]2)C(C)C1 C(CNC(=O)CCC1CCCCCC1)(CC(F)(F)F)NC(CN(C)C(N)=O)=O CC(CCNC(=O)CC1(C)CCCO1)CCNC(c1coc(Br)n1)=O C1(CN(C(=O)C(CCC2CCC2)NC(=O)OC(C)(C)C)C)CCC2(CCC2)O1 N1(C(CSc2n(C)cnn2)=O)CCC(NC(c2csc(CO)n2)=O)C(F)C1 N1(C(C2CC(OCC)C2)=O)CCC(N(C(=O)CCN2CCC2)CC(C)C)CC1 CCC(C)N=c1[nH]c2c(c(=NCc3ccccc3-c3cnn(C)c3)[nH]1)CCC2 c1(NC(C)=O)cc(C(=O)NC23CCN(C(C4CC45CC5)=O)CC2C3)ccc1C C1(NC(=O)NCC2=NOC(C)C2)CCCN(Cc2ccccc2)C1C C1(CC(=O)OC(C)(C)C)(NC(C)CCC2CCCO2)CCOC1 c1(C(N2CCCC(C)(NC(C(C(C)(C)C)SC)=O)C2)=O)cnn2c1NCC(C)C2 C1(NC(c2ccc(OCOC)cc2)c2nnnn2C(C)(C)C)COCC(C)(C)O1 C1(NC(CC(C)N(C)C)=O)CCCCC1NC(=O)Cc1cnco1 C=C(Cl)CC(C(=O)NCC1(COC)CCCC1)NC(=O)C(C)CO N1(C(CC(=C)C)=O)C2CCCC1CN(C(c1cccnc1NC(C)C)=O)C2 C1(N(C)C(c2cccnc2O)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1 N=C1NC(=O)C(CC(N2CC3C(CNC(=O)CC4(c5ccon5)CC4)C3C2)=O)S1 C1(N(C(Cc2cnc(C)o2)=O)C)CCCCN(C(C2CN3CCC2CC3)=O)C1 c1(C(=O)NCC(C)(CNC(c2cnn3ccsc23)=O)OC)nc2ccccc2[nH]1 N1(C(CSC)=O)CC2(CC(C(N3CCC4C(C(N)=O)C4C3)=O)CO2)C1 C1(C(=O)NC(C2CCN(C(C(CC=C)(F)F)=O)C2)(C)C)CCc2ncncc2C1 N1(C(C2C(CCOC)C2)=O)CCC2C(C(=O)N(C3CC3C)C)C2C1 C1(OC)CCn2cc(C(=O)NC(CNC(=O)C=Cc3nccs3)C(C)C)nc2C1 CC1CCCC(C)N1C(=O)COC(C1CCCN1C)=O N1(C(c2c(CC)n(C)cc2)=O)CC2CC(C1)N2C(C1(CC2CC2)CCC1)=O c1(C(C)(C)NC(CC2CC(NC(=O)OC)C2)=O)nnc(N)o1 C(CCCCNC(=O)Cc1cnc[nH]1)N(C(=O)CSCc1ccccc1)C O=C(CS(=O)(=O)C1CC1)N1CCC2(NC(=O)CNC(C3CCC3)=O)CC2C1 C1(NC(C2C(CNC(C)=O)CCC2)=O)CCC(NC(=O)CC(O)CC2CC2)CC1 N1(C(c2c(OC)cncc2)=O)C2CCC1C(CNC(c1cc(C)nc(O)n1)=O)C2 Cc1cc(-c2ccccc2F)nnc1N1CC(CCO)C(CCO)C1 c1(OC)ccc2c(n1)NC(C(N1CCC(CNC(c3ccc(F)cn3)=O)C1)=O)C2 C1(CN(C)C(c2ccccn2)=O)C2CC(CC2F)N1C(=O)C(c1cccn1C)=O C(CC(C)(C)CC(=O)NCC(N1CC1CO)=O)OC C1(C(=O)NC(CN(C)C(c2cccc(O)n2)=O)(C)C)CCCCN1CC(F)F C(C(C)(C)CC(=O)N(C(CO)C(C)C)C)NC(C(COC)OC)=O C#Cc1ccc(C(N2CC(N(C(=O)Cc3ccc(F)cn3)C)C(F)C2)=O)cc1F C1(COC)CN(C(C2CCCC2NC(=O)C=NOC)=O)CCO1 C1(C(=O)NCC)CC2CCC1N(C(=O)CCc1ccccc1C#N)C2 c1(CC)ccc(CC(=O)N(CC(O)CN(C(=O)C(C(C)OC)N(C)C)C)C)cc1 C1(C(=O)NC2CC(C)(NC(c3ccncc3C(F)F)=O)C2)CCc2nc[nH]c2C1 C(=O)(CCCC(C)(C)C)NC12C(CN(C(C(C)(c3ccccc3)N(C)C)=O)C1)C2 N1(C(C(CCC)C)=O)CCC2(CCOCC2)C(NC(=O)C(CC(C)C)OC)C1 N(C(=NCCC(=O)N(C)C)N1CCC(CS(C)(=O)=O)C1)C(CC)C c1(C(=O)NCC23C(CN(C(CC(C)C)=O)C2)C3)cc([N+](=O)[O-])c(Cl)cc1F C(=O)(C1=NOC(CNC(c2cccc[n+]2[O-])=O)C1)N(CC(C)(C)O)CC N1(C(C(C=C)OC)=O)CCC12CN(C(=O)CC1CCCN1C)C2 CCCS(=O)(=O)CC(=O)N1CC2CCOC2(CNC(C2CC2(C)C)=O)C1 C(c1ccncc1)=C(C)C(=O)NCC1CN(C(c2oncc2C)=O)C2CC12 N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(C2C3CCN2CC3)=O)CC(C)(C)C1 C[Si](C)(C)c1cccc(-c2ccc(C(=O)Nc3cc4sccn4c3)c(F)c2)c1 c1(CC(=O)NCC2CCC(NC(=O)C(F)=C3CCCC3)C2)ccc(F)c(Cl)c1F c1(NC(=O)Nc2c(N3CCN(C)CC3)ccc(F)c2)cc2ccc(O)nc2s1 O=C(C1=CCCCCC1)NC1CC12CCCN(C(=O)C(Cl)=CCl)C2 c1(C(=O)NCC(C)CNC(=O)CCCCCF)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCC2C(C)CCN2C(C2C3(CC3)C23CC3)=O)nc2cc(O)ccc2[nH]1 c1(C(N(CCC(C)NC(c2cn(CC)nn2)=O)C)=O)cccc(N)n1 C1(NC(c2ccc(CC)cc2)=O)CCN(C(c2csc(CC)n2)=O)CC1O CCC(C(F)(F)F)NC(CC(C)C1CCCC1)c1nnnn1C1CCCCC1 c1(NC(=O)NCC(CC)(C)c2ccccc2)ccc(F)c(OCCN(C)C)c1 C(C1=CCCN(C(=O)C(=Cc2ccccc2)C)C1)NC(CN(C(C)=O)C)=O C1(CNc2[nH]cc(C(C)(C)C)n2)CN(C(=O)CCCCn2ccnn2)CCO1 c1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CCC2)cnc(OC)cn1 Cc1cnccc1C(C)C(=O)NC(CNC(c1ccc(CSC)o1)=O)C1CC1 C1(C(=O)Nc2n(C)nnn2)COc2ccc(-c3ccc4c(c3)NCCO4)cc2C1 c1(C(N2C3(CNC(CN=S(C)(C)=O)=O)CCCC(C2)C3)=O)ccnc2ccccc12 C1(CC)CCC(C)N(C(C23CC(N)(C2)C(C)O3)=O)C1 C1(C(=O)NC(C=C)(C)C)CN(C(C2CC23CCOCC3)=O)CC12CCC2 c1(OC)ccc2cc(NC(=O)NC(C)Cc3cnccn3)ccc2c1 C=CC(C)(O)C(=O)NC1CCCC(NC(=O)C(F)(F)C2CC2)C1 C(c1cccc(O)c1)=CC(=O)NCC1(O)CCN(C(=O)C(F)=CC2CC2)C1 C1(NC(CC(=O)NCC)=O)(CO)CCCN(C(C2CSCCS2)=O)C1 C(=O)(C#CC1CCCO1)N1CCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 c1(C(=O)NC2CN(C(C(CNC(C)=O)(C)C)=O)CC2(C)C)ccc2cncn2c1 c1(CC(N2C(CNC(CN(CC)CC)=O)CC(C)(C)C2)=O)noc2ccccc12 c1(C(N(C2CCCC2)CCCNC(C=CCCC)=O)=O)cc(CSC)on1 N#CC1=C(C(=O)NCCOCCNC(c2cnc(O)c(Cl)c2)=O)CCC1 C1(NC(C2(C(C)(F)F)CC2)=O)COCC1n1cc(C(C2CC2)C2CC2)nn1 c1(C(=O)NC(N2CC(CO)CC(C)C2)=O)ccc2cccnc2c1 C1(CC#C)(C(=O)N(C)CCN(C)C(C2CN(C3CCC3)C2)=O)CCOC1 N1(C(=O)OC(C)(C)C)CC2C(COC(C3CC(O)(c4ccncc4)C3)=O)C2C1 CCC(CC(=O)N1CC=CC1(C)C(=O)NCC1(O)CC(C)(C)C1)C(C)C n1(CCOC)nc(-c2ccc(F)cc2)nc1-c1ccc(CC(C)C)cn1 C1(NC(c2c(OCC)ccs2)=O)CC(NC(C2CC=CCC2)=O)CC1O N1(C(C2(C(C)C)CCN(C(=O)C(C3CC3)C3CC3)C2)=O)CC(CO)OCC1C CCCN=C(NCC(C)CNS(C)(=O)=O)NCc1cc(C)on1 N1(C(C23CN(C(CCC(C)SC)=O)C(C2)CO3)=O)CC2(CCC(O)CC2)C1 Cc1cc(C(=O)NCC2CN(C(C3CCCCS3)=O)CCO2)c(C)nc1C c1(C(=O)NCCC(C)N(C(=O)C(C)CC(F)F)C)cnc2sccn12 CCCCCCCC(=O)N1CC(O)CCC1C(=O)NCc1nnc(O)n1CC c1(CC)cc(C(=O)NC(Cc2cn[nH]c2)C(N2CCOC(C)C2)=O)nn1C C=CCCCC(=O)NCCC1CCCN1C(c1cc(Cc2ccccc2)c[nH]1)=O N1(C(C2CCCN(C(C)=O)C2)=O)CCOCC(C)(CNC(=O)Cc2ccco2)C1 N1(C(C2C(=C)C2)=O)CCCC(CNC(c2ccc(CC(C)C)cc2)=O)C1 C1(NC(=O)CONC(=O)C2CC(OC3CCC3)C2)CC2CCCC2C1 N1(C(C(CC=C)CC)=O)CCC2C1CCCN2C(=O)CNC(=O)NC C(=O)(C1CCCc2ncnn21)N1CCC(NC(C)=O)CC1 C1(C(C)C)(C(=O)NC(CCO)C(C)C)CCCN1C(c1csnn1)=O N1(C(C2C(C)C2)=O)CC=C(CNC(=O)C(CN2CCCC2)c2ccccc2)CC1 c1(C(=O)NC(C2OCCN(C(c3scc(OC)c3)=O)C2)C)ccc(S(N)(=O)=O)o1 C1(NC(c2cn(CCO)nn2)=O)CC2(CCN(C(=O)C=C3CCSCC3)CC2)C1 CC(C)(CC1CCOC1)C(=O)NCCC1(O)CCN(C(=O)C=Cc2cc[nH]n2)C1 C1(F)(NC(=O)OCC)CCN(N2CCn3c(cnc3-c3ccccc3)C2)CC1 C12(CC)CN(C1)C2=O.c1(CNC(C(CC2CC2)NC(=O)OC)=O)ccccc1 c1(NCc2ccc(CNC(c3cc(CC)n(C)n3)=O)cc2)ncnc2scnc12 N1(C(c2cc(C)oc2C)=O)CCc2ccccc2C1CNC(c1cn[nH]c1)=O C(C)(C(=O)NCC1(NC(=O)CCc2ncccc2C)CCCCC1)(C(C)C)OC Cc1nn(C)c(Cl)c1C(=O)COCCSc1ccc(Br)cc1 CC1CCC(NC(N2CCC(Cc3ccnn3C)CC2)=O)c2ccccc21 N1(C(c2c(C)nccc2)=O)CC2ON=C(CNC(C3(CC4CC4)CC3)=O)C2C1 C(c1cccc(Br)c1)=CC(=O)OC1C(SCCOCC)CCC(C)C1 Cc1cc(C)c(C(=O)NC2(C(=O)NC(CO)CC(C)(C)C)CC(F)C2)cn1 c1(C(C2CC2)NC(C2N(C(C(CC)C)=O)CSC2)=O)ccccc1COC c1(C(=O)NCCN(C)C(c2cc[nH]c2)=O)n[nH]c(C2CC2)c1Cl Cc1ccc(COC(C)C(N2CCC(n3cc(C(O)C4CC4)nn3)C2)=O)cc1 c1(CNC(Cn2c(C)cc(C)n2)=O)cc(O)nc(CNC(=O)C(C)NC(N)=O)n1 C1(CNC(C2(N)C(C)(C)C2)=O)CS(=O)(=O)CCO1 CC(C)CC(O)C(C)C(=O)NCCC1(C(N2CCC(O)C(C)(O)C2)=O)CCCC1 c1(C(N2C(CNC(CN(C(C)=O)C)=O)CCC2)=O)cnc(C(C)(C)C)nc1C N1(C(COC)=O)CC(C)CN(C(c2ccc3nc[nH]c3c2)=O)CC1C N1(C(CC(=O)OC)=O)CC2CC2(C(=O)N(C(C)CO)C2CC2)C1 c1(C(N2CCN(C(C(C=CC)O)=O)CC2COC)=O)cnc(O)c2ccccc12 CC1CN(C2CCC2)CC1(c1nnnn1C1CCCC1)Nc1c(Cl)nsc1Cl c1(C(=O)NCC=CCNC(C(CC)n2nccc2C)=O)cc(SC)ccc1C C(=O)(C(O)CCCC)N1C(C(N2C(CC#C)COCC2)=O)CSCC1 c1(C(=O)NC2CCN(CC(=O)NCC(C)(C)OC)CC2)ccc(C)nc1C C1(NC(c2ccc(SC3C(C)C3)cc2)=O)CC2CC1CN(C(c1cccs1)=O)C2 N1(C(C(C(C)C)NC(C2N(CCC)CCC2)=O)=O)CCCCCCC1CC Cc1c(NC(C)CS(N)(=O)=O)ncnc1N1CCN2C(=O)CC12 c1(OC)cc(CC(N2CCC(C)(CNC(=O)CS(C)(=O)=O)C2)=O)cc(OC)c1O C(=O)(C1=CCC2(COC2)OC1)N(CCCN(C)C(c1ccnn1C(F)F)=O)C c1(CNC(c2cc(CC)oc2C)=O)ccc(CNC(C2(C)CC(C)C2)=O)c(F)c1 CC#CCC(C)N=c1nc(N2CC3C(C2)C3(F)F)c2c([nH]1)CCC(C)C2 C12(CCNC(c3ccc(CC)s3)=O)CCC(C1)N(C(C1CCOC(C)(C)C1)=O)C2 C(C)(CNC(=O)C1=CCOC1)(CC(C)C)NC(C(CCSC)NC(C)=O)=O C1(CNC(=O)Cn2cccn2)CC2CCC1N(C(c1ccc(CO)o1)=O)C2 N1(C(COCCCCC)=O)CCC2CN(C(C3CCOC(C)C3)=O)C(C)C12 C1(CC(N2C3C(CNC(Cn4nc(C)oc4=O)=O)C(C3)C2)=O)CCC(C)(C)CO1 C1(NC(c2cnc(Cl)c(Cl)c2)=O)CN(Cc2cc(O)c(F)c(F)c2)CCC1(F)F c1(NCC2(NC(C3CC4C=CC3C4)=O)C(C)CCCC2)ncnc(Cl)c1[N+](=O)[O-] n1(CCC)nccc1C(=O)N(CCC(=O)N(CC(C)C(C)C)C)C1CC1 C(=O)(C(C)CC1CC1)N(CC(=O)NC(c1ncc[nH]1)CC)CC1CC1 C1(NC(C2CC(NC(c3cc[n+]([O-])cc3)=O)C2)=O)CC2CC3C(C2)C13 C1(CC)CN(C(C2(C)CCCS2(=O)=O)=O)CC(C)N1 C1(C#N)(c2nc(NC(c3ccnc(SC(C)(C)C)n3)=O)sc2)CCOCC1 O=C1CCC(CC(N2CCCC2CN(C(=O)C2=NOCC2)C2CC2)=O)CN1 C(CC1CC1)(C(=O)N1CCCC1CC1CC1)NC(CC1CC(=C)C1)=O CC1CCc2[nH]c(C(=O)NC(C)CNC(=O)COCC3CCCO3)cc2C1 Cc1ccc(O)c(C(N2C3CCC2C(C(=O)NC2(C)CCC(C)C2)C3)=O)c1 N1(C(C2CCC(C3CC3)CC2)=O)CCC2OCCN(C(=O)COCC3CC3)C2C1 n1(CCCC)ncc(C(=O)NCCN(CC(C)O)C(c2occ(C)c2C)=O)c1C N1(C(C)=O)CCCC(NC(=O)C(Cn2ccnn2)NC(c2coc(C(N)=O)c2)=O)C1 C1(CC)(NC(=O)CC2CCCCN2C(c2cnn(C(C)C)c2)=O)CCCCC1 CCCCC(CC(=O)N1CCC(C)(CC)CC1)NC(c1coc(C)n1)=O C(CC(C)(C)C(=O)Nc1ccccc1F)NC(C(C)n1cccn1)=O C12CCN(CC1O)C(=O)CCc1nc(no1)CC(=O)N2.C1(O)(C(C)C)CCC1 N1(C(C2CN(CCC)C(=O)C2)=O)CC(CO)C2(C1)CN(C(=O)Cn1ccnn1)C2 C=CC1CCCN(C(c2cccc(C(c3ccccc3)=O)c2)=O)C1 C(=O)(C(C)CCCC)NC(CNC(C1(C=C)CCC1)=O)C1CC1 C#CC(CC(C)(C)C)NC(=O)CC(C(C)C)NC(C1(O)CCCCCC1)=O N1(C(C(C)S(N)(=O)=O)=O)CCC(CNC(=O)CCC(F)F)C(F)(F)CC1 Cc1cc(C(=O)NCC2CCCCC2NC(C2(F)CCS(=O)(=O)C2)=O)ccc1N c1(C(=O)NCC=CCNC(C2C(CC)C2)=O)ccc([N+](=O)[O-])cc1C(F)(F)F c1(CC(=O)Nc2cccc(-c3ccco3)n2)cn2cc(-c3cccs3)ccc2n1 C1(NC(=O)C=CI)CC(N=c2[nH]nc(-c3ccccc3)s2)C12CCOCC2 N1(C(C(CC)CC)=O)CCN(C(=O)Cn2[nH]cnc2=N)CC2CCCCC12 CC(c1ccccc1C)=CC(=O)N(C1CC(NC(=O)CCc2nncs2)C1)C c1(SCCC(=O)NC(C(C)NC(CCCC)=O)CO)ccc(F)cc1F Cn1ncc2cc(CN3CCC(NC(=O)C(=O)NCC(F)F)C3)cnc12 N1(C(=O)CC2CCN(c3c(F)cnc(C)n3)CCC2CO)Cc2ccccc2C1 c1(NCC2CCC(C)C2)ccc(S(=O)(=O)N(C)Cc2ccnn2C)cn1 N1(C(c2c(CC)csc2)=O)CCN(C(=O)CC2CCN(C)CC2)CC1CC(F)F C1(C2CCN(C)CC2)(C(=O)NCCCN(C(=O)CCCC(C)(C)C)C)CC1 N1(C(C(CC=C)CC)=O)CCC(C)(C)C(C=O)C1.N1(CC)CCC1 c1(CC)cc(C(=O)NCC2CCCN2C(C2CC23CCOC3)=O)c2c(c1)CCO2 C(CCC(C)C)(C(=O)N1CC2(CCC2)CC1CNC(=O)C(F)(F)CO)NC(C)=O N1(C(c2cn(C3C(OCC)COC3)nn2)=O)CCN(CCC(Cl)Cl)CC1 CCC(CC(=O)NCC1(NC(C2(CO)CCCCC2)=O)CCC1)OC C(=O)(CC(=O)NC(C(=O)NCC(F)C1CCC1)c1cccs1)OC c1(OC)ccc(C(=O)NCC2(O)CCCN(C(=O)C(C)n3ccnc3)C2)c(Cl)c1 C(CCC(=O)N(C)CC=CC(N1CCC(CC2CC2)C1)=O)=C(C)C C1(C#CC(=O)N(CCC(C)NC(c2cc[n+]([O-])cc2)=O)C)(CC)COC1 c1(N(C(=O)C2=CCC2)C)ccnc(-n2cncn2)c1.C12CCCN1C2=O c1(C(C(N2CCCC(c3cn(CC(=O)OC)nn3)C2)=O)C)ccc(F)c(OC)c1 c1(C(=O)OC)cc(CCC(=O)NC(C(C)(C)C)c2cccs2)c[nH]1 c1(C(=O)NC(CC(C)NC(c2cccc(OC)c2N)=O)C)ccc2c(n1)CCC2 Cn1nc(CC(=O)NC2CCC(NC(c3csc(C#N)c3)=O)C2)cc1Cl N1(C(c2cnn(CC)c2Cl)=O)CCN(C(=O)CC(C)(C)C#N)CC2CCCCC12 C(=O)(C(CC(C)CC)NC(=O)Cn1nc(C)cc1C)N1CCC(C=C)C1 C1(NC(c2scnc2Cl)=O)CC(F)CN(C(=O)CCc2cnc[nH]2)C1 C1(C(=O)NC(c2cccs2)C)CC(C)(C)CCN1C(c1cnn[nH]1)=O c1(OC)cc(F)c(CC(N2CC(NC(C3CCCCC3)=O)C(O)C2)=O)c(F)c1 CC1C(NC(c2cccnc2N2CCCC2)=O)CCN1C(=O)C(=O)NCC(F)F C(=O)(C1=CC(C)CC1)NC(CNC(C(c1ccccc1O)OC)=O)(C)C c1(C(=O)NCC2CN(C(CCc3cnc(C)o3)=O)C2)cncnc1C1CC1 CC1(C)C(CO)CN1C(=O)CSCCNC(C1CC(F)C1)=O CC1CC(NC(c2cc(N3CCCC3)ccn2)=O)CN(Cc2ccccc2F)C1 CC(C(=O)NC1(CCC(=O)N(CC(Cl)Cl)C)CCC1)NC(=O)C1CC1 C1(NC(c2c(C)cns2)=O)CCN(C(C2CCSC2)=O)C1(C)C N1(C(CS(CC)=O)=O)CCN(C(=O)CCCOc2ccc(Cl)c(C)c2)C(CO)C1 c1(C(=O)NC2CC(NC(C3CC(C)C3)=O)C2)c[nH]c2ccc(Br)cc12 N1(C(c2cncc(N(C)C)n2)=O)CC2(C1)CN(C(C1CC1c1ccc(Cl)s1)=O)C2 CCCC(C(=O)NC1C=CC(CNC(c2nccnc2C(F)(F)F)=O)C1)OC N1(C(CC(CCC)O)=O)C2CCCC1CN(C(c1c[nH]nc1C(F)F)=O)C2 C1(C(N(CCCSC)C)=O)CC12CCN(C(c1ccc(C)nc1C)=O)C2 C1(C2CC2)(CNC(c2cc(OC)nn2C)=O)CCN(C(=O)CC(C)C2CC2)C1 c1(C(N2CCC(C)(NC(C(CC)SC)=O)C2)=O)cc(C)c2c(O)nc(O)nc2n1 C1(CCNC(=O)CC2CCCO2)CCCN(C(=O)C=Cc2ncc[nH]2)CC1 C1(NC(c2cnc3sccn23)c2n(CCOC)nnn2)CCCCC12CCC2 C(=O)(CCC(=O)NCC(C)(F)CNC(c1nnc(S)n1C)=O)N(C)C N1(C(c2cc(C(C)C)no2)=O)CCN(C(C2(C)C=CCCC2)=O)CC(O)C1 Oc1nnc2n1CCN(CC(c1cccc(F)c1)NCc1ccccc1)C2 C1(N(C(c2ncc(C)nc2)=O)C)CCCN(C(=O)Cc2nc(C)c(C)s2)CC1 N1(C(C2(CC#C)CCCCC2)=O)CCCC2(NC(c3cncc(C)c3)=O)CC2C1 c1(NC2CN(C(C3(COC)CC=CC3)=O)CC2C)nc(C)nc2n[nH]cc12 Cc1cc(C(=O)NC2C3CN(C(=O)CN4CCCCC4)CC23)c2ncccc2c1 CC1CCC(C(=O)O)N(C(C2CN(c3ccc(C#N)cn3)C2)=O)C1 Cc1ccc(CC(=O)N(C)CC2CCN(C(c3nscc3C)=O)CC2)c(F)c1 O=C1CC(NC(=O)CCCCc2cn(C3CCS(=O)(=O)C3)nn2)CCCN1 NC(=O)CCC(=O)N1CCC(NC(=O)C=CCOC2CCOCC2)C1 c1(C(N(C2CCCC(NC(c3ccc(CC)[nH]3)=O)C2)C)=O)cc(N)nc(Br)c1 C(=O)(CCCCCC(=O)NC1C=CC(CNC(=O)C(C(C)O)N(C)C)C1)OCC C(C1CCOCC1)=CC(=O)N(CC(C(=O)NC(CCC)c1ccco1)C)C1CC1 CC1CC(CNC(=O)Cc2ccc(CO)cc2)CN1C(c1cccc(Cl)c1)=O S(=O)(=O)(c1c[nH]ccc1=NC1CC(N)CC1(C)C)N(CCN(CCN(C)C)C)C c1(OC)cc(Cl)c(C(N2CC3CCC(C2)N3C(C2CC2C2CC2)=O)=O)cc1OC N1(C(CC2CC(C)(C)C2)=O)CC(NC(=O)CC2CC(=O)NC(=O)C2)CC12CCC2 C1(C)(C(=O)NC2CCC(CNC(C(C)OC3COC3)=O)C2)CC(F)(F)C1 Cc1ncnc(C)c1CC(=O)NCC(=O)NCC1C=CCOC1 C1(O)(COC)CCN(C(c2n[nH]c(C)n2)C(=O)NCC2CCCO2)C1 c1(OC)ccc(OCC(=O)NC2(C3CCCN3C(=O)C(C)CN(C)C)CC2)cc1 CC1(CNC(C2(C)CC2Br)=O)CCCN(C(C2CC(=O)N2)=O)C1 c1(C(=O)NC2C(CNC(c3cc(C)cc(Cl)c3)=O)CCC2)c[nH]c2nccc-2c1.C C1(NC(C(C(CC)O)C)=O)CN(C(c2cc(C3CC3)ncn2)=O)CC(C)(C)C1 N1(CC)CC(NC(c2conc2CNC(=O)CC2CCCC(=O)C2)=O)CCC1=O c1(OC)ccc(=NC(=O)C2(C)CCCN2C(=O)C=Cc2ccccc2OC)[nH]n1 CC(O)CCCCCC(=O)N1CC(NC(=O)Cn2cnnc2O)C2(CCC2)C1 c1(C(=O)NC(CNC(c2c(SC)ccs2)=O)C)ccc2c(c1)CCCO2 C1(C(=O)NC2C(CC)C2)CCC(NC(c2ccnn2C2CC2)=O)CC1 Cc1sc(C)c2sc(C(=O)NCC3CCCCC3NC(=O)CC(F)F)cc12 c1(C(N2CCC(NC(c3cnc(-n4cccn4)s3)=O)C2)=O)ccc(C(F)F)nc1 C(C(C)(C)CNC(=O)Cn1ccnn1)N(C)C(c1cnn(-c2ccccn2)c1)=O N1(C(CCC2CC(SC)C2)=O)CCc2ccccc2C(O)C1 CC(C)CCC(=O)N1CC(CF)(NC(=O)C(N2CCCCC2=O)C)C1 c1(CC)[nH]c(Cl)nc(=NC(C)CNC(C2(C)CCOC2)=O)c1C#N C1(NC(CS(=O)(=O)NCC)=O)CN(C(=O)C=Cc2cc[nH]c2)CCC1O c1(NC(=O)CC(c2ccc(O)cc2)NC(COC(C)C)=O)cn(C)c(C(=O)O)n1 N1(C(c2c(COC)scc2)=O)CCOCC(NC(=O)Cc2ccns2)C1 CCC(CC)CC(F)C(=O)NC(c1cn(C)nn1)C(N1CCC(F)(C(N)=O)C1)=O CC(CC(=O)N1CCN(C(=O)C(F)=CC2CC2)C2CCC12)C(F)(F)F c1(NC)c(C(N2CC(COC)(NC(c3cc(C)cc(C)c3)=O)C2)=O)cccc1F c1(C(N2CC(CCO)(NC(c3nc(C)n(C)c3)=O)C2)=O)cc2cnccc2[nH]1 N1(C(CCc2c(C)nccc2)=O)CCN(C(=O)C(=O)Nc2ncc[nH]2)CC1CF C1(N(C(CCOCC)=O)C)CCN(C(c2csc(COC)n2)=O)CC1C C(N=c1nc(N2CC3CC2CS3(=O)=O)c2ccccc2[nH]1)c1n(C)cnn1 N1(C(=O)NC2C(C)CCCC2)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CCC1C N1(C(C=C(C)c2ccco2)=O)CC2CCC(N(C(=O)C(C)n3cccn3)C)C2C1 C1(CC(=O)NCc2c(C)noc2C)N(C(=O)CC2CC(F)(F)C2)CCC1(C)C CC(CNC(c1cccnc1-c1ccccn1)=O)(C(F)(F)F)C1OCCO1 N#Cc1ccc(S(=O)(=O)N2CCC3(CC2)CC3COC(F)F)cc1NCCO O=C(C1=COCCC1)NCCn1cc(C(=O)NC2C=CCC2)nn1 N(C(=NCCCC1CCCCO1)NCC1(C)CCCCC1)C(c1cccs1)C Cc1nc(-c2nc[nH]n2)sc1C(=O)N(CCCCNC(C1CC12CCCC2)=O)C C1(C(=O)NCC(C)NC(=O)C(c2ccccc2F)C)(OC)CCCCC1 CCS(=O)CC(=O)NC(C)(C)C=CC(=O)NC(c1n[nH]c(C)n1)C C#Cc1cncc(C(=O)NC(CCNC(c2cnc(N(C)C)o2)=O)C(C)C)c1 N1(C(CCOCCC)=O)CCC(N(C(=O)CCc2cscn2)C)C2(CC2)C1 O(NC(=O)C(C)N1CCOCC1)c1c(C(C)C)nsc1 c1(C(c2nnnn2CC2CCOC2)NCc2c(I)c[nH]n2)cc(F)c(Cl)c(F)c1 CCC(C)C(C(=O)NCc1cnco1)N(C)C(c1cccc[n+]1[O-])=O C(=O)(C(CC(F)F)N(C(=O)C1=COCCC1)C)NCP(OCC)(C)=O N1(C(CC2(OC)CN(C(C3CCCC4(CC4)C3)=O)C2)=O)CCC2(CCCCO2)C1 N1(C(C(CC)CO)=O)CCN(C(=O)C2=CCSC2)CC1CCOC N1(C(c2nn(CC)nc2C)=O)CC(C(N2CCC2(C)CCO)=O)CC12CCC2 N1(C(c2cnc(SC)s2)=O)CCN(C(C2CCOC2(C)C)=O)C(CCO)C1 CN1CCN(C(c2cc(CCNC(=O)CCc3cnco3)on2)=O)CCC1=O CC1CCCc2cc(C(N3CCC(CC(C)NC(=O)C4CC4)CC3)=O)nn21 C(=O)(CC(C)CC(=O)OC)N1CCCC(CN(C(=O)C(C)(C)C(N)=O)CC)C1 c1(OC)cc(NC(c2cccc(NCc3ccc(F)nc3)c2)=O)ccc1Br CCC(O)C(C)(C)C(=O)NC(C)CC(=O)Nc1ccccc1C c1(C(N2C3CC(C(N4CCCC(C#N)C4)=O)C2CC3)=O)cc2ncccc2[nH]1 Cc1cc(Cl)c(C(=O)NC2CC3CC2N(C(=O)CCc2cn[nH]c2)C3)cc1F Cc1cc(C(=O)NC2CCCCC2CNC(c2cc(C)n(C)n2)=O)ccc1F C1(NC(C2CC2F)=O)(CO)CCCN(C(=O)CCC2CCCCO2)C1 c1(C(N2CC(C(C)(C)O)(CNC(c3nc(C)c(C)s3)=O)C2)=O)ccc(Cl)nc1N N1(C(C2CCN(C)C(=O)C2)=O)C2CCCC1CC(NC(=O)CCc1nccs1)C2 c1(C(N2CC(SC)C(NC(C3C=CCC3)=O)C2)=O)cnc(C)cc1C C12(CNC(c3cc(=O)cc(Cl)[nH]3)=O)CCC(C1)N(C(=O)CCc1ccncn1)C2 C1(C)(C(=O)NC(CCCNC(c2c(CCC)n[nH]c2)=O)C)CCC(C)=C(C)C1 CC1CC(C(=O)NCC2CN(C(c3occc3-c3ccccc3)=O)C2)CO1 C1(CNC(c2[nH]cc(C#N)c2)=O)CN(C(C2CC3CCC3C2)=O)CC12CC2 Cc1cc(OCC(=O)NCCCOCCNC(=O)Cc2csc(C)c2)no1 CC(C(N)C(=O)NC1CCC1NC(c1ccccc1)=O)C1CCCCC1 c1(C(=O)NC2CCC(NC(C3(COC)CCCO3)=O)CC2)cc(=O)c(O)c[nH]1 c1(OC)cc(NC(C2CCCC2NC(c2cccnc2)=O)=O)c(F)cn1 Cc1oc2ccccc2c1C(=O)NC1CC1NC(=O)CCc1cc[nH]n1 N1(C(CCCCC)=O)CCC(C2CCN(C(=O)C(c3cnn(C)c3)O)CC2)C1 Cc1cc2ncc(C(N3CCC4(CCCN4C(=O)Cc4cnc[nH]4)C3)=O)cn2n1 C1(CNC(C(COc2ccc(CC)cc2)C)=O)CCCCN(C(=O)C(=O)NC)C1 c1(OC)ccc2[nH]cc(C(N3CCC(CNC(=O)C(C)OCC4CC4)C3)=O)c2c1 C1(C(=O)NCc2n(C)cnn2)CC(O)CN1C(=O)CC1CC(C)(C)CO1 C=CC(C)(C)C(=O)NCCC1(NC(c2cnn(CCC)c2C)=O)CC1 C(C(=O)N1CCCC1C(C)(C)NC(=O)Cc1cc(C)no1)(C(C)C)SCC C1(C)(C(N(CCC(C)NC(c2csc(C)c2C)=O)C)=O)COC(C)(C)CO1 C(=O)(CCS(C)=O)N1C(Cc2cn(CNC(CCN(C)CCO)=O)nn2)CCC1 c1(C(=O)NC2C3(CNC(C=CCOC)=O)CCC(C2)C3)cccc2nc[nH]c12 CCCC(C(=O)NCCCc1cc(C)no1)NC(c1ccc(C#N)o1)=O c1(C(N2CCC(C(C)NC(=O)Cc3cc[nH]c3)C2)=O)c(F)cc(C#N)cc1F C1(NC(c2c(C)cn(C)c2)=O)CC2CCC(C1C)N2C(c1ccoc1)=O c1(OC)ccc(CC(N2CC3CC3(CNC(C)C)C2)=O)cc1C(F)(F)F c1(C(N2C(COC)(CNC(=O)Cn3cc(C)cn3)CCC2)=O)cn(C)ccc1=O C1(C)(OC)CN(CC(=O)N(CCC(=O)N(CCCCOC)C)C)C1 N1(c2nnc(C(C)C)o2)CCN(C2CCCN(C(C3CC=CCC3)=O)C2)C(=O)C1 C(Cc1ccccc1)(C(=O)N1CCC(CCNC(=O)CCc2nc[nH]n2)C1)OC c1(C(=O)NCC2C(NC(CSCC#C)=O)CCC2)ccccc1S(C)=O CC1CN(C(C2CS(=O)C2)=O)CCC1NC(=O)C1=CSCS1 CC1(C(=O)NC2CC3C=CC2C3)CCCN1C(=O)CN1CCCC1=O CC1CN(C(C2(C)CC(=O)C2)=O)CC(C(=O)N(CC(O)CF)C)O1 N1(C(c2cnc(OCC)c(Cl)c2)=O)C2CCC1CN(C(c1cccs1)=O)CC2 N1(C(CC2CC(=O)NC2)=O)CC(NC(=O)COc2cccc(F)c2F)C2(CC2)C1 C1(NC(C(C)NS(C)(=O)=O)=O)CCCOC12CCN(C(c1cscn1)=O)CC2 CC1(C)CCC(C(N2CCOC3CC23)=O)CN1C(C1C2CC3C(C2=O)C13)=O C1(C)(C(=O)NC(C)CCCNC(=O)Cn2ccnn2)COC(=O)OC1 c1(CCNC(c2n(CC=C)nnn2)c2ocnc2C2CC2)ccc(OCC)cc1 C1(CNC(c2cc[nH]c2)=O)COCCN1C(C1(c2ccc(Cl)nc2)CC1)=O C(=O)(C(CC)C(=O)N1CCC(C)(C(=O)NCC(O)CO)CC1)OCC C1(C2CC2)(C(=O)NCC(CC)NC(c2cnn(C)c2F)=O)CC=CC1 C1(CNC(CN(CCC)C)=O)CC2(CCN(c3cc(C)ccc3[N+](=O)[O-])C2)CO1 N1(C(C(CSC)OC)=O)CCN(C(C2CCC(OC(C)C)CC2)=O)C2(CCC2)C1 N1(C(c2cc(CCNC(=O)C(O)CC(F)(F)F)on2)=O)CC2CCCC2C12CC2 c1(C2(C(=O)NC(C3CN(Cc4sncc4Br)C3)C)CCC2)ccccc1 C1(C(=O)NCC2(C(C)(C)O)CN(C(c3n(CC)nnc3)=O)C2)CCCN1N=O N1(C(CC(CC=C)NC(=O)CCCN(C)C)=O)CCC(O)CC12CC2 N1(C(CNC(CCC)=O)=O)CC(C)N(C(=O)CCc2ncccc2OC)CC1C C1(C(=O)NCC2N(C)CCN(C(=O)CCc3cc[nH]n3)C2)C2CCCCCCC12 CC(CN1CCCC1)CN=c1[nH]c(=NCC2C3CCCCCC23)[nH]c2c1SCC2 C1(CNC(C2CN(C(C)=O)C2)=O)CCC(NC(c2ccoc2Br)=O)C1 C1(CNC(c2c(CC)ncs2)=O)CC(F)(F)CN1C(C1CCCC(C2CC2)O1)=O Cn1nc(C2CC2)c(Br)c1CNC(c1cncc(-c2ccoc2)c1)=O O=C(CC1=CCOCC1)NC1COCCN(C(C2C3CCN2CC3)=O)C1 C1(C(N(C2(CC)CC2)C)=O)CC2C=CC1N(C(=O)CN(C(=O)COC)C)C2 CC(O)CC(C(=O)O)N(c1ccc(C(F)(F)F)cc1)C(=O)CCN1CCCCCC1 Cc1cc(C(=O)NCC2COCC2NC(=O)CCF)c(O)c(C)n1 c1(C(N2CCCN(CC(C)O)CC2)=O)ccc2ncc(=O)n(C)c2c1 CC(O)C(F)(F)C(=O)N1CCOC(CN(C)C(c2cncs2)=O)C1 c1(C(N2CCN(C(C#CC(C)(C)O)=O)C(CN(C)C)C2)=O)ccn2cccc2c1 N1(C(c2n[nH]c(O)n2)=O)CCCC(CNC(=O)C(c2ccc(F)cc2)(F)F)C1 c1(C(=O)NCC2(CO)CCCNC2)cnn2c1NCCC2C(F)(F)F N1(C(c2ccc(-c3ccc(C)s3)s2)=O)CCN(C(C)C(=O)O)C(=O)C1 N(C(=NCCCC(F)F)NCc1cc(C)ccc1Br)CCOCC Cc1nc(Br)sc1C(N1CCC(C)(C(F)(F)F)C1)C(=O)NCCC1CC1 C(=O)(C1=CCCC1)N1CC(CCC=C)(C(=O)N(C)Cc2ccn(CC)n2)C1 C1(NC(CCSCCCC)=O)CC(CNC(=O)CCCc2cncs2)C12CCC2 c1(C(N2C(CNC(C3(OC)CC3)=O)CC2)=O)cccn(CC(=O)N(C)C)c1=O C#Cc1cccc(CC(=O)NC(CCC2CC2)C(=O)NC2(C)CC2(C)C)c1 Cc1oc(CO)cc1C(N1CSCC1C(N1CCSCC1C)=O)=O c1(CC(=O)NC(C)CNC(C2CCOC2=O)=O)ccc2nc[nH]c2c1 C(=O)(C1CCCc2nncn21)NCC(CC(C)C)NC(CN1CCC(C)C1)=O C(C(C)(C(=O)N1CC(c2nncn2C)C1)NC=O)OC.C(C)(C)C c1(C(=O)NC(CNC(c2cc(C)c(C)nc2)=O)(C)C)cc(F)cc2c1NCCC2 N1(C(C(C)c2ccsc2)=O)CCN(C(=O)C=CSc2ccccc2)CC1C(F)F N1(C(CNC(=O)OC)=O)CCN(C(=O)C(CC(C)C)OC)CCC1C N1(C(C2CN(C)C2)=O)C2CCC1CC(N(C)C(C1(O)CC(C)(C)C1)=O)C2 c1(OC)ccc(C(=O)NCCC2CCCN(C(=O)CCCC3CCCC3)C2)nn1 N1(C(C(C)CS(C)(=O)=O)=O)CC2(CCCN(C(=O)CCOC3CCCOC3)C2)C1 C=CCCC(C)(C)C(=O)N1CCC=C(C(=O)NC(c2snnc2C)C)C1 C1(CCC(=O)NC2CCCC2(F)F)CCN(C(C2CCC(F)(F)C2)=O)CC1 N1(C(CCOCCNC(C(C)(C)C)=O)=O)CCCc2cccc(F)c21 N1(C(c2nc(C)oc2)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)CCO2 Brc1cc2ncnc(N3CCC(c4ncc[nH]4)CC3)c2s1 c1(C(=O)NC2CN(C(c3ccc(OC)cc3)=O)CC(O)C2)c(F)ccc(C)c1F N1(CC2(NC(c3c(C)onc3)=O)CC2)CCN(C(C2CCC(F)C2)=O)CC1 N12CCC(CC1)COC1CC(C1)C2=O.C1(C(=O)NC(C)(C)C)OC2CCC1C2 c1(C(N2CC(CC(N3CCOC4CC34)=O)C2)=O)cc(Br)cc2[nH]ccc12 CN1CC=C(CC(=O)N2CC3CCCC(C2)N3C(=O)Cc2ccc(O)nc2)CC1 c1(OCC)cc(NC(=O)NC(C)CS(N)(=O)=O)c(Cl)cc1Br CC(C)(CNC(=O)C(O)C1CCC1)CNC(C1CCN(S(C)(=O)=O)C1)=O c1(OC)cc(C(=O)N(C)CC2CCCN2C(=O)CCC2CC2(C)C)n(C)n1 C1(CNC(C(CC)F)=O)CCCCN(C(=O)Cn2ccc(O)nc2=O)C1 C(CC)(CC)(CCNC(=O)C(C)C(F)F)NC(c1cccc(SCCCC)c1)=O C1(O)(C(CC)C(=O)NC2CCC2CNC(C2(C(=O)NC)CC2)=O)CCCCC1 c1(C(=O)NC(C(C)C)CCNC(c2cccnc2CO)=O)cccc2c[nH]nc12 CC(=NOCC#N)C(=O)NCCC(O)C(=O)NCC(Cl)C(C)(F)F c1(C(N(C)CC2CN(C(=O)C3=CCCS3)CCO2)=O)nccc2cc[nH]c12 C1(CCC=C)(C(=O)NCc2ccc(C)nc2)CCN(C(=O)C(C)OCCOC)C1 C1(C(N2CC(O)(CNC(C3(NC(C)=O)CCCC3)=O)C2)=O)CCOC2(CCC2)C1 C(=O)(C(C)(C)C(F)F)N1CCC(C(CNC(C(C=C)OC)=O)O)CC1 C(=O)(CC(C)(C)C(F)F)NC1C(OC)CCN(C(c2cc(OC)c(O)cc2)=O)C1 C1(C(=O)NCc2ncc(OCC)nc2)CN(C(=O)C(C(C)O)N(C)C)CCCO1 C(=O)(CC(F)(F)C(F)(F)F)NCCCC(c1ccco1)NC(CC(=O)NC1CC1)=O c1(C(N2C3CC(NC(CCC#N)=O)CC2CC3)=O)ccc(F)c2occc12 N1(c2cc(NCc3scc(C)c3)nc(C)n2)CC(C)CC(C)(C)C1 C#CC1CC2(CC(C(N3CC(NC(=O)Cc4cccc(F)c4)C(O)C3)=O)C2)C1 Cn1nc(Br)nc1C(c1nnnn1CC(F)F)NCCc1cc(Br)no1 C1(O)(CC(=O)OC)CCN(C(=O)NC2CCC(C)CC2)C1 c1(CN2C(C(=O)Nc3c(C)occ3)CCCC2)ccc2cc[nH]c2n1 c1(NC(c2cncc(NCc3c(N)cccc3F)c2)=O)ccc2c(c1)OCCO2 c1(NCC)ccc(C)cc1C(N1CCC(CN(C)C(C2C3CCCC23)=O)C1)=O N1(C(C(CC)CC2CCCC2)=O)CCN(C(=O)C(C)(F)F)C(C(C)C)C1 c1(NC(C(C#N)c2ccccn2)=O)ccnc(O)c1 N1(C(CSCCCC)=O)CC2C(CNC(=O)CCn3ccnc3C(C)C)C2C1 c1(N(C)CC2N(C(CN(S(CC)(=O)=O)C)=O)CCC2)cc(Cl)ncn1 CC#CCC(C(=O)N(C1CC(C)CC(C)C1)C)NC(C1CCCCC(=O)C1)=O CCCCC(CC)CC(=O)NCCC(O)CNC(C1CC(n2cnnc2)C1)=O Cc1ccc(C(=O)N(C(C)CCNC(=O)CC2CC(CN(C)C)C2)C)cc1 Cc1cc(C)c(CC(=O)NCC(C)N(C)C(c2cnc3[nH]cnc3c2)=O)c(O)n1 C(C)(CCCCNC(C1(CS(C)(=O)=O)COC1)=O)NC(CC(C)OC)=O N1(C(CCNC(C)=O)=O)CC2CCOC2(CNC(=O)C(C)(C)CC(F)F)C1 N1(C(C(=O)Nc2cccc(NC3CCC3)c2)=O)CC2CCC1C(CO)C2 c1(OC)cccc(C(=O)NC(C)C(C)(C)NC(=O)C(C2CC(F)(F)C2)O)n1 c1(C(N2CC(O)(CN(C)C(C3CC3F)=O)C2)=O)ccccc1-c1cncnc1 N1(C(c2c(C)snc2)=O)CC(C)C(NC(C2CC(C)(O)C2)=O)C(C)C1 c1(C(N(C)CCOCCCNC(=O)CC2CCCC2)=O)cccn2cnnc12 Cc1cc(C(=O)N(C2CCC(NC(=O)CCN(S(C)(=O)=O)C)C2)C)nn1C1CC1 CC1(C)CN(C(c2cc(Cl)c(F)c(Cl)c2)=O)CC(C)(C)C1NC(=O)C1=CCCS1 Cc1cc(C(N2CC(CC(=O)Nc3ncc(Br)c(O)n3)C2)=O)cc(O)n1 C=CCC(CNC(C1CCSCC1)=O)NC(c1cc(C(F)(F)F)ns1)=O Cc1nc(O)[nH]c1C(=O)NC(C1CCN(C(c2cc(O)nn2C)=O)C1)(C)C c1(C(=O)NC2C(NC(CCc3scc(C)n3)=O)CC2)ccc2c(c1)C(=O)CCC2 C1(CC(=O)NCC(CNC(C=CCN(C)CC)=O)F)CCCN1C(C)=O C1(NC(c2n(C=C)nnc2)=O)CCN(C(c2ccccc2)=O)CC1C c1(CC)cc(C(=O)NC(Cn2cccn2)C(=O)N(CC(C)(C)C#N)C)no1 CCCCC(C(=O)NCCOCC(F)F)NC(=O)C(C(C)C)NC(C)=O C(C(C)(O)CNC(=O)C(Cc1cn[nH]c1)NC(=O)CCCNC(C)=O)OC C1(C(=O)NC2CN(C(CCCCSC)=O)C2)CC(C)(C)CCO1 C#Cc1ccc(C(=O)NC2CCC2C(=O)N(C(CO)CO)CC)cc1C C=C(C)C(C)(C)C(=O)N1CCC(C=CC(=O)NC2CC(C)OC2=O)CC1 N1(C(C2(C=C)CC2)=O)CCCC(C2CCN(C(=O)C3=CCC3)C2)C1 C1(CC)CCc2nc(NC(=O)NCc3c(F)cncc3Br)ncc2C1 N1(CC(=O)NCC2(CN(C(=O)C(N3CCCC3)C3CC3)C)CC2)CC(=O)N(C)C1=O N1(C(c2c(OC)cccc2C)=O)CC2CCCC2(CNC(C2CC(SC)C2)=O)C1 C(C1=CCN(C(=O)CC2CCCC(C(C)C)O2)CC1)NC(c1cnn(CC)n1)=O CON=CC(=O)NC(CNC(C1CC1(F)F)=O)C1CCC1 Cn1ncc(C(=O)OC2CCC(OC3CCC3)CC2)c1C(F)(F)F c1(C(=O)NC2(CNC(=O)C(F)(F)c3ncc[nH]3)CCOC2)cccc(OCF)c1 C(CCN=C(NC(C)C)N1CCC(F)(c2ccccc2Cl)C1)=CC Cc1ccoc1S(=O)(=O)NCC(c1cccnc1)C C(=O)(C(C)(O)CNC(c1nnsc1C)=O)OC.C12CCC1C(=O)N2 C(=O)(C(CC(F)(F)F)c1ccccc1)N1CC2C(COC(C)(C)C)C2C1 c1(CC(=O)NC(CC)(C)CNC(c2nc(Cl)sc2C)=O)c(C)cc(C)cc1C C1(NC(C23C(NC(Cn4c(C)nc(C)n4)=O)C4CC2C3C4)=O)CCC(=O)N(C)C1=O c1(OC)cc(C(=O)NC2CCCCN(C(c3ccsc3)=O)C2)c([N+](=O)[O-])cc1F CON(C(=O)c1c[nH]nc1CCNC(c1cc(C2CC2)on1)=O)C1CCCC1 C1(NC(c2ccc(C(C)(C)C)[nH]2)=O)CCC(NC(C2CC2C(F)F)=O)CC1 N1(Cc2cn(CC(CNC(c3cc[nH]c3)=O)(F)F)nn2)CC=C(CO)CC1 c1(-c2c(C(C)(F)F)cccc2)ncnc2[nH]cnc12 c1(C(=O)NCCC(=O)NC2CC3CCCC3C2)ccc2ccccc2c1 C12(C(N3C(C4(NC(CCC#C)=O)CC4)CCC3)=O)CCC(N(C)C)(CC1)CC2 C1(CC(=O)NCCNC(c2ccc(C(C)(C)C)cc2)=O)Cn2ccnc2NC1=O c1(CC(N2C(CCCNC(C3CC=CCO3)=O)CCC2)=O)ccc(O)c(F)c1 c1(C(=O)NCCCN(C(CC(CC)CN(C)C)=O)CC)cc2scc(C)c2[nH]1 C1(NC(c2c(C(C)C)n[nH]c2)=O)CC(C)CN(C(c2cn(C)nc2Br)=O)C1 c1(C(=O)NC2CC(CC(=O)NCCCn3cncn3)C2)c[nH]c2ccccc12 c1(CC(N2CC(OCC)C2)=O)nc([N+](=O)[O-])n[nH]1 C(=O)(CC1=CCOCC1)N1C(CN(C(=O)CC2CCCS(=O)(=O)C2)CC)CCC1 C1(OC)CC(C)CN(C(=O)C=CC(C)NC(C2C3CCCC(=O)C23)=O)C1 c1(C(=O)NC2CC(CNC(C(C=C=C)C)=O)C(O)C2)ccc(Cl)cc1C N1(C(c2cc(C)[nH]n2)=O)CCC(C(=O)NC(C2CCCC2)C)(C(C)C)C1 c1(OC)cc(F)ccc1C(N1C2CCC(C2)C1C(=O)NCc1nc(Cl)cs1)=O C1(CNC(CS(=O)(=O)N(C)C)=O)CCC2(CN(C(c3cccc(F)c3N)=O)C2)O1 C1(NC(CN2CCC(OC)C2)=O)CN(C(=O)CCCN=[N+]=[N-])C2(CCCC2)C1 C1(CNC(C#CC(C)C)=O)(NC(=O)CN(C)S(N)(=O)=O)CC2CCC1CC2 C1(CC=C)(NC(=O)CCCCCCN)CCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CNC(CCN(CCC(C)(C)C)C)=O)CCC(NC(c2cnc(Cl)s2)=O)CC1 c1(NC(Cc2c(C(C)=O)cccc2)=O)ccc(NC(c2ccco2)=O)cc1Br C1(NC(c2ccc(C(=O)OC)o2)C)CC2(CCCN(C(=O)CN(C)NC(C)=O)C2)C1 N1(C(C(C(CC)CC)C)=O)CC2(NC(c3cncc(N)n3)=O)CCCC2(F)C1 CC(CC(=O)NC12CC(CNC(=O)C(O)Cc3ccccc3)(C1)C2)CC(C)(C)C C(=O)(C(F)CC(C)(C)C)NCCN(CCNC(c1cccc(CO)c1)=O)CC c1(C(=O)NCC(F)(F)C(F)(F)F)ccc(F)c(Br)c1F C1(C(=O)NC(C)CNC(=O)CCCCN2CCOC2=O)Cc2cccc(F)c2O1 c1(SC)nc(Cl)cc(=NCCC2CCN(C(c3cc(C)nc4ncnn34)=O)C2)[nH]1 c1(OC)nc(C(N2CCCC2CNC(C2CCCCC2C(N)=O)=O)=O)sc1C c1(-c2nc(C3C(C)CCN3)on2)c[nH]c2cc(OC(F)(F)F)ccc12 c1(C(=O)NCCNC(c2ccc(C)c(O)c2)=O)ccc2cnnc(O)c2c1 C1(CNC(C(CC)C)=O)CC2CCC(C1)N2C(C1CCS1(=O)=O)=O C1(C)(N(C)C)CC=CC1.C12CC(C1)CN(CC1CCCO1)C(=O)CONC2=O c1(C(N(C)CC)=O)ccc(C(=O)NC(C)CNC(C2(N=[N+]=[N-])CC2)=O)cc1 CN1CC(C(=O)NCC23CC(NC(c4csc(Cl)n4)=O)(C2)C3)CC1=O C(c1nc(C)co1)=CC(=O)NC1CCC(CNC(Cc2c(C)con2)=O)C1 Cc1noc2cc(C(N3CC(NC(c4cccc(N)c4)=O)C3)=O)ccc12 C(=O)(C(O)CC(F)F)NCC12OCC(CNC(c3ccc(NC(C)=O)s3)=O)(C1)C2 C1(C(=O)NCc2cc(C(=O)NC(COC)C(=O)OC)n[nH]2)CN2CCC1C2 C=CC(C)(O)CC(=O)NC(CO)C(C)NC(C1(C(F)F)CC(=C)C1)=O N1(C(c2cn(C)c(O)n2)=O)CC2(C1)CN(C(C1CC(S(C)(=O)=O)C1)=O)C2 Nc1cc(C(=O)NCCC2CCN(C(=O)CN(c3ccncc3)C)C2)ccc1F CC(C)(C)C(=O)C1(C(N2CC(c3cn(Cc4cccnc4)nn3)C2)=O)CCC1 CCC(C)(C)C(C)CC(=O)NC1CCCC(CNC(=O)CCC(C)C)C1 c1(-c2n(CC(=C)C)nc(C(C)O)n2)cn2cc(C)nc2s1 c1(C(CCC)NC(=O)C(C)N(C(=O)C(C)C)C)ccc(Cl)cc1 CCC(O)C(C)C(=O)NCC1CC1CNC(c1n[nH]cc1Br)=O N1(C(c2c(C(C)C)occ2)=O)CCC(F)C(NC(=O)C=C2CCCCC2)C1 CC(CC(F)F)C(=O)NCC1CC(F)CN1C(c1coc(CO)c1)=O c1(C(N2CCC(NC(CCOCCC)=O)C2(C)C)=O)cc(Cl)cc2c1CCC2 CN1CC2CCC(C1)N2C(C1CC=CCC1NC(C1(F)CC=CC1)=O)=O N1(C(CCNC(=O)OCC)=O)CCCC(N(C(=O)C(C)(COC)OC)C)C1 C1(NC(CCC=CCC=C)=O)(CF)CCN(C(c2snnc2C2CC2)=O)C1 C1(C(=O)NC2(CC=C)CN(C(c3ccc(C#N)o3)=O)C2)CC2C(C1)C2(F)F N1(C(COCCOC)=O)CCC(CCNC(c2ccc(OC)cc2Cl)=O)CC1C CCC(CC(=O)NCC1COCCN1C(=O)C=Cc1cc(C)no1)C1CCC1 C(C#Cc1cccc(C(=O)OC(C)(C)C)c1)NC(C1C(C)(COC)C1)=O C1(NC(Cc2ccc(C)c(F)c2)=O)CN(C(=O)C(C)C(C)O)C2(CCC2)C1 c1(C(N2CCCN(C(c3c(C)n(C)nc3)=O)CC2)=O)csc2ccccc12 Cc1[nH]c(C(=O)NCCOc2ccc(Br)nc2F)c(C)c1C(=O)OC(C)(C)C c1(CC(=O)NCC2(NC(C(C=C=C)C)=O)CC2)cnn2c1CCCC2 C12(C(=O)NCC#CCNC(C(C(C)C)NC(C)=O)=O)CCCN1CCC2 N1(C(CCN(CC)CC)=O)CC(N(C)C(c2ccc(C)cn2)=O)C(O)C1 c1(C(=O)NCCCN(C(C2CCN(C)CC2)=O)C)c(O)ccc(Cl)c1F c1(OC)ccc(C(=O)NC(C)(C)CC(=O)NCC=CCl)cn1 c1(NC(CCCOC)C)ncc(S(=O)(=O)NC(C)CCCC(F)(F)F)cc1Cl c1(C(=O)NC(CC(C)NC(c2n(CCC)ncc2)=O)C)cc(F)cc(F)c1 N1(C(C(=O)NC2(CO)CCS(=O)(=O)CC2)=O)CCC(C2(O)CNC2)CC1 N1(C(c2c(C)coc2)=O)CCC(C(=O)NC2CCCSCC2)CC1 C1(C(=O)NC(C2CCCC2)C)CCN1C(c1cc[nH]c1)=O C1(C2CCCN(c3nccc(C#N)n3)C2)(NC(c2ncc(OCC)nc2)=O)CC1 CC1(C)CN(C2CC2)CCC1NC(=O)C=Cc1nc[nH]n1 c1(C(=O)NC2CCCC(CNC(C3CCCCC3)=O)C2)cc2occc2[nH]1 C#CCCCC(C)C(=O)N1CCC(C)(C)C(C(N2CC(=O)NC(CC)C2)=O)C1 C=CC1(CC(=O)NC2CCC(O)C2)CN(C(=O)Cc2ccc(C)nc2)C1 c1(C(=O)NC2C(OC)CN(C(=O)COCP(C)(C)=O)C2)nc(Cl)ccc1N c1(CN2CCOCC2)cccc(C2(O)CCC2OC(F)(F)F)c1 c1(C(=O)NCC2CCCC(CNC(=O)CCCCCF)C2)cc2n(c1)CCCC2 CN1CC(C)(C)CC1C(N1CCCC(O)(CNC(=O)CC2(N(C)C)CCC2)C1)=O C1(Nc2c(C3c4nnnn4CCCO3)ccnc2)CC(C)(C)C12CCC2.CC.SC c1(C(=O)NCC2C(NC(c3[nH]cc(CS(C)(=O)=O)c3)=O)COC2)cc(O)nc(O)n1 C1(C(=O)NCCN(C(C(C)(C2CC2)OC)=O)C)CCC(CCC(C)C)CC1 C(CC(=O)Nn1cccn1)C1CCN(C(c2c(CC)ccs2)=O)C1 C1(NC(c2c(C)noc2C(C)C)=O)CN(C(C2CN(C(C)C)C2)=O)CC1(C)C C1(C(C(=O)NCCSC)N2CCC2C(C)C)CCC(CC2CC2)CC1 CC1C(NC(=O)CC2CCCCCCC2)CCCN1C(=O)Cc1ccsc1 c1(C(N2CC(NC(C(C)=C3CC3)=O)CC2(C)C)=O)sc(S(N)(=O)=O)c(C)c1Cl N(C(=NCc1ccnn1C)NCC1(C)CCCOC1)CC1(SCC)CC1 C1(NC(CC(=C)C)=O)CCCCC12CCN(C(=O)C(F)CC)C2 N1(C(c2c(Cl)ncc(OC)c2)=O)CCN(c2nnc(C3CC3)o2)CC(O)C1 c1(C(N2CCC(CCNC(C(C)C#N)=O)C2)=O)ccnc(CSCC(F)(F)F)c1 C1(C(=O)NC2(CNC(c3c(C)nc(CC(C)C)s3)=O)CC2)CC2CCC1CC2 C1(NC(C(N2CCCCC2)C)=O)COCC1C(=O)NCCn1cnnc1 C1(CNC(C(C=C)OC)=O)CN(C(=O)Cc2cnn(C)c2)CC1(F)CO CCCC(C(=O)NCC1CCCCN1C(c1oc(C)nc1CC)=O)OCC C1(CNC(C(CC=C)C)=O)CCC(C)(C)CN1C(=O)C(C)C(C)COC c1(C(N2CCCC(c3cc[nH]c(=N)n3)C2)C)cc(I)cc(I)c1 c12nc3ccc(nc3s1)O2.C1(NC(COC)=O)(CO)CCN(CC2CC2)CC1 CC(CO)CCN=c1[nH]c(=NC2CCCC2C(N)=O)[nH]c2c1COCC2 C=Cn1nccc1C(N1CCCC(C2CCCN2C(c2cnc(O)o2)=O)C1)=O C(=O)(CCCCC(=O)NCC1CCC2(CN(C(c3c(C)n[nH]c3C)=O)C2)O1)NC c1(C(=O)NC2CCN(C(c3ccncc3Br)=O)CC2O)ccn2ccnc2c1 N1(C(CCNC(C)=O)=O)CC(NC(c2nccnc2N)=O)CC(C)C1 N1(CC(=O)NC(CNC(C(C(C)C)O)=O)C2CC2)CCP(C)(=O)CC1 C1(C)(NC(C(CNC(C2C(C)=CCS2)=O)N(C)C)=O)CCCCCC1 CC1(C)CN(CCC(=O)NCCC(O)CNC(C23CCCC2C3)=O)CCS1 c1(CC(=O)N(CC(CC)NC(=O)C=CC(C)C)CC)ccc2nsnc2c1 c1(C(=O)NCCCN(C(=O)Cc2cncnc2)C)nccc2ccn(C)c12 C1(C(=O)NC(C=C)(C)C)CCCN(C(C2Cc3nccn3C2)=O)CC1 c1(C(c2nnnn2-c2ccccc2)(C2CCOC2)NCCCOC)ncc(Cl)cc1Cl c1(CCOCC)nc(C(=O)NCC(C)CNC(C2CCN(CC(C)C)C2)=O)co1 C1(CC(=O)N(c2c(C)nsc2)C)CCCN(C(=O)CC(C)C)C1 c1(C(=O)NCC(CNC(c2ncc(C)nc2)=O)O)ccc2c(C)cc(O)nc2c1 c1(C(N(CC)Cc2cc(C)on2)=O)cn2c(n1)CCN(CC1(CO)COC1)CC2 C(=O)(CS(=O)CCC(F)(F)F)NCC1CN(C(C2C(OC)(OC)CC2)=O)C1 N1(C(c2c(CC)ocn2)=O)CCCC2CN(c3cnc(C#N)c(C#N)n3)CCC12 C1(NC(C2C(CC)CCC2)=O)CCCC12CCN(C(=O)C(C1CC1)SC)CC2 c1(C(=O)NC(CN(C(C2C(C)C2C)=O)CC)C)cc(C(F)(F)F)ccc1Cl N1(C(C2N(C(c3c(C)ncs3)=O)CCOC2)=O)CCCC(C)(O)C1 c1(C(=O)NC(CCCNC(CC=C=C)=O)C)c(OC)ncnc1C Cc1oc(-c2ccsc2)nc1CC(=O)NCC(C)CNC(C1COCCO1)=O C1(NC(C2(N(C)C)CC2)=O)CN(C(=O)CCn2cccc2)CC2(CCC2)C1 c1(C(=O)NCC(CCCC)NC(C2C(=C)CC2)=O)cnc2onc(C)c2c1 N1(C(C2(C3CCCO3)CCOCC2)=O)CC2COCCC2(N)C1 C1(C(=O)NCC(CCOC)NC(c2occc2CN(C)C)=O)CCN(OC)CC1 Cc1ccc2nonc2c1C(=O)NC1(CO)CCN(C(C2CCOC2)=O)C1 C1(CC)CN(C(=O)CC2CC=CC2)CCC1NC(c1c(Cl)c(C)nn1C)=O c1(C(=O)NCC(C(C)C)(C)NC(=O)C(O)CN(C)C)ccc(=O)n(C)c1 N1(C(c2c(C(C)C)ncs2)=O)CCC(C(F)(F)F)C(CNC(C2(F)CC2)=O)C1 Cc1cccc(-n2cc(C(c3nnnn3C)NC(C3(C)CC=CC3)=O)cn2)c1 N1(C(CC2C(OC)(OC)CC2)=O)CCC(N(C(=O)COc2ccsn2)C)C1 CC1CCCCN1CCC(=O)NC1CCC1CNC(=O)Cc1ccsc1Cl c1(C(=O)OC)ccc(Br)cc1S(=O)(=O)N1CC(c2cccc(F)c2)C1 c1(CC(N2C(CCNC(C(C(CC)O)C)=O)CCC2)=O)noc2ccccc12 CCCC(CCCNC(c1nc(Br)sc1C)=O)NC(C12CCC(C1)C2)=O C(CC(C(=O)NCCc1ccccc1O)NC(C1COCCN1C)=O)SC N1(C(c2nn(C)c(F)c2)=O)CC(C2CN(C(C3CC3c3ccnn3C)=O)C2)C1 c1(C(N2C(CNC(=O)Cn3cccc3)CCCC2)=O)ccc(OC(F)F)c(F)c1 c1(C(C)C)c(C(=O)NC2CN(C(=O)Cc3ccns3)CC2F)cnn1C N1(C(C(CCC)F)=O)CCC(CNC(=O)C2=C(C)CC2)C12CC2 C1(CC(=O)NCCCC(C)O)CCN(C(C2CC2C2(C)COC2)=O)C1(C)C c1(CCCNC(CCN(C(C2CCC(F)C2)=O)CC)=O)nc(C)no1 c1(OC)ccc(F)cc1C1CCCN1CCCNS(C)(=O)=O c1(NC(=O)CC2COCCO2)cccnc1CC(N1CCOCC1C1CC1)=O C(C(C(=O)NCCCCCN(C)C)C(C)(C)C)NC(C(COC)COC)=O Cc1sc(Br)cc1C(=O)NCCC1CCN(C(C2CC(N(C)C)C2)=O)C1 N1(C(C(=O)NC(c2ccc(Cl)s2)COC)=O)CCC(CC(=O)N(C)C)CC1 c1(C(N(C2CN(C(CC(COC)C)=O)CC23CC3)C)=O)ccc([N+](=O)[O-])n1C N1(C(c2ccnc(Cl)c2Cl)C(=O)NCc2cccnc2)CCOCC(C2CC2)C1 C(=O)(C#CC1CCOCC1)N(CCCCC(=O)NCC1(O)CCCOC1)C c1(CNC(C2(CC)COC2)=O)cnn2c1CN(c1ccc(C(N)=O)cn1)CC2 C1(NC(c2cnc(C(C)C)o2)=O)CN(C(C2CC=CCO2)=O)CC1(C)C c1(C(=O)NCC2CC(C)(C)N(C(c3ccncc3)=O)C2)ccc2c(c1)COC2 CC(C)CCC(F)C(=O)N1CC(N(C(=O)CCc2ccncn2)C)C(F)C1 c1(C(=O)NCCCC(C)NC(C=C(C)c2ccsc2)=O)cccc2nsnc12 N1(C(=O)CC2(CO)CC2)CCN(C(c2csc(-c3ccccn3)n2)=O)CC(O)C1 c1(C(N2CC(CC(N3CCOCC3C3CC3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 C1(NC(c2ccnc(C)n2)=O)CCN(C(=O)CC2CCC(=O)N2)C12CCC2 n1(CC(N2CC(N(C(c3c(COC)noc3)=O)C)C2)=O)cnc2ccc(C)cc12 N1(CCCCNCC(c2ccccc2C)OC)CCN(CCO)CC1 c1(C(=O)NCC2(CCNC(CSCC(=O)OC)=O)CC2)cc2c(F)cccc2[nH]1 C#CCC(C)(CC)C(=O)NC1CC1NC(=O)CCCC#CC C1(C(=O)NC(C)CCO)C2CC(CC2F)N1C(c1ccc(C(F)(F)F)cc1)=O C=CCCCCC(=O)NC(C)CN(C(=O)Cc1n[nH]cc1Br)CC c1(NCC(C)CC2CC2)nc(N(C)Cc2c(F)cccc2Br)c2c(n1)CCC2 c1(C(=O)NCC2C(NC(C=CCOC)=O)CCCC2)ccc(F)c(C#N)c1 C1(C(=O)NC(CC)(C)C)CN(C(C2CCC(F)CC2)=O)CC1CC(C)(C)C C1(COCC)CCCN(C(C2CCC3(c4ccc(COC)cc4)CC23)=O)C1 Cc1ccnnc1C(=O)N(CC(CO)(CO)NC(C1CCSC(C)C1)=O)C C1(NC(C(COC)O)=O)CCN(C(=O)Cc2cccc(F)c2)CC1F N1(C(Cc2c(C)noc2C)=O)CCOCC(C(=O)NC(C)CCO)C1 C(C(C(CS)(C)CC)CCCCC)NC(CC)COC N1(C(=O)NCc2cn(C(c3ccn(C)n3)=O)nn2)CCCS1(=O)=O c1(NC(c2csc(NC(c3ccc(Br)nc3)=O)n2)=O)cccc2ncsc12 c1(C(=O)NCC(CC(=O)N(C)CCN(C)CCO)OC)ccc(=O)n(C)n1 c1(C(N2CC(N(C(=O)C(C)(F)c3ccccc3)C)C2)=O)ccccc1OC(F)F CC(C)C(O)C(C)C(=O)NC(C)CN(C(=O)CCc1cnc(C2CC2)o1)C C(=O)(C(CNC(=O)CC(C)C)CC1CN(C(C2CC2(F)Cl)=O)C1)OC C(=O)(CCCN=[N+]=[N-])N1CC2C(CN(C(CN(CCOC)C)=O)C)C2C1 c1(C(N2C3(CCN(C(C4C(C=C)C4)=O)C3)CCC2)=O)ccnc2cc(F)cnc12 N1(C(Cc2c(C)nc[nH]2)=O)CC2CCOC2(CNC(=O)Cc2ccsc2)C1 C1(CC(N2CCC3(CCCN3C(=O)CCBr)C2)=O)COc2ccccc2O1 CCS(=O)(=O)CC(=O)NC1CCN(Cc2ccc(Br)c(C)n2)CC1C C1(C(=O)NC(CC)C(C)(F)F)CC1C1CN(C(=O)C(C)c2ccco2)C1 C(=O)(CC1=Cc2ccccc2C1)N(C)CCN(C)C(C1CCCCC(F)(F)C1)=O C1(OC)CCC(NC(C2(NC(c3nccn3C)=O)CCSC2)=O)CC1 C1(C(=O)NCc2ccc(OC(C)C)nc2)CCCN(C(=O)CNC=O)CC1 c1(C(=O)OC)ccc2c(c1)CN(C(C1(C#N)CCC1)=O)CC2 C1(C2CN(C(C3Cc4cscc4C3)=O)C2)(NC(c2cc(C3CC3)ns2)=O)CC1 c1(C(N2CC(=C(CNC(c3cc(C)sn3)=O)F)C2)=O)c(C(F)F)nn(C)c1C c1(C(N2C3CN(C(=O)CCCCBr)CC32)=O)cccc2c1CCC2 c1(C(=O)NCCCNC(Cc2cc(C)on2)=O)cnccc1N1CCCC1 C(=O)(C1CSc2ccccc21)NCCC1(O)CCN(C(C#CC(C)(C)C)=O)CC1 n1(CC)nc(C(N2CC3C(N(C4(C)CCC4)C)C3C2)=O)cc1C(=O)OCC N1(C(C2(CC=C)CC=CC2)=O)CC2(CC(C(=O)Nc3cncc(OC)c3)CO2)C1 C=CCCCC(C(=O)NCCC(F)(F)CO)NC(c1csc(Cl)n1)=O C12CCC3(CCC3)N(C1)C2=O.O=C1NCCN1CCC1CC1 c1(CNC(NCC(=O)NCC#C)=NCCCCl)noc2c1CC(C)CC2 c1(CC)c(C(=O)NC2CN(C(=O)C=C3CCC3)CC2(C)C)cccc1C C(=O)(CC(F)(F)F)NCc1cccc(CN(C)C(c2nnn(C)n2)=O)c1 C(=O)(C(C)C(C)NC(=O)C(C)c1ccco1)NCc1cn(CC)nc1 C(CCCCC(=O)NC(C(=O)NC(C)Cc1cccnc1)C1CCOC1)OC C1(CC=C)(NC(C2CC(n3ccnn3)C2)=O)CCN(C(=O)C(C)SCCCC)CC1 N1(C(C23N(C(c4n(CCC)ncc4)=O)CCC2C3)=O)CC2(CCNC(=O)O2)C1 C1(NC(C(c2cnn(C)c2)NC(C(C)c2ccsc2)=O)=O)CCCC(O)C1O C=CC(C(=O)N(C)CCOCCNC(c1n[nH]cc1F)=O)c1ccccc1 c1(C(N2CC(C(=O)NC(CC#C)C(N)=O)C(CC)C2)=O)ccc(C=C)cc1 C1(NC(CC=CCC)=O)CN(C(=O)CC(C)F)C2(CCCCCC2)C1 N1(C(c2c(C)cco2)=O)CCC2CCN(C(=O)CCCc3cccnc3)CC2C1 OC1c2ccccc2CC1CCCCN1CCN(c2ncnc(C(F)F)c2Br)CC1 C12(CNC(C(C)NC(C)(C)C)=O)CN(C(c3ccc(N)cc3F)=O)CC1CCO2 c1(CC)cc(OCC(=O)NC2(C)CCN(C(=O)CC=C(C)C)C2)ccc1Cl CC1C(=O)CCC1CC(N1CCC(C2CCCN2C(c2ccn(C)c2)=O)CC1)=O Cc1ccc(CC(=O)NCC2CCN(C(=O)CN(c3ccccc3)C)CC2)cc1 Cc1nc(C)c(CC(=O)NCC2C=CC(NC(=O)Cc3cncc(F)c3)C2)s1 c1(C(=O)NCC2CCC(C)N(C(c3ccoc3)=O)C2)cc2sccc2cn1 C(=O)(N1CC2COCC2O1)C1N(C(CC(C)F)=O)CCCCC1 C(=O)(C(F)C(C)(C)O)N(C(CNC(c1c(OC)n(C)nc1)=O)C)C C(=O)(N=c1ncn(Cc2cccc(F)c2)[nH]1)c1ccc(N(CC#N)C)cc1 c1(C(N(C2C3CCOC3C2(C)C)C)=O)ccc(S(N)(=O)=O)c(N)c1 C(=O)(CN=c1ccnc[nH]1)NC(CCCC)CNC(=O)Cc1ccc(OC)nc1 N1(C(C(=O)Nc2nc(CSC)c(C3CC3)s2)=O)CC2CC(C1)C2(F)F c1(C(N(C(c2ccccc2)CNC(C(F)=CC)=O)C)=O)cc(C)c(C)[nH]1 C1(C(=O)NC2(C(F)(F)F)CCC2)C2CCC(C2)N1C(c1cccc(Cl)c1F)=O c1(C(N2CC(C(=O)NCC)C2)=O)ccnc2c1CCC2 c1(C(N2CCC3CCN(C(c4ccco4)=O)CC32)=O)cc2ncccc2cc1Cl N1(C(Cc2c(OC)noc2C)=O)C(C)C2CC1C2NC(c1c[nH]c(Br)c1)=O C1(C(N2C(C)CN(C(=O)CC3CCC(O)C3)CCC2)=O)CC(C)(C)OC(C)(C)C1 C1(C(=O)NCCOCC(N2C(C)(COC)CCC2)=O)CC2CC1CC2O N1(C(CCC=CC)=O)CCC(CCF)(C(=O)O)C1 C1C(C(C)(C)C)C(=O)N1C1CC1.C1(C)(C(C)C)CC1C(=O)NCCC(C)C C(CN=c1[nH]c(=NC2COC(C(C)C)C2)[nH]c2cccnc12)SCC C1(CNC(C(C)C(F)F)=O)CCC2(CCC2)C1NC(c1ccc2occc2n1)=O C1(CNC(C(C#N)C2CC2)=O)CC2CCC1N(C(C1CCC(=O)N1)=O)C2 C1(CC(C(=O)NCCCSC)N(CC(C)C(=O)OC)C)CCCCN1C(C)=O c1(C(N2CC(NC(c3cnncc3O)=O)C(CO)CC2)=O)nc2cnccc2s1 c1(N(CC(=O)OCC)CC2CC2)cc(C(N)=O)nc2ccc(Br)cc12 CCC(CCC(=O)N1C(CO)CC1C)NC(c1ccncc1)=O C1(NC(C(C)n2cccn2)=O)CC2CC1N(C(c1ccn(C)c1)=O)C2 c1(CC)c(C(=O)NCC(C)CNC(c2c(Cl)c(C)nn2C)=O)cccc1C C(=O)(CC(C(CC)CC)C(COCCOC)=O)NCC(C)(C)N.C(=O)(N)NC(C)C C1(CNC(CCC#CC)=O)CCCCCN1C(=O)CNC(=O)Nc1ccccc1 C1(CC(=O)NCC(CC)N(C)C)CC(C)(C)CN1C(=O)CC1CNC(=O)O1 C1(C(=O)NCC(CN(C(CCOCC#C)=O)C)C)CCCCC1n1cccc1 C1(CCOC)CN(C(=O)C(C)OCC(C)C)CCN1C(c1cc(=N)[nH]n1C)=O C1(C(=O)NCc2cn(C3CN(C(c4ccno4)=O)C3)nn2)CC2CCC1O2 CC1(C)COCC(C(=O)NC2CN(C(=O)CCC3CC3(C)C)CC2(C)C)O1 C1(OC)CC2CC(OC)C2C1.N1(C(Cc2cn(CC)nn2)=O)CC2CC1(CO)C2 c1(C(N)=O)cc(C(=O)NC2CCC2NC(c2cc(-c3ccco3)[nH]n2)=O)co1 N1(C(c2c(I)ccc(C)c2)=O)CCc2cc(-c3ccnc(C)c3)ccc2C1 c1(C(=O)NC2C(CNC(c3cc(C)on3)=O)CCC2)csc2c1CCCC2 N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)COCP(C)(C)=O)CC1CC(F)F c1(OC)ccc(-n2nnnc2C(c2occc2Br)NCC(C)C2CCC2)c(C)c1 N1(C(c2c(=N)[nH][nH]c2)=O)CCC2(CCC2)C(NC(C2CCCC(F)(F)C2)=O)C1 c1(C(=O)NCC2=CCN(C(c3c(C)nc(N)cn3)=O)CC2)cccc2nn[nH]c12 N1(C(CC=C=C)=O)CCCC2CN(C(C3(OCC)CCSCC3)=O)CCC12 Cc1cnnc(O)c1C(N1CC2(NC(C3CCC(N(C)C)C3)=O)CC1C2)=O C1(COC)C=CCCN1C(C1(NC(=O)CNC(=O)NC)CCCC1C)=O S(=O)(=O)(c1cc(CN=c2ccc(OC3CCCCC3)n[nH]2)ccc1Cl)CC(=O)O CC(C(=O)NCCN(C)C(C1CC1c1cnn(C)c1)=O)C(C)(F)F c1(CC)ccc(C(=O)NC2CC(C)N(C(=O)CCC(C)CN(C)C)C2)c(C)c1 NCCCC(=O)NCc1cc(C(F)(F)F)cs1 CCC(C(=O)NCCCOCCC(=O)N(C)CCOCCO)C(C)(C)CC CC(C)(C(=O)NCC(CNC(C1CC2C=CC1C2)=O)C(F)(F)F)C1=CCSCC1 N1(C(COCC#C)=O)CC(CNC(=O)C(C=C)c2ccccc2)CC1(C)C C1(O)(CC)CCCN(C(=O)CC2COCCN2C(c2ccncc2O)=O)C1 CCC(CC(=O)NCCC(O)C(C)C)NC(c1ccn(CCF)n1)=O c1(C(N(C(C)CNC(=O)CNC(=O)NCCCCCC)CC)=O)ccc(CO)s1 C(CC(=O)NC1CCC(C(N)=O)CC1)(C(C)(C)C)NC(c1cn(CC=C)nn1)=O C1(NC(Cc2c(C)ncs2)=O)CCCC(N(C)C(c2ccc(C(F)F)cc2)=O)C1 CC1(C)CCc2onc(C(=O)NCCC3CN(C(=O)C=Cc4ccsc4)C3)c2C1 Cc1sc(C(N2CCC(C)(NC(c3cc4occc4[nH]3)=O)C2)=O)c(C)c1C CN1CCCC1CCNC(C1CC(N(C(=O)CC2CC2C2CC2)C)C1)=O C1(NC(Cc2cccc(OCC)n2)=O)CCCN(C(C2CSC2)=O)C1CC C1(C(=O)NCCCc2ccco2)(CC)CCCN1C(c1cn(C)c(C)n1)=O C(C)(C)(CC(F)C(=O)N1CCN(C(C)(C)C)CC1)NC(C(C(COC)C)C)=O C1(c2cn(CCCC(C)(F)CNC(c3c(C)nns3)=O)nn2)CCCNC1=O N1(C(C(C(C)(C)C)O)=O)CCC(C2CN(C(=O)CCCNC(=O)C3CC3)C2)CC1 N1(C(c2cccc(C#C)c2)=O)CC2CC(C1)CN(C(c1cnn3ccsc13)=O)C2 N1(C(c2c(C)ccs2)=O)CC2CCN(C(c3cnn4c3CCC4)=O)CC2C1 n1(CC(=O)NCC(CNC(C2(CC)CCC2)=O)(C)C)nnc2c1CCCC2 Cc1ccc(C(N2CC=CC2CNC(C2(C)CCC(=O)N(C)C2)=O)=O)c(N)c1C N1(C(C2CCC(C)(C)C2)=O)CCOC(C)(CNC(=O)Cc2csnn2)C1 C1(C2CN(C(=O)CCF)C2)(NC(=O)CC2CCCCC2F)CC1 c1(C(N2CC(OC)(CNC(=O)CNC(=O)CN(C)C)C2)=O)ccc(Cl)cn1 N1(C(CCS(N)(=O)=O)=O)CC2CCN(C(c3cnc4[nH]ncc4c3)=O)CC12 C1(C(=O)NC(CC(=O)NCc2c(C)cncc2)C2CC2)CCOC(=O)CC1 CCC(C)(COC)C(=O)NCCOCC(N1CCCC(O)C1)=O Cc1cc(C)c(C(=O)NC2CCN(C(c3ccc(F)c(N)c3)=O)CC2F)c(O)n1 N1(C(CCC=C)=O)CC(C)CCC1C(=O)Nc1cccc(C(C)=O)c1 c1(C(C(=O)NCC(=C)C)N(C2CCC2)CC)cnn2c1CCC2 c1(C(N2CCC(NC(=O)C(O)C3CC3)C2)=O)ccc(-c2ccncc2)cc1F c1(C(=O)NC2CC2)occ2c1CCC2.C12CN(C1)C(=O)CN2CC#C Cc1cc(C(=O)N(C2CC(C(=O)NC3CC(O)C(F)C3)C2)C)cc(C)n1 Cc1cc(C(=O)NCCCNC(=O)CC(=O)OC(C)(C)C)c(S(N)(=O)=O)s1 N1(CC(=O)N(C2CCN(CC(=O)C3CC3)CC2)CC)CCC(C)(C#N)C1 C(N=c1cc(NCc2nc(-c3ccc(Cl)cc3)no2)nc[nH]1)c1n(CC)cnc1 c1(C(N2CC(NC(C3(C(F)(F)F)CC(=C)C3)=O)C(OC)C2)=O)ccc(F)c(C)c1 C1(N(C(C)(C)C)C)CCn2cncc2C1.c1c2cn(c(=O)c1)CC2 CC1=C(C(=O)NCC2CC(C)N(C(c3cnccn3)=O)C2)CCCC1 C12(CNC(CC3(C)CC3)=O)CCC(CC1)N(C(c1cn(C3CCOC3)nn1)=O)C2 CC1=C(C)CC(C)(C(N2C3CCC2CC(NC(c2cnc(C)cn2)=O)C3)=O)CC1 C1(CC=C)(NC(c2ccc(OCC)cc2C)=O)CCCN(C(c2cn[nH]c2)=O)C1 Cc1nn(C)c(Cl)c1CC(=O)NC1(CNC(c2cccc(OCF)c2)=O)CCC1 C(=O)(CS(=O)(=O)CC(C)C)NCC1C(NC(CSCC#C)=O)CCC(C)(C)C1 N1(C(Cc2n[nH]c(=N)s2)=O)CCCCC(CNC(=O)C(c2ccccc2)F)C1 c1(CCNC(=O)NC2N(CC(CCC)C)CC2)noc(=O)n1C Cc1c(NC(=O)NC(C)C(C)(C)CO)cnc(F)c1Br C(=O)(C(O)C(C)(C)C)N(CCCNC(=O)CC1CCCOCC1)CCC N1(C(C(C)(C)CC2CC2)=O)CC2CCC1CC2NC(c1ccnn1C1CCC1)=O c1(C(N2CC(NC(=O)C(O)c3ccco3)C3(C2)CC3)=O)cccc2nc(O)[nH]c12 C1(C(=O)NCCCNC(c2ccnc(N3CCCC3)c2)=O)CCN(C2CC2)C1=O C1(O)(CC(C)N(C2CC3(C(=O)O)CC23)C)CN(C(=O)OC(C)(C)C)C1 C1(CNC(Cc2c(C)ocn2)=O)C(O)C(O)CN1C(c1cncc(Br)c1)=O n1(CC(=O)NC(CNC(c2ccnnc2)=O)C2CCC2)cc(Cl)c(O)nc1=O c1(C(=O)NCC2CC(NC(CC(CC)C)=O)C2)cccc2[nH]c(=N)oc12 C(=O)(C1=CCC(C)(C)CC1)N(CCC(=O)N(C12CC(C1)C2)C1CC1)C(C)C c1(C(=O)NCC(C2CCCCC2)C)cc(C2CC2)nn1-c1ccc(Br)cc1 Cc1c[nH]c2cc(C(=O)NC3CCN(Cc4c(F)cccc4Br)CC3F)ccc12 C1(C(N(C2CCCN(C(C(F)=C(C)C)=O)C2)CCO)=O)CCc2c[nH]nc2C1 C1(O)(NC(N)=O)CCN(C(=O)C(O)C2CN(C(C3CN(C4COC4)C3)=O)C2)C1 c1(C(N2C(CNC(=O)COCC3CCOC3)CC2)=O)c[nH]nc1[N+](=O)[O-] CCCCCCCCCC=CC(=O)NCCCN(C(=O)Cc1cnns1)C C12(CC(=O)N(CCC)CC3CC3)CC(CO1)N(C(=O)CC(=O)OC)C2 CC1CCC=C1C(=O)NC1CN(C(c2cc(Br)cs2)=O)C(C)(C)C1 C1(C(=O)NCc2c(C)coc2C)CN(C(c2cnsc2)=O)C2(CCC2)C1 CC(C)(C(=O)N1CC2CC2(CNC(c2c[nH]nc2C(C)(C)C)=O)C1)C(N)=O C1(C)(NC(COCC#C)=O)CCN(C(C2CC2c2ccccc2)=O)C1 C=CC(CCC)CC(=O)NC(CNC(c1ccc(CC)[nH]1)=O)CC(C)C c1(OC)ccc2cc(C(=O)NC(C)CNC(c3cccc(F)c3)=O)c(=O)oc2c1 c1(C(N2C(c3ccc(C)cc3)CCCC2)C(=O)NCC2CC2)cccc(Cl)c1C c1(NCC(CC)(C)CO)ncnc(N2CCN(C(=O)NC)CC2)c1C C1(NC(C(=O)NCC(C)C)C)CCC(NC(=O)CCNC(=O)CO)C1 c1(C(N2CC(C(C)NC(c3n(C=C)nnc3)=O)OCC2)=O)ncn2ccccc12 c1(OCC)ccc(C(=O)NC2CSCCN2C(=O)C(O)CC)cc1[N+](=O)[O-] Nc1c(C(N2CCNC(C(F)(F)F)C2)=O)ccc(F)c1Br Cc1ccc(C(=O)NC2CCC(NC(=O)CN3CCCCCC3)CC2)c(F)c1F Cc1ccc(N(C(=O)CN(C)C2CC2)Cc2ccc(C)s2)cc1 N1(C(c2cc(CC)on2)=O)CCCN(C(=O)C(N2CCCC2CC)=O)CCC1 C(=O)(CCC(C(N)=O)NC(N1CCN(C(C)C)CC1C)=O)OC(C)C C1(C(=O)NCC2(F)CN(C(c3cnc(C)nc3C)=O)C2)C2CCC(C2)S1(=O)=O c1(NC(c2c(C3CC3)ccc(OC)c2)=O)cccc(S(C)=O)c1 C1(O)(C(=O)NC2C(NC(C3(C)CC4CCC3O4)=O)CCC2)CC2(CCOCC2)C1 C1(C(=O)NC2(CC(N)=O)CCN(C(c3ccc(C4CC4)o3)=O)C2)CCCCC(=O)N1 c1(C(=O)NCC2N(C(c3cn(C)c(=O)n3C)=O)CC=C2)cnc2c(n1)CCCC2 C(=O)(CCCCCC(C)C)NC(CC#C)(C)C(=O)N(C)CC1CCN(C)C1 n1(CC(=O)NCCC2CCC(NC(C3(CC)CC3)=O)C2)ccc2cc(F)ccc12 C1(C(N(CC(CC)NC(c2cnn(CC)c2C)=O)C)=O)C=CC=CC=C1 C1(C)(C(N2CC(C)N(C(C3CCOC(C)C3)=O)CC2)=O)Cc2ccccc2C1 c1(N2CCC(NCC3(OC)CCSCC3)C2)c(OC(C)C)cccc1Cl C(=O)(CC1=CCCCC1)N1C(C2(NC(C(c3cccc(C)c3)C)=O)CC2)CCC1 c1(C(C)C)ccc(C(=O)NC2CCCCC2NC(=O)CC(C)(C)C)cc1Cl C12(C(N(CCCOC)C)=O)CCC(CN1C(c1cccnc1OC(C)(C)C)=O)C2 O=C1CCc2cc(C(N3CC4CC3CN4C(C3CC3(Cl)Cl)=O)=O)ccc21 c1(C(=O)NCC(N2CC(CNC(CC(C=C)C)=O)(OC)C2)=O)ccc(F)cc1F Cc1ccc2cc(C(=O)NCC(N3CCC(O)CC3)c3ccccc3)ncn12 C1(NC(c2ccc(CSCC)cc2)=O)CCCN(C(c2conc2C)=O)CC1F N1(C(c2c(CC)occ2)=O)CC2CCN(C(c3ccc(C(F)F)cc3F)=O)CC12 CCC(F)(F)C(C)(C)NC(=O)CC1C=CC(NC(=O)C(C)OC(C)(C)C)C1 c1(CN(CCCP(C)(C)=O)C(C)(C)C)ccc(F)cc1Cl C(=O)(CC(F)(F)CC(=O)OC)N1C(C)(C(=O)Nc2cc(OC)cc(Cl)n2)CC1 C1(NC(C=CC=C)=O)CCCN(C(c2cncn2C(F)(F)F)=O)C1 C(N=c1[nH]c(Cl)ncc1Cl)C1CCN(C(C2ON=C(C)C2)=O)CC1C c1(NC(C(C)N(C(CC#C)C(=O)OCC)C)=O)cccc2ccoc12 Cc1ccc2c(=NCC3CC4(C3)CC43CCC3)[nH]c(=NC(C)CN(C)C)[nH]c2c1 C1(NC(c2ccc(C(=O)NCC3CC3)cc2)=O)CC(O)C(O)CO1 c1(C(=O)NC2CCC2)cccnc1CNC(C1CCCCC1F)=O CCC(C)(C(=O)N(C)C(C1CN(C(=O)C(C)C2(O)CCC2)C1)C1CC1)OC C1(CN(C(C)(C)C)CC=CC(=O)OC)CC(NC(=O)C(F)CC2CCC2)C1(C)C c1(CC(=O)NC2CC(NC(c3cccc4nncn34)=O)C2)ccc2c(c1)COC2 c1(C(N2CC(NC(CCCN(C)C)=O)C(F)(F)C2)=O)cc([N+](=O)[O-])c(F)cc1F c1(CNc2cncc(-c3c(C#N)nccc3)c2)c(Cl)ccc(F)c1F C1(CNC(Cn2c(C)nnn2)=O)CC2(CCC2)CN1C(c1ccc(F)c(N)c1)=O C=Cc1ccc(C(=O)NC2CN(C(c3csc(Br)n3)=O)CC2OC)cc1 CC1=CC(C)=NS(=O)(=O)N1CC(N1CC2C(NC(=O)C(C#N)C(C)(C)C)C2C1)=O c1(C(C(=O)NC2CC(NC(=O)Nc3cc(OC)ncn3)C2)OC)c(Cl)cccc1Cl n1(CC(=O)N(C(C)CNC(=O)C(C)(C)CCOC)CC)nc(Cl)ccc1=O c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccc(F)cc1OC N1(C(C(C)=C(CC)C)=O)CCC(NC(=O)Cc2ccc(F)cc2)CC1C N1(C(C=C2CCN(C)C2)=O)CCOC2(C1)CN(C(=O)CCn1cnnn1)C2 N(C(=NCc1ncc(Br)cn1)NC(C)Cc1ccccc1)Cc1c(C)ccs1 N1(C(CN(CCCC)C)=O)CCCC1C(O)CO C1(C)(CNC(c2cnc(OC)s2)=O)CC(F)(F)CN1C(=O)CN(C1CCSC1)C C(C(O)CC(F)(F)F)NC(C(CNC(c1cc(CO)on1)=O)N(C)C)=O N1(C(CC(CC)C)=O)CCCC2C1CCN2C(=O)CCCCCl C(=O)(N=c1[nH]n(C)cc1P(C)(C)=O)NC1C(CC)CN(S(C)(=O)=O)CC1 Cc1csc2c(CC(=O)NC3(C4CN(C(=O)C(C)(Cl)Cl)C4)CC3)cccc12 N1(C(C2C(CC)CN(C(=O)C=Cc3ccoc3)C2)=O)CCCSCC1C c1(C(=O)NCCC(CNC(c2csc(S)n2)=O)O)c[nH]c(=O)c2ccnn12 C1(C(=O)NCC(CC(C)C)NC(=O)CCc2cncnc2)CN2CCC1CC2 C1(NC(C(c2ccccc2Cl)C)=O)CC2(C1)CC(CNC(=O)CC1CC(F)C1)C2 S(=O)(=O)(c1ccc(C)c(C)c1)NCC(N1CCCC(CNC(CSCC)=O)C1)=O C(c1cncc2ccccc12)=CC(N1CC2NCCOC2C1)=O c1(OC)cnnc(C(N2CCCCC2C(N2CCCC2CN=[N+]=[N-])=O)=O)c1 C#CC1CN(C(=O)NC(c2cc(C)on2)C)CCN1C(=O)OC(C)(C)C C1(=O)CCCC(=O)N2CCCC(CC2)N1.C(=O)(C(C)(C)C)N(C)C C1(CNC(c2c(OC)csc2)=O)CC(NC(=O)C=C(C)Cl)C1(C)C Cc1ccc(C)c(C(N2CC(CNC(=O)Cc3csc(Cl)n3)CCC2C)=O)n1 c1(CC(N2CC(F)(CNC(C3C(C)CCC3)=O)C2)=O)ccc(Br)c(Cl)c1 C1(NC(CC(C)SC)=O)CC2(C1)CC(NC(=O)Cc1c(Cl)cccc1Cl)C2 c1(C(N2CC(CNC(c3c(C)nc(C4CC4)s3)=O)C2)=O)ccc(S(C)(=O)=O)cc1 c1(C(=O)NC2CCN(C(CSCC)=O)C(C)C2)ccc(C)c(Cl)c1Cl N1(C(c2ccc(C(C)=O)cc2)=O)CCC2C(NC(c3ncn(C)n3)=O)C2CC1 c1(C(N(C)CCN(C)C(c2cnc(C3CCCO3)s2)=O)=O)cc(=O)cc(Cl)[nH]1 N1(C(CNC(CCC)=O)=O)CCCC1C(C)(C)CNC(=O)Cc1ncc(Br)s1 N1(C(=O)OC(C)(C)C)CC(O)CC1C(N1CCC(NC(c2cc[nH]n2)=O)CC1)=O C1(C(N2CCC(C(=O)OC)CC2)=O)CNC(=O)CN1C(c1cc(C2CC2)cs1)=O Cc1nn(C)c(F)c1C(=O)NCc1ccccc1CNC(C1COCC(C)O1)=O N1(C(c2cc(OC)c(Br)s2)=O)CCC(C)(c2cn(-c3cncc(Cl)c3)nn2)CC1 c1(C(C)O)cn(CC(=O)NCC2(NC(c3cc(Cl)no3)=O)CCCC2)nn1 CC(Cc1ccccn1)C(=O)NCCCNC(=O)CNS(=O)(=O)CCOC1CC1 N1(C(C(C=CCCC)O)=O)C2CCC1CN(C(c1cccc(CC#N)c1)=O)C2 C(CNC(c1cnn(C2CCC2)n1)=O)(C(C)(C)C)NC(CCC1C(C)C1)=O C1(C(=O)NC2C(OC)CN(C(c3cc[nH]n3)=O)C2)CC(=O)NC(=O)N1 C(=O)(C1CCc2c(Cl)cccc21)N1CC(O)(CNC(C(C(C)(C)F)(C)F)=O)C1 c1(CCC(=O)NCC2CCC(NC(=O)CNC(=O)C3CC3)C2)cccnc1Cl C1(F)(C(=O)NC2CCN(C(Cn3c(C)c(Cl)cn3)=O)C2)CCC2(CCC2)C1 C1(CNC(CC(C)SC)=O)CC(C)(C)CN1C(c1coc(N(C)C)n1)=O C1(CC(=O)NCCOC2CCN(C(=O)CC3CC3)C2)CCCOCC1 C(C(=O)N1CC=CC(C(=O)NCC2(N(C)C)CCCC2)C1)(C(C)(C)C)OC c1(OC)cc2c3c([nH]c2cc1Cl)CCN(C(=O)NCC1CCOCC12CCC2)C3 N1(C(c2nccc(OC)c2)=O)CCC2CN(C(=O)CCCCCC(C)C)CCC12 N1(C(c2cc(CC)on2)=O)CCCOC(CNC(=O)Cc2ccco2)C1 C1(C2N(C(CCOC(C)=O)=O)CCC2)CCCN(C(c2ccn(C)n2)=O)C1 C(=O)(C1CCc2snnc21)NC(CCCNC(CC(CC)(C)C)=O)CO c1(C(=O)NC(CNC(COC(C)C)=O)(C)C)coc(C(N)=O)c1 C(=O)(C1=CC2CC=CCC12)NCCC1(NC(c2c(CCC)nco2)=O)CC1 c1(OC)cc(C(=O)NC2CC(F)CN(C(=O)CCOC(C)=O)C2)c(Cl)cc1Cl CC1CN2CCN1C(C(N1CC(CNC(C3CCS(=O)(=O)N3)=O)CC1(C)C)=O)C2 N#CCCCCCC(=O)N1CC(F)CC1CNC(=O)C=Cc1cccc(Cl)c1 c1(C(=O)NC2C(NC(C3N(C(C)C)C(=O)CC3)=O)CCC2)ccccc1[N+](=O)[O-] C1(C(N2CC(COC)C2)=O)COC(CNC(=O)C(C)CO)C1 C(=O)(CCCCC(F)F)N1C2CC(CNC(=O)C3=CCCCO3)(OC2)C1 Cc1ccc(C(N2CCC(C)(NC(c3cccc(O)c3C)=O)C2)=O)cc1C N1(c2nc(SC)c(C)cn2)CCOCC12COCCN(C(C1CCCOC1)=O)C2 CC(C)C(C#N)C(=O)N1CCC(CNC(=O)CCc2nncn2C)CC1C c1(C(=O)NC(CN(C(c2cc(C(C)C)ccc2F)=O)CC)C)cnc(N)c(N)c1 C=CC(CC)CC(=O)NC1CCN(C(c2ncsc2C)=O)CC1CC N1(c2cc(N(C)CC3CC=CCC3)nc(COC)n2)CCCC2(C1)CC2(F)F CC1COCCC1CN(C=O)Cc1ccc(C(F)(F)F)cc1 C(=O)(C(C(=O)NCC1CCCC1C(=O)NC1(c2ccccc2)CC1)OC)OC N1(C(CCCn2c(C)ncc2)=O)CCN(C(=O)CC2(C(F)(F)F)CC2)C(C)C1C S(=O)(=O)(c1sc(Cl)nc1-c1ccccc1)N(C(C)C)C(C)C CC(C(=O)NC(CCF)C(=O)NC(CCO)C1CCCC1)C(F)(F)F N1(C(c2ccc(OC)o2)=O)CC2(CC1CNC(c1occ(C)c1C)=O)CC2(F)F C1(N(C(C2CC3(CC3)C2)=O)CCF)CCCN(C(c2csc(C(F)F)c2)=O)C1 N1(C(=O)Nc2cnc(C)s2)CC2CN(C(=O)CCC(C)(C)NC(C)(C)C)CC2C1 CC#CCCC(=O)N(CCNC(=O)Cc1cc(C)sc1C)Cc1ccccc1 N1(C(CNc2n(C)c(S)nc2)=O)CC2CC(NC(C3CC4COCC4C3)=O)C1C2 Cc1nn(Cc2ccccc2)cc1C(=O)Nc1cnn(C2CC2)c1 C1(C(=O)NC2CC(C(C)(C)C)C2)CCN(C(c2cnc(O)o2)=O)CC1O C1(C(=O)NCC(CC)(C)NC(=O)CCc2ccnc(C)n2)CSCC(=O)N1 C=CC1CN(C(=O)CN(C)CCC)CC1NC(c1ccc(-n2ccnc2)nc1)=O C1(CC=C)(NC(=O)C=CCF)CN(C(=O)C(CC)n2ccc(C3CC3)n2)C1 C1(CNC(C2CC2(Cl)Cl)=O)CCN(C(c2csc3nnsc23)=O)C12CC2 CCC(C(=O)NC1(C(=O)NCC2CC2Cl)CCCC1)n1ccnc1 C(CC(F)F)(C(=O)N(CCCCCO)C)NC(C(C=C)C)=O C12(CNC(C(N)=O)=O)CN(C(c3ccc4cnoc4c3)=O)CC1CCO2 C1(NC(C2C(C)C2)=O)CCN(C(=O)Cc2coc3cc(F)ccc23)CC(C)(C)C1 C1(NC(CCCCN(C)C)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1F C1(C(=O)O)(C(=O)O)CC=CCC1.CC(C=O)OC1CN(C)C1 c1(CCCC(=O)NCC(CN(C)C(C2CC3CCC3C2)=O)O)ccc(Cl)cc1 C1(C(=O)NCC2CCN(CCCC(F)(F)F)C2)C2CCN1CC2 C(C(C(C)C)NC(=O)COCC(=O)NC(=O)C(C)=C(C)C)OC c1(C(=O)NCCOC2CCN(C(C3C(CC(C)C)C3)=O)C2)ccc[n+]([O-])c1 CCCCCCCC(=O)N1CCCCC(NC(=O)CN2CCOCC2)CC1 c1(OCC)ccccc1OCC(=O)NCC1CCN(C(c2nn(C)cc2Cl)=O)C1 C1(NC(=O)CC2OCCCO2)CCCC(NC(c2cc(C(F)(F)F)cs2)=O)C1 c1(C(=O)NC2CCN(C(c3cc(C)ncc3)=O)C(C)C2)c[nH]nc1S(N)(=O)=O c1(C(=O)NCC(C)(C2CC2)NC(C2N(CC)CCC2)=O)cc(N)c(F)cn1 N1(Cc2cn(C(COCC)C(=O)NC)nn2)CCN(C)CC1c1ccccc1 c1(C(N2CCC(CNC(CCCC(=C)C)=O)C2)=O)ccc(N)c(F)c1Br c1(C(=O)NCCC(CNC(COCCCC#C)=O)O)cnn2cccc(Cl)c12 C(=O)(C(O)CCN(C)C)NC(CC)CN(C(=O)CCc1ccncc1)C C1(O)(c2cn(CCC(C)C)nn2)CCN(C(C2COC(C)(C)CO2)=O)CC1 c1(C(=O)NCC2CN(C(C(C)SC)=O)CC(C)(C)C2)ccc(S(C)(=O)=O)cc1Cl C1(NC(c2cc(OC)ncc2F)=O)COC2(C1)CN(C(c1ccc[nH]1)=O)C2 N1(C(C(CCC#C)O)=O)CC2CCC(C1)N2C(=O)C(CCC)NC(N)=O c1(C(=O)NCC2C(NC(c3c(C)onc3)=O)CCC2)c(C)nc2ccnn2c1C C(=O)(CCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(C(F)F)CCC2)=O)C1)OC Cc1ccc(C(N2CC(N(C)C(C3CC34CCC4)=O)C2)=O)nc1 c1(OC)cccc(NC(=O)C(c2ccc(Cl)nc2)N(C2(C)CC2)C)c1 C1(CC)(NC(c2sccc2OC)=O)CCCN(C(c2ccns2)=O)C1 CCC(CNC(=O)C(C)CSC)(CC)NC(C1OCCOC1C)=O CC1CC(CCNC(c2cc(O)cc(Cl)c2)=O)CCN1C(=O)Cn1cnnn1 N1(C(c2onc(C)n2)C)CCC(NC(C2(C)CCCC2C)=O)C(C)(C)C1 N1(C(C(CC)C(C)C)=O)CCN(C(c2cc(C)n(CCO)n2)=O)CC(O)C1 O=C1COc2cc(C(=O)NC3CCN(C(c4ccc(Cl)nc4O)=O)C3)ncc2N1 C=CCCC(C(=O)NCC(Cl)=CCl)NC(C1CC(C)CC(=O)N1)=O C1(CN(C(C2CCCOCC2)=O)CC)CCN(C(=O)C#CC(=O)N(C)C)CC1 C1(NC(c2nc(COC)oc2)=O)CC2CC1CC2C(N1CCCC(C#N)C1)=O C1(C(=O)NCCN(C(=O)C(c2c(C)noc2C)CC)CCC)CCOC(C)(C)C1 Cc1nn2c(c1C(N1CCC1CNC(=O)CC1(CO)CCCO1)=O)NCCC2 N1(C(C2OCCN(C)C2)=O)CCN(C(=O)COc2ccccc2O)C2COCC12 C(=O)(C(C1CCCC1)NC(=O)C(=O)NC1CC1)NC(c1ccns1)C C12(CC)CN(C(=O)C(O)COc3ccc(OC)cc3)C(CNC(=O)C(C)O)(C1)C2 N1(C(C(C)=C2CCC2)=O)CCCC1(C)CNC(c1ccnc(C(N)=O)c1)=O C(C(C)(C)CC(=O)N1CC(O)(C(F)C(N2CCOC(COC)C2)=O)C1)OC N1(C(CCC#CC)=O)CC2CCCC2(NC(c2cc(OC)ns2)=O)C1 C1(NC(c2c(C)ccs2)=O)CC(O)CN(C(=O)CC2CCC2)C1 C(C1=CCCOC1)NC(C1CCC(NC(C(C)(C)n2cnnn2)=O)C1)=O c1(CC)ccoc1C(=O)NC(c1cn(C)nn1)C(=O)NCCC1(C)CCCO1 c1(CC)cc(C(=O)NC(C(=O)NCCc2nccc(C)n2)C2(O)CCC2)c(C)o1 c1(CC(=O)N(CCOCCNC(C2(CN(C)C)CC2)=O)C)ccc[nH]1 N1(C(CCC)=O)CC(NC(=O)C(C)NC(=O)Cc2ccccc2)CC(C)(C)C1 CC1C(C)N(C(=O)CN(C)S(=O)(=O)N(C)C)CCN1C(C1CC(O)C1)=O CCC(C)(C)C(C)CC(=O)N(CCCNC(=O)C(Cl)=CCl)C1CC1 c1(CC(=O)NCCCCNC(c2cn(C)nc2Cl)=O)coc2cc(O)ccc12 CC1CCCC(C(N2CC(CCNC(C3(CO)CCCCC3)=O)C2)=O)C1 N1(C(C2C(CC)OCC2)=O)CCC2(CCCN2c2ncc(F)cn2)C1 c1(OC)ccc(C(=O)O)c(C(F)(F)F)c1.c12ccc(cc1)CC(=O)N1CCC2C1 N1(C(C(C2CCC2)OCC)=O)CCC(C(C)(C)NC(=O)C(C)n2ccnc2)CC1 c1(OC(C)C)cc(C(N2CCC(CNC(C3CCC(C)S3)=O)CC2)=O)ccn1 CC(C)(C(F)(F)F)OCC(=O)NCC1CC1NC(=O)CCc1cccc(Cl)c1 c1(C(=O)NCC(C)(C2CC2)NC(C(C)CC(N)=O)=O)cc(Br)c2[nH]nnc2c1 CC(C)CC(CC(C)C)C(=O)N(C1C2CN(C(=O)C(C)N3CCC3)CC12)C N1(C(C2(CC)CCOC2)=O)CCCCCC1CNC(c1cc(C)cc(Cl)c1)=O Cc1cc(C(=O)NCC2CCN2C(=O)C=CCOc2ccccc2)cnc1O C1(CNC(C2(CC(C)C)COC2)=O)(NC(C2CCCCO2)=O)CCCCCC1 C1(C(=O)NCCc2cc(C)n(C)n2)CCN(C(c2cncc(Cl)c2)=O)CC1O c1(C(N2CCC(NC(Cc3c(C)ccc(Br)c3)=O)C2)=O)cc2cccc(C)c2[nH]1 c1(CC)cncc(C(=O)NC(CNC(c2cnn(C)c2)=O)(CC)CC)c1 Cc1ncc(S(N)(=O)=O)cc1C(=O)NC1C=CCN(C(=O)COC2CCOC2)C1 Cc1cccc(C)c1C(=O)NC1CN(C)CC1C.n12cc(nn1)C(=O)NOCC2 C1(C(N)=O)CCN(C(=O)CC2CC(NC(=O)CCCc3ccc(O)cc3)C2)CC1 C=CC(C(F)(F)F)NC(C1CC(O)CN1C(=O)CCC1CCCCO1)=O N1(C(C=CC(CC)=CC)=O)CCN(C(c2cc(C)n(C)n2)=O)CC1CC(F)F c1(OC)cc(C)cc(C(=O)NCC(C)CNC(c2ccnc(C(C)C)n2)=O)c1N Cc1cc(O)ccc1C(=O)NCC1CCN1C(=O)C(F)n1cccn1 c1(C(N2CC(CNC(C(C(=O)OC)C)=O)C2)=O)csc2ccc(F)cc12 c1(C(=O)OC)nn(C)c2ncc(S(=O)(=O)NC(CCCCCO)C(=O)O)cc12 c1(C(=O)NCC(CNC(C(C=C)O)=O)F)sc2cccc(F)c2c1COCC c1(C(N2CC(C)CC(NC(c3c(OC)cccc3)=O)C2)=O)ccc2c[nH]nc2c1 c1(Oc2c(Cl)ccc(C)c2)ccc(C#N)cc1Cl C(=O)(C1CCCn2ncnc21)NCC1CN(C(CCCSC)=O)CC1C(F)(F)F Cc1ccn(C)c(=NC(=O)N2CCC(C3CCCO3)CC2)n1 CC#CCC(C(=O)NC1CC2CC1CC2COC)NC(=O)CN(C)C(C)=O N1(C(c2c(CCC)n(C)nc2)=O)CCCC(NC(c2occc2C)=O)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)NCC(CC)NC(c1cccc(Cl)c1C)=O N1(C(c2cc(C)cc(C)c2N)=O)CCN(C(=O)CC(=O)NC2CC2)CC2(CC2)C1 C1(CNc2cccc(NC(C)(C)C)c2C)CC2C=CC1N(CC)C2.C(=O)(OO)SC C1(NC(COC(CC)C)=O)CCCCCC1NC(c1nc[nH]c1C(C)(C)C)=O c1(C(=O)NC(CC)(CNC(=O)CCCC2CCCC2)CC)ccc2ccnn2c1 c1(N(C(N(CCC)CCc2nc[nH]n2)=O)C)ccc(C)cc1Cl N1(C(C2(C(=O)OCC)CC2(F)F)=O)CCC(N(C)C(c2cc(Cl)ccn2)=O)CC1 C1(NC(C(COCC)NC(c2n(C=C)nnc2)=O)=O)CCn2cnnc2C1 C(C(=O)NCCOC1CN(C(=O)C(c2ccccc2)O)C1)(C(C)C)NC(=O)OC CC1CN(C(=O)CC23CCC(CC2)OC3)CC(C)N(C(=O)CC(O)C(C)(C)C)C1 N1(C(C(F)OC)=O)CCC2(CCOC2)C(CNC(=O)COc2ccc(F)nc2)C1 C(C(=O)N=c1cc2n([nH]1)CCCC2)C1CCN(Cc2n(C)cc([N+](=O)[O-])c2)C1 c1(C(N2CCC(NC(C(C)=C3CC3)=O)C2C(C)(C)C)=O)ccc(C)c(C)c1N C#Cc1cn(C)nc1C(=O)N(CC(C)O)CCNC(=O)C=CC1CCCC1 CC1(O)CCN(CC(N2CC=CC(NC(=O)CCN3CCCS3(=O)=O)C2)=O)C1 N1(C(C(C)Oc2ccccc2)=O)CC(CN(C(=O)Cn2nccn2)CC)C(F)(F)C1 CCN(Cc1nccs1)N1CCN(c2cc(Cl)ccn2)CC1 C1(CNC(C(C)(C)OCC)=O)CCC2CN(C(c3cc(C)ns3)=O)CC12 c1(-c2nc(C)on2)ccn2ccccc12.c12ccc(n1C)C1CCCN1C2=O.c1(CC)ccccc1 C1(CNC(C(CCCC)C)=O)CCN(C(=O)CSCC(N)=O)CCC1(F)F C1(C(=O)NC(C2(O)CCN(C(=O)CN3CCOCC3=O)C2)C)CC2(C1)CC2F c1(NC(C(COC)N(C)C)=O)cc(C)ccc1F CC(C)C(CO)ONC(=O)C=CCC1CC1.C1(C)(N(C)C=O)CC1C c1(C(=O)OCC)c(NCC(c2ccc(F)cc2)N)oc2c1COCC2 C1(C(C)(C)F)CCN(C(c2cc(Br)sc2Cl)=O)CC1 N1(C(CCN(C(=O)Cc2nnc(C)o2)CC=C)=O)CCN(C)CC1C C1(C(=O)NCC(CC)(CC)NC(=O)CC2SC(=N)NC2=O)CC(C)(C)CN1C CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1ccccc1C(F)(F)F)=O Cc1cc(CNC(=O)CC2CCSCC2)oc1C S(=O)(=O)(CC(=O)NCCC(C)CCO)N.C(CC(=O)N)NS(C)(=O)=O C1(C(=O)NCC2CC(NC(C=CC(C)C)=O)CC2O)Cc2c(F)cccc2O1 Cc1nc(CC(=O)NCC#CCNC(=O)CSC(F)F)c(C)s1 N1(C(C=C(C)Cl)=O)CCCC2CN(C(C3COc4ccccc4C3)=O)CC12 C(CC(=O)N1CC2(CC(N(C)C)C2)C1)(C(F)F)NC(C(CC#C)O)=O C1(CS(C)(=O)=O)(CN(CC(=O)O)C(=O)Cn2cc(CN(C)C)nn2)CC(F)(F)C1 C1(C(=O)NC2CN(C(c3nc(Cl)c(Cl)s3)=O)CC2O)CC2COCC2C1 c12cccc(n1)C(=O)N2.N1(C(C2CCC(C(=O)OC)C2)=O)CCCC(F)C1 Cn1nnc(=NS(=O)(=O)c2cccc(NC(=O)C3CCCn4cnnc43)c2)[nH]1 Cc1ncc(Cl)cc1C(=O)OCC1CCCCC1(C)C C1(C(C)=O)CC(C)CN(C(c2cnc(Cl)c(F)c2)=O)C1.c12n[nH]cc1NC2=O C12CCC(C=CC(=O)N1)C2.c1(C2C(N(C)C)CCC2)ccc(C(F)(F)F)cc1 C1(C(C)NC(=O)CC2CC(=O)C2)CCN(C(C2(CF)CC2)=O)C1 C1(NC(C=CCNC(CSC(C)(C)C)=O)=O)CCNC(=O)CC1 C1(CC(=O)NCC2N(C(C(c3ccccc3)OC)=O)CC2)CCCNC(=O)C1 c1(C(N(CCCn2cc(CN(C)CC)nn2)C)=O)cnc2scnc2c1 C1(OC)(CNC(=O)C(CO)N(C)C)CCN(C(=O)C(c2cncn2C)O)C1 C1(NC(Cc2c(C)noc2)=O)CCCN(C(=O)Cn2cnnc2)CC1 C#Cc1ccccc1CNC(=O)C(C)N(C(C1CN2CCN1CC2)=O)C1CC1 C1(NC(CCCC#C)=O)CN(C(C2CCCC(C)(C)O2)=O)CC2(CCOCC2)C1 CC(C)C(C(C)NC(c1coc(Cl)n1)=O)NC(c1cn(CCC2CC2)nn1)=O C1(C(=O)NCC2(CN(C(C(CC)OC3CCCC3)=O)C)CC2)CCCC12CC2 c1(N2CC3C(C(=O)NCC(C(C)C)(F)F)C3C2)ncc2ccccc2c1N N1(C(CCSCC)=O)CCCC(O)(CNC(C2CC2C)=O)C1 CCCC(C(=O)N1CCC(NC(c2nc(O)sc2C)=O)C1)NC(C)=O N1(C(c2c(C)nco2)=O)CC(NC(c2ncnc(O)c2Cl)=O)CC(C)(C)C1 c1(C(N(C2CC(NC(C3(F)CC3C)=O)C2)C)=O)nsc2cc(Br)ccc12 c1(Sc2ccccc2)ccc(Cl)cc1CN(CC=C)C1CC1.OC C#Cc1cc(F)c(C(N2CCC(NC(c3ccsc3Cl)=O)C(C)C2)=O)cc1F c1(NC(c2ccccc2)CC)cccc(N(Cc2cnn(C)c2)CC)c1 C12(NC(CCC)=O)COCCC1CN(C(=O)CCc1cn(C)nn1)C2 N1(C(C(=O)NCCOCCCC)=O)CCC(C)(NC(=O)C2=COCC2)C1 c1(OC)ncnc(N2CCCC(CO)(NC(C3CCCC3O)=O)C2)c1OC N1(C(C2C(C=C(C)C)C2(C)C)=O)CCN(C(c2ccsc2C)=O)C2(CCC2)C1 N(C(=NCC1CCCN1Cc1cnccn1)NC1CCCC1)C1CCN(CC)C1 C1(NC(C2C(C(C)O)C2)=O)CCC2CC1CN2C(C12CCCC1C2(F)F)=O c1(C(=O)NC2C(C)N(C(c3[nH]nc4ncccc34)=O)CC2)nnn2ccccc12 C#Cc1ccc(Cl)c(C(=O)NCCN(C(=O)C(O)CC(C)(C)C)CCOC)c1 c1(NC(C2CC(NC(CSc3nc(C)[nH]n3)=O)C2)=O)n[nH]c(C)c1F Cc1ncnc2c1CC(C(N1CCN(C(=O)CP(C)(C)=O)C(CCO)C1)=O)CC2 N1(Cc2c(OC)cc(Br)cn2)CCc2c(C(=O)Nc3cccc(C)n3)n[nH]c2C1 C(CCCCCNC(C1(C2CC2)CCCO1)=O)N(C)C(c1cn[nH]c1)=O Cc1ccc(-c2n[nH]cc2C(=O)NCCOCCN(C(=O)CC(C)(C)F)C)cc1 c1(CN2C(CC(=O)Nc3cc(C)c(Br)cc3F)COCC2)ccc(O)c(C#N)c1 c1(CC(=O)NC2C(NC(CC(CCC)O)=O)CC2)cc(F)c(C)cc1F C1(C(N2CCCC(NC(c3nn(C)c(Cl)c3)=O)C2)=O)CCCOC1(C)C CCCC(CCCNC(c1c[nH]nc1CC)=O)NC(C1ON=C(C)C1C)=O Cc1cccc(-c2cn(C3CC(NC(=O)CCCF)C3)nn2)c1N(C)C Cc1cc(F)ncc1NC(=O)CC1CCN(C(=O)CNC(C)C)C1 N1(C(C2N(C(C)C)C(=O)CC2)=O)CC2CCN(C(c3cc(Br)n[nH]3)=O)C2C1 CCCC(CC)C(=O)NC(C)(CNC(C1(CF)CC1)=O)CC(C)C N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)Cn2nc(C)cc2C)C1(C)C N1(C(CC)=O)CCCC(C2CN(C(=O)COc3ccc(C)cc3)C2)C1 C1(C(N2CC(C)(CCC(=O)NCCCCCN=[N+]=[N-])C2)=O)OCC2CCCC12 c1(C(=O)NC2CC(CNC(CC3CCC(=O)C3)=O)C2)ccc2ncsc2c1 c1(C(=O)NCC(C2CCOC2)NC(c2n(CC#C)ccc2)=O)csc(C)c1C c1(C(=O)NC(C)CN(C)C(C2(C)CCSCC2)=O)cc2cccc(F)c2s1 c1(C(N2C(C(C)NC(=O)C=C3CCC3)CCC2)=O)cncc2[nH]ccc12 c1(CNC(C23CC(Nc4cc(OCC)ncn4)(C2)C3)=O)ccc([N+](=O)[O-])c(O)c1 c1(C(N2CC3CC3(CNC(C34CCCC3OCC4)=O)C2)=O)n[nH]c2c1COCC2 C1(CC)CN(C(=O)CC(C)N(C)C)CCN1C(c1ccc(OC(F)F)cc1F)=O N1(C(c2c(C)n(C)cc2)=O)CCOC2(C1)CN(C(c1cccc3c1OCC3)=O)C2 CCCCC(O)CCC(=O)N1CC(NC(=O)C#CC2CCCCO2)C(C)C1 N1(C(CSN(CC)CC)=O)CCC2CN(C(=O)CSc3cccs3)CCC2C1 C(=O)(NNc1cc(CC(N)=O)ccc1Br)C1N(C(=O)OCC(C)(C)C)CCC1 C(C(O)CN(C)N1CCC2(Cc3ccccc3C2)C1)OC(C)C CC[Si]1(CC)CCN(C(=O)NC(c2cccc(C)n2)C)CC1 c1(C(=O)NC2(CC)CN(C(=O)CC(C)(C)O)C2)ccccc1Oc1cccnc1 C1(C(N(CC(=O)Nc2cnn(CCF)c2)C)=O)CCC(=O)CC1 N(C(=NCc1ccnc(OC(C)C)c1)NC1CCC(C(F)(F)F)CC1)C(C=C)C C1(C(=O)NCCC(C)NC(=O)CSc2n[nH]c(=N)s2)CCCCCCC1 C1(NC(CNC(C)=O)=O)CN(C(=O)CC2CC3(COC3)C2)CC1S(C)(=O)=O N1(C(C2=NOC(C)(C)C2)=O)CC(NC(c2cn(C3CC3)nn2)=O)CC12CCCC2 CC(C)(C)C1=NOC(C)(C(=O)NC2CC3CCC2(NC(=O)COC2CCC2)C3)C1 N1(C(c2c(F)ccc(C)c2)=O)CCOCC(C)(CNC(C2C3(CC3)C23CC3)=O)C1 CCC(CC(=O)NCC(CC(=O)NCC1(CC(=O)OC)CC1)OC)C(C)C n1(CC(=O)N(CCNC(CN(CCOC)C)=O)C)ncc(Cl)c1C c1(CC(=O)NC2(CO)CCN(C(=O)CCc3cnn[nH]3)CC2)ccc2c[nH]nc2c1 C1(NC(CCC#C)=O)CCN(C(c2ccc(OC)cc2OC)=O)C12CCC2 CN1CC(C)(C)CC1C(N1CC(CNC(=O)CSc2cccs2)C1)=O N1(C(c2c(OC)ccc(F)c2)=O)CCc2sc(CNC(=O)C(C)(C)OC)nc2C1 C1(NC(c2ccn(CCC)n2)=O)CCC2CN(C(=O)C(C)COC)CCC2C1 CC(C)C(C)N(C)CCN(C)CCN(C)C.C1(=O)C(C)O1 c1(C(=O)NCC2(NC(C3C(OC)C3)=O)CCCC2)[nH]c2ccc(F)cc2c1C n1(C(C)C)ncc(C(N2CCCC2C(C)NC(C2(C(F)(F)F)CCC2)=O)=O)c1N c1(C(=O)NCCCOCCN(C)C(C2CCC3(CCC3)C2)=O)cc(F)cc(Cl)c1 c1(C(N2C(CO)CC(NC(C3(C)COC(=O)C3)=O)C2)=O)cc2ncccn2n1 c1(C(N(C2CCN(C(=O)CCn3ccnn3)C2)CC#C)=O)csc(CCC)n1 C12(NC(CCCOC(C)C)=O)CCN(C(c3cncc(N(C)C)n3)=O)CC1C2 c1(C(=O)NC(C)C(C)NC(c2ccc(F)cn2)=O)cc(N)nc(Br)c1 C1(CCCC)CN(C(C2CC(C3CC3)=NO2)=O)CCN1C(c1sc(C)cc1Cl)=O c1cnc(N2CCNCC2)c(-c2nc(-c3cnc(-c4ccccc4)s3)no2)c1 C(=O)(CCS(N)(=O)=O)N1CCC(C(CNC(C2N(C(=O)OCC)CCC2)=O)F)C1 Cc1[nH]c(=N)[nH]c(=NCCC2CC(C)(C)NC2=O)c1Cl C(CC(=O)N(CCCC(C)C)C)(C(F)(F)F)NC(C(CC)C(C)C)=O C(=O)(C1=CCCOC1)NC1CCN(C(c2c(C(C)C)ncnc2)=O)C1 C1(C(=O)Nc2cccc(CNC(C=C(COC)C)=O)n2)CCC=CCCC1 c1(C(N2CC(NC(=O)C#CC3CC3)CC(C)C2)=O)ncnc2sccc12 CC(C)CC(CNC(c1cn(CC(F)(F)F)nn1)=O)NC(=O)C(F)C(C)C c1(OCC(=O)NC2CCN(C(CC)=O)CC2O)cc(F)c(F)cc1F N1(C(=O)OC(C)(C)C)CCC(CO)(CNC(=O)CC2CC=CCC2)C1 N#CCCCCCC(=O)N1CCC2CN(C(=O)CN3CC4CC4C3)C2C1 c1(C(=O)NC2CCN(C(Cc3scc(CC)n3)=O)C(C)C2)ccc2ccsc2c1 c1(C(N2CC(C(C)NC(C3C(C=C)C3)=O)C2)=O)cc(OC)cc(Br)c1N CC1CCN(C(c2cn(C(C)(C)C)nn2)=O)C1CNC(c1ncoc1C1CC1)=O CC1(C)OCC2CC12C(N1CCOCC(NC(=O)CCCC2CCCC2)C1)=O CC(C)CC(C)C(=O)N1CCCC(CCNC(=O)Cc2ccn(C)n2)C1 c1(C(=O)NC(C2(CNC(C3(C)CCCCC3)=O)CC2)C)ccnc2ccncc12 C(=O)(CC1=CCN(C)CC1)N1C(C)CCN(C(=O)CC2(C)CCOC2)CC1 c1(OC)cc(C(=O)N(CC(C)NC(C2CSCN2C(C)=O)=O)C)ccc1F C1(NC(c2cnc(Cl)[nH]2)=O)CN(C(c2scc3c2CCCC3)=O)C2(CCC2)C1 C(=O)(C(O)CC(N)=O)NCC1(O)CC(CNC(c2cnn(C)c2C(F)(F)F)=O)C1 C(=O)(C1CCc2cccc(F)c21)N1CCN(C(C(CCSC)OC)=O)C2(C1)CC2 c1(CC(C)C)nccc(C(=O)NCC2(C)CCN(C(C3(F)CCOC3C)=O)C2)n1 N1(S(CCOC(=O)CCc2ccc(F)cc2)(=O)=O)CCN(CC)C(C)C1 N1(C(c2n(CC=C)ccc2)=O)CCC2(CCN(C(C3CCCN3C)=O)C2)C1 c1(NC(C2N(C(c3c(C)nc(Cl)s3)=O)CC2)=O)c(Br)cc(Br)c2ccccc12 C(C(C)(C)CC(=O)O)NCCCc1c[nH]c(C)c1CCC(=O)OC.C(C)C c1(C(=O)NCC2(CNC(COCC=C)=O)CC2)ccc(F)c(C(=O)CCC)c1F C1(CNC(c2n(C)ncc2)=O)COC(C)(C)CN1C(=O)Cc1cn(C)nc1Cl C1(C(=O)NC2CC(NC(CC(C=C)(C)O)=O)C2)CCC2C(C1)C2(F)F C1(O)(CNC(=O)CC2CC2)CC(C(=O)NC2CC(N(C)C)C2)C1 c1(C(=O)NC2(CCNC(CC3C(C)C3)=O)CCC2)ncccc1C(F)F N1(C(C2N(C)C(=O)OC2)=O)CCOCC(C(=O)NCC2CCCS2)C1 c1(SC)ccc(NCC(N2CCN(c3ncccn3)CC2)=O)c(Cl)c1 c1(CC(=O)Nc2c(C)nn(CC(=O)OC)c2C)ccc2c(cnn2C)c1 CCC(C)C(C)C(=O)N1CCOCC1CN(C(=O)C(F)CC1CCCC1)C c1(NC(N2C(C(=O)NC3CCN(C(C)=O)C3)CC3CC32)=O)cnccc1C(F)(F)F Cc1cc(C)c(C(N2CC(NC(=O)CC3CCC(F)(F)C3)C(C)C2)=O)c(=O)o1 Cc1nnc2n1C(C(=O)NCCC1CCN(C(C3CCS(=O)(=O)N3)=O)CC1)CC2 c1(C(C(=O)NCCCNC(Cn2c(C(=O)OC)cnc2)=O)CC)cccc(Cl)c1 C(C1CCN(C(=O)COC2CC3CC3C2)CC1)=CC(=O)N(C)C c1(SC(C)C)ccc(C=CC(=O)Nc2cc(C(F)(F)F)ccc2C)cc1 n1(CCOC)nnnc1C(CC1CCOCC1)NC(C1(n2cc(Br)cn2)CC1)C CC1CN(C(c2sccc2Cl)=O)CC1NC(c1ccc(C2CC2)cn1)=O N1(C(c2c(C)cncc2Br)=O)CCC2CN(C(C3CCCCC3O)=O)CC12 c1(CC(CNC(=O)CCSC2CCCC2)NC(=O)CC2C=CCC2)ccccc1 CCC(C)C(C(=O)NCc1cncc(OC)n1)NC(=O)CCC(C)(C)F Cc1cc(F)cnc1C(N1CCCCC1CCC(C)(C)NC(=O)C(C)O)=O C1(n2cc(C3(N4CCCC4)CCOC3)nn2)(C(=O)OC)CN(C(=O)C(C)=O)C1 C1(NC(C2CC(SC)C2)=O)CC(NC(C2(C(C)(F)F)CCC2)=O)CC1O CN1C(=O)C(=O)N(CC(=O)NCC2C=CC(NC(c3ccc(Cl)o3)=O)C2)C1=O C(=O)(CCCCC(N)=O)N1CCC(C)(NC(c2ccc(COC)cc2)=O)C1 c1(CC(=O)NCCCCc2cn(C3C(C)(O)CCC3)nn2)cc(F)c(Cl)cc1F C1(C(N(C)CC2COCCN2C(c2ccnc(S)c2)=O)=O)CCCCC2(CC2)C1 Cc1nc2ccccn2c1CC(=O)NCC1C2CN(C(=O)CN(C)C(N)=O)CC12 C1(C(=O)NCc2occ(C(N(C)CC3NC(=O)NC3=O)=O)c2)CC2C(C1)C2(C)C C1(CC)CC(C(=O)NCc2c[nH]nc2C(=O)Nc2ccc(C(C)C)nc2)CCO1 C(C(O)CNC1C2CCCC12)(OCC)OCC N1(C(c2c(C)ccc(O)c2)=O)CCC2CCN(C(c3cc(C(C)C)no3)=O)C2C1 C1(C(=O)NC(C(N2CCCC(CCF)C2)=O)C2CCOC2)CC2CC1CC2O c1(C(N(CCCNC(=O)C=C2CCSCC2)C(C)C)=O)ccn2nccc2n1 C1(CC(=O)OC)COC(CNC(=O)CC2CSCCO2)C1 c1(CSCC(=O)NCCC(C)NC(c2ccccc2)=O)csc(=N)[nH]1 C(=O)(CC(C)CC(C)C)NC1(CNC(C2CCCN(C(CC)=O)C2)=O)CCCC1 c1(C(=O)NC(CNC(c2ccc[n+]([O-])c2)=O)C2CC2)cccc2c1COCC2 C(CCS(C)(=O)=O)(C(=O)NCC1CCCCN1C(C1(SC)CCC1)=O)OC C=CCCCC(C(=O)NCC12CC(CN1C)C2)NC(=O)Cn1ccc(C)n1 C1(NC(CN(C2CC2)CC)=O)CCC2CN(C(C3CCCS(=O)(=O)C3)=O)CC2C1 CC1CCN(CCC(=O)NC2CC2NC(=O)CC2CC(=O)NC2=O)CC1 C1(C(=O)NCCCCC(N)=O)CCN(C(=O)CC2(O)CCOC2)C12CC2 C(C(=O)NCc1ccc2c(c1)OCO2)(C1=NOCC1)N1C(C)COCC1 N1(Cc2c(C)ncc(Br)c2)CC(NC(C2(CO)CC2)=O)CC2(CCC2)C1 N1(C(C2OCCN(C)C2)=O)CC2(CC2)CC1CNC(=O)CC1CC1 N1(C(C(CC)(F)F)=O)C(CC(=O)NCCS(C)(=O)=O)C2CCCC12 C1(O)(C(=O)NC(C2CN(C(C3CCc4nc[nH]c4C3)=O)C2)C)CCCC(C)(C)C1 O=S(=O)(c1cncc(Br)c1)NCC1C=CC(NC23CC4CC(CC(C4)C2)C3)C1 c1(C(=O)NCC2(C)OCCN(C(C(C(CC)C)C)=O)C2)cccc2sccc12 C1(NC(CSCC(=O)OC)=O)CCC(NC(=O)CC2CCC(C)CC2)CC1 c1(COC)cccnc1C(=O)NCC1(CNC(=O)Cc2scnc2C)CC1(F)F C1(C(=O)NC(CNC(CCOCC#C)=O)COC)CCC2(CC2)C1 N#Cc1cc(C(N2CC(NC(=O)COCC(F)(F)F)C(F)C2)=O)ccc1O N1(C(C(CC#C)C)=O)CCC2(CCCN2C(=O)CC2(COC)CC2)C1 C1(NC(c2ccc(NS(C)(=O)=O)cc2)=O)CCN(C(C2(CO)COC2)=O)CC1O N1(C(c2ccc(C=C)cc2)=O)CCC2(CC(NC(C3CS(=O)(=O)C3)=O)CO2)C1 c1(CN(CC(C)NC(C2(CCOC)CCC2)=O)C)ccc(C(=O)OC)cn1 CC1CCCC(CC(N2CCC(CC(=O)NOCCF)C2)=O)O1 CC(C)CC(C(=O)NCc1cn(C)nn1)NC(c1nnc(O)nc1O)=O C(=O)(C(C)(C)C(C)(F)F)NC1CC(NC(c2nc(C(C)C)sc2)=O)C12CCC2 C1(COC)(NC(=O)CCC2(C)CC2)CCN(C(=O)C#CC2(C)CC2)CC1 N1(S(CC)(=O)=O)CCC(Oc2ccc(NC3CCCC3C3CC3)cc2)CC1 c1(CC(=O)NC(C)CCCNC(c2ccc(F)cc2)=O)ccc(OCF)c(F)c1 N#Cc1ccc(C(=O)NCCC2CCCN(C(=O)Cn3ccc(C4CC4)n3)C2)o1 C(=O)(CCCCCC(C)O)NCC(CN(C(C=CC(CC)C)=O)CC)(C)C C1(NC(C(CC)CC)=O)CC(CNC(=O)CC=CCc2ccccc2)C12CCC2 CC1CC(C(=O)N(CCCn2cc(COCC(N)=O)nn2)C)CO1 c1(C(=O)NCC2(CCNC(C(CSC)C)=O)CC2)ccc2n[nH]cc2n1 c1(C(=O)NC(C)(C)CCNC(C2CCCS2)=O)ccnc(-c2nccs2)n1 C(CC(=O)N1CC2CC1CN2c1nc(C2CC2)nc(=N)[nH]1)(C(F)(F)F)OC N1(C(C2C(C#C)C2)=O)CC(NC(C2(n3cncn3)CC2)=O)CC(F)C1 C1(C(=O)NCC2CC(NC(CCCC#C)=O)C2(C)C)SC2C=CC1CC2 C(CC(C(C)(C)C)NC(=O)CP(C)(C)=O)N(C(=O)CN1CCCCC1)C c1(OC)cc(CCC(N2CCC(C)CC2CNC(=O)C=CS(C)=O)=O)ccc1F c1(CC)c(C(=O)NC2CCOCC2NC(c2[nH]cnc2C)=O)sc2ccccc12 C1(C(N2CC(N(C(CN(C3CC3)CC)=O)C)C2)=O)CCOC1(C)C c1(C(=O)NC(CCCCNC(C(CC)(C)OC)=O)C)ccc(C)c(OC)c1 C1(C(=O)NCC)CCN(c2cc(NCC(F)C3CCC3)ncn2)CC1 n1(CC)ccnc1C(=O)NC12CC(C(=O)Nc3cnsc3)(C1)C2 C1(C(=O)NCC(C)(C)NC(C(CC)=CC)=O)CCC2(CC2)N1C(=O)OC(C)(C)C N(C(=NCc1ccccc1C)N1CCC(F)(C(=O)OC)C1)CC(C)(C)OCC NS(=O)(=O)CCC(=O)N1CCCC1CNC(=O)CC1CC(O)C12CCC2 CCC(C)CC(C(=O)NCCc1ccns1)NC(=O)C(C#N)C(C)C C1(C2(O)CCCOC2)(C(N2C(C)CN(C(c3ccco3)=O)CC2)=O)CC1 c1(CC)cnccc1C(=O)NC(CCF)C(=O)NC1(COC)CC(O)C1 C(=O)(C#CC(C)(C)CNC(c1cccn1C)=O)NCc1cc(OC)nn1C C1(C(C)C)CCC(C)CC1C(=O)NC1CC12CC(NC(C1(F)CCCOC1)=O)C2 c1(C(c2nnnn2C(C)(C)CC)NC(CC)(C)C)nc2ccc(Br)cc2o1 N1(C(c2c(CC)n[nH]c2)=O)CCCC(C(=O)NC2CC(CCC(=O)O)C2)C1 n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N2CCC(SC)C2)c(C)n1 C1(NC(C(CNC(C2(C)CC=CC2)=O)OC)=O)CN(C)C(=O)C12CC2 CCCC#CC(C)(C)NC(C1CCOCC1NC(=O)CC1CC=CC1)=O C1(N(C)C)CCCCC1(c1nnnn1C1CC1)Nc1cncs1 C(=O)(C1=NOCC1)N1CCC(NC(=O)COCCF)C1 C1(C)(CNC(CC2(C=C)CC2)=O)COCCN(C(c2cnc(Cl)n2C)=O)C1 n1(CC)ncc(C(=O)NC2CCCC2NC(c2csc(C(=O)OC)c2)=O)n1 C(=O)(C1Cc2ccccc21)N1C(C)CC(C(N2CC(Cc3ccco3)C2)=O)CC1 CCCC(C(N)=O)NC(=O)CC(CNC(=O)C=CC(C)(C)C)OC Cc1cc(C(=O)NC(CNC(C2CC2(C)C(F)F)=O)C(C)C)cc(C)c1F O=C(C#CC1CCOCC1)N1CCN(C(C2CCCC3(CC3)C2)=O)C(CCO)C1 CC(C)CS(=O)(=O)CC(=O)NC12CCOCC1CN(C(=O)C#CC(C)(C)C)C2 C(=O)(CCCCN(C)C)NCCCOCCN(C(CC(C)C)=O)C C1(NC(c2c(Cl)cnc(C)n2)=O)CN(C(C2CC2CC(C)(C)C)=O)C2(CCOC2)C1 C1(NC(C2CCCC(=O)N2)=O)CCN(C(C23CCC(CC2)CC3)=O)CC1F c1(C(=O)NCC2(F)CCC(NC(C(CCC)(C)C)=O)C2)cnn2ccnc(N)c12 c1(C(N2CC(NC(C(CCC)NC(N)=O)=O)C3(C2)CC3)=O)ccnc2cc[nH]c12 C1(C(=O)NCC(CN(C(C2CCCN2N=O)=O)CC)(C)C)(N(C)C)CCCSC1 C1(C(N(C(CC(C)C)C)C)=O)CCN(C(c2ocnc2C2CC2)=O)C12CCC2 c1(OCC(=O)N(CC=CC#C)CC2CC2)ccc(CO)cc1.C1(C)CC1 C(=O)(NN1CCCOC1=O)NC(=O)COCCc1cn(-c2cccc(F)c2)nn1 C1(CC(=O)NC2CC2)CCC2(CC1)CCN(C(=O)C(F)(F)c1ccncc1)CC2 C(CCCCC(=O)N1CC(NC(=O)CP(C)(C)=O)C1)=CCCC C1(C(=O)NC23CC(C)(C2)C3)CCN(C(=O)CC2OCCC2(C)C)C1(C)C C(=O)(CCS(=O)(=O)N(C)C)N(C)CC1C2CN(C(C(CC#C)C)=O)CC21 c1(NC(N2CC(C(=O)Nc3ccc(N(C)C)cc3)C(O)C2)=O)cc(Cl)ccc1Cl N1(C(c2c(CC)nco2)=O)CCCC(NC(C2CN(C(=O)N(C)C)C2)=O)C1CC N1(C(CCN(C2CCC2)CC#C)=O)CCOC(C(=O)N(CC(=O)NC(C)C)C)C1 CCCC(C)(O)CC(=O)N1CCCC(C)(CNC(C2CN(C)CC(C)O2)=O)C1 C(C(=O)NCC(C)NC(=O)CCc1cn[nH]c1)(C(C)C)NC(C)=O c1(CNC(c2ccccc2)CCc2cn(C)nn2)nc2cnccc2s1 c1(N2CCCC(F)(CO)C2)nc(N2CCC(C)(CO)CC2)c2c(F)cccc2n1 CC(C)C(CO)CCNC(=O)C=CCC1(NC(=O)CCc2nncs2)CCC1 C1(NC(CCc2c(C)cccc2)=O)CCN(C(=O)C(C)(C)n2cccn2)CC1O c1(C(N(C(c2ccccc2)CNC(C(CO)OC)=O)C)=O)cccn2ccnc12 N1(C(C2(C)CC2)=O)CCC2CCN(C(=O)CCC(=O)NC3CC3)CC2C1 C(CC(C)(C)C)(c1ccccc1)NC(c1n(C(C)(C)C)nnn1)c1ccno1 c1(OC)ncc(F)c(=NCc2ccc(C(N3CC4CC4C3)=O)[nH]2)[nH]1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NC1CC1CNC(=O)CC1CCCO1 Cc1ccnc2sc(C(=O)N(C)CC3(CNC(=O)C4=COCC4)CC3)c(C)c12 N1(C(c2c(C)[nH]nc2C(C)C)=O)C2CCCC1CC(NC(c1ccoc1)=O)C2 CCC(C)C(C(=O)NCC1CC(C)(C)CO1)N(C)C(c1n[nH]c2c1COC2)=O c1(SC)c(C(=O)NC2CCOC(c3cccs3)C2)cccc1Cl c1(C(N2CC(O)(CNC(C(CCOC)C)=O)C2)=O)cc(OC)cc(C(F)F)c1 Cc1ccncc1C=CC(N1CCC(F)(CNC(=O)CC2NC(=O)NC2=O)C1)=O C1(CC)(CC)CC(C(N2CCCC2C(C)NC(c2ccn(CC(F)F)n2)=O)=O)C1 C(=O)(C(CN(C)C)C(C)C)N1C(C(=O)NCc2cc(C)sc2C)(CC)CCC1 C(C(C)(O)C(=O)NCCCOCCC(=O)NCCc1ncnn1C)OC N1(C(C(C)C)=O)CC2CC1CC2CNC(C1CC(C(C)C)C1)=O c1(C(N2C(C)C(NC(C3CN(C4CCOC4)C3)=O)CC2)=O)ccc(F)cc1O CC(CC(=O)NC(C1CCCCCC1)CNC(c1nocc1C1CC1)=O)C(F)F C1(CNC(C2(CC#C)CC2)=O)C(C)CCCN1C(c1cc(C)sn1)=O N#Cc1cc(F)c(F)cc1NC(C1CC(F)CN1Cc1sccc1Br)=O CC(C)CC(CNC(C1CC1C)=O)NC(=O)CN1CCS(=O)CC1 Cc1cc(C(=O)NCC(O)CNC(C2CN(C)C(=O)N2)=O)cc2ccoc12 N1(C(C)=O)CC(C)CCC1Nc1cc(OC(F)(F)F)cc(Br)c1 c1(OCC(=O)NCC(CNC(C2(COCC)CC2)=O)F)ccc(OCCF)cc1 C1(C2CC2)(NC(c2csc(C)c2C)=O)CCN(C(=O)C(c2cccc(F)c2)C)C1 C1(COC)(CNC(=O)CCCC2CCC2)CCCN1C(c1ocnc1C1CC1)=O n1(CC(=O)OC)nc(C)c(S(=O)(=O)Nc2csc(Br)c2)c1C c1(OC)cc2ccccc2cc1CN1CCC(O)C(C(N2CCOCC2)=O)C1 c1(Cn2cc(CC(CC)C(=O)O)nn2)ccc2c(c1)CCCS2 c1(CNCC2N(C(CCc3c(C)ncs3)=O)CCOC2)cc2ccccc2[nH]1 c1(NC(Cc2cnn(C)c2Cl)=O)cccc2c1CCCN2C(=O)CSC1CC1 n12nc(cc1C)NC(=O)C2.c1(N2CCC(CC)C2)c(OC)nsc1OC c1(C(N(C2CCC(C(N3CCCC(F)C3)=O)CC2)C)=O)ccc([Si](C)(C)C)cc1 C1(C(N(CC(=O)NCCC2CCC(C)O2)CC)=O)CC2(CSC2)C1 Cn1c(C(N2CCC(C(F)F)(CNC(C3CC(F)C(=O)N3)=O)C2)=O)nnc1S C12(C(N3C(CNC(C4C=CC=CC=C4)=O)COCC3)=O)CC1CCC2(F)F c1(C(N2CC(NC(CC=C)=O)C(O)C2)=O)cc2cn[nH]c2cn1 c1(C(N2CCC(F)(C(=O)Nc3nccc(I)n3)C2)=O)cc(Cl)c2cn[nH]c2c1 c1(C(=O)NC(c2cccnc2O)C)cnc(CNC(=O)C#CC2CC2)nc1 CCCN=C(NCC(C1CCN(C)CC1)(C)C)N1CCN2C(=O)CCC2C1 C1(CNC(CCC=C(C)C)=O)CCN(C(=O)CCc2cn[nH]c2)C1(C)C C1(COC)CC2(CCN2C(=O)C(CN(C)C)NC(c2occ3c2CCC3)=O)C1 c1(NC2C(C)CN(C(c3ccc(Cl)cc3)=O)C2)ncnc2c([N+](=O)[O-])cccc12 n1(CCC(=O)Nc2cc(C(F)F)nc3ncnn23)c(=O)oc2ccccc12 C1(C(N(CCN(C(CSCC(=O)OC)=O)C)C(C)C)=O)CC2C=CC1C2 N1(C(CCCOC(CC)=O)=O)CCN(C(c2cc(OCC)n(C)n2)=O)CC2(CC2)C1 C1(C(N(CC(=O)OCC)C)=O)CN(C(=O)C(O)CCSC)CC(C)(C)C1 c1(OC)cc(CC(=O)NCC2CCCN2C(c2n[nH]c(C)n2)=O)ccc1C Cc1nn(C)c2c(NCc3csc(Br)c3)nc(N3CCc4[nH]c(=N)sc4C3)nc12 N1(C(c2ccc(Cl)o2)=O)CC(CO)C2(C1)CN(C(=O)C1=CC3(CCOC3)C1)C2 c1(C(C)=O)ccc(NNC(=O)NC2CCS(=O)CC2)cc1 C12(C(N(CC(C)C(=O)N3CC(C4CCCOC4)C3)C)=O)CCC(C1)OC2C c1(C(=O)NC2CN(C(C3CCCC3)=O)CC23COC3)cc2ncccc2[nH]1 S(=O)(=O)(c1cc(C)cnc1NC(CO)C1CC1)N(C)Cc1ccc(OC)cc1 N1(C(CC(C)CN(C)C)=O)CCCCC12CN(C(C1CC1C1CCC1)=O)C2 C1(C(C(=O)N(CC(C)CNC(C2(CO)CCC2)=O)C)F)CCCCC1 O=C1Cc2cc(CN3CC(=O)N(Cc4nccn5nccc45)C3=O)ccc2CN1 CC(CC(=O)N1CCC(C)(NC(=O)C(O)C(F)(F)F)CC1)P(C)(C)=O C(c1ccc(Cl)cc1Cl)=CC(=O)NC(C1CN(c2nnnn2C2CC2)C1)C C=C1CC(C(F)(F)F)(C(=O)NCC2CCN2C(=O)CSc2cnn(C)c2)C1 CC1=C(C(=O)NC2(CN(C)C(c3nc(C)nn3C)=O)CC2)CCC(C)(C)C1 C1(CCNC(C(C)NC(CC)=O)=O)CCCCN1C(=O)CCc1ccc(C)s1 Cc1nc2ncc(C(=O)NC3CC3CNC(=O)Cc3nn(C)cc3Cl)c(=O)n2[nH]1 CC(C)(C#N)CCC(=O)NCC1CN(C(C2Cc3cccnc3C2)=O)C1 C1(CC=C)(C(=O)N(CCCOC)C)CN(C(=O)C(CC)=CCCC)C1 CCC(C)(C)CC(=O)N1CCCC1C(=O)NCc1oc(CSC)nc1C N1(C(CCC#C)=O)CCN(C(C2C=CC2C(=O)OC)=O)CC1CC(F)F c1(C(N2C(CCNC(Cc3c(C)nccc3)=O)COCC2)=O)ccc(=O)n(C)n1 C1(CC(=O)NC2CC(C(C)NC(c3cnsn3)=O)C2)CCC2(CC1)CCC2O N1(C(=O)Cc2csc3ccccc23)CCN(C(C2CC=CCC2)=O)C2CCCC12 C1(C(=O)NCCC(CC)CO)C2CCCC2CN1C(=O)C(C(=O)OC)OC Cc1cnc(F)cc1C(=O)NCC1CCCC1NC(c1cn(C)nn1)=O N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CN(C(=O)C(N3CCOCC3)C)CC2C1 C1(CC(=O)NC2(CNC(C3(F)CCC3)=O)CCCC2)CCc2ncc(Br)n2C1 c1(COC)ccnc(C(=O)NCC23CC2CN(C(=O)C=CC2CCC2)C3)c1 C1(OC)CCCC(CC(=O)NC2CCCC2NC(=O)CCCCn2ccnn2)C1 c1(C(=O)NC2CC(CNC(C3CC3CF)=O)C2)nccn2nccc12 c1(C(N2C(CNC(CC(COC)C)=O)CC(C(F)(F)F)C2)=O)ccc(S(N)(=O)=O)s1 c12cc(sc1C)NC2.c1(C(c2nnnn2C)OCC)cn(C)nn1 CCCCS(=O)(=O)CC(=O)NCC1CCN1C(=O)CCCCC#N c1(NCC2CC(NC(c3cc(C)sc3C)=O)C2)ccc(C#N)cc1[N+](=O)[O-] N1(C(C(C2CCCC2)OCC)=O)CCC(NC(c2nc(C)n(C)n2)=O)C1C c1(C(N2CCC(C)(CNC(CC(CC)C3CCC3)=O)C2)=O)cnc(OC)c(C)n1 N1(C(CSC)=O)CCCCC(CNC(c2ccncc2Oc2ccccc2)=O)C1 N1(C(CC2(C)OCCO2)=O)CCCC(C)(NC(=O)C(F)CC2CCOC2)C1 c1(C(N2OCC(n3cc(C(C=C)(C)O)nn3)C2)=O)cc(S(N)(=O)=O)ccc1Br N1(C(c2ccc(CC)cn2)=O)C2CCC1C(NC(=O)Cn1cc(C)cn1)C2 c1(OC)cccc(Br)c1NC(=O)CC1CCN(Cc2cccc(C3CC3)c2)CC1 c1(C(=O)NCCCN(C(=O)C(c2cccnc2)O)C)cc(=O)c(Br)c[nH]1 C(C)(CCC(=O)N(CCCCCNC(c1ccnc(S)c1)=O)C)OC C12(NC(CC3CCCC(OC)C3)=O)CCCC1N(C(C1(C)CC=CCC1)=O)CC2 C1(CC(=O)NCCNS(CC)(=O)=O)CCN(C(C2CN(C(C)C)C2)=O)C1(C)C CC1(CNC(=O)C(C#N)CC2CC2)OCCc2ccccc21 N1(C(CC=C)=O)CC2CCC1CN2Cc1ccc(Br)c(C)n1 C(CC1CCCCC1)(C(=O)NC(C)CCCNC(C1(C)CC=CC1)=O)OC N1(C(CC2(C=C)CC2)=O)CCC(C2CCN(C(=O)C(C)OC)CC2)C1 c1(C(=O)NCCC2CN(C(C(C)NC(C)=O)=O)C2)cccc2cccc(Cl)c12 C1(CC=C)(NC(C2CC(=O)N(C3CC3)C2)=O)CCN(C(c2ccn(C)n2)=O)C1 CC1CCC(NC(c2sc(Cl)cc2Cl)=O)CN1C(c1ccc(F)cn1)=O N1(C(c2nn(CC)c(O)c2)=O)CC2CC(NC(c3cc(C(F)F)on3)=O)C2C1 c1(C2(NC(=O)NCC(C)N(CC)CC)CCC2)cccc(C#N)c1 c1(CNC(=O)CC2OCCCO2)cccc(NC(c2ccc(F)o2)=O)c1 C1(C(=O)NCC2(OC)CC(C)C2)CC12CCN(C(=O)CC1CCSC1)CC2 CC1(C)COCCC1CNC(=O)CC(C(F)F)NC(=O)CC1CCCCCC1 c1(C(N(CCC(C)NC(COC(C)C)=O)C)=O)cnc2c(c1)c(O)nc(=O)n2C Cc1ccc(C(=O)NC2CC(C(=O)Nc3ccc(Cl)c(Cl)c3Cl)C2)c(I)c1C C1(NC(c2cccn2C2CC2)=O)CCCCC1C(=O)NCc1cccnc1O Cc1cc(F)cnc1C(=O)NC1(CCCC(=O)N2CC(CC(N)=O)C2)CCC1 C(=O)(C1CCc2cc(F)ccc21)NCCCN(C(COCCC=C)=O)C1CC1 c1(C(=O)NC2CCCN(C(c3nnc(CC)s3)=O)CC2)c(O)nnc(C)c1C C1(NC(c2cccnn2)=O)CCN(C(C2(CC3CC3)CCCO2)=O)CC1O S(=O)(=O)(c1ccc(Cl)cn1)N1C(CC(=O)NCc2cn(C)nc2)CCC1 Cc1cc2c(C(=O)NCCC3CN(C(=O)CCc4cnn(C)c4)C3)nccn2n1 CCC(CC(=O)NCC1(O)CCN(C(c2cc(N)ccn2)=O)CC1)C(C)(C)C C#Cc1ccc(C(N2CCCC2CN(C(=O)C(O)C=C)C)=O)cc1Cl N1(C(C)C(=O)NC(N)=O)CC2CC1CN2C(C1CC12CCCC2)=O C(=O)(C(CO)NC(=O)C1CC1)N(CC(CC)NC(=O)C(CC)C1CCOCC1)C N(C1c2ccc(OC)cc2CC1(C)C)C(=O)NCCc1ccc(C(=O)OC)s1 c1(C(N2C(C(N3CCC(c4ccccc4)C3)=O)CCC2)=O)ccc(F)cn1 C1(C(N2C(C)(C(=O)NCc3cc(Br)ccn3)CC2)=O)C=CC(=O)N=N1 C1(NC(CSCCC)=O)COC2C(NC(=O)CCc3nc(C)cs3)COC12 N1(C(c2c(C(=O)OC)scc2)=O)CCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C(F)C1 N1(C(c2cnn(C3CC3)c2)=O)CC2(C1)CN(C(C1(CC(F)(F)F)CC1)=O)CC2CO Cc1c(C(=O)NCC(O)CN(C(=O)Cc2cccc(C(N)=O)c2)C)cccc1F c1(C(N(C(C)CCNC(C2(C)CCCOC2)=O)C)=O)c(O)cccc1Cl N1(C(C(C)CN(C(=O)C=CCO)C)=O)CC2C3CCC(C3)C2C1 n1(CC(=O)NC2C(C)N(C(C34COCC3C4(F)F)=O)CC2)ncc(C#N)c1N N1(C(CC=C)=O)CC2(CCC(C(N3CCCCC3CCO)=O)O2)C1 c1(OC)cccc(C(C)=CC(=O)N(CCC(C)NC(=O)CC23CCCC2C3)C)c1 C(=O)(CCCCCC#N)N(CCNC(C1(OC)CC(C)CC(C)C1)=O)C1CC1 CC1CN(C(C2COCCOC2)=O)CC1(C)CNC(=O)CN(C)S(N)(=O)=O c1(CNC(C2CCc3n[nH]cc3C2)=O)cnn2cc(Br)ccc12 c1(OC)ccc(-n2nc(C3CC3)nc2-c2cc(C3CCOCC3)on2)cn1 C=CC1(CC(=O)NC(C)CC(C)(C)O)CN(C(=O)C2CC2)C1 CN1CCC(CCC(=O)NCC(C)(CO)NC(c2ccc(F)s2)=O)C1 c1(CC)cc(CC)[nH]c(=NCCC(C)NC(=O)C(N2CCCCCC2)C)n1 C1(C(=O)NC(C(=O)NC(C)Cn2cccn2)c2cccs2)CCCC1C1CC1 C(=O)(CCCC(F)(F)F)NC1(CF)CCN(C(C(=Cc2ccccc2)OC)=O)C1 CCCCC(CC)CC(=O)NC1CCC1CNC(c1ccc(Cl)c(N)c1Cl)=O C(CC(C(=O)Nc1nccs1)N1CCC(CO)CC1)C1CC(=O)NC1 c1(C(=O)OC)ccc(C=CC(=O)NC(CNC(C23CCCC2C3)=O)C2CC2)cc1 C1(COC)CN(C(C2CC=CC(n3cc(-c4cncnc4O)nn3)C2)=O)CCO1 c1(C(C)NCC(=O)NCC2CCOCC2)n[nH]c(C(C)(C)C)n1 c1(C(=O)Nc2cnc(F)cc2CNCC(O)C(F)(F)F)ccc(O)c([N+](=O)[O-])c1 Cc1coc(C)c1C=CC(=O)NCCC1(C)CCN(C(=O)C(C)C2CC2)C1 c1(C(=O)NCC2N(C(C#CC(C)C)=O)CC(C)CC2)ccc2cnoc2c1 Cc1cc(CC(=O)NCCN(C(C2CCC(C(N)=O)C2)=O)C(C)C)sn1 c1(COC(C2(n3ncc(C)c3)CCCC2)=O)ccc(C(C)C)nc1O O=S(=O)(c1ccnc(C(F)(F)F)c1)NCCOc1ncccc1Br C#CC1(CNC(C2CC2CCNC(C2(CC3CC3)CC2)=O)=O)CC2CCCC12 C#CCC(CC(F)F)C(=O)NCCC(C)(C)NC(=O)CC1CCCCC1 C12(C(N3CCN(C(CCC)=O)CC3CF)=O)CCCCCC1OCC2 c1(C(=O)Nc2scc(-c3c(C)noc3C)n2)cc(F)ccc1O N1(C(c2c(CC)ncs2)=O)CCC2(CCN(C(c3cc(C)c(F)cc3O)=O)C2)C1 c1(C(=O)NCC(C2CCOC2)NC(c2c(C#N)ccs2)=O)ncnc2sccc12 C1(C(=O)NCCCCC(C)NC(=O)C(C)Cc2cnco2)CCc2c[nH]nc2C1 C1(C(N(C)CC2CCN(C(c3c(OC)csc3)=O)C2)=O)Cc2c(C)cccc2O1 C(C(C)(C(=O)NC(c1nc(C)no1)C)NC(=O)CCCc1ccco1)SC Cc1cc(F)ncc1NC(C1(CNC(=O)C(O)Cn2cncn2)CC12CCC2)=O N1(C(CCOCC#C)=O)CCC2CCN(C(c3cnc(OC)c(C)c3)=O)CC12 N1(C(C(N2CCSCC2)C)=O)CCN(C(=O)CCCc2cncs2)C(C2CC2)C1 S(=O)(=O)(c1ccc(I)cc1)NCC1(C(=O)NC2(C#N)CCC2)CC1 c1(C(N2CC3C(NC(C(C)OCC=C)=O)(C3)C2)=O)cnn2c1CC(F)(F)C2 c1(C(=O)NC2C3(NC(C(C)OC)=O)CCC(C2)C3)nc2ccccc2cc1Cl N1(C(C(CC)C)=O)CCC2(CC1)CC2C(=O)Nc1ccnc(C(=O)OC)c1 N1(C(c2cccc(CC)n2)=O)CC=C(CNC(C2CCC=CCCC2)=O)CC1 CCCC(C#N)C(=O)NCC(CC(=O)NC1C2CCC(F)(F)C12)C1CCC1 C1(C(=O)OC(C)(C)C)CCCC(NC=O)C1.C12(C(=O)NC(C(C)O)=O)CC(C1)C2 c1(C(=O)NC(C2(O)CCN(C(=O)C(O)CC3CC3)C2)C)cn(C)c2ncccc12 CC1CCc2nc(S(=O)CCNS(=O)(=O)c3cc(Cl)c(F)cc3F)sc2C1 c1(CNC(c2cc3c[nH]cnc-3n2)=O)cccc2c1CCN(c1ncns1)C2 C(C(C)CC(=O)N=c1cc(C2CC2)n(C)[nH]1)NC(C(CCC(C)C)O)=O C1(CNC(CCCC(=C)C)=O)CN(C(c2cccn2C(C)C)=O)CCC12CCC2 N1(C(CCCN(C(=O)CC2CCCC(=O)C2)C)=O)CCC2(CC1)N=N2 c1(C(N(CCCN(C(C(C)OCCC#C)=O)C)C)=O)cc(C(C)(F)F)ccn1 CC(CC(=O)NCC(C)CNC(C1(C)CC1(C)C)=O)N1CCCC1=O C1(NC(CC(C)NC(N)=O)=O)CC(CNC(c2cncnc2)=O)C(O)C1 C1(C(N2CCC(NC(C(C)(C)OC(C)C)=O)C(O)C2)=O)CCC2(CCC2)CC1 C1(CC)(NC(=O)CC2(N(C(=O)CCc3cccnc3)C)CC2)CCNC1=O CC1(C)CCCCC1CC(=O)NCC(C)(C)NC(=O)CC1CCCNC(=O)C1 CC(C(=O)NCC1CCC(NC(C2COC(=O)N2)=O)CC1)C1=CCCC1 C12(C(=O)NCCOCCCNC(c3n[nH]c4c3CCC4)=O)OCCCC1C2(F)F C1(C)(C(=O)NCCCn2c(C)nnc2)C=CCN1C(=O)CCC1CCCO1 c1(C(=O)NCCCC2(NC(C3C(C=C)C3)=O)CC2)cc(O)nc(C2CC2)n1 C1(C(N2CCC(N(C)CC)C2)=O)CCC2CCC1N2C(=O)CCN1CCCCC1 c1(C(C(N)=O)NC(N(C)CC2CC2c2cn[nH]c2)=O)ccc(Br)cc1 c1(C(C)C)nnc(N2CC(C(C)CN(C)C(=O)OC(C)(C)C)C2)o1 CC1(C)CCCC(C(=O)NCC2CCN2C(=O)CCC2CCOC2)CC1 c1(OC(C(=O)NCC2C3CN(C(=O)CC4CCC4)CC32)F)ccc(Cl)c(F)c1 c1(C(=O)NC(C(C)C)CNC(=O)Cc2cnccn2)ccc(N)c2ccncc12 N1(C(C(C)(C)OC(C)C)=O)CCCC2(C1)CN(C(=O)CCn1ccnc1)CCO2 c1(C(=O)NCCN(C(=O)C(C)NC(c2ccco2)=O)CC)cncnc1.C1CC1 CCC(CC)(CC)C(=O)N1CC2CC1C2NC(C1OCCC1C)=O CCC(CC(=O)C1C(C(=O)NCCC2(CO)CCCCC2)CC1(C)C(C)(C)C)SC.OCC N1(C(CCc2n(C)c(S)nn2)=O)CCC2(NC(c3cscc3Cl)=O)CC2C1 N1(C(C2(CC)CCCO2)=O)CC(CCNC(c2cnc(O)n2C)=O)C(C)C1 c1(C(N2CC(CNC(C(C)(Cl)Cl)=O)OCC2)=O)cc(S(=O)(=O)NC2CC2)c[nH]1 C(CF)(C(=O)NC1CC(CNC2CN(C(C3(Cc4ccncn4)CC3)=O)C2)C1)OC c1(CC(N2C(CNC(CCCSC)=O)C(C)CCC2)=O)c[nH]c2cc(Cl)ccc12 C1(N(c2n(C(C)C3CC3)ncc2)C(=O)C2CC2)CCC2CCC12 N1(C(C2(C#C)CCCC2)=O)CC(C)OC2(CCN(C(=O)COC(F)(F)F)C2)C1 C1(NC(C(=C)Cc2ccccc2)=O)COCCN(C(=O)CSC)C1 C1(C(C)NC(c2cscc2C(F)F)=O)CN(C(=O)CC2(N3CCCC3)CC2)CCO1 c1(C(N2CCC(C(C)NC(Cc3ccc(SC)cc3)=O)C2)=O)cn2ccnc2s1 c1(C(=O)Nc2nc(Br)cs2)cccc2c1CN(Cc1ccn3ccnc3c1)CC2 c1(C(N(CC(C)N(C(C(CCC)C)=O)C)C)=O)ccc2cc(C)ccc2n1 NC1CCOCC1C(=O)NCC(F)(F)CN1CCCC1 c1(CNC(c2cc(C)on2)=O)csc([N+](=O)[O-])c1.C12(CCOCC1)C(=O)N2 C(=O)(C(C)CC(F)F)N1CC(CC(C)NC(C2CCC(CCCCC)CC2)=O)C1 C1(NC(C(N(C)C)C2CC2)=O)CN(C(c2cc(F)c(F)c(F)c2)=O)CC2(CC2)C1 C1(C(=O)NC2(CNC(c3nc(C4CC4)cs3)=O)CC2)CC2C=CC1C2 N1(C(c2nc(NC(C)=O)sc2)=O)CCN(C(=O)C2=CCCS2)CC1C c1(OC)cccc(C2=NOC(C(=O)OCc3cnsc3)C2)c1 O=CN1CCCC1C(=O)NCC12CC(CNC(=O)Cc3ccnnc3O)(CO1)C2 N1(C(C2CCN(C)C2)=O)CC2(CNC(c3cccc4nncn34)=O)CCC1CC2 N1(C(=O)CC2CCCCO2)CCC2CCN(C(c3nccc4occc34)=O)C2C1 N1(C(Cc2n[nH]c(=N)s2)=O)CCOC2(CCN(C(C3CCCC(F)C3)=O)C2)C1 N1(C(CCCCC=C)=O)CC(C(N2CCOC(C(C)(C)C)C2)=O)C2(CCC2)C1 C12(C(N3CCC(NC(C(C)(C)C)=O)C(CO)C3)=O)CC(C)(C1)OC2(C)C C1(C)(CC)CC(NC(c2c(F)cccc2F)=O)CN1C(c1cncnc1C)=O C(=O)(C(O)C(F)(F)F)N1CC(CC)C1.c12n[nH]cc1C(CN(C)CC1CC1)NC2=O c1(CC(=O)NC(c2cnn(C)c2)C(=O)N(C(C=C)C2CC2)C)csnc1C C[Si](C)(C)C1(C(N2CCCC2C2CCCCC2O)=O)COC1 c1(C2(NC(C(c3ccccn3)OCC)C)CC2)ccccc1F c1(C(N2CC3N(C(COCCC)=O)C(CC3)C2)=O)cc(C)nc(O)c1[N+](=O)[O-] N1(C(COCCC#C)=O)CC2CC(C1)N(C(c1sc(C(C)(C)C)nc1C)=O)C2 c1(NC)cnc(F)cc1C(N1CCOC(CNC(c2csc(C3CC3)n2)=O)C1)=O N1(C(c2cccc(COC)n2)=O)CCC(NC(C2CC(OC)C2)=O)C12CCC2 NC1C=CC(NCC2CCCC2OCc2ccccc2)C1 c1(-c2onc(CC(N3CCN(C(CC)(C)C)CC3)=O)n2)coc2cc(O)ccc12 C1(C(=O)NCCC(=C)CO)CC(C)(C)CN1C(=O)CC(C)(C)O CON(CCC(=O)NOCc1nc[nH]n1)C(=O)C(C)CC(F)(F)F c1(CC(=O)NC23C(n4cc(C(C)(C)C)nn4)CC(CC2)C3)ccc(C#N)c(Cl)c1 N1(C(CC2(OC)CCC2)=O)CCC=C(C(=O)NOCC(C)(C)C)C1 N1(C(=O)NCCCCN(CCCCC)C)CCCC1C(=O)NCC.C(C)(C)(C)O N1(C(CC2(C)CCCC2)=O)CCC(O)(CNC(c2coc(C3CCC3)n2)=O)C1 N(C1CC(C)(C)Oc2ccc(F)cc21)C(c1c(OC)cns1)=O CC(O)CCCCCC(=O)NC1CC12CC(NC(=O)CCC=CBr)C2 N1(C(C(c2n(C)ccc2)=O)=O)CC=C(C(=O)NC2CCC(C)(C)C2)CC1 C1(CC(=O)NC2C(C)=C2)CCCC(NC(=O)CCCOC(C)(C)C)C1 N1(C(C2CC(C)(C)C2C(F)(F)F)=O)CCC(CO)(NC(c2ccnnc2)=O)CC1 C(C)(CO)(C(=O)NCC(C(=O)NCC(=O)NOC)N(C)C)OC C(C(CC1CC1)C(=O)Nc1cnccc1CO)NC(C(C)OCOC)=O C(N=c1[nH]c(N(CC(C)(C)CO)C)nc2c1CCC2)C1C(CCC)CCC1 N1(C(c2cc(OC)c(Cl)cc2)=O)CCC(C)C(NC(c2cccnc2)=O)C1C c1(N2CCC(CNC(C)=O)C2)cc(N2CCC(C(F)F)CC2)ncn1 c1(C(N2C(C(=O)NC(CC=C)CO)CC3CC32)=O)c[nH]c2nccc-2c1 N1(C(C(C)=CCC)=O)CCC2(CC1)CC2C(N1CCOCC1c1ccccc1)=O c1(CC)cnc(NC(C2CC(n3cc(CCN(C)C)nn3)C2)=O)s1 C1(NC(c2cc(C)no2)=O)CCN(C(=O)Cn2ccc(=O)n(C)c2=O)CC1(C)C c1(C(N(C(C)CCNC(C2CCC(C)O2)=O)C)=O)cccn(C2CCC2)c1=O CC1C(c2ccccc2)CCN1Cc1cn(C2(C)CCC(C)C2)nn1 N1(C(C2N(CC)CCC2)=O)CCCC(CC)C1C(=O)NCCCSC c1(-c2cn(C)c(=O)cc2)nc(C(=O)Nc2cccc(C#N)c2Cl)n2ccccc12 N1(C(C=Cc2n(C)ncc2)=O)CCN(C(=O)CCc2cncs2)C(CO)C1 N1(C(CC2C(C)=NNC2=O)=O)CC2(C(=O)NCc3cnn[nH]3)CC1CCO2 CCC(CCCO)N=c1[nH]c(=NC2CCOc3c(OC)cccc32)c2ncccc2[nH]1 C1(NC(C2(CC)CCNC2=O)=O)CC=C(C(=O)NC2(CF)CC2)C1 N1(C(c2cccc(-c3cn[nH]c3)c2)C(=O)NCC(=C)C)CCC(O)C(F)(F)CC1 C(=O)(C1=NOC(C)C1C)NC1C(SC)CN(C(C2CCCOC2)=O)C1 c1(NC(c2ccccc2F)CNC(C(C(C)C)NC(C)=O)=O)ncccc1C#N n1(CC(=O)NCC(CNC(CC2C(CC)C2)=O)OC)cc(Cl)c(C)n1 c1(Cc2cc(C(N3CCCC(C(=O)OCC)C3)=O)no2)cc(Cl)ccc1[N+](=O)[O-] c1(CC(=O)NC2CN(C(C(c3ccc(C)cc3)=O)=O)C(C)C2)cc(O)nc(O)n1 C(CC(C(=O)NCC1CCCO1)NC(=O)CCOCC(C)(C)C)=CC C(C(O)CC(=O)NCC12CCC(CC1)O2)NC(CN(CC(C)(C)C)C)=O C1(C(=O)NCC(C)CNC(=O)CCn2cncn2)CC2OC1C1CC21 C#CC1(C(=O)NCC(c2ccccc2)C)CCN(C(=O)C(O)c2ccsc2)C1 N#Cc1ccc(O)c(NC(=O)C(Cn2ccnn2)NC(c2c[nH][nH]c2=N)=O)c1 c1(OC)ccc2[nH]cc(C(=O)NC3CCOCC3NC(C3CSC3)=O)c2c1 C1(C)(CC)CCC(CNC(=O)C(C)(CO)NC(c2csnc2OC)=O)O1 c1(C(N2CCCC(C(C3CC3)NC(CN3CCC(C)C3)=O)C2)=O)ccnc2[nH]cnc12 N=c1nc(Cl)cc(C(N2CCCC(CNC(=O)CCN3CCCCC3)CC2)=O)[nH]1 Cc1nn(C)c2sc(C(=O)NC34CCCC3CN(C(=O)C=C3CCC3)C4)cc12 CCC(CC)C(C)C(=O)NCC1(F)CCCN(C(c2sc(C)cc2C)=O)C1 c1(C(C(=O)O)N(C(CC#C)C)C2CC2)cccc(N2CCCC2=O)c1 C(=O)(C1=CCCO1)N1C(CN(C(CCSCC)=O)C2CC2)CCC1 CC1CCC2(CC1)CCN2CC(=O)NCc1ccc(F)c(Cl)c1F C1(C2CCC2)(C(N(C(C)CN(C(=O)CC(C)n2cccc2)C)C)=O)CC1 N1(C(C=CC(C)(C)SC)=O)CCCCC1C1CCN(C(c2ccc(Cl)s2)=O)C1 C1(OC)CN(C(c2ncc(F)cn2)=O)CC1NC(=O)C(c1ccc(Cl)s1)=O c1(N(C2CCN(C(c3nc(O)n[nH]3)=O)C2=O)C)cccc(N)c1F N1(C(C2C(C=C)C2)=O)CC2CC2(CNC(C2(C3CCCO3)CCCC2)=O)C1 Clc1cscc1CNC(c1ccnn1CCF)c1nnnn1C1CCC1 c1(CC)ccc(O)c(CNC(C2CC2NCc2csc(Br)c2)=O)c1 Cc1cc(C(N2CC(C3(NC(=O)Cc4nccn4C)CC3)C2)=O)c(C)n1C(C)C Cc1cc(=NC(=O)CN(C(C)(C)C)C(c2cccc(F)c2C)=O)[nH]o1 c1(C(CNC(=O)NC2CCC(N(C)C)CC2)(F)F)c(F)cccc1F N1(C(COCCC(C)C)=O)CCC2(NC(=O)CCCn3c(O)nnc3O)CC2C1 C(=O)(C(C)(C)CC(F)F)NCC1C(NC(CCOCC#C)=O)CCCC1 c1(C(=O)NCC2(C)OCCN(C(C=NOC)=O)C2)cccc2c1CCS2(=O)=O C1(CCNC(=O)CCc2ccc(C)o2)(OC)CN(C(c2ccoc2)=O)C1 CCS(=O)(=O)CC(=O)N1CCC(n2cc(-c3ccccc3O)nn2)C1 C1(CC)CCCN(C(c2cc(C3CC3)n(C)n2)C(=O)NCC2CCCO2)C1 C1(NC(C(c2ccoc2)NC(C(C)CO)=O)=O)CCCC(C2CC2)C1 c1(C(N2C(CCNC(c3c(C)cnnc3)=O)COCC2)=O)ccc(Br)c(F)c1 C1(C(N(C2CCN(C)C2C)C2C(CC)C2)=O)COCCN1C(=O)Cc1cocn1 c1(NC(C2C3CN(C(C(CCC)CCC)=O)C2C3)=O)ccc2c(c1)OCCO2 c1(C(=O)OCC)c[nH]ccc1=NCCC1CCN(C(c2conc2C2CC2)=O)C1 N#Cc1cc(C(N2CCCC(CS(c3ccccc3)(=O)=O)C2)=O)sc1Br C1(C(N2C(CNC(CCNC(N)=O)=O)CC2)=O)CCNC(=O)C1 c1(C(C(C)NC(=O)NCc2c(I)ccnc2F)OC)cc(Cl)cc(Cl)c1 C1(C(=O)NC(C2CCN(C(=O)CC(C)(C)O)C2)C)COC2CCCCC12 CCC(CC)CC(F)C(=O)NC(C)CC(=O)N(C)CC1CCCN(C)C1 c1(NC(C(C=C)N(C)C)=O)ccc(C(N2CC(OCC)C2)=O)cn1 c1(C(=O)NCC2(C)CC(NC(C(CCOC)C)=O)C2)cc([N+](=O)[O-])c(C)s1 C1(CC)(NC(=O)CN2CCCOC2=O)CCCN(C(c2cc(Cl)nnc2O)=O)C1 CC(C(=O)N1CC(CN(C(=O)C(c2ccccc2)O)C)C1)C(C)(C)C C1(NC(c2ccc(Cl)s2)=O)CN(C(=O)Cc2ccc(Br)cn2)CC2CC12 c1(N(C)Cc2cc(F)cc(Cl)c2)nc2ccc(Cl)cc2c(=NCC2CC23CC3)[nH]1 C1(C(F)(F)F)(NC(C2CCN(C(COC)=O)C2)=O)CCCCC1 CC(=O)CCCC(=O)NC1CCCC(CC(=O)Nc2ccccc2F)C1 c1(C(N2CC(OC)(CNC(C3CC4CC3C3CC43)=O)C2)=O)scc2c1OCCO2 C1(NC(C(C2(O)CN(C(C3(C)CCNC3=O)=O)C2)F)=O)C2CCC3C(C2)CC13 CC1CN(C(c2cc(C3CC3)cs2)=O)CCC1N(C)C(c1cn(C)ccc1=O)=O CS(=O)(=O)c1cnn(CCNC(=O)C(=O)NC2CC2(F)F)c1 c1(C(N2CC(NC(C3CCN(C(C)=O)C3)=O)C2)=O)cc(Br)nn1C CCC(CC)CCC(=O)N1CCOCCC1C(=O)NC(C)CC(F)(F)F CC1CCCC=C1C(=O)N1CCC2CN(C(c3ncc(C#N)cc3Cl)=O)CC12 N1(C(C23C(NC(c4c(C)cccc4)=O)C4CC2C3C4)=O)CCOC2(CCC2)CC1 N1(C(C)=O)CCCCC1C(=O)N(C)CC1CN(C(C2CN(C)C2)=O)C1 C1(C(N(CCC)CCNC(=O)C=Cc2ccc(Cl)cc2)=O)Cc2ccncc2C1 C(=O)(C1=C(C#N)CCC1)NC1CCCC(CC(N2CCC(C)C2)=O)C1 CC(C)(CCNC(=O)CC1CCSC1)C(=O)NC1CCN2CCC1C2 C(=O)(CC(C)C(C)C)N1CCC(C)(C(NOCCC(=C)C)=O)C1 C1(C(N2CCCC(NC(CC(CC)CN(C)C)=O)C2=O)=O)CNC(=O)CC1(C)C C(=O)(C1CCc2cccnc21)N1C(C)(CC)CC(NC(=O)COC2CCC2)C1 Cc1nn(C)c(C(N2CC3CC3(NC(=O)CC3CCC(C)(C)C3)C2)=O)c1Br c1(C(N2C(C)(CNC(C34CCCN3CCC4)=O)CCC2)=O)ccc(Cl)c(F)c1 c1(C(=O)NC2(CN(C(CCC(CC)OC)=O)C)CC2)cc2nccnc2cc1F CC1(C)C2CCC(C2)C1C(=O)NCC1(NC(=O)CC2CCCSC2)CCC1 C1(C(N2CCCC(CC3CC3)C2)=O)CCCCN1C(c1ccc(Cl)cc1)=O C1(C(N2CCC(NC(C(N3CCCC(C)C3)=O)=O)CC2)=O)CC2C(C1)C2(F)F c1(NC(N2CC(C(CC)C)C2)=O)ccn2nccc2n1 CC(C)C(F)(F)CC(=O)N1CCC1NC(=O)CNS(=O)(=O)C1CC1 N1(C(=O)NC2CN(C(C)=O)CC23CCC3)CCCc2ccccc2C1 C(C(=O)NCC(c1ccc(F)cc1)C(=O)OC)(C(CC)CC)N(CCC)CCC c1(CNC(CC)C(=O)OC(C)=O)ncccc1C(N1CCCCC1C(N)=O)=O C(=O)(C(C)(C)C(C)(C)C)NCC(CC(F)(F)F)NC(Cc1cc(C)c(F)cc1)=O C(=O)(C1COc2ccccc21)NC1CCCC(NC(C(CSC)(C)C)=O)C1 CCC(CC)(CCC(=O)NC1COCC1NC(C12CCC(OC)C1C2)=O)[N+](=O)[O-] C(=O)(C(CNC(=O)C(C1CCC1)OCC)CC1CCCC1)N(CCCF)CC C(c1ccccc1F)=CC(N1CCC(C)(NC(=O)CCC2CC(F)(F)C2)C1)=O C1(OC(C(=O)NCCC(=C)CNC(=O)C(CO)N(C)C)C)CCCCCC1 c1(C(N2CC(CNC(CC(CC)C)=O)N(C)CC2)=O)ccc2c(C)[nH]nc2c1 C1(NC(C)=O)CCCN(C(=O)CCn2cc(-c3ccc(N(C)CCO)nc3)nn2)C1 c1(NC(C2C(O)CCN2C(c2cc(Br)ccc2F)=O)=O)ccnc(Cl)c1I N1(C(Cc2cnc(C)s2)=O)CCOCC1CC(=O)NC1CN(C2CCC2)C1 Cc1occc1C(N1CCCC1C1CCN(C(=O)CNC(=O)C(F)(F)F)C1)=O c1(C(=O)NC2(CF)CCN(C(C(C)OCC=C)=O)C2)cc(=O)c(Br)c[nH]1 c1(C(N2CCC(CNC(c3c(OC)scc3)=O)C2(C)C)=O)nc2ccccc2[nH]1 c1(C(N2CCCC3CC23)C(=O)NCSc2ccc(F)cc2)nc2ccc(F)cc2s1 N1(C(C=C(C)C)=O)CC(CC(=O)NCC2CC(F)C2)C2(CC2)C1 C1(C(=O)NCC(C)N(C(c2c(Cl)c(C)n(C)n2)=O)C)CC(C(C)(C)C)=NO1 N1(C(Cc2ccc(C)o2)=O)CCN(C(=O)CC2=CCCC2)C2CCCCC12 c1(CNCC2CCN(C(COCC)=O)C2c2cccnc2)scc2c1OCCO2 C#CCCC(C(=O)N1CCC(CN=[N+]=[N-])C1)NC(c1cnc(C)nc1C)=O C(=O)(C1=NOC(CNC(c2cnnc(O)c2)=O)C1)NCCC#CCC C1(CNC(C2C=CCC2)=O)CCCC2(CN(C(=O)CCC3CCC3)C2)O1 CC1CN(C(c2ccc(F)c(Cl)c2)=O)CCN1C(=O)CC1CC1C C=CC1(C(=O)NCCCCC(CO)NC(=O)CCn2ccnc2)CCOCC1 S(=O)(=O)(c1cnn2ccc(=NCC(C)(C)C3CC3)[nH]c12)NC(C1CCCC1)CC c1(C(C)C)conc1CC(=O)NCC(C)N(C(=O)C(F)(F)C1(O)CCC1)C N1(C(Cc2cnc(C)s2)=O)CCC2CN(C(c3cccc(Br)c3F)=O)CC12 C1(NC(c2nc(CC)oc2)=O)CN(C(c2c(Br)cncc2Br)=O)CC12CC2 CC(C)C(O)C(=O)N1CCC(C)(CNC(=O)CCc2cccc(O)n2)C1 C(=O)(N=c1cnc(I)c[nH]1)C1C(O)CCN(C(C2CCCC(C)CC2)=O)C1 Cc1cc(Cl)ccc1OCC(=O)N(CC(C)NC(C1CCC(C)(C)C1)=O)C C(C1CN(C(C2(C#N)CCCO2)=O)CC1C(=O)NC1(C)CCCC1C)=CC Cc1c(C(=O)NCCOC2CCN(C(=O)CCS(N)(=O)=O)CC2)cccc1F C1(NC(=O)CC2C3CN(C(c4coc(C5CC5)n4)=O)CC23)CCN2CCC1C2 N1(C(C2(CC#C)CCCO2)=O)CCC2(CCCN(C(=O)Cc3nccn3C)C2)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC2CC(O)C1C2NC(c1c(OC)csc1)=O c1(CNC(CC2(N(C)C)CCC2)=O)ccc(C(=O)NCC2CSCCO2)cc1 c1(C(=O)NCC2CC(C)N(C(=O)CC34CNC(=O)C(C3)C4)C2)ccc(F)c(O)c1 N1(C(c2c(NCC)cccc2)=O)CCCC(C)(CNC(C2CCC(F)C2)=O)C1 N1(C(C2C(=C)CC2)=O)CCC(CN(C)C(c2cn(CC3(C)COC3)nn2)=O)C1 c1(C(=O)NCC(CNC(c2ccc(C(N)=O)o2)=O)O)cccc2ncnc(O)c12 N1(C(C2CCCN(CCC)C2)=O)CCC2(CCCN2C(=O)C=Cc2cscn2)C1 C12(C(=O)OCC)CCC(NC(c3cc(Cl)cnc3F)=O)(CC1)C2 c1(C(N(C2CC(NC(C(Cc3c(C)cccc3)C)=O)C2)C)=O)ccc(F)c(Cl)c1 C1(C(C)NC(CC2(C=C)CCC2)=O)CCN(C(C2CCCCC2)=O)CC1 O=S(=O)(c1cnc(N2CCOCC(O)C2)c(Cl)c1)NCC1(CCCO)CCCC1 C1(NC(Cc2c(C)nc[nH]2)=O)CCN(C(C2CC2CC(C)(C)C)=O)C1(C)C C1(c2cccs2)(N(C(=O)CC(C)(C)C2CCCC2)CC(=O)OC)CCCCC1 CN1CCC(CNCc2cc(C3CC3)ns2)C1c1ccc(F)cc1 C1(c2ccccc2Cl)(C(=O)NC2C(NC(C3(CCC=C)CC3)=O)C2)CCCCC1 C(c1nc2ccccc2s1)=CC(=O)NCCN(C)C(C1CCC=CCC1)=O C1(NC(C(C)N(C(C=CC(C)C)=O)C2CC2)=O)C2CCCCCC12 C#Cc1cnn(C)c1C(=O)NC(CC(C)C)C(=O)NCC12CCC(CO1)C2 c1(C(=O)NC)ccc(NC2CCNC2Cc2ccccc2)c(F)c1 c1(CC(=O)NCC23CC(CNC(C=CCC)=O)(OC2)C3)cn2cccc(C)c2n1 c1(NCC(CC)(CC)NC(=O)CC2CC=CC2)ncc2ccnc-2[nH]1 C1(NC(CCCOCC=C)=O)COCCN(C(=O)C(c2ccccc2)C2CC2)C1 C(=O)(CC(=O)Nc1cnn(CC2(C(C)(C)C)CCCO2)c1)OC c1(OC)ccc(C(=O)NCC2CCCCN2C(=O)C=CCO)cc1C1CC1 C12(C(N3CC(C=C)C(NC(=O)CCCCC)C3)=O)CCC(OC)(CC1)CC2 CCC(C)CC(=O)N1CCCCC1CCNC(=O)Cn1cnc(C(N)=O)n1 CCCCC(CC(=O)N1CCCC(N(C)C)CC1)NC(=O)CCC(C)OC Cc1cc(C(=O)NCCCN(C(=O)CC(C)(C)C)CC2CCCC2)nn1C C1(CN(c2nccc(N3CCC(CC)(CO)C3)n2)C)CCC2(CCOCC2)CO1 c1(C(=O)NC(c2c(CC)cccc2)CNC(C2C(C)C2C)=O)c(N)cccc1Cl CN1CCN(C(C2CC3(C2)CC(O)C3)=O)CC1C(N1CC(F)(F)C1)=O N1(C(c2cnn(C)c2Cl)=O)CCCCCC(NC(c2n[nH]cc2Cl)=O)C1 c1(OC)cnc(Cl)cc1C(=O)NCC1CCCC(CNC(=O)C2=C(C)CCC2)C1 c1(CN2C(C(N3CCC(O)C(F)C3)=O)CC(F)C2)c(Br)cccc1[N+](=O)[O-] C1(CNC(C(C2CCCCC2)C)=O)CN(C(c2cnc(O)n2C)=O)CC1O C1(CCNC(c2cncc(OC)n2)=O)CCN(C(c2nccnc2N)=O)C(C)C1 C1(C(=O)Nc2ccccc2)CCN(CC(O)COCCC2CCCC2)C1 c1(OC)ccc(Cl)cc1C(=O)NCC(C)(C)CN(C)C(C1CCOC1C)=O C(CC(=O)N(C(CO)C(C)C)C)(C(C)C)NC(C(C)NC(CC)=O)=O Cc1scc(C(=O)NCC(O)CN(C(=O)CN2CCN(CC(F)F)CC2)C)c1N C(CC(C)(C)C(=O)NCC(C)O)NC(c1c(C)cccn1)=O N1(C(C(C)OCCC=C)=O)CCC(CNC(c2coc(Br)n2)=O)(OC)C1 c1(C(=O)NC2CCC(N(C(c3cc(C)sn3)=O)C)C2)c(Cl)ccc(C)c1O C(=O)(C(O)C1=CCCCC1)NCCC(C(=O)NCC(CC)(CC)CO)(C)C c1(OC(C(N2CC(O)(CNC(C=CC)=O)C2)=O)C)ccc(C)cc1C CS(=O)(=O)c1ccc(C(c2nnnn2C2CCC2)NCc2ccnc(Cl)c2)o1 CCN=c1cc(C(=O)NC2(CNC(=O)C(F)(F)c3ccncc3)CCC2)cc[nH]1 c1(C(C)OC(C(C)Sc2ccc(NC(C)=O)cc2)=O)cc(=O)n2c(C)cccc2n1 C1(C2CCN(C3C(=O)N3)C2)COCCC1(C)O.c1(CCCSC)sc(Cl)nc1Cl C1(CNC(C2C(C)(C)COCC2)=O)CCN(C(C2(O)CCCC2)=O)CCC1(F)F C(CCN=C(NCCC(C)(C)C)NC1C(C)(C)C1(C)C)SC N1(C(C(C)SC(C)C)=O)CCOC2(CCN(C(=O)CC3CCC(F)(F)CC3)C2)C1 O=C1CCC2(CCC(NC(=O)CNC(=O)NCc3cccc(O)c3)CC2)N1 c1(SC(C2CCCN(C(C(C(C)(C)C)NC(N)=O)=O)C2)C)ccccc1S(N)(=O)=O N1(C(C(C(C)C)N(C)C)=O)CC2OCC(NC(=O)CCc3cccc(F)c3)C2C1 Cc1ncnc(C)c1CC(N1CCC(OCCNC(=O)C=CC2CCCC2)C1)=O C1(NC(C(CC)OC)=O)CCCC12CCN(C(=O)COc1ccccc1F)CC2 c1(-c2nc(C3C(C)C3)n(Cc3cncc(F)c3)n2)cccc(S(C)(=O)=O)c1 N1(CC)CCCC(ONC(=O)C2CC2C(C)NC(C2CCC(=O)O2)=O)C1 c1(C(=O)NCC(C)NC(C2(CCC)CCNC2=O)=O)ccnc(O)c1F Cc1cc(C(=O)NC(C)CNC(=O)CC2NC(=O)NC2=O)n(-c2ccccn2)n1 C(=O)(CC1=CCN(C(=O)C(C)C(F)F)CC1)NC(CC(C)C)C CC(C)C(CCCC(=O)O)NC(c1ccc(-n2cc(C(C)(C)O)nn2)cc1)=O CC1=C(CNC(C2CN(C(=O)C(C)N3CCCC3)CC(C)O2)=O)COCC1 C1(CNC(=O)CCC2CC2)CC2(CCOCC2)CN1C(=O)CCCC1CC1 c1(-n2c(CCOC)nc(CCN3CCCC(C)C3)n2)ccc(S(C)(=O)=O)cc1C Cc1ccc(C(N2CCC(C)C(CC(=O)NCC(C)N(C)C)C2)=O)cc1C#N Nc1c(CC(N2CCNC(=O)C2c2cccc(Br)c2)=O)cccc1Br n1(CC)ccnc1-c1cn(C(C)C(=O)NC2CC(CC(=O)OC)C2)nn1 c1(CCNC(CC2N(C(C3CN(C(=O)NC)C3)=O)CCC2)=O)nnc(C)n1C c1(CNC(CC(CC)N(C(=O)CCC(C)(C)N(C)C)C)=O)ccc(F)c(O)c1 c1(CC(N2C(CNC(C3CC(C(F)F)(OC)C3)=O)CCC2)=O)ccc(O)c(F)c1 c12cccc(c1)C(=O)N2C.C1(OC)CCCC1NC(C)C N1(C(C2C(C(C)C)C2)=O)CCC(NC(c2cn3c(n2)CCCC3)=O)C12CCC2 C1(CC(=O)NC2C(C(N(C(CC(=O)OC)C)C3CC3)=O)C2)CCCCC1O c1(C(N2CCC(CNC(C=COCC)=O)(CO)C2)=O)cnc2nccn2c1 Cc1cc(F)cc(C(=O)NC2CN(C(c3c(O)cccc3F)=O)CC23CC3)c1C Cc1nc2cc(C(=O)NC(C3CN(C(=O)Cc4cnco4)C3)C)ccc2o1 Cn1nc(-c2ccncc2)cc1CN(C(N1CC(c2ccc(F)cc2)(C)C1)=O)CCl C1(C2CC2)(NC(CC(CC)C2CCC2)=O)CCN(C(=O)COC2CCC2)C1 C1(CNC(C(C2CC(NC(c3cnn(C)c3Cl)=O)C2)F)=O)CC2(CCC2)CO1 C1(CN(C(=O)CCc2ccccn2)C)COCCN1C(c1ncc[nH]1)=O N1(C(c2c(CC)n(C)nc2)=O)CCC(NC(C2(C)CC2Br)=O)C(CO)CC1 N1(C(c2cc(CC)[nH]n2)=O)CC2(C1)CN(C(c1cccc3scnc13)=O)CCO2 Cc1cc(C)c(C(N2CC(CN(C)C(c3cnc(C)o3)=O)C3(CC3)C2)=O)c(C)n1 N1(C(C2C(CC)C2)=O)CC(O)(C(C)NC(=O)Cc2cc(C)no2)C1 C1(CC=C)(NC(=O)CSC(C)C)CCN(C(c2c(C)nn(C(C)C)c2C)=O)CC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CO)NC(C(C(C)(F)F)(C)C)=O C1(C(N2CCC(NC(C3(F)C(C)C3)=O)C2c2ccccc2)=O)CCC2(CC1)CC2 C(=O)(C(C)C(=O)OC)NC1CC(C(=O)NC(CCC=C)C)C1 C1(O)(C(=O)NCC2CC(COC)CN2C(=O)CCSC)CC2CCC1C2 CC1(C)CC=C(C(=O)N2CCCC(CO)(NC(C3CCS3(=O)=O)=O)C2)CC1 Cc1ccc(CC(=O)NCCOCCNC(c2occc2C)=O)c(Br)c1 C(=O)(CCN=c1[nH]ccs1)NC1CCCN(C(C2C(C)C2)=O)CC1 C1(OC)CC(C)CN(C(C2(C)CCN(C(=O)Cc3nocc3C)C2)=O)C1 c1(C(=O)NCC2(NC(C(C)n3cncn3)=O)CCOC2)csc2nccn12 CCCCC(C)CCC(=O)NCC1CCC(NC(c2ccc3n[nH]cc3n2)=O)C1 C1(CC(N2CCC(C)C2c2cn(CCF)nn2)=O)CCC2(CC1)OCCO2 N1(C(CCC)=O)CCCN(C(C2(n3cc(Br)cn3)CC2)C2CC2)CC1 C1(NC(CCC(=O)NCCC)=O)CCN(C(=O)C(OC)OC)CCC1CO C=C(Cl)CC(C(=O)NCC(CC1CC1)CO)NC(=O)CNC(=O)CC C1(C)(C(N2CCC(N(C(CN(C(C)C)C)=O)C)C2)=O)Cc2ccccc2C(=O)O1 c1(CC)c(C(=O)NCC(C)NC(=O)C=CC2C(C)C2(Cl)Cl)[nH]c(C)c1C(N)=O CC1(C)COC(C)(C(=O)NC2CCCN(C(=O)CCCc3ccncc3)C2)CO1 c1(C(=O)NC2(CF)CCN(C(=O)CN3CCCCCC3)C2)cc2c(s1)CCCC2 C1(CNC(CC2ON=C(CC)C2)=O)CC2CCC(C1)N2C(=O)C(C)(C)CC(C)C c1(C(N2CC3C(C(=O)NC)(C3)C2)=O)cc2cc(O)ccc2cc1O N1(C(C(CC=CCC)C)=O)CCC2(C1)CN(C(c1ccc(O)c(F)c1F)=O)C2 CCCC(CC)C(=O)NC1CCC(C)N(C(=O)Cn2ncccc2=O)C1 c1(C(c2n(CCSC)nnn2)Nc2cnc(O)c(Br)c2)cccc2sccc12 C1(F)(CNC(c2cnc(CC)[nH]2)=O)CCC(NC(c2cncc(SC)c2)=O)C1 c1(CNCCOCCN(C(C(C(=O)OCC)F)=O)C)c(C(F)(F)F)cc[nH]c1=N N1(C(c2cnn(-c3cccc(F)c3)c2)CC)CCOCC1c1n[nH]c(C)n1 N1(C(Cc2ccc(OC)cc2)=O)CC2(CNC(=O)C=C3CCCC3)CCC1CC2 c1(C(=O)NC2C(NC(CSCCC)=O)CCOC2)ccc2nncn2c1 CCCCCC(O)CC(=O)N1CCCC1CCNC(c1ncsc1CC)=O Cc1nccc(Cl)c1C(N1CC(Cn2cc(-c3ccnn3C(C)(C)C)nn2)C1)=O c12nc(nc3sccc13)CN2CCCN(C)C.C(CC(C)(C)C)Sc1cocn1 N1(C(CC2C(C)(C)C2)=O)CCC(CCNC(c2csc(F)c2)=O)C1 c1(NC(c2scc(C(=O)Nc3c(I)ccc(C)c3)n2)=O)cc(F)cc([N+](=O)[O-])c1 N(C(=NCCC1=CCCCC1)NCc1ccco1)Cc1nc(C(=O)OCC)on1 CCC(CC(=O)N1CC(C(N2CC(C)(C)CC2C)=O)C(C)(C)C1)C(F)F C1(C(=O)NCC2C(C(=O)NCCc3c(C)ncs3)CCO2)CC12CCOCC2 c1(CNC(C23N(C(c4c(C)nc(CC)o4)=O)CCC2C3)=O)ccc(O)cc1C c1(C(N2CCC(C(C)NC(C3CSC3)=O)C2)=O)ccc(Br)nc1O C(=O)(C1=CCC(NC(c2sc(F)cc2C)=O)C1)NC(C#C)(C)C1CC1 c1(C(N2CCC(N(C(CNS(CCCC)(=O)=O)=O)C)C2)=O)c(C)cccc1F c1(CCCNC2(CNCC3CCC(F)C3)CCC2)cc(O)ccc1Cl c1(C(N(C2CN(C(=O)COC(F)F)CC2F)C)=O)cc(F)cc2nn[nH]c12 C1(CNC(C=CC(C)(C)NC(c2ccc(CC)s2)=O)=O)CCC(C)(C)CC1 N1(C(C2CC(C(=O)OC)C2)=O)CC2CCCCC2C1C.N12CCOC(C1)C2=O c1(CCC(N2CCC(C3N(C(C4(C=C)COC4)=O)CCC3)C2)=O)ccnc(Cl)c1 N1(C(CCC=CC)=O)CCCC(NC(=O)Cc2cc(C)no2)CC1 c1(C(=O)NC2CC3(CN(C(C(CC)C(C)O)=O)C3)C2)cc(C)c(C)c2ncsc12 Cc1c(C(N2CCCC(CN(C(=O)CCN3C(=O)C=CC3=O)C)C2)=O)ncn1C N1(C(c2cc(C#N)no2)=O)CC2(CC2)CC1CNC(=O)CCc1nncs1 C1(C)(C(=O)NCCCN(C(C2CC2(C)C(F)(F)F)=O)CC)CC=CC1 N1(C(CCN(C)CCO)=O)CC2CC(N(C(=O)CCc3ccsc3)C)C1C2 N1(C(C(C(C)(C)C)NC(C)=O)=O)CCC(C)N(C(=O)CC2CCCCCC2)CC1 Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)Nc1cc(Cl)cc(F)c1O C1(NC(c2cnc(OC)nc2)=O)C2CC1N(C(c1cc3n(n1)CCC3)=O)C2C C(CCCCC(=O)N1CCCC(NC(=O)CCP(C)(C)=O)C1C)OCC C12(NC(C3CCN(C)C3)=O)COC(CNC(c3cn(C)nc3C(C)(C)C)=O)(C1)C2 c1(CNC(=O)NC(COC)C)ncccc1OCC1CC1(Cl)Cl Cc1oc(C(=O)N(C2C3CN(C(=O)C(C)(C)CO)CC23)C)cc1CO c1(NC(N)=O)ccc(CC(CC(=O)NCC(CNC(c2nnc(C)o2)=O)O)=O)cc1 n1(CC)nnnc1CNC(=O)CCN(C(=O)CC1CC1CC)CCO C1(CNC(c2snnc2C2CC2)=O)CN(C(=O)C2=COCC2)CC1C(F)(F)F O=C(CCCC1CC1)N(CCc1cc(C(=O)NC2CCOC2=O)no1)CCO C(=O)(C(CC(F)F)N(C(=O)C=Cc1cc[nH]c1)C)N(CCC(N)=O)CC N1(C(CC2C(C)C2)=O)CCC(NC(=O)C(N2CCCCCC2)=O)C(CO)C1 C1(CNS(C)(=O)=O)CN(C(=O)CCOCCOCCO)CCC12CCC2 CC#CC1CCN(C(=O)C(C2CCC2)NC(C2COCC2(C)C)=O)CC1 c1(C(N(C2CCN(C(C3CC(C)OC3)=O)CC2)CCO)=O)cnc2[nH]ncc2c1 CCC(CC)(CN=c1[nH]nc(C)o1)NC(c1cn(CCC(C)C)nn1)=O Cc1ccc(C(=O)NC2CCCCN(C(c3ccn(CC#N)n3)=O)C2)cc1F c1(CC(N2CCC(N(C(C=CC=CC)=O)CC)C2)=O)cc(Cl)ccc1Br c1(C(=O)NCC2CN(C(C3CC(=C)C3)=O)C3C2C3)cc(F)c(C)cc1Cl N1(C(CNS(N)(=O)=O)=O)CCC(N(C(=O)C(F)CC2CCCC2)CCO)C1 c1(CCSC)nc(-c2cc(-c3ccccc3)no2)n(C2COC(C)(C)C2)n1 C(CCCCC(=O)NC(c1nn(C)cc1O)C)NC(C1CC(C)SCC1)=O N1(C(C=CC(C)C)=O)CCOCC1C(=O)NCc1cnn(CCO)c1 C1(F)(CNC(C(n2cc(Cl)cn2)C)=O)CCN(C(C2CCC(=O)N2C)=O)CC1 c1(N(C(=O)NC(C2CCCO2)(C)C2CC2)CC)ccccc1[N+](=O)[O-] c1(C(N2CC3(CCN(C(C(C)OCCN(C)C)=O)C3)C2)=O)cc2c([nH]1)CCC(C)C2 c1(C(=O)NCC2(OC)CN(C(CCN(C)CC)=O)C2)cc(OC)c2c(c1)OCO2 C(=O)(C1CCc2nccn21)N1CCC(C(C)(C)NC(=O)Cc2cnoc2)C1 N1(C(C(C)OC)=O)CCN(C(C2(C3CCCO3)CCC2)=O)CCC1C C1(N(C)C(C2(C)CCCCO2)=O)CCCN(C(c2[nH]ncc2C2CCC2)=O)CC1 CCC(C)(C)CCCC(=O)NCCC1(C)CCN(C(C2CCOC(=O)N2)=O)C1 Cc1cc(NC(=O)C(=O)Nc2ccc(-c3ccc(CO)o3)c(F)c2)cc(Br)c1C CC1(C(N2CCCC2CCNC(=O)COc2ccc(Cl)cc2)=O)CCCNC1=O O=C(C(O)CC(F)(F)F)NCC1CCN(C(=O)CCCN2CCOC2=O)CC1 CC(CNC(=O)C(=O)N(C)C)CN(C)C(C1(CNc2cnn[nH]2)CCC1)=O C1(NC(=O)C2CC2)CN(Cc2cnc(-c3ccccn3)s2)CC1CCC(C)(C)C C1(C(=O)NC23CC(NC(c4c(COC)cco4)=O)(C2)C3)CN2CCN1CC2C c1(C(N(C(C(=O)NC(C)Cc2cncs2)=O)C)C)ccc(F)c(F)c1 C1(F)(CNC(C=C(C)C(C)C)=O)CCCN(C(c2cc(C(N)=O)cn2C)=O)C1 N1(C(=O)CC2CC2)CC(NC(C2(C3CC3)CCOCC2)=O)C(c2ccccc2)C1 CC1CN(C(=O)Cn2ncnn2)CC1(C)CNC(c1ccc(=O)n(C)n1)=O N1(C(C(C2CCCC2)OCC)=O)CCOCC1CNC(=O)CC1COC2CC1C2 C1(CNC(CC2C(CC)C2)=O)CC(C(=O)N(CC(C)C#N)C)C1 N1(C(C(C)OCCN(C)C)=O)CCCC(CNC(=O)C(C2CCCCC2)O)C1 Cc1ncnc(C)c1CC(=O)NCC1CC1CNC(c1ncccc1F)=O N1(C(C(C)(Cl)Cl)=O)CC2CS(=O)(=O)CC2(NC(=O)C=CC2CCC2)C1 c1(CNC(C(CC)NC(=O)CSC)=O)n[nH]c2c1CCC2 Cc1nc(CO)sc1C(=O)N(CC(O)CN(C(=O)C(O)Cc1cn(C)cn1)C)C N1(C(COCCC#C)=O)CCCC1(C)CNC(C1(F)CC(C(=O)OCC)C1)=O CC1CCN(C(C23CCCC2C3(F)F)=O)CCN1C(=O)CCC(=O)N(C)C c1(OC)nn(C)cc1C(N1CCCC1CNC(=O)C(F)(F)c1ncccn1)=O C1(OCCNC(C=CC(=O)OC)=O)CCN(C(C2CC23CCC3)=O)CC1 C(Cc1ccccc1)(C(=O)NCCC(N1CCOCC1)C)OC C1(C(=O)NCC(CC(C)C)NC(C(CC)N(CC)CC)=O)CC=C(C(C)C)CC1 C1(NC(COC(C)(C)CNC(=O)CC(Cl)Cl)=O)CCN2CCCCC12 c1(N2CCC(NC(C(CC)C(C)O)=O)C(O)C2)cc2nnc(C)n2cn1 C(=O)(CC(C)C(=O)NCC1CCC(C)CN1C(c1ccc(C)n1C)=O)OC N1(C(C(C=CC)O)=O)CC(F)(F)CC1CCNC(c1cc(C)sn1)=O CCC(C(=O)NCC(F)(F)CNC(=O)OC(C)(C)C)C(C)(F)F N1(C(C2N(CC)CCC2)=O)CC(CNC(c2cncnc2C(C)C)=O)CC1(C)C C(=O)(C(C)(C)C(=O)NCC1(CNC(c2ncn(C)n2)=O)CC1(F)F)NC n1(CC)cnc2[nH]c(=NCC(C)C(F)F)nc(N3CCC(CC)(CO)C3)c12 c1(SC)ccc(C(=O)NC(C)CCCCNC(=O)C=Cc2sccc2C)c(Cl)c1 CC(N=[N+]=[N-])C(=O)NC(c1cn(C)nn1)C(=O)N(C(C)CC(N)=O)C C1(CC)(NC(C2C3CC2N(C(=O)CNC(=O)NC)C3)=O)CC(F)(F)C1 Cc1nnc(O)c(C(N2CC(NC(=O)C(C)(O)C3CCC3)CC3(CC3)C2)=O)c1C c1(NC(C2CN(c3cccc(C)c3)C(=O)C2)=O)ccc2c(c1)CCN(C)C2 c1(C(C(=O)N(CCN(C(C(C2CCOC2)OC)=O)C)C)(C)O)ccc(Cl)cc1 N1(C(C2CCC2)=O)CCC(C2CCN(C=O)C2)C1.c1(C=O)cc2cn[nH]c2cn1 C(=O)(CC(C)(C)C(C)(F)F)N1CCC(C)C1CNC(=O)C(=O)NCC(F)(F)F C1(NC(C2CCN(C(N)=O)CC2)=O)COC2(C1)CN(C(C1CCCC1O)=O)C2 C(=O)(C(O)CC(C)(C)C)NC1C(CNC(c2cn(CCC)nc2C)=O)CCC1 C1(CC)CN(C(=O)C(=O)NCc2cc(Br)ccc2Br)CC(CC)O1 c1(CC)cc(C(=O)NC2CC(CNC(C3CCOC(C)C3)=O)C2)c(C)nn1 c1(C(CC)C(=O)NCC(CO)NC(c2cnc(C)o2)=O)ccc(Br)cc1 C(=O)(C(CCS(C)=O)N(C)C)N1CC(C(C)NC(Cc2c(C)cccc2C)=O)C1 Cc1cccc(NC(C2(F)CCN(Cc3cc(C(=O)O)ccc3O)C2)=O)c1Cl C1(C(=O)NC2CCCN(C(C=CCC)=O)C2C)CCOCC12CCCCC2 c1(C(CNC(CCSC)=O)NC(=O)C(C)OCCc2ccccc2)ccccc1 Fc1ccc2c(c1)CCN(c1nc(Br)cs1)C2 c1(NC(C2CC3CC3N2C(=O)COCC2CCCC2)=O)nccc2nc[nH]c12 Cc1cc(C2(C(=O)N(C)CC3CCCN(C(C4CC4(Cl)Cl)=O)C3)CC2)cc(C)c1 c1(OC)ncc(C(N2CC3CC(N4CCC4N)C2C3)=O)cc1Br.N1CCCC1 c1(OC)ccc(CCC(=O)NCC23CC2CN(C(c2cc(F)n(C)n2)=O)C3)cn1 C(=O)(C(C)CCC)NC(CNC(C1(CC=C)CCCC1)=O)CCOC CCC(C(C)O)NC(C1(CCNC(c2cn(C3CC3)cn2)=O)CCCC1)=O N1(C(c2n[nH]c(C)c2F)=O)CCC(CNC(=O)C(N2CCSCC2)C)C12CCC2 C(CC)(CCCO)NC(N(C(CC(=O)OCC)c1ccccc1)C)=O C1(=O)CCC2(CC2)NC(=O)C=CC(=O)C(=O)NCCN1.C1(C(=O)N)CCC1.CO c1(C(N2CCCC(C)(CNC(c3cn(C)nc3O)=O)C2)=O)nc2ccccc2[nH]1 C1(O)(NC(N2CC(F)(F)C2)=O)CCN(C(=O)COc2ccccc2)CC1 C(C1CN(C(C23CCC(C2)C3)=O)CC1C(=O)NC1CC(N2CCC2)C1)=CC C1(NC(C(C)(C)C2CC2C2CC2)=O)CCC(NC(=O)CC2CCOC2)CC1 CCCC(C(=O)N1CCC(C(=O)NCCc2cc(C)on2)(CC)C1)NC(N)=O C#CCC(C)(CC)C(=O)NCC1(CC(=O)NCc2cnn(C)c2C)CC1 C1(NC(C2(C(C)C)COC2)=O)CCCN(C(C2CC(O)CN2C)=O)C1 C1(NC(C(C)OCCC(C)C)=O)CC(NC(c2c[nH]nc2C2CC2)=O)CC1O C1(C(=O)NC(C2CN(C(c3ccc(N)c(Cl)c3)=O)CCO2)C)CN2CCN1CC2 c1(SCc2nc(-c3c(OC)ccnc3)on2)ncnc2sc(C)nc12 c1(C(=O)NCC(CNC(C(C)C2CCC2)=O)F)nc[nH]c2ncc(Br)c1-2 C(C(N=c1[nH]ccn2nnnc12)C(C)C)NC(c1nc(C(C)C)sc1)=O N1(CCNC(C2CC2CSc2cnn(C(F)(F)F)c2)=O)CCOCC1 c1(CN(CC(=O)NC2CCCOC2)C)coc(Br)n1 c1(SCC(=O)NCCN(C)C(c2cn(C3CCCCC3)nn2)=O)n[nH]c(=N)s1 Cc1cc(=O)n(CCC(=O)N(c2cccc(C#N)n2)C(C)C)cn1 C1(NC(c2c(C(C)C)occ2)=O)CCC2CCN(C(=O)C(C)(C)CF)C1C2 C(=O)(C=C1SCC(=O)N1C)N1C(CNC(C=CC)=O)CCCC1.C(=O)N c1(NC=O)ccc(N(C(=O)C2=CSCS2)CC2CC2)cc1.C12C=CC(C1)NC2=O C1(C(C(N2C(CNC(C3CCN(CCO)CC3)=O)CC2)=O)O)CCCCCCC1 N1(C(C(C)OC2CCCC2)=O)CCC2(CN(Cc3ccncc3Cl)C2)C1 N1(C(c2c(CC)noc2)=O)CCCC(CNC(C2(CO)CCCC2)=O)CC1 N1(C(c2cc(C)oc2C)=O)CC2CCOC2(CNC(C2CCN(C)S2(=O)=O)=O)C1 C1(NC(C=COCC)=O)CC2CN(c3nc(C(F)(F)C(F)(F)F)nc(=N)[nH]3)CC12 C(=O)(C(CC)CC)NCC1(CC=C)CN(C(=O)Cc2ccccc2SCC)C1 CC1CN(C(c2cnc(S)nc2)=O)CC(C)N(C(c2ccc(Cl)c(F)c2N)=O)C1 N1(C(CSC(C)C)=O)CCOCC1CNC(=O)C=Cc1ccc(C(N)=O)o1 c1(NC(C2CCCN(C(c3ccc(Br)nc3)=O)C2)=O)cc(Cl)ncc1Br CC(CC(=O)NC1(CC(N2CCC(CC(F)F)C2)=O)CCCCC1)C(F)F C1(C(=O)NCC2C(C)CN(C(C3CC3(C)C)=O)C2)COC2COCC12 Cc1ccc(CNC(=O)C(C)NC(=O)CN2CC3CC3C2)c(O)c1 N1(CCNC(=O)C=Cc2nccs2)CCCN(C(C2CCC2CF)=O)CC1 c1(C(=O)NCC2CC(NC(c3c(C(C)=O)ccs3)=O)C2)ccnc(F)c1Cl c1(C(N2CC(N(CC=C)C)C2)=O)cn2cccc(Br)c2n1 Cc1cnc2n1CCN(C(=O)Oc1ccccc1F)CC2 C1(C(=O)NC23CC(CNC(c4n(CCC)ccc4)=O)(C2)C3)CCC(C)(F)CC1 CC1(C)CC(CNC(C2CC(O)C2)=O)CN(C(=O)CC(C)(O)c2ccccc2)C1 c1(NCC(c2ccc(OC)cc2)OC)cc(P(C)(C)=O)ncn1 N1(C(C)=O)CCCC(CCN2CCCC2CC(N2CCCCC2)=O)C1 C1(CN(C)C(C2C3CCC2(c2ccco2)C3)=O)COCCN1C(=O)CC1CC(F)C1 C(=O)(C1=NNC(=O)C1)NCCN(C(c1nc(C)c(C)s1)=O)CC C1(NC(c2ccc(C)o2)=O)CN(C(c2cnc(Cl)s2)=O)CCC1CO Fc1ccc(CNCC23CCCCC2NCC3)c(OC(F)F)c1 c1(C(=O)NC2CN(C(c3nccc(C(F)F)n3)=O)CC2O)cc2n(n1)CCCC2 N1(C(CC2CCCC(C)(C)C2)=O)CCC2CCC(NC(c3cc(N)ccc3F)=O)C12 CC(Cc1ccccc1)(C(F)F)NCc1nnc(-c2ccccc2)s1 c1(OC)cc(C(=O)NCC2CCN(C(=O)C(C)(C)c3nccs3)C2)ccc1O c1(CC(=O)N(C(CNC(c2cnc[nH]c2=N)=O)C2CC2)C)ccc2c(c1)OCO2 C1(C(C)(C)NC(CC(C)O)=O)CCN(C(c2cc(C3CCCCC3)on2)=O)CC1 C(=O)(CC(C)C(F)(F)F)NC1CC(CC(=O)NC(COC)(C)C)C1(C)C C=CCC(C)(CC)C(=O)NC1CCCC(N(C)C(c2cnc(OC)c(Cl)c2)=O)C1 N1(CC)CCc2cc(-c3cccc(CC(C(=O)OCC)NC(=O)CSC)c3)ccc21 c1(OC(C)C)ncccc1CC(=O)NCC1(F)CC(NC(=O)CC2CCCO2)C1 C1(CNC(C=CC(CC)C)=O)(CO)CN(C(=O)CCNC(=O)OC(C)(C)C)C1 N1(C(CCSCCCC)=O)CC(C(=O)NC(=O)C(CCC)N(C)C)CC1(C)C N1(C(CC2N(CC)CCC2)=O)CCC2CC1CN2C(=O)CCCN(C)C(C)=O S(=O)(=O)(c1csc(C2CC2(F)F)n1)N(CC(CC)O)Cc1ccccc1 c1(C(=O)NC23CC(C(NOCC4C(OC)CCC4)=O)(C2)C3)c(C)ncnc1C N1(C(c2nnn(CC)c2C)=O)CC(CCNC(=O)CC(=O)N(C)C)OC(C)C1 N1(C(C(CC#CC)NC(C23CSCC2C3)=O)=O)CC2(CCC(=O)N2)C1 c1(C2C(C(=O)Nc3n(CC(=O)OC)ncc3)C2)ccc(OC)c(OC)c1 c1(C(=O)NC2CC3CC2CN3C(C2CCCCC2)=O)csc2c1CCCC2 C1(NC(C2(NC(c3cc(Cl)cn3C)=O)C(C)C2)=O)CCCN2CCCC12 C1(OC)CCCCC1C(=O)NC(C)CNC(C)=O CN1CCCC1(C)C(N1CC(CNC(c2ncnn2C2CCOCC2)=O)C1)=O C1(C(=O)NCC2(C(N)=O)CN(C(=O)CCC3CCCC(=O)N3)C2)CC(F)C(=O)N1 C=CC(C(F)(F)F)NC(C1C(NC(=O)CCNC(=O)COC)C1(C)C)=O c1(NC2CC(C)N(C(c3cnc(Cl)s3)=O)C2)ncc(C#N)cc1Br C1(CNC(C(COCC)(C)C)=O)CC2CC(C1)N(C(c1c[nH]cc(Cl)c1=O)=O)C2 C(=O)(C(C)CC(C)CC(C)C)N1CCC(CC)(NC(c2cc(OC)no2)=O)CC1 n1(CC)nnnc1C(CC)(C1CC1)NCC1CC12CC2 CC(CC1CCOCC1)N=c1cc[nH]cc1S(=O)(=O)NC1(c2cnn(C)n2)CC1 CC12COC(C(=O)NCC(C)(C)NC(c3cc(C4CC4)[nH]n3)=O)(C1)C2 C12(C(=O)NC3CC(n4cc(CCCOC(=N)O)nn4)C3)CCCC(CC1C(=O)O)C2 N1(C(c2cccc(CC)c2)=O)C(C)CC2CN(C(C3OCC4CCCC34)=O)CC12 Cn1c(O)nc2cccc(C(N3CC(CCNC(C4CCCC(O)C4)=O)C3)=O)c12 C(=O)(C1=CCCCC1)N1CC(C=C)(CC(=O)NCC2(F)CCOCC2)C1 N1(C(C2(CNC(c3c[nH]c(=N)o3)=O)CC(=C)C2)=O)CCC(F)(C(N)=O)C1 CC1(C(N2CCCC(CNC(=O)Cc3ccc(F)cc3)CC2)=O)CCNC(=O)C1 Cc1cc(N)ccc1C(=O)NCC12CC1CN(C(=O)OC(C)(C)C)C2 C1(N(C(CCC2(NC(C=NOC)=O)CCC2)=O)C)CC2CCC1CC2 C(=O)(C#CC1CCCCC1)NC(COC)CC(=O)NCC(N1CCCCC1)C C(=O)(C(F)CCC(C)C)NC1CN(C(C2CCC(C(=O)OC)CC2)=O)CC(O)C1 N1(C(CN(C)C)=O)CCCCC1CC(=O)N(CC(C)(C)CO)C CCCCC(O)C(C)C(=O)C(CC(C)N(C(=O)C(O)CCC)C)C(=O)N N1(CC(=O)NC2C(CNC(c3c(COC)nn[nH]3)=O)CCC2)CCNC(=O)C1 c1(CC(C)C)ccc(C(=O)NC2CCC2NC(=O)CCc2ccc(O)nc2)cc1 C1(OC)CC(NC(c2ccc(C(F)F)o2)=O)CN(C(C2CC2(F)F)=O)C1 c1(N2CC(C)(C)C(NC(C3(C(F)F)CCOCC3)=O)C2)c(Cl)cncc1[N+](=O)[O-] n1(CC)cnnc1CNC(=O)C(=O)Nc1cnnn1Cc1ccccc1 n1(CCC)cc(C(=O)N(CC(C)NC(C2CCCC2O)=O)CC)nn1 N1(C(c2n(CC=C)ccc2)=O)CCN(C(c2cscc2C)=O)C(C)C1 Cc1nc(C(N2CCC(C(=O)NC3CCCC3N(C)C)C2)=O)co1 C(CC1=CCC2CC1C2(C)C)OC(c1c(C(C)C)n(-c2cccc(Cl)c2)nn1)=O Cc1nc(Cl)ccc1C(N1CCCC(n2cc(CN3CCOCC3)nn2)CC1)=O C1(C2CN(C(C3CN(C(=O)NC)C3)=O)C2)(NC(C2(C(C)C)CNC(=O)C2)=O)CC1 c1(CC(CNC(C(=C)Cc2ccccc2)=O)C(=O)OC)c[nH]c2cc(F)ccc12 c1(C(N2CCC(O)(CNC(=O)CCn3cccn3)C2)=O)cnc2ncccc2c1 C(=O)(C(CO)C(C)(C)C)NC1CN(C(C(C(C)O)NC(C)=O)=O)C1 N1(C(CC2CCCC(NC(C(C3CCOCC3)C)=O)C2)=O)CC(N(C)C)C2(CC2)C1 C1(NC(c2c(CCC)nns2)=O)(CNC(=O)Cc2ccno2)CCOCC1 c1(C(N(CC(C)(C)NC(C2C(CC)OCC2)=O)C)=O)nc(C)n(C)c1C N1(C(CC)=O)CCC2(C1)CN(C(=O)C(C)NC(S(=O)(=O)Cc1ccccc1)=O)C2 N1(C(C23CCC(NC(CC4C(C)(C)C4)=O)(CC2)C3)=O)CCN2CC(O)CC2C1 c1(C(C(=O)NCC(Cn2cc(CN(C(C)=O)C)nn2)(F)F)C2CC2)ccc(Cl)cc1 c1(NC(c2n(Cc3nnn(C)n3)nnn2)C2CC2)cn(C)nc1Oc1ccccc1 C12(C(=O)NCCc3c(CNC(COCC)=O)cccc3)CCCC1C2(F)F C(c1ccc(C)cn1)=CC(N1CC(C(C)NC(CC2(OC)CC2)=O)OCC1)=O CC(F)CC(=O)N1CCC(CCNC(=O)CCCF)C1 c1(NCCC(C)C)[nH]c(=NC2CSCC2C)nc2scnc12 C(=O)(CC(O)CNC(c1ncncc1Cl)=O)NC(C(=O)NC)(C)C c1(CC)ncc(C(=O)NC(C2CC(NC(C3CC(CC(C)(C)C)C3)=O)C2)C)cn1 Cc1nc([N+](=O)[O-])cn1CC(N1CCOC(CCNC(=O)C(C)CC(F)F)C1)=O C#Cc1ccc(C(N2CCC(CC(N)=O)(NC(C3CC3COC)=O)CC2)=O)cc1 C1(NC(C=CCC)=O)CC2CCC(C1)N2C(C1(CO)CCC1)=O N1(C(C2C(CC)CCO2)=O)CC2CC1C2CNC(=O)Cc1ccn(CC(C)C)n1 C(=O)(C1c2ccccc2Oc2ccccc21)NC1C(NC(=O)CCF)C1 C1(C(=O)NCC(CO)NC(=O)CC(=O)NC2CC2)(C(F)F)CC(F)(F)C1 C12(C(N(CCC)CCNC(C34COC(C3)C4)=O)=O)CCCC1(C(N)=O)C2 CC1(C)CCC(C(=O)NCC2CCC2)(NC(C23C(=O)C4CC2C3C4)=O)C1 c1(C(N(CCN(C(C2CC2F)=O)CC)CC)=O)cc(C)nn1CC(=O)OC C1(SCC)CCC(C)N(Cc2ccc(Nc3cn(C)nc3C#N)cc2)C1 Cc1cccn(CC(=O)NCC2CC(C)CCN2C(C2CCCC23CC3)=O)c1=O CC1CN(C(=O)NCCc2cnco2)CC(C)(C(F)F)O1 C1(CCNC(CC2(OC)CN(C(C3CCS(=O)CC3)=O)C2)=O)CCC(C)(C)C1 C(=O)(CCCC(CC)CC)NCC(CCC)C(=O)N1CCC1C1CCCCC1 c1(OC)ccc(C2CC2)c(C(=O)NCCC(C(C)C)NC(=O)C2=C(Cl)CCC2)c1 c1(C(N(C2CC(NC(C3(OC(C)=O)CC3)=O)C2)C)=O)cc2c(C)c(Cl)ccc2[nH]1 Cc1ccc2oc(N3CCC(C(C4C5Cc6ccccc6C45)=O)CC3)nc2c1 N1(C(c2c(C)cc(C3CC3)cc2)=O)CC2CCC1CC2NC(C1SCCCS1)=O c1(C(=O)NCC(CC)NC(=O)CCC=C(C)C)cnc(C)[nH]c1=N C1(CNC(c2c(OC)c(C)sc2)=O)CCC(C)N(C(C2OCCN(C)C2=O)=O)C1 C1(C(=O)OC)Cc2ccc(S(=O)(=O)NC(c3ccoc3C)=O)cc2C1 CCCC(C(=O)NCC(O)CC(=O)NCC(=O)NOC)OCC C1(NC(CCc2scc(C)c2)=O)CC2(C1)CN(C(C13CCC(CC1)CC3)=O)C2 C1(CNC(c2c[nH]c(=N)o2)=O)CCCC(NC(=O)C(c2ccccc2)O)C1 C1(OC)CC(OC)CN(C(C2CCCCN2C(=O)C(C)C)=O)C1 c1(OC)ccc(OC)c(C(N2CCCC(CCNC(=O)C=CC(C)C)C2)=O)c1 c1(NC(C)=O)ccc(CC(=O)NC(C)CNC(c2c(C)ncn2C)=O)cc1 N1(C(C(CC)n2cncn2)=O)CCC(C(=O)NCc2ccc(Cl)nc2)C(C)(C)C1 N1(C(C(C)Cn2ccnc2)=O)CCN(C(c2cncc(O)c2)=O)CC(C)(F)C1 c1(C(N(C2CCN(c3nnc(O)s3)C2)C)=O)c[nH]nc1C1CCOCC1 C1(NC(=O)NC(CC(C)C)c2ccccn2)CC2CCCC2C1 c1(C(=O)NC(CN(C(=O)C(=O)N(c2ccccc2)C)CC)C)nn(CC)nc1C C1(CC)CN(C(C23CC(CCO2)C3)=O)CCN1C(=O)Cn1nc(C)cc1C C=CCC(CNC(=O)CNC(=O)C(C)(C)C)NC(=O)CSc1ccccn1 CCCCC(F)C(=O)N1CCC(C)(NC(C2CCCN2C=O)=O)CC1 C1(C(C)C)CN(C(=O)CC2CCCC(NC(C3CCC4(CC4)C3)=O)C2)CCN1C N#CC1CCCC(C(N2CCCN(C(c3ccc(C4CC4)s3)=O)CC2)=O)C1 C1(CN(C(c2cc(CO)[nH]n2)=O)CC)CCCCN1C(=O)CN1CCCCCC1 c1(C(N2C(CN(C(=O)C3=C(Cl)CC3)C)CCCC2)=O)ccc2c(O)n[nH]c2c1 N1(C(CC(CC)C)=O)CCCC(NC(C2(C)CCOCC2)=O)C1C c1(C(N2CCCC(NC(C3CCC(OC)CC3)=O)C2)=O)ccc2ncccc2c1 C12(C(=O)NCCOCCOCC)COCC1CN(C(=O)CC1CCC(=O)N1)C2 CC1(CO)CC(NC(=O)CCOCCNC(C2(O)CCC2)=O)C1 c1(-c2onc(CC3Cc4c(nc(C)s4)CC3)n2)cc(C)cc2c1NCCC2C N1(CC(=O)N(C(CCNC(C2ON=C(C)C2)=O)C)C)CC2CCC1C2 c1(CC)nn(C)c(Cl)c1C(=O)NC1(COC)CN(C(C2CC(SC)C2)=O)C1 c1(CC)cccc(CC(N2CCN(C(=O)CN(CC)CC)CC2)=O)c1 C1(CNC(c2cc(C)on2)=O)CC(C)CN(C(C2(CN(C)C)CC2)=O)C1 S1(=O)(=O)c2ccc(cc2)CN1C.C1(OCC(F)F)CC1CC Cc1cc(C(=O)NC(CNC(=O)C(F)(F)c2cncs2)C(C)C)co1 Cc1cc(C(=O)NCCC(C)NC(C2(CN(C)C)CC2)=O)on1 C=C1CCC(C(=O)NCc2nocc2C(=O)NC(C)(CO)CCF)CC1 N1(C(C(c2c(CC)cccc2)(F)F)=O)CCCC(O)(CNC(C2CC2(C)C)=O)C1 N1(C(COCCCC)=O)CCCC(NC(c2cccc(C3(C)CC3)c2)=O)C1C C12(CNC(c3ccncc3)=O)CC1CN(C(=O)CNC(C1CCCCC1)=O)C2 C(CCC(C)C(=O)N1CCCC(NC(c2nonc2N)=O)C1)OC C1(C(=O)NC(CC=C)CC)(CC)CCN(C(C2CCCCC2O)=O)CC1 c1(C(N2CCC(C)(CNC(CC3CC(C)C3)=O)C2)=O)ccc2c(=O)ccoc2c1 c1(OC)noc(-c2nc(C3CCCC3)nn2-c2cccnc2)c1Br C1(CNC(c2c(OCC=C)cccc2)=O)CC2CCC1N2C(=O)CC1(OC)CC1 C1(C(=O)NC2CC(NC(=O)CCCn3cccn3)C2)(OC)CCOC1 c1(C(=O)NCC(C)CNC(=O)CSc2cccc(F)c2)cccc2nonc12 N12CCCC1(C1CC1)C(=O)NOCC2=O.CCCC(C)OCC N1(CCC)CC(CNC(c2ccccc2I)c2nnnn2C)CC1=O C1(C(=O)NC2C(C)CN(C(c3cnn(CC(F)F)n3)=O)C2)CCCCC1(F)F c1(C(N(CC(CC)NC(=O)C(c2cnn(C)c2)OC)C)=O)[nH]c(C)nc1C N1(Cc2c(C)nc(-c3ccc(OC)cc3)s2)C(=O)CCN(CC2C3CCC23)C1=O c1(C(=O)NC(Cn2cccn2)C(=O)O)ccc(C(F)(F)F)c(Cl)c1 C1(NC(C(CC)OCC)=O)C2CC3C1C3C2C(=O)N(CCF)C1CC1 c1(C(N2C(C(CNC(c3cn(C)nc3)=O)(C)C)CCC2)=O)cc(O)cc(C#N)c1 c1(C(N2CC3CC(CNC(=O)COCCF)C3C2)=O)ccc2cncn2c1 C(=O)(CC(C(F)F)C(=O)OC(C)(C)C)NCCCC(C)NC(C1(C)CC(=C)C1)=O C1(C(N2CCC(F)(C(N3CC4C(CO)C4C3)=O)C2)=O)CCCC2(CC2)C1 C1(CNC(Cc2cn(CC)nc2)=O)CCCCN(C(c2nnc(C)s2)=O)C1 C1(C(=O)Nc2cccc(C)c2)CN(Cc2csc(-c3ccco3)n2)CC1(F)F c1(C(=O)NCCC=C)n[nH]c2ccc(-c3cnn(CCCNC(C)=O)c3)cc12 C(=O)(CC(O)CC(C)(C)C)N1CCCCC(N(C(C(=O)NCC)=O)C)C1 N1(C(C(C)N(C(c2ccc(C)[nH]2)=O)C)=O)CCC2CCN(C)CC12 c1(C(N(CCN(C(C2CC(=O)N(O)C2)=O)CC)CC)=O)cc(CC(C)C)nc(O)c1 c1(C(C(N2CCCC(CN(C(c3cc(C)on3)=O)C)C2)=O)O)ccc(C#N)cc1 c1(CNC(c2ccc(C)cn2)=O)nc2c(s1)CN(C(c1csc(S)n1)=O)CC2 C#CCC(C)(C)C(=O)NCC(CC=C)C(=O)N1CC(N2CCC2)C1 CC1Cc2n[nH]cc2CN(CN(c2ccc3c(c2)CC(SC(C)(C)C)CC3)C)C1 c1(C(=O)NC(CCCNC(c2c(CC)occ2)=O)C)ccc2ccccc2n1 N1(C(C2CCN(C)C2)=O)CCCC2CN(C(=O)Cc3ccc(F)c(Cl)c3)CC12 C1(CN(C(C2C(C)C2C)=O)C)CCN(C(=O)CC2(N(C)C)CCCC2)C12CCC2 CC(C)CC(C(=O)NCC1CNC(=O)CO1)NC(c1cccc(=O)o1)=O c1(OCC)ccc(C(=O)Nc2nccc(C#N)c2OC)c2ccccc12 c1(C(=O)NCC(CN(C(C(CC)(F)F)=O)C)O)cccc(F)c1C C(CCCCCNC(C1CCCCO1)=O)N(C(C(c1cccc(Cl)c1)OC)=O)C C(=O)(CCC(=O)NC(CO)C(=O)NC(C1CCCC1O)C)NCCC Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(C)(C)Cl)cnn1 N1(C(C2(C)CCC(F)(F)C2)=O)CC2(CCCN(C(c3nocc3Cl)=O)C2)C1 C1(NC(c2n(CCCSC)nnn2)(C)CCBr)CC12CCCCC2 C1(NC(CCC(=C)Cl)=O)CCN(C(=O)C(C)NC(=O)CC)C2CC12 C1(C(N2CCC(COC)C2)=O)CC(F)CN1C(c1ccc(Cl)o1)=O C(=O)(C1=CCCSC1)NCC1(OC)CCN(C(c2cccc(F)c2F)=O)C1 C(=O)(C1=NOC(CNC(=O)C(F)(F)CC)C1)NCCN(CCO)CC c1(NC(=O)NCCN(CC(c2ccnn2C)O)CC)c(C)noc1C C1(S(C)(=O)=O)(C(=O)NCCN(C(=O)CC2CCCS2(=O)=O)C)CCC1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC(O)CNC(=O)CC1CCCC(=O)N1 CC(C)C(C(=O)NC12CC1CN(C(=O)CCCCn1ccnn1)C2)c1cccs1 C1(C(=O)NCC2(CNC(CC)=O)CCCC2)CCCCC1C1CC1 c1(C(=O)NC2CC(CCNC(C3CN(C(C)=O)C3)=O)C2)ccnc(C2CC2)c1 CC1CN(C(c2cnc(O)o2)=O)CC(CCNC(C23CC(F)(C2)C3)=O)O1 CCC(C)CC(C(=O)NC1CC(CO)C2CC12)NC(c1c(CO)n[nH]c1C)=O Cc1cnc(C(=O)NC2COCC2NC(=O)CSc2ccc(C(C)C)cc2)cn1 N1(C(CCC=C)=O)CC(C(F)(F)F)OCC1CNC(=O)Cc1cccc(O)c1 C1(C(N2CC(CC=C)C(O)C2)=O)CN(C(C2CC3(CCC3=O)C2)=O)CC1(F)F C(=O)(C1CCCc2cccnc21)N1CC(OC)(CNC(=O)C=C2CCC(C)C2)C1 N1(C(C(CC#C)O)=O)CC2(C1)CN(C(c1cc(CC)ccn1)=O)C2 C(=O)(C1CCCc2cncn21)N1CCC(NC(c2ccnc(S)c2)=O)CC1 N1(C(=O)CC2COCCN2C(c2cccnc2Br)=O)CCc2ccsc2C1 N1(C(CC)C(=O)NC2(CO)CC(O)C2)CC(C)OC(C)C1 C1(C(=O)NC(CC=C)C2CC2)CCCC(NC(C2CC(C)=NO2)=O)CC1 N1(C(CCC(C)SC)=O)CCOCC(CNC(c2ccc(C(N)=O)o2)=O)C1 N1(C(c2snc(C)c2Cl)=O)CC(F)(F)CC1Cn1cc(CC(C)O)nn1 c1(C(=O)NCCN(C(c2c(C)snn2)=O)C)ccnnc1NC1CC1 c1(NC(C2CC3CC3N2C(c2sc(Br)cc2Br)=O)=O)cc(Cl)cc(Cl)c1F c1(CC(=O)NCC2N(C(c3cccc(OCC)c3)=O)CC2)ccc(C)c(F)c1 CCC(CCCC(=O)NCC1(C2(O)CCC2)CC1)NC(=O)CSC CC(c1ccsc1)=CC(=O)NCCCN(CCO)C(C1CC1c1cccnc1)=O N1(C(=O)Nc2cnn(-c3cccc(C)c3)n2)CCCc2c(N(C)C)cccc21 C1(NC(c2ccnn2CC(F)F)=O)CCN(C(=O)C2=COCCC2)C12CCCC2 c1(CNC(=O)NC2C(OC(C)(C)C)CCCC2)cccc([N+](=O)[O-])c1 C1(C2CCN(C(c3nncs3)=O)CC2)(NC(=O)COCCF)CCC1 C1(=O)CC(C(F)(F)F)N1.c1(C(=O)NCc2sc(C)c(CO)n2)cc(Cl)cc(F)c1N C1(OC)CCC2CN(C(=O)CCCCN(C(=O)CCCC3CC3C)C)CC12 c1(C(=O)NC(CNC(c2ncn(C(C)C)n2)=O)C)ccccc1F c1(CN(C)C(=O)OC(C)(C)C)ccc(C(=O)Nc2ccccc2C2CC2)cc1 C1(C(=O)NC(CNC(C2(CCN(C)C)CC2)=O)C(C)C)(CC)CCCO1 c1(C(N(C)CC2CCCC(NC(c3c(C)nn[nH]3)=O)C2)=O)cc(Cl)c(Cl)cc1N Cc1c(C(=O)NCC2CN(C(=O)C(C)(O)C3CC3)CCO2)ccn1C(C)C C(=O)(C(O)CC[S+](C)C)NC1C(NC(Cn2ncc(C)c2)=O)CCC1 C(=O)(CC(C)CNC(c1cc(OC)nn1C)=O)N1CC(O)(CCC)C1 C1(OCC)CC(NC(=O)N(C2(C)CCCC2)C)C12CCCO2 C1(CC)(CNC(C2CCN2C2CCCC2)=O)CCN(C(C2CC3CC3C2)=O)CC1 C1(CNC(c2cnc(NC(C)=O)s2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 c1(-c2ccc(CN3C(C)(C(=O)OC)CCC3)s2)cc(C(F)(F)F)ncc1F N#CC1(CC(=O)NCC2CC2CNC(C2(OCc3ccccc3)CC2)=O)CCC1 C1(CC(=O)N(CCC(C2CCCC2)NC(C(C)=C(CC)C)=O)C)CSCCS1 CCC(C)(CC)C(N)NCc1c(C)nn(C(C)(C)C)c1C C=CCC(CC)C(=O)NCCOCCN(C(=O)Cc1cc(C)cc(C)c1)C C1(NCc2nccc(C)n2)CC(=O)N(c2cccc(C(C)C)c2)C1=O c1(SC)cccc(CNC(c2nnnn2C2CC2)c2ccno2)c1 CC(C(=O)NCC(F)CNC(C1(CO)CCCC1)=O)C(=O)N1CCOCC1 C(CNC(C1C=CC=CC=C1)=O)(CC(C)C)NC(C1(OC)CCC1)=O C1(N(CCC)C(C2CSCN2C(C)=O)=O)CCN(C(=O)C(CCO)N(C)C)CC1 N1(C(C(=O)Nc2c(OC)cc(SC)cc2)=O)CCC(O)(C2CCC2)CC1 c1(C(N2CCC(O)(C(C)NC(C(C)N(CC)CC)=O)C2)=O)ccn2nccc2c1 N1(C(c2ccc(C)o2)=O)CCCC2(C1)CN(C(=O)CC1CCC13CCC3)CCO2 c1(OC)ncnc(C(N2CCC(NC(C3(C#N)CCCC3)=O)C(C)C2)=O)c1F C1(NC(COCCOC)=O)CC12CCN(C(c1cnc(Br)o1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NC1(COC)CCN(C(=O)Cc2sc(O)nc2O)C1 C(=O)(C(C)(C)C1=CCN(C(c2ccsn2)=O)C1)NCC(C)Cc1cn[nH]c1 c1(C(F)F)ccc(CNCc2sc(-c3ccccc3)cc2Br)cc1 Cc1n[nH]c(=NCC(C)N(C)C(c2ccc(OCC(N)=O)cc2)=O)o1 N(C(=NCc1cc(C(F)(F)F)cs1)NC(c1nnc(C)s1)C)C(CC)C C1(CNC(c2sc(CC)c(C)c2)=O)CC(C)(C)CN1C(C1CCCC(C)(C)C1)=O Cc1cc(NC(C2CC(F)CN(C(=O)Cc3cnc(C)s3)C2)=O)cc(Br)c1 CC(CC(=O)NCC(c1ccccc1F)NC(=O)C#CC1CCC1)C(C)(C)C C1(C(=O)NCC2(SC)CCC2)CCC(C(F)(F)F)N1C(=O)CN1CCSCC1 c1(C(=O)NCC(C)N(C)C(C2CC(C)(C)CN2C)=O)nc[nH]c2ncnc1-2 C1(NC(=O)Nc2cccc(O)c2)CCCN(C(c2cnccn2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CCOCC(CNC(c2cnsc2C)=O)C1 Cc1cnc(C(=O)NC2C3CC2CN(C(=O)CCc2nc(=N)[nH][nH]2)C3)cc1C c1(C(N2CCN(C(c3ccc(C(C)=O)[nH]3)=O)CC2CO)=O)csc(S(N)(=O)=O)c1 Cc1nc(F)ccc1-c1cn(CC(C)NC(=O)CCCN(C)C)nn1 c1(CC)cc(NC(=O)C(C)(C)CCNC(=O)CN2CCCC2C)cc(O)c1 N1(C(CCC#C)=O)CCC2(CC2C(=O)NC(CN(C)C)C(C)(C)C)C1 C(=O)(C(O)C1=CCCCC1)NC(C(NOCC(=O)OC)=O)C1CCC1 O=S1(=O)C=C(CNS(=O)(=O)c2cnn(-c3ccccc3F)c2)Cc2ccccc21 C1(C(C)(C)C)CCCCN1C(C1(NC(=O)CC2(O)CCCCC2)CCC1)=O C=CCC(C(=O)NCc1cc[nH]c1C(N1CC(O)(CCC)C1)=O)C(C)C C1(NC(C(C)SC(F)(F)F)=O)C2CC3CN(C(=O)C=C4CCN(C)C4)C1C3C2 n1(C(CC)CC)ccc(C(=O)NCC(C)(O)CNC(c2ccc(C(C)C)[nH]2)=O)n1 N1(C(CC=CCC)=O)CC2(CCC(CNC(C3CC(O)CN3C)=O)O2)C1 c1(OC)ccc2oc(C)c(C(=O)NC3CCCCN(C(=O)C(C)(C)OC)C3)c2c1 N1(C(C(C)(C2CC2)OC)=O)CCOCC(C(=O)NC2(CCO)CCCC2)C1 CC1(C)CN(C(=O)C2=COCC2)CC1CNC(=O)C=Cc1cnccn1 S(=O)(=O)(c1cccc2c(N(C)C)cccc12)NC1CCN(C(C(CC)CC)=O)C1 c1(C(N(C(CNC(c2ccnc(C)c2C)=O)C)C)=O)cnc2ccoc2c1 Cc1ccc(C(=O)N(C(CO)C(=O)N(C)C)C)cc1.C1=CCNC1=O C(=O)(C(C)(CCC)CCC)NC(CC#C)CC(=O)NCc1cncn1C N1(C(C2CCC(NC(C)=O)CC2)=O)CC2CN(C(c3ocnc3C)=O)CC12 Cc1cnc(N2CC3CN(C(=O)C(O)C4CCC4)CC3C2)nc1S(C)(=O)=O Cn1ccc(C=CC(N2C(C(=O)NCCOCCN=[N+]=[N-])CCC2C2CC2)=O)c1 c1(C(N(CC(CC)NC(=O)CC2CCCOC2)C)=O)ccc2cnccc2c1 C1(C(=O)NCCCCCN(C(c2cc(OC)no2)=O)C)CNC(=O)C(C)(C)C1 c1(N(C)C)ncc(C(=O)NCCC2CCN(C(C3CCOCC3)=O)C2)cn1 C1(CC(C)(C)C)COCCN1C(=O)Nc1ccncc1F c1(C(c2nnnn2CCC2CC=CC2)NC(=O)OC(C)(C)C)nc(C2CC2)no1 C(CCC(=O)NC1(C(=O)N(CC(N)=O)C)CC1)SC C1(NC(CSCC(C)C)=O)CCC(CNC(c2ccsc2)=O)C1 C1(C2(O)CN(C(=O)C(CO)C(C)C)C2)(CNC(c2c(C)ccc(N)c2)=O)CC1 c12ccc(cc1)COC2=O.c1(CC(=O)NCC)ccc(OCCO)cc1 C1(C(=O)NCC(CNC(COCCC)=O)(C)F)CCc2nc(C)cn2C1 c1(C(=O)NC(CNC(C(C=C)O)=O)C2CCC2)cccc(C(F)(F)F)c1 C(=O)C(O)CCC(C)C.n1(CCNCC)cc(C(c2cccnc2)O)nn1 C1(CNC(CNC(C)=O)=O)CC2(CCN(C(=O)C=C(C)c3cnn(C)c3)C2)CO1 Cc1noc2nc(C(C)C)cc(C(=O)NCCN(C(=O)C(=O)NC3CC3)C)c12 c1(N(CCOC)C)nc(NC2CC(C)(C)C2OC)nc2c1CCC2 c1(C(=O)NC2(C)CC(NC(CCNC(=O)NC)=O)C2)cnc2c(cnn2C)c1 c1(OC)ccc2cc(C(=O)NC3CN(C(c4cc(C)c(C)o4)=O)CC3C)[nH]c2c1 c1(NC)cc(C(=O)N(CCCNC(=O)C(C)C(F)F)CCO)cc(Cl)n1 c1(C(N)=O)nccnc1C(=O)NCCOCCCNC(=O)CC1CSCCS1 C(=O)(C(C)(C)CC#N)N1CCCC(N2CCN(C(Cc3cnn(C)n3)=O)CC2)C1 c1(C(=O)NCCN(C(c2cc(C(N)=O)co2)=O)CC)cc(C(C)(C)C)no1 Cc1ccc(-n2cc(CCNC(c3cc(C(F)(F)F)on3)=O)nn2)nc1 c1(CC)cc(C(=O)NC2CC3CC2N(C(C24COC(COC)(C2)C4)=O)C3)cc(O)n1 C1(C2CCN(C(=O)CN3CC4CC4C3)CC2)(NC(=O)C(O)C2CCCC2)CCC1 C1(NC(=O)COCC2CCOC2)CCCCCC1.C12CN(C1)C2 C1(NC(C2(C)CC=CCC2)=O)CCN(C(c2ccc(O)c(N)n2)=O)CC1F C1(C(=O)NC(CN(C(C2CN(C(=O)OC(C)(C)C)C2)=O)CC)C)CCCC(F)(F)C1 CCCC(C)(CCC)C(=O)NC(CC1CC1)C(=O)NC(c1cccc(O)c1)C N1(C(c2c(OCC=C)cccn2)=O)CCCCC(NC(=O)CCCC(=O)OC)C1 N1(C(c2[nH]cc(C)c2)=O)CCC2CCCN(C(c3nnn(C)c3N)=O)C2C1 C1(C(C)C)CC(C(=O)N(C)Cc2cn(-c3ccccc3Cl)nn2)CCO1 c1(C(=O)NCCN(C(=O)CC2(COC)CC2)CC)ccc(C(C)C)nc1C N1(c2nc(C)cc(OC)n2)CC(NC(=O)CN2CCCCCC2)C2CCCCC12 C(=O)(CCOC1CN(C(=O)CSc2nc[nH]n2)C1)NCCCC1C(C)C1 C1(C)(CC)C=C(C(=O)N2CCC(CC(=O)NCC(O)C(C)(C)O)CC2)C1 c1(N2CCC(c3ccc(C(C)C)cc3)(C)C2)c(F)cc(C#N)cc1F c1(C(N2CC(NC(CC(=O)OCC)=O)C3(C2)CC3)=O)c(F)ccc(I)c1F N1(C(c2cc(OC)ncc2Cl)C(=O)NCCCSC)CCCC2(CCNC2=O)C1 N1(C(C2CCC3(CC3)N2C(C2CC(O)C(F)C2)=O)=O)CC=CC12CCOCC2 C1(C(N2CC(N(CCOC)C)C2)=O)OCCC1CNC(C1CCC1COC)=O C1(NC(C2(C)C(C)C2)=O)CCN(C(C2CC2c2ccnn2C)=O)C1 C1(CC)CCN(C(c2ncn(C)c2C)=O)C1C(=O)NCC(C)(C)n1cccn1 c1(OCC=C)cccc(CN2CC(NC(c3ccc(CO)o3)=O)C(F)C2)c1 c1(C(=O)NCC(CNC(CCCCOCC)=O)C)ncc2[nH]ncc2n1 n1(CCC)nnc(NC(=O)C(C(C)O)NC2CC2C2CNC2)c1C#N c1(C(N2C(C(=O)O)CSCC2)=O)sc2sccc2c1Cl N1(CC)CC(C(=O)NC2CC(CCF)C2)CC1=O.C(=O)(CN)NC(=O)NC1CC1 Cc1nc(CC(C)C)oc1C(=O)N(C(C)CCNC(=O)CNC(N)=O)C N1(C(CC2(OC)CCC2)=O)CC2CC1CN(C(c1c(C)ccc(F)c1O)=O)C2 C(=O)(CN=c1ccc(C#N)c[nH]1)N1C(C)CN(C(=O)Cc2ccnn2C)C(C)C1 C1(NC(c2cc(OC)ncc2)=O)CCCCCN(C(=O)C(C2CCCCC2)=O)C1 C1(C(N(CCCCNC(CCc2cncc(C)c2)=O)C)=O)CN2CCN1CC2C C1(C#N)(C(N(CCCN(C(=O)C(C)(C)c2cnco2)C)C)=O)CC2CCC1CC2 c1(SC)cccc(CC(N2CCCC(CCc3cnc(N(C)C)nc3)C2)=O)c1 c1(CCOCCC(=O)N(CCNC(C2(SCC)CC2)=O)C)ccc(C)cc1 C12(C(=O)NCC3CN(C(CC4CC(C)C4)=O)CC3O)CCC(C)(CC1)OC2(C)C CCCCC(O)CC(=O)NCCN1CCCN(C(c2cc3scnc3[nH]2)=O)CC1 C1(CC(N2C(CN(C(CCOCC)=O)C)CCC2)=O)CCC(=O)CC1 c1(OC)cc(C(N2CCCC(NC(C3CC(C)C3)=O)C2)=O)ccc1C CN1CCC(C#N)(C(=O)N(C2CC(NC(=O)C(C)(F)F)C2)C)CC1 C1(C(N2CC(SC)(CNC(c3cccc(OC)n3)=O)C2)=O)CC2CC1CC2=O c1(CC(C)C)c[nH]c(C(=O)NC2COCC2n2cc(C3(C(=O)O)CC3)nn2)c1 c1(CC)cc(NC2(CCSC)CCC2)ccc1O CCC(C)(C)C(O)C(=O)NCC1(CNC(c2cc(CO)[nH]n2)=O)CC(F)(F)C1 CC(CC(=O)NCC1CCCCCN1C(=O)Cn1cnnc1O)CC(F)(F)F Cc1ccc(SCC(=O)NCC(C2CC2)N(C(=O)CCc2cccs2)C)cc1 C(=O)(C#CC1CCOCC1)N1CCN(C(CN(C2CC2)CC)=O)CC1C(F)F N1(C(CC)=O)Cc2ccccc2C(CNC(c2cnc(O)n2C)=O)C1 N1(C(C=CC(=O)N(C)C)=O)CC(OC)C(C(=O)NC2(C(N)=O)CC2)C1 C1(CCNC(c2cnc(C(C)C)[nH]2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC(C)O1 N1(C(CCSCC)=O)CCC(C2CCN(C(c3cn[nH]c3)=O)C2)C1 C1(C(=O)Nc2ccc(C#C)nc2)CCCCCCN1C(=O)CC1CCCOC1 N1(C(c2c(NC)cccc2)=O)CCOC(C)(CNC(=O)CCn2ccnc2)C1 C=CCCC(F)(F)C(=O)NC(CCC)CCCNC(c1[nH]nnc1C1CC1)=O c1(C(=O)NC(CNC(c2c(OCC)n[nH]c2)=O)C)ccc(C)c(F)c1Br c1(CN(C2CCN(C(C)=O)C2)C(=O)OC(C)(C)C)nccc2c(C)cccc12 N1(c2sc3cccc(C)c3n2)CC(C(=O)N(C)C)Oc2ccccc21 c1(C(=O)NC(C)CN(C)C(C2C3(CC3)C23CC3)=O)cc([N+](=O)[O-])cc(Cl)c1Cl N1(C(CCCOC)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C(C2CC2)C1 c1(OCC(=O)N(CC(C)NC(CSCC#C)=O)CC)ccc(F)nc1 C1(CC(=O)N(C2CCCCC2)C(=O)OCC2CC(F)(F)C2)COC(C(F)(F)F)C1 C1(CNC(C(CC)OC)=O)CC2CCCCC2N1C(=O)CCOC1CCCCC1 C12(CC(=O)NC(C3CCCN(C(=O)CS(N)(=O)=O)C3)C)CC3CC(CC(C3)C1)C2 Cn1nc(C(=O)NCC(C2CC2)NC(c2c(Cl)n[nH]c2C2CC2)=O)cc1CO c1(C(N2C(CN(C)C(C3COC4COCC34)=O)CCCC2)=O)cc2c(s1)CCC2 CCC(N=c1[nH]c(=NCCCc2cnn(CC)c2)[nH]c2c1CCCC2)C1CC1 C(=O)(C1=C(C2CCCCC2)N(CC(F)F)C(=S)NC1c1cnn[nH]1)OCC c1(C(=O)NCCOCCn2cc(C3(C)CCOCC3)nn2)cnn2c1OCC(F)C2 c1(C(N2CCCC(C(C)NC(=O)CCC(=O)N(C)C)C2)=O)cc(N(C)C)ccc1F C1(C(=O)NC(C2(O)CCN(C(c3cnc(N)cn3)=O)C2)C)Cc2ccccc2O1 C1(C(C(=O)N(CCCCN(C(C(c2cnccn2)C)=O)C)C)F)CCCCC1 CCCC(C(=O)OC)C(=O)NCC#CC(N1CCC2C(C(N)=O)C2C1)=O c1(C(=O)NCC2N(C(CC3OCC(C)(C)C3)=O)CC(O)C2)cnc(S(C)(=O)=O)s1 O=C(CC1CCc2ccccc21)NC1(CNC(C2CC2C2CCCC2)=O)CC1 c1(CC(=O)NC2(CN(C)C(C3CC(F)C(=O)N3C)=O)CCC2)c(F)cncc1Cl N1(C(C(C)OC2CCCC2)=O)CCN(C)C(C(N2CC(F)CC(F)C2)=O)C1 N1(C(c2n(C)ncc2C2CC2)=O)CC2CN(C(C34CCCC3(CO)C4)=O)CC2C1 N1(C(CC(CC)C2CCC2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1C(C)C C(=O)(CCC(C)(C)F)CC(C)N(C(=O)C(c1ccccc1)F)CCNC c1(C(N2CC(CNC(c3n(OC)cnc3C)=O)OCC2)=O)cnc2[nH]cnc2c1 Cc1cn(CC(=O)NC2CCN(C(C3CCC3(C)C)=O)C23CCC3)c(=O)nc1O C(=O)(C1=CCSC1)N(CCCOCCNC(=O)C(=O)NCC(N1CCCCC1)=O)C C1(N(C(=O)CCc2cnco2)C)CCCN(C(=O)C(c2cccnc2)N(C)C)C1 Cc1nn(C)c(NC(=O)CC2COCCN2C(c2cc(CO)ccn2)=O)c1C=O CC1CN(C(=O)CCc2nccs2)CC(C)N(C(c2ccc(C3CC3)nc2)=O)C1 C(=O)(C(C)(C)CC(=O)N1CCC(CN(C)C(c2nccc(F)c2Cl)=O)C1)OC c1(C(N(C)CCN(C(=O)C(=Cc2ccccc2)C#N)C)=O)nnc(O)cc1O c1(OC)cccc(CC(N2CCCC2CN(C)C(c2cc(N)ccn2)=O)=O)c1 C(C(=O)N1CCC(C(N2CC3CC3(CO)C2)=O)(CC)C1)(C(C)C)SCC c1(C(=O)NCC(C)N(C(CNC(CCNC(C)=O)=O)=O)C)cnc(N(C)C)cn1 N1(C(C=C(C)C2CC2)=O)CCOC(CCNC(C2CCN(C)C2)=O)C1 N1(C(=O)CC2CC(Cl)(Cl)C2)CCc2ccc3ccccc3c2C1 N1(C(C(=O)NCCC2C=CCOC2)=O)CCOCC1CC1CC1 C(=O)(C(F)C(C)C(F)(F)F)N(CCCNC(c1cncc(Br)c1)=O)CC c1(CC(=O)NC2C(NC(C3(CC=C)COC3)=O)CC2)csc(N2CCCC2=O)n1 C12(C(=O)OC)CCCCC1(C(=O)N(Cc1ccco1)CC1CCCO1)CC2 CCC(C)CCCC(=O)N1CCOCC1CNC(=O)CCCC(N)=O CCCC(CC(C)C)C(=O)NC1(C)CC(C(=O)N(CC(C)C#N)C)C1 C(=O)(C1c2c[nH]nc2CCC1C)NCCC(C)NC(c1cc(Cl)ccc1Cl)=O C#Cc1cncc(C(=O)NC(C)C=CC(=O)NC(c2ccccc2)CC)c1 C1(C(c2ccc(Cl)nc2)N(CCNC(C2(CCC)CC2)=O)C)Cc2nncn2C1 C(=O)(CC(C)(C)C#N)N1C(C(C)(C)NC(C(C)Cc2ccc(F)cc2)=O)CCC1 C(=O)(NNc1cc(Cl)cc(Cl)c1)NC(C#C)Cc1ccc(Cl)cc1 c1(OC)ccc(C(N2CCC(NC(c3cc(Cl)cc(I)c3)=O)C2)=O)c([N+](=O)[O-])c1 CC(C)(O)C(F)C(=O)NCC(O)CC(=O)NCC(O)CNC(N)=O C1(CCC(C)C)CCC(C(N2CC(CNC(c3nncs3)=O)C(C)C2)=O)CC1 CC1CC(C(N2CC(CN=[N+]=[N-])C2)=O)CN1C(=O)CC1CSC1 Cc1ncc(C(=O)NCC2(F)CCN(C(=O)CN3CC(=O)NC3=O)C2)n1C c1(C(=O)NCC2(C(N(C(C=C)C)C)=O)CC23CCC3)cn(C)c(=O)n1C CC1CC(NC(=O)CCSCC2CCCCO2)CN(C(c2ccncc2F)=O)C1 OCC1(c2ccccc2)CCC(NCCCOC2CCOC2)CC1 C(C(CO)(CO)NC(=O)C=Cc1ccccc1)N(C(C1C(C(=O)OC)CC1)=O)C C1(NC(c2c(C)n(C)nc2)=O)CC1C1CCN(C(C2CCOC(C)C2)=O)CC1 c1(NC)ccc(F)cc1C(=O)NC(CNC(=O)C(C)Cc1ccnn1C)C(C)C N1(C(c2occ(C)c2C)=O)CCCC(CNC(c2cccc(C(N)=O)n2)=O)CC1 c1(C(=O)NCC2CN(C(C3(CC(C)=O)CC3)=O)CC2C)cc(F)c(F)cc1F C(CC(C(C)C)NC(C1OCC1(C)C)=O)NC(CC=CCC)=O C(=O)(C(=O)CC(C)C)NCCC(CC)(CC)NC(CCC(C)OCC)=O c1(C(=O)NCCC2(CNC(C3C(CC)C3)=O)CC2)cc2n(n1)CCCC2O CCCCC(O)C(C)C(=O)N1CC(F)(F)CC1CNC(c1cnc(CC)[nH]1)=O N1(C(C(C)OC)=O)CC2CN(C(C3(c4cc(C)no4)CCOCC3)=O)CC2(C)C1 Cc1cc(CN=c2[nH]c(NC(c3nc4ccccc4[nH]3)=O)cs2)c(F)cc1Cl C(CCCC(=O)N(CCC(c1cccs1)NC(c1scnc1C)=O)C)OCCC=C c1(CN2CCC(CNC(C(CCC)OCC)=O)C2)ccc(Cl)nc1C c1(C(=O)NCC2(CNC(C3(F)C(C)OCC3)=O)CC2)ccc2cccc(F)c2n1 CCCCC(C(=O)NCC1(F)CCN(c2cc(OC(C)CC)ncn2)CC1)C(C)C C1(C(=O)NCC2CN3CCC2C3)CCC(O)CN1C(C1CCC1(F)F)=O N1(C(c2nn(CC)c(C)c2)=O)CC(NC(C2CCOC(=O)N2)=O)CC1(C)CC Cc1nc(C)c(C(=O)NCC=CCNC(c2cc([N+](=O)[O-])c[nH]2)=O)c(C)n1 N1(C(C(C(C)C)CO)=O)CC(C)OC2(CCN(C(=O)CC3CC(C)(C)CO3)C2)C1 C1(C(=O)NCC(C(=O)NC)C)CCC2CCC1CN2C(=O)CCc1ccco1 c1(C(N2CCC(N(C(CCC(=C)Br)=O)C)C2)=O)cc(-n2ccnn2)ccc1F C1(NC(N2CCOC(C3CC3)CC2)=O)CC[Si]2(CCCC2)CC1 c1(C(N2CCCC(CCNC(C3COC(=O)O3)=O)C2)=O)ccc(Cl)nc1O N1(C(c2c(=O)ccn(C)c2)=O)CC2CCC(NC(C3CCC(=O)NC3)=O)C2C1 c1(OC)ccc2c(CCNC(=O)C(N3CCCC3c3ccc(Br)s3)=O)c[nH]c2c1 C1(C(=O)NC2(C)CC(F)(F)C2)CC(NC(=O)Cc2ccco2)C12CCC2 N1(C(C2(NC(C)=O)CCC2)=O)CCC(CCC(C)(C)NC(=O)C(O)C(C)C)CC1 C(CN=[N+]=[N-])(C(=O)NC1CCCN(C(C)=O)C1)NC(CN(CCC)C)=O c1(C(N2C(CCCC)CCC2)=O)cc(CNC(C2(F)CCOC2C)=O)ccn1 c1(CNC(C(CN(C)C)NC(COCCC=C)=O)=O)ncc[nH]c1=O C1(CCC=O)CCCN(C(=O)C(O)C2CC2)C1.N(CCF)(CC)CC CN1CC(CNC(=O)C(O)C2(O)CNC2)C(F)(F)C1 C1(C(N(CCCNC(C2C(CCC)C2)=O)C(C)C)=O)CS(=O)(=O)CC(=O)N1 CCC(O)C(C)(C)C(=O)N1CCC1CNC(c1c(-c2ccccc2)c[nH]c1C)=O N1(C(C(=O)N(C)C)=O)CCC(NC(c2ccc(C3CC3)cc2F)=O)C(F)C1 c1(OCCCCC)ccc(C(=O)NC2CC(NC(C3(C)CC3(C)C)=O)C2)cc1 C#CCCCCCC(=O)NC1CCC1CNC(=O)Cc1cnccc1OC C1(NC(C2(NC(C)=O)CCCCC2)=O)CC2CN(C(=O)Cc3cc[nH]n3)CC12 C(N=c1nc(N2C3CCC2CN(C)CC3)c2c([nH]1)CSC2)c1cccc(C)c1Cl S(=O)(=O)(CCCC(CCCCC)OCC(F)F)NCC1(C=C)CCC1 C(c1ccc(F)cc1F)=CC(=O)N(CCCNC(=O)CC1CC1(C)C)C(C)C c1(C(c2nnnn2C2COC2)NCCCCOCCO)ccc(F)cc1 c1(C(=O)NC(CC=C)CNC(=O)Cc2ncc(C)o2)cc(F)cc2cc[nH]c12 c1(C(N2C(C)(CCC)CC2)=O)c(CNC(c2cccnc2CC)=O)cnn1C c1(CC(=O)NC2CC(F)(CNC(C(=C(C)C3CC3)F)=O)C2)ccc(C)c(Cl)c1 c1(NC(C2CCC(C)N(C(=O)CCCCC(N)=O)C2)=O)ccn2nccc2c1 C1(=CC(=O)NC2(CO)CN(C(CCCC)=O)C2)CN2CCC1CC2 c1(OCC(N2CC(C)C(NC(=O)CC3CC4(CC4)CO3)C2)=O)ccc(Cl)cc1Cl N1(C(=O)NC2CCC(CC(N)=O)C2)CC2(CCC2)C12CCC2 C1(NC(COCC=C)=O)CN(C(c2cc3scnc3[nH]2)=O)C(C)(CC)C1 C(=O)(CP(C)(C)=O)NCCN(CCOC)C(c1cnc(COC)nc1)=O C=CCCCCCC(=O)N1CC(OC)CC1CCNC(C1CN(C2CCC2)C1)=O C1(C)(C(N2CC(OC)(CNC(=O)C(C)CCN(C)C)C2)=O)C(C)(C)C1(C)C CC1(C)CCCN(C(=O)NC(c2cccc(O)c2)(C)C(=O)NCCCl)C1CO c1(CCNc2ccccc2)cn2c(n1)CCCC2.CC1(C)CC12CO2 Cc1c(C(N2CCCC2C2CCCN(C(=O)C(C)CO)C2)=O)cccc1[N+](=O)[O-] CC1=NOC2(C1)CC(c1nc(-c3ccccn3)nn1C1CCOC1)C2 C1(C(N(C)C)=O)C2CCC(C2)C1NC(c1ncccc1NC1CCCC(N)C1)=O C(CS(=O)(=O)c1ccc(F)cc1)NC(C(C(=O)OCC)OC)=O C1(NC(COCC)=O)CCCC(NC(c2nn(CC(F)(F)F)cc2Cl)=O)CC1 N1(C(C2(OCC)CCOCC2)=O)CC2(CNC(C3CC(C)CO3)=O)CCC1CC2 c1(C(=O)NCC2CC(C)(C)CN2C(=O)CNC=O)cnc2ncnc(O)c2c1 C(=O)(CCCC(=O)NCCC1CCCN(C(=O)Cc2nc(C)sc2C)C1)OCC C1(C(N(CCC(C)NC(CCC(=C)C)=O)C)=O)C(C2CC2)C1(F)F c1(SCc2c(OC)c(Br)cc(Cl)c2)nc(Cl)nc2c(F)cc(C)cc12 C1(CNC(c2cc(OC)ns2)=O)CCN(C(=O)C(C)=CC(C)(C)C)C(C)C1 C(N=c1ccnc(-c2cccc(C(N)=O)c2)[nH]1)C1CN(C(C2C(=C)C2)=O)C1 C1(C)(C(C)C)CCN(C(=O)CONC(=O)CN2CCC(F)CC2)CC1 CC(CC(=O)N1C2CCC1CC(NC(c1nc(C3CC3)cs1)=O)C2)P(C)(C)=O N1(CC(=O)NCCN(C(=O)C(F)CC2CCOC2)C)CCOCC1 N1(C(c2ccc(CC3CC3)o2)C(=O)NC(CC)C)CC(c2ccccc2)C(C)(C)C1 Cc1c(CC(C(C)C(C)C)=O)cnn1C.N c1(CC)nc(C(=O)NC2CC(NC(c3cnc(OCC(F)F)cn3)=O)C2)c(C)o1 C(=O)(C(CC)CCOC)N(CC(CC)NC(c1ccc(O)c(Cl)n1)=O)C C#CC1(C(=O)NC2CC(=O)N(CC)C2)CCN(C(=O)CCN(C)CCC)CC1 C(=O)(CC(C(C)C)C(C)C)N1C(C(C)NC(c2ccnc(CO)c2)=O)CCC1 CN1CCN(C2CCC(C(N3CCCCC3COc3ccccc3)=O)C2)CC1 c1(C(=O)NCC2C(C)CN(C(=O)C(C)(C)C3CCC3)CC2)ccc(F)c(C#N)c1 C(C)(C)(CCC(=O)N1CCCC(NC(=O)C=CC(=O)NC2CC2)CC1)OC C1(NC(C23CC(c4ccc(F)cc4)(C2)C3)=O)CCCC12CCN(CC#N)C2 c1(CC)nc(C)[nH]c1C(=O)NC(C)CN(C(=O)CC1CCCO1)C c1(C(=O)NCC(C)CNC(=O)CC2COC3CC2C3)ccc(F)cc1C(F)F C1(C(N2CC(NC(c3n(CC)ccn3)=O)C(C)C2)=O)CCc2ncnc(C)c2C1 C1(CC=C)(NC(=O)CCCCCO)CCCN(C(=O)Cc2ncccc2C)C1 n1(CC2CCN(C(=O)NC3CCC(C(=O)O)C3)CC2)cnc2ccccc12 N1(C(CN2C(C)CCC2C)=O)CCN(C(=O)C=Cc2cccc(CO)c2)CC1C CC1(C)OCC2CNCC12NCCCOC1CC1(F)F C(=O)(C(C)C(C)C1CCCC1)N(CCCCN(C(C)=O)C)C.C12CC(F)(C1)C2 N1(C(C2CC(N(C)C)C2)=O)CC2CCC1CN2C(c1csnc1Br)=O N1(C(CCNC(=O)NC)=O)CCC(C)(C)C1CNC(=O)CC1C(=O)N(C)N=C1C C12CC3CCC1CN(C3)C(=O)C1(CC1)C(=O)N2.C1(CN(C)C)CCCC1(C)C c1(OC)ccc2[nH]c(=NC(C)CCSC)[nH]c(=NC3CC(O)CC(C)(C)C3)c2c1 Cn1cc(C#N)cc1C(N1CCC(CCNC(c2c(Cl)nsc2Cl)=O)C1)=O C(N=c1[nH]nc(CC(C)C)s1)C1OCCN(C(C(=Cc2cn[nH]c2)C)=O)C1 N(C1CCCc2ccc(O)cc21)C(=O)SCC=CCc1cn(C)nc1 Cc1cn(C)cc1C(=O)NC1CCC(CNC(=O)Cc2ccccc2CC#N)C1 c1(C(N2C(CNC(C=NOC)=O)CN(C)CC2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(NC(C(CC)CCOC)=O)CN(C(C2(C)CC(C)(C)C2)=O)CC2(CCC2)C1 C(=O)(C(O)CCCNC(C1(O)CC1)=O)NC1CCN(CCC)C1 CC1CC(=O)NCCN1C(c1cc(CNC(=O)CC2CCCN2C)on1)=O CC(C)CS(=O)(=O)CC(=O)NCC(C)CNC(=O)CSc1cccc(O)c1 N1(C(c2nc(C)[nH]n2)=O)CC(NC(C2CCC2(F)F)=O)C(C(F)F)C1 c1(C(=O)NCC(C2CCOC2)NC(c2cnc(C)o2)=O)c(C)nn(C)c1C(F)F C1(CN(C(=O)NCc2n(CC)ccn2)CCO)CCC(C(F)(F)F)CC1 C1(NC(C(C)N2CCC2)=O)CCCC(CNC(=O)CN2CCS(=O)CC2)C1 C(C(C)(C)CCNC(c1ccc(C(C)(C)C)o1)=O)NC(C1(CCC)CCC1)=O c1(C(C(=O)NCC)N(C2CCC(C)C2)C)ccc(OC)c(OC)c1OC.C1CCC1 CC(=O)CCCC(=O)N1CCN(C(c2ccnnc2O)=O)CC1CC(C)(C)C c1(-c2c(F)ccc(NC(c3c(OC)ccc(C)c3)=O)n2)ccc2occc2c1 N(C1COc2c1ccc(Cl)c2Cl)C(C(=O)NC(C)(C)CN1CCC(O)C1)=O C12(NC(c3c(OC)ncc(Cl)c3)=O)CCCCC1N(C(=O)CCC(F)(F)F)CC2 C1(NC(C(C2CC2)OC)=O)CCN(C(=O)CCc2ccn(C)c2)CC1O C(=O)(C(C(=O)NC1(CNC(=O)C(F)C2CCC2)CCCC1)C(C)C)OCC c1(OC)cnc(Br)cc1C(N1CC(CC(N2CCC3CC23C)=O)C1)=O N1(C(C)C)CCOC(C(=O)NCC(O)CNC(c2ccccc2C2CCC2)=O)C1 c1(C(=O)NCC(CNC(c2c(C)snn2)=O)CO)ccc2c(c1)CC(=O)NC2 N1(C(C(C(CC)O)C)=O)CC(NC(=O)CC(C)(C)C(C)(F)F)CC12CCOCC2 C1(CNC(CC(C=C)C)=O)Cc2ccccc2CN1C(c1cc(F)cnc1O)=O c1(C(N2CC(NC(CC(COC)C)=O)C(SC)C2)=O)c(C)nn2cc[nH]c(=O)c12 C(C(=O)N1CC(O)CCO1)(C1CCCO1)NC(Cc1c(C)ncs1)=O N1(C(c2c(C)csc2Cl)=O)CC(C2CCCN(C(c3ccc(Cl)[nH]3)=O)C2)C1 C1(C(=O)NCCOCCN(C(=O)C(CCSC)N(C)C)C)(CC)CCNC1=O C1(S(N)(=O)=O)(C(=O)NCC2N(C(Cc3c(C)n(C)nc3)=O)CCOC2)CCCC1 c1(C(N2C(CNC(=O)Cn3cnnc3)CCC2)=O)ccncc1Cl c1(NC(C2OCC(C)OC2)=O)ccc2ncnc(O)c2c1 Cc1cc(C(=O)NC2CC2NC(c2cccc3c2CCCC3)=O)cc2ccoc12 c1(C(=O)NC(CC)CO)cc(O)nc2c1CN(C(C1(O)CC1)=O)CC2 c1(CC(c2ccccc2)NC(C2(NC(=O)OC(C)(C)C)COC2)=O)ccc(O)nn1 c1(C(N2CCOCC(CNC(CCOCCC)=O)C2)=O)cc2ccncc2[nH]1 c1(C(=O)NC(CNC(Cc2cc(C)no2)=O)(C)CC(C)C)cc2c[nH]cnc-2n1 N1(C(C(COC)C)=O)CCC(NC(=O)C(=Cc2cnn(C)c2)C)C12CCCC2 C1(C(C)C)CCN(S(=O)(=O)NC(C2(C(F)(F)F)CCCCCC2)=O)CC1 c1(CCCCC)cc(C(=O)N(CCC(C)NC(=O)CC2(C)CCOC2)C)n[nH]1 C(=O)(CCCC(=O)NCC(C1CC1)NC(=O)CCc1ccc(Cl)s1)NCC c1(CCC(=O)N(CC(CNC(C(C)C2CCOC2)=O)(C)C)C)ccc(F)c(F)c1 c1(C(=O)NC(CC(C)NC(c2cc(CCOC)on2)=O)C)cnc2n1CCOC2 C1(CCNC(C2CC23CCCC3)=O)CCCN(C(=O)C(=C2CCCCC2)F)C1 C1(C(N2CCN(CCc3cccc(Cl)c3)CC2)=O)C2CC3C(C2=O)C13 C1(C(=O)NCC(C2(O)CCN(C(=O)C=Cc3cnc[nH]3)C2)C)(CC)CCOCC1 C1(NC(C=CCN(C)CC)=O)CCN(C(c2cc(O)nc(Cl)c2)=O)CC(C)(C)C1 C(=O)(CN=S(C)(C)=O)NCC(C)(CO)NC(C1CC1c1ccccc1F)=O C(=O)(C(CC(C)C)C(C)C)N1CC(OC)(CNC(=O)Cc2cccn2C)C1 C(=O)(CCCC(C)C)NC1CCN(C(C(C)OCc2cccc(C)c2)=O)C1 c1(C(=O)NC(CC)CNC(c2csc(Cl)c2Cl)=O)cc2c(s1)COCC2 c1(OC)ccc(OC)c(C2CC2)c1.N12CCCC1CNC2=O c1(OC(C)C(=O)N(C2CCC(NC(C3CCC3(F)F)=O)CC2)C)ccc(F)cc1 c1(C(c2nnnn2CC(F)F)N(c2ccccc2I)C)cc(C(=O)OC)cn1C CC1CC=CCC1NC(=O)C(c1ccco1)NC(=O)C=CC(F)(F)F CCCCCCC(C)C(=O)NC(Cc1ccccc1)CCOC(F)(F)F C1(C(N2CCCC(C(C)NC(Cc3cc(CC)no3)=O)C2)=O)CCC(=O)NC1=O c1(C(=O)NCC2C(NC(c3cnc(C(=O)OC)s3)=O)CCC2)ccc(C)cn1 CCC(CC(=O)NC1CN(C(C2CCC=CCCC2)=O)C2(CCC2)C1)CC(C)C c1(OC)ncc(Cl)cc1C(=O)NCC(C)CNC(C1CC(N2CCOCC2)C1)=O C1(C)(NC(CSCC=C)=O)CCCN(C(c2nc(Br)c(C)s2)=O)C1 C12(NC(c3cnc(SC)n3C)=O)CC3CCC(C1C2)N3C(C1(C)CCC(=O)C1)=O Cc1cn2cccc(C(=O)NC(C)CC(C)NC(=O)C(C)Cc3cnc[nH]3)c2n1 c1(N(C2c3nc(oc3)NC2=O)C)ccccn1.C(=O)(CC1CCO1)OC c1(C(=O)NCCNC(c2c(CC)noc2)=O)ccc2c(ccn2C)c1 c1(C(N2CC(C3(NC(C(C=C=C)C)=O)CC3)C2)=O)cn2c(Br)c(C)nc2s1 N1(C(c2scc(C(N)=O)c2)=O)CCC(CNC(=O)C(F)=CCCF)CC1 Cc1scc(C(N2CCN(C(=O)COCC3CCCO3)CC2)=O)c1C1CC1 Cc1cc(CC(=O)NC(CNC(C2CCOC2c2ccnn2C)=O)C2CC2)n[nH]1 c1(C(=O)NCC2N(C(C(C=C)O)=O)CC(F)(F)C2)c(C)cc(C#N)cc1C C1(N(C(C=CC)=O)C)CCCC(N(C)C(c2cnc(-c3cccs3)o2)=O)C1 C1(CC(C)C)(C(=O)NC(C)Cc2nc(-c3ccccc3)no2)CCCNC1 c1(C(c2n(CC(=C)C)nnn2)NCC2(CCO)CC2)cnn(C)c1C(F)(F)F C=CCC(C)(CC)C(=O)N1CC(CNC(c2csc(C)n2)=O)C(F)(F)C1 N1(C(C2(CCC=C)CN(C(=O)C(=O)CCCC)C2)=O)CCN(C)CC(C)C1 c12ccc(cc1)NC(=O)CO2.C1(C(=O)OC)(CF)COC1 c1(C(=O)NCCOC2CCN(C(C(C)SC)=O)CC2)ccnc(O)c1Br C1(C(=O)Nc2n(C)nc(Br)c2)CC(F)(F)CN1C(c1cc(F)ncc1Br)=O Cc1cccc(F)c1CC(=O)N(CC(C)N(C(=O)COc1ccccc1F)C)C CC(C)(CN(C(=O)CC1CCN(CCc2ccccc2Cl)C1)CCO)C(=O)O c1(C(C)C(=O)NC2CC(CNC(C3CCC(C)O3)=O)C2)ccc(Cl)c(Cl)c1 C(=O)(C1=CCCSC1)NC(c1ccnn1C)C(=O)Nc1c(CC)cccc1 C1(CNC(C2CCC(CC)O2)=O)CN(C)CCN1C(=O)CC12CCC(CC1)OC2 c1(C(=O)NCC2CN(C(c3ccc(C)nc3C)=O)C3C2C3)ccc([N+](=O)[O-])cn1 N1(C(C(=O)N(CC(=O)NCCC(N)=O)C)=O)CCC(NC(=O)CN(C)C)CC1 C(=O)(C1CCc2c[nH]nc21)N1CC(NC(c2c(N)sc(C)c2C)=O)CC1(C)C C(C(N=[N+]=[N-])C(=O)N1CCC(NC(c2ccc(OC(C)C)nn2)=O)C1(C)C)OC c1(-c2nn(C)c(Cc3cccc(O)n3)n2)ccc(Cl)cc1O C1(C(=O)NCC2CC(NC(C3CC(F)(CO)C3)=O)C2)CCCCCC1(F)F c1(C(=O)NC2(C)CN(C(C3CCn4nncc4C3)=O)C2)cc2cccc(Cl)c2s1 C1(c2cn(CC(CC)C)nn2)CN(C(=O)CCCOC(C)=O)CCN1C O(NC(=O)C(CCC=C)CC(C)C)C(C(=O)NCC(CCCC=C)(C)C)CC N1(C(COCCC=C)=O)Cc2n[nH]cc2C1C(=O)NCCCc1cc(C)[nH]n1 c1(C(=O)NCC2CN(C(CSC)=O)C(C)C2)ccc(C)c(O)c1 C(C(C)(C)C(=O)NC1(c2cn(CC3CCCO3)nn2)CC1)N(C)C Cn1cc(C(N2CC(F)(CNC(C3CCC(C)(C)OC3)=O)C2)=O)n(C)c1=O c1(C(N2CC(NC(C(C)C#N)=O)C(CC(C)(C)C)C2)=O)cc2cnccc2o1 c1(C(=O)NC(CNC(c2cnc(C)o2)=O)(C)C(C)C)cccn2ncc(Br)c12 c1(C(N2CCCCC2C(O)CC(F)(F)F)=O)cccc(Br)c1Cl C12(CNC(c3ccns3)=O)CC1CN(C(=O)Cn1ncc(Br)n1)C2 c1(C(=O)OC)cc(C(N2CC(O)CC2C(=O)Nc2sccc2CO)=O)cc(F)c1 Cc1ccc(C(=O)NCCNC(=O)C(c2cccc(Br)c2)(C)C)c(N)c1 C(C1CC(C)Oc2ccccc21)NC(C1(c2c(OC)cccc2)CC1)=O C1(O)(CC(N2C(C(=O)NCc3ccc[nH]3)CC2)=O)CCCOC1 C1(C(N(CCN(C)C)CC)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O C1(CC(=O)NC2CN(C(C(C)(C)OCC)=O)C2)CC(F)(F)C1(F)F C(=O)(C(C)(C)CCC#N)NCC1(CCNC(C(n2c(C)cc(C)n2)C)=O)CC1 Cc1nc(N2CCC(C(C)NC(C3(O)CC3)=O)CC2)c2scc(C)c2n1 N1(C(CC2C=NN(C)C2=O)=O)CCCC(F)(C(=O)NCC(C)(CO)CO)C1 c1(C(N(CCN(C(C(C=CCCC)O)=O)C)C)=O)csc(C)c1Br c1(CN(C(=O)C(C)(C)CCl)C)ccc(CCCCc2cc(C(C)C)[nH]c2)cc1.N C(=O)(CC1=CCCCC1)NC(C1CN(C(C2(C(=O)NC3CC3)CC=CC2)=O)C1)C C1(C)(C(=O)NC(C2(CNC(=O)C(C)N(CC(F)(F)F)C)CC2)C)C=CCC1 C(=O)(C(C#N)C(C)(C)C)N1C(C)CC1C(N1CC(c2ncccn2)C1)=O C=CCC(CNC(=O)CCC(C)(C)OC)C(=O)NCC(C)CC(C)(C)C C(=O)(C(C)(C)CCC(=O)NC1COCC1CNC(C1CN(CC(C)C)C1)=O)OC N1(C(CC2(C)CCOCC2)=O)CC2(C1)SCCC2NC(c1cscc1Cl)=O c1(C(=O)NC23CC(C(=O)NCC4CC4c4ccsc4)(C2)C3)cc2ccccc2[nH]1 CC1CC(C)N(C(=O)CSC2CC2)CCN1C(=O)C#CC1(C(F)(F)F)CC1 N1(C(C2CC(NC(C=CC3(C)COC3)=O)C(O)C2)=O)CCCCC(F)(F)C1 C1(CNC(c2c(C)n(C3CCOC3)nn2)=O)CCC(C)CN1C(=O)CC1CC1 C1(COC)(NC(c2c[nH]c(C)c2)=O)CCCN(C(=O)C(C)C2CC2)C1 C1(CN(C)C(C2COC2)=O)CCN(C(c2sc(Br)cc2F)=O)CC1 C1(CN(C(C(CC=C)c2nn[nH]n2)=O)C)CCC(C)(C)CC1 C1(NC(c2ccn(CC#N)n2)=O)COCCN(C(=O)Cc2ccc(F)cc2Cl)C1 CC1(C)CN(C(C2CCCC(F)C2)=O)CC1NC(C1C2CCC(=O)C12)=O Cc1nccnc1C(C)NC(=O)C(C1CCCN(C(=O)CC2(C)CC2)C1)C C(C(=O)N1CCN(C(c2cc3sccc3[nH]2)=O)C(CC2CC2)C1)(C(C)(C)C)SC Cc1cccc(C(C(c2ccccc2)CC#N)CNC(=O)N(C)C)c1 C1(C2CCN(C(C3CCCS3(=O)=O)=O)CC2)(NC(c2c(C)nn(C)c2)=O)CC1 c1(SCC(=O)NC2C(C(=O)Nc3cc(OC)ns3)C2)ccc2c(c1)OCCO2 N1(C(CS(CC)=O)=O)CCC(C2CC2)(CNC(c2conc2C2CCC2)=O)C1 C1(NC(Cc2c(C)nc(Cl)cc2)=O)CC2CC1CN(C(=O)CCc1ccoc1)C2 C(=O)(C(C)(CCc1ccccc1)N(C)CCOCCOCC1CC1)OCC c1(C(C(=O)NCC2CC2)N(C)CC2CCN(C)C2)csc2c(F)cccc12 c1(OC)cccc(NC2=CCCCC2)c1.C1C(=O)OCCN1C(C)=O C1(C(=O)NCC2(CC3CC3)CCC2)CC2C=CC1N(C(=O)C=Cc1ccncn1)C2 C(c1cocn1)=CC(=O)N(CC(C)NC(C1CC2(CC2)C1)=O)C CCCCC(F)C(=O)N1CC2CC1CN2C(=O)C(CN(C)C)C(C)C c1(C(=O)NC(CC(=O)NC(CC)CCO)COC)nnc(O)nc1O c1(C(N2CCN(CC(=O)Nc3ncc(Br)s3)C(=O)C2)=O)ccc(Br)c(Cl)c1F c1(OC)ccc(CC(=O)NC2CC23CC(NC(C2CCCO2)=O)C3)cc1O c1(C(N(C(CC)CC(=O)NC2CCCC2OC)C)=O)coc2c1COC2 O=C1C2CC3C(C2)C13C(=O)NC(C(=O)NCc1ccc2c(c1)CC2)C1CCCO1 Cc1cnc(OCC(=O)OC2C=CCC2)nc1 N1(C(CC2CC(CC)C2)=O)CCC(C(=O)NCC(C)CC2CC2)(CC)C1 n1(CC)nccc1C(=O)NC1(CNC(=O)CN2CCC(C)C2)CCC1 C(=O)(N=c1nco[nH]1)NC1(COC)CNCCO1 c1(OC)ccc(C2CCCN2C(c2ccccc2SCc2cccs2)=O)cc1F C1(CC(=O)NC2C3CN(C(c4c(CC)nns4)=O)C2C3)CC2(CCCC2)CO1 c1(SC)ncc(N)c(C(=O)NCC2CCCC2NC(c2cc(C)ncn2)=O)n1 C=C(Cl)CC(C(=O)NCC(CO)N(C)C)NC(C1CC1c1cccs1)=O c1(C(N(C)CC2CCCN(C(C3(C)CCCCO3)=O)C2)=O)nccc(N)c1Cl N(C(=NCCC1CC(F)C1)NC1CCC1)C(COC)C C1(C(=O)OC)CC12CN(C(=O)CC(C)CNC(=O)CNC(C)=O)C2 C(=O)(C1CCCc2cccnc21)NC(CNC(CCC(=O)NCCC)=O)C(C)C C(c1ccc(OC(F)F)c(OC)c1)=CC(=O)NC1CCN(CC(=O)NCC)CC1 C1(NC(c2cccc(N=[N+]=[N-])c2)=O)CCC2CN(C(C3C=CCC3)=O)CCC2C1 CC1C(NC(C2CC(N(C)C)C2)=O)CCCN1C(c1cc(N(C)C)ccc1N)=O C1(C(N(CC(=C)C)CCOC)=O)CCCN1NC(=O)CCC1CC1C Cc1ccc(Br)c(F)c1C(=O)NC1(CNC(C2(C#N)CCC2)=O)COC1 c1(C(=O)NCC2CC(NC(c3c(NC)snc3C)=O)C2)nccn2cc(C)nc12 C1(NC(C2(NC(=O)C=CCO)CC(O)C2)=O)CC2(CNC(=O)O2)C1 c1(OC)ccc(F)cc1CC(N1CCCC(NC(C2C3COCC23)=O)C1)=O c1(C(=O)Nc2ccc(CN3C(=O)CSC3=O)cc2)ccc2nccc(Cl)c2c1 N1(C(C(n2ccc(C)n2)C)=O)CC(NC(C2CC2c2oncc2C)=O)C2(CC2)C1 O=C1NCC2(CCCN(C(=O)C3=CCNC3)C2)O1 c1(N2C(CNC(C3(CO)CC3)=O)CC3(CC3)C2)cc(C(F)(F)F)nc2ncnn12 C(=O)(CCCCC(N)=O)NC(C)CN(C)C(c1cc(-c2ccco2)c[nH]1)=O c1(C(=O)NC(CC(=O)NC2CC23CCCCC3)C2CC2)c(F)cncc1F C12(NC(C3(C(F)(F)F)CC3)=O)CC(CNC(c3ccc[nH]3)=O)(C1)OC2C.CCC CC1(C(=O)NC2CN(C(=O)CN3CC(=O)NC3=O)CCC2F)CCC(F)(F)CC1 c1(OC)ccc(NC(C2CC(NC(c3cccc(C)c3)=O)C2(C)C)=O)cc1C c1(C(=O)NCCC(C)N(C(C(C=C)c2ccccc2)=O)C)ccccc1C(C)C N1(C(C(C(C)C)NC(CCOC(C)=O)=O)=O)CC2CC1CN2C(C)C C(=O)(C(C)(C)CC(=O)N1CCCC(NC(=O)CNC(=O)C2CC2)C1)OC CC1OCCCC1C(=O)NCCCN(C(=O)CCOC1CCCC1)C C12(NC(c3n(CC)c(O)nc3)=O)CCC(C1)N(C(=O)COC1CCC1)C2 CC(CC(C)(F)F)C(=O)NC1CCC1NC(=O)CCc1c(F)cccc1Cl c1(CN(C2CCCN(C(=O)Nc3cn(C)nc3CCC(=O)O)C2)C)ccc(F)cc1 c1(C(=O)NC2CC(C)(NC(C(CCCC)C)=O)C2)ccc(OC)c(F)c1N c1(C(=O)NC(CNC(C2C(C)CCC2)=O)(C)C)cc2ncccc2cc1Cl CC(C)CC(CNC(C1(CCF)CCC1)=O)NC(C1CC1(C)C)=O.C1(C)CC1 C(=O)(CCCCCCn1cc(C2CC2)nn1)NCCOC1CCCC(C)C1 NS(=O)(=O)c1ccc(C(=O)NCC(CO)NC(=O)Cn2cnnn2)o1 N1(C(C=CCC)=O)CCCC(O)(CNC(=O)C(c2c(Cl)cccc2Cl)C)CC1 C(=O)(C1CCCNc2ccccc21)NCC1N(C(c2cc(C)sn2)=O)CCC1 c1(C(=O)NOCCO)n[nH]cc1CNC1(C2CCCCO2)CC1 c1(CCC(=O)NCC2(NC(C34CC(C)(C3)C4)=O)CCOCC2)ccc(F)cc1Cl N1(C(CCC=C)=O)CC(CC(=O)NC2(CN3CCCC3)CC2)C2(CC2)C1 c1(C(=O)NC2CCC(NC(C(C)OCC)=O)CC2)c(C)[nH]c2ccc(Cl)cc12 Cc1cc(C(N2CC=C(C(=O)Nc3cnn(C)c3)C2)=O)nnc1C N1(C(c2n(CC#C)ccc2)=O)C(C)CN(C(=O)C=C(Cl)Cl)CC1C N1(C(C2C(C)(C)CO2)=O)CC(CO)C2(C1)CN(C(c1cncc(Cl)c1Cl)=O)C2 c1(CC(C)(C)C)ccc(C(=O)NCCC(O)CNC(=O)C(CO)N(C)C)cc1 c1(CCCC)nc(C(=O)NCC2CCN2C(c2ccsn2)=O)cs1 C(=O)(C1=C2CCCN=C2NN1)N1CCN(C(Cn2ncn(C)c2=O)=O)CC(O)C1 N12CCOC3CC(CCC13)C2=O.C1(NC(C)=O)CCOC(C)(c2ccccc2)C1 c1(C(=O)NC(C(=O)NC(CCC)C(=O)NC)CN(C)C)cc(C)n(C)c1C C=CC1(O)CCN(C(C2CCCN(C(c3cncc(OC)n3)=O)C2C)=O)C1 C1(CCC)CN(C(c2c(Cl)c(CC)nn2C)=O)CCN1C(=O)CCOC C1(OCCCNC(C2C(C)C2C)=O)CCN(C(C2(N(C)C)CCC2)=O)CC1 c1(C(=O)NCCCOCCNC(C(C(CC)CC)C)=O)n[nH]c2nccc(Cl)c12 C=CCC(C)C(=O)NCC1(OC)CN(C(c2ccc(CN3CCCC3)cc2)=O)C1 c1(OC)cncc(CNC(C2CC(C)N2C(c2cccc(CO)c2)=O)=O)c1 C12(CNC(CSCCC#N)=O)CCCC(CN(C(c3ccc([N+](=O)[O-])s3)=O)C1)C2 C1(NC(C(COC)O)=O)CCCCC1CNC(C1CCCC1)=O c1(OC)ccc(C(c2cn(CC(O)CCC3CCCOC3)nn2)OC)cc1 N1(C(c2c(CC)[nH]cc2)=O)CCCC1(C)CNC(C1(C)CNC(=O)C1)=O c1(C(=O)NC(CNC(C(C2CC2)OC)=O)(C)CO)cc(C)ccc1Br c1(OCC)ccc2c(c1)C(C(=O)NCCNC(=O)Cc1nc(=N)[nH][nH]1)CC2 C(=O)(CC1=CCCCC1)NC(CC(C)C)CN(C)C.C12(CC1)C(=O)NCC2 C1(NC(CNC(COCCOCC)=O)=O)CN(C)CCC1O C1(NC(C2CC(CCC)C2)=O)CN(C(=O)COC2CC2)CC1C1CC1 c1(OC)ccc(F)c(C(=O)NC2CC2NC(=O)C(O)C(C)(C)C)c1F Cc1cc(C(=O)NC(CC2CC2)CC(=O)NCCCCN2CCC2)c(C)o1 CC1(NC(=O)C(=O)NCC(F)(F)F)CN(C(C2CCC2(F)F)=O)C1 N1(C(C(N2CCNC2=O)C)=O)CCC(CF)(NC(c2cncc(CO)c2)=O)C1 Cc1cc(C(=O)NC(C(=O)NC(C)CN(C)C(C)C)C2CC2)nn1C C(=O)(CC(C)(C)CC(C)=O)N1CC2(CN(C(C3CCC(CC)O3)=O)C2)C1 c1(C(=O)NC2CCCC(CN(C(c3c(C)nns3)=O)C)C2)cc2n(n1)CCC2 c1(SC(C)C(N2CCC(NC(=O)CC3CCCCCO3)CC2)=O)ccc(Cl)cc1 C1(C(=O)NCC(CNC(COCCOCC)=O)OC)CCOCC1(C)C c1(NC(CC2CCN(Cc3ccc(OC)cc3)C2)=O)c(C)nn(C(F)(F)F)c1C CC1(C)CCc2c(C(N3CCCC(CNC(=O)Cc4cscn4)C3)=O)n[nH]c2C1 C=CCC(C)(C)CC(=O)N1CCC(=CCNC(c2nnc(C(C)(C)C)s2)=O)CC1 c1(C(=O)NC2CC(F)(CNC(C(F)OC)=O)C2)nnn(-c2ccn(C)n2)c1C C12(CCCC1)C(=O)N2.C(=O)(C(=O)N1CC(C(N)=O)C1)N(C)C N1(C(CC(C)C)=O)CCOCCC1C(=O)NCC(C)(O)C1CCC1 C(=O)(C1=CC2CCC=CCCC12)N1CC(Nc2nccc(SC)n2)C(C)C1 N1(C(CCc2ccc(OC)cc2C)=O)CC(NC(=O)C(N)=O)Cc2ccccc21 c1(C(N2CCN(C(c3c(C(C)C)onc3)=O)CC2)=O)cc2c(F)ccc(Cl)c2[nH]1 Cc1ccc(F)c(C(=O)NC23CCCC(NC(=O)C(C)CS(C)=O)(C2)C3)c1 C(=O)(C1=CS(=O)(=O)CCC1)NC1CC(NC(c2c(C)nc(CC)s2)=O)C12CCC2 N1(C(C)C)CCC2(CC1)CC2(C)C(N1CCN(C2CCOCC2)CC1)=O c1(C(=O)Nc2scc(-c3c(F)ncc(OC)c3)n2)nn(C)cc1[N+](=O)[O-] c1(CN2CC(=O)N(CCCN(CCOCC)C)C2=O)c(F)ccc(Br)c1Cl c1(C(=O)NCc2cn(CC(=O)NCC3CNC(=O)C3)nn2)ccncc1F C1(=O)C(F)CC2CN1C2.N1(CC)CCC1CNC(C1(n2cnnn2)CC1)=O Cc1[nH]c(=NCc2cccc(O)n2)sc1C(=O)Nc1cccc(Br)n1 Cc1nsc(C(N2CCC2CNC(C2COCC2(C)C)=O)=O)c1N N1(C(COCCSC)=O)CCC(F)CC1C(N1CCSCC1C)=O C1(CC)CCCN(C(c2cnc(C)nc2C)=O)C1C(=O)NCCC[Si](C)(C)C C1(CC)CC(CC(=O)NC2C=CCN(C(=O)CC#N)C2)CCO1 CCCC(CCCO)C(=O)NCC1CCCC1NC(c1cc(OC)ncn1)=O c1(NC(C(CC)(C)O)=O)ccc(NC(=O)CCC(=O)N2CCOCC2)c(F)c1 N1(C(CC=CC=C)=O)CC2CCC2(NC(c2ccnc(CC)c2)=O)C1 C1(C(N2CC(OC(=N)O)C2)=O)(NC(C(C2CCC(=O)N2)C)=O)CC1(C)C N1(C(C=C2CCC(C)CC2)=O)CC2CCC1C(CNC(C1CCC(O)CC1)=O)C2 c1(C(=O)NCC2N(C(C(C)OC)=O)CC(F)(F)C2)c(C)sc2ccccc12 Fc1ccc(C(c2nnnn2C2CC(F)(F)C2)NCCc2ncccn2)cc1Cl C(c1ccc2occc2c1)=CC(=O)NCC(CNC(C=C(C)C1CC1)=O)(C)O Cc1cccc(C(=O)NCC(CC2CC2)C(=O)NC(Cc2cnc[nH]2)CO)c1N c1(OC)cc(C(=O)NC2CCC(NCc3c(F)cccc3Cl)C2)c(OC)cc1Cl c1(C(N2CCCC(O)(CNC(CCOC(C)C)=O)C2)=O)cn(C)c2ccccc12 c1(C(C(=O)NC(CC)C)N(C)Cc2c(I)cnn2C)c(C)nn(C)c1Cl C1(CC)CN(C(c2cnc(O)cc2C)=O)CCC1NC(=O)CCc1ccco1 C(=O)(CCCN=[N+]=[N-])N(CC(O)Cc1ccccc1F)C(C)(C)C Cc1cc(C#N)nc(N2CC(CNC(=O)Cn3ncnn3)CC2C)n1 CC(Cc1cnc[nH]1)C(=O)NCC(C1CCOC1)NC(c1ccn(C)n1)=O C(=O)(C(CC(C)C)CC(C)C)NCC(CC)NC(C1Cc2cc(F)ccc2O1)=O c1(C(=O)OC)ccc(N2CCN(CCCOC3CCOC3)CC2)nc1C Cc1[nH]c(=N)sc1CC(N1CC=CC(NC(c2ccc(C(N)=O)[nH]2)=O)C1)=O CC1CC(C(N2CC(c3ccccc3)(NC(C3CC4CCC3C4)=O)C2)=O)CCO1 Cc1ccsc1CC(=O)NC(CN(C)C(C1CC1F)=O)Cc1ccccc1 c1(C(CC)NC(C2CCN2Cc2noc(C)n2)=O)cccc(C(F)(F)F)c1 C1(C2CCCCC2)(C(=O)NC(CCNC(C(C(C)C)OC)=O)C(C)C)CC1 N(S(N)(=O)=O)CC(=O)N(CC(C)NC(c1cnc[nH]1)=O)C N1(C(C(C=C)(C)O)=O)CCC2(CCC2)C(NC(c2oc(CC(C)C)nc2C)=O)C1 c1(C(=O)OC)c(C(N2CC(n3cc(CNC(=O)CNC=O)nn3)C2)=O)n[nH]c1C C1(NC(c2c(C)cc[nH]2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC1C C1(CCC(=O)N(CC(CC)NC(c2c(CC)nns2)=O)CC)CCC(=O)NC1 c1(OC)ccnc(OC)c1C(=O)N(C1CC2CC1N(C(=O)C(C#N)C(C)C)C2)C CCC(C#N)(CC)C(=O)N1CC(NC(=O)C(C)Cc2ccnn2C)C(O)C1 CCC(CNC(c1c(Br)c(C)nn1C)c1nnnn1C1CCOC1)(CC)C(N)=O c1(C(=O)NCC(C)(CO)NC(C2CCC(=O)N2)=O)cccc2c(O)nncc12 c1(CCC(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2O)nc2ccccc2[nH]1 c1(C(N(CCC(c2cccs2)NC(C(C2CC2)SC)=O)C)=O)csc(=NC)[nH]1 C(=O)(C(F)n1ccnc1)NCC(=O)NCC(c1ncc[nH]1)O N#Cc1ccc(CC(N2CC3CC3(CNC(=O)CC3NC(=O)NC3=O)C2)=O)cc1 C1(C(c2n(CC)nnn2)NCC2CC(CC(C)(C)C)C2)C(C)(C)C1(C)C c1(C(N2CCC(C(N(C(CC(=O)NC)C)C)=O)C2)=O)cccc(C)c1C N1(CCNC(N(CC(CC)O)C)=O)CCOC(C)C1 CCC(C)C(CC(=O)NC1CCCC(O)CC1)NC(c1ccnc(OC)c1)=O c1(C(=O)NCCCNC(C2CCC(C(N)=O)O2)=O)ccc([N+](=O)[O-])s1 c1(NC(C2(CNC(c3cnc(Cl)nc3)=O)CC2)=O)cnn2ccc(Cl)nc12 N1(C(C(CC2CC2)NC(C(n2c(C)ccn2)C)=O)=O)CC2(C1)NC(=O)NC2=O Cn1nc(C(=O)NC2COCCC2NC(=O)Cn2cnnc2)cc1C(F)(F)F C=CCCC(C)(C)C(=O)NCc1cccc(NC(C2CCN(C)S2(=O)=O)=O)c1 C1(COC)CN(C(c2ccc(Br)cc2)=O)CCN1C(=O)COCC(C)C C1(n2cc(-c3c(C)nsc3)nn2)CC2(CC2)CN1C(C1CC(C)(C)C12CC2)=O Cc1nc(C2CCCC2)sc1C(=O)NCC1CC(NC(C2CN(C(N)=O)C2)=O)C1 CCCCCCC(CNC(c1ncoc1C(F)(F)F)c1nnnn1CCC1CC1)CC c1(C(N(CC(=O)N(CC(F)F)CCOC)C2CC2)=O)nc(C)sc1C N1(C(CCCC(=C)C)=O)CCC2(CC1)CC2NC(=O)CCN(C)CCO c1(C(=O)NC2CC(C)(NC(CCC(C)(C)C#N)=O)C2)cc2ccncc2cc1F c1(C(N(CC(CNC(C(COC)(C)C)=O)C)C)=O)cc(OC)ccc1F c1(C(N2CCCN(C(C(C)NC(=O)NC)=O)CC2)=O)ccc2nn[nH]c2c1 c1(CC=C(C)C)cc(C(=O)NC2CCN(C(C3(C)CC3C)=O)CC2O)ccc1F C1(C)(NC(C(CCC)O)=O)CCN(c2nc(OC)cc(OC)n2)CC1 CC(C)C(CNC(=O)CC1CCC(=O)N1)N=c1[nH]c2cc(F)ccc2o1 C1(C(=O)NCC2CC[Si](C)(C)C2)CC(C)(C)S(=O)(=O)C(C)(C)C1 N1(C(C2C(C)(Br)C2)=O)CCC(c2cn(Cc3cc(C4CC4)no3)nn2)C1 C(C(CC(F)(F)F)NC(c1c[nH]cc1Br)=O)NC(CCCN(C(C)C)C)=O O=C1CN(C(=O)NC2CC2C(=O)Nc2ccc(C(F)(F)F)cc2)c2ccccc2N1 c1(C(N(CC(CN(C(C(CCC)C)=O)C)O)C)=O)cccc(C#N)n1 c1(C(N(CC(N2C(CC)C(O)CC2)=O)C2CC2)=O)c[n+]([O-])c(C)cn1 c1(-c2c(CN(CCN(C)C)C)cc(Cl)cn2)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NC(C(=O)NC(c2n(C)ncc2)CO)C2(C)CC2)cc(Cl)cn1C c1(C(N2C(C(=O)Nc3cnn(CC)c3)CC(=C)C2)=O)cnc(Cl)cc1OC C1(C(=O)NCCN(C)C(C2CC(=O)N(C3CCCC3)C2)=O)CCC2(CCC2)CO1 C1(=O)C(C(C)O)N1.N1(CCC)CCC(C(=O)N(C2CCCN2C(C)C)C)C1 Cc1cn2c(n1)C(C)CC(C(=O)NCC1CN(C(c3cnn[nH]3)=O)CCN1C)C2 c1(C(C(=O)NCCN2CCC(O)CC2)Nc2ccco2)ccc(F)c(Cl)c1 C(=O)(CCC(=O)NN(C)C)N1C(C)CN(C(c2cnc(SC)n2C)=O)C(C)C1 Cc1nc(C)c(C(=O)NC(c2nc(C(F)(F)F)n[nH]2)C)c(C)n1 c1(C(=O)NCC(C2CCCC2)NC(c2c(CC)occ2)=O)ccn2ccnc2c1 C1(N(C)C(c2ccc(C3CCC3)nc2)=O)CCCC(NC(=O)Cc2cscn2)C1 N1(C(COCCNC(c2c(C)nc(C)s2)=O)=O)CCN(C)C2(CC2)C1 C12(NC(=O)COc3cccnc3)COCCC1CN(C(=O)CN1CCCC1)C2 Cc1c(C(=O)NCCC(O)CNC(=O)CC2CCCOC2)sc2[nH]cnc(=O)c12 N1(C(C2CCCOC2)=O)CCN(C(=O)CCc2cnco2)C(CC2CC2)C1 C12(C(=O)NC3CC(C)N(C(=O)COCc4ccncc4)C3)CCCC(C1)OC2 CC(CC(=O)NC1CCN(CCNC(=O)C(c2cncnc2)C)CC1)C(C)(C)C C(C(CO)(CO)NC(=O)C(F)CC1CCCC1)N(C(=O)CNC(C1CCC1)=O)C c1(CCC)cnnc(C(N2CC(CC(C)(C)CNC(C3CC(CC)C3)=O)C2)=O)c1 c1(C(N(C(C)C)CCNC(=O)C(c2ccccc2)F)=O)cncc(C(F)F)c1 O=C(C#CC1CCCC1)N1C(C(=O)Nn2cnnc2)CCC1CF C(CCCC(=O)N(CCCCC(=O)NCCN(C)C)C)OC CC(C)(C)C(=O)NC1CC1C(=O)NCC1COC(=O)N1 c1(C(N2CCC(N(C(=O)C(F)C(C)C)CC)CC2)=O)cncc(Cl)c1C C(C(=O)N1CCC(C)C1CNC(c1cc(C(N)=O)c[nH]1)=O)(C(C)C)NC(=O)OC Cc1noc(C(=O)NC(CNC(=O)CCC2CC2(F)F)C2CC2)c1C C1(NC(=O)OC(C)(C)C)CCN(Cc2cccc(CO)c2)CC1CC#N C(C1=NOC2CN(C(c3nocc3C(C)(C)C)=O)CC12)NC(COCCC=C)=O C(=O)(C(C)(C#N)CC)N1CCC(C(C(=O)N(CCN(CC)CC)C)C)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(C(=O)NCc2cn[nH]c2)C(C)(C)C1 c1(C(N(CC(CNC(CC(C)c2ccncc2)=O)O)C)=O)ccc(=O)n(C)n1 C(=O)(CCCC(C)=O)NCC1(C(=O)NC(C)COC(F)(F)F)CC(=C)C1 N1(C(C(c2cccc(C(F)(F)F)c2)(C)O)=O)CCCNC(=O)C1 C(C(=O)NC1CCN(c2cc(C)ncn2)C1C)(C(C)C)NC(C)=O c1(SCCCCN(C(=O)CCN2CCOC2=O)CCOC)c(C)noc1C c1(C(=O)NCC(C)(C2CC2)NC(C(C)n2cccn2)=O)ccc(C#N)[nH]1 C1(NC(C2C(C)(CC)C2)=O)CC2(CCN(C(=O)CC3=CCCC3)CC2)C1 C1(COCC)(CNC(CNC(=O)CSCC2CCCO2)=O)CCCCC1 N1(C(C(C)NC(=O)NC)=O)CC2CCC(C1)C(NC(=O)CC1CCC(=O)C1C)C2 N1(C(CC2N(C(CCC(CC)OC)=O)CCOC2)=O)CCCNC(=O)C1C N1(C(C(C(C)C)C2CCC2)=O)CCC(C)N(C(C2SC3C=CC2C3)=O)CC1 Cc1cc(C(C(=O)NCC(C)C)N(CCC(=O)N(C)C)C)c2ncccc2c1 N1(C(c2c(C)cco2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2(CC2)C1 N1(C(C2C(C)C2C)=O)CC2CCN(C(c3cc(Cl)c(Br)cn3)=O)CC2C1 c1(CNC(C(C2CCCCC2)C)=O)cc(C(=O)N(C2CC(C)(C)C2)CCO)cs1 CC(C)CC(C(=O)NCC1(F)CCC(NC(c2ncoc2C2CC2)=O)C1)C(C)C C1(OC)(CO)CCN(C(C2(N(C)C(C3CC(C)CCO3)=O)CCC2)=O)C1 N1(C(CC(C)OC)=O)CCC2(CC1)C(NC(=O)CC1(CO)CC1)CS(=O)(=O)N2C N1(C(COCCNC(c2c(CC)cncc2)=O)=O)CCCC2(CC1)CC2 c1(C(=O)NCC(CCCC)NC(=O)CCC(C)(C)C)cnc(N)c([N+](=O)[O-])c1 CCC(CC(=O)NC1CC2CC(NC(c3ccoc3Cl)=O)C2C1)CC(C)C C1(C(C)C)CCCN(C(=O)C(N2CCCCC2C(O)N(C)C)=O)CC1 C(S(=O)(=O)CCCC(=O)NCCc1ccco1)c1ccc(C)o1 C1(C(N(CC=C)Cc2cccc(-n3cncn3)c2)=O)Oc2ccccc2OC1C N1(C(C2N(C)CCCC2)=O)CC2(CCC2NC(=O)CN2CCCCC2=O)C1 C1(CNC(C2CN(C(C)C)C2)=O)CCOC1C(N1CC(N2CC=CC2)C1)=O C(N=c1cccc(S(=O)(=O)N2CCOCC(C)C2)[nH]1)c1c(OC)ccnc1 N1(C(C(CC)n2cccn2)=O)CCOCC(NC(C2CC(C)(F)C2)=O)C1 c1(OCC)n[nH]cc1C(=O)NC1(CCNC(=O)Cc2cnnn2C)CCC1 C(CC(=O)N1CC=CC(NC(C2(OC)CCC2)=O)C1)(C(C)C)OCC c1(C(N2C(C(=O)NC(c3ccc(F)cc3F)CO)CC2)=O)c(Cl)cc(Br)cc1Cl C1(CC(C)NC(c2cncc(F)n2)=O)CCN(C(=O)Cc2cc[nH]n2)CC1 C(=O)(C1=CCN(C(=O)CC2CC2(C)C)CC1)NC(CCOC)C N1(C(C2CCCCO2)=O)CCCN(C(C2CC3CC3C2)=O)CC1 C1(OC)CCN(C(c2cncc(F)c2Br)=O)C(C2CC2)C1 C(=O)(CCCC1OCCO1)NCCC1(NC(C(C)SC(C)C)=O)CCC1 c1(C(=O)NC2CCCN(C(CCCOCCC)=O)C2)ccc(O)c(CO)c1 c1(C(N2CCCC(NC(C3C(C)CC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1Br c1(C(=O)NCCN(C(c2ccc(OC(C)C)o2)=O)CC)ccc2n[nH]cc2c1 N1(C(C23OCC(C)(C2)C3)=O)CCCC(F)(CNC(c2cscc2F)=O)C1 c1(C(N2CCN(C(C(c3scc(C)n3)C)=O)C(C)C2)=O)ccc(N)c(Cl)c1O C(=O)(CCCC(C)(F)F)N1C(CCCNC(c2c(NC)ccc(Cl)c2)=O)CCC1 C(CCCCC(=O)NC(C1CC=CCC1)C(=O)NC1C(O)C2CCOC12)OC C(=O)(C1CCCc2cncn21)N1CC2CCC(NC(Cc3c(C)non3)=O)C2C1 S(=O)(=O)(c1ccc(Br)cn1)N1CC(NC(C2(C(=O)OCC)CC2)=O)C(C#N)C1 Cc1ccc(S(=O)(=O)NC(=O)CCc2ccccc2N)cc1C C1(C#CC(=O)NC2(C)CCN(C(=O)COC(F)F)C2)(CC)CC1 C=CCC(C(=O)N1CCCCC(N(C)C(c2nnn3c2CSCC3)=O)C1)C(C)C C1(C(C)C)CN(C(C2CCC(N(C)C)CC2)=O)CCN1C(=O)C(=O)N(C)C C1(NC(COC2CCC(C)CC2)=O)CC2(CCCN(C(c3cc(Cl)no3)=O)C2)C1 C(=O)(C(CNC(C1CC(F)(CF)C1)=O)C(C)(C)C)NCCc1n(C)cnc1 c1(C(=O)NC(C(C(=O)OC)(C)C)c2ccccc2)ccc2nccc(=O)n2c1 N1(C(CC(C(C)C)(F)F)=O)CC2CCCN(C(c3cn4c(n3)COCC4)=O)C2C1 CC1CCC(NC(c2ccc(C(F)F)o2)=O)CN1C(c1ncc(Cl)nc1Cl)=O c1(C(C)C)c(C(=O)OC(C)(C)C)cnn1-c1ccccc1.C1CNC(=O)O1 Cc1c(CC(N2CCC(CC(=O)N(C3CC4(CC4)C3)C)C2)=O)ncn1C c1(C(=O)NCC2(O)CC(C(=O)NCC(C)C(C)(C)C)C2)ccn2cncc2c1 CCCCCCC(CC)NC(=O)CC1CCN1C(C1(C)CC2CCC1C2)=O CCC(CC(=O)N1CC2CC2(CNC(=O)CC(=O)NCC(F)(F)F)C1)C1CCC1 C1(CNC(c2c(C)ccc(C)c2)=O)CN(C(C2COCCOC2)=O)CCC1(F)F c1(C(=O)NCC2(NC(c3cc(CO)cc(F)c3)=O)CCC2)cc2cccn2cn1 Cc1cc(C(=O)NCCC(C)N(C(=O)C(n2ccc(C3CC3)n2)C)C)ccc1Cl C1(C(=O)NCC(CC)NC(=O)C(C)CC(C)(C)C)Cc2ccccc2N1C(C)=O n1(CC)ncc(Cl)c1C(=O)N(C)CC1COCCN1C(C1CC(F)C(=O)N1)=O C(C)(N(C)N1CCOC(CCO)C1)c1ccc(OC)nc1 CN1CCOCC1C(=O)NCC1(C)N(C(=O)C(C)(C)N2CCCCC2)CCC1 C1(NC(Cc2ccc(C)s2)=O)CC2CCC(C1)N2C(=O)COC1CCOCC1 C1(CNC(C=CC)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1C C1(CCN(C)C(C23CCCC2C3)=O)CCCCN1C(=O)COc1ccn(C)n1 Cc1ccc(C(N2CC(NC(=O)Cc3sc(O)nc3O)C(C)C2)=O)c(O)c1 N1(C(C2C(C=C)C2)=O)CCN(C(c2cccc(SC)n2)=O)C(C(C)C)C1 Cc1ccnc2ccc(C(N3CCCC(NC(=O)CCOCC4CC4)C3)=O)cc12 C(C(C)(F)C(C)(C)F)(c1n(CCSC)nnn1)NC(N1CCCCCC1OC)=O N1(C(C)C(=O)N(C2CCCOC2)C)CCN(C(c2ccoc2Cl)=O)CC1 c1(C(N2CCC(CCNC(c3c(C)cc(SC)o3)=O)C2)=O)ncc(C)cc1C C(=O)(CC(C(F)(F)F)NC(C1(CO)CCC1)=O)N(C)Cc1ncccn1 CC1CCC(CNC(=O)Cc2cccs2)N(C(=O)C(=O)Nc2ncc[nH]2)C1 C1(C(N2CCCC(CCCCNC(c3cc(C)sc3)=O)C2)=O)CC12CCOCC2 c1(OC)cc(C(=O)OCc2ccc(O)c(Cl)c2)nc(C(C)C)n1 CCCC(CCC)C(=O)NCC1(CNC(C2CCN(C3CCSC3)CC2)=O)CC1 C(=O)(C(CC(C)C)N(C)C)N(CCCOCCNC(CC)=O)C c1(C(N(CCC(C)NC(=O)Cc2cnns2)C)=O)ccc([N+](=O)[O-])cc1F Nc1cc2c(cc1C(N1CCC3C(NC(=O)C4=COCCC4)C3CC1)=O)CCC2 C1(C2CCCC2)(C(=O)NC(C(C)(C)O)C(=O)O)CCNC1=O N1(C(c2oc(CC)c(C)c2)=O)CC(NC(=O)C(COC)OC)CC12CCC2 CCCCCC(=O)N1CCC(CCOC)(NC(=O)CCCn2ccccc2=O)C1 c1(OC)c(NC(CNC(=O)CC2CC(C)(C)C2)C2CC2)ccc(Br)c1F c1(C(c2nnnn2Cc2ccccc2)NC(COCC)(C)C)c(C)cncc1C O(NC(=O)C(O)CCCNC(c1cccc2c[nH]nc12)=O)CCC(=C)C c1(C(CC)C(=O)NCC(C)(C2CC2)NC(C2CSCCS2)=O)cccc(Cl)c1 C#CCCC(C(=O)NCC1CC2CCC(C1)C2)NC(c1nocc1Cl)=O N1(C(C(CCCCC)F)=O)C2CCCC1CN(C(=O)CC(C)F)C2 c1(CNC(=NCCC)NCC2(SC)CCOCC2)ccc2ccccc2n1 C(C(C)(C)CC(=O)NC1(CCCCO)CC1)NC(C1N(CC)CCOC1)=O c1(C(N2CCC(N(C(C3CCC(=O)O3)=O)CC)CC2)=O)cnn(C)c(=O)c1 c12ccccc1OCC(=O)NCC(OC)CNC2=O.c1(CC)ccc(Cl)cc1 c1(OC)nc(N)cc(C)n1.N1CCCC(F)(CNC(C2C3C4CCC(C4)C23)=O)C1 Cn1ccc2cc(C(=O)NCC3CCCN3C(C3(C)CC3(C)C)=O)cnc12 C#CCC(C)(CC)C(=O)NC1CCCC1NC(=O)COc1cnn(C)c1 C1(C)(C(=O)NC(C)(C)C)CC12CCN(C(=O)Cc1ccccc1O)CC2 C(=O)(CC(C)(C)C(=O)OC)N(CC(N1CC(C)(C)CC1CO)=O)CC#C c1(C(N2C(CNC(c3c(CCC)nco3)=O)C(C)CC2)=O)cccc2c1CCC2 c1(NC(c2sc3n[nH]c(C)c3c2)=O)ccc([N+](=O)[O-])c(OC(C)C)c1 C(=O)(CC1CC(=O)Nc2ccccc21)NCCN(C(=O)Cc1ccn(C)n1)CC Cc1cc(C(=O)NC2CC(NC(C3(CO)CCOC3)=O)C2)c(F)cc1Cl Cc1ccc(CC(=O)NC2CCCC2NC(C2(C)COC(=O)OC2)=O)cc1Cl N1(C(CC(C)CN(C)C)=O)CC(C)(CNC(=O)CNC(N2CCCC2)=O)CC1(C)C CCC(C)C(O)CC(=O)NCCCCN(C)C(C1(C2(O)CCC2)CC1)=O C(=O)(CC(C)(C(F)(F)F)N(C)C)N(C(CCCC)COC)C.C(=O)(C)NCCSCC CC1CCN(Cc2nc(C(C)(C)C)cs2)CC1NC(=O)CSCCOc1ccccc1 c1(C(N2C3C(NC(C(CC)CC)=O)CC(C3)C2)=O)cc2ccccc2s1 C(=O)(C(C)(O)C(C)C)N(CCOC)CCNC(=O)C(c1cccc(C)c1F)O c1(CNC(C2CCN(C)C2)=O)ccc(CNC(=O)CC2CC3CC3C2)cc1F N12CCOCC(C1)C2=O.c1(NC)n[nH]cc1C(N1CCCC1CN(C)C)=O N1(C(CC(C)(O)c2ccccc2)=O)CCC(NC(=O)C=CI)C(CO)CC1 c1(C(N2CC(OC)C(NC(c3ccc(C(F)(F)F)o3)=O)C2)=O)ccc(N)c(F)n1 C(=O)(CCCn1cc(COc2ccccc2)nn1)N(CC(=O)OCC)CCOC C1(NC(C(C2CCCCC2)NC(C(C2CCOC2)OC)=O)=O)(CO)CCOCC1 CCCC(CNC(=O)C(C1CCOC1)OC)NC(c1c[nH]nc1C(C)(C)C)=O C(=O)(C1=NOC(C)C1C)N1CCC(CCOC)(C(=O)NC2(CF)CC2)C1 N1(C(c2cc(C)sn2)=O)CCCC2(C1)CN(C(c1ccnc(C)c1C)=O)CCO2 c1(OC)cc(NC(=O)CC2CCN(Cc3ccc(Cl)nn3)CC2)c(C)cc1[N+](=O)[O-] C1(C(N2CCC3C2CCCN3C(c2ccccc2)=O)=O)CCc2nccn2CC1 c1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CCC2)cccc(OC)c1O N1(C(C=C(C)C)=O)CCC(F)(C(=O)NC2(C(N)=O)CCOC2)CC1 c1(C(N2CCCC(NC(C3CC(=C)C3)=O)C2C)=O)cccc(SC)c1[N+](=O)[O-] CC(C)(C)CC(C)(C)C(=O)N1CCN(CCCNC(=O)C2=CCCCO2)CC1 Cc1ccc(-c2cc(NCC3(O)CCN(C(=O)OC(C)(C)C)C3)n(C)n2)cc1C C(=O)(C(CC(F)F)NC(C1CC(C)(C)CN1C)=O)NCc1cc(C)on1 C1(CC(=O)NC2(CNC(CC3CC(CC)C3)=O)CCC2)CCC2(CC2)CO1 C=CCCCCCCC(=O)NCc1n[nH]c2cc(Br)ccc12.C12CC(C1)NC2=O N1(C(CCC)=O)CCCN(C(c2nnc(S)n2C)=O)CC1C(C)C C1(C(N(C)Cc2ccc(Cl)s2)=O)C2CCC1(c1ccc(Br)cc1)C2 O=C(CC1CCc2ccccc21)NC1CCN(C(=O)Cn2cc(Cl)cn2)CC1F C1(CC(=O)NCCOCCNC(=O)CC23CCCC2C3(F)F)CN2CCN1CC2 n1(CCCOCC)cc(CC(=O)OC)nn1.n12nnnc1C1(COC1)NCC2 c1(C(N(C2CCN(C(c3cnc[nH]3)=O)C2)CCC)=O)cnc(NC)cn1 C1(CC)CCCN(C(C2CC2CCC=CCNC(=O)CC2CCCN2C)=O)C1 c1(C(N2C3CCC(NC(C(C#N)C4CC4)=O)(C3)C2)=O)cc2ccnc(Cl)c2[nH]1 N1(CCNC(C2CC(C)(C)OCC2)=O)CCN(C(C2CCC2(F)F)=O)CC12CCC2 O=C1CC2CC(C(N3CC(O)(c4ccccc4)C3)=O)C1O2 Cc1cc(C(=O)NC(c2ccccc2)CNC(C2CC3(CCC3)C2)=O)oc1C N1(C(c2cn(CC)nc2)=O)CC(CNC(=O)C(N2CCSCC2)C)C(F)(CO)C1 C1(C(=O)NCc2scc(CNC(C(C)n3cncn3)=O)n2)CC2CCC1O2 c1(CN(C2CCCC(n3ccnc3)C2)CC)ccc(C#N)cc1F C1(NC(c2c(OCC)oc(C)n2)=O)CN(C(=O)C(C)(O)CC)CC1S(C)(=O)=O C1(C)(C(N2CCC(N(C(Cn3c(CCC)ncc3)=O)CC)C2)=O)CC(C)(C)C1 c1(NC(C=CCN(C(C(C=CC)O)=O)C)=O)cnn2c1OCCC2 C1(NC(CCC)CC)CCOCC1C(=O)OC(=O)CC1(CS(C)(=O)=O)CC1 c1(SC)cnc(OC(C)C)nc1.C1(C)(C)CN(C)CC(=O)N1 c1(C(N2CC(CC(C)NC(=O)CC3CCCCC3)C2)=O)ncoc1-c1ccon1 c1(OC(C)CNCC(c2ccccc2)C)ccccc1C(F)(F)F c1(COC)cc(=NCC2CCC(NC(=O)CCCC3CCC3)C2)[nH]cn1 CCCC(C)(C)CC(=O)NCC(CNC(C1C2CCCOC12)=O)C(F)(F)F CCC(CC)C(C(=O)N1CCCOC(CCNC(C2(C)CC=CC2)=O)C1)OC C1(NC(CCc2n(C)ncn2)=O)CC2CCC1N2C(=O)COCC1CCCOC1 CN1CC(C)(C)CC1C(=O)NC1CCCCN(C(C2(C)CCC2)=O)C1 c1(C(N2CCC(C)C2CNC(C2CCC(O)C2)=O)=O)cccc(C#N)c1 C(=O)(C(C(=O)N1CCC(C(C)NC(=O)CCCOC(C)=O)C1)C(C)(C)C)OCC N1(C(COCCC)=O)CC2CCC1C1CN(C(c3csc(C)n3)=O)CC21 c1(OC)ccc(C=CC(=O)NC=CC=C)nc1.C1CC(NC(=O)C=CC2CC2)C1(C)C CCCC(C)C(=O)Nc1ccccc1Br.N12CCSCC1NC2=O CN1CC(NC(=O)C(C2(C)CC2)NC(c2ccc(=N)[nH]n2)=O)C(=O)N1 c1(C(=O)NCCCCNC(C(CCSC)O)=O)cc2ccccc2nc1C(F)F C1(OCCNC(C2C(=C)C2)=O)(CNC(=O)COC2CC2)CCOCC1 C1(OCC)CCCCC(c2nnnn2C(C)COCc2sccc2C(=O)OC)C1 CC1CCN(C(=O)CC2CCC(=O)NC2)C(CNC(=O)CCc2cnco2)C1 c1(NC)ccccc1C(=O)NCCC1CC(C(=O)Nc2ccsc2C(C)C)C1 N1(C(CSCC#C)=O)CCC(NC(=O)CN2CCc3sccc3C2)CC(O)C1 CC(CCCCCO)NC(=O)C(C1CCCO1)NC(=O)CCc1ccccc1 c1(CCC)nc(C)c(C(N2CC(N(C)C(c3ccn(C(C)C)n3)=O)C(F)C2)=O)s1 Cn1cccc(C(=O)NCC2CCCCN2c2nnc(-c3ccccc3)o2)c1=O CC1C2C(CCN2C(c2csnc2Cl)=O)CN1C(=O)C(F)CC1CCOC1 C1(C(N2CC(C3(NC(C4CSC4)=O)CC3)C2)=O)CCOC2(CCCC2)C1 CC1CN(C)CCN1C(=O)C(C(C)(C)O)NC(=O)COCCCN(C)C c1(OC)ccc2ncnc(N3CCCC4C3CCN4c3ncncc3F)c2c1 Cn1cnc2c1CCC(C(N1CC(NC(C3CCCC(=O)N3)=O)C(O)C1)=O)C2 Cc1cc(=NCCCOCCO)[nH]cc1S(=O)(=O)NC1CCCOc2ccccc21 C1(Nc2nc(C(CC)OC)cc(C)n2)CC12CCc1ccccc12 c1(CC(=O)NCC2(O)CCN(Cc3n(C)cnc3)C2)ccccc1[N+](=O)[O-] c1(C2N(C(=O)Nc3c(C4(OC)CCC4)cccc3)CCC2)cc(F)cc(F)c1 c1(C(C(=O)NCC=C)NC(C)(C)C)ccc(C)c(Br)c1C.c1(OCC)ccc(F)cc1 c1(-n2c(C(C)OCC)nc(-c3ccc(Cl)s3)n2)ccc2nccnc2c1 S(=O)(=O)(c1ccc(COC)cc1)C(CSCCC(=O)N(CCC)CCC)=O C(=O)(C1=C(Cl)CCOC1)NC(C1CCCN1C(c1cc(C(N)=O)c[nH]1)=O)(C)C c1(C(=O)NC2C(C)CCN(c3ncnc(CC)c3F)C2)ccc2ccnn2c1 Cc1c(C(N2CC(CNC(c3ccc(N(C)C)nn3)=O)CC2C)=O)n[nH]c1C1CC1 Cc1ccc(CC(N2CCN(CC(=O)NCc3cc(C4CC4)n[nH]3)CC2)=O)cn1 C12(C(N(CC(C)(C)NC(C3(C(=O)NC)CC3)=O)C)=O)CCCCC1CCC2 C(CCC(C(=O)NN1CC(C)(CNC(=O)C2CC2)C1)NC(=O)C1CC1)OC Cc1cc(=O)n(C)cc1C(=O)NCC(O)CNC(c1cn(CCO)nn1)=O c1(CCNC(C(C)SCCCC)=O)ocnc1CNC(C1CCC(CC)O1)=O C1(NC(COC(C)(C)C)=O)C2COCC1CC(NC(C1(CO)CC1)=O)C2 N1(CC(=O)NCCCC)CCC2(CCN(C(c3cccc4ncccc34)=O)C2)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(CO)C1 CC1CCC(CNC(C2CCSCC2)=O)N(C(c2ccc(C(F)F)c(F)c2)=O)C1 c1(C(=O)NC2CC(C(C)NC(Cc3cc(C)[nH]n3)=O)C2)ccccc1Br c1(C(C(=O)NC(C)CC)N(CC(C)C)CCC)cc2c(cc1OC)CCC2 C(CN=c1[nH]nc(C(F)F)o1)(CC(C)C)CN(C1CCN(CC)CC1)CC C1(N(C(c2c(C)snn2)=O)C)CN(C(c2cc(-c3ccccc3)no2)=O)CC1O c1(OC)nc(Cl)ccc1C(=O)NCCC1(O)CN(C(=O)C(O)Cc2cnc[nH]2)C1 c1(C(N2CCCC(NC(=O)CC3CS(=O)(=O)C3)CC2)=O)cc2c(O)cccc2[nH]1 c1(Nc2cnn(CCOC)c2C)nc(=NC2CCC3(CC3)C2)[nH]c2c(C)nn(C)c12 c1(C(N(C)CC2CN(C(CC=CCC)=O)CC23CC3)=O)nn(CC)cc1[N+](=O)[O-] N1(C(C(CC)C2CC2)=O)CCC2C(CCCN2c2cc(SC)nc(SC)n2)C1 c1(NC(C2CC(NC(c3c(CC)n(C)nc3)=O)C(O)C2)=O)cc(C)c(C)c(C)c1 N1(C(C=CC2(C)COC2)=O)CCCC(CNC(=O)CC2CCC23CCC3)CC1 CC(O)(CNC(=O)CCCC1CCCC1)CNC(C1CCCCC1)=O Cc1nnc2n1C(C(=O)NC1CC1CNC(c1cccc3c1CCCC3)=O)CC2 C1(COC)(NC(C2CCOC2)=O)CCCN(C(=O)C=Cc2cnccc2C)C1 C1(NC(=O)CC2(N3CCCC3)CC2)CC2(NC(C3C4COCC34)=O)COC1C2 C#CC(CNC(=O)CCCCCN(C(=O)Cc1ccccn1)C)CC(C)(C)C CC1(C)CC2(CC(C(N3CCC(CCNc4nccnc4F)C3)=O)C2)C1 C1(C2=CCCCCC2)(C(=O)NCC2(O)CCN(C(C(CCC)(C)C)=O)CC2)CC1 c1(C(=O)NCC2C(NC(CC(C)CF)=O)CCCC2)cc(F)c(Cl)cc1Cl C1(C(CNC(c2cncs2)=O)F)CCN(C(=O)C(c2ccc(F)cc2)F)CC1 C(CC)(C(=O)NC1(CNC(c2cc(C(C)=O)on2)=O)CC(OC)C1)OCC.C1CC1 C1(NC(c2c(C)noc2)=O)CC(F)CN(C(c2ccc(OC(C)C)cc2)=O)C1 N1(C(c2c(CC)c(C)sc2)=O)CC2C3CCC(C2C1)N(C(=O)C(F)(F)C1CC1)C3 n1(CC(N2CCC(C)(NC(C(C)C(C)(C)C)=O)CC2)=O)cc2ccccc2n1 N1(c2ccc(S(=O)(=O)NCC(C)F)cc2Cl)CCc2ccc(C#N)cc2C1 c1(CC(N2C(CNC(C3(C)CCC(=O)NC3)=O)C=CC2)=O)c[nH]c2cnccc12 N1(C(Cn2ccc(C)n2)=O)CCC(C)(C)C1C(=O)NCCC1(CN(C)C)CC1 Cc1nc(C)c(CC(N2CCCC(C)(NC(C3CCCC(F)C3)=O)C2)=O)c(O)n1 c1(C(N2CC(n3cc(C4CCN(C)CC4)nn3)C2)=O)cc2c(Br)cccc2s1 C1(C(=O)OC)C=CCCN1C(C1CCN(C(c2cscc2OC)=O)C1)=O c1(C(N(CCCNC(c2nc(Cl)oc2C)=O)CC)=O)ccc(F)c(C#N)c1 C(=O)(C1CCSc2ccccc21)NC1CCC(NC(CCC(C)(C)O)=O)CC1 c1(C(=O)NC2CC(F)(CNC(C(C)NC(CC)=O)=O)C2)ccc(Br)c(N)c1 C1(C(=O)NC(C2CCOCC2)C)CC(NC(=O)C(F)(F)C(F)F)C12CCC2 Cc1nccc(C(=O)NC2CC2CNC(=O)CCCSc2ccccc2)n1 N1(C(CC2CN(C(C(CCC)C#N)=O)C(C)(C)C2)=O)CCCC(C2(C)CC2)C1 c1(C(=O)NCC(C=C)(C)C)coc2c1CN(C(=O)CCN(C)CCC)C2 n1(CC)c(C)cc2c1CCCC2NCCCc1c(C)oc2cc(C)ccc12 C1(CC(=O)NC2CCN(c3nc(C)cc(OC)n3)C2)Cc2ccccc2C1 c1(C(N2CCCC(N(C)C(C3CC(=O)CCO3)=O)C2)=O)[nH]cc2c1CCCC2 c1(C(N2CCOCC(NC(C=CC(C)C)=O)C2)=O)nnc(O)c2ccccc12 C(=O)(C1CCc2c[nH]nc21)NCCCCNC(c1cncc(OC)c1)=O c1(CC=C)cccc(C(=O)N(CCC(=O)NCC2C3COCC23)CC)c1 C12(CNC(C3CCN3C(=O)COC3CC=CC3)=O)CCC(CC1F)C2 CCC(C)CCCCC(=O)NC1CN(C(c2cccc3c2OCCO3)=O)CC1O C1(CC=C)(NC(C(C=C)(C)O)=O)CCN(C(C2CN(C(C)=O)C2)=O)CC1 N1(C(c2c(C)nn(C)c2)=O)CCOC2(CCC(NC(=O)Cn3cnnc3)CC2)C1 C(=O)(CCCC(F)(F)C(F)(F)F)NC1COCCN(C(C(C(C)C)C#N)=O)C1 c1(C(=O)NC2CCN(C(C(C)C(C)O)=O)C2C)coc2c1CCCC2 C1(CC(N2C(C)CC(CCNC(C(CSC)C)=O)C2)=O)CCCCC1(F)F C#CCN(OC)C(=O)C(O)CC1CCCN1C(=O)CC(C)(C)C C12(CCNC(C(F)=C(C)C)=O)CCC1CN(C(C1(c3cccs3)CC1)=O)C2 c12cnc(cn1)C(=O)NC(C1CC1)CNC2=O.c1(C(=O)OC)cc(C(F)F)cs1 C1(CNC(CC(C)(C)N(C)C)=O)CN(C(=O)C(F)(F)C2(O)CCC2)CC12CCC2 CC(CNC(=O)CC1CCC1)C1CC1.C1(C2(C(=O)NCC(F)(F)F)CC2)CCCO1 c1(NC(c2cscn2)C)[nH]c(=NC2CCCC(O)C2)nc2c1cnn2C C1(C)(CC)CCC(c2nnnn2CCCSC)(NCc2ncn(C)n2)CC1 c1(C(=O)NC(CC(C)NC(c2ccc3sncc3c2)=O)C)cc(S(N)(=O)=O)co1 C#CCCC(C(=O)N1CCC(F)(CO)C1)NC(c1cccc(C)c1O)=O c1(OC)cnc(NC(c2ccsc2COC)=O)nc1SC(C)C C(=O)(C(C)(C)C#N)NC1C(NC(C(C)CSCc2ccccc2)=O)C1 C(CCCN=c1[nH]c2cc(Cl)cc(Cl)c2o1)NC(C1CCCC(NC(C)=O)C1)=O C1(CNC(C=NOC)=O)CC(C)(C)CN1C(=O)CS(N)(=O)=O O=C(N=c1cccn[nH]1)C1CC(O)CN(C(c2ccnc(-c3cccs3)c2)=O)C1 C1(CNC(C(CC#C)(C)C)=O)COCC2(CCN(C(=O)CC(C)(C)SC)CC2)O1 CCC1=NOC(CC(=O)NCCN(CC(C)O)C(=O)C=C(C)c2ccco2)C1 C1(C(=O)NC(CCC)CNC(c2cc(C)sc2C)=O)CCc2nc(C)[nH]c2C1 C1(c2nnnn2C2COC2)(NC(CC=C)CC)CSCCSC1 C1(C(=O)OC)(C(=O)NCC=CCC(=O)NCC2CC2)CC1C.c1(C2CCC2)ncc[nH]1 C1(C)(CNCc2n(C)ccn2)CNCCO1 C1(CCNC(c2cnc(C(C)O)s2)=O)CCCCN1C(C1CCC=CCC1)=O CC(C)(F)C(C)(F)C(=O)NC1CC(NC(c2cnc3ccnn3c2)=O)C1 N(C1CCCc2c1cnn2-c1ccccc1)C(=O)NCc1c(C)scc1 CC1COCCCN1C(=O)C(CC(F)F)NC(=O)Cc1ccon1 C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])c1c(CNC(c2c(C)noc2)=O)cccc1 C=CCC(CNC(=O)Cc1nc[nH]n1)NC(=O)CC1CCSCC1 N1(C(C2(COC)CC=CC2)=O)CC(NC(C2CCC(F)CC2)=O)C(C)(C)C1 c1(C(N2C(C)CN(C(C3(C)CC3Br)=O)CC2)=O)ccc2ncsc2c1 c1(C(N(CCN(C(=O)COc2ccc(Cl)nc2)C)C)=O)cccc2nc(O)[nH]c12 N1(C(c2cn(C(C)C)nn2)=O)CCOCC(NC(C2(CCF)CCC2)=O)C1 S(=O)(=O)(c1csc(C(=O)NC(C(C)NC(C23CCC(CC2)C3)=O)C(C)C)c1)NC N1(C(C2C(C)CCC2)=O)CCCC(C)(C)C1CNC(C1CCCSS1)=O C1(NC(C(=O)NCC)=O)COC2C(NC(C3CNC(=O)N3)=O)COC12 c1(C(=O)OCc2ncccc2Oc2ccc(F)cc2)cc2cccnc2cn1 c1(C(=O)NC(C)CN(C(=O)CCc2nccs2)C)sccc1S(N)(=O)=O N1(C(C=NOC)=O)CC2CCCC(CNC(c3cc(O)nc(O)n3)=O)(C2)C1 c12c(cccc1C)NC(=O)NC2.C(CCO)N(CCC)CCOC N1(C(C(COCC)C)=O)CC(OC)CC1C(=O)NCc1c(C)cnn1C C1(C(F)(F)F)(C(N2CCC(N(CCC)C(C3COC(C)C3)=O)C2)=O)CCOCC1 c1(C(N2CC=CC(C(N3CC(OC)C(O)C3)=O)C2)=O)cc(O)ccc1C c1(CC(CC)C)nc(-c2nnn(CC)c2C)n(C2CCOC(C)C2)n1 c1(OC)cc(CC(=O)N(C)CCN(C(=O)C(C)(C)CF)C)cc(F)c1 c1(C(=O)NC(C(=O)N(C)CC2(O)CN(C(CC(C)C)=O)C2)C)ccc(F)cc1F S(=O)(=O)(c1ccc(NC(=O)NNC(=O)c2ccccc2N(C)C)cc1)NC C(=O)(CCC(=O)N1CCC(C)C1CNC(=O)CCCc1sccc1C)NC c1(SC)cc(C(=O)NC2CC(CNC(c3[nH]cnc3C#N)=O)C2(C)C)c(C)o1 C1(C(=O)NC(c2ccco2)C)CC(O)CN1C(C1C=CCC1)=O Cc1nnc(C(N2CC(c3ocnc3Cn3cc(C4CC45CC5)nn3)C2)=O)s1 N1(C(=O)OC(C)(C)C)CC2CC1CN2C1CCCC1.c12ccccc1CS2 c1(CC)cc(C)c(C(=O)NCCCN(C)C(C2C3CC(=O)CC23)=O)o1 c1(C(N2C(C)CC(CNC(C(CC#C)CC#C)=O)C2)=O)cnc2cnccc2c1 c1(C(=O)NCCC2CN(C(CCCC(N)=O)=O)C2)cccc2[nH]ccc12 C1(C)(C(=O)NCC2C(C)CN(c3ncnc(=N)[nH]3)CC2)CCCNS1(=O)=O N1(C(C2CC2C2CCC2)=O)CCC(NC(C2(Sc3ccccc3)CCC2)=O)CC1 c1(C(=O)NC(C(C(C)C)C)CNC(C2(CO)CCCC2)=O)ccc(C#N)cc1F c1(NC(C2(C(N(C3(C#C)CC3)C)=O)CC2)=O)nn(C)cc1C C=CC(C)CC(=O)NC(CCNC(=O)C(CCC)N(C)C(C)=O)C(C)C NS(=O)(=O)C1(C(=O)NCC2(F)CCC(NC(C3CCNC3=O)=O)C2)CCCC1 N1(C(CC)=O)CC2CN(C(c3cc(C4CC45CC5)ccc3Cl)=O)CC2C1 C(=O)(C1=C(Cl)CCOC1)N1CC(CCNC(c2ccc(F)s2)=O)OCC1 C(=O)(C1=CN=C2N=CNN2C1)N1C2CN(C(C3=CC(C)(C)C3)=O)C(C2)C1 C1(NC(C(C(CC)C)OC)=O)CC2CN(C(=O)C(=Cc3ccccn3)C)CC2C1 C(=O)(C(CCCN)NC(c1ccc(NC(=O)C2CC2)nc1)=O)OC Cn1c(C(N2CC3CC2C3CNC(C2C=CC=CC=C2)=O)=O)cccc1=O c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)C(C)C)ccc(O)nc1Cl C=CC(CCC)CC(=O)NC(C(=O)NCC1([Si](C)(C)C)CC1)C1CCCC1 C1(C(N2CCC(CNC(c3cc(F)n[nH]3)=O)C2)=O)CC2CCC(C1)S2 c1(C(N2C(C(C)NC(CC)=O)CCC2)=O)cnc2ccncc2c1 CCCC(O)C(=O)N1CCC(CN(C(=O)CCc2c(C)noc2C)CC)CC1 N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC2CC2(C)C)C(O)C1 C(CCC(C)C(=O)NC1CC(NC(c2ncoc2C)=O)C1)OC C1(C(N2C(C=C)CCC2)=O)C2CCC(C2)N1C(=O)C=C(C)COC N1(CC(=O)N(CCC(=O)NCC2(O)CSC2)C2CC2)C(=O)CNC1=O CN1CCCC(CNCC2NCC23CCCC3)C1c1ccccc1 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)CC2CCCO2)cn(C)nc1C C1(NC(c2c(C)nc[nH]2)=O)CCC(NC(=O)CCNc2ccccn2)CC1 N#Cc1cc(C(N2CCCC2CC(=O)N(CCO)CCO)=O)ccc1O C(CC1=CCN(C(=O)CN2CCC2)CC1)NC(=O)CC(c1ccccc1)C1CC1 c1(OCC(=O)NC(CN(C(C(C)OCC#C)=O)CC)C)cccc(Br)c1 c1(C(=O)NC(c2cncnc2)C)coc(CNC(=O)CCCSC2CC2)n1 c1(C(N2CC3CC(NC(c4cnsc4)=O)C3C2)=O)cncc2c(O)nccc12 S(=O)(=O)(c1ccc(Cl)nc1)N1C(CC)CN(C(C2CN(C)C2)=O)CC1 C1(C(=O)NCCC(C)NC(C2CCN(CCC)CC2)=O)CCc2n[nH]cc2C1C c1(C(C(=O)NCC(C)N(C(=O)CC2CCC(O)C2)C)(C)C)cc(Cl)ccc1F N1(C(C(CC=C)C)=O)CCC2C(NC(=O)Cc3ccsn3)C2C1 C1(COC)(NC(=O)CC=Cc2ccc(C)cc2)CCCN(C(C2CCSC2)=O)C1 C1(C(N(CC(CC)NC(=O)CC2(O)CCCC2)C)=O)C(c2ccccc2)C1(F)F N1(C(c2ccn(CCCF)c2)C(=O)Nc2ccccc2)Cc2ccc(Br)cc2C1 c1(OC)ccc(C(N2CC(CC(C)NC(=O)CCc3cnc(C)o3)C2)=O)c(F)c1 n1(CC(=O)NCCN(C(=O)C(C)CC(F)F)CC)c(C)cc(C)nc1=O CC1CCC(F)(C(=O)NCC2CCN(C(c3ncoc3C3CC3)=O)C23CC3)CC1 N1(C(C)C(=O)N(C)CCN(C(=O)C(C)Oc2cccnc2)C)CCCCC1=O N1(C(C(C)(C(C)C)OC)=O)CCN(C(c2csc(C(C)(C)C)n2)=O)CC(O)C1 N1(C(C2(O)CCC(C)CC2)=O)CC(C)N(C(C23CC(F)(C2)C3)=O)C(C)C1 n1(CCNC(C(CCOCCO)NC(COC)=O)=O)ccc([N+](=O)[O-])n1 C(=O)(C(F)CC(C)(C)NC(=O)CC1CSCCO1)N1C(CC(=O)OC)CC1 Nc1ncc(Br)nc1C(=O)NCC1CCC(NC(=O)CCOCC2CC2)C1 C(=O)(C1=CCCN(C(C2CCCSC2C)=O)C1)N1CCC(C=C)(O)C1 N1(C(c2cnn(CC)n2)C(=O)NCCCF)CCc2oc(C)nc2C1 c1(C(N(C(C)C(C)(C)C)C)=O)cc(CNC(=O)CC(C)C2CCCO2)nn1C C1(C)(N(C)CC)CCN(C(c2coc(CN(C(=O)C(C)(C)CF)C3CC3)n2)=O)C1 C1(OC)CC2CCCCN2C1=O.c12cc(C#N)ccc1[nH]c(=O)[nH]2 c1(OC)nn(C)cc1C(=O)CNC(c1cnn(C)c1F)=O C1(C(=O)Nc2cccc(OCC(=O)OC)c2)C2CCC1N(C(=O)CCN(C)C)C2 N1(C(CN(C(COC)=O)C)=O)CCC(C)N(C(C2CNC(=O)C(C)(C)C2)=O)CC1 N1(C(C(C)NC(C)=O)=O)C2CN(C(C3CCC(=O)N3c3ccccc3)=O)CC12 c1(C(=O)NCC(=C2CN(C(c3cnc[nH]3)=O)C2)F)cnn2ncccc12 C1(NC(CC2CN(C)C2)=O)CC2CCCC(C1)N2C(c1csnn1)=O C1(NC(C(c2ccn(CCF)n2)C)=O)C2CC(NC(C3(C)C=CCC3)=O)CC12 CC(C)CC(C(=O)NCC(O)CCNC(c1ccc(C#N)o1)=O)C(N)=O c1(C(C(F)F)NC(c2ncc(Cc3cccc(Cl)c3)s2)=O)ccccc1Br c1(OC)cc(C)c(C(=O)N(C)CC2CCN(C(c3cnoc3C)=O)C2)cn1 C1(CCC)CN(C(=O)CC2OCCO2)CC1C(N1CC2(CC2)C1)=O C1(CC(=O)NCC2CCCC2NC(c2cncn2C2CC2)=O)CC(=O)NC1=O C(=O)(CC(C(C)C)C(C)C)N1CC(OC)C(NC(=O)CCC2CCN(C)CC2)C1 c1(C(=O)NC2CCCC(NC(=O)COC(F)F)C2)ccc(C(C)(C)C)cn1 Cc1cn(C(C)C)cc1C(=O)NCCCC1(NC(=O)Cc2ccc(F)cn2)CC1 C1(C2CCN(C(C3CSCCS3)=O)C2)(NC(=O)C(CC(F)F)C2CCC2)CC1 c1(C(=O)NCC2CN(C(C)=O)C(C)C2)coc2c(C)cccc12 C1(C(=O)Nc2cc(OC)nc(C(=O)O)c2)CC12CCN(C(=O)CCN(C)C)CC2 CS(=O)(=O)c1ccc(CC(=O)NCC2(F)CCN(C(=O)Cn3cncn3)CC2)cc1 O=C(CCCCCO)NCC1(NC(=O)CC2(N3CCOCC3)CCOCC2)CC1 N1(C(C2(CF)CCN(C(C(C(C)C)O)=O)C2)=O)CC2(COC(C)(C)C2)C1 c1(C(N(CC(C)NC(C2CCC2C(F)F)=O)C)=O)c(C(F)(F)F)ncn1O N1(C(=O)NC(c2ccc(C#N)cc2)CC(C)C)CCN(C2CCOC2)C(=O)C1 CC1=CC(C)CN(C(C2C(C)CN2C(C2CCN(C)C2)=O)=O)C1 Cc1cccnc1CNC(=O)CC1CCC(NC(=O)C=CC2CCOC2)C1 C=CC1(CC(N2CCOC(CNC(=O)CCOCCOC)C2)=O)CCCCC1 N1(CC(=O)N(C(C#C)C)C)CCN(C(c2cnccc2OC)=O)CC1 C1(NC(CSc2cccc(C)c2)=O)CS(=O)(=O)CC1NC(c1cc(C#N)on1)=O c1(OC)ccc(C)c(C(N2CC3CC(NC(=O)C=CC(C)(C)C)C2C3)=O)c1N N1(C(c2ccc(CC)cc2N)=O)CCN(C(c2cn(CCO)nn2)=O)C(C)C1C N1(C(=O)CC2CCCS(=O)(=O)C2)CCC2CCC(NC(C3(Br)CC3)=O)C1C2 C1(CC(=O)NC2CCC(CNC(CN(c3ccccc3)C)=O)C2)COC2CC1C2 Cc1ccccc1C(C)CC(=O)N1CC(N(C)C(c2cc(O)n(C)n2)=O)C1 c1ccc(NC2(CCCC3CCCCO3)CCC2)cc1 c1(C(N(CCNC(C2CC(=C3CC3)C2)=O)CC)=O)ccc(C2CCCO2)[nH]1 c1(COC(C)(C)CNC(=O)NC(C)CCCc2ccccc2)cccc(F)c1O C1(NC2C(C)(CC)CC2OC(c2cnn3c2CCC3)=O)CC(S(C)(=O)=O)C1 C=CC1(CC(=O)NCc2cccnc2F)CN(C(=O)C=C2CCOCC2)C1 c1(NCCC(=O)NC(CC)C)nc(N2CC(O)CC(F)C2)cc(C)n1 C1(C(=O)NCC(CNC(COCCC)=O)F)CCSCC1 N1(C(C23CN(C(C4CCO4)=O)C(C2)CCO3)=O)CC2C3CCC(O3)C2C1 C(=O)(C#CC1CCCCO1)NCC(CNC(C1N(C(C)=O)CCC1)=O)C c1(SCC(=O)NCCC(C)(C)NC(CC=CC)=O)nc2ccc(C)cc2[nH]1 CC1CCN(C(=O)Cc2c(C)noc2Cl)C(C)C1NC(=O)C1=COCC1 N1(C(CN(C(C(C)C)=O)C)=O)CC2(CC2)CC1CNC(C1CC12CCSCC2)=O c1(OC)cccc(C2CCN(C(=O)NCCc3cn(C4CCCCC4)nn3)C2)c1 CCC(CN(C)C)CC(=O)NCC(C)(C)NC(=O)C=Cc1cncs1 c1(C(=O)NC(CC=C)CNC(=O)C=C2CCC(C)CC2)cncc2ccccc12 CN1C(=O)NCC1C(N1CC2C(NC(C3CC(CF)C3)=O)C2C1)=O C(N=c1[nH]cnc(NCC23CCC(CC2)CC3)c1C)c1scc(CC)n1 N1(C(c2c(CC)nc[nH]2)=O)CCC(C)C1CNC(=O)C(=O)NCCOC CC(C(C)C(=O)NCCN(C1CCCC1)Cc1cc(F)ccc1F)S(C)(=O)=O c1(CN(C)C)cc(C(=O)NCC2(CN(C(=O)CCC3CCCOC3)C)CC2)no1 C1(N(C(C2CCCC2)=O)CC)CCCN(C(=O)CC2CCS(=O)(=O)C2)CC1 CCCC(C#N)C(=O)NCCCCc1cn(-c2ccc(C)c(Br)c2)nn1 c1(C(N(CCNC(C(F)(F)C2(OC)CCC2)=O)C2CC2)=O)cnc2cccnn12 C1(NC(c2cncc(C)n2)=O)CC2CN(C(C3CN(C)CC(C)O3)=O)CC12 c1(C(N2C(CNC(C3N(C(C)(C)C)CC3)=O)CC2)=O)cc2c(s1)CCCCCC2 C1(C(=O)NCCCCCCNC(C2CC2F)=O)CS(=O)(=O)c2ccccc2O1 c1(OC)cccc(C2CCN(Cc3cc(Cl)ccc3N(C)C)C2)c1F c1(CNC(=NCC)NC2CC(OC(C)(C)C)C2)nnc(O)c2ccccc12 CN1CCc2[nH]nc(C(=O)NC3CC(NC(=O)C(CC(F)F)C4CCC4)C3)c2C1 c1(C(N2CCC3(CCC3)C2)=O)csc2c1CCN(Cc1cccc(F)c1Br)C2 C1(SCC(=O)N(C2CN(C(c3cc(Cl)ccn3)=O)C2)C)CCS(=O)(=O)C1 c1(-c2cncc(C3CCN(C(CCOCC)=O)CC3)c2)ccc2sc(C)nc2c1 C(C(C)(C)C(=O)N1CCOC(C(=O)NCCSC(F)F)C1)OC(C)C Cc1nc(C(N2CC(O)(C(F)C(=O)Nc3ccccc3F)C2)=O)sc1C N1(C(COCC(=O)NC)=O)CCCC2C(CCCN2C(c2ccc(F)cn2)=O)C1 N1(C(C2N(Cc3c(OCC)ccs3)CC(C)C2)=O)Cc2ccccc2C1 N1(C(c2nc(CC)sc2)=O)CCCC(C2(NC(C3(OC)CC3)=O)CC2)C1 N1(C(C2CC(OCC)C2)=O)CCC(NC(=O)CCN(CC(C)C(C)C)C)C(O)C1 O(NC(=O)C(F)C(C)(F)F)C(C(=O)NCC(NOC)=O)CC(C)C c1(C(CC)C)nc(NC(=O)CCOC)cc(C)n1 CCC(CC)(CC)C(=O)Nc1ccc(CC(C)NC(=O)NN2CCCC2=O)cc1 C1(C(N(CCS(C)(=O)=O)C)=O)CC2CC2N1C(C1(C#N)CCCC1)=O C(N=c1cc(C(F)(F)F)nc[nH]1)C1(NC(C2CCC(C)C2)=O)C(C)CCCC1 Cc1cccc(C(N2CCOC(C(=O)NC(c3ccc(Br)cc3)CO)C2)=O)c1O C1(CCNC(C2C(C)CC(C)O2)=O)CCCN(C(c2nnn(C)c2N)=O)CC1 C(=O)(CCCCC(C)(C)OC)NC(CC)CNC(=O)C(COC)NC(C)=O C1(C(=O)NCC(C)C(=O)O)CCCN(C(C)Cc2ccco2)C1 c1(CC)cc(C(=O)NC2(CNC(c3ccc(-n4cncn4)cn3)=O)CC2)sc1C O=C(CC(F)(F)C(F)(F)F)NC1CCC12CN(C(c1cccc3[nH]ncc13)=O)C2 C1(C)(C(N2CCC(C)(NC(CCCCCOC)=O)C2)=O)CCCC(F)(F)C1 C(=O)(CC(C(=O)OC)OC)NCC1c2ccc(cc2)OC1.C(C)(C)(C)OCC=C N1(C(C(CSC)O)=O)CCC(C(O)CNC(C2CC(F)(F)CS2)=O)CC1 Cc1ccc2sc(NC(CNC(=O)C(=O)N=S(C)(C)=O)C(C)C(C)C)nc2c1C Cc1nn(Cc2ccccc2)cc1CN(C(=O)C(F)C(=O)O)CCN(C)C c1(C(=O)NC(c2cnn(C3CCCC3)c2)C(=O)OC)csc2cncn12 C1(CC(C)(C)C)(C(=O)N(CCCO)C2CCC2)CCNC1 c1(CNC(=O)NC2(CCO)CCCOC2)ccc(Cl)c(F)c1F c1(CNC(=O)NCC2CCC(C(F)(F)F)C2)cccc2ccc(Cl)cc12 C(N=c1[nH]c(N2CCOC(CCF)C2)nc2c1COC2)C1(C)COCCO1 CCCC(O)CCNC(C1(CNC(c2sccc2F)=O)CC(C)(C)C1)=O N1(C(c2c(OC)ncnc2OC)=O)CCC2(CCCN2C(=O)C(C)C(C)C)C1 C(CCC(C)(C)C(=O)NCC1(O)CCCC1(C)C)NC(CCc1ccn(C)c1)=O C1(O)(C(=O)NCCN(C(C(C)CC(F)F)=O)CC2CC2)CN2CCC1CC2 c1(NCC2CCCN(C(C(CC)(CC)CO)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 N1(C(C(C(C)C)OCC)=O)CCC2C1CCCN2C(c1ccc(C#N)cc1F)=O Cc1ccc(F)cc1N(C=O)C(COCc1c(F)cccc1Cl)Cc1ccccc1 c1(C(=O)NC(CN(C(=O)CC(C2CC2)C2CC2)CC)C)sccc1Br c1(Nc2cccc(CNC(=O)Nc3c(C)coc3C)c2)ccc2c(c1)CCCO2 C(=O)(C1=CCCCC1C)NC1CC(C)(CNC(Cc2c(C)cco2)=O)C1 CCC(CC)C(C)C(=O)N1CCC(CNC(C2CCCCS2(=O)=O)=O)C12CC2 CC1N(C(C2(C(C)NC(c3ncccc3O)=O)CC2)=O)CCOC1(C)C c1(COC)ccc(C(=O)N(CC(=O)NC(CC)C(C)O)C2CC2)o1 c1(C(=O)NCC(O)CCNC(c2ccc(O)nc2Cl)=O)ccc2c[nH]nc2n1 C12(C(C(=O)NCCC(O)CNC(=O)C(C)CN(C)C)OC)CCC(CC1)C2 CCCCCC(C(C)(C)C)NCc1cnc(CCC(F)(F)F)s1 c1(C(N(CCN(C(c2ccc(C(=O)OC)[nH]2)=O)C)C(C)C)=O)cc2n(n1)CCCO2 c1(C(N(C)CCNC(C2CCCC(C(N)=O)C2)=O)=O)cc(C(C)(C)C)ccc1N c1(C(N2CCN(C(CS(CCC)(=O)=O)=O)CC2)=O)cc2cccc(C)c2s1 c1(SC)ncc(C(=O)N(C2CN(C(=O)C(C)C3CCC3)C2)C)n1C c12ccc(cc1)[nH]c2=O.C12CCC(CC1)OCC(=O)N2.C1(CO)CCCO1.CC CN1CCc2cc(C(=O)N(C3CCC(NC(=O)Cc4nccn4C)C3)C)sc2C1 C1(C(N2CCC(CC)C2)=O)CN(C(=O)C2=CCCOCC2)CC(C)(C)C1 Cc1ncc(CC(=O)NC2CCCC(NC(c3cc(CCO)on3)=O)C2)c(O)n1 N1(C(C(=CC2CCCC2)C)=O)CC2CCCN(C(c3cnncc3O)=O)C2C1 C1(CCNC(CC2C(C)C2(F)F)=O)CCCCN1C(c1cc(C(F)F)no1)=O N1(C(=O)NC2(c3ccc(OC)c(Br)c3)CCOCC2)CCCCCCCCC1 C1(=O)CCN1.C(=O)(C(C)=CC(C)(C)C)N(CCN(C(=O)NC)C)C(C)C C1(NC(C(COC)O)=O)CN(C(=O)C=Cc2cncc(O)c2)C(C)(C)C1 C1(N(C(=O)C(=O)Nc2nnc(O)s2)CC)CC(N(C)C)C1(C)C c1(C(=O)NCC2CCN(C(C(CC(N)=O)O)=O)CC2)[nH]nc2ncccc12 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CC2CC2(NC(=O)CCC2CCC(=O)NC2)C1 C1(NC(=O)CN2C(=O)CCC2=O)CCC2CN(C(C3CCOC3)=O)CC2C1 C1(CC(N2CCC(C(C(N3CC(N(C)CC)C3)=O)F)C2)=O)CCC(=O)NC1 C(=O)(C1=Cc2ccccc2C1)N1CCC(NC(c2ncc(Cl)cc2Cl)=O)C(O)C1 C1(CN(C(CC2CC(SC)C2)=O)CC(=O)O)CCc2ncnc(C)c2C1 Cc1ccc(C(=O)NCCCNC(=O)CC2(C)CCCO2)c2c1NCCC2 Cc1cc(S(N)(=O)=O)oc1C(=O)NC1CCN(C(=O)Cn2cnnc2O)C(C)C1 C(=O)(C1=NOC2(CCC2)C1)N1C2CC(NC(Cc3ccc(C)cc3)=O)CC1CC2 CC1(C)COC(CCC(=O)NC2CC3(C2)CC3NC(c2coc(CO)c2)=O)C1 c1(C(N(C)CC2CCN(C(CSCC#C)=O)CC2)=O)cc(C(=O)OC)ccc1Cl N1(C(=O)NC2CC(Cc3n(CC)ncn3)C2)CCCC2CC12 C(CCCC)(CC(=O)NCC1(C)CCCC(=O)N1)NC(C(CC=CCC)C)=O C1(CCC)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN1C(=O)CC(C)O C(C(=O)Nn1cnn(CC)c1=O)N(C(=O)COC)CCC.C1CCCOC1 Cc1nc(Cl)sc1C(N1CCC(CC(=O)NCc2nccnc2Cl)C1)=O C12(C(=O)NC3CC(C(N4CC(C(F)(F)F)C4)=O)C3)CCCCC1C2 c1(C(=O)NC2(C(N(CCC(=O)NC3CC3)C)=O)CC2(C)C)cc(N)cc(F)c1 N1(C(C(CCC)N(C)C)=O)CC2CC(CNC(C3(SC)CCC3)=O)C2C1 C1(COCC)CC(F)(NC(=O)C(C)(C)c2cnsc2)C1.C1(C2CCC2)C(=O)N1 CC(CC1CCCCC1)C(=O)NC1(CNC(=O)COc2cccnc2)CCOC1 c1(COC)cccc(NC(=O)NCC(c2cccc(OC(F)F)c2)SC)c1 c1(C(N2CC(CNC(CN(C3CCC3)C)=O)OCC2)=O)cccc(N=[N+]=[N-])c1 N1(C(c2cc(CC)sn2)=O)C(C(=O)N(CC(C)N(C)C(C)=O)C)CCC12CC2 c1(CC(N2C(CCCNC(=O)C=CC(F)F)CCCC2)=O)ccn2cncc2c1 n1(CC)ncnc1C(N1CC(O)(CCNC(C2(C3CCCO3)CC2)=O)C1)=O CC1(C)CC(=O)NCC1C(=O)NCC=CCNC(c1ocnc1C1CC1)=O c1(C(=O)NC2(C3N(C(CCCC#C)=O)CCCC3)CC2)cnn(C)c(=O)c1 c1(CC)noc(CC)c1CC(=O)N(C(C)CN(C(=O)CCCCNC(N)=O)C)C C1(NC(C)=O)CC12CCN(C(=O)COC(c1ncsc1)=O)C2.C1(SC)CCCCO1 CN(C)S(=O)(=O)NC1CC1NC(=O)C(c1ccc(F)cc1)O C(CC(C)(C)C(=O)NCC1CCC(NC(C2CCCC3CC23)=O)CC1)OC N1(C(C(C2CCCCC2)OC)=O)CCCC(CC(N2CCC(C(C)O)CC2)=O)C1 O=C1Cc2cnc(N3CC4CC4(C(=O)Nc4cc(Br)ncc4F)C3)nc2N1 CCCCCC(O)C(=O)NCC12CCC(CC1)N(C(=O)CC(C)(C)O)C2 c1(C(N(CC(C)NC(C(C)C2CCC2)=O)C)=O)sc(Cl)cc1Br C1CCCCN1C(=O)CNC(=O)NC1CC1.C12(CCCC1)C(=O)N2.C(COC)OC c1(C(=O)NCC2(C)OCCN(C(C(C)OCOC)=O)C2)cccc2c1CC(=O)N2 c1(C(N2CCC(NC(c3nc(C)oc3)=O)C(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(CCCC)CCCN(C(c2ncoc2C2CCCNC2)=O)C1 Cc1c(C(=O)NC(CO)C(C)NC(c2cc(C3CC3)no2)=O)nn2ccccc12 c1(C(=O)NC(C(=O)NC)(C)C)ccc2c(n1)CCN(C(=O)C(O)C(C)C)C2 c1(OC)cncnc1C(=O)N(C)CC1(O)CN(C(=O)C(C)(C)c2ccccn2)C1 C1(C(=O)NCCC2(NC(c3c(CC)non3)=O)CCC2)CCCC1S(C)(=O)=O C1(CC(=O)NCC2COCC2O)CCN(c2ncccn2)CC1 Cn1cc2c(n1)CCCC2NC(=O)NCC(C(F)(F)F)n1cncn1 c1(N(C)CC2CCN(C(=O)CC3CCCOCC3)CC2)nc2ncc(Cl)cc2o1 C1(C(=O)NCC(CSC)OC)(CF)CCN(C(=O)CN2CC=CC2)C1 C1(CC(=O)N(CC(CC)NC(=O)C(C)(C)n2cccn2)C)CC(C)(C)CO1 c1(CCC(=O)NCC(CC)NC(C2CC2C(=O)OC)=O)ccccc1Cl c1(OCC)ccccc1C(C(C)CCCC1(CO)CC1)NC(=O)C(=O)N(C)C CC1(CS(=O)(=O)NC2COC(c3ccccc3)C2)CCCCO1 C(=O)(CCC(C)(C)C)N1CCC(CC=C)(NC(C2CC(=O)N(C(C)C)C2)=O)C1 N1(C(c2ncc(OC)nc2)=O)CC=C(C(=O)NCC2(O)CC(O)C2)CC1 c1(NC(=O)NC(C)C(=O)Nc2ccccc2)ccc(Cl)cc1CN(C)C CCC(C)CC(C(=O)NCCC1(OC)CCC1)NC(c1ncccc1CC)=O C=Cc1ccc(C(=O)NC(CN=[N+]=[N-])C(=O)NCCC2CCCC2(C)C)cc1 CC(CC(=O)NCC1CCN(C(C2CCC3(CCC3)CC2)=O)C12CC2)C(C)(C)C C(N=c1[nH]c(=NCc2ccc(F)cc2F)[nH]c2cc[nH]c12)C1N(CC)CCCC1 N1(C(c2c(C)non2)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(F)(F)C(C)(C)O c1(SC)nc(C(=O)NCCCCCN(C(=O)CSC2CC2)C)c2ccccn12 CC(F)(F)C(F)(F)CC(=O)NC1CCCC1NC(=O)CCc1ccccc1 c1(CC(N2CC(C)N(C(=O)Cc3cnn(C)c3)CC2)=O)cc(F)c(Br)cc1F N1(C(C2N(CC)CCC2)=O)CCCC(O)(CCNC(=O)CCc2cccnc2)C1 N1(CC)CCCC1CC(=O)NCCC(C)N(C(=O)CCc1nc(C)cs1)C N1(C(C2(S(C)(=O)=O)CCC2)=O)CCN(C(=O)C(C2CCCCC2)F)CC12CCC2 O=C(CC1OCc2cc(Cl)ccc21)NC1CN(C(C2CCCC2)=O)C1 C1(NC(c2cc(C(C)NC(C3CCC3CN)=O)on2)=O)CCCC1C1CC1 c1(OC)cc(N)c(C(=O)NCCN2CCN(C(=O)C=CC3CCC3)CC2)cc1F c1(OC)cc(C(=O)NCCN(CC(C)O)C(=O)Cc2cn(C)nn2)cc(Cl)c1 c1(C(=O)NC2CCC(NC(c3cn(CC=C)nn3)=O)C2)noc(C)c1C(=O)OC C(=O)(CCCCCC#N)N1C(CN(C(c2cnc(C)c(N)c2)=O)C)CCC1 c1(C(=O)NCC2CC(N3CCCC3)C2)cccc(S(=O)(=O)CC(F)(F)F)c1 c1(CCC(N2CC(C(=O)OC)C(N)C2)=O)c(I)ccnc1O C(CC)(CCCC(=O)NCc1nn[nH]c1C1CC1)NC(CSCCC)=O c1(C2(C(C)NCc3ccnc(Br)c3)CC2)c(F)cccc1F C(=O)(CC(C(F)F)NC(C1(C)CCN1C(=O)C(=O)N(C)C)=O)NC C1(C(=O)NCCc2c(C)nn(C)c2)CCN(C(c2cc[nH]c2)=O)CC1O N1(C(C2CC(C)C2)=O)CC=C(CC(=O)NCCn2cnnc2C)CC1 Cc1cn(C)cc1C(=O)NCCn1cc(-c2cccnc2C)nn1.C12CCCC1C2 CC1CCn2ncc(C(=O)NCCCC3(NC(=O)CCc4cc[nH]n4)CC3)c2C1 C(=O)(C1CCCn2cnnc21)NCC(CO)NC(CCNC(=O)NC)=O C1(NC(C2(SCC)CC2)=O)CN(C(=O)CNC(c2ccnc(O)c2)=O)CCC1C N1(C(CC=C)=O)CCC2(CC1)CCN(C(=O)C=C(C)C1CCCCC1)C2 Cc1nc2c(N3CC4(C3)CN(C(=O)C(O)Cc3ccc(O)cc3)C4)ncnc2[nH]1 C(C)(CO)(C(=O)NC1CC=CCC1)NC(Cc1c(CC)con1)=O C1(CNC(C2(C=C)CCCC2)=O)CCC2(CCC2)C1NC(c1cccnc1C)=O c1(C(N2CCC2CSc2ocnc2CO)=O)csc(-c2ccsc2)n1 c1(OC)cc(OC)nc(CC(N2CCC3C(NC(c4cn(C)cn4)=O)CC23)=O)n1 C(CN=c1ccc([N+](=O)[O-])c[nH]1)N(C(NNC(C)=O)=O)CCO C(=O)(CC(C)(C)C)NC(C)(CSC)CC.C1=CCNC1=O.CC=C C1(C(=O)OC)CCS(=O)(=O)C12CN(C(c1c3c(c[nH]c1=N)CCC3)=O)C2 C1(NC(C(=O)NCC(CC=C)NC(=O)OC(C)(C)C)(C)CO)CCS(=O)(=O)C1 N(C(=NCCCS(=O)(=O)c1ccccc1)NC1CCCn2nc(C)nc21)CC c1(C(=O)NC2(CNC(C3CCC4CCC34)=O)CCC2)nccc2[nH]ccc12 N1(C(C2N(C)CCC2)=O)CC2CC1CN2C(=O)Cc1ccncc1 C=CCCC(C(=O)NC1(c2ncc[nH]2)CC1)NC(C1CC(=O)N(C)C1)=O CN(C)S(=O)(=O)N(C)CC(N1CCCC(O)(CCNC(c2ccns2)=O)C1)=O c1(NC2(CC#C)CCC2)ccc(-c2ccon2)cc1 N1(C(c2ccc(C=C)cc2)=O)CCCC2CN(C(c3cccc(=O)n3C)=O)CC12 C1(CC(N2CCC2(C)CC(N2CCC(OC3CCC3)CC2)=O)=O)CCC(C2CC2)C1 C1(CNC(=O)CC2CC=CC2)CC2COCC2N1C(c1ccc2cc[nH]c2c1)=O C(CN1C(=O)C(=O)c2cc(F)ccc21)N1CCN(C(C(C)(C)C)CN)CC1 N1(C(C(C)n2cccn2)=O)CCC2(C1)CN(S(=O)(=O)c1ccn(C)n1)C2 c1(OC)ccc(C(=O)NC2CC2CNC(C2(F)C(C)(C)C2(C)C)=O)c(N)c1 N1(C(C(C=C)CC)=O)CCC(NC(c2ccc(C)o2)=O)CC1C1CC1 c1(N2CC(CC)SCC2)ncnc(NC(COC)COC)c1C C(=O)(CCC(C)(F)F)NCC1(COC)CN(C(c2cc(C)nc(C)n2)=O)C1 C=CCC(C(=O)N1CC(C(C)NC(C2(F)CCCCC2)=O)C1)c1ccccc1 c1(C(=O)NC2CC3C(NC(=O)CCn4ccnn4)C3C2)ccnc2ccsc12 CCC(CCCC(=O)N1CC(NC(=O)CC(C)C)C(F)C1)NC(=O)OC(C)(C)C c1(NC(C2CCNC(c3ccc(F)cc3Cl)C2)=O)cnc2c(c1)CCC2 C1(C(=O)NCCC2CCN(C(C3(CCC)CCC3)=O)C2)CC2COCC(C1)C2 N#Cc1ccc(C(N2CCN(C3CC3)CC2)C(=O)NCCC2CCC2)c(F)c1 C12(CNC(C(C#C)(C)C)=O)CCCC1N(C(c1nn(C)cc1C#C)=O)CCC2 CCCCCCC(F)C(=O)NC1CN(C(=O)Cn2cc(F)ccc2=O)CC1F N1(c2ccc3c(c2)CCC3)CCN(C(=NCCc2cnccn2)NC2CC2)CC1 c1(C(=O)OCC)ccc(C(N2CC3C(C2)C3(C)C)C(=O)NCCOC)c(Cl)c1 c1(C(=O)NC(CCC)C(=O)NCC(C2CC2)SC)nccc(C)c1F C1(C)(C(=O)NCc2cn(CC)nc2)CCCN1C(=O)CCC(=O)OC C(CC(C(=O)NC1(CCNC(=O)CCc2cn(C)nc2C)CCC1)N(C)C)SC N1(C(C(C)OCC(C)C)=O)C2CCC1C(CNC(=O)Cc1ccsc1Cl)C2 O=C(C1=CSCCO1)NC1CCCCC1CNC(=O)COc1ccccc1 Cc1ccc(C)c(OCC(=O)N(C2CCN(C(=O)C=CC3CCOC3)C2)CCO)c1 c1(C(=O)NC(C)CN(C(=O)CCSc2ccc(Cl)cc2)C)cccn(C)c1=O c1(C(=O)NCc2c(=N)cc[nH]c2)cnn2cnnc2c1 C12(C(=O)OCC(CCC(=O)OC)(C)C)CCCC1CC(F)(F)CC2 CN(C)S(=O)(=NCC(=O)O)NC(C1COC(C)(C)OC1)=O Cc1ccc(C(=O)OCC(=O)N(C(c2ccc(F)cc2)C)C(C)C)cc1 C1(C(=O)NCCC)CCCN1CCC(=O)NCCC(C)(F)F C12(CC)CN(C(c3coc(CO)c3)=O)C(CNC(=O)Cc3ccsc3)(C1)C2 N1(C(C=CCNC(C(C(C)C)C#N)=O)=O)CCCNC(=O)C1C(C)C C(C(C)(O)CNC(=O)COCC1CCCO1)N(C)C(c1cnn(C2CC2)c1)=O c1(OC)cccc(CCC(=O)NCCN(CC(C)O)C(C2CC(F)(F)C2)=O)n1 CN1N=C(CC(=O)N(C)CC2CN(C(c3ccc(F)c(C#N)c3)=O)C2)CC1=O CC(C)CCC(C(=O)NCC1C(CO)C1(C)C)NC(=O)CC(C)O C12CCCN(C1)C(=O)NCC2.C(CS(=O)(=O)Nc1ccn(C2CC2)n1)OC C1(F)(CNC(=O)C=CCn2cncn2)CCCN(C(C2CCS2(=O)=O)=O)C1 C1(C)(C(=O)NCCC2N(C(c3cccc(OC)n3)=O)CCOC2)CCC(=O)NC1 c1(CC)ccc(C(=O)N(CC(CC)NC(=O)C(C)C2(O)CCC2)CC)cc1 Cn1nc(O)cc1C(N1CC(CCCCNC(C2CCC(=O)NC2)=O)C1)=O C1(CC(N2CCCC2)=O)C2CCCC2N1C(=O)C(O)Cn1cncn1.CC(C)N CCCCC(CC(=O)NC1CC=C(C)CC1)NC(=O)CC1(CSC)CC1 C1(CCC(=O)NCC2(NC(C3CNC(=O)N3)=O)CCOCC2)CCC(F)(F)CC1 CCCCC(COC)NC(c1cn(CCNC(c2nnn(C)c2N)=O)cn1)=O C(=O)(CCC(=O)C(C)(C)C)NCCN(CCC)C(c1ccc(CN(C)C)nc1)=O N#Cc1cccc(Cl)c1C(=O)OCc1ccnc(O)c1 c1(C(N(CCNC(=O)CCCc2ccc(F)cc2)C2CC2)=O)cc(Cl)ccc1F CC1CC(NC(C2COC3(CCC3)C2)=O)CCN1C(=O)CC(F)(F)F N1(C(c2c(C)nc(CC)s2)=O)CC2CCC1CN2C(c1cc(F)c(F)cc1O)=O C1(C)(C(C)C)CCCN1N(CC1CCCO1)Cc1ccc2c(c1)CCC2 c1(CC(C)C(=O)NC2CCCC(CNC(=O)CC(C)(C)O)C2)ccc(Cl)cc1 CCC(CC)(CC)C(=O)NCC(C)NC(c1sc(-n2cccc2)nc1C(C)C)=O c1(C(N2C(CCCNC(COCC(=O)NC)=O)CCCC2)=O)cc2scnc2[nH]1 Cc1nn(C)c(=O)c(C(=O)NC2CCCN(C(=O)C(C(C)O)N(C)C)C2)c1C c1(C(=O)NC2CCCC(NC(C3C(=C)CC3)=O)C2)ccc2c(c1)CCCO2 n1(C(C)C)cnc(C(N2CCCC2CNC(C2CC2F)=O)=O)n1 c1(C(=O)NCCC(CNC(c2cnc3c(c2)CCC3)=O)O)cc2c(nn1)CCC2 C(N=c1nc(N2CCC(C)CC2)c2c([nH]1)CSC2)C1N(CCS(CC)(=O)=O)CC1 C1(C(=O)NC2CC(CNC(c3cc(COC)on3)=O)CC2O)CC12CCOCC2 N1(C(CC(CC)O)=O)CCCC(CNC(c2ccc(-c3cnco3)cc2)=O)CC1 C1(C(=O)NCC(CNC(COCC(=C)C)=O)CO)CC2CC(=O)C1C2 c1(NC)snc(C)c1C(=O)NC1CCC(NC(=O)CC2CCCC(C(F)(F)F)C2)C1 C(=O)(CC1CCc2cc(Br)ccc21)NCC(CNC(CCCC=C)=O)CO N1(C(c2cccc(CC=C)c2)=O)CCCN(C(=O)C(C)n2cccn2)CC1C c1(OC)ccc(C(N2CCN(Cc3cc4n(n3)CCC4)C3CC23)=O)cc1C C(C)(CCNC(=O)C=CCOCC(F)(F)F)N(C(C=CCC)=O)C N1(C(c2n(C(C)C)ccn2)=O)CCC2(CCCN2C(c2cc[nH]n2)=O)CC1 CCC(C)(C#N)C(=O)NC1CC(C(=O)NCc2ccc(N3CCNC3=O)cc2)C1 c1(C(=O)NC(CC(=O)NC2C(C)(C)C2C#N)C2CC2)cc2occc2[nH]1 c1(C(=O)NCC(CNC(c2c(C)c(Br)no2)=O)C)c[nH]c2cccnc12 c1(C(=O)NCCC2CCCN2C(=O)Cc2cc[nH]n2)sc(F)cc1Br Cc1ccc(NC(=O)C(C)NCCC2CCCC2(F)F)cc1 N1(C(C(CC)O)=O)CCC2(CCN(C(=O)CCN3CCc4ccccc4C3)C2)C1 C(C)(CN=c1[nH]c(=N)[nH]c(=NC2CCCC(C(C)(C)C)C2)[nH]1)c1ncc(C)s1 c1(C(=O)NC(CC=CC)C(=O)NCc2n[nH]cc2CC)cc(C#N)nn1C S(=O)(=O)(c1cc(C(=O)NCC2(NC(C3CC3CF)=O)CCCC2)ccc1F)NC CC1CCC(C)N1CC(N1CC=CCC1C(=O)NOCC1CCCO1)=O c1(C(=O)NC(CCCNC(CN(S(CC)(=O)=O)C)=O)(C)C)ccc2occc2n1 Cc1ncc(Cl)cc1NC(C1CCCC1NCc1ccc(-c2ccccc2)o1)=O C(CC(C)C)(C(=O)Nc1ccc(N(C)C)nc1)ONC(CCc1ccc(C)o1)=O c1(C(=O)OC)cnc(N2CC3CC2CN3C(=O)Cc2cnn(C)c2)nc1C C1(C)(C(N2CC(OC)(CNC(c3cn[nH]c3)=O)C2)=O)C=CCCC1 C1(CC(=O)NCc2c(C)cco2)CC(C)(C)CN1C(C12CC1CNC2=O)=O N1(C(=O)C=CC2CC2)CCC2(C1)c1[nH]cnc1CCN2C(C1CCCOCC1)=O c1(CCC=C)ccc(C(=O)N(CC(C)N(C(=O)C=Cc2ccncn2)C)C)cc1 c1(C(N2CCC(C)C2CNC(=O)C2=CCSC2)=O)ccc2c(c1)C(=O)NC2 c1(OCC=C)cccc(COC(C)=O)c1.C1CCSCCO1 C1(CNC(c2c(C)nc(C(C)C)o2)=O)CN(C(=O)C(F)CC2CCC2)C(C)(C)C1 O=C(C1=CCC(F)(F)CC1)NC1CCC(O)CN(C(=O)C2CC2)C1 c1(CC(N2CCCC(NC(C(CC)OC)=O)(CC)C2)=O)noc2ccccc12 C1(C(=O)NCC(C)NC(c2c(F)ccc(C)c2)=O)CCN(S(=O)(=O)N(C)C)C1 c1(C(=O)NCC2OCCCN(C(C=NOC)=O)C2)nc2ncc(Br)cn2n1 c1(CC)ccc(C(N2CCC(C(C)NC(C3(C)CCN(C)C3)=O)CC2)=O)c(O)c1 C1(C(=O)OCC)C2CC(CN(C(=O)C(C)(C)O)C2)N1Cc1csnc1C C#CCCN=C(NCC#CC1CC1)NC(C1CCCO1)C c1(C(=O)NC2CC(CNC(CC3C(C)CCC3)=O)C2)cccc(=O)o1 C1(NC(CC=CCC)=O)CCC2(CCN(C(c3n[nH]c(CC)n3)=O)C2)C1 C1(OCC)CCCCC1NC(C1(NC(=O)CCC2CCCCC2)CC1)=O c1(C(=O)OCC)cncc(C(=O)NC2CC(NC(c3nn(C)cc3Cl)=O)C2)c1 c1(CN2CCC(NC(c3ccccc3CO)=O)C2)ccc(Cl)cc1-n1ccnc1 N1(C(CSC)=O)CCCC(CCNC(C2CCN2C2CCCC2)=O)C1 c1(C(=O)NCC(CC)(C)NC(C2(N(C)C)CCC2)=O)cc(OC)cc(OC)c1 C(C(CC(C)C)C(=O)NC1CC2(C1)CC2C(N1CC(N(C)CCO)C1)=O)OC CCC(C)C(C(=O)NC1CNC(=O)C12CC2)NC(c1csc(=N)[nH]1)=O C1(CNC(C(c2ccccc2)C)=O)(CNC(C2CCSC2)=O)CC1(F)F N1(C(=O)OC(C)(C)C)CCC(C(=O)NC2CCCCC2)C(F)C1O C1(OC)(CNC(C2COCCN2C)=O)CCN(C(c2nc(Cl)cs2)=O)CC1 Cc1ccc(F)c(C(N2CCC3CN(C(C4(C)CCC(=O)CC4)=O)CC23)=O)c1F c1(C(N(C(CCNC(C(C(CC)O)(C)C)=O)C)C)=O)cc(C)c2c(O)n[nH]c2n1 CC1(C)CN(CCC(N2CC(O)(CCNC(=O)Cn3cnc(=N)[nH]3)C2)=O)CCS1 N1(C(C2C(C)CCC2)=O)CC2(CCCCN2C(=O)CCn2ccnc2)C1 c1(C(=O)NCCNC(CC2N(C(C)=O)CCC2)=O)cccc2c1CCC2 N1(C(c2c(C)con2)=O)CCCC2(C1)CN(C(=O)Cc1ccns1)C2 N1(c2cc(SCC)ncn2)CC2CN(C(c3ccncc3O)=O)C2C1 CC1(C(=O)NC2(C(F)(F)F)CC2)CC(O)CN1C(c1ccsc1)=O C(=O)(C(CCCC(C)C)N1CCOC(c2cccc(S(N)(=O)=O)c2)C1)OCC C12COCCN1C(=O)CC(C)NC2=O.C(CC(=O)NC(C)(C)C)N(C(C)=O)C CC12CC(C(N3CCC(NC(c4ccccc4F)=O)CC3)=O)(C1)C1(CCC1)O2 C1(C(N(CCC)CCO)=O)CC12CCN(C(c1sc(F)cc1C)=O)C2 N1(C(c2ncc(OC)cn2)=O)CC(NC(c2cc(Br)c(C)o2)=O)C2(CC2)C1 CCCCC(CNC(c1ccccc1OC(C)C)=O)NC(=O)CCCF C(=O)(CCCCCC#N)NCC(C(=O)NCCN1CCC2CC12)N(C)C C1(C2CCCN(C(c3ccc(N)cc3)=O)C2)(NC(CCC=C(C)C)=O)CC1 C(=O)CCCCCC(C)O.C(CC(=O)N1CC(NC)C1)OCC(C)C CC1(CNC(=O)C(CNC(C2CCC=CCC2)=O)CC2CCCC2)CCCC1O C1(CNC(CC(c2ccc(C)cc2)C)=O)CC(F)(F)CN1C(=O)C(C)CF N1(C(c2c(=O)ccn(C)c2)=O)CCC2(NC(=O)Cc3ccsc3)CCCCC12 C1(CNC(C(CCOC)C)=O)(NC(=O)CCC(C)SC)CCC(C)(C)CC1 CC1(NC(=O)Nc2ccc(N3CCC(C(F)(F)F)CC3)cc2)CCC(CO)CC1 N1(C(CC2CCN(C(C(=O)NC3CC3)=O)CC2)=O)CCC(O)C(F)(F)C1 c1(-n2ncc(OC)c2)nc2ccc(C)cc2s1.C12(CO)CCCN(C1)C(=O)C2 N1(C(C2CC(CC)C2)=O)CCCCC(NC(c2cccnc2SC(F)F)=O)C1 n1(CC)nc(C(=O)NC2COCC2C(N2CCSCC2CO)=O)cc1O CCCCC(C)C(=O)NC1CN(C(c2cnc(Cl)cn2)=O)CC1(C)C N1(C(C23CC(CC)(C2)C3)=O)CC2CN(C(C3(C)C=CCC3)=O)CC2C1 C12(C(=O)NC3C(CNC(=O)CCCCC4CC4)CCCC3)CCCC1OCC2 CCC(CC)C(F)C(=O)NC(CNC(=O)CSC)C1CC1 Cc1cc(C(N2CCCC(CO)(Nc3ncnc4sccc34)C2)=O)cc(C)c1F CN1CCCCC(C(N(CCOCCC(=O)NCC2(C)CCC(=O)C2)C)=O)C1 C(=O)(C(CCC(N)=O)N(C)C)N(CC(CC)NC(C1CN(C)CC1C(F)(F)F)=O)C Cc1cc(=NC2CCCN(C(=O)C(F)C3CCOC3)C2)[nH]cc1C#N Cc1nccc(C(=O)NC(C)CCNC(c2ncsc2Br)=O)c1Cl C1(C(=O)NC2CC(CNC(c3ncccn3)=O)C2)CCn2ncnc2C1 C(CC(C)N=c1cc(C)nc(N2CCC(Oc3ccc(CO)cc3)CC2)[nH]1)SC CCC(CC)(CCNC(C1CCCC1C(F)(F)F)=O)NC(c1cnnn1C)=O N1(C(=O)CSC2CC2)CC(NC(C2(C3CCCCO3)CCOCC2)=O)CC(F)C1 n1(CC(=O)NCCN(C(=O)C(F)CC2CC2)C)c(C(F)(F)F)nc2ccccc12 c1(C(=O)NC2C(C(=O)NC(c3cn(CC)nc3)C)OCC2)sc(C)cc1C c1(NCCN2CCN(C(C3(C)CCN(C(C)=O)C3)=O)CC2)ccc(Cl)nc1O N1(C(C(=O)Nc2cc(F)cc(Br)c2)=O)CCc2nc3ccccn3c2C1 Cn1cc(NC(=O)C(c2ccco2)NC(=O)C(N2CCOC2=O)C)cn1 CN1C(=O)COCC1CNC(C1CN(C(C2CCCCC2F)=O)C1)=O Cc1nc(N2CCC(C)C2CNC(c2cc(C(N)=O)[nH]n2)=O)cc(O)n1 c1(CCC(=O)NCC(CNC(Cc2ccc(C)o2)=O)C)ccc(=N)[nH]c1 C=CCCCCCCC(=O)NCC1CCCCN1C(=O)CC1CC2CCC1C2 N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(CCC(NC(C3CC3c3ccco3)=O)C2)C1 C(=O)(C(N)CN(c1ccco1)CCCN(CCCO)Cc1ccccc1)N(C)C C(C(C(=O)N1CCC(C(C)NC(C2CCN(C)C2)=O)C1)C(C)(C)C)OCC(=C)C C=CC1CN(C(c2cccc(N)c2)=O)CC1NC(c1csc(-c2cnc[nH]2)n1)=O c1(C(=O)NC(CN(C(C(C)OCCCC)=O)C)(C)C)ccoc1Br C1(C(=O)NCC(CNC(c2n(C)ncc2)=O)(C)O)CC2(CO1)CC(F)(F)C2 C1(C(C)C)CN(C(=O)C(O)C(F)(F)F)CCCN1C(c1ns[nH]c1=O)=O C(=O)(C(F)(F)CC)N1CCC(OCCNC(C23CC(CC)(C2)C3)=O)C1 c1(CC(N2CC3C(NC(c4csc(Br)c4)=O)(C3)C2)=O)n[nH]c2c1CCCC2 C1(C(C)NC(C=C(C=C)C)=O)CCCN(C(=O)C(c2cccc(OC)n2)(F)F)C1 c1(C(=O)NC(C)CN(C)C(c2cccc(C(N)=O)c2F)=O)cc(Cl)c(N)c(Cl)c1 C(C(C(=O)NC1CC(O)C1OC)NC(c1cnns1)=O)OC CC1CN(C(=O)C2=CCCSC2)CC(C(=O)Nc2ccc(F)cc2Cl)O1 c1(OC)ccc(-c2ccc(CNC(=O)CCc3ncccc3Cl)cn2)cc1OC Cc1nc(C(=O)NC(C(N2CC(S(C)(=O)=O)C2)=O)C2CCC2)ccc1C#N c1(CC)oc2ccccc2c1C=CC(=O)NCCNC(=O)C=C(C)C1CC1 C(C(C)(O)C(=O)N1CCC(CF)(NC(=O)CSc2ccncc2)C1)OC C1(C(C(=O)NCCCC(C)NC(Cc2c(C)scc2)=O)(C)C)CCCN(C)C1 c1(NC(CC2CC(C)N(C(=O)CC3C(C)(C)C3(C)C)C2)=O)cc(Cl)cnc1O Cc1cccc(OCC(N2CCCC(C(=O)Nc3ccc(Br)nc3)C2)=O)c1 c1(C(=O)NC2(CC)CCCN(C(=O)CC(C)CF)C2)nccc2occc12 C(=O)(C(C)(C)CCC#N)NCC1C(C)CN(C(=O)COCC(F)F)CC1 C(=O)(CCCCCCNC(C1CCCS1)=O)NCC(C)Cn1cccn1 Cc1nn(-c2ccc(Cl)cc2)cc1C(=O)NC1CCCN(C(C2CC23CC3)=O)C1 C1(CC)C(NC(c2cc(C3(C)CC3)on2)=O)CCCN1C(=O)Cc1ccc(C)s1 N1(C(C=C(C)Cl)=O)CCC(NC(=O)CCSc2ccc(F)c(F)c2)C(F)(F)CC1 N1(C(C(C)=O)=O)CCn2c(C(N3CCC4(CNC(=O)O4)C3)=O)cnc2C1 N1(C(C2(C)ON=C(C)C2)=O)CCC(C)(NC(C2CCCC(C(F)(F)F)O2)=O)CC1 C(=O)(C1CCc2c[nH]nc21)NCCOC(C)(C)CNC(c1cncc(Cl)c1)=O N1(C(COCCC)=O)CC2(CCCCN(C(C3CC34CC(C)(C)C4)=O)C2)C1 Cc1c[nH]c(C(=O)NCC2(CCNC(c3c[nH]nc3C(F)(F)F)=O)CC2)c1 N1(C(c2ccncc2Cl)C(=O)NC)CCN(C2=NCC(C)S2)CC1 Cc1ccc(C(=O)N(C)CCN(C(=O)C(c2ccc(Cl)c(F)c2)O)C)cc1Cl c1(NC2CCC(NC(C(C)C3CCCC3)=O)CC2)ncc2c(n1)CCCC2 C=C1CCC(C(=O)NCCSCc2ncc(C)s2)C1 N1(C(CCN(CCCO)C(c2c(CC)n[nH]c2)=O)=O)CCC(C)C(C)C1 c1(C(=O)NCC=CCNC(C(CC)N(C)C)=O)cnn2c1CCCC2 N1(C(CC(COC)C)=O)CCC(F)(CNC(=O)CC(C)C(F)F)CC1 c1(CN(C(=O)CC2(C)CCN2C(=O)CSC(F)(F)F)C)ncccn1 c1(NC(=O)NC(CNC(C2CCN(C(CC)=O)C2)=O)CO)scc(C)c1Cl C1(C(=O)NCC2CC3CN(C(c4scc(C)c4C)=O)CC32)CN2CCN1C(C)C2 Cc1cn2c(C(=O)C(=O)NC3(C(=O)N(CC(C)N)C)CC3)c(C)nc2s1.C(C)(C)N C1(NC(c2c(CC)c[nH]c2)=O)CC2C1CCN2C(=O)CCC1C(=O)ON=C1C c1(C(=O)NC2CCCCN(C(C=C(COC)C)=O)C2)c(Cl)ccc2ncccc12 Cn1nnc2cc(C(=O)NC3CCCC3NC(=O)Cc3cccnc3Cl)cnc12 CCCCCC(O)CC(=O)N(C)CC1CCCN(C(=O)CC(C)(C)F)C1 c1(OC(C(=O)NC(CC=C)CNC(c2ccoc2Cl)=O)C)ccccc1OC C1(CC(C)Nc2ccn(C3CCCNC3)n2)CCCCN1 C(=O)(C(C)OC)N(CCNC(=O)CCNC(=O)OC)CC N1(C(C(C)n2ccnn2)=O)CC(C2CC2)(C(=O)NCC2CCOCC2(C)C)C1 Cc1ccc(C=CC(=O)NC2C3CN(C(=O)CCc4nc(=N)[nH][nH]4)CC23)o1 c1(C(=O)NCCC2N(C(c3ncn(C)n3)=O)CCC2)nn(C)c2ccc(F)cc12 C=CC1(CC(=O)NC2CN(C(C)=O)C2)CN(C(=O)NCCN2C(=O)CCC2=O)C1 N1(C(C(c2ccc(Cl)s2)C)=O)CC(F)(CNC(=O)C=CC2CCCO2)C1 C=CC1(CNC(=O)CC2CCN2C(c2cc(COC)on2)=O)CCOCC1 C(C(=O)Nc1cc(C)ccc1O)(C(C)CC)N(C(c1c(CC)[nH]cc1)=O)C N1(C(c2ccc(OC)cn2)=O)CCC(C)(C)C1C(=O)NCCN1C(=O)CNC1=O C1(C(N2CC(OC)C(F)C2)=O)CCCC12CCN(c1ccnc3ccnn13)C2 c1(C2CC(=O)NN2)ccc(F)c(NC(=O)CCc2cnccn2)c1 C1(CNC(C(CC)(C)CO)=O)CCC2(CN(C(C3CSC3)=O)C2)O1 N1(C(C=CCC)=O)CCN(C(c2cncnc2CC)=O)C(CCC)C1 C1(NC(c2cc(OCC)c(C)cc2)=O)CCN(C(=O)CNC2CC2C)CC1(C)C C1(OC)CCC(C(=O)NC2COCC2F)N(C(=O)OC(C)(C)C)C1 CCC(O)C(C)C(=O)NCCN(C)C(c1cc(C)n(C)c1C)=O c1(C(=O)NC2CCCC(NC(=O)Cc3cnc[nH]3)C2)cc2ccc(Cl)cc2[nH]1 c1(C(N(CC(CC)(C)OC)C)C)cccc(F)c1F C1(NC(CS(=O)(=O)NCC)=O)CC2CCC(C1F)N2C(C1CC1C#N)=O C12(C(=O)NC3(C)CC(NC(Cc4c(C)noc4Cl)=O)C3)CCC(F)(CC1)C2 C12(CN3C(C(=O)NCc4cnn(CCO)c4)(CC)CCC3)CCC(F)(CC1)C2 c1(CC(=O)OCCc2ccsn2)c(F)ccc(Cl)c1Br c1(CC)ncc(C(=O)NCc2nc(C(=O)NCc3nc(=O)o[nH]3)co2)cn1 C(C1CCOCC1)=CC(=O)N(C(C(N1CC(C)(C(=O)OC)C1)=O)C)C1CC1 C1(C(N2CC3(CN(C(C)(C)C)C3)C(CO)C2)=O)CCN(C(=O)CCS(C)(=O)=O)O1 CC1(C(=O)NC(CC(=O)NCCC2(C)CC2(F)F)C2CC2)CC(=O)C1 C12C(C1(C)C)C(=O)N2.C(C(C)(O)CSC)NC(CN(CCOC)C)=O c1(CNC(CC)=O)ccc(-c2nnc(CN(C(=O)C(C)O)C)n2C(C)C)cc1 N(C(=NCCN1CCCC1)N1CCC(C2(O)CC2)CC1)C1CCCC(OC)C1 c1(OC(C)C)ccc(F)c(C(N2CCC(NC(=O)C(C)C(F)F)C2)=O)c1F C(C(C)N=c1[nH]c(=NCC2CC2)[nH]c2ncn(C)c12)(c1ccc(C)cc1)C1CC1 CCCC(C(=O)N1CC(OC)C(NC(c2cc(F)n[nH]2)=O)C1)OCC CCCC(C)(C)CC(=O)NCCCOCCN(C)C(C1(CO)CCOC1)=O CN1CCCCC(CNC(C23CC2CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C3)=O)C1 C12(NC(c3c(C)nc(O)[nH]3)=O)CCCN(C(C3(CC(C)C)CC3)=O)CC1C2 c1(OCC)ccc(N2CC2=O)cc1.n1(CC(=O)N(C(CC)C)C)cnnn1 N1(C(C(C)NC(=O)Cn2cnnn2)=O)CC=CC1CNC(=O)Cc1ccon1 C1(C(=O)Nc2c(C(=O)OCC)occ2)CN(C(=O)Cc2cccc(C)c2)CC1C Cc1n[nH]c(C)c1SCC(=O)NC1CCCC(NC(=O)CC2CCC(C)CO2)C1 C1(CCNC(c2c(CC)csc2)=O)CCCCN1C(=O)Cc1nncn1C(C)C Cc1nc2cc(NC(=O)CC3COCCN3C(c3sccc3F)=O)ccc2o1 c1(CC(C(=O)NCC(CN(C(=O)COC2CC2)C)(C)C)(C)C)ccc(C#N)cc1 N1(C(CC)=O)CCC(C)(NC(=O)NC2CC(OC(C)(C)C)C2)C1 N1(C(C2(NC(CCOCCOC)=O)CCCC2)=O)CC2(CC(CO)CO2)C1 CC1CN(C(c2ccc(Cl)cn2)=O)CC(C)C1Nc1nc(Cl)ncc1Cl C1(C(=O)NCC(CN(C(Cn2c(C)ncc2)=O)C)O)CC12CCC1(CC1)CC2 CC(C)CS(=O)(=O)CC(=O)N1CC(CNC(c2csc3cccnc23)=O)CC1C Cc1ccc(C)c2c1N(c1ccc(Br)cc1C(F)(F)F)CCC2 N1(C(CCNC(COC)=O)=O)CC2CC(NC(=O)CCc3ccncc3)C1C2 C1(CNC(CC(COC)(C)O)=O)CC2(CCC2)CN1C(=O)CCc1cc(C)on1 C(=O)(C(F)(F)Cc1ccc(Cl)cc1)N1CC(C(C)(C)C)C1 N1(C(=O)NC(c2ccc(O)cc2)C)CCC(Cc2ccccc2Cl)CC1 CCCC(CCC)CC(=O)NCC=CCNC(=O)CCc1ncc[nH]1 C(CCC(N)=O)(C(=O)NC(C)(CNC(=O)CCCCCF)C1CCC1)NC(C)=O c1(C(=O)NC23CC(NC(=O)C(O)C(F)F)(C2)C3)cc(F)cc(F)c1O C1(NC(C(C)SCCCC)=O)CC(NC(C2CC=CCO2)=O)C(O)C1 Cc1c(C(=O)NC2C3CN(C(c4cc(F)ncc4Br)=O)CC23)cncc1Br N1(C(c2cc(OC(F)F)cc(F)c2)=O)CCCC1C1CCCN1C(=O)C(Cl)=CCl c1(OCC)nc(N2CC(C(C)NC(=O)C(C)(C)c3ccccc3)C2)ncc1Cl N1(C(CC2(C)CCOC2)=O)CCCN(CCNC(C2CCCN2C(N)=O)=O)CC1 N1(C(CCSC)=O)CCC2CCCC(C1)N2C(=O)CCc1cnn(C)c1 C1(CC(=O)NC2CN(C(CC(CC=C)(C)C)=O)CC2F)Cn2ccnc2NC1=O c1(C(N2CCN(C(c3c(CC)[nH]c(=N)s3)=O)CC2)=O)cc(C)ncc1C CS(=O)(=O)c1c[nH]ccc1=NC(=O)N(CCN1CCOCC1)CCO C(=O)(C1CCc2c(Cl)cccc21)NCC1N(C(CC2CC=C(C)CC2)=O)CCC1 N1(C(C(CC)(C)OC)=O)CCN(C(c2ccc(C3CC3)s2)=O)CC12CC2 C1(NC(c2ccc(OC)nc2Cl)=O)C2CCC1CN(Cc1ccnn1C)C2 N1(C(C=C2CCC(C)CC2)=O)CCN(C(C2CCC(=O)CC2(C)C)=O)CC(O)C1 Cc1ccc(S(N)(=O)=O)c(C(=O)NCC2C3CN(C(C45CC(CO4)C5)=O)CC23)c1 N1(C(C2(OC(C)C)CCC2)=O)CCOCC2(COCCN2C(c2ccc[nH]2)=O)C1 c1(C(=O)NCCC(=C)CNC(C2CC2C)=O)cc(Br)cc2scnc12 CC1(C)C(CC(=O)NCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1O N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC1(C)CN(C(=O)CN2OC(C)(C)CC2=O)C1 C1(C(=O)NCCN(C(c2cc3cnccc3[nH]2)=O)CC)OCC2COCCC12 C(CCC(O)C(=O)NOCCN(C)C)NC(c1cnc(OC)s1)=O CC(C)(CO)C(CNC(=O)C(=O)Nc1cccc(F)n1)c1ccco1 C(=O)(C(C)(O)CSc1cccc(F)c1)N(CCCNCC)NC(=O)C(C)OC CCC(CC)C(C)C(=O)NCC1CN(C(=O)Cc2cc(F)ccc2OC)C1 N1(C(c2c(C)nc(C(C)C)cc2)=O)CC2CN(C(c3cnoc3C)=O)CC2(C)C1 N1(C(CCC(N)=O)=O)C(C(=O)NCc2cc(O)cc(F)c2)CCC12CC2 C1(C(N2CC(CC#C)OCC2)=O)N(C(c2cc[nH]n2)=O)CC12CCCC2 C1(CC(=O)NCCC(C)N(C(c2cn(CCC=C)nn2)=O)C)CCCC(=O)C1 Cc1cc(C)n2ncc(C(=O)N(C)Cc3nc4ccccn4n3)c2n1 c1(CC(=O)NCCN(C(CC(C(C)C)OCC)=O)C(C)C)ccccc1[N+](=O)[O-] C(=O)(C1=C2CCN=C2NC=C1)N1CC2OCC(NC(CCSC)=O)C2C1 C1(C(=O)NCC(CCOC)NC(c2ccc(C(N)=O)cc2)=O)CC=C(C)CC1 N1(C(C2(CC)CC2)=O)CCC(C)C(NC(c2cc(C3CCCCC3)[nH]n2)=O)C1 c12ccc(cc1)CN1CCC(C1)CNC(=O)CCO2.CCCCCOC(F)(F)F c1(CC(=O)NCC(N(C(C2C(=C)C2)=O)C)C2CC2)c[nH]c2cccc(OC)c12 CC1(CO)CC(O)CN1C(C1CCC1)=O.O1NC(=O)CNC(=O)C1 CCCC(CC)C(=O)N1CC(CNC(=O)CNC(C)=O)C(C)C1 C1(CNC(c2c(CC)occ2)=O)CN(C(=O)CSc2n[nH]c(C)n2)CCO1 C1(C(N(CCCNC(c2ccc(C(C)C)o2)=O)C2CC2)=O)CC2(C1)CC21CCC1 CCCCC1CC(=O)N1.C12(NC(=O)C=C(C)COC)CC(C1)C2 c1(OC)ccc(Br)cc1NC(=O)NC(c1nc(C2CC2)no1)(C)C N1(CCN(C(=O)C(=O)Nc2scc(C)c2)C)CCc2c(Br)cccc2C1 N1(C(C(C)n2cnnn2)=O)CC2(CCC2CNC(c2cc(Br)no2)=O)C1 c1(C(C)C)ncoc1C(=O)NCC#CCNC(c1cc(Cl)ns1)=O C(=O)(C(O)C(C)(C)CC)N(C1CC2CN(C(CN(C(=O)OC)C)=O)C1C2)C C1(OC)CCCCC1C(N1CC(C(C)NC(c2cc(CC(C)C)nn2C)=O)C1)=O CCCCC(F)C(=O)NCC1CCCCC1C(=O)NOC1CCC(O)C1O CN1CCC2CN(C(=O)CC3(CNC(=O)C=Cc4ccoc4)CC3)CC2C1 Cc1c(C(=O)N(C)CCNC(=O)CCCc2nccs2)cccc1F C1(CC(=O)NCC2(C)CC(NC(c3c(SC)ccs3)=O)C2)C(=O)NN=C1C CC(CC(F)(F)F)C(=O)NC1CCC(CNC(c2ccc3[nH]ccc3n2)=O)CC1 c1(C(=O)NCC(CNC(c2cc(C)nc(O)n2)=O)F)ccnc2cc[nH]c12 Cc1nc(=NC2CC(NC(C34CC5CC(CC(C5)C3)C4)=O)C2)[nH]c2ccccc12 C#Cc1cccc(CC(=O)N(CCCCN(C)C(C2(C)CC2(F)F)=O)C)c1 N1(C(C=Cc2ccn(C)c2)=O)CCCC12CCN(C(C1CCC(C)(C)CO1)=O)C2 N1(C(c2[nH]cc(C#N)c2)=O)CCC(O)CC1C(=O)NC1CCC(F)(F)CC1 C1(C(=O)NCC2(C(N3CC(CN(C)C)C3)=O)CCCO2)COCC1(C)C C1(C)(NC(C(C)SCC)=O)CCN(C(=O)C2=C(C)OCC2)CC1 c1(C(=O)NC2(C)CC(NC(c3cnc4ccnn4c3)=O)C2)cnc2[nH]cnc2c1 N1(C(c2c(C)snc2)=O)CCCC(O)(CNC(c2ccc(CCF)cc2)=O)CC1 C1(CNC(C(C=C)(F)F)=O)(CO)CC12CCN(C(c1coc(OC)n1)=O)CC2 c1(C(=O)NC(CC)(CNC(C2(C)COC2)=O)CC)cc(Cl)c2ccncc2n1 c1(C(=O)NC2C(OC)CN(C(C3C(C=C)C3)=O)C2)cc2c(F)cccc2s1 Cc1cccnc1C=CC(=O)NCC(C)N(C(=O)CC(C(F)F)n1ccnc1)C c1(CC)cscc1C(=O)NC1CCCC1CC(=O)NCC1SCCS1 C1(CNC(C2(CC)CN(C(C3CC(O)CN3C)=O)C2)=O)COCC(C)O1 C1(NC(c2ccc(COC)o2)=O)CN(C(=O)C(F)CC2CCOC2)CC1C c1(C(=O)NCC(CO)NC(c2ccc(C)cc2O)=O)cc([N+](=O)[O-])c(C)cc1C C1(CC2CCN(C(=O)NC3(C)CNC(=O)C3)CC2)CCC(F)(F)CC1 c1(C(=O)NCC(F)CNC(C2CC=CCC2)=O)c[nH]cc1Br C12(NC(=O)C3=COCCO3)CCCC(CN(C(C3CC4(C3)CC3(CC3)C4)=O)C1)C2 c1(C(N2CC(C)C(CNC(=O)C(C)N(C)C)C2)=O)cc2cccc([N+](=O)[O-])c2[nH]1 N1(c2cc(NC(c3ccc(F)c(Cl)c3)(C)C)ncn2)CCOCC(O)C1 N1(C(C2CC2N(C)C(C2CCCCC(=O)N2)=O)=O)CC2(CC(NC(C)(C)C)C2)C1 Cc1[nH]c(Cl)nc(=NC2CN(C(C3C4CC5C(C4)C35)=O)CC3(CCC3)C2)c1C#N N1(C(=O)Cc2cc[nH]n2)CCC2(CC1)CN(C(c1cc(F)cc(Cl)c1O)=O)C2 Cc1cc(C(=O)NC(c2cccc(C(=O)O)c2)Cc2ccccc2)nn1C Cc1cc(NC(=O)C(=O)NC(c2cnn(C)c2)CN(C)C)c(C)s1 CCC(C(=O)NCc1csc(C(=O)NC(c2ncc(C)s2)C)c1)OC N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCC(C(C)C)CC2)=O)C1 N1(N(c2ccccc2)C(CC(CCCC(N)=O)(F)F)=O)CCC(c2cccnn2)C1 C1(OC)(CNC(C2CC2CNC(C2CCC2)=O)=O)CCCC1 N1(C(C2(C#C)CCCC2)=O)CC2CC(NC(C3(C)CCN(C)C3)=O)C1C2 C1(CN(C(=O)CC2CC(F)C2)CC)CCN(C(=O)CC2(N(C)C)CCCC2)CC1 C(=O)(C(C(C)C)n1ncc(N)n1)NCC(=C)CCNC(C1C=CCC1)=O c1(Cn2cc(-c3c(COC)c(Cl)cc(Cl)c3)nn2)n[nH]c2cccc(C(N)=O)c12 C1(C(=O)NCC(CC)(CC)NC(=O)C(C)N2CC(C)C2)CC2C=CC1C21CC1 C1(CNC(C=CCOC)=O)CN(C(c2sc(OC)nc2Cl)=O)C2COCC2O1 Cc1ccc(C(N2CCC2(C)CC(=O)NC23CCC(CC2F)C3)=O)c(C)c1 C(=O)(C1Cc2ccc(Cl)cc21)NCC1N(C(c2ccc(OC)cc2O)=O)CCC1C N1(C(c2c(N)non2)=O)CCOC(CNC(C2CC3CC3C2)=O)C1 C(CC(CNC(=O)C(C)(C)NC=O)NC(=O)C(Cc1ccsc1)NC=O)OC c1(C(=O)NCC2C3CN(C(C4CC(=O)N4)=O)C2CCC3)ccc2cnccc2c1 C12(NC(CC3(C=C)CN(C(=O)CC(C)C4CC4)C3)=O)CCCC1OCC2 CC1=NOC(C(=O)N(C2CC(C(=O)NCCc3cnc(C)[nH]3)C2)C)C1 CC(C)C(Cc1ccccn1)N=c1cc[nH]c(=NCCCCF)[nH]1 N1(C(c2cccc(C)c2O)=O)CCC(C2(NC(=O)C(n3cc(Cl)cn3)C)CC2)C1 Cc1cc(C(N2CCN(CCNC(c3ccc(F)s3)=O)CC2)=O)c2c(c1)CCC2 CC(CS(C)(=O)=O)C(=O)NCC(C1CCC1)NC(=O)CCc1ccc(O)nn1 CC1CN(C(=O)CC2CC2C(F)(F)F)CCCN1C(=O)C=CCO C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC1(O)CC(NC(C(=O)N(C)C)=O)C1 CCC(CC(=O)N1CCCCC(NC(C2CCC2)=O)C1)C(C)(C)C.C(C)=O C12(C(=O)NC3CCC(NC(CC(CN(C)C)O)=O)C3)CC3CC1C2C3(F)F n1(CCC)nccc1C(=O)NC1CCCC1CNC(=O)C(C)Cc1cnc[nH]1 c1(C(=O)NC(CCNC(c2cc(OCC)no2)=O)C)cnn(C)c1CC c1(NS(CCC2CC(OC)(OC)C2)(=O)=O)cc(Cl)c(F)cc1[N+](=O)[O-] O(N(C(=O)C1CCCCN(C(=O)C(C)C(C)C)C1)C(C)C)CC N1(C(C2(OC)CCC2)=O)CC(C(F)(F)F)C(CNC(C2CCN(C(C)C)CC2)=O)C1 C1(CCNC(c2n(CCCC)nnn2)c2cscc2F)CCCS1(=O)=O Cc1ccc(C(CCO)Nc2cc(NCC3CCCS3(=O)=O)ncn2)cc1 CC1(C)CC=C(C(=O)NC2CC2NC(C2CC3(C2)CC(C)(C)C3)=O)CC1 CCC(C)CC(C(=O)N1CCCCC1CCCO)NC(=O)CC(C)(C)C(C)=O c1(C(N2CCCC(N3CCN(C(C4CCC4)=O)CC3)C2)=O)ccc(F)cc1F C12(C(N3CCC(C#N)(F)C3)=O)CCCC1CN(C(=O)CC1(O)CCOC1)C2 c1(OC)ccccc1NC(=O)C(c1cccc(Br)n1)N1CC=CCC1 c1(NC(=O)CC2C3CN(C(c4ccc(CO)o4)=O)CC23)ccc2n[nH]cc2c1 N1(C(C(C(C)C)O)=O)CCC(n2cccn2)(CNC(c2cc(C#N)cs2)=O)CC1 N1(C(c2ccc(C(C)=O)s2)=O)CCOCC1CNC(=O)C(C1CCOCC1)C c1(NC(C)=O)cc(S(=O)(=O)NC(C2CCOCC2)C(=O)OC(C)=O)ccc1N c1(C(N(CCNC(C=CC(=O)OC)=O)C2CC2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 c1(NCC)ncccc1S(=O)(=O)NC1(c2nnnn2C)C(CC)CCOC1 N1(c2nc3ncn(C)c3cn2)CC2C3CCC(C2C1)N(C(=O)C1=CCOCC1)C3 C1(C(N2CCCC(CCNC(C3(C)CC3(F)F)=O)C2)=O)CCCC12CCOCC2 C(CN=C(NCC(c1cccs1)(C)C)N(C)CC1CCC1)N1CC(C)CC(C)C1 c1(N(CC(CN(CC)CC)O)CC)cccc(C#N)c1 c1(C(=O)NC(CCC)CC(=O)N(CC(C2CC2)OC)C)cccc2[nH]ncc12 N1(C(C(=O)NC2CC(C)N(C3CC3)C2)=O)CCc2cc(F)c(F)cc2C1 c1(C(=O)NC2(COC)CN(C(=O)CCc3nc(C)cs3)C2)nnccc1C Cc1cc(C(=O)NC(Cn2cccn2)C(N2CCN(C(C)(C)C)CC2)=O)ncn1 C1(NC(C(C)C(F)F)=O)CN(C(c2cccc(OC3CC3)c2)=O)CC(C)(C)C1 C1(C(=O)NCc2c(C)occ2)COCCC1NC(c1csc(F)c1)=O c1(CC)n[nH]cc1C(=O)NC1CCC(N(C)C(c2cc(-c3ccco3)on2)=O)C1 c1(NC(c2cc[nH]n2)C)[nH]c(=NCCCCO)nc2c1cnn2C C1(C(=O)NCC2(NC(=O)CC3CCCC3)CCOC2)CC2(CCCC2)CO1 C(CCCCCCO)(C(=O)NCCC#N)N(CC(=O)NC1CC1)CCC c1(CC)cccnc1C(N1CCC1CC(=O)NC1CCC(CO)CC1)=O C1(C(=O)NC2C(F)CCN(C(Cc3c(C)scc3)=O)C2)CCc2[nH]nc(O)c2C1 c1(C(=O)NC(CC=CC(=O)NCC2(OC)CC(C)(C)C2)(C)C)cn(C)c(=O)n1C c1(CC)cc(C(=O)NC(C)(CNC(C2CCS(=O)(=O)N2)=O)C2CCC2)ccc1F N1(C(c2cnc(C(C)C)s2)=O)CCC(NC(=O)CCN2CCCC2)C(O)C1 CC1(C)CCC(CC(=O)NC(C)(C)C(=O)ON)N(C(=O)OCc2ccccc2)C1 C1(NC(CCC(=O)NC)=O)CCN(C(=O)Cn2cnc(C(N)=O)n2)C12CC2 C(=O)(CCCCCCCCCO)N1CC2CN(C(C(C(CC)O)C)=O)C2CC1 CC1CN(C(=O)Cc2ccccc2I)CC1C(=O)NCC1C=CC(=O)N=N1 Cc1nn2c(c1C(=O)NCC(C)CNC(=O)CC1CCCCO1)CCCC2 c1(C(N2C(C(C)NC(C3CC(C)(C)C3C(F)(F)F)=O)CC2)=O)ccc(Cl)c(C#N)c1 c1(OCC(=O)NCCN(CCC)C(c2[nH]cnc2C#N)=O)cc(Cl)ccc1Cl c1(CC(N2CCC(C(=O)Nc3ccc(O)nc3)CC2)=O)cccc2ncccc12 N1(C(C2(OC)CCOC2)=O)CC(F)CC1CNC(=O)COCc1ccnn1C CN1CCN(C(=O)NCCC2COCCN2Cc2ccc(O)cc2Cl)C(CO)C1 C12(C(=O)OCC)COC(C(=O)N(C)CC3CCCN3C(=O)C3=COCC3)(C1)C2 C1(C(=O)NCC(=C2CN(C(C3CCCN3C3CCCC3)=O)C2)F)CC2CCC1C2 C1(C(N2CCC(N(C(CCc3c(C)noc3C)=O)C)C2)=O)CCCC(F)(F)CC1 Cn1cnnc1CCCC(=O)NC1COCC1NC(c1cc[nH]c1C1CC1)=O C1(C(=O)NC2CCN(C(=O)CN3CCCC3CO)CC2)CCCC2(CC2)C1 CC(F)(F)C(C)(C)C(=O)NC1CS(=O)(=O)CC1NC(=O)C(O)(C1CC1)C1CC1 c1(-c2ccc(CNC3CON(CC)C3=O)s2)ccc(SC)c(C)c1 C(C)(C)(CC(F)C(=O)NCc1csc(CO)n1)NC(C(C(C)C)SC)=O c1(C(N(C(C)C(N2CCC(CCOC)C2)=O)CC)=O)cc2ccccn2c1 Cn1cc2c(C(N3CCCC(NC(=O)C4=CC5C=CC(C4)C5)C3)=O)cccc2n1 Cc1ncccc1CC(=O)NCCCOCCNC(=O)CN1CCCC1=O C1(NC(C2(OCC)CCC2)=O)CN(C(=O)Cn2ncccc2=O)CCC1CO C1(C)(C(=O)NC(CNC(CCSC)=O)CO)CCN(C)C1=O C1(NC(NCC2CCC(C(N)=O)O2)=S)CCC(=O)NC1 c1(C(N2CCC(CNC(C(C(C)(C)C)OC)=O)CC2C)=O)c(C)cc(O)cc1C C1(NC(C(C=CC)O)=O)CC2(CCN(C(c3cccc4nncn34)=O)C2)C1 c1(N(CC(CCC)C)C)cc(NCc2ncoc2C(=O)NC)nc(C)n1 C(CC(=O)NNC(=O)C(C)N)NCC(C)C(C)C.CCO C1(NC(C2CN(CCC)C(=O)C2)=O)CCN(C(c2c[nH]nc2OC)=O)CC1O C(CCC(=O)NC(c1n[nH]c(CO)n1)C)(C(C)C)NC(C(c1ccc(C)o1)C)=O C1(N(CC(=O)N(CC(C)NC(=O)NC)C)C)(C=O)CC1.CCOCC CC1CCCC(C)C1NC(c1cc(CNC(c2cc(Cl)cn2C)=O)no1)=O C1(C(N2CC3C(CNC(C4C(C)C4C)=O)(C3)C2)=O)CC2CCCC2C1 C1(C)(NC(C2C3N(C(c4c(C)csn4)=O)C(CC3)C2)=O)CN2CCC1CC2 C1(CCNC(c2nc(C)oc2)=O)CCCCN1C(c1cnnn1C)=O Cc1cn2c(n1)CC(C(N1CC(NC(=O)Cc3c[nH]nc3O)CCC1C)=O)C2 N#Cc1ncc(Br)cc1NC(C1C2CCC(C2)N1C(c1ccc(O)c(Br)c1)=O)=O CCCC(CNC(c1c(C)nsc1N)=O)C(=O)NC(c1nc[nH]n1)C1CC1 c1(Oc2cccc(-c3ccc(NC(C4CCCCO4)=O)s3)n2)ccc(Br)cc1F N1(C(C2CN(C(c3ccc(C)cc3)=O)C2)=O)CCc2c(n(C)c3ncccc23)C1 CN1CC(C(=O)NCC2CCN2C(=O)CNC(c2ccccc2)=O)OCCC1=O C(CC(C(C)(C)C)NC(C1CCCC1C1CC1)=O)N(C(=O)Cc1ccsc1)C C1(C)(CNC(CC(C)NC(N)=O)=O)CCCN1C(=O)COc1ccon1 N1(C(Cc2ccc(C)s2)=O)CC2(C1)OC1(C)CC2(NC(C2CCCCN2C)=O)C1 CC1OC(=O)NC1C(N1CCCC(CNC(=O)CC2C=CCC2)C1)=O c1(NC2CC(NC(c3c(C)[nH]nc3Cl)=O)C2)ncnc2cccc(Br)c12 C1(C(=O)NC(CC=C)C2CC2)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C(=O)OCC)cnc2nc(OC)ccn12.C12(C(F)F)CCN(CC1)C2=O N1(C(c2nc(CNC(CCC=C)=O)oc2)=O)CCN2CC(C)CC2C1 N1(C(C(COC)OC)=O)CC2(C1)OC1(C)CC2(NC(c2cn(C)nn2)=O)C1 CP(C)(=O)c1cccc(S(=O)(=O)NC2(C(F)(F)F)CC3C=CC2CC3)c1 Cc1cc(C)c(C(=O)N(C(CNC(c2ccc(C(N)=O)[nH]2)=O)C2CC2)C)c(S)n1 C1(C(N(C)CC2CCCN2C(C2(C)CCC(=O)N2)=O)=O)CSC(c2ccccc2)=N1 C1(NC(CCC)=O)CCCN(C(c2ccnn2C)C(=O)NCCC2CC2)C1 CCC(CC(=O)NCCC1CCOC1(C)C)NC(=O)CC(C)n1ccnc1 c1(-c2cc(C(=O)NCC(CN(C(CC(C)N(C)C)=O)C)O)n[nH]2)cccc(Cl)c1 NS(=O)(=O)c1ccsc1C(=O)NCC1CCC(NC(C2CC(F)(CO)C2)=O)C1 Cc1cccc2c1CC(C(=O)NC1CN(C(C3(C)CCCCCC3)=O)CC1C)N2 C1(C(=O)NCCN(C(C)C)C(C2(CN(C)C)CC2)=O)COC(C)C1 c1(N2CC(NC(C3(C)CC=C(C)CC3)=O)C(C)C2)cc(C#N)ccc1[N+](=O)[O-] c1(C(=O)NCC2CC(OC)CN2C(=O)CC(C)OC)ccc2nc(C)cn2c1 N1(C(C2C3(CC(NC(C4CC(=C)C4)=O)C3)C2)=O)CC2CC=CC1C2 C1(C(N2CC(NC(c3cc(O)ccc3F)=O)C(F)C2)=O)CCCCNC1=O N1(C(CNC(CCC)=O)=O)CC2CN(C(c3ccc(N)cc3F)=O)CC2(C)C1 c1(C(=O)NCCCN(C(=O)C(F)C2CCC2)CCC)coc(C)n1 CCCCCCN(CC(=O)NC1CC(NC(=O)Cn2cc(C(=O)OC)cn2)C1)C C12CCN(C1)C(=O)C(C)(C)CC(C)NC(=O)C2C.C(C)(=O)NC(N)=O C1(OCC(=O)NC(C2CCN(C(Cc3cc(C)ns3)=O)C2)C)CCN(C)CC1 CON=Cc1ccc(C(=O)NCC2CN(C(=O)CC=C(C)C)CC23CC3)cc1 C1(C(F)F)(NC(c2cscn2)=O)CCN(c2ccnc(C(F)F)n2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1C2CN(C(C3N(S(C)(=O)=O)CC3)=O)CC1CC2 C1(C(N2CC(N(C(=O)CC3(C)CCOC3)C)C2)=O)CC(OC(C)(C)C)C1(C)C N1(C(Cc2ccc(C)o2)=O)CCCC2(NC(c3cnn(C)c3F)=O)CC2C1 C1(NC(C(C)Sc2ccc(Cl)cc2)=O)CC2C1CCN2C(=O)Cc1c[nH]nc1O N1(C(C2CC(=C)C2)=O)CCC2C(CCN2C(c2ccc([N+](=O)[O-])cc2I)=O)C1 C1(OC)CC(CC(=O)NC2(CO)CN(C(=O)C(F)(F)CN(C)C)C2)C1(C)C C12(C(N3CCC(CC)C3)=O)CC(CNC(=O)CC3(C)CC3(F)Cl)(C1)OC2C Cc1cc(C(=O)N(C)CCNC(c2c[nH]nc2C2CCC2)=O)c(N)c(F)c1 CC(C)C(CN(C)C)N=c1[nH]c(=NCc2c(Cl)cccc2Cl)[nH]c2cccnc12 C1(C(N2CCC(NC(CCc3ccc(SC)cc3)=O)C2)=O)CN(S(N)(=O)=O)C1 c1(C(N2CC3N(C(C(CC#C)C)=O)CC(C3)C2)=O)[nH]c2ccc(OC)cc2c1C C(=O)(N=c1ccn(CC(N)=O)[nH]1)C1N(C(C2N(C(=O)OC)CC2)=O)CC(O)C1 C(=O)(C(C(C)C)NC(N)=O)N1CC(O)(CCNC(C(C)NC(COC)=O)=O)C1 C1(=CC(=O)NCCOCCNC(C2C(C)OC(C)C2)=O)CCC(C)(C)CC1 N1(C(c2c(CC)ccs2)=O)CCN(C(=O)C2=CCC(C(F)(F)F)OC2)CC(O)C1 C12(CC)CCCN1C(=O)C(C1CCC1)CN(C)C2=O.N1(C(COC)=O)CCCC1 N1(C(C(COC)OC)=O)CC(OC)CC1CNC(=O)CCCN1CCCCC1 CC1(C)CC(CC(=O)NC2CCN(C(c3cnc(C(N)=O)s3)=O)C2)CCO1 O=C(C1=CCN(C(=O)C=C2CCCCC2)CC1)NCC12CCCCC1C2 C1(CNC(C2(C)CC(C)C2)=O)CN(C(c2ccoc2C(C)C)=O)CCO1 O(S(=O)(=O)c1ccccc1)c1ccc(N2C(=O)N(c3ccccc3Cl)CC2)s1 c1(C(=O)NCC2CC(NC(=O)Cc3cncnc3)C2)cc2c(cc1F)NCCC2 C1(CNC(=O)CCc2cnoc2)CN(C(=O)C2CC2)C2CCN1C2 c1(C(N2C(CNC(C(C)SCC)=O)C(CC)CC2)=O)nccc(N)c1Cl Cc1cc(NC(C2CN(C(c3c(C)nn(C)c3C)=O)CC2(F)F)=O)ccc1F C1(NC(C2(C)CCSCC2)=O)CCN(C(C2CC=CCC2)=O)CC1CO N1(CC)CCCCC1c1nc(O)n[nH]1.C(CC)(CF)N C(=O)(C(C)(F)CCCC)N1CCC(CN(C(C(C=C)(C)C)=O)C)C1 c1(CN(C(=O)NCC2C(C)OCC2)C)ccc(-n2cccn2)nc1 N1(C(CC(CC)(C)C)=O)CCN(C(=O)CCn2ccccc2=O)C(C)C1C C1(C(N(CCC(=O)NCC(c2nccs2)C)C)=O)CC1C1CCCC1 C1(CNC(c2cnn(C)n2)=O)CN(C(c2cnn(CCO)c2)=O)C2CC12 N1(CC(=O)NCCCCCNC(=O)CNC(=O)Nc2ccccc2)CCOCC1=O C1(C(=O)NCC(C)(CO)NC(c2coc3c2COC3)=O)CCc2[nH]nc(O)c2C1 c1(C(=O)NCC(CN(C(c2cncc(OC)c2)=O)C)C)ccc2oc(C)nc2c1 N1(C(C(C)C#N)=O)CC(C(=O)Nc2cc(C#N)ccc2F)C2(CCC2)C1 c1(C(=O)NC23CC(NC(=O)CSC(F)(F)F)(C2)C3)ncc(Br)cc1F CC(C(Cc1ccsc1)CO)NC(=O)NCC1(C(F)F)CC1 CC(C)(CO)C(C)(C)NC(C1CCCCN(C(=O)C=Cc2ccncc2)C1)=O C1(OC)CC(F)CN(C(=O)CC2CCCN2C(=O)CC2(C)CC2)C1 N1(C(C(CC)C)=O)CCC(F)C(NC(=O)C(c2ccccc2Cl)O)C1 C1(=CC(=O)NCC2(F)CCN(C(C(=O)NC(C)C)=O)C2)CCC(C)(C)CC1 c1(OC)ccc(NC(C2(NC(=O)CC3CCOC3)CCSC2)=O)cc1 N1(C(C(C)(C2CC2)OC)=O)CCC(CNC(c2c[nH]cc2C(C)(C)C)=O)C(C)C1 C1(C(N2CCOCC(F)(CNC(=O)C(C3CC3)C3CC3)C2)=O)CCOCC12CCC2 C#CC1(C(=O)NC2CCN(C)C2=O)CCN(C(c2cnn(C)c2CC)=O)C1 c1(OC)ccc(O)c(OCC(O)CN(C)CC2C3COCC23)c1 C(=O)(C(N=[N+]=[N-])C(C)C)N1C(CN(C(C2CC(CC(=O)OC)C2)=O)C)CCC1 N(C1CC2(CN(C(c3c(C)cnn3C)=O)C2)n2ccnc21)C(CCCC(=C)C)=O Cc1cc(C(=O)NC2CC(CNC(=O)C(F)=C3CCC3)C2)c2[nH]cnc2c1 CC1(C)CN(C(=O)Cn2cnnn2)CC(CNC(c2cc(Cl)ns2)=O)O1 C12CCCC(C1)N(C)CC(C)CNC2=O.c1(N(C)C)cc(-n2ccnc2)ncn1 c1(C(=O)NCCCN(C(C2(C(C)C)CCCO2)=O)C2CC2)cnnc2ccccc12 C(=O)(C(=O)CC(C)CC)NC1CCCC(C(=O)NC(CC#C)CO)C1 c1(C(=O)NCC(CC)NC(=O)C(O)CCC(C)C)c(C)cc(C)cc1C CCCCCC(O)C(=O)NC(C)(CN(C)C)CNC(=O)C(O)CN(C)C(C)=O CC1CC(=O)NCC1C(=O)N(C)CCN1CCN(C(C2OCCCO2)=O)CC1 C=CCC(C)C(=O)NCC1(C(N)=O)CN(C(C2(CF)CC2(F)F)=O)C1 C1(NC(c2c(C)noc2)=O)C2CC3CN(C(=O)CS(=O)(=O)C(C)C)C1C3C2 c1(C(N(CC(C)NC(=O)C(C)NC(c2cnccn2)=O)C)=O)ns[nH]c1=O Cc1nc2cc(C(=O)NCC(C)(CO)NC(=O)CC3CCC(=O)N3)cnc2[nH]1 Cc1cc(C(=O)Nc2cnc(Cl)cc2C(=O)Nc2c(C)cccc2Br)ccc1O c1(N(C)C)ccc(NC(c2cccc(C(C3CN(CC(F)F)C3)=O)n2)=O)cc1 C(=O)(C(O)CC[S+](C)C)NC12CC(NC(c3nccc(OC)c3N)=O)(C1)C2 C(N=c1nc(N2C3CCC2CC(F)C3)c2c([nH]1)CCC2)c1ccc(Cl)c(Cl)c1 N1(C(c2c(CC)cccc2)=O)CC2CN(C(=O)C(C)OC3CCCC3)CC2(C)C1 C#CC1(C(=O)NC2CN(CC)CCO2)CCN(C(c2cccc(O)n2)=O)C1 c1(SC)ncc(Cl)c(C(N2CCN(C(c3cc4ncsc4[nH]3)=O)CC2C)=O)n1 N1(C(=O)NCC(C)(C)Oc2ccc(Br)cc2)C2CCC1C(N)C2 c1(N(S(C)(=O)=O)CCn2cc(C(C(N3CC(SC)C3)=O)=O)nn2)ccc(C)cc1 CCC(C)C(O)C(C)C(=O)N(C1(C(=O)NCCC(Cl)Cl)CCC1)C1CC1 N1(C(=O)Cc2cccnc2Cl)CCC2CCN(C(=O)C(n3cccn3)O)C2C1 C1(NC(N(CCC)Cc2cccc(Br)c2)=O)CC2CC3C(C2)C13 N1(C(C2(C)CN(C(CCn3ccc(C)n3)=O)C2)=O)CCC(F)(COC(C)C)CC1 C1(C(=O)NCC(CC(=O)NCc2cnns2)C2CCC2)CC2(CCO1)CC2 c1(C(=O)NCC2C(NC(c3ccc(N(C)CC)cc3)=O)C2)ccc2nncn2c1 c1(N(C)CC2CCN(C)C2)nc(N2CC3(C)COCC3(C)C2)nc2c1COCC2 C1(C(c2ccccc2)C)CN(C(=O)Cn2cc(C(=O)OC)nn2)CC1N(C)C.C(=O)O N1(C(C2C(CNC(CC=CCCCCC)=O)OCC2)=O)CCC(COC)C(C)C1 N1(C(C2C(C=C)C2)=O)CCN(C(c2ccn(CC)c(=O)c2)=O)C(CC)C1 C1(NC(c2c(C)n(C)c(C3CCCC3)c2)=O)CC(=O)N2CCCCC12 C1(CC)CN(C(c2sc(C(C)OC)nc2C)=O)CCC1NC(=O)CCF O=C(NNc1ncnc(Cl)c1CO)C1CCOC12CCOCC2 Cc1nc(Cl)ccc1S(=O)(=O)N(CC1CC1c1ccccc1)CC1COCCN1 S(=O)(=O)(c1ccc(N2CCCC(C(F)F)C2)c(F)c1)NCCCOCC(C)C C(=O)(CCCC(CC)NC(=O)CCOC(C)=O)N1CCC(OCC=C)C1 N1(C(C2N(C(c3ccc(C#N)[nH]3)=O)C(C3CC3)CC2)=O)CCC2C(C(N)=O)C2C1 N1(C(COCCN(C)C)=O)CCC(C=CC(=O)N(CC(F)F)CCO)CC1 Cc1ncnc(C(=O)NCCC2(C(=O)N(C)CC3CCCOC3)CCC2)c1C N1(C(C2ON=C(C)C2)=O)CCC(NC(c2cc(Br)no2)=O)C(C)(C)C1 CCCC(C(=O)NC(CCC)CC(=O)NCCN(CC(F)F)C)C(C)C c1(CC(C(=O)NCCCNC(C(C=C)O)=O)NC(=O)OC(C)(C)C)ccccc1Cl C(=O)(C(C)CC(C)C)NCCC1N(C(c2n(CC)ncc2)=O)CCSC1 C1(NC(c2c(CSC)cccn2)=O)CCCN(C(=O)CCC2CCN(C)C2)CC1 N1(C(C(C)=C(C)C)=O)CC(C)CCC1CNC(=O)Cc1cnn(C)c1C C(=O)(C(O)P(C)(C)=O)N(CCC)CCC.C(CC)NC(=O)COC(C)CC c1(N2CC(C)(CC(=O)Nc3c(OC)cc(Cl)nc3)C2)ncc2cn[nH]c2n1 C1(CNC(C2CCC2)=O)C2CC1N(C(=O)CCC1CCCC1)C2.O=C1C(CO)N1 Cn1cc(C(=O)NCCN(C(C2C3COCC23)=O)C2CC2)c(C(C)(F)F)n1 c1(C(=O)NC(CCCC)CNC(=O)CC2(C)CC(F)(F)C2)cc(O)nc(O)n1 Cc1nc2ccc(C(N3CC4CCCN(C(C5CC(C)CO5)=O)C4C3)=O)cc2o1 C1(CC(=O)NCC(CN(C(c2cnc(CCCC)s2)=O)C)(C)C)CCCCC1F c1(C2(C(=O)NCC3(F)CCN(C(=O)C(F)(F)CO)C3)CC2)ccc(F)c(Cl)c1 N1(C(C(=O)NC(C2(O)CN(C(C3N(C(C)=O)CCC3)=O)C2)C)C)CCCC(O)C1 c1(NCc2cccc(C(=O)OCC)c2)cc(-c2n[nH]c(C)n2)ccc1C c1(C(=O)NC(C2CCCN(C(C(C#C)(C)C)=O)C2)C)cccc(C)c1F CC1CCN(CCC(=O)NC(CCN(C(C2(C(F)(F)F)CC2)=O)C)=O)C1 C(CNC(=O)CC1(O)CCCOC1)(C(C)(C)C)NC(CN1CC(C)C1)=O C1(CNC(N(C(c2c(C)cccn2)C)C)=O)COc2ccccc2O1 C1(OC)CC2CC1CN(c1nnc(-c3ccc(F)c(F)c3)s1)C2 C(=O)(C1CCCc2n[nH]cc21)N1C(CNC(c2ccc(C(C)C)cc2F)=O)CC1 CC1c2ccccc2CC1C(=O)NC1(C)CN(C(=O)Cc2cc[nH]c2)C1 C1(CC(N2C(CNC(C=C(COC)C)=O)CCC2)=O)Sc2ccccc2NC1=O N1(C(C(CC(=C)C)C)=O)CC(NC(=O)Cc2ccccc2Cl)CC2(CC2)C1 c1(CCC)cc(C(=O)N(CC(C)NC(=O)C(c2cccnc2C)C)C)ccn1 CCC(C(=O)N1CCCC1CC(=O)NCc1cnc(C)[nH]1)N(C)C c1(OC)ccnc(C(=O)NCC(C)CC(=O)N2CCC2CO)c1 CC#CC1CCN(C(C2CCCN(C(=O)CCC(=O)NC)C2)=O)C1 N1(C(C(CCC(C)C)F)=O)CCCC2C1CCCN2C(=O)CCN1CCCC1 CC1=C(C(=O)N2CC(F)(C(=O)NCC3CCOC3)C2)CCC1 n1(CC(=O)N(C2CCN(C(C3CCC(F)(F)C3)=O)C2)C)ccc2ccc(F)cc12 c1(C(N2CC3CC(CN(C(C(CC)F)=O)C3)C2)=O)nc(C2CC2)n2ccccc12 C1(C(=O)NCC2CCCN(C)C2)CN(C(=O)C(O)CN2CCCC2)CC12CCC2 C12(C(C)C)CCC(NC(=O)NC(C)(Cc3ccccc3)C(F)F)C1C2 CCCCCC(=O)NCC(=O)NC(CNC(C1CC1C(F)F)=O)CC(C)C N1(C(CC(CC)NC(=O)C2=NOC3COCC23)=O)CCC2(CCN(C)C2)C1 CC(O)(CC(=O)N1CC2=C(C1)CN(C(=O)COCCCN=[N+]=[N-])C2)C(F)(F)F N1(C(C(C)S(C)(=O)=O)=O)C2CCC1CC(O)(CNC(=O)CCCNC(N)=O)C2 c1(C(=O)NC2CCN(C(C3C(CC)N(C)CC3)=O)C2)cc(O)nc2cnccc12 Cc1cc(N)cc(C(N2CCCC2CNC(=O)C(C)(C)c2cnco2)=O)c1F C1(CCNC(C(C)(C)C2CCC2)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1 C1(CNC(c2nc(NC(C)=O)sc2)=O)COCCN(C(=O)C#CC(C)C)C1 Fc1ccc(Br)c(-n2nnnc2N2CCN(CC3C4CCCCC4CN3)CC2)c1 c1(CN(C2CCCN(C(c3ccn(CCOCC)n3)=O)C2)C)ccc(F)nc1C C1(C(N2C(COC)C(C)(C)C2)=O)CNC(=O)CN1C(=O)Cc1cncn1C c1(C(N2C(C)CC(NC(=O)CC3CCC(=O)N3)C2)=O)ccn2nncc2c1 N1(C(C(C2CC2)OCC)=O)CC(CC)CC1C(=O)NCC(=O)N(C)OC C1(CCNC(c2cn(C(F)(F)F)cn2)=O)CCCN1C(=O)CNc1ccccn1 C(=O)(C1CCc2sc(NC(=O)NC3CCC(S(=O)(=O)NCC)CC3)nc21)OCC CC(C)C(N=[N+]=[N-])C(=O)NCC1COC(CNC(=O)CCc2cncs2)C1 C1(NC(=O)Cc2ccsc2Cl)CCC12CN(C(c1cccn(C3CC3)c1=O)=O)C2 c1(C(N2CC(CC(C)NC(C(CCOC)(C)C)=O)C2)=O)cc(C)c(F)cc1Cl c1(OCCC(=O)NC(CC)(CNC(C2(O)CCCC2)=O)CC)cc(Cl)ccc1Cl N1(C(c2cc(C)[nH]n2)=O)CCC2CN(Cc3c(Cl)ccnc3Cl)CC12 Cc1cc(C(=O)C(=O)NCC2CCC(F)C2)c(C)o1 N1(C(C2C(C(=O)OC)CC2)=O)CCC2CCCC12C(=O)NC(C)CN=[N+]=[N-] C(=O)(CC(C(F)F)NC(=O)CCC(N)=O)N1CCC(NC(C)=O)CC1 c1(-c2ccc(C(=O)NCCN(CC(F)(F)F)C)o2)ccc(F)c(F)c1 c1(C(N2CCC(N(C(c3csc(CC(C)C)n3)=O)CC)C2)=O)ccc(F)nc1F c1(CC)c(C(=O)NCCCOCCNC(C2CCCO2)=O)oc2ccccc12 C1(C(N2CC(=C(CNC(c3cccc(C4CC4)n3)=O)F)C2)=O)CC(=O)CC2CC12 C1(C(=O)NCC(C)(C)OCCO)CCN(C(C2CC2Cl)=O)C1 C(c1cccc(Cl)c1)=CC(=O)NC1(CO)CN(c2nc(C3CC3)ns2)C1 C12CCC(CC1)n1cc(nn1)C(C)(C)NC2=O.c1(CC)ncoc1C(=O)N(C)C c1(OCC)ccc(CNC23CC2CN(C(c2cc(Cl)nc(Cl)c2)=O)C3)cc1Br C1(NC(c2ccccn2)=O)CN(C(=O)Cn2cncn2)CC1C1CCCC1 Cc1nn2ccccc2c1C(=O)NCC1(F)CC(NC(=O)C(C)(C)C(C)C)C1 c1(C(N(C2CC2)Cc2ccc(OC(C)=O)cc2)=O)cc(C)nc(Cl)c1 C(=O)(C(C)C(=O)N1CCOCC1c1ccc(C(=O)NCCC2(C)CC2)n1C)OC C(=O)(CC(C)CC(=O)NC(CC1CC1)C(=O)Nc1cccc(F)c1)OC C1(CC(=O)N(C2CCN(C(C=CC=CC)=O)C2)CCC)SC2=NCCN2C1=O C(=O)(CCCn1cc(CCCO)nn1)N(C(C)(C)C)NC(=N)N c1(CNC(C2(C)CC=C(C)CC2)=O)nc2c(s1)CN(C(c1ccoc1)=O)CC2 N1(C(C2(C(F)F)CC(=C)C2)=O)CC2C(NC(c3cnc(C)[nH]3)=O)C2C1 C1(NC(C(c2cccc(C)c2)C)=O)CCC(C)N(Cc2cc(C)on2)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CCC(CNC(CCC=C)=O)C(F)(F)C1 c1(C(=O)NCC2(F)CN(C(C34CCC(CC3)CO4)=O)C2)cc2ccc(Cl)cc2o1 N1(C(CCCN(CCC)CCC)=O)CC2(CC(NC(C3CCN(C)C3C)=O)C2)C1 C1(C(=O)NC(CNC(C2(C(C)C)CCC2)=O)(C)CO)CS(=O)(=O)CC(=O)N1 CC(C)(C)C(=O)C(=O)NCC1CCCN1C(C1(Cl)CC12CCC2)=O C1(CCOC)(C(N2CCC(O)(CCNC(=O)C(C)(C)CF)C2)=O)CCN(C)CC1 S(=O)(=O)(c1ccc(Br)cc1)NC1C(C)(C)CN(S(=O)(=O)CC2CCC2)CC1 N1(C(CC(C)C2CC2)=O)CCC2(CCN(C(=O)CC(C)(C)C)CC2)C1 N1(C(CC2(COC)CC2)=O)CC2C3CCC(C2C1)N(C(=O)C(C)(O)C1CC1)C3 CCC(C)(C)CC(C(=O)NCCCF)N1CCOC(CN=[N+]=[N-])C1 C=CC1(CC(=O)OC2(OC)CCC2)CCC1 C1(C(N2CC(NC(C(C)(C)N(C)C)=O)C(F)CC2)=O)Cc2ccccc2S1 S(=O)(=O)(c1nc2c(s1)CCCC2)NC(C1(C2CC2)CC1)=O C(=O)(C(C)N(OC)C(=O)C1COCCC1NC(C12CC(F)(C1)C2)=O)OC C=CCC(C(=O)N(C)CCN(C)Cc1nnc(C)n1CC=C)NC(C)=O c1(C(N2CCN(Cc3ccc(C)o3)CC2CC#N)=O)cccc2ccnn12 C(CNC(=O)C(C(C)OC)NC(c1c(C)csc1C)=O)(CC(C)C)OC c1(C(=O)NCC2CCC(C(=O)NC(CC(CC)C)C)O2)cc2cccn2cn1 CC(C)C(=O)NC(=O)CNC(CC(CO)NC(N1CCCC1)=O)=O N1(C(c2cc(C)cc(Br)c2)C(=O)NC(C(=O)OC)C)CCc2ccc(F)cc21 N1(Cc2n(CC(F)F)ncc2)CCC(F)(F)CC12CCC2 N1(C(C(C)OCC=C)=O)CCC(C)(C)CC1C(=O)Nc1cnc(CO)nc1C C1(C(N2CCN(C(c3cc(O)cs3)=O)CC2)=O)CC12CCC(F)(F)CC2 CC(C)(O)C(O)C(C)(C)C(=O)NC1CC2(CCC2)CN1 c1(C(C)=O)ccc(CC(=O)NCCC(C)(C)NC(=O)C(=Cc2ccco2)C)cn1 CCCCCCC(C)C(=O)NC12CCC(C(=O)NCCCn3cnnc3)(CC1)C2 C12(NC(C(CCCC)F)=O)CCCC1N(C(c1cnn(C3CC3)c1)=O)CC2 C=Cc1ccc(C(N2CCC(CNC(c3cc[nH]c(=N)n3)=O)C(O)C2)=O)cc1 N1(C(C2(C)CCCS2(=O)=O)=O)C2CCC1CC(CN=c1ncc(F)c[nH]1)C2 Cc1ccc(Br)c(CN2CCC(F)(C(=O)NC(C#N)C(N)=O)C2)c1 CC1CCCC(C(=O)NCCC2(C(=O)NC3CCCCC3CCO)CC2)O1 C1(C(N(CC(C)NC(c2nccc(C)n2)=O)C)=O)CC(C2CCC2)C1 C1(NC(CCCOC(C)C)=O)C2CCC1N(C(=O)CC1CCCCN1C)C2 c1(CNC(=O)C(O)Cc2ccccn2)cccc(NC(C2CCC3(CC3)C2)=O)c1 C(CCNC(C1COCC1C(F)(F)F)=O)(CNC(=O)C(=O)N(C)C)OC CCC1=NOC(C(=O)NC2(C)CC(NC(c3cc(C)c(C)[nH]3)=O)C2)C1 c1(CC)ccc(C(C)=CC(=O)NCCN(C(=O)C(=O)NC2CC2)CC2CC2)cc1 C1(CCOC)(NC(=O)C(C)NC(C2CCC2)=O)CCN(C(c2csc(C)c2)=O)C1 C1(Cc2cc(NC(C3(c4oncc4C)CC3)=O)no2)CCCC(NC(=O)NC)C1 c1(CNC(C(c2nc[nH]n2)N(CCC)C)=O)nncn1CC1CC1.OC Cc1cnccc1N1CCN(C(=O)NC(c2ccc(Br)cn2)C(F)(F)F)CC1 CC(CC(=O)N1CC(S(C)(=N)=O)C1)CC(C)(C)C.C12(CCCCC1)C(=O)NC2 c1(C(=O)NC2C(CNC(C(C)CS(C)=O)=O)CCC2)ccc(F)c(O)c1F C(=O)(C(C)(O)CC(C)C)NC1CCN(c2nnc(-c3cnc(C)s3)o2)CC1 c1(C(=O)NCC(CC(=O)OCC)C)cc(I)ccc1O Cn1nnc2c1CC(C(=O)NCC1(O)CCCN(C(C34CC(C3)C4)=O)CC1)CC2 CC1CC(c2ccccc2F)C(C)CN1CC(=O)Nc1ccco1 C(N=c1[nH]c(=NCC(C)OC2CCCCC2)[nH]c2c1COC2)C1C(CCC)C1 C1(F)(C(=O)NC(C2CC(NC(C3CCC(C)CC3)=O)C2)C)CCCN(C)C1 CCS(=O)(=O)N(CC(=O)N(CCNC(=O)COC(F)(F)F)CCOC)C C(=O)(CCCS(C)(=O)=O)N1CC(N(C(C2CC=C(C)CC2)=O)C)C2(C1)CC2 c1(CC)cnccc1C(=O)NCC(C)CN(C)C(c1nc(Br)c[nH]1)=O C(=O)(C(CC(F)F)NC(C1C=CCC1)=O)NCC(C)(O)CO C(=O)(CC(C)n1cccn1)NC(C(=O)NCCC(=O)N(CC)CC)c1cccs1 C1(C(=O)NCC(CCOC)NC(=O)CC2CN(C)C2)CC(C)CC(C)C1 c1(C(N2CCN(C(=O)Cn3ccnn3)C(C(F)F)C2)=O)cnc2ncccc2c1 c1(OC(C)C(=O)N(c2ccc(I)cc2)C(C)(C)C)ccc(Cl)c(F)c1 C#CCC(CC(F)F)NC(C1(F)CN(C(=O)C(C)(O)CCC)C1)=O n1(CC(=O)NC2CCC(NC(CN3C(C)CC3)=O)CC2)cc(C#N)c(O)nc1=O Cc1cc(=NCC2(S(=O)(=O)NC(C)(C)C)CC2)[nH]c(=NCC2OCCC2C)[nH]1 N1(C(Cc2cnc(C)s2)=O)CCC12CN(C(=O)C(C1CCS(=O)(=O)CC1)(C)C)C2 C1(C(=O)NC(C)(CNC(c2ccc(CO)nc2)=O)CO)CCc2nc(O)[nH]c2C1 c1(C(=O)NC(C(C)C)CNC(C2CCOC2=O)=O)cc(F)c2[nH]nnc2c1 C1(CNC(c2ccc(CC(F)F)cc2)=O)COCCN(C(=O)CC2CCCC2)C1 C1(NC(c2ccn(C(F)F)n2)=O)CCOCC1NC(C1CC(CF)C1)=O CC(C)C(=O)C(=O)N1CC2C(NC(=O)C(C)Oc3ccc(Br)cc3)C2C1 C=C1CCN(C(c2ccsc2)=O)C(C(=O)NCC2CC(O)C(O)C2)C1 c1(CN(C2CCN(CC)CC2)CCO)ccc(S(C)=O)cc1.C12CCN(C1)C2=O c1(NCC(=O)NCC2CCC(NC(=O)COC3CC=CC3)C2)ccc(F)c(F)c1 c1(C(=O)NCC2(F)CC(NC(CCOCCOC)=O)C2)nccc2c1CNC2=O C1(CNC(c2n[nH]c(C)c2O)=O)CN(C(=O)C(C)N2CCC2)CCC1(C)C C(CC(F)(F)F)N(C(C)C(=O)NC1CC1CNC(=O)CSc1ccccc1)C CC1CN(C)CCCN1C(C1CC2CC1CN(C(C1SCCS1)=O)C2)=O C1(C(=O)NCCN(C2CC(C#N)C2)C(C2CC(F)(F)C2)=O)CCC(C(F)F)CC1 C1(NC(C2CCSC2)=O)CC(C(=O)NCC2(CO)CCC2)CC1O C1(C(=O)NCc2c(C)ncs2)(NC(=O)CC23CCCC2C3)CCN(C)C1 N1(C(=O)CCCSC2CC2)CCN(C(C2CC=CC2)=O)C2CCCCC2C1 C(=O)(C1CCCc2ncnn21)NC1C(CNC(=O)CCn2cccnc2=O)CC1 N1(C(C2CCN(CC)C2)=O)CC(C)C(C)(CNC(c2[nH]cc(C)c2C)=O)C1 C1(NC(C2C(CC)C2)=O)CCN(C(c2cc(C)c(O)c(Cl)c2)=O)CC(C)(C)C1 C1(NCCC2(C)CCNC2)C=CC2(CCCCCC2)CC1 Cc1ccccc1-c1cnc(CN2CCC(NC(c3cn(C4CC4)nn3)=O)C2)o1 C1(C(=O)NC2C3CCN(C(=O)CCc4cnccn4)C23)COCC2(CCC2)O1 c1(C(=O)NCC#CCNC(C(=Cc2cccs2)C)=O)c(Cl)cccc1[N+](=O)[O-] C1(CC(N2CCC(CCNC(CCCN=[N+]=[N-])=O)CC2)=O)CCn2cncc2C1 c1(C(N(C(C)C(=O)NCCC2CCC(C)O2)C)=O)cccc(CO)c1 Cc1c(Cl)cc(Cn2ccccc2=O)c(Cl)c1C.C1(C(=O)O)(CN)CCC(C)(C)C1 Cc1cc(Cl)c(C(=O)NC2CC(C)CN(C(=O)CSC3CCOC3=O)C2)cc1C N1(C(c2cc(CCC)nn2C)=O)CCN(C(C2(CC)CCCC2)=O)CCC1C CC(=O)CCCC(=O)N1CCC(C)CC1CNC(c1cc(F)n[nH]1)=O Cc1cccc2c1C(C)CC2CNc1c(F)cc(Br)cc1F N1(C(CCN(CC)CC)=O)CC(NC(c2c[nH]c(Br)c2)=O)C2CC12 c1(C(=O)NC(CC)CNC(=O)C(C)OCC2CC2)cccc(CC(C)C)c1 n1(C(C2CCCCC2)C)nc(-c2cccs2)nc1-c1ccon1 CC1CN(C(C2(C)CC3CCC2C3)=O)CCC1NC(C1(C#N)CC1)=O C1(C)(CC(=O)OC2CCC(OC)CC2)Oc2ccccc2O1 N12CC3CC(C3)(C1)CNC2=O.C1(C)(OC)CN(Cc2ccccc2)C1C1CC1 Cc1cc(F)c(C(N2C(C(=O)Nc3cnn4cccnc34)CCC2C)=O)c(F)c1 C1(NC(C(CCC)F)=O)CCCN(C(c2cccc(F)c2N)=O)C1C c1(Sc2nnc(S)s2)ccnc2cc(Cl)ccc12.C12CCN(C1)C(=O)CNC2=O c1(-n2ncc(CN3CC(O)(c4nnc(C)o4)C3)c2)cccc(Cl)c1 c1(C(CNC(C2(CC3CC3)CC2)=O)NC(c2cc(Cl)cs2)=O)ccc(F)cc1 N1(C(CC(N)Cc2csc3ccccc23)=O)CC2(CCC2)CCC1CO C(=O)(C(C)(C)C(O)C(C)C)NC1CC=C(C(=O)NC2C(CC=C)CCC2)C1 C(=O)(C(C)(C)CC(=O)OCC)NC1CC(=C)CN1Cc1cc(C)cc(OC)c1C(N)=O N#Cc1ccc(C2CCN(CC3(C(F)(F)F)CC3)C2)s1.c12ccc(cc1)s2 c1(C(N(C2CCN(C(c3cc(C(N)=O)cs3)=O)C2)C)=O)c[nH]c2ncnc(O)c12 C1(CNC(C(C=C)(C)O)=O)CC(C)(C)CN1C(=O)C(c1ccc(Cl)cc1)C c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CS(=O)(=O)C2)cccc2c1oc(=O)n2C C1(NC(c2c(C)noc2)=O)CCCCN(C(C2CCC2)=O)C1 N1(C(c2nnc(C)s2)=O)CCOC(CNC(c2c(C)nsc2Br)=O)C1 Cc1sc(C(=O)N(C2(Cc3cc(C(F)(F)F)nc(C)n3)CCC2)C2CC2)c(C)c1C c1(CNCCC)ccc(C)c(O)c1.C1C(O)CN(C)CC(=O)N1C n1(CC)cccc1C(=O)NCC1(F)CC(NC(C2CC(=C3CC3)C2)=O)C1 CC(C)CC(C(=O)NCC(CNC(=O)CCCN(C)C(C)C)CO)C(N)=O N1(C(CN(C(C)=O)C)=O)CCC2CCN(C(=O)CCc3nc(C(C)C)no3)CC12 c1(SCC(=O)OCC(CCCC)OC)c(C(C)=O)oc2ccccc12 CC1OC2(C)CC1(C(=O)NC13CCC1CN(C(c1ccc(N)c(Cl)c1)=O)C3)C2 c1(SCC)cccc(CC(=O)NC(C)Cn2cc(Cn3cc(Cl)cn3)nn2)c1 N1(c2nnc(COCC)n2CC2(OC)CCC2)CCC2C(C1)C2(F)F.C1(C)CC1 C(=O)(C1=NOC2COCC12)N1C2C(NC(c3c(CC)[nH]cc3)=O)CC(C2)C1 C1(NC(c2cnc(CC)o2)=O)CC(NC(C23CCC(CC2)C3)=O)C(O)C1 C1(C(=O)OCC)CCC2(CC(C(=O)OC)C2)N(CC)C1.c12cnc(O)c(c1)NC2 C1(C(N2CC(C)CC(CC)C2)=O)CC2(CCN(C(=O)CCCCC(C)C)C2)C1 N1(C(CCSCC(N)=O)=O)CCCN(C(c2cnc3nccn3c2)=O)CCC1 c1(C(N2CC(C(Cn3cc(C(CCCC)CC)nn3)F)C2)=O)ccc(F)cc1N c1(C(=O)NCCOC2CCN(C(c3c(CC)nc[nH]3)=O)C2)ccc(C)nc1O C1(CC)C(C(=O)NCc2c[nH]nc2C2CC2)CCCN1C(c1c[nH]c(=O)cn1)=O CC1=C(C(=O)NCC2CCN2C(C2CC3(C2)OCCO3)=O)COCC1 N1(C(C2C(C)(C)N(C(=O)C(F)CC3CCOC3)CC2)=O)CCc2cccc(O)c21 O=S(=O)(c1cccc(N2CCC(CCO)CC2)n1)NCC1CC12CC2 C1(O)(C(C)NC(C=CCCC)=O)CCN(C(=O)CC2CCC(C)CO2)CC1 Cc1cc(C(=O)NC(C(N2CC3(CCCO3)C2)=O)C2CC2)ncc1N C1(C(F)(F)F)(N(C(=O)OC)C)CCCN(S(=O)(=O)N=S(C)(C)=O)C1 c1(C(=O)NC2CN(C(C3N(C)CC(O)CC3)=O)CC23CC3)ccnc2c1CCO2 C(=O)(C(C)CC(C)C)N(CC(C)NC(C1CC(OC)C1)=O)CC C(C)(C)(C(C)NC(=O)CCc1nc(C2CC2)no1)NC(C(=O)NCCOC)=O C(=O)(C1CC(C)(C)Oc2ccccc21)NC1(C)CN(C(C(COC)OC)=O)C1 c1(C(=O)NC23CCN(C(c4c(C)nc[nH]4)=O)CC2C3)cc2c(o1)CCCNC2=O c1(C(=O)O)ccc(CNC2CCC(N3CCOCC3)C2)cc1 C1(C(=O)NC(C)CSC(F)F)CCCCCC1NC(c1cc(O)nc(O)n1)=O C(=O)(CCCC(F)(F)CO)N(C1CCCN(C(=O)CC2CCC(C)CO2)C1)CC c1(OC)nc(C)c(Br)cc1C(C(=O)NCC(C)C)N(C)CC1CCCC(F)(F)C1 c1(C(N2C(CCC(=O)NC3CC(O)C3)CCC2)=O)cc(F)c([N+](=O)[O-])cc1F c1(OC)ccccc1CCN(C1CC(OC)CC(Nc2ccc(C(F)(F)F)o2)C1)C=O c1(C(N2CCC(NC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)c(Cl)nn(C)c1Cl C1(NC(c2ccn(CC)n2)=O)CC2CC(C1)N(CC(N1CC(C)CC(C)C1)=O)C2 c1(C(N2C(CCNC(=O)COC(F)(F)F)CCCC2)=O)c(F)ccc2n[nH]cc12 N1(C(C2CC(C#N)C2)=O)CC(F)(F)CC1CCNC(=O)CC1C=CCC1 c1(CC)c[nH]c(C(=O)NC(C2CC=CCC2)C(=O)NCC(=O)N(C)C)c1 N1(C(CC(C=C)C)=O)CCC2(CC2NC(c2cnn(C3CCC3)c2)=O)C1 c1(OC)ccccc1C(CNC(C1CC1CF)=O)NC(=O)Cc1nc(C)sc1C c1(OC)cc(CNc2ccc(C(=O)Nc3cncs3)nc2)ccc1C c1(C(C)(F)F)ccc(Cl)c(C(=O)NC(CC2(O)CCC2)C(F)F)c1 C(CC(C)(C)C(=O)N1CCC(N(C)C)C(C)C1)NC(CC1C(C)OCC1)=O N1(C(N(C)C)=O)CCCC(C(N2CC3CC2C3NC(=O)C(C)(C)N(C)C)=O)C1 Cc1cc(S(=O)(=O)N2CC(C)(C)OC(C)(C)C2)ccc1-c1cccnc1 C#Cc1ccc(C(=O)NCC2CCN2C(=O)C(C)N(C)C(C)=O)cc1 N1(C(Cn2ccc(C)n2)=O)CCC2(CCN(C(c3cnc(N)c(Cl)c3)=O)CC2)C1 c1(C(N(C2CC(NC(C3C(=C)CC3)=O)C2)C)=O)cc(Cl)cs1 Cn1ccc(C(N2CCC2CNC(c2cn(CCO)nn2)=O)=O)cc1=O N1(CCNC(C2CC(CNC(CC3CC(=C)C3)=O)OC2)=O)CCCC(O)C1 c1(C(C(=O)N(C(CNC(C2(C(=O)NC)CC2)=O)(C)CO)CC)C)ccccc1C c1(C(=O)NCc2nc(-c3cccc4c3COC4=O)no2)ccc2c(c1)C(=O)NCC2 C1(C2CN(C(C3CC3Cl)=O)C2)(NC(C2CCCCC2)=O)CC1 C1(C(N2C(CN(C(=O)CN3CCCCC3)C)COCC2)=O)CCn2nncc2C1 CCCC(C(=O)OC)C(=O)NC1(CC)CCCN(Cc2ccc(C)nn2)C1 c1(C(C)(C)C)cccc2c1CCN2C(c1cccc(-c2cc(Cl)ccc2Cl)c1)=O c1(N(C(=O)CN2CCCC2)C=O)cccc(F)c1N.C(=O)(OC)OC c1(CCC(=O)NCC2CC2CNC(=O)CSCC(C)C)cc(SC)c(C)o1 c1(C(=O)NC(CC)CNC(=O)CC2CCC(=O)N2C)cc(C)c(O)c(C)c1 C(CCC)(CC(=O)NC(C)CC(C)C(F)F)NC(CCC)=O N1(C(CCCN(C(C)C)C)=O)CCN(C)CC1C(=O)NC1CN(C(N)=O)C1 N1(C(CC(CCN)O)=O)CC(NC(=O)CN2CCCC2)CC12CCC2.C(C=O)SC c1(C(=O)NCCC(=O)NCc2c(C(C)C)ocn2)cnn(C)c1N c1(C(N2CC(O)CC(NC(C3CC4(CSC4)C3)=O)C2)=O)c(Cl)ccc2ccoc12 C=CCCC(C)(C)C(=O)NC(C)CC(C)NC(C1(c2cc[nH]n2)CC1)=O N1(C(Cc2ccc(CC(C)C)cc2)=O)Cc2[nH][nH]c(=NC(=O)c3cnco3)c2C1 c1(NC(=O)COCC2CCC2)cccc(CN(C(COCCOC)=O)C)c1 N1(C(=O)NCCOC2CCS(=O)(=O)C2)CC2CCCN2Cc2ccccc21 Cc1cc(Cl)c(C(=O)NC2CN(C(=O)C(F)CC3CCC3)CC2O)cc1C C1(C=O)CCCN(CC#N)C1.C1(N(C(C=CCC)=O)CCCC(F)(F)F)CCCC1 Cc1cc(C(=O)NCCC(O)C(=O)NCC2(C)CC=CCC2)c(C)cn1 CC1NC(=O)CCC1CNC(=O)C(O)CNC(C1(F)CC=CCC1)=O CC1OCCC1C(N1CCC(C(=O)NC2(CCF)CCC2)C1)=O C(C(C)(CC(=O)O)NC(=O)C(C(C)C)OCc1cccs1)OC c1(C(=O)NCCC2CC(C(=O)NC(CSC)(C)CO)C2)nc(C)ccc1C C#CCCCCS(C)(=O)=NC(=O)C(=O)C1CC(C)(C)CC(C)(C)C1 CC1CCN(C(c2cnc(S)n2C2CC2)=O)CC1NC(=O)C=Cc1cccnc1 C1(C(=O)NC2CON(CC)C2=O)CN(C(=O)CC(C)OC)CCC1(C)C C1(C(=O)NCC2C(NC(C(CCC)OC)=O)C2)CCC(N=[N+]=[N-])CC1 c1(C(c2n(CCOC)nnn2)NC(C(N)=O)C2CC2)ccccc1C(C)(F)F Cc1ccc(-c2cc(C)n(CC(=O)NCc3cc(-c4ccco4)[nH]n3)n2)cc1 c1(-c2cc(C(=O)NC3C(NC(C(CSC)O)=O)C3)on2)ccc(Cl)cc1 N1(C(c2cn(CC)nc2C2CC2)=O)CCC2C(CCN2C(=O)C(F)C2CC2)C1 S(=O)(=O)(c1c(F)ccc(C)c1F)Nc1sc(CCC)c(-c2nn[nH]n2)c1 CC(C)C(C(=O)N(CCCNC(c1ccc(C(F)F)cc1)=O)C)NC(N)=O C1(CN(C=O)Cc2cccc(OC(F)F)n2)CC2OCCC2O1 c1(C(=O)NC(C2CC3CCC2C3)C#N)cc(C(=O)O)c(Br)cn1 c1(C(N(C2CCN(C(c3nc(CCC)oc3)=O)C2)COC)=O)nnn2c1CCC2 N1(C(c2c(F)ccc(OC)c2)=O)CCCCC(NC(=O)CC(C)SC)CC1 c1(CCC2CCCN(NC(C(N3CCCCCC3)C)=O)C2)nnn2c1CCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CC23CCCC2(C1)CN(C(=O)CSC(F)(F)F)C3 C(=O)(CC(C)(C)C(F)F)N1CC(C)C(CNC(=O)CSc2nnc(S)s2)CC1 C1(SCC)CCC(C(=O)N(CCNC(C2(C)CC3CC3C2)=O)CC)CC1 Cc1cccc2nc(CCC(=O)NC3(C)CCN(C(=O)CCCC4CC4)C3)[nH]c12 Cc1nn(C)c2cc(C(=O)NCc3cn(-c4cnc5c(c4)CC(=O)N5)nn3)ccc12 C1(COC)(CNC(c2n[nH]c(C)c2C)=O)CCCN1C(c1[nH]cnc1C)=O Cc1cc2[nH]c(C(=O)NC3C4CC3CN(C(c3ccc(F)cc3Cl)=O)C4)cc2o1 C=CC1OCCCC1C(=O)NCC1CCN(C(=O)C=C(C)Cl)C(C)C1 CCC(CCC(=O)NC(C)CC(C)O)NC(c1cccc(OC)c1)=O c1(SC)nc(N2CCC(NC(C3(C)CCCS3(=O)=O)=O)C(C)C2)cc(Cl)n1 C(CC(=O)NC1CC1c1cncs1)(CC(C)C)NC(c1c(C)nncc1)=O C(c1ccccc1C)=CC(N1CC(CC)C(C(N2CC(C3CC3)C2C2CC2)=O)C1)=O c1(OC)ccc(CCCNC(Cc2ccccc2)C(C)C)cc1O C=CCC(C)C(=O)NCCCC1(NC(=O)CCc2nc(-c3nc[nH]n3)no2)CC1 c1(C(N2CCC(C3N(C(C(N4CCCCCC4)C)=O)CCC3)C2)=O)cncc(N)n1 CC(C)(C(=O)N1CC2(CCN(C(c3coc(CS(C)(=O)=O)n3)=O)C2)C1)S(C)(=O)=O c1(C(=O)NC(CNC(C(C)NS(C)(=O)=O)=O)(C)C)ncc(F)cc1N c1(CC(=O)N(CCCCN(C(=O)C(O)CF)C)C)ccn2cncc2c1 C1(CNC(c2cnc(CC)s2)=O)CCN(C(C2CC2c2cccnc2)=O)CC1C C=C1CC(C)(C(=O)NCC2OCCC2C(=O)NCc2nc(C(C)C)n[nH]2)C1 Cc1csc(CCC2CC2NC(N2CCC(Cc3cccs3)C2)=O)n1 c1(C(C(=O)NC2C(NC(C(CSC)(C)C)=O)C2)C)ccc(F)c(Cl)c1 Cc1nc(C)n(CCCC(=O)NCCC(C)NC(=O)C=CC(=O)N(C)C)n1 c1(SC(C(=O)NCC#C)CCF)cc(C)nc(C)c1.C12(CC1)C(=O)N2 BrC1=CC=CCC2C3(CCOC1CNCCC2)CC3 C1(COC)CC(C)CN(C(C2CS(=O)C2)=O)C1 c1(OC)cc(C(=O)N(C)CC2CCCN2C(C2CC2C(N)=O)=O)c(Cl)cn1 CC(C)(O)C(C)(O)CNC1CC(c2ccccc2)CN1 CC(F)(F)C(C)(C)CC(=O)N1CCC2CC1CN(C(c1ccc(Cl)c(F)c1)=O)C2 N1(C(c2n(C)ccn2)=O)CCOC2(CCN(C(C3CCC(C(N)=O)CC3)=O)C2)C1 Cc1c(C(N2CCC(CNC(=O)CSC(C)C)CC2)=O)ncn1C C1(CC)CN(C(c2ccc(OC)nc2Cl)=O)CCN1c1ncccn1 CC1CCCCC1CC(N1CCC(C)(NC(N)=O)C1)=O.c12cn(nn1)C1CC23CC13 c1(OC)cc(C(=O)NCC2CN(C(c3cnc(C)[nH]c3=N)=O)C2)ccc1[N+](=O)[O-] c1(C(C(=O)NCC(=C)C)N(C(C)C)C2CC2)cncn1C C(=O)(C1CCCc2ccccc21)NC(C(C)NC(CCCOC(C)C)=O)CO CC(C)(CNC(C1CCCO1)=O)CCNC(c1ncoc1C1CC1)=O C#CCC(C(=O)NC(CCF)C(=O)NC(c1ncc(C)cn1)C)C1CC1 c1(C(=O)NC(CC)(C)CNC(C2CC2C(C)(F)F)=O)cncc(C#N)c1 C12(NC(c3c(C)cc(F)cc3)=O)CCCN(C(c3ccsc3C#N)=O)CC1C2 C(=O)(C(CCCCC)C(C)C)NCC1CCC(CN(C(C(CC#C)O)=O)C)CC1 c1(CC)ncc(C(=O)N(C2CCC(NC(c3nc(O)sc3C)=O)CC2)C)c(O)n1 C(N=c1[nH]cnc(Cl)c1OC)C1CCCC(NC(CC(C)SC)=O)C1 c1(C(N2C3CN(C(c4c(C)cn(C)c4)=O)C(C3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(C)(CCNC(C2(NC(=O)OC)CCCC2)=O)CCN(C(c2cnn(C)n2)=O)C1 c1(C(N2CC(C(C)NC(C(C)OCC)=O)C2)=O)cc(C#N)c(F)cc1F C1(NC(C=CSC)=O)(CNC(=O)CCC2CCCC(O)C2)CCCCC1 C1(OC)CCCCC1NC(c1cc(CN=C(NCc2ccco2)NC)c(C)o1)=O C1(C)(C(NOCCC=C)=O)CCCN(C(C2CC(=O)OC2(C)C)=O)CC1 N(C(=NCCc1ccsc1)NCCSC)C.Cn1nc(C(F)(F)F)cc1C1CCCC1 C(=O)(CC(C)C(F)(F)F)N1CCC(OCCNC(C2(COC)C=CCC2)=O)C1 CCCC(O)C(CO)NC(=O)C1=CCN(C(c2n[nH]c(C)c2C)=O)C1 N1(C(Cc2nn(C)c(Cl)c2)=O)CC(NC(=O)CCS(C)=O)C2CCCCC12 N1(C(c2c(CC)n(C)cc2)=O)CC2CCCC1CN(C(=O)Cn1cnnn1)C2 C1(NC(c2ncc[nH]2)=O)CC2(CCN(C(C3C4CCCCCCC34)=O)C2)C1 N1(C(c2ccn(C)c2CC(=O)O)=O)CCn2cc(C(=O)NC3CCOC3)nc2C1 N1(C(C2(CCC)CCCC2)=O)CC2(C)CN(C(C3(NC(N)=O)CC3)=O)CC2(C)C1 N1(C(C2CCC3(CCC3)O2)=O)CCC2(C1)CN(C(C1(c3cc[nH]n3)CCC1)=O)C2 N1(C(CC=CCC)=O)CCC(CNC(c2ccn3ncnc3c2)=O)C12CCC2 N1(C(c2cc(Cl)ns2)=O)CCC2(C1)CN(C(=O)CCc1ccc[nH]1)C2 C1(NC(=O)Cc2cc(Cl)cs2)CC2CCC1(NC(=O)CC1(O)CCCC1)C2 N1(C(C(=O)Nc2cn(CC)nc2)C)CCC(N(C(=O)COCC(=O)OC)C)CC1 C1(CNC(c2nccc(C)n2)=O)COCCN(C(=O)C(C)C2CCC2)C1 c1(CC(=O)NC2CC3CC2N(C(c2ccco2)=O)C3)ccc(Br)cc1F Cc1ccc(CC(=O)N(C)CC2C3CN(C(=O)C(C)(C)CO)CC23)cc1Br CCC(CCC(=O)N1CC(C(F)Cn2cc(CS(=O)(=O)CC)nn2)C1)OC(C)=O c1(CNCc2cc(Br)sc2)cc(N2CCCC2)ccn1 C(CCN=C(NCCCN(C1CCN(C)CC1)C)NCC1CC1)SC N1(C(C(C)CNC(c2ccc(CO)cn2)=O)=O)CCC(=C(F)F)CC1 N1(C(CC=CC)=O)CC(NC(C2(OC)CCSCC2)=O)CC1C N(C1CCCn2cnnc21)C(=O)NCc1ncccc1-c1nn[nH]n1 N1(c2nc(C)nc(Cl)c2)CC(NC(=O)C2=C(Cl)CC2)C2CCCCC12 C1(C#C)(C(N2C(C#C)CC2)=O)CCN(C(=O)C(C)C(C)COC)C1 c1(OC)cc(C(=O)NCc2ncccc2C(=O)NC(C)CC(C)(C)OC)ncn1 N1(C(CCC(C)(C)NC(C(n2ccc(C)n2)C)=O)=O)Cc2cccc(F)c2C1 c1(N(C(C2C(NC(CCSC)=O)CCC2)=O)C)cc(C)cc(F)c1 C#CCCCCCCC(=O)N1CCC(NC(c2cnc(C)[nH]2)=O)C1 c1(NC(=O)NC(C(=O)OC)C)ccc(C(F)(F)F)cc1[N+](=O)[O-].C12CCCN1C2 CC1CN(C(=O)CCOCC2CC2)CCC1NC(C1(C)CCSCC1)=O C1(C(=O)NCC(CC=C)CC=C)CN(C(c2cc(C)cc(C)n2)=O)CCC1(C)C N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)Cc2ccc(Cl)cc2Cl)CC1C(C)(C)C N1(C(c2c(CC)c[nH]c2)=O)CCC2C1CCCN2C(C1CN(CP(C)(C)=O)C1)=O C1(C(=O)NCC(C)N(c2ncc(C)c(O)n2)C)CC2(C1)NC(=O)NC2=O N1(C(CC(C(=O)OC)(C)C)=O)CCC2(CCC(NC(C3CC4(CCC4)C3)=O)C2)C1 N1(C(CN(CC(C)C)C(c2ccn(C3CC3)n2)=O)=O)CCCC2(CC2)C1 N(C)(S(=O)(=O)N(C)C)CC(=O)N(CC(CO)(CO)NC(c1cc(C)oc1C)=O)C C1(N(C(C(C(C)C)SC)=O)C)CCCCN(C(c2ccc(C)nc2O)=O)C1 C1(C(=O)NCC2CCN(C3CC3)C2=O)CCN2CCOCC12 c1(C(=O)NCC(=C)CCNC(=O)CCc2ccccn2)ccc(Cl)c(F)c1 C12(CC(N3CCC(OC)CC3)=O)CCC1CN(C(C1CCC(N(C)C)C1)=O)C2 c1(NC=O)ccc(C(=O)NC2CN(C(c3cc[nH]n3)=O)CC2F)cc1 N(C1c2ccccc2CC1NC(=O)C=CC=C(Cl)Cl)C(c1cncn(C)c1=O)=O N1(C(c2nc(C3CC3)n[nH]2)C)CC(O)CCC1c1ccccc1.C1(C)(C)CN1 c1(C(N(CCNC(C(C2CCC2)OCC)=O)C2CC2)=O)cc(I)c[nH]1 C(N=C(NN(C)CC1(O)CCOC1)NC1CCC1)c1ccc(N(C)C)s1 N1(C(c2n(CCOC)ncc2)=O)CCC(C)(NC(c2cc(Br)ccc2F)=O)CC1 c1(C(=O)NC2(CC=C)CN(C(C3CCCN4CCCC34)=O)C2)cncc(C)c1C N(C1CCCc2c1cnn2C)C(=O)NCCc1c(C)n(C)nc1 C12(NC(CC(C=C)(C)C)=O)CCCCCC1N(CC(=O)NC1CCCC1)CC2 CCCC(CCCNC(C1CC1C)=O)NC(=O)C=Cc1cncs1 c1(NC)cncc(C(N2CCC(C(C)NC(c3cc(C(F)(F)F)no3)=O)C2)=O)c1 N1(C(CSC)=O)CCC2(CCOC2)C(CNC(c2n[nH]c3cc(C)ccc23)=O)C1 c1(CC(=O)NC(C)CCNC(C2(CO)CCOC2)=O)ccc(Cl)cc1Br CC1(CNc2cc(CC#N)ncn2)CCN(C(=O)CCC2CC2)CC1 n1(CC)nc(C(C)C)cc1C(N1CCN(C(=O)NC=O)CC1)=O.C1(=O)CC(C)O1 CC(CC(=O)N1CC(C)(NC(=O)CC2C=CCCC2)C1)C(F)F N1(C(CC(C)N(C(=O)C=Cc2ccoc2)C)=O)CCCC(C)(O)C1 C(C)(C)(C(C)CC(=O)NOC(CO)C(C)C)NC(CC1CC(=C)C1)=O C1(C(N2CC(CNC(C(C)OCC3CCCCO3)=O)C2)=O)CCC(C)(C)CC1 CCCCC(CCCC)NC(C1C(C)OCCN1C(c1ccnn1C(C)C)=O)=O N1(C(CCCOCC=C)=O)CC2(CC2)CC1CNC(=O)C(C)(C)c1cnn(C)c1 C1(CC(N2CCC(CNC(C3(OCC)CCCC3)=O)C2)=O)CCCC(C)(C)CC1 N1(C(C2CC=C(C)CC2)=O)CC(O)C(O)C1CNC(=O)CCCN1CCCC1 c1(C(N(Cc2cn(C(C(OCC)OCC)C)nn2)O)=O)cc2c(Cl)cccc2[nH]1 c1(C(=O)NC2CCN(C(C34OCC(C)(C3)C4)=O)CC2)ccc2c(c1)OCCO2 C1(CC)CN(C(=O)CCC[N+](=O)[O-])CCC1NC(=O)C(c1ccccc1)O N1(Cc2cn(C(C)C)nn2)CC2C(NC(=O)CC3CCCOC3)C2C1 c1(CC(=O)N(CCNC(=O)CNS(=O)(=O)N(C)C)CC)c(C)[nH]c2ccccc12 CCC(C)C(C(=O)N1CCC(NC(=O)CC2(C(=O)OC)CCCCC2)C1)OC CC1CN(C(C2(CO)CCC2)=O)CC1(C)C(=O)N(C)CCOC(F)F C1(NC(c2c(C)cns2)=O)CCC(F)(CNC(=O)Cn2cnc(C#N)n2)C1 CON1CC(NC(CCC2(C)CN(C(C3CC4(CCO3)CC4)=O)C2)=O)CC1=O c1(C(=O)NC2(C)CN(C(c3coc(C(F)F)n3)=O)C2)cccc2c1OCC(=O)N2 c1(C(=O)NCCc2c(CNC(CC=C)=O)nco2)sc(F)cc1Br S(=O)(=O)(CCC(F)(F)F)N1CC2CN(S(CC#N)(=O)=O)CC21 N1(C(C(CCC)c2ccc(Cl)cc2)=O)CC2(CNC(=O)CSC)CC1CCO2 c1(CCCNC(=O)C(=O)NC2CCCC2)ccc(F)cc1Cl N1(C(C(C)OC)=O)CCCCC1C1CCN(C(C2CN(C)C2)=O)CC1 C12(CCCSC1)NC2.S(=O)(=O)(CCN(C)C)N(CC)CC C12CN(C)C3CC(OC)(CC13)OC2.c1(OC)ccc(Oc2ccccc2)c(OC)c1 CC(CS(C)(=O)=O)C(=O)NC1CC2(CCN(C(c3cn(CC(N)=O)nn3)=O)C2)C1 CCCC(C)C(=O)NCCN(C(C)C)CC1CCCCCC1 CCC(CC(=O)NC1(CN(C(=O)C(C(C)C)n2cccc2)C)CC1)C1CC1 C1(O)(CNC(CCCN(C(C)=O)C)=O)CCCN(C(c2cncc(N)c2)=O)CC1 c1(OC)ncc(C(=O)NC(C)CCCNC(c2coc(C(C)=O)c2)=O)c(C)n1 c1(C(=O)NCC2(NC(CC3CCCN(C)C3)=O)CCOC2)cc(F)c(Cl)cc1Cl c1(C(=O)NCc2c(C(N3C(C)(CCO)CC3)=O)[nH]cc2)cc(CO)ccn1 N1(C(C2N(C(c3ccn(C)c3)=O)CC(O)CC2)=O)CC2(CCCCC2)C1 N1(C(CCCN(C(C)=O)C)=O)CC(O)CC1CNC(=O)CC1CCSC1 N1(C(C(CC#C)NC(c2ccc(CC)cc2)=O)=O)CCN(CC)C(C)C1 CCC(C)C(=O)NCC(C(C)C)NC(C1CC(CC(=O)OC(C)(C)C)C1)=O N1(C(CC(C)(C)F)=O)CCC2C(CCN2C(C2CCC(=O)N2)=O)C1 S(=O)(=O)(c1ccc(N(C)Cc2cc(C)ccc2C)cc1Br)NC(CCC)C C1(C(=O)NCCN(C(=O)C(C)(C)C2CCOC2)C)CC(=O)OC1(C)C C1(C(N(CCO)CC)=O)CCc2nc(-c3cccc(C)c3OC)sc2C1 N1(C(C2N(C(C3N(C)C(=O)CC3)=O)CC=C2)=O)CC(F)(F)C(F)(F)C1 C1(C(N(C2CCCN(C(C3(C=C)CCC3)=O)C2)CC)=O)CCc2ccccc2C1 c1(NC2C(SCC)CCC2)cc(N2CCCC(F)(CF)C2)nc(C)n1 CC1CCCn2c(CC(=O)NC3C4CC3N(C(C3CC3C(C)(F)F)=O)C4)cnc21 C12CCN(C(C(=O)NC(CO)C3CC3)C1)C2=O.C1(CC)C=CCC1 C(=O)(CC(CNC(=O)CC(Cl)Cl)OC)NCC1(OC)CCC1 Cc1nn(C)c(C(=O)NC23CC2CN(C(=O)CNC=O)C3)c1[N+](=O)[O-] c1(C(N2C(CNC(=O)C=CC(=O)N(C)C)CC(OC)C2)=O)ccc2ccsc2c1 c1(CCC(=O)NCC2CC3CC3N2C(=O)CC2CC2)ccc([N+](=O)[O-])cc1Cl N1(C(=O)OC)CCS(=O)(=O)CC1.c12cccc(c1)NC(=O)CO2.C12CN(C1)C2=O N#Cc1c[nH]c2c(F)cc(F)cc2c1=NCC(O)CNC(=O)Cc1cscn1 c1(OC)c(C(=O)N(C)CC2CCCN2C(C2CC23CCOCC3)=O)cccc1Cl C1(NC(C2CCC(=O)C2)=O)CC2CCC1CC2NC(c1ccncc1Cl)=O n1(CCCOCCOC)ncc(-c2nc(COc3ccccc3)no2)c1C(F)(F)F N1(C(C2CN(C)C(=O)CC2)=O)C2CCC1CN(C(=O)Cc1cnns1)C2 c1(C(N2CC(n3cc(CCCCC)nn3)C2)=O)cccc2nn[nH]c12 c1(CN2CCC(NC(c3n[nH]cc3[N+](=O)[O-])=O)C(F)C2)cc2ccccc2cn1 C(=O)(C(C)C(O)C(C)C)N1C(CNC(c2ncc(OC)cn2)=O)CCC1 C1(C(C(=O)N(CC(C)NC(C2(CCC)CCC2)=O)C)C)CCOCC1 Cc1cc(N)c(C(N2CCCC(NC(=O)CC3CC3(Cl)Cl)C2C)=O)cc1C C1(NC(C2CC(OCC)C2)=O)CC(C)(NC(=O)C=C(CC)CC)C1 c1(OC)cncc(C(=O)NC2CC(N(C)C(c3ccc(C(N)=O)nc3)=O)C2)c1 Cc1[nH]cc(C(N2CCC(CCNC(=O)CCC3CCCC3)CC2)=O)c(=O)c1Cl C1(SC)CC(C(=O)NCCN(C(=O)NC(C)(C)C)CC2CC2)C1(C)C N1(C(c2cnc(OC)c(Cl)c2)=O)CC(C)CN(C(C2(C#N)CCCC2)=O)CC1C C1(CNC(COCCN(C)C)=O)(CO)CCCN(C(C2CCCO2)=O)C1 C1(NC(C(c2cnn(C)c2)NC(c2ccc(C)[nH]2)=O)=O)CCC=CCCC1 c1(N(C)CCC2CCCCN2C)nc2c(c(=NC3CCN(C)C(=O)C3)[nH]1)SCC2 CC1CCC1CC(=O)N(CCC(=O)N1CC(N2CCCC2)C1)C CCCCCC(C)(C)C(=O)NCC(C)(O)CNC(c1c(C)[nH]c2ccccc12)=O c1(C2C(C)C2)[nH]c(=NCc2cn(C)c3ccc(C4CC4)cc23)nc2sccc12 C1(CN(C(C2CCN(C(C)=O)C2)C(=O)NCCOC)CC)CCS(=O)(=O)C1 C1(N(C(C2CCC(C)(CC)O2)=O)C)CCC2CN(C(c3ccc(F)s3)=O)CC12 C1(CC(=O)NCC2(CN(C)C(c3ccccn3)=O)CC2)CCCCCCC1 N#CC1(C(=O)NCCC2CCN(C(=O)C(F)=C3CCCC3)CC2)CCCO1 Cc1cc(CNC2CCCN(CCF)C2)c2cn[nH]c2c1 CC1=NNC(=O)C1CC(N1CCC(CCC(=O)N(C(CF)CF)C)CC1)=O CCCCCC(CC)C(=O)N1CC(NC(c2cc(CC)on2)=O)CC12CCOC2 c1(-c2onc(-c3c(CSC)cccc3)n2)ccc(S2(=O)=NCCC2)cc1 CC(C)(O)C(F)CNC(=O)Cn1cc(-c2nc(Cl)cs2)nn1 CS(=O)C=CC(=O)NCC(c1cccc(C(F)(F)F)c1)NC(=O)CC1CSCCS1 Cc1cc(C(N2CCC(N(C(=O)COC(F)(F)F)C3CC3)CC2)=O)c(C)n1C N1(C(CN(C)C(N)=O)=O)CC2(CCC2)CC1C(=O)NCc1ncsn1 N1(C(C(=O)NC2CCOC2)c2cccs2)CCC(C2(O)CCOC2)CC1 C1(CCOC)(NC(=O)C(F)C(F)(F)F)CCN(C(c2coc(C(N)=O)c2)=O)CC1 c1(NC2CC(NC(C3N(C)C(=O)OC3)=O)C2)ncc2ccsc2n1 c1(C2(C(=O)NC(c3ccsc3)CO)CC2)cccc2c([N+](=O)[O-])cccc12 c1(OC)ncnc(OC)c1CNc1cnc(F)cc1C(=O)Nc1ccncn1 N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC(NCc2c(C(=O)O)cccc2F)C(F)(F)C1 c1(C(=O)NCC2C(NC(c3cncn(C)c3=O)=O)C2)cn2cccc(F)c2n1 Cc1ccc(C(=O)NC2CS(=O)(=O)CC2NC(=O)CC2CC=CC2)c(C)c1 C(C)(C1=CCN(C)CC1)NC(CN(C(=O)Cc1cn(C)cn1)C(C)C)=O C1(NC(CNC(C2C(C)C2)=O)=O)CC=C(C(=O)N2CC(O)(C(N)=O)C2)C1 N1(C(C2C(C)=C2)=O)CCN(C2CCN(C(c3cnc(Cl)cc3Cl)=O)CC2)C(=O)C1 C1(O)(CNC(C(C)N(CC)CC)=O)CCCN(C(c2cc(CO)on2)=O)CC1 N1(C(Cc2n(C)ncc2)=O)CC(NC(C2CC2[N+](=O)[O-])=O)CC1(C)C C=CC1(CO)CCN(C(=O)C(c2cccs2)NC(c2cn[nH]c2)=O)CC1 c1(NC2(CNC(c3ccc(O)nc3Cl)=O)COCCC2O)ccc([N+](=O)[O-])c(O)n1 N1(C(Cc2cc(C)nn2C)=O)CCC2(CC2C(N2CCS(=O)(=O)CC2)=O)C1 CCCC(C(=O)NCC1CC(NC(=O)CC23CCC(CC2)C3)C1)NC(N)=O C(C(C)(C)C(=O)NCC1CC(NC(=O)C(c2cncc(F)c2)C)C1)OC c1(C(N(C2CN(C(C(C)SC)=O)CC2(C)C)C)=O)c(C)ccc2n[nH]cc12 CS(C)(=O)=NC(=O)C(=O)N1CC2(C1)CN(C(c1c(N)cccc1F)=O)C2 N1(C(c2ccn(C)c2)C(=O)NCCCSC)CCN(CCNC2CCC2)CC1 CN1CCN(C(C2CCCO2)=O)C(CNC(=O)CCn2cc(Cl)cn2)C1 C1(NC(c2scc(C)c2)=O)CN(C(C2C3CCC2(c2ccco2)C3)=O)CCC1F N1(C(c2c(C)ncc(Cl)c2)=O)CCN(C(=O)CNC(c2ccoc2)=O)C(C)C1C N1(C(=O)COCC2CCCC2)CCC2CN(C(c3ccc4[nH]ccc4n3)=O)C2C1 C1(CNC(CCC(C)SC)=O)CC2(CCN(c3cc(=O)n(C)c(=O)n3C)C2)CO1 CN1CC2(CCN2C(c2c(CNC(C3(C)CCOC3)=O)nnn2C)=O)C1 N1(C(c2c(CC)cno2)=O)CCC(C(N2CCOCC2CC)=O)(CO)C1 c1(C(N(C2(CC(=O)N(C3CC(O)C3)C)CC2)C)=O)ccc(C#N)[nH]1 c1(C(=O)NC2CCCC(CCC)C2)cc(C)ccc1N(CC)CC N1(C(C(C)CC2CCC2)=O)CCN(C(c2cc(O)cnc2N)=O)C(C)C1 C1(C(C)N(C(=O)COC2CN(C(=O)CC3(C)CC3)C2)C)CC(F)(F)C1 c1(NC(C2N(Cc3cccc(N(C)C)c3)CCC2O)=O)c(F)ccc(Br)c1F N1(C(c2c(C)oc(CO)c2)=O)CCOC2(CCN(C(=O)C#CC3CCOC3)C2)C1 C1(C(N2CCC(COC)CC2)=O)C2CCC1CN(C(C1(F)CCCC=C1F)=O)C2 N1(C(c2cnc(CC)nc2C)=O)CCC2CC1CN(C(=O)C(C)(C)C(C)O)C2 C1(NC(c2n(CC)ccc2)=O)C2CCN(C(C3SCCCS3)=O)CCC12 C1(C(N2CC(O)C(O)C2)=O)CN(Cc2cc(F)cc(Cl)c2O)CC(F)(F)C1 C1(C(N(C)Cc2cc(CNC(=O)C(O)c3ccsc3)[nH]n2)=O)COCCN1C C(=O)(C(C)(C)CN(C)C(C1CCCN1C=O)=O)NCCC1CC(C)C1 CC(CF)CC(=O)NCC1(C(C)(C)C)CCNC1=O C(=O)(C1c2c[nH]nc2CN1C(=O)CCC1CCC(=O)NC1)N(CCOCC)C c1(C(=O)NCCN(C)C(C2CC23CCOCC3)=O)cccc(Br)c1Cl c1(NC(C(=O)Nc2ccc(NCC(F)F)cc2)=O)nc2c(s1)CC(O)CC2 n1(CCOC)cc(C(=O)NCc2nc(CNC(=O)CC(C)F)cs2)nn1 c1(NCC23CC2CN(CC2(C(C(CC4(C=C)CC4)=O)=O)CC2)C3)ccc2c(c1)OCO2 C(C)(CCCC(=O)N1CCN(C)CC1)NC(C1(CCC)CC(=O)C1)=O N1(C(CCC(C)(F)F)=O)CC2(CNC(=O)C(CO)C(C)(C)C)CC1CCO2 C(=O)(C(F)C(C)(C)O)N1C(C2(O)CN(C(Cn3c(C(C)C)nnn3)=O)C2)CCC1 Cn1ncc(S(C)(=O)=NC(=O)C2CC3CC2(c2cccnc2)C3)c1C(N)=O Cc1cnnc(NC(c2nnnn2C2CC(F)(F)C2)CC2CCC2)c1 c1(OC)c(Cl)cc(C(=O)NC2CCN(C(C3COC(=O)O3)=O)C2)nc1Cl Cc1ncc(C(N2CCC=CC2C(=O)NCCCOC2CC2)=O)cc1C#N C1(c2nn[nH]n2)(N(C(=O)C(C)(C)C)C(C)C(=O)NCc2ccco2)CCCCC1C N1(C(c2ccc(CC)cc2)=O)CCN(C(C2CCCCO2)=O)C(c2ncc[nH]2)C1 c1(OC)ccc(C(=O)NC2CC(C(=O)Nc3ccnc(C)n3)C2)c(F)c1F C(=O)(CC(F)(F)CC(=O)N1CCOCC(F)(CNC(C2(C)CCCO2)=O)C1)OC C1(CNC(=O)C(c2ccccc2)O)CC2(CO1)CN(C(=O)Cc1cc[nH]c1)C2 C(c1ccccc1)=C(OC)C(N1CC2CC1C2NC(=O)CSc1nnc(C)n1C)=O c1(C(N2CC(C(=O)Nc3cc(OC)c(Br)cc3)OCC2)=O)cc(F)cc(C)c1O C(CC(C)(C)C(=O)NC)N(C1CC(C(F)C(=O)C(N)=O)C1)C.c1(N)cc(C2CC2)no1 Cc1c(NC(C2C(C)CCN2c2nccc(C(C)(C)C)n2)=O)ccc2n[nH]cc12 C(=O)(CC(C)(C)CC(F)F)N1CCC(C2(NC(CCS(C)=O)=O)CC2)C1 CC1(C)CCC(CNC(c2cncnc2C2CC2)=O)N(CCC2CCC2)C1 c1(C)ccccc1CC.n1(CCOC)nnnc1C(c1cccs1)NCCSC c1(C(=O)NCC2C(NC(CCCC(N)=O)=O)CCC2)coc2c1C(O)CCC2 CCC(C)CCCCC(=O)N(C(C)CNC(c1cc(C)c(F)cn1)=O)C O=C1OCc2cc(C(=O)NC3CCCCN(C(c4c[nH]c(=O)cn4)=O)C3)ccc21 N1(C(C2(CC)CCC(O)CC2)=O)CCC2(CCC2CNC(=O)C(C)(C)CF)CC1 C(=O)(C(F)C(C)(C)O)N(CC(N1CCCC(OCC)C1)=O)C1CC1 Cc1csc(C(N2CC(CNC(=O)C=C3CCCCC3)C3CC23)=O)c1C C1(CN(C)C(c2ncn(C)n2)=O)CCCCN1C(=O)C(F)=C1CCCC1 N1(C(c2c(C)cnn2C)=O)CC2CCC2(CNC(=O)CSCCC(C)C)C1 N1(C(CCC=C=C)=O)CCC(NC(=O)COc2cncc(Cl)n2)C(CO)CC1 C(=O)(C1=CCc2ccccc21)NC1CC2CN(C(C(=O)NC(C)C)=O)CC(C1)C2 c1(C(=O)NC(C)CC(C)NC(C2(NCCO)CCC2)=O)cccc(=O)n1C c1(CSCC)cn(CCN(C(=O)C(CC)N2CCCC2=O)C)nn1 N1(C(C(C(C)O)C)=O)CCN(C(c2nccc3cc[nH]c23)=O)C2(CCC2)C1 N1(C(C2(OC)CCSC2)=O)CCCN(C(=O)C(C)c2ccsn2)CC1 C1(NC(CC2C(C)C2)=O)CC2CC(C1)N(C(c1cc(O)c(F)cc1N)=O)C2 Cc1cc(C(=O)NC(c2ccc(CNC(C3(Br)CC3)=O)cc2)C)cc(N)c1O C1(NC(C(CC=C)C)=O)CC2CC(C1)N(C(c1ccc(OC)s1)=O)C2 Cc1ncc(C=CC(=O)NC(CNC(=O)Cc2nnc(C)o2)C(C)C)c(O)n1 c1(C(CNC(c2c(CCC)n[nH]c2)=O)NC(=O)C(C)SC(C)C)cccc(C)c1 c1(CNC(C(C)CN(C(=O)CCN2CCCC2=O)C)=O)ccccc1C#N C(=O)(CC(c1ccccc1)C1CC1)NCC(C)NC(=O)CCC1(C)CCCN1 c1(OCCOC)ccc(CNC(=O)C(=O)Nc2cnc(CCN)nc2)cc1 CC1CN(CC(=O)NCC(C)(C)NC(=O)COCC(F)F)C1 N1(C(C=CC=CC)=O)CCCC(C)(C)C1C(N1CC2(CO)CC2(CO)C1)=O N1(C(C=C(CCC)CCC)=O)CCOC2(CCN(c3ccc(C#N)nc3)C2)C1 C1(C(N2C(CNC(CCOC)=O)CC(F)(F)C2)=O)CC2CC1C1C2C1(F)F N1(C(Cc2nc(C)sc2)=O)CCN(C(c2coc3c2COC3)=O)C(CF)C1 c1(C(N(CCNC(C2CCN(CC)C2)=O)CC)=O)cc2n(c1)CCC2 C1(C(N(C2CCN(C(c3nc(CCC)sc3)=O)C2)CC)=O)CCC(=O)NC1 c1(NC(C)=O)ccc(NCC(n2cc(C3(OC(C)C)CCOC3)nn2)C)c(F)c1 N1(C(C(C(C)C)O)=O)CC2CS(=O)(=O)CC2(NC(=O)C(F)=CCCF)C1 Cc1ccc(NC(=O)NCc2ccnc(N3CCCCCC3)c2)nn1 C=CCC(CC=C)C(=O)NC(CC=C)C(=O)NCCC1CC=CC1 c1(C(N(CC(C)(C)NC(C2CC(C)(C)CCO2)=O)C)=O)n[nH]c2ccccc12 c1(-n2ccc(CCNC(=O)NC34CC(CO)(C3)C4)n2)cccc(F)c1 c1(NCC(CC)C(C)C)[nH]c(=NCC(C)(C)N(CC(F)(F)F)C)nc2sccc12 C1(CNC(C(C)CNC(=O)C(C2(O)CCCC2)F)=O)CC12CCOCC2 C#Cc1ccc(C(N2CCN(C(=O)CCCc3cccs3)CC2C)=O)cc1C S(=O)(=O)(c1cccnc1)NC(C(=O)NCC1(NC(COC(C)C)=O)CC1)C(C)C C(=O)(CCC(C)(C)C(=O)OC)N1C(CNC(C(C(CC)O)(F)F)=O)CCCC1 N1(C(C2ON=C(C)C2)=O)CCC(O)CC1C(=O)NCC1CCCCN1C C1(NC(C=CC(C)C)=O)CCCC(CC(=O)NCC2(F)CCOCC2)C1 C=C1CC(CONC(=O)C2CC(NC(=O)CNC(=O)NC3CC3)C2)C1 S(=O)(=O)(c1c(OCOC)ccc(Cl)c1F)CCOc1ccc(C(=O)OC)cc1 C1(C)(C(=O)NCC(C(C)C)NC(c2ccccn2)=O)CC(C2CC2)=NO1 c1(-c2scc(C(=O)NC(c3ncc(F)cc3F)C)n2)c(Cl)cccc1Cl CC(F)(F)CC(=O)NC1CCC(NC(=O)CC2CCC23CCC3)C1 Cc1cc(C2CC2)ccc1C(=O)N(C)CC1CCCN1C(c1ncoc1C)=O Cc1c[nH]ccc1=NC(=O)c1cc(NC(C2CCC(F)(F)CC2)=O)cn1C C(CNC(=O)Cn1nnc(C2CC2)n1)(CC(F)(F)F)NC(Cc1c(C)n[nH]c1C)=O c1(C(=O)NC2C(C)CCN(C(c3cccn3C)=O)C2C)cccc2c1nnn2C c1(C(=O)NCCCOCCNC(C(C)C2CC2)=O)ccc(N(C)C)cc1 C1(C)(C(N2CC(O)(CNC(C3(OC)CCCOC3)=O)C2)=O)CCC(C)C1(C)C C(=O)(C1CCCn2cncc21)NC(CC=C)CNC(c1cn(C)ccc1=O)=O c1(C(=O)NC2(C#N)CCN(Cc3ccc(Cl)cn3)C2)cc2ccoc2cn1 CC(c1cnn(C)c1)=CC(=O)NCC1C2CN(C(=O)CCc3ccoc3)CC12 c1(NC(c2nc(C(=O)Nc3ccc4c(c3)OCO4)cs2)=O)cccc2ccnn12 c1(CC(N2CC(NC(C3(C#C)CCCC3)=O)C(OC)C2)=O)cnc2ncccn12 C1(CNC(c2c(CC)nco2)=O)CN(c2ccnc(Cl)n2)CCN1C C1(NC(Cn2ncc(CC)c2)=O)CCCN(C(C2CCC=CCCC2)=O)CC1 Cc1sc(C(N2CCC(C3CCCN3)C2)=O)cc1[N+](=O)[O-].C12=CC=C(C=C1)C2=O CCC(CC(=O)NC1CC(NC(C2CCCN2C2CC2)=O)CC1O)SC N1(CC)CCC(C(N2CCSCC2CCNC(c2cnn(C(F)F)c2)=O)=O)CC1 c1(C(=O)NCC(C)(C2CCC2)NC(C2Cc3nccn3C2)=O)cc2n(n1)CCC2 c1(C(=O)NC2CC3CN(C(c4cn(CC=C)nn4)=O)CC32)cnn2ccn(C)c12 C1(C(N(CCC(C(C)C)NC(CCCC=C)=O)C)=O)CC12CC(C)(C)C2 N1(C(C2CN(C)C(=O)CC2)=O)CCC2C(CCCN2C(c2cnc(S)nc2)=O)C1 c1(C(=O)NC(C(=O)N2C(CC)CC2)CO)ncncc1OC C1(C(N2CCN(C(C(C(CC)C)=O)=O)CC2C(C)C)=O)Cc2cccnc2C1 O=C1C2Cc3ccc(F)cc3N2C(=O)N1CC1(Br)CCOCC1 N1(C(C=COCC)=O)CCOC2(CCC(NC(=O)C(C)CSC)CC2)C1 CC(=O)CCCC(C)C(=O)NC(Cn1cncn1)C(=O)NCCCCC(C)(F)F C(C)(CCC(=O)NC1(CO)CN(C(=O)Cc2cccnc2Cl)C1)OC c1(C(C(=O)NCCSC)N(C2CCCC2(C)C)C)cc(S(N)(=O)=O)cs1 C1(C(N2CC(C(C(=O)NC3C(C)C3C)OC)C2)=O)(COC)CCCC1 C1(CN(S(=O)(=O)CCN(C)C(C)C)CC)C2CCC1(c1ccnn1C1CCC1)C2 C12(NC(=O)CSCc3ccc(N)cc3)CCC(C1)N(C(C1CCCCS1)=O)C2 C1(NC(CCCCCN(C)C(c2cc(C(F)F)[nH]n2)=O)=O)CCn2cnnc2C1 c1(C(N(C(C)C(=O)NC(CO)CCCO)CC)=O)ccc(=O)n(C)c1 C1(C(=O)NC2(CC(C)C=CCc3ccncc3)CCC2)CCCCCC1 C(=O)(CCCCN(C(=O)CCC1CC(F)(F)C1)C)N(C)Cc1cncn1C Cc1ccc(C(=O)NCC(=O)Nc2cn[nH]c2)cc1Br.C12CCCN1C2=O c1(C(=O)NC(C(C)NC(C(CCC)OCC)=O)CO)cc2ccncc2s1 CC(F)(F)C(=O)NC1CCCC1NC(=O)CNC(c1ccco1)=O Cc1ccc(C(=O)NCC(C)(F)CNC(=O)C(C)C#N)cc1F C12(NC(=O)Cc3cnns3)CCCCC1N(C(=O)CS(=O)(=O)C1CC1)CC2 c1(C(=O)NC2CC(NC(=O)CC(c3ccc(F)cc3)O)C2)ccnc2ncnn12 N1(C(=O)NC2C(c3c(-c4c(C)n[nH]c4C)cncc3)C2)CCc2cccnc2C1 C(=O)(C(O)CCC(C)C)NC1(C(N2CC(CCCCC)C2)=O)CCSC1 c1(NC(CCCC)(COC)c2nnnn2C)ccc2oc(C(F)F)nc2c1 C1(C(N(C)CCc2ccccc2)=O)CC12CCN(c1nnc(C(F)(F)F)o1)CC2 c1(OC)ccc(Cl)cc1C(N1CC2CC1CC2NC(c1ccnnc1O)=O)=O C=CCC(CNC(C1CCCN1CC(C)C)=O)NC(c1cc(CO)[nH]n1)=O c1(CC(=O)NCCN(C)C(c2ccc3nonc3c2)=O)cncc2ccccc12 C1(SC)CN(C(C2CC(n3cccn3)C2)=O)CC1NC(=O)CNC(C1CCC1)=O C(=O)(CCCCC(F)(F)F)NCC1N(C(C=C(C)Cl)=O)CCC1(C)C C1(NC(CC(n2ccc(C)n2)C)=O)CN(C(c2cc(C#N)cs2)=O)CC(C)(C)C1 C1(NC(CCC(C)OCC)=O)CCC(C)N(C(=O)Cn2ccsc2=N)C1 C1(O)(C(C)NC(c2occc2C(C)C)=O)CCN(C(=O)CCSc2ccccn2)C1 C1(CNC(C(C=C)O)=O)CC12CCN(C(=O)CCCCC#N)CC2 C1(CC(=O)NCC2(F)CC(NC(CCC3(C)N=N3)=O)C2)CCC(F)(F)C1 Cc1ncnc(O)c1C(N1CCC(CCCNC(C2(CO)CCCO2)=O)CC1)=O Nc1cc(CC(=O)NCC(CNC(C2(C(F)F)CCC2)=O)CO)ccc1[N+](=O)[O-] n1(CC)cc(Br)c(C(=O)Nc2ccc(NC(=O)CNC3CC3)cc2)n1 C1(C)(C(=O)NC2C=CC(C(=O)NC(c3cn(C)nc3)CO)C2)CCSCC1 c1(CC)cccc(OCC(N2CC(O)(CN(C(=O)CCC(C)OCC)C)C2)=O)c1 Cc1cc(C(=O)NCC(CC(F)(F)F)NC(=O)CC2CCCCN2C)cc(C)n1 N1(C(C(C)(C)CF)=O)CCC(C2(O)CC(NC(C3C=CCCC3)=O)C2)CC1 N1(C(C(CCCC)O)=O)CCN(C(=O)Cc2ccoc2)CC(C)(F)C1 c1(CC2C(C(=O)NC(c3n(C)ccn3)C(F)F)C2)cccc(I)c1 c1(C(=O)NCCC)ccc(-c2cncnc2C(N2CCN(CCC)CC2)=O)cc1F CC(C)CC(O)C(=O)N(C)CC1(O)CCN(C(=O)Cc2ccc(F)cn2)C1 Cc1cc(Cl)n[nH]c1=NC(=O)C1CCN1C(=O)C1=NOC(C)(C)C1 C1(NC(C2N(C(C)C)CCC2)=O)CCN(C(C2CC3(CCC3)CO2)=O)CC1F c1(CN(c2n(CCC=C)c(CC3CC3)nn2)C)ncc2n1CCCC2 N1(CC)C(=O)CCC1CC(=O)N(C1CCN(C(c2cc(C)sn2)=O)CC1)C C1(NC(c2c(C)cnn2C(C)C)=O)CC2CCC1N2C(=O)CCC1CC1 N1(C(C2C(CC)CCO2)=O)CC2(NC(=O)C(=O)Nc3ncc[nH]3)CCC1CC2 C1(CNC(c2c(C)oc(-c3ccccc3)n2)=O)C(C2CC2)CCN1C(=O)CC#N Cc1c(C(N2C3CN(C(=O)CCC(N)=O)CC23)=O)ccc2c1OCCO2 C(=O)(C(C)(C)CCC(C(=O)NCCC#N)N1CCOCCC1C(C)C)OCC c1(C(=O)NC(C(C)NC(C(=O)NCCOC)=O)C)ccc(OCC(F)F)cc1 c1(CC)ccc(F)cc1NC(=O)CCCCNC(=O)C=Cc1ccn(C)c1 C1(NC(C2(S(C)(=O)=O)CC2)=O)CCCN(C(=O)C2=COCCO2)CC1 c1(C(=O)NCC2C(NC(c3c(C)nc(C)s3)=O)C2)cc(N)c(F)c(O)c1F c1(C(c2n(CC=C)nnn2)NC(C2CC2)C2CC2)ccc(-n2cncn2)c(F)c1 N1(Cc2ccc(N(C)C)cc2O)CC2CN(C(c3ccc(F)c(Cl)c3)=O)CC2C1 c1(C(=O)NCC2CCC(NC(c3cnc(COC)s3)=O)C2)c(C)nc(C)o1 C1(CC(=O)NC(CC#C)CCOC)N(C(c2ncc(CC)cn2)=O)CCC1(C)C c1(C(=O)NCC2CCN(C(Cc3cccc(OC)c3)=O)C2)nc(Br)cnc1N N1(C(C2(COC)CC2)=O)CCC(C(C)C(=O)N(C2CC(C)C2)C)CC1 c1(C(=O)NC(CC(C)NC(c2cn(CCF)nn2)=O)C)cccc2sncc12 CCCCCCC(F)C(=O)N(CCNC(=O)CS(=O)(=O)N(C)C)C1CC1 Cc1c[nH]cc(C(N2CCC(OC3CN(C(C4CNC(=O)C4)=O)C3)CC2)=O)c1=O C1(CC(N2C(C)CC2)=O)COCCN1C(C1CCCC(=O)C1)=O c1(N(CC(C)(C)CO)C(c2ccccc2OC(F)F)=O)ncnc2cc[nH]c12 c1(CC)ncc(C(=O)NC(C2CN(C(=O)CCc3cc[nH]n3)CCO2)C)c(O)n1 c1(C(C)C(=O)NC2CCCC(C(F)(F)F)C2)cccc(-c2nn[nH]n2)c1 C1(CC(=O)NCC2(COC)CN(C(=O)CCc3nccn3C)C2)COC(C)(C)C1 c1(C(N(CC(O)CNC(=O)CN(C2CCCC2)C)C)=O)cc(=O)n(C)cn1 N1(C(C(CC)(C)C)=O)C2CCC1CC(CC=C)(NC(c1ccn(C)c(=O)c1)=O)C2 c1(CC(C)C)cc(C(=O)NC2CCC(NC(C3(C(N)=O)CC3)=O)CC2)cc(O)n1 O=C(CCCCC(F)(F)F)NCC1CC2(CCC2)CN1C(=O)Cn1cccc1 C12(NC3CCN(c4cn(C)nc4)C(=O)C3)CCN(C1)C(=O)NC2=O N1(C(C(CCC)n2cccc2)=O)CCOC(C(=O)NCCCOCC)CC1 c1(NC(C(N2CCC(F)(C(=O)OC)C2)=O)=O)ccc(F)cc1C1CC1 C1(CNC(COCCSC)=O)CCN(C(=O)Cn2cccn2)CC1(F)F c1(NC(N2CC(C(C(=O)OCC)F)C2)=O)ccccc1OCC c1(N2CCC(N(C(=O)C(F)=C3CCC3)CC)C2)ncc([N+](=O)[O-])cc1C(F)(F)F N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCN(C)c2ccc(C)cc21 N1(Cc2ccccc2)C(=O)CN(CCC2(C)CC2)C1=O.CCC1(C)CN1C C(CCN(C)C(c1ccc(C(F)F)o1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O N1(C(c2ccc(CC)s2)=O)CCC(C)(C)C1C(=O)NCCF C1(NC(C2CC(C3CCC3)C2)=O)CCCCN(C(c2ccco2)=O)C1 Cc1cc(C(=O)N(CC(C)NC(c2ccnnc2C)=O)C)cc(C)c1F C1(NC(CC2N(C)CCC2)=O)CCC12CCN(C(c1cscn1)=O)CC2 CC1(C)CCN(C(=O)C#CC2CCC2)C1C(=O)NCc1ncc(F)cc1F c1(COC)ccoc1C(=O)N(C)CC1CCCN1C(=O)C(F)Cc1ccccc1 c1(C(=O)NCC2(O)CCN(C(CCCCOC)=O)C2)cc(Cl)c2ccccc2n1 C12(CNC(CC3OCC(C)(C)OC3)=O)CCCC1N(C(c1csc(Cl)c1)=O)CC2 CC(C)C(C)(CNC(=O)CSC1CCCO1)NC(c1cccn(C2CC2)c1=O)=O C(=O)(CC(C)(C)CCOC)N1CC(N(C(c2c(CC)nccn2)=O)C)C(O)C1 C(=O)(CC(=O)N(C)C)N(C(C)C(=O)NCC(CC1CCCCC1)(C)C)C N1(C(C(n2ccc(C)n2)C)=O)CC(O)CC1C(=O)NCC(C)(C)CC1CC1 C(C)(C(C(=O)NCCC1CCOC1)NC(c1cc(C)sc1N)=O)OC c1(C(N2CC(C(C)NC(c3ccc(Cl)s3)=O)C2)=O)cn2c(n1)CCCC2 c1(CC)cc(F)cc(C(=O)NCC#CC2CCCCO2)c1C N1(C(C2CN(C(N)=O)C2)=O)CCCCC1C1CCN(C(=O)CCc2cn[nH]c2)C1 C1(C(N2C(C(C)C)CC2)=O)CN(C(=O)C(C)C2(O)CCC2)CCN1C C(=O)(CCCCCC#N)NC(C1CCN(C(C2CCCC(F)C2)=O)C1)C Cn1cnc(C=CC(=O)NCCCCC2CN(C(c3cc(C(F)F)cs3)=O)C2)c1 C1(CN(C(C2CC2c2cccnc2)=O)CC)CC(F)CN1C(=O)C(Cl)=CCl CN1CCN(C(=O)CCC2(C#N)CCC2)CC1CNC(c1cnn(C)c1N)=O c1(C(=O)OC)ccc(=NC(=O)CCc2ccccc2OC)[nH]c1F N1(C(C2(C)CCSCC2)=O)CC2CCC(C1)C(NC(=O)CC1CSCCO1)C2 C1(NC(=O)Cc2csnn2)CC2(C1)CN(C(c1cnc(-n3cccn3)cn1)=O)C2 C1(C(=O)NC(C(C(=O)OC)C)C)CC2CC1CN(C(=O)C(c1ccn(C)n1)C)C2 C1(NC(C2C(=C)C2)=O)C(C)(C)CN(CC2CN(C(=O)C(C)(C)C)CCO2)CC1(C)C c1(C(=O)NC(CNC(C2(CC)CCCCC2)=O)CO)cccc2c1COCCN2 N1(CCNC(=O)C(O)CF)CCCN(C(c2ccn(-c3ccccc3)n2)=O)CC1 c1(OC)cc(CO)ccc1CCNC(N1CC(CO)OCC1C)=O N1(C(C(C)(CO)OC)=O)CCOC2(CCN(C(c3cc(Cl)cnc3C)=O)C2)C1 C1(C(=O)NCC#CC)(NC(=O)C(=Cc2ccco2)C)CCSC1 Cc1cncc(C)c1C(=O)NCCCC1CCN(C(C2C(C)C2C)=O)CC1 c1(OC)cc(F)c(C(N2CC(=C(F)CNC(C3(O)CCC3)=O)C2)=O)cc1N S(=O)(=O)(c1ccc(=NCc2ccno2)[nH]c1)NCc1cccc(OCC)c1 c1(CC(=O)O)ccc(-c2csc(CN3CCCC3CCOCBr)n2)cc1 C1(C)(C(=O)NC(CN(C(=O)CSS(C)(=O)=O)CC)C)COCCO1 C(=O)(C1=NN(CCO)C(=O)CC1)N1CC2(CC(CNC(C(CC)C(C)O)=O)C2)C1 C12(CC(=O)NC3(COC)CN(C(C4CC5CCCC45)=O)C3)CCCCC1C2(F)F N1(S(CCC=CCOc2c(C(C)(C)C)ccc(Cl)c2)(=O)=O)CC(C(=O)O)C2(CC2)C1 C1(C(=O)NCC2(NC(CCN3CC(=O)NCC3)=O)CC2)CCC(C2CC2)C1 CC1CN(C(c2coc(O)n2)=O)CC1NC(c1ccc(SC(F)F)cc1)=O C(C#Cc1cn(C2CCCC2(C)O)nn1)NC(Cn1ncc(C)c1)=O C(=O)(CC(O)CNC(C1CN(C)CCO1)=O)Nc1c(CC)csc1 CCC(C(=O)NC1(CNC(C2(C)CC2(C)C)=O)CCCCC1)C(C)C c1(C(=O)NC2CN(C(C(C)NC(N)=O)=O)CC2C)cc(O)nc(N(C)C)n1 C(=O)(CC(C)(C)C(F)F)N1CCC(C(N(CC)CC2CC2)=O)OCC1 Cn1c(=O)oc2cc(CN3CC4C(NC(c5ccc(O)cc5)=O)C4C3)ccc12 N1(C(C2(N(C(c3nc(C)c(C)s3)=O)C)CC2)=O)CCCC2(CCC2)C1 N1(C(C(c2ccncc2)OC)=O)CCCC2(CCN(C(C3(F)CCCC3)=O)C2)C1 N1(C(C2(NC(C3CN(C)C3)=O)CC(O)C2)=O)CC(CO)C2(CCC2)C1 Cc1cccc(C)c1OCC(O)CNCc1ccnc(NC(=O)OC(C)(C)C)c1 C1(CNC(=O)C(N2CCC(CO)C(O)C2)c2cncc(F)c2)CCC(F)(F)CC1 CCCCC(C(=O)NC)N(C)CC.C(=O)(C(C)(C)N1CCCC1)N1CC(=O)OCC1 N1(C(C(N)=O)=O)CCN(C(C2CC3CCC3C2)=O)CC1CF C(CCC(C)(C)O)NC(C1C(NC(C(C)N2CCC2)=O)COC1)=O N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(=O)C(Cl)=CCl)C(C)(C)C1 C1(C(N2CC(CC(C)NC(=O)CC(C)(C)C3CC3)C2)=O)CC2(CCOCC2)C1 N1(CCCC)CCC(NC(c2cn(-c3ccc(C)cc3OC)cn2)=O)C(O)C1 c1(-c2cn(CC)nc2)ccc2cc(C(=O)NC(C)(CO)CO)cn2c1 N1(C(C)C)CCOC(C(=O)NCC(C2CC2)NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 CC1CN2CCN1CC2C(=O)N(CCCCCNC(=O)Cc1ccsc1Cl)C CC1(C)COC(CC(=O)NC2(CF)CCN(C(=O)CC3CCCCC3O)C2)C1 N1(C(c2c(C#N)scc2)=O)CCCC2(NC(C3CCCOCC3)=O)CCCC12 c1(C(N2CCC(N(CCC)C(c3cccc(OC)c3)=O)C2)=O)ccc(N)c(N)n1 C12CCN(C13CC3)C(=O)CC1CC(C1)C(=O)N2.Cc1nccn1CCC(=O)N(C)C c1(NC(c2nnnn2C2CCOC2)C2(CO)CCC2)cc(Cl)c(Br)cn1 CC(C(=O)N1CC(CNC(=O)C(=O)N(C)C)C1)n1ccnn1 c1(SCCC(=O)NC2CC(NC(C3CCC(OC)C3)=O)C2)ccc(F)c(F)c1 C1(CCNC(C(=O)NC2(C#N)CCC2)=O)CCC(F)(F)CC1 c1(C(N2CC=CC(NC(C3CCC3(F)F)=O)C2)=O)ccc(F)c(O)c1 c1(C(=O)NCC(C(C)(C)C)NC(CCC#C)=O)cc2n(n1)CC1(CC1)C2 C(=O)(CC1=CCN(C(=O)CC(C)F)CC1)N1CCCC(C)(OC)C1 c1(C(=O)NC2(C)CC(NC(C3C(CC)OCC3)=O)C2)cc[n+]([O-])cc1 Fc1ccc(C(C2CC3CC3C2)Nc2nnnn2CC2CC2)nc1 N1(C(CCCOCC)=O)CCN(C(=O)COc2ccc(OC)cc2)C2CC12 CC(C(C)C(=O)NC1CC2(CCN(C(c3coc(O)n3)=O)CC2)C1)S(C)(=O)=O CCC(CNC(c1c(CNC(c2cc(C3CC3)[nH]n2)=O)nnn1C)=O)CCO C(CCCCC(=O)N1CC(C)OC(C)C1)N(C(CC(C)OC)=O)C c1(NC(CC2N(CC3(C)CC3(Cl)Cl)CCCC2)=O)ncncc1C#N n1(C2CCN(C(C(N3C(=O)CCCCC3)C3CC3)=O)CC2)cnc2cc(Cl)ccc12 c1(C(=O)NC2(CC)CN(C(C34CCC(OC)C3C4)=O)C2)ccc(F)cc1 CCC(C)C(CS(=O)(=O)c1ccccc1)NC(=O)C(C1CCCCC1)C CC1=CCC(NC(=O)C(Cn2cncn2)NC(C23CSCC2C3)=O)CC1 Cc1nnccc1C(=O)NC(C1CCCC1)CNC(C1(C2(C)CC2)CC1)=O N1(C(c2cc(C)c(Cl)cc2)=O)CCC(C)N(C(c2nocc2Br)=O)CC1 C(=O)(C1=Cc2cccc(OC)c2OC1)NCC1CCC(NC(CC)=O)C1 c1(OC)cc(CN(C)C(C2CNCCO2)=O)cc(Br)c1OC C1(NC(CN(C(C)C)C)=O)COCC1CNC(C1CCOC1)=O c1(N(C)CC2CCCN2C(Cc2cccc(OC)c2)=O)ccc([N+](=O)[O-])c(C)c1 CCC(C)(CC)C(=O)N1CCN(C(c2cccc(OC(C)C)c2N)=O)C(CO)C1 c1(NC(N2CC3CCCC(C3)C2)=O)cnc2[nH]cnc2c1 C1(OC)(CNC(=O)CN2CCNC(=O)C2)CCN(C(=O)CCCn2ccnn2)C1 c1(C(CCC(=O)NC2(C)CCN(C(CCOCC#C)=O)C2)=O)ccc(O)c(F)c1 c1(SC)ncc(C(=O)NCC2CCC(NC(=O)CCC3CC3)C2)s1 C1(N(C(=O)CCCF)CCC)CCN(C(=O)CC2(C)CCCO2)CC1 Cc1ccc(C=CC(=O)NC2CCC(CNC(=O)COCc3nc[nH]n3)CC2)s1 c1(-c2cc(CNC(Cc3nc(C(=O)O)sc3)=O)no2)c(Cl)cccc1Cl C(=O)(CCC(CF)CF)NC(CC(=C)Cl)C(=O)N1CC=C(CO)CC1 O=C(CC(F)(F)C(F)F)NCCCNC(c1ccnn1CCF)=O N1(C(CC=CCC)=O)CCC2CCC(NC(=O)CCNC(=O)CO)C1C2 C1(C(=O)NCC(C)(C2CCC2)NC(CC=CCC)=O)Cc2nn(C)cc2C(=O)N1 C(=O)(C(C)CCC(C)(C)C)N1C(CNC(c2cc(OC)n[nH]2)=O)CC2CC21 N1(C(c2cccc(C)c2N)=O)CC2CCCC2(C(=O)NOC(C)C)C1 C1(C(NOCC)=O)C(C)OCCN1C(=O)C(C)OC(C)=O Cc1ccc(N(C)C)c(N2CCNC2=O)c1.c12cc(ccc1O)NC2 N1(C(C(=O)NCCCC=C)=O)C2CCC1CC(F)C2 C1(C(N(CC(C)(C)NC(c2cc(C(F)(F)F)n[nH]2)=O)C)=O)CCn2ncnc2C1 C1(C(N2CCCC(C(=O)NC)C2)=O)COCCN(C(C2CN(C(N)=O)C2)=O)C1 C#Cc1cnc(N2CCC(CNC(c3cnc(F)c(F)c3)=O)C2(C)C)nc1 C1(C2CN(C(=O)CCCC(F)F)C2)(NC(C2CCCC(C)C2)=O)CC1 N1(C(C(CC)COC)=O)CCCN(C(c2cc3sccc3[nH]2)=O)C(C)C1 c1(N2C(C)(CNC(C3(C)CCCS3(=O)=O)=O)CCC2)nccn2nnnc12 N1(C(c2csc(Cl)n2)=O)CCC(CNC(C23CC2Cc2c[nH]nc23)=O)C12CCC2 c1(CN(C)C(=O)NCC2CCOC(C(=O)OC(C)(C)C)C2)c(Cl)cncc1Cl N1(C(c2ncc(C)cc2C)=O)CC(C)(C)OC2(C1)CN(C(c1[nH]cnc1C)=O)C2 C(c1ccc(C)cn1)=CC(=O)N(CC(CC)NC(C1CCC=CCCC1)=O)CC Cc1ccc(F)c(C(N2CC(NC(=O)CCOC3CCCOC3)CC(O)C2)=O)n1 CCCCC(CNC(c1sccc1OC(F)F)=O)NC(C1(CF)CC1(F)F)=O CCC(CC(=O)NC(COC)C(C)C)N(C)C(c1cc(C)c(C)[nH]1)=O C1(C(N2CC(F)(CNC(C(C)OCC)=O)C2)=O)CCC(C(N)=O)CC1 Cc1ccn(CC(=O)NC2(C)CC(NC(=O)CCCN(C)C(C)C)C2)c(=O)c1 Cc1cc(CC(N2CCC(CNC(c3cnn[nH]3)=O)C2)=O)no1 N1(C(COC)=O)CC(CC(=O)NCC(C2CCC2)OC)CC1(C)C Cc1nnn(CC(=O)NC(C(=O)NC(C2CCCO2)CO)C2CCCC2)n1 C1(NC(C2(NC(=O)CN3CC(=O)NC3=O)CCN(C)C2)=O)CC1C1CCOCC1 N1(C(C2(C(=O)OC(C)(C)C)CCC2)=O)CCC(F)(C(N2CC(N3CCCC3)C2)=O)C1 C12(NC(=O)Cc3ccc(CO)cc3)CCCC1CN(C(=O)C1=COCC1)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCC2CN(C(=O)Cc3cc(C)sc3C)C2C1 CCCCCCN(CC(N1CCC(N(C(=O)CC2CCCSC2)CC2CC2)C1)=O)C C12(NC(COCCC#C)=O)CCC(C(=O)NCC3CCCC3CF)(CC1)C2 C(CCN=c1[nH]c(=NCc2cccnc2N(C)C)[nH]c2ccsc12)N(C(C)=O)C N1(C(C(c2cnccn2)C)=O)CC(NC(=O)CN(C)Cc2ccco2)CCC1C c1(CCC)ncc(C(=O)NCC2CC(NC(=O)CCc3ccc(C4CC4)o3)C2)s1 c1(C(N(CCC2N(C(C=CC(CC)C)=O)CCCC2)C)=O)cc(Cl)ccc1C c1(C(N)=O)nccnc1C(=O)NC(c1ccccc1F)CNC(=O)C(O)C1CC1 N1(C(C(=O)NC)=O)CCOCC(C(=O)NCCC(C)N2CCCC2)C1 c1(C(=O)NC2CCCC(N(C(CCOCC#C)=O)C)C2)ccc([N+](=O)[O-])cn1 C1(OC)CN(C)C(C)(C(=O)NC2CCN(C(c3nccnc3C)=O)CC2)C1 C1(C(=O)NC2(CCNC(C=CC(C)(C)C)=O)CC2)CCN(C2CC2)C1=O c1(OC)ccc(COCC(=O)NC23CC(C2)N(C(C2CC24CCOC4)=O)C3)cc1 N1(C(Cc2c(C)noc2C)=O)CCC2(CCCN2C(=O)CC2CCC(C)(C)C2)C1 c1(C(N2CC3N(C(C(CC)=O)=O)C3C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1Cl Cc1cc2[nH]c(C(N3CCCN(C(=O)CC(=O)NCC4CC4)C(C)C3)=O)cc2o1 c1(CC(=O)OCC)cc(Cl)ccc1NC(c1csc(N(c2ccccc2)C)n1)=O C1(c2n(C)ncc2)CC(CNC(=O)C(=O)N(CCCCCCO)C)C(O)C1 c1(OC)cc(C=CC(N2CC3CCN(C(=O)C(C)CBr)C3C2)=O)ccc1O N1(C(c2cc3nc[nH]c3cn2)=O)CCN(C(c2cnns2)=O)C2CCCCC2C1 CC(C)C1=CCC(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])o3)=O)C23CC3)CC1 C1(NC(c2c(OCC)cccn2)=O)COC2(CCCN(C(=O)CC3(C)CC3)C2)C1 C1(NC(=O)COC2CC=CC2)CCC(NC(=O)Cc2ccnc(O)c2)CC1 c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)C)c[nH]c2c(F)c(F)ccc2c1=O c1(NC(c2c(-c3cnn(CC)c3C)csc2)=O)cccc([N+](=O)[O-])c1Cl N1(C(c2n(CC=C)ccn2)=O)CCCC2(C1)CN(C(=O)CC(O)C(C)C)CCO2 N1(CC)CCOCC1CC(=O)NC1CN(C(=O)C=CSC)CC1C(=O)O N#CC1(C(N2CCCN(C(=O)COCC3CCCO3)CC2)=O)CCSCC1 c1(OC)ccccc1C(=O)NC1CCCC1C(=O)Nc1ccccc1N(C)C C(c1c(C)nn(C)c1Cl)=CC(=O)NCCCCNC(CC1CC(CC)OCC1)=O CCC(COCC1CC1)N=c1[nH]c(=NC)[nH]c(=NCC2(C)CC2(C)C)[nH]1 N1(C(CC2N(C(C3(C(=O)NCC(=O)OC)CC3)=O)CCCC2)=O)CCC(O)C(C)C1 C(=O)(CC1=CCN(C(C2CCCN2C(C)C)=O)CC1)NCC1N(C(C)=O)CCC1 c1(C(=O)NC2CN(C(C(CC)C)=O)C2)cc(Br)c(Cl)s1 C1(C(=O)NCC(C2CCCC2)NC(C(C(C)C)(C)C)=O)CCCCN1S(N)(=O)=O N1(C(C2CN(C(CCCCSC)=O)CC23CC3)=O)CCC2(CCCC2)C1 C1(NC(C2CCCC23CCC3)=O)CC2CCC(C1)N2C(=O)Cc1cc(C2CC2)on1 c1(C(=O)NCC2(NC(CS(CC)=O)=O)CCCCC2C)cn2c(n1)COCC2 c1(C(=O)NCCCCC(C)NC(=O)C=C2CCN(C)C2)ccn2ncccc12 C12(C(=O)NCC3CC(C)N(C(C4C(C)(C)C4(F)F)=O)C3)CCC(F)(CC1)CC2 N1(C(C(=Cc2cn[nH]c2)C)=O)CCCC(CNC(C2C(C)C2C)=O)C1 C=C=C(C)CC(=O)NCc1cccc(NC(C2CCC(C(F)(F)F)O2)=O)c1 C(=O)(C1=CCN(C(c2cnn(C3CC3)c2C)=O)C1)NCCC1ON=C(C)C1 c1(OC)cc(NC(c2n[nH]cc2NC(c2ccc(Cl)c(F)c2)=O)=O)cc(Br)n1 Cc1cc(=NCc2cccc3c2CCN3)[nH]c(NC2CCCC(C)(C)C2)n1 Cc1nn(C)c(C)c1C(=O)NCC1(F)CCCN(C(C2C3CCC(=O)C23)=O)C1 c1(N2CCN(C(C)=O)CC2)nc(=N)nc(N(CCC#N)C)[nH]1 CC(C)=C=CC(=O)N1CC(O)CC1CNC(C1CC2(CC2)CO1)=O CCC(CC)CC(=O)NC1(CNC(C2CC23CCCOC3)=O)CCCC1 Cc1cc(F)c([N+](=O)[O-])cc1NC(C1CCN(C(c2cc(F)ncc2Br)=O)C1)=O Cc1cc(C(=O)NC2CN(C(=O)C(C)(C)O)CC2F)c(S(N)(=O)=O)s1 N1(C(C2CCN(C(CC(CC(C)C)O)=O)C23CCC3)=O)CCc2cccnc2C1 Cn1cc(C(F)(F)F)c(NC(C2CC2NC(C2(c3cn[nH]c3)CC2)=O)=O)n1 N1(C(C(C=C)O)=O)CCCC2C1CCN2C(c1cc(Br)cn1CC)=O Cc1nc(F)ccc1NC(C1CC(C)N1C(C1CC(=C2CC2)C1)=O)=O c1(C(=O)NC(C(=O)N(CC(CC)(F)F)C)CC(F)F)cncc2[nH]ccc12 N1(C(C(CCC=C)NC(C23CC(CN2C2CC2)C3)=O)=O)CCOC2COCC12 C#Cc1cc(C(=O)NC2(C)CCN(C(c3ccnn3C(F)F)=O)C2)cc(F)c1 C1(NC(Cn2nc(C)c(Cl)c2)=O)C2CC1N(C(c1cn(C3CC3)cn1)=O)C2C CC(C(=O)N1CCC(CNC(c2ncn3c2CCC3)=O)C(C)C1)P(C)(C)=O CC1CCCCN1CCCC(N1CCC(N(C)C)C1)=O.c12ccc(cc1)c(=O)[nH]2 CCCC(C)(O)C(=O)N(CC(O)CN(C(=O)Cn1nc(O)ccc1=O)C)C c1(CCC)ccc(C(=O)NC2CCC(NC(=O)CCc3ccc(Cl)cc3)C2)cc1 C1(C(N2CC(C=C)C(OC)C2)=O)CC2CCC(C1)N2C(=O)Cn1ncnn1 c1(CC(=O)NCC2(F)CC(NC(CCCN(C)C)=O)C2)c[nH]ccc1=O N1(C(C2(C)C(C)CCCC2)=O)CC=C(CC(=O)NC2CC(CCF)C2)CC1 N1(C(c2cc(C3C(C)C3)no2)=O)CCC(c2cn(-c3ccncc3)nn2)C1(C)C Cc1cccc(C)c1NC(N(C)Cc1ccc(F)cc1Br)=O c1(SCC(N2CC(CCC(F)(F)F)C2)=O)scnc1C1CCCC1 CC(CCNC(=O)CCc1nc[nH]n1)CCNC(=O)C=Cc1nnc(C(C)C)o1 N1(C(c2cnc(Cl)s2)=O)CCC2(CCCN2C(C2CCC23CCCO3)=O)CC1 N1(C(C2(CC=C)CN(C(=O)CNC(=O)OCC)C2)=O)C2CCCC1CN(C)C2 c1(C(N(C)CCOCCN(C)C(C2CC(F)C(=O)N2)=O)=O)cc(N)ccc1Cl c1(C(=O)NC(C)CCCNC(=O)C(F)=C2CCC2)ccc(C(F)F)cc1Cl c1(C(=O)NCC2(CSC)CCC2)cn(C2CCN(C)C2)nn1 N1(C(CNC(=O)Nc2ccco2)=O)CC2CCC(NC(=O)C3=CCOC3)(C2)C1 S(=O)(=O)(c1cccnc1NCc1cn(C)c(=O)n1C)N1CCCC(CC)CC1 N1(C(c2ccn(CC)n2)=O)CCC(C2(O)CN(C(=O)C3=C(C)CC3)C2)CC1 N1(C(C(C(=O)OC)C)=O)CCC2(CCCN(C(=O)Cc3ccnc(F)c3F)C2)C1 CC(O)(CNC(=O)CSC1CCCO1)CNC(C1CCCC1)=O CCCCC(CNC(c1oc(Br)cc1C)=O)NC(=O)C(C)Cn1cccn1 c1(C(N2CC(CNC(C(COCC)(C)C)=O)OCC2)=O)cnc2n1CCOC2 C1(CC(N2CCCC2CNC(c2n(CC)ccc2)=O)=O)CCCC(OC)C1 c1(C(=O)NCC(CNC(c2c(C)n(CCC#N)nc2)=O)(C)C)cc(O)nc(O)n1 C1(NC(C2(CCNC(c3c(C)nc(C)[nH]3)=O)CC2)=O)CC(C)CC(C)(C)C1 N1(C(c2c(C(C)C)ocn2)=O)C(C(=O)NCCNC(=O)C(C)C)C2CC(O)C1C2 Cc1c(C(=O)NCC2CCCCN2C(C2CC(O)C2)=O)[nH]c2c1CCCC2 C(N=c1cccc(NC(=O)C(F)(F)F)[nH]1)c1ncn(C(C)(C)C)n1 N1(C(c2nc(C(CC)NC(c3coc(C)n3)=O)oc2)=O)CCCC(F)(C(N)=O)C1 N1(C(c2nn(CC)nc2Br)=O)CC2(CCCC2NC(C2CC2C(C)C)=O)C1 N1(C(C2(C)CCN(C(c3cccc(C=C)c3)=O)C2)=O)Cc2ccnn2CC1C N1(C(C(C)(C)C2CC2)=O)CC2(C=C(C(=O)NCC3CC3Cl)CO2)C1 C1(CNC(=O)CSCC(N2CC(F)C2)=O)CCCC(F)C1 N1(C(c2nccc(CNC(CCCC3C(C)C3)=O)c2)=O)CC2C(C1)C2(C)C c12ccc3c(c1)C(C(=O)N2)CCC3.c1(-c2cn(C(C)C)nn2)cnc(C)n1C C(CNC(=O)Cc1ccn(C)c1)(CC(=O)Nc1ccc(SC)nc1)OC c1(CCC(=O)NCCN(CCOC)C(C2COCC(C)O2)=O)ccc(C)cc1C CC1CC(C)CN(C(C)(C)COC(c2cnoc2C2CC2)=O)C1 c1(SC)ncc(Br)c(N(C(=O)Cc2ccc(Cl)cc2F)CC2CCCNC2)n1 c1(C(N2CC(CC(=O)NC(C=C)C)OCC2)=O)ccc(OC)cc1O N1(C(Cc2n(C)cnc2)=O)CCC2(CC(C(=O)NOCC3C=NNC3=O)C2)C1 c1(C(=O)NC2CCN(C(c3c(C)c(Cl)ccc3)=O)C(C)C2)cc2cnccc2[nH]1 c1(C(=O)NC(C2CCCC2)CNC(=O)CCOC2CCC2)ncoc1C1CCCO1 N1(C(C2(C)C=CCC2)=O)CCC(CN=c2[nH]nco2)C(F)(F)CC1 CC(C)C(F)(F)CC(=O)NC1CCN(C(c2cn(Cc3ccccn3)nn2)=O)C1 c1(C(N2CC3C(NC(C(CC(C)C)F)=O)C3C2)=O)cccc2nccnc12 C1(CCC)CN(C(c2ccc(CC)cc2)=O)CCN1C(=O)C(CC#N)n1ccnc1 CC1CCN(C(=O)CCC2CC2)C(CNC(c2ccc(C(C)(C)C)o2)=O)C1 N1(C(C(CC)OC)=O)CCC2(CCCN(C(=O)CNC(C3CCC3)=O)C2)CC1 c1(OCCC(=O)NCc2nc(-c3cccc(F)c3)no2)ccc(Br)cc1 c1(C(=O)NCC2(NC(C3CC4CC4C3)=O)CC2)ccc(CO)o1 C1(C(=O)NC(C)C(CO)NC(=O)Cc2ccsc2C)(CC)CC(C)(C)C1 C1(C(=O)NC2(CNC(=O)COC3CCC3)CCC2)CC(F)C(=O)N1 CCC(CCC(=O)NCc1cccc(C)c1C)NC(=O)C(C)(COC)OC Cc1cnc(C(=O)NC2CCCCC2C(N2CCC2C2CCC2)=O)c(F)c1 Cc1ccc(C)c(C(N2CCC(CNC(C3(C)CCC(=O)NC3)=O)C2(C)C)=O)c1 c1(OC)c(C)cc(CN2CCC3(CC3C(=O)Nc3nc(Br)ccc3C)C2)cc1C N1(C(Cc2c(OC)nccc2)=O)CC(NC(=O)C=Cc2cscn2)C(C2CC2)C1 c1(C(N(C=O)CC2CN(C)C2)C2CC2)ccc(F)cc1 C1(N(C(=O)CCn2cccn2)CC)CCCN(C(c2ncccc2C)=O)C1 C=CC(CCC)CC(=O)N1CCC(NC(c2ccccc2N2CCCC2=O)=O)C1 C#Cc1ccc(C(N2CCCC(CC)(NC(=O)CCNC(=O)C=CCl)C2)=O)nc1 N(C1c2ccccc2CC1C)C(N1CCCC(COC)C1)=O C1(CC)CN(C(=O)CC23CCC(CC2)CC3)CCC1NC(c1cscn1)=O CCCC(O)C(C(=O)O)NCC1CC(CC(C)(C)C)C1 N1(C(CNC(c2c(C(C)C)onc2)=O)C)CCN(C(=O)CC2(O)CCOC2)CC1 C1(NC(c2cnc(C)nc2)=O)CCN(C(c2cccc(N(C)C)c2)=O)C(C)C1 N1(C(C=Cc2c(N)cccc2)=O)CCC2(CCN(c3nnnn3C3CCC3)C2)C1 C=CCC(CC(C)C)C(=O)N1CCCC1CN(C)C(c1n[nH]cc1CC)=O C1(C(=O)NC23C(CN(C(C=C(C)C)=O)C2)C3)CCC(F)(F)CC1 N1(C(c2c(C(C)C)[nH]cc2)=O)CCCCC1C1(NC(C2CCN(C)C2=O)=O)CC1 C(=O)(C(C)(CNC(c1n[nH]cc1C#C)=O)CC)N1C(C#C)CCC1 Cn1ncc(C(=O)NC2CN(C(=O)Cc3cccnc3O)C3CC23)c1Cl N1(C(CCS(C)(=O)=O)=O)CC2CCC(C1)N2C(c1ccc(F)cc1Br)=O n1(CCN(C(C(F)=C(C)C)=O)C)cc(CC(C(=O)N(C)C)C2CC2)nn1 c1(C(N(C2CCCC(NC(Cc3c(C)scc3)=O)C2)C)=O)ccc(N)c(F)c1 C1(CNC(c2cccc(OC(F)F)c2)=O)CC2CC2N1C(=O)C=Cc1ccco1 N1(c2nccc(C(=O)OCC)n2)CCS(=O)(=O)C(CCNC(=O)CSCC)C1 c1(C(=O)NC(C2N(C(C(=O)NC(C)C)=O)CCC2)C)ccnc2c1nnn2C CCC(CNC(c1sc(NC2CC2)nc1C)=O)(CC)NC(C1CC=CCO1)=O N1(C(=O)C2=CCOCC2)CC2CCC(NC(C3CC4CCC(C3)S4)=O)CC2C1 c1(CC)c(C(N2CCCC(CCNC(=O)C(O)C(F)F)C2)=O)cccc1C c1(C(=O)NCC(CNC(CC=CC=C)=O)C)cc2cccnc2s1 C(=O)(C(CC=C)C(C)C)N1C(CN(C(c2nccc(C#C)c2)=O)C)CCC1 C1(C=O)C2CCC(F)(F)C12.N1(C(CCC2(OCC)CCC2)=O)CCC(C(C)N)C1 C1(CC(=O)NC(C)CCN(C(=O)CSc2ccccc2O)C)CC2(CCC2)CO1 Cc1n[nH]c(C)c1S(=O)(=O)N(C1(C#N)CCNC1)Cc1ncnc2c(Br)csc12 c1(C(=O)NC2CCC(C(N=c3cc(C)o[nH]3)=O)CC2)c(F)ccc([N+](=O)[O-])c1F N1(CC(=O)NC(C2CCN2C(=O)C=CSc2nc[nH]n2)C)CCCC1C(=O)NC c1(OC)ccc(C(=O)N(C(=O)CC2CCC(C(F)(F)F)N(C)C2)C2CC2)nc1Br c1(CC)cc(F)ccc1C(=O)NCC1CCCC1NC(=O)C1=C(Cl)CCC1 C(C(F)(C(=O)Nc1cc(C)c(F)cc1O)C(C)C)NC(C1(OC)CCOC1)=O c1(C(=O)NCC2CCC(NC(C3(CC)COC3)=O)C2)ccc(-c2ccsc2)cc1 C1(CC(=O)NC(CN(C(c2ncn(C)n2)=O)CC)C)CCc2ccccc2C1 C12CCN(CC1)C2=O.c1(CC(N2CCC(C(CC)=O)C2)=O)cccnc1 O=C(C1=CCOC1)NC1CN(C(c2cccc(-c3ccccc3)n2)=O)C2CC12 Cc1csc(=O)n1CCC(=O)NCC1CCC(NC(=O)CSC2CC2)C1 CC1=C(C(=O)NCC2CN(C(=O)C(C)CC3CCC3)C(C)(C)C2)CCO1 c1(N(C)CCN2CCCCC2)ccc(-c2cc(CN)[nH]n2)cc1 C1(NC(c2ccc(C(F)F)cc2)=O)CN(C(=O)Cc2sc(O)nc2O)C2CC12 CC(C)C(C)(CNC(c1cc[nH]c1)=O)NC(C1CC1F)=O C1(C(=O)NC2CCN(CC)C2)(CC)CCN(C(=O)C=CC2CCC2)CC1.CCF Cn1nc(Br)cc1C(=O)NCC1(C)CCCC1NC(C1CC1(C)C)=O C1(C)(C(NOCCCOC)=O)CC(O)CN1C(c1c[nH]nc1C1CC1)=O c1(C(N(C(C)CNC(=O)CCN2CCCCC2)C)=O)cc(N)cc2ccccc12 C1(NC(C#CC(C)(C)C)=O)CN(C(=O)CN(C2CCSC2)C)C2(CCC2)C1 C=CCCC(=O)NC(CC1CC1)C(=O)NCC(=O)NC(C)C c1(CC(=O)NC2C(C)(CNC(CNS(NC)(=O)=O)=O)CCC2)c[nH]c(=N)nc1O C1(NC(C=C(C)C(F)F)=O)CCN(C(=O)C=Cc2ccoc2)CCC1(F)F N1(C(C(CCC)CCC)=O)CCc2sc(CNC(=O)COCC(=O)OC)nc2C1 N1(C(=O)OC(C)(C)C)CCC(CN(CC(F)(F)C(=O)O)CC(=O)O)C(F)(F)CC1 N(C(=NCC1C(C)(C)C1(C)C)NCC1(C#N)CC1)C(c1cccs1)C c1(C(C(=O)NC(C)C)N(c2ccccc2C)C(C(C)SC)C)nc(Cl)ccc1Cl CCN=c1[nH]c(C)c(C(=O)NC2CN(C(=O)C(C)=CC)CC23CC3)s1 c1(CN=[N+]=[N-])c(N2CCS(=O)(=O)CC2C2CC2)nc2n1CCCC2 C=CC(C)(CCOC)C(=O)N1CC(C(C(N)=O)NC(c2ccc3nccn3c2)=O)C1 c1(C(=O)NCCC(C)NC(c2cc[nH]c2-c2ccccc2)=O)ccc(F)cc1Cl C(=O)(CC1=CSC2=NCCN12)NCC1COCCN(C(C(CC)CO)=O)C1 N1(C(c2[nH]ccc(=N)n2)=O)CCN(C(=O)C2=CCC2)C2CCCCC2C1 C(=O)(CCCCCC(C)(C)C)N1CC(C)CN(C(COc2cc(C)on2)=O)CC1C N1(C(C(CC(N)=O)O)=O)CC2CN(C(c3cc(O)nc(O)n3)=O)CC2C1 N(C1CCCn2cnnc21)C(=O)CC1CCN(C(C2CC3CCCC3C2)=O)CC1 c1(NCC(CC)C)ccc(S(=O)(=O)N2CCOCC2CC2CC2)cc1Cl C=CCCCCCCNC(C1(NC(C2C(C)(C)C2(F)F)=O)CCC(C)(C)C1)=O C(CCCC(=O)NC(C)CCF)NC(C(C)C1CCOC1)=O C(=O)(CC(C(F)(F)F)NC(c1ccc(F)c(C2CC2)c1)=O)OC C1(COC)(NC(=O)CCc2cnn(C)n2)CN(C(=O)Cc2ccc(C)o2)C1 c1(C(=O)NC(CC)CN(C(=O)CNS(=O)(=O)N(C)C)CC)ccc2cnnn2c1 C1(CNC(c2cc(C)ncn2)=O)N(C(=O)CN2CCCC2C)CCC1(C)C N1(C(C(c2ccccc2)OC)=O)CCC(C2CC(NC(c3cc(C)c[nH]3)=O)C2)C1 C12(C(=O)NCC3CCN(C(CC(OCC)OCC)=O)C3)CCCCC1NC(=O)C2 C1(C(=O)NCCCC(C)NC(c2c(C)ccs2)=O)COCCN1CC(F)F c1(OC)cc(C(F)(F)F)c2cc(C(N3CC(P(C)(C)=O)C3)=O)[nH]c2c1 Cc1cccc2cc(C(=O)NCC3CN(c4cncc(Cl)n4)CCO3)[nH]c12 N1(C(C2(CC#C)CC=CCC2)=O)CCN(C(c2ncc(Cl)n2C)=O)C2(CCC2)C1 N1(C(C(N2C(CC)CCC2)=O)=O)CCC(C)(NC(C2CCCS(=O)(=O)C2)=O)CC1 O=C(Cc1csc2ccccc12)NNC(=O)N=c1cc2n([nH]1)CCCC2 CCC(O)C(C)C(=O)NCC1(O)CCN(C(c2cnc(C(C)=O)s2)=O)C1 N1(C(c2c(OC)ccs2)=O)CC(C(=O)NC2(C)CCC(=O)N(C)C2)C2(CCC2)C1 C(N=c1[nH]c(N2CCC3C(C2)C3(F)F)nc(=N)[nH]1)c1cc(C(C)C)no1 N1(C(c2ncccc2Cl)=O)CCC2C(C1)CN2C(=O)CCSCc1ccccn1 C(C(O)CCNC(c1coc(Br)n1)=O)NC(c1cc(CO)[nH]n1)=O c1(OC)cnc(Cl)cc1C(=O)NC1CC(C)CN(C(c2cc(C)nc(C)n2)=O)C1 C(CC(C(=O)NCC1(C(C)(F)F)CC1)NC(C12CC(F)(C1)C2)=O)N(C)C c1(C(N2C3(CN(C(c4cc(OC)c(I)cc4)=O)C3)CC2)=O)ccc2c(c1)OCC2 c1(C(N2CC3(CCN3C(c3ccc(C4CC4)c(F)c3)=O)C2)=O)cnc(O)cc1O C(C)(C)(C(C)CC(=O)N1CCC(C2CC2)CC1)NC(C1CN(CC)C(=O)C1)=O CC(=O)CCCCC(=O)N1CC2(CCCC2NC(c2sc(C)cc2C)=O)C1 N1(C(C(CCOCC)NC(C2C=CCC2)=O)=O)CC2(CC=CC2)C1 C1(CNC(C2C(CC)C2)=O)C(C)CCN1C(=O)CCN1CCNC(=O)C1 Nc1cccnc1C(=O)NC(CC1CCCC1)C(N1CCCC(F)C1)=O c1(N(CCC(C)N)C(=O)NCc2c(Br)nnn2C)ccc(F)cc1 C(=O)(C(F)(F)CO)N1CC(CC(C)NC(c2cnc(-c3ncccn3)s2)=O)C1 CCCS(=O)(=O)C(C)C(=O)N1CCCCC1CNC(=O)C(C)c1ccco1 C(=O)(CCCC(=O)NC(C)C)N(C1(C)CC(NC(=O)CC(O)CC)C1)CCC C(C(CNC1(c2nnnn2CCN2CCOCC2)CCOC1)C(C)C)OC C12(CNC(CCC)=O)COCCN1C(=O)CN(C(c1cccc(CO)c1C)=O)C2 C(=O)(C(Cc1cccnn1)OC(c1ccsn1)=O)OC C(=O)(CC(C)(O)CCC)N(C1CCN(C(=O)C(CC)N(C(N)=O)CC)C1)CC#C c1(NC(N(CC)Cc2c(F)cccc2F)=O)ccc(OC)c2c1OCC2=O C1(NC(C2(C=C)CCC2)=O)CCN(C(=O)C(C)=CC(C)(C)C)O1 N1(C(=O)CCC2CCCO2)CCC2CCC(C1)N2Cc1cccc(F)c1F N1(C(COC(CC(C)c2cccnc2)=O)=O)CC(O)C(O)C1 Cc1n[nH]cc1CCNC(C1(NC(c2csnn2)=O)CC1(C)C)=O c1(N(C)CC2CC2)nc(N2CCS(=O)C3(CCC3)C2)nc2c1CCCCCC2 C1(C(=O)NC(C2CCCN2C)C)CC2CC2N1C(C1CCN(C)CC1)=O C12(C(=O)NC(C)C(CO)NC(=O)C(C)OC3CCCCC3)CCC(CC1)CC2 c1(CC)c(C(=O)NC2CCCC2CNC(=O)C(C)C(C)(C)C)cccc1F Cc1nc(NC2CCN(C(=O)CC3CC4CCC(C3)N4C)C2)c2c(C)csc2n1 N1(C(C(CC=C)NC(C)=O)=O)CCC2(CC1)CC2C(=O)N(CCCF)C N1(C(C2(C)CN(C)C(=O)C2)=O)CCN(C(C2CC(F)(F)C2)=O)CC12CC2 C=CCC(C(=O)NCCNC(=O)CCOCC1CCCO1)c1ccccc1.COC CCC(C)(C)C(O)C(=O)NCC(CC1CC1)C(=O)N1CC(C(F)(F)F)C1 C1(C(=O)NCC(C)NC(=O)C(c2cccnc2)C)CCC2CC2CC1 c1(C(=O)NCCC2(N3CCCC3)CCC2)ccnn1CC1CC1.C12(CC1)C(=O)N2 C(C(COC)C(=O)NCC(c1ccc(C)cc1)NC(c1sc(F)cc1Cl)=O)OC N1(C(C2(COC)CCOC2)=O)CCC2C(C1)CN2C(c1cccc2scnc12)=O C1(NC(C=C(C)C(F)F)=O)CN(C(c2ccc(C3CC3)c(F)c2)=O)CCC1C C1(NC(c2ccc(CNC(=O)C=Cc3ccsc3)s2)=O)CC2C=CC1CC2 Cc1ccc2occ(C(=O)NCC34CC3CN(C(c3ccc(Cl)cc3)=O)C4)c2c1 CN1CC(O)CC1(C)C(N1CCCC(NC(c2cc(O)ccc2F)=O)CC1)=O C1(N(C(C(COC)C)=O)C)CN(C(C2(O)CCC2)=O)CC1F C1(CNC(Cc2c(C)cccc2C)=O)CC2CC(C1)N(C(=O)CC1CC(F)(F)C1)C2 N1(C(c2ccn(CCF)n2)C(=O)NCCCOC)CCN2C(CNS2(=O)=O)C1 c1(NCC2OCC(CNC(c3cc(C)c(CSC)o3)=O)C2)cnc(C#N)cn1 C1(C(C)=O)CC(C(=O)NC2CC(NC(=O)C(C)(C)c3cccs3)C2)C1(C)C C1(O)(CN(C(COC)=O)C)CCCN(C(C2CCC(=O)N(C3CC3)C2)=O)C1 CCC(CCC(=O)Nc1cnn(C)c1C)NC(c1cnn(C)c1CC)=O c1(CC(N2C(CNC(=O)Cc3cnsc3)CC(F)C2)=O)coc2ccc(F)cc12 N1(C(C2C(c3n(C)cnc3)C2)=O)CCC(F)(NC(c2cccc(Br)c2F)=O)CC1 N1(C(C2CC(N(C(=O)CC3(O)CCCC3)C)C2)=O)CCc2ccsc2C1 CC1CC2(CCN(C(=O)C3=COCCC3)CC2)CN1C(C1CCCC(C#N)C1)=O c1(OC)c(NC(C2C3CCC2(c2ccccn2)C3)=O)cccc1C(=O)O c1(CN2C(C(C(=O)OC)(C)C)CCCC2)cn2c(n1)CCCCC2 C1(SC)CCCC1n1cc(C2(C)CN(C(C3CCCN3C(C)C)=O)C2)nn1 C1(CN(C(C(C)n2cccc2)=O)C)CN(C(c2cc(C(N)=O)c[nH]2)=O)CCO1 C1(NC(C(CCCC)=O)=O)CN(C(c2cn(C(F)F)cn2)=O)C2(CCC2)C1 C1(NC(c2coc3c2COC3)=O)CC2CN(C(C3CN4CCN3CC4)=O)CC2C1 O=C(C1=C(c2ccc(F)cc2)CCOC1)NCC(CO)C(F)(F)F C1(C(=O)OC)CCC(C)(C(=O)NCC2CCCN2C(C2(C)C=CCC2)=O)C1(C)C c1(C(=O)NCC(c2ccccc2)NC(CSC(=N)N)=O)[nH]cc2c1CCCC2 CN1N=C(C(=O)NC2CC(NC(c3c[nH]nc3Br)=O)C23CCC3)CCC1=O CC1(CC(=O)O)CCN(CCNC(C2(c3ccccc3)CCC2)=O)C1 C(C)(CCC(=O)N1CCOC(CNC(c2cn(CCC(C)C)nn2)=O)C1)OC N1(C(C(C)n2ccnc2)=O)c2ccccc2CC1CN c1(C(C)C)cc(O)nc(SCC(=O)NCCc2ccc(N3CCOCC3)nc2)n1 c1(OC)ccc(C(=O)NC(C)CC2CCN(C(c3cccs3)=O)CC2)c(C)n1 N1(C(c2nc(C)oc2)=O)CCC(NC(=O)C(c2cnn(C)c2)=O)CC1C c1(OCCC(=O)NCCN(CCC)C(C2CCN(C)C2)=O)ccccc1C(C)C c1(C(=O)NCCC2CCN(C(c3cc(C(=O)OCC)n[nH]3)=O)C2)cncc(C)n1 C1(C(N2C(CNC(CCN(C)CCO)=O)CCCCC2)=O)CCc2nccn2C1 C1(NCCC2(C)N=N2)CN(C(=O)OC(C)(C)C)CC12CCC2 CN1CC=C(CC(=O)N2CCC(C)(C(=O)NCC(c3cccnc3)O)CC2)CC1 C12(C(=O)OC)CCN(C)CC1CN(c1nnc(C(C)(C)O)n1CC(C)C)C2 N1(c2snc(CCC)n2)CCC(C)C(NC(=O)C(C)(c2ccccc2)OC)C1 Cc1csc(C=CC(=O)NC23CC2CN(C(C2(c4ncco4)CC2)=O)C3)n1 N(C1CCOc2ccc(O)cc21)C(C(c1ccccc1-c1ccccc1)OC)=O c1(CC(C)=O)cccc(C(=O)NC(C)CN(C)C(c2nnc(C)o2)=O)c1 C(=O)(C1CCCc2ncnn21)NC1(C)CCCN(C(CCC#C)=O)C1 c1(C2(NC(C(Cc3ccc(OCC)cc3)C)=O)CCC2)cc2ccccc2o1 CCCC(C#N)C(=O)N1CC(NC(c2cc(-c3cnn(C)c3)on2)=O)CC1(C)C N1(C(COCC#C)=O)CC(NC(=O)C(CC#C)C2CC2)C(O)C1 N1(C(C=CCOC)=O)CC2CCC1C(CNC(=O)C(F)CC1CC1)C2 N1(C(CC2(CNC(Cc3nc(C)sc3)=O)CC2)=O)CCc2cc(F)c(F)cc2C1 c1(OC)ccc(C(=O)NCC2CC(OC)CN2C(C2CNC(=O)N2C)=O)cc1F c1(CN(C(=O)NCC(=O)OCc2ncc[nH]2)CC2CCOC2)ccc(Cl)cc1 CC1(C)CCC(C(=O)NC2(C(=O)Nc3cc(F)ccc3O)CCSC2)CO1 N1CCCC12CCN(C(C1N(C)CCC1)=O)C2.c1(C2(CC)CC2)cc(O)cc(Cl)c1 N1(C(CC(C)(C)NC(=O)CCN=[N+]=[N-])=O)CCC12CCC(O)CC2 Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(=O)CC=C(Cl)Cl)C(C)C1 C(C)(c1ccccc1C)=CC(N1CC(CC)C(NC(C2CC(C)=NO2)=O)C1)=O CC1(C)COC(CCNC(C2(NC(=O)C(F)F)CCCC2)=O)C1 C(=O)(C(COC)CC)N1CCC(CN(C(c2c(CCC)nco2)=O)C)C1 Cc1cccnc1C=CC(=O)NCCN1CCN(C(C2(C)C=CCCC2)=O)CC1 N1(C(CNC(c2n(CC)ncc2)=O)C(F)F)CCN(C(=O)CC2CCOC2)CC1 c1(OC)cc(N2CC3CC(NC(c4csnn4)=O)CC2C3)ccc1[N+](=O)[O-] C1(C(=O)NC2CCC23CN(C(c2cc(Cl)c[nH]2)=O)C3)CCc2nccn2C1 C1(COC)CN(C(c2ccnn2-c2ccccc2)=O)CCN1C(C1CC1(F)F)=O CC(O)C(C)(C)C(=O)NC1CN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 NS(=O)(=O)c1n[nH]cc1C(N1CCC12CN(C(c1ccnc(Cl)c1O)=O)C2)=O C1(O)(CNC(=O)NCCN2CC(C)OCC2)CCC(C)(C)C1 N1(C(c2cccc(C(=O)OC)n2)=O)CC2(CCC(CNC(C3CC3CF)=O)O2)C1 C(c1cncc(F)c1)=CC(=O)NC1CC(NC(c2cccc(Br)c2)=O)C1 C(C)(C)(CC(=O)NC12CCN(CC1)C2)NC(C(C)c1cccs1)=O N(C(=NCCN1CCN(C)CC1)NCC1CC1)C(c1ccc(N(C)C)cc1)C c1(C(=O)NCC(C)N(C(C(C)OCC#C)=O)CC)cnc(CCC(F)(F)F)s1 C(=O)(CCC(=O)N1CCC(F)(CNC(C2CCC(C)(C)O2)=O)C1)NC N1(C(C2C3CN(C(C(C)Sc4cccc(C)c4)=O)C2C3)=O)CCCC2(COC2)C1 N1(C(C(CCSC)O)=O)CCN(C(=O)C=Cc2ccc(F)cc2)CC1CC(F)F C1(CNC(C=CCC)=O)CCCC(OC(=O)C=Cc2ccncc2)C1 C(=O)(CCC(C)(C)C)N1C(CN(C(C2CCCN(C(CC)=O)C2)=O)CC)CCC1 N1(C(C2CCC(C(C)(C)C)CC2)=O)CC2CCC(NC(=O)C=C3CCC3)CC2C1 C12(C(N(CCCNC(=O)CC3C=CCCC3)C)=O)CCC(CC1)C2 c1(C(N(C(C(=O)NCC2N(C)CCOC2)CC(F)F)C)=O)cc(C#N)ccc1N c1(OC)nscc1C(=O)NC1CC(O)C1CC(=O)NCC1CCC(C2CC2)O1 C1(NC(c2cn(CC=C)nn2)=O)CCN(C(=O)Cc2c(Cl)cccc2Cl)C(C)C1 CCC(CC)(CCC(=O)OC1CCCC(S(C)(=O)=O)C1)[N+](=O)[O-] C(=O)(C(O)C(F)(F)F)NCC(C)(C)CNC(=O)CC1(n2cccn2)CCC1 c1(C(N2C(CCNC(CC#C)=O)CCCC2)=O)ccc(NS(C)(=O)=O)cc1Cl c1(COC)nc(C)c(C(N2CC(C)(NC(=O)C(C)NC(=O)COC)C2)=O)s1 N1(C(C(C2CC2)OC)=O)CC(C2CN(C(c3ncc(Cl)cc3Cl)=O)C2)C1 CCC(C)(CNC(=O)C(F)(F)C1CCCC1)NC(c1cccnc1)=O C1(C(=O)NCC=C2CCN(C(c3c(C)ccnn3)=O)CC2)CCC2(C1)CC2(F)F Cc1ccnc(CNC(=O)N(C)Cc2nnn(C(C)C)n2)n1 CC1(C)CCOC1C(=O)NCCC1(C)CCN(C(c2cccc[n+]2[O-])=O)C1 CCCCC(CC)C(=O)N1CCN(C(c2cc3n(n2)CCOC3)=O)CC1CCC O=C1COc2cc(F)c(C(N3CCC(NC(C4CNC(=O)N4)=O)C3)=O)cc2N1 C1(C(=O)NCC(C)NC(=O)C(=O)NCC(F)(F)F)CCCN1C1CCCC1 C1(CNC(c2ccc(C)cn2)=O)COCCN(C(=O)CC2(C)CCCO2)C1 c1(OC(C(=O)NCCN(C(=O)C(C)(O)CC)CCC)C)ccc(F)c(F)c1 c1(C(=O)NCC2CCN(C(C(n3c(C)ccn3)C)=O)C2)nnc(Cl)cc1N c1(C(N2C(CNC(=O)C3=CCCC3)CC3(CC3)C2)=O)cnc2[nH]ccnc1-2 O=[N+]([O-])c1cnn(CCN2CCOC(c3cn(CC(O)CO)nn3)C2)c1 c1(-c2nc(C)c(F)cc2)n[nH]c2c1CN(C(c1c(F)cc(O)cc1F)=O)CC2 c1(OC)ccc2ncc(C(=O)NC3CN(C(=O)CN(C)S(N)(=O)=O)CC3F)n2n1 N1(C(CCC2CC(OC)C2)=O)CC(C2CN(C(=O)C(C(C)(C)C)NC(N)=O)C2)C1 c1(C(=O)NN(CC=CC(=O)NC(C23CCC(CC2)C3)C)C)ccnc(C2CC2)c1 Cc1cc(-c2cn(CCCC(=O)NC3CCCOC3(C)C)nn2)c(C)cc1Cl CCC(C)(COC)CNC(=O)C(c1cn(C)nn1)NC(=O)C(C)=CC1CC1 C(=O)(C1CCc2cccnc21)N1CCCCC(N(C)C(c2csc(CO)n2)=O)C1 C1(C(=O)NC(C)(CNC(=O)CC2C=CCC2)C2CC2)CC2(C1)CC(F)(F)C2 N1(C(c2nnn(CC)c2C)=O)CCN(C(c2csc(Cl)n2)=O)CC1CC(C)(C)C C1(C)(C(=O)NCCCNC(c2c(OCC(C)C)nccc2)=O)CCCC1(F)F C(=O)(C(C)Cc1ccncc1)NCC(C1CCCCC1)NC(CC=CCC)=O CC1CCC(C(N)=O)CN1C(C1(C)CCCN1C(=O)CC1(C)CCC1)=O CCCC(C)CC(=O)N(CC(=O)NCC(C)OC)CCn1cc(C)cn1 c1(C(=O)NC2CC(F)(CNC(CC(C)C)=O)C2)cnn2c(=O)cc[nH]c12 C(C(C(C)(C)C)NC(=O)Cn1ccc(C(F)F)n1)NC(C1(C)C(C)C1)=O C(C)(C)(CCCNC(=O)C(C)(C)F)NC(C1C(C(=O)OC)COC1)=O C1(CNC(C(n2ccc(C)n2)C)=O)CC2(CCC2)CN1C(=O)OC(C)(C)C N1(C(C=C(C)C(C)(C)C)=O)CCC(O)(CNC(=O)CCc2ccnc(Cl)c2)C1 C1(NC(=O)C=C2CC2)CC12CCN(C(=O)Cc1ccc(F)cn1)CC2 c1(CC2CCCN(CCCl)C2)cccc2ncnn12.C12(CC1(F)F)C(=O)N2 c1(CC)ccoc1C(=O)NC(CNC(C1CC1(F)F)=O)C(C)C c1(COC(C2C(NCc3cccc(SC)c3)C2)=O)ccc(OC(F)F)cc1Cl C1(C(=O)NCc2cccnc2F)CCC2(CC2)N1C(c1csc(Cl)c1)=O CC1(C)CN(C(=O)COCC2CC2)C(CNC(c2coc(Cl)c2)=O)CO1 N1(C(c2c(C)[nH]cc2)=O)CCC(C)CC1C(=O)NC(C1(CO)CC1)C N1(C(C(C)(C)SC)=O)CCCC(F)(CNC(c2cc(C)c(O)nn2)=O)C1 C#CC1(C(=O)NCCCC(O)CO)CCN(C(=O)C(C)CSC)C1 C1(COC)CC2(CCN2C(=O)CC(CNC(C2CN(C3CCC3)C2)=O)C2CCC2)C1 N1(C(C(C)OCCOC)=O)CC(C2CN(C(c3sc(F)cc3Cl)=O)C2)C1 C1(NC(Cc2cn(C)nc2)=O)CCN(C(=O)CN2C(=O)CNC2=O)CC12CCC2 C1(C#N)(C(=O)NCCN(C(c2c(N(C(C)=O)C)cccc2)=O)C)CCCOC1 N1(C(C(C)=C(C)C)=O)CCCCC1CC(=O)NCc1nn[nH]n1 c1(C(N2CC(C(=O)Nc3ccc(CC#N)cc3)C2)=O)cc(Cl)cc(Cl)n1 C1(NC(c2cc(C(C)=O)sc2)=O)CC(C(=O)N(C2CCOC2)CCF)C(O)C1 c1(CC(=O)NC(C)CCCNC(c2c[nH]cc2Br)=O)noc2ccc(F)cc12 c1(C(N(C2CCN(C(c3cc(C(N)=O)no3)=O)CC2)C)=O)cc2cccnc2s1 N1(C(C(CCC)C)=O)CC2CC(NC(c3cccn(C)c3=O)=O)CC1C2 C1(CC=C)(C(N2CCOCC2C)=O)CCCN1C(=O)C(O)C=CC C1(S(C)=O)(C(=O)OCC)CCN(C(C2CC(=O)N(c3cccc(C)c3)C2)=O)CC1 CC1(C(=O)NCC2(CCNC(c3cc(F)ccc3F)=O)CC2)CCC(=O)CC1 C(=O)(C1=CC2CCC(C1)C2)NCC#CC(N1CC(C)CN(C)CC1)=O c1(CC)ocnc1C(=O)N(C(C)C(=O)NCCCN1CCOCC1)C c1(CCN(C(C(=O)N(C)CC2CCCO2)=O)CC(F)F)cccc(F)c1 C(C(O)CN(C(=O)CCC1CCCO1)C)N(C)CC1CCOC1 C1(C2CC2)(C(=O)NC(c2cn(C)nc2)C(=O)NC2C3CCC(F)C23)CCC1 c1(C(=O)NC2(CF)CCN(C(=O)CCCC3CCCCC3)C2)n[nH]c2c1COC2 C1(CNC(CC2CC(CC)C2)=O)CC12CCN(C(=O)COc1cncc(C)n1)CC2 N1(C(c2c(C)nncc2)=O)CCC2CN(C(c3oc(Br)nc3C)=O)CC12 N1(C(COCC=C)=O)C2CCC1(CNC(=O)Cc1c(C)cccc1C)CC2 c1(C(=O)NCC(CCCC)NC(C2COCC2(C)C)=O)ccc2nccnc2n1 N1(C(C)C)CCCC1C(N1CCC1C(=O)NC1CCCC1F)=O c1(OCC(=O)N(CCCC(=O)NC(c2ccnn2C)CC)C)ccccc1C C1(CN(C)C)CC(O)CN1C(C1CCOCC1NC(c1cnn(CCO)c1)=O)=O C(C)(CCCC(C)C)NC(C=C1CCN(Cc2onc(C)n2)CC1)=O N1(C(c2c(C(=O)O)cn[nH]2)=O)CCC2CC1CN(Cc1ccccc1)C2 Cc1cc(CCC(N2CCCC(CNC(=O)C(C)(C)c3cncs3)C2)=O)n(C)n1 c1(C(=O)NC(C(C)C)C)occc1CNC(=O)CC1(C(=O)O)CCC1 C1(NC(C(C)CO)=O)CCN(C(=O)C(c2ccc(F)cc2F)(C)C)CCC1CO Cc1csc(C(=O)NCCC(O)CNC(c2ccccn2)=O)c1 C1(C(N(CCCCCCCC)C)=O)CN(C(=O)C(CCC)OCC)CC12CCC2 C(=O)(C1=NOC(C)C1C)N1CC(C(=O)Nc2cnn(CC)c2C)(CC)C1 CC1(C)CCN(C(=O)CP(C)(C)=O)CC1C(=O)NC1CCCSCC1 N1(C(C2C(C)CC(=O)NC2)=O)Cc2[nH]nc(C(=O)NCCCC3CC3)c2C1 N1(C(c2c(C(C)(C)C)ocn2)=O)CCOCC1CC(=O)NC1CC(CC2CC2)C1 CC1CC(NC(C2CCC(F)CC2)=O)CN1C(C1CC(=O)N(C)C1)=O C(=O)(C(CC1CCCC1)NC(=O)C(C)OCOC)NCCCC c1(CC(N2CC(C(N(c3csc(Cl)n3)C(C)(C)C)=O)C2)=O)ccccc1C(F)(F)F C1(CCNC(CSCCC)=O)CN(c2cc(C)nc(CO)n2)CCS1(=O)=O C(CCCCCC(=O)NCC1(C2CC2)CC1)NC(c1n(C)c(Cl)nc1)=O N1(C(C2C(C(C)(C)C)C2)=O)CC2(CNC(=O)CCCOC(F)F)CC1CO2 C1(CC(N)=O)CN(CC(=O)NC2CCNC(=O)C2)CCO1 c1(N2CCC(N(C)C(C3CCCN3C3CC3)=O)C2)ncnc2c(Br)nn(C)c12 C=CCC(C)(C)CC(=O)N1CCCC(C)(C)C1CNC(c1cc(=O)n(C)cn1)=O C(CC(C)C)(C(=O)NCC(C)C)N(C(COC)=O)C N1(C(c2scc(C)c2)=O)Cc2c([nH][nH]c2=NC(=O)c2ncccc2Br)C1(C)C N1(C(C2N(CC)CCCC2)=O)C(CC(=O)NCC2OCCC2C)C2CCCC12 N1(C(C(C)OCC)=O)CCC2(CCCC2NC(=O)Cc2csc(Cl)n2)CC1 n1(C(C)(C)C)ccc(C(=O)NCCC2CC2CNC(=O)CC2CCOCC2)c1 C1(NC(C2C3CCCC23)=O)CC2(CCN(C(c3cc(CO)ccc3O)=O)CC2)C1 CC1ON=C(C(=O)N2CCN(C(c3cnc(N)c(Br)c3)=O)CCC2C)C1C Cn1ncc(Cl)c1CC(=O)NC1CCC(F)(CNC(=O)Cn2nnc(=O)[nH]2)C1 C1(NC(C(C#C)(C)C)=O)CCN(C(=O)CCN(CC(F)(F)F)C)CC1(C)C Cc1ncc(Cl)c(C(=O)NC2CCC(NC(C3CC34CC4)=O)C2)n1 N1(CC(=O)N(CC#C)CCN)CCCC(NC(=O)OC(C)(C)C)C1.CO C#Cc1ccc(C)c(NC(C2CC(NC(=O)CCc3cncnc3)C2(C)C)=O)c1 CC(CCNC(=O)CCc1cccc(F)c1)CCNC(C1CC1(C)C(F)F)=O c1(N2CC(C)(C(F)F)OCC2)ccc(S(=O)(=O)NC(C)(CO)CCF)cc1C#N CC(C(C)(C)C)=CC(=O)NC(C1CCCN1C(=O)C(C)n1cccc1)C N1(C(c2ccn(CCC)n2)=O)CC2CCC(C1)N2C(c1cncc(C(F)F)c1)=O CCC(CC)CC(=O)N(C1CCC(NC(c2cnc(C(=O)OC)cn2)=O)CC1)C Cc1ccc(O)c(CC(=O)NCC2(NC(C3CC(C(F)(F)F)C3)=O)CCOC2)c1 CON=CC(=O)N1CCC(CCNC(=O)CCC2CC2(Cl)Cl)C1 c1(NC(C(C)N(C(COC(CC)C)=O)C2CC2)=O)cc(C)cc(Cl)c1 N1(C(COCc2c(C)cccc2)=O)CCC(NC(=O)CN=S(C)(C)=O)C(C)C1 Cc1cc(C)c(C(N2CC3(CCN3C(=O)C(C)C(O)C(C)C)C2)=O)cc1N C12(C(=O)NCCCC(c3ccccc3)NC(C(C)SC)=O)CCCC1C2(F)F C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CC2CCC1CN(C(C1CSCCS1)=O)C2 c1(C(Cc2nc(CC)sc2)=O)cc(C(=O)NCC2CC2)nn1C.C1=CCNC(=O)C1 C(CCC[Si](C)(C)C)N(C(=O)C(C)(C)n1cccn1)C.c1cccc(F)c1 C1(NC(=O)CSc2ccccn2)CC2CN(c3cncc(Cl)n3)CC12 C1(NC(C(C)C2CCC2)=O)CCCCN(C(=O)C(c2ccccc2)O)CC1 N1(C(C2CC(OC)(OC)C2)=O)CCC(CC(=O)NCC(F)(F)Cl)CC1 N1(CC(=O)NC(CNC(c2c(C)ncs2)=O)C(C)C)CCCCCCC1=O c1(C(=O)NCC2N(C(C(C)(C)C)=O)C3C(C2)C3)cnc2c(Cl)cccn12 Cn1nc2c(c1C(=O)NCC1C=CCN1C(=O)CC1CCOC1)CSCC2 c1(NCC(=C)Cl)cc(Br)ccc1S(=O)(=O)NC1CCOC(c2ccncc2)C1 c1(C(N2C(CC(=O)NCCC3=CCCCC3)CC(F)C2)=O)cnc2c(c1)COC2 c1(C(=O)NC2CCC(C)(CNC(C3(COC)CCC3)=O)C2)cccc2[nH]ncc12 C(=O)(CCCCN=[N+]=[N-])N1CC2C(CC(=O)NC(c3nc[nH]n3)CC)(CC2)C1 c1(OC)nccc(NC(=O)COCC2CC2)n1.C12CCCC(C1)NC1CC(C1)N2 C(F)(C(=O)N(CC(=O)N(CC(C)OCCOC)C)C)=C(C)C.CCO Cc1cccc(C(N2CCCC(NC(=O)CC3CN4CCN3CC4)CC2)=O)c1O N1(C(C2CCCCO2)C(=O)NCCCOC)CC(C)CSc2ccccc21 C1(CNC(C(c2c(C)cccc2)C)=O)CN(C(c2cc[n+]([O-])cc2)=O)CC1(C)C C1(C(=O)NC(C2CN(C(=O)CC(C)(C)O)C2)C)CCC2(CC1)CC2 c1(CCN(C(NNC(c2cncc(CC)c2)=O)=O)CC)cn(C)c2cc(F)ccc12 N1(C(CCC=C)=O)CCC(C)C1CNC(c1cnccc1OC)=O N1(C(=O)OC(C)(C)C)CC2(C1)CN(C(C1(Cc3ccc(C#N)cc3)CC1)=O)C2 C1(N(C(C2CCCCC2)C(=O)NC2CC2)C)CCCN(C(=O)CSC2CCC2)C1 c1(CC(=O)NCC2(C(N)=O)CN(C(=O)CCC=CBr)C2)ccccc1[N+](=O)[O-] C1(C(C)C)CC(NC(N2CCOCC2CC(c2ccccc2)O)=O)CCO1 c1(C(N2CCC(NC(C3CC(OC)C3)=O)C2)=O)cccc2c1COCC2 c1(CC(=O)NCC(C)N(C(=O)C(C)SC)CC)csc(C(C)OCC)n1 c1(C(N2CCC(C)(CNC(Cc3c(C)ocn3)=O)C2)=O)ccc(C(F)(F)F)nc1N N1(C(CC(=C)C)=O)CCC(CNC(c2sc(Cl)c(Cl)c2OC)=O)C12CCC2 C(CC(F)CN=[N+]=[N-])NC(C(CC=CC)NC(C1CCCCN1C)=O)=O C1(NC(C2N(C(=O)OC(C)(C)C)CC(C)OC2)=O)CCOCC12CCC2 C1(C)(CNC(CCCC=C)=O)CN(C(=O)C=Cc2cncs2)CCO1 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCCNC(c1sc2cc(C)sc2c1)=O C1(C(N2CCC(N(C(=O)CC3CC(C)(C)C3)CC)C2)=O)CC(=O)OC1(C)C N(C1CS(=O)(=O)c2ccccc21)Cc1nc(-c2ccc(SC)s2)sc1 C1(CNC(CCc2ccc(C)cc2)=O)N(C(=O)C2=CCCC2)CCC1(C)C C=CC1COCC1NC(c1ccoc1CNC(=O)C(CN(C)C)CC)=O C(C(C)(C)CC(=O)N1CCCC1(C)CNC(=O)CCC=C(C)C)OC C=C(C)CC(=O)N(CC(CC)NC(C1CCCC1)=O)C N1(C(C)C(=O)NC2CC2)CCCC(NC(c2ccc(C3CCCO3)[nH]2)=O)C1 N1(C(CC(C)(C)OC)=O)CC(C)N(C(=O)Cn2ccc(C(=O)OC)n2)CC1C C1(N(C(c2ccc(C)n2C)=O)C)CN(C(=O)C(F)(F)C2CCCC2)CC1(C)C CC(C(=O)NN1CCCC1C(=O)N=c1ccn(C)[nH]1)C1CCCC1 c1(COCC2C=CC(Nc3ccc(C(CF)OC(C)=O)cc3)C2)ccc(C)cc1 C1(C2CCN(C(=O)CC3CC=CC3)C2)(NC(c2c(Cl)ccc(OCC)n2)=O)CC1 C1(OCc2cn(CC(COC)O)nn2)CCCN(C(=O)COCC(=O)NC)C1 C1(C(=O)NC(CC)(C)CNC(=O)Cn2ncnn2)CNC(=O)C(C)(C)C1 n1(-c2ccc(C(=O)NC(C)C(c3ccccc3)C)s2)nnc2ccccc12 C(=O)(C1CCc2cccnc21)N(C)CC1(O)CN(C(C2CC(F)C2)=O)C1 CS(=O)c1cc(C(=O)NC2CC(F)(CNC(C3CCC(=O)O3)=O)C2)ccc1F C1(C(=O)NCC2(O)CN(C(C3CC4CCCC34)=O)C2)(COC)CCOCC1 Cc1cc(C(N2CCC(NC(=O)C=CC3CCC3)C2C(C)(C)C)=O)ncc1C#N N1(C(C(C)NC(=O)NC)=O)CCC(NC(C2(C)CC3CCC2C3)=O)C(F)C1 CC(C)(CC(=O)O)NC(=O)CC1CCCC1(C)C CC(C(=O)NCCCCC(C)NC(C1CCC2(CCC2)O1)=O)S(C)(=O)=O CN1CCN(C(C2COCCN(CC(O)CO)C2)=O)CC1c1nccn1C C(=O)(C(C)C(O)C(C)CC)N1CCCC(F)(CNC(CC(=O)NCC#C)=O)C1 C(=O)(C1CCCc2nc[nH]c21)NCC#CCNC(C1=NOC(C)C1)=O C1(NC(=O)C2=COCCO2)CCOC2(CCN(C(C34CCC(C3)C4)=O)CC2)C1 C(C(C)(O)CC(=O)N1CCN(CC(=O)Nc2c(C)cccc2O)CC1)OC c1(OCC(=O)NC2N(C(C(C(=O)OC)C)=O)C3C(C2)C3)ccc2c(c1)CCC2 N1(C(=O)C(N2CCOCC2)Cc2cccs2)CCCC1C=Cc1ccccc1 N1(C(CCC=CC)=O)CC2CC2(NC(=O)CSc2ccccc2Cl)C1 C=CCCC(C(=O)NCCCCC(C)(F)F)NC(=O)CCCN=[N+]=[N-] N1(C(c2csc(C)c2C)=O)CC(C)CCC1CNC(c1ccc(C(N)=O)s1)=O CC1(C)C2CC(C(N3CCCC3(C)Cc3ccccc3Cl)=O)CC12 C1(C(=O)NCCC2CCCCN2C(=O)CSCCC(C)C)(CC)CCC(O)CC1 c1(C(N2CCC(=CCNC(C(C)SCCCC)=O)CC2)=O)coc2c1CCCC2 N1(C(C(CC(CC)C)=O)=O)CCC2(CCCCC2NC(=O)C=C2CCC2)CC1 Clc1ccccc1C1CCN1Cc1c(CNc2nccc(N3CCCC3)n2)n[nH]c1 C1(NC(c2cn(C(C)C)nc2)=O)CCC12CCN(C(=O)CN1CC3CC3C1)CC2 c1(C(N2CCN(Cc3cccc(OC)c3)CC2)C(=O)NCCC)cccnc1C C1(C(=O)OC(C)(C)C)N(C(=O)OCC(N2CCCC2)=O)CCC1(C)C.CC1CO1 c1(C(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)c(Cl)sc2nnsc12 C(C(=O)NCC(F)CNC(=O)CNS(N)(=O)=O)(C(C)C)OCC Cc1noc(C)c1C(C)C(N1CCC(Cn2cc(C(C)CC3CC3)nn2)CC1)=O O=C1OC2CCN(C(=O)Nc3ccc(N4CCCCC4)c(Cl)c3)CC2O1 c1(NC(C(CCCOC)NC(C2OCCC2(C)C)=O)=O)cnc2ccnn2c1 C12(NC(=O)Cc3sc(O)nc3O)CCN(C(c3cc(Cl)sc3Cl)=O)CC1C2 CCCCC(=O)C(=O)NC1CCN(C(=O)C(C)(C)Oc2c(F)cccc2F)C1 CC1CN(C(c2ccoc2)=O)CCC1CNC(C1(CC#N)COC1)=O C(=O)(C(C)(C)N=[N+]=[N-])NCC(CC(=O)N(CC(C)(C)O)C)O c1(CC)cnc(C(=O)NC2(C(=O)NC3CC4(CCC4)C3)CC(F)C2)nc1 c1(NC(N2CCC(CC3CCNCC3)CC2)=O)cc(-c2cccc(F)c2)ccn1 C1(C(N(CC(COCC)O)C)=O)CN(C)CCN1C(c1cnc(O)c(C)c1)=O C1(C(=O)NC2(CC)CN(C(c3cnn(C)c3)=O)C2)CCCC(C(N)=O)CC1 C1(C(N(CCCC)CC(=O)NCC(C2CCCCC2)C)=O)Cc2nccn2C1 N1(C(CC2(C)OCCO2)=O)CC2CCC1C(NC(C1(F)CCOCC1)=O)C2 c1(C(=O)NCCN(C(C)C)C(C2CC3CCC2O3)=O)ccc(N2CCCC2)cc1 C(C(C(C)(C)C)NC(=O)C(C)(C)N(C)C)NC(c1ccc(C(C)=O)o1)=O N1(C(C=Cc2n(C)ncc2)=O)CCC2CN(C(c3nocc3Cl)=O)CCC2C1 c1(C(N2CC(C)C(NC(c3cccc4nonc34)=O)C2)=O)cc2ccncc2s1 c1(C(=O)NC2C(SC)CN(C(=O)C(C#N)C(C)C)C2)cc2cccc(N)c2cn1 N1(C(c2c(C)ccnc2)=O)CCN2CCN(C(c3ccsc3C(F)F)=O)CC2C1 c1(OCC)cccc(NC(C2CCCN(C(C)=O)C2)=O)c1 N1(C(C2(OCC)CCOC2)=O)CC2(C)CC1(C(N1CC3CC3C3CC13)=O)C2 C=C(Cl)CCC(=O)NC1C(C(N2CCCC2C(C)(C)CO)=O)C1(C)C N1(C(Cc2nc(CC)sc2)=O)CCOCC1CN(C)C(C1(C)CCCOC1)=O N1(C(c2ccc(C#C)o2)=O)CCC(NC(=O)C2=CCCCC2C)C(CO)CC1 C(=O)(C1=CCOCC1)N(CCN(C(c1cnc(C(C)C)nc1)=O)CC)CC N1(C(C(C=C)C)=O)CCN(C)C(C(N2CCC(C(C)O)CC2)=O)C1 N1(C(c2c(CC)noc2)=O)CCC(C)C1CNC(C1(NC(C)=O)CCC1)=O C(CC(C(=O)OC(F)(F)F)NC(=O)C=CC(=O)Nc1ccccc1F)SC C1(C(N2CCC(N(C(=O)Cc3cscn3)C)C2)=O)CCS(=O)(=O)N1 N1(OC(C)C)C(C)CN(C(c2cccc(C#N)c2)C(=O)N(C2COC2)C)CC1C c1(C(=O)NC2C(CNC(CCSC)=O)CC2)ccc(C2(F)CC2(F)F)cc1 CC1(C)C2CCC1(CC(=O)NC1CC=CC1)CC2.C1CCOCCNCC(=O)N1 c1(C(N2CC(CC(C)NC(CCOCCOC)=O)C2)=O)noc2cc(Cl)ccc12 CC1(C)CC2(CC(C(=O)NCC(F)CNC(C3CC4CCCC(C3)C4)=O)C2)C1 c1(CC)ccccc1C(=O)NC(C)C(C(C)C)NC(c1cnc(C)s1)=O C1(NC(c2cc(CC)on2)=O)CN(C(=O)OC(C)(C)C)CC(C)(C)C1 C(=O)(CC(O)CC(C)(C)C)NC1CCCN(C(C2(CCCC)CCC2)=O)C1 c1(CC(=O)NCC2CCCCC2NC(c2ccon2)=O)ccc(F)cc1C(F)F CC(CF)N=c1ccn2ncc(S(=O)(=O)N3CCOC(C)CC3)c2[nH]1 CS(=O)(=O)c1cccc(Cl)c1CNCC1CCC2(C1)CC2(F)F C(=O)(C(O)CC(F)(F)F)N1CC(O)(CCNC(C2N(C=O)CCC2)=O)C1 C1(O)(CCNC(C2(CCOC)CCC2)=O)CN(C(=O)C(C)C2CCC2)C1 N1(C(C2(C#N)C(C)C2)=O)CCN(C(=O)CC(=O)N(C)C)CC(C)(C)C1 c1(CNC2N(C)S(=O)(=O)CC2)ccc2c(c1O)CCCC2 c1(C(=O)NC2C(C)N(C(c3ccc(C(C)(C)C)nc3)=O)CC2)ccc(F)cc1F C1(C(C)C)CCCN(C(=NCc2cccc3c2OCCO3)NCC2CCCO2)C1 c1(C(=O)NC(CCN(C(CC(C=C)CC)=O)C)C)ccn2cc(C)nc2c1 Cn1ncc(C(N2CC(n3cc(-c4cccc(N(C)C)c4)nn3)C(O)C2)=O)c1C#N Cc1cccc(Cl)c1C(N1CC(NC(c2cnnc(O)c2)=O)C(F)C1)=O c1(C(N2CC(NC(C=C(CC)C)=O)CC2(C)C)=O)ccc(Br)c2c1OCCC2 c1(C(=O)NCCOCCNC(c2cc(C)on2)=O)nc(Cl)c(Cl)s1 C1(NC(CCOCCN(C)C(C2CCS(=O)CC2)=O)=O)CCCC(O)C1O C(CC(O)C(=O)NC(C1CCOC1)CO)NC(Cc1cnc(C)s1)=O C(N=C(NCc1cncs1)NC1CCOc2ccccc21)c1cc(C)c(Cl)cn1 c1(C(N2CCC(C(N3CCC(COC)C3)=O)(CF)C2)=O)cccn(C)c1=O c1(CC(=O)NC(C2CCN(C(=O)C(N)CC(N)=O)CC2)C)ccc(F)c(Br)c1 C1(C(c2ccc(Cl)cc2)NCCOCCCC)CCCC(C)CC1 N1(CCNC)CCC(N=c2[nH]c(N(C)CCc3c[nH]c(=N)s3)nc3c2COC3)C1.CS C(=O)(C#CC1CCOC1)N1CCC(CC(=O)NC(c2nncn2C)C)CC1 C(CC(=O)NC1(CC(C)C)CC1)OCCN(C(CSCC=C)=O)C C1(F)(C(=O)OCC(=O)Nc2n(C)cnn2)CCS(=O)(=O)C1 N1(C(c2c(C)nc(C)s2)=O)CC(C)CN(C(C2CC3C=CC2C3)=O)C(C)C1 CC1=C(COC(=O)C2=NNC(C(F)(F)F)C2)C(C)(C)CCC1 c1(C(N2CCC(=Cc3cccnc3)CC2)=O)ccc(Cl)c(C(F)(F)F)c1 c1(OC)ccc(NC(=O)C(C)CCOC)cc1OCC(F)(F)F N1(C(C(C(CC)C)O)=O)CCC2CN(C(c3cc(C(N)=O)co3)=O)CC2C1 CC1(C)CCN(C(C2CCOC2(C)C)=O)C1C(=O)NCc1ncc[nH]c1=O CCCN=C(NCc1cc(C)cc(Cl)c1)NC1CC(=O)N(c2ccccc2F)C1 CC(C)CC(C(=O)N(C1CCC1)C(C)C)ONC(C1(C)CCC(=O)C1)=O c1(C(=O)NCc2cccc(CNC(C(C)=CC)=O)c2)ccc2nc(Cl)nn2c1 N1(C(c2ncc(C3CC3)cn2)=O)CC2CC(C(N3CCCC3)=O)(C2)C1 N1(C(Cc2nnc(C)o2)=O)CC2CCC2(CNC(C2CC(C(C)C)=NO2)=O)C1 C1(n2cnnn2)(C(=O)NCC(CO)NC(=O)C(C2CCCCC2)O)CCOCC1 C(=O)(C(O)CC(F)(F)F)NCC1(OC)CCN(C(c2cc3ccncc3[nH]2)=O)C1 C1(NC(COCC#C)=O)CCN(C(c2cccnn2)=O)C1 C(=O)(C(CC(F)F)NC(c1coc(C(F)F)c1)=O)N(CC(COCC)C)C Cc1csc(C(N2CCCC(C(=O)Nc3cn(C)nc3C)C2)=O)c1C c1(C(=O)NC2CCN(c3cccc(C)c3)C2=O)cc(C)c(Br)c(C)c1 N1(C(C(C)NS(C)(=O)=O)=O)CCCC(NC(=O)CCC2(O)CCC2)C1C N1(C(C2(C)ON=C(C)C2)=O)CCCC2(C1)CN(C(=O)CC1OCCC1C)CCO2 N1(C(c2nc(C)[nH]n2)=O)CCC(C2CCN(C(=O)C=C3CCC(C)(C)CC3)C2)C1 N1(C(CCCC#C)=O)CCC2(CC1)CCN(C(=O)CN=c1cc[nH]cc1)C2 C1(CNC(CC=CC=C)=O)CN(C(=O)CC(c2ccc(F)c(F)c2)C)CCN1C c1(C(N2CC(C)C(NC(c3cc(C(C)C)ccc3N)=O)C2)=O)cn2c(n1)SCC2 c1(C(N2CC(C)(NC(=O)CC3(C)CCS(=O)(=O)N3)C2)=O)cc(Cl)c(F)cc1O C1(C(N(C)CC2CC2(C)C)=O)N(C(c2cnn[nH]2)=O)CCC1(C)C CC1CCn2cc(C(N3CCCC(F)(CNC(C4CC(O)C4)=O)CC3)=O)nc2C1 C#CCC(C(=O)NC1CC1C(F)(F)F)NC(=O)C=CC(C)C C1(CC(N2C3CN(C(c4n(C)ncc4)=O)C(C3)C2)=O)Cc2cccc(Cl)c2O1 C(C(=O)NCCCC1CCCN1C(=O)CCn1ccnc1)(C(C)C)OCC(C)C N1(C(C(CCC)C(C)C)=O)CCC2CCN(C(c3nn[nH]c3Cl)=O)CC12 c1(NC(C(C)S)=O)n[nH]c2c1CN(C(=O)CN1CCNC1=N)CC2 Cc1c(F)ccc(C(N2CCC3C(NC(=O)CCCCC(N)=O)C23)=O)c1C#N c1(NCC(CCCC)NC(C2CCN(C)C2=O)=O)nc(Cl)nc2[nH]cnc12 CCCC(C)C(=O)N(C1CC(NC(c2c(C(F)(F)F)noc2C)=O)C1)C Cc1ccc(NC(C2CN(C(=O)C(C)(C)C(C)O)C2)=O)cc1CO Cc1cc(C2CCC2)ccc1C(=O)NCC(C)N(C)C(C1CN2CCC1CC2)=O N1(CCN2C(c3ncc(-c4ccccc4)o3)CCC2)CCCC1(C)C1CCCCC1 C1(C(N2CC(C(C)NC(c3cc(Br)c[nH]3)=O)C2)=O)Cc2cncn2C(=O)N1 CCC(CC)CC(F)C(=O)N1CC(NC(c2cncnc2)=O)CC(F)C1 c1(NC(=O)NCc2cccc(OC)c2OC(F)F)c(Cl)cc([N+](=O)[O-])cc1Br C1(NC(C(CCSC)O)=O)CCN(C(c2cc(N)cc(O)n2)=O)C(C)C1 C(=O)(C(C)CC1CCCCC1)NCC(C)NC(c1coc(-c2ccccc2)n1)=O C1(C(=O)NCC2CC(NC(c3c(C)snn3)=O)C2)SC2C=CC1CC2 C1(N(C(C2CCN(C(C(CC=CCC)C)=O)CC2)=O)C2CC2)CCCN(C)C1=O Cc1cc(F)ccc1C(=O)CNC(=O)C(F)CC1CCOC1 CCC(C(=O)OC)C(=O)N1CSCC1C(=O)NC1(C)CCC(C)(C)C1 C12(CNC(c3c(C)noc3N)=O)CCCCC1N(C(=O)CN(C)CCO)CC2 N1(C(C(C)(CO)NC(C)=O)=O)C2CCC1C1CC1(NC(c1cc[n+]([O-])cc1)=O)C2 C(CCCC(CO)NC(=O)C(COC)CC)NC(CNS(NC)(=O)=O)=O c1(NC(c2n(C(C)C)ncc2)=O)ccc(NC(C2CC(O)CN2)=O)c(F)c1 c1(C(=O)NCC(CN(C)C(C2CCC(F)(F)C2)=O)O)cc2cccnc2nc1O CCC(C(=O)N1CCN(C)C(CNC(C2CNC(=O)O2)=O)C1)C(C)(C)CC C1(NC(c2cnc(C)s2)=O)CC(CNC(=O)C(C#N)C2CC2)C(O)C1 c1(CN2CCN(C(CC)C(=O)NC3CC3)CC2)c(Cl)nc2ccccn12 n1(CC(=O)NCC(=O)Nc2ccc(Br)cc2)cccnc1=O N1(C(CCCSC)=O)CCN(C(c2ncc(C(F)(F)F)s2)=O)C(CCO)C1 c1(C(=O)NC(CCOC)Cc2cccc(Br)c2)cc(C(F)(F)F)ccc1C(=O)O N1(C(C(CNC(=O)OCC)(C)C)=O)CC(C(=O)N(CC(=O)OC)C)CC(C)(C)C1 CCCCCC(C)(C)C(=O)NCCC1CN(C(=O)Cc2cc(F)ccc2Cl)C1 C1(NC(C2CC3(CC(=O)N3)C2)=O)CCCC12CCN(C(c1ccco1)=O)CC2 c1(-c2cn(C(c3ccc(OCC)cc3)CC=C)nn2)cc(F)cc(Cl)c1 C(=O)(CC(C)C(C)(C)NC(c1cccc(C)c1F)=O)NCc1ccc(C)nc1O N1(CC)Cc2ccc(NC(C3CCNC3c3ccccc3)=O)cc2C1 C12(NC(C3CN(C)C3)=O)CCC1CN(C(c1ccc(NCC(N)=O)cc1)=O)C2 C(=O)(C(CNC(=O)CC1OCCCO1)CC1CC1)NC(c1n[nH]c(CO)n1)C C1(C(=O)NC2C(SC)COC2)CCCCCCN1C(=O)CCCc1ncco1 C1(NC(=O)CNC(C2CCCCO2)=O)CN(C(C2OCCCO2)=O)C2(CCC2)C1 c1(CNC(C(N2CCCCCC2)C)=O)cc(O)nc(CNC(=O)CC2CC2C)n1 CCC(O)(C(=O)N1CC(CNC(=O)CC2(C)CC2(F)Cl)C1)c1ccccc1 CCCCC(CCCC)C(=O)NC1CC(CNC(=O)Cc2ccc(OC)cc2)C1 C1(N(C(c2occ(C)c2)=O)C)CCC(NC(C2CC2c2ccsc2)=O)CC1 C(=O)(CC(C)(C)C)NCC(=O)NCC(C)N(C)C(c1cnc(-c2cccs2)o1)=O c1(CC)ccc(C(=O)NC(CNC(c2cnn(C)c2C)=O)CC(C)C)c(Cl)c1 C(=O)(C(O)CCC(C)C)N1C(C(=O)NCCN(CCC)CC)CC(OC)C1 c1(OC)cnc(N(CCc2c[nH]c(=N)s2)CC2CN(C)CCO2)nc1C C1(C)(CC)CC(NC(=O)CCOC2COC2)CN1C(c1c[nH]cc(Cl)c1=O)=O C1(C(=O)NCC2C(C(C)(C)C)C2)(NC(=O)Cn2ccnc2)CCC1 Cc1c(Br)ccc(-c2noc(CSc3cccc(F)c3Br)n2)c1F O=S(=O)(c1ccc2[nH]c(=NCc3ccsc3)sc2c1)NCC1CSCCS1 O=C(CC1OCc2cc(Cl)ccc21)NC1CCN(C(C2CSC2)=O)CC1O Cc1ccc(SCC(=O)N(CC(O)CNC(=O)COC2CCC2)C)c(C)c1 C12(NC(c3n(C)c(S)nc3)=O)CCC(CC1)N(C(C1CCC3C(C1)C3(F)F)=O)C2 N1(Cc2c(C(=O)O)c3c(s2)cccc3)CC2CS(=O)(=O)CC(C1)C2(F)F S(=O)(=O)(c1c[nH]c(C(=O)NC2(C)CCN(C(=O)C(C)S(C)(=O)=O)C2)c1)NCC c1(C(N2CC(O)(CN(C(C(CC#C)CC#C)=O)C)C2)=O)n[nH]c2ccc(F)cc12 c1(-c2cn(C3CCN(C(C4CCS(=O)(=O)C4)=O)C3)nn2)ccc(F)nc1 C1(NC(c2n[nH]cc2F)=O)CN(C(c2cnn3c2CCC3)=O)CC12CCOCC2 N1(C(CCCCOCC)=O)C2CCC1CN(C(=O)CC(n1nc(C)cc1C)C)C2 c1(COC)nc(C(=O)NCCC2(OC)CN(C(c3conc3C)=O)C2)co1 CC1(CNC(C2CCC(OC(F)F)CC2)=O)CCCN(C(c2c[nH]c(=N)s2)=O)C1 c1(C(=O)NC(CNC(CCCC#C)=O)CC(C)C)c(OC)cc(OC)cc1N Cc1ncc(C(=O)NCC2CN(C(c3cc(C(F)F)on3)=O)C2)n1C N=C1NC(=O)C(CC(N2CCN(C3CCCN(C(=O)CC4(O)CC4)C3)CC2)=O)S1 CC1CN(C(c2cscc2C#N)=O)CCC1C(=O)N(C1CC(C(N)=O)C1)C S(=O)(=O)(c1ccc(Cl)c2nonc12)Nc1ccc(NC(c2ccc(Cl)cn2)=O)cn1 C1(NC(CS(CC)(=O)=O)=O)CCC2CN(C(c3ccc(C)nc3OC)=O)CC2C1 c1(C(=O)NC2CC(NC(C(CC)(F)F)=O)C(O)C2)ccc2cc(C#N)ccc2c1 N1(C(C2(C(=O)OCC)CCC2)=O)CC2CCC2(CCNC(c2cscn2)=O)C1 N1(C(CC2C(CC)C2)=O)CCC2(CCCC2NC(c2ccc3c(c2)CCC3)=O)CC1 c1(OC)cc(N2CCC(NC(C3CC3C3CC3C)=O)CC2C)c(Cl)cc1[N+](=O)[O-] CC(C)C(C(=O)N(CC(C)CNC(C1CCCC1C(C)C)=O)C)n1cccc1 C1(CNC(=O)CCc2ncccn2)CCC2(CCC2)CN1C(=O)C=CCF C(=O)(CC(C(F)F)n1cccn1)NCc1ccc(CNC(C(C)=C(C)C)=O)cc1 Cn1ccc(=O)c(C(=O)N(CC(=O)NCCC(=O)NC2CC2)CCO)c1 C1(C(N(C(CNC(=O)CN2CSCC2=O)C2CC2)C)=O)CCCC2(CCC2)C1 C1(C(=O)NC2CCN(C(c3cc(Cl)ns3)=O)CC2O)(OC)CCC(C)(C)CC1 N1(CC(N2CCCCC2c2cc[nH]n2)=O)CCN(Cc2ccc(F)cc2)CC1=O N1(C(C2(C3CCCCO3)CC2)=O)CC2=C(C1)CN(C(C13CC(F)C1C3)=O)C2 C1(CNC(C=CCC)=O)C(C)CCN1C(C1CCCN(C)C1)=O c1(C(=O)NC2CC(CNC(c3cccc(C)n3)=O)C2)cnc(C)c(N)c1 c1(CC)cc(Cl)ccc1C(N1CCCC1CCNC(c1cnnn1C)=O)=O C1(C)(OC)CC2CC1CC2NCC1CC2(C1)N=N2 N1(C(C2(NC(=O)CN3CC(C)(C)C3)C(C)CCC2)=O)CCCNC(=O)CC1 C12(CC(C)(C)C1)C(=O)NC2.C1(C(=O)NC2C=CCC2)(OC)CC(C)C1 Cc1csc2nc(CC(=O)NCC3(O)CC(CNC(C45CC(F)(C4)C5)=O)C3)cn12 c1(NC2C(C)C2)nc2c(c(=NCC3Cc4ccccc43)[nH]1)CCC2 C1(CNC(CNC(C)=O)=O)CN(C(=O)COc2cncc(Cl)n2)C2CCCC2O1 N1(c2nc(C)cc(OC)n2)CC(NC(=O)CC(C)(O)C2CC2)CC2(CCC2)C1 c1(C2C(CNC3(c4n(CCSC)nnn4)CC(C(C)C)C3)C2)ccc(C)cc1 Cc1cc(C)c(CN(C(CC2CCN(CC(=O)NCc3nc(O)n[nH]3)C2)=O)C)s1 C(=O)(CC1=NN(C)C(=O)C1)NC(CCC)CCCNC(=O)CCCN1CCCC1 N1(CC)CCOCC1C(=O)NCCCN(C(=O)C(n1ccnc1C)C)C(C)C C1(CNC(=O)COC2CCCCC2)C(C2CC2)CCN1C(=O)C(F)C1CCC1 c1(CNCC(C)(CC2CCOCC2)NC(C)=O)cn(C)c(=O)n1C c1(C(=O)NCC2(F)CCC(NC(C3(C)ON=C(C)C3)=O)C2)cccc(N)c1O C1(C(N(C)CC2(CNC(CCOC)=O)CC2)=O)(OCC)CCCCCC1 CC(C)CCC(O)C(=O)NCC(C)CNC(=O)C(F)(F)c1cnccn1 c1(CC)cc(C(=O)NC(C(=O)NC2CCCN(C)C2)c2ccco2)c(C)o1 c1(C2(C)CC2CNC(c2cnn(CCc3ccccc3)c2)=O)cn(C(C)C)nn1 c1(C(N2CCC(CNC(C(CN(C)C)N(C)C)=O)C2)=O)c(F)cccc1[N+](=O)[O-] Cc1cc(C(N2CC(C(=O)NC(=O)CNc3cccc(Cl)c3)C2)=O)cnc1O c1(C(=O)NCCOCCN(C(C2C(OC)C2)=O)C)cnn2cc(C)cnc12 C#CCCCC(=O)N1CCC(NC(c2cn(-c3ncccn3)cn2)=O)C1C C1(CC(=O)NCCC2CC(NC(C(C)OCC3CC3)=O)C2)COCCN1C c1(CC)nc(C)c(CNC(C2CCN(C(=O)C(C)NC(C)(C)CC)C2)=O)o1 Cc1nnccc1C(=O)NC(C)C(C(C)C)NC(C1(C)COC1)=O C1(C)(C(=O)NC(C2CCN(C(=O)C(C)=CC3CC3)C2)C)CCCC1 c1(C(N2C(CNC(C(CCC)OC)=O)CC(O)C2)=O)sc2ccc(Cl)cc2c1C c1(C(N2C3CC(NC(C4CCNC4=O)=O)CC2CC3)=O)cc([N+](=O)[O-])ccc1O c1(C(=O)NCC2CN(C(CNC(CC)=O)=O)C(C)C2)cnc(N)c(CO)c1 N#Cc1cccc(C=CC(=O)NC2CC2C(=O)NCc2cc[nH]n2)c1 C=C(Cl)C(C)(C)C(=O)N1CCC(NC(=O)CSc2c(C)noc2C)C(F)C1 C=C(Cl)CCC(=O)NCCOC(C)(C)CNC(=O)C(CC1CCCCC1)CC c1(C(N(CC(C)NC(=O)CC2CC23CC3)C)=O)ccnc(N2CCCC2)c1 c1(C(N2CC(CCNC(=O)CSCC(F)(F)F)OCC2)=O)cc(C(F)F)cnc1O CC(C)C(CC(=O)O)NC(=O)Cn1cc(-c2ccc(C(N)=O)nc2)nn1 c1(C(=O)NCC(CCOC)NC(c2[nH]c(C3CC3)nc2C)=O)ccc(C)nn1 C(CC(=O)N1CCCC1(C)C(=O)OC)(C(F)(F)F)NC(C1(CC#C)CCC1)=O N(C(=NCC(C)c1ncc(C)s1)NCN1CCOC(CC)C1)C(CC)CC c1(N2CCC(N(C(c3cc(SC)sc3Cl)=O)C(C)C)C2)cccc(Cl)c1Cl O=C1CCC(C(=O)NCC2COCCN2C(=O)CC2CCC(=O)NC2)=NN1 CC(c1cccc(C)c1)=CC(N1CCC1CNC(c1cn(C2CC2)nn1)=O)=O N1(C(c2cc(-c3c(OC)cccc3)no2)=O)CC(=O)N(C2CC2)C1=O c1(OC)cc(C(=O)NC2(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)cnc1O C=CCCCC(=O)NC(C)CCCNC(=O)Cc1nncn1C c1(SC)cccc(F)c1C(N1CCC(C)C1CNC(=O)Cc1cnn(C)c1)=O Cc1ccc(N)c(C)c1C(=O)N(CCCCN(C(=O)C(C)C(F)(F)F)C)C CC1=C(C)CC(C(=O)NC2CCCCN(C(=O)CN(C)C(=O)C3CC3)C2)CC1 c1(CNC(=O)C(C(C)C2CCOC2)OC)cc(F)cc(F)c1.c1(O)ccccc1F c1(C(N2CCC(COC(CC)(C)C)CC2)=O)cc(C(F)(F)F)cc(C(C)C)c1 N1(C(C(C(C)C)NC(C)=O)=O)CC2CC(C1)N(C(=O)C(C)(C)OC(C)C)C2 CC(CC(F)F)C(=O)N1CCC(C(=O)Nc2cccc(OCF)c2)C1C N1(C(CCC=CCC=C)=O)CC(NC(c2conc2C(F)(F)F)=O)C(C)(C)C1 C1(NC(C2CCCC(C)(C)C2)=O)CCN(C(c2csc(Cl)c2Cl)=O)CC12CCC2 CCC(CC)(CO)C(=O)NCC1CCCCC1NC(c1nc(=O)n(C)[nH]1)=O N1(C(C)=O)CC2CCN(C(C3CC3Cl)=O)CCC2C1.NC(C=O)=Cc1cccs1 c1(-c2cn(C(C)CNC(=O)C(F)C(F)(F)F)nn2)c(F)cccc1F c1(CC)cnc(C(N2CCC(NC(c3cnn(C(C)C)c3Br)=O)C2)=O)cn1 C1(C(N2CC(C)C(C)C2C)=O)(CC)CCN(C(=O)C=CC(=O)NC2CC2)CC1 c1(C(N2CCC(CC(=O)NC(C)C(F)(F)F)C2)=O)cc(Cl)nc(Cl)c1F c1(CC)[nH]nc(C(N2CCC(CO)(NC(=O)Cc3cncs3)C2)=O)c1Br C(N=c1nc2sccc2c(N2CCCCC(C)(F)C2)[nH]1)c1nn(C)c(Br)n1 C1(C(NOCCC)=O)CN(C(=O)CC23CCCC2C3)CC1CCCC.C(CCO)O C(=O)(C(C(C)(C)C)NC(=O)CCCC)NCC1(CO)C(C=C)C1 N1(C(CC2(C(=O)OC)CCOCC2)=O)CCCC(CNC(c2ccns2)=O)CC1 C1(NC(=O)NCC(C)S(C)=O)CCCC1P(C)(C)=O CC1CN(C(=O)C=C2CCC2)CC2(CCN(C(C3CC(=O)N(C4CC4)C3)=O)C2)O1 C1(CC)CN(C(=O)C(C)CC(=O)OC)CCN1C(c1cccc(C)c1F)=O c1(CN(CCN(C)C)C(c2ccnc(CN)c2)=O)ccc(F)nc1 N1(C(CNC(C(C)(C)C)=O)=O)CCC2(CCC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 C=CCCC(O)CNC(C1CC1C(C)NC(c1c[nH]nc1C(C)C)=O)=O C1(NC(CCN(S(C)(=O)=O)C)=O)COCCN(C(c2cncnc2)=O)C1 CC1(C)CCN(C(=O)CCF)C1CNC(c1ccc(C(F)(F)F)nc1)=O CC(C)C(CNC(=O)C=C1CCCC1)C(=O)NCCCN1CCCC1C c1(NC(C(C)C)C)ccc(S(=O)(=O)NC2CN(C)CC2O)cc1C#N C1(C(=O)OC)CN(C(=O)C(=O)N(C)Cc2c(C)nn(C)c2C)CC1(C)C C12(C(N(C(CC)CCOC)C)=O)CC(CN1C(=O)C(C)(C)COC)C2 CC12CC3CC(CC(C(N4CCCC(O)(CNC(C5CC5F)=O)CC4)=O)(C3)C1)C2 c1(C(N2C3C(NC(C(C)NS(C)(=O)=O)=O)CC(C3)C2)=O)ccc([N+](=O)[O-])cc1N c1(C(=O)NC(CCCNC(C(C)NC(CC)=O)=O)CO)c(C)cccc1Cl N1(C(C2(C(=O)NC)CC2)=O)CCC(NC(C2CSC2)=O)CC1C Cc1nc(NCCc2nc(Br)n[nH]2)cc(=NCC2(c3ccccc3)CC2)[nH]1 CC(CC(C)C(F)F)NC(C1(NC(=O)C(C)SC(C)C)CCC1)=O c1(CS(C)=O)c(C(=O)NC2(CO)CCN(C(=O)CO)CC2)oc2ccccc12 c1(C(=O)OC)c(C)[nH]c(C(N2CC(NC(c3ncc(C)cn3)=O)C2)=O)c1C C1(COC2CCN(C(=O)NCCC)C2)(Cc2ccccc2)CCCC1O N1(C(C=COCC)=O)CCC2CC1CN(C(c1sccc1OC)=O)C2 CP(C)(=O)CCC(=O)N1CCCC1C1(C(=O)Nc2ccc(SC3CC3)nc2)CC1 Cn1nc(C(=O)NCC2CC3CN(C(=O)C=C4CCC4)CC23)c2c1CCCC2O C1(C(=O)NCc2ccc(CNC(C(C)NC(C)=O)=O)cc2)CC(=O)N(OC)C1 c1(NC(=O)CCNCC2NCCC23CC3)ccc2c(c1)CCCO2 C1(CNC(c2cn[nH]c2)=O)(NC(c2scc(Cl)c2Cl)=O)CCC(F)(F)CC1 C1(CC)(CC)CC(NC(=O)C#CC(C)(C)C)CN1C(=O)CN(C)C N1(C(C)C(=O)NC2COCC2CNC(c2cc(Cl)cs2)=O)CCCCC1=O C(CC(CC)C(=O)N1CCC(CNC(=O)Cc2ccsc2Cl)C1(C)C)=CC Nc1ccc(NC(=O)C(F)CC2CC(C(=O)NCCCN)C2)cc1 Cc1noc(C)c1C(=O)NCc1ncoc1C1CN(C(C2C=CCC2)=O)C1 C(CC1CCCC1)(C(=O)N1CC(OCC(N)=O)C1)NC(COCC#C)=O N1(C(C2N(C(C(C)Oc3ccccc3)=O)CCCC2)=O)CCNC(=O)CC1 Cc1cccc(C(C)C(=O)NC(C2CCCN(Cc3ccc(CO)cc3)C2)C)c1 N1(C(c2cc(C(=O)OCC)c(C)[nH]2)=O)CC2(CCC(NC(C3(C)CC3)=O)CC2)C1 N1(C(C(C)OC)=O)CCN(C(=O)C(F)(F)CCn2ccnn2)CCC1C Cc1nc(C(=O)NC(C)CCNC(c2coc(Cl)n2)=O)c(C(F)(F)F)[nH]1 c1(NCC(C)CCO)cc(Br)ccc1S(=O)(=O)NC(C1CCCCO1)(C)C c1(NC(c2c(CNC(C3(C)CCNC3=O)=O)noc2)=O)cc(C#N)ccc1O N1(C(C(CO)NC(N)=O)=O)CCN(C(=O)CCc2ccc(F)cc2)CC12CCC2 c1(CCC(=O)NC(C(C)NC(c2n(CC)ccc2)=O)C)ccc(C)nc1 c1(C(=O)NCC2C(CNC(Cc3cn(CC)nn3)=O)C2)ccc2nn[nH]c2c1 C1(CC(=O)NCC2N(C(CC)=O)CC2)SC(=N)NC1=O CC1(CO)CCN(C(=O)CCOC2CN(C(C3CC(=O)CCO3)=O)C2)C1 c1(OCCCCC)cc(C)ccc1CNc1ccc(NC(=O)C2CC2)cn1 C1(CNC(C(C)Nc2scc(C)n2)=O)CCCN(C(C2(CC(C)C)CCC2)=O)C1 C1(NC(CCc2c(C)ncs2)=O)CCN(C(C2(COC(C)C)CC2)=O)CC1C c1(CC)ccc(C(=O)NC(C)C(CO)NC(C2(C(F)F)CCC2)=O)c(C)n1 c1(CNC(c2n(CCCSC)nnn2)C2CCCSC2)cn2cccc(F)c2n1 C#CCC(C(=O)N1CCC1C(N)=O)NC(c1csc(CO)n1)=O Cc1nc2c(o1)CCN(C(C1CC1NC(=O)Cc1noc(C)c1C)=O)C2 C12(CC3CCCC13)C(=O)NOC2.CCC(C)(C)NC(C)C(=O)NC1CCCO1 c1(C(=O)NC2(CCNC(C(C)n3ccnn3)=O)CCC2)ccc(N)c(F)c1F C1(NC(c2cc(OC)c(F)cc2)=O)CCC2(C1)CN(C(=O)C=C(C)C)C2 Cc1nn(C)c2c(NCC3CSC3)nc(=NCCC3(C(F)(F)F)CC3)[nH]c12 CCC(C)(CNC(c1ncoc1CCC#N)=O)NC(c1cnc(C2CC2)[nH]1)=O C1(NC(c2cc(-c3cn(C)nc3)no2)=O)CCN(C(C2(C)CC=CC2)=O)CC1O C1(NC(C(N2CCOCC2)C)=O)CC2CC(C1)N(C(C1CC1C)=O)C2 C(=O)(C(C)CC(C)(C)C)N1CCCC(NC(C2COCCN(CCCC)C2)=O)C1 c1(COC)nc(CC2CCCCC2)n(-c2ccccc2F)n1 C1(O)(C(CNC(C2(COC)CC=CC2)=O)C)CCN(C(c2csc(C)n2)=O)C1 C1(C)(CNC(C(C)Cc2ccncc2)=O)CCN(C(c2ccncn2)=O)C1 S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1C2C(N3CC(C)C4(C3)CNC4)CC(C2)C1 N1(Cc2cnc(C)o2)CC2CCC(NC(=O)CCC3CCCCO3)CC2C1 N1(C(CC(C)n2ccnc2)=O)CC2CC2(CNC(C2CC(O)CN2C)=O)C1 N1(C(CCCC=C)=O)CC(NC(C2(C)CCC2C(=O)OC)=O)CC12CCOCC2 C1(C(=O)NCCC2CCCCN2C(=O)CN2CCCCC2)CC2CCCCCC12 c1(CC(=O)NCCCC(C)NC(Cn2cc(C(=O)OC)nc2)=O)ccc(C)cc1F Cc1ccc(CSCC(=O)OCC(=O)N(C2CCCC2)C)nc1Br C1(CC(=O)NCCN2C(C)CCC2)CCN(C(c2scnc2Cl)=O)C1(C)C CC(C)CC(CNC(C1(C)CCC(=O)N1)=O)NC(=O)CCSCc1ccccn1 Cc1ccc(C=CC(=O)NC(C)C(C)NC(c2ccc(Br)s2)=O)cc1C C(C1CCOCC1)=CC(=O)N(C)CC1CCCN1C(C1CCC1(F)F)=O c1(CCC(=O)NCC2(O)CN(C(C3C(C)CC3)=O)C2)ccc(Br)c(Cl)c1 C(CCCCn1cc(C2(n3nccn3)CC2)nn1)NC(C1CC2CC2C1)=O c1(C(=O)NC(CCN(C(C(CC)(C)O)=O)C)C)oc(P(C)(C)=O)cc1C N1(C(C(C)SCC)=O)CCOCC(CNC(=O)C(C2CC(F)(F)C2)OC)C1 C1(NC(C2CCCS2)=O)(CO)CN(C(=O)CNc2ncccn2)C1 c1(C(=O)NC(C)C(CO)NC(=O)C(c2ccccc2)O)cc(Cl)ccc1O N1(C(Cc2c(C)ccs2)=O)CCCC(CCCCNC(C2OCC2(C)C)=O)C1 N1(C(C(C)N2CCC2)=O)CC2CCN(C(C3CCOC3c3ccncc3)=O)CC12 c1(C(=O)NC(C(=O)N2C(COC)CC2)CCF)cc2occc2[nH]1 C1(COC)CC(CNC(c2csc(C)c2C)=O)N(C(=O)CCc2cncn2C)C1 c1(C(=O)NCC(C)CNC(=O)CCOCCN(C)C)ccc(C2CC2)nc1 c1(C(N2CCC3C(NC(C(C)C(C)(C)C)=O)C32)=O)cccc2sncc12 c1(CN(C2CCCC2)C(CC2CCN(C(C(CC)C)=O)C2)=O)n[nH]c(C)c1Br C(CCCC(C)NC(C1(F)CCCCC1)=O)NC(c1c(C)scc1)=O O=C(C1=C(Cl)CC1)NC1CCOC(C(=O)NCCC(O)CO)C1 c1(C(N2CC(CNC(C(C3CCOCC3)C)=O)C(C)C2)=O)ccn(O)c(=O)c1 C=C=C(C)CC(=O)NCC1CCCCC1C(=O)Nc1cnc(C)nc1 C#Cc1ccnc(C(=O)NC2CN(C(=O)CNS(=O)(=O)N(C)C)C(C)(C)C2)c1 C1(NC(C2CCC(C)O2)=O)CCC2CCN(C(c3ccc4nc[nH]c4c3)=O)C12 c1(NC)nc(C)cc(=NC(CNC(c2cccc(Cl)c2)=O)C2CCC2)[nH]1 C1(C(N(C2CCN(C(C3CC=CCC3)=O)CC2)CC)=O)CC(C(C)=O)C1(C)C N1(C(C(=O)NC(c2ccncc2Cl)C)=O)CCC(C)C(N)C1 c1(C(N2CCC(F)(CNC(c3n(C)ccn3)=O)CC2)=O)ccc2ncncc2c1 c1(CCNOC)nc(N2CC(C(N3CCOC(C)C3)=O)C2)c(F)c(Cl)n1 C1(C(=O)NCC(CC)NC(C=CC(=O)NC)=O)CCC(CN2CCOCC2)O1 N1(C(C(C)OCOC)=O)CCCN(CCNC(=O)CCc2cscn2)CC1 c1(SC)ccc(N2CC(C(=O)NC3CCN(C(=O)C=C4CCC4)C3)CC2=O)cc1 C1(C(N(C(C)CNC(=O)C(C)(C)n2cc(Br)cn2)C)=O)CC2CCC1C2 c1(OC)ccc2c(c1)CCN(C(C1CCC3(CC3)C1)=O)C2C N1(C(c2n[nH]c(CC)c2Cl)=O)CC(CNC(C2CC(C)C2)=O)C(F)(CO)C1 C(N=c1[nH]nc(OC(F)F)s1)C1OCCN(C(C(N2C(C)CCC2C)C)=O)C1 c1(OC)cc(C(N2CC(C)(CC(=O)Nc3cc(F)cc(F)c3)C2)=O)ccc1I CCC(CC)C(C)C(=O)N1CC(CCNC(=O)CC23CCC(CC2)OC3)C(C)C1 C1(C)(OCC)CCN(C(C2CC(C)CN2C(c2cc[n+]([O-])cc2)=O)=O)CC1 C1(NC(COCC#C)=O)CCCC(NC(c2nnc(S)n2C)=O)C1 C1(CN(C)C)(NC(=O)C(C2CC2)N(C(=O)C=C2CCOCC2)C)CCCC1 C(=O)(C(CC(C)C)C(C)C)NCC1C(NC(C(C)N(C(C)=O)C)=O)C1 C(=O)(CCCCCCCCCO)N(C(C)CN(C(=O)C(Cl)=CCl)C)C c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC2O)ccc2ccc(Cl)cc2n1 N1(C(c2c(OC(C)C)nccc2)=O)CCCN(C(=O)C(C)n2ccnc2)CCC1 c1(C(C)C)ccc(F)cc1C(c1ccccc1)OCN1CCNCC1C(=O)NCCF c1(CCC(=O)NC2C(C)CCN(C(CC(CCC)O)=O)C2)c(C)nc(O)nc1C C12(CCCCC1C)C(=O)N2.C(CC(=O)NC)OC.S(C)(=O)(=O)N(CCN)C CCCC(C(=O)NC(CO)C(C)NC(c1ncn(-c2ccccc2)n1)=O)OC N1(C(c2cn(C(C)C)nc2)=O)CCC(C(=O)NCCn2ccnn2)C1C c1(C(=O)NCC2CCC(NC(C3(C4CCC4)CCC3)=O)C2)cc2c[nH]cnc-2n1 N1(C(c2c(CCC)nns2)=O)CCC2CN(C(C3CCSC3)=O)CC12 N1(C(=O)OC)C2CCC1CN(c1nnc(-c3n[nH]c(C)c3Cl)n1CC1CC1)C2 c1(C(=O)NC2C(NC(COC(C)C)=O)CCCC2)nn(C)c2c1CC(F)(F)CC2 N1(C(c2nnn3c2CCC3)=O)CC2CCN(C(=O)C(C3CCCCC3)F)CC2C1 c1(CCNC(c2n(CCSC)nnn2)c2nc(C)cs2)cncc2ccccc12 C1(C(C)C)CCCC(N=c2[nH]c(=NCC3(C)CCN(C)CC3)[nH]c3c2SCC3)C1 C(=O)(C1=CCCOCC1)N1CC(C)(C)C(NC(=O)Cc2ccc(Br)s2)C1 Cc1nc2sccn2c1C(=O)NC(=O)Cc1c(C)noc1C.C12CC1C2 CCC(CC)CCC(=O)NCc1ccc(C(N2CCc3ccsc3C2)=O)nc1 C1(C(N(CCCCN(C)C(c2ccc(-c3ccco3)o2)=O)C)=O)CC2CCC1C2 c1(C(N2CCC(CCNC(c3nc(C4CC4)cs3)=O)C2)=O)ccc(O)cc1 C1(N(S(=O)(=O)Cc2ccccc2)C(C)=O)CC2(C1)CN(Cc1ccc(O)nc1)C2 Cc1ccc([N+](=O)[O-])c(CC(=O)NCCCN(C)C(c2c(N)sc(C)c2C)=O)c1 N1(C(C(=Cc2ccco2)C)=O)CCCC2CN(c3ncc(C#N)cc3Cl)CCC12 N1(C(c2sc(CC)c(C)c2)=O)CCC2CCC12CNC(c1cnc(O)c(F)c1)=O C(C(F)(F)C(F)(F)F)n1c(-c2csc(CO)n2)nc(C(CC)C)n1 C#Cc1ccc(C(=O)NC2CN(C(c3ccc(SC)s3)=O)CCC2C)nc1 C1(C(=O)NCCCC(C)(C)NC(c2nc(C)oc2C)=O)CCOC(=O)CC1 N1(C(CC2C(=O)NC(=N)S2)=O)CC2CC1CN2C(=O)CCc1cncnc1 C1(CNC(C=C(CCC)C)=O)CCCC(NC(=O)CCSCC(C)C)C1 c1(C(=O)NC2CC(NC(CN(CCOC)C)=O)C2)cccc2[nH]nc(O)c12 C12CCCN(CC1)C(=O)C1(CC1)N(C)C2=O.C1(C(=O)OC)CCNC1=O CC#CCCCC(=O)NC1CCC(N(C(=O)CCCc2sccc2C)C)C1 N1(C(C2CC(C)CN(C(=O)C3=CC(C)(C)C3)C2)=O)C2CCCC1COC2 C1(c2ccc(OC)cc2C)NC(=O)N(CCC2CC2)C2=C1C(=O)NCC2 N1(C(N(C)Cc2ccccc2)=O)CCC2CCNC(=O)C2C1 c1(-c2ccc(C(=O)NCC(CCOC)OC)o2)ccc(F)c(OC)c1 Cc1ccc(C(N2CC3CC(C2)N(C(=O)CCCC(C)(F)F)C3)=O)c(=O)n1C C1(CNC(c2c(C)ccn2C)=O)C(O)C(O)CN1C(c1cnc(CC(C)C)s1)=O c1(CNC(C2(C=C)CCC2)=O)nc2c(s1)CN(C(=O)Cc1ccsc1Cl)CC2 O=C(CCCC1CCCO1)NC(c1ccccc1)C(=O)NC1C=CCC1 C12(C(N(C(CNC(c3cc(C4CC4)on3)=O)C3CC3)C)=O)CCC(F)(CC1)CC2 C1(C2CN(C(C3(C)CC=CCO3)=O)C2)(NC(CC=C(C)C)=O)CC1 N1(C(C(c2cnn(C)c2)C)=O)CC(C)N(C(=O)CC2COCC(C)O2)CC1C N1(C(C(C)(C)SC)=O)CC2(NC(c3cc(N)c(F)cn3)=O)CCC1CC2 CC(CC(=O)NC1CC(O)(CNC(c2cc(C(N)=O)co2)=O)C1)N1CCCC1=O C1(C)(C(=O)NCCN(C)C(c2ccnn2C2CC2(F)F)=O)CCNC1=O CCC(COC)C(=O)NCCCC(=O)Nc1cnn(C(C)(C)C)c1 O=NN1CCCC1C(=O)Nc1cccc(NC(C2CCCCNC2)=O)c1 N1(C(C2N(CC)CC2)=O)CC2CC1C2CNC(=O)CCC(C)N(C)C c1(C(=O)NC(C(C)(C)C)CNC(c2cccc(O)n2)=O)cc2sccc2n1C c1(SCCNC(=NCC)NCCC(c2ccccc2)O)ccccc1S(N)(=O)=O C1(CCC)(NC(c2cn(C)cc2C)=O)CCN(C(c2cnnn2CC)=O)CC1 C1(OC)CCN(C(=O)CSCCNC(=O)Cc2ccnc(O)c2)CC1C C1(C(=O)NCC(C)(C)NC(C2CCN2C2CCCC2)=O)CCC2(CC2)C1 N1(C(CCN(CC(F)(F)F)C)=O)CCC(CF)(NC(c2cnc(Cl)[nH]2)=O)C1 c1(C(N2C(CNC(C3(C)C=CCC3)=O)CC2)=O)cccc(C(OCCN(C)C)CC)c1 CC1CC(C(=O)N2CCCC(NC(=O)CCS(C)(=O)=O)C2C)=NO1 c1(CC(=O)O)coc2c1CN(C(C1CCC(Oc3ccncc3)C1)=O)C2 c1(N2CCC(NC(C34C(C)(C)C(CC3)CC4)=O)C2)nnc2c(c1C#N)CCCC2 C1(C)(C(=O)NCC2C(C)CN(C(C3CCC(O)CC3)=O)CC2)CC2(C1)CC2(F)F n1(CC(=O)N(C)CC2N(C(C3C(C)=C3)=O)CCC2)ccc2c(N)cccc12 Cc1ncc(Br)c(C(=O)NCCN2CCN(C(=O)CC3CCCCCC3)CC2)n1 C1(NC(CCc2c(C)nccc2)=O)CC(C(=O)O)C12CCC2 c1(NC(N(CCC)C(c2ccccc2)C)=O)c(Cl)cc(Cl)nc1C c1(OC)cc(C(=O)NC2CC(C)N(C(c3ccc(SC)o3)=O)C2)nn1C CC1CN(C(C2CCS(=O)CC2)=O)CC(C)N(C(c2cnc3n2CCS3)=O)C1 c1(CN(C)C)cc(NC(=O)NCCCCCN(C)C)cc(Br)c1 c1(SC)cc(C(=O)N(C)Cc2ccccc2CNC(=O)CC(F)(F)F)c(C)o1 NC(=O)CCC(=O)NCCC1(O)CN(C(=O)C=CC(=O)NCc2ccccc2)C1 c1(C(N2CCN(C(c3[nH]cc(C)c3)=O)CC2CCO)=O)ccc2nc(O)sc2c1 C1(C(=O)NC(CC=C)CO)CC(NC(=O)CC2CC(OCC)C2)CCO1 c1(C(N2CC(OC)C(NC(=O)C(C)(C)c3ccsc3)C2)=O)nnn2c1CCCC2 C(=O)(CC(CC=C)NC(=O)C(C(C)OC)N(C)C)N(CCC=C)CC C(=O)(C(F)C(C)C)OCc1nnc(CC)s1 C(C(=O)N(CCCNC(=O)CCSC1CCCO1)C(C)C)(SC)SC C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(=O)C(F)C(C)(C)O)C2(CCCCC2)C1 C1(C)(NC(c2nccc(CC)c2)=O)CCCCC1C(=O)NCC(C1CCCC1)OC N1(C(CC(C)c2cnn(C)c2)=O)CCC2CN(C(=O)CC3CCC3)CC2C1 N1(C(C(C)NC(C)=O)=O)CC2(C)CN(Cn3ccc(C4CC4)n3)CC2(C)C1 c1(C(=O)NCC(CCNC(=O)CC2CCOC2)O)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC2(C)CN(C(c3cc(OC)cc(OC)c3)=O)C2)cc2sc(F)cc2[nH]1 CC(CC(=O)NC(C1CCN(C(c2scnc2C(C)(C)C)=O)CC1)C)P(C)(C)=O CCC(CC(C)C)C(=O)N1CCC(CC(=O)NCC2(CN(C)C)CC2)CC1 C12(C(=O)NCCN(CCO)CC)CCCCC1N(C(=O)C(C)CCOC)CCC2 Cn1cnc(C=C(F)C(N2CCCC2CC2C(C)(C)C2(C)C)=O)c1 c1(C(N(C2CCCN(C(C3CS(=O)C3)=O)CC2)CC)=O)cccc2occc12 C12(C(CNC(Cn3ncc(C)c3)=O)NC(=O)CC3CC3(Cl)Cl)CCC(CC1)C2 Cc1nn(CC(C)C)c(C)c1CN1CCN(C(=O)NC(C)(C)C)CC1C(F)(F)F c1(N2CCN(C(C(C(=O)OC)(C)F)=O)CC2)cc([N+](=O)[O-])ccc1Br CC1CC(C(=O)N2CCC(C)(C)C2CNC(=O)CC(C)(C)C)=NO1 CCCC(C)(O)CC(=O)N1CCOC(C(=O)NCCc2ocnc2CO)C1 c1(C(=O)NCC(c2ccccc2)N(C(C(C)C2CC2)=O)C)cnn(C)c1 C12(C(=O)NCCCN(C(c3ccc(COC)cc3)=O)CC)CCC(O)(CC1)CC2 N1(C(c2cc(C(C)C)no2)=O)CCC2C(CCN2C(=O)CC2(C)CCCCC2)C1 Cc1nocc1C(=O)N(C(C)CC(=O)N1CC(c2cccnc2)C1)C C(=O)(CC(C)CC(C)C)NCCC1(OC)CN(C(c2nnsc2N)=O)C1 c1(C(N2CC(NC(c3cnn(CCC)c3C)=O)C(O)C2)=O)ccc(C#N)cc1C c1(C(=O)NCCC(C)(C)NC(CN(C2CC2)CC)=O)cc2cc(F)cc(F)c2[nH]1 C1(C(=O)NCC2(CC(=O)NCCCN3C(C)CCC3)CC2)CC(=O)OC1(C)C CC1CN(C(=O)CN(C)CCO)CCCN1C(c1ccc(OC(F)(F)F)nc1)=O c1(OC)cc(C(=O)Nc2cccc(F)c2Cl)c(NCc2cc(Cl)cnc2Br)cn1 N1(c2ccnc(NCCCc3c(OC)cccc3)n2)CC2(C1)CN(C)CCO2 CC1CC(C(=O)NC2COCC2CO)CN(C(c2ccnc(O)c2)=O)C1 CC1(C)CCN(C(c2nc(Cl)cs2)=O)C1C(=O)NC1CCCC1N=[N+]=[N-] Cc1cccn2cc(CC(=O)NCC3CCC(NC(=O)C(O)C(F)(F)F)C3)nc12 Cn1cc(C=CC(=O)NC2(C)CC(NC(c3cn(CC(F)(F)F)cn3)=O)C2)cn1 N1(C(C2N(C(C)=O)CSC2)=O)CCCC(N(C)C(C2COCCO2)=O)C1 C(=O)(C(C(C)C)OC(c1cncc(-c2cccnc2)c1)=O)NC C=CC(C)(CC)C(=O)N1CC(CNC(C2CCC3(CC2)CC3)=O)C(F)(F)C1 C=CC(CCC)CC(=O)NCCN(C)C(c1c(F)cc(OC)cc1Cl)=O CC(O)(Cc1ccccc1)C(=O)NCC(CC(F)(F)F)NC(C1(CO)COC1)=O N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2cccc(F)c2C)=O)CC1CC(C)(C)C C1(OC)CN(C(=O)C(C)(CSC)NC(C2CC(SC)C2)=O)CC12CC2 Cc1cc(Cl)c(C)c(C(N2CC(CO)(NC(=O)CCC=CC(C)C)C2)=O)c1N CC1(C)CN(C(C2CCNC(=O)CC2)=O)CC1c1cn(-c2ccc(F)cc2)nn1 c1(NC(C(N2CCC(CNC(C3CC(=C)C3)=O)C2)=O)C)ccc(Br)cc1 c1(NCC2CCN(CC)CC2)nc[nH]c(=NCC2(F)COCCOC2)c1C Cc1cn2c(C(=O)NCC3CCN(C(C4CCCS(=O)(=O)C4)=O)C3)c(C)nc2s1 CC(=O)CCCC(C)C(=O)NCCC(=O)N(C)C(c1nccs1)C NS(=O)(=O)c1ccc(F)c(NC(c2ccccc2CF)=O)c1 C=C(Cl)CCC(=O)NC1C2CC(NC(c3cn(CCC)nn3)=O)CC12 C(=O)(CCC(CF)CF)NC1C(C(N2C(C(=O)NC)CC(O)C2)=O)COCC1 C#Cc1ccccc1CNC(=O)CC(C(C)OC)NC(=O)C(C)OC NC12CCOCC1CN(C(=O)C=CCN1CCOCC1)C2 C1(C)(NC(Cc2nc(C(C)(C)C)sc2)=O)CCN(C(=O)C(=O)NCC(F)F)C1 N1(C(Cc2ccc(C)o2)=O)CC(CCNC(=O)CC2(C#N)CC2)OC(C)C1 C12(CNC(c3ccc(CC)cc3)=O)CC(NC(c3ncccc3Br)=O)(CCO1)C2 C1(NC(C2(N(C)C)CCC2)=O)C2CC1N(C(C1CC1c1cccc(Cl)c1)=O)C2 CCC(C)C(O)CC(=O)N1CCCC(C)(C(=O)NC2CCN(C)C(C)C2)C1 c1(C(N2C(CNC(C3N(C(C)=O)CCCC3)=O)C=CC2)=O)nccc2n[nH]cc12 N1(C(C(C)=C2CC2)=O)CCC(F)CC1C(=O)N(C1CC(C)C1)C N1(CC(C)(C)NC(C(CN(C)C)O)=O)CCN(C(=O)CC2CCC(=O)N2)CC1 S(=O)(=O)(c1cccnc1N1CC(F)C(F)C1)NC(C)C(C1CCCCC1)C C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(Cc2nc(CC)sc2)=O)CC1C1CC1 Cc1cccn2cc(C(=O)NC(C)CCCNC(=O)C(CO)C(C)C)nc12 CCCCCCCC(F)C(=O)NC1CCCCC1CNC(=O)C=C1CCOCC1 C1(NC(c2nc(C)oc2)=O)CN(C(c2cnsc2)=O)CCC1C C(=O)(C(C)(CC)C(N)=O)NCC(C1(O)CCN(C(C=CC=CCC)=O)C1)C C(C)(C)(C(C)CC(=O)N1CC(C)(O)C1)NC(c1nc(C)oc1)=O C1(C(=O)NC2C(C)(C)CN(C(c3cnc(O)n3C)=O)C2)CCCC2(C1)CC2(F)F c1(C(N2CC=C(CCNC(CC(C)(C)SC)=O)CC2)=O)ccc2cn(C)nc2c1 C(CC(C)(C)C)(C(=O)Nc1cnc(F)c(C)c1)NC(C12CCC(OC)C1C2)=O c1(C(=O)NCCC(C)NC(C(C)C#N)=O)cc(Cl)ccc1OCC(F)(F)F c1(CC(N2CCC(CNC(C(F)=CCC)=O)C23CC3)=O)ccc2nc[nH]c2c1 c1(N(CCCCOC)C)cccc(S(=O)(=O)NC2CCS(=O)(=O)C(C)C2)n1 CC(C)CCC(=O)N(C(C)C(N1CCC1(C)CCO)=O)C1CC1 c1(OC)ccc(CCC(=O)NC2CC2NC(=O)CNS(N)(=O)=O)cc1OC C12(NC(C=C(C)C)=O)CC1CN(C(=O)CCc1ccccc1OC(F)(F)F)C2 C1(CC)CN(C(C2CCC(C(=O)NCc3ccc(CC(=O)O)cc3)C2)=O)CCO1 C1(CC(N2C(C)(C(=O)OC)CC2)=O)CC(NC(=O)CNC(=O)CC(C)C)C1(C)C CN1CCC(C(=O)NCCC2(O)CN(C(c3[nH]ccc3-c3ccccc3)=O)C2)C1 c1(OC)ccc(CCC(N2CCCC2c2cccc(Br)c2)=O)cc1 C1(NC(C(C)OCCCCCC)=O)CC(CNC(c2cc(=O)n(C)o2)=O)CC1O c1(CC)c(C(=O)NC2CCN(C(C34CCCC3CC4)=O)CC2)oc2ccccc12 N1(C(c2c(COC)scc2)=O)CCC(N(C(=O)C2=CCSC2)C2CCOCC2)CC1C Cc1nc(N2CC3(CCCC3NC(=O)C3=C(Cl)CCOC3)C2)c2ccsc2n1 C=C(Cl)CCC(=O)NC(C)CCCCNC(=O)C(C)COC(C)=O C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CCC(NC(CCSCCC)=O)CC1 c1(CC(N2CCC(N(C(C=CC)=O)C)C2)=O)ccc(OC)cn1 C12(NC(C(CC=C)(F)F)=O)CCC(CNC(=O)COCCOCC)(CC1)OC2 c1(C(=O)OCC)cc(NCc2cn(C)nc2C(F)F)ccc1C C(=O)(C1CCc2nnc(C)n21)NCCC1N(C(Cc2cc(C)no2)=O)CCSC1 N1(C(CC2CCC(OC)CC2)=O)CC2CC(C1)CN(C(=O)Cn1ccc(C)n1)C2 C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(CNC(CCC(CC)OC)=O)C N1(Cc2cc(C(=O)OC)n[nH]2)CCC2C(C1)NC(=O)CCN2C C(CNC(C1COC(C)(C)C1)=O)(CC)(CC)NC(c1nc(CCC)oc1)=O C1(CNC(CCC#C)=O)COC(C)(C)CN1C(c1ccc(-n2cccn2)c(C)c1)=O c1(C(=O)OC)cc2c(s1)CCN(C(c1cccnc1C)C(=O)NC1CCCC1)C2 C#Cc1cccc(CC(=O)NC2CC3C(NC(C4(OC(C)=O)CC4)=O)C3C2)c1 C(=O)(CC(C)C(C)(C)C)NCC(C)(CC(C)C)NC(c1c(CCC)sc(S)n1)=O C(=O)(C1=CC(C)(C)C1)NC(C1(C(N(CC)Cc2cnn(C)c2)=O)CC1)C N1(C(CCC)=O)CCCC(C(N2CCCC2COC)=O)C1CC C=CC(C)CC(=O)NC(CCOC)C(=O)NC1CCCC1CCOC c1(CNC(=O)Nc2ccc(OC)c(F)n2)c(O)cc(F)cc1F C1(C(N2CC(OCCOC)C2)=O)CC12CCN(C(=O)Cc1ccsc1C)CC2 C1(C(=O)NC(C(C)F)C)CCC(C2CC2)N1C(=O)C=Cc1nccs1 CCCCC(C(=O)NC1CCN(C(N)=O)C1)NC(=O)C(CCC)N(C)C CC1CC(C(=O)NC2CC3CN(c4ccnc(C#N)n4)CC23)=NO1 C12(C(=O)NCC(N(C(C3(OC)CCSC3)=O)C)C3CC3)CC(C)(C1)OC2C N1(C(c2ccc(C3CC3)cc2)C)CC(Cc2c(C)cccc2)CCC1C N1(C(C2(CSC)CC2)=O)CCC(F)(C(=O)NC2(CF)CC2)C1 C1(C(=O)N(C)CC2CCCC2(C)C)(SC)CCN(C(=O)C(C)SC(C)C)C1 c1(CN2CC3N(C(c4c(C)cnn4C(C)C)=O)C3C2)ccc2ncnn2c1 N1(C(C(CC)C2CCOCC2)=O)CCC(C)(CCNC(c2c(C)ncn2C)=O)C1 c1(NC(C(=O)N(CCC2CCOC2)CC)=O)cc(OC)c(OC)cc1OC N1(C(c2ccccc2)C)CCC(C)(NCc2cn(-c3cccc(Br)c3)nn2)C1 CC(C)(C(=O)NC1CCCC(CNC(c2c[nH]nc2Cl)=O)C1)C(F)F C(=O)(C(C)(C)CCCO)NC1(CC=C)CN(C(=O)C=CC(c2ccccc2)=O)C1 c1(OCC)cc(C(=O)NCC(C)N(C(=O)Cc2cnccc2C)CC)ccc1C c1(C(=O)NCC(C)CNC(=O)C(C)C2CCCO2)ccc(C2CCC2)nc1 C1(C(=O)NC2C(C)N(C(c3cnn(C)c3N)=O)CC2)CNC(=O)CC12CCOC2 c1(SC)ncc(N)c(C(=O)NC(C)CCNC(=O)Cc2cc(F)cc(Cl)c2)n1 C(=O)(N=c1cc(C(=O)NC2CCC3(CC2)CNC3)[nH][nH]1)c1c(N(C)C)nccn1 CC(C)CC(=O)C(=O)NCCC1(C(N2CCC(CCCO)C2)=O)CCC1 C1(CC(=O)NC2CCC(CCNC(c3c(C)ccs3)=O)C2)CCCC(C2CC2)O1 C(N=c1ccnc[nH]1)c1nc(CNC(=O)C=Cc2cc[nH]n2)nc(O)c1 C(=O)(CC(CC)C(C)(C)C)N1CCC(N(C(c2ncc(C#C)cc2C)=O)C)C1 c1(CCC(=O)NC(C2(O)CN(C(c3cc[nH]c3)=O)C2)C)ccc(Br)s1 c1(OCCC)ccc(N(C(c2ccnc(F)c2)C(=O)NC)C)cc1 c1(C(=O)OC)ccccc1CNC(=O)CC1(C(N(C)C)C2CC2)CC1 O=C(CCS(=O)(=O)C(F)(F)F)NCC1CC(O)CN1C(=O)CCC(F)(F)F C1(C(=O)NCC2CCC23CCC3)CCC2(CC2)N1C(=O)CN1CCSCC1 N1(C(C(CCC)OC)=O)C2CCC1CC(F)(CNC(C1(CC)CCC1)=O)C2 Cc1cc(C(N2CC3CC2C3CNC(=O)C(C)(C)COC(C)C)=O)c(C)n1C1CC1 C1(OC)(CNC(=O)C=CCCc2ccccc2)CCN(C(C2(C)CC2C)=O)C1 C1(C(N2CC(C(=O)NCC(=O)OC(C)C)(COC)C2)=O)CC2CC(=O)C1O2 C(=O)(C#CC1(C)CCCO1)N1CCC2(CC(C(N(CC(F)F)C)=O)C2)C1 c1(C(=O)NCCC(C)NC(=O)COC2CC2)ccc(Cc2cccs2)cc1 c1(NC(CCCCC)C2CC2)nc2ccccc2nc1NC1CCN(CC)C1 C1(C(=O)NC2CN(C(C(CC)OC3CCCCC3)=O)C2)CC(S(C)(=O)=O)C1 C1(NC(c2ccc(OC)nn2)=O)CCCCN(C(C2OCCC2C)=O)C1 c1(NCC2C(C(=O)OC)C2)cccc(NC(C2CC(F)CN2C(C)=O)=O)c1 c1(C(=O)NCCCC(C)NC(=O)C=CCN(C)C)ncnc2c1cnn2C c1(C(N(C2CN(C(c3c(SC)csc3)=O)CC2(C)C)C)=O)cccn2nncc12 C1(CC(=O)NC2CN(C(C3CCC(=C)CC3)=O)C2)CCCC2CCCCC12 c1(C(=O)NC(CN(C(=O)CC2CC3CC3C2)C)(C)C)ccc(S(N)(=O)=O)s1 C1(NC(CSc2ccc(OC)cc2)=O)CN(C(=O)CC2CCN(C)C2)CCC1F Cc1ccc(CC(=O)NC2CC2CNC(c2cn(C(C)(C)C)nc2C)=O)c(C)c1 c1(N(CC=C=C)C)nc(-c2ccccc2)nc(=NCCCOCCCO)[nH]1 C1(c2nnnn2C2(C)CC2)(NC(c2cccc(NC)c2)=O)CCOCCC1C c1(CC(C2CC2)NC(=O)NC2CCCCC2)ccccc1 CC(C(=O)NC1(C)CC(NC(=O)CCOc2ccc(F)c(F)c2)C1)S(N)(=O)=O CCCC(C)(CC)C(=O)NCC(C)(C)CNC(c1ccc(=O)n(CC(C)O)c1)=O N1(CC)CC(NC(=O)C(c2ccco2)NC(c2cc(C(F)F)[nH]n2)=O)CCC1=O C#Cc1cncc(C(=O)NCC2CN(C(=O)CC(=O)NCC3CC3)CC2(F)F)c1 C1(CNC(CC(C)SC)=O)CCN(C(c2cc(Cl)nn2C)=O)C1(C)C N1(C(C(COC)(C)C)=O)CCC2CN(C(=O)C=CC(=O)N(C)C3CC3)CC2CC1 c1(C(=O)OC(C(=O)NCCC2C(C(=O)OC)CC2)=O)ccc(C(F)(F)F)cc1 C1(C(N2CCC(F)(CNC(C(C)(C)CF)=O)C2)=O)CC2CCC1CC2 C1(NC(C(C)NC(N)=O)=O)CCC(CNC(=O)CCCn2ccnn2)CC1 C(C)(CN=c1nc(C(C)(C)C)nc[nH]1)N(C(CC(CC)CNC(C)=O)=O)C c1(NC(CC)=O)ccc(C)c(C(=O)NC2CCCC2NC(=O)C(Cl)=CCl)c1 c1(C(C)C)n[nH]cc1C(=O)NC1COCC1C(=O)N(C)Cc1ccon1 CCC(CC(F)F)C(=O)N1CCOCC(NC(C2(C)CCC(=O)NC2)=O)C1 C1(NC(c2c(C)nc(CO)s2)=O)COC2(CCN(C(c3ncn(C)c3C)=O)C2)C1 C(CCCCCCCC1CC1)(N(C)Cc1ccc(F)cc1)C1CC1 C(c1cccc(C)c1)=CC(=O)N(CCNC(=O)CC(C)(O)C1CC1)CC N1(CC)CCN(CCC(=O)NCC#CCNC(C2(O)COC2)=O)CC1 C(C)(C)(C(=O)NCCCCCNC(C1CC(O)C1)=O)OCC C1(CNC(C2CN(C(C)=O)C2)=O)CC(C)CCN1C(=O)C(O)C1=CCCC1 c1(NC(c2ccc(NS(=O)(=O)CCCl)cn2)=O)cc(Cl)nc(Cl)c1Cl c1(C(N2CCCCC(CNC(=O)Cn3cncn3)C2)=O)ccn2c(O)nnc2c1 C1(C(N(CCCC)CC)=O)(NC(c2cncn2C)=O)CC(O)C1 CCC(C)C(CC(=O)NC1CCC(=O)NC1(C)C)NC(=O)C(C(C)C)N(C)C C1(C)(C(=O)NC2C(NC(C3(CCOC)CC3)=O)CCC2)CC2(C1)CC(F)(F)C2 c1(C(=O)NC2C3CN(C(c4cocn4)=O)CC23)ccc(Br)cc1I N1(C(CCOC(CC(C)C)C)=O)CCCC(N(C)C(C2(O)CCOCC2)=O)CC1 CCCCC(CNC(=O)CCC(C)OC)NC(C1CCCN1C1CC1)=O C1(NC(c2cnc(CC)o2)=O)CN(C(C2CC(C)CC(=O)N2)=O)C(C)(C)C1 Cc1cc(C(=O)NCC2(NC(=O)CSc3cn[nH]c3)CC2)c(C)n1C(C)C c1(NCC)ncccc1C(N(C1CC(NC(=O)CCCCNC(=O)OC)C1)C)=O N1(Cc2ccc(C(=O)OC)cc2)CCC(CN2CCCC3(CC3)C2)CC1C C1(C(C)CO)CCN(C(C2C3CN(Cc4cc(Cl)ccn4)CC23)=O)CC1 C1(C(CNC(C=C(CCC)C)=O)(C)C)CCN(C(=O)CCC(C)SC)CC1 C1(C(C)(C)C)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CCN1C(C1CCOC1)=O C#CCC(O)C(=O)N(CCCOCCNC(c1n[nH]c(C)c1Br)=O)C N1(C(=O)N(C(C2CC2C(C)(F)F)=O)C2CC2)CCCCC1C(O)C1CC1 C1(CCCC)(C(=O)NCC2CCN2C(C2CC3CC3C2)=O)CCCC1 Cc1cc(C(N2CC(NC(c3c(C)ncn3C)=O)CC(C)C2)=O)ncc1N N1(C(C=Cc2cn(C)nc2)=O)C2CCC(C2)C1C(=O)NCC1CC(=O)N(C)C1=O c1(C(=O)NC2(COC)CN(C(C3CCCS3)=O)C2)ccc2nnc(S)n2c1 C(CO)(C(=O)NCC1(NC(=O)CN2CC3CC3C2)CCCC1)N(C)CC N1(C(CC(C(C)C)O)=O)CCC(C(=O)N(c2cccc(C#N)c2)C)C(C)(C)C1 c1(C(N2CCC2CNC(C2C(=O)NCCC2C)=O)C)cccc2ccccc12 N1(C(c2cnc(C)nc2)=O)CCC2(CC1)CCN2C(c1cc(Br)c(C)cc1O)=O C#CCC(C)(CC)C(=O)NCC(C)(C)C#CC(=O)Nc1ccc(F)nc1 Cn1nc(Br)c2cnc(N3CCCC34CCN(C(=O)CC3C=CCCC3)C4)nc12 CC1SCCCC1C(=O)NCCNC(c1cc(-c2ccn(C)n2)on1)=O c1(C(N2CCC3CN(C(C4C5CCCOC45)=O)C3C2)=O)cccc2nc(Cl)cn12 C(=O)(CC(C)(C)CC(=O)NCc1cn(C2CC2)cn1)c1ccc(C)cc1 c1(C(N2CC3C(N(C(C=CC=CC)=O)C)C3C2)=O)cc(O)ccc1CC C1(NC(=O)Cc2ncc(Cl)s2)CC2CC1CN2C(=O)CN1CCOCC1=O CCCCS(=O)(=O)CC(=O)NC1CCCC(NC(c2nc(C)c(N)cc2C)=O)C1 C1(CNC(CC=CCC)=O)CN(C(=O)COc2cc(C)on2)CC1(F)F C(C1(C)Cc2ccccc21)NC(C)(C)C.c12nc(SCC)cc(n1)N(C)C2C C1(CNC(CCCNC(C)=O)=O)CCN(C(c2cc(C(F)F)nn2C)=O)CC1C C(=O)(C1CCc2nccn21)N1CCN(C(C2(C)CSC2)=O)CC1CO C#CCC(C)(CC)C(=O)NCC(C)(CC)NC(c1ncc(C(N)=O)cc1Cl)=O C(=O)(CC(C)(C)CC=C)NC1CCC(C(=O)NCC2(C#C)CCC2)CC1 c1(C(=O)NC2CC(NC(COc3cccc(C)c3)=O)C2)cn(C)c(=O)nc1O C(=O)(CCC1(NC(c2ccon2)=O)CCC1)NC(C1(C)CC1)CO C1(NC(COC(C)=O)=O)CCCC12CCN(C(c1cccc3nsnc13)=O)CC2 N1(C(c2c(C)ccnc2)=O)CC2CCC(C1)C2NC(=O)C(C)Cc1ccccn1 C(=O)(C1=NNC(C(F)(F)F)C1)NCC1C2CN(C(c3nn(C)c(Cl)c3)=O)CC21 c1(CNC(C2(COC)CN(C(=O)CC3CC4CC4C3)C2)=O)cc(OC)ncn1 Cc1ccccc1C(C)CC(=O)NC1(CN(C(=O)C(C(C)C)N(C)C)C)CC1 N1(C(C23C(NC(C4C(CC(C)C)C4)=O)CC(CC2)C3)=O)CCC(=C(F)F)CC1 CN1C(=O)CSC1=CC(=O)N1CC2C(CNC(C3CCCS3(=O)=O)=O)C2C1 CCCC(CC(C)C)C(=O)N1CCOC(C(=O)NCCCCCC(C)C)CC1 c1(C(N2CCC(C)(CNC(C(C)SC(C)C)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(=O)NC(CNC(CCOCC)=O)(C)C)ccnc(OCCO)c1.CC(F)(F)F c1(N(C(c2cccc(Cl)c2Cl)C(=O)NC(C)C)C(C)C)cccc2ccccc12 N1(C(CCCCCNC(=O)C2=C(Cl)CCC2)=O)CCC2C(C1)C2(F)F c1(OC)ccc(-c2cnccc2C(=O)Nc2sncc2C(N)=O)c(OC)c1 c1(C(=O)NCC(C)CNC(C2CC2c2ccccc2F)=O)cc2cccnn2n1 N1(C(C(C2CCC2)NC(Cn2ncc(C#N)c2)=O)=O)CC(=O)NC(=O)C1 n1(CC)cc(Cl)cc1C(=O)NC(C1CCN(C(C2(C3CCCO3)CCC2)=O)C1)C C1(C(N2CCCC2CC2CC2)=O)(OC)CCN(C(c2cnco2)=O)C1 C1(NC(c2c(C)c[nH]c2)=O)CC(O)CN(C(c2cn(C)nc2-c2ccoc2)=O)C1 c1(C(=O)NCCNC(C2N(CC)CCCC2)=O)c(Br)nc2n1CCC2 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CC(CNC(=O)Cc2cn[nH]c2)C2(CC2)C1 C(CCC(C)CC(=O)NC1C2CN(C(=O)CS(=O)(=O)N(C)C)CC12)=C(C)C C(C1CCCc2ccccc21)NC(C1N(c2nc(OC)c(C#N)cn2)CCOC1)=O c1(C(n2cc(-c3ccc(Br)s3)nn2)COC)ccccn1 c1(C(=O)NCCC2CCCN2C(C2C=CCCC2)=O)ncncc1Br N1(C(C(CC=C)NC(c2cc(CC)no2)=O)=O)CCCN(C)CC1CC c1(C(=O)NC2CCN(C(C=NOC)=O)C2)nc2c(cc1Br)OCCO2 C=CCC(CC(C)C)C(=O)Nc1ccccc1OCc1cccs1 c1(C(=O)NCC(C(C)(C)C)NC(c2ccc([N+](=O)[O-])s2)=O)cnc2[nH]ccc2n1 Cc1cc(C)n(C(C)CC(=O)NC(CCNC(=O)Cc2cnc(C)s2)C(C)C)n1 CC(CC(=O)N1CCCC1CN1CCCCC1)C(=O)c1cccc(F)c1 c1(CC)cc(F)ccc1C(=O)NC(CNC(=O)C(CSC)c1ccccc1)CC Cc1cc(F)c(NC(=O)CC(=O)c2ccccc2)c(Br)c1 Cc1ccc(OC(C)C(=O)NC2C=CCN(C(c3c[nH]nc3C)=O)C2)c(C)c1 N1(C(c2ccn(C)c(=O)c2)=O)CC2=C(C1)CN(C(C1CCc3ncsc3C1)=O)C2 CC1CC(=O)NC(C(N2CCCC(CC(=O)NCC3CNC(=O)C3)C2)=O)C1 C(=O)(C(C)(C)C(F)(F)F)NC(CC1CN(C(CC2CC(OCC)C2)=O)C1)C c1(N)nc2cc3ccccc3cc2s1.C1(CN)CC(=O)N1.C(C(=O)O)OC c1(C(=O)NCCC(C)NC(C23CCC(CC2)C3)=O)cc(N)cc(S(C)(=O)=O)c1 N1(C(=O)OC(C)(C)C)CCCCCCC1C(=O)NCC1(O)CC(CN)C1 c1(OC)ccc(CC2CCCN2C(C2CCN(C)CC2)C(=O)NC)c(Br)c1 C1(C2(NC(CCNC(N)=O)=O)CC2)CCCCN1C(=O)CC1CC2(CC2)CO1 C1(C(C(=O)NCCCN(C(=O)C(C)N=[N+]=[N-])CC)(F)F)(OC)CCCCC1 c12ccnc(c1)NC(=O)C2.CC1(CC2CC2)CN(C(=O)CCC2CCCC2)C1 c1(C(=O)NCC=CCCNC(c2cc(OC)ncn2)=O)cc2sccc2[nH]1 c1(C(=O)NC(C(C)NC(=O)C(C2CCOCC2)O)CO)c[nH]c(=N)c2[nH]ccc12 Cc1sc(NC(c2cnc(NCCc3c(Cl)ccc(Cl)c3Cl)s2)=O)cc1[N+](=O)[O-] O=C(C1=CNC2=NCCCN12)N1CC2CCN(C(C3CC34CC4)=O)C(C2)C1 c12ccc(cc1)s2.N#CC(C(=O)NCC1CCN(S(C)(=O)=O)C1)C1CC1 c1(C(=O)NCC2N(CCC)CC2)sc(Cl)nc1C N1(CC(=O)NC)CCCC2(CCN(C(=O)C3CCCc4c3ncn4C)C2)C1 C(=O)(CCC(C)(C)NC(=O)COCCN(C)C)NCC(C)(C(N)=O)OC N1(C(c2ccc(O)cc2Br)=O)CCCC2(C1)CN(C(c1cc(O)no1)=O)C2 CCCCC(CC)CC(=O)NC1CC(CC(=O)NCCOCC)C1(C)C N1(CC=C)CCC(C(C)(C)CNC(=O)C(c2ccc(F)cc2)C)CC1 C(=O)(CCCC(=O)N(C1CN(C(C2CC(F)(CO)C2)=O)CC12CC2)C)OCC C1(CCC(=O)N(C)Cc2snc(C)n2)CCCCN(C(=O)C(C)c2ccsc2)C1 N1(C(C2N(CC)CC2)=O)CCC2CN(C(c3cc(C)cnc3F)=O)CC2CC1 CN1CCC2(CC1)CC2CNC(c1ccc(C(F)F)nc1)=O Cc1ccnc2c(C(N3CCC4(CCN(C(=O)C(C)(C)C)CC4)C3)=O)cccc12 N1(C(CC2C(SCC)C2)=O)CCN(C(C2CCSC2)=O)C(C2CCC2)C1 c1(OC)noc(C)c1C(=O)NCC1(F)CN(C(C2CN(C)CC2C)=O)C1 C1(N(C)C)CCCN(N(C)C2CN(c3ccccc3)CC23CCC3)C1 N1(C(CC(C=C)C)=O)CCC2(CC1)CN(C(=O)CCc1cc(Cl)no1)C2C(C)C Cc1ccnc(N2CCCC2c2cnc[nH]2)c1-c1ccc(CO)cc1 C(=O)(CC(CC)NC(c1ccn(COC)n1)=O)N(CC#C)Cc1ccco1 c1(C(C(=O)NC(CC)CNC(=O)CCc2cccs2)C)ccc(OC)cc1C c1(C(=O)NC2CC(CNC(C(C)(C)OC(C)=O)=O)C2)n[nH]c(C)c1Cl CC(CC(N)=O)C(=O)N1CCC(CCN(C)C(c2ncncc2N)=O)CC1 C1(C(=O)Nc2c(OCC)nccc2)CCC2(COC2)N(C(=O)OC(C)(C)C)C1 c1(COC)ccnc(C(=O)N(C2CCN(C(=O)C(C)SC3CCCCC3)C2)C)c1 c1(CC(C(=O)O)NC(CC2CCC(C)C2)=O)cc(F)ncc1Br C(=O)(CCCC(C)C)NC(c1c(OC)cccc1)C(C)NC(c1ccoc1)=O N1(C(C(C)(F)F)=O)CCCC(N(CCO)C(C2CCN(S(C)(=O)=O)CC2)=O)C1 N1(C(CCCCCC)=O)CCc2nc(CNC(=O)C(CC(C)C)C(C)C)sc2C1 c1(C(=O)NC2CN(C(COCCC#C)=O)C(C)C2)cc(Cl)c2ccccc2c1O N1(C(c2c(C)cc(C)[nH]2)=O)CC2CC(NC(c3ccc4c(c3)CCC4)=O)C(C2)C1 c1(C(N(C2CCN(C(c3cc(C)[nH]c3C)=O)C2)CC)=O)cc(C)n(C)n1 C1(NC(CCc2n(C)ccn2)=O)CC(C(=O)NCc2ccnnc2O)C12CCC2 C1(=CCNC(Cc2cc(C)on2)=O)CCN(C(C2(CC(C)C)CCNC2=O)=O)CC1 Cc1cccc(C(O)C(=O)NCCOCCOCCNC(C2CC2(F)Cl)=O)c1F CC(CC(=O)NCCC1(CNC(C2CC(=O)NC(=O)N2)=O)CC1)C(F)F C12CCN(CC1)C(=O)C2N1CCC1Cc1cncn1C.N1(CC)CCC1C(=O)OC C(=O)(C1=CCCCC1C)NC1CN(C(C(COC)C)=O)CC(C)C1 N1(C(Cc2cc(C)no2)=O)CC(N(C(=O)Cc2c(C)n[nH]c2C)C)C2(CC2)C1 C1(CC(=O)OC)CCCN(C(c2cn(C)nn2)C(=O)NC2CCOC(C)C2)C1 C1(NC(C2CCC(=C)CC2)=O)CC2CC(NC(=O)CC(O)CN(C)C)C1C2 c1(OC)nc2ccccc2c(=NCC2CC2CN2C3CCC2c2ccccc23)[nH]1 CC(C(=O)N1CCC1CNC(c1ccc(C(N)=O)o1)=O)C(C)(C)C C(CC(C(=O)NCCNCCN=[N+]=[N-])NC(=O)C(C)CC1CCC1)SC C1(N(C(Cc2c(C)occ2)=O)C)CCN(C(=O)C(F)=CCCF)CC1C c1(OC)ccc(C(N2CC3CC(NC(=O)C(C)C4CCC4)C2C3)=O)cc1O CN1CCCC(C)(C)C1CNC(=N)N1CCC1 O=S(=O)(c1[nH]c(=NCC23CCCC(CO2)C3)ccc1Br)NCC12CCCC1C2 C1(C(=O)NCCC(=C)CNC(=O)CCCOC)CN2CCN1CC2C C1(NC(C=C(C)C2CC2)=O)CCCC(CNC(=O)C=CC2CCOCC2)C1 CC1(O)CCCC(CC(N2CCCC2c2ccccc2Br)=O)C1 c1(C(=O)NCC2(C)CCN(C(c3c(CC)[nH]cc3)=O)CC2)cc(F)c(F)cc1N Cc1nc2ccc(C(=O)NC3CCC4CN(Cc5cncs5)CC4C3)cc2n1C Cc1c(C(=O)N(CCCCN(C)C(C2CCCOC2)=O)C)sc2cncn12 Cc1ccncc1C(=O)N(C1CCCN(C(=O)Cc2ccoc2)C1)C c1(OC)ccccc1C1(C(=O)NCC(C)NC(=O)CC2CCC(C)(C)C2)CC1 C(=O)(C(O)CC(C)(C)C)NCC(CC)NC(c1nc(CC)oc1C)=O N1(C(CC=CC=C)=O)CCN(C(c2[nH]cc(C)c2C)=O)C(c2ccc(F)cc2)C1 C(C(C)(CC)CC)(c1n(CCOCC)nnn1)NCC1(C(=O)NC)CC=CCC1 c1(SSC)c(F)cc(C(=O)O)cc1F.C1(C2CC2)(C)CCCN1OC c1(C(N2CC(NC(C(C=C=C)C)=O)C(F)C2)=O)ccc(Cl)c(OC)c1F C1(C(=O)NC(C2CN(C(C(C3CC3)SC)=O)C2)C)CCN(C(N)=O)CC1 C12(NC(CC=C)=O)CN(C(c3cccnc3)=O)C(COC)(C1)C2 Cn1nc([N+](=O)[O-])cc1C(N1CCC2CCCC12CNC(c1ccc(F)o1)=O)=O C1(C(=O)NC2C(CC)CN(C(C3(F)CCOC3)=O)CC2)Cc2ccc(C)cc2S1 N1(C(CC2CC(OC)C2)=O)CCSCC1C(=O)NC1CC1(C)C c1(NC(CCN(C(=O)C2=C(C)CCOC2)CC=C)=O)cc(C#N)ccc1F C(C(CC(F)(F)F)NC(c1cccc(C(F)F)n1)=O)NC(c1ccccn1)=O c1(C(=O)NC2(C3CCCN3C(=O)CC3CCOC3)CC2)nc[nH]c2ncnc1-2 N1(C(C(C2CCC(=O)N2)C)=O)CC2(C1)CN(C(=O)CCc1nc(O)n[nH]1)C2 C(C1=CCCN(C(=O)Cc2ccc(OC)cc2)C1)NC(CC=CC=C)=O C1(C(=O)NC)(NC(C2CN(C(C(CC)(C)C)=O)CC2F)=O)CCC(C)(C)CC1 O(N=C1CCCCCC1)CC(N1C2CC(NC(c3ccc(OC)nn3)=O)(C2)C1)=O C(CC(=O)N1CCC(NC(c2cccc(N)c2O)=O)CC1C)(C(F)(F)F)OC c1(CC)cc(C(=O)NCC2COCC2NC(C2(OC)CCSC2)=O)cc(O)n1 C(=O)(C1CCc2cc(Br)ccc21)NC1C(CNC(c2cn(CC)nn2)=O)CC1 C(C(C)(O)CC(=O)N1CC2C(CNC(C34CC5CC3C4C5)=O)C2C1)OC c1(CNC(C2CSCCN2)=O)cccc(F)c1Br C1(C(=O)NCCCN(C(=O)CN2CCCCCCC2=O)C)OC(C)(C)OC1(C)C C(c1ccc2c(c1)OC(F)(F)O2)=CC(=O)OCC(c1c(Cl)ccc(Br)c1Cl)=O c1(C(=O)NCC(C(C)C)NC(CC(c2ccc(C)cc2)C)=O)cc(Cl)ccc1F C1(CC(=O)NC(c2cscn2)=O)CCN(Cc2ccccc2F)CC1 c1(C(N(C2CCN(C(C=C(CCC)C)=O)C2)C)=O)cc(=O)n(C)cn1 C1(C(N2CC(O)(C(C)NC(C(C3CC3)OCC)=O)C2)=O)CCC(=C(F)F)CC1 c1(C(C(=O)NC)(F)F)ccccc1C.N12CCC(C1)NS(=O)(=O)CC2 C(N=c1ccnc(N(C)Cc2cc(OC)ncc2F)[nH]1)C1CC(CC)(CC)C1 CN1CCC(C(=O)NC2CC3CC3C2)CC1.C12CCC1C(=O)N2CCO C12(C(N(CCCCCNC(C(C)Cc3ccccn3)=O)C)=O)C=CC(CC1)C2 Cc1c(Br)sc(C(N2CCC2CNC(c2cc3sccc3[nH]2)=O)=O)c1C C1(CNC(CN(C2CCSC2)C)=O)COCCN1C(=O)Cc1cncc(F)c1 C12(NC(=O)CC3CC4(CC4)CO3)CCCC1N(C(=O)CCn1cccc1)CCC2 c1(C(N2CC(O)(C(C)NC(C3CCC3(F)F)=O)C2)=O)cccc(C(F)F)c1F C(CC)(CC)(CCNC(C1(CF)CC1)=O)NC(C1CC(O)(CC#C)C1)=O c1(C(N2CC(Cc3cn(CCCO)nn3)C2)=O)cc(Br)ccc1N1CCOCC1 N1(CC)N=C(C(=O)NC2(C3CC3)CCN(C(=O)CCc3cc(Cl)no3)C2)CCC1=O c1(C(=O)NC2CC2NC(=O)CSc2ccccc2)ccnc(O)c1Br C(CCCNC(=O)C(C)N(C)C)(c1ccccc1)NC(C1C(COC)C1)=O N1(C(C=CC(C)(C)C)=O)CCC2CCCC12CNC(c1ncc(C(F)F)s1)=O C1(C#N)(C(N2CC(C(C)(C)O)(CNC(CCNC(COC)=O)=O)C2)=O)CC(C)C1 c1(C(=O)NCCN(CC(=O)NCCCC)C(C)C)cc(C(C)(C)C)nn1C Cc1oc(C#N)cc1C(=O)NCC(C)C(=O)NC1(C)CS(=O)(=O)C1 c1(CNC(=O)NC(CC(=O)OCC)C)ccc(OC)cc1 C1(C)(CNC(c2n(CCC3(C)CC3)nnn2)c2ccns2)C=CCCC1 CC1(CNC(C2CCCN2C(=O)CCc2cc[nH]n2)=O)CCCCCC1 c1(C(=O)NCC(CO)NC(C(C)Cc2ccccc2F)=O)cc2cccnc2o1 C(=O)(C1=CCCOCC1)NC1CCN(C(c2n(CC#N)ncc2)=O)CC1O CCCCCC(=O)N(C1CCN(C(=O)CC2OCCC2C)CC1)C C1(C(N(C)CC2(Br)CC2)=O)CCCCC1CNC(=O)CN1CCSCC1 C1(C(N2CC(O)CCC(NC(=O)CC3(C4CC4)CC3)C2)=O)CC2C=CC1C21CC1 C1(C(=O)NCc2c(C(N(CC(N)=O)CC)=O)nco2)CCC(C2CC2)C1 C1(C(=O)NCC(CCC)NC(=O)C(C)(C)O)CCCC(F)(F)C1 C(c1cccc(N)c1)=CC(N1CCC(C)(NC(C(C2CC2)SC)=O)C1)=O C12(C(N(C3CCN(C(c4cnccn4)=O)C3)CCCOC)=O)CC(C1)C(C)O2 C1(NC(CC2C(C)(C)C2)=O)C2CC3C(C2)C13C(=O)N1CC(O)CO1 CC1(C)CC(C(=O)NCCOCCC(=O)NCC2CC3CCCC3C2)CCO1 c1(C(=O)NCC(CC=C)NC(=O)CCC2CC(C)(C)CO2)ncc(N(C)C)cn1 c1(C(=O)NCC2C(NC(C=C(CCC)C)=O)C2)cc(C)nc2[nH]nc(O)c12 CN1Cc2c(-c3nc(COc4ccc(F)c(F)c4)no3)cccc2NC1=O N1(C(C2N(C(C(CCOC)OC)=O)CCC2O)=O)CC2(CCOCC2)C1 N1(C(CC2COCC(C)O2)=O)CC2CCN(C(=O)C3=NNC(=O)CC3)C2C1 c1(OC)c(Br)cc(CN2CCCC(C(=O)NCc3ccc(O)nc3)C2)cc1Br O=C(CCC(=O)N1CCCC1C1CCCCCC1)c1ccncc1 CC1(C(=O)NCCC2CCC2)C=CCCC1.N12CC3CC1C3C2=O C(=O)(CC(C)CC(F)(F)F)N1CCCC(C)(NC(c2ccc(C(C)C)cn2)=O)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)CC2C(C)(C)C2(C)C)noc2ncccc12 N1(C(C2(c3ccc(OC)cc3)CCC2)=O)CC2CC(CO)CC(C1)C2O c1(C(=O)NC2(C)CN(C(C3CC=C(C)CC3)=O)C2)cc2n(n1)C(C)CCC2 C1(C(=O)NCC2(C(=O)NC)CCC2)CN(C(C2CN(C)C2)=O)CCC1O C1(NC(C(=O)NCC(CCSCC)N)=O)CCC(C)(C)CC1CN N#CC1(F)CN(C(C2N(C(C3C4CCC(F)C34)=O)CC23CC3)=O)C1 c1(C(=O)NC2CCCN(C(C3CC34CCSCC4)=O)CC2)scc2c1CCCC2 C1(NC(C2CCC(C(C)C)CC2)=O)CCCCN(C(C2(F)CCOCC2)=O)C1 C1(C)(CNC(c2c(C)onc2)=O)CCN(C(C2CCC(CC(C)C)CC2)=O)C1 N1(C(C2CCN(SCCCOC)CC2)C(=O)NCC)CCCCC1c1ccon1 c1(NC(C2N(Cc3ccc(C)c(Cl)c3)CC(C)C2)=O)cccc([N+](=O)[O-])c1Br C1(CNC(C(C)NC(CC)=O)=O)(CO)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C1 C=CCC(C)(C)CC(=O)NC1CCN(C(c2cc(C)cc(Br)c2)=O)CC1F N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CC1CN2C(=O)CC(=O)c1ccco1 CC1(C)CCCC(C(C2(C)OCCO2)O)O1.C1(C(=O)O)CCC(CC)CC1 c1(C2C(C(=O)NC3(CC(=O)NC4CN(C)C4)CCC3)C2)ccc(Cl)c(C#N)c1 C1(CNC(=O)CC2CCSCC2)C2CCC1(c1cccs1)C2.C12CCN1C2=O c1(OC)c[nH]c(C(N2CCCC2N(CC(F)(F)F)C)C(=O)NCCCF)cc1=O N1(C(C2CCCN2C(=O)C(F)Cl)=O)CCOC2(CCC2)C1.c12cccc(c1)NC2=O C(=O)(C(O)CCC(C)C)N1CCC(N(C(c2nc(OC)c(F)cn2)=O)CCO)C1 CCCC(CC)CCC(=O)N1CCC(OC2CN(CC3CC3[N+](=O)[O-])C2)CC1 n1(C(C)C)ccc(C(N2CCC(Cc3cn(CC(=O)O)nn3)C2)=O)n1 c1(NC(=O)NC2CCC(NC(Cc3ccc(C)cc3)=O)C2)cc(C)c(O)cn1 C(N(O)C(=O)Cc1cccc(Cl)c1)c1cn(C(C)C(=O)N(C)C)nn1 N1(C(C2N(C(C3N(C)C(=O)CCC3)=O)CC(O)C2)=O)CC2C=CCC(C2)C1 CC1(CC(N2CC(CNC(c3cn(C(F)(F)F)cn3)=O)C(O)C2)=O)CCCCC1 C1(OC)CCCC(NC(c2nc(C(c3ccccc3)(F)F)no2)C)C1 CC12CCC(C(=O)NC(CNC(=O)C=C3CCC3)CO)(CC1)CO2 N1(C(CCN(CCOCCOC)C)=O)CC(NC(=O)C(F)(F)CO)C(C)C1 C1(C2CC2)(NC(CC(C=C)C)=O)CCN(C(c2noc3c2CCCC3)=O)C1 CC1(C)CCC(C(=O)Nc2cnn(CCO)c2)(NC(C2CCC3(CCC3)O2)=O)C1 Cc1ccnn1C(C)C(=O)NC(C1(O)COC1)C c1(C(=O)OC)ccc(NC23CC(C2)N(C(=O)C(C)(C)N(C)C)C3)cc1OC C1(CNC(c2c(OC)c[nH]n2)=O)CCCC2(CN(C(=O)C(F)C(F)(F)F)C2)O1 C=C1CCN(C(c2cc(C(C)C)no2)=O)C(C(=O)NCC2C=CCCC2)C1 c1(Cc2nc(-c3nccc(OC)c3)nn2C)onc2ccccc12 C1(C(C)C)CN(C(N)=O)CCN1C(=O)C(Cc1ccc(O)cc1)NC(N)=O CC1(C)CC(CC(=O)NCCCNC(c2cccc(C(C)(C)C)c2)=O)NC1=O C1(CNC(C(C(C)C)NC(COC)=O)=O)COCCN(C(c2cc(C)c[nH]2)=O)C1 N1(CC=C)CCC(NC(=O)NC(C)CC(C)c2ccco2)CC1 C1(NC(c2ccc(-c3ccco3)o2)=O)CCCN(C(C23CC(O)C2C3)=O)CC1 c1(C(N(C2CN(C(Cc3cc(C)[nH]n3)=O)CC2F)C)=O)cc2nccn2c(O)n1 C(=O)(CCCc1sccc1C)NC1(CN(C(=O)CC2(CO)CC2)CCC)CC1 C12(CNC(CC(CC)CC)=O)CCCC1N(C(=O)C=C1CCCCC1)CCC2 C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NC(C)CCNC(c1ccccn1)=O CC(C)S(=O)(=O)C(C)C(=O)N1CCC2(C1)CN(C(c1cc(Cl)c(F)c(Cl)c1)=O)C2 Cc1cccc(C)c1C(=O)NC1CC1C(=O)OC(=O)C(C)N(C)C CCC(C(=O)NC(c1ccccn1)C)N(C(=O)Cc1cnsc1)C C(CCCC(=O)NCc1ocnc1C(N1CCOC(C(N)=O)C1)=O)OCC C1(NC(c2c(OC)cc(C)cn2)=O)CC2CC1CN(C(C1CCC(C)C1)=O)C2 C1(C(=O)NC2CCN(C(CC3(C=C)CCC3)=O)CC2F)C2CCCCCCC12 c1(CCC)nc(C)c(C(=O)NCC2CC(NC(=O)C(F)(F)CC3CCCO3)C2)s1 c1(NC)ccc(C(N)=O)cc1C(=O)NCC(C)NC(C1CC=CCC1)=O c1(CC)nc(C)oc1C(=O)NC12CC1CN(C(c1csc(O)n1)=O)C2 C(=O)(CCC(F)(F)F)N1C(C(=O)NC(COC)C2(C)CC2)CCC1 C(=O)(CCCC(CC)NC(c1c(C)ncnc1C)=O)NCC(CCC=C)O C1(O)(CCNC(=O)COC2CC=CC2)CCN(C(C2CC3CCC3C2)=O)C1 C1(C(N(C2CCN(C(=O)CCc3cnccn3)CC2)C)=O)CC(=O)N(C2CC2)C1 c1(C(=O)NC2CC(CNC(CSc3n(C)nnc3)=O)C2)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC(C)CCNC(=O)C(c2cccc(F)c2)C)cnc2n(c1=O)CCS2 c1(C(=O)NCCC(=C)CNC(c2n[nH]cc2F)=O)cncc2[nH]ccc12 C=CCCCC(C(=O)NCC(C)C(F)(F)F)NC(C1COCOC1)=O c1(CNCC2(C(=O)Nc3ccc(C#C)cc3)CC2)n[nH]c2ccc(Br)cc12 c1(CC(N2C(CNC(CC=C)=O)C=CC2)=O)ccc(F)c(Br)c1 c1(NC(C)CNC(=O)C(C2(O)CCCCC2)(F)F)nc(O)n(C)c(=O)c1[N+](=O)[O-] c1(C(C(=O)OCC)N(c2ccccc2)C(C)=O)cccc(Cl)c1 C(c1ccc(OC)c(F)c1)=CC(=O)NC(C(=O)OC)Cc1cn(C(C)(C)C)nn1 CC1=C(C(=O)N2CCCOC(CNC(c3nc(C)nn3C)=O)C2)CCO1 N(C1CCc2cc(CNC(c3cc(CO)on3)=O)ccc21)C(c1cn(C)nn1)=O N1(C(CC(=O)N(C)C)=O)Cc2ccccc2C1CNC(=O)CCC(C)(C)F c1(SC)c(C(=O)N(CCCNC(c2cnc(NCC3CC3)s2)=O)C)csc1C C(C)(C(=O)NCCCCO)N(CCC)C(C1CCO1)=O C1(NC(C(CSC)c2ccccc2)=O)CCCCC1NC(=O)C=Cc1cncn1C C1(NC(Cn2ncc(CC)c2)=O)CCC(C)(C)CC1CNC(c1nnsc1C)=O C(=O)(C1CCCCc2ccccc21)NC1CC(CNC(=O)C2=CCOC2)C1 C12(CNC(C(C)(C)CF)=O)CCC(C1)N(C(=O)C(F)CC1CCC1)C2 CC(=O)C(C)CC(C)C(=O)N1CC(NC(c2ccc(O)nc2)=O)CC12CCC2 C1(CNC(C(CCOC)C)=O)CCCCN(C(c2cc(C3CCC3)no2)=O)C1 c1(OC)ccc(-c2n[nH]cc2C(=O)N(C(C)CNC(=O)C(CO)N(C)C)C)cc1 c1(NC(=O)C(C2CCCCC2)F)nc(C(N(c2ccccc2)CC#C)=O)oc1C C(N=c1ccc2ncc[nH]c-2n1)C1(C)CCN(C(C2CC(F)(CO)C2)=O)C1 C1CCCCCNC(=O)CC(=O)N1CC.C1(C(=O)NC)CCOC(C(C)C)C1 Cc1nc(CC(=O)NC(C2CN(C(c3ccc(C4CCCCC4)[nH]3)=O)C2)C)cs1 c12nocc1C(=O)NC2C.C(CC(C1CC1)C1CC1)NC(C1C(CC)C1)=O C1(NC(C(=O)NCC2CC2)=O)CCCC2CN(C(c3nccc(Cl)c3F)=O)CC12 N1(C(c2c(CC)nc[nH]2)=O)CCN(C(=O)CC2=CCN(C)CC2)C(C)CC1C CC1(C)CC(NC(c2cccc(Cl)c2F)=O)CN1C(C1CCC(=O)C1)=O CCS(=O)(=O)CC(=O)NCC(CC#N)C(=O)NC(CF)C(F)(F)F c1(CNC(C2(NC(c3n[nH]c(C)c3Cl)=O)CCOCC2)=O)ccnc(F)c1F C(=O)(C(C)CC(N)=O)N(C(c1ccccc1)CNC(CC1(C(=C)F)CCC1)=O)C CC1CN(C(c2ccnc(N(C)CCOCCO)c2)=O)CCC1CO C(C(F)(F)CCNS(=O)(=O)CC1(C(=O)OC)CCC1)n1cc(C(C=C)(C)O)nn1 N1(C(C(C)N(C(Cn2ccc(C)n2)=O)C2CC2)=O)CCCN(C)CC1 c1(C(=O)NC(CC)CC(=O)NC(c2ncn(C)n2)C)ccnc2cc[nH]c12 Cc1n[nH]c(=NCC(C)(C(C)C)NC(=O)CC2CCNC2=O)s1 c1(C(N2CC=CC(C(N(CCSC)CC)=O)C2)=O)cnn2cccc2c1 CC1CN(Cc2ccccc2)CC(C)N(C(c2ccc3ocnc3c2)=O)C1 C1(NC(C2(c3ccn(C)c3)CC2)=O)COCCN(C(=O)Cc2ccsc2)C1 CC1CC(NC(c2cc(Br)c[nH]2)=O)CCN1C(c1ncccc1Cl)=O CC1=NN(C)C(=O)C1CC(N1CCCN(CCNC(=O)CN(C)CCO)CC1)=O C(=O)(CCCCC(=O)NC1CC(F)(CNC(C2CCc3cnnn3C2)=O)C1)OC C12(C(=O)NC3CC(C)N(C(=O)C(=O)Nc4ccccc4O)C3)CC3CC1C2C3O CC1(C(=O)NCC2(F)CCC(CNC(=O)C3=NOCC3)C2)CCC(O)CC1 c1(C(N2C(=O)C2)=O)cnc2c(Br)n[nH]c2c1.c1(C(C)(C)C)cnc(C2CCC2)o1 C(=O)(C(O)CC(C)(C)C)N1CCN(CC2CN(C(CCC(=C)Cl)=O)C2)CC1 C(=O)(CCCC(=O)N(C)C)NC(C(=O)NCC1(O)C(C)CCC1)Cn1ccnn1 c1(OCCC(=O)NC(C)C=CC(=O)N(C)CCO)ccc(F)cc1Cl Cc1cc(CNc2ccc(-c3ccc(N(C)C)nc3)cn2)cc(C#N)c1 c1(OC)cnc(F)c(C(=O)NCC(n2cc(-c3cnccc3Cl)nn2)C)c1 C1(NC(CNC(C(CC)CC)=O)=O)CCN(C(=O)C(=O)C(C)(C)C)C(C2CC2)C1 C1(C(C(=O)N(CCCN(C(Cc2c(C)n[nH]c2)=O)C)C)(C)C)CCCN(C)C1 C1(CC)C(NC(c2cccnc2C)=O)CCCN1C(=O)CN1CCC(OC)C1 C1(C(N2C(COC)C=CC2)=O)CC2CC2N1C(=O)C(n1ccnc1C)C c1(N2CC(NC(CCN(C)CC)=O)CC3(C2)CC3)nc(CC)nc2c(C)csc12 C1(NC(c2c(CC)cccc2)=O)CC2CCC(C1)N2C(C1(Br)C(C)C1C)=O N1(C(C(C)CCO)=O)CCN(C(=O)Cc2csc(NC=O)n2)CC(O)C1 C1(C(=O)N(CCCCN(C(=O)Cc2c[nH]nc2O)C)C)(OC)CC(C)CC(C)C1 Cc1cn2c(C(=O)NCC3(NC(c4cc(O)nc(C)n4)=O)CC3)c(Cl)nc2s1 C(=O)(C(C)CCO)NCC(CN(C(c1cc(COC)on1)=O)CC)(C)C c1(C(=O)NCC(C)NC(C2COC3(C)CC2C3)=O)cccc(C(F)(F)F)c1O C1(CC(=O)NC(CN(C(c2ccoc2CC(N)=O)=O)CC)C)CCCS(=O)(=O)C1 C1(CCNC(C2CC(OC(F)F)C2)=O)CCN(C(=O)CSC2CCCCO2)C1 C1(C(=O)NCC(C)CNC(C2(C)CC2C(F)(F)F)=O)CS(=O)(=O)CC(=O)N1 C1(NC(c2ccc(C)c(O)c2)=O)CN(C(=O)C(O)C2CCC2)C2(CCOCC2)C1 S(=O)(=O)(c1c[nH]ccc1=NCC1CCOC1C)N(CCCSC)C N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCC(NC(=O)CC(C)N(C)C)C1(C)C C1(NC(C2(Oc3ccccc3F)CC2)=O)C2CN(C(c3ccccc3)=O)CC12 N1(C(CCSC)=O)CCC(NC(C2CN(C)CC(C)O2)=O)CC1C CC(C(=O)NNc1ccc(Br)nn1)c1c(F)cccc1Cl c1(-c2onc(CC(c3ccc(CC4CC4)cn3)=O)n2)ccc(OC(F)F)cc1Cl C1(C(c2cn(Cc3c(C(=O)O)cco3)nn2)O)CCN(C(C2(Br)CC2)=O)CC1 C1(NC(c2ccc(SC)cc2)=O)CN(Cc2cccnc2)CCC1(F)F N1(C(C(C)OCCOC)=O)CCC(C)(Cn2cc(COC(C)C)nn2)CC1 C1(O)(CCC(=O)NCC=CCNC(C2C(C)(C)C2N2CCC2)=O)CCCOC1 CN1CCN(C(=O)C(CNC(C2OC3CCC2C3)=O)N(C)C)CC1CO c1(C(=O)NC2C3CN(C(CC=C(C)C)=O)C2C3)cc(S(N)(=O)=O)c(Cl)cc1Cl c1(CNC(C2C(C)C2)=O)ccc(CNC(=O)C(C)CC2CCCC2)cc1 C#Cc1ccc(C(N2CCCC(NC(=O)C(C)N(C)C)C2C)=O)cc1 CCCCC(CNC(=O)C(C)CCOC)NC(c1onc(CC)c1C)=O C1(C(N(C2CCN(C(C(c3cn(CC)nc3)(F)F)=O)C2)C)=O)CCCS1(=O)=O N1(c2nnc(-c3c[nH]c(Br)c3)n2CCC2CCOC2)CCNCC1.CSC CCC(CC(F)F)C(=O)N1CC(CNC(c2cnoc2CC(C)C)=O)CC1(C)C N1(C(C(C)OCCOCC)=O)CC2(C1)CN(C(=O)C(C)OC1CC1)C2 c1(-c2c(NC(C(C)S)=O)c3c(nc2)cccc3)cccc2c([N+](=O)[O-])cccc12 C1(C(=O)NCC2N(C(C3(F)CC3)=O)CCC2)CC12CCOc1ccccc12 c1(OC)cc2ccc(Cc3ccc(C#N)cc3)cc2cc1OC c1(C(=O)Nc2ccc(-c3cnn[nH]3)cc2)ccc(O)cc1Cl c1(OC)cccc(COCC(=O)NC2CCN(C(=O)CCC(C)SC)C2C)c1 c1(CNC(=NC)NC2CCC(C(F)F)CC2)ccc(F)c(OC)c1F.C1(=O)CO1 c1(C(N2CC(OC)CC(NC(C(C=C)(C)C)=O)C2)=O)ccc2nn[nH]c2c1 N1(c2c(Br)cn(C(C)C)n2)C(=O)C2c3ccccc3OCCN2C1=O CC(C)(C)CS(=O)(=O)NCCc1c(Cl)cccc1Cl C1(C(=O)NC(C)CNC(=O)Cc2nnco2)CCCC12OCCO2 N1(CCNC(Cc2cc(C)no2)=O)CCN(C(C2CCCC23CC3)=O)CC1 c1(C(=O)NCC(CN(C(C)=O)C)O)n[nH]c2ccc(Cl)cc12 c1(CC)ccc(C(N2CCC(NC(c3cc(COC)no3)=O)C2(C)C)=O)cc1F N1(C(C2CC3(ON=C(C)C3)C2)=O)CCCCC2(C1)CN(C(=O)CSCCC#N)C2 NS(=O)(=O)c1cc(C(=O)NCCOC2CCN(C(C3CNC(=O)N3)=O)C2)c(Cl)o1 C1(C(=O)NC(C2(C(=O)OC3CC3)CC2)C)C(C(C23CCC(C2)C3)=O)C1(C)C CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(C2COCCO2)=O)C2CC12 c1(C(N2CC(C(C)NC(c3c(C(C)C)nns3)=O)C2)=O)cc2ccsc2[nH]1 Cc1ccc(C=CC(=O)NCC(C)CNC(=O)CC2CCCS(=O)(=O)C2)cn1 N1(C(c2cnc(C)nc2C)=O)CCCC2(NC(c3cnc(C)[nH]3)=O)CCCC12 Cc1ccc(N)cc1OCC(N1CCC1CNC(=O)C(c1ccc(Cl)s1)C)=O N1(C(C2(OC)CCC2)=O)C(C(=O)NC2CCC3CCC23)CCC12CC2 N(C1CCc2c(Cl)cccc21)C(c1c2ncc(C(N)=O)c(N)n2nc1)=O C1(C(=O)NCCC2CCN(C(C3CC(C(=O)OC)C3)=O)C2)CCC(C)(C)OC1 c1(N(CC(C)C(F)(F)F)C)ccc(S(=O)(=O)NC2CC2C2CCOCC2)c(Br)c1 C=CC1(C(=O)NCC2(OC)CN(C(=O)CC(C)(O)COC)C2)CCCCC1 c1(NC(C)=O)ccc(C(=O)NC(C)CNC(C2(C#N)CC(C)C2)=O)c(Cl)c1 C1(C2(NC(Cc3ncc(C)s3)=O)CC2)CCCCN1C(C1C2CCCC12)=O N1(S(CC(=O)OCC)(=O)=O)CCCC2(CCN(C(c3ccc(S)cc3)=O)C2)C1 c1(NCCCC(N)=O)nc(N2CCSCC2)nc2scnc12 C1(NC(CCC2(C)CC2)=O)CC2CCC1N2C(=O)Cc1ccc(OCC#N)cc1 C(=O)(CCCS(C)(=O)=O)NCC(c1ccccc1)CNC(CC(CC)SC)=O CC(C)C(C(=O)NC1CN(C(=O)C(C)C2CCC2)CC1C)NC(c1cccs1)=O N1(CC(C)(C)NC(CCCOCC)=O)CCN(C(c2ccc(F)cn2)=O)CC1 CCC(C)(C(=O)NC(C)CCCCNC(=O)CCc1ccc(O)nn1)OC N1(C(c2c(C)n(C)cn2)=O)CC2CN(C(C3CC3c3ccncc3)=O)CC2(C)C1 c1(C(=O)NCCSc2ccc(C)cc2)c[nH]c2ccccc2c1=N c1(OC)cc(Cl)c(C)cc1C(=O)COC(=O)C(F)(F)CC(C)C c1(CCNC(C2(OC)CCCCCC2)=O)c[nH]c2cc(C(C)C)ccc12 CC1CN(C(=O)CC(F)(F)F)CCN1C(C1CC(O)C(F)C1)=O N1(C(c2cc(C#N)sc2)=O)CCCC2(CCCN2C(c2ccc(Cl)nc2O)=O)C1 N1(C(Cc2cc(C)nn2C)=O)CC(C2CN(C(c3cc(F)c(F)cc3Cl)=O)C2)C1 Cc1cncc(OCC(N2CC(CN(C)C(c3ccn(C(C)(C)C)n3)=O)C2)=O)n1 CCCC(C)(C)C(=O)N1CCC(C)(NC(C2CCC23CCOCC3)=O)C1 CCCC(CCC)CCCC(=O)N1CC(CCNC(=O)CN(C2CCSC2)C)C1 C1(C(=O)OC)CC(=O)CN1C(c1c(O)n[nH]c1-c1ccccc1)=O c1(CCC(=O)NCC(CNC(C2=C(C)OCC2)=O)C)cccc(S(N)(=O)=O)c1 O=C(C1CCCc2nc[nH]c21)NCC1C2CC1N(C(=O)CCC1CCCCO1)C2 CCC(C(=O)OC)C(=O)NC(C)CNC(c1ncc(Br)cc1C(F)F)=O CN1CCc2c(NC(=O)NC3(c4ccncc4)CCC3)cccc2C1=O Cc1ncc(CCNC(=O)C(C2(O)CN(C(C3CC3[N+](=O)[O-])=O)C2)F)[nH]1 C1(CCC(=O)NCC(C2CCCC2)NC(C2(CC)CC2)=O)CCC(=O)N1 C(=O)(C1=CCCOC1)NC(C(C)C)CCN(C)C(c1cnc(C(F)(F)F)cn1)=O c1(N2CCCC(CNC(=O)CC3CCCS3(=O)=O)CC2)c(Br)cccc1[N+](=O)[O-] c1(NCc2cc(C)ns2)cc(NCC(Cl)=CCl)ncn1 c1(-c2cn(C3C(C)CN(C(C4(CCF)CC4)=O)C3)nn2)ccc(F)cc1Cl CC(C)CCN=C(NCc1ccc(Br)o1)NC(C1CCCO1)C C(=O)(C(C)(C)CC(=O)NC(C)CNC(c1ccccc1C(C)(C)C)=O)OCC CCC(C)CCCCC(=O)N1CCC(N(C(=O)CCSC)CCO)C1 CC1(C)C2CCC1(C)C2C(=O)NC1CN(C(c2cc(F)ccc2F)=O)CC1F c1(CC)cc(C(=O)NCC2CCC(C(=O)NCCC(C)(C)F)O2)n[nH]1 O(C=C(C#N)C(=O)N1CC(NC(c2cc(C3CC3)cnc2Cl)=O)C(C)(C)C1)CC C1(C(N2CCCC(c3ccccn3)C2)=O)COc2ccccc2C1 c1(SCC(=O)NCCN(C(=O)C(C)(C)C)CC)nc(C)nc2sc(C)c(C)c12 C1(C(=O)NC2(CN(C(=O)Cn3cccn3)C)CC2)CCC1C(C)(C)C C(C(COC)C(=O)NC1CC2(C1)CC2C(=O)NCC(C)(C)OCCO)OC C1(NC(=O)Nc2c(C)cccc2)CC(F)CN(C(C2CCCS2)=O)C1 c1(C(=O)NC2C(NC(C(C)NS(C)(=O)=O)=O)CCOC2)cn2c(n1)CCC2 C(C)(C(=O)NCCCN(C(=O)CNC(=O)Cn1cncn1)C)=CC Cc1ccc(C(=O)NCC2CN(C(c3cnnn3C(C)C)=O)CCO2)c(C)n1 C#Cc1ccc(C(N2CCC3CC23C(=O)NC(CC2CC2)C(=O)NC)=O)cc1 N1(C(CC(CCC)C)=O)CC2C3CCC(C(NC(c4sccc4C)=O)C3)C2C1 C#CCCCC(=O)N1CCCC1C(N1CC(NC(=O)C2CC2)C1)=O CC1CC(C(=O)NCC2CCN(C(=O)CCc3cn[nH]c3)CC2)Cc2nn[nH]c21 C1(C)(C(=O)NCCC(CC)(C)NC(C2COCCO2)=O)CCCN(C)C1 C1(OC)CCN(C(C2CSCCN2C(C2CCCC(=O)C2)=O)=O)CC1(C)C C1(NC(c2cc(C(F)F)cs2)=O)CCC12CCN(C(=O)C(F)CC1CCC1)CC2 c1(N(CCOCCNC(C)=O)C)nc(N2CCCC(F)C2)c2c(n1)CCC2 c1(OC)cccc(CN2CC3CC(C2)N3C(=O)C2=CCC2)c1Oc1ccccn1 CCC(CC(F)F)C(=O)NCC1(NC(c2ccn(C(C)(C)C)n2)=O)CCOC1 C1(C(N(CCCNC(=O)Cc2cncc(C)c2)CC)=O)CC(C)CC(C)C1 C1(C(N2C(CNC(COCCCCC)=O)CC2)=O)CCCC(F)(F)C1 C1(NC(CC)=O)CC(C2CCN(C(=O)CN(C3CCSC3)C)C2)C1 CC1C(C)N(C(c2cccc(C#N)c2Br)=O)CCN1Cc1ccccc1 c1(CNC(CNC(=O)OC)=O)nc(OC(=O)C(F)C(F)(F)F)cc(O)n1 n1(C(c2nc(CC(C)C)on2)C)cc(Br)cn1 C1(CNC(c2[nH]cc3c2CCC3)=O)CN(C(=O)C(F)(F)CO)CCC1(F)F C1(CNC(N(C)CC2CC2C)=O)C=CCC1 O=C1CCC(CC(=O)NC2CN(C(C3CCS(=O)(=O)N3)=O)C2)CN1 C(=O)(C(O)CCC(C)C)NCC(CC(N1CC(CC)C(F)C1)=O)C1CCC1 C1(OCCC)CCCCC1Cc1nc(-c2cc(C)oc2C)nn1CCC(C)(C)C Cn1cc(-c2nnc(C3CC3F)o2)c(Oc2ccccc2)n1 c1(C(=O)NC2C(NC(Cc3ccc(C)c(Cl)c3)=O)C2)cccc(S(N)(=O)=O)c1C CCCCC(C)(N=c1ccn(C2CC2)[nH]1)c1nnnn1C1CCC1 C1(C(N(C2CCN(C(C3(SC)CCC3)=O)CC2)CC#C)=O)CCC(=O)NC1 Cc1n[nH]c(=NC2=CCCC2)o1.N1(C(C(=O)N2CCC2)C)CCCC(O)C1 C1(NC(=O)NC(C)C(=O)NCc2ccco2)CCNC(=O)C1 c1(C(N(C(CN(C(C(CC=C)N(C)C)=O)C)C)C)=O)cccc2[nH]ccc12 c1(C(N2C(C)CC(NC(c3c(C)c(N)n(C)n3)=O)C2)=O)ccc2cncn2c1C c1(C(=O)NCC2CC(F)CN2C(c2cc(Br)n[nH]2)=O)csc2ccncc12 C1(C(=O)NCCC(C)(C)NC(c2cc(C(C)(C)C)ccn2)=O)CCC2C1C2(F)F C1(CN(CC(=O)NCCC)C)CCN(C(=O)C(CC)SC)CC1 C1(OC)C(NC(C2(CNC(=O)Cn3cncn3)CC=CC2)=O)CC12CCC2 N1(C(CCCOCC)=O)CC2(CCCCN(C(C3(Cl)CC3(F)F)=O)C2)C1 CC(C)(C(=O)N1CCC(NC(c2cnn(C(C)(C)C)c2)=O)C(CO)C1)S(C)(=O)=O C1(NC(C(CC)NC(N)=O)=O)CCC2CCN(C(C3(CO)CCC3)=O)C1C2 C1(C(N(CC)Cc2cnc(Br)cn2)=O)CN(C(=O)OC(C)(C)C)CCS1(=O)=O CC1(C)CC(=O)NC1CNC(C1CCC(CNC(=O)C(Cl)Cl)O1)=O CC1CCCC(CNC(=O)C(=O)NCc2ccsc2)CC1 C1(CN(C(=O)Cc2ccccc2C(F)(F)F)C)CCCCN1C(=O)CC1(C)CC1 C1(NC(CC2N(C(c3c(C)n(C)cn3)=O)CCCC2)=O)CC1C1CCCC1 C1(CC)(CO)CCN(CCC(=O)Nc2cnn(C3CCCCC3)c2C)C1 N1(C(COCCC=C)=O)CCCC(CCC)(NC(c2cccn2C)=O)C1 n1(CC)c(N2CCC(c3ccon3)CC2)nnc1C1CCC1c1ccsc1 C1(NC(C(=O)NCC(c2ccncc2)C)=O)CCCN(Cc2cccc(F)c2)C1 Cc1sc(C)c(C(=O)NCC2(NC(C34CC(F)C3C4)=O)CCOC2)c1C#N C(=O)(C(F)(F)c1cscc1Br)N(C1CN(C(C2(C)CC2(C)C)=O)C1)C C=CC(F)(F)C(=O)NCCCC(C)NC(C1CSCN1C(C)=O)=O Cn1cncc1C(=O)NC1CC(NC(=O)CC2C(C(F)(F)F)C2(F)F)C1 N1(C(C(C)=C(CC)C)=O)CC(OCC)C(NC(=O)CNC(=O)C(C)(C)C)C1 Cc1ccc(C(N2CC3CC3(NC(C3(C4CCCO4)CC3)=O)C2)=O)cc1Cl c1(C(C)=O)ccc(Cl)cc1S(=O)(=O)Nc1cc(C)nc(N2CCOCC2)n1 C(CN=c1cc(C)c(S(=O)(=O)N2CCN(c3ccncn3)CC2)c[nH]1)SC C1(C)(NC(C(CCN(C)C)NC(COCCOCC)=O)=O)CN2CCC1CC2 c1(OCC(C)(C)NC(C(CC)N(C)C)=O)cccc(C)c1.C1(=O)COC(C)N1C c12ccc3c(c1)n(CC(F)(F)F)c(=O)n3C2.CCCCC(C(=O)O)OC c1(C(=O)OCC)ccc(CNC(=O)CC2(C)CCN2C(c2ccsc2C)=O)cc1 N1(C(c2c(C)nc(COC)s2)=O)CCN(C(=O)CC(C)SC)CC1CO N1(C(CSC)=O)CCN(C(C2CCCN(C(C)(C)C)C2=O)=O)CC1C(C)C C1(C)(C(N(C)CC2CC(O)C2)=O)COCCO1.c12cn(nn1)C1CN(C1)C2=O N1(C(C2(C=C)CCN(C(=O)Cn3cccc3)C2)=O)CCCC(C)(C)CC1 C(C(=O)C(=O)NC(COCC)C1CC1)(c1ccco1)NC(=O)OC.C1(=O)C(C)N1 c1(C(=O)NCC(CCCC)NC(=O)C(C(C)C)NC=O)nc(C)c(C)nc1C C1(CCC)CN(C(=O)CCC(=O)NC)CC1NC(=O)COCc1nc(C)no1 CC1CCC(NC(c2cccc(C3CC3)n2)=O)CN1C(C1COC2(CCC2)C1)=O Cc1c(C(N2CCCCCC2c2ccc(Cl)cc2)=O)oc2ccc(F)cc12 C#CCCCCC(=O)NC1(CNC(c2c[nH]nc2CC)=O)CC2CCC1C2 c1(SC(C(=O)NC(CNC(CCCc2onc(C)n2)=O)C)C)ccc(F)cc1 c1(C(N2C(C)CC(CNC(c3cccc(OC)n3)=O)C2)=O)ncc(Cl)cc1Cl C#CC1CCC(C(=O)N(C2CN(C(C3OCCC3C)=O)CC2(C)C)C)CC1 N1(C(c2c(C)[nH]nc2Cl)=O)CC(NC(=O)C(C)NC(c2cccs2)=O)C(C)(C)C1 c1(OC)nccc(Sc2noc(C34CC3CN(C(=O)C(C)CC(N)=O)C4)n2)c1F c1(C(C)C)ccc(C(=O)NCC2CN(C(=O)C(C)OCCN(C)C)CCO2)cc1 C1(CC)(CC)CN(Cc2ccccc2)CCS1(=O)=O.c1(C)nccn1C(F)F C1(CNC(c2c(OC)nsc2)=O)N(C(C2CC2C(C)(C)C)=O)CCCC1(C)C C=CCC(CC(C)C)C(=O)N1CCN(C(=O)COCC=C)CC1C1CCC1 c1(CNC(c2n(C)ccc2)=O)nc(CNC(C2C(C3CC3)C2(F)F)=O)cc(O)n1 Cc1cc(C)c(COC(C2Cc3ccccc3C2)=O)c(C)c1O N1(C(=O)CCC2CCOC2)CC2(CCCCN2C(=O)COC2CCCOC2)C1 Cc1cc(CN(C=O)Cc2ccc(O)c(Br)c2)ccc1N(C)C Cc1ccc(C)c(CC(=O)NC(C2CCCCN2C(=O)C(C)OCC2CC2)C)c1 N1(C(c2ncc(OC)cn2)=O)CCc2sc(CNC(C3CC3C(C)C)=O)nc2C1 c1(C(=O)OC(CC(=O)N(CCN(CC(=O)OC)C)C2CC2)=O)cccn2nncc12 c1(CCC(N2CC(O)(C(C)NC(C3CCCOC3)=O)C2)=O)cccc(N(C)C)n1 c1(C(=O)NCC2(OC)CCN(C(c3cncs3)=O)C2)cc2c(F)cc(F)cc2[nH]1 C=CC(C)(CC)C(=O)NCc1cn(C2CN(C(=O)CSCC(N)=O)C2)nn1 N1(C(CNC(=O)OCC=C)=O)CCC(NC(C2CCCCN2N=O)=O)C(C)C1 c1(C(N(CCOCCNC(C2(COC)CC2(F)F)=O)C)=O)cc(Cl)ccc1OC c1(C(=O)OC)ccc(C)nc1NC1CCN(C(c2cc(C)cs2)=O)C1C CC1CCCCN1S(=O)(=O)N1CCN(C(c2cc3c(Br)c(Cl)ccc3[nH]2)=O)CC1 N1(C(CN(CCC#C)C)=O)CC(NC(C2CCC2C(=O)OCC)=O)CC(C)C1 C#Cc1cccc(C(=O)NCC2CCN2C(=O)Cc2cc(F)ccc2C)c1Cl c1(CNC(C(C)(C2CC2)OC)=O)ccccc1CN(C)C(c1c(C)cnn1C)=O Cc1cnncc1C(=O)NOCC(N1CCOCC1c1ccccc1OC1CC1)=O c1(C(N2C(C)CCN(C(=O)C(F)OC(F)(F)F)CC2)=O)c[nH]c2cc(F)ccc12 Cc1nc2ccccn2c1CC(=O)NCCN(C(=O)C(C)C(C)(F)F)C N1(C(C(C(=O)OC)C)=O)CCC2CCN(C(=O)C(=O)NC(C)C)CC12 c1(C(=O)NC2C(NC(CC(C=C)(C)O)=O)C2)cccc2c1COCC2 c1(CC)cc(C(=O)NC2CC2CNC(c2cc(Br)n[nH]2)=O)c(C)o1 Cc1ccc(-c2nc(C)sc2CC(=O)N(C(C)(C)C)CCOCCO)cc1 c1(C(=O)NCCCC2N(C(C3CC(OC)C3)=O)CCCC2)cc(Cl)c(F)c(Cl)c1 CC1CN(S(=O)(=O)N2CCC(NC(N)=O)CC2)CCO1 C12(C(N(C)CCC3CCN(C(C4(N=[N+]=[N-])CC4)=O)CC3)=O)CCCC(CO1)C2 C1(C2CCC2)(CNC(=O)C=CC2CCOC2)CCN(C(=O)COCCCF)CC1 C12(CN(C(C(c3ccc(N(C)C)cc3)C)=O)CCO)CCCC1OCC2 Cc1nn(CC(N2CC(C)CCC2CNC(=O)CC(C)C)=O)c(C)c1Cl C1(CC(=O)NCC(=O)N(C)C)CCN(S(=O)(=O)CCc2ccno2)CC1 N1(C(Cc2ncc(C)nc2)=O)CCC2CCCC12CNC(=O)C(C)(C)CC#N C1(C(=O)NCCCCCNC(c2cn(CC)nc2C)=O)CCc2[nH]nc(O)c2C1 c1(OC)ccc(CC(=O)NCCn2cc(CCC#N)nn2)cc1O c1(C(=O)NC2CC3(C(C(=O)NC(C(=O)OCC)C)C3)C2)cnc(C)nc1C C1(CN(C(=O)CC2COCC2(C)C)C)C2CN(C(C3CC(F)(F)CS3)=O)CC12 N1(CC)CCC(CCNC(=O)CC2CC(C)=NO2)CC1.C12C=CC(C1)CNC2=O c1(C(=O)NCC2C(C(=O)OC)CCC2)ccc(-c2ncco2)cc1F c1(C(=O)NC(CC)CNC(=O)CCC2CCC(=O)N2)cncc2[nH]ccc12 C(=O)(CCS(C)(=O)=O)NC(C)C(C)NC(=O)C(F)(F)c1ccsc1Cl C(=O)(C(CC(=O)O)n1cc(-c2cn(CC(=O)O)nc2)nn1)NN1CCOC(CO)C1 C1(C(N2CCC(NC(c3cc(C)on3)=O)C(O)C2)=O)CC(O)c2ccccc2O1 c1(NC(C23CC(C(N(CC(C)C)CCC)=O)(C2)C3)=O)c(Cl)c(F)nc(F)c1Cl c1(NC(c2nc(-c3c(C)ccc(OC)c3)sc2C)=O)ccc2scnc2c1 n1(CC(=O)NC2(C)CC(NC(C(C)(C)OC)=O)C2)c(O)nc2ccccc12 C1(C(=O)NCC2CCCN(C)C2)CCN(C(=O)Cc2ccccn2)C12CC2 Cc1nc(Cl)ccc1CC(N1CCN(C(=O)CC2CCCOCC2)C(CO)C1)=O O(NC(=O)C(CC(N)=O)NC(=O)CCCOC)CCOCC#C Cc1cc(C(N2CC(O)(C(F)C(=O)NCC(CC3CC3)CO)C2)=O)ccc1F C1(CC(C)CNC(=O)C#CC2CC2)CCN(C(=O)Cc2ccon2)CC1 c1(NC(=O)CC2CCCN(C(=O)CC3CCOC3=O)C2)cccc(F)c1F CCC(C(=O)NC1CC(CCNC(=O)CCc2cncn2C)C1)OC C12(NC(c3c(Cl)cncc3Cl)=O)CCCC1N(C(=O)CC1CC1)CCC2 c1(C(N2CC(COC)N(C(=O)C=Cc3cccs3)CC2)=O)cc(C)c(Cl)c(C)c1 C1(C(=O)NC2CC(=C)CN2c2cc(O)nc(C)n2)CCc2nc[nH]c2C1 c1(N2CC3(C(NC(C4CC45CC5)=O)CCS3)C2)c(Cl)cncc1[N+](=O)[O-] CC1CN(C(c2cc(Cl)no2)=O)CCCN1C(=O)CCCCC1CC1 N1(C(C2C(C(C)C)N(C(c3cnc(S)nc3)=O)CC2)=O)CC(O)CC1(C)C C(=O)(C(=O)C(F)(F)F)NCCC1CCN(C(C(C)CC2CCC2)=O)CC1 c1(C(=O)NCC2(O)CCN(C(c3c(C)nn[nH]3)=O)CC2)cc(S(N)(=O)=O)oc1C c1(C(=O)NCCN(C(=O)Cn2cnnc2O)CC)cnn(CCC(F)(F)F)c1 C1(C(=O)NC(COC)CNC(C2CC(OC)C(OC)C2)=O)CCn2c(O)nnc2C1 C1(NC(C2C(C)CCC2)=O)CCCC2CN(C(c3cccc(C4CC4)c3)=O)CC12 C12(C(=O)NC3CCN(C(C(c4ccc(F)cc4)CC)=O)C3)CCC(C1)OC2 c1(NC(C(C)(C2CCC2)NC(N)=O)=O)ccc2cccnc2c1 N1(C(c2ccc(OC)c(F)c2)=O)CC(NC(=O)CCC(C)N(C)C)C(C2CC2)C1 C1(C(N2CCC(CNC(c3csc4ccccc34)=O)C2)=O)COCC2(CCC2)O1 C#CC1(O)CCN(C(=O)CC2CC2CNC(=O)C(COC)CC)C1 c1(C(=O)OC)ccc(NCCCNC(=O)CC2CC3(CCC3)CO2)c([N+](=O)[O-])c1 c1(C(N2CC(OC)C(CNC(C3(C#N)CC(C)C3)=O)C2)=O)ccc(F)c(C)c1C N1(C(c2n(C)c(Cl)nc2)=O)CC(F)(F)CC1C(=O)NC1(C)C(C)(C)C1(C)C c1(C(=O)NCC(C)(C2CCC2)NC(=O)CCS(C)(=O)=O)cccc2[nH]nc(O)c12 c1(C(N2CC(NC(CC(n3c(C)ncc3)C)=O)C(C)C2)=O)cc(Cl)ccc1F CC(C)CCCC(C)NC(c1cc(CCNC(c2cnncc2O)=O)on1)=O c1(N(C2CNCC(F)C2)C(c2scnc2C(F)(F)F)=O)ncc(Cl)cn1 O=C1NCC2(CCN(C(=O)CC3(NC(C4CC(O)C4)=O)CCCCC3)C2)O1 N1(CCOCC)CCC(N=c2[nH]c(=N)[nH]c(=NCCCn3cccn3)[nH]2)CC1 N1(C(C(C)OCC)=O)CCCC(N(C)CC2CCOC(C)C2)C1 C1(CNC(C2=CCC(C)CC2)=O)CN(C(=O)C=Cc2cc[nH]n2)C2COCC2O1 N#Cc1cn(CC(N2CCCC23CCN(C(=O)C2=CCCC2)C3)=O)c(=O)nc1O c1(C(N2CCC(C(=O)NC)C2)C(=O)NC2(C)CC2)cc(Cl)ccc1C C(=O)(C(C)C(F)(F)C(F)F)N1CCC(CCNC(C2(CC#C)CCOCC2)=O)C1 C1(NC(c2c(CC)nns2)=O)CCN(C(C2(N=[N+]=[N-])CC2)=O)CC1CC N1(C(CCOC)=O)CC(C)CCC1C(=O)N(C)CCc1cnn(C)c1 c1(CNC(COCC(=C)C)=O)cn(C2CN(C(=O)CCc3ccncc3)C2)nn1 c1(COC)nc(C(=O)NC2(C)CC(NC(c3snnc3CC3CC3)=O)C2)cs1 C(c1ccc(NC(=O)C(=O)NC2C3CCC(O3)C2N)cc1)=CC(=O)OC(C)(C)C c1(C(=O)N(C)C)ncc(F)cc1N.CC1C(N(C)C)C(=O)N2CCC2C(=O)N1 C(=O)(CS(=O)(=O)CC)N1CCC(N(CC#C)C(C2C3CN(C)CC23)=O)C1 N1(C(Cc2cnc(C)[nH]2)=O)CCCC(C)C1CNC(=O)CCc1ccn(C)n1 C1(NC(c2n(CC)ccn2)=O)C(CNC(=O)C(C)=CC2CC2)CCC12CCC2 c1(OC)sc(C(=O)NCC2CC2CNC(c2ccnc(C)c2)=O)cc1Br N1(C(CS(CC)=O)=O)CCCCC(NC(c2cncc(C(N)=O)c2)=O)C1 c1(C(=O)NCc2c(C)cccc2)csc2c1CCN(C(=O)C(C)(C)F)C2 C1(NC(c2nc[nH]c3nccc2-3)=O)CCCCCN(C(=O)CC(F)(F)Cl)C1 c1(C(=O)NCC(C)CNC(=O)COCc2nc[nH]n2)ccc(F)c(N)c1 c1(CNC(CC2(OC)CCC2)=O)ncccc1CNC(c1cnccc1C)=O N1(c2nc(=NC)[nH]c(=NCc3ncc(C)cn3)[nH]2)CCOc2ccc(Br)cc2C1 N1(C(=O)COCCO)CCOC2(CCCN(C(C3CCC=CO3)=O)C2)C1 Cc1cc(=NC(=O)C2CCN(C(c3cc(Br)cc(I)c3)=O)CC2O)[nH]c(Cl)n1 Cc1ncc(CC(=O)NCC2(C(=O)NCC3CCCN3C)CC2)s1 C(=O)(CCC1=CCCCC1)NC1CC2(CC(C(=O)NCC(COC)(O)CO)C2)C1 C(CCCCC(=O)NCC1CC(NC(c2ncc(Cl)cc2F)=O)CC1O)SC S(=O)(=O)(c1ccc(C#N)cc1Cl)N1CC2N(S(CC(=O)OC)(=O)=O)C(COC2)C1 c1(-c2n(C(COCC)C)nc(C(C)O)n2)cc(C)c(Br)cn1 CC1C(C)N(CC(F)F)CCN1C(c1cc(Cl)nc(Cl)c1)C(=O)NC1CCOC1 C1(N(C)C(c2cc(=O)cc(Cl)[nH]2)=O)CN(C(=O)COC2CCCCC2)CC12CC2 C1(CNC(CCOC)=O)COCCN1C(c1nccc(SC)n1)=O N1(C(CC2CC(C)C(C)CC2)=O)CCCC2(CCN(C(=O)CSC(F)F)CC2)C1 c1(OC)ccc(O)cc1C(N1CC(O)(C(C)NC(c2csc(Cl)c2Cl)=O)C1)=O c1(CN(C(C2CCOCC2)C)C)ccc([N+](=O)[O-])c2cccnc12 CCC(CN(C)C)CC(=O)NCC1C2CN(C(c3ccnc(Cl)c3OC)=O)CC12 C(C(C(=O)NCCCc1ncco1)NC(=O)Cn1ccnn1)SCC C1(C(=O)NC2(CC=C)CCN(c3nnc(C(N)=O)s3)C2)CCC(C)(C)CC1 N1(C(c2cc(C)n(C)n2)=O)CC2CN(C(C3CCN(CC(C)C)CC3)=O)CCC12 CC(C(=O)NCC1CC2CCC1N2C(c1cc(Cl)ccc1F)=O)C(C)(F)F C(=O)(C(C(C)O)NC1CCN(C(C)Cc2ccccc2)C1)OC C1(N=[N+]=[N-])(C(=O)NCc2nccc(C)c2F)CCN(C(=O)CC2CCC(=O)C2)C1 c1(C(N2CCC(C)(CCNC(c3ccc(C)cc3)=O)C2)=O)ccc(F)cc1C c1(C(N(CCC(C)NC(c2c(C)cccn2)=O)C)=O)ccc(C#N)cc1O C1(OC)COCC1n1cc(C(N2CCCC2CNC(c2cscc2Cl)=O)=O)nn1 c1(C(N2C(C)CC(NC(c3cc(F)c(F)c(F)c3)=O)C2)=O)cc(Cl)cc(F)c1N Cc1cc2c(C(N3CCCC(CO)(NC(c4cnns4)=O)C3)=O)ccc(C)c2[nH]1 C1(C(N2CC(c3ccccc3)(NC(CC3(C=C)CC3)=O)C2)=O)COC2(CCC2)C1 c1(C(c2nnnn2C2CC2)NCC2(CCF)CCC2)ccc2ncsc2c1 c1(SC)nocc1CCNC1CC1.C1C(=O)N1CCO C1(C(=O)NCCCCNC(c2ncc(Br)cn2)=O)CCCC(F)(F)C1 N1(C(=O)OC(C)(C)C)CCC(O)C(C)(C(=O)Nc2cc(Br)ccc2C(C)(C)C)C1 C1(CC(=O)NC2(CNC(c3cnn(C)c3N)=O)CCC2)CCC(C)(C)CO1 c1(C(CC)C)ccc(C#N)c(N2CCCN(C(c3c(Cl)csc3Cl)=O)CC2)n1 c1(CNC2(CO)CC2)ccccc1C(C)(C)N(C(C1C(C(=O)OC)C1)=O)C1CC1 N1(C(C2(OC)CC2)=O)CCC(C(F)(F)F)C(NC(=O)C=CC2CCC2)C1 CS(=O)CCC(O)C(=O)NC1CCN(C(=O)Cn2nnc3ccccc23)CC1 N1(C(c2c(C)ccs2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C2(CCC2)C1 CS(=O)(=O)c1cccc(Cl)c1NCC1=CCN(C(=O)NC2CC2)CC1.c1(SC)ccccc1 CC1(CCNCc2ccc(-c3cccc(Cl)c3)cc2)CCNC1=O C1(C)(C(N2CC(CC)C(CNC(c3cc(C)ns3)=O)CC2)=O)CC(C)OC(C)C1 C1(NC(C(N2CC(C)C2)C)=O)CC=CCC1C(=O)NCC1(CO)CCCO1 N1(C(C(C(C)O)N(C)C)=O)CCN(C(=O)C=Cc2cccc(F)c2)CC(CO)C1 c1(C(C(=O)NCCC(CNC(c2c[nH]nc2C(C)C)=O)OC)C)c(C)n[nH]c1C c1(C(=O)NC2CCSCC2)cccc(CN(C)C)c1.CC1C=CC(=O)N1 Cc1nc(CC(=O)N(CC(O)CN(C(=O)CN(c2ccccc2)C)C)C)cs1 c1(CC(=O)OCC)cc(Br)c2c(c1)CCO2.c12ccsc1COC(=O)C2 C(=O)(C(F)(F)C(C)O)NC1CN(C(C(CC=C)OC)=O)CC1F O=C(C(O)C(F)(F)F)NCc1cccc(-c2cn[nH]c2)c1 N1(C(C(C2CCOC2)NC(CC=CCC)=O)=O)CCCC(CCC)CC1 Cc1noc2ccc(NC(C3CC(Nc4ncnc5cc(I)sc45)C3)=O)cc12 C1(OC)CCCC1C(=O)NCC(C)N(C)C(C1CC(C)(C)C1)=O c1(CN(C(C(=O)NC(C2(C)OCCO2)C)=O)C)nc(Br)cs1 C1(C(=O)NCC2CCC(NC(C(C)OCCN(C)C)=O)C2)COC2COCC12 CC1CCN(C(C(=O)NCc2ccccc2)C2CC2(Br)Br)Cc2ccc(O)cc21 C(=O)(CCS(=O)(=O)NC)N(CCCCN(C(CCCN(CCC)CCC)=O)C)C CCC(C)C(O)C(=O)N1CC(C)(NC(c2cccc(C(F)(F)F)c2O)=O)C1 c1(NC(C2(CNC(c3cccnc3CO)=O)CC2)=O)cc(F)c(Cl)cc1F Cc1nc(N2CCCC(C(=O)N(C(C)C)Cc3cccc(Cl)c3)C2)nc(O)c1C Cc1nc2c([nH]1)CC(NCc1c[nH]nc1-c1ccccc1Br)CC2 Cc1c[nH]c(C(=O)NCC2(C(=O)NC3CC(CC(N)=O)C3)CCCO2)c1C c1(CNC(C2CC3(C2)CN(Cc2cccnc2)C3)=O)cc(Br)cc(Cl)c1F C(C)(C(CC(=O)NCC1CCOC1C)NC(C1CCC1C(C)(C)C)=O)OC N1(C(COC(CC)(C)C)=O)CC(N(C(=O)CN2CCC(O)CC2)C)C(O)C1 C(=O)(CCC(N)=O)NCC1(NC(c2n(C(CC)C)ncc2)=O)CCOC1 N1(C(C)C)CCC(C(N2CC(N3CCN(c4ccc(F)cn4)CC3)C2)=O)C(C)C1 c1(C(=O)OC)ccc2c(c1)C(NC(=O)NC(C)C(=O)N(C)C1CC1)CC2 N1(C(CCC(C)(C)C)=O)CC2(CNC(=O)CC3CC=CCC3)CC(F)(C1)C2 C1(CN(C(=O)C(N2CCCC(F)CC2)=O)C2CC2)CCC2(CCCCCC2)O1 N1(C(CC2(NC(CCC)=O)CC2)=O)CCC(CCCO)C1.C1C(=O)N1 CS(=O)c1ccc(CC(=O)NCC(=O)NC2CC2)cc1.c1ccc(N)c(Cl)c1O C=C(F)C1(CC(N2CCN(CC(=O)NCc3n[nH]cc3C)CC2)=O)CCC1 C(=O)(C(F)(F)C(C)(C)O)NCC12OCC(NC(C(CC)NC(N)=O)=O)(C1)C2 c1(OCCC(=O)NCCCCNC(c2ccc(C)cn2)=O)ccccc1[N+](=O)[O-] N1(C(c2c(CNC(C(C(C)C)C3CCC3)=O)cc[nH]2)=O)CC(CO)CC1(C)C c1(CC(=O)N(CC(CNC(C(CC)C)=O)(C)C)C)c[nH]c2cc(F)ccc12 c1(COC(CN(C(C)=O)C)=O)ccc(O)cc1.C12CC(CO1)NC2=O C1(C)(C(=O)NCC(n2cc(C3(C)CCCC3)nn2)C)CCCS1 N1(C(=O)C=CC2CCCCCC2)CC2CCN(C(C3C=CCCC3)=O)C2C1 Cc1cc(C(=O)NC2(C(=O)N(C3CCN(C4CC4)C3)C)CC(F)C2)sc1C c1(CCc2c(C)c(N3CCC(C4CCCC4)C3)ncn2)ccc2oc(=O)n(C)c2c1 c1(C(=O)NCCCOCCCNC(C(C(C)(C)O)F)=O)cn2cccnc2n1 Cc1cc(C(=O)NCC(C)CC(=O)NC2CC(n3cccn3)C2)nc(O)c1 n1(CCC(=O)NCCN(C(=O)CC2CCC3CC23)C)cc([N+](=O)[O-])cn1 N(C(=NCCC(C)C)NCc1cn(C2CCOC2)nn1)CC1CCC(=C)CC1 c1(C(=O)NCCC2CC(OC)CN2C(c2ccc(C)s2)=O)cc(C)c(C)c(F)c1 C=CCCCCCC(=O)N1CCN(C(=O)C(C)(CC)OC)CC(CO)C1 N1(Cc2cn(CC(=O)NC3(C(N(CCC)CC)=O)CC3)nn2)CC2CCC1C2 N1(C(C(c2cccc(C)c2)O)=O)C2CCC1CC(O)(CNC(=O)CCF)C2 c1(OCC(=O)N(C)C)ccccc1NC(CNC(c1snnc1C1CC1)=O)CO C1(C)(NC(C(C)Oc2ccc(O)cc2)=O)CCCN(C(=O)CCP(C)(C)=O)C1 C1(NC(C=Cc2scc(C)n2)=O)CCCC(NC(c2cn3c(n2)CCC3)=O)CC1 CC1=C(C)CC(C)(NC(=O)CNC(c2ccc(C#N)n2C)=O)CC1 C(=O)(CC(C)C(C)(C)C)N1CCC(C=C)(C(=O)NCC(c2cnc[nH]2)C)C1 C1(C2CCN(C(=O)Cc3cc[nH]c3)C2)(NC(c2cc(CCC)c(C)s2)=O)CC1 N(C(=NC)N1CCC(n2cc(C)cn2)C1)Cc1nc(C(=O)OCC)nn1C C1(COCC)CN(c2ncncc2OC2(C(=O)NC)CCCC2)CC(C)(C)O1 CC(CC(=O)NC(C1CCN(C(=O)CC2CC2C)C1)C)CC(C)(C)C Cc1cc(F)sc1C(=O)NC(C)CNC(C1CC12CCC2)=O CC(C)C(O)C(=O)N(CC(C)CNC(=O)Cc1ccc(SC2CC2)cc1)C c12cccc(c1)NC2=O.C1(SCCC(=O)OCC)CCCCC1 N1(C(C2C(C)C2C)=O)CCCC1CN(C(=O)CO)C1CC1 C1(c2ccc(C)cc2)NC(=O)N(CCCNC(c2nnnn2C)=O)C1=O c1(C(N2CCN(C(C=CC=CC)=O)CC(O)C2)=O)ccnc2c1ccn2C c1(C(N2CC(=C(CNC(C3C(OC)CCC3)=O)F)C2)=O)ccc(C(C)C)cc1 C12(C(=O)NCC(CO)NC(c3cccc(OC)c3)=O)CC=CCN1CCC2 CC1CCN(C(c2ccc3n[nH]cc3c2)=O)C(C)C1NC(C1CCC(C)O1)=O C1(C(=O)NC(CSC)(C)C)C2CN(C(c3cc(Cl)n[nH]3)=O)CC12 c1(C(N2CCC(OC)(CNC(=O)C(O)C(C)C)C2)=O)cc(C)nc(CC(C)C)n1 C1(OC)(COC)CCCC(C)C1.c12cncc(n1)C(=O)N1CCC1c1cn-2nn1 C=C(C)C(CC(=O)NCCOC1CCN(C(=O)CS(N)(=O)=O)C1)OCC CN(CCCC(=O)NCC1CC1NC(=O)Cc1cc2ccccc2o1)N=O C1(CC=C)(C(=O)Nc2ccc(SC)nc2)CCCN(C(=O)C(O)C=CCC)C1 CC(F)(F)C(F)C(=O)N1CC=CCC1C(=O)NCC1Cc2nccn2C1 N1(C(C2CC(F)CN2C(c2cc(F)c(F)c(Cl)c2)=O)=O)Cc2ccc(F)cc2C1 C1(CC(=O)NCC(CC)NC(c2ccc(OC)c(C)c2)=O)CCCC2(CCC2)O1 c1(C(=O)NC23C(CN(C(CC(C)F)=O)C2)C3)cc(N)c(Cl)cn1 N1(C(C2(CC)CCC2)=O)CC(NC(c2cc(N)ccc2Cl)=O)C2(CC2)C1 N1(C(CN(C(C(C)C)=O)C)=O)CCC(C)(CCCC2(C(=O)O)CCCO2)C1 C1(NC(C2(C(C)C)CCCC2)=O)CCN(C(c2cnoc2C2CC2)=O)CC(O)C1 CC(CCN=c1ccc(Br)c(S(=O)(=O)NCCC2=CCN(C)CC2)[nH]1)N(C)C O=C(C1=C2CCN=C2NC=C1)NCC(C1CCCCC1)NC(=O)CSc1cccs1 C1(C)(C(=O)NC2(C(C)NC(C3CCC3C(F)F)=O)CC2)CCCC1O N(C(=NCC(C)(C)CC1(C)OCCO1)NCC1CC1)C(c1ccc(Cl)c(F)c1)C N1(C(c2cc(C)[nH]c2)=O)CCCC(C(=O)NCCc2cc(C)[nH]n2)CC1 C(=O)(C1=CCCN(C(=O)CC2C=NN(C)C2=O)C1)NCC(C#C)C(C)C C1(C(=O)NC(C)CNC(c2cccc3c2OCCO3)=O)Cc2c(F)cccc2O1 C1(c2cn(CC(F)(F)CO)nn2)(NC(C2CCC(F)C2)=O)CCCCC1 N1(C(C(CC)Sc2nc(C)cs2)=O)CCC(C2CN(C(=O)CCSCC)C2)CC1 Cc1c(C(F)(F)F)cc(NC(N2CCN(CCC(=O)O)CC2)=O)cc1O C1(NC(c2c(C)cc[nH]2)=O)CCCN(C(c2cc(C3CC3)on2)=O)CC1F Cc1cc(CNC(C)(CCCl)c2nnnn2-c2ccc(F)cc2)cnc1C c1(C(=O)NC2C(CNC(CCC(C)OC)=O)CC2)sc(C#N)cc1Cl N1(C(CC(C=C)C)=O)CCCC(CO)(CNC(c2ccc(OCCO)cc2)=O)C1 c1(N2CC3N(C)C(CCC3)CC2)nc(=NCC23CCC(CO2)C3)[nH]c2ccsc12 c1(C(N(CC(C)NC(C2COC(=O)N2)=O)C)=O)cnn(C2CC2)c1Cl C1(C(CNC(COCC(=C)C)=O)(C)C)CCN(C(C2CCCC2OCC)=O)CC1 c1(C(=O)OCC)c(NC2CC(C)N(C(=O)CC(C)(C)OC)C2)cc(C)nc1O CCCCC(=O)C(=O)N(CCCN(C(=O)C(C)c1cc[nH]n1)C)C N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)C(C)(O)C3CC3)C(C2)C1 c1(SCC(N2CCCC(CNC(C3(CC=C)CC3)=O)C2)=O)ccsc1[N+](=O)[O-] N1(C(c2cc(C)oc2C)=O)CC2CCC1C(CNC(C1CC1F)=O)C2 C12(C(N(c3cccn3C)CCNC(C)=O)=O)CC3CC(C1)CC(O)(C3)C2 c1(CNC2(CC(=O)NC(c3ccccc3F)C)CCC2)ccc2[nH]ccc2c1 Cc1cc(C)c(CC(=O)N(C2CCN(C(=O)COc3ccc(F)cc3)C2)CC)s1 C1(c2cn(CCC3CN(C(C4OCC(C)C4)=O)C3)nn2)CCCC(F)(F)C1 CCC(CCC(=O)NCC1CCCC(NC(=O)CCc2cc(C)nn2C)C1)OC N1(C(c2c(OC)cnnc2)=O)CCCC(CC(N2CCC2C)=O)CC1 NS(=O)(=O)CCCC(=O)NC1COCC1NC(c1cc2c(s1)CCOC2)=O CCC(CC(=O)NCCNC(C1(C)CCC(=O)N1)=O)C1CC1 Cc1cn(C)cc1C(=O)NC1(C(=O)NC(C(N)=O)C2CCCC2)CC1C Cn1[nH]c(C2CCN(CCN3CCOCC3)CC2)nc1=N N1(C(CC2(C)OCCO2)=O)CCC(CF)(NC(=O)Cc2cc(C3CC3)no2)C1 Cc1ccc(CNC(N2CCN(C(c3cn(CC4CC4)nn3)=O)CC2)=O)cc1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)Cn2ccsc2=N)c2c(c1)CCO2 CCC(C)C(O)C(C)C(=O)N1CCOC(CN(CC(=O)NC)C2CC2)C1 c1(CC)cccc2c(F)c(C(N3CC4C(NC(=O)C=C(Cl)Cl)C4C3)=O)[nH]c12 Cc1ccc(Cl)cc1C(=O)NC1(CNC(C2CCN(CC(C)C)C2)=O)CCCC1 N1(C(c2c(F)ccc(N)c2)=O)CCCC(C2CCCNC2)C1 c1(OC(C)C)n[nH]c(C(=O)NC2CN(C(=O)Cn3cccc3)CC2F)c1Br C=CCCC(C(=O)NC(c1cnns1)C)NC(=O)CCC(C)OC c1(C(=O)NCC(C)NC(C(C)NC(CC)=O)=O)ccc(C(F)(F)F)cc1[N+](=O)[O-] N1(C(CCCc2ncc(C)o2)=O)CCC(CNC(=O)CSCC(C)C)C(C)C1 C1(C(N(CC(C)NC(c2ccc(SCC)cc2)=O)CC)=O)CCCCC(F)(F)C1 c1(C(N2CCC(F)(CNC(C3(CF)CCC3)=O)C2)=O)cccnc1F C=CCCCC(C)(C)C(=O)N1CCC(C)N(C(=O)CC2CCS(=O)(=O)CC2)CC1 C1(C)(CNC(C2C(CC=C)CCC2)=O)COCCN(Cc2cn(C3CC3)nn2)C1 c1(C(C(=O)NCC2N(C(CCOCC)=O)CCCC2)C)ccc2ccccc2c1 C(=O)(CC(F)(F)C(C)C)N1CC(CC)N(C(c2nnn(C)c2C(F)(F)F)=O)CC1 C1(C(C)NC(c2ccc(C3CC3)o2)=O)CN(C(C2CCCC2)=O)CCO1 CC(CS(C)(=O)=O)C(=O)Nc1ccc(Cl)c(C#N)c1.C12CN(CC1O)c1cn2nn1 c1(C(N(C2CN(C(C3CC4(CSC4)C3)=O)C2)C)=O)nnc2ccccc2c1N C1(CNC(C(COCC)C)=O)CN(C(c2ccccc2OC(C)CC)=O)CCN1C c1(C(N2CC(NC(CC3(C)CC3(F)F)=O)C2)=O)ccc(C(=O)CF)cc1 c1(C(N2CCC(OCCNC(C(C)n3cncn3)=O)C2)=O)cc(C2CC2)nn1C c1(C(N(CC(C)N(C(=O)CC2CCN(C)C2=O)C)C)=O)cc2n(n1)CCC2 Cc1nc(N2CC3CCCC(NC(C4CC(C(C)C)C4)=O)C3C2)ccc1[N+](=O)[O-] N1(C(CN(C(C(C)C)=O)C)=O)CCC2CN(C(=O)CN3CCN(C)C(=O)C3)C2C1 C1(C(N(OCC(=O)OC)C)=O)CC(NC(c2cc(OC)n[nH]2)=O)CCO1 CC1(C)COCC1C(=O)NC1CN(C(C2CC3CCC(C2)C3)=O)C1 CCC(C)(CNC(C1CCC(=O)O1)=O)C(=O)NC(c1nnc(C)o1)C C1(CNC(C2CN(C(C3C4CCC(F)C34)=O)CCO2)=O)CC2(CCC2)C1 c1(OC)cc(C(N2CCC(F)(CNC(=O)C=Cc3nc(C)co3)C2)=O)c(F)cn1 c1(OC)ccc(C2CCN(C(c3csc(-c4cccc(F)c4)n3)=O)CC2)nc1 CCC(CC(F)F)C(=O)NCC1CN(C(=O)CC(C)C(=O)OC)CC(C)(C)O1 C(CC(C)(C)CC(=O)NC(c1nc2ccccc2o1)C(C)C)OC C1(C(=O)NC2CC(CC(=O)NC(CC(C)O)C)C2)CCC(C)(C)OC1 c1(CCC)nc(=NCC2(O)CCCN(C(=O)CC(=O)N(CC)CC)C2)s[nH]1 Cc1cc(C)c(NC(C23CC(CN(C(c4cnc(N)c(N)c4)=O)C2)C3)=O)cc1O C1(C(=O)NCC2CCC(C(N(c3ccc(OC)cc3)C)=O)C2)CCOC(=O)CC1 c1(CC(=O)N(C(C)CNC(=O)C(c2cncnc2)C)C)cccc2ncccc12 Cc1ncc2n1CCC(C(=O)NC(C)CNC(C1CC1C(C)O)=O)C2 N1(C(C(CCN(C)C)N)=O)CCC(OC(F)F)C(O)C1 c1(C(=O)NC23CCN(C(=O)C=Cc4nccs4)CC2C3)cccc2[nH]nc(O)c12 N1(C(C(=Cc2cn[nH]c2)C)=O)CCOC(CCNC(=O)CC2CCC(=O)N2)C1 c1(CNC(C(C)SCC)=O)ccc2c(c1)CCN(C(=O)Cc1cc(C)nn1C)C2 C(CC(C(C)(C)C)NC(C1CC1c1ccco1)=O)N(C(C(C=C)(C)C)=O)C C1(=CC(=O)N(C(C)CNC(=O)C=CCN(C)C2CC2)C)CC2CCC(C1)N2C C(CCC)(C(=O)NCC1CCC1N(C)C)NC(COCC(=C)C)=O C(=O)(C1CCCc2n[nH]cc21)N(CC(C)CNC(=O)Cc1cccnc1Cl)C c1(C(N2CC3(CCN(Cc4cc(F)cc(Br)c4Cl)C3)C2)=O)nc2ccccn2n1 Cc1nc(C)c(C(=O)NCC(O)CN(C(=O)COCCCN(C)C)C)o1 c1(C(=O)NCC)ccc(OC(C2CCC(C#N)CC2)=O)c([N+](=O)[O-])c1 C=CCC(CC)C(=O)NC1(C)CN(C(c2cc(OC(F)F)cc(F)c2)=O)C1 c1(OCC)ncccc1N(C)C(c1cccc[n+]1[O-])=O c1(C(C(=O)N(CCCCN(C(C2CC(=C)C2)=O)C)C)=O)cc(Br)cs1 CCC(C)C(O)CC(=O)NCCC1CC(NC(=O)CNS(=O)(=O)C2CC2)C1 c1(C(N(C2(C#N)CCN(S(=O)(=O)c3cn[nH]c3)C2)C)=O)cccc2c(O)nccc12 C(C(CC(C)C)C(=O)NCc1ccc(C(=O)NC(C2CCCO2)C)nc1)OC c1(C(=O)NC(CNC(Cc2c(C)n[nH]c2C)=O)CO)onc2ccccc12 N1(C(CCCCC)=O)CCC2(CC1)CC(NC(=O)CCn1cncn1)CO2 c1(CC(=O)NC2C=CCN(C(c3cc(O)ncn3)=O)C2)cc(F)cc(Br)c1 C(C(=O)N1CC(O)(C2CCCN2C(=O)COCC2CC2)C1)(C(C)(C)C)NC(C)=O CC(CCC(=O)N1CCC(CNC(=O)Cc2cncnc2)C12CC2)S(C)(=O)=O C1(C)(CC)CN(C(c2[nH]cnc2C)C(=O)Nc2ccc(F)cc2C)CCO1 CCCC(C(=O)N1CCN(CC(C)NC(c2cn(CC)nn2)=O)CC1)NC(N)=O C1(CNC(CCCC(C)=O)=O)COC(C)(C)CN1C(=O)CC1CCOC1(C)C C(C(O)C(=O)NC(C)CC(=O)NCCc1ccon1)=CC N1(C(CCC2(NC(=O)CCc3ccsc3)CCC2)=O)CC(O)(C2CCC2)C1 C(=O)(C(CC1CCCC1)NC(=O)CC(C)N(C)C)NCCCNC(C)=O c1(N2C(CNC3CN(c4ccc(C(N)=O)cc4)C(=O)C3)CC2)ccnc2ncnn12 N1(C(C2(CC)CCOC2)=O)CC(CCNC(C2C(CN=[N+]=[N-])C2(C)C)=O)C(C)C1 N1(C(=O)C=C2CCCC2)CCC(O)(C2(NC(C34CCC(CC3=O)C4)=O)CC2)CC1 CC1(C)CCCCCC1S(=O)(=O)Oc1cnnn1-c1ccccc1 Cc1cnc(C(N2CCOCC2CNC(=O)CCS(C)(=O)=O)=O)c(C)c1 N1(C(CCCOC)=O)CCCC(CO)(CNC(=O)CC2CCSC2)C1 C1(NC(c2cscc2F)=O)CC2CCC1CN(C(=O)C1CCc3c[nH]nc31)C2 N1(C(C(C2CCCCC2)C)=O)CC2CC(NC(c3ccc(Cl)s3)=O)CC1C2 c1(OC)cnc[nH]c1=NCC1(O)CCCN(C(=O)CSc2cccc(F)c2)C1 C(=O)(C(C)(C)C(C)O)NCC(=O)NC(C)C(C)C(=O)O n1(CC)nnc2c1C(C(=O)NCc1ccc(F)cc1F)CN(C(C1CC1C)=O)C2 Cc1cc2nc(NC(=O)N(c3ccc(=N)[nH]c3)C)sc2cc1F O=C(C#CC1CCCO1)NCC1CCCN1C(c1scnc1C1CC1)=O c1(C(N2CC(C)(O)C2)=O)nc(-c2cccc(F)c2C#N)c2ccccn12 n1(CC(=O)NCC2CC(NC(C(CCCC)O)=O)C2)ncc2ncccc12 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2SCCS2)=O)CCC1C C(C(F)(F)CO)N(C(=O)C(c1cccs1)NC(c1cccn1C1CC1)=O)C N1(C(c2c(C)cn(C)n2)=O)CC2CC1CCC2NC(=O)Cc1c[nH]nc1C Cc1cnc(C(N2CC(NC(=O)Cc3cc(C4CC4)on3)CC2C)=O)cc1C#N N1(C(C(C)Cc2ccc(Br)cc2)=O)CCOC2C(C(=O)OC(C)(C)C)CC12 c1(C(N2CCC(C)(NC(C(C(=O)OCC)F)=O)C2)=O)nc2ncc(C)cn2n1 N1(C(=O)Nc2cc(CC(C)C)ncc2)CCC2C(CC(=O)N2C)C1 NS(=O)(=O)c1coc(C(N2CCC(NC(=O)CC3CCC(=O)N3)C2)=O)c1 C1(NC(C(C2CC2)OC)=O)COC2(C1)CN(C(c1c(N)cccc1F)=O)C2 N1(C(C)C)CCOC(C(=O)NCCCC2CN(C(c3cc(F)n[nH]3)=O)CCO2)C1 C1(NC(c2c(NC)cncc2)=O)CCN(C(=O)C(F)(F)CN(C)C)CC1F c1(CCC(=O)NCCC2CCN(C(C3(F)CCOC3)=O)C2)ccc(F)cc1 c1(OC)ccc(C2C(C(=O)Nc3nccs3)C2)cc1OCC(N)=O C1(NC(c2c(C)occ2)=O)CC2CC(NC(c3cnc(Cl)c(N)c3)=O)C1C2 C(=O)(C(C)C(C)COC)NC1CC(NC(c2n[nH]c(CC)c2Br)=O)C1 Cn1cnc(=N)[nH]c1=NCc1cc[nH]c1-c1ccncc1 Cc1cccc2c(N(C(=O)C=Cc3ccc(F)cc3)CC3CCNC3)ncnc12 C(=O)(CC1=CCCC1)N(C(C)CNC(=O)C(c1cc(Cl)ccc1F)(C)C)CC Cc1ccc(CNC(C2CC2C(=O)Nc2oncc2C#N)=O)c(F)c1 Cc1cc(C)nc(N2CC(NC(c3cn(CC4CCCOC4)nn3)=O)CC2C)n1 N1(C(CCC2CC(NC(C3(C)N(C)CCC3)=O)C2)=O)CC2CC3CC2C1C3 C1(CCC(=O)NCCN(C(=O)Cc2nc(C3CC3)nn2C)CC)CCN(C)CC1 C1(CNC(c2c(C)n(C3CC3)nc2)=O)CN(C(c2cnc(N)cn2)=O)C(C)(C)C1 c1(C(=O)NC2C(C)N(C(=O)CC3CC3(C)C)CC2)c(Cl)c([N+](=O)[O-])nn1C C1(NC(c2cc(Cl)no2)=O)CC2CC1CN2C(C1(C(c2ccccc2)=O)CC1)=O CCCCN=C(NCC1(C)CCC(=O)N1)NC(C)CC.C12CCN1C2 C(=O)(C(CC(C)(C)C)NC(=O)CC1CC(C)C1)N1CC(CC(C#C)C)C1 C(C(=C)C1CCOCC1)NC1(c2n(CC=C)nnn2)CC(C2CCNC(=O)C2)C1 C1(N(C(=O)COCc2ccccn2)C)CN(C(=O)CN2CCSCC2)CC1(C)C C1(N=[N+]=[N-])(C(=O)NCC(C#C)C(C)C)CCN(C(=O)C(N)=O)C1 C(CC1=CCCCC1)N(C1CCCN(CCC)CC1)CCCS(=O)(=O)CC c1(C(C(=O)NC(CNC(C2(C(N)=O)CC2)=O)(C)CO)=O)cc(F)ccc1C C1(C(=O)NCC2(NC(CCC=C)=O)CC3CCC2CC3)Cc2c(C)cccc2O1 c1(C(=O)NC2CCN(C(c3cc(CC)on3)=O)CC2)cc(C)c(O)c(C)c1 CN1C(=O)CCC1C(=O)NOCCCC(F)(F)F.c12ncccc1C(=O)NC2 c1(C(=O)NCCOCCNC(CCC2CCN(C)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(CC(=O)N(C)CC2CCCN(c3nnn(C)n3)C2)CCOC(C)(C)C1 C1(C(=O)NC(Cn2cc(C(C=C)(C)O)nn2)C)CC2(CCNCC2)CO1 Cc1cc(C(=O)NCC2CC2NC(=O)CC2(n3ccnn3)CC2)cnc1C(F)F C(=O)(C1=NN(C)C(=O)CC1)N(C)CC1(CNC(c2nc(CC)oc2C)=O)CC1 C(C(C)N=c1[nH]c(CC#N)nc(Cl)c1C)(C1CC1)NC(C(C)C)=O C1(NC(C2(CO)CCN(C(C(C)OCCN(C)C)=O)C2)=O)C(C)(C)C(O)C1(C)C C1(C2(O)CCN(C(=O)C=CCN(C)C)CC2)(NC(C(C)NS(C)(=O)=O)=O)CC1 C(=O)(CCCC(C)=O)N1C(C(=O)NCC2(F)CCCCC2)(COC)C=CC1 c1(OCC)cccc(C(=O)NC2CCC(CNC(=O)CNC=O)C2)c1N C1(COC)CN(C(c2ncc(C(C)(C)C)cn2)C(=O)NCCCSC)C(C)(C)C1 C(C1(O)CCc2ccccc21)NC(CC(C=C)(C)C)c1nnnn1C1COC1 c1(SCC(N2C(c3cc(C)[nH]n3)CSCC2)=O)cccc(F)c1[N+](=O)[O-] C1(C(C)N(C)C(C2CC(CCNC(=O)CC(C3CC3)C3CC3)C2)=O)CCOCC1 CC1CN(C(=O)CCC2(C)CN(C(C3CCN(C)CC3)=O)C2)CC1(F)F CC1COc2c(C(=O)NC3CCCC3NC(=O)CCCC(N)=O)cccc21 CC1(C)C=C(C(=O)N2CC(NC(c3cc(-c4cccs4)[nH]n3)=O)CC(F)C2)C1 N1(C(c2c(CC)onc2C)=O)CCCC(C2(NC(=O)C(F)=C(C)C)CC2)C1 C12(CC(=O)NCC3C(CNC(c4nn(C)c(F)c4)=O)C3)CCC(CC1)CC2 c1(C(N2CC(C)C(CNC(=O)CCCC(F)F)C2)=O)coc2c1C(=O)NCCC2 C1(C(=O)NC2(CSC)CCC2)CCN(C(c2cnnc(O)c2)=O)CCO1 C1(OC)CC(CCNC(C)=O)N(C(C2CCN(CCC3CC(F)C3)CC2)=O)C1 C1(C(=O)NCC(CCC=C)O)CN(C(=O)Cc2c(C)noc2C)CCN1C c1(OC)cccc(C(=O)NC(C)CC(C)NC(=O)CCNC(C)=O)c1F N1(C(c2cnc(C)c(N)c2)=O)CCC2CN(C(=O)Cc3cccn3C)CC2C1 c1(SC(C(=O)OC(CCC)C)C)ccc(Cl)cc1 C1(C)(NC(C(CNC(C2N(CC)CCC2)=O)N(C)C)=O)CC(C)(C)C1 C1(NC(CC2(C)N(C(c3cc(C)cc(O)n3)=O)CCC2)=O)CCn2ncnc2C1 c1(C(=O)NCC(CC(C)C)NC(C(C(CC)O)C)=O)nc(N)cc2ccccc12 CC1(CNC(N)=O)CN(C(=O)C(C2CCCC2)NC(=O)CCCCO)CCO1 C1(NC(C2CCN(C)C2)=O)CN(C(c2cc(C(C)(C)C)on2)=O)CC2(CC2)C1 C1(C(=O)NCC(CSC)(C)C)C2CCC(C2)N1C(=O)C(C1CCCCC1)C c1(NC(C2CC(NCc3cccc4cc[nH]c34)C2)=O)c(Cl)cc(Cl)cc1[N+](=O)[O-] C#CCCCCCC(=O)N1CC=CC1C(=O)NCc1cc(F)ccc1Cl N1(C(c2c(C)c(Cl)ccn2)=O)CCC2(CCCCC2NC(c2cc(Cl)no2)=O)C1 N1(C(C2C=C(C)CS2)=O)CC(C(=O)Nc2cc(C)cc(O)c2)CCC1(C)C c1(N2CCCC(CC)C2)nc(N(CCS(=O)(=O)NC)C)nc2ccc(Cl)cc12 c1(CC(CC(F)(F)F)NCC2C(C)(C)COCC2)ccc([N+](=O)[O-])cc1F N1(C(C(n2c(C)cc(C)n2)C)=O)CC(NC(=O)CC2OCCO2)CC12CCC2 C1(NC(c2c(SC)ccs2)=O)CCN(C(C2(C)COCCO2)=O)CC1CO Cc1cc(-c2csc(C(N3CCn4cccc4C3)=O)n2)c(F)c(F)c1 C1(CC)CN(C(C2CN(C(C)C)C2)=O)CC1C(=O)NCCSC c1(C(C(=O)NCC(C)(C)NC(C2(CC)COC2)=O)O)cccc(OC)c1 O=C(CCCC(=O)c1ccc(F)cc1)NCC(F)CNC(C1CCCC12CC2)=O C1(C(=O)NC2CN(C(=O)CC3CNC(=O)O3)CC2O)(CC)CCCC1O C#CCC(C)(C)C(=O)N1CC(CNC(c2ccccc2C(C)C)=O)C(O)C1 Cc1ccc(F)c(C(N2CCC(C)(NC(C3CC34CC4(F)F)=O)CC2)=O)c1 c1(C(=O)NCCOC2CCN(C(CC3(C)CCCO3)=O)C2)cc(Cl)ccc1CO Cc1cc(C(=O)N(C2CC(NC(=O)Cc3cc(C)on3)C2)C)c(C)cn1 CC#CCCCC(=O)NC(CC#CC)C(=O)NCCC(=O)NC(C)CC N1(C(c2cnc(C(C)C)s2)=O)CCOC(CNC(=O)C=Cc2cnc[nH]2)C1 Nc1cc(F)cnc1C(N1CC2CCC2(CC(=O)NCc2cnsc2)C1)=O C1(C(=O)NC2CC(OC3CCCC3NC(CC)=O)C2)CN(C(C)=O)CCO1 CC1(C)CCCC(C(=O)NCC2CN(C(c3ccnc(F)c3N)=O)C2)CC1 C1(CCC)(NC(=O)COc2cn[nH]c2)CCCN(C(C2CCC(CC)O2)=O)C1 c1(CCC(=O)N(C(=O)CSc2ccccc2)CC)cc(C)nc(C)c1 C(=O)(CCCC1CC1)N(CC(C)O)CCNC(C(C)OC1CCCC1)=O C12CC(CN1C)OC2=O.c1(C(C)CN(C)C)ccc(CN2CCCCC2C)cc1 C(C)(C(=O)N1CC(NC(=O)C(C)=CCO)CC(F)C1)(C(C)C)OC N1(C(C(C)OCCC#C)=O)CCC(CCCCNC(C2C3CC4C(C3)C24)=O)CC1 c1(N(C(=O)C(C)=CC2CC2)CCOCC)nc(CC(=O)OC)cs1 CCC(C)C(C(=O)NCC(C1CCCC1)C)N(C)C(c1cnccc1C#N)=O N1(C(c2c(CC)nco2)=O)CC(CNC(C2CCC(C)(C)CC2)=O)C2(CCC2)C1 Cc1cc(=O)oc(C)c1C(N1CC2CC1C2NC(C1(Br)CC1)=O)=O C1(O)(CCNC(=O)CCF)CCN(C(c2ccccc2C(F)F)=O)C1 C1(OC)CC2(C1)CN(C(=O)CNC(=O)C(F)CC1CCC1)C2 C(C(C)(O)CC(=O)NCC1CC(NC(c2cnc(C3CC3)s2)=O)C1)OC N1(C(C(C(C)C)(C)C)=O)CC(NC(C2(C)CC2(F)F)=O)CCC(O)C1 c1(C(=O)NCCSCC)cc(-n2cc(C)cn2)cc(F)c1.O(C=CC(=O)NCCO)CC c1(C(=O)NC(CC)CNC(c2c(C)nn(C)c2C(F)F)=O)nn(C)c2c1CCC2 c1(C(=O)NC(c2ccccc2)CNC(C(C(C)C)O)=O)csc2ncnc(O)c12 N1(CCOC)CCN(c2nnc(-c3cc[nH]n3)n2CCc2cccs2)CC1 N1(C(c2n(COC)ncc2)=O)CC=C(C(C)(C)C(=O)N2CCC(F)(C#N)C2)C1 c1(OC)cc(C)c(C(=O)NC2CCCCN(C(=O)C(F)C(F)(F)F)C2)c(F)c1 N1(CC)CCC(NC(c2sccc2CNC(C2COC(C)C2)=O)=O)CC1 c1(C(=O)NC(CNC(C2CC(C)=C(C)CC2)=O)CO)n[nH]c2c1CCSC2 C1(C(=O)NC2CCN(C(CCOCCCOC)=O)CC2C)CCC(C2CC2)CC1 c1(C(C(=O)NC2(CN(C(=O)CN3CCOCC3)C)CC2)F)ccccc1 N1(C(CNC(C(CC)C)=O)=O)CCOC(C)(CNC(=O)CCS(C)(=O)=O)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(C(C)C)NC(C1CC1C#N)=O Cc1cccc2cc(C(=O)NCC3CCCN3C(c3cc(Cl)ncc3O)=O)sc12 CCC(O)C(=O)N1CCC(C(=O)NC2CSC2)C1 c1(SCC(=O)OC(C)=O)ccc([N+](=O)[O-])c(OC)c1.C1(=O)C=CCN1 c1(CC)ccc(C)cc1NC(=O)C(O)C(C)(C)NC(=O)OC(C)(C)C N1(C(c2nccc(-c3ccccc3)n2)C)CCN(CC(O)CNC(C)(C)C)CC1 c1(CC(=O)NC2C=CCN(C(c3ncc(F)cn3)=O)C2)c[nH]c2cccc(F)c12 C1(C(N2C(CN(C(Cn3c(C)nnn3)=O)C)COCC2)=O)CC2(C1)CC21CC1 N1(C(CCCC)=O)CCC2(CCOCC2)C(CNC(=O)CCCCC(F)F)C1 C1(CNC(c2ccc(Cl)nn2)=O)CCN(c2ncc(C(F)F)cn2)CC1(F)F C(=O)(C1=Cc2ccccc2C1)N1CC(C(=O)NCC(COC)(F)F)CC12CCC2 CC1C(CC(=O)NCCC2CC2)CCCN1C(c1cc(F)cc(Cl)c1)C(=O)N(C)C C1(C(N(CC(N2CCC3(CC3)C2)=O)CC)=O)CCn2ccnc2C1 Cn1cc2c(n1)CC(C(=O)NC1CCC(CCNC(=O)CNC=O)C1)NC2=O CC(F)CC(=O)N(C(c1ccccc1)CNC(=O)Cn1ncnn1)C c1(C(N(C)CCNC(c2cc(C(N)=O)ccn2)=O)=O)ccn2ccnc2c1 CC1CCC2(CC2)N(C(C2CC3CC2CN(C(c2cnccn2)=O)C3)=O)C1 c1(C(=O)NC2C(CNC(c3c(C)n[nH]c3)=O)CCC2)cc2cccnc2nc1O C#CCC(C)C(=O)NCCCNC(c1ccoc1I)=O c1(N2C(CCCNC(C(C)NC(COC)=O)=O)CCC2)nc(Cl)nc2[nH]cnc12 c1(CC)nocc1C(=O)NCC(CCNC(=O)Cc1ncoc1C)OC N1(C(Cn2cc(CNC(=O)Nc3cccc(N)c3)nn2)=O)CC2COCC2C1 CC1(C)COCC1C(=O)NC1CC2(C1)CC2NC(C1CC1c1ccccc1)=O C1(C(N)=O)CCCN(N2CCC(SCC(F)(F)F)CC2)C1 CN1CCOc2ccc(-n3cc(CC4(C(=O)O)CCC(CO)CC4)nn3)cc21 c1(C(C)=O)cc(CNC(CC2N(C(C34CC(CSC)(C3)C4)=O)CCC2)=O)oc1C CON(C)CCCNC(=O)C(CNC(c1ncoc1C(C)C)=O)N(C)C C(=O)(C(CCOC)NC(C12CCCC1C2)=O)NCC1CC(CN(C)C)C1 Nc1cc(C(=O)NC2CCC2NC(c2n[nH]cc2Cl)=O)c2ccccc2c1 N1(C(Cc2ccc(C)cc2)=O)CCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1 C1(C(=O)NCC2(C(N3C(CCC=C)CCC3)=O)CC23CCC3)CC(=O)CC(=O)N1 c1(OCCC)cccnc1CC(=O)NCCC1(O)CN(C(=O)CCC=C(C)C)C1 N1(C(C(CC)CCOC)=O)CC(NC(C2CCc3ccnn3C2)=O)CC12CCC2 c1(C(=O)NC2C3CN(C(c4c(C)cc[nH]4)=O)CC2C3)ccc2[nH]c(C)c(C)c2c1 c1(C(N2CCOCC(NC(C3C(=C)CC3)=O)C2)=O)cc(C)nc(Cl)c1N c1(CCC(=O)OC(CN(C)Cc2c(OC)cccc2)C)ccc(Cl)c(Cl)c1 CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(C2CCCCS2)=O)C(C2CCCC2)C1 N1(C(c2cnc(CC)s2)=O)C2CCC1CC(CNC(=O)C(O)C(F)(F)F)C2 C1(O)(C(=O)NCCNC(=O)Cc2cncs2)CCC(C(F)F)CC1 c1(C(=O)NC2CN(Cc3cncs3)CC2(F)F)ccc2ccccc2n1 C1(NC(C2CC(C)(CC)C2)=O)CCN(C(c2ccc(C(N)=O)cc2)=O)CC1 C1CC(=O)N=C2C=CN(N2)C12CC2.C(CC)(C(=O)NC)=CC CCC(C)(C(=O)N1CC2CCC1CN2C(=O)C=C1CCCCC1(C)C)C(N)=O C12(NC(C(CC)=CCCC)=O)CCCC(CN(C(c3cnc(C4CC4)s3)=O)C1)C2 N1(C(C(C(C)C)NC(C)C)=O)CC2CCC1C(NC(C1(O)CC1)=O)C2 C=CC(C)CC(=O)NC(C)(CNC(c1cscc1Cl)=O)C1CC1 c1(OC(C)C(=O)NCC(F)CNC(=O)CC2CC(=O)C2)ccc(Cl)cc1Cl C1(C(=O)NCC2CC(C)(NC(CSCCC)=O)C2)CNC(=O)CC1C C1(NC(c2c(CC)nco2)=O)CCN(C(=O)Cc2ccoc2)CC1CO N1(C(c2c(OC)scc2)=O)CCN(C(=O)C=CC=C(C)C)C(c2cn[nH]c2)C1 C1(NC(C(c2ccnn2C)C)=O)CCC(NC(c2cn(C(C)(C)C)nn2)=O)CC1 n1(CC)cc(C(=O)NC2CC(CNC(C3CCC(OC(F)(F)F)C3)=O)C2)c(C)n1 CCC(Cc1nc(CCN2CCCCCC2)no1)C(C)(C)C c1(C(N2CCC(O)(CN(C(c3c(OC)noc3C)=O)C)C2)=O)cc(C)cc(C)c1 C(=O)(CS(=O)(=O)c1ccccc1C)NC1CC(NC(CC2CC(CC)OCC2)=O)C1 c1(CNC(C2N(C(CCc3ccc(OC)nc3)=O)CCC2)=O)ccnc2[nH]ccc12 C1(C(=O)NCC(C)NC(=O)C(F)=CC2CC2)CCc2nnnn2CC1 Cc1nc2[nH][nH]cc-2c(=NC2CCC3CN(C(=O)C(F)(F)C(C)(C)O)CC23)n1 CC(C)(O)C#CC(=O)NC1CC1CNC(c1ccccc1N1CCCC1)=O C1(NC(C(Cc2ccc(C)cc2)C)=O)CCN(C(=O)CCC2CC2(C)C)C(C)C1 C1(O)(C(=O)NCCN(C(c2cccnc2)=O)C2CC2)CC2(CCOCC2)C1 c1(N2CCC(=C)CC2)ncnc2n[nH]cc12.C12CCCCC1N2 c1(OC)cc(C(=O)N(C)CC2(O)CN(C(=O)C(O)CN3CCCC3)C2)ccc1C N1(C(=O)NC)CCC(N=c2cc[nH]cc2S(=O)(=O)N2CCC(F)C(O)C2)C1 c1(-c2cccc(CC(=O)NC(c3cccc(F)c3Br)=O)n2)c(O)cccc1F N1(C(c2c(C)c[nH]n2)=O)CC2(CCCN(C(c3ccc(C(C)(C)C)cc3)=O)C2)C1 N1(C(c2ccc(COC(C)C)cc2)=O)CCC(O)(CNC(=O)C(C)O)CC1 C1(CNC(C(C)N(C)C)=O)CCN(C(=O)C(CO)N(C)C)C(C)C1 N1(C(c2ncc(OC)nc2)=O)CCCCC(C(=O)N(C(C)C(C)SC)C)C1 c1(C(=O)NC2(C)CC(NC(C3CC4COCCN4C3)=O)C2)cnn2c1NCCC2 C1(NC(C(C(C)C)CO)=O)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CC2(CCC2)C1 NC(=O)CCCCC(=O)N1CCC2(CC1)CC2NC(c1ccc(=O)oc1)=O C(=O)(C(O)CCC(C)C)NCC1C(CC(=O)NCc2ncc(C)[nH]2)C1 c1(C(N2CCN(C(C=CSC)=O)C(C)CC2)=O)ccc(C#N)c(F)c1Br Cn1cc(S(=O)(=O)NC(C2(C)C=CCC2)=O)ccc1=O N1(C(c2cc(CC)c(CC)o2)=O)Cc2nccn2CC(NC(C2CC2(Cl)Cl)=O)C1 CC(C)CCCCC(=O)NC1CN(C(=O)C(C)(C)Oc2ccc(Cl)cc2)C1 N1(Cc2cn(CC(CNC(C#CCOCC)=O)(C)C)nn2)C(=O)CNC1=O c1(C(N2CC(N(C(C(C(C)C)n3cnnc3)=O)C)C2)=O)cc(F)cc2nn[nH]c12 C(=O)(C(C)(C)C(C)C)N1CCC(CC=C)(NC(=O)C=Cc2ccc(C)s2)C1 S(=O)(=O)(c1ccccc1F)N1C(C(=O)OCc2nc(Br)c[nH]2)CCC1 N1(Cc2nccc(OC)c2)CCC2(CC1)CN(C(c1ccoc1C1CC1)=O)C2 Nc1ccc(F)c(F)c1C(N1CC(NC(=O)Cc2cnns2)CCC(O)C1)=O Cc1sc(Br)cc1C(=O)NCC(C)(CO)NC(C1CCS(=O)CC1)=O C1(CNC(C(COC)NC(c2ccoc2)=O)=O)(CO)CCN(C)C1 c1(C(=O)NCCCC(=O)NC)ccc2nnc(C(F)F)n2c1 C1(CC(N2C(CNC(c3c(C)cc(C)s3)=O)CC2)=O)OCCCC1(C)C CC(CC(C)(C)O)C(=O)NC1CC(N2CCN(C)CC2)C1 C#CCC(C)(C(=O)NCC(c1ccnn1C)O)NC(C1CC(F)(CF)C1)=O N1(C(C2(C(C)C)CC2)=O)CC(F)(CNC(=O)C(F)(F)Sc2cnn(C)c2)C1 N1(C(CSCCCC)=O)CC2CC2(CNC(C2CC2F)=O)C1 CC(C)(Cc1nn[nH]n1)C(=O)NC1(c2cccc(Br)c2)COC1 Cc1cccc(C(=O)NC2CC2CNC(c2cncc(N(C)C)c2)=O)c1C S(=O)(=O)(c1cccc(F)c1)N1CC(NC(c2c(C)ccc(C(=O)O)c2)=O)C(O)C1 C1(C(=O)NCC2(CCC)CC2)CC(NC(C2CCC(F)CC2)=O)CCO1 N1(C(c2ccncc2Cl)=O)CC2CCC1CN2c1nc(Cl)ncc1F CCC(CC)C(C(=O)NCC1COCCN1C(C1OCCCO1)=O)OC c1(SCC(=O)NCC2CN(C(C=CC)=O)CC2O)ccc(NS(=O)(=O)CC)cc1 C1(O)(C(=O)NC2CC3CC2N(C(=O)CC2CCCC2)C3)CC2(CCOCC2)C1 c1(CC)ncc2c(n1)CCC(C(N1CCCC(CNC(=O)C(C)(C)F)C1)=O)C2 C(C(C)(O)CC(=O)NCCCCCCn1cc(C2CC(F)(F)C2)nn1)OC CC1CC(NC(c2cc(OCC(F)F)ccn2)=O)CN1C(c1csnn1)=O C1(CC)CCC(C(N2CCOC(CNC(=O)C(O)CSC)C2)=O)CC1 C1(NC(=O)CCCn2ccnc2)COC2(C1)CN(C(C13CCCC1C3(F)F)=O)C2 N1(C(c2c(C)ccc(F)c2)=O)CC(C2CN(C(c3cc(C(C)(C)C)c[nH]3)=O)C2)C1 C=C=C(C)CC(=O)N=S(C)(=O)c1cnn2c1CN(C(C13CCC(C1)OC3)=O)CC2 C(=O)(CC1=NNC(=O)C1)N1CCC(NC(CCCN(C(C)=O)C)=O)C12CC2 CC1CN(C(=O)C(C2(C)CC2)NC(C2CCC2C)=O)C(C)C(C)(C)O1 C(=O)(C(F)(F)C(F)F)NC1CN(C(C2C(C(=O)OCC)C2)=O)CC1C(F)F CCC(CC(C)C)C(=O)NCC#CC(=O)N(CCCF)C c1(C(C)NCCCF)cccc(N2CCOCC2=O)c1 c1(CNC2CC3CC(CC(=O)OC)C2C3)c(C)cc(CN)cc1C C1(CC(=O)NCC2CC(O)CN2C(c2cccnc2S)=O)(COC)CCOCC1 C1(C(C)(C)C)CN(C(=O)CC(F)(F)F)CCN1C(=O)C(F)CC1CCCC1 C=CC(C)(C)NC(C1(NC(=O)CCOCCN(C)C)CC1)=O c1(C(=O)NCCCCNC(C2C(C)(C(C)C)C2)=O)cnnc(C2CC2)c1 CCC(CC(=O)NCCCc1cccs1)N(C(=O)C(CSC)OC)C c1(-c2cncc(C)c2)ccc(C(=O)Nc2ccnc(CC3CC3)c2)c(C)n1 c1(C(N2C(CNC(=O)CCC3CCOC3)C3CCC2C3)=O)cccc2c1OCO2 C(=O)(C1=CCS(=O)(=O)C1)N1CC2(CC(NC(=O)C(F)CC3CCCCC3)C2)C1 c1(CN2C(C)(C(=O)NCc3nc(Cl)ccc3F)CCC2)ccncc1[N+](=O)[O-] CN1CC(=O)NC12CCN(C(C1CCC(=O)CC1(C)C)=O)CC2 c1(NC2C3(CN(C(C4C(C)(C)CC4)=O)C3)CCC2)ncc2cccnc2n1 Cc1cc(C)n(-c2ccc(CC(=O)NC(C3CN(C(=O)C(C)(C)O)C3)C)cc2)n1 CC(C)(CCCNC(C1CCCO1)=O)C(=O)NC1C2CCCCC12 Cn1c([N+](=O)[O-])cnc1C(=O)OCC1CCCC(C)(C)C1 Cc1ccncc1C=CC(=O)NC(C1(O)CN(C(C2CC3CC3CC2C)=O)C1)C N1(C(C(COC)C)=O)CCN(C(c2ccccc2-n2ccnn2)=O)CC(O)C1 c1(SCC(=O)NCCC(O)CNC(C2CCCCO2)=O)ccc(F)cc1 C#CC1CCCN(C(=NCCF)NCc2cccc(C(F)(F)F)c2O)C1 C(C)(N=c1[nH]nc(C(N)=O)s1)C1(O)CN(C(Cc2c(C)nc(C)s2)=O)C1 c1(C(N(CC(CNC(CC(C(=O)OC)C)=O)O)C)=O)cnc2cc[nH]c2c1 c1(C(=O)NCCC2N(C(CC(CC)C)=O)CCSC2)ccc(F)cc1C#N c1(C(N2C(C)CCC(NC(c3cc(OC)ns3)=O)C2)=O)cccn2nccc12 c1(C(=O)NC2CN(C(C3CNC(=O)O3)=O)C(CO)C2)cc2ncsc2[nH]1 C1(CC#C)CCCN(C(C2C(C)CCN2C(=O)COCC(=C)C)=O)C1 N1(C(C(C)OCCOC)=O)CC2CCC2(NC(=O)C=CBr)C1 C1(CNC(c2nnc(CC)s2)=O)CCN(C(=O)CSC(F)(F)F)CC1C C1(NC(CCC(C)(C)N(C)C)=O)CN(C(=O)OC(C)(C)C)C(C)(CO)C1 C(C)(CC(=O)NC1CC(=CC(=O)NOC(C)C(=O)OC)C1)OC CCCCC(O)CC(=O)N1CCC(F)(CNC(=O)CCc2cc[nH]n2)C1 c1(C(=O)NCCC(CNC(c2cn(C3CC3)nn2)=O)OC)ccccc1C c1(C(=O)NCC(CNC(c2cc(Cl)cc(C)c2N)=O)O)ccc2c(c1)CCC=C2 CCC(C)CC(C)C(=O)N1CCC(CCNC(C2CC(C)(C)C2)=O)CC1 c1(C(N2C(C(=O)Nc3cc(OC)ncc3)CCC2)=O)ccn2cncc2c1 Cc1cc(N)c(C(N2CCC(OC3CN(C(C4CC(F)C4)=O)C3)CC2)=O)cc1C CCCC(C(F)(F)F)NC(C1CCCN(C(c2cc(C)nn2C2CC2)=O)CC1)=O C1(C#N)(C(=O)NC(CN(C(c2ccsc2C)=O)CC)C)CCC1 C1(CNC(C2C(OCC)C2)=O)CC2(CC2)CN1C(C1CC12CCSCC2)=O N1(C(C(CC)OCC)=O)CCC(N(CCO)C(c2cnoc2CC)=O)CC1 c1(C(N2CC(NC(C(CC)(C)OC)=O)C(C)C2)=O)c(N)cccc1Cl Cc1cc(CC(=O)NC(C)CCCNC(=O)C(C)Cc2cnc[nH]2)c(C)s1 S(=O)(=O)(c1ccc(Cl)c2cccnc12)NC(C(c1ccc(CC)cc1)N)=O CC1CCc2[nH]nc(C(N3CC4CC(NC(=O)CCCC(N)=O)C3C4)=O)c2C1 C1(COC(C)C(=O)OCc2ccccc2)CCCN1Cc1nc(C(C)(C)C)no1 C(=O)(C1=Cc2ccccc2C1O)N(CCNC(c1cc(C2CC2)nn1C)=O)CC C1(C(=O)NC(C)CCNC(=O)C(C)CCO)CC(=O)CC1(C)C c1(CC(=O)NCCc2cn(-c3cc(C)cc(N)c3)nn2)cccc2cccnc12 S(=O)(=O)(c1nccs1)NC1CCCN(C(c2cccc(Br)c2F)=O)C1 N1(C(CCCCN(C)C)=O)CC2CC(C1)N2C(C1CC2(CC2)CN1C)=O C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(CNC(C(C(CC)C)O)=O)C12CCC2 N1(C(C2CCC(NC(C(CCC)C)=O)C2)=O)CC(C2CC2)(CC)C1 C12(C(=O)NCC3(NC(Cc4c(C)n[nH]c4C)=O)CCOC3)COCC1C2(F)F c1(C(c2nnnn2CC)NC(c2ccccc2)(CSCC)C)ccc(F)c(Br)c1 N1(CCNC(CCC2(NC(C(C)c3cccs3)=O)CCC2)=O)CCCCC1 c1(C(N2CC(NC(C(C)C3CCCO3)=O)(CO)C2)=O)cc2c(Cl)cc(F)cc2[nH]1 C(=O)(C(F)C(C)(F)F)N1C(C(N2C(C)(C(=O)NC)CCC2)=O)CC(O)C1 C=C(C)CN=C(NCC1CCOC1)N(C)CC(=O)NC(C)(C)C C1(CC)CN(C(c2nn(CC)cc2Cl)=O)CCC1NC(C1(O)CCSCC1)=O N1(CC)CC(C(=O)NC2CN(C(=O)CCc3nc(C)no3)C2)CCC1=O c1(C(=O)NCCC(C(C)C)NC(c2cscn2)=O)c(F)cccc1[N+](=O)[O-] N1(C(c2cc(C)nnc2)=O)CCN(C(=O)CCCCCF)CC1CF C(=O)(CC1=CSC2=NCCN12)NCC(C)NC(=O)C(C)CS(C)(=O)=O CC(=O)CC(C)(C)CC(=O)N(C)CCN(C)C(C1CCC(=O)N(C)C1)=O C12(CC(N3C(C(=O)OC)CC3)=O)CCC1CN(C(=O)CCC1CCCCC1)C2 c1(NC(CCSC)C)ccc(S(=O)(=O)N(C)CCc2c(F)cccc2Cl)c(Cl)c1 C(N=c1[nH]c(=NCc2ccoc2)[nH]c2c1CC(C)CC2)c1cc(OC)c(C)cc1 CCC(C(=O)NCC1COCCN1C(=O)C(C)C1(O)CCC1)C(C)(F)F c1(CC(=O)NCCC(C)NC(C(C(CC)C)NC(C)=O)=O)ccc([N+](=O)[O-])c(N)c1 N#CCCCCC(=O)N1CCC(NC(C2CC3CCC2O3)=O)CC1 c1(NCC#C)nc(C)sc1C(=O)N(CCO)CCc1cccc(Br)c1 CCCCC(O)CC(=O)NC1CCN(C(=O)CCc2c(C)noc2C)C12CCC2 Cc1cc(NC(=O)C(C2(O)CCC2)NC(=O)C#CC2CCC2)cnc1Cl c1(C(=O)NC(CNC(CSCC=C)=O)C(C)C)cccc(C)c1N N1(C(C2CCN(CC(C)C)CC2)=O)CCN(C(=O)CC2CC2(C)C)CC(CO)C1 CCCCC(O)CC(=O)N(CCCNC(c1ccc(C)nc1)=O)CCC c1(C(=O)NC(CN(C(=O)CCn2cccn2)CC)C)cnn(C(C)C)c1Br C(CC(C)C)(C(=O)NCC(O)C(=O)NC)N(C(C1CC(=C)C1)=O)C N1(C(CC(=O)NCC)=O)CC2(CNC(=O)CC(C)(C)CC)CC2(C(F)(F)F)C1 O=C1C2COCC1CC(C(=O)NC1CCN(C(C3CCC3)=O)CC1CO)C2 c1(C(N(CCC(C)NC(c2cc(N3CCCC3)ccn2)=O)C)=O)ccncc1O C1(C(=O)Nc2ccc(F)cc2CO)CC2(C1)CN(C(=O)CC1CC1)C2 C1(OC)CN(C(=O)C(CCC(C)C)NC(C2COC(=O)N2)=O)C2(CCC2)C1 CN1CCC(C(=O)NCC2CCC(NC(c3cc(C(F)(F)F)cs3)=O)C2)CC1=O C(N=c1ncc(F)c[nH]1)C1N(C(CCCC(=C)C)=O)CCCC1 c1(NCC(CNC(CC(C)C(F)F)=O)O)ccc([N+](=O)[O-])cc1F C(COC)(CC(=O)N1CCC(O)(CO)C1)NC(C1CCC(CC)O1)=O N1(C(C2(C#N)CC2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C2(CCC2)C1 CC(CCC(C)(C)C)C(=O)NCC(c1ccccc1)N(C(=O)CP(C)(C)=O)C c1(N2CC3CN(C(=O)Cc4cc(F)ccc4Cl)CC32)ncc2cc(Br)cnc2n1 N1(C(c2cccc(C)c2)=O)CC2CC(CNC(=O)CN3CCOCC3)CC1C2 c1(OC(C(=O)NCC2CC(NC(C(C)C)=O)C2)(C)C)ccc(F)cc1 C(CC1=CCCCCC1)NC(CC1CC(NC(C2(CC(C)C)CC2)=O)C1)=O c1(CC(=O)N(C2CCCN(C(c3c(CC)nns3)=O)C2)C)ccc(C#N)cc1 C=Cn1nncc1C(=O)NC(c1ccccc1)CNC(=O)C=CCOCC c1(C(=O)NC2C(NC(C(C=C)(C)C)=O)CC2)c(F)ccc(C)c1Cl C1(C(N(C2CCN(Cc3cnsc3)CC2)CC#C)=O)CCCC(F)C1 CC1(C(=O)NCC2(NC(c3cccc(CC(F)(F)F)c3)=O)CCC2)COCCO1 Cn1nc(CNC(=O)NCC2(NC(=O)OC(C)(C)C)CCC2)cc1Br c1(CNC(=O)NCC2(C(=O)OCC)CC2C(F)(F)F)c(C)ccc(C)c1O Cc1cc(C(N2CCCC2(C)C(=O)Nc2cncnc2O)=O)ccc1Br c1(C(N(CCNC(=O)COc2ccsn2)C2CC2)=O)ccn2ccnc2c1 c1(C(N(CCC(=O)NC(C2CCCC2)CC)C)=O)ccc(O)nc1 c1(NC(C(=O)NC2(CCCNC(C=CC=CCC)=O)CC2)C)ccc(F)cc1 C1(NC(=O)OC(C)(C)C)CC2CC(NC3CCN(C4CC4)C3=O)CC12 c1(SC)ccc(C(N2CC3C(NC(c4cn5c(n4)SCC5)=O)C3C2)=O)c(Cl)c1 CC1(NC(c2ccncn2)=O)CN(C(=O)C(C)(C)c2ccc(Cl)s2)C1 C(C(O)CC(F)(F)F)NC(C(C(C)NC(c1cccc(CO)n1)=O)C)=O Cc1nc(CC(=O)NC2CC(O)(CNC(c3ccsc3CN(C)C)=O)C2)sc1C CCCCC(CNC(c1ccc(C(F)(F)F)nn1)=O)NC(=O)C=CCF c1(C(=O)NCC2(COC)N(C(C(CCCC)O)=O)CC2)ccc2c(C)noc2c1 CCCC(CNC(=O)C(C)(C)C(C)(C)O)C(=O)NCC1CC(O)C12CCC2 C1(NC(c2ccc(OC)s2)=O)CCCCC1CNC(c1c(C)[nH][nH]c1=N)=O c1(NC(C2(C)N(c3cc(OCC)ncn3)CCC2)=O)ccnc(Cl)c1OC c1(C(N2C(CNC(c3c(C)snc3)=O)CCCC2)=O)cc2c([nH]1)CCC(C)C2 c1(C(=O)NCC2CC(CC(=O)OC)C2)c(Br)ccc(F)c1I C12(NC(=O)NCC3CCC(N4CCOCC4)CC3)CCCC1C2(F)F C1(C(N2CC3(CCNC3=O)C2)=O)N(C(C2CC23CC3)=O)CC12CCCC2 C(C)(CNC(c1ccsc1CC)=O)(CC(C)C)NC(c1cccc(CCC)c1)=O N1(Cc2nc(-c3ccn(C)n3)nn2CCN(C)C)CCC2(CC1)N=N2 c1(C(N)=O)cc(C(=O)NCC(O)Cn2cc(CC(C)(C)O)nn2)c[nH]1 C1(NC(CSCCCCC)=O)C=CC(CC(=O)NC(C)CC(C)O)C1 CCC(C)CC(=O)N(CCNC(=O)C(N1CCC(O)CC1)C)C(C)C c1(C(=O)NCC(F)(F)F)c(-c2ccccc2C(=O)NC2CCCC2)cncc1F N1(C(C2(CC)CCOCC2)=O)CCC(C)C(NC(c2ccncc2)=O)C1 CCC(CC(=O)NCC(O)CN(C)C)N(C(=O)C(F)n1ccnc1)C C1(NC(C2(CNC(C(CC=C)NC(C)=O)=O)CC3(CC3)C2)=O)CCOC(C)(C)C1 C1(NC(c2nc(C)sc2)=O)CN(C(=O)CCc2ccc(F)nc2)CC2CCCC12 c1(C(=O)NC(C(C)C)CNC(=O)CC2CC=CCC2)ccc2c(=O)cc[nH]c2c1 c1(C(=O)NCCC2CCCN(C(COCCC)=O)C2)ccc(C(C)CC)nc1O C1(=CC(N2CC3C(NC(=O)C=CCn4cncn4)C3C2)=O)CN2CCC1CC2 c1(C(N2CCC(CC=C)(NC(=O)C(O)CCSC)C2)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(CC2N(C)CCC2)=O)CCCCN(C(c2cncnc2)=O)CC1 CC(CN(C(=O)C(F)C(C)C)C)N=c1ccn2c(Br)cnc2[nH]1 c1(OC)cc(Cn2nc(C(C)O)nc2CC(C)P(C)(C)=O)cc(OC)c1OC CCN(C(C)c1cccc(C(F)(F)F)c1)N1CCN(C)CC2(CCCCCC2)C1 N1(C(c2[nH]cc(CN(C)C)c2)=O)Cc2ccccc2C(NC(=O)C=CCF)C1 c1(Nc2ccccc2)ccccc1O.n1(C(CN)=O)nncc1C(CCC(F)(F)F)=O C#CC1(C(=O)NC(CNC(=O)C(F)(F)c2nc(CC)cs2)CC)CCCC1 Cc1noc(Cl)c1CC(=O)NCCN(C(c1conc1C(C)C)=O)CC1CC1 c1(C(=O)NCC(CNC(c2cc(CCC)ncc2)=O)(C)OC)cc(C)cc(C)n1 C1(N(C(C(=O)NC2COC2)c2cscn2)C)CCC(C)(C)C1 CN1CCC(CNC(=O)N=c2ccn(CCS(C)(=O)=O)[nH]2)c2ccccc21 c1(C(=O)NC(C)CN(C)CCOC2CCOC2)ccc2ccc(Cl)cc2n1 C=CC1CCCCN1C(=O)C(C(C)(C)C)NC(C1CC(C)N(C)C1)=O Cc1oc(CNC(=O)CCCC#N)nc1C(N1CCC(C(C)C#N)CC1)=O Cc1cn(C(C)(C)C(=O)NCC(C)NC(=O)CCc2nncn2C)cn1 C(CC(O)CCO)NC(C(C1CCCC1)NC(=O)CCc1ccccc1)=O c1(C(=O)NCC2CCN2C(=O)C=C(Cl)Cl)ccc(=O)n(CC(F)(F)F)c1 CC(C)(CCCF)C(=O)NC1CC(CNC(C23CCCC2C3(F)F)=O)C(O)C1 [N-]=[N+]=NCCC(=O)N(CCC(=O)NC1CCCC(C(N)=O)C1)CCCO CC(O)(CC(F)F)C(=O)N1CCCC(NC(C2(C(F)(F)F)CCOCC2)=O)C1 C(CC(C)C(=O)N1CCCC1C=CC(=O)NCC1C=CCOC1)=CC c1(C(C(=O)NC(C)COCC(F)(F)F)F)ccc(Cl)nc1 c1(C(N2CCCC(CNC(c3c(OC)csc3)=O)C2)=O)ccc(O)nc1Cl N1(C(CC#N)=O)CCC2(C1)CN(C(=O)Cc1csc3cccc(F)c13)CCO2 C1(N(C(C2CN(C)C(=O)N2)=O)C)CCC2CN(C(c3csc(O)n3)=O)CC12 c1(COC)ncc(C(N2CCCC(NC(c3n[nH]c(SC)c3Cl)=O)C2)=O)c(O)n1 Cc1cc(C(=O)NCC23CC2CN(C(c2ccc(C(F)F)cn2)=O)C3)cc(F)c1 CC(F)(F)C(=O)NCC1CC(NC(C2CC2[N+](=O)[O-])=O)C1 CC(C)C1=CCC(NC(=O)COC(C)(C)C)CC1.c12ccccc1SC2 C1(Nc2ncn(C)c(=O)c2)(CNC(=O)C(=O)NC2CC2)CCC(F)(F)CC1 n1(CC(=O)NCC2(NC(=O)CSC3CCCC3)CCCC2)ncn(O)c1=O N12CCC(CC13CC3)CC(=O)COC2=O.c1(C2C(C(C)(C)C)C2)ncco1 CC1CN(C(=O)C(F)F)CC1CCc1cn(Cc2nc(C(N)=O)cs2)nn1 C(C(=O)O)(C(O)c1cccnc1)NC(C(n1cc(Cl)cn1)C)=O c1(C(=O)NC(C2(O)CN(C(C=CCC)=O)C2)C)cc(C)c(Cl)cc1C N1(Cc2cccc(OCC)n2)CC2(CCC(NCc3cc(C)cc(Cl)c3)C2)C1 c1(CC(=O)NCCC2CC(NC(C(C)c3ccco3)=O)C2)ccc(Cl)cn1 C(CCCCC(=O)NCC1(O)CC(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1)SC C1(NC(c2cn(CCOC)nn2)=O)C=CCN(C(=O)C(F)C2CCC2)C1 Cc1c(C(N2CC(O)CC2CNC(C2CC3(CC3)CO2)=O)=O)nn(C)c1Br C1(c2ccc(CC)cc2)CN(C(C2(CCF)CC2)=O)CCN1C(C1SCCS1)=O C(C)(C)(CC(F)C(=O)NC(C)C(=O)N(C)C1CC1)NC(c1c(CC)cco1)=O c1(C(=O)OCC)c(C)nc2scc(C(=O)NC)c2c1C.N12CC(C(C)C1)NC2=O C(=O)(CC(CC#N)c1ccccc1)NCC(C)NC(C1(c2ccccc2F)CC1)=O Cc1ccc(C(F)(F)F)cc1C(=O)NCC1CC1NC(c1ccc(F)cn1)=O C1(C(=O)NC(C)C(C)(C)NC(=O)CS(=O)(=O)C2CC2)Cc2cc(Cl)ccc2O1 c1(CC)noc(C(N2CCC(N(C(=O)Cc3ccoc3C)C)CC2)=O)c1C Cc1cccc(C(=O)NCC(C)C(=O)NC(C2CCC2)C2CC2)c1F N1(C(c2c(C)cccc2N)=O)CC(C2CCCN(C(c3cn(C)nc3O)=O)C2)C1 C1(CCNC(Cc2nnc(C)s2)=O)CSCCN1C(=O)CSC(F)F c1(C(=O)NC(C)Cc2cccc(C(F)(F)F)c2)cc2nccc(C(F)F)n2n1 n1(CC)nc(C(=O)NCC(O)CNC(=O)CCc2csc(=N)[nH]2)c(Br)n1 c1(OC)cnc(C(C)C)c(C(=O)NCCNC(=O)CNC(c2ccoc2)=O)c1 c1(C(=O)NCC(CC(=O)NCC(C)CN(C)C)C2CCC2)ccc([N+](=O)[O-])o1 c1(CC(N2CC3CN(C(c4c(C)c[nH]n4)=O)CC3C2)=O)ccc([N+](=O)[O-])cc1F N1(C(c2cn(CCC(F)(F)C(F)F)nn2)C(=O)NC)CCCC1C1OCCO1 c1(C(=O)NC2C(CNC(C=CC(=O)OCC)=O)C2)c(C(F)(F)F)cccc1F c1(C(N2CC(C(C)NC(=O)C(C)(Cl)Cl)OCC2)=O)ccc(=O)n2c1CCC2 c1(NC(C2(CNC(c3ccc(OC)cc3)=O)CC2)=O)scc(O)c1C#N C#CCCCC(C)C(=O)NC1C2CCN(C(=O)CCc3ccncc3)CC12 c1(C(C(=O)NC(CNC(Cc2nc(C)[nH]n2)=O)CO)(C)O)ccc(F)cc1 CCC(Cc1cccc(F)c1)C(=O)NCC(c1cn(C2CC(O)C2)nn1)(C)O c1(C(=O)NCC(CC(C)C)NC(=O)CSC(F)F)ccc2nc(O)[nH]c2c1 C#CC1(C(=O)NCc2nonc2C)CCN(C(=O)C(O)C2CC2)CC1 N1(C(C2(F)CCN(C)CC2)=O)CCC2(CNC(=O)Cc3ccsc3)CCCC12 CC(C)(CNC(=O)C(C1CCOCC1)N1CCCC1)Cn1cc(C2CC2)nn1 CC1(C)CC(NC(=O)C=CCO)CCN(C(C2CC3(CCCC3)CO2)=O)C1 C(=O)(C(C)C(F)(F)C(F)F)N(CCNC(C(C(CC)(C)C)O)=O)C(C)C c1(CC(N2CCN(C(COCCCC)=O)C3C2C3)=O)c[nH]c2c(CC)cccc12 N1(C(C(CCCC)C)=O)CC2(C1)CN(C(=O)CCCOCCOCC)CCO2 C1(NC(c2c(C)nc[nH]2)=O)CN(C(c2cncc(Cl)c2)=O)CCC1F Cc1ccc(O)cc1CN1CC2(CC2)CC1C(=O)NCCC(C)CO Nc1c(C(=O)NC(c2ccccc2Cl)CCO)cc(F)cc1Br C#CCCCC(C)C(=O)N1CC=C(C(=O)NC(C)(C)CCO)CC1 O=C(C1=CCCCO1)NC1CCN(c2ncnc(O)c2Br)C1 C(=O)(C1=COCCO1)NCC1(CNC(=O)CCc2cn[nH]c2)CC12CCC2 c1(N2CCC(C(C)NC(c3cnc(Cl)cn3)=O)CC2)nc(C(C)(C)C)nc(=N)[nH]1 N1(C(C(CCSC)NC(C)=O)=O)C2CCC1C(F)C(NC(c1coc(Cl)c1)=O)C2 C=CC1(C(=O)N(C)CC)CCN(C(c2ccc(N)c(F)n2)=O)C1 c1(C(=O)NC(CNC(CN2CC(C)C2)=O)C)ccc(-c2ncno2)cc1 N1(C(C2C(OC)(OC)CC2)=O)CC(CNC(c2ncoc2C)=O)CC1(C)C CC1CCN(C(=O)CCCc2cnn[nH]2)C(C(=O)NCCCC2CCCCO2)C1 C1(C(=O)NC2C(NC(=O)CCc3ccsc3)C2)CCCC2(CCC2)O1 c1(C(N2CC(C(N(C)CC3C(C)C3)=O)OCC2)=O)cc(F)ccc1F c1(C(=O)NCC)ccc(C(CC)NC(C2CCCN2N=O)=O)cc1 c1(CN(C)CC2(C)CC2(F)F)cc2cc(Cl)ccc2s1 CC(C)CCCN=c1[nH]c(N2CCC3(CCCN3C)C2)nc2ccc(Cl)cc12 c1(OC)cc(-c2nc(CCCOC)nn2C(C)C(F)(F)F)c(C)cc1C1CC1 C1(C)(CC)C=C(C(=O)NCC2CN(C)CCN2C(c2csc(C(C)=O)n2)=O)C1 C(C(=O)N(C1CCCN(C(c2c[nH]c(Br)c2)=O)C1)CCO)(C(C)C)OC C=C(C)CC(C(=O)N(CCCNC(c1ccc(C(=O)OC)s1)=O)C)NC(C)=O c1(C(=O)NCC2CC(NC(c3c(N)ccc(O)c3)=O)C2)ccnc2c1CCC2 N1(C(c2ccc(SC)o2)=O)CCCC(O)(CNC(=O)Cc2cc(C)cc(C)c2)C1 N1(CC(=O)N(C(=O)Cc2ccc(F)c(Cl)c2)C(C)C)CCCCC(C(C)(C)C)C1 C1(CNC(CNC(=O)OC)=O)CC(OC)CN1C(=O)C(C)(C)NC(=O)C=COC C1(OC)CC(NC(c2cncc(C(C)C)c2)=O)CN(C(=O)C(F)OC(F)(F)F)C1 N1(C(c2c(C)nc(=N)[nH]c2)=O)CC2(NC(=O)CC3CCN(C)C3=O)CCC1CC2 C1(NC(CNC(c2ccc(C)s2)=O)=O)CC2CN(C(C34CC(C3)C4)=O)CC12 C1(NC(C2N(C)CCC2)=O)CN(C(c2cc(O)ccc2F)=O)C2(CCOCC2)C1 N1(C(c2scc(OC)c2OC)C(=O)NCCC)CCCC(C)(C)C1C(=O)OC C1(NC(CSCC)=O)CN(C(=O)C=Cc2cncc(O)c2)C(C)(C)C1 N1(C(C(C)OCCC=C)=O)CCC2(CCOCC2)C(NC(=O)CC(C)CCC)C1 C(=O)(C(C#N)CC)NC(CCC)CNC(c1ccncc1OC(C)C)=O CCC(C(=O)NC1(CO)CCN(C(=O)C(=O)NC)C1)C(=O)NCCOC c1(C=C(COC(c2c(CCC)n[nH]c2)=O)C)ccc(OC)c(OC)c1OC N1(C(=O)Nc2cnc(C)s2)CC2(CCN2C(=O)Cc2ccc(Cl)cc2)C1 c1(C(=O)NCC(C(C(C)C)C)NC(c2ccc(Cl)cn2)=O)cnc2[nH]ncc2c1 C(C(O)(C(=O)NC1CC2C1CCN2C(C1CCCC(=O)N1)=O)C(F)(F)F)N(C)C C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(C)C2CC2)CC1F c1(C(=O)NCCOC2CN(C(C(C)SCC)=O)C2)csc2cc(OC)ccc12 C1(NC(Cc2c(C)cccn2)=O)CC(F)CN(C(C2CCC(=O)N2)=O)C1 CC1C(=O)N(C)CCN1C(=O)CCC1(NC(c2ccncc2O)=O)CCC1 C(=O)(C(C)(C)C(=O)NCC(C1CCN(C(c2cnc(O)c(C)c2)=O)CC1)O)NC N1(C(c2c(CC)ncs2)=O)CCCC2CN(C(=O)C(c3ccccc3C)C)CC12 c1(C(=O)NC2(CN(C(C3C(OC)C3)=O)C)CC2)cc(=O)c2ccccc2[nH]1 C1(NC(C(CC)OC2CCCCC2)=O)CN(C(=O)C=CC=C(Cl)Cl)CC1SC c1(C(=O)NC2C(NC(C3(C(F)(F)F)CC(=C)C3)=O)COC2)cc(F)cnc1OC N1(C(CNC(C2CCCCCC2)=O)=O)CCOC2CCCCC12 c1(C(=O)NC(C2CCCCC2)CNC(C2N(CC)CC2)=O)cscc1Cl C=CCC(CC=C)C(=O)NCC(CCCC)NC(c1ccnc(CN(C)C)c1)=O CC1=C(C)CC(C(=O)NCC(C(=O)NC2CN(C(N)=O)C2)N(C)C)CC1 CC1Cc2cc(C(=O)NC34CCC(C3)N(C(=O)CN(C)C3CC3)C4)ccc2O1 C1(CN(C(=O)COCCCF)C)CCCC(NC(c2ncccc2F)=O)C1 c1(C(=O)NC(C2CCN(C(c3c(C)c[nH]n3)=O)C2)(C)C)nn(C(F)F)cc1Cl C(=O)(C(CCC(C)C)CC(=O)OC)NCC1CC(F)(C(=O)NC)C1 C1(CN(CC)CC)CCCCN1C(=O)CCc1ccc(N(C)C)nc1 N1(C(C(C)(C)OC(C)C)=O)CCN(C(C2(C)CCCS2)=O)CC12CCC2 n1(CC)cc(Cl)c(C(=O)NC(C(C)NC(c2conc2COC)=O)C(C)C)n1 c1(C(=O)NCc2cc(C(N(CC(C)O)CCF)=O)on2)cc2occc2[nH]1 c1(CC(=O)NCCN(C(=O)C2=C(C)CCC2)CC)ccc2ocnc2c1 c1(COC)ccccc1CC(=O)N(CCNC(c1cc(=O)cc[nH]1)=O)CC1CC1 C12(NC(COCCSC)=O)CCC(CC1)N(C(=O)CC1CCCS1(=O)=O)C2 n1(C(C)C)nccc1-c1cn(C2CC(NC(C3CCC(C(N)=O)C3)=O)C2)nn1 c1(CC(N2CC(CC(C)NC(c3c(CC)cno3)=O)C2)=O)ccc(F)cc1 c1(C(=O)NC2CN(C(C(CC)C(C)O)=O)CC2(C)C)ccnc2[nH]ncc12 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CN(C(=O)C(F)C1=CCCCC1)CC2CO N1(C(c2c(C)cccn2)=O)CCn2c(CNC(c3cccnc3N)=O)nnc2C1 C1(NC(C(c2ccccc2)OC)=O)COCCC1NC(c1nc(C)oc1C)=O C(CCCC(=O)N1CCC(F)(CNC(C2C3CN(C)CC23)=O)C1)SC C1(CNC(c2ccc(SCC)nc2)=O)CCC(C)CN1C(=O)CNC(N)=O c1(SC)cc(C(=O)NCCC2(O)CCCNC2)cc(SC)c1 N1(C(c2cc(C)ns2)=O)CCN(C(=O)C(n2nccc2C)C)C2CCCC12 C1(CCNC(c2cc(OCC)no2)=O)CC(F)(F)CN1C(=O)C(N)=O C1(NC(C2(CC)CC2)=O)CC2CC1CN2C(C1(c2ccccc2)CC1)=O C1(C(=O)NCC2CCCN(C(c3ccccn3)=O)C2)CC12CCC(F)(F)CC2 C1(OC)(CNC(=O)C(O)CNC(c2cc(C)ns2)=O)CCOC1 C1(CCOC)(NC(C(=O)NC(c2ccccc2)CSCC)=O)CCCC1 C(=O)(C(C)C(O)C(C)C)NCCN(CC(C)O)C(c1nc(C(C)C)oc1)=O CC1(C)CCC(CC(c2nnnn2C2(C)CC2)NCc2cc(C(C)(C)C)no2)C1 CCC(CC)C(C)C(=O)NCC1(C(N2CCCC3C(=O)NCC23)=O)CC=CC1 c1(C(N(C2CC(NC(CC3(CC)CCC3)=O)C2)C)=O)nc(C)oc1C N1(C(C(CC(C)C)C)=O)CCCN(C(C2(n3cc(Cl)cn3)CC2)=O)CC(CO)C1 c1(C(=O)NCC2(C(C)(C)O)CN(C(C3C(CC)CCC3)=O)C2)cccc(CO)n1 N(C1CCCc2sccc21)C(CCCCCO)c1n(CC(=C)C)nnn1 C1(C)(CC)CC1C(=O)NCC1CC(C(=O)NCC(C)(C)n2ccnc2)C1 CCC(CC(=O)NCC1CN(C(C2OCCC2(C)C)=O)CCO1)OC C1(OC)(CNC(C2CC(F)(CO)C2)=O)CCN(C(=O)CC2OCCC2(C)C)C1 C(=O)(C(C#N)C(C)C)NCC(c1ccccc1)N(C(c1[nH]cc(C)c1)=O)C c1(OCC)cnc(C(=O)NC(CNC(=O)CCOC2COC2)CC(C)C)cn1 c1(OC)nccnc1C(=O)NC1CC(C)(NC(C2CCCN2C(C)=O)=O)C1 C1(C(=O)OCc2coc(Cc3ccccc3)n2)CNC2(CC2)CO1 CC(C)CC(C(=O)Nc1cc(Cl)cnc1O)NC(=O)C(C)CC#N Cc1c(F)cc(C(=O)NC2CCCCN(C(=O)C=Cc3cscn3)C2)c(F)c1N Cc1ncsc1C=CC(=O)Nc1cccc(NC(=O)C(F)(F)c2cncs2)c1 C1(COC)CCC(C(=O)NCC(C(=O)NCC2(C)CCOC2)N(C)C)O1 N1(C(C(CC)C)=O)CC2(C(=O)NC3CC(n4cncn4)C3)CCC1CC2 N1(C(C(C)=NOCC#N)=O)CCCC(CC(=O)N(C(C)CO)C2CC2)CC1 C(=O)(C(C)(C)CC(=O)N1CC2CCCC2(NC(c2ccoc2C)=O)C1)OCC C#CC(C)(C)C(=O)N1CC2CC2(CNC(=O)COCC2CCCCO2)C1 c1(C2(C(=O)NC3C(NC(c4[nH]cc(C)c4)=O)C3)CC2)cc(F)cc(C#N)c1 c1(C(=O)NCC2(CNC(C(C(C)O)N(C)C)=O)CC2)cc2cc(O)ccc2[nH]1 c1(C(N2CC(CNC(C(C)(C)OCC)=O)C3C2C3)=O)nc(C)ccc1C C1(CC(=O)NCCC(CNC(CC=CCC)=O)O)CCC(C(=O)OCC)CC1 N1(C(COCCCC#C)=O)C(CNC(=O)C2=C(Cl)CCOC2)CC2CCCC12 c1(OC)ccc(C(=O)N(CCC(C)NC(C2CC23CCCC3)=O)C)c(O)c1F C1(C(N(CC(C)(C)CNC(=O)Cc2ccoc2)C)=O)CCCCS1(=O)=O CCN=c1ccc(C(=O)NCC(C)(C(C)C)NC(=O)CC2CC23CC3)c[nH]1 C1(NC(C2C(CC)OCC2)=O)CC12CCC(NC(=O)C=C1CCN(C)CC1)CC2 Cc1cc(C)c(C(=O)CCCC(=O)OCCc2cc(C)n(C)n2)c(C)c1 O=S(=O)(c1c[nH]ccc1=NC1CCC(F)C1)NC1CCN(c2cccc(Cl)c2)C1 N1(C(CC(C)C(=O)c2cccc(F)c2)=O)CC2CCC1CN2C(=O)C=CC1CC1 c1(C(=O)NCC2CCN(C(C3(CC#C)CCCO3)=O)C2)cc(C)c(C)c(C)c1 Cn1nc(CN2CCC(O)(c3ccccc3Br)C2)cc1C1CC1 [N-]=[N+]=NCC(C(=O)N1CCSC2(CC2)C1)NC(=O)C(O)C1CCCC1 CC1CC(CNC(c2ccn(-c3ccccc3)n2)=O)CN1C(=O)CSCCC#N c1(OC)ccccc1C(CNC(c1ncc(F)cn1)=O)NC(=O)Cc1ccon1 N1(Cc2ccc(OC)c(Br)c2)CCn2c(nc3c2CCCC3)C1 CCC1CC(=O)N1.C1(CCNC(=O)COC)(OCCOC2CC2)CCOCC1 C1(C(N2CC(O)(CCNC(COC3(C)CCC3)=O)C2)=O)CC(C2CCCC2)C1 c1(C(=O)OC)cnc(C(=O)NC(C)CCCNC(=O)C(C)n2ccnc2)cn1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(COC)(CNC(=O)C(C)CC(C)C)C1 c1(C(=O)NCCN(C(C(c2ccccc2)SC)=O)C)cc2cc(Cl)ccc2s1 C(=O)(C#CC1(C)CCCO1)N1C(C(=O)Nc2c(OC)n(C)nc2C)CC=CC1 C1(NC(c2cnc(C3CC3)s2)=O)COCCN(C(c2ccccc2Br)=O)C1 c1(C(=O)NCC2C(CNC(c3nncn3C3CC3)=O)C2)cn(CCO)nn1 C1(CC(=O)NCCCC2N(C(CCC(=O)OC)=O)CCCC2)CCCCC1(F)F c1(C(=O)NC(C(C)NC(c2csc(S)n2)=O)CO)ccc(Cl)c(Cl)c1 c1(C(=O)NC(c2nocc2C(=O)NCc2ccncn2)C)cccc2cncn12 C#Cc1ccc(NC(C2CN(C(C3(C#N)CCCCC3)=O)CCO2)=O)cc1 c1(SC)ccc(CN(C)C(N2CCOCC2C2CCC2)=O)cc1 C=C(C)CCCC(=O)NCc1nc(C2CCN(C(C3CC3(F)F)=O)CC2)n[nH]1 N1(C(c2c(C)nc(Cl)cc2)=O)CCC2(CCCN2C(=O)C(C)n2cccn2)CC1 CC(C)C(C)(CNC(C12CC(C)(C1)C2)=O)NC(=O)CCc1ccsc1Cl CC1CC(=O)NCCN1c1nnnn1C1CCC2CC2CC1 CN1CC(C(=O)NCCNC(=O)CN2CCOCC2=O)CC1=O c1(N(C)CCC2CC2)ccc(S(=O)(=O)NCC(O)CCC2CC2)c(Br)c1 C=C(CNC(=O)C(c1ccccc1)OC(C)C)CCNC(=O)CC1CSCCS1 c1(NC(=O)CCF)ccc(Cl)c(CNC(c2cnccc2N2CCOCC2)=O)c1 C=CC(C)(CCOC)C(=O)NC(C)CCCNC(C1(F)CCCN(C)C1)=O C1(CNC(c2c(CC)n[nH]c2)=O)CN(C(=O)C(=Cc2cccnc2)C)C(C)(C)C1 N1(C(C2C(=C)C2)=O)CC(F)CC1CN(C(=O)C(CC)=CCCC)C C=Cn1nccc1C(=O)N(C1CCC(O)C1O)Cc1c(OC)nsc1OC c1(-c2nccc(C(C3CCN(C)CC3)(C(C)C)C)c2)ccc(Cl)c(Cl)c1 C(=O)(CCCN=[N+]=[N-])NC(C=CC(=O)Nc1c(C)n(C)nc1)C C1(C(N2CCC(N(C(c3ccc(F)s3)=O)CC)C2)=O)CCCC(OC)C1 N1(S(CC)(=O)=O)CCC(C(N2CC(CNC(c3cn[nH]c3)=O)(OC)C2)=O)CC1 CCC(CC)CC(=O)NCC1CCC1C(=O)NC1(C(C)(F)F)CCC1 CCC(C(=O)NC(C1CCN(C(c2cnc3n2CCC3)=O)C1)(C)C)C(C)C C1(NC2(CNC(CCN(C)C3CC3)=O)CC2)C2CCCCC12.C12(CC1)N(C)C2=O C(CCNC(C1(C#N)CC1(C)C)=O)(C(=O)NCc1nn[nH]n1)OC CC(C)C(C)(CN=c1[nH]c(=NCCC(C)CO)[nH]c2cc(CO)ccc12)NC C(=O)(C(C)(C)CC(F)F)NC1C(C(=O)NCC(CSC)(C)C)CCC1 c1(OC)cccc(C(CNC(C)=O)NC(C2C3CCC2(c2ccncc2)C3)=O)c1 c1(C(N2CCC(CN(C(C(C(CC)CC)C)=O)C)C2)=O)cc2c(cc1Cl)OCO2 c1(C(N2CCCC2)=O)ccc2c(c1)CN(N1CCC([N+](=O)[O-])CC1)C2 O(NC(=O)CCCC(C)NC(C1CCOC1C(C)C)=O)CC(=C)C C1(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)CCCCC(C)(C)C1 N1(C(c2nc(CCC)sc2)=O)CC(C2CN(C(c3cccc(F)c3C)=O)C2)C1 CC(CC(=O)N(CCCCN(C(=O)CN1CC2C=CC1C2)C)C)CC(C)(C)C c1(C(N2CC(OCCNC(CC(C)CF)=O)C2)=O)cc(F)c(O)c(F)c1 c1(OC)n[nH]c(-c2nc(CC(C)OC)nn2-c2ccnn2C)c1Cl c1(C(N(CCCNC(CCN(CC)CC)=O)CC)=O)ccc(C)c(P(C)(C)=O)c1 c1(-c2occ(C)n2)cc(CN2CCCC(C(F)(F)F)(CO)C2)ccc1C C1(OC(=O)CN(C)C(c2ccc(C)cc2)=O)CC(O)CN(C(=O)OC(C)(C)C)C1 CC(C)CC(C)(C)C(=O)NCC1CCC(C(N2CCCCCC2C)=O)O1 O(NC(=O)CC(C1CC1)NC(=O)CNc1ncccn1)CCCC#C C12(CNC(CC(C)SC)=O)CC1CN(C(c1cnn(CC(C)C)c1)=O)C2 Cc1cc2c(C(=O)N=c3ccn(-c4ccc(F)cc4C#N)[nH]3)cccc2[nH]1 C1(NC(c2nc(C(=O)OC)sc2)=O)CC2CC(NC(=O)C(C)N(C)C)CC2C1 N1(C(C)=O)CC2CCN(C(C3CCN4CCC3C4)=O)CC12.C(=O)CCS(C)(=O)=O C1(=CC(=O)N(C(C2CCCCC2)CNC(=O)C(N)=O)C)CCCCC1 C1(O)(CCOC)CCN(C(=O)Cn2nc(C)nc2C)CC1 N1(C(CCC(C)N(C)C)=O)CCC2(CC(NC(c3ccsc3)=O)C2)C1 c1(C(N2CC3CC2CN3C(c2cccc3cncn23)=O)=O)ccc2ncsc2c1 N1(C(C#CCNC(C2(C)CC(=C)C2)=O)=O)CCC2(CCOC2=O)C1 C(CC(C(=O)NCC(O)CCO)NC(=O)C=CC1CCCC1)OCC c1(C(N(C2CCCCN(C(C(C=C)C)=O)C2)C)=O)cc(C)cc([N+](=O)[O-])c1 c1(NC(COC)=O)cccc(C(=O)NCc2ccc(CC(F)(F)F)cc2)c1O c1(OC)ccc2c(=NCCC3CC=CC3)[nH]c(=NCc3cccc(O)n3)[nH]c2c1 C1(CNC(c2ncccc2CO)=O)CC(O)CN1C(c1cnc(C2CC2)s1)=O N(C1CCc2c(C(F)(F)F)cccc21)C(C1C(CC)OCC1)=O c1(C(N2CCN(C(CS(CC)(=O)=O)=O)CC2CCO)=O)nccn2nccc12 C1(C(=O)NCCn2cc(C3(OC)CCOC3)nn2)CCS(=O)(=O)CC1 C1(CNC(c2cnc(C)nc2)=O)COC(C)(C)CN1C(C1CCCN(C)C1)=O C(=O)(C1=C(Cl)CC1)NC(CC)(C)CNC(=O)CCc1ncc[nH]1 N1(C(C2C=CCC2)=O)CCC2CCC(C1)N2C(c1ccc(O)cc1Cl)=O N1(C(C)=O)CCCC(C(N2CC(O)(CNC(C34CC(CCO3)C4)=O)C2)=O)C1.OC CC1CN(C(=O)Cc2cn[nH]c2)CC(C)CN1C(=O)C(C(F)(F)F)C(F)(F)F N1(C(Cc2cnc(C)s2)=O)C2CCC(C(N3CCCCC(CO)C3)=O)C1CC2 Cc1nc(=N)[nH]c(=NCC2CC(CNC(c3ccncn3)=O)CO2)[nH]1 N1(C(C2C(C)C2)=O)CCOC2(C1)CN(C(=O)CN1CCCC(C(F)(F)F)C1=O)C2 C1(NC(c2sccc2C2CC2)=O)CC2CC(C1)CN(C(C1(CO)CCCO1)=O)C2 C1(OC)CC(C)CN(C(C2CCCN(C(=O)CC3CCC(=O)C3)C2)=O)C1 N1(C(C(c2cn(C)nn2)OC(c2c(C(=O)NC)ccs2)=O)=O)CCC(C)C(CO)C1 CC1(C(=O)NCc2ccc(C(=O)N(CC3CC3)CC3CC3)cn2)CCC(O)CC1 C1(C(N2C(CC(N3CC=C(C)CC3)=O)CC(F)C2)=O)CC12CCCCC2 Cc1nn(-c2cccc(F)c2)cc1C(=O)NCC1(NC(C2CC23CC(O)C3)=O)CC1 c1(C(C(=O)NCCC2(CO)CCC2)NC(=O)Cn2ccnn2)cccnc1 C(N=c1[nH]c(=NCC(CC)(CC)CCO)[nH]c2c1COCC2)c1c(CC)c[nH]n1 Cc1ncsc1C=CC(N1CCCCC1CCCNC(C12CC(F)C1C2)=O)=O O(N(C)C(=O)CCN(C(c1cc(Cl)cn1C)=O)C1CC1)CC(=O)OC N12CCC(CC1C(=O)O)C2.c1(C(=O)OC)ccc(-c2ccc(C(F)(F)F)s2)cc1 CN1CC=C(CC(=O)NC2CCC(C(N3CCC4NCCC4C3)=O)CC2)CC1 c1(C(N(C2CCCN(C(CN(C)CC)=O)CC2)C)=O)cnn2c(=N)[nH]cnc12 N1(C(CCOCC)=O)CCN(C(=O)CNC(C2CCC2)=O)CC1c1ccccc1 C1(CNC(C(CC)OC)=O)CC2(CCC2)CN1C(=O)Cc1cn2c(C)csc2n1 N1(C(CNC(C)=O)=O)CC2(C1)CN(C(C1CN(C3COC3)C1)=O)CCO2 C1(NC(Cc2ncn(C)c2)=O)CN(C(=O)CC2=CCCC2)CC2(CC2)C1 C=CC(C)(C)CC(=O)NC1CCN(C(c2ccc(CN(C)C)nc2)=O)C1(C)C N1(C(C=C(CC)CC)=O)CCc2[nH]nc(CNC(c3ccncc3Br)=O)c2C1 c1(-c2cc(C(=O)NC(CCC)CCC)c(F)nc2)cc([N+](=O)[O-])ccc1F Cc1cc(C(N2CC3(C2)CN(C(C2Cc4nccn4C2)=O)C3)=O)ccc1C#N n1(CC)cc(CC(=O)N(C(=O)CCc2cocc2Br)CC2(O)CC2)cn1 c1(C(=O)NCC(C)NC(c2cc3cc(F)ccc3[nH]2)=O)n[nH]c2c1CN(C)CC2 CCCC(C)C(=O)N1CCC(C(=O)Nc2ccccc2C(C)(C)C)C1 c1(C(=O)NC2CCCN(C(C3CCN(C)CC3)=O)CC2)ccc2nccnc2c1 C1(c2ccccc2)(C(N2CC(N(C(=O)CC3(C(F)(F)F)CC3)C)C2)=O)CCCC1 C1(C(=O)NC2CCC(C(=O)NC3C(C)(C(F)F)C3)CC2)CC12CCOCC2 N1(C(CC(=O)OC)=O)CC(CNC(=O)C(C)CN2CCCCC2)OC(C)(C)C1 Cn1nnc(C(=O)NC2CCN(C(C3CC(O)(c4ccccc4)C3)=O)C2)n1 c1(NC(C2CCC(NC(c3c(Br)cnc(C)n3)=O)C2)=O)ccc2nn[nH]c2c1 C1(O)(C(=O)NCC2C(NC(c3cnc(CC)s3)=O)CCC2)CCCC(C)(C)C1 CC1(CNC(=O)CC2(NC(c3ccncc3F)=O)CCC2)CCC(=O)N1 c1(C(=O)NC2(C)CC(NC(COC(CC)C)=O)C2)cccc(C)n1 N1(C(=O)NCCCOC(C)(C)C)CC(F)(F)C1C1CC1 c1(OC)ncc(Cl)c(=NCC2CC(NC(c3cccc4cnccc34)=O)C2)[nH]1 C(=O)(CCCC(F)(F)C(F)(F)F)N(CCCNC(c1c(C)con1)=O)C CCC(CC(=O)N1CCC(C(C)(C)C(=O)NCC(Cl)=CCl)C1)C(C)(C)C CC1(NC(=O)C(C)(C)NC(C23CC2CNC3=O)=O)CCC(=O)NC1=O C(CCC(C)C)(C(=O)NC1CCN(C(c2cnc(N)c(N)c2)=O)C1C)NC(C)=O C(N=c1nc2c(cnn2C)c(NCc2cnc[nH]2)[nH]1)c1c(CC)con1 N1(C(c2nccc(CC)c2)=O)CCC2CN(C(=O)CSCCC(C)C)CC12 n1(C(C)C(=O)NCCC2CC2(Cl)Cl)cc(C2(C)CCCO2)nn1 N1(C(COCC(=C)C)=O)CCCCC(NC(c2ccnn2C(C)CC)=O)C1 CCCC(C(=O)N1CCCC(CCNC(C2(CO)CCOCC2)=O)C1)S(N)(=O)=O N1(C(C(CC(=C)C)C)=O)CCCCC(C2CN(C(c3cncc(Cl)c3Cl)=O)C2)C1 c1(C(=O)NC2C3CN(C(C(C)(F)F)=O)C2C3)cnc2c(n1)CCCC2 N1(C(CC2CCC(C)CO2)=O)CCC2(CC2)CC1C(=O)NCc1cc(CO)on1 C1(NC(c2c(CSC)cccc2)=O)CC2(CCN(C(=O)CC(=O)NC3CC3)C2)C1 N1(C(C(CC)F)=O)CCN(C)CC1CNC(c1sc(-c2ccc(C)o2)nc1C)=O c1(C(=O)NC(C)CCCNC(=O)CC#N)ccc(-c2ccccc2)cc1F C1(NC(CCC(C)NC(Cc2c(C)ocn2)=O)=O)CC12CCCCCC2 CC1CCN(C(c2cccnc2O)=O)CC1CC(N1CCC(C(N)=O)CC1)=O c1(CC)ccc(NC)cc1.O1NC(=O)CN(C)C(=O)C1 C12(NC(=O)C3=COCC3)CC(C(C)NC(=O)C(O)Cn3cncn3)(CO1)C2 n1(CC)ncc(C(=O)NC2CCC(CNC(=O)CCC(C)SC)CC2)c1C C=CCN(OC)C(=O)c1cn(CCN(C(=O)C(CCC)OCC)CC)nn1 C(CC(C)C)(C(N)=O)NC(CC(CC)NC(c1sccc1C#N)=O)=O c1(C(=O)NCC(CN(C(c2c(C)cccc2O)=O)C)C)cc2c(C)sc(C)c2s1 C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CC(NC(c3cc(C)c(C#N)cn3)=O)C2)C1 C1(NC(C2C(C)OCC2)=O)CN(C(c2cnn3cccnc23)=O)C2CCCC12 N1(C(CC2CCN(C(C3CC(O)(CC#C)C3)=O)C2)=O)CCC=CC1COC C1(C(C)(C)O)CC(NC(=O)C(c2ccc(-c3ccccc3)cc2)(C)C)CCN1 N1(CCNS(CC2(C)CCNC2=O)(=O)=O)CCCOC(c2ccc(C)cc2)C1 Cc1cc(C(=O)NC2CC(C)CN(C(=O)C(C)NC=O)C2)cc(O)n1 C1(C(=O)NC(C(=O)OC)C(C)O)CCCN(C(c2cc(C3CC3)on2)=O)CC1 C=CCN=c1[nH]cc(C(=O)NC(CN(C(=O)Cn2ccc(C)cc2=O)C)CC)s1 CC1=C(C(=O)NC2CCC(NC(c3cncc(C(F)F)c3)=O)C2)CCO1 C(=O)(C1=CCC2(COC2)OC1)NC(C(C)NC(=O)Cn1ccc(C(F)(F)F)n1)C N1(C(C(CSC)O)=O)CC2CC3CC2C1C3NC(C1Cc2cc(C)ccc2S1)=O N1(C(C(C)n2ccnc2)=O)CCC(CNC(=O)COCCOCCO)C(O)C1 CC1CN(C(=O)CC2(N(C)C(c3ncc(F)cc3N)=O)CC2)CC(CO)O1 c1(OC)c(F)ccc(C(N2CC3CN(c4ncc(C)c(C)n4)CC3C2)=O)c1F N1(c2n(C)c(=O)n(C)c(=O)c2)CCC2CCC(C1)N2C(C1CC1(C)Br)=O c1(C(=O)OC)cc(NC(c2ccc(C#N)c(O)c2)=O)cc(OC)c1OC C1(CC)C(=O)NCCCN1C(C1CC(C)CN(C(c2cccc(Cl)c2)=O)C1)=O Cc1ccc2ncc(C(=O)NC3CCC(NC(=O)CC45CCCC4C5)C3)n2c1 C(=O)(CC(C(=O)NCCC(C)CCNC(c1cncc(C)c1)=O)NC(C)=O)OC c1(SC)ccc(C(=O)NC(C)CCNC(=O)C(C)(C)c2ccsc2)s1 C(c1ccc(F)cc1)=CC(=O)NC1CCC(NC(=O)CC23CCCC2C3)C1 N1(C(CCN(C)CCO)=O)CCC(C2CC2)C1C(=O)NC1CC2(CCOC2)C1 C1(CNC(c2ccc(COC)o2)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1(F)F C(N=c1cc[nH]cc1[N+](=O)[O-])C1CN(C(Cc2c(C)non2)=O)CC12CCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CCCN(C(C2CCN(C3CC3)C2=O)=O)CC1 c1(OCC)ccncc1C(=O)N(c1ccccc1)CC(F)F CC(O)C(C)(C)C(=O)N1CC(n2cc(-c3ccc(Cl)cn3)nn2)C1 CCCC(CC(=O)NCC(C)NC(c1cccc(F)c1C)=O)NC(=O)OC(C)(C)C c1(C(N(C2CC(C#N)C2)CC(=O)NC(c2ncc[nH]2)CC)=O)ccc(Cl)o1 C1(C(=O)NC(C)CCCNC(=O)C(C)(C)O)CCC2CCCCC2C1 c1(Cc2nn(-c3cccc(OC)c3)c(CCCF)n2)coc2c(C)c(Cl)ccc12 C1(CNC(C(C)(C)SC)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 N1(Cc2cccc(C#N)n2)CCC2(CC(C(=O)N=c3cncc(Br)[nH]3)=NO2)C1 N1(C(C=COCC)=O)CCC(c2ccccc2)(NC(=O)C(C)SCC)C1 C(=O)(C1CCNc2ccccc21)c1onc(-c2c(C)cc(F)cc2Cl)n1 O=C1CN(CC(N2CCC3CC23CC(=O)NOCCOCCO)=O)C(=O)N1 C1(c2cn(CCC=C)nn2)CN(C(C2CC=CCO2)=O)CCO1 C(=O)(C(C)(C)N(C)C)N(CCC(=O)NCCC1CCNC1=O)C C(=O)(CCC(C)NC(c1ncn(C)n1)=O)NCc1ncc(C)o1 C=CCC(C)(C)C(=O)NCc1occc1C(=O)NCc1nocc1C(C)C C1(N(C)C(c2csc(C3CC3)n2)=O)CN(C(C23CC(F)(C2)C3)=O)CC12CC2 N1(C(C(CC)C)=O)CCCC2(CCCN2C(c2n[nH]c3c2CCC3)=O)C1 C1(C(=O)NC(C#C)C2CC2)(CNC(=O)Cn2nnc(C)n2)CCCO1 CC1(C)CC(=O)N(CC(=O)NC2CN(C(C3CC4CCC4C3)=O)CC2C(F)F)O1 C1(NC(CC2(C)CC2(F)Cl)=O)CCC(NC(=O)C=CCOC2CCOCC2)CC1 C1(C)(NC(C(CCC)NC(=O)C(C(C)C)SCC)=O)CC(F)(F)C1(C)C c1(C(=O)NCC2(C)CCCN(C(C3(CC)COC3)=O)C2)cc2c(=O)[nH]ccn2n1 N1(C(C2CC=C(C)CC2)=O)C2CCC1C(NC(c1cc(C)[nH]n1)=O)C2 c1(CC(N2CC3(CN(C(=O)CCc4cnn[nH]4)C3)C2)=O)cncc2ccccc12 C1(CC(=O)N(CC(N2CC(CCC)C2)=O)C2CC2)CC2CCC1C2 c1(C(N(C)CC2CCN(C(=O)C=CCF)CC2)=O)cccn2ncnc12 C1(CC)CN(C(c2cc(C)c[nH]2)=O)CCC1NC(C12CC3CC1C2C3)=O N1(C(c2c(COC)nn(C)c2)=O)CCOCC(C(=O)NC(CO)C(C)(C)C)C1 N1(C(c2ccc(N)cn2)=O)CCC(NC(=O)CC2CC(O)C23CCC3)C(O)C1 c1(C(N(C)CC2CCN(C(c3c(C)nc(CC)o3)=O)C2)=O)cc(F)cc(Cl)c1N O=C(C#CC1CCCCO1)N1CCC(F)CC1c1ccco1 CCCC(C(=O)NCC(CC)N(C(c1ccn(CCC)n1)=O)CC)C(C)C N1(C(COCCOC)=O)CC(C(=O)NC(C2CCCO2)(C)C)C(C(C)C)C1 C1(NC(C(C)=C(CC)C)=O)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1C C(CCO)(C(F)F)N(C(CNC(CN1C(C)CCC1)=O)=O)C C1(C(C)NC2CCOC2)CCCN(C(=O)CN2CCOCC2)C1 N1(C(C2(OCC)CC2)=O)CC2C(CN(C(=O)CC3COCCN3C)C)C2C1 N1(C(CCSCC)=O)CC(NC(C2CCCCCN2C)=O)CC1(C)C C12(C(=O)NC3CC(OCC(=O)N(CCC(O)CO)C)C3)CC(CO)(C1)C2 C(CN=c1[nH]c(=NCCc2nc(-c3cccs3)n[nH]2)[nH]c2ccsc12)SC(C)C N1(C(=O)C(=O)NCCOC2CCOC2)CCC(c2cccnc2)C1 c1(C(=O)NC2CCC(NC(COCC#C)=O)C2)c[nH]ccc1=NC(=O)C(C)(C)C C1(N(C(=O)Cn2cccn2)C)CCCC(NC(c2cscc2F)=O)C1 c1(OCc2cn(C(C)CNC(=O)Cc3cc(Cl)cs3)nn2)ncc(C#N)cc1Cl Cc1ccc(C=CC(N2CCC(F)(CNC(=O)CCc3ccc(CO)cc3)C2)=O)s1 C1(C)(CC)CCC(C(=O)NC2CC2CNC(=O)CCc2cn[nH]c2)O1 c1(OC)ccc(Br)c2c1C(NCC1CCNC3(CCC3)C1)CC2 C(=O)(C(C)CS(C)=O)N(CCCNC=O)C.c1(C(=O)OC)ccc(N2CCC2)nc1 Cc1cc(C(=O)NC(CNC(=O)Cn2nccc2C)C(C)C(C)C)cc(C)c1Cl CC(C)CCC(=O)O.C1(CC(=O)NC)CCOC1=O.C1C(=O)N1.C1C(=O)N1 c1(C(N(CCNC(C(C(C)C)SCC)=O)C)=O)cc(F)cc2cnccc12 O(NC(=O)C(CCC(C)C)NC(=O)C(C)NC(N)=O)C(CC)CC c1(OC)ccc(C(CNC(=O)NC(C(F)(F)F)C2CC2(C)C)N(C)C)cc1 C=CCC(C(=O)OC)NC(=O)Cn1cc(-c2cccc(SC(F)(F)F)c2)nn1 C=CC1(C(=O)NCc2cnns2)CCN(C(=O)CC(C)C(F)F)C1 N1(C(C(COC)N(C)C)=O)CCN(C(=O)Cc2ccsc2C)C(CCOC)C1 N1(C(C(CCC)CNC(C2CC2Cl)=O)=O)CCC2(CC(CO)C2)C1 Cc1cc(=NC(=O)C(C(C)NC(=O)C(c2cnn(C)c2)C)C(C)C)[nH]n1C1CC1 C(CCO)(C(C)(C)C)NC(CCN(C)C(c1cnc[nH]c1=N)=O)=O N1(C(C(C)(C)CO)=O)CC2CN(C(C3(S(C)(=O)=O)CCCC3)=O)CC2(C)C1 CC1CN(C(c2ccccc2CO)C(=O)NCCCC2CC2)CC1(C)C(N)=O c1(C(=O)NC(CNC(CC2CC(C)OC2C)=O)C)c2c(nn1C)CCOC2 N1(C(C(COCC)N=[N+]=[N-])=O)CCCC(C2CN(C(c3cc(=O)cc[nH]3)=O)C2)C1 Cc1nc2c(s1)CCCC2C(=O)NCC1CC(F)(NC(=O)CCCS(C)(=O)=O)C1 c1(CC(=O)N(C(CCNC(C(C)OCCC#C)=O)C)C)cc(C)n(C)n1 n1(C2(C(CCCC)=O)CC2)cc(CN2CCOCC2)nn1.C1COO1.C1(CC)CC1.O.C C1(NC(c2c(F)cc(OC)c(F)c2)=O)CC12CCN(C(C1CCCC1)=O)CC2 CCCC(CCC)C(=O)N(CCNC(C1CCCC1C1CC1)=O)CCOC c1(C(=O)NCCCN(C(C(C)OCC#C)=O)Cc2ccccc2)cc(O)ncn1 C#Cc1ccc(F)c(C(=O)NCCC(CC)(CC)NC(=O)CC2CCOCC2)c1 c1(CC(N2CCC(C(C)NC(=O)C(C)C3CC3)C2)=O)c(F)cccc1F C1(C(=O)NCC(CCCC)NC(C=COCC)=O)CCOC(=O)CC1 C(CC(F)CN=[N+]=[N-])NC(C(C1(O)CN(C(c2cn(C)nc2)=O)C1)F)=O C12(C(=O)NC(CC=C)C3CC3)CC1CN(C(=O)CC1CCCCN1C)C2 c1(C(N2CCC(C)(CNC(C(C)N(C)C)=O)C2)=O)c(C(F)(F)F)cccc1Cl C1(NC(CN(CCC#C)C)=O)CCCN(C(c2cccc(N)n2)=O)C1C C(C)(C(=O)NC1CCOC(C(=O)NC2CC(O)C2O)C1)(C(C)C)OC C#CCCCCCCC(=O)N1CC2CC1(c1cn(-c3ccccc3SC)nn1)CO2 Cc1ccc(C(N2CC(NCc3cc(C)n(C)c3)CC(C)C2)=O)cc1C(F)(F)F c1(SC)ccc(Cl)c(C(=O)NC2CCN(C(=O)Cc3ccc[nH]3)CC2C(C)C)c1 c1(C(C(=O)NC2CN(C(c3cc(C)cc(F)c3)=O)C2)C)cn(C)c2ccccc12 N1(C(c2c(CC)ccc(F)c2)=O)CCC2(NC(=O)Cc3cccnc3)CCCC12 C1(NC(=O)NCc2nc(COC)sc2)(COc2ccccc2)CCCC1C1CC1 C1(C(=O)NC(CCNC(C2CCC(CCC(C)C)CC2)=O)C)CC(C)CC(=O)N1 c1(C(N2CCCCC(NC(CN(C)C)=O)C2)=O)cc([N+](=O)[O-])c(Br)cc1F C1(N(C(=O)Cn2cccn2)C)CN(Cc2sccc2OC(F)F)CCC1O C1(C(N(C)CC2CN(C(c3ccc(C)o3)=O)C2)=O)CCC(=O)NC1 Cc1nc(C(=O)NCC2CN(C(=O)Cc3sccc3C)CC2C)ccc1[N+](=O)[O-] CN1CC(C(=O)NC2(CCNC(c3nc[nH]c3C(F)(F)F)=O)CCCC2)NC1=O c1(C(=O)NCC2C(NC(C(n3ccc(C)n3)C)=O)C2)cc(Br)c(C)cn1 C(CCCC(=O)NCC(C(=O)N1CCC(CO)C1)N(C)C)SC c1(C(=O)NC2C3CN(C(c4c(N(C)C)ccnc4)=O)CC32)ccc(F)c(F)c1F C12(C(=O)NC(C(C)F)C)CCCC1CCN2C(=O)C(c1cnn(C)c1)C C1(NC(C2COCCOC2)=O)COC2(C1)CN(C(c1cnc3nccn3c1)=O)C2 C=CC(CC)C(=O)NC(C(=O)NCC1(OC)CCC1)c1ccco1 N1(C(c2noc(CSC)n2)=O)CCC2(NC(=O)Cc3cnn(C)n3)CCCC12 N1(CC)CC(NC(=O)C(CC2CCC2)NC(=O)C=CC2CCCC2)CC1=O c1(C(C(=O)NC(C2(O)CN(C(C3(O)CC(C)(C)C3)=O)C2)C)CO)ccc(F)cc1 C1(C(=O)O)CCC(C(=O)NC(c2cccc(Cl)c2)CF)CC1 c1(C(=O)NC2C(NC(COC)=O)CCCC2)ccc(C)c(OCC(C)C)c1 C1(C(N(CC(C)NC(c2c(C(=O)OC)n(C)nc2)=O)C)=O)CN2CCC1(C)CC2 N1(C(C(C(C)C)SC)=O)CCC2C(C1)CN2C(=O)CC(C)(C)CN1CCOCC1 c1(CC(C(=O)NCC(C)NC(CC(=C)C)=O)C)ccccc1Cl Cn1cc2c(n1)CCCN(C(C1C3CN(C(=O)C(C)(C)n4cccc4)CC13)=O)C2 Cc1coc(C(=O)NC2CCC(CNC(=O)C(F)(F)c3nccs3)C2)c1 N1(C(C(=O)N(C)C)=O)CCC(NC(c2nc(Cl)sc2Cl)=O)C(CO)CC1 C=C(C)CCCC(=O)NCCC1CN(C(=O)C(C(=O)OCC)OC)CCO1 C1(C(=O)CC2(c3ccccc3Br)CC2)CNC(C2CC2)CO1 Cc1cc2cc(C(=O)NCC3CN(C(=O)C(C)(F)C(F)(F)F)C3)[nH]c2cc1Cl C1(CC(=O)NC2C(N(C)C)COC2)CCOC1(C)C S(=O)(=O)(c1ccsc1C(N1CCC(NC(=O)C=Cc2cncs2)C(O)C1)=O)NC Cc1ccccc1C(=O)NCC(=O)NCC(F)CNC(c1sccc1Cl)=O c1(C(N2CC(OC)C(NC(c3cnnc(C)c3)=O)C2)=O)cccn(C)c1=O c1(NC(C(CNC(C2CC(COC)C2)=O)C)=O)c(C)[nH]c(C)cc1=O N1(C(C=C(C)Cl)=O)CCC2CC(NC(c3cnc4nccn4c3)=O)CCC2C1 c1(C(=O)NC(CNC(c2ccc(C)o2)=O)C)cnc2c(c1)c(C)nn2C S(=O)(=O)(c1ccc(F)c(Br)c1)N1CCN(C2CCN(C(=O)C(F)F)C2)CC1 C1(NC(CCC2N(C(C=CC(CC)C)=O)CCC2)=O)COC2(CCCC2)C1 N1(C(COCC=C)=O)C(C(=O)N(C(C)C(C)(C)O)C)C2CC(O)C1C2 C1(CC)C(C(=O)NCCCC(C)(C)OC)CCN1C(c1ccccc1NC)=O c1(NC2C(C)C(c3ccccc3)C2)ccc(Cl)c(C2=CCNCC2)c1 c1(C(N2C(C(C)NC(c3cnc(O)o3)=O)CCCC2)=O)cccc2oc(O)nc12 N1(C(c2c(C)nco2)=O)CCCC(N(C)C(c2cc(F)c(N)cc2F)=O)CC1 N1(C(c2c(C)cccn2)=O)CC2CCC(CNC(C3CC3Cl)=O)C2C1 C1(n2cc(C(C(C)(C)C)O)nn2)(CNC(C2CCC(F)(F)C2)=O)CCCCC1 c1(C(=O)NC2CC(N(C)C(c3nccnc3C(N)=O)=O)C2)ccnc2c1CCO2 Cc1[nH]nc2cc(C(N3CCN(C(=O)CC(C)CF)CCC3C)=O)ccc12 c1(C(=O)NC2CCCN(C(C3CC34CC4)=O)CC2)c[nH]c2cc(O)ccc12 C1(NC(=O)CC2COCCOC2)CC(NC(=O)Cc2ccsn2)C12CCC2 CCC(CC(C)C)C(=O)NC(CNC(c1sc2ccsc2c1C)=O)CO C1(NC(C2CCN(C(C)C)CC2)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)C1(C)C C1(S(C)(=O)=O)(C(=O)NCC2(NC(CCC(C)(F)F)=O)CCOC2)COC(=O)C1 c1(C(=O)NNC(=O)C23COC(C2)C3)cccc(S(=O)(=O)C(F)(F)F)c1 c1(CC(=O)NCCCCCCNC(CCS(=O)(=O)NC)=O)ccc(C)c(F)c1F Cc1nn(CC(=O)NC(C(C)NC(C2(O)CCC2)=O)C(C)C)c(C)c1[N+](=O)[O-] CC(C)(C)C(CNC(=O)CCC(F)(F)F)C(=O)NC1CCC2CCC12 c1(OC)cccc2c1CCCC2NC(=O)C(C)(C)c1ccns1 C1(NC(C(Br)=C(C)C)=O)CN(C(=O)CCC(C)C#N)CCC12CCC2 CCCCCS(=O)(=O)CC(=O)NCC(C)CN(C(=O)CC12CC(C1)C2)C C(C(F)(C(=O)NCCCC(=O)NC1CC1)C(C)C)NC(c1c(CC)cccc1)=O CC(C)C(C(=O)NC(C)CN(C(=O)Cc1n[nH]c(=N)s1)C)c1ccncc1 c1(OC)ccc(NCC2(C)CCC(C(=O)OC(C)(C)C)C2)cc1N1CCOCC1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(C2CN(C(c3c[nH]c(=N)o3)=O)C2)C1 CN1C2CCC1CN(C(=O)C(CO)NC(c1ccncc1N)=O)CC2 Cc1cc(C(C)(C)C)ccc1C(=O)NCCN(C(C1CC1(F)Cl)=O)C(C)C c1(OC)cnncc1C(=O)NC(C1CCN(C(C2CCC(=O)N2)=O)C1)(C)C CC1CCC(NC(c2cnc(-c3ccccc3)[nH]2)=O)CN1C(=O)CNS(N)(=O)=O c1(CNC(C=C2C(C)(C)CCCC2)=O)c(F)ccc(N)c1F CCCC(C)CCCC(=O)NCCCNC(=O)C(c1cccnc1)O C(=O)(CCCCCF)N1CCC(C(C)NC(CCc2cccc(OCC)n2)=O)C1 C(CCC(C(=O)N(C1COCC1OC)C)NC(c1scnc1Cl)=O)OC C(Cn1cncn1)(C(=O)NCCC1COCCO1)NC(CCOC(C)=O)=O CCCC(CC(C)C)C(=O)N(CC(C)NC(=O)CN(CC)CC)CC N1(C(c2c(C(C)C)ccs2)=O)CCC2CCN(C(C3CC(=O)N3)=O)CC2C1 C(CCCCCCO)NC(C(C1CCCN(C(=O)C=CC(=O)N(C)C)C1)C)=O Cc1cc(NC(=O)CSCCC(C)C)ccc1NC(C1CCCC(C)O1)=O N1(C(c2cnn(C)c2N)=O)CC2CCN(C(=O)CC3CC4(CCC4)C3)C2C1 c1(OC)c(NC(C2CC(C)CN2C(c2nc(C(C)C)cs2)=O)=O)c(C)nn1C Cc1cccc(C(=O)NC2(CCNC(=O)C(F)C(C)(C)O)CCCC2)c1C C(C(C)(C)C#CC(=O)NCCC1COC(C)(C)C1)NC(C(C)S(C)(=O)=O)=O c1(CC(=O)N(C(CNC(C2(C(=O)OCC)CCC2)=O)C)C)cscc1Br C(=O)(C(C)(C)n1cc(Cl)cn1)NCC(C)(C)OCC(=O)N(C)CC1CCCO1 N1(C(c2n(CC#C)cnn2)=O)CCN(C(c2scnc2Cl)=O)C(CC)C1 C1(C(=O)OC)CC(C(=O)OC)CC(C(N2CCC(CCF)CC2)=O)C1 Cc1cc(C(=O)NCC2CCCC(NC(=O)COCc3scnc3C)C2)n(C)n1 C1(C(N2CCC(C)(CC)CC2)=O)CCC(C)(C)N(C(=O)Cc2nc(=N)[nH][nH]2)C1 C(CC(C)C)(C(=O)N(C1CN(C(C)C)C1)C)ONC(c1cc(CC)[nH]n1)=O c1(NC(C2(C(C)C)CCNC2=O)=O)cc(Cl)cc2c1OCC(=O)N2 CN1CCOC(C(=O)NC23CC(NC(C4CCCC(C(=O)N(C)C)C4)=O)(C2)C3)C1 CCC(O)C(C)C(=O)N1CCC(C(C)(C)NC(c2cnn(C(C)(C)C)c2)=O)C1 C1(C(=O)NCCOCCOC)CCCC(NC(c2nccn2C2CC2)=O)CC1 C(C1CCCCCC1)=CC(N1C(CO)CC(NC(Cc2c(C)noc2)=O)C1)=O C1(NC(c2cncc(CNC(=O)Cc3cnccn3)c2)=O)CCCCC1(F)F C1(CNC(C2N(CC)CC2)=O)CC2(CO1)CN(C(=O)CCC1CCC(=O)C1)C2 c1(OC)ccc(C=CC(=O)NC2(CN(C(=O)CC3CCC(C)CC3)C)CC2)cc1 c1(C(=O)NCC(CC=C)NC(=O)CC2COCCN2C)cc2c(C)nn(C)c2s1 C1(CNC(COCCCCC)=O)COC(C)(C)CN1C(c1cccc(C)c1)=O C12CN(CCC1C)C(=O)C2.C1(CCC)(CC)CCCN1C(=O)CCC1CC1 Cc1ccc(C(=O)NCC2CN(C(=O)CC(c3cccc(F)c3)O)CCO2)nc1 C1(NC(Cc2c(C)n[nH]c2C)=O)CC2CC(C1)N(C(=O)Cc1cncnc1O)C2 c1(CC(=O)NC(c2nn[nH]n2)C2CC2)ccccc1OCCCC#N CC(C)C(O)CC(=O)NCC(F)CNC(c1cc(-c2ccncc2)no1)=O C=CC(CC)CC(=O)N1CCCC(CNC(c2coc(-c3cn[nH]c3)c2)=O)C1 C1(C)(C(=O)NCC2N(c3ncc(OC(C)C)cn3)CCC2C)CCCCCC1 c1(C(N(CC(N2CCN(CC(C)C)CC2)=O)C)=O)cc2cccnc2o1 c1(C(N2C(C)CC(NC(=O)Cn3nccn3)C2)=O)cc(=O)c2ccc(O)cc2o1 N1(C(=O)NC(C)CN2CCCN(C)CC2)CCNc2cc(Br)ccc2C1 C1(NCCNC(Cn2cnc(C(=O)OC)n2)=O)CCCSC1 C1(C(N(CCCCCNC(C(CSC)OC)=O)C)=O)CC2(C)CC1CO2 C1(CNC(C2CC(CC)C2)=O)C2CN(C(=O)CN(C3CCC3)C)CC12 N1(C(C(C)Oc2ccc(C)cc2Br)=O)CCCC2CCCCC12 N1(C(C(CSC)O)=O)CCC2(CC1)CCN(C(C1CCC3(CCOCC3)C1)=O)C2 c1(C(N2CC(F)(CNC(CC(C)C(C)(C)C)=O)C2)=O)cc2c(F)c(F)ccc2[nH]1 c1(C2(COC)CC2)ccc(C(N)=O)nc1.C1(CCN)(NC(=O)C=CC)CCC1 CC(O)(C(=O)N1CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C(F)C1)C(F)(F)F C(=O)(C1=CCc2ccccc21)NCCC(CCNC(CC(=O)OCC)=O)C c1(CC(=O)NC2CC(C(C)NC(=O)CCC3CCCOC3)C2)cc(C)nn1C c1(C(=O)NCC2(F)CCN(C(c3ncc(OC)nc3)=O)C2)ccc2c(c1)CCC2 c1(C(=O)NC2C3(CC(NC(CCNC(=O)NC)=O)C3)C2)cccc(C)c1C C1(CNC(c2ccc(C(F)(F)F)[nH]2)=O)CC(O)CN1C(C1CCC(F)(F)C1)=O C(=O)(C(C)(C)C(=O)NCC(CC(F)(F)F)NC(=O)C=Cc1ccc(F)cc1)NC C1(c2n(C)ccc2)CN(C)CCN1C(c1ccc(C2CC(C)(C)OC2=O)cc1)=O C#CCCCC(C)C(=O)NC1(CC=C)CN(C(c2cc[nH]c2)=O)C1 c12cccc(c1)CNC2=O.C1(C(=O)NCC(C)(C)OCCO)OC2CCC1C2 c1(C(=O)NC(C)C)nnc(N2CCOC3CC23)n1Cc1cccc(Cl)c1 c1(C(=O)Nc2ccc(-n3c(C)ccn3)cc2)cc2cccc(C)c2s1 C1(CCNC(CCCOC)=O)C(C)CCCN1C(C1CCCCC1)=O N1(C(C(CO)OC)=O)CCCN(CCNC(=O)C(F)CC2CCCC2)CC1 N1(C(=O)CC(F)(F)C(=O)O)CC2CCN(C(c3cscn3)=O)CC2C1 C1(CNC(CSCCC)=O)CC2(CCC2)CN1C(c1sccc1C)=O C(C)(C(C)(C)C(=O)NC1(c2cccs2)CC1)NC(C(CO)OC)=O CN1CC(C(=O)NC2CN(C(=O)C=Cc3ccc(=N)[nH]c3)CC23CC3)CCC1=O N1(C(c2c(C)cc(F)s2)=O)CCC2CC(NC(c3csnn3)=O)CCC2C1 c1(CN2C(CC(C)C)CCCC2=O)cc(=O)[nH]c2ccccc12 C1(CNC(C(C)OC(C)C)=O)CCC2(C1)OCCO2 N1(C(c2c(CC)n[nH]c2)C(=O)NC2(C)CC2)CC2CC3CC2C1C3C(=O)OC c1(Cc2occc2)ccc(F)c(-c2ccc(C)cc2)c1.n12nnnc1C2.C1CCC1 CCCC(C)(CCC)C(=O)NCC1C=CC(NC(=O)Cn2ccnc2C(C)C)C1 N12CCCC(C)(C1)C2.N1(C(=O)OC(C)(C)C)CCC2CC12C(F)(F)F c1(NC)c(C(=O)NCCN(C)C(c2c[nH]cc2C(C)C)=O)cccc1F C1(C(=O)NC(C)CCN(C(=O)CCc2ncco2)C)OCCN(C)C1=O c1(C(=O)NCC2(C(=O)Nc3c(C)cc(Br)cc3Cl)CC2)ccc2nc(O)oc2c1 c1(NC(C2C(NC(c3c(O)ccc(C)c3)=O)C2)=O)cc(Cl)c(Cl)cc1[N+](=O)[O-] C12(NC(=O)COC(F)F)CCCC1N(C(=O)C(c1cc(F)c(F)cc1F)O)CC2 Cc1cc(CC(=O)NCC2CCN(C(c3ccccc3)C)CC2)n(C)n1 CC(N=c1nc2scnc2c(NCCOc2ccncc2)[nH]1)C1CCOC1 c1(C(=O)NCCC2OCCN(C(CC3(C)CC3(F)F)=O)C2)cccc2c1CCC2 C1(OC)CC2CC1CN(C(c1conc1CNC(c1cnccn1)=O)=O)C2 N1(C(C(CSC)OC)=O)CCCC(C)(C)C1CNC(=O)C(=O)N=S(C)(C)=O C1(O)(CN(C)C(C2(F)CCOC2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1 c1(C(=O)NCCC(C)NC(c2cnc(NC(C)=O)o2)=O)nn(C)c(N)c1C c1(C2(C)CC2)ccc(C(=O)NCC2(NC(c3cc(C)c[nH]3)=O)CCOC2)cc1Cl C(=O)(CCC(=O)N1CC(NC(=O)Cc2c[nH]nc2O)CC1C)N(CCC)CCC N1(C(C(CC(C)C)O)=O)CCN(C(=O)C(=CC2CCCCC2)F)C2CCCC12.CC=CC C1(C(C)NC(C2(C(N)=O)CC2)=O)CCN(C(c2ccc(CCF)cc2)=O)CC1 CC1(C)CC1(c1ccccc1)C(=O)NCC1CN(C(C2(CF)CCC2)=O)C1 c1(CCOC)ccc(OC(C)CCF)c(C)c1 N1(C(Cn2ncc(CC)c2)=O)CCCN(C(=O)CCCC(=O)N(C)C)CC1C Cc1cc(F)c(C(N2CCC(C)C(NC(=O)Cc3csc(S)n3)C2)=O)cc1F c1(C(N2C(CO)CC(NC(CN(CCOC)C)=O)C2)=O)ccc2nnc(O)n2c1 C1(O)(CCC2(C)CN(Cc3cccc(N4CCOCC4)c3)C2)CCCCC1 C(=O)(CCC(C)C#N)N(CCC(=O)OCC)C1CC1 N1(CCNC(C(n2cc(-c3cc[nH]n3)nn2)C)=O)CCCC1CO C1(C)(NC(C2C(OC(C)=O)C2)=O)CCN(C(c2cc(CC(C)C)on2)=O)C1 N1(C(Cc2cn(C(C)(C)C)nc2)=O)CC(CO)C(CCO)C1 N1(C(C(C)(C)N(S(C)(=O)=O)C)=O)CC2CC1CN2C(c1cncn(C)c1=O)=O c1(CC)ccc(C(F)(F)F)c(C(=O)OCC23CC(OC)(C2)C3)c1 C1(S(N)(=O)=O)(C(N(C)CC2CN(C(C3CCCCN3C)=O)C2)=O)CCC1 C1(CNC(Cn2ncc(CC)c2)=O)CCC2CN(C(=O)C(F)=CC3CC3)CC12 N1(C(CC(C)SC)=O)CCC(CCC(=O)NC2CN(C)CC2C)CC1 C1(CCCNC(c2ccc(CCC)s2)=O)CN(C(c2cc(C)co2)=O)CCO1 N1(C(Cc2c(SC)cccc2)=O)CCC2(CC1)CN(C(=O)CC1CCOC1=O)C2 C#Cc1cccc(C(=O)NC2CC(CCNC(c3ncccc3F)=O)C2)c1F c1(C(N2CC(CCC)N(C(=O)C(C)=C(C)C)CC2)=O)oc2cc(Cl)ccc2c1C C1(CNC(CCCC#C)=O)C(C)CCCN1C(=O)C(C)SCCCC N12CCCN(CC1)C(=O)C2.c1(CCC(=O)OCC(=O)NC)nnc(C)n1C C1(NC(c2cc(CO)[nH]n2)=O)CCC2CCN(C(C3(CO)CCC3)=O)C1C2 N1(C(C2C(C)(COC)C2)=O)CC2CC(C1)C2NC(c1cc(O)cc(F)c1)=O Cc1[nH]cc(C(N2CC(NC(C3CC4CSCC(C3)C4)=O)C2)=O)c(=O)c1Cl C1(N(C)C(C2(C)CC(C(F)(F)F)C2)=O)CCC(NC(=O)Cc2ccco2)C1 C1(C(=O)N(c2ccncc2)Cc2ccccc2)CSc2ccccc2O1 c1(CCCC(=O)NCC(C)(C2CC2)NC(CC(C)O)=O)ccc(F)c(F)c1 C(=O)(CCCC(=O)NC1(C)CCN(C(=O)CC2CCCN2C(C)C)CC1)OCC N1(C(=O)CCC2CCCC2)CC2CC(NC(C3(COC)CC(=C)C3)=O)C(C2)C1 c1(C(c2nnnn2CCCC)NC(CCCC)CCC)sc2ccccc2c1Cl N1(c2ncc(C)cn2)CC(NC(=O)C(CO)c2ccccc2)CC(C)C1 CC(C(=O)NCC(O)CC(=O)N1CCCC1CCCO)C(C)(C)C c1(C(=O)NCC2N(C(CN(C(C)C)C)=O)CCCC2C)c(F)cccc1[N+](=O)[O-] c1(CC(=O)N(C)CC2N(C(CC3(C=C)CCC3)=O)CCC2)cn2c(n1)CCCC2 C1(C(=O)NC(CNC(c2ccnc(CO)c2)=O)C2CCC2)CC2(C1)CC(F)C2 C1(C(=O)NC2C3CC2N(C(C2CCO2)=O)C3)CC(c2ccccc2[N+](=O)[O-])=NO1 C(C(C)(COC)C(=O)NCc1cccc(NC(C2CCC(C)(C)OC2)=O)c1)OC N1(C(c2ccc(OC)nn2)=O)CCCC(NC(=O)CC2(C)CCCCC2)C1C c1(CCC(N2C(CCCNC(C3CCSC3)=O)CCC2)=O)nc2ccccc2[nH]1 N1(C(C2(OCCOC)CC2)=O)CCN(C(c2conc2C(C)(C)C(F)F)=O)CC1 N1(C(C(C)OCC=C)=O)CC2CCC1CN2C(c1c(C)[nH]c(C(=O)O)c1CC)=O Cc1cc(C(N2CCCC(CNC(=O)C(F)C(F)(F)F)CC2)=O)c2occc2c1 N1(C(C(C)O)=O)CC2(CCN(C(c3ccc(F)cc3Br)=O)CC2)C1 C1(C)(C(N(C)CCNC(=O)CC2CCC(=O)N2C)=O)CCCCNC1=O C1(N(C)C)CCCC(C(N2CC(O)(CN(C(=O)CC3CCOC3)C3CC3)C2)=O)C1 C(=O)(C(C)(O)C(F)(F)F)N1CC2C(N(C(=O)CCCCCc3cccs3)C)(C2)C1 C(=O)(C(F)CC(C)(C)C)NCCn1ncc(C(=O)NC(C)CC(N)=O)c1 N1(C(CC(CC)N(C(c2c(CC)c[nH]n2)=O)CC)=O)CCN(C2CC2)CC1 Cc1sc(C)c(C(=O)NC(CNC(C2CCCN2C)=O)C2CCC2)c1C#N c1(OCC)ccc(-c2cc(C(=O)Nc3cnccc3Br)n[nH]2)c(C#N)c1 C(=O)(C1=NOC(C)C1C)NC(C(N1CCC(O)(CC)CC1)=O)CCN(C)C CCC(C)(C(=O)O)N(c1ccccc1F)C(=O)CCCC1(c2cccc(Cl)c2)CC1 c1(NC(=O)NCC2CC(NCc3ccc(OC)cc3)C2)cc(F)c(C)cc1Cl C(C)(CCC(=O)NC1(CCNC(=O)C(=O)NC2CC2)CCC1)OC c1(OC)ccccc1CCC(N1CCOCC1CNC(=O)C=CC1CCOC1)=O C(=O)(C1COc2ccc([N+](=O)[O-])cc21)NCC(CC)(C)NC(=O)C(N)=O N1(Cc2nccc(OC)c2)CCOCC(C2CCC2)C1 C(C(C(=O)NC(c1ccon1)(C)C)C(C)C)NC(c1c(C)coc1)=O N1(C(CCP(C)(C)=O)=O)CCN2C(=O)C(NC(c3cnc(=N)[nH]c3)=O)CC2C1 C(=O)(C1=NNC(=O)C1)NCC1CN(C(c2c(COC)cco2)=O)C1 CC1(C)CC(C(N2CC=CCC2)=O)CCN1C(=O)CCn1cccc1 N1(c2nc(C)nc(C#N)c2)CCC2CCC(NC(=O)C=CC=C(Cl)Cl)C1C2 c1(C(=O)OC)ncccc1NC(=O)C(=O)NCC1CCCSCC1 C1(COC)CN(C(c2ccnc(CNC(C3CCCS3)=O)c2)=O)CCO1 c1(CNC(c2c(CNC(C3(COC)CCOC3)=O)cco2)=O)nn(C)cc1SC c1(C(N(C2CCC(NC(C3CC34CCC4)=O)CC2)C)=O)cc(Cl)cc(F)c1N C(=O)(CN=c1[nH]c(=NCCC2CC2(Cl)Cl)c2ccc(OC)cc2[nH]1)OCC=C C=C(C)C1OCCCC1C(=O)NC1CCC1NC(c1cc(Cl)cs1)=O CC1OCCC1C(=O)NCC(=O)OC1CC(C(=O)N(C)C)C1 Cc1c(F)ccc(C(=O)NCC2CCCN2C(=O)Cc2ccc(Cl)cc2F)c1Cl c1(C(N(CC(CN(C(C2C(CC)C2)=O)C)O)C)C)nc(C(C)C)no1 n1(C(C)C)ncc2cc(NC(=O)C3=CC(C)CC3)ccc12 CS(=O)(=O)c1ccnc(N(C2CC2)CC2CN(C(C3CCCC3)=O)C2)n1 C1(CNC(C2N(C(Cc3n(C)ccc3)=O)CC=C2)=O)CC12CCOCC2 C(C1=CCN(C(=O)CCN2CCCC2)CC1)NC(c1cncc(CC)c1)=O C1(NC(c2ncn(C)c2)=O)CCC(CNC(=O)CCC2NC(=O)NC2=O)CC1 C1(C)(C(=O)NC2CCC(N(C(CCC=C)=O)C)CC2)CCCN(C)C1 C1(CC(=O)NC2(CNC(c3n(CC#C)cnn3)=O)CCC2)CC(C)(C)C(=O)N1 N1(C(CCC=C(C)C)=O)CCC(C(=O)NCc2ccnc(C#N)c2)CC1(C)C N1(C(C2(F)CCN(Cc3cc(OCC)c(Br)cc3)C2)=O)CCCC(F)C(F)(F)C1 C1(N(CCCSC)C)CC2CC1CN(C(=O)CCOc1cccnc1)C2 C1(CNC(c2ccn(CCC)n2)=O)CC(C)CN(C(c2ccc[nH]2)=O)C1 c1(C(=O)NC2CCC(CNC(Cc3nn(C)c(Cl)c3)=O)C2)cnn2c1CCCC2 c1(C(N2CCC(C(CC)NC(=O)C(c3cnn(C)c3)C)C2)=O)ccc(C)nc1N c1(CS(=O)(=O)NCCCNC2CCCN2CCN2CCOCC2)cccc(Br)c1 CCC(C(=O)N1CCC(n2cccn2)(CNC(=O)C2=COCC2)CC1)C(C)C c1(NC(C2CC(CC(C)(C)C)C2)=O)c(CO)cnn1C.C12CC(C)(C1)CNC2=O C1(C(=O)NCCC2(O)CCN(C(=O)C(O)CCSC)C2)(CC)CC(C)(C)C1 N1(C(C(C)CO)=O)CCC(O)(C2(NC(=O)CC3COCC(C)(C)O3)CC2)CC1 Cc1cccc(CCCN(C(=O)CC2CCCC(O)C2)C)c1.C(=O)(CO)N c1(C(C23CCCC2NCC3)N2CCC(c3nnc(C)o3)CC2)cccc(Cl)c1F N1(C(C(C(C)C)C)=O)CCn2ncc(CNC(C3(c4cccs4)CC3)=O)c2C1 C1(OC)(NC(C2CC2c2ccc(Cl)cc2F)=O)CCC(C)CC1 N1(C(c2cc(CC)no2)=O)CC2CCCC2(Nc2cc3nncn3cn2)C1 C1(NC(c2[nH]cc3c2CCCC3)=O)C2CC3CN(C(C4CC=CCC4)=O)C1C3C2 CC(Cc1cnc[nH]1)C(=O)NCC1CN(C(c2ncoc2C2CCC2)=O)C1 C(=O)(CCCC(=O)N(CCCN(C(=O)CC1CCCCN1C)C)C)OC C1(Cl)(C(N2CCCC(N(C(CCCCOCC)=O)C)C2)=O)CC2CCC1O2 CCC(CC(F)F)C(=O)NCC1CCCN1C(=O)Cc1cccc(C(=O)OC)c1 N1(C(CCc2n(C)cnc2)=O)C2CCCC1CN(C(C1CCCCS1(=O)=O)=O)C2 Cc1nc2sc1NC(=O)C(C)CN1CCC2CC1.C1(C2(C(=O)O)CC2)CCCO1 N1(C(c2nc(C)co2)C(=O)NCC)CC(Cc2ccccc2)OCC1C C1(C(=O)NCC2N(C(CCCNC(N)=O)=O)CCC2)Cc2ccc(F)cc2O1 Cc1[nH]nc(C(F)F)c1C(N1CCCC(NC(=O)Cc2ccc(Cl)s2)C1)=O c1(C(=O)NCCNC(=O)CC2(O)CCCOC2)cc2cscc2s1 c1(C(=O)NCC2C(C)CN(C(=O)CC(O)CN(C)C)CC2)c(N)cc(Cl)cc1F CCCCCCC(=O)N(C)CC1C2CN(C(c3nc(C)c(C)[nH]3)=O)CC12 C(=O)(C(C)CC(C)(C)C)NC1CCCN(C(c2nc(CCC)sc2)=O)C1 Cc1cnc2n1CCC(C(=O)NCCCN(C(=O)C(C)Oc1ccccn1)C)C2 N1(C(c2cc(NC(C)=O)ncc2)=O)CCC2(CCCC2NC(c2cscn2)=O)C1 Cc1ccc2nc(C(=O)N(C)CCN(C)C(C3CCCO3)=O)ccc2c1 c1(SC)cc(C)ccc1C(=O)NC(C1CCCN1C(C1COCOC1)=O)C c1(C(=O)NC2(C(=O)N(C)Cc3c(C)noc3C)CC(F)C2)cncc(CC)c1 C1(C(N2CCC(C)(CNC(c3cncnc3C)=O)C2)=O)(CC)CNC(=O)C1 Cn1ccc2[nH]c(C(=O)NC3CC(NC(c4c[nH]c(=O)cn4)=O)C34CCC4)cc12 N1(C(C2CCN(C(C(CCC)O)=O)CC2)=O)CC2CC1CS2=O c1(CC)ccc(C(=O)N(CCNC(=O)C(C)OCCOC)C(C)C)c(N)c1 C1(Nc2cc(N(C3CCC(O)CC3)CCCC)ncn2)CC2(CCC2OC)C1 C12CCN(CC1)C2=O.C1(C(C)(C)C)(CN(C(=O)Cc2cn(C)nn2)C)CCCC1 c1(SC)ccc(C)c(C(=O)NC(c2ccccc2)CNC(c2cc(Cl)no2)=O)c1 C1(C2CC2)(NC(COCC(=C)C)=O)CCN(C(=O)C(C)SC(C)C)C1 c1(CC)conc1C(=O)NC1COCC1C(=O)NCC(C)O n1(CC)ccc(CC(=O)NC2CCC2CNC(=O)CC2(SC)CCC2)n1 C#CCC(C)(C(=O)N=c1ccn(C2CC2)[nH]1)NC(C1C2CCC(=O)C12)=O C12(C)CCN(C1)C2=O.CC1(N2CCCC2)CN(C(C2CCCOC2)=O)C1 c1(C(=O)OCC)ccccc1COC(=O)C(F)(F)c1nc(C)cs1 C1(CN(CCCN(c2ccncc2)C)CC)CCCCN1C(=O)CCCF CCCCCCCC(O)C(=O)NCc1c[nH]nc1C(=O)O C1(CC(=O)NC(C)Cn2ccnc2)CCN(C(=O)C(C2(O)CCCCC2)O)CC1 C1(COC)(CNC(=O)CCn2ccc(C)n2)CCCN1C(c1ccccc1)=O c1(C(=O)NC(C(=O)NCCCNC(C)=O)C(C)O)ccc(=O)n(C)n1 c1(C(=O)NC(CNC(c2cc(C)ncn2)=O)C(C)C(C)C)ccc(C)c(Cl)c1Cl C1(O)(CNC(c2c(CC)nn(C)c2Cl)=O)CCCN(C(=O)CSS(C)(=O)=O)CC1 C1(CC)(CC)CCN(C(=O)C(CC(C)C)NC(=O)C(C)N=[N+]=[N-])CC1 N1(C(C(COCC)NC(CCC=CCC=C)=O)=O)CC2CC1CN2C(=O)NC C1(C(=O)NCCNC(CC(C)C(F)F)=O)CC2CCC(C1)C2F c1(C(=O)NC(C2CCCCN2C(=O)C2=CSCS2)C)cccc[n+]1[O-] C#CCCC(C(=O)NC(c1ccc(C)cn1)C)NC(=O)CCn1ccnc1C C1(C(=O)NC(C2CCCC2)CNC(CNC(COCC#C)=O)=O)CCSC(C)C1 C1(C(=O)NCC2CCN2C(C2CCC(=O)O2)=O)(OC)CCC12CCC2 C1(O)(C(C)NC(C=CSC)=O)CCN(C(C2CC(C)CO2)=O)CC1 C(=O)(C(CC(C)C)n1ccnc1)N(CCCCN(C(C(F)=CCC)=O)C)C c1(C(=O)NCC(CNC(C(COC)C)=O)O)cn(CCO)c(=O)nc1O C(=O)(C1=C(c2ccccc2)CCCC1)N1C(CNC(CC(CC)(C)C)=O)CC1 CC(CNC(N1CCOCC(C(=O)O)C1)=O)CC(F)(F)F c1(CC)cc(C(=O)NC2CC2NC(=O)CN(C)C(C)=O)ccc1F N1(C(C2CCC(CC)O2)=O)CCC2CCCC(C1)N2c1nnc(CC(=O)NC)s1 CC1=C(C(=O)NC(C(=O)NCC2=CCCC2)C(C)(C)C)CCC1 C1(NC(C(C(=O)OC)C)=O)CC2CCC1CN2C(c1cnc(OC)nc1C)=O C1(NC(C2CCN2C(=O)CC2C=CCC2)=O)C(O)CC1O CC1(C)CCC(C)(C)c2cc(S(=O)(=O)N3CCC(OCC(F)F)C3)ccc21 c1(C(=O)NC(C2CC=CCC2)CNC(C)=O)cccc(C(N)=O)c1F C(CCC(=O)N(CCC(=O)NC(C)(CO)C1CC1)CCO)C1C(C)C1 CCC(O)C(C)(C)C(=O)N1CCN(C(c2ccnc(S)c2)=O)C(CO)C1 N1(C(CCC=C)=O)CCN(C(=O)C=Cc2ccoc2)CC1CC1CCCC1 CC(C)C(O)C(C)(C)C(=O)NCCC(C)(C)CNC(=O)CCCCC1CCCC1 N1(C(C(C(COC)C)C)=O)CCCN(C(=O)Cc2cc(OC)ccc2Cl)CCC1 C1(c2n(C)nnn2)(NCCc2ccc3c(c2)CC3)CCCC(OC(C)(C)C)C1 C1(C(=O)NC2CCCN(C(C3(CC(=O)OC)CC3)=O)CC2)CCN2CCOCC12 CC1(C)NC(=O)CC1C(N1CCCC(C)(CNC(C2CC2c2ccoc2)=O)C1)=O N1(C(C2(CC)CCOCC2)=O)CC2CCC(CNC(=O)C3=C(Cl)CCOC3)C2C1 CCC(CC(=O)NCCCC(O)C(=O)N1CC2CCC(C1)O2)C(C)C N1(C(C(=O)NC(C)(C)C)CCc2ccco2)CCCC(C(F)F)(C(=O)OC)C1 c1(C(=O)NC(CCC)C(=O)NCC2CCC(C)C2)ncc(F)cc1C C(C(C)(COC)C(=O)N1CCC(CO)C(NC(=O)CCc2cnccn2)C1)OC N1(C(C(C)NC(c2ccco2)=O)=O)CCC2CCN(C(=O)CSC3CC3)CC12 CCC(CC(=O)N(CC(C)(C)CNC(C1CC(=C2CCC2)C1)=O)CC)SC C1(NC(C=CCC)=O)COC2C(NC(c3c(F)ccc(F)c3OCC)=O)COC12 S(=O)(=O)(c1ccc(Br)cc1)N(C(CN(C1CCSCC1)C)=O)CC1CC1 C(CCC1CCC1)(C(=O)NC(c1cccs1)C)NC(c1ccc(SC)o1)=O Cc1nn(C)c(Cl)c1C(=O)NCCN(C(=O)CCOc1cccc(C#N)c1)C1CC1 N(C(=NCCOC1CCSCC1)NCc1ccccc1)C1CC(CN)C1 CCC(C(C)C)S(=O)(=O)NCC1CCCC2(CCC2)C1 c1(C(=O)NC(C2(C)CN(C(=O)CCc3cn[nH]c3)C2)C)cc(O)cc(F)c1 c1(NCC2(CNC(C3(C)CC4CCC(C3)S4)=O)CC2)nccc(S(C)(=O)=O)n1 N1(C(c2ccn(C(C)C)n2)=O)CCC(CO)(NC(=O)C(c2cnn(C)c2)C)CC1 C1(N(CC(=O)NC2(C)CC=CCC2)C)C2CC(O)C1N(C(c1ccncc1)=O)C2 C(=O)(CCCC(=O)NC1CC1NC(c1ccc(C2CCC2)cc1)=O)OCC C1(C(=O)NC(COC(C)=O)CO)CC(F)(F)CN1C(C1OC2CCC1C2)=O c1(-c2c(CC)ncs2)nc(CC(C)OC)nn1C.n1(CC)ccnc1 C1(C2(O)CCOC2)(NC(C(C(C)NC(CSCC)=O)C)=O)CC1 Cc1ccc(CC(C)C(=O)N(CCC(C(C)C)NC(c2csc(F)c2)=O)C)cc1 C(=O)(C#CC1CCOCC1)NC(C1(C2C(C(C)(C)C)C2)CCC1)=O.C1(C)CCCC1 N#CC1CCCC(CC(N2CCCC(CCC3CCC(OC(F)(F)F)C3)C2)=O)C1 c1(C(C(N2CCCC(CNC(CC(C)OC)=O)C2)=O)(F)F)ccc(=O)n(C)c1 Cc1cc(CC(=O)NCCC2(O)CCCN(C(=O)C(C)N(C)C)C2)ccc1Cl N1(C(CCCOCC)=O)CCC(O)(C(C)CNC(c2cccc[n+]2[O-])=O)C1 N1(C(c2c(C)n(C)cn2)=O)CCN(C(c2ccsc2C#N)=O)CC1C c1(C(N2CCCC(N(C(C34CC(OC)C3C4)=O)C)C2)=O)cc2n(n1)CCNC2=O c1(OC)cc(Cl)c(Cl)cc1CNC1C=CC(C(=O)Nc2cc(CO)cc(C)c2)C1 c1(CCCC(=O)N2CC(=C(CNC(C3CC(C)(F)C3)=O)F)C2)ccc(F)c(F)c1 Cc1ccc(C(=O)CN2CCN(C(=O)Cc3ccsc3)CC2C2CC2)cc1Cl CON1CCC(C(=O)NC2CN(C(=O)CSC(C)(C)C)CCC2C)CC1 N1(C(CC(C)OC)=O)CCC(C)(C(=O)NCCC(F)(F)F)C1 CC1CCN(C(=O)C=Cc2cnc[nH]2)CC1NC(=O)C=CCN1CCCC1 c1(NCC2OCCN(C(C3(COC)CCOC3)=O)C2)ncc([N+](=O)[O-])cc1F c1(SCC(c2ccccc2)OCC)cccnc1-c1ncccc1Cl C(C(F)C(=O)NCCNC(=O)NC1(c2cccnc2)CCCC1)N(CC)CC C1(C)(C(=O)NCc2onc(C)n2)CCCN(C(C2CCC=CCCC2)=O)C1 C1(NC(CCC(=O)NC)=O)CCC2CN(C(c3ccn(C)c3)=O)CC2C1 N1(C(C(C)OC)=O)CCC2C1CCN2C(=O)C(c1ccccn1)Nc1ccccn1 c1(C(N2CC(COC)N(C(=O)CCS(C)=O)CC2)=O)cc2c(C)ccc(F)c2o1 Cc1cc(CC(=O)NCCC2CN(C(C3(C#N)CC3C)=O)C2)nn1C C=C(Br)CCC(=O)N(C1CN(C(C2(O)CCC2)=O)C1)C CC(C)(CNC(=O)NC1(Cl)CC1(F)F)CSc1ccccc1 C1(NC(CC(CC)(C)C)=O)CC2CN(c3cc(C)c([N+](=O)[O-])cn3)CC2C1 n1(CCC)cc(C(N2CCC(N(C(=O)C(C)CC(C)C)C)C2)=O)c2ccccc12 c1(C(=O)NCC2C(NC(C(C)c3cccs3)=O)COC2)cnn(C)c1Cl c1(C(=O)NCC(CNC(c2c(CCC)nsc2N)=O)C)cccc2cncn12 N1(C(C(CCCC)N(C)C)=O)CCC2(CCN(C(c3ccnnc3)=O)C2)C1 c1(C(=O)NC2CCCN(C(c3cnc(CC)[nH]3)=O)C2)cnc2ccnn2c1N N1(C(CCC=C)=O)CCOC2(CCN(C(c3cnc4cc(C)nn4c3C)=O)C2)C1 c1(C(=O)NC(C(=O)OC)C)n[nH]cc1CNC(=O)CCOC1CCCC1 C(C)(C)(CC(F)C(=O)NCC(C)(O)COC)NC(C=C(CCC)CCC)=O C1(CNC(=O)CSc2cccnc2)CC(F)(F)CN1C(=O)C(C1CC(F)(F)C1)O c1(OC)cc(N2CC(C)(C)OC2=O)cc(OC)n1 C1(C(=O)NCC(CC=C)NC(c2oc(C)cc2C)=O)(N(C)C)CCCOC1 CCCC(O)CC(=O)NC1CCN(C(=O)Cn2ccc(C)n2)C1 CC1CCC(=CC(=O)NCC2CN(C(=O)Cc3ccc(C(F)(F)F)cc3)C2)CC1 N1(C(C2CCN(C)CC2)=O)CCCCC12CN(C(c1cc(C(N)=O)c[nH]1)=O)C2 c1(-c2cc(C(N=c3[nH]nc(SC)s3)=O)n[nH]2)ccc(S(=O)(=O)NCC(C)C)cc1 n1(CC)ncc(C(=O)NC2(CF)CCN(C(=O)Cc3cc(C(C)C)no3)C2)c1Cl N1(C(CC)CC)C(=S)NC(c2cc(OC)c(O)cc2F)C2=C1C1(CCC1)NC2=O C1(CSC)(CO)CCCN(C(C2(NC(C(CCC)NC(N)=O)=O)CC2)=O)C1 C(C(=O)NC1(CNC(=O)C2=CSCCO2)CCC1)(C(C)(C)C)OC O=S(=O)(c1nc(N2CCC3(CCCCC3)C2)ccc1Br)N.N1CC2CC2C1 N1(C(c2c(C)c(Br)no2)=O)CCOCC(NC(C2(C)CCCS2)=O)C1 N1(C(CN(C2CCSC2)C)=O)CCC(CO)(CNC(=O)Cc2cncs2)CC1 N1(C(CCC2OCCN(C(CCC(=O)NCCC)=O)C2)=O)CCCC(C)(O)CC1 c1(C(C)=O)c(C)[nH]c(C(N2CCCC(N(C)C)C2C)=O)c1C(C)C N1(C(c2nccc(NC(c3cccc(N(C)C)c3)=O)c2)=O)CCN2CCCC2C1 CCC(CC(=O)OC)NC(c1oc(CNC(=O)Cn2nnnc2C)nc1C)=O c1(C(N2CC(CNC(CNC(CCC)=O)=O)N(C)CC2)=O)cc2nnn(C)c2s1 C#Cc1cn(C)nc1C(N1CCOC(C)(CNC(C2CCCCS2(=O)=O)=O)C1)=O C1(NC(CCC=C)=O)CCN(C(=O)C(c2ccc(F)cc2)F)C(C)C1 c1(C(=O)NCCC2(CNC(c3n(CC)nnc3)=O)CC2)cc2c(s1)CCCC2 CC1CN(C2CC2)Cc2cccc(Br)c21.N12C(=O)OC(C(F)(F)F)C1C2 C(=O)(C1=CC(O)C(NC(C2CC3CC3C2)=O)C1)NCC(=O)NCC1CC1 C1(NC(C=CC=CCCCCC)=O)CCN(C(c2ccc(C)cc2Cl)=O)CC1C C(CCC(C)C)(C(=O)N(C)CC1CCOCC1)NC(CC(CC)C1CC1)=O C1(C(N(CC(O)C(F)(F)F)C)=O)CC2CCC(C1)N2C(C1(F)CCCC1)=O c1(CN2CC(NC(CC(CC)O)=O)C(F)(F)CC2)ccc(C)cc1[N+](=O)[O-] C=CCCCCCCC(=O)NCCOCCC(=O)NCCc1cnc(C)[nH]1 FC(F)(F)C(CC(F)F)c1nc(-c2cccc(Br)c2)nn1CC(F)F C(=O)(C1CCc2cc(F)ccc21)N1CCC(NC(c2n(CC)nnc2)=O)CC1C CCCCCCNC(C1(NC(=O)CC2C=CCCC2)CC(F)C1)=O c1(C(=O)NCCCN(CCC)C(c2cc(C)nn2CC)=O)ncc(C)cc1C N1(C(C(CC)F)=O)CCCC(CC)(NC(c2cc(C)c(C(=O)OC)o2)=O)C1 c1(CNC(C(CC)SC)=O)cncc(CNC(=O)C(C)Cc2ccccc2F)c1 Cc1ccc2sc(C(N3CC4CC(C3)C4NC(=O)CC3CCCO3)=O)c(C)c2c1 C(=O)(C1=C(Cl)CC1)NC(C)CCCNC(c1cc(Cn2cccn2)on1)=O N1(C(C(CNC(=O)NCC#C)O)=O)CCC(CNC(C)=O)(NC)CC1 C#Cc1cccc(NC(C)C(N2CCN(C(=O)C(F)n3cccn3)CC2)=O)c1 C1(NC(COc2cc(C)on2)=O)CCC12CN(C(=O)Cc1cc(Cl)cnc1C)C2 N1(Cc2cn(CCCCOCC(=O)OC(C)(C)C)nn2)CCCCC1C(=O)O O=C1CC(=O)NC(C(=O)NC2C=CC(C(=O)NCc3ccncc3Cl)C2)C1 Cc1cc[nH]c1C(=O)N(C1CN(C(=O)C(F)n2cccn2)C1)C c1(N(C(=O)CN2C3COCC2C3)C(c2cn[nH]c2)=O)ccccc1F C1(CNC(c2cocn2)=O)C(C2CC2)CCN1C(c1csnc1Cl)=O C12(CNC(c3ccc(C)cn3)=O)CCC1CCN2C(=O)CSc1nncn1C C=CC1CN(C(=O)CNS(=O)(=O)CCCC)CC1NC(=O)Cc1ncccc1C c1(CC)cccc(CC(=O)NCCN(C(c2cc(C)c(Br)o2)=O)C2CC2)c1 c1(C(N2CCC(C(C)NC(=O)Cn3nccn3)C2)=O)cnc2[nH]nnc2c1 C(=O)(C1CCCc2nc[nH]c21)NCC1(F)CC(CNC(=O)CCOC2CC2)C1 CC1C(=O)OC2C1CCC1(C)CCC3(C=CCCN(C)C3)CN2C(=O)C2CC1CCN2 C1(CNC(Cc2ccn(C)n2)=O)CC2COCC2N1C(c1ccncc1)=O Cc1ccc(CN2CC3(CC3)CC2C(N2CCOC(C#N)C2)=O)cc1O C(CCC(=O)N1CCCC1CC(=O)NCC(C1CC1)SC)OC C1(C(=O)NCCC#C)CC(O)CN1C(=O)C(c1ccccc1Br)OCC.C(C)(=O)O N1(C(c2c(OC)c(C)sc2)=O)CC2CN(C(c3cc(C)c(O)nn3)=O)CC2(C)C1 c1(OC)c(C(=O)NC(CNC(c2ccoc2)=O)C(C)C)cccc1C(F)F c1(C(=O)NC2C3CN(C(C4C(C)C4)=O)C2C3)ccn2c(C(F)(F)F)nnc2c1 N1(C(C(CC)CC)=O)C2CCC(C2)C1C(=O)NC1C=CC(C(=O)NC)C1 Cc1nnn(CC(=O)NCC(C2CCCC2)NC(C2(O)CCOC2)=O)n1 C1(C(=O)NCC2CC(NC(C(CC(C)C)C)=O)C2)CN2CCN1CC2C C1(NC(c2ccc[n+]([O-])c2)=O)CCN(C(=O)Cc2ccnnc2O)CC1 c1(OC)ccc(CC(=O)NCC2CC(C)N(c3nnc(O)s3)C2)c(C)c1 c1(C(N2C(CO)CC(NC(C3CCCS3)=O)C2)=O)c(Cl)ccc2c[nH]nc12 C(=O)(C(O)CCCc1ccccc1)NC(CC)CNC(C1(N(C)C)CCC1)=O FC(F)(F)C(F)(F)N(CC(O)Cn1cnnc1O)Cn1ccnc1 C1(CC(C)NC(=O)CC2(C)CC2(Cl)Cl)CCN(C(c2nnn(C)n2)=O)CC1 CC1(C)CCCC(C(=O)NC(Cc2ccccc2Br)Cc2c(Cl)cccc2Cl)C1 C1(C(=O)O)CCN(N(C(CC)C)C)CC1.c1(C=O)ccncc1F C(=O)(C1=CCCCO1)NC1CN(C(=O)C2=CCCC2)CC1c1cccc(F)c1 C(=O)(C1=C(C#N)CCC1)NC1CCC(N(C(=O)CC2CC(F)(F)C2)C)C1 c1(C(=O)NCC2COCCN(C(CC3C(C)C3)=O)C2)cccc(C#CC2CC2)c1 C1(CN(C(=O)C2=CCOC2)C)COCCN1C(=O)CCCc1ccsc1 N1(C(CCC)=O)CCC(NC(=O)COc2ccc(Br)cc2CC)C(C)C1 S(=O)(=O)(c1ccc(NC2CC3CC3C2)c(Br)c1)N(CCCO)CC CC(=O)CCCC(C)C(=O)NCC1(C(N2CCC3(CCC(O)C3)C2)=O)CCCC1 c1(SCC)cnc(O)c(C(=O)NC2CCN(C(c3cc(C)n(C)c3)=O)C(C)C2)c1 C1(C#N)(C(=O)NCCNC(C2C(=C)CC2)=O)CC12CCC2 C1(C(N2C(C(=O)NC)CCC2)=O)CC(C2CNC2)C1 c1(CNC(C2(F)CCN(C(C)=O)C2)=O)ccc(F)c(C#N)c1 C1(C)(C(=O)NCCC2CCCN(C(C3C(C)OCC3)=O)C2)CCN(C)C1=O N1(C(C(Br)=C(C)C)=O)CCC(C(C)CNC(=O)C(C)Cn2cccn2)CC1 c1(C(N2CCC(C(C)N=c3nc(C(C)(C)C)[nH]s3)C2)=O)ccc2ccncc2n1 C1(NC(c2ccc(C)nn2)=O)CCC12CN(C(=O)CC1CCCC1)C2 N(C1CCCc2c1cnn2-c1ccccc1)C(C1CC(CS(C)(=O)=O)C1)=O CC1=C(C(=O)N2CCSCC2c2ccc(C(F)(F)F)o2)S(=O)(=O)CCO1 CCC(CC)CCC(=O)N1CCCC1C1CCN(C(=O)CCCC(N)=O)C1 C(C(C)(F)C(C)(C)F)n1cc(C2CN(C(C3(C)CCN(CCO)C3)=O)C2)nn1 c1(C(C(=O)NCCCC2CC2)N(CCCO)C(C)C)ccc(C2CC2)cn1 c1(CC)ccc(C(=O)N(C2CCN(C(C3C=C(C)CS3)=O)C2)CCOC)s1 CC(C)CCCC(C)C(=O)NCC(C)(C)C(=O)NC(C1CCOCC1)C C1(CNC(C)=O)C2CCC1CN(C(=O)Cc1cncnc1)C2.C1CCCC(=O)N1 N1(C(CC2CC(=C)C2)=O)CC2(CO)CC1(C(=O)NC(CO)CCC1CC1)C2 CCC(CCC(=O)N(CC(O)C(F)(F)F)C)NC(=O)CCNC(C)=O n1(CC)nc(C)c(NC(C2CC23CCN(C(=O)CN2CCCCC2=O)C3)=O)c1C C1(NC(Cc2c(C)nc(S)s2)=O)CC(O)CN(C(=O)COCC2CC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC(CNC(=O)Cc2cncs2)OCCC1 Cc1ccc(F)cc1-c1nnc(CN2CCCC2c2ccco2)o1 C(C1CC1)(C1CC1)=CC(=O)N(CC(C)C(=O)NC1CCN(CC2CC2)C1)C Cc1cccc2c(C(N3CCC(CNC(=O)CC(C)(C)C)C3)=O)coc12 CC1CN(C(=O)C(F)(F)c2cccnc2)CCN1C(=O)CC1CCCC1 N(C1CCCc2ccoc21)C(C1CN(C(C=CC=CC)=O)CC12CC2)=O c1(C(=O)NC2CCC2NC(c2cccc(C3CC3)c2)=O)ccc2oc(S)nc2c1 CC(CC(C)(C)C)C(=O)N1CC(C)(C)CC1C(N1CCOC(C)(CO)C1)=O C(=O)(C(C)(C)CS(=O)(=O)N1CC(N=[N+]=[N-])CC1C(=O)OC)OC C1(NC(CCNC(C)=O)=O)CCN(C(C2CSC2)=O)CCC1CO n1(CC)nc(C(N2CCCC(CC(=O)N(CC(C)O)C(C)C)C2)=O)cc1C C12(Nc3ncc(C)c(C)n3)CCCC1CN(C(c1cc(C)c(C)nc1O)=O)C2 CC1CC(NC(c2cc(C(F)F)nn2C)=O)CN(C(c2nn(C)cc2N)=O)C1 C1(OC)CSCC1.C1(C(F)(F)F)(C(=O)OC(C)(C)C)CC1 C1(C(N2CC(C(=O)NCC3CCCC3C)(COC)C2)=O)CCCC(=O)C1 N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)CCC1CCC(=O)N1)C2C(C)C Cc1cc(NC(=O)C(O)CCNC(C2(C)CCC(=O)NC2)=O)cnc1O C(=O)(C(O)CC(C)(C)C)NCC1N(C(c2nc(C)c(C)s2)=O)CC1 C1(C#N)(C(N2CC(C(C)NC(=O)Cn3cc(Cl)cn3)C2)=O)CC1(C)C CCCCC(CC)C(=O)N1CC2CCC(C(=O)NC3CCC(N(C)C)C3)(C2)C1 N1(CC(=O)NC(C2CCCCC2)CNC(COCC(=C)C)=O)CCOCC1 N1(C(C(CC=CC)C)=O)CC2(CC(NC(C3(CSC4CC4)CCCO3)=O)C2)C1 CCCCC(CNC(=O)CC(C)n1cc(Br)cn1)NC(=O)CCSC Cc1[nH]c(C#N)cc1C(N1CCC(CF)(NC(=O)Cn2cccn2)C1)=O C1(O)(CNC(C#C)=O)CCN(C(=O)C(c2ccc(F)cc2)F)CC1 c1(OCCC)ccccc1C(N1CC(NC(=O)Cc2ccsc2)C(O)C1)=O N1(C(C2(N(C(c3ncc(C)[n+]([O-])c3)=O)C)CC2)=O)CC2(CNC(=O)C2)C1 C1(CNC(c2cc(C)ns2)=O)CCC2CN(C(c3ncoc3C(C)C)=O)CC12 Cc1ccn(C)c1C(N1CCCC(CNC(c2cc(Cl)ccn2)=O)C1)=O O=C(C1=CC2CCC(C1)C2)N(CCC(=O)NCC1CCC(F)C1)C1CC1 Cc1cnc(C(N2CCOCC2c2cn(Cc3nccs3)nn2)=O)c(Cl)c1 C1(C(=O)NCC2(O)CC(NC(=O)CSC(F)F)C2)CN2CCC1(C)C2 c1(C(N)=O)ccccc1C(N1CCC(C(=O)NCC(CO)CO)C1)=O C12(CC(=O)N(C3CCCN(C(c4snc(C)c4N)=O)C3)C)CCCN1CCC2 N1(C(C(C(C)C)n2cccc2)=O)C2CCC1CC(NC(=O)C(F)(F)C(C)O)C2 Cc1cc(C(=O)N(CCCC(=O)NC2CCN(C(C)(C)C)C2)C)c(C)n1C CC(N=c1[nH]c2c(c(=NCc3cn[nH]c3)[nH]1)SCC2)c1ncnn1C c1(C(=O)NC2(C)CCCN(C(C3(CO)CC(F)(F)C3)=O)C2)cnn2cnnc2c1 c1(C(N2CCC(CCNC(C(CC)OC)=O)C2)=O)ccc(OC2CC2(F)F)cc1 N1(C(C(F)=CC)=O)CCC2(CC1)CC2CNC(c1ccc(CS(C)(=O)=O)cc1)=O C1(NC(C(CC)=CC)=O)CC2CCC1CC2NC(=O)CCOC(C)CC(C)C N1(C(CCCOC)=O)CC(CNC(=O)C(C)Cc2ccccc2)CC(C)(C)C1 C(C1=CCCN(C(=O)CC(C)c2ccco2)C1)NC(C(CO)OC)=O CCC(CC)C(=O)NCC1CCCN1CC.c12ccccc1CNC2=O C1(CC#C)(C(N2CC(OC3C=CC(CCC(=O)NCC(N)=O)C3)C2)=O)CCOC1 c1(C(N)=O)cocc1C(=O)NCC1CCCN1C(=O)CC1CC2(CC2)C1 C1(O)(CCNC(C2C(C=C)C2)=O)CCN(C(C2(C)CS(=O)(=O)C2)=O)C1 C#CCCCC(=O)NC(C1CCCCN1C(=O)C=C(CCC)CCC)C C1(NC(c2c(OC)ccs2)=O)CCCC(C(=O)NCC2(CCO)CN(C)C2)CC1 C(N=c1nc2sccc2c(N2CCc3c[nH]nc3C2)[nH]1)C1N(C(CC)=O)CCC1 CCCCCC(O)CC(=O)NC1CN(C(c2cocc2C)=O)C(C)(C)C1 Cn1cc(CC(N2CCCC2C(C)(C)NC(C2(F)CC=CC2)=O)=O)cn1 N1(C(C(CCC)NC(C)=O)=O)C2CCC1CN(C(C1CC(OC)C1)=O)C2 c1(C(=O)NCC(C(=O)NC2CCC(F)(F)C2)N(C)C)ccc(O)cc1 C1(NC(c2cc3nc(C)sc3[nH]2)=O)CCN(C(=O)COCCF)CC(C)(C)C1 c1(CC)nc(=N)[nH]cc1C(=O)N(CC(O)CN(C)C(C1CC(=O)NC1(C)C)=O)C C(=O)(C1CCCn2cnnc21)N(C1CCC(C)(C)C1)CCOC c1(OC)cc(C(N2CCCC2CCCNC(=O)CSCC2CCCCO2)=O)sn1 C1(C(=O)NCc2c(SC)c(F)ccc2)CC2COCC(C1)C2 O=[N+]([O-])c1ccn(-c2ccc(F)c(CNC3CCOC3c3ccccc3)c2)n1 c1(C(N2CCC(C(C)C(=O)N(C)Cc3cncs3)C2)=O)ccc(O)c(F)c1 C1(c2nnnn2C)(NC2(CCOC)CCOC2)CC2CC(O)C(C1)N2C c1(N(CCC)C(=O)Oc2ccc(-c3cccs3)cn2)ccc(-c2cscn2)cc1 C1(COC)CCN(C(=O)Cc2c[nH]c(C(N3CCC3C(=O)OC)=O)c2)CC1 N1(C(CCS(=O)(=O)NC)=O)CCC(C)(C)C(C(N2CCCC2CO)=O)C1 C(=O)(C(C)(C)C(C)(C)O)NCC(C(C)(C)C)NC(c1ccc(Br)o1)=O C(=O)(C1CCc2c[nH]nc21)N1CC(CC(CNC(c2c(C)sc(O)n2)=O)(C)C)C1 C1(NC(c2n(CC)ncn2)=O)CC2CC(C1)N(C(c1ccnc3c1CCC3)=O)C2 c1(C(=O)NCC(CC)NC(C2C3CCC(F)(F)C23)=O)cc([N+](=O)[O-])cnc1N C(CC(O)CNC(=O)CCN(CCC(C)(C)C)C)NC(C1(CC(C)=O)CC1)=O C1(OCCCN(C)C(c2cnc(Cl)[nH]2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1 CC(=Cn1ccnn1)C(=O)NCCC1CN(C(=O)CC2CCCCN2C)CC1C C#Cc1cccc(C(=O)NC2(C)N(Cc3cccc(CC)c3)CCOC2)c1 C1(CC)CN(C(C2CCCCN2C)=O)CC1NC(c1ccc(C(N)=O)cn1)=O C(CCCC(=O)NC(C1CCCN1C(=O)C(C)C)C)(OC)OC C1(C(N2CC(O)CC2C2CC2)=O)CCN(C(=O)CC2(O)CCCCC2)C12CCC2 CC1CC(=O)NC1C(=O)NC1(CNC(c2[nH]c(O)nc2C)=O)CCC1 C1(OC)CCCN(C(C2CCCC2CNC(=O)C(C)(C)n2cccn2)=O)C1 C(=O)(C(O)C1=CCCCC1)NCC(CCCC)NC(c1cccc(Cl)c1F)=O N(C1CCC(NC(=O)C(CC)(CC)OC)c2ccccc21)C(CSCCC)=O C1(NC(COC(C)=O)=O)CCC(C#N)CC1.C12CCC1NC2=O N1(C(C(C)OCCC(C)C)=O)CCC(C2(NC(C3CC4(CC4)CO3)=O)CC2)CC1 N1(C(C2CCCC(C)C2)=O)CC2CC(NC(c3cccc(N(C)C)n3)=O)C(C2)C1 C1(C(=O)NCC(CO)NC(C2OCCO2)=O)(OC)CCCOC1 C1(NC(C2(CC)CCCC2)=O)CCCCC1NC(C1CCC(C)CC1)=O C1(SC)CN(C(c2ccc(C#N)[nH]2)=O)CC1NC(C1CS(=O)C1)=O c1(C(N2CC(NC(CC(CC)C)=O)CC2(C)C)=O)cc(=O)n(C)cc1Br C1(N(C(C(C)C#N)=O)CCF)CCCN(C(=O)C(=O)NCCC(N)=O)C1 c1(NC(N2C(C)(CNC(c3c(OC)cccc3)=O)CCC2)=O)oc(C)nc1C#N C(CCCCC(=O)NC1CCCC1(C)CN(C(=O)CC(C)(C)SC)C)SC C1(C(=O)NC(C2CCC2)C)CN(C(C2CC(F)(CF)C2)=O)CC1C1CC1 c1(CNC(=O)NC(c2ccccc2F)C)ccc(C(C)(C)C)cn1 c1(NCc2cc(C)[nH]n2)nc(N2CCC(N(C)C)C(C)C2)nc2c1cnn2C NC(=O)C1=NOC(CNC(=O)CCNC(c2csc(Cl)n2)=O)C1 N1(CC2(NC(C(C3CCSC3)N(c3cc[nH]n3)C)=O)CC2)CCCCC1 c1(NC(C(C)N(C(c2n(CCC)ncc2)=O)CC)=O)ccc(F)cc1CO c1(C(C(=O)Nc2ccc(OC(F)F)cc2)(F)F)c(F)cccc1Cl.N1CCCC1 Cc1ccc(C)c(C(=O)NCCCCCCNC(c2occ3c2CCC3)=O)c1C c1(CC(=O)NCC(C2CC2)NC(C=CC2N(C)CCC2)=O)ccc([N+](=O)[O-])c(N)c1 CN1CC(C(N2CCOCC2C(=O)Nc2cccc(CCF)c2)=O)CCC1=O C(N=c1cc(C)nc(NC2CCCCN2CC)[nH]1)C1(OCC)CCCSC1 C1(O)(CN(C(c2c(C)nns2)=O)C)CCN(C(c2ccncn2)=O)C1 C1(OC)CN(C(c2cn(CCO)nn2)=O)CC1C(NC[Si](C)(C)C)=O C1(CNC(=O)C=C(C)CNC(C2(COC)CC(=O)C2)=O)(OC)CCCCC1 C1(NC(C=CSC)=O)CCOC2(CCN(C(C3CC3CC(C)C)=O)CC2)C1 c1(N2C3CN(C(C(CC)CCOC)=O)C(CC3)C2)nc2ccc(Br)cc2s1 c1(C(=O)NCC2C(C)CN(C(C3CNC(=O)N3)=O)CC2)cnn2ccccc12 C(C(C(=O)N(C)Cc1cnc(C)s1)NC(=O)Cc1cnnn1C)OC c1(CC)cnccc1C(=O)N(C)CC1C2CN(C(=O)CSCC(N)=O)CC12 c1(C(N(CCCN(C(c2c(C#N)cnn2C)=O)CC)C)=O)ccc(=O)n(C)c1 N1(C(CN(CCCCCC)C)=O)C(CNC(=O)CCN(C)CC)CC2COCC12 N1(c2n(C)c(C(c3cccnc3)O)nn2)CCC(C2CC2)C1c1nnc(O)o1 C(CCCCCC(=O)N1CC(SC(F)F)C1)NC(=O)CN1CCCCCC1 C1(CNC(C(CC)C(C)(F)F)=O)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)CC2)O1 CCC(C)(CO)C(=O)N1CC(NC(=O)COc2ccc(F)cn2)C2(CC2)C1 C12(C(=O)NC(CC)C)CC(CO1)N(C(c1c(C)coc1CN)=O)C2 CC1C(C(=O)NCc2nc(N(C)C)n[nH]2)CCCN1C(c1cccnn1)=O CC(C#N)C(=O)N1CC(N(C)C(c2cc(C3CC3)no2)=O)C1 C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(=O)CC(F)(F)F)C2(CCC2)C1 C1(C(N2C(CNC(c3cc[nH]n3)=O)CCC2)=O)CCCCC12CC2 C(CNC(C1CC(OCC)C1)=O)(CC)(CC)NC(c1ccccc1-c1ncc[nH]1)=O c1(NC2CCC(C(=O)NC(C(=O)N(C)C)(C)C)OC2)ncnc(C(F)(F)F)c1Br C1(C(N(CC(CC)NC(COC2(C#C)COC2)=O)CC)=O)C(F)(F)C12CC2 C1(C(C)C)CN(C(c2cnc(OC(C)C)cn2)=O)CCN1C(=O)CCS(C)=O c1(C(=O)OCC)cncc(CN(C2CCCC2)CC2CCNC2=O)c1 CC1CCC(NC(c2cc(C(F)F)n(C)n2)=O)CN1C(c1cnsc1)=O N1(C(CCCCOCC)=O)CC(C)(C)OC2(C1)CN(C(C1CCC(F)CC1)=O)C2 C(=O)(C(C)(F)C(=O)NCCC(C)(C)NC(=O)COC1CCCC1)OC c1(-c2n(CC)cnn2)cccc(NC(C2CCC(NS(=O)(=O)C3CC3)C2)=O)c1 c1(NC(C2CCCO2)COCCCOC)nccc(=NCCC#N)[nH]1 c1(C(N2C(CC=C)CCCC2)C(=O)NCCCC)csc2ccccc2c1=O C1(NC(C2CCC(NC(C3(C=C)CCCC3)=O)C2)=O)CCCCNC1=O n1(CCC)ccc2cc(NCCC3COC4(CCC4)CO3)ccc12 c1(C(N2CC(NC(=O)Cc3cnc[nH]3)C2)=O)cnc(COc2ccccc2)s1 N1(C(c2cc(C(=O)OC)ncc2F)=O)CCC2CN(C(c3ccoc3)=O)CCC12 C1(C(=O)NCCCSCC)(NC(c2conc2C2CC2)=O)CC(O)C1 CC1(C)CCC(C(=O)NC2CCN(C(C3CCCS(=O)(=O)C3)=O)C2(C)C)CC1 CCCC(C(=O)N(C(C)CNC(c1nsnc1O)=O)C)S(N)(=O)=O CS(=O)(=O)c1cc(C(N2CCC(NC(C3CC=CCC3)=O)C23CC3)=O)cc(N)c1 C(=O)(CCCCCNC(c1coc2c1COC2)=O)N(CC(C)(C)C)C1CC1 O=C(CCC#Cc1ccccc1)NCC1COCC1NC(C1(CO)CC1)=O C(C)(CCC(=O)NC(C)C(CO)NC(=O)C(c1ccnn1C)C)SC C(C(CC(C)O)c1ccccc1)NC(N(CCCCC)CCO)=O c1(OC)cc(N)c(C(=O)NCC2CCN(C(C3(C)CCCC3(F)F)=O)C2)cc1F N1(C(C2CC3CC3C2)C(=O)NCCCSC)C2CCC1CN(CC(F)F)C2 c1(CN(C(C)C(O)Cc2ccccc2)C=O)ccc(CC#N)c(F)c1 C(=O)(C1CCCn2cc(C)nc21)NC(C(C)(C)NC(CSCCC)=O)C C1(CC(=O)NC(CC(=O)NC2C(OC)CC2O)C2CC2)CCC(C)(C)O1 CCN(OC)C(=O)C(C)N(C)C(c1nscc1C)=O c1(OC)ccc(C(N2CCCC(O)(CN(C(=O)Cn3cnnn3)C)C2)=O)c(O)c1 c1(-c2cn(C(C)(C)CO)nc2)cccc2[nH]c(C(=O)Nc3coc(Cl)n3)cc12 N1(C(C(=Cc2ccccn2)C)=O)CC2CCC1C2NC(=O)C1=COCC1 CCCCC(CNC(=O)C=C(CC)CC)NC(=O)CC1(O)CCOC1 c1(NCC(N2CCN(CC)CC2)(C)C)ccc(Cl)c(C)c1Cl c1(C(=O)NC(CCNC(c2cc(C)nc(O)c2)=O)(C)C)cc(F)c(C#N)c(F)c1 c1(NC(CNC(C(C)OCC=C)=O)=O)sc2c(c1C(N)=O)CCC2.c1(N)cnsc1 C12(CNC(CCCCCSC)=O)CCC(CN(C(=O)C3=CCC(C)CC3)C1)C2 N1(C(COC)=O)CC(C(=O)NCCCCc2cnn(C)c2O)C(C)(C)C1 C1(CC)(CC)CC(C(=O)NC(COC(C)C)C(=O)NC2CCN(CC)C2)C1 C1(C(N2C(CN(C)C(c3ncc(Cl)nc3Cl)=O)CCCC2)=O)CC2C(C1)C2(C)C Cc1cccc(Cl)c1C(=O)N(C1CCC(NC(c2cc(Cl)cn2C)=O)CC1)C Cc1cnn(C(C)C)c1C(=O)N(C)CC1CCN(C(=O)CC(C)(C)C2CC2)C1 c1(OC)cc(NC(c2ccc3c(cnn3C(F)F)c2)=O)cc([N+](=O)[O-])c1 C1(C(N2CC(C)C(NC(=O)C(C)NC=O)C2)=O)CCCCCN1C N1(C(CCCOCC)=O)CCCC(NC(c2cn3ccsc3n2)=O)C1C N1(C(CCC(=C)Cl)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1C1CCCC1 N1(C(c2cccn3nccc23)=O)CCn2c(n[nH]c(=O)c2=O)C1 Cc1nc(C(C)NC(=O)CC(C2CC2)NC(c2cc(Cl)cs2)=O)n[nH]1 c1(OC)ccc2cc(C(=O)NC3CN(C(c4cnn(C)n4)=O)CC34CC4)[nH]c2n1 C1(O)(C(N(C)CC2CCCN(C(C3(CSC)CC3)=O)C2)=O)CCC(C)(C)CC1 C=C(Cl)CCC(=O)NC(CN(C)C(c1coc(-c2ccccn2)n1)=O)CC CC1C2CCN1C(=O)C1(CC1)CN2.C1(C(=O)ON)CCCCC1c1cccnc1 C(=O)(CCCC(C)NC(=O)CCC1CCC(=O)C1)N(CC(=O)OC)C1CC1 Cc1cccc(C(O)C(N2CCC(NC(c3nccn3C)=O)C2)=O)c1 C(c1nc2ccccc2s1)=CC(=O)NC1CCC1NC(C1CCCCC(=O)N1)=O N1(CC(CC)CC)CCCC(C(=O)NC2CONC2=O)C1 Cc1cc(F)c(C(=O)NC(CO)CCCNC(c2ccn(CCF)n2)=O)cc1F c1(C(n2cc(C3CC4CC4N3C(=O)C(O)C(C)(C)C)nn2)C)c(F)cc(Cl)cc1F CCC(C)(C)C(O)C(=O)NCC(C)NC(c1coc2c1CCCC2)=O c1(C(=O)NC2CCC(NC(CC(CC)C3CC3)=O)CC2)cc2c(Cl)cccc2s1 C1(C)(CNC(c2c(C)n[nH]c2)=O)CN(C(C2CCOC2=O)=O)C(C)(C)C1 C1(CNC(COCCCCC)=O)CN(C(c2cc(CC)[nH]n2)=O)CCC1(F)F NS(=O)(=O)c1n[nH]cc1C(N1CC=CC(NC(=O)C(F)OC(F)(F)F)C1)=O N1(C(CC(C(C)OC)NC(C(CC(CC)(C)C)=O)=O)=O)CCCC(N=[N+]=[N-])CC1 N1(C(C2(C)CCCO2)=O)CCN(C(=O)CNC(C2CC2C(F)(F)F)=O)CC1 N1(C(c2cnn(C)c2Cl)=O)CCC2C(C1)CN2C(=O)Cc1csnn1 c1(NC(COCc2ncc(C)o2)=O)cccc(NCc2c(C)coc2C)c1 C1(CC(=O)NC(C2(C(=O)N(C)CC3CCCC3)CC2)C)CCCCC1 C=C(Cl)C(C)(C)C(=O)N1CC2(C1)CN(C(C1CCCCC1(C)C)=O)C2 N1(C(c2c(C)ccc([N+](=O)[O-])c2)=O)CCC2C(CCCN2C(c2ccsc2)=O)C1 c1(C(N(C2CCN(Cc3nc(CC)sc3)C2)C)=O)cnn2cccnc12 c1(CC(=O)NC2C(CNC(CC(=C)C)=O)CC2)c(F)cccc1Br c1(C(N(CC(=O)NC(CC=C)C)CCOC)=O)cnc(COCC)s1 c1(C(N2CC3(CC(NC(C4CCCCS4)=O)C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1O C(C(C)(C)C(C)(F)F)NC(C1(NC(CCSC)=O)CC1)=O.C(C)(=O)O Cc1nn(C)c(C(N2CCC(N(C)C(c3cncc(N)c3C)=O)C2)=O)c1Br C=CCC(C)(C)CNC(=O)C(C1CCN(C(=O)CN(C2CC2)CC)C1)F C1(N(C(=O)C(C)(C)C2CCOCC2)C)CCN(C(c2ccc(Cl)o2)=O)CC1 c1(C(C(=O)NC2CC(C)(NC(C(C)SC)=O)C2)C)ccc(CC(C)C)cc1 N1(C(CSc2n(C)cnn2)=O)CCCC12CCN(C(c1c[nH]c(C(N)=O)c1)=O)C2 c1(C(N2C3CC(NC(C)=O)CC2CC3)=O)cc2nccc(Cl)c2s1 c1(CO)nc2n(n1)Cc1cc-2nn1C.C1(C)(C2CC2)CC1 N1(C(C(CC)C)=O)CC2(C)CC1(C(=O)N(C)CC)C2 N1(C(Cc2c(C)non2)=O)CC(NC(=O)C(C)OCC2CC2)CC12CCCC2 C1(NC(c2cc(C)c(C)[nH]2)=O)COCCN(C(C2CC23CC(O)C3)=O)C1 c1(CC)nc(=N)[nH]c(=NCCC2CCN(C(c3ccccc3COC)=O)C2)[nH]1 C1(CC(=O)OC)CC2(CCC2)CN1C(=O)NC1CC1C1CCC(N)CC1 C1(NC(CC2C=CC(NC(CC=CCC)=O)C2)=O)CCCCNC1=O C#CCCCC(=O)NC1C2CN(Cc3sccc3Br)CC12 Cc1c(C(=O)NCC=C2CCN(C(=O)CC3(C)CC3(F)F)CC2)cnn1C1CC1 c1(C(N2CC=CC(NC(CCc3c(C)n[nH]c3C)=O)C2)=O)ccc2nccn2n1 c1(C(=O)NCCC2CC(NC(CNS(CC)(=O)=O)=O)C2)ccc(SC)nc1 N1(C(C)C)CCC(C(=O)NC2CN(C(C3CC4CC4C3)=O)CC2O)CC1 c1(CC(N2C(C)CCC(NC(=O)CC(C)(C)C)C2)=O)ccc2nc(O)[nH]c2c1 CN1C2CCC1CC(C(=O)NCC1CN(C(c3ccncc3F)=O)CC1O)C2 N1(C(CCN(c2ccccc2)C)=O)CC(CO)(NC(=O)Cc2n[nH]c(=N)s2)C1 CC(C)C(O)CCN=c1[nH]c(=NCc2ccnc(OCCO)c2)c2[nH]ccc2[nH]1 c1(OCC(N2C(CNC(c3c(C)ocn3)=O)CCC2)=O)ccc(Br)cc1 c1(C(N2CC(O)(CNC(c3c(C)n(C)nc3Cl)=O)C2)=O)n[nH]c2c1CC(C)CC2 Cc1ccc(C(=O)NCC2C=CCN2C(=O)Cc2nncn2C)cc1C C1(C(=O)NCC2(CO)C(C=C)C2)CCN(C(c2c[nH]c(=NC)s2)=O)C12CC2 C(=O)(C1=CCCN(C(=O)CCc2cnc(C(C)NC(=O)OC(C)(C)C)o2)C1)NC c1(C(C(=O)NCC2C(NC(CCC3CC(OC)C3)=O)C2)OC)ccccc1Cl C1(NC(C2C(NC(c3cc(OCC)no3)=O)CC2)=O)CC(C)OC1=O N1(C=O)CC(F)(F)OC(F)(F)C1.N1(N(c2ccccc2)COCC)CCOCC1 C1(CNC(C=C(CCC)C)=O)CC(CNC(c2cnc(CC(C)C)[nH]2)=O)CO1 c1(CCC)nc(C(=O)NCC(C2CCCCC2)NC(=O)COCC(F)F)cs1 C(=O)(C(C(=O)N(C1CCCCC1NC(C12CC(C)(C1)C2)=O)C)C(C)(C)C)OCC C1(C(=O)NCC(C2CCCCC2)NC(c2ccc(C(C)C)s2)=O)CC=CCC1C CCCCCC(F)C(=O)NCC1CC(C)CCN1C(=O)C(C)SC N(C1c2ccccc2CC1O)C(N1CC(C)N(CC(N2CCOCC2)C)CC1)=O N1(C(CNC(c2ccccn2)=O)=O)CC=C(CNC(C2CNC(=O)N2)=O)CC1 Cc1oc(C(C)C)nc1C(=O)NCC1CCCCN1C(C1CCCC(=O)N1)=O c1(C(N2CC3C(CCNC(CC=C)=O)(CC3)C2)=O)nc2ccccc2cc1Cl C(C1(C)CCOCC1)=CC(=O)NCCNC(CN1CCC(C)C1)=O Cc1nccc(C(=O)NC2C=CC(CC(N3CCC(C)(C(N)=O)C3)=O)C2)n1 C1(N(C(c2cncnc2)=O)CC)CCCN(C(=O)C(C2CC2)C2CC2)C1 C1(O)(C(N2CCC(NC(C(=O)NCC)=O)C2)=O)CCSCC1 c1(C(=O)NC(CN(C(C2C(C)OCC2)=O)C)(C)C)ccc(C#N)[nH]1 c1(C(C)C(=O)NCC2CC(NC(=O)C(F)(F)c3ccnn3C)C2)ccc(F)cc1 C1(C(=O)NCCC(C)NC(=O)C(C)(C)c2cc[nH]n2)CCC2(CC1)COCCO2 Cc1cc(CNC(C2CCCC(NC(=O)Cc3cnoc3)CC2)=O)cc(C)n1 CC1(C)CCC1C(=O)NCC1(CNC(C2CS(=O)(=O)C2)=O)CCC1 c1(NC(C23CC(NCc4ccc(OC)c(C)c4)(C2)C3)=O)ccc(C#N)c(Cl)c1 C1(NC(Cc2ncc(C)s2)=O)CCCN(C(c2c(Cl)c(C)nn2C)=O)CC1 c1(C(C)(C)C(=O)NC2CCC(NC(C3CCOC3C)=O)C2)cccc(O)c1 c1(C(=O)NCC2(O)CN(C(C3CC(=O)N3)=O)C2)ncc(Br)cc1F C#CC1CCC(C(=O)NCC2CN(C(=O)Cc3ccc(F)c(CC)c3)C2)CC1 N1(CC(C)C)CC(C(=O)NCC(F)CNC(C2(n3cccn3)CC2)=O)CC1=O c1(C(=O)NC2CCC(C)N(C(c3nccnc3N)=O)C2)c[nH]c2cc(Cl)ccc12 N1(C(C(C(C)c2ccccc2)O)=O)C2CCC1CC(c1cn[nH]c1)C2 c1(NC(C23CC(C(N4CC5CC4CO5)=O)(C2)C3)=O)ccc(Br)c(C(F)(F)F)n1 C(=O)(C1=C(C)OCCS1)N1CC(NC(CCOCC#C)=O)C(OC)C1 Cc1cccc(CC(=O)NCC2CC(F)(CNC(=O)CC3CCCSC3)C2)c1C CC(C)C(O)C(C)C(=O)NCCCCCN(C)C(C1(O)CCCC1)=O C1(NC(c2c(C)cno2)=O)Cc2ccccc2C1NC(=O)C(C)CS(C)(=O)=O CCC(C)CC(=O)C(=O)NC1CCCC(C(=O)NCCSC(F)F)CC1 C1(NC(C2(NC(CC3CCN(C)C3)=O)CCCCC2)=O)CCC(=O)N(C)C1=O C(=O)(C(O)CCNC(=O)C=CCN(C)C)NC1(CC=C)CC1 C1(NC(C2C(C)=CCS2)=O)CCC(C)(CNC(=O)CN2CCNC(=O)C2)CC1 c1(OCC(=O)NC(CCN(C(C)=O)C)C(C)C)ccc2c(c1)CCCC2=O C12(CNC(CC3(C=C)CC3)=O)CC3CC(CC(C3)C1NC(=O)C(F)CC1CC1)C2 Cc1cn2c(n1)CCC(C(=O)NC1CC3CC(O)C1C3)C2 C1(C(N2CCN(CCN(C(c3c(C)occ3)=O)C)CC2)=O)CCC2(C1)CC2(F)F c1(CC(=O)NC2CCC(C(N(CCCC)CCCO)=O)CC2)cccc(C#N)c1 N1(S(C)(=O)=O)CCN(CC(=O)NC2CC(NC(C3(N=[N+]=[N-])CC3)=O)C2)CC1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)NC1CN(Cc2cn(C)nc2)CC1C#N c1(N2CCC(NC(CC(CC=C)(C)C)=O)CC2C)cc(S(C)(=O)=O)ncn1 c1(C(C)=O)ccc(C(N2CCC(N(C(=O)CSCC3CCCO3)C)C2)=O)[nH]1 Cc1ccc(F)c(C(=O)NC(CCN(C(=O)CCCCCF)C)C(C)C)c1O CCCC(C)(CCC)C(=O)NC(c1ccc(C)cc1)CNC(c1cocn1)=O NC1CCc2cccnc2N(C(c2cc(C(F)(F)F)c(Br)s2)=O)C1 C1(CNC(=O)CCF)CC=CCN1C(=O)C(O)CC1CC1 c1(C(C(=O)NC2(C#C)COC2)O)ccc(OC)c(OC)c1 C=CCCCCCC(=O)NC(C)CC(C)NC(c1cc2sccc2[nH]1)=O N1(C(c2cnc(OCC)s2)=O)CC(NC(=O)CC2CNC(=O)O2)C(SC)C1 C=CCCCC(C(=O)NCC(=O)NC(C)(C)C)NC(C1CC12CCCC2)=O c1(C(N2CC3CCN(C(c4[nH]n(C)c(=O)n4)=O)C3C2)=O)cc2ccc(Cl)cc2o1 c1(C(N2CCCC(C)(NC(COCCCOC)=O)C2)=O)cc2c(s1)CCOC2 C1(NC(C=CSC)=O)CC(NC(C2CC2c2cncn2C)=O)C(O)C1 C(=O)(C(Cn1cccn1)NC(=O)NCCC1CC1)OC(C)(C)C N1(C(c2c(OC)cccc2)=O)CCC(C)C(CC(F)(F)F)C1.C1CC(=O)O1 C1(CNC(c2nnn(C)n2)=O)CCC(CNC(C2C3CCC(F)C23)=O)CC1 N1(C(c2cc(C)c(N)cn2)=O)Cc2nccn2CC(NC(=O)CC2CC2(C)C)C1 Cn1cc(C(=O)NCCN(C(C2CCO2)=O)CS(C)(=O)=O)c(C2CC2)n1 Cc1ocnc1C(N1CC(NC(=O)CCN(C)C(=O)OC(C)(C)C)C1)=O C1(NC(C(=O)NC2C(OC)COC2)=O)CCN(C(=O)NCc2ccccc2)CC1 CC1(C)CC(NC(C2CN(C(=O)CC3CC3(C)C)CC2F)=O)CO1 N1(C(c2occ(C)c2)=O)CC2(CCN(C(=O)C=Cc3ccccc3Cl)C2)C1 N1(C(C(c2ccccc2)N(C)C)=O)CCC(N(C(=O)CC2CC=CC2)CCO)C1 CN1CCOC(CONC(c2cccc(C(=O)NS(C)(=O)=O)n2)=O)C1 C(=O)(CN=c1[nH]c2ccccc2s1)N(CCN(C(C(COC)C)=O)C)C CC1CC(NC(=O)CSc2ccccc2)CN(C(=O)Cc2n[nH]c(=N)s2)C1 C(CCCCC(=O)N1CCN(C(c2n[nH]cc2C(C)C)=O)CC1)SC C(CCC(=O)NCC(O)CCC)N(C(CCSCCCC)=O)CCC O=C1NCC2(CN(C(c3nccc4[nH]ccc34)=O)C2)N1.C1(=O)C2=CCN(C2)N1 N1(C(C(CC)Nc2ccccc2)=O)CCCC(NC(=O)CC2CCNC2=O)CC1 N1(C(COCCCC(C)C)=O)CCC(NC(C2CC(C(C)(C)C)C2)=O)CC1C CC(N=[N+]=[N-])C(=O)N(C(C)(C)CC(=O)N1CCN(C(=O)CCO)CC1)C c1(SC)cc(N2CCN(C(c3sc(C)nc3C)=O)CC2)nc(SC)n1 C(=O)(C(CC(F)F)N(C(=O)C=Cc1cnccn1)C)NCC(n1cccn1)C O=C(CCS(=O)(=O)c1ccc(F)cc1)OCc1cscc1C(F)(F)F C1(CNC(C(C)c2ncco2)=O)CC12CCN(C(c1ccoc1Cl)=O)CC2 C(C(CC(=O)N(C)CCS(C)(=O)=O)C(F)F)NC(C(C)(C)NC(C)=O)=O C(=O)(C1Cc2c(Cl)cccc21)NC1CCN(C(c2c(OC)cnc(F)c2)=O)C1C C(Cc1ccccc1)(CC(F)(F)F)NCc1nc(N(C)C)sc1 N1(C(c2cc(C)sc2)=O)CCC(Nc2ncc(C#N)c3ccsc23)C2(CCC2)C1 N1(C(C(COC)O)=O)CC2CCC1C2NC(c1ccc(N2CCCC2)cc1)=O Cc1nc(N2CCC(CCNC(=O)NC3CC(C)OC3C)C2)c(C)c(Cl)n1 C(C)(c1ccccc1OC)=CC(N1C2C(CNC(C(CC)(C)CO)=O)C(C2)C1)=O C=CCCC(C(=O)NCC1CN(C(=O)OC)C1)NC(c1cn(CC)nc1C)=O c1(NC(N2CCCC(CCCC)C2)=O)sc(OC(=O)C2CC2)cc1C N1(C(C=COCC)=O)CCC(C2CCN(C(c3cn(C4COC4)nn3)=O)C2)C1 CCC(C)(CN=c1[nH]c(NCCCc2cnccn2)nc(=N)[nH]1)C(C)O c1(C(N(CC(C)O)CCNC(C2(C)CCCCC2)=O)=O)ccc2c(c1)nnn2C C(=O)(C1=Cc2ccccc2OC1)NC1C2CCN(C(C(C)CC(N)=O)=O)C2C1 C1(NC(C(n2c(C)ccn2)C)=O)CCCC(NC(=O)C(C)OCOC)C1 O=C(CS(=O)(=O)CCO)NCCC1CCCN(C(C2CC3C=CC2O3)=O)C1 c1(NC(COC)CC2CCOCC2)cc(C(=O)NC(C)C)ccc1[N+](=O)[O-] CC1(C)CC(C(=O)NCC2(CNC(C3CC(=C4CC4)C3)=O)CC2)CNC1=O N1(C(CSc2c(C)n[nH]c2C)=O)CCN(C(=O)C(N2CCCCC2=O)C)C(C)C1 C(CC(=O)NC1CCOC1=O)(C(F)(F)F)NC(CCCC=C)=O S(=O)(=O)(c1cnn2ccc(NNCC3CCOCC3C)nc12)N(CC#CC)C C1(CC(=O)N(CCOC)CCNC(c2ccn(C(F)F)n2)=O)CC2CCC1O2 C1(CCCNC(CCN(C(C)=O)C)=O)CCN(C(c2ncsc2N(C)C)=O)CC1 CN=c1[nH]cc(C(N2CC(OC)CC2CNC(=O)C2=CCOC2)=O)o1 c1(-c2nc(C)c(NS(=O)(=O)c3ccc(Cl)s3)s2)c(C)ccc2ncccc12 c1(C(=O)NC2CCCN(C(CC=CCC)=O)C2)ccc2c(c1)oc1ccccc21 c1(C(N2CCC(C(CNC(C(CC)O)=O)(C)O)CC2)=O)ccn2cncc2c1 N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2ncncc2Cl)=O)C2COCC12 CCC(C)(O)C(=O)NCc1c[nH]nc1C1CCN(C(c2cc(C(F)F)n[nH]2)=O)C1 C(=O)(C(F)C(C)(F)F)NC(COC(C)C)C(=O)N1CC=CC1CF N1(C(CC(CCC)O)=O)CCC2CC1CN(C(=O)Cc1cccc(C3CC3)c1)C2 C(=O)(C(CCS(C)=O)N(C)C)N(CC(C)CNC(C1CCC(CC#N)CC1)=O)C c1(CNC2CCC(C(=O)Nc3cc(C)c(Cl)cn3)OC2)c(O)cc(F)cc1F C1(C)(C(=O)OC)CCN(C(=O)CC2CCCN(C(c3cccn3C)=O)C2)C1 O=C1Cc2c(C(=O)NCC(F)CNC(=O)Cn3cnnn3)ccnc2N1 N12CC(O)CC1C2=O.C1(NC(=O)OC)(CNC(=O)C(=O)NCC(F)F)CCC1 c1(CN2C(C(=O)NCCC(=O)OC)CSCC2)ccc(Cl)cc1OC N1(C(C2=C(C)CCC2)=O)CC2=C(C1)CN(C(=O)C(C)(C)C(C)C)C2 C(=O)(C1CCCc2sccc21)N(C1CN(C(CC=CC=C)=O)C(C)(C)C1)C1CC1 C(CC(N)=O)(C(=O)NCC1(F)CCCN(C(=O)C(=O)NC2CC2)C1)NC(CC(C)C)=O c1(C(=O)NCC(CC)NC(c2cccc(=O)o2)=O)c(OC)c(Cl)cc(O)c1Cl C1(C(=O)OCC)CN(C(=O)CC2COCC(C)O2)CCC1=O S(=O)(=O)(c1ccc(Br)cc1N)N(C)Cc1ccc(SC)o1.N12CCCCC1C2 c1(OC)ccc(OCC(=O)NCC2CC(O)CN2C(C2CCCNC2=O)=O)cc1 C#CCCCCCC(=O)NC1CCN(C(c2cnc(C)[nH]c2=N)=O)C1(C)C c1(C(N2CCC(NC(Cc3ncc(C)s3)=O)C(F)C2)=O)ccc2oc(S)nc2c1 N1(C(CCC(C)=O)=O)CC(NC(C2CC2C2CCCC2)=O)Cc2ccccc21 C1(NC(C2CCN(C(C)=O)C2)=O)(CF)CCN(C(c2cncnc2)=O)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(C)(CNC(c2n[nH]c(C)c2F)=O)OCC1 C1(CNC(C2(C#C)CCCC2)=O)CC2COCC2N1C(c1ccco1)=O C1(CNC(C(C2CC2)SC)=O)CCC(NC(c2ccc(C3CC3)o2)=O)C1 c1(C(N2CCOC(C3CC3)C2)C(=O)NCCCF)cnn(C(C)C)c1F C1(C(N2CC(n3cc(CN(CC(C)(C)C)CC)nn3)C(C)C2)=O)CC(=O)NC(=O)N1 C(=O)(C(O)C(C)(C)CC)N1CC(NC(CC(CC)CNC(=O)OC(C)(C)C)=O)C1 N1(C(COCC)=O)CCC(N2CCN(C(c3csnc3Br)=O)CC2)CC1 N1(C(c2cc(OC)ns2)=O)CCC(C2CCN(C(c3ccnn3C)=O)C2)CC1 N1(C(=O)NCc2csc(N3CCCCC3)n2)CC(CC)OC1=O N1(C(CCOCC#C)=O)CC(CC(=O)NCC2(C)CC(C)(C)C2)CC1C c1(C(c2nnnn2-c2ccccc2)NCC(C)OC)cc(F)c(F)c(F)c1 c1(OCC)ccc(NC(=S)Nc2cnc(C(C)O)cn2)cc1OC(C)C c1(C(=O)NCC2CCN2C(=O)CC2(CSC)CCCC2)ccc(F)cc1Cl c1(C(c2nnnn2C2CCOC2)NCCCOC(=N)O)occc1Br c1(NC(C(CC)(C)O)=O)ccc(CNC(=O)C(C)(C)N2CCCC2)c(C)c1 N1(C(C2(SCC)CC2)=O)CCC(C(C)NC(=O)Cc2cc(-c3cccs3)on2)C1 c12ccc3c(c1)C(=O)N(C3=O)COC21CCCC1.COCC C1(NC(C(C=C)OC)=O)CN(C(=O)Cc2cccc(OC(F)F)n2)CC12CC2 N1(C(CN(C)C)=O)CCCCC(NC(=O)COc2ccccc2C(N)=O)CC1 Cc1cc2c(CC(=O)NC3CCNCC3c3ccccc3)csc2s1 c1(C(=O)NC2CC(CCCN(C(=O)C(F)C3CCCC3)C)C2)ccc(C#N)cc1 Nc1c(C(=O)NCC2(NC(C3CC4(CCC4)CO3)=O)CCCCC2)cccc1F N1(C(c2n(C(C)C)ncn2)=O)CCCC1(C)CNC(c1sccc1CC#N)=O c1(-n2cc(CCC3N(C(CCS(C)=O)=O)CCC3)nn2)ccc(Cl)cc1Cl C12(CNC(C(CC)C(C)C)=O)CCC(CNC(=O)CC34CCCC3C4)(CC1)CO2 c1(C2N(C(=O)Cc3n[nH]cc3Br)CCC2)nnc2n1CCC2 Cc1cc(C(N2CC(CNC(=O)CN3C(=O)CNC3=O)C3CC23)=O)cn(C)c1=O CC(C)CC(C)(CO)NC(=O)COC1CN(C(C2CCCCCCC2)=O)C1 Cc1oc(-c2ccco2)nc1C(N1CCOC(CS(N)(=O)=O)C1)C(=O)NC1CC1 c1(C(=O)NCCN(C(c2cn(CCC)nc2C)=O)C)cnc(O)c2cccnc12 N1(C(c2cn(C)[nH]c2=N)=O)CCC(CO)(CNC(C2(Cl)CC23CCC3)=O)CC1 c1(OC)ccc(C(N2CCOC(C(C)Nc3cc(C(N)=O)ncn3)C2)=O)c(C)c1 C1(COC)(NC(=O)Cc2cccn2C)CN(C(=O)CCC2CCOC2)C1 C#CCCC(=O)NC(C1CC1C(=O)NC(c1nn[nH]n1)C1CC1)C N1(C(C2C(C(C)(C)C)CC2)=O)CCCC(C(=O)NCC2CCCC23CC3)CC1 C1(NC(C2C(C=C)OCC2)=O)CCN(C(=O)CC2CCC(OC)CC2)CC1CC C(=O)(C(O)CC1CCOCC1)NCCN(C(=O)C(O)CC1CCOCC1)C(C)C c1(C(N2C(CCOC)CN(C(=O)C=C(C)Cl)CC2)=O)cnn2cc(C)cnc12 O=C(N=c1ncnc2[nH][nH]cc1-2)C1CC12CCN(Cc1cccc(F)c1O)C2 C1(NC(c2c(OC)ncc(Cl)c2)=O)CN(C(=O)CSCCC#N)C2(CCC2)C1 N1(CC#N)CCC2(CCCCN(C(C3(C4CCCO4)CCCO3)=O)C2)C1 c1(C(=O)NCC(n2cc(Cc3nn[nH]n3)nn2)C)cccc(C2(F)CC2(F)F)c1 C(CC(O)C(=O)NCC(CC(C)C)NC(C1CC1C(=O)OC(C)(C)C)=O)SC c1(CCC(=O)OCC(c2c(OC)ccc(F)c2)=O)ccc2ncccc2c1 N1(C(=O)Cc2nc[nH]n2)CCN(C(c2ccc(OC(F)F)c(F)c2)=O)C(C2CC2)C1 N1(C(CCN(C)CC)=O)CC2CCC2(CC(N2Cc3ncsc3C2)=O)C1 N#Cc1cccc(S(=O)(=O)Nc2cc(C(N3CCC(O)(CF)CC3)=O)n(C)c2)c1 CC1CN(C(=O)C(C2CC2)N(C(=O)Cc2ccccn2)C)CCS1=O C1(C(=O)NCC(CNC(c2cnn(CCN(C)C)c2)=O)OC)CCCCO1 c1(N2CCC(NC(C3CN(C)C3)=O)C(F)C2)nc2ccc(O)cc2s1 Cc1cc(C(N2CC(F)(CNC(=O)C(N3C(=O)CCC3=O)C)C2)=O)cc(N)c1 N1(C(c2nc(C(C)C)oc2)=O)CC2CC1C2NC(=O)COc1ccsc1Cl c1(C(C(N2C(CNC(C(C)(C)OC)=O)C=CC2)=O)C)ccc(C(C)(C)C)cc1 CCC(C)(C(=O)NCCCNC(c1ccc(Oc2ccccn2)cc1)=O)OC c1(C(=O)NCC2(NC(C3C(C(C)(C)C)C3)=O)CCC2)ccc2nccn2c1 C(c1ccncn1)=CCc1csc(CNC(CCC(CC(C)(C)CO)(C)O)=O)n1 C1(CC(=O)NCC2C3CC2N(C(c2nocc2Br)=O)C3)CCS(=O)(=O)C1 C1(OCC)CN(C(=NCCN)NCC2CCCCN2C)CC1N(S(C)(=O)=O)C c1(OC)cc(O)ncc1C(=O)NCC(C)CNC(c1cccc(C2CCC2)c1)=O C12(C(=O)NCC3N(C(CCC(CC)CC)=O)CC(O)C3)CCCC(=O)N1CCC2 c1(SCC(=O)NC2(CCCNC(C3(CC)CC3)=O)CC2)ccc(O)cc1 N1(C(C(N2CCOCC2)C)=O)CCC(CNC(=O)Cc2cncn2C)(OC)C1 c1(OC)ncc(Br)c(C(N2CC3CC(C2)N3C(=O)CC2CCCC2O)=O)n1 C1(C(=O)NCC2(CC(=O)NCCCCC#C)CC2)CCCCC1O C(CC(=O)NCc1cccc(C)n1)(C(C)CC)NC(c1c(C#C)c[nH]n1)=O c1(SC)ccc(C(=O)NC2CC2NC(c2n[nH]cc2C(F)(F)F)=O)s1 N1(C(C(CCN(C)C)NC(=O)C#CC(C)(C)C)=O)Cc2cccc(O)c2C1 CCCC(CC(C)C)C(=O)N1CCC(C(=O)N(C2CCCC2)C)C(C)C1 C1(NC(c2sc(CC)c(C)c2)=O)CCN(C(=O)COCC2CCCCO2)C1(C)C c1(C(N2CCN(C(CC=C(C)C)=O)CC2CF)=O)[nH]c2ccc(C)cc2c1Cl c1(CN2CC(NC(c3ccc(O)c(O)c3O)=O)C(F)(F)C2)cc(F)c(Cl)c(Cl)c1 N1(C(C=CC(C)C)=O)CC(NC(c2ccc3nn(C)cc3c2)=O)CC12CCCC2 c1(NCCOCCN(C)C(C2CCC3CC3C2)=O)ncnc2c1nnn2C1CC1 C1(C(C)C)CCc2[nH]nc(C(=O)NC(=O)C3CC3)c2C1.C12CN(CCN1C)C2=O CN1C(=O)CCC1CNC(c1cc(C2CCCC2)nn1C)=O c1(NCC(=O)NCC2CCC(N(C(C(CCC)O)=O)C)CC2)c(C)cccc1Cl C1(C(N(CC(CC)C)C)=O)CCN(C(C2CCCOCC2)=O)CC1 c1(OC)ccnc(C(=O)NC2CCCCN(C(C3CC4(C3)CC4F)=O)C2)c1OC C1(OC)CN(C(C2NC(=O)OC2C)=O)CCC1NC(c1sccc1C1CC1)=O C1(CNC(C2CC(N(C)C)C2)=O)CCC(NC(=O)C(O)CC2CC2)CC1 O=C(C1=CCCOCC1)NC12CCCC1N(C(c1cnns1)=O)CC2 O=C1CCN(C(c2cccc3ncnn23)=O)C2CCCCC12 C1(OC)CC(CC(=O)NC(C(=O)NCCC(=O)NC(C)(C)C)C2CC2)C1 c1(C(N2C(CNC(CC3(C)CC3)=O)COC(C)(C)C2)=O)cc([N+](=O)[O-])ccc1N N1(C(c2ccc(C(C)C)o2)=O)CCCC(O)(CNC(c2nnn3c2CCC3)=O)C1 c1(C(=O)NC2C(NC(C(c3ccccc3O)OC)=O)CCC2)ccc([N+](=O)[O-])[nH]1 C1(NC(=O)Nc2ccnc3c2CNCC3)CCc2nnc(-c3ccccc3)n2C1 C(=O)(C1=NOC2COCC12)NC(CCNC(C=CC)=O)C(C)C C(=O)(C#CC1CCOC1)N1CCC(C(=O)Nc2cccc(F)c2)OCC1 C1(NC(c2n(CC)ccn2)=O)(CO)CCN(C(=O)C(c2ccccc2Cl)O)C1 CC(CC(=O)NCC12CCC(CC1)O2)C(C)(C)NC(=O)C1=NOCC1 CC1CCC(CC(=O)NC2CCCC2CC(=O)Nc2ccc(N(C)C)cc2)OC1 c1(C(=O)NC2CC(C)(CNC(C3(C(=O)NC)CC3)=O)C2)c[nH]c2c(Cl)cccc12 CCC(CCC(=O)NCCOc1ccncc1)NC(=O)C(C)CC(F)F C1(CC)CNC(=O)CN1C(=O)C(CC(C)C)NC(=O)CC1CCCSC1 CC1=C(C)CN(C(=O)CC2CC3(C2)CN(C(c2ccoc2Cl)=O)C3)CC1 c1(C(=O)Nc2c(C(C)(C)C)cccc2)ccc2c(=O)c(C(C)(C)C)c[nH]c2c1 CS(=O)(=O)c1ccc(Br)cc1CC(=O)OCC(=O)N(c1ccccc1)C1CCC1 C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC=CCNC(C(C)C(F)(F)F)=O Cc1nc(C2CC2)ncc1C(=O)NC1CCN(C(C2(C3CC3)CC2)=O)CC1O C1(CC(=O)NCCN(CCC)C(C2CCCCCC2)=O)CCC(F)(F)CC1 C(=O)(CCCCC(=O)NC1CC(CO)N(C(=O)CCNS(C)(=O)=O)C1)NC c1(OC)cccc(Cl)c1C(N1CCN(CCN(C(=O)C(C)CC(C)C)C)CC1)=O c1(C(=O)NCC(CC=C)NC(c2c[nH]cc(C)c2=O)=O)c(F)ccc(C#N)c1F C1(NC(CCCN(C)C)=O)CC(NC(C2OCCC2C(F)(F)F)=O)C(O)C1 c1(C(=O)NCC2(CNC(C(c3c(C)noc3C)C)=O)CC2)nn(C)cc1[N+](=O)[O-] C1(C(C)C)CN(C(=O)C(=O)C(C)(C)C)CCCN1C(c1ccnc(N(C)C)c1)=O N#Cc1cc(C(=O)NCC=CCC(=O)Nc2cccc(CCO)c2)co1 C1(C(=O)NC2CC(OCC(=O)NCc3ccc(F)c(O)c3)C2)CCCC12CCC2 C1(NC(C2(C=C)CCOCC2)=O)CCN(C(=O)CC2CCCN(C)C2)CC(O)C1 CCCC(C(=O)NC1CCOCC1NC(C1(C(C)C)CC1)=O)C(C)C C1(OC)CC(NC(=O)C=C(Cl)Cl)CN(C(c2nn(C)cc2Cl)=O)C1 c1(CSC)ccc(C(=O)NCCCCNC(C2(n3cncn3)CC2)=O)cc1 N1(C(C(COCC)N=[N+]=[N-])=O)Cc2n[nH]cc2C1C(=O)NCC=CCOC C1(CNC(c2c(COC)cc[nH]2)=O)CCCN(C(c2c(Cl)cnn2C)=O)C1 CN1CCn2nc(C(=O)N(CCc3nn[nH]n3)CC3CNC3)cc2C1 N1(C(C2C(NC(c3cnn[nH]3)=O)C3CCC2C3)=O)CCC(C2CCC2)C1 c1(C(N2CC3CC(NC(C4(CCF)CCC4)=O)CC3C2)=O)ccn2cncc2c1 CC1=NC=COCCN2N=NN=C3C=CC(OC(F)F)=CC=C1CCC2NC3 Cc1cc(CC(N2CCN(C(=O)CC3(O)CCCN(C)C3)C(C)C2)=O)ccc1Br c1(C(=O)NCC2C(CNC(c3ncn(CC)c3)=O)C2)cccc(N2CC=CC2)c1 C(=O)(C(C)(C)C(=O)N1CC(NC(=O)CC(C)NC(C2CCCC2)=O)CC(F)C1)NC N1(C(C(C)CSc2ccccc2)=O)CCCC(CO)(NC(=O)C2=CSCCO2)C1 C1(C)(CC)CC(NC(C2CC=CC(NC(=O)CCC3CC3(C)C)C2)=O)CCO1 C1(N(C(C(CCC)N(C)C)=O)CC)CCCN(C(c2nn(C)cc2C)=O)CC1 c1(OC)ccc(C=CC(=O)NCC(O)CNC(=O)C(C(C)C)NC(C)=O)c(C)c1 c1(N2C(C)CC(F)C2)ccc(S(=O)(=O)NCCN2CCOCC2)cc1Cl Cn1ncc(C(N2CC(NC(=O)C3=CCCC3)CC(C)(C)C2)=O)c1S(C)(=O)=O C(=O)(C(F)(F)C(F)(F)F)N(CC(C)(C)NC(c1cc(C)[nH]c1C)=O)C CC(C(=O)N1CC2(CC(NC(C3(OCCNC)CCOCC3)=O)C2)C1)C(C)(C)C c1(C(C(=O)NC(C2CCCN2C(=O)Cc2cocn2)C)(C)C)ccc(Cl)cc1 N1(C(CNS(C)(=O)=O)=O)CCC(C)(C)C(NC(C2(O)CCSCC2)=O)C1 c1(C(=O)NC2CCCC(NC(c3cc(C)c(C)[nH]3)=O)C2)cnc2nccn2c1 Cc1nn2c(c1C(N1CC(NC(c3nccn3C)=O)CC1C)=O)NCCC2 C(=O)(CC1=CCCC1)NCC1C(C)CCN1C(=O)CCOC1CC1 c1(CN2CC(CC(=O)Nc3cccnc3F)OCC2)ccc2c(Cl)ccnc2c1 C1(NC(Cc2cc(C)n(C)n2)=O)CCN(C(c2nnn(C)c2C(F)F)=O)C12CC2 C1(C(=O)NC(C2CCCC2)CNC(c2ncnc(O)c2F)=O)CC12CCSCC2 C1(C(=O)NCCCN(C(CC2C(C)(C)COC2)=O)CCO)CC12CCOCC2 C1(NC(=O)CC2CCOC2)CCN(C(=O)CNC(C2CCC2)=O)CC1CO c1(C(=O)NC(CC2CCN(CC(CC)OC)CC2)C)cnc(C2CC2)nc1C N1(CCC(CC)(C)C)CCC(=O)N(Cc2ccc(CC(N)=O)cc2)C1=O CCCC(C(=O)NCC(C)(C)C1CC1)N1CCNC(=O)C1 N1(C(C2C(NC(C(C)OCOC)=O)COCC2)=O)CCn2ccnc2C1 C#CC1CCN(C(=O)C(CC)NC(c2c[nH]c(C(N)=O)c2)=O)C1 c1(NC(C2CCCC(NC(c3scc(C)c3C)=O)C2)=O)c(F)c(F)cc(F)c1F S(=O)(=O)(c1ccccc1[N+](=O)[O-])NCCCNC(=O)C(=O)NC1CCCC12CC2 c1(N2CCN(c3ccnc(C(C)C)n3)CC2)ccc2c3c(cccc13)CC2 C#Cc1ccc(C(=O)NCC2CC2CNC(=O)Cn2cc(Br)c(C)n2)c(C)c1 CCC(C)C(=O)C(=O)NCC1CC2(CC(NC(=O)CC3CC=CCC3)C2)C1 N1(C(C2(CCC)CCC2)=O)C(C(=O)NCCNC(C2CCCS2)=O)CCC12CC2 C1(NC(C23CC(NC(C(CC)OC)=O)(C2)C3)=O)CCCC(C(C)(C)C)C1 N(C(=NCCCCl)N1CCC(C(=O)NC(c2c(CSC)ccs2)=O)C1)C(C)C N1(C(CCC)=O)CCCCC1C(N1CCC(N(C(c2ccncc2)=O)CC)C1)=O C(=O)(CC1OCc2ccccc21)N1CCC(CCNC(CC(C)O)=O)C1 N1(CC(=O)NC(C)CCN(C(=O)C(F)=CC2CC2)C)CC(=O)Nc2ccccc21 N1(C(C2CCCC23CCC3)=O)CC(C2CC2)(C(N2CCOC3CC23)=O)C1 C1(NC(CC(C2CC2)SC(C)C)=O)CCCCC1NC(C1C(C(N)=O)C1)=O c1(C(=O)NCC2(NC(C(C(C)C)NC(COC)=O)=O)CC2)c(O)nnc(C)c1C C(=O)(C1=CCCCC1)N1C(CC=C)(C(=O)OC)CCC1.C(=O)CCCn1ccnc1 C1(c2cn(CCc3cn(C)nn3)nn2)CCC(N)CC1 CC1CCC(CO)(NC(=O)CCN(C)C(c2cccc(CC#N)c2)=O)C1 N1(C(COCCC)=O)CC2CCN(C(=O)Cc3csc(S)n3)CC2C1 C1(C(N(C2CCCC2)CCC=C)=O)Cc2c(F)ccc(F)c2CN1 Cc1oc(C(N2CCC(CNC(=O)C(O)Cn3cncn3)C2)=O)cc1Br Cc1cc(C#N)nc(N(C2CCNCC2F)C(c2ccc3c(c2)CCO3)=O)n1 N1(c2cc(N(CC)Cc3ccccc3Cl)ncn2)CC2CC(C1)C2C(=O)O c1(-c2cn(CC(=O)NCC(CC)(C)CO)nn2)ccc(C)c(F)c1 CC1=C(C(=O)N2CCC(CC(=O)N(C(C)C)Cc3cnccn3)C2(C)C)CCO1 N1(C(c2cc(C)nc(O)c2)=O)CCC2CN(C(c3cc4sccc4cn3)=O)C2C1 c1(C(=O)NC2CC(C)(CNC(C3CC4CC4C3)=O)C2)cccc2[nH]ncc12 N1(C(C2(CC)CCCC2)=O)CC(N(C(=O)Cc2n[nH]cc2Br)C)C(O)C1 C1(CC=C)(C(=O)NCC(=O)OC)CCN(C(=O)CCCOCCC)C1 c1(CC)nn(C)c(C(N2CCC2CNC(=O)CC2CCC3(CCC3)O2)=O)c1Cl N1(C(C(=O)NCCOC)C(C2CCC2)OCC)CCC2OCCCC2C1 N1(C(C(C)n2ccnc2)=O)CCC2(NC(=O)Cc3ccc(O)nc3)CCCC12 Cc1ccc(Cl)cc1NC(=O)C(C1CCN(C(C2C(C)(C)C2(F)F)=O)C1)F C1(NC(CC=C)=O)CCC2(CC1)CC2NC(=O)CC(CN(C)C)CC c1(C(N(C(CNC(c2nnc(C)s2)=O)C)C)=O)ccc(=O)n2c1CCCCC2 N1(C(c2sccc2I)C(=O)NC(CC)(C)C)CC(=O)NC(C(C)C)C1 c1(N2CCC(NC(c3cc(SC)c(F)cc3)=O)C(O)C2)ncc2c(n1)COC2 c1(N(C)CC2N(C(C(C)OCCN(C)C)=O)CCC2)nccc(S(C)(=O)=O)n1 c1(C(N(CCCCNC(C(C)NC(C)=O)=O)C)=O)c(Cl)cc(C#N)cc1Cl Cc1oc(C(=O)NC(CCN(C)C)C(=O)NC2CCN(C(C)(C)C)C2)cc1CO CCS(=O)(=O)CC(=O)NC1CCCC1CN(C)C(c1ncnc(C)c1C)=O C(=O)(C(C)CS(C)(=O)=O)N1CC2(N(C(COCCCCCCOC)=O)CC2)C1 C1(CC(N2CC(C)(NC(=O)CC3CCCC(C#N)C3)C2)=O)CC2CCC1C21CC1 Cc1c(C(=O)NCCC2(O)CN(C(C3(C)CC=CCC3)=O)C2)[nH]c2ccccc12 N1(CC(=O)NCCSCCCl)C2CCCC1CC(=O)NC2.CC(C)(C)S C1(C(=O)Nc2cnc(-c3ccccc3)s2)CCS(=O)(=O)CC1.C12CCN(CC1)C2 C12(C(=O)Nc3cc(SC)n[nH]3)CC1CN(C(c1ncoc1C)=O)C2 Cc1c(Cl)ccnc1C(=O)NCCC1CCCN(C(=O)COCP(C)(C)=O)CC1 C1(CNC(CC2CCC2)=O)CC(O)C(O)C1.C12CCOC1CNC2=O.CCOC C(CCC(=O)NC(C)CNC(=O)C(C)(C)C1CC1)NC(=O)OC CC1CN2CCN1CC2C(=O)NC1CCCCC1CNC(C12CCCC1C2)=O C1(OC)CC2(C1)CC(C(C(=O)NC1COC1)N(C)Cc1nccn1C)C2 N1(C(C2(CC#C)CCC2)=O)CCC(C(O)CNC(=O)CSC(C)(C)C)CC1 c1(C(=O)NCC2(OC)CN(C(C3CCC(F)C3)=O)C2)cnn2c1CCC2 C1(C(N2C(CCC)COCC2)=O)CC(C)(C)CCN1C(C1CC(=O)CCO1)=O c1(C(=O)NC(C)CF)ccnc(CNC(C2CCCC(F)C2)=O)c1 c1(C(=O)NCCC2CCCN2C(=O)CCc2ncc[nH]2)cc2n(n1)CC(F)C2 N1(C(C(C2CCC2)OC)=O)CCN(C(=O)CCc2conc2C)CCC1C c1(CNC(=NCCOCC=C)NCCC(O)C(C)(C)C)c(C)cc(C)cc1C Cc1cccc2ccc(C(=O)NC3CCC(NC(=O)C(C)O)C3)nc12 Cc1cccc(N)c1C(=O)NC1CCCC(NC(=O)C=C(Cl)Cl)CC1 CCCCC(CCC)NC(=O)C(=O)Nc1cccc(COC)c1 C1(CNC(C(CSC)(C)C)=O)CN(C(=O)CC(F)(F)F)CCC1C c1(N(CCCF)C)nc2c(c(=NCC3(CO)CCCO3)[nH]1)CCC2 Cc1cnc(C(=O)NCC2CN(C(C3CC34CCSCC4)=O)CC2(C)C)cc1Cl c1(OC)ccc(C=CC(=O)NC2CN(C(c3nocc3C)=O)CC2C)c(C)c1 c1(C(=O)OC)ccc(C(CO)N(c2cncc(C(F)(F)F)n2)CCO)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C2C(CNC(C(C(C)C)O)=O)CC(CC2)C1 c1(NC(C2(CC)CN(C(c3cc(O)ccc3C)=O)C2)=O)cnc2ncnn2c1 N1(C(Cc2c(C)cccc2C)=O)CCC2CN(C(c3ccnnc3S)=O)C2C1 N1(C(C(CC=C)C)=O)CCN(C(c2cc(C)c(C)o2)=O)C(C2CC2)C1 C1(CNC(C2(OC)CCC2)=O)CCC(C)(C)CN1C(c1ccncc1)=O c1(NCC2(C)CCCN(C(CC(CN(C)C)O)=O)C2)ncc2c(n1)CCCCC2 C1(NC(C2CC23CCC3)=O)CCCCCN(C(=O)C(F)(F)c2nccs2)C1 Cc1cc(C(F)(F)CNCC2(N)CCOC2)cnc1Cl C=CCC(CC)C(=O)NCCOC(C)(C)CNC(=O)C(C1CCC(C)(C)CC1)C C12(C(C=Cc3cc(C(=O)OC)c(OC)cc3)=O)CCC(C#N)(CC1)CC2 CC(C)C(C(C)NC(=O)COC1CCCCCC1)NC(=O)CCc1cnc[nH]1 c1(C(=O)NC(C)CNC(=O)CC2CCC(=O)N2)cc(=O)n(C)o1 c1(C(=O)NCC(CCNC(c2ccc(C(C)=O)[nH]2)=O)O)ccc(C(C)C)nc1O C(=O)(CC(O)C(C)(C)C)N1CCN(C(C(C(C)C)NC(=O)OC(C)(C)C)=O)CC1C C=CC(CCC)CC(=O)NCC1CCC1NC(c1cc(C#N)c[nH]1)=O C(=O)(C(F)(F)C1=CCOCC1)N1CCC(CCN(C)C(c2ccsn2)=O)CC1 N1(C(CC(CCC)O)=O)CCN(C(=O)CSc2cccs2)C2COCC12 C12(NC(C=CCCC)=O)CC(CNC(=O)C(N3CCN(C)CC3)C)(C1)OC2(C)C c1(C(N(C(c2ccccc2)C(=O)OC)C)=O)ccc(OC(C)C)cc1OC N1(C(C(F)=CCC)=O)CC(OC)CC1(C)CNC(=O)CSc1n[nH]c(C)n1 C1(C(=O)NCCN(C(C)C)C(c2cnn(-c3ccncc3)c2)=O)CCCN(C)C1 c1(C(C(=O)NC(C)CC)N(CCCOC)C)sc(C(=O)OC)cc1C Cc1cccc(OCC(=O)NCC2C3CN(CC4CCCCO4)CC23)c1C c1(SCC(N2CC(C(C)NC(=O)CCn3cccc3)C2)=O)ccncc1 C=CC(CC)CC(=O)NC1CN(C(c2cc(C(F)(F)F)cnc2N)=O)C(C)(C)C1 Cc1cc(CC(=O)NC(C)CC(C)NC(c2cnsn2)=O)ccc1CO CCCCC(C)C(=O)NCc1cccc(CN(C(=O)C=C(C)C(F)F)C)c1 N1(C(C(C)N2CCC2)=O)CC(C(C)(C)O)(CNC(C2CC2(C)Br)=O)C1 CCC(C)(C)C(C)NC(=O)C(C)(C1CCC1)NC(=O)Cn1ccnc1 c1(C(=O)NCC2(CNC(C(CSC)O)=O)CC2(F)F)cc2c(F)ccc(F)c2[nH]1 C(=O)(CC1=CCCCC1)NCCC(=C)CNC(=O)C(F)(F)c1ccnn1C C12(NC(CC(=O)OC)=O)CCN(C(=O)CSc3ccc(C)cc3)CC1C2 N1(C(c2c(Cl)cc(C)s2)=O)CCC(C)C(NC(C2CC3CCC2CC3)=O)C1 C1(CNC(c2cnc(CCCC)s2)=O)CCCC2(CN(c3ncc(O)cn3)C2)O1 S(=O)(=O)(c1ccc(NCc2csc(CO)n2)c(F)c1)NCC1C(C)OCC1 N1(c2n(C(C)C)nnn2)C(C)CCCC1C.C(=O)CCN=[N+]=[N-] C#CCCCCCCCNC(=O)C1=CCC(NC(=O)C(C)=CC=C)C1 C=CC1(C(=O)N(CC(C)(C)COC)C)CCN(C(=O)C(C)CC(=O)OCC)CC1 N1(C(c2c(OC)nsc2)=O)CC2CC(C(=O)NC(C)(C)CNC(N)=O)C(C2)C1 C1(NC(=O)Nc2ccc(OC)cc2)CC2(C1)CC(Nc1nccnc1C#N)C2 CC(C)CCCCCC(=O)N1CCC(C)C1C(=O)NCCN1CCOCC1 C1(C)(CNC(CC2CC(OCC)C2)=O)CN(C(c2cnc(C)c(N)c2)=O)CCO1 C1(C(N(C2CCN(C)CC2)C)=O)CCC(O)CN1C(c1nnc(S)n1C)=O C=CC(C)(C)CC(=O)NC(C)CCN(C(=O)C(O)C1CCCC1)C O=C(CC1=CCCCC1)NCC1CCCC(NC(=O)CCCc2cnccn2)C1 C1(CNC(c2cnn(-c3nccs3)c2)=O)CC(F)CN1C(=O)CO CN1CCC(C(N2CCCC(CCCO)C2)=O)(NC(c2scnc2C(F)F)=O)C1 C1(NC(c2ccc(C)c(C)c2)c2nnnn2C(C)C)CC2(CCCOC2)C1 N1(C(C(COC)OC)=O)CC=CC(NC(C2(CC3CC3)CCC2)=O)C1 N1(CCCc2ccccc2Sc2ccc(Cl)cc2)CCOC2(CCCC2)C1 C1(CSC)CCCCN1C(C1CC1C(C)NC(c1cn(C(C)C)nc1C)=O)=O c1(CCN(C2CCN(C(=O)CC3COCCO3)C2)C)c[nH]c2ccccc12 Cc1cncc2nc(CC(=O)NCC3(C4=CCOCC4)CC3)cn12 CC1(C)CCC1C(=O)NCC1(NC(C2(c3ccccc3)CC2)=O)CCC1 CN=c1ccc(Br)c(C(=O)NC(C)CN(C(=O)CCC=CC(C)C)CC)[nH]1 c1(C(N2CC(CC(N3CCC(CO)C3)=O)C2)=O)c(OC)cccc1CC C(=O)(CC(C(=O)N1CCC(C2CCCN2C(c2ccns2)=O)CC1)N(C)C)OC N1(C(CCC2(NC(CCCC)=O)CCC2)=O)CCN2CCCC2C1 C1(OC)CC(NC(C2(C3CCC3)CC2)=O)CN(C(=O)COC2CCCC2)C1 C=CCC(CC)C(=O)N1C(CC(N2CC(C)CCC2CC)=O)C2CCCC12 Cc1ccc2c(C)c(C(=O)NCC34CC3CN(C(=O)CCC3CC3)C4)[nH]c2c1 c1(CN=C(NCC2(CC)CCC(=O)N2)NCCSCC)ccc2c(c1)oc(=O)n2C C1(C(N2CC(CNC(=O)Cc3ccno3)C2)=O)CC12C(=O)Nc1ccccc12 C(=O)(C(CO)C(F)(F)F)NCC(=O)NCc1nccc(OC)c1 C(=O)(CC(c1ccccc1)Nc1ccc(SC(=O)OC)o1)OCC C(=O)(C(C(=O)OCC)C(C)C)NCC1(F)CN(C(CSCC(=O)NCCOC)=O)C1 C1(NC(C2(C)CC(N(C)C(c3cc(C(N)=O)co3)=O)C2)=O)CCN(C)C1=O C(CC(C)(C)C(=O)N1CCCOC(CNC(c2cc(C)sn2)=O)C1)OC c1(CC(=O)NC(CN(C(C2C(OC)CCC2)=O)C)C)ccc(Cl)cc1 C(C1=CCN(C(C2(C)CCCC2)=O)CC1)NC(C(CC)Oc1ccccc1)=O C(CCCC(=O)N1CCC1C(C)C)N(C(C(C)(C)OC(C)=O)=O)C C1(C(N(C(C)C)CCN(C)C(C2CCC(F)C2)=O)=O)CCn2ncnc2C1 C1(CC#C)(C(=O)NCCCCCNC(c2cnc(COC)[nH]2)=O)CC=CCC1 N1(C(C(=O)NCCOC)=O)CCC12CN(C(c1ccc(C(C)=O)nn1)=O)C2 C1(NC(c2c(C)cno2)=O)CCCC(NC(c2c(Br)n[nH]c2C)=O)C1 C1(C#CC(=O)NC2COCCN(C(=O)CC(C)C3CC3)C2)(CC)COC1 c1(C(N2C(CC)C(NC(c3csc(C)c3)=O)CC2)=O)csc2ccccc12 C1(C2CCOCC2)(C(N(C)CCN(C(=O)C(C)(C)C(N)=O)C)=O)CCOCC1 N1(N(C(=O)Cn2cccn2)CCC2(C(F)(F)F)CC2)CC(C=O)CC1=O.C C1(CC)CCCN2C1C(=O)NC(C(C)OC)C2=O.C1(C)CCCN1C(C)=O Cc1cccc(C(=O)NC(C2CN(C(c3cc(Cl)ccn3)=O)C2)C)c1[N+](=O)[O-] C1(NC(C(COC)(C)C)=O)CC12CCN(C(C1CC(CF)C1)=O)CC2 N1(S(c2c(CC(=O)OC)cccc2)(=O)=O)CCS(=O)(=O)N2CCOCC12 CC1(C(N2CC=CC(NC(=O)Cc3ccsn3)C2)=O)CCC2(CC1)OCCO2 C12(C(=O)NCC#CCNC(c3nc(C)n(C)c3)=O)CC(CO)(C1)OC21CCC1 c1(CNC2C(C(=O)Nc3nc(C)c(Cl)s3)C2)ccc2cc[nH]c2c1 CCCCCCCCCCOc1c(Cl)cc(C(=O)OC)cc1Br C1(CN(C(=O)CCC2CCCCO2)C)COCCN1C(=O)Cn1cnnn1 C1(O)(CCC)CCN(C(c2c(CNC(=O)C(C)NC(C)=O)nnn2C)=O)CC1 N1(CC)N=C(C(=O)NCC(O)CCNC(=O)CC2CSCCS2)CCC1=O Cc1nc(NC(c2sc(Br)nc2C)=O)sc1C(N1CC2C(CO)C2C1)=O C1(NC(N)=O)CCN(C(=NCC2CCCN(CC(F)F)C2)NC2CCC2)C1 c1(C(N2CCC(NC(C(C)SCCCC)=O)C2)=O)cccc(C)c1[N+](=O)[O-] N1(C(C2(COC)CC2)=O)CC2CCC1C(CNC(=O)C(O)CC(C)C)C2 CC1CCN(C(c2nncn2C2CC2)=O)CC1NC(=O)CSCCC(F)(F)F c1(SC)cc(C(=O)NCC2CN(C(=O)CCC3CC3(C)C)CCO2)c(C)o1 N=c1nnn(CC(=O)NC2CC(CNC(c3ccsc3Br)=O)C2)[nH]1 CC12CN(C(c3ccc(OC(F)F)cn3)=O)CC1CN(C(C1CCCCS1)=O)C2 C1(CNC(C(C=C)O)=O)CN(C(C2CSC2)=O)CCN1C c1(N(CCCCCNC(C2C(C(=O)OC(C)(C)C)CCO2)=O)C)c[nH]ccc1=N CCC(CC(=O)NC1CC=C(C(=O)NCCCCS(C)=O)C1)C(C)C c1(C(=O)NC2CCCN(c3nnc(C)o3)C2)ccc(O)nc1C N1(C(C23N(C(C#CC)=O)CC(CO)(C2)C3)=O)C2CCC1CC(OCC)C2 C(c1ccc(F)cc1)=CC(=O)NC1CC(CNC(C(COC)C)=O)C(O)C1 N#Cc1cc(N(CCNC(c2csc(Cl)c2Cl)=O)C2CC2)nc(C2CC2)n1 Cc1cc(C)c(S(=O)(=O)N2CCC(N(C)Cn3nc(C)cc3C)C2)c(C)c1 Nc1ccc([N+](=O)[O-])c(C(N2CCN(C(=O)Cc3cocn3)C3(CC3)C2)=O)c1 C1(C(=O)NCCN(C(=O)C=C2CCCC2)CCC)CCCN(c2nccn2C)C1 CC(C)CC(CC(=O)NCC1(NC(=O)CC2(C)CCC2)CCCC1)CC(N)=O Cc1ccnc(-n2cc(C3(F)CN(C(C4CC5(C4)CC5F)=O)C3)nn2)n1 C1(NC(C2CC(=C)C2)=O)CCCCC12CCN(C(C1CCCN1C(C)=O)=O)CC2 c1(C(N2C(C)CC3CNCC23)C(=O)NC(C(=O)OC)C)ccc2ncccc2c1 c1(C(N2C(C)CCC(NC(c3c(C)cncc3)=O)C2)=O)cc(C)cc2c1CCC2 Cn1ncc(C(=O)NC2CC(F)(CNC(c3ccc(C(F)F)cn3)=O)C2)c1F C(=O)(CS(=O)(=O)C1CC1)N1C(C(C)C)C(NC(c2cc(F)cnc2O)=O)CC1 c1(C2C(C(N(C(C(=O)N3CC(COCC)C3)C3CCC3)C)=O)C2)ccccc1F N1(C(C)=O)CC(F)(F)CC1C(=O)N(CCc1ccccc1)Cc1ccccc1C C(=O)(C1CCCc2nn(C)cc21)NCC1(O)CC(NC(c2n(CC)ccc2)=O)C1 CC(C(=O)NN1CCCCC1=O)NCC.c1(O)ccc(Cl)cc1 C(CCC(O)CO)NC(C=CCN(C(c1ccc(COC)s1)=O)C)=O n1(CC(=O)NCC(CCNC(CC(C)CN(C)C)=O)O)sc(=O)c2ccccc12 c1(C(N(CCCNC(c2c[nH]cc2-c2cnn(C)c2)=O)C)=O)ccc(N)cn1 Cc1ncc2n1CC(C(=O)NC(C)CC1(O)CCC1)CC2 N1(C(C2(C(C)(F)F)CC2)=O)CCCCC(NC(c2ccc(CO)cn2)=O)C1 c1(C(N(CCNC(c2cccc(OC)n2)=O)CC)=O)ccc2c(c1N)CCCC2 N1(C(CCC=C(C)C)=O)CCN(C(=O)C#CC(C)(C)C)C(C)C1 C1(C(=O)NC(C2(O)CN(C(=O)CCCn3cncn3)C2)CC)CCCCC1OC N1(Cc2c(C)scn2)CC2C(C(=O)Nc3n[nH]c(C)c3Cl)C2C1 c1(CC(=O)NCCCNC(=O)Cc2cn[nH]c2)c(F)cccc1F c1(C(N2CC(CC(=O)NCCOc3ccccn3)C2)=O)ccc(C(F)F)cc1F c1(C(N(C)CCC2CCN(C(c3cnc(Cl)cn3)=O)CC2)=O)cnc(O)nc1O Cc1cc(Br)c2nc(CNCc3cc(F)c(C#N)c(F)c3)ccc2c1 C(CNC(=O)Cc1cncc(C)c1)(CC(C)C)NC(C1CCC(OC)C1)=O C1(NC(c2ncccc2CO)=O)COC2(CCN(C(=O)C3=CCOCC3)CC2)C1 c1(OC)cc(C(=O)NCC(F)CNC(=O)C(C(C)O)N(C)C)cc(Cl)c1O N1(C(c2nc(CC)oc2C)=O)CC(OC)CC1(C)CNC(c1cc(C)cc(C)c1)=O C1(CNC(c2cnn(C(C)C)c2Cl)=O)(NC(C2CCC2)=O)CCCCC1C N1(CC(N2CC(O)(CN(C)C(c3n[nH]c4c3COC4)=O)C2)=O)CCS(=O)(=O)CC1 C(=O)CC(C)(O)CCC.N1(CCCC)CCC(NC(=O)CC)CC1 CCC(C)CCC(=O)NC1CCN(C(c2cc(Br)cn2CC)=O)C1C C1(OCC)CC2CN(C(=O)C(C(C)CC)NC(c3nscc3C)=O)CC12 Cc1cc(C(=O)NC2C3CN(C(c4nocc4Cl)=O)CC23)cn1C(C)C Cc1cc(Br)cnc1C(=O)N(C)CCN(C(=O)CC1OCCC1(C)C)C C1(CC(=O)NC(C2(NC(=O)CN3CCCC3)CCC2)C)COC(C)(C)C1 CCCCC(C)C(=O)NC1(COC)CCN(C(=O)C(C2CCCCC2)O)CC1 C=C(C)C(C)(O)C(=O)NC1CCCC1NC(c1ccn(C(C)C)n1)=O C(=O)(C1Cc2ccc(F)cc21)N1CCC(CNC(CCC(C)C)=O)C(C)C1 c1(OC)ccccc1C(=O)NCC(C(C)(C)C)NC(=O)CCc1cc(C)[nH]n1 c1(N(C(CC)(C)C)C(CCOC(C)C(C)CC)c2nn[nH]n2)nc(C)c(C)o1 N1(C(CCCCCCCSC)=O)CCN(C(=O)CSC)C2CCCCC12 C(=O)(CCN(C)CCNC(=O)CSC)NC(C#C)C1CC1 N1(C(c2cnc(OCC)nc2)=O)CCOCC(NC(=O)CC2CC(C)C2)C1 N1(C(C2CC(NC(c3c(C)cn(C)c3)=O)C2(C)C)=O)CCS(=O)CC1C c12ccc(cc1)C(c1ccccc1)Nc1cc-2cs1.c1(S(C)(=O)=O)ccccc1 c1(C(=O)NCc2cn(C3N(C(C=CC)=O)CCC3)nn2)ccc2cnc(C)n2c1 C12(OC)CCCC1N(C(=O)CC1CCOCC1NC(=O)OC(C)(C)C)CC2 C(=O)(C1=CNS(=O)(=O)N=C1C)N1C(C)CCC(CNC(CCCOCCC)=O)C1 c1(C(=O)NC(CN(C(=O)Cc2ccc(Cl)c(F)c2)CC)C)cc(N)ccc1C C(=O)(C(O)CC(F)(F)F)NC(C)CC1CN(C(C2CCCCN2C)=O)C1 N1(C(C(C)(C)c2ccno2)=O)CCCC(CNC(=O)CSc2ccccc2O)C1 c1(CC)ccc(C(=O)N(CCCCCNC(=O)Cc2cnccn2)C)c(F)c1 c1(C(=O)NCC(CNC(CCC(C)OC)=O)OC)ccnc(C)c1C C1(C(=O)NC2CCN(CCCNC(C(C)(C)C(F)F)=O)C2)CCOC2(CCC2)C1 N1(C(C2(C)CC2(F)F)=O)CCOC2(CCCN(C(=O)Cc3cnns3)C2)C1 CCC(C(=O)NCC1CCCN1C(C1CCC=CCCC1)=O)C(C)C N1(C(CCCCC(N)=O)=O)CCC(C2(NC(C3(F)CCCCC3)=O)CC2)CC1 Cc1ccc(O)c(C(=O)N(CC(C)C(=O)NCC2CC(C)(C)CO2)C)c1 c1(C(=O)NC2CC(NC(c3c(OC)c(Cl)ccc3)=O)C2)cc2ncn(C)c2cn1 c1(C(=O)NCC2C(C)CCN2C(c2cccc(N)n2)=O)cnc(O)n(C)c1=O CCCC(O)CC(=O)NC1CC(C)CN(C(=O)CCC(=O)c2cnn(C)c2)C1 c1(CC(=O)N(C(C(=O)N(C(C(C)SC)C)C)(C)C2CC2)C)ncccc1F C=C(C)CN=C(NCC(c1ccncc1)C)N1CCC(NC(=O)NC)C1 c1(C(C(=O)NC2CCN(C(c3nn[nH]c3Cl)=O)CC2)(F)F)cc(Cl)ccc1F c1(C(=O)NC(CCC)C2CC2)sccc1CNC(=O)CCc1ncnn1C c1(N(CCC(CC)O)C(=O)C(N2CCC(O)CC2)=O)ccc(C(=O)OC)cc1 CCC(C)CCC(=O)NC(C)(C(=O)N(CC(C1CC1)OC)C)C1CCC1 c1(CC(=O)N(C)CC2N(C(CN3C(C)CC3)=O)CCOC2)noc2ccccc12 C(=O)(C1CCCc2ncccc21)NCC(CNC(c1scc(C)c1C)=O)C C1(C#CC(=O)NCC2C3CCC(C3)N2C(=O)COCCOC)(CC)CC1 C1(C(C2(O)CCOCC2)C)NC(=O)N(CCc2nccs2)C1=O c1(CC(N2CCC(Sc3cc(C(=O)OC)c(O)cc3)C2)=O)cc(C)cc(C)c1C C(=O)(C(O)CC[S+](C)C)N1CCC(N(C(=O)COCC2CCC2)C)C1 C1(C(=O)NCC2=CCN(C(c3c(C)nco3)=O)CC2)CCC2C(CC1)C2(F)F Cc1cc(NCCC#CCN=[N+]=[N-])cc(C)c1S(N)(=O)=O c1(NC(C(C)NC2(C(=O)NC34CC(C)C3C4)CCCC2)=O)ccccc1Cl c1(C(c2n(CCCC)nnn2)NCc2cnn(CCF)c2)cnc(OC)c(F)c1 C1(n2c(COC)ncc2)CCN(C2CNC(C)C2)CC1 C1(COC)(CNC(=O)CCF)CN(C(C2(C)CCCO2)=O)C1 N1(C(=O)C2CC2)CCN(C2CCN(C(=O)C(=O)Nc3n(C)ccn3)CC2)CC1 S(=O)(=O)(c1cccc(N2CCCC(CC(F)(F)F)C2)n1)NCCC(=O)N(C)CC C1(CNc2n(C(CCC)C)ncc2)COCCN1Cc1ccccc1 C1(C)(CC(=O)N(CC#C)CC2CCCC2)CCN(C(=O)C(C)CN(C)C)C1 c1(C(=O)NCC23N(C(CCC)=O)CCC2CCCC3)cc2ccccc2c(O)n1 C(N=c1[nH]c(=NCCCCS(N)(=O)=O)[nH]c2c1SCC2)C1CCCC(CC)C1 C(=O)(N=c1ccn(CC2CC2)[nH]1)C1N(C(C=CC2C(C)C2(Cl)Cl)=O)CC(C)(C)C1 C1(CCCNC(C(C2CCC2)OC)=O)CN(C(=O)CC2CCCC(C)O2)CCO1 CCCC(O)C(=O)N1CC(CNC(C2CCCN(C(C)=O)C2)=O)C(C(F)(F)F)C1 Cc1cc(C(N2CCC(C)(NC(=O)Cn3ccnn3)C2)=O)ncc1Br C1(C(=O)NC(CC)CNC(c2ccnn2CC2CCC2)=O)CC2C=CC1C21CC1 C(CCC(=O)N(C)CC1(CSC)CN(C(=O)C=CC(=O)N(C)C)C1)OCC c1(C(C)C)cc(-c2nc(CN3CCC(CC(=O)N(C)C)CC3)cs2)ccc1F N1(C(c2c(CC)occ2)=O)CC2(C1)CN(C(c1cnn(C)c1Cl)=O)CCO2 c1(OC)cccc(C(=O)NC2(C3CN(C(C4NC(=O)CC4C)=O)C3)CC2)c1O C(Cc1cc[nH]n1)(C(=O)NCC(C)CC1CCC1)NC(C=CCC)=O CCCCCC(C)CC(=O)NC1CC(F)(CNC(c2cnc(C(C)(C)C)o2)=O)C1 N#Cc1cc(S(=O)(=O)N2CCC(F)(C(=O)O)C2)ccc1NC1CC1 N1(C(C2N(C(c3ncc(OC)nc3)=O)CC(O)C2)=O)CC2(CNC(=O)N2C)C1 Cc1cc(C)c(C(=O)NC2CCN(C(C3COC4(CCC4)C3)=O)CC2O)c(S)n1 c1(OC)cc(C(F)(F)C(=O)NC2CC(CNC(C3CCCO3)=O)C2)ccc1C C1(CNC(c2ccc(CC=C)s2)=O)CCCCN1C(=O)C(C)CC1CCCC1 C(C(C)(CC(C)C)NC(c1cnc2n1CCC2)=O)NC(c1c(C)sc(Cl)n1)=O Cc1c(C(=O)NC(CC2CC2)C(=O)NCC(c2ccsc2)C)nnn1C C(=O)(CCC(=O)N1CCCC(N(C(=O)CCCc2cc[nH]n2)C)C1)NCC c1(C(N2CC(NC(C(C)NC(=O)NC)=O)C(C)C2)=O)n[nH]c2cccc(OC)c12 C(C)(CC(=O)NCC1C2CC1N(C(=O)C=Cc1cc[nH]c1)C2)(C(F)F)N(C)C C(N=c1[nH]c(C(=O)Nc2ccnc(Br)c2F)cs1)c1cc(OC)ncc1 c1(C(=O)NCCC(C)NC(=O)Cc2nnc(O)s2)cc(Cl)cc(Cl)c1 C1(C(=O)OC)CCC(C(N2CCCC2CCNC(=O)C(C)SC(F)(F)F)=O)CC1 N1(C(C(N2CCOC2=O)C)=O)CC2CCC(C1)C2CNC(=O)C(C)C1CCCC1 N1(C(C2(C#N)CC3(CC3)C2)=O)CC2COCCC2(NC(=O)CC2CCCC2)C1 C1(C(=O)NCC(C)(C)CNC(=O)CCC(=O)N2CCC2)CCC(C(F)(F)F)N(C)C1 N#CC(C(=O)N1CCCC1C(=O)NCCCc1ccccc1)c1ccccc1 N1(CC(C2CCOCC2)OCC)C(=O)CN(CC(n2cc(Br)cn2)C2CC2)C1=O C1(c2n(CC=C)nnn2)(NCc2n[nH]c(C3CC3)n2)CC2CCCCC12 N1(N(c2n[nH]cc2I)C2CCN(C(C)=O)C2)CCC2(CCOC2=O)C1 N1(S(=O)(=O)c2cc(Br)c(Br)s2)CCc2cc(F)ccc2C1 C(=O)(CCC(C)NC(c1cnn(C)c1N)=O)NC(C)C(=O)NCC(F)F c1(CNC2(C(C)O)CCOCC2)[nH]nc2c1CNC2(C)C C(c1ccccc1)=CC(=O)NC(C)C(=O)N(C1CCN(C)C1=O)C C1(C(N2C(C(N3CC(F)C(F)C3)=O)C=CC2)=O)C2Sc3ccccc3C12 c1(C(N(CCNC(c2cnn(CCOC)c2)=O)CC)=O)cc(Cl)sc1Cl C(=O)(C1CC(=O)c2c(F)cccc21)NCC(CO)NC(C(CC)=CC)=O c1(C(=O)NCC2(NC(C3CC(=O)NC3)=O)CCOC2)ccc2nc[nH]c2c1F c1(CCC(=O)NCCN(C)C(C2CC2Cl)=O)ccc2ncsc2c1 C(=O)(C1=CCCOC1)NCC(c1ccccc1)NC(C12C(CN(C(C)=O)C1)C2)=O C1(C(N2CCN(C(CC(C)C)=O)C(C3CCC3)C2)=O)CN(S(=O)(=O)N(C)C)C1 Cc1c(C(=O)NCC2CCC(NC(c3occc3C(C)C)=O)C2)c(Cl)nn1C C(=O)(CCCC(=O)N(C)C)NCC=CCNC(CCC=CC(C)C)=O S(=O)(=O)(c1cc(Br)c(F)cc1F)N1C(C)(C(=O)Nc2c(Cl)ccc(OC)n2)CC1 c1(CC(N2CC(NC(C(CC=C)C)=O)C(CC)C2)=O)cc(Br)ccc1C N1(C(CCc2cn(C)nc2)=O)Cc2[nH]nc(NC(C3CCSCC3)=O)c2C1 c1(OCC(=O)NCC(C)(C)CNC(c2csc(O)n2)=O)ccc(F)nc1 c1(CC(=O)NCC2CCCC(NC(=O)CSC(F)(F)F)C2)cccnc1Cl CC(C)CC(C(=O)N(C(C)C(=O)NCC1CNC(=O)CO1)C1CC1)C(N)=O CC(C)(C(=O)NCC1(F)CC(NC(=O)CCc2cnco2)C1)n1cnnn1 C1(OC)CCCC(C(N2CC(CO)(NC(=O)Cc3conc3C)C2)=O)C1 c1(C(N2C(CNC(C(C)Cc3cnc[nH]3)=O)CC(F)C2)=O)c[nH]c2ncccc12 c1(NCC2CC(F)C23CCC3)ncnc2[nH]c(I)cc12 CCN=c1[nH]cc(C(=O)NCC(C2CC2)NC(c2cccc(C3CC3)c2Cl)=O)s1 c1(CN2C(C)CCC2C(=O)NC2CN(C)C2)ncn2ccccc12 c1(CCC(=O)NCCCCN(C(=O)CC2CC(O)C2(C)C)C)cccc(F)c1F C(=O)(C(O)CC(N)=O)NC(C1CN(C(=O)CCc2cncs2)CCO1)C c1(SCC)ccnc(NS(=O)(=O)CCCn2cnnn2)c1.C=O c1(CCC(N2CC(NC(C3C4CNC(=O)C34)=O)C2)=O)cc(Br)ccc1F C=CC1(CNC(=O)C(C2(O)CCC2)NC(C2CCC(=O)N2C)=O)CCOCC1 c1(NC(C(COCC)C)=O)ccc(O)c(C)c1C C(=O)(CCP(C)(C)=O)N(C1CCCCC1NC(=O)CCc1csc(=N)[nH]1)C c1(CC)ccc2c(c1)C(NC(C13CCCCC1NC(=O)C3)=O)C(=O)N2 C1(CNC(C2(NC(CCCOC(C)=O)=O)CCOCC2)=O)CC1C1CCCC1 c1(C(=O)NC2(CCNC(C(C)=Cc3ccsc3)=O)CC2)cc(C2CCCC2)on1 c1(C(N(CC(C)NC(c2cc(C(C)=O)cn2C)=O)C)=O)c[nH]cc(F)c1=O c1(C(N2CC3CC2CN3C(c2cnc(Cl)s2)=O)=O)cc2ncccn2n1 CC(C(=O)NCc1ccc(CNC(c2cnc(S)[nH]2)=O)c(F)c1)C(C)(C)C c1(CC)nn(C)c(OC)c1C(c1nnnn1C1COC1)NCC1CCSC1 Cc1cn2cc(C(N3CCCC(NC(C4CC(C)C4)=O)CCC3)=O)cc(C)c2n1 c1(C(N2CCC(NC(CCC=C)=O)CC2C2CC2)=O)ccnc2c1cnn2C Cc1cc(C(N2CCC(O)(CCNC(c3ccco3)=O)CC2)=O)c(Cl)cc1F C(N=c1cc[nH]cc1S(=O)(=O)NCC1CC12CCOC2)c1c(OC)cccc1F c1(COCCSCC(=O)NCC(CNC(C2(C)CCC2)=O)O)ccccc1 Cc1cc(NC(=O)CCC2CCCN2C(=O)Cc2ccccn2)cc(C)c1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC2CN(C(=O)Cn3cc(OC4CC4)cn3)CC12 N1(C(C2(CC)CCCN2C(c2ccc(C)o2)=O)=O)CCC(OC)C(C)(C)C1 c1(OC)nc(C(N2CCC(NC(c3ccc(C)c(C)c3)=O)CC2C)=O)cc(O)n1 c1(C(N(CC(C)O)CCF)=O)cc(Br)c2occc2c1 C(=O)(C(C)CC(C)C)N(CCCNC(C(=Cc1cnc[nH]1)C)=O)C1CC1 CCCCC(C)(F)C(=O)NCC1CCCCN(C(c2cn(C)nc2C)=O)C1 N1(C(CCC(=O)N(C)C)=O)CCCCC(C(=O)NCc2ccc(CO)cc2)C1 N1(C(C(COCC)C)=O)CC(C)(C)CCC1CNC(c1cscc1C(F)(F)F)=O C1(C)(CNC(C(C)(C)N(C)C)=O)COCCN(C(=O)C2=CCCCC2)C1 N1(C(c2cc(F)c[nH]2)=O)CC2(CCN(C(c3ccccc3C3CC3)=O)CC2)C1 C=C1CCC(C(=O)NC2CC3(C2)CC3NC(=O)CNC(=O)OC)CC1 CC1CC(CNCCCN2CCCN(C(=O)OC(C)(C)C)CC2)CC(C)C1 c1(CC(=O)NCCCCCCNC(CSS(C)(=O)=O)=O)ccc2cccnc2c1 c1(N2CC3CN(C(C4CCN(C(C)=O)C4)=O)CC3C2)ccc2nccnc2n1 CC1=C(F)CN(C(=O)CNC(c2cc(C)n(C)n2)=O)CC1 c1(C(N(CCCNC(C(C(C)C)SCC)=O)CCO)=O)cn(C)c(=O)cc1OC CCCCC(O)C(C)C(=O)NCC(CNC(c1cnc2cc[nH]c2c1)=O)CO N1(C(C2C(C)(C)C2C#N)=O)CCOC(C)(CNC(c2coc(C(F)F)c2)=O)C1 c1(CNC(C2CC(F)CN2C(C2CCCS2)=O)=O)c[nH]c2ccc(Br)cc12 N1(C(c2ccc(C)nc2)=O)CC(O)CCC1C(N1CCC(C(C)C)CC1)=O N1(C(C2CC(C(=O)OC)C2)=O)CC(CNC(=O)CC2CCCN2C)CC1(C)C N1(C(C(c2ccc(C)s2)C)=O)CC(NC(C2CC2C)=O)CC(C)(C)C1 c1(C(=O)NC2CC(CNC(C3(C)CCCCO3)=O)C2)cc(N)ccc1Br c1(OC)nc2ccc(CC(=O)NC(C(F)F)c3ccco3)cc2s1 C1(NC(CC(=O)NC2CC2)=O)CC(NC(=O)CCN2CCCCC2=O)CC1O N1(C(C2CNC(=O)N2)=O)CC(CNC(c2cccc3[nH]ccc23)=O)C2(CCC2)C1 C1(NC(c2ccsc2C(F)F)=O)CC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 N1(C(C2(CC#C)CCC2)=O)CCC2(CC1)CC2C(=O)NC1CCC(O)(CC)CC1 CCC(CN(C)C)C(=O)N(C(C)CCNC(=O)CSc1ccc(OC)cc1)C c1(CNC(C(c2ccsc2Br)N(C2CCC2)C)=O)cccc(Br)c1 c1(SC)nc(N2CCOC(C(C)NC(C3(C4CCC4)CC3)=O)C2)cc(C(F)F)n1 N1(C(C2(CCN(C)C)CCCC2)=O)CC2CC(NC(=O)C3=CCCC3)CC2C1 CCCCC(O)C(=O)Nc1cccc(-c2c(OC)cccc2O)n1 N1(C(CC(C(=O)OC)(C)C)=O)C2CCCC1CC(CNC(=O)Cc1cn[nH]c1)C2 c1(C(=O)NCCC(=O)NC2CC2CF)c(F)cccc1F C1(NC(CCOCCN(C)C)=O)CCC12CN(C(=O)CCn1ccc(O)nc1=O)C2 C1(C)(C(C)(C)C)CC(C(=O)NC2CC2CNC(C2CC3CC3C2)=O)C1 N1(C(=O)NC(CC(C)C(F)F)C)CCCCC(C)(F)C1 C1(N(CCC(=O)NC2CCOC2)C)CCN(C(C2CN(S(C)(=O)=O)C2)=O)CC1 C1(C(=O)Nc2c(CNC(CC=CC)=O)c[nH]n2)CC(SCC(F)(F)F)C12CCC2 c1(C(N2CCC(NC(C(CC)=CC)=O)(CF)C2)=O)cc(OC)cc(C)n1 c1(C(N(C2CCN(C(C(COC)C)=O)C2)C)=O)cncc2[nH]ccc12 CC(C)(CC(F)(F)F)C(=O)NCCC1CCCN1C(=O)CN1CCOCC1 C(=O)(CC(C)C(C)(C)C)N1CCC(O)(CCNC(C=COCC)=O)C1 C1(C(=O)NCCc2ncccn2)(NC(C(C)C2CC2)=O)CC1(C)C C(=O)(C1=NOC2COCC12)N(C1CN(C(=O)CCn2cccn2)CC1(C)C)C N1(C(C(=CC2CCCC2)C)=O)CCCCCC1CNC(c1snnc1C1CC1)=O C1(NC(CCNC(CC(C)C)=O)=O)CC(CNC(=O)CC=C(Cl)Cl)C12CCC2 c1(C(N2C(CNC(c3cnn4cc[nH]c34)=O)CCC2)=O)cccn(O)c1=O c1(OC)ccc2c(c1)NCCN(C(c1ccn3ncccc13)=O)C2 N1(c2nc(C)cc(CC)n2)CC2CCC1C1CN(C(=O)CCS(C)=O)CC21 c1(N2C(=O)CC(C(=O)NCC(CNC)(C)C)C2)ccc2nc(CN)oc2c1 C1(O)(CNC(C2(C)CC2(Cl)Cl)=O)CCCN(C(=O)C(F)(F)C(F)F)C1 CCC(CC(C)C)C(=O)NCCN(C(C1C(F)(F)C12CC2)=O)CC1CC1 N1(C(C(C)(C)OCC)=O)CCCC(C(C)C(=O)NC(c2cn(C)nn2)C)C1 C1(C(N2CCC(CNC(C34CCC(F)(CC3)C4)=O)C2)=O)CCCCC(F)(F)C1 c1(NC(=O)NC(C(=O)OC)OC)ccc(CS(C)(=O)=O)cc1 C(=O)(CC1COc2ccccc21)NC(CNC(C(C(=O)OCC)(C)C)=O)C c1(N2CC3C(C(F)(F)F)(C3)C2)nccc(-c2ccncc2)n1 c1(C(N2CCC(NC3C(OC)COC3)CC2)=O)ccnc2c1CCC2 c1(CCNC(c2cnc(C)o2)c2nnnn2C(C)(C)C)c(C)noc1C CC1=C(C(=O)N2CC(NC(=O)C3=NOCC3)CC2(C)CO)SCCO1 C1(CC(=O)NCC(CNC(Cc2n[nH]c(=NC)s2)=O)(C)O)CCCC12CC2 c1(CC)nc(C(=O)NC(CNC(=O)C(CC)CC)C2CC2)c(N)s1 c1(NC(=O)NCc2cc(N(C)C)ncc2)sc2ccccc2c1C#N CCCCC(CNC(=O)C(c1ccc(Cl)cc1)=O)NC(c1cnn(C)c1)=O CC(C)C(C(=O)Nc1cncc(C(=O)NC(C2CCOC2)C)c1)c1ccccc1 CCCC(CC)CC(=O)NCC(CNC(c1ccc(CO)c(Cl)c1)=O)CO c1(CN2CCC(NC(c3ccc(Cl)cc3)=O)CC2)c(F)ccc(F)c1Cl N1(C(CCCC(C)=O)=O)CCC(O)(C2(NC(c3cc(Br)no3)=O)CC2)CC1 C1(N(C(C(C)OCC#C)=O)C)CC2CCC(C1)N2c1ncns1 C1(OC)CC(CNC(=O)C(C2CC2)N(C)C)N(C(C2CC3(CC3)CO2)=O)C1 CNS(=O)(=O)N1CCN(C(=O)C2CCc3ccc(Br)cc32)CC1 N1(C(C2N(C(C)(C)C)CC2)=O)CCCC(C2CC2NC(c2ccsc2)=O)C1 N1(C(C2C3(CC(NC(C(C)SC)=O)C3)C2)=O)CCCC(C)(C)C1 C1(C(=O)NC2C(OC)COCC2)COCCN(C(C2(Cl)CC2(F)F)=O)C1 c1(C(N(CC(CNC(CCOCC(C)C)=O)C)C)=O)sc(=N)[nH]c1C1CC1 c1(CCC(=O)NC2C(NC(C(C)NC(CC)(C)C)=O)C2)ccc(OC)c(O)c1 C1(NC(c2cc(SCC)ncc2)=O)CCCCN(C(C2(CO)CCCO2)=O)C1 C(=O)(C1CCc2nccn21)NC(C(=O)N(CC(CC)C)C)C(C)(C)O NS(=O)(=O)c1cccc(CCC(N2CC3(CCCCC3)C2)=O)c1 Cc1ccc(C(=O)NC23CC(NC(=O)Nc4ccc(COCO)cc4)(C2)C3)cc1 C1(C(N(C)CC2(CNC(c3cnco3)=O)CC2)=O)CCCCS1(=O)=O C12(C(C)NC(N3CCC(NCCC(C=C)(C)C)CC3)=O)CC3CC(CC(C3)C1)C2 C1(CNC(c2c(SC)snn2)=O)CCC(N(C(=O)CCc2nncn2C)C)CC1 C1(CNC(C2N(C(C)C)CCC2)=O)CCCCN(C(=O)C(C)c2cccs2)C1 C1(NC(CCNC(COC)=O)=O)CCC12CN(C(=O)C(F)C(F)(F)F)C2 N1(C(CCOc2ccc(OC)cc2)=O)CC2CC1CC2NC(=O)C(C)=C1CCC1 C(=O)(CCCCC#N)NCCOCCCN(C(=O)CCC1(C)CC1)C c1(C(N2CC(NC(c3ccc(OC)c(O)c3)=O)C(F)C2)=O)cc2ccccc2o1 Cc1ccc(-c2cn(-c3ccccc3C(=O)N(C)C(C)C)nn2)c(C)n1 N1(C(c2cc[n+]([O-])cc2)=O)CC2(CCCN2C(c2ncn(-c3ccccc3)n2)=O)C1 N1(C(C(CSC)(C)C)=O)CC=C(CC(=O)NCC2(O)CC3C=CC2C3)CC1 c1(N2CCC(C)(C(=O)NC3CC3)C2)ccn2nccc2n1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2(CC1)CC2C(=O)NC1CCCC(O)C1 c1(C(CO)NC(C2CCCCC2O)=O)ccc(C(F)(F)F)cc1 c1(CC(=O)NCc2nc(C(C)(C)C)sc2)c[nH]c2ncc(Br)cc12 C1(C(N2CC3CC3(CNC(C3(CF)CCC3)=O)C2)=O)Cc2nccn2C1 CC(C)(C)C(=O)C(=O)NCCCCCCNC(=O)COc1cccc(C#N)c1 S(=O)(=O)(c1ccc2ccccc2c1)NC(C)C(=O)NC1CCCNCC1 C1(NC(C2C(CC)C2)=O)C2CCCN(C(=O)CCOCC(C)(C)C)C2C1(C)C Cn1nc(-c2cccnc2)cc1C(=O)NC1CC1NC(c1ccon1)=O CC#CCC(CO)NC(=O)CC(C)CNC(c1ocnc1CCC)=O C1(C(=O)OC)CCCCN1C(c1nc(C(C)NC(c2ccc(F)nc2)=O)cs1)=O c1(CNC(C2C(CC)N(C(=O)Cc3ccn(C)c3)CC2)=O)ccc(C)cc1O N1(C(C2(CC)CC2)=O)CCN(C(=O)Cn2cc(C3CCOC3)cn2)C(CCO)C1 C1(C)(C(N(CCOCC)C)=O)CN(C(=O)CSc2ccc(F)cc2)C(C)(C)C1 Cc1ccc2c(c1)CN(C(C1C(O)CCN1C(C1C3C4CCC(C4)C13)=O)=O)C2 C1(C(=O)NC(C)C(=O)O)CC2CCN(C(=O)CSCC3CCCC3)CC12 c1(CCNC2(c3n(-c4c(C)cccc4)nnn3)CCC2)cc2[nH]nc(C)c2cn1 c1(C(=O)NC2(CNC(c3ccoc3Cl)=O)CCC2)cc2c(Cl)cccn2n1 N1(C(C2C(OC)CCC2)=O)CCOC(CNC(=O)C(c2nc(C)cs2)C)C1 C12(C(=O)OCC3CCCCN(C(=O)OC(C)(C)C)C3)CCCCN1CCC2 c1(CNCCP(OCC)(C)=O)c(F)ccc(Cl)c1Br CC(C)(C(=O)NCc1cc(C(=O)NC2CCN(C(N)=O)C2)n[nH]1)C(F)F Cc1nc(NCc2nc(C3CC3)cs2)cc(=NCC2(C)C=CCCC2)[nH]1 N1(C(=O)NCCc2cccc(CC)c2)CC(=O)OCC1c1ccccc1 c1(CC2C(C(N(CC(C)(C)NC(=O)C(C)(C)c3ncco3)C)=O)C2)sccc1C#N C1(NC(=O)CCF)CC2CC(C1)CN(C(=O)C(c1ccc(F)cc1Br)O)C2 C1(NC(C(CC=CCC)C)=O)CCCN(C(C2CCC(=O)CC2)=O)CC1 CC1=C(C(=O)N2C(C(=O)Nc3cc(CO)ccc3C)CC2C)CCO1 c1(C(C(=O)N(CCCNC(=O)C(CSC)OC)CC)(F)F)cccc(C)c1 C1(NC(COC2C(C)CCCC2)=O)CCSC12CN(C(=O)C(C)(C)C1CCC1)C2 c1(CNC(NC(CC)C)=NCC2CCCC(=O)N2)c(C)ccc(Br)c1F C12CN(CC1(C)C)C2=O.c1(NC(C)=O)ccc(NC(c2cccn2C)=O)cn1 C1(NC(c2nc(-c3ccccc3F)cs2)=O)NCCCC1C(F)(F)F c1(C(CNC(C(CC)SC)=O)NC(=O)Cc2nn(C)cc2Cl)ccc(F)cc1F C#CC1(C(=O)NCC2(O)CC(CNC(=O)CSCC)C2)CCC1 C1(C(=O)NCCCc2cc(C(=O)OC)c(C)o2)CC12CCC(C)(C)CC2 c1(NC(C(=O)NCc2c(C)cccc2)=O)ccnc2c1CCO2 C(CC(C)(C)C)(C(=O)NCCc1ccncc1)NC(C(C(C)C)C1CCC1)=O C1(C(=O)NC(c2cccc(OC)c2)c2ccccn2)CC(C)(C)OC1=O C1(NC(c2cnn[nH]2)=O)CCCC12CCN(C(c1cc3n(n1)CCCN3)=O)C2 C1(C(N(CCC(C(C)C)NC(C(C=C=C)C)=O)C)=O)CC2CC(C1)CC(F)(F)C2 Cc1n[nH]cc1CC(=O)NC(C)(C)CNC(=O)CCOCC1CC1 C(=O)(C1=CCCC1)N1CCC(N(C(=O)COCC(=O)NC)CCOC)C1.CC CC(c1ccccc1F)=CC(=O)NC(Cc1ccccc1)CCC(=O)O CCC(C)(CCNC(=O)C(C)COC)NC(=O)C=Cc1ccnn1C C(CC(C(=O)N(C)CP(C)(C)=O)NC(=O)Cc1cnccc1C)=CC N1(C(C(=O)NC(C)C)=O)C(C)CC2CN(C(c3ccc4ncncc4c3)=O)CC12 C1(C(N2CCC(CC(N3CCOC(CN=[N+]=[N-])C3)=O)C2)=O)CC2(CC2)CO1 C1(CC(=O)NCC2C=CCN2C(c2ccnnc2O)=O)(OC)CCCCC1 c1(C(=O)NCC(C2CCCC2)NC(c2c(CC)ocn2)=O)c(O)cccc1O N1(C(C(CC#C)O)=O)CCCC(NC(c2cccn2Cc2ccncc2)=O)C1C C1(CNC(C2CCS(=O)(=O)C2)=O)CC2(C1)CN(C(=O)Cc1cccnc1)C2 C1(CC=C)(C(N2CCC(CN(C)C(C3CC(O)C3)=O)C2)=O)CCOCC1 O(NC(=O)C(CC(C)(C)C)NC(=O)CC1CC2CC2C1)C(CC)CC CCCC(C)(O)C(=O)NC1CC(N(C(=O)CCCc2ccc(C)cc2)C)C1 Cc1cccn2ncc(C(=O)NCC(C3CC3)NC(=O)C(C)(O)CC(C)C)c12 c1(C(N2C(=S)NC(c3c(C)cccc3)C2=O)=O)c[nH]c2c(F)c(Cl)ccc2c1=O Cc1ncnc(N2CCN(C3CCN(C(c4cc(F)ccc4Cl)=O)C3)CC2)c1Br c1(NC(C)C(C2CCCCC2)NC(=O)CCC2CCCCCC2)ncc(I)cn1 c1(C(=O)NC2(CNC(=O)CC3(O)CCOC3)CCC2)sc(Cl)cc1Cl CCC(CC)CCC(=O)OCC(C1CCN(C(=O)C(COC)N(C)C)CC1)C c1(C(=O)OC)ccc(N2CCN(C)CC2)nc1C.c12nccnc1C(=O)N2 C(c1ncco1)=CC(N1CCC(C2CCCN2C(=O)Cc2cscn2)C1)=O Cc1c(N)ccc(C(=O)NC2CS(=O)(=O)CC2NC(c2coc(O)n2)=O)c1Cl C=CCC(C(=O)N1CC(CC(=O)NC2(CO)CCOCC2)C1)c1ccccc1 C1(C(N2C(C)C(NC(=O)C(F)=C3CCCC3)CC2)=O)CCCS(=O)(=O)C1 CCCCCCCCC(=O)N1CC2(C1)CN(C(C1CC(OC)C1)=O)C2 CC1CCC(NC(c2cn[nH]c2)=O)CN1C(c1cc(Cl)cc(Cl)c1)=O Cn1nc(Br)c2ncnc(N3CCC(NC(=O)CC4CC(O)C45CCC5)CC3)c12 N1(C(C=C(CCC)CCC)=O)CC(N(C)C(c2[nH]c(=N)ccc2C)=O)C2(CC2)C1 c1(OC)cccc2cc(C(=O)NC(C)CC(C)NC(=O)C(C)(C)N3CCC3)[nH]c12 C1(C(N2CCC(CC(C)NC(c3occ(C)c3)=O)CC2)=O)CCC(N=[N+]=[N-])CC1 c1(CC(C)C(N(C(c2ccc(F)nc2)C)C)=O)ccc(F)cc1F C1(NC(CCN(C)CC)=O)C(CNC(=O)Cc2ccccc2Cl)CCC12CCC2 c1(CC)cc(C(=O)Nc2cccc(NC(=O)CN3CCCCC3C)c2)oc1CC N1(C(C2(COC)N(C(C3C(=C)C3)=O)CC=C2)=O)CCC2(CCOCC2)C1 N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCN(C(=O)C#CC2CC2)CC(C)(F)C1 c1(C(=O)NCC(C2CCCCC2)OCC)nc(Cl)ccc1Cl S(=O)(=O)(C1CN(C(C2(O)CC2)=O)C1)N1CCN(C(C2CCCC(C)C2)=O)CC1 c1(CNC(CC2(C)CN(C(C3COC3)=O)C2)=O)ccc(Br)c2ccccc12 C1(C(=O)NC2(CNC(c3c(C)n[nH]c3)=O)CC2)CC2CCCC12 C12(C(=O)NC(C3(O)CCN(C(CC(C)CF)=O)C3)C)CC3CC(C1)CC(O)(C3)C2 Cc1cc(C)c(C(=O)NCC2CC(O)CN2C(c2cnn3c2OCC3)=O)cc1N C=CC(F)(F)C(=O)N(CC(C)N(C(=O)OC(C)(C)C)C)C.C1(OCC(=O)N)CCCC1 C1(F)(CNC(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)CCCN2CCCC2)C1 C1(O)(CNC(c2cn(C3COCC3F)nn2)=O)CCN(C(=O)Cc2cnsc2)C1 c1(C(=O)NC2C3CN(c4nc(C#N)c(F)cn4)C2C3)ccc2[nH]nc(Br)c2c1 c1(NCC(O)CC(C(C(C)C)n2cncn2)=O)ccc(Cl)c(Cl)c1 C1(CC)(NC(=O)CN(c2ccccc2)C)CCCN(C(=O)Cc2ccc(C)o2)C1 CON=C(C(=O)N1CCCC(N(C(=O)CSC(F)(F)F)C)C1)c1ccco1 CCC(C)(O)C(=O)N1CC(CCNC(=O)C(C)CC#N)C(C)C1 N1(C(C(CC)(C)CNC(=O)CCc2ccoc2)=O)CCCC2C(=O)NCC12 c1(CC(=O)NC23CC2CN(C(C2(C(F)F)CC2)=O)C3)nsc2ccccc12 C(=O)(C#CC1CCOC1)N1C(CC)C(C(=O)NCc2cc(C)cnc2O)CC1 CCC(C)C(C(=O)NC1CCC(O)CC1)N(C(=O)C1=CCCCC1)C c1(C(N(C2CCC(F)(F)C2)CC)=O)cccnc1O N1(C(C(CC)(C)C)=O)CCC2(NC(c3cn(CCCC#N)nn3)=O)CCCC12 C1(NC(C(CC=CC)C)=O)CCC2CN(C(=O)CNc3ccccc3Cl)CC2C1 N1(C(C2C(=C)C2)=O)CCC2(CC1)CC2c1cn(CCc2ccc(O)c(O)c2)nn1 C(=O)(CCC(C)(C)F)N(C1CCCC(NC(CCCc2scc(C)n2)=O)C1)C c1(C(N2CCN(C(c3ccc[nH]3)=O)CC2c2cn[nH]c2)=O)cc2c(s1)CCOC2 C1(C(=O)NC2C(C(=O)NCc3n(C(C)C)ncc3)C2)C2CCCOC12 N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(=O)C(C)CCC(C)(C)C)C2(CCC2)C1 C1(CNC(c2n(CC)cc(Cl)c2)=O)N(C(=O)C(F)=C2CCCC2)CCCC1(C)C N1(C(C(=O)Cc2ccc(F)cc2)=O)CC2(CC2)CC1CNC(=O)Cn1nccn1 C1(NC(C(C)SC)=O)COC2(CNC(=O)C(c3ccc(C)cc3)(F)F)CC1C2 c1(C(=O)NC(C)CNC(C2CC2CF)=O)cn(-c2ncccn2)cn1 c1(C(N2C3C(C(=O)NCCC4C(C)CCCC4)C(C3)C2)=O)cc(F)c(F)cc1Cl N1(C(CCC=C=C)=O)CC2CCC(N(C(=O)COCC(C)(C)C)C)C2C1 c1(COC)cccc(NC(C2CC=CC(NC(=O)C(C)(CO)OC)C2)=O)c1C N1(C(CC(=O)OC)=O)CCC(C)C1CNC(=O)CC1CCC(C)CO1 C1(NC(c2cc(CCO)on2)=O)CN(C(=O)C2=C(Cl)CCC2)CCC1O C1(CC(N2CCC(CCN(C(=O)C(C)CC)C)CC2)=O)(COC)CCOCC1 S(=O)(=O)(c1ccc(CCC(=O)O)cc1)N(c1ccccc1)CCC(=O)O C=CCCC(O)CN(C)C(C1(C)C=CCN1C(=O)Cc1c(C)noc1C)=O CCN=c1[nH]c(C)c(C(=O)NC2CCCCCC2NC(=O)C(C)=CC(C)(C)C)s1 Cc1cccc(OCCC(N2CC3CC3(NC(=O)Cc3ccc(F)cn3)C2)=O)c1 c1(C(=O)NCCC2(O)CCN(C(C3C=CCCC3)=O)C2)noc2ccc(Cl)cc12 O=C1CCC2C(C(=O)NCc3ocnc3C(=O)NCC=CCl)C12 c1(C(C(=O)NCC(C)N(C(=O)CC2CCC2)CC)(F)F)ccc(C(C)C)cc1 C(=O)(C1CCCc2n[nH]cc21)NCCC(C)Nc1nccc(CC(=O)OC)n1 CC(CC(C)(C)C)C(=O)NC1CCC1C(N1CCC(O)(C(N)=O)CC1)=O C(=O)(C1=C(C)OCCS1)N(CCC(=O)NCCOC(CC)CC)CCO CC1CCC(NC(c2cn3c(n2)SCC3)=O)CN1C(c1nnn(C)c1N)=O C(=O)(CCCCCOC)N1CCC(CN(C(C2C(C(=O)OC)CCC2)=O)C)CC1 C1(NC(CC2(C)CCC2)=O)CCCC(CNC(c2cc(Cl)ns2)=O)C1 c1(C(=O)NC2C(NC(c3nc(C)oc3C)=O)CCC2)ccc2c(c1O)CCCC2 c1(NC(=O)NCC2CC3C(C2)C3(F)F)nc2c(s1)CC1(CCCCC1)CC2 n1(C(C)C)ncc(-c2noc(C3CCCO3)n2)c1F C1(C(=O)NC2C(NC(C(C)(C)Cc3cccc(Cl)c3)=O)CC2)NC(=O)OC1(C)C C#Cc1ccc(C(=O)NCCN(C)C(c2cnc(CC)[nH]2)=O)nc1 O=C(CC1=CCCC1)NCC1C2CN(C(=O)CCN(CC(F)(F)F)C)CC12 c1(-c2cn(C)nn2)nc(CCn2cc(Br)cn2)nn1CC(N)=O C1(NC(CCSCC#C)=O)CC(C(=O)NCc2cccc(C=C)c2)C12CCC2 c1(CC(C)C(=O)NCC2CN(C(C3(C#N)CCC3)=O)C2)ccc(Br)cc1 Cc1ccn2nc(C(N3CC(CNC(=O)CC4CC4C)C3)=O)nc2n1 c1(C(N2CCCC(N(C(C(CC)NC(N)=O)=O)C)C2)=O)cc2occc2[nH]1 C12(C(=O)NCC3CCN(C(c4ccoc4)=O)C3)CC3CC1C2C3 CCC(C)(C)C(C(=O)N1CCOCCC1c1cccc(C(F)(F)F)c1)NC(C)=O CCCCC(CNC(c1ccc(-c2cccs2)s1)=O)NC(c1nc(O)sc1C)=O C1(F)(CNC(c2cnc(O)s2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1 c1(CNC(=NC)NCc2c(F)cc(F)c(F)c2F)cccc(S(N)(=O)=O)c1 c12ccc(cc1Cl)[nH]c2=O.c1(CC(=O)Nc2ncc(CC)s2)ccc(Br)cc1C Cc1cnc(C)c(C(=O)NCCC2CCN(C(=O)CC3CCCC(C)O3)C2)c1 C1(CNC(C(C)(C)C)=O)CC2(CCC2)CN1C(C1CC=CCC1C(F)(F)F)=O N1(C(c2n(CC(C)C)ncc2)=O)CC2CCC(NC(=O)Cc3cn[nH]c3)CC2C1 C=CC(CC)CC(=O)NCCCCC1CCCN(C(=O)Cc2cn[nH]c2)C1 c1(C(=O)NCC2N(C(c3ncc(NC)nc3)=O)CC(OC)C2)c(C)[nH]c(C)c1C c1(OC)c[nH]c(C(=O)NCCN(C(C2CCOC(C)C2)=O)CC2CC2)cc1=O c1(C(=O)NC)ccc(C(=O)N(C)CC2(O)CN(C(=O)C=CCCC(C)C)C2)cn1 N1(CC2CN(C(C3CN(C(C(C)SCCCC)=O)C3)=O)C2)CCN(C)CC1 C1(C(=O)Nc2cccnc2C)(CC)CCN(C(c2cn(C3CC3)cn2)=O)C1 C(c1ccc(I)o1)=CC(=O)NC(C(=O)NC(C)C)C C(=O)(CC(C)(C)CC(=O)OC)NC1CC(F)(CNC(c2c(COC)noc2)=O)C1 C1(NC(C(CC#C)O)=O)CN(C(=O)C(CSC)c2ccccc2)CCC1O c1(CCC)cc(C(=O)NC2CCN(C(=O)CCCC3CCC3)C2C)cc(O)n1 Cc1cc(C(=O)NCC2CC(C(=O)NN3CCC3C)C2)ccc1N1CCOCC1 N1(C(=O)CC(F)(F)F)CCC2CCN(C(C3(F)CC4(CCC4)C3)=O)CC2C1 N1(C(C=COCC)=O)CCC2(CCC(CNC(C3CN(C)C3)=O)O2)CC1 C(=O)(C1=CCSC1)NCCNC(C1CN(C(C(N2CCCCC2=O)C)=O)C1)=O C1(CNC2C=CC(C)(C)CC2)CCCC(C2CC2)C1 c1(CCC(=O)OCc2n(CCC)ccn2)cccc(F)c1Br c1(OC)c(NC(C2CCCN2C(=O)CC2CCCN2C(C)=O)=O)cnn1C C1(C(C)C(=O)NCC(O)CO)CCCN(C(C2(CF)CC(=O)C2)=O)C1 N1(C(C(C(C)C)(C)O)=O)Cc2ccccc2CC1CNC(=O)CC1CCN(C)C1 Cc1oc(C)c(C(N2CC(NC(=O)CCc3cnoc3)C(C)C2)=O)c1C c1(C(N2C(CN(C(CCOCCOCC)=O)C)COCC2)=O)cccc(C)c1F C1(NC(Cc2nnc(C)o2)=O)CC(O)CN(C(=O)CC2(n3ccnc3)CC2)C1 C1(C#N)(C(N2CCC(OC)(CNC(C3CCC3(F)F)=O)C2)=O)CCCCCC1 C1(C(N2CCC(NC(Cn3nnc(=N)[nH]3)=O)(CO)C2)=O)CCc2nc[nH]c2C1 C1(NC(COC(CNC(C2(C(C)(F)F)CC2)=O)(C)C)=O)CC(F)(F)C1(C)C CS(=O)(=O)C(C(=O)Nc1ccc(NS(C)(=O)=O)cc1Cl)C1CC1 N1(C(c2c(C)n(C)nn2)=O)CCN(C(C2COCCN2C(=O)N(C)C)=O)CC1C c1(C(N2C(CN=c3nnn(C)[nH]3)(C)CCC2)=O)csc2c1CCCC2 C(=O)(CC(C(C)C)OCC)N1CCC(N(C(C2(CC)CC(OC)C2)=O)C)CC1 C1(CNC(COCCOCC)=O)CNCCN1C(C1CN(C2CCOC2)C1)=O c1(C(=O)NC(C)CCC2CCCC2)cc(CNC(=O)CC(C)C2CC2)on1 CCCCC(CC)CC(=O)NC1CCC(N(c2nc(C)nc(Cl)c2C)C)CC1 c1(C(=O)NC(C)CNC(C2CCOC(=O)N2)=O)ccc2c(c1)NC(C)CC(=O)N2 C(c1ccc(F)cc1)=CC(=O)NC1CCC(N(C)C(c2ccco2)=O)CC1 N1(CC(=O)NCC)CCCC1C1CCCCN1C(=O)C=C1CCCCC1 c1(C(=O)NCCN(C(=O)CCN2CCCC(C(C)(C)C)C2)CC)cccc(NC)c1 C1(C)(CCC)CCN(C(=O)C(C)(C)CNC(C2CC=CCO2)=O)C1 c12ccnc(c1)NC2=O.C1(=O)C(C2CCOC2)N1.N(CCC1CC1)(CC)CC c1(C(=O)NC2(C(=O)O)C(C)C2)cccc(Cn2cc(-c3ccccn3)nn2)c1 CC1(C)CCCCC1C(N1CCCC1CN(C(C12CCC(CC1)CO2)=O)C1CC1)=O N1(C(CCCC#C)=O)C2CCC1C(F)C(NC(C1CCC(N(C)C)CC1)=O)C2 C1(C(=O)NCC(CO)NC(C)=O)CCN(C(c2cc(CO)on2)=O)CC1 C1(NC(C2(C)CC(C)C2)=O)CCC(CNC(=O)Cc2ccsn2)CC1 CCCCC(C)C(=O)NC12CC1CN(C(c1coc(C(F)F)n1)=O)C2 c1(C(N2C(C(=O)Nc3cc(C)cc(O)c3)CC2C)=O)cc(C#N)ccc1C c1(C(C=CC(=O)NCCN(CC(C)C)CCOCC)C)ccccn1 N1CCC(CCn2nccn2)CC1.n1(CC)ccnc1 CC(C)S(=O)(=O)C(C)C(=O)N1CC(NC(=O)Cc2nc[nH]n2)C(CC(C)(C)C)C1 N1(C(C2N(C)CCCC2)=O)CCN(C(c2cnc(-c3ccsc3)s2)=O)CC1CF C1(CN(C(CC(C)n2cccn2)=O)C)C2CN(C(c3ncccc3F)=O)CC12 C(=O)(C1CCCc2sccc21)NC(C)CNC(C1(C2CCC(=O)NC2)CCC1)=O C(=O)(C(=O)N=S(C)(C)=O)NC(CCCNC(CN1C(C)CCC1C)=O)(C)C C(=O)(C(F)C(C)(F)F)N1C(C2(C(=O)NCc3n(C)cnc3)CC2)CCC1 C(=O)(CCCC(=O)NC1CC1)NCC1CC(C)N(C(=O)Cc2ccnc(O)c2)C1 CS(=O)(=O)c1ccnc(NCCCC(CC)Nc2cc(C#N)ccn2)n1 N1(S(CC)(=O)=O)C2CCC1CC(C(=O)NCC1(O)CCCN(CCO)C1)C2 Cc1cnc2ccc(C(=O)NC3(CNC(C4(Cl)CC4(C)C)=O)CC3)cn12 Cc1nn(C)cc1C(=O)NC1CCN(C(C2CCN(Cc3ccsc3)CC2)=O)C1 c1(CC)cccc(C(=O)NCC2C=CC(NC(c3ccc(C4CC4C)o3)=O)C2)c1 N1(C(CCC)=O)CCCCC1C(=O)NCC(c1scnc1C)N1CCOCC1 Cc1nc(-c2c[nH]cc2C(=O)NCCC2CCCN2C(C2CC2C)=O)cs1 C12(C(=O)NCC3(NC(CCN4CC(=O)NCC4)=O)CC3)CCCC1C2(F)F N1(C(c2cn(CCC)nc2C)=O)CCCN(C(C2CCCCO2)=O)C(CO)C1 c1(CNCC2N(C(C3CCO3)=O)CCC2)ccc(Oc2ccccc2)cn1 Cc1cncc(C)c1C(=O)NCC(C)(C(C)C)NC(C1CC2CCC1CC2)=O C1(F)(NC(C2CCOCC2)C)CCN(Cc2cccc(C(F)(F)F)c2)C1 N1(C(Cc2ccn(C)c2)=O)CCC(C(=O)NC(CO)CC(F)(F)F)C1(C)C c1(OCC(=O)NCC(CO)NC(c2nc(C)sc2)=O)ccccc1O.C(C)C CCCC(CCC)NC(C1CCC(C2CC2)N1C(=O)CCCOC(C)=O)=O C=C1CCC(C(=O)NCCC2CCN(C(C3CC(OC(C)(C)C)C3)=O)C2)CC1 C1(NC(C(C)OCCC#C)=O)COC2(CCN(C(c3ccnnc3O)=O)CC2)C1 CCC(C)CCCCC(=O)NC1C(C)(C)C(NC(c2ocnc2C)=O)C1(C)C c1(C(=O)NCCCC(C)NC(C2(CC#C)CCCCO2)=O)nccc(C)c1F N1(C(C(C)c2ncco2)=O)CC2(NC(C3CC(=O)N(CC(F)(F)F)C3)=O)CC2C1 Cc1ccc2sc(C(=O)NCCNC(=O)Cc3ccc([N+](=O)[O-])cc3Cl)cc2c1 N1(C(CN(C(=O)OC)C)=O)C(C(=O)N(CC(O)C2CCC2)C)CCC12CC2 C1(NC(c2c(SC)scc2)=O)CCCCC1NC(c1[nH]c(C)nc1C)=O O=C(CCCCCc1ccc(O)cc1)NCC1(CNC(c2nsnc2O)=O)CC1 Cc1csc2ncnc(N3CCC(C)(C)C(CNC(=O)CCCS(N)(=O)=O)C3)c12 N1(C(C(C)OCC)=O)CCCC(N(C(=O)Cc2ccccc2Cl)C)C1 CC(C)CC(CNC(=O)CCC(C)(C)N(C)C)C(=O)NC(c1ccc(F)cn1)C C12(C(=O)NCC3N(C(C4CCCC(O)C4)=O)CCC3)CCCN(CCC1)C2 CC(CCN1CCC(CS(C)(=O)=O)C1)C(=O)NC1CCCCC1 C12(CCNC(C3N(CCC)CCC3)=O)CCC1CN(C(=O)Cc1c[nH]nc1O)C2 c1(N(C(C2CCCCC2)C(=O)NC2CCCCC2)C)cncc(C(N)=O)c1 C1(NC(C(Cn2ccnn2)NC(Cn2nnc(C)n2)=O)=O)CCN(C)CC1 c1(C(=O)NC(C(=O)NCC2N(C(C)=O)CCCC2)CO)cc2ccsc2s1.C(N)=O c1(OC)cc(OC)nc(C(N2CCC23CC(c2ncc[nH]2)C3)=O)c1 c1(C(C)OCC)noc(CC(=O)N(C)CCCCCNC(=O)Cn2ncnn2)n1 c1(SCCCC(N2CCCC(NC(C(CSC)O)=O)C2)=O)ncnc2[nH]cnc12 C#CC(CC(C)(C)C)NC(C1C=CCN(C(c2cc(O)cc(F)c2)=O)C1)=O C(CN=c1nc(N2CCC3(CCCC3)C2)c2[nH]ccc2[nH]1)OCCC(C)C C(=O)(CCCCCC(C)O)NC1C(CNC(c2ccc(CC)cn2)=O)COC1 N1(C(C)C)CCC(CC(=O)NC(C)(CNC(=O)CC2CC2C2CC2)CO)CC1 CC(C)C(C)C(=O)N1CCC(CNC(C2CCCC(CF)C2)=O)CC1 CCC(C)(CC(=O)NCCN(CC(C)O)C(c1cccc(COC)c1)=O)C(=O)OC N1(C(C2C(C)C2)=O)CCCC12CCN(C(c1cc3c(s1)CC(C)(C)C3)=O)C2 C(c1ccc(S(C)(=O)=O)o1)=CC(N1C(C#C)CN(C(C2CCC2(F)F)=O)CC1)=O C(C(C(C)(C)C)Nc1cc(CN2CCC(O)CC2)ncn1)NCc1ccc(C)o1 c1(OC)cccc(NC(=O)CCN(CC2CC2)CC2CCCO2)c1 N1(C(C=C(C)C)=O)CC(C)CN(C(c2ccnc(O)c2Br)=O)C(C)C1 CC(CNC(=O)C(F)(F)c1ccccn1)(Cn1cccn1)N=c1cc(Cl)c(O)n[nH]1 O=C1CC2(CCN(C(=O)C(c3cccc(Oc4nccs4)c3)(F)F)C2)CN1 c12cc(Br)ccc1S(=O)(=O)N2.c1(CCN(CCOCCC=C)CC)ccncc1 Cc1noc(C(F)(F)F)c1C(N1CC(CC(=O)NC2COCCC2C)C1)=O c1(C(N2CCC(N(CCC)C(C3CC3CC)=O)C2)=O)ccc2cn(CC)nc2c1 CCC(O)C(F)(F)C(=O)NC(C1CN(C(c2cc(=O)n(C)cn2)=O)C1)C CCC(CCC(=O)NCCc1ccncc1F)NC(C1CNC(=O)O1)=O CC#CCCC(=O)NC1CC(CNC(=O)CCCCC2CCCCC2)C1 C(=O)(C(C)(C)C(=O)NC1CCN(C(=O)CN2CCC(F)(F)C2)CC1C)NC CCC(C)(CNC(=O)CCC1CCCN1C(=O)C(C)N1CCCC1)CO C1(C(N(C2CCN(c3ccc(C#N)nc3)C2)CC)=O)CCc2cncn2C1 CC12CC(C(=O)NC3CC(NC(c4cccnc4O)=O)C3)(C1)C1(CCC1)O2 c1(-c2cn(Cc3ccc(N4C(=O)NCC4)cc3)nn2)ccc2nccnc2c1 C1(C(=O)NC2C(NC(c3cc(C(N)=O)[nH]c3)=O)CCC2)Cc2ccccc2C1 c1(C(=O)NCC(CCNC(C(C)(C)OC)=O)O)[nH]cc2c(=O)n(C)ccc12 C1(C(N2CC(C#C)(F)C2)=O)CC(F)CCN1C(c1ncoc1C)=O c1(NC(C)=O)ncc(S(=O)(=O)NC2CN(Cc3nccs3)CC2F)s1 N1(Cc2cccc(CC)c2)Cc2[nH]nc(NC(c3cccc4[nH]ccc34)=O)c2C1 c1(C(=O)NCCCCCN(C(c2c(CC)ccs2)=O)C)cc(OC)cc(C)n1 C=CCC(CC)C(=O)N1CCC(CCN(C(=O)Cc2sc(C)nc2C)C)CC1 c1(N(Cc2c(C)cccn2)CC2(C)CCCC(=O)N2)ccccc1[N+](=O)[O-] CC1CCCN(C(=O)CCn2ccnn2)C1CNC(=O)CN1CCN(C)CC1 C1(C(=O)NC(C)C(C)(C)O)CCN(C(=O)C(F)C2CCC2)O1 CCC(C)C(O)C(C)C(=O)N1CCC(CCNC(=O)CCc2ccsc2)C1 Cc1cc(C(=O)NCCC2(O)CN(C(c3cn(C)nc3Cl)=O)C2)cc(C)c1F C1(C(=O)NCC(C)(C)CNC(=O)C(F)F)CC12C1CC3CC(C1)CC2C3 c1(C(CNC(c2ccnn2CC(C)C)=O)NC(C(=O)NCC)=O)cccc(C)c1 C1(OC)CN(C(=O)C(C)(C)OCC(F)(F)F)CC1NC(C1CCCCCS1)=O C1(N(c2c(SCC)cccn2)C(c2ccnc(C(N)=O)c2)=O)CCCN(CC)C1 c1(C(=O)NCC(C)CNC(=O)C(C(C)(C)C)n2ccnn2)ccc([N+](=O)[O-])cc1 C1(NC(CCCC#N)c2n(C)nnn2)CC2CC3C(C2)C13 N1(C(CNS(CC)(=O)=O)=O)CC(NC(=O)Cn2cc(C3CCC3)nn2)C(C)(C)C1 c1(OCC)nc(Cl)ccc1C(=O)NCCC(C)NC(C1CCCC1O)=O CC1CCN(C(c2c[nH]c(=N)nc2O)=O)CCN1C(c1noc2c1CCCC2)=O Cc1ncn(C)c(=O)c1C(=O)NCCNC(C1(C#N)CC2(CC2)C1)=O C1(OC)CC2(C1)CC(C(=O)NCC(CO)NC(=O)CC1CCC(F)(F)CC1)C2 C=C(C)C(C)(C)C(=O)NCCC1(NC(c2cc(C#N)n(C)n2)=O)CCC1 N1(C(CC(CC)(C)C)=O)CCCN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1C N1(C(C(CCC2CCC2)NC(c2ccn(CC)n2)=O)=O)CCc2ncncc2C1 C(c1c(Cl)cccc1Cl)=CC(=O)N(CC(C)(C)NC(c1c(C)snc1)=O)C Cc1nsc(N2CCC(N(C(=O)C=C3CCCCC3)C)CC2)c1C#N CCCCC(O)C(=O)NCC1CN(C(c2ccccc2O)=O)CC1O c1(OC)ccc2[nH]cc(CC(=O)OCc3noc(COCC(C)C)n3)c2c1 N1(C(CC(CCC)C)=O)CC(NC(=O)Cn2ncc(Br)n2)CC(C)(C)C1 c1(C(=O)NC(c2ccc(C)cc2)CNC(=O)CN2CCCC2)cc(N)c(F)cc1C C1(CC(=O)NCC(C)NC(C=C)=O)CC(=O)NC(=O)C1 C(=O)(CC1(O)CCOc2ccccc21)NC1CCN(C(C(CCC)CCC)=O)C1 N1(C(CC2(OC)CCC2)=O)CC2(CC(NC(c3ccccn3)=O)c3nccn32)C1 C1(C(=O)NCC2(O)CN(C(c3cc(OC)c(F)cc3)=O)C2)CC2C=CCC(C1)C2 c1(C(N2CC(C(C)(C)O)(CNC(CCCCCC)=O)C2)=O)cc2n(n1)CCCO2 c1(CNC(COCC#C)=O)cc(C(=O)NC2(C(N)=O)CC(CO)C2)n[nH]1 c1(N2C(CCC=C)CCC2)nc(=NCC23CCC(C2)C(C)(C)O3)[nH]c2ccsc12 Nc1cc(Cl)nnc1C(=O)NC1CS(=O)(=O)CC1NC(c1c[nH]cc1C1CC1)=O C(CC(=O)N(CC(O)CN(C(=O)Cc1c(C)cccc1F)C)C)(C(C)C)OCC CCC(N=c1cc(NCC(=O)N(C)C)nc(C(C)C)[nH]1)C1CCOC1 c1(C(N2CC(CCNC(C(C(C)C)O)=O)C2)=O)cc2ccnc(Cl)c2s1 C1(CCNC(c2ccc(C)nc2)=O)CN(C(c2ncsc2C2CC2)=O)CC(C)O1 c1(OC)cc(C(N2CC(CNC(c3ccsn3)=O)CC2C)=O)cnc1O CCCC(C(=O)OC)C(=O)NC(CO)C(=O)NCCc1cnn(C)c1C C(=O)(CC1=CSC2=NCCN12)NC1C(C2CCN(C(c3cc(C)on3)=O)CC2)C1 S(=O)(=O)(c1c(C)cccc1Cl)N(C(C=CCCC=C(C)C)=O)CC(F)F N1(C(c2nnn(C)n2)C(=O)NC(=O)OC(C)(C)C)CCn2cncc2C1 Cc1c(C(=O)NC(C2CCCN2C(=O)CC2CCCC(C)(C)C2)C)cccc1F C1(CC=C)(C(=O)NCC(=O)N2CCCO2)CCN(C(=O)C(F)C(C)C)C1 c1(C(=O)NC2CCCC(CNC(CCC#CC)=O)C2)cc(OC)c(S(N)(=O)=O)s1 C1(C(N(C)CCC2CCCCN2C(=O)CS(C)(=O)=O)=O)OC2CCC1CC2 c1(OC)ccc(NC(=O)C(=O)NC(C)C(=O)NO)cc1S(C)(=O)=O CC(C)(C)C(C(=O)NCC1CNC(=O)CO1)NC(=O)CCn1cnnn1 c1(C(N2CCCC(N(C(C(C)NC(N)=O)=O)C)C2)=O)cc2ccccc2s1 CC1CC2(CCO1)CC2C(=O)NC1CCCCN(C(c2ncn(C)n2)=O)C1 C1(C(=O)NCC2C=CC(NC(c3cc(OC)no3)=O)C2)CCCOC1C c1(C(N2C(CNC(CC3C(C)C3)=O)CC2)=O)cccc(-c2cnn(C)c2)n1 C1(O)(CNC(CC(C)C(F)(F)F)=O)CC2CCC(C1)N2C(=O)C(O)C(C)(C)C N1(C(c2ccc(CSc3scc(C)n3)cc2)=O)CCN(C)C(=O)C1C C12(C(N3CC(O)(C(C)C)C3)=O)CCCC1CCN2C(=O)CC1=CCCCC1 C1(NC(C(C)Cc2ccc(F)cc2)=O)CN(C(=O)C(F)=C2CCC2)CC2(CC2)C1 c1(CC2(C(=O)NN3CCC(C(=O)OCC)(CO)C3)CC2)ccc2c(c1)OCO2 C1(NC(C(=O)NCCC(N)=O)=O)CC2CCC1N(C(=O)Cc1ccc(O)cn1)C2 N1(C(C)=O)CCC2(CCCN2c2nc(N3CCOCC3)c3sccc3n2)CC1 CC1CCN(C(=O)COCc2ccccc2Cl)C(CNC(c2cc[nH]n2)=O)C1 N1(C(c2cnc(O)c(F)c2)=O)CCC(C2CN(C(C3CC3(F)Cl)=O)C2)CC1 N1(C(C(C)N(C(CCCOCC)=O)CC)=O)CCC(F)(F)C(C)C1 c1(C(N(CCC(C(C)C)NC(=O)CC(C)(C)C)C)=O)ccc2c(c1)CN(C)CC2 Cc1sc2ncnc(N3CCCC(C)(CNC(=O)C=Cc4cnc[nH]4)C3)c2c1C N1(C(c2nc(Br)sc2C)C(=O)NCC(=C)C)CCOC(C)(CC)C1 C(=O)(C1CCCc2c[nH]nc21)NC1(CC)CCN(C(C2CCC(C)C2)=O)CC1 Cc1ccc(C)c(C(=O)NC2CC(C)(CNC(=O)CC3CCCOC3)C2)c1 N1(C(c2c(C)ocn2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)C(CC(C)(C)C)C1 c1(C2C(NC(c3c(Br)n[nH]c3Br)c3n(CC=C)nnn3)C2)ccc(F)cc1 CCCC(C)(CCC)C(=O)NCC(C)CNC(c1cnn2c1OCC2)=O Cc1cc(C(=O)N(C2CN(C(=O)C(c3cccnc3F)(C)C)C2)C)c(C)s1 C1(NC(C(C)OCC#C)=O)C2CC1CN(C(=O)C(N1CCC(C)C1)=O)C2 C1(N(C(c2ccc(SC)s2)=O)C)CN(C(c2ccc(F)cc2O)=O)CC12CC2 C1(C(=O)NCC2CC(C(=O)NCC3CC(OC)C3)CO2)(CC)CCCCO1 Cc1cnc(C(=O)NC2CC(NC(c3cn(CCO)nc3C)=O)C2)cn1 C=CCCCCCN=c1[nH]c(N2CCC3CCCC3C2)nc2cccnc12 C1(CC=C)(NC(c2nc(Cl)ccc2Cl)=O)CCCN(C(C2(Br)CC2)=O)C1 C(CO)(C(C)NC(c1cc(CNC(=O)CSCCC(C)C)[nH]n1)=O)SC c1(C(=O)NCc2c(C(=O)NC(CCSC)CO)n[nH]c2)cnn(C)c1Cl CC1(C)CCOC1CC(=O)NC1COCC1CNC(c1cccnc1C(F)F)=O C1(CNC(C2(CC)CCNC2=O)=O)CN(C(C2(C)CCC(=O)N2)=O)CCC1(F)F C(=O)(C1CSc2ccccc21)NC1C(NC(C=Cc2c(C)n(C)nc2)=O)COC1 C1(CC)(CNC(=O)C(=O)Nc2cc(I)ccc2N(C)C)CCCC(=O)N1 N1(C(CC(C=C)C)=O)CC(CNC(c2cncc(NC)c2)=O)CC1(C)C C1(C(=O)NC(C#C)CC2CC2)CCc2nc(C#N)sc2C1 c1(CC)ccc(Cl)nc1NC(=O)C(C)NC(C(=O)OC(C)(C)C)C(C)C CCCCC(CNC(C1CN(C(c2ncncc2Cl)=O)CC(C)O1)=O)CCC N1(S(C)(=O)=O)CCN(C(=O)COC(C2(C)C=CCC2)=O)CC1 c1(OC)ccc(CCCNS(C)(=O)=O)cc1Cl.c1(C(=O)O)cnn(C)c1 C1(NC(c2cccc(=O)o2)=O)CCC2(CC1)CC(NC(=O)C(O)CC1CC1)C2 c1(C(N(CC(C)N(C(=O)C(C)OCCN(C)C)C)C)=O)cnc(C(C)(C)C)o1 c1(CC)cc(C)c(C(=O)NCCC(C)(C)CNC(=O)CC2(O)CCCCC2)o1 c1(C(=O)NCC(CC)(CC)NC(=O)C(O)C(C)OC)c(Cl)nc2ccccn12 c1(C(N(C2CC(C(F)C(=O)NCC(C)(O)C3(C)CC3)C2)C)=O)ccn(C)n1 N1(C(c2c(C)nc(COC)nc2C)=O)CCC2(CC(C(=O)NC(CF)CF)C2)C1 N=c1c(C(=O)NC2CCCCN(C(C3CCC=CCC3)=O)C2)c[nH]c2ccc(Br)cc12 NC(=O)CC(O)C(=O)NC1CC2(C1)CC2C(=O)NCCOc1ncccn1 C1(C(N(C2CCN(C(CCc3n[nH]c(=N)s3)=O)C2)CCO)=O)CC12CCCCC2 N1(C(c2ccc(C)cc2F)C(=O)NCCC#N)CCCSc2cc(C)ccc21 C1(O)(C(=O)NCCNC(C2CCC3(CCOCC3)C2)=O)CCc2ccccc2C1 N1(C(Cn2cc(COC)nn2)=O)CC(NC(C2(C(C)(F)F)CC2)=O)CCC1C c1(N2CCC(N(C(=O)C(C)CSSC)CC)C2)cc(SC2CC2)nc(C)n1 Cc1ccc(C(=O)Nc2cc(Cl)ccn2)cc1Cl c1(C(C2CCCCC2)C(=O)N(C)CCN(C)C(C2CCO2)=O)ccccc1F c1(C(=O)NC(c2ccc(F)cc2)CNC(C2(C=C)CCC2)=O)csc(=NC)[nH]1 CCC(C(=O)NCC(C)CN(C(=O)CCc1ccc(C)s1)C)OC Cc1ccc(OCCC(=O)NCC(C(C)(C)C)NC(c2nn(C)cc2N)=O)cc1 CC(C(=O)N1CCC(CNC(=O)COCC2CCCC2)C1)S(N)(=O)=O N1(C(Cn2c(C)ncc2)=O)CC(NC(c2cc(C(F)(F)F)cc(F)c2)=O)C(C#N)C1 C1(CCOC)(NC(=O)C(C)CS(C)=O)CCN(C(c2ccnc(CO)c2)=O)CC1 C(CCCCCNC(c1ccc(Cl)cn1)=O)NC(c1c(COC)ncs1)=O C(c1ccc(F)cc1)=C(C)C(N1CC2CC1(CNC(=O)CC(C)C1CC1)C2)=O C1(CC(=O)NC(CC)C(=O)NC23CC(F)(C2)C3)CCOC1(C)C N1(C(C)C)CCNC(=O)C1.C1(CO)C(=O)N1 N1(C(c2c(CC)c[nH]c2)=O)CC(N(C(=O)CC2CC(C)(C)C2)C)C(F)C1 CC(C(=O)NCC1CC(C(=O)NC2(CN(C)C)CC2)C1)N1CCCC1 Cc1c(NCC(F)(F)CC2CC2)ncnc1N1CCC(CO)CC1 N1(C(CC(c2ccc(OC)cc2)C)=O)CCN(C(=O)CCCOC)C2CSCC12 CC(CC(=O)N(C)CC1(O)CCN(C(=O)CN2CCOC2=O)CC1)P(C)(C)=O C1(O)(CNC(=O)CN2CCCS2(=O)=O)CCCN(C(=O)C(c2ccccc2)O)C1 N1(C(C(N)CC2CCOC2)=O)CCC2(CC1)NC(=O)N(Cc1ccccc1)C2=O C=C(C)CC(C(=O)NCC#CC(F)(F)F)NC(=O)CCn1ccnn1 c1(C(N2CC3(CC(NC(C(C)n4cccn4)=O)C3)C2)=O)cc2cccnc2[nH]1 c1(C(=O)NC2CN(Cc3cc[nH]n3)CC2O)ccc2c(c1)OCCO2 C(=O)(C(C)CCC(C)(C)C)NC(CNC(C1CCN(CC(C)C)C1)=O)C C1(NC(C(CC)N(C)C)=O)CC1C1CCCN(C(c2cc(C)n(C(C)C)n2)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCCC(O)(CCNC(C2CC(OC)C2)=O)C1 O=C(CC1=Cc2ccccc2C1)N1CCCC(NC(C23CCC2C3)=O)CC1 CCCC(CC)C(=O)N(C)CC1CCN(C(=O)C2=CSCS2)CC1 c1(CC)ncncc1C(=O)NC1CC1CNC(c1ccc(CO)s1)=O CN1CCCC2C1CCN2C(=O)CC1CC2CCC1O2 N#Cc1ccc(CN2CCC(F)(C(N3CCC(O)(C(F)(F)F)C3)=O)C2)c(O)c1 CC(CCC(=O)N1CCC(C)(O)C1)NC(=O)CSC1CC1 C1(NC(c2c(CC)nns2)=O)CN(C(C2CC(F)C2)=O)C2(CCOC2)C1 c1(C(=O)NCCC2CCN(C(C)=O)C(C)C2)c(F)ccc2[nH]ccc12 CC1(C)OCCC1C(N1CCSCC1C(=O)NC1C=CC(CO)C1)=O c1(C(=O)NC2CC3(CC(NC(C(COC)C)=O)C3)C2)nc(Cl)c(Cl)c(N)c1Cl C1(CCCNC(CC2CC(=C)C2)=O)CCN(C(=O)CC2(N(C)C)CC2)CC1 C1(CC(=O)NCC2CC(NC(C3(CC=C)CCCC3)=O)C2)CC(CC)=NO1 c1(C(C(=O)N(CCC)CCNC(C2(COC)CC2(F)F)=O)C)cc(F)cc(F)c1 C12(C(=O)NCCCCCNC(C(CC=C)CC)=O)CC(CO)(C1)OC2(C)C c1(NC(COC)=O)ccc(NC(=O)C(C)(C)OC2(OCC(F)(F)F)CC2)cc1 c1(NC2CCCN(CC)C2)ccc(S(=O)(=O)NCCC#CC(C)C)cc1Cl.C1CS1 c1(C(=O)NC(c2ccccc2)CNC(=O)CCc2nccs2)cc(Cl)nnc1O CC1CCCC(CCNC(=O)CCC(=O)C2CCCCC2)C1 c1(C(=O)NCC23CC2CN(C(c2cnc(S)[nH]2)=O)C3)ccc2oc(O)nc2c1 C1(NC(C(c2cncn2C)C)=O)CCC(C(=O)NCCCn2ccnc2)C1 n1(CC)ccc(CNC(=O)CC2CCN(C(C3(CCN=[N+]=[N-])CC3)=O)C2)n1 C1(NC(C2(C)CC=CCO2)=O)CCN(C(c2scnc2Cl)=O)CC1O c1(C(=O)NC2C(N(C)C)CC2)cccc2cncn12 N1(C(c2noc(CC)c2C)=O)CC2CCCC2(C(N2CC(SC)C2)=O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC2OCCN(C(=O)C(C)C(F)(F)F)C2C1 C1(C(C)(F)F)(C(=O)NCC(C)CNC(=O)C(F)=C2CCCC2)CCOCC1 c1(OCC)cncc(C(=O)NCC2C3CN(C(=O)C(O)C(C)C)CC23)c1 C1(C(=O)NCC2C(NC(c3ccc(-c4ccccn4)s3)=O)C2)CCC(F)CC1 CC(C)CCCCC(=O)NCC12CN(C(=O)C(C)OC(C)(C)C)CC1CCO2 c1(NC)ncccc1C(=O)NCC1CC(C)N(C(=O)CCN2CCC2)C1 N1(C(c2cncc(C)c2)=O)CCC2CCC(NC(C3CC(C)CCO3)=O)C12 C1(C(C)C(=O)NC(c2scc(CC)n2)(C(C)C)OC)CCN(CC)CC1 C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CC2CN(C(CCSCCC)=O)C1C2 CCCCC(CNC(c1cc(C)n(CCO)n1)=O)NC(C1CCCO1)=O CCC(CC)C(=O)N1CCCC1CC(=O)N(c1cncc(C(=O)OCC)c1)CC c1(C2C(C(=O)O)C2)ccccc1C(=O)Nc1ncc(CCN2CCOC3CC23)s1 C(=O)(C1CCCc2c(O)cccc21)NC1(COC)CN(C(=O)C(O)C(F)(F)F)C1 c1(N(CCNC(c2ncoc2-c2ccon2)=O)C2CC2)ncc2scc(Br)c2n1 C(CCN=c1ncc(C2CC2)c[nH]1)NC(c1ccc(C)nc1)=O Cc1nn(C)cc1CC(=O)N(C1CN(C(c2nn[nH]c2C(F)(F)F)=O)C1)C CCC(CC1CC1)C(=O)N1CCC(C)(NC(c2cc(COC)on2)=O)C1 C(=O)(CCC(F)F)NC(C)CCCNC(C1(C)CC1C(F)(F)F)=O Cn1nc([N+](=O)[O-])cc1CNC(=O)NCC(=O)NCC1(C)CCC1 N1(C(C(C)OCC)=O)CCOC2(C1)CN(C(c1cccc(Cl)c1F)=O)C2 N1(C(CCC(N)=O)=O)Cc2ccc(CNC(=O)CCn3ccnn3)cc2C1 c1(C(N(C(CNC(CSCC=C)=O)C)C)=O)ccc(NS(=O)(=O)CCCC)cc1 Cc1cc(C(=O)NCCCN(C)C(c2cn(C)nc2C2CC2)=O)nnc1O N1(C(c2ncn(C)c2)C(=O)NC2CC2)CCSC2CCCCC12 c1(OCC(=O)NC2(CN(C)C(c3cnn[nH]3)=O)CC2)ccc(F)cn1 c1(C(=O)NC2C(NC(C3(OC)CCOC3)=O)C2)sc(C#N)cc1C N1(C(C(c2cccnc2)OC)=O)CC(NC(=O)C(O)CC(N)=O)C2(CC2)C1 C1(CC#C)(C(=O)N(C2CCC3CC23)C)CCN(C(C2CC2(F)F)=O)C1 N1(C(C2C(C)CCCC2)=O)CCCC2(CCN(C(C3CCC(C)(C)OC3)=O)C2)C1 C1(NC(=O)CC(O)CNC(C2CCN(CCC)C2)=O)CCC(=O)N(C)C1 CC1C(NC(c2cccc(S(C)=O)c2)=O)C(C)CCN1C(c1cnn[nH]1)=O N1(C(c2c(O)ccc(C)c2)=O)CCC(N2CCCC(Cn3cc(Br)cn3)C2)C2(CC2)C1 CC1CN(C(=O)Cc2nccn2C)C1C(=O)NC(C1CCCCC1)C C1(CNC(C2ON=C(C)C2)=O)(CO)CC12CCN(C(c1sccc1F)=O)CC2 N1(C(C2(O)C(C)(C)C2)=O)CC(C2CCCCN(C(c3ccc(C4CC4)s3)=O)C2)C1 N1(C(c2c(O)cncc2F)=O)CC=C(c2ccnc(Cl)c2F)CC1 N1(S(C(C)C)(=O)=O)CCOC2(CCCN(C(c3cc(Br)cc(F)c3C)=O)C2)C1 CCC(CC(=O)NC(C)C(=O)NCC(C)(F)F)OC C1(C(N2C(C)CN(C(C3(O)CCOCC3)=O)CC2)=O)CC2CSCC(C1)C2 C1(C(N2CCC(N(C(=O)C=CCO)CCO)C2)=O)CCc2nnc(C(F)(F)F)n2C1 c1(C2C(C(=O)NC3C(NC(C=C(C)Cl)=O)CC3)C2)cnn(C(C)C)c1 c12cn(nn1)C(C)C(=O)N2.C(C)(C(C)(C)C)N(CC(=O)OC)C1CC1 C1(CNC(CCS(C)=O)=O)CN(C(=O)CC(F)(F)Cl)C2(CCC2)C1 Cc1ncc(CNC(=O)C(CC2CCOCC2)NC(=O)Cc2nonc2C)[nH]1 N1(C(C(N2C(C(=O)O)(Cc3c(C)cccc3)SCC2)C)=O)CCS(=N)(=O)C(C)C1 N1(C(C=CCC)=O)CCC2(CC1)CN(c1ccnc(C(=O)OC)n1)CCO2 N1(C(c2c(SC)cn(C)n2)=O)CCCC(NC(=O)CC2CCOC(C)(C)C2)CC1 N1(C(Cc2cnc(C)s2)=O)CCC2CCC12CNC(=O)C#CC(C)(C)C c1(C(N2CC3CCN(C(=O)CCC(F)F)C3C2)=O)cc(Cl)c(F)cc1F CCC(C)C(C(=O)N1CCCOC(CNC(c2cc(C)c(C)[nH]2)=O)C1)OC N1(C(c2c(CCC)n(C)nn2)=O)CC(NC(=O)CN2CCSCC2)C(C2CC2)C1 c1(OC)cnc(Cl)cc1C(N1CCC(N(C(=O)CCC(F)(F)F)C)C1)=O CC#CCCC(=O)NC(C)CC1CCN(C(C2(c3cc(C)no3)CC2)=O)CC1 CC(C)C(CCC(=O)NOCC(O)CO)NC(C1CCCCC1O)=O CCC(C(=O)N1CCCC1CNC(=O)C(C)=C1CCC1)SC N1(C(CC(C)(C)SC)=O)CC2CC(C1)N2C(C1CC1C(F)F)=O c1(C(N2CCC(C)C(N(C(=O)Cc3cncnc3)C)C2)=O)cc(F)c(O)c(F)c1 c1(C(N(CC(O)CF)CC)=O)ccc(CNC(C2CC(=O)N(C)C2)=O)cn1 Cn1ncc([N+](=O)[O-])c1N1CCC(NC(=O)C=Cc2ccsc2)C(CO)CC1 C1(NC(C2C(OCC)C2)=O)COC2(CCN(C(=O)C=Cc3cnc[nH]3)CC2)C1 n1(CC)[nH]cnc1=NC(=O)C(=O)NCC1=NOCC1 N1(C(c2nc(C)n(C)n2)=O)CC2(CCN(C(C3CCCNC3=O)=O)CC2)CC1C C(=O)(C1=CS(=O)(=O)CCC1)N1C(C)CCC(NC(=O)C=Cc2ccc[nH]2)C1 C1(CC)CC(CC(=O)N(CC(C)(C)CNC(=O)CC(=O)N(C)C)C)CCO1 N1(C(C2CC(n3cc(CNC(=O)NC)nn3)C2)=O)CCOC(C(C)(C)C)C1 CCC(C)(CO)C(=O)N1CC2CC2(CNC(=O)CNC(c2ncccc2O)=O)C1 N1(C(C(C=C)c2ccccc2)=O)CCCCCC(NC(=O)CCc2cscn2)C1 c1(SC)cccc(N(C(C)C(=O)NC2CN(C(C3CC(NC(C)=O)C3)=O)C2)C)c1 N1(C(CSc2ccc(C)cc2)=O)CC2=C(C1)CN(C(=O)CCc1cncnc1)C2 c1(CCC(=O)OC)ccc(F)c(CN2CCN(C(C)CN)CC2)c1 C1(NC(C2(CCNC(C3CCC(=O)C3)=O)CCC2)=O)CCC2(CCC2)C1 CC1=C(C(=O)NCC2(CNC(=O)C(O)C3CC3)CCC2)Cn2nnnc2N1C c1(C(N2CCC(NC(c3c(C)cc(F)cc3)=O)C2)=O)cnn2c(C)cccc12 C(=O)(C1CCCc2nc(C)[nH]c21)NCC(C)(CO)NC(c1cncc(C)c1)=O c1(CN2CCC(C)(C(N3CCS(=O)CC3)=O)C2)cc([N+](=O)[O-])ccc1Br c1(SCC)ccc(C(N2CCCC2C2(c3ccc(C(=O)NC)cc3)CC2)=O)cn1 CN1Cc2ccc(C(N3CCC(CNC(c4ncc[nH]4)=O)C3(C)C)=O)cc2C1 c1(C(=O)NCCC2(O)CCN(C(CN=S(C)(C)=O)=O)C2)scc2c1OCCO2 N1(C(C(CCC)OC)=O)C2CCC1CC(F)(CNC(C1(C(=O)NC)CCC1)=O)C2 N1(C(c2c(C)cccc2Cl)=O)CCC2(CCC(NC(=O)CC34CCCC3C4)C2)C1 Cc1ccn(C(C)C(=O)N(C(C)CN(C(=O)CN(C)C(N)=O)C)C)n1 c1(C2N(CC(=O)NC(C3CC(F)(F)C3)C)CCC2)ccc(C(F)(F)F)cc1 c1(NC(Cc2cn(CC(CC(C)C)OC)nn2)=O)ncc2nccnc2n1 Cc1cc(C(N2CCOCC2CN(C(=O)Cn2cncn2)C)=O)c2n[nH]cc2c1 C1(NC(CCSC)=O)Cc2ccccc2C1NC(c1ccc([N+](=O)[O-])cc1F)=O CC(=O)CCCC(C)C(=O)NC1CN(C(c2cc(CO)oc2C)=O)CC12CC2 c1(C(N2CCC(C(=O)Nc3ncccc3F)C2)=O)cc2c3c(ccc2[nH]1)NCC3 C1(C(=O)NC(C(O)CO)C2CC2)CC(O)CN1C(=O)CCc1cncnc1 N1(c2ccnc(NC(c3csnn3)C)n2)CCC(C)(C2CC2)C1 C1(NC(=O)Cn2cnnc2O)CCCC2CN(C(c3ccc(F)nc3F)=O)CC12 c1(C(=O)NCC2CCN(C(C(N3C(CC)CCC3)=O)=O)CC2)cc2scnc2[nH]1 c1(C(N2C(CC(=O)NC(C#C)C(C)OC)CCC2)=O)cccc(CC)c1 C1(CN(C(=O)CN(S(C)(=O)=O)C)C)CC(F)CN1C(C12CCC1C2)=O C(CCCC(=O)N1CC(N(C(=O)C(C)CCOC)C)C1)OCCC=C c1(C(=O)NCC(CNC(c2c(CCC)nco2)=O)O)cncc(OC(C)C)c1 N1(C(c2c(OC)cccc2I)=O)C2CCCC1CC(NC(C1CCCOC1)=O)C2 c1(OCC)ccc(C(N2CCC(F)(CNC(=O)CNC(=O)OC)C2)=O)cn1 C(=O)(CC(=O)NCC(C)N(C)C(c1cnn(C2CC2)c1)=O)OC c12ccc(cc1)S(=O)(=O)N2.C1(N(C)CCO)CCN(CC2CNC2)CC1.C1C(=O)N1 C(=O)(C1=CCCCN1C(=O)OC(C)(C)C)N1CC(N(CC(F)(F)F)C(C)=O)C(C)C1 c1(NCC(C)(C2CC2)OC)ccc2c(C)[nH]nc2c1 C(C1=CCN(C(=O)C(c2ccccn2)O)CC1)NC(C=C(C)Cl)=O C(=O)(C(O)P(C)(C)=O)NC1CC(NC(c2cc(NC(C)=O)ncn2)=O)C1 c1(CC(=O)NCC2CC(F)(CNC(CN(C)CC)=O)C2)ccc(C)cc1 N1(C(C(C)(C)c2cc[nH]n2)=O)CC2CC2(NC(c2cncc(C(F)(F)F)c2)=O)C1 C1(NC(C2CCCN(C(C(CO)OC)=O)C2)=O)CC12CCOCC2 C1(NC(C2CCN(C(C)C)CC2)CC)CCCC(C)(C)C1 C#CC1CCCN(C(C2CCN2C(=O)CN(C)CCOC(C)=O)=O)C1 CC(CNC(=O)Cc1ccc[nH]1)C(F)C(=O)NC1CN2CCCC1C2 N1(C(COCP(C)(C)=O)=O)CCOCC(NC(=O)C(c2cccnc2)O)C1 C1(C(N2CCCC(C)C2CCO)=O)(OC)CCN(C(=O)CCc2ccoc2)CC1 Cc1cc(CC(=O)NC2CN(C(=O)Cc3nocc3C(C)C)C2)sn1 C1(CC)CC(C(=O)N(CC(=O)N(CC(C2CC2)OC)C)CC2CC2)CCO1 c1(C(C(=O)NCCC(=O)OCC)N(C(C)CCC(C)C)C)nn(C)nc1Br c1(CC(N2CCCC(C(=O)NC3CCN(CC=C)CC3)C2)=O)c(Cl)cccc1Cl C1(CNC(C2CCN(CC)C2)=O)CC2(C1)CN(C(=O)COc1ccon1)C2 C12(C(N(CCN(C(C(CC)COC)=O)C)C)=O)CCC(C(F)F)(CC1)CC2 CCCC(CCC)C(=O)N1CCCC1C(C)NC(=O)COCc1nc(C)no1 C1(C(N2CCC(C(CNC(CCSC)=O)O)CC2)=O)C2Cc3ccccc3C12 c1(OC)cccc(CCCn2nnnc2C2(NCCF)CCC3CC23)c1 c1(CC)ccc(F)c(C(=O)NCC2(C)CCN(C(C3CC4CCC3O4)=O)C2)c1 Cn1ncc(C#N)c1NC(C1CC(O)CCN1C(c1ccc(Cl)cc1F)=O)=O N1(C(c2cncc(OCC)c2)=O)CCC2(CC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 c1(CN2CC(C)(CC(=O)Nc3c(C(=O)OC)ccs3)C2)nc(Cl)ccc1F c1(NCCN(CC)CC)cc(=NC(C)c2ccc[nH]2)[nH]c(C(C)C)n1 c1(Cc2nnc(-c3ccc(OC)cc3OC)o2)cn2cc(Cl)cc(Cl)c2n1 N1(C(C2C(CNC(c3ccc(O)nc3)=O)CC2)=O)CCC2CCCC2CC1 N1(CC(N2CC(CC(F)C(=O)NCc3ccc(O)cc3)C2)=O)C(=O)CCCC1=O CC1(C)CC(=O)N(CC(=O)NCCNC(C2(C3CCCO3)CCCO2)=O)C1=O c1(C(N(C2C(C)(C(=O)O)CCC2)C(=O)CCN2CCC2)=O)cc(Br)cnc1O c1(Oc2c(CNC(CC(C)C3CC3)=O)cccc2)ccc(Cl)cc1Br C12(CNC(C3(C)COC3)=O)CCC(CNC(=O)C#CC(C)(C)C)(CC1)CO2 C=CC(C)(O)CC(=O)N1CCC(C(C)(C)NC(=O)CCc2ccc(C)c(C)c2)C1 C1(CN(C)C(C2(C(F)F)CC2)=O)COCCN1C(=O)C(O)C1CC1 C(CC(=O)NCC1(F)CCOCC1)(C(F)(F)F)NC(C(COC)C)=O C#Cc1ccccc1CC(=O)NC(C)(C)CCN(C(=O)CCCC#CC)C CC(C(=O)NCC1(NC(C2CSC2)=O)CCOC1)C(=O)N1CCOCC1 C1(NC(c2cc(CNC(C3CCCC3)=O)oc2)=O)CC2CC1OC(=O)N2 CC(O)C(C)(C)C(=O)NCCC(C)NC(C1CCN(C)C1)=O Cc1ccc(Cl)c(N)c1C(=O)NC1CC1CNC(C12CC(C(F)(F)F)(CO1)C2)=O C1(NC(c2csc(Cl)c2)=O)CCOCC1NC(C1CC(F)(F)C1)=O c1(CNC(C2C(C)CCCC2)=O)ccc(C#N)cc1F.C12CC(C)(C)CN1C2=O N1(C(CNS(C)(=O)=O)=O)CC2ON=C(CNC(c3ccc(C(N)=O)cn3)=O)C2C1 CCC(C(=O)NN(C(=O)NC(=O)OC(C)(C)C)S(C)(=O)=O)C1CCOC1 C(=O)(C1c2ccccc2C2CC1C2)NC1CC(NC(C(CC=C)CC)=O)C1 C(=O)(C1(C)CCCc2ccccc21)N(C)C.C12CC3CCCC(C1)N3C2=O c1(C(=O)NCCN(C(C)C)C(c2cccc(N)c2F)=O)ccc(F)cc1F C1(NC(CSC(=N)N)=O)COC2(C1)CN(C(c1cc(C(F)(F)F)on1)=O)C2 C1(NC(=O)NC2(c3cccc(Cl)c3)CCC2)CC2C(C1)C2(F)F c1(C(=O)NC2C(C)CCN(C(c3c(C(C)C)ncs3)=O)C2)n[nH]c2ccccc12 CC1CCN(C(C2CCSC2)=O)CCN1C(c1ccc(CO)c(F)c1)=O C1(NC(C=C(COC)C)=O)CC2C1CCN2C(c1nnn(-c2ccccc2)n1)=O Cc1cc(C(=O)NCC2CCN(C(=O)CCc3ccoc3)C(C)C2)cc(N)c1O N1(C(c2c(N)nccn2)=O)CCC2CN(C(=O)CC3CS(=O)(=O)C3)CC12 CC1C2C(CCN2C(=O)C2=CCCC2)CN1C(=O)CC1(O)CCCCC1 C1(CCC)(NC(=O)COC)CCCN(C(c2cc(C)ccc2-n2cncn2)=O)C1 c1(C(=O)NCC(CNC(Cc2nc(C)sc2)=O)CO)nnc2n1CCCCC2 C(CC1=CCCCCC1)NC(C1N(C(CCCOC)=O)CCC(C)C1)=O C1(C(C)NC(C2(O)CCC2)=O)CCN(C(=O)Cc2ccccc2)C1 c1(C(=O)NC2CN(C(C(=CC3CCCC3)C)=O)C2)ccc(Br)cc1O C12CCCC3CN(CC13)C(=O)N2.CC(CCC1CC1)NC(=O)OC(C)(C)C c1(C(N2CCC(C(=O)NCC3CN(CC)C(=O)O3)(CF)C2)=O)cncc(F)c1C c1(NCC2CC(C)(COC)C2)ncnc2onc(C)c12 CCC(C(=O)NC1CC(NC(c2c(Br)ccc(F)c2F)=O)C1)C(C)(F)F C(=O)(C(CC(C)=O)NC(=O)C(C)CN1CCCC(C=O)C1)OC.c1(C)ccccc1 N1(C(CCC(=C)Cl)=O)CCCC(NC(=O)C(O)Cn2cncn2)CC1 c1(C(C)=O)cc(=NCc2ccccc2CNC(C2CCc3nncn3C2)=O)[nH]cn1 c1(CCN2CC(=O)N(CCc3nnn(C)n3)C2=O)nc2cc(F)c(F)cc2[nH]1 Cc1ccccc1C(C)C(=O)NCC1COCCN1C(C1CC1(C)C)=O Cc1nncc(CNC(C2CN(C(C3(C)CCCOC3)=O)CC2(F)F)=O)c1C C1(C(N(C2CN(C(=O)C(F)=C3CCC3)C2)C)=O)CCC(=O)N2CCCC12 C1(C(=O)NC2CC(O)C2)CN(C(c2ccc(Br)cn2)=O)Cc2cccn2C1 Cc1cc(-c2cn(CC3CCCN3C(=O)CCOC(C)C)nn2)sc1C N1(C(=O)OC(C)(C)C)CCC2(CCC(C(N3CCC(C)(NC(=O)C4CC4)C3)=O)C2)C1 Cc1nnn(NC(=O)CC2CN(C(=O)CCN3CCOC3=O)CC23CC3)c1C CC1(C)CCC(=CC(=O)NCCC2CN(C(C3(Cl)CC34CCC4)=O)CCO2)CC1 c1(OCCC)ccccc1NCC(O)CNC(=O)C1CC1.C1(=O)C(C)(C)CN1 c1(-n2c(-c3nc(OC)ccc3Cl)nc(CCCCC)n2)cc(Cl)ccc1OC c1(C(=O)NCC2(C)OCCN(C(Cc3cn(C)nc3)=O)C2)cnc2[nH]nnc2c1 CC1=C(C(=O)NCC2CCCN(C(=O)CCc3ccoc3)C2)CCCC1 c1(C(=O)NCCCC(C)NC(c2c(OC)n[nH]c2)=O)nn(C)nc1C C1(C(=O)OCC)(CO)CN(N2CC(CO)C(C)(COC)C2)C1 C1(C(=O)NCC(=C)C)CCC2(CN(C(c3cc(F)c(Cl)cc3C)=O)C2)O1 c1(C(=O)NC2C(CNC(Cc3cc(C)ns3)=O)C2)c(C)cc[nH]c1=N CC(CC(N)=O)C(=O)N1CC2(CCN2C(=O)C(O)CC(=O)c2ccccc2)C1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(CC(C)NC(C(C(CC)C)OC)=O)C1 Cc1ccc(C(c2nnnn2C2COC2)NC2CC(=O)N(O)C2)c(C)c1C N1(C(=O)OC(C)(C)C)CCCC12CCCN(c1ccc([N+](=O)[O-])cc1C#N)C2 Cc1cc(C#N)ccc1NC(c1cnn(-c2ccccn2)c1C)=O N#Cc1cc(C(=O)NCC2CCN(C(c3cc(F)c[nH]3)=O)CC2)ccc1[N+](=O)[O-] c1(C(=O)NCC2CN(C(CC=CCC)=O)C(C)C2)cn(C)c2ncccc12 c1(C(N2CC(NC(C(CN(CC)CC)F)=O)(CO)C2)=O)cc2ncccc2o1 CC1(CCNC(C2(F)CC2)=O)CCN(C(c2cccc(O)c2F)=O)CC1 C1(C(C)(C)C)C(NC(C2CCC(C)(C)C2)=O)CCN1C(=O)CNc1ncccn1 Cc1nc(C(=O)NCCn2cc(CCc3ncccc3F)nn2)c(C)o1 c1(C(=O)NCC2CC(NC(C(C)N(CC(F)(F)F)C)=O)C2)c[nH]nc1C(C)(F)F c1(C(N2CCN(CCCNC(C)=O)CC2)=O)c(C)nc2ccc(N(C)C)nn12 c1(NC(N2CC(CC)(CO)C2)=O)ccccc1OC(c1ccc(Cl)cc1)C(C)C N1(C(c2oc(C)c(Br)c2)=O)C2CCC1CC(CNC(C1CC1(C)C)=O)C2 C1(NC(CCOCCOCC)=O)CCC(CNC(=O)C=CC2CCCO2)CC1 Cc1nc(Cl)[nH]c(=NC(C)C2CN(C(c3cccc(OC(F)F)c3)=O)C2)c1F C1(C(N2CCC(CNC(=O)CC3OCCCO3)C2)=O)(OC)CC(CF)C1 c1(OC)nc(N(CC(O)CN(C2(C)CC2)C)C)nc2[nH]cnc12 c1(C(C)(C)C)cc(C(=O)NCCC2(NC(C3(C)CCCO3)=O)CC2)no1 N1(C(C(F)=CC)=O)CCC(CNC(c2nc(-c3cccs3)oc2C)=O)CC1 C=CCC(C(=O)N1CC=CC1C(=O)NC1CCOC(C2CC2)C1)NC(C)=O C1(NC(c2cnnc(O)c2)=O)COC2(C1)CN(C(=O)Cc1cscn1)C2 C12(CNC(C(CC=C)(F)F)=O)CCCCC1CN(C(c1cc(OC)n[nH]1)=O)C2 C1(C(=O)Nc2c(CC)nn(C)c2)C(C)OCCN1C(=O)C(N1CCOC1=O)C c1(C2CCN(C(c3ccc(-c4ccc(F)cc4)nn3)=O)C2)ccnc(Br)c1 c1(C(=O)NC(C)CN(c2nc(-c3ccccc3)ns2)C)coc(C2CCC2)n1 C(=O)(C(F)C(C)(C)O)N1C(CCNC(c2c(C)oc(C(F)(F)F)n2)=O)CCCC1 c1(C(N2C(C3(NC(CCCOC)=O)CC3)CCC2)=O)cccc2c1NCC(C)C2 Cc1nc(O)sc1C(=O)NCC(C)NC(=O)C(C)CN(C)C C(=O)(C1Cc2ccccc21)NCC(C(=O)NCC1CCN(C(CC)=O)C1)O C1(C(N(CCOC)CC)=O)CCCCCN1C(c1cnncc1OC)=O C1(CC(=O)NC2CC(C(C)C)OC2)CCN(C(=O)CN2CC3CC3C2)C1(C)C N1(C(C(C2CCOC2)NC(=O)CC2CCCC2)=O)CCCC2(CC2)C1 c1(C(=O)NC(CSC)(C)C(=O)N(C)CCOCCCO)ccc(C)c(O)c1 C1(CNC(C(C=C=C)C)=O)CN(C(c2ccnc(CC(C)C)n2)=O)CCC1(F)F C1(NC(=O)C=Cc2ncc[nH]2)CC2CCC(C1)N2C(c1ccc(F)c(Cl)c1)=O N1(C(c2ccc3nc(C)sc3c2)=O)CCC(N=c2[nH]c(C(C)C)ncc2Br)C(C)C1 C(=O)(Nn1ccccc1=O)C1(NC(C2CC(C)OC2C)=O)CCCC1 CC(O)CCC(=O)N1CC(C)CC1C(=O)Nc1ccnnc1O c1(CN2CCC(CC(=O)Nc3c(C)c(Br)ncc3)C2)ccc2c(c1)OC(F)(F)O2 N1(C(C)=O)CCCC1CC(=O)N(C(C)CNC(C1OCCCO1)=O)C N=c1[nH]cnc2c1CN(c1nc(N3CCC(CCO)C3)c3c(n1)COC3)CC2 c1(CC(=O)Nc2cccc(NC(C(CCCC)O)=O)c2)ccc2c(c1)CCCS2 N1(C(CC(C)F)=O)C2CCC1CC(CNC(c1ccc(Cl)cc1C(F)(F)F)=O)C2 C1(NC(C2N(C(Cc3c(C)n[nH]c3)=O)CC=CC2)=O)COC2(CCCC2)C1 C(CCC(O)C(=O)NC1(CSC)CCCC1C)NC(CCSCCCC)=O C(=O)(C(CO)C(C)(C)C)N1CCC(NC(COCCCCCC)=O)C1 C(C(CC1CC1)C(=O)N1CCC(N(C)C)C1)NC(c1cnc(CC)o1)=O C1(CC)(NC(c2cnc(OC(C)C)cn2)=O)CCCN(C(c2occc2C)=O)C1 CC1(C)CN(C(c2cccc(Br)c2F)=O)CC1NC(c1ccncc1N)=O C(=O)(C(C)(C)C(=O)NC1(CNC(C2(OC)CCSC2)=O)CCCCC1)OC CC1(C)CN(C(C2CC3CCC3C2)=O)CC1CNC(c1ccnc(C(N)=O)c1)=O c1(C(N(CCCCNC(=O)COC2CC=CC2)C)=O)ncccc1N(C)C C1(OC)CCC(C(N2CCC(F)(CO)C2)=O)CC1.C12(CC1)C(=O)N2 c1(CCC(=O)N(C)CCNC(C2(F)CC(C(=O)OC(C)(C)C)C2)=O)ncccc1F c1(OC)ccc(Br)nc1CNC1C=CC(C(=O)NCCOC(F)(F)F)C1 c1(C(N2C3CC(NC(C(C)=C4CCC4)=O)(C3)C2)=O)ccc(Br)cc1Cl CC(CC#C)(C(=O)N1CCCc2ccnn21)NC(=O)Cc1ccc[nH]1 N1(C(c2ccc3n[nH]cc3n2)=O)CCC2CN(C(C3(CF)COC3)=O)CC2CC1 N(C1CCCc2ccc(F)cc21)C(c1cc(CC)on1)c1nnnn1CCSC CC1(C)C(NC(=O)CCc2cc(F)c(F)c(F)c2)C(C)(C)C1O Cc1cc(C(=O)N(C2CCC3CC23)C)c(O)c(C)n1 C1(O)(CCNC(=O)Cc2nc[nH]n2)CCN(C(=O)CC2CC(=O)NC2=O)CC1 N1(C(c2ccn(CCCC)n2)=O)CC(C)N(C(=O)CCN2CCOCC2)CC1C C1(C(N(CC=CC(=O)N(C)Cc2ccn(CC)n2)C)=O)CC(=O)CC(=O)C1 c1(CNC(C2(CC)COC2)=O)ccnc(C(=O)NOC2CCC(O)C2O)c1 N1(C(CC(=O)OCC)=O)CCN(C(c2cc3sc(CC)cc3s2)=O)CCC1C C1(CC(=O)OC(C2CC(OCC)C2)=O)CCC2CN(C(=O)OC(C)(C)C)CC12 C#CCC(C)C(=O)NCC1C(C)CCN1C(=O)CN(S(C)(=O)=O)C c1(C(=O)NC(C2N(C(CC(CCC)C)=O)CCC2)(C)C)cc2ccccn2c1 c1(OC)ccc2c(c1)N1CCN2Cc2ncc(s2)C1=O.C(CN)SC c1(C(=O)NCC(C)N(C(=O)C(O)C(F)F)C)ccc2c(c1)CCCC(=O)N2 c1(OC)ccc2ccccc2c1CN1CCC1C(=O)NCc1cn[nH]c1 C(C1=Cc2ccccc2OC1)NC1C(SCc2c(F)cccc2)CC1 C(=O)(C(CCNC(c1cc(CO)oc1C)=O)OC)NC(C1CCCOC1)CC N1(CCS(N)(=O)=O)CCC(NC(=O)NC(CC(=O)O)c2ccccc2)CC1 CCCCC(C)C(=O)NCC1(CCNC(C2CCC(N(C)C)C2)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)NC1CCC(CNC(=O)CC2CCNC2=O)C1 Cc1[nH]nc2c(C(N3CCCC(C(N4CCOC(C(=O)O)C4)=O)C3)=O)cccc12 C1(NC(CN(C(c2ccc(Cl)cc2)C(=O)NC(CC)C)C)=O)CC(N=[N+]=[N-])C1 C1(C(=O)NC(CC(C)C)C(=O)NC)(NC(C(C=C)CC)=O)CCC(C)(C)C1 N1(C(C23N(C(=O)OC(C)(C)C)C(CC2)CC3)=O)CC(C2CCCCC2)C1 c1(N2C(C(C)O)CC2)nc(=N)c2ncc(Br)n2[nH]1 C=CCC(C)(CNC(=O)C(c1ccoc1)NC(=O)C(F)n1ccnc1)CO N1(C(c2c(C)scc2)=O)CCC(OCCNC(=O)CC23CCCC2C3)CC1 N1(CCC)CCCC(C(=O)NCC2CC(F)CN2C(c2cn(C3CC3)nn2)=O)C1 C(=O)(CC(C)CNC(C1(C)CC1(C)C)=O)NCCN1CC(OC)C1 N1(C(COCCOCC)=O)CC(N(C)C(C2CC3CCC2CC3)=O)C(C)(C)C1 C1(C(N2CC(CNC(CN(CCCCCC)C)=O)C2)=O)CC(C(C)=NO)C1(C)C C1(C)(CNC(c2c[nH]c(=NC)s2)=O)CN(C(C2(C)C=CCCC2)=O)CC1C Cc1nc(NC2C(C)CCC(C)(C)C2)c2cc(C)sc2n1 C1(NC(c2ccc(SC)s2)=O)(CO)CCN(C(c2nc(C)ccc2C)=O)CC1 c1(C(N2C(=O)NC(CC(C)C)C2=O)C)ccccc1[N+](=O)[O-] c1(C(=O)NCCCN(C(=O)Cc2ccc(C)cc2)CC)nn(C(C)(C)C)cc1Cl c1(C(N2CC(NC(c3sccc3Cl)=O)C(O)C2)=O)cc(F)c(F)cc1Cl C1(NC(c2ccccc2Cl)c2n(CCC)nnn2)CCCCC12CC2 N1(C(CN(c2ccccc2CO)C)=O)CCCC2(C1)CN(C(c1cc[nH]c1)=O)C2 c1(C(N(CC(C)(C)NC(C(=O)NCCOC)=O)C)=O)cc(Cl)c(OC)c(Cl)n1 c1(C(N2CCC(N(C(=O)CCn3cnnn3)C)CC2)=O)cc(F)c(CO)c(F)c1 N1(C(c2sc(C)c(O)n2)=O)CC(NC(=O)C(O)C2CCCC2)C2CCCC12 N1(C(c2cccc(CC=C)c2)=O)CC2CCN(C(c3cc(C)c(Cl)s3)=O)C2C1 Cn1cc2c(n1)CCCC2C(=O)NCC1(C)CCN(C(c2ncc(F)cn2)=O)C1 C(C(F)(C(=O)NC(C)(C)CCCO)C(C)C)NC(CCNC(=O)OCC)=O c1(C(N(CC(CO)(CO)NC(Cc2c(C)non2)=O)C)=O)cccc2ncsc12 N1(C(C2N(C(=O)NC)CCC2)=O)CCCCCCC1C(=O)NC1CCNC(=O)C1 N1(C(c2c(OC)scc2)=O)CCCC(C2(NC(C3COC4COCC34)=O)CC2)C1 C1(CC)CCCCCCN1C(=O)CNC(C1CC(=O)C12CCC2)=O N1(C(CC(C)c2ccco2)=O)CCCOC(CCNC(=O)CC2CCN(C)C2)C1 N1(C(CCCOCCC)=O)CC(C(F)(F)F)CC1CNC(=O)C(CC)SC C1(CC(=O)N(C2CCN(C(c3cnco3)=O)CC2)CC#C)CCCS1(=O)=O C(=O)(C(CC)CC=C)NC(CCC=C)C(=O)NCCCCC(C)(F)F CCC(C(C)C)NC(=O)C#CCNC(c1cnc(C)o1)=O C1(N(CCNC)C(C2(C)CC2C(C)C)=O)CCNCC1 C1(C(=O)NC)CCCCN1C(=O)CSC1CCN(c2cccc(F)c2)C1=O C(=O)(C1=C(C)CCOC1)N(CCCN(C(CCC(=C)C)=O)C)CC CCCCCC(C)(C)C(=O)NC(C1CC=CCC1)C(=O)NCCc1cnn(C)c1 CCC(CC(=O)N(CC(O)CN(C(=O)CCn1ccnc1)C)C)C(C)(C)C c1(N(C(C(CC(=O)OC)CC2CC2)=O)C(C)C(=O)N2CCCC2)ccnnc1O Cc1ccc(C(=O)NCC(C)(C)CN(C)C(C2CS(=O)(=O)C2)=O)cc1Cl C(CCCCNC(C1CC(C)C1)=O)N(C(CCSCC)=O)C c1(C(=O)NC(CCNC(c2nn(C)c(Cl)c2)=O)(C)C)ccc(O)c(Cl)n1 N1(C(C2(COC)COC2)=O)CCC(C)C(NC(c2ccncc2C(F)F)=O)C1 C1(CC(=O)NCC(F)(F)F)(OC)CN(C(C2(c3ccccn3)CCC2)=O)C1 C12(C(C(F)(F)F)NC(C3CC3OCC3CC3)=O)CC3CC(CC(C3)C1)C2 c1(C(N2C(C(=O)Nc3cnc(C(N)=O)nc3)C(O)CC2)=O)cccc(F)c1F Cc1cc(NC(C2CC2)=O)ncc1-c1nc(C2CCC3CC3CC2)no1 N1(C(COCCCCC)=O)CC2CC2C1C(=O)N(C)CC1(COC)CCC1 C1(NC(c2cc(C(N)=O)oc2)=O)CC(=O)N(C2CN(C(C3CC3C(N)=O)=O)C2)C1 c1(CNC(=O)NC(CCOC)C)c(C)cccc1O N1(C(=O)NC(c2ncc(C)[nH]2)C(C)(C)C)CCOc2ncccc2C1 c1(C2C(C(=O)NC(CNC(CS(C(C)C)(=O)=O)=O)C)C2)ccnc2ccccc12 Cc1ccc(C)c(C(N2CC(CC(=O)NOCC(O)C(C)C)CC2C)=O)c1 C1(C(=O)NCCc2c(C)cnn2C)CCC(=O)N(C2CC2)C1 C1(C(=O)OC(C)(C)C)(CF)CCN(N2CCC3CCN(C)C3C2)C1 c1(OC)ccccc1C1CNCCN1Cc1noc(-c2ccccc2)n1 c1(CNC(c2ccncc2-c2ccc(CO)cc2F)=O)cccc(Cl)c1Cl c1(C(N2CCOCC(CNC(C3CC34CCCC4)=O)C2)=O)cc(Cl)cc(F)c1F c1(CCC)c(C(=O)NC(C)C(CO)NC(c2csc(C(C)(C)C)n2)=O)nnn1C C(CCCCC(=O)NCc1c[nH]nc1C(=O)NC1COCCC1(F)F)OCC CC1OCCC1CC(=O)NCc1cc(C(=O)NCCc2c[nH]nc2O)co1 c1(NCc2c(CC)nns2)ccc2ccccc2c1 C1(C(N2CC(OC)CC(CO)C2CO)=O)CCC2(CC1)CC(CN)C2 N1(C(C)C)CC2CC1CN2C(=O)CCC1CCN(C(C2CCOC(C)(C)C2)=O)C1 c1(CCOC)cc(Cl)cc(Cl)c1NC(c1cccc(F)c1-c1c(OC)cccc1)C N1(C(CCCNC(C)=O)=O)C2CCC1CN(C(C1COCC1C(F)F)=O)C2 C1(CNC(CCCN(C(C(C)CC2CC2)=O)C)=O)CCCOC1(C)C n1(CC(=O)NC(C)CC2CN(C(=O)CC3CCC3)C2)cnc(Br)c1 C1(NC(CC2C=CC(NC(c3cnn(C)c3C#N)=O)C2)=O)CC12CCCCCC2 n1(CC(N2CC(CCCCNC(CCOCCOC)=O)C2)=O)ccnc1C CCCC(C(=O)NCCC1(O)CN(C(c2ncsc2C2CC2)=O)C1)NC(N)=O C=C1CCN2C(C1)C2=O.N1(CCC(=O)NC)CCC(C)CC1 C1(NC(C(CC)Oc2ccccc2Cl)=O)CCN(C(=O)CC(C)C)CC1(F)F CC1(F)CCN(c2nnc(-c3cccc(Br)c3)n2CCN2CCCCC2)C1 c1(NC(c2n(C(CC)(C)C)nnn2)C2CN(CC(F)F)C2)ccc2nccn2c1 n12cc(nn1)C2.n1(NC(C2CC(N(C(C)=O)CC)C2)=O)cc(C)cn1.C1(=O)CCO1 C1(CNC(c2cncc(Cl)c2)=O)CC2CN(C(=O)C(F)n3cccn3)CC12 O=C(C1=CCSC1)NCC1(CNC(=O)CCc2ccoc2)CC1(F)F c1(CC)nnc(N2CC3C(CNC(=O)CN4C(C)CCC4C)C3C2)c(C#N)c1CC c1(CN(C)Cc2c(F)cc(Cl)cc2F)cccc2c[nH]nc12 N1(C(C2C(CCC)C2)=O)CCCC(C(=O)N(C)CCC)C1CC CCCCC(O)C(=O)NC1C2CC1N(C(C1CCN(C3CC3)CC1)=O)C2 c1(C(=O)NC(C2CCN(C(CSC)=O)C2)(C)C)cc(C(=O)OC)oc1C CCCC(O)C(=O)N1CCC(CN(C)C(c2ccc(-c3ncnn3C)cc2)=O)C1 CC1OC2(C(=O)NC3CN(C(=O)Cc4cnccn4)CC3C)CCC1CC2 C(CC(C)(C)CC(=O)NCc1cnc(OC)cn1)OC c12ccc(OC)c(c1)ON(C(C1C(C)(C(=O)OC)C1)=O)CCNC2=O.C1(C)CC1 CCCCCCC(CC)C(=O)NCC1CCN1C(C12CCC(CC1)C(C)O2)=O C1(NC(C(N2CCC(O)CC2)C)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1F C1(OC)CC(C(=O)NCC2CCC2NC(=O)COc2ccccn2)N(C(C)=O)C1 C1(NC(C(C(C)C)OC)=O)CCN(C(=O)C=Cc2cnn(C)c2)C12CCC2 c1(C(=O)NC2C(NC(C3N(C)C(=O)OC3)=O)CCC2)ccc([N+](=O)[O-])cc1F C=CCCCC(C)(C)C(=O)N1CC2CC2(CNC(c2oc(C(F)F)cc2C)=O)C1 CC1=C(C(=O)NCC2CC(C)CN(C(=O)CCC3CCCO3)C2)CCC1 C1(CC=C)(C(=O)NCC(=O)NOC)CCCN1C(=O)CCC1CCCCO1 c1(OC)c(Cl)nc[nH]c1=NCC1(NC(=O)COC(=O)C2CC2)CCCC1 c1(C(=O)NCC(CC)NC(=O)CCF)cc(OC)c(Cl)cc1Cl CCC(C)(COC)C(=O)NC1CC(O)CN(C(=O)C(C)(C)COC)C1 c1(OC)cccc2c1OCCC2OC(=O)CS.c1(CC#N)ccc(F)cc1 C1(NC(C(CC)O)=O)CN(C(=O)C(c2csc(C)n2)=O)CCC12CCC2 c1(C(C(=O)NCCC(C)N(C(=O)C(C)=C(C)C)C)OC)ccccc1SC c1(OC)nc(C(N2CCC(OCC(=O)N(CC(C3CCCC3)O)C)C2)=O)co1 CC1CC(C(=O)NCC2CCN(C(c3cnn(CCF)c3)=O)CC2O)CC(=O)N1 C1(CC(N2C(COC)CC2)=O)N(C(c2csnc2OC)=O)CC1(C)C N1(C(CCC=C)=O)CCC(C(=O)NCc2ccnc(F)c2)C(C)(C)C1 c1(C(=O)OC)cc(S(=O)(=O)NC2CCS(=O)(=O)C2)ccc1C c1(C(=O)NC2(C(=O)NCC#CCN(C)C)CCCO2)cccc(OC2CC2)n1 C(CC(C)(C)C)(C(=O)N1CC(C(=O)NCc2ncc(CO)o2)C2(CCC2)C1)OC N1(C(CC=C=C)=O)CC2CCN(C(c3scnc3C(C)C)=O)CCC2C1 C1(NC(c2cnc(OC)nc2)=O)CCN(C(=O)C(C)CSC)CC(C)(C)C1 CC(C(=O)O)C(C)(C)CC(=O)NC(C)CCNC(c1ccccn1)=O c1(C(N2CC(C(=O)Nc3cc(C)c(F)cc3)CC2(C)C)=O)cc2cccnn2c1 N1(c2ccn(C)n2)CCCCNC(=O)C(F)(F)C1.C1CCCCCC(=O)N1 C(=O)(C1=CCCCC1)N1CCC(C)(C(=O)NC(CCO)C(F)F)C1 CCC(C)CC(=O)C(=O)N1CCC1CC(N1CCCC(C)(C)C1)=O C#CC1CCN(C(C2COC(CNC(=O)C(O)C3CCCC3)C2)=O)C1 N1(C(C=CC(CC)C)=O)CC(C(F)(F)F)CC1CNC(=O)C(c1ccccc1)O C(=O)(CCC(C)=O)NCC1C(C(=O)NCC(COC)(F)F)OCC1 C#Cc1cnn(CC(N2CCC(C(=O)NC(C)Cc3cccs3)(CF)C2)=O)c1 C(=O)(C(C)(C)C(C)(C)O)NCC1N(C(Cc2c(C)cccc2Cl)=O)CCCCC1 c1(C(=O)NCC(C(C)C(C)C)NC(CCCSC)=O)c(C)ccc([N+](=O)[O-])c1C c1(OC)ccc(-c2cn(C3CCN(C(C4CC(O)C(F)C4)=O)C3)nn2)cc1Br c1(C(=O)NC(C2CCN(C(=O)Cc3sc(O)nc3O)C2)C)cncc(C2CC2)c1 c1(C(=O)NCC(CC=C)NC(c2cn(C)c(C)n2)=O)cccc2c1CCC2 c1(C(N2CC(NC(=O)OCC)C2)=O)cc(CNC(c2csc(Cl)c2)=O)ccn1 N1(C(CCCOC)=O)CCCOC(CCNC(=O)CC=Cc2ccccc2F)C1 C1(C(C)C)CCCN(C(=O)CCN(CCO)C(C2(Cl)CCC2)=O)CC1 c1(C(N2C(C(=O)NC(C#C)C)CC3CC32)=O)cc(Br)c(C)c(Br)c1 NS(=O)(=O)c1ccc(-c2csc(CNC(=O)COCC3CCCO3)c2)cc1 N1(C(=O)Nc2nn(CC)c(O)c2)CCC2(CC1)CC(NC(=O)OC(C)(C)C)C2 C(CCN(C)C(c1ccc(C)nc1O)=O)(C(C)(C)C)NC(CC(=C)C)=O c1(CC(=O)NC2C(C)CN(CCc3ccc(F)cc3)CC2)cccc2nsnc12 c1(C(=O)NCc2ccc(C(=O)OCC)cc2)n[nH]c2cc(OC)c(OC)cc12 Cc1nc(C)c(F)c(=NCC2C(C)CCCN2C(c2scnc2C)=O)[nH]1 C1(CC)CCOCCN1C(C1CC2C(C1)C2(F)F)C(=O)NC C1(CNC(CCCCCC)=O)(NC(=O)CC(C)CN(C)C)CCC(F)(F)CC1 C(CO)(CCCCNC(C1CCCC1)=O)NC(CCNC(C)=O)=O CN1CC=C(CC(=O)NCC2CCN(C(=O)CC3CCCC34CC4)CC2)CC1 CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC(C(=O)NC1CC(=O)NC(=O)C1)C2 C1(C(=O)N(CCCCNC(=O)CCC2CCCCO2)C)(COC)CC(=O)C1 Cc1cncc(C(=O)NCC2C(C)CCN2C(c2cnn(C(C)C)c2)=O)n1 C#CC1(C(=O)NCCCNC(C)=O)CCN(C(=O)COC(=N)O)C1 C12(C(N3CCCC3CCSc3ccccc3)=O)CCC(CC1)CC2.C12CCCN1C2 N1(C(CSCCC(C)C)=O)CCCC1CNC(C1(CCN(C)C)CCC1)=O C1(NC(C2(CC(C)C)CC2)=O)(CO)CCCN(C(=O)Cc2ccno2)C1 N1(C(CCC(=C)Cl)=O)CCCC2(NC(c3ccc(C4CC4)c(F)c3)=O)CC2C1 c1(C(NOCc2cn(CC3CC(C(C)C)OCC3)nn2)=O)c(Cl)nnc(Cl)c1O C(=O)(C1=NNC(=O)CC1)NCC1C2N(C(C3C4CC(C)(C4)OC3)=O)C(CC2)C1 Cc1ccc(-c2noc(C3CN(C(=O)OC(C)(C)C)C(C(F)(F)F)C3)n2)cc1F C1(NC(C(CC#C)C)=O)CC2CC(C1)N(C(C1(c3cccc(OC)c3)CC1)=O)C2 C#CCCCCCCNC(=O)C(C)CNC(=O)CC1(O)CCOCC1 CC1CCN(C(c2ccno2)=O)C1CNC(c1cc(Br)n[nH]1)=O C1(C(=O)OC)CC(CNCc2cccn2CF)N(S(C)(=O)=O)C1 N1(C(CC#C)=O)CCCCC1CCNC(c1cncc(Br)c1)=O c1(NC(c2n[nH]c(=N)s2)C)ncc(S(=O)(=O)NCCc2cccnc2)cc1Cl N1(C(C(C)CN(C)C)=O)CC2(CNC(c3ccc(CC4CC4)o3)=O)CCC1C2 c1(C(=O)NC2CCN(C(c3ccn(C(C)C)n3)=O)C2)n[nH]c2c1CCOC2 C=CCC(CNC(c1cnc(=N)[nH]c1)=O)C(=O)NC(C)(C)CCF c1(C(C)C(=O)NC2CC2NC(=O)CC2=NNC(=O)C2)ccc2ccccc2c1 N1(C(Cc2n(C)ccn2)=O)CC(O)CC1C(=O)NC1CN(C(N)=O)C1 C1(NC(C2(CC=C)CCCCC2)=O)CC(NC(C2(OC)CCCC2)=O)C12CCC2 C1(CNC(C=CCC)=O)CC(NC(c2ccn(CC)n2)=O)C(O)C1 c1(OC)c(C(=O)NCC(C2CC2)NC(c2ccc([N+](=O)[O-])o2)=O)cc(Cl)cc1C N1(C(CC2(OC)CC2)=O)CCCC2(C1)CN(C(=O)C(C)N=[N+]=[N-])C2 C=CCC(C)(C(=O)NC1(CNC(c2cc(OC)nc(Cl)c2)=O)CCC1)N(C)C N1(C(c2occ(C)c2C)=O)CCC2CC1CN(C(=O)CC(C)c1ccncc1)C2 C12(C(=O)NC(CCNC(c3cc(C(C)C)nn3C)=O)(C)C)CSCC1C2(F)F c1(C(=O)NC(CN(C(C(C=C)(F)F)=O)C)C)cncc2ccccc12 c1(C(=O)Nc2ccc(NC(c3cccc(C)n3)=O)cc2C)c(C)cc(O)cc1C Cn1cc(C(=O)NC2CCN(C(C3(C#N)CC3)=O)CC2)c(C(C)(C)C)n1 CCC(CCOC)C(=O)NC(C)(C)C(C)NC(c1csc(C(F)F)n1)=O C1(C=O)CC1C1CN(N(CCC(=O)OC)C2CC2)C1.C1(C=O)CC2CC(=O)C1C2 Cc1cccc(C2(CC3(C4CC4)CCCC3)CCC2)c1 c1(C(N(C(CNC(c2cc(C(C)C)n(C)n2)=O)C)C)=O)nn(C)c2c1CSCC2 C1(NC(C=Cc2c(C)ncs2)=O)COCCN(C(=O)C=CSCc2ccco2)C1 N1(C(C)=O)CCN(C(=O)Cc2cc(=O)n(-c3ccc(C)cc3)[nH]2)C2CCC12 CCC(CC)C(C)C(=O)N1CC2CC2(CNC(C2CC(n3ccnn3)C2)=O)C1 C12(CNC(C(CC)F)=O)CCCC1N(C(c1ccc(Br)c(F)c1)=O)CC2 C(=O)(C(CC(F)F)NC(c1nccnc1N)=O)NC(C#C)CC(C)C C(=O)(C(CC(=O)OC)NC(C)=O)N(C1CC(NC(COCCCC)=O)C1)C c1(OC)ccc(C(N2CC(C(C)NC(C3CC(OC)C3)=O)C2)=O)cn1 CC(F)(F)C(F)C(=O)N1CCCC1(C)CNC(=O)CCc1cn[nH]c1 C1(C(N(C(C)C(=O)N(C)CCn2cncn2)CCC)=O)CCN(C)C1 C(=O)(CCC1=CCCCC1)NCC(CCNC(C1(C)CCC(C)CC1)=O)O C1(CN(C(c2cnc(CC(C)C)[nH]2)=O)C)CCCN(C(=O)CC2CCNC2=O)C1 CCS(=O)CC(=O)NC1CCN(C(c2cccc(C(C)(F)F)c2)=O)C1C(C)(C)C N1(C(C2(F)CN(Cc3ccncc3Cl)C2)=O)CCc2nc[nH]c2C1 c1(C(=O)NCC(CC=C)NC(c2cc3ccccn3n2)=O)ccc2c[nH]nc2c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC2CCCN(C(=O)CN(C)C(C)=O)C2C1 c1(C(N2C(CCC)CN(C(C3(CO)CCCC3)=O)CC2)=O)ccc2occc2c1 c1(CC)nc(C(=O)N(C)CC2CCCCN2C(=O)CC(C)C2CC2)c(N)s1 c1(C(=O)NCC23N(C(C4(c5n(C)ccn5)CC4)=O)CC(C2)C3)cnc2n1CCC2 C1(CNC(C(CC)OCC)=O)(NC(=O)CCCSC(C)(C)C)CCCCC1C N1(C(c2c(C)ncn2C)=O)CCC(NC(=O)C=C2CCN(C)C2)C(CO)CC1 C1(C(N(C2CCN(C(CCc3c(C)nn(C)c3)=O)C2)C)=O)OCCN(C)C1=O c1(C(=O)NC(C2CCCN2C(C2CCC(=O)N2)=O)(C)C)cccn2ccnc12 C1(C(N(C2CCN(C(=O)C(C3(O)CCCC3)F)C2)CC)=O)CCCCN1C C(C(C)(C)C1=CCCC1)NC(C(Cc1ccoc1)NC(C(SC)SC)=O)=O C(C)(CO)(C(=O)N(CC(O)CN(C)C(C1CCC(F)(F)C1)=O)C)OC c1(C(C(=O)NCc2ccc(F)cc2)N(CC(CC)O)C)nc(Br)ccc1OC CC1OCCC1(C)C(N1CC(OCCNC(=O)Cc2ccnc(O)c2)C1)=O c1(N2C(CCCNC(c3cccc(F)c3F)=O)CCC2)ncnc2c1SCCC2 N#Cc1cn(CCC(=O)NCCCC2NC(=O)NC2=O)c(=O)nc1O N1(CCNC(CC(CC)C2CCC2)=O)CCCN(C(c2snc(O)c2Cl)=O)CC1 C(=O)(CCC(C)S(C)(=O)=O)NCC(C)(C)NC(CC(COC)C)=O Cc1cccc(C)c1N1CCN(C(=O)CC(O)C(C)C)CC1 N#Cc1cc([N+](=O)[O-])ccc1N1CCC(CN(C(=O)COC2CCOC2)CCO)C1 C12(NC(=O)CCSC(F)(F)F)CCCN(C(=O)Cc3cnoc3)CC1C2 CC1SCCC1(c1nnnn1CC1CC1)NCCCc1cccs1 CC1CC(O)CCN(C(C2CCCN(C(C3C4CN(C)CC34)=O)C2)=O)C1 C1(C(=O)NCCN(C(CCSCC(C)C)=O)CC(C)O)CCCC(O)C1 N1(C(C(CC)N(C)CC)=O)CCC(C2CCCCN2C(=O)CC2OCCO2)CC1 CC(=O)CCCC(=O)N(C1CCCN(C(c2cnc(C)nc2C(C)C)=O)CC1)C C1(C)(C(=O)NC2CCC(NC(c3c(C)c(=O)cc[nH]3)=O)CC2)CCC(F)(F)CC1 Cc1cc(C(N2CC(O)CC2(C)C(C)(C)C)=O)ccc1S(=O)(=O)C(C)C C1(NC(CCCCC)=O)CCCCCN(C(=O)CCc2ccncn2)C1 C1(NC(CCN(C)CC)=O)CCN(C(c2ccccc2C)=O)C12CCC2 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCc2ccc(C)cc2)=O)CC1C c1(OC)ccccc1C(C1CC1)NC(C1CC2(CCC2)C1)=O c1(NCC2(NC(C(CC(CC)C)C)=O)CCCCC2)nc2c(cc1C#N)CCC2 c1(C(=O)NCC(CNC(Cc2ccc(C)o2)=O)F)ccc2ncccn12 N1(C(C(C=C)C)=O)Cc2occ(C(=O)N(C(C)COC)C)c2C1 CCC(CC(=O)NCCCCCCNC(=O)CCCC(OC)OC)C(F)F N1(C(c2n(CC)ncc2)=O)CCC2(C=C(C(=O)NCc3cccc(OC)n3)C2)C1 CCC(CCOC)C(=O)NCC1CCN(C(=O)COc2cc(C)cc(C)c2)C1 CC1(C)CCC(NC(C2COCCC2NC(=O)Cc2cncs2)=O)C1 c1(NC(C2CCN(C(c3ccccc3F)=O)C2)=O)ccc2cc[nH]c2c1 C1(C(N2CCC(C)(NC(C(C)c3ccco3)=O)C2)=O)CCc2ncnn2C1 C1(CCC)CN(C(=O)C(C)CSC)CCN1C(c1[nH]nc(OC)c1Cl)=O c12cc(C#N)ccc1NC2.Cc1ccc(N2CCCCC2c2nncn2C)cc1 N1(C(c2ccc(=N)[nH]c2Cl)=O)CCC2(CC1)CN(C(C1CCCCC1F)=O)C2 c1(OC)nccc(C(=O)N(CC(C)CNC(=O)CNC(N)=O)C)c1Br c1(C(=O)NC(C)CCN(C)C(C2(C#N)CC23CCC3)=O)c(F)cccc1Cl C(=O)(C(C)(C)S(C)(=O)=O)NCC(CCOC)NC(C12CCC(CC1)O2)=O Cc1ccc(-c2cc(C(=O)NC3CC3CNC(=O)C3CC3)n[nH]2)c(C)c1 c1(C(C)C)cc(C(N2CCC(F)(CNC(=O)C(C)(C)N3CCCC3)C2)=O)nn1C c1(CC(=O)NCC2CC(NC(=O)C3=C(Cl)CC3)C(O)C2)ccc(C(F)F)c(F)c1 c1(CC(C(=O)NCC2C(CNC(C3CN(C)C3)=O)C2)O)ccccc1Cl C1(NC(CNS(N(C)C)(=O)=O)=O)CC2CC1N(C(=O)CC1CN3CCC1CC3)C2 c1(OC)c(C(N2C3COCC2C3NC(=O)CC2CCCCC2)=O)nc(O)nc1O C1(C(=O)NCC=C2CCN(C(=O)CC=C(Cl)Cl)CC2)(OC)CCC(C)C1 c1(C(C)NC(C2CCCN(CC(C)C(C)(F)F)CC2)=O)ccc(F)cc1Cl C1(NC2(c3n(C(C)C)nnn3)CC3CCC(C3)C2)CCCC2(CC1)CC2 CC1(C(=O)NCc2ncoc2C2CN(C(C34CCC3C4)=O)C2)C=CCC1 C#CCCCC(C)C(=O)N1CCN(C(c2occc2COC)=O)C(C)C1 N1(C(C(C)OCCC(C)C)=O)CCCN(C(C2CC3CCC2O3)=O)CC1 N1(C(CCN(C2CCCCC2)C)=O)CC2CCN(C(c3ccc(Cl)cn3)=O)C2C1 C(=O)(C(C#N)C(C)(C)C)N1C2CC(NC(c3cc(CC)no3)=O)C1CC2 c1(C(N2CCC(CN(C(C(c3ccccc3)C)=O)C)C2)=O)cccc(O)c1F C1(N(C)C)CCC(C(=O)NC2CCCC2(C)CNC(C2CCN2C2CC2)=O)CC1 c1(CC)ccc(C(=O)NC2CCC(CCNC(c3sccc3OC)=O)C2)c(F)c1 N1(C(C2N(C)C(=O)CC2)=O)Cc2ccccc2CC1CNC(=O)C=CI C1(CC(=O)NCCN(C(=O)OC)C)CCN(C(C2CC(=O)N(C)C2)=O)CC1 Cc1nn(C(C)(C)C)cc1C(N1CCC(NC(=O)C=Cc2cc[nH]n2)C1C)=O C(=O)(CCC(=O)NCC1CC(C)N(C(c2cc(COC)oc2C)=O)C1)NCC C(=O)(C1=C2CCCN=C2NN1)N(C)CC1CCN(C(C2CCCC(C)C2)=O)CC1 C(C)(C(C(=O)Nc1cnn(CCF)c1)C(C)C)NC(CCC)=O c1(C(C)C)ccccc1C(NC(=S)NC(c1ccccc1)C1CCOCC1)=O C1(N(C(=O)C(CC)N(C)C(c2cnc(Cl)s2)C)CC#C)CCN(C(C)=O)CC1 C12(NC(CCCC)=O)CCN(C(c3ncc(Br)cn3)=O)CC1C2 CCCCC(CC(=O)N1CCC(C)CC1)NC(c1[nH]nnc1CC)=O C(CC(=O)NC(C1CCN(C(=O)CCC2CCC(=O)N2)CC1)C)(C(F)(F)F)OC c1(-c2nc(C(C)O)nn2C2CCCOC2)ccc2ncn(C)c(=O)c2c1 C1(O)(CN(C(CN(C(COCCCC)=O)CCOC)=O)C)CCCCC1 C1(CCC#C)CCCCN1C(=O)CN(C(=O)CN1CCCC(O)C1)C c1(CC)nc(C)c(C(N2CCCC2(C)C(=O)N(CC)CC2(O)CCC2)=O)o1 O=C(C1=CS(=O)CCC1)N1CCC2CN(C(=O)CCC3CCCCC3)C2C1 C(CC(=O)N=c1ccn(C)[nH]1)C12CN1C2.C12(OC)CCCC1C2(F)F C(C(CC(=O)NCC1CC(NC(c2ccc3nn[nH]c3n2)=O)C1)C(F)F)N(C)C C1(C(N2C(C(=O)NC3(COC)CCOCC3)CCC2)=O)CC2C(C1)C2(F)F C1(CC)CCCCC1C(=O)NCCOCCOCCNC(c1n[nH]c(C)n1)=O C1(C#N)(C(=O)NC(CNC(c2cccc(OC)n2)=O)CCOC)CC2(CCC2)C1 CC1C(NC(C2(C)CCCCC2)=O)CCN1C(C1CCC1CF)=O C1(C(=O)NC(c2cccnc2)C(=O)NCCOCC(F)(F)F)CC2(CCC2O)C1 N#CC1CCN(C(=O)COC2CCN(C(=O)CC3CCC(=O)N3)C2)C1 N1(C(C2CCC(=O)NC2)=O)CC2CC(CNC(=O)Cc3ccc(O)cn3)C2C1 NC(=O)C(F)(F)CNC(=O)CNC(c1cn(CCO)nn1)=O C(=O)(C(F)CCC(C)(C)C)NC(c1nc(-c2noc3ccccc23)no1)C c1(C(=O)N)cc2c(C3CC3)cccc2[nH]1.C1(CC)CCN(C(c2coc(CO)c2)=O)C1 C1(CNC(C(CC)NC(N)=O)=O)CC2CCC(C1)N2C(=O)CC(C)(C)OC C1(C(N2C(CCC#C)CCC2)=O)C(C)CCN1C(=O)Cn1nnnc1CC N1(C(CC2C(CC)C2)=O)CCCN(C(C2(CF)CC2)=O)CC1 c1(C(C)(C)C)cnc(CCC(=O)NCC2(NC(C3CSCCS3)=O)CCOC2)o1 c1(OC)ccc(C(=O)NC(C)(C)CNC(C2CCC(NC(N)=O)C2)=O)nc1N c1(C(=O)NC2CC(CNC(C3C(CC)C3)=O)C2)cn(C)c(C)cc1=O N1(C(c2c(CC)cccc2)=O)CCC(C(=O)N(C2CCC(CC)CC2)C)C(C)C1 C1(CC)(NC(c2c(C(=O)OC)cnn2C)=O)CCN(C(c2cn(C)cn2)=O)CC1 C#CCCCC(C)C(=O)NCCCCCCN(C(=O)C=CC(C)(C)C)C C1(CC)CC2(CCN2C(=O)C(C)(CSC)NC(=O)C(F)C(C)(F)F)C1 Cc1cnc(Cl)c(S(=O)(=O)NC2CN(C(c3cc(Br)c(C)s3)=O)CC2F)c1 c1(CCC(=O)NC(CC)CNC(=O)C(CO)N(C)C)n[nH]c2c1CCCC2 CCCCCS(=O)(=O)CC(=O)N1CCCN(C(c2ccc(Cl)c(C)c2)=O)CCC1 CCC(C)(C)CCCC(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C Cn1ncc(C(N2CCOCC2CC(=O)NCC2=CCCCC2)=O)c1Cl c1(CNC(C2N(C(CCCC)=O)CSC2)=O)c(C)cnn1COC c1(C(=O)NC2CC(C(=O)Nc3ncc(F)cc3Cl)C2)c(Cl)cnc(Cl)c1Cl C(=O)(CCC(C)(C)C(=O)NC1CC1CNC(c1ccc2c(C)noc2n1)=O)OC CC1(C)CN(S(=O)(=O)COc2ccc(Br)cc2)CCC1CNc1ccccc1 CCC(C(=O)N1CCN(C(=O)CSCC(N)=O)CC12CC2)C(C)(F)F C(=O)(CC(C)(C)C(F)F)NCC(C1CCN(C(=O)Cc2ccsc2Cl)CC1)(C)O CC(C)C(C)(CNC(=O)OC(C)(C)C)NC(c1ncc(Br)cn1)C S(=O)(=O)(c1cccnc1NC1CCCCC1C(F)(F)F)NCC(CN(C)C)(C)C C1(c2n(CC)ccn2)CCCCN1C(c1conc1CC)C(=O)NC1(C)CC1 C(=O)(C(C(C)(C)O)NC(c1cnn2c1CCC2)=O)NC(c1nccs1)C N1(C(c2cccnc2C2CC2)=O)CCN(C(c2cc(F)n[nH]2)=O)C(C2CC2)C1 C(CC(C(=O)N(C1C2CN(C(C34COCC3C4)=O)CC12)C)NC=O)SC S(=O)(=O)(c1ccc(=NCC(O)c2ccnn2C)[nH]c1)N(CCN(C)C)CCO c1(C(=O)NCCNC(C2CC=CCC2)=O)ccnc2cc(F)cnc12 c1(OC)c(CC(=O)NCC(O)CCOC)cccc1F c1(C(C)C(=O)NC(C(=O)NCc2ccon2)C2CCC2)ccnn1C Cc1cn(C)nc1CN1CC(C)(O)C1.N12CCC(CC1)C(=O)N1CC2C1 Cc1cc(NC(=O)CCc2cnn(C)c2)ccc1NC(=O)CC1CCC1C C1(C(C)C)CC(C(=O)NOCC(O)C(F)(F)F)CCO1.C1C(=O)N1C(C)C C1(NC(=O)NCc2nccc(C(C)C)c2)CCc2nnc(C(F)F)n2C1 CC(CC(=O)NC1CCCC1CNC(c1cccnc1OCC(F)F)=O)C(F)F C(=O)(CCCCCCN=[N+]=[N-])NC1(C2N(C(C(CCC)OC)=O)CCCC2)CC1 N1(C(CNC(C(C)N(C(C)=O)C(C)C)=O)=O)CCN(C(=O)CSC(F)F)CC1 C1(C)(CNC(c2c(CC)oc(C)c2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CCO1 c1(C(C(=O)NC(CNC(C2CC=CCO2)=O)CO)(F)F)cccc(Cl)c1 N1(C(C2(CCNC(c3cccc(C)c3F)=O)CC2)=O)CCCCC(F)(F)C1 N1(C(CC(C)c2cccnc2)=O)CCCC(CNC(C2(CO)CCCO2)=O)CC1 c1(C(C(C)O)NC(=O)CCC2CCOC2)cccc(OCCN(C)C)c1 C1(CNC(C(CC)SC)=O)(NC(=O)C=Cc2cnn(C)c2)CCCCC1 C(=O)(N=c1cc(C2CC2)n(C)[nH]1)C1N(C(C(C)OCCC(C)C)=O)CC1 c1(C(=O)OC)c(Cl)nc[nH]c1=NCCC1CCCCN1C(=O)CC1CCOCC1 c12cnccc1NC1CCN(C1)C(=O)c1cc(n[nH]1)C(=O)N2.C(C)(C)(C)OC Cc1cccc(N)c1C(N1C2CCC1C(CNC(=O)CCF)C2)=O C1(NC(c2c(C)cns2)=O)CCOC(C(=O)NCCS(N)(=O)=O)C1 c1(CC)cc(NC(C2(CNC(=O)CN3CSCC3=O)CC23CCC3)=O)ccc1F C1(OC)CC(CNC(c2c[nH]nc2C(C)C)=O)N(C(=O)C(F)CC2CCCC2)C1 c1(C2CCN(c3ccnc(NCC4(C(C(C)C)O)CC4)n3)C2)cc(F)cc(Cl)c1 C(=O)(CS(=O)(=O)c1cccc2nsnc12)N1CC=CC(NC(C2CC2(F)F)=O)C1 C1(C)(C(=O)NC2C(NC(c3cc(COC)on3)=O)CCC2)CCNC(=O)C1 CCCC(CC)N=c1cc(C)[nH]c(=NCc2cc(C)cs2)[nH]1 C1(O)(CN(C(c2c(NC)cccc2)=O)C)CCCN(C(C2C=C(C)CS2)=O)C1 CCCCC(C)NC(C1CCN1C(c1cncnc1)=O)=O c1(C(=O)NC23CC(CNC(C(C(C)C)(C)O)=O)(OC2)C3)sccc1S(N)(=O)=O C1(C(N2CC(C(=O)NCC)C2)=O)CC2CCCC2N1C(=O)CON(CCO)CC Cc1ccc(C(C)C(=O)NC2CC(CNC(c3c(Br)noc3C)=O)C2)cc1 c1(CN(C(=O)CC2CCC3CC23)C(N)=O)nnnn1C1CC1.C12CCCN1C2=O c1(C(=O)NCC(CC(C)C)NC(C(CC=CC)C)=O)cc(C(C)C)n(C)c1C c1(CNC2C(C)CN(C(=O)C(c3cnn(C)c3)=O)C2)ccc(F)c(O)c1F CCC(C)CC(C)C(=O)N1CC(CC)(NC(=O)CN(c2ccc(Cl)cn2)C)C1 c1(CNc2cc(C)nnc2)cnn2cccc2c1 C1(OC)CCN(CC(=O)N(C)CCNC(c2csc(Br)n2)=O)C1 CC1CN(C(=O)C(F)(F)C(O)C2CC2)CCC1CNC(=O)CSC(C)(C)C C#CCCCC(C)C(=O)NC(CC(C)(C)C)C(=O)Nc1ccc[n+]([O-])c1 c1(OC)ccc(CN2CCC2(C)C(N2CCOC(C)C2)=O)cc1-c1ccccc1 c1(C(=O)NCC2CCC2NC(C2CCC(=O)N2C2CC2)=O)cccc2occc12 CC1CN(C(c2cnsc2)=O)CC(C)CN1C(=O)C(N1CCCCC1=O)C N1(C(C2COCCN(C(C(C(C)C)C)=O)C2)=O)CC2CCCCC12C N1(C(c2csc3ccccc23)=O)CC(CO)C2(C1)CN(C(C13COCC1C3)=O)C2 C1(CNC(CSCC(=O)OC)=O)CCN(C(=O)Cc2cc[nH]n2)C1 C1(O)(CNC(C(CCNC(C(C)(C)CO)=O)O)=O)CC2CCC1O2 C=Cn1nccc1C(=O)NC1CCCN(C(=O)C(c2cnn(C)c2)=O)C1 S(=O)(=O)(c1cccc(S(=O)(=O)N(n2cccn2)C)c1)N(C(CN(C(C)C)C)C)C C1(NC(C(F)=CC)=O)CCCC(NC(=O)C(c2cccc(OC)c2)(F)F)CC1 C12(C(=O)NCC(C)OCC)CC(CN)(C1)OC2(C)C.c12cccc(c1)N2 C(=O)(CCN=C(NCc1cc2cc(Cl)ccc2[nH]1)NCC1(SC)CCC1)NC C(=O)(C1=NOC2COCC12)N1C(C)CC(NC(=O)CC2CCN(C)CC2)CC1 Cc1cc2ncnc(N(C)CC3CCCN3C(=O)COCC(C)(C)C)c2[nH]1 N(C1c2ccccc2CC1NC(c1ccc(CO)o1)=O)C(C1C(C)CCO1)=O N1(C(C(C)OC)=O)CCC2(CCN(C(c3cc(N)ccc3C(F)(F)F)=O)C2)C1 C1(CC(=O)NCC(C)(C2CC2)NC(CCSC)=O)C(=O)ON=C1C CCCCCCCCCCC(C)NC(=O)C(=O)Nc1cc(Cl)cc(Br)c1F C1(NC(c2c(C)ccs2)=O)CC12CCN(C(c1c(F)ccc(O)c1F)=O)CC2 n1(CC(=O)OC)c(C)cc(C(=O)NC(CNC(=O)CC23CCC(CC2)C3)CO)c1C C(c1ccncc1)=C(C)C(N1CCOC(CN(C)C(C2CC2C(F)(F)F)=O)C1)=O C1(NC(C(C)CC2CC2)=O)(CO)CCN(C(c2coc(CO)c2)=O)CC1 c1(C(CC)C(=O)N2CC(NC(c3ccc(CN(C)C)o3)=O)C2)ccc(F)cc1 C1(C(=O)NCCn2c(C)cc(C)n2)CC12CCN(C(=O)C(C)(C)C1CC1)C2 N1(C(c2cc(Cl)ccc2C(F)(F)F)=O)CCn2ncc(C3=CCCC3)c2C1 c1(C(N2CCCC(NC(c3cc(O)ccc3Br)=O)CC2)=O)ccc2sccc2c1 N1(C(c2cc(C(=O)OC)n(C)c2)=O)CCN(C)C(CNC(=O)C(F)OC)C1 N1(C(C(C)Cc2ccncc2)=O)CCN(C(=O)CSc2cn[nH]c2)CC(C)(F)C1 N1(C(=O)NC(c2cccc(Cl)c2)C(C)C)CC(O)C2(CCCC2)C1 c1(C(N2CCN(C(c3ccc(C)c(O)c3)=O)C(CF)C2)=O)[nH]nc2ncccc12 c1(C(=O)NCC2N(C(CC)=O)CC2)cc(C2(C)COC2)no1 c1(CCCC)cc(=NC(=O)CC(=O)N(C)Cc2ccc(OC)cc2C(=O)O)[nH]o1 CC1CN(C(C2C(C)(C)C2(C)C)=O)CC(C)C1NC(c1cc(Cl)c(Cl)s1)=O C1(C(CC)C)CCCN1C(=O)C(C)N(C(=O)CCNC(=O)C1CC1)C N1(C(C2CC(O)(CC#C)C2)=O)CC(C)(C)OCC1CNC(C1(CC)CCCO1)=O c1(C(N2CCC(CCNC(C(C)CC(N)=O)=O)C2)=O)cnn2c1CCCC2 C1(CC=C)(NC(=O)CC(C)N(C)C)CCN(C(=O)Cc2cc(C)ccc2F)CC1 C1(C(=O)NCC(C(C)(C)C)NC(c2c(CC)nco2)=O)CC(C2CC2)=NO1 N1(C(c2c(C)n(CCO)nc2)=O)CC(C2(NC(=O)C=Cc3ccncc3)CC2)C1 c1(C(N2CCC(CNC(CCCCCSC)=O)C2)=O)cc2n(n1)CC(C)NC2=O N1(C(CCCC=C)=O)CC2CN(Cc3ccc(O)c(C)c3)C2C1 c1(C(=O)Nc2c(C)nc(F)cc2)n[nH]c2c1CN(Cc1sc(Br)nc1Br)C2 N1(C(Cc2c(C)nc[nH]2)=O)CC2CC(C1)CN(C(C1CCCNS1(=O)=O)=O)C2 CCCCCC(C)(CC)C(=O)NCCCCCCn1cc(CC2CCCC2)nn1 N1(C(CC(CC)CC)=O)CC2(CCC2)CC1CNC(c1c(C)ccc(C)c1C)=O C(C(C(F)(F)F)n1cccn1)NC(=O)NC(c1ccncc1)C C1(CC(=O)NC(C(=O)OCC)C)CC2(C1)CN(C(=O)CN(C)C(N)=O)C2 CCCCC(C)(CO)NC(=O)CC(C(F)F)NC(=O)CC(CC)CC C(=O)(N=c1cnn(C2CCC2)[nH]1)c1cccc(NC(=O)OCc2ccccc2)c1 C=C=CCCC(=O)NCCC(=C)CNC(c1occc1Br)=O c1(CN(C)C(c2ccc(O)cn2)=O)ccccc1CNC(c1cn(CCO)nn1)=O C1(NC(c2cnc(C(C)C)nc2)=O)CC(C)CN(C(c2cc(Cl)ccc2N)=O)C1 C=CCCCCC(=O)N1CCC1CNC(C1(CF)CC1(F)F)=O C=C(C)CC(C(=O)NC(C)CCC(=O)NCCc1ncoc1C)OC Cc1ccc2c(c1)CC(C(=O)OCC1CCCN1)S2(=O)=O CC1=C(C)CC(C(=O)NC2CN(C(C34CSC(C3)C4)=O)CC2C)CC1 CC1(NC2c3nnnn3CCOCCC23CCC3)CC(F)(F)C1.C1(CF)CC1 c1(COC(CSC)=O)nc(C)c(NC(c2ccccc2C)=O)s1 c1(C(N2CC(NC(C(C)OCCOCC)=O)C2)=O)cc2c(nc1O)CCOC2 N1(C(C2CN(C(N)=O)C2)=O)CC(C2CC2)(C(N2CC(O)(CO)C2)=O)C1 N1(C(C=C(C)C(F)F)=O)CCOC2CN(C(c3cc4[nH]ccc4s3)=O)CC12 c1(-c2cnc(CNC(c3cccc(CO)c3O)=O)nc2)cccc2c1OCC2 C(=O)(C(O)C(F)(F)F)NC(C(=O)NC1CCC(C(N)=O)C1)CC1CCC1 c1(C(N2CC(CC)C(NC(C3CCSC3)=O)CC2)=O)cncc2sccc12 N1(C(CCC(=O)NC)=O)CCCC(OCCNC(CCOCC)=O)C1C N1(C(C=CSC)=O)CCN(C(c2nnccc2C)=O)C(C)C1C C1(NC(c2c(C)nsc2C)=O)CC2CC(C1)N(C(C1CN(C3CCCCC3)C1)=O)C2 S(=O)(=O)(c1cc(C(=O)O)cs1)NCC(=O)Nc1c(C)noc1-c1ccccc1 c1(CC(=O)N(CCC(C)NC(CSCC)=O)C)nc(Br)n(C)c1C C1(CC(=O)NCC2(NC(CCc3cc(C)[nH]n3)=O)CCCC2)CCCCC1(C)C c1(OC)cccc(CC(N2CCCC2C(c2cn(CCC(C)C)nn2)(C)C)=O)n1 C1(C(N2CC(Nc3ncncc3F)CC(F)C2)=O)CN2CCC1CC2 C(N=c1[nH]c(N2CCCC3(C=CCO3)C2)nc2cccnc12)c1nnc(C)o1 Cc1c(C(N2CC(NC(c3ccsn3)=O)C(C)C2)=O)cnc2ccnn12 c1(C(=O)NC(c2ccccc2)C(C)NC(CCCOCC)=O)cc(C)n(C)n1 CC1(C)CC(NC(=O)CC(CNC(=O)CC2OCCO2)C2CCC2)C12CC2 Cc1cc(CC(=O)NCC2(CO)CCN(C(C3OCCC3(C)C)=O)C2)cc(F)c1 c1(C(N2CC(NC(C(C)(CO)OC)=O)C(F)C2)=O)cccn2nccc12 C(=O)(CCC(C)(C)C)NC(C)CCNC(=O)CNC(c1ccccc1)=O N1(C(C(CC)C2CCC2)=O)CCN(C(C2(C#N)CC2)=O)CC(C)C1 N1(c2nc(Cl)nc(C)c2F)CCC(C2CCCN(C(C3(Cl)CC3)=O)C2)C1 C(=O)(C1=C(C2CC2)N(C)C(=O)N(C)C1c1cncc(C(=O)OC(C)(C)C)c1)OC Cn1cnc2c1C(C(=O)NNC(=O)c1ccc(Br)cc1OC(F)(F)F)CCC2 C1(C)(CC)CC(NC(=O)CNC=O)CN1C(c1oc(C)nc1C)=O c1(C(=O)NC2C(NC(CC=C=C)=O)CC2)ccc(C#N)c(Cl)c1 c1(C(=O)NC(C(C)NC(=O)CC2CCCC2)C)ccc2c(c1)NC(=O)CCN2C C1(c2n(C(C(=O)OC)C)nnn2)(NC2CC(C)CC(C)C2)CCC=CCC1 c1(-c2ccc(SC)cn2)nc2ccc(C(=O)Nc3ccc(C#N)cc3Cl)cc2s1 CCCC(CCC)CC(=O)NC(C)C(=O)Nc1ccc(CCO)cc1 CCCCCCCC(=O)NC1CC(C(=O)N(CC(=O)OC)C)=CC1O c1(C(=O)NC2CCC(C(=O)NCC3CCN(CC)CC3)C2)cc(F)cc(Br)c1F C1(C(=O)NC(CC)COC)CC2CCCC2N1C(C1CC(=O)N(C)C1)=O C1(NC(c2cc(C)sc2C)=O)C2CCCN(Cc3snnc3C)C2C1(C)C c1(CNC(C2CCCN2Cc2cc(O)ncc2Br)=O)cc(Cl)cc2nc[nH]c12 C12(CNC(C3C(C=C)C3)=O)CCC(NC(=O)CC3(NC(C)=O)CC3)(CC1)CO2 c1(CCOC(C)C(=O)NC2CN(C(=O)C(c3ccccc3)F)C2)ccccc1 c1(CN(CC(=C)F)C(C2(n3nccn3)CC2)=O)cn(CC(=N)O)cn1.c12cn-1nn2 c1(OC)ccc(C(N2CC(CNC(=O)CCc3cnc(C)s3)C2)=O)cc1C1CC1 N1(CC(=O)NC2CCCN(C(=O)Cc3cc[nH]c3)C2)CCCCC(O)C1=O c1(C(N(CCOC)CCNC(=O)Cn2cccn2)=O)c(F)cc(C)cc1F C12(C(=O)NC(C=C)(C)C3CC3)COC(C1)C(NC(c1cnc(C3CC3)o1)=O)C2 c1(OC)oc(C)nc1C(=O)NC(C1CN(C(=O)C2=C(C)CC2)CCO1)C CC1(C)CCN(C(=O)C(C2CC2)C2CC2)C1CC(=O)NCC(F)CO C1(CNC(C(F)=CC)=O)CC2(C1)CN(C(c1cnc(OCC)s1)=O)C2 C(=O)(C(CO)C(F)(F)F)N1CC2C(CC(=O)N(C(C(=O)NC)C)C)C2C1 C(=O)(C(O)COC)NCC1(CC(=O)NCC(C)OC)CC1 c1(C(=O)NC2(CNC(c3cccc(Cl)c3F)=O)CCOC2)ccc2c(c1)NCC2 C(=O)(CC(C(=O)NCC(O)CNC(=O)CCN1C(=O)CCC1=O)NC(C)=O)OC c1(C(N(C(C)CCNC(c2cc(Cl)cnn2)=O)C)=O)ccnn(C)c1=O c1(C(=O)NC2C(CNC(Cc3cn(C)nc3)=O)CCC2)cc2n(n1)CCCC2=O C1(C(=O)NCC(C)Cn2ccnc2)CN(C(C2(C(N)=O)CCC2)=O)CCO1 C1(C(=O)OCC)CCCN(S(=O)(=O)N2CC(CNC(=O)NCC3CC3)C2)C1.OCC CCS(=O)CC(=O)N1CCC(C)(CCNC(c2ccnn2C2CCCC2)=O)C1 c1(C(=O)NCC(C)CN(C(=O)CSc2cnn(C)c2)C)ccoc1Br N1(C(c2cn(CC)nc2)=O)CCC2CCN(C(=O)CC3=CCCC3)C2C1 C1(NC(C2C(C)CCO2)=O)CCCC(CNC(c2cccn2C2CCCC2)=O)C1 c1(-c2nc(O)cc(C)n2)nc(C2COc3ccccc32)nn1CC1CCCO1 Cc1nc(O)ccc1C(=O)NC1COCCN(C(C2CC2C)=O)C1 n1(CC(C)C)[nH]c(CC(=O)NCCCC(C)NC(C2CCCOC2)=O)cc1=O C1(C(N2CCC(CNC(C3(O)CCOC3)=O)C2)=O)CN2CCN1CC2 C#CCCCCC(=O)NCCN(C(=O)Cc1ccc(F)cc1C)CCOCCO S(=O)(=O)(CC(=O)NCC(C1CC1)NC(=O)C(=O)C(C)C)NCC N1(C(C2C(CC)CCC2)=O)CC2CC(C1)CN(C(c1cnc(S)nc1)=O)C2 C(=O)(C1CCCc2ccnn21)N(C1CCCN(C(c2c[nH]c(=N)s2)=O)C1)CCF CCC(C)(CNC(c1n[nH]cc1Cl)=O)NC(C1CC(=O)C1C(C)(C)C)=O c1(N(C)C)cnc(C(N2CCCC(CNC(c3cocc3C(N)=O)=O)C2)=O)cn1 c1(OC)cc(Cl)c(Br)cc1NC(CCC(C)C)C(=O)OCCCF C1(C(C)(CNC(C2CCSC2)=O)NC(=O)OC(C)(C)C)CCOCC=C1 N1(C(CC(C)(C)C)=O)CC2(CCCC2NC(c2noc3ccccc23)=O)C1 Cc1c(C(N2CC(CNC(C3(C)CC(C)OC(C)C3)=O)C2)=O)cccc1[N+](=O)[O-] N1(C(c2c(C)nn(C)c2)=O)CC2(C)CC1C2NC(c1c[nH]ccc1=O)=O N1(C(C2CCN(CC)C2)=O)CCC(NC(c2snnc2C2CC2)=O)C12CC2 C(=O)(C(C)S(N)(=O)=O)N1CC(C(=O)NC(c2ccncc2)C)C(C)C1 c1(C(=O)NC)ncc[nH]c1=NCc1ccc(-c2cccc(C(=O)N(C)C)c2)cn1 c1(C(C)C)ccc(C(=O)NC(C)CC(C)NC(c2ccc(C3CC3)cc2)=O)cc1 N#CC1(C(=O)CCCc2nc(-c3sccc3CO)no2)CCC1 n1(CCC(=O)NCCC2(OC)CN(C(=O)CCC3CC3(F)F)C2)cnccc1=O C1(CN(C(c2sc(C(C)(C)C)nc2C)=O)CC)CCCCN1C(=O)C1=COCC1 c1(C(=O)NCCCCN(C(=O)CCc2cnc(O)[nH]2)C)cccc2nsnc12 c1(C(N2CCC(CNC(C3(C)CC(=C)C3)=O)C2)=O)cc2c([nH]1)CCC2 c1(CNc2c(CC(N3CCC(F)CC3)=O)cccc2)cccc2nccnc12 C1(C)(C(N2CC3C(NC(c4ccc(CC)s4)=O)(C3)C2)=O)CC(C(F)(F)F)=NO1 C(=O)(C(C(C)(C)C)OC)N1C(C(N2C(C=C)CC2)=O)CSCC1 c1(C(N2CC(NC(C3CC(=C)C3)=O)C(OC)C2)=O)ccc(C(F)(F)F)cc1SC CCC(CNC(=O)C(CN(C)C)N(C)C)(CC)NC(C1OC2CCC1C2)=O C1(CNC(CC2(CSC)CC2)=O)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 C1(N(C(Cc2scc(C)n2)=O)C)CCCN(C(C2CNC(=O)N2C)=O)CC1 N1(CCS(CC(C)OC)(=O)=O)CCC(C(=O)NC(C)C)c2ccccc21 N(C(=NCC1CCC1c1cncnc1)N1CCc2c(F)ccc(F)c2C1)CC(F)F C(=O)(CC(F)(F)CS(C)(=O)=O)N1C2(CCN(C(C(CC)C)=O)CC2)CC1 N1(C(C2N(C(C)=O)CC(O)C2)=O)C2CCC1CC(NC(c1ncccc1Cl)=O)C2 C1(CNC(C(C)SC(C)C)=O)CCC2(CN(C(C3CCC4(CCC4)CC3)=O)C2)O1 C1(C(=O)NCC2(CN(C(C(F)=C(C)C)=O)C)CC2)OCCC1(C)C Cc1sc(C(=O)NCCOCCNC(=O)Cn2[nH]cnc2=N)c(C)c1C Cc1cc(C(=O)NCC(C)(F)CNC(=O)CC2=CCOCC2)c(C)c(C)c1 N1(C(CC(CCCCC)O)=O)CCC(C2CCCN(C(c3cnn(C)c3)=O)C2)C1 C1(C#CC(=O)N2CCC(C(C)NC(c3nc(C)ccc3C)=O)CC2)(CC)COC1 c1(C(=O)NC(C2CN(C(C3(O)CC(C)(C)C3)=O)C2)C)cccc(-c2ccc[nH]2)c1 C(CC(C)C)(C(=O)N1CCCC(N(CCF)C(c2ccc(Cl)s2)=O)C1)OC C12(NC(c3nc(C(C)(C)C)oc3)=O)CC(C1)N(C(C1CCCOC1)=O)C2 c1(C(N(C2CN(C(C(C)=C(CC)C)=O)CC2F)C)=O)cc(F)c(F)cc1OC c1(C(=O)NC(C)(CO)C(=O)N2CCC(n3ccnc3)C2)cccc2cc[nH]c12 C1(CCC)CN(C(c2cn(C)nc2OC)=O)CCN1C(=O)CC1CCC(=O)N1C c1(OCC)cccc(CNC(c2c[nH]nc2CNC(=O)C(C)C#N)=O)n1 c1(CC(=O)NCCC2CC(NC(=O)C(O)CC3CC3)C2)cccc(OC(F)F)c1 c1(C(N2CC(CCNC(c3n[nH]c(C)c3Cl)=O)OCC2)=O)cc(Cl)c(F)cc1F c1(C(N2CCC(C(=O)NC(COC)C(C)C)C2)=O)c(OC)cccc1C N1(NC(=O)NC(C2CCN(C(C)C(=O)N3CCCC3)C2)(C)C)C(=O)CCC1=O S(=O)(=O)(c1cccc(F)c1C#N)NC1C(C)(C)CN(C(=O)C2CC2)C1 CCC(CC)CCCNC(c1c(O)cccc1F)c1nnnn1CC N1(C(C2(C)CC=C(C)CC2)=O)C2CCC1CN(C(c1nnn(C(C)(C)C)n1)=O)C2 c1(C(=O)NCCC2OCCCN(C(C(C=C)O)=O)C2)cc2ccccc2c(=O)o1 CCS(=O)c1ccccc1NC(=O)NCCC(C)(O)C1CCCCC1 C1(NC(c2ccc(CCC)s2)=O)CC2CCC1C(NC(=O)C#CC(C)(C)C)C2 C1(CCC)CCN(C(=O)C(F)C2CC(NC(C3CC3Cl)=O)C2)CC1 N1(C(CC2C(CC)C2)=O)CC(NC(C2(C)CCCN(C)C2)=O)C(N=[N+]=[N-])C1 c1(NCC2C(C)C2C)[nH]c(=NCc2ccccc2C(C)(F)F)nc2ncn(C)c12 C1(C(N(CCNC(C2CN(CCC)C(=O)C2)=O)C)=O)COc2ccccc2C1 C1(NC(c2cccc(CC)c2)=O)C(CO)C2CCCCC12 c1(C(=O)NC23CC(NC(c4n(C)ncc4)=O)(C2)C3)nccc(F)c1Cl N1(CCC)CCN(C(=O)C(C(C)O)NC(C2CC(C)(F)C2)=O)CC1 c1(C(N2C(C(=O)NCC(CC)C(C)C)CC(OC)C2)=O)cc(C)nc(C)n1 N1(CC(=O)CC2CCOC2)CCN(C(C2CCCC2(F)F)=O)CC1 CC1=C(c2ccco2)CN(N(C)CC(O)C2CC2)CC1 c1(N2CC(OCCNC(c3c(C(C)C)noc3)=O)C2)ncccc1C#N C1(CNC(=NCC=C)NCC(C2CCOCC2)(F)F)CCc2ccccc2O1 N1(C(CCCCCC)=O)C2CCCC1CC(CNC(=O)Cc1cncc(F)c1)C2 C1(C)(CNC2(c3n(CC=C)nnn3)CCSC2)CCCCC1 Cc1cc(C(=O)N(C2(CC(=O)NOCC3CCOC3)CC2)C)ns1 c1(C(=O)NCCCCNC(c2ccccc2OC2CCC2)=O)ccc(Cl)cn1 c1(C(N2CCC(O)(C(C)NC(CNC(C)=O)=O)C2)=O)c(C)ncc2ccccc12 c1(N2CCC(c3nc[nH]n3)CC2)nc(N2CCN3CCCC3C2)nc2ccsc12 CC1=NN(C)C(=O)C1CC(=O)NC1CC(NC(c2cn(C)cc2C(F)(F)F)=O)C1 c1(C(=O)NCC2(C)CCC(NC(c3cc(CC)[nH]n3)=O)C2)cnn2cnnc2c1 C(c1ccncc1)=CC(=O)NCC(CC)N(C(=O)C(CC1CCCC1)OC)C N1(C(CCC2N(C(C(c3ccn(C)c3)C)=O)CCCC2)=O)CCOCC(O)C1 C1(C(=O)NC2(CNC(COC3(C)CCC3)=O)CCCC2)CC12CCOCC2 Cc1cc(Cl)c(Cl)cc1C(N1CCOC(C(C)NC(=O)C=CCN(C)C)C1)=O N1(C(C(=O)NC(C2COC2)C)C)CCN(C(=O)C2CC2)CC1 C1(C(=O)NC(C2CN(C(=O)C(c3ccccc3)F)C2)C)CCCOCC1 c1(C(C)C(=O)NC2C(NC(=O)C3=C(C)OCC3)CCOC2)c[nH]c2ccccc12 C=CCC(CC(C)C)C(=O)NC1(C(=O)NC2CC2O)CCC1 c1(CCNC(C2CCC(C)C2)=O)ccc(CNC(c2n[nH]c(C3CC3)n2)=O)cc1 C1(CN(C(CN(C)C)=O)C)COCCN1C(=O)CC1CCC(O)C1 c1(C(N2C(C)(CNC(Cc3ncc(C)o3)=O)CCC2)=O)ncnc2c1CCCC2 CN1CC2(CCN2C(C2(F)CCN(CC)C2)=O)C1.C(=O)C=CC(F)F C1(NC(c2c(C)n(C)nc2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 N1(C(C(c2ccncc2)C)=O)CCC(C)C(CNC(c2cccc(Cl)c2)=O)C1 c1(C(N)=O)cnc(Cl)[nH]c1=NC1CCC2CN(C(c3c[nH]c(=O)cn3)=O)CC2C1 C1(C(=O)NC(CNC(C(c2nc(C)sc2)=O)=O)C(C)C)CC2CCC1O2 Cn1nc(C(=O)NCC2CN(C(c3ccc(C(N)=O)cc3)=O)CC2O)ccc1=O CC(CCC(=O)N1CCC(O)(CCC(=O)O)C1)NC(c1cnns1)=O C1(C2CCN(C(C34CC=CC(C3)OC4)=O)CC2)(NC(C(C)C2CCCC2)=O)CC1 C#CCCCC(C)C(=O)N1CCC(C)(NC(=O)Cc2sc(C)nc2C)C1 N1(C(C(=O)NCC)=O)CCn2c(CNC(C3CC(=O)C3)=O)nnc2C1 N1(C(c2nn(C)cc2I)C(=O)NCCOC)CCCCCC1c1cccc(C)c1 N1(C(c2nc(C)n(C)n2)=O)CC2CC(NC(c3ccc(N=[N+]=[N-])cc3)=O)CC1C2 CN1CCN(C(N2CCOCC2CCCc2ccccc2)=O)CC1C1=CCN=C1 C(=O)(C1=CCCSC1)NCCC(C(=O)N1CC(COC)C1)O C1(NC(c2cncc(NC)c2)=O)CC2CC(NC(c3cc(C)n(C)c3)=O)CC2C1 c1(CC(=O)NC2N(C(CC3C(=O)NC(=N)S3)=O)CC2)coc2cc(F)ccc12 CCCCCCC(C)NC(C1(F)CCCN(C(c2cnc3n2CCC3)=O)C1)=O C1(CC=C)CCCCN1C(=O)C(Cc1ccccc1Br)NC(=O)Cc1ccsn1 C1(C2CCCCC2)(C(N(C)CC2CN(C(C3(CCN(C)C)CC3)=O)CCO2)=O)CC1 c1(NC(C2C(NC(c3ccc(C)cc3F)=O)CCC2)=O)ncc2ccccc2n1 C(=O)(C1CCc2nccn21)NCCN(C)C(C1CN2CCN1CC2)=O C=C(Cl)C(C)(C)C(=O)NC1CCN(C(=O)CCCN(C)C)C1 CN=c1[nH]c(=NCC2(C)CCCCO2)[nH]c(=NCc2ccnc(SCC)c2)[nH]1 CCC(CN=c1nc2c(ncn2CC)c(NCC(C)(CC)OC)[nH]1)OC c1(C(N(C2CCCN(C(=O)CCOC3CCC3)C2)C)=O)cc(C2CC2)ccn1 Cc1ncccc1C(=O)NC(c1ccccc1)C(=O)NCCn1cccnc1=O c1(CN2CCN(C(c3c(CC)c(Br)ccc3)=O)C(CC)C2)cc(F)cc(C)c1O CC1(C(N2CCCC2c2cn(Cc3cccc(Cl)n3)nn2)=O)Cc2ccccc2C1 Nc1ccc(C(=O)NCCN(C(c2ncc(Br)cn2)=O)CC2CC2)c(Cl)c1 O(NC(=O)C(C)(C)C(C)NC(c1cnn2c1CCC2)=O)C(CC)C C12(NC(c3ccc(CC)cc3O)=O)CCC(CNC(=O)C=CCOC)(CC1)OC2 N1(C(C)=O)CCC2(CC1)CN(C(=O)C(c1ccccc1)=O)C2 N1(C(=O)CC2CNC(=O)O2)CC2CC(C1)N2C(C1(F)CCCC1)=O c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCCOCC)=O)ccc(N)c(Cl)c1 CC1N(C(=O)CN(C)C(C2COC2)=O)CCCC1(C)C N1(C(c2ncc(OC(C)(C)C)nc2)=O)CC2CCC1CN2C(c1cnccn1)=O C1(SC)CCCC1C(N1CC(C(N)=O)(CNC(=O)CC2(NC(C)=O)CC2)C1)=O C1(C(C)OCC)CCN(CCC(=O)NC(=O)NCc2ccccc2Br)CC1C C=C1CCC(CNC(C2CCCN(C(=O)Cc3nc[nH]n3)C2)=O)CC1 C12(C(=O)NCC(CCOC)NC(c3nnc(C)s3)=O)CCC(CC1)CC2 C1(NC(C2(NC(C)=O)CCC2)=O)CC2(CCCCN2C(C2SCCC2C)=O)C1 N1(C(C2(CC(=O)OC)CC2)=O)CCC2CCCN(C(=O)CCc3nc(=N)[nH][nH]3)C2C1 C1(C(=O)N(C2CC2)C(C2CC2C(=O)N(CCO)CCO)=O)CCC(O)CC1 c1(C(C)C)cc(C(=O)NCC2CC(C(=O)NCc3cn(C)nn3)C2)on1 c1(CCC(=O)NC2C(NC(CCC#CC)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] N1(C(c2c(C#C)c[nH]n2)=O)CCC2(CC1)CN(C(=O)C(C)CCCCCC)C2 N1(C(CCCNC(C)=O)=O)CCC(C(=O)N2CC(C)C2(C)C)=C(F)C1 N1(C(C(=O)Nc2ccc(OC)cc2)=O)CCC(C)C(NC(C2CSCCS2)=O)C1 C(C(=O)NCC1(NC(=O)C2=CCCS2)CCCCC1)(C(C)C)SC C1(NC(c2cnc(C)[nH]2)=O)CN(C(C2Cc3nccn3C2)=O)C2CCCC12 c1(C(CC(=O)NC(C)CCNC(C2CC(=C3CC3)C2)=O)C)cccc(F)c1 N1(C(C2CCN(C(=O)C3(C4OCCO4)CC3)O2)=O)CC23CCC2(COC3)C1 C=CCC(C)C(=O)NCc1ccc(CN(C(=O)CC(C)COC)C)cc1 C(N=c1[nH]c(N2CCCC(CF)C2)nc2ccccc12)C1(CO)CCC(C)(C)C1 Cc1nc(C)c(CN2CCC(NC(c3cc(I)c(F)cc3Cl)=O)C(F)C2)nc1C N1(C(C(CCC)NC(c2ncn(C)n2)=O)=O)CCC(C)=C(F)C1 c1(C(=O)NCC(C2CCOC2)NC(c2cc(C(=O)OC)on2)=O)ncncc1Cl N1(C(C(CC#C)NC(C)=O)=O)CCC(NC(C2CC3CCC2CC3)=O)C(C)(C)C1 c1(C(=O)NC2CCCC(Nc3ncc(I)cn3)C2)cc2ccccc2oc1=O c1(C(=O)NC(CCOC)C(=O)N(C)CC2CCCO2)cnn2ccccc12 N1(C(C(C=C)CC)=O)CCC(CCOC)(NC(c2ccc(=N)[nH]n2)=O)CC1 c1(CC(=O)NC(CCNC(CC)=O)(C)C)ccc(F)cc1Br Cc1ccc(C(N2CC(O)(CN(C)C(c3c(C)coc3C3CC3)=O)C2)=O)c(C)c1 CC1CCCCN(C(=O)C(C(C)(C)O)NC(=O)COC(C)(C)C)C1 C1(C(=O)OCC)CN(C(=O)OCc2c(C)nn(COC)c2C)CCC1O C#CCCC(O)C(=O)NC(C)C(C)(C)NC(c1ccn(CC(C)C)n1)=O C(=O)(C(C)(C)CC(F)F)NC(CCN(C(=O)C=Cc1cnc[nH]1)C)C(C)(C)C CCCC(CCCNC(C1CC12CCC2)=O)NC(c1ccc(OC)cc1Cl)=O N1(C(CCOC)=O)CCC(C(C)(C)C)(CNC(=O)C(C(C)C)c2cccnc2)C1 C1(C(=O)NCc2n(CCC)ccn2)CN(C)CCN1C(=O)CC1(N(C)C)CCC1 c1(C(=O)NCc2c(C(N3CCC(C(N)=O)C3)=O)scc2)ccccc1Cl C1(c2cc(C)sc2)CCN(C(=NCC2CCC2)NCc2cccc(Br)c2O)C1 N1(C(CC(C)C2CCCC2)=O)CC2CCCCC2(NC(=O)Cn2ncnn2)C1 c1(-c2cn(CCC(=O)NC(C)CCN(C)C)nn2)ccc(C(F)(F)F)cn1 CC(C)(C)CC(C)(C)C(=O)NC1CCCN(C(=O)CCCc2cnccn2)CC1 CCCC(O)C(CO)NC(=O)CN(C(c1cc(C)nnc1C)=O)CC1CC1 N1(CC(C)(C)NC(=O)C=Cc2cccnc2)CCN(C(C2CCNC2=O)=O)CC1 C1(NC(C2(CC=C)CCOCC2)=O)CCN(C(C2(C#N)CC2)=O)CC1F S(=O)(=O)(c1cccc(NCC(C)Oc2ccc(F)c(Br)c2)c1)N(CCC(C)C)C c1(OC)cc(C(=O)N(CC(c2c[nH]c3ccccc23)=O)C)cc2c1OCO2 C1(NC(c2c(C)cc(F)nc2)=O)CCN(C(=O)CC2CCC3CC23)CC(O)C1 n1(CC)c(-c2nc(CCCO)nn2CCN2CCC(O)CC2)cnc1O CC1(C)CCCCCC1NC(C1CCC(C(=O)NCc2cc[n+]([O-])cc2)O1)=O Cc1cnccc1C(N1CC(c2ccccc2)(NC(C2COC(=O)C2)=O)C1)=O C=CCC(CC)C(=O)C(C)=O.C(=O)(C(C)C)N(CCCOCCN)C N1(C(CN2CC(C)C2)=O)CC2CC(C(=O)NC3CC3)CC(C2)C1.C1(=O)C=CCN1 C1(CC(=O)NCCN(C(=O)CCc2cnn(C)c2)CC)Cc2ccccc2C1=O CC1CCN(C(=O)CC2(CO)CC2)C1CNC(c1c[nH]ccc1=N)=O c1(C(CC)N(CCNC(=O)C(C)(C)C)Cc2occc2Br)ccccc1F c1(CC(=O)NC(CNC(C(C)OC)=O)C2CCC2)ccsc1Cl O(NC(=O)CN(C(=O)CC)CCN(C)C)CCC.C1(C)CCCO1 CN(CCCC(=O)N1CC(NC(c2cnn(CCC#N)c2)=O)C2(CC2)C1)N=O CC1CN(C(=O)CS(C)(=O)=O)CCC1N(C(=O)C(F)(F)C1CCOCC1)C c1(C(C(C)NC(c2c[nH]c(C(C)(C)C)c2)=O)C)ccc(C(F)(F)F)cc1 c1(NC(N(C(C(C)SC)C)C)=O)ccc(OCCCF)cc1 C1(NC(C2C(CC)OCC2)=O)CCS(=O)(=O)C12CN(C(=O)C=C(Cl)Cl)C2 C(=O)(CCCC(F)F)N(C(CNC(C1CCN(C)C1)=O)C1CC1)C CCCCCC(C)(C)C(=O)NC1CCCCN(C(=O)C(CCSC)OC)C1 CC1CN(C(C2CCC(F)CC2)=O)C(C)CN1C(=O)CCc1ccccc1C#N CCC(CC(=O)N1CCC(C)(C)C(C(=O)N(C)Cc2cnc[nH]2)C1)C(C)(C)C N1(C(=O)C2=CCOC2)CCN(C(c2ccc(-c3cccs3)o2)=O)C(C2CCC2)C1 C1(CC(=O)NCC(CNC(C2(C(C)C)CCCO2)=O)(C)C)CCCCCC1 N1(C(C2(O)C(C)(C)C2)=O)CCC2(CCOCC2)C(NC(=O)Cc2cn[nH]c2)C1 N1(C(CCCOC(C)C)=O)CCC(C(C)(C)NC(C2CC(N(C)C)C2)=O)CC1 n1(CC(=O)OC)c(C)cc(C(=O)C(Cl)(Cl)Cl)c1C.C1(C2C(=O)O2)CCCCO1 c1(-c2ccc(CN3C(CC(=O)NC4CCCCC4)CCC3)o2)ccc(F)cc1 Cc1cnc(O)c(NC(=O)C(C2CC=CCC2)NC(=O)C=CC2CC2)c1 C1(NC(c2cnn(C)c2Cl)=O)CN(C(C2CC(=O)N(CC3CC3)C2)=O)CC1(C)C C1(N(C)C(=O)OC(C)(C)C)CC2CC(NC(=O)C(c3ccc(O)cc3)=O)C1C2 C1(CNC(CCN(C(=O)C=Cc2cocn2)CC#C)=O)(CF)CC(=O)C1 C1(C)(CSC)CCN1C(=O)C(F)CC1CN(C(=O)COc2cc(C)on2)C1 C1(N(C(=O)Cn2nnc(C)n2)CC)CCCN(C(C2CC3CCC2O3)=O)C1 C1(CNC(CC(=O)OC)=O)CCN(C(c2nn(C(C)(C)C)cc2Cl)=O)C1(C)C c1(NC(C2CC2NCc2ccc(F)s2)=O)ccc2sc(Cl)nc2c1 C(=O)(C(C)(C)C(=O)OC)NC12CC(NC(COCCCC#C)=O)(C1)C2 C1(CC)CN(C(=O)C(CC2CCC2)NC(=O)C(=O)NC(C)C)CC1O N1(C(C2N(C(c3c(C)cccc3O)=O)CCC2)=O)CC(=O)NC2(CC2)C1 N1(C(c2cncc(O)c2Cl)=O)CCCC(C2CN(C(=O)C(O)C(F)F)C2)C1 CCCC(C)(C)C(=O)NC1CC(F)CN(C(C2(C)CCC(=O)NC2)=O)C1 CCC1=NOC(C(=O)NC2(C)CCN(C(c3nnn(CC)c3C(C)C)=O)C2)C1 CCCC(C#N)C(=O)N1CCC(C)C1c1cn(CCOCc2ccccc2)nn1 c1(COC)nc(Cl)cc(=NC2CC(NC(C3Cc4ccccc4CO3)=O)C2)[nH]1 C1(NC(c2onc(C)c2C)=O)CCCCC12CCN(C(C1(CF)COC1)=O)CC2 c1(C(=O)NCCCN(C(C(C=CCCC)O)=O)C)cc2c(Cl)nccc2s1 N1(C(C(CC)OC)=O)CCC(C2CC2)(NC(c2csc3ccccc23)=O)C1 N1(C(Cc2cc(C)sc2)=O)CC2CC(NC(=O)CC3CCOC3(C)C)CC1C2 n1(CC)cc(C(=O)NC(C)(C)C=CC(=O)NCC(F)(F)CC2CC2)nn1 Cc1cccc(F)c1C(=O)NC1C=CC(C(=O)NCc2nocc2C(C)C)C1 C#Cc1ccc(C)c(NC(=O)C(=O)NC(CSC)C(=O)N2CCCCC2)c1 c1(OCC(=O)NCC(C)NC(C(C(C)C)O)=O)c(Cl)cccc1F Cc1cccc(CC(=O)NCc2cc(C(N3CCCC3CN(C)C)=O)co2)c1 C1(CCC2N(C(c3nc(C)[nH]n3)=O)CCC2)CCN(C(=O)CC2CC2C)CC1 c1(C(=O)NCC2C(C(=O)NC(C=C)CO)C2)cccc(CN2CCSCC2)c1 C1(CNC(C2N(N=O)CCC2)=O)CC2CCC1N2c1cc(C(F)(F)F)nc(Cl)n1 C(C(C)(CNC(=O)CCN(C(c1ccc(C#N)s1)=O)CC1CC1)CO)OC N1(C(C(C(C)C)F)=O)CCC(O)(C(C)NC(=O)CCCCCn2cnnn2)CC1 CC1CCN(C(=O)N(C)Cc2ncnn2C)c2ccccc21 C1(C(=O)NC(C2CCN(C(C3(C)CCCC3)=O)C2)C)CCC1(C)C C1(NC(CCC(=O)NC)=O)CCCC12CN(C(C1CC3(C1)CC3F)=O)C2 N1(C(C2(CC)COC2)=O)CC(CO)(NC(=O)CSc2cccs2)C1 C12(NC(c3c(C)cc(SC)o3)=O)CCCC1N(C(c1ccc(Cl)cc1C)=O)CC2 C12(C(N(C)CC3CN(C(C4OCC4(C)C)=O)CCO3)=O)CCC(CC1)CC2 CC1(C)CCCC(CC(N2CCC(C(C)(C)NC(=O)Cn3cnnc3O)C2)=O)C1 c1(CC)cc2c(NC3(CNC(c4coc(CC)n4)=O)CCC3)ncnc2s1 n1(CCC)cc(C(=O)NCC2(CN(C(=O)CC(C)OC)C)CC2)c(C)n1 c1(CN2C(C(=O)NCC3(O)CCOCC3)CC(=C)C2)c(Cl)cccc1B(O)O Nc1cc(F)c(-c2cccc(C(=O)NC3(CO)COC3)c2)c(F)c1 N1(C(C(CC=CC)C)=O)CC(CC(=O)NCC(C)(O)CSC)CC1(C)C CCCCCC(O)CC(=O)N1CCC(C(C)NC(C2CC3(C2)OCCO3)=O)CC1 C1(CNC(C(CC)CCOC)=O)CN(C(=O)COC(C)=O)C2COCC2O1 CC(CC(=O)N1CC2CN(C(c3nc(Cl)ccc3N)=O)CCC12)C(F)(F)F CC1(O)CCN(CC(=O)NC2(CNC(=O)CN3C(=O)CNC3=O)CCCCC2)C1 C(CC(N=c1cc[nH]cc1C#N)C(C)C)N(C(c1ccc(C)nc1)=O)C C(CCC(C)C)(C(=O)NCc1ccnc(Cl)c1)NC(Cc1cc(C)n(C)n1)=O C1(C(=O)OC)CCCCC1(C)C.c1(CCC23CN(C2)C3=O)ccc([N+](=O)[O-])s1 c1(C(N2C(C)CN(C(=O)CC3CCCNC(=O)C3)CC2)=O)nc2cccnc2s1 O=C(N=c1nn[nH]n1-c1ccccc1Cl)NC1CC1C(=O)Nc1ncccn1 N1(C(C2CC2c2c(Cl)cccc2Cl)=O)CC2(CCOCC2)C1c1ccco1 c1(OCCOC)ccc(-c2cncc(C(=O)NCCc3ccccn3)n2)cc1 C1(C(=O)NCc2c(C(C)C)con2)CCN(C)CC1.C12(CCCO1)C(=O)NC2 Cc1nn(CC(=O)NC(C2CCCN2C(=O)CC2CCSC2)C)c(=O)o1 c1(CNC(=O)NC2C(CC(C)C)CCCC2)ccc(F)cc1O C1(C2CCOCC2)(NC(C2CC(CNC(=O)C=Cc3nccs3)OC2)=O)CC1 C1(NC(=O)CCCC(=O)N2CCC2)CN(C(=O)C=CC2CCC2)CC12CCOCC2 C1(C(=O)NCC2(F)CC(CNC(c3nnsc3C)=O)C2)(OC)CCCOC1 c1(CN(CC(O)CNC(C2CC2C(C)(C)O)=O)C)ccccc1 c1(C(C(F)(F)F)OC)ccccc1NC(c1nc(C)cn1C)c1ccccc1Cl c1(C(=O)NC2C(C)(CNC(c3coc(CO)c3)=O)CCC2)ccnc2[nH]cnc12 c1(C(N(CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC)CC)=O)ccc(Cl)c(C)c1 N1(C(CCOC2CN(C(CC(C)N(C)C)=O)C2)=O)CCC(C2=NOCC2)C1 C=CCCN=C(NCc1cc(C)ccc1Br)NC1CCC(=O)NC1 N1(C(c2cc(C)c(C)o2)=O)CC(C2CCN(C(C3CCOC3(C)C)=O)CC2)C1 C1(OCCNC(C(C)c2cncs2)=O)CCN(C(c2coc(Cl)n2)=O)C1 c1(C(=O)NC(C)C(=O)N(CCCNC(C2C(Cl)(Cl)C23CC3)=O)C)ccccc1Cl N1(C(CCOCC)=O)CC(NC(c2nscc2C)=O)C(n2ccnn2)C1 CCCC(C(=O)N1CCCCC1CNC(=O)C(C(C)CC)OC)S(N)(=O)=O CC1CN(C(=O)COc2cccc(F)c2)CC1NC(=O)C=Cc1cnc[nH]1 Cn1ccc(-c2noc(C3(C4CCNCC4)CCC3)n2)n1 N(C)(S(=O)(=O)N(C)C)CC(=O)NC1CCC(CCNC(COCCC#C)=O)C1 c1(C(=O)NC(C)CCNC(=O)C(c2ccccc2F)O)cccc(P(C)(C)=O)c1 CC(=Cn1ccnn1)C(=O)NCCCCN(C)C(C1CCC(F)(F)CC1)=O C1(C(N2CC(OCCNC(C(C)S(C)(=O)=O)=O)C2)=O)CCc2nn(C)cc2C1 N1(C(C2C(=C)C2)=O)CCC2CC12C(=O)NCCN(C)C(C)C CC(C)C(CCN(C(=O)CCc1cc[nH]n1)C)NC(C1(O)CCCC1)=O C1(CNC(CCSC)=O)CN(c2nccc(C(C)(C)C)n2)CCCO1 C(CCN(C(=O)C(c1ccc(F)cc1)CO)C)(C(C)C)NC(c1c(C)cc[nH]1)=O N1(C(C2C(CC)N(C(c3ccc(F)cc3)=O)CC2)=O)CC(OC)CC(C)C1 C1(C(N(CCCN(C(C2C(C(=O)OC)C=C2)=O)C)C)=O)CCCCN1C Cc1ccc(C(C)(C)C(=O)NCC2CN(C(=O)C3=CCC3)C3CC23)cc1 c1(C(N(C2CCC(NC(C3CC34CCOC4)=O)CC2)C)=O)c[nH]c2cnccc12 Cc1ccc(S(=O)(=O)NC(c2ccccc2)C(=O)O)cc1.N12CCC(C1)CC2=O c1(CCNC(C2CC2F)=O)ccc(CNC(C2CC(F)C2)=O)cc1 C(CCF)(C(=O)NCCCc1nccs1)NC(C1C(C)OCC1)=O c1(C(N(CC(CC)NC(c2cc(C(CC)CC)no2)=O)C)=O)nnc(O)cc1O C(=O)(C(=O)NCC(C)CNC(C1CCN1C(=O)OC(C)(C)C)=O)NC c1(C(N2CC(O)(CC=C)C2)=O)ccc(CNC(=O)CN2CCSCC2)cc1 C1(C(N2CCC(COC)(CNC(=O)C(O)C(C)C)CC2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NC(c2ncc(C)o2)C)CC(C)CN(C(C2C=CC=CC=C2)=O)C1 C=CCN(OC)C(=O)C12C(NC(=O)CCc3csnn3)C3CC1C2C3 C1(NCCCC(C)OC)CC12CCN(C(=O)OC(C)(C)C)CCCO2 c1(OC)ccnc(OC)c1C(=O)NC1CCN(C(C2COC(=O)O2)=O)C1 C1(CC(N2CCN(CCNC(CS(CC)(=O)=O)=O)CC2)=O)COC2(CCC2)CO1 N1(C(c2c(COC)cco2)=O)Cc2ccccc2C(NC(=O)C(F)C(C)(C)O)C1 c1(SCCC)cccc(C(=O)NC2CN(C(=O)C=NOC)CC2C(F)(F)F)c1 S(=O)(=O)(c1cscc1F)Nc1c(CC(=O)OC)cccc1 c1(OC)c(C(=O)NC2CCC2CNC(C2CCC(O)CC2)=O)cnn1C C1(CC(=O)NC(C=C)(C)CC)CC2(CC2)CN1C(=O)CSC(C)(C)C c1(OC)cc(NC2CN(C3CN(C(C4C=C4C)=O)C3)C(=O)C2)nc(OC)n1 C(c1cnc2ccccc2c1)=CC(=O)NCc1cnn(C)c1Br C1(NC(CSC(C)C)=O)CN(C(c2cnc(N)c(Cl)c2)=O)CC1S(C)(=O)=O C(=O)(CCC(F)F)NCC(CNC(=O)Cn1ccc(C(F)(F)F)n1)O [N-]=[N+]=NC1CC(C(=O)NC2CC3CCC2O3)N(C(c2ccc(C#N)cc2)=O)C1 Cc1ccc(-c2ccc(C(=O)NC3CC(F)(CNC(c4ccsn4)=O)C3)s2)s1 C1(OC)C(NC(=O)CC(C)(C)n2cc(CC(C)(C)O)nn2)CC12CCC2 c1(C(N2CCC(CNC(c3cn[nH]c3)=O)C(F)(F)C2)=O)ccc2nc(O)[nH]c2c1 C(=O)(C1=Cc2ccccc2C1O)NC1C(C)(C(C)C)C1 C1(C(N(C)Cc2n(CC)cnn2)=O)CCN(C(C2CC(=O)N(C)C2)=O)C1(C)C c1(OC)c(C(c2nnnn2CCC2(C)CC2)NC(C)(C)CF)ccc(Br)c1F C1(NC(CN(c2ncccn2)C)=O)CC2CC(C1)N(C(=O)Cc1ccc(Cl)s1)C2 C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)CSc2nnnn2C)CC1C C#CCC(O)C(=O)N(C)CC1CC(F)CN1C(=O)CSc1nnnn1C1CC1 N1(C(C(c2ccc(F)cc2)C)=O)CC2CC2(CNC(c2ccsc2C#N)=O)C1 C1(CC)CN(C(=O)C(c2ccccc2F)O)CCC1NC(C1(Br)CC1)=O C1(C(N2CCC(C(=O)OCC)C2C)=O)CC(n2cc(CC3CCC3)nn2)C(O)C1 Cc1ccc(C(=O)NC2CCCC2NC(C2(C(C)(F)F)CC2)=O)c(Cl)c1.C1(C)CC1 N1(C(C(CCOC)C)=O)CCN(C(c2ccc(C)cn2)=O)C(C)C1 Cc1cc(C(c2nnnn2C2COC2)Nc2cn(CCO)nc2C)sc1C C1(C(=O)NCC2(CN(C(=O)C=C3CCC(C)C3)C)CC2)(OC)CCC(C)(C)CC1 c1(OC)ccc(Cl)c(C(=O)NCCC2CCCCN2C(c2cccnc2C)=O)c1 N1(C(C(CC(C)C)O)=O)CCCCCC(NC(c2ccc3ncnn3c2)=O)C1 c1(NCCCCOC)cc(=NCC2CNC(=O)CO2)[nH]c(C(F)(F)F)n1 c1(C(N2CC(F)CC(NC(C(C=C=C)C)=O)C2)=O)ccc2cc(O)ccc2n1 CCCCCC(O)C(=O)NCC(C)(CC(C)C)NC(=O)CCNc1ccccn1 CCC(CCC(=O)N1CCC(SC)C1)NC(c1cc(Cl)cs1)=O N1(C(C(C)=C(C)C)=O)CCC(C(C)C(=O)NCC2CN3CCC2C3)CC1 C=C=CC(C)C(=O)NCC(C(C)C)NC(c1c(C(F)(F)F)coc1CC)=O c1(C(=O)NC2CN(C(C(C)(C)NC(C)=O)=O)CC(C)C2)c[nH]c2ccc(Br)cc12 C1(NC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)COC2(C)CCCC2)CC1F C1(CCC)CC(C(=O)N(C)CCNC(c2nc(C)n(C)n2)=O)CCO1 N1(C(C(CC2CCCC2)NC(C(CC=C)(F)F)=O)=O)CCC2(CC1)CN(C)C2 C1(CNC(CN(C(C)C)C)=O)CCC(CNC(C2CC3C=CC2C3)=O)CC1 C1(NC(C(C)OC2CCCC2)=O)CC2(C1)CC(NC(C1CNC(=O)N1)=O)C2 C(=O)(C(CC(C)C)C(C)C)N1CC(CC)C(CNC(c2cnnc(C)c2)=O)CC1 c1(C(=O)NCCC(CNC(CCOCC#C)=O)=C)nc(C)c(C)[nH]c1=O N1(C(C(C)=C(CC)C)=O)CCCC1(CNC(C1(CC)CCOCC1)=O)COC c1(C(N2CC(NC(c3cc(CCOC)on3)=O)(CO)C2)=O)cc(O)ccc1C S(=O)(=O)(c1cccc(Cl)c1)N1CC(CC(N2CCC(F)C2)=O)OCC1 C12(CCNC(C3C=CCN(C(C4(Cl)CC4)=O)C3)=O)CC(CCO1)C2 C#CC1(C(=O)NCC2(N(C)C)CCC2)CCN(C(=O)CC(C)(O)C=C)C1 N1(C(C2(CC(N)=O)CC2)=O)CC(CNC(=O)CC2CC(N(C)C)C2)C(O)C1 c1(C(N(CC(CC)NC(C2CC2c2ccsc2)=O)C)=O)ccc(F)cc1[N+](=O)[O-] C1(NC(c2cc(CC)no2)=O)CCC2(CCN(C(C3(CF)CC(=O)C3)=O)C2)C1 c1(C(C)C)conc1CC(N1CCC(CNC(c2cc(C3CC3)[nH]n2)=O)C1)=O N1(C(c2cccc(NC(C)=O)c2)=O)CC(C)N(C(c2cccc(=O)o2)=O)CC1C C1(CNC(c2nccc(C)n2)=O)CN(C(C2CC(=C3CC3)C2)=O)CCC1(C)C C(C(C)N=c1[nH]c(Cl)nc(C)c1F)NC(Cc1ccc(C)cc1Cl)=O c1(C(N(C(C)C(=O)NOCC(O)CO)CC)=O)n[nH]nc1OC N1(C(c2cc(CC)c(C)s2)=O)CCCC1C1CCCCN1C(=O)COC(C)(C)C C(CC(=O)NCCCCCC(C)C)(C(F)F)NC(c1ccc(C(C)=O)[nH]1)=O c1(CCC)ccc(C(=O)NC2COCC2CNC(=O)C(C)(O)CC)cc1[N+](=O)[O-] S(=O)(=O)(c1ccc(Cl)cc1Cl)N1C2CN(C(c3cc(Br)cnc3F)=O)CC21 CCC(O)CC(=O)NC1CCN(C(c2nc(Cl)sc2C)=O)C1 C1(C(C)(C)O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C.C12CCN1C2=O N1(C(CC2CN(C(Cc3ccc(C)s3)=O)C(C)C2)=O)CC2CCC(C1)C2O N1(C(CC(C=C)CCC)=O)CCCCC2(C1)CN(C(=O)CC(F)(F)F)C2 C1(C(N(CC(C)OC)C)=O)CN(C(=O)Cn2cc(CO)nn2)C(C)(C)C1 c1(CCCCC)cc(CN2CC(CNC(=O)Cc3ccnn3C)(COC)C2)n[nH]1 Cc1cccc(OCC(=O)OCc2cn(Cc3cccnc3)nn2)c1C c1(C(N2CC3CN(C(C4(n5ccnn5)CC4)=O)CC3C2)=O)cc(Cl)c(F)cc1Cl N1(C(C2CC(C)(C)C2)=O)CCC2(CCCN(C(c3ccc(F)c(F)c3)=O)C2)C1 c1(C(=O)NCC(CN(C(=O)C2=C(C)CCC2)CC)(C)C)c(F)ccc(F)c1O CCC(C)CCCCC(=O)NC(CCCOC)C(=O)N(C)CC1CCCCCC1 c1(C(=O)NCCC(C)NC(=O)CC2COC(=O)C2)ccnc2[nH]cnc12 c1(CCC(=O)NCCN(CCOC)C(C2CC23CCCC3)=O)ccccc1Br C(=O)(C(CO)c1ccccc1)N(CC(C)(C)NC(=O)C(N)=O)C n1(CCNC(=O)OC(C)(C)C)cc(C(N)=O)cn1.C1(=O)C(=O)NCCCN1 c1(OC)cccc(N(CC(C)C)C)c1.c1(C2N3CCCC3NC2=O)nocc1C Cc1ccc(OCC(=O)NCC(O)CN(C(=O)CSc2cnnn2C)C)cc1 CC1(C(N2CC3C(CNC(=O)CC4CCCCCC4)C3C2)=O)COC(=O)N1 c1(CCC)cc(C(=O)N(C)CC2CN(C(c3cnn(CC)n3)=O)CCO2)nn1C C(=O)(C1=CCCSC1)N1CCC(CCCCCNC(Cc2c(C)ocn2)=O)CC1 N1(C(CN(C)C(N)=O)=O)CC2CCCC(C1)N2C(C1CC12CCOCC2)=O c1ncc2c(n1)CC1CCC2N1C(=O)C.C1(C(C)(C)C)CCC(C(F)(F)F)CC1 C12(C(=O)NC3C(NC(=O)CCc4cnco4)CC3)CCCC1C2(F)F C1(NC(c2c(C(C)C)occ2)=O)CCC2(CCCN(C(=O)Cc3cncs3)C2)C1 c1(C(=O)NC(CNC(C=C(C)C(C)C)=O)C(C)C)nc2n(c1Br)CCC2 c1(OCC(C)C)ccc(C(N2CC(O)(CCNC(C3(C)CSC3)=O)C2)=O)cc1 C1(NC(=O)CCc2ccccn2)(CNC(=O)C(F)F)CCc2ccccc2C1 C1(CC(N2CC(n3cc(NC(=O)CN4CCCCC4)cn3)C2)=O)CCS(=O)(=O)C1 C(C=CC(=O)NC1(CNC(=O)CNS(N)(=O)=O)CC1)(CC)=CC C1(C(=O)OCC)CCNCCC1Nc1c(N(C(COCC)=O)CC)cc(Cl)cc1 N1(C(CC=C)=O)CCC2CN(C(=O)C(=Cc3cnn(C)c3)C)CC2CC1 C(CC(F)(F)CC(F)(F)F)ONC=O.C=CCCCn1cc(C(O)C2CC2)nn1 C1(CNC(C(C)NC(CC)=O)=O)CC2CN(C(=O)C=C(C)C(F)F)CC12 CC1CCN(C(=O)OC(C)(C)C)C1C(=O)NCCC(O)C(F)F Cc1n[nH]c2cnc(C(=O)NC3CN(C(C4CC5CCCCC45)=O)CC3C)cc12 n1(CC)ccnc1C(N1CC(O)(CNC(=O)CC2CCOC2C)C1)=O S(=O)(=O)(c1ccc(Cl)cc1Cl)N1CCC2CN(C(C=CC)=O)CC21 C1(c2cn(CC3C(C)C3C)nn2)(NC(CC2CC(CC)C2)=O)CCOCC1 C(C)(C(O)C(=O)NC1CC(CNC(c2cccc(N)n2)=O)C1)OC N1(C(C(CC)=CC)=O)CCC(CNC(c2csc(C(F)F)c2)=O)C1(C)C c1(NC)ccccc1C(=O)OCC(C)C(=O)Nc1ccccc1OC n1(CC=C)c(N(CCO)Cc2cccc(Br)c2)nnc1C(C1CCOCC1)C C1(N(C)C)CCCC(C(=O)NCC2CCN2C(C2CCCO2)=O)C1 c1(C(C)(C)NC(=O)NC(C)C(C)(C)C#N)ccc2c(c1)OCCO2 C1(CNC(CC(CCC)O)=O)CCN(C(=O)Cn2ccnc2C)C12CCC2 c1(CNC(CC(=C=C)C)=O)c(C)nn2c1CN(C(=O)CN1CCCC1CO)CC2 C(=O)(C1=C(Cl)CCCC1)N1C(CCCC(=O)NC2(C(=O)OC)CCCCC2)CCC1 c1(C(N2CC(NC(c3[nH][nH]c(=N)c3Br)=O)C2)=O)ccc2sncc2c1 c1(C(=O)NC2(CC)CCN(C(c3cc(C)n(C)c3)=O)CC2)cc(F)c(C)cc1F c1(NC(C(F)F)Oc2cccnc2)nccc(=NCC2=CCCOC2)[nH]1 Cc1nc(-c2ccccc2)[nH]c1C(=O)Nc1ccccc1OC(C)C N1(C(COC2(C)CCC2)=O)CCCC(NC(=O)C(C)(F)c2ccon2)C1 C1(CNC(Cc2ccc(C)cc2C)=O)CC2CCCC2N1C(=O)CCC1(C)CC1 C(CCC(C)(C)C(=O)N1CC2CCC(CNC(=O)C3=C(Cl)CCC3)C2C1)OC C(=O)(C1=CC2CCCCC12)N1CCN(C(c2cnn(C)c2Cl)=O)C2(C1)CC2 Cc1ccn(CC(=O)NCC2(CNC(c3cncc(Cl)c3Cl)=O)CC2)c(=O)c1 c1(C(=O)NCC2C(CNC(CC(COC)COC)=O)C2)cn2c(n1)CCC(C)C2 N1(C(CCC2CC(NC(c3cncc(C)c3)=O)C2)=O)CC2COCC2C1 N1(C(C(c2ccc(C)o2)C)=O)CC=CC(NC(c2ccc(Br)s2)=O)C1 c1(OC)ccc2[nH]c(=NCCCCCCCO)nc(N3CCC(F)C3)c2c1 N1(C(C2CC3CCN(CC(C4CCCCC4)O)CC23)=O)CCCC2C1CCN2CCO C=C(C)C1OCCC1C(N1CCC(CCC(N2CCCC2C(O)CO)=O)C1)=O c1(C(=O)NC2C(C)CCN(C(c3c(C)c(O)ccc3)=O)C2)cc2ncccc2o1 Cc1cccc2cc(C(=O)NC3C4CCN(C(=O)CC(C)(C)O)C34)oc12 N1(C(c2cc(SC)oc2)=O)CCCC(CNC(=O)C(c2ccccc2)F)C1 c1(C(N(CC(CNC(Cn2ncc(C)c2)=O)O)C)=O)cc(F)c(Cl)cc1F Cc1ccc(Cl)c(OCC(N2CC3CC3(CNC(C3(CF)COC3)=O)C2)=O)c1 C(=O)(CCC1=CCc2ccccc21)N1CCC(NC(C=CC=CCC)=O)C(F)C1 c1(C(=O)NCCC2(NC(c3csc(CN4CCCC4)n3)=O)CC2)ccc(Cl)cn1 c1(C(=O)NC2CN(C(C)(C)C)C(=O)C2)cc(Cl)c(Cl)c(C(N)=O)c1Cl c1(C(N2C(CNC(=O)CC3C=CCC3)CC2)=O)ccc(-c2ccccc2)nc1 C1(CC(=O)NC(CSC)CO)CN(C(C2(OC(C)=O)CCOC2)=O)CC12CC2 Cc1cc(Br)cc(C(N2CCOCC2C2CCC2)C(=O)NC2CC2)n1 Cc1cc(C(=O)N(C2CN(C(=O)Cn3nccn3)CC2F)C)nn1C(C)C N1(C(CC(C(C)C)OCC)=O)CC2(CCC(NC(c3cnc(Cl)s3)=O)CC2)C1 c1(C(C)OC)ncc(C(=O)NC2CC(N(C)C(c3cccn3C(C)C)=O)C2)s1 c1(C(N2CCC(F)(CNC(=O)C=CCF)CC2)=O)ccn2cnnc2c1 c1(CC(=O)N(C2CCC(NC(CCCC)=O)C2)C)ncn2c1CCC2 C1(N(C(C(C2CCC2)OC)=O)C)CCCCN(C(c2ccc(C(N)=O)cn2)=O)C1 C1(CC(=O)NCC2C=CCN2C(c2cc(C3CCC3)[nH]n2)=O)CCCC2CC12 C(CN=C(NCC(OC)OCC)NC1CC(O)C12CCC2)C1(CNCC)CC1 c1(NC(C2CCN2Cc2cc(F)c(F)cc2Br)=O)cc(Cl)c(O)cc1Cl CC1CC(NC(=O)CCOC2CCCCC2)CN1C(=O)CCc1cncc(F)c1 c1(C(=O)NC2C(SC)CN(C(c3cc(Cl)no3)=O)C2)cc(C)c(C)cc1C c1(C(=O)NCCCCNC(C(C)NC(CC)=O)=O)ccc(S(=O)(=O)NOC)cc1 C=CC(CC)CC(=O)N(CCCNC(=O)Cc1ccc(CC)c(F)c1)C c1(CNC(C2(C=C)CCC2)=O)cc(C(=O)NCC(C2CCCC2)O)ccn1 C12(C(=O)NC3CN(C(CNC(=O)CC(F)(F)F)=O)CC3O)CCCC(C1)OC2 CC#CCCCC(=O)NCC=CC(=O)NCC(CC)C(C)(F)F c1(C(N2CC(C3N(C(CC=C)=O)CCC3)(O)C2)=O)cc([N+](=O)[O-])nn1C C(=O)(CCCC(=O)N1CCC(C(=O)NC(c2ccccc2C)C)C1C)OC N1(C(C2CCC(=O)N2)=O)CC(NC(c2cc3cccnn3n2)=O)CC12CCOC2 C1(CNC(CC)=O)CN(C(c2cccnc2OC(C)C)=O)CC1C CC1=C(C(=O)NC(CC2CC2)CC(=O)NC(CN(C)C)CCO)CCCO1 C(C1(O)CCc2cc(F)ccc21)NC(c1cc(C2CCC2)[nH]n1)=O N1(C(CCC)=O)CC(NC(=O)CCc2ccoc2)CC2(CCC2)C1 N1(C(CC2C(C)(C)COC2)=O)CC2CC1CN2C(=O)CCOCC(F)(F)C(F)F C12(C(N3CC(O)(CN(C(=O)CC4C=CCC4)C)C3)=O)CC3CC(CC(C3)C1)C2 N1(C(c2nc(C)oc2)=O)CCC(C)(C)C(NC(c2ccc(OC(F)F)nc2)=O)C1 CCCCCC(=O)OC(C)(C)C.C(CCCCCn1cc(C(C)N(C)CCO)nn1)N c1(C(N2CCC(CN(C(c3c(C)scc3)=O)C)C2)=O)ccc2c(c1)CC2 CC1(C)CC(CO)N(C(c2ccc(CNC(C3CC3[N+](=O)[O-])=O)nc2)=O)C1 C(=O)(CCC(C)O)NC(CNC(CCN(CC)CC)=O)C(C)C c1(OCC)ccc(C2(C(=O)NC)N(C(C3CC4CC4C3)=O)CC2)c(C)c1 C1(C(=O)NC(C(=O)OC)CC#N)C=C(c2ccc(Cl)cc2)CC1 C1(C(N2C3CC(C(N4CCCC5(CC5)C4)=O)C2CC3)=O)C2Sc3ccccc3C12 N1(C(C(CC)C)=O)CCC2(CCCN2C(=O)CCNC(c2cccs2)=O)C1 N1(C(C2C(C)=CCC=C2)=O)CCCCC(N=c2nc[nH]cc2C#N)C1 c1(N(C)C)nc(Cl)c(C(=O)NCCCCCNC(C2(CO)CCOC2)=O)s1 C1(NC(c2n(CC)ccc2)=O)CC(O)CN(C(=O)CC2CCC=CCC2)C1 N1(C(C(CC)(F)F)=O)CCCC(F)(C(=O)NCCNC(=O)NCC)C1 N1(C(=O)CC2CCCCO2)CC2(CCCN2C(c2cccc3ncsc23)=O)C1 c1(C(C)C)cc(C(=O)NCC(CO)NC(c2sccc2OC(F)F)=O)n[nH]1 C1(NC(c2nc(C(C)C)oc2)=O)CC2CC(C1)N(C(C1(C)CC(O)CN1C)=O)C2 C1(NC(=O)C(F)C2CCOC2)CC1C1CCCN(C(c2c[nH]cc2C2CC2)=O)C1 N1(C(C2C(C)C2(F)F)=O)CC(NC(=O)C=C2CCN(C)CC2)C(O)C1 C1(CC)(Nc2nccc(CO)n2)CCN(C(C2(CF)CC2)=O)CC1 CCC(C)(COC)C(=O)NN1CCCC1C(=O)NCCC1CC(C)C1 C1(NC(=O)CCN2CCCCC2)CCCC12CN(CC(=O)N(CCO)CC1CC1)C2 N1(C(C2C(CC)CCC2)=O)CCC(C)C(NC(=O)CC(C)(C)CC)C1C Cc1cnc(CCC(=O)NCC2CCN2C(C2CSCCS2)=O)[nH]1 N1(C(N2CC(C)C(C(=O)OC(C)(C)C)C2)=O)CC(C)C(F)(F)C1 C=CCC(CC(F)F)NC(C1C(CC)CCCN1C(=O)COC1CCOCC1)=O CC(C)CCC(C(=O)NC1(C(=O)N(C)C)CC1)NC(=O)CCC(C)(C)N(C)C N1(C(Cc2c(C)ocn2)=O)CCOC(CN(C)C(C2CCC(=O)N2C)=O)C1 N1(C(Cc2cc(C)n(C)n2)=O)CCN(C(c2ccn(C(C)C)n2)=O)CC(C)(F)C1 C1(NC(C2(CC#C)CCCC2)=O)CCC(C)N(C(=O)Cn2cc[n+](C)c2)C1 CC1CN(C(=O)Cn2cc(C#N)cn2)CC1NC(=O)C(C1(O)CCCC1)F Cc1ccc2c(=NC(=O)NCC3CC3C3CC3)[nH][nH]c2n1 N1(C(c2c(C)n(C)c(-c3ccccc3)c2)=O)CC23CCCC2(COC3)C1 C(=O)(C1CCc2cccc(OC)c21)NC(CC=C)CNC(=O)Cn1cc(Cl)cn1 CC1(C)CC(C(=O)NC2CNC(=O)C2)CCN1C(=O)C(F)=CC1CC1 Cc1[nH]cc(C(=O)NC2CN(C(=O)C(C)C3(O)CCC3)CC2(C)C)c(=O)c1Cl C1(C(=O)NC(CN(C(c2occ(C)c2)=O)C)(C)C)CC12CC(O)C2 C#CC1(C(=O)Nc2ccc(OC)nc2)CCN(C(=O)C#CC2CC2)CC1 C(=O)(CCCCNC(C1CCCCN1C(c1ccc(F)s1)=O)=O)OCC N1(CC)CCC2(CC1)CC(Cn1nc(-c3ccsc3)nc1C(=O)OC(C)C)=NO2 C1(C(=O)NCCN(C(C2(O)COC2)=O)C2CC2)CCCC1n1cccc1 C1(CNC(C2COC3COCC23)=O)CCC2(CN(C(=O)CC3CCOCC3)C2)O1 C1(SC)CN(C(=O)CC2CCCCC2O)CC1NC(=O)CCc1ccncn1 c1(C(=O)NC2CN(C(C(C(CC)O)(F)F)=O)CC2O)sc2cccc(F)c2c1Cl C1(NC(c2cnc(S)[nH]2)=O)CC2CC(C1)N(C(c1ncsc1Br)=O)C2 Cc1nccc(CNC(=O)C=CCC(C)(C)NC(=O)Cc2cc[nH]n2)n1 C(=O)(CCCC(CC)NC(=O)C1=C(C)OCC1)N(C1CC(SC)C1)C c1(C(N2C(CNC(C(C=CC)O)=O)CCC2)=O)cnc2cnn(C)c2c1 C1(C(=O)Nc2scc(C)n2)CC12CCN(c1ncnc(C)c1Br)C2 N1(C(c2cn(C)cc(Br)c2=O)=O)CCCC(N=[N+]=[N-])CC1 C(=O)(C=C1SCC(=O)N1C)N1CC(NC(C(CC=CCC)C)=O)C(OC)C1 C12(C(=O)NC3C(C=C)OCC3)COCC1CN(C(=O)Cc1cccc(F)c1)C2 c1(N2C(C)(CNC(C(C)NC(C)=O)=O)CCC2)ncc([N+](=O)[O-])cc1F CCCC(C)(C)C(=O)NCC1(O)CCCN(C(c2nccc(Cl)c2O)=O)C1 C1(C(=O)NCC2CCC(NC(COCC(C)C)=O)C2)CC2CCC(C1)C2(F)F C1(OC)CC(CCNC(=O)CN2CCC2C)N(C(C2CCC=CCC2)=O)C1 n1(-c2c(C)ccc(C)c2)nc(-c2cccc(Br)n2)nc1C1CCc2c[nH]nc21 c1(CC(=O)N(CC(C)N(C)C(C2CCC23CCC3)=O)C)c(F)cccc1F c1(NC(C2(C)N(C(c3cc(C)on3)=O)CC2)=O)ncc(Br)nn1 C1(C(N2CC(C(=O)NCC(C3CCCCC3)C)(SC)C2)=O)CC2C(C1)C2(C)C C1(N(C(c2c(OC)csc2)=O)C)C2CN(C(C3CC(F)(CF)C3)=O)CC12 C(=O)(CCCCC(C)(C)C)N1CC(NC(C(CCCC)CC)=O)C2(C1)CCC2 C1(CCC=C)(C(=O)NCC(O)CO)CN(C(=O)Cc2ccc(Cl)s2)C1 C(C1CCCC1)=C(C)C(=O)NC(C)C(=O)NC(C)Cc1nn[nH]n1 c1(CN(C(CN2CCC(CCCC)C2)=O)C)ccccc1Cl C1(NC(c2cc(C)nn2C)=O)CCN(C(c2sc(Cl)cc2Cl)=O)C(C)C1 N1(C(C)C(N2CCCC2CNC(=O)CC2CCN(C3CC3)CC2)=O)CC2CCC1C2 N(C(=NCCC(=O)OC(C)C)NC1CC(=O)N(C(C)C)C1)CC(CC)(C)OC N1(C(Cc2c(C)nsc2)=O)CC2CC1CN2C(=O)Cc1sc(=N)[nH]c1-c1cccs1 Cc1nn(C2CCCCC2)cc1C(=O)NCC12CC(CN1C(=O)C=C(Cl)Cl)C2 C1(NC(CC2C(C)OC(C)C2)=O)CCN(C(=O)Cc2nncs2)CC1(C)C c1(N2C(C3CCN(C(CC=C)=O)C3)CCC2)cc(OC)nc(OC)n1 C1(CCC(=O)NC2CC(N(C(=O)C(N3CCOCC3)C3CC3)C)C2)CCCN1C CCC(C(=O)NC(C1CCN(C(c2[nH]nnc2C2CC2)=O)C1)C)c1ccccc1 C1(CNC(c2c(C)nn[nH]2)=O)CN(C(=O)CCc2nncs2)CC1O C(=O)(CCC(F)F)N(CCNC(C(C)SC(C)C)=O)C(C)C c1(C(N2CC(NC(c3cnc(CC)[nH]3)=O)C(C)CC2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(C(N2C(C3(NC(C=CC=CC)=O)CC3)CCC2)=O)CN2CCC1(C)CC2 CC1(C)CCCC(C(=O)NCCC2(NC(c3cnc(O)s3)=O)CCC2)CC1 C1(NC(C(c2ccc(C)cc2)(F)F)=O)COCCN(C(c2cn(C)cc2C)=O)C1 C(CC(=O)OCc1ccco1)(C(F)(F)F)N1C(C)CCC1 c1(NC(C)CCN2CCOCC2)nc(N(CCC#CCO)C)nc2c1CCC2 c1(NCCN(C(C2CC(C#C)(O)C2)=O)CCC(C)=O)ccc(Cl)c(Cl)c1 C1(NC(c2ccc(CN(CC(N)=O)C)cc2)=O)CCOC12CCOCC2 c1(C(=O)NC(C)C(C)NC(C2CN(C)C2)=O)cnn(-c2ccccc2)c1 C1(NC(CCc2c(C)n(C)nc2)=O)CCN(C(c2nonc2N)=O)CC(C)(C)C1 Cc1c(C(N2CCOCC(CNC(C3(C)CCCN3C)=O)C2)=O)sc2cncn12 CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CC1(C)CNC(=O)C(c1ccccc1)F C1(CC(=O)NC(C(C)n2cccn2)C)CCCCN1C(C1OC2CCC1C2)=O c1(C(=O)NC(c2ccccc2)CNC(C2(C(C)C)CC2)=O)ccc(N)cc1Cl N1(C(CSC(C)(C)C)=O)CC2CCC1C(CNC(=O)C1CC1)C2 CCCC(C(=O)N(C)Cc1ccc(C)cn1)NC(c1ccccc1)=O C1(C(=O)NC2(C)CCN(C(c3nn(C)c(Cl)c3Cl)=O)C2)Cc2cc(F)ccc2O1 C(=O)(C(CC(C)C)C(N)=O)N1CC(C(C(=O)N(CC=C)CCOC)OC)C1 Cn1nc2c(c1C(=O)Oc1c(F)cc(OC)cc1F)CN(Cc1ccc[nH]1)CC2 CC1CCCN(C(=O)C2=CCOC2)C1CNC(c1ccoc1C(F)(F)F)=O c1(C(=O)NC2CN(C(C(CCC)OC)=O)CC2C)cc(S(N)(=O)=O)cs1 CCCC(CC)CCC(=O)NC1CN(C(c2ccc(C#N)o2)=O)CC1O N1(C(C(CO)NC(C2N(C)CC(O)C2)=O)=O)CCC(C2CCC2)CC1 C1(C(C)NC(c2coc(CO)c2)=O)CN(C(C2CSCC(=O)N2)=O)CCO1 C(=O)(CC1=NNC(=O)C1)N1CC(C)C(CNC(c2cc(Cl)cc(F)c2N)=O)C1 Cc1cc(F)c(C(=O)NCCCNC(N)=O)cc1Br.C(C)(CCSC)NC C1(CCC(=O)NCCOCC#C)CCN(C(c2c[nH]nc2OC)=O)C1 C1(CNC(CN(C(C)=O)C)=O)(NC(c2ccnc(C(F)F)c2)=O)CCCCC1 c1(CO)ccc2ccccc2c1C.C12CC1C(=O)N(CCC)CCN(CC)C2=O CC(=O)CCCC(=O)NCC1CCN(C(c2coc(C(N)=O)c2)=O)C1 c1(C(=O)NCC(C)C(=O)O)ccc(F)c(-c2cn(CC3(O)CCSC3)nn2)c1F c1(C(=O)NCCC(C)NC(c2cc(C)oc2)=O)oc2c(C)ccc(C)c2c1C C#CCC(C(=O)N(C1(C)CC1)C)NC(C1CCCN1C)=O C1(F)(C(=O)NCC(c2ccccc2)N(C(C=C(CCC)C)=O)C)CC1(F)F CC(O)CCCCCC(=O)Nc1ccccc1CN1CN(C)C(=O)N(C)C1 C1(NC(C2(CCCC)CCC2)=O)CN(C(=O)Cc2cccc(C(F)F)c2)CC1O c1(C(=O)NCCC(CNC(c2c(C)ccnn2)=O)O)c[nH]c(=N)nc1C N1(C(CNC(=O)NC)=O)CCN(C(c2cc(O)nc(C)n2)=O)C(C(C)C)C1 CC(C)CCCC(C)C(=O)N(C)CC1CCN(C(C2COC(=O)N2)=O)CC1 C1(NC(=O)CCC2CCC2)CCCC2CN(C(=O)CNS(N)(=O)=O)CC12 CCCC(C)C(=O)N1CCC(F)(C(=O)Nc2nccnc2C)C1 c1(NC(C2CCCN(c3cc(C)nc(C)n3)C2)=O)ccc(C(F)(F)F)c(F)c1C C1(NC(C(CCN(C)C)O)=O)(CO)CCCN(C(=O)C(c2cccc(N)c2)O)C1 N1(C(C(C(CC)CC)C)=O)CC(CNC(=O)C=Cc2ncc[nH]2)OC2COCC12 C1(C(=O)NCCN(C(c2cc(COC)on2)=O)CC)CCOC(C)C1 CC1CCN(C(C2CC(NC(c3cc(Br)c(F)cc3F)=O)C2)=O)CC1(F)F C1(NC(=O)CCC2CCCC2)CN(C(C2(CC3CC3)CCCO2)=O)CC1F c1(OC)ccc(CC(=O)NC2CC(F)CN(S(=O)(=O)C(C)COC)C2)cc1F C1(NC(Cc2c(C(=O)OC)csc2)=O)C(C)CCN(C(=O)CNC=O)C1C C(C1=CCN(C(C2(F)CCCCCC2)=O)CC1)NC(c1ncc(Cl)cc1F)=O C(CC(=O)NC1CCC(CO)CC1)(C(C)C)NC(c1c(CC#N)cccc1)=O C1(C)(C(=O)NC(C23CCC(CC2)C3)CNC(CCNC(C)=O)=O)CCCS1(=O)=O C1(NC(C2CC(CCC)OCC2)=O)CCCC2CN(C(=O)C(C)=CC3CC3)CC12 C1(NC(COCC)=O)CS(=O)(=O)CC1N=c1ccnc(-c2cccc(Cl)c2)[nH]1 N1(C(c2c(NC)snc2C)=O)CC(NC(=O)CCc2ccccc2)CC(O)C1 C1(CNC(Cn2cc(C(C)=O)nn2)=O)CC(NC(C2C3COCC23)=O)CCO1 c1(C(=O)NC(C(C)C)C(=O)NC(C)CS(C)(=O)=O)cccc2ccoc12 N1(C(CC2(C=C)CC2)=O)CC(CNC(c2nnc(S)n2C)=O)OC2(CCC2)C1 C(c1ccc(C#N)cc1)=CC(=O)NC1CCC(C)N(C(c2cccc(=O)o2)=O)C1 N1(C(C=C(C)CCc2ccccc2)=O)CC2OCC(NC(=O)C3=CCCS3)C2C1 CCC(O)C(F)(F)C(=O)NC(C1CC(NC(c2coc(C3CCC3)n2)=O)C1)C c1(NC(C(c2cc(O)cc(Cl)c2)N2CCC(C(=O)NC)C2)=O)ccc(Cl)cc1F C1(C(N(CC(C)N(C(C(C2CC2)SC)=O)C)C)=O)CC2(C1)OCCO2 c1(C(N2C(CNC(c3c(CC)non3)=O)C(C)CC2)=O)cncc(S(N)(=O)=O)c1 N1(C(c2c(C)n(C)nc2)=O)CC(F)(F)CC1(C)CNC(=O)Cc1ccnnc1O C1(NC(C=CCC)=O)CCC(N(C(=O)C(C(C)C)Oc2ccc(Cl)cc2)C)CC1 C12(C(N3CC(C)(NC(CC(C=C)C)=O)C3)=O)CCCN(CC1)S2(=O)=O c1(C(=O)NC(C2(O)CCN(C(=O)CSCC(N)=O)CC2)C)ccccc1[N+](=O)[O-] C12(CNC(=O)Nc3c(C)c(Cl)ncn3)CCC(CC1)C(C)(C)O2 N1(C(C)C)CCOC(CN2CC(CNC(c3cccc(C(N)=O)n3)=O)C2)C1 Cc1[nH]nc2c1CC(C(N1CC(CNC(=O)CCCCNC(N)=O)C1)=O)CC2 CCCC(C)(CCC)C(=O)NCC12CC(CN1C(=O)C(C)CCC(C)(C)C)C2 Cc1ccnc(C(N2CCOC(C(C)NC(C3CC(C)(C)C3)=O)C2)=O)n1 CC1CN(C(c2c(Cl)nsc2Cl)=O)CCCN1C(c1ccc(C(N)=O)cc1)=O C1(CC)CCCCN1C(=O)CC1C=CC(NC(=O)Cc2ccc(C)o2)C1 Cc1cc(C(=O)NC2COCC2NC(C2(C)CCC(C)C2(C)C)=O)cc(C)c1N CCC(CS(C)(=O)=O)NCc1cccc(-c2nncn2CC)c1 c1(C(N(C2CN(C(C(CC=CC)CC)=O)CC2(C)C)C)=O)[nH]cc2c1CCCC2 c1(C(N2CC(C)(NC(C(CC)C(C)C)=O)C2)=O)cc2c(o1)CCCNC2=O C12(C(=O)NC(c3cn(C)nn3)C)CCC(CC1)N(C(C1CCOC1(C)C)=O)C2 CCCCCCNC(=S)NC(C)C c1(C(=O)NCC(CC=C)NC(c2ccc(COC)o2)=O)ccc(Cl)nc1 Cc1ccc(C(=O)NC2CCOCC2NC(=O)CCNC(C2CCC2)=O)c(F)c1 c1(OC)cc(C(=O)NC(C)CN(C(=O)CCc2ccc(N(C)C)cc2)C)ccn1 C(CC(C)C(F)(F)F)NC(=O)NCC1CC(C)SCC1 C1(NC(c2ccc(C)cn2)=O)CCC2CN(C(c3cc(Cl)cnn3)=O)CC2C1 c1(C(=O)NCCCCC(C)NC(c2c(C)sc(O)n2)=O)cnn2c1CCCN2 N1(C(C(COC)O)=O)CC2(CC(NC(c3cnc(OC)cc3C)=O)CO2)C1 c1(C(=O)NC(C2(O)CN(C(C3CC(F)CN3C)=O)C2)C)c[nH]c2ccc(F)cc12 C(=O)(C1=Cc2ccccc2OC1)N1CCN(C(CC(C)N(C)C)=O)C2(C1)CC2 Cc1ccn2ncc(C(=O)NC3CC(NC(c4cc(CO)[nH]n4)=O)C3)c2c1 C1(NC(CN2C(C)CC2)=O)CCN(C(C2CCN(CCC3CC3)CC2)=O)C12CC2 C1(C(=O)NC23C(NC(C(C)=C4CC4)=O)CC(CC2)C3)CCn2nnnc2C1 C#CC(CC(C)(C)C)NC(=O)C(C)N(C(C1(C)CC(C)(C)C1)=O)C1CC1 N1(C(c2cc(C3CCCC3)no2)=O)CCCC(N(C(=O)CCC(F)F)CCO)C1 c1(N2CCC(COC)CC2)ccncc1S(=O)(=O)NCC1COC(C)(C)O1 N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(c3c(C)[nH]c4ccccc34)=O)CC12 c1(NCC2C(NC(C(CC)OC)=O)CCCC2)cc2nncn2c(C)n1 Cc1nc(-c2ccccc2)oc1C(=O)NC(C)CNC(=O)CC(C)CN(C)C Cc1ccnc2c1N(C(c1cc(Cl)ccc1CN1CCCC(O)C1)=O)CCO2 CCCC(O)CC(=O)N1CC(NC(c2ccc(OCC)cc2)=O)CC1(CC)CC C1(CNC(CCSCCN(CC)CC)=O)C(O)C(O)CN1C(=O)CCS(C)(=O)=O N1(C(C2N(C)CCC2)=O)CC2CC2(CNC(=O)C(C)(C)c2ccns2)C1 C=C(C)C1OCCC1C(=O)NC1C2CC1N(C(c1cnncc1C)=O)C2 C1(NC(c2cc(C(F)F)[nH]n2)=O)CCC2CC1CN2C(c1cnn(CCF)c1)=O C(=O)(CC(C(=C)C)OCC)NC1(CO)CCN(C(CCC(=C)Br)=O)C1 C1(C(N2CCC(CN(C(=O)Cc3cnsc3)C)C2)=O)CC(c2ccncc2)=NO1 C1(CNC(c2c(C)n(C)nn2)=O)CN(C(=O)CC2CCCOC2)CCN1C N1(C(C=C(C)CCc2ccccc2)=O)CC(NC(=O)CC(C)C)CC(C)(C)C1 C1(C2CCCC2)(NC(C2C=CC(NC(=O)CC3CCC=CCC3)C2)=O)CC1 c1(NC2CCCN(C(C(CC)NC(N)=O)=O)C2)ncnc2c1ncn2CC C=CC1CCCN1C(=O)C(C)(CO)NC(C1COCC1C(N)=O)=O C(=O)(C(O)C(F)(F)F)N(C)CCN(C(=O)CCc1cc[nH]n1)C c1(C(c2n(CCC)nnn2)NCc2nnc(C(F)F)s2)ccc(S(C)(=O)=O)s1 CC1CN(C(C2OCCC2NC(=O)CC2CC(F)C2)=O)CCC1(F)F C1(C(C)NC(C=CCC)=O)CCN(C(=O)CC(=O)NCC)CC1 N1(C(C(C)OCC=C)=O)CC(C)(CNC(C2CC2c2ccnn2C)=O)CC1(C)C c1(C(=O)NC(CNC(C2(CC=C)CCOC2)=O)C)sc(C2CCCC2)nc1C C(=O)(C1=NOC(CNC(c2ccc(C(N)=O)[nH]2)=O)C1)NC(CN(C(C)C)C)C N1(C(C(=O)NCC)=O)CC(C)C(NC(=O)Cc2c[nH]c3ccccc23)C(C)C1 C1(CSC)CCCN(C(c2ccc(Br)cn2)C(=O)NCCCSC)C1 CCC(CNS(C)(=O)=O)N=c1[nH]c(=NCC(CC)n2cccn2)[nH]c2cc[nH]c12 N1(C(C(C)OCC2CC2)=O)CC(O)C(O)C1CNC(=O)C(C)(F)F N1(C(=O)OC(C)(C)C)CCCCC12CCCN(C(C1CC1(C)C)=O)C2 N1(C(C(C=C)(C)CC)=O)CC2CCN(C(=O)CC3(OC)CC3)CCC2C1 C1(NC(c2ccc(CC)nc2)=O)COC2(C1)CN(C(c1cc(N)ccc1C)=O)C2 c1(CC(=O)NCCCCCNC(c2ccc(C(C)=O)o2)=O)ccc2[nH]ccc2c1 O=C(CCCc1ccncc1)NCCCNC(c1cc(CO)on1)=O c1(OC)cc(C(=O)NCC#CCNC(=O)COC(C)C)c(Cl)cn1 C(=O)(C1=CCC2CCC1N2C(C1(C)CC2CC2C1)=O)NCc1cc(OC)no1 c1(OCC(=O)NCCN(C(C2CC(N3CCCC3)C2)=O)CC)cccnc1 CCCCCCCCCC(O)C(=O)N1CCCC(NC(c2cnc(C)[nH]2)=O)C1C C1(CNC(c2cc(SC)ncc2)=O)C(C)CCCN1C(c1occc1C)=O C(=O)(C(C)CCC(C)(C)C)N1CCC(O)(CN(C(c2c(C)nc[nH]2)=O)C)C1 c1(OC)cncc(CCC(=O)NCC(O)CCNC(C2CCCC2C(C)C)=O)c1 N1(C(Cn2ccc(C)n2)=O)CCC2(CCCN(C(c3cc(C#N)[nH]c3C)=O)C2)C1 N1(C(c2cncc(OC)n2)=O)CCC(NC(=O)CC2CCC(=O)N2C)CC1C c1(C(=O)NCC(CC)NC(c2ccccc2COC)=O)c(C)nn(CC(C)C)c1Cl Nc1c(C(=O)NCCNC(c2[nH]nnc2-c2ccccc2)=O)cccc1F C1(C(C(C)NC(=O)CN(C)C(C)=O)OC)CCCCC1 c1(-c2cccc(CN(C(C)C)C)c2F)ccc([N+](=O)[O-])cc1O C1(C(=O)NC(CC)CNC(=O)Cc2cnn(CC)c2)C(C(F)(F)F)C1[N+](=O)[O-] c1(NC2(C(=O)NCCNC(C)=O)CC2)cc(C(C)C)cc(N)c1 C(=O)(C(F)C1=CCCCC1)N1CC2CN(C(c3c(C)nsc3N)=O)CC2C1 C1(C(=O)NCC2CC(C)(C)C2)CCN(C(=O)CCCCN(C)C)CC1O N1(C(c2c(CC)nco2)=O)CCN(C(C2CCC(=O)N(CC)C2)=O)CCC1C c1(C(N2CCC(COC)(NC(=O)CCc3nnc(C)o3)C2)=O)cc2n(n1)CCC2 c1(NCc2c(-n3cccn3)c(C)n(N)n2)nn(C)c2ccccc12 N1(C(C(COC)(C)C)=O)CCCC2(C1)C(NC(=O)C1=CSCCO1)CCN2C C#CCC(C)(C(=O)N1CCCCC1C)NC(c1cc(C)ccc1C)=O N1(C(c2n(C)ccn2)=O)CC2CCC1C1CN(C(=O)CCc3ccnn3C)CC21 c1(C(N2CC(CNC(c3c(C)csc3)=O)OCC2)=O)cc(Br)c(F)cc1F C1(C(=O)NCCC2(NC(c3cnc(O)s3)=O)CCC2)(CC)CCCCC1 c1(NC(c2c(C(=O)OCC)c[nH]n2)=O)ccc(NC(=O)C(C)C2CCOC2)cn1 C(CCCCC(=O)N(C(C)(C(=O)NCc1ccc(F)cc1C)C1CC1)C)OC NS(=O)(=O)c1cc(C(N2CC(OCCNC(=O)C(F)(F)CO)C2)=O)co1 n1(C(C)C(=O)N(C2CCCS2)C)cc(C(C)(C)CC2CC2)nn1 N1(C(C2C(C)CCO2)=O)CCOC(C(=O)NC(C2CCOC2)CO)C1 N1(C(C(=O)NC2(C)CC(C)(C)OC2=O)=O)CCC2C(CCCC2(F)F)C1 N1(C(C(=C)F)=O)CCC12CN(C(=O)CCc1ccccc1OC(F)(F)F)C2 c1(OC)nscc1C(N1CC(O)(C2CCCN2C(c2ccsc2Cl)=O)C1)=O c1(C(=O)NCC(C(=O)Nc2ccc(OC)cc2)OC)ncnc(O)c1F C(CC(C(=O)N(C1CCCC1C#N)C)NC(=O)C1=CCCC1)OCC c1(C(=O)NC(CN(C(=O)CCN2CCOCC2)C)(C)C)snc(Cl)c1Cl c1(C(=O)NC2(CF)CCN(C(CCNS(C)(=O)=O)=O)C2)ccc2c(c1)B(O)OC2 c1(SC)c(NC2(c3nnnn3C3CCCC3)C(OC)CCC2)cnnc1COC N1(C(=O)Nc2csc(Br)c2)CC(CO)CC12CCOCC2 CC1(C)CCN(CCNC(c2ccc(CNC(C3CC3(F)Cl)=O)o2)=O)C1 c1(C(N2CCC(F)C2)C(=O)NC2CCOC2)ncc(C2OCCO2)s1 C1(c2nc(C(c3ccoc3)OC)on2)(c2cccs2)CCCCC1 c1(OC)ccc(C(=O)NC2CC3CC2N(C(=O)C(C)(C)C#N)C3)cc1C(F)F CCCCCCCCC(=O)N1CCOCC1CN(C(=O)C(C)(CC)CO)C CC1(C)CCCC1CNC(c1[nH]ccc1-c1cccs1)=O C=CCCCC(C(=O)NC(CC)C(C)(C)C)NC(=O)COCCF c1(NC(=O)NNC(=O)c2ccccc2)cc(F)c(F)c(F)c1 C(=O)(CCCNc1cccnc1)N1CC(OCCNC(c2cnns2)=O)C1 c1(C(N2C(COC)CN(C(=O)C=CBr)CC2)=O)ccnc2ccccc12 C#CC12CCC(C(=O)NC3CN(C(C4COC4)=O)CC(C)(C)C3)(CC1)CC2 C(CNC(C1CN(C2CCC2)C1)=O)(CCOC)NC(C1(OC(C)C)CCC1)=O C1(C(N2CC3CC(CN(C(CNS(N)(=O)=O)=O)C3)C2)=O)CCCC2(C1)CC2(F)F CC(C)S(=O)(=O)c1ccccc1NC(=O)CC1(C)CCN1Cc1cccnc1Cl N1(C(c2cccc(N)n2)=O)CCC2(NC(c3ccn4ccnc4n3)=O)CCCC12 c1(CC(=O)NC2CCN(C(C3CC(C)N(C)C3)=O)CC2)c[nH]c2ccncc12 c1(C(C(=O)NCCNC(C2CCC2)=O)C)cccc(C(=O)OC)c1 N1(C(c2cc(C)ncc2C)=O)CCCC2(CCC2NC(c2cnccc2C)=O)C1 C12(NC(=O)CN3CC=CC3)CCOCC1CN(C(c1cccc(C(F)F)c1)=O)C2 c1(OC)ccc(-c2cc(CN(C3C4CN(C(=O)C(O)CCl)CC34)C)n[nH]2)cc1 CC(C(=O)NCCC1CN(C(c2cc(Cl)c(Br)cn2)=O)C1)C(C)(C)C CCC(C)C(C(=O)NC1CC(NC(c2coc(-c3ccccc3)c2)=O)C1)OC c1(C(=O)NC2C(NC(c3cn(CCC=C)nn3)=O)COC2)cncn(C)c1=O N1(C(CCCOCCC)=O)CCCC(CO)(NC(c2oc(CC3CC3)nc2C)=O)C1 C1(COC)CN(C(c2c(C3CC3)noc2C)=O)CCN1C(c1cscc1C)=O C(=O)(C1CCc2nccn21)NC1(CC=C)CCN(C(c2coc(C(F)F)c2)=O)C1 C1(NC(C2CC(NC(c3ccccn3)=O)C23CCC3)=O)CCc2nncn2C1 C1(NC(C(C(C)C)OC)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1F Cn1cnc(CC(=O)NCC(C2CCOC2)NC(=O)COC2CCC2)c1 c1(C(N2CC(CCNC(C(C(CC)C)O)=O)C2)=O)ccc(F)c(S(N)(=O)=O)c1 c1(CC)ccccc1CCNC(C1CC1CCCC(=O)OC)=O.C(F)(F)F CC(C)CCC(=O)NCC(=O)NC1C=CCN(C(=O)COCC2CCOC2=O)C1 n1(CC)c(CNC(=O)CN(C(=O)CC2CCOCC2)C2CC2)nnc1O C(=O)(C(CC(C)C)OC)N1C(C2(NC(c3c(CC)nc(C)o3)=O)CC2)CCCC1 c1(OC)ccc(C(F)(F)F)cc1CNC12CC(C(N3CCC3(C)C)=O)(C1)C2 c1(C(=O)NC2(CC=C)CCN(C(C3CC(N(C)C)C3)=O)C2)ccc(S(C)(=O)=O)s1 C1(C(c2cn(CCNC(C(C=CCCC)O)=O)nn2)C)CCN(C)CC1 Cn1ncc(C(=O)NCC(c2ccccc2)NC(=O)Cc2sc(O)nc2O)c1Cl c1(C(C)C)ccc(CC(=O)NCC(C)(CO)NC(=O)C(C)C2CCCC2)cc1 C1(CCNC(c2cc(C(F)(F)F)no2)=O)CCCN(C(=O)CC2CCOC2=O)C1 CC1CCCCC1(CO)NC(c1cncc(CNC(=O)CCCN=[N+]=[N-])c1)=O c1(C(=O)NC2CCC(CNC(c3occ(C)c3C)=O)CC2)ccc2nccn2c1 c1(C(N(C2(CNC(=O)CC3(C(F)(F)F)CC3)CC2)C)=O)cnco1 C1(C(=O)NCCC2CC(NC(c3ccc(=O)oc3)=O)C2)CC2CCC1O2 C(C)(C(=O)NCCCn1cc(-c2ccc(C)cc2Cl)nn1)(C(C)C)OC C#CCC(C)(C)C(=O)NCCOCCNC(=O)CCC(N)=O C1(C(=O)NCC2CN(C(C3CCN(C(CC)=O)C3)=O)CC2C)CN2CCC1CC2 CC1(C)CCC(C(=O)NC2(CNC(=O)CCC3CC(F)(F)C3)CCC2)O1 c1(C(c2nnnn2C)NC(CCC)Cn2cncn2)ccncc1COC CC(CN(C)C)C(=O)N1CC(C(O)C(=O)N(C)CCF)C1 c1(C(=O)NCC(CC)(C)NC(c2ccn(C)c2)=O)cc(COC)c(C)s1 C1(C(=O)NC2C(CNC(COC3(C)CCC3)=O)CCCC2)CC(C)(C)C12CC2 C(CC(=O)NCCC(C)OC)(C(F)F)NC(C1(CC)CC(C)(C)C1)=O C1(C(=O)NCC2(C)N(C(c3cc(C)sn3)=O)CCC2)CCc2ccnn2C1 c1(N(CCOC)CCNC(=O)CCN2C(=O)CCC2=O)nccc(C)c1[N+](=O)[O-] c1(NC(C2C3CC2N(C(c2ccc(Br)c(F)c2)=O)C3)=O)ncc(Cl)cc1O c1(C(=O)NCC2CCN(C(=O)Cc3ccc(Cl)cc3F)C2)ccc(Cl)c(Br)c1 c1(C(=O)NC2C(NC(C3CCN(C)C3=O)=O)COC2)cc(F)c2ccccc2c1 N1(C(C(C=C)(C)C)=O)CC(CC(=O)NC2CN(C)CC2C)C2(CC2)C1 C1(NC(COC)=O)CCN(C(c2cc(Br)sc2Cl)=O)C(C)C1 O=C(C1=CC2CCCC12)Nc1ccc(C(=O)OCc2cc(F)cc(F)c2)c(Cl)c1 C(=O)(CCCCCS(N)(=O)=O)NCC1CN(C(c2ccc(OC(C)C)nc2)=O)C1 C(=O)(CC(O)CC(C)(C)C)N1CC2N(C(c3n(CC)ncn3)=O)C(CC2)C1 C(C(C)(C)CC(C)O)NC(C1CN(C(C2(CC=C)CCCC2)=O)CC1F)=O N1(C(C(=O)NC(c2c(Cl)nn(C)c2Cl)C)C)Cc2ccccc2C1CCO CCCCC(CC)CC(=O)NC(CCC)C(O)C(=O)Nc1ccc(OC)cc1F N1(C(C2C(C)OC(C)C2C)=O)CCC(NC(=O)CCCCCO)C2(CCC2)C1 C1(NC(=O)CC(=O)OC(C)(C)C)COCCN(C(CC2CCCC(OC)C2)=O)C1 N1(C(C(CC)SC)=O)CCCC1(CNC(=O)C(C)(C)c1cccnc1)COC C12(CNC(=O)CC3=CCCC3)CCCCC1N(C(=O)COc1ccccc1)CC2 N1(C(C2CC(=C)C2)=O)CCC(O)C(NC(c2c[nH]nc2-c2ccoc2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CC(CNC(c2cnc(SC)s2)=O)CC1(C)C N1(C(C2CCC3(CC3)C2)=O)CCCCC2(C1)CN(C(C1CCCCO1)=O)C2 C1(NC(=O)C(F)CC2CCCC2)CS(=O)(=O)C2CN(C(=O)Cc3ccco3)CC12 Cc1cc(C(N2CCC(CN(C(=O)COCCCF)C)CC2)=O)c(C)nc1C c1(CNCC(C)C2CNC2)ccccc1CNS(C)(=O)=O CCC(C)C(O)CC(=O)NC1(C(=O)NC2CN(C(C)C)CC2C)CCCC1 c1(C(N2CCC(N(C(C=CC(CC)C)=O)C)CC2)=O)ccc(Cl)c(F)c1 C(=O)(CCCCC(F)F)N1CC(F)(CNC(C2(C)N(C)CC(OC)C2)=O)C1 c1(C(N2CC3C(N(C)C(C4CCS(=O)(=O)N4C)=O)C3C2)=O)cc(O)cc(C#N)c1 C1(CC(N2C(C)CN(C(=O)CCc3nncn3C)CC2)=O)CC2(CCCC2)CO1 C(=O)(CCCS(N)(=O)=O)NC1CCC(NC(C(C)Cc2ccncc2)=O)CC1 C1(NC(c2c(OC)csc2)=O)COC2(C1)CN(C(=O)C(C)(O)c1ccccc1)C2 C12(C(=O)NCC(C)CN(C)C(c3cc(F)cnc3O)=O)CCCC1CC(=O)CC2 c1(CC(N2C(COC)CN(C(=O)CCC(=O)NC)CC2)=O)nnc2n1CCCC2 C1(C(=O)Nc2cc(OC)n[nH]2)CCCCN1Cc1cnc(C)cn1 C(C(N)=O)(C(C)CC)N.n1(CC#C)ccc(-c2nccn2C(C)C)c1 Cc1n[nH]c(C)c1C(C)C(=O)N(CC(C)NC(c1ncccc1C(F)F)=O)C C1(C(=O)NC2CCC(CNC(c3scnc3C3CC3)=O)C2)C(F)(F)C12CCC2 N1(C(c2cccc(N(C)C)c2)=O)CC2CC1CC2NC(c1cc(O)cc(Cl)c1)=O C1(C(=O)NCC2C(OC)CC2)CC(c2ccccc2)(NC(C2CC23CCC3)=O)C1 C=C1CCC(C(N2CC3CC3(CNC(=O)C(C)Nc3nc(C)cs3)C2)=O)CC1 C1(C(=O)NC2CC2(F)F)COC2(CCN(C(c3ccncc3Br)=O)CC2)C1 c1(C(=O)NC2(CNC(C)=O)CCCC2)c(F)c(F)cc(F)c1F C1(C(=O)NCC2CCN2C(=O)CN(C(=O)C(C)C)C)(SC)CCC1 C(=O)(C(=O)NOC)NC(c1ccccc1)C(=O)NC1(C=C)CCC1 c1(C(=O)NCC(C2CCN(C(=O)CN3CSCC3=O)CC2)(C)C)ccncc1Cl N1(C(C=CCNC(c2cscn2)=O)=O)CCC(n2cncn2)C1 C1(C(=O)OCC(=O)N(CC#N)Cc2cccc(Br)c2)COC2(CCC2)C1 CCCC(C(=O)NC(C)(CNC(C1(F)CCCCC1)=O)CO)c1ccc(Cl)cc1 c1(-c2n(C(COC)C)nc(-c3ccc(N)cn3)n2)cnn2c(N(C)C)ccnc12 c1(C(C)C)cc(C(=O)NCC(C)(C(C)C)NC(=O)CCc2cocn2)cc(O)n1 CC1(C)CC(C)(C(=O)NC2CC=CCC2)CN1C(c1ccc2[nH]ccc2c1)=O Cc1cccc(C(=O)NC(C)(C)CCNC(=O)C(C)CSc2ccccc2)c1F C(C(C(=O)Nc1cnn(C)c1)NC(C1CC(N(C)CC)C1)=O)SCC C(=O)(C(C)CC(C)(C)C)NC1(C2N(C(CCc3cc(C)no3)=O)CCCC2)CC1 O(NC(=O)CCC(C(C)C)NC(=O)C(CC(C)C)C(C)C)CCOC(C)C c1(CC)nc(C(C)NC(c2nnnn2Cc2ccco2)C2(CC)COC2)cs1 Cc1c(C(=O)NC2CC2NC(=O)C(F)(F)C2(O)CCCC2)cncc1Cl c1(SC)cc(C)c(C(=O)NC(C2CN(C(=O)Cc3cnccc3C)CCO2)C)o1 c1(C(N2C(CC(=O)Nc3c(OCC)cccc3)CC2)=O)ncc(F)cc1N Cc1nnc2n1CCC2(C)C(=O)N(C)C.n1(CC(=O)N2CC2)ncnn1 c1(C(=O)NCC2(NC(CCCC3C(C)C3)=O)CC2)cccnc1F O=C(NNc1ccc(Br)cc1O)c1ccc(CC(=O)N2CCC2)cc1 N1(C(CS(C)(=O)=O)=O)CCCC2(C1)CN(C(C1CC3CC1C3)=O)CCO2 N12CSCC1C2=O.CC(O)(CC(c1ccco1)=O)C1CCNC1 c1(C(N2C(OC)C=CCC2)=O)cc(O)nc2c1CN(C(=O)C(C)CC1CC1)CC2 N1(CC)CC(C(=O)NCCCNC(C2CCCN(C(=O)OC(C)C)C2)=O)NC1=O CC(CC(=O)NC(C)CN(C)C(c1ccnc(Cl)c1)=O)C(F)F CC(C)CCCC(=O)NC(CCN(C(=O)CC1CC1(C)C)C)C(C)C N1(C(=O)COC(F)F)CCN(C(c2ccc(CO)nc2)=O)C(C2CC2)C1 N1(C(C2CCCC(=O)O2)=O)CC(NC(=O)C=Cc2cncnc2O)CC2(CC2)C1 c1(C(=O)NCC(CC(C)C)NC(C2CNC(=O)N2C)=O)c(O)cccc1Cl C(C(=O)N=c1cc(C)o[nH]1)N1CCCC(CN(C(CC(C=C)CC)=O)C2CC2)C1 c1(C(N(C)CC2N(C(C(N3CCCC(O)C3)C)=O)CCC2)=O)nc(Cl)c(Cl)s1 c1(OC)cc(C(=O)NC2CCN(C(=O)C(C)(C)CF)CC2CO)c(Cl)cc1Cl c1(CNC(=O)NC2N(C(CN(CCCN(C)C)C)=O)CCC2)sc(Br)cc1Br c1(CC(=O)Nc2cc(=O)oc3cc(O)ccc23)cc(S(=O)(=O)N2CCCC2)ccc1Cl N1(C(CC(CC)C(F)F)=O)CC(NC(c2ccc(=O)oc2)=O)CC12CCOCC2 C1(c2n(-c3c(C)cccc3)nnn2)(N(c2ccc(Br)nc2)C2CC2)CCCCCC1 C1(COC(C)C(=O)NCCNS(=O)(=O)C2CC2)(CO)CCN(C(C2CC2)=O)CC1 c1(C(N2CCC(NC(c3c(C)nn(C)c3)=O)C2)=O)ccc(=O)n(C(C)C)c1 c1(C(N2C(C)C(O)CC2)=O)cc(O)nc2c1CN(C(C1CCN(C)C1C)=O)CC2 Cc1ncnc(C)c1CC(=O)NC(C)CCCCNC(C1CC1c1cnc[nH]1)=O N1(CCC)CCCC1C(N1CCC(C(=O)NCc2cccs2)C1)=O C1(NC(C(C)OCCC=C)=O)CC2(C1)CC(C(=O)NC1CCN(C)C1C)C2 C1(C(=O)Nc2cccc(COC)c2)N(C(=O)CCc2cccs2)CCC1(C)C C(=O)(C(CC)C(C)(C)CC)N1CCN(C(c2cn(CCOC)nc2)=O)CC(O)C1 C1(CC(=O)NC)CN(C(c2conc2C)=O)CCN1C(=O)C(=O)NC(C)C CC1(C)CN(C(=O)CNC2CCCC2)C1C1CCCO1 CCCCCC(O)CC(=O)NC1CCN(C(=O)C#CC(=O)N(C)C)C12CC2 C1(CC)CN(C(C2CC(=O)N(C)C2)=O)CC1NC(c1cccc(OC2CC2)c1)=O CC1(NC(c2cccc(OCC3CCCO3)c2)=O)CCCN(C(=O)CCC#N)C1 N1(C(C(C2CCOCC2)OC)=O)CCOCC(NC(c2cccc(CO)c2C)=O)C1 Cc1nnc2cc(NCC3CCC(NC(c4cccc5nncn45)=O)C3)ncn12 CCCCCC(C)CC(=O)NCC#CC(=O)Nc1cccc(CO)c1 CC1CCC(CNC(=O)CCCCC2CC2)CN1C(=O)CCc1cocn1 C1(C(N(C)Cc2c[nH]ccc2=O)=O)CN(C(=O)CC2CC(=O)NC2=O)CCO1 N1(C(c2cnn(C)c2Cl)=O)CCC2(CCN(C(C3CC(=O)CCO3)=O)C2)C1 CC(F)(F)CCC(=O)N1CCC(N2CCN(C(=O)Cc3ccsn3)CC2)CC1 c1(C(N2CCC(NC(C(C)C3CC3)=O)C2)=O)ccc2c(c1)OCCO2 C1(O)(CN(C)C(C2CC(=O)CN2C(C2(C)CCCO2)=O)=O)CCCCC1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(CNC(c2cncc(OC(C)C)c2)=O)C1 O=C1CCN(CC(=O)OCC2CC3(CCC3)C2)C(=O)C(CC(F)(F)F)N1 C1(C(=O)NCC2CN(C(Cc3c(C)ncs3)=O)C(C)C2)CCc2n[nH]cc2C1 C(CN=c1cccn[nH]1)NC(N1CCC(n2ccnn2)C1)=O N1(C(CCS(C)=O)=O)C2CCCC1CN(C(=O)CCC1CCC(=O)NC1)C2 c1(N2C(C)CN(C(c3cccc(=O)n3O)=O)CC(C)C2)ncnc2c1SCCC2 Cc1ocnc1C(N1CCC1CNC(c1cn(-c2ccn(C)n2)cn1)=O)=O N1(C(CCCC)=O)C2CCC1C(F)C(NC(C1CCSC1)=O)C2 C1(C(N(CC(O)CNC(=O)CCc2ccon2)C)=O)CC(C)(C)SC(C)(C)C1 c1(N(C)CC2CCN(C(=O)COc3ccsn3)C2)ncc(S(C)(=O)=O)cc1Cl C=CC(CCC)CC(=O)N1CC2(CC2)CC1CNC(c1cc(F)ccc1CC)=O n1(CC(C)NC(C2(C(F)F)CCCO2)=O)cc(CCC2CCCCO2)nn1 c1(CNC(C(=O)NC2C(C)CCC2)=O)ccc(NC2CC=CCC2)cc1 c1(C(C)NC(=O)NC(CCN(C)C)C(F)(F)F)ccc2c(c1)CCC2 N1(C(C2(C#C)CCC2)=O)CC(NC(=O)CCc2cc(C)cc(C)c2)C2(CC2)C1 c1(C(CC(=O)OCCCCC(=O)N(C2CCC2)C)N)ccc(C(F)(F)F)cc1 C1(C(=O)NC(C2CCN(C(c3ccoc3)=O)C2)C)C2CCC3(COC(=O)C13)O2 N1(C(C2CC(OCC)C2)=O)CCCC1c1cn(C2CC(O)C2)nn1 N1(C(CNS(CC)(=O)=O)=O)CC2CC1CN(C(C1CCC(C(N)=O)CC1)=O)C2 N1(C(C2CCC(C(=O)OC)CC2)=O)CCCC(F)(F)C1O C(=O)(C(CCC)OC)N1CCC(C(C(=O)NC(C=C)(C)CC)(C)C)C1 Cn1nc(Br)cc1C(=O)NCC1CCCC1NC(=O)CCC1CCC1 N1(C(CCOCCNC(C(COCC)N=[N+]=[N-])=O)=O)CC=CC12CCOCC2 c1(C(=O)NC(CCNC(CC(CC)OC)=O)C(C)C)cc(F)c2[nH]nnc2c1 C(CCC(=O)NC1(CNC(c2ccc(CN(C)C)s2)=O)CCOC1)=C(C)C C(=O)(C#CC1CCCOC1)NCC(C)(CNC(=O)CC(Cl)Cl)OC C1(CC(=O)NCc2c(C(=O)NCc3onc(C)n3)cco2)CCCC(=O)N1 N1(C(C2(F)C(C)C2)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C(F)(F)CC1 C12(C(=O)NC(C34CCC(CO3)C4)C)COC(C1)C(NC(=O)C#CC1CCC1)C2 C1(OC)CN(C(c2cc(Br)c3[nH]c(C)nc3c2)=O)CC12CCOCC2 c1(C(N2CCC(F)(CNC(C3(C)C(C)C3)=O)C2)=O)ccc2c(c1)CC(C)(C)C2 c1(C(N2C(CNC(C(C)NC(C)(C)C)=O)CC2)=O)c2n(c(=O)n1C)CCCC2 Cc1ccc(C)c(C(=O)NC(C)C(C)NC(c2nn(C)c(C)c2Cl)=O)c1N N1(C(c2cn(C)nc2O)=O)CC(NC(C2C=CCS2)=O)CC2(CCC2)C1 c1(CC)cc(C(=O)NCCCN(CCO)C(c2cnsc2)=O)ccc1C C1(NC(c2sccc2-n2cccc2)=O)COC2CN(C(c3ccnnc3)=O)CC12 C(=O)(CCC(C)N(C)C)NC(C1N(C(C(=O)NCC)=O)CCC1)C c1(CC)noc(CC)c1CC(=O)NCC1CCCC(NC(=O)C(C)(CO)OC)C1 C1(O)(CNC(C2C(C)(COC)C2)=O)CCN(C(c2cnc(C3CC3)s2)=O)CC1 c1(C(N2C(C)(CNC(c3cc(CF)on3)=O)CCC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nn(-c2ccccc2)cc1NC(C1(N2CCOCC2)CCCC1)=O C1(C(=O)NC2C=CC(C(N3CC(CSC)C3)=O)C2)CC12CCOCC2 C(=O)(CCCCC(C)(C)C)N1CC2C(C(=O)NC(C)C(=O)NO)(CCC2)C1 N1(C(c2c(CSC)cccn2)=O)CC2CCN(C(C3CC(SC)C3)=O)CC2C1 c1(OC)ccc(-c2cn(CCNC(=O)Cc3cccc(Cl)c3Cl)nn2)cc1F C(=O)(C(C)(C)c1cncnc1)N(CCC(=O)O)CCCC(c1ccccn1)O CC1COC(C)(C)CN1C(c1cc(O)nc2c1CCC2)=O N1(C(C(CC)(CNC(c2ccc(N)cn2)=O)CC)=O)Cc2ccc(C)nc2C1 N1(C(C(C)OCCCCCC)=O)CCCCC1CNC(=O)C(C)CC C(c1cncc(C(F)(F)F)c1)=CC(N1C(C)CCC1C(=O)Nc1ccccn1)=O C1(NCCc2cccc(C(F)(F)F)c2)CCC2CNCC2C1 c1(C(N(C)CC2CCN(C(=O)Cn3cccn3)CC2)=O)cc([N+](=O)[O-])cnc1O CCC(F)C(=O)N1CCC(N(C(=O)CCC=CCC=C)CC)C1 C1(C(=O)NCC(CC)NC(=O)COCC2(F)CC2)CCC(C(C)(C)C)CC1 c1(NC(C(=O)N(C2CCOCC2)C(C)C(C)n2cccn2)=O)ccc2nccn2c1 Cc1oc(C(=O)NC2CCC2CNC(=O)C(N2CCCC(O)C2)C)cc1CO C(=O)(C(C(=O)N1CCCC(NC(c2cc(C(C)(F)F)on2)=O)C1)C(C)C)OCC N1(C(C2(C)COC2)=O)CCC2(CCCN(C(c3cc4ccnc(Cl)c4s3)=O)C2)C1 c1(C(N2CC3(CC(NC(=O)CC4CS(=O)(=O)C4)C3)C2)=O)noc2cc(Cl)ccc12 c1(OC)c(C(=O)N(CCCCN(C)C(C2CCCC(C)O2)=O)C)nc(O)nc1O N1(C(c2c(COC)ccs2)=O)CC2CCN(C(=O)Cc3cscn3)CC12 c1(CCNC(=O)NC2CCCC2n2cccn2)cccc(F)c1 c1(SCNC(C)CCN=[N+]=[N-])ccc(S(N)(=O)=O)c(C)c1 CC1(C)CCCC(C(=O)NC2CCCCC2CNC(=O)C=CCN2CCC2)C1 c1(OC)ccc(F)c(C(N2CCCC2CNC(c2cncn2C2CC2)=O)=O)c1 C(CC(=O)NOC1CCC1)C1CN(C(CN(C(=O)OCC)C)=O)C1 Cc1cc(F)c(C(=O)NC(C2CCOC2)CNC(=O)CC(C)(C)C)cc1F C1(OC)CC(CNC(=O)Cc2ccc(C(=O)O)cc2)C1(C)C C#CC1(C(=O)NC2C3CC2N(C(=O)CC2OCCCO2)C3)CC(F)(F)C1 C1(O)(CN(C(=O)COC(F)(F)F)C)CCCN(C(=O)C(=O)N(C)C)C1 c1(C(C(=O)NCC2CCN(C(C(CC)F)=O)C23CC3)=O)c[nH]c2ccccc12 CC(C)CC(O)C(=O)N1CCN(CCCNC(c2cc(Cl)no2)=O)CC1 n1(CC)c(C(N2CCNCC2C(=O)O)=O)cc2ccccc12 c1(C(=O)NC2CCN(C(c3c(C)cns3)=O)CC2F)cc(S(C)(=O)=O)c(C)o1 C(=O)(C(O)CCCNC(C1(C#N)CC1)=O)NC(C)(C)C(N)=O c1(OC)ccc(C(=O)NCCN(C(=O)C(CCSC)NC(C)=O)C(C)C)cc1C N#Cc1ccncc1C(=O)NCC1OCCC1C(=O)N(CCCO)CCCO c1(OC)cncc(C=CC(=O)N(CCNC(c2ccc(F)c(Cl)c2)=O)C(C)C)c1 N1(C(C(C)n2ccnc2)=O)CCOC(C(=O)Nc2ccc(F)cc2)CC1 C(=O)(CCN=C(NCc1cccc(SC)c1)NC1CCOC(C)(C)C1)NC N1(C(C(=O)NCCOC)=O)CCN(C(=O)CCc2cnco2)CC1C1CC1 C(=O)(C1=CCC(NC(c2cc[nH]c2)=O)C1)NCCC1C(C)CCO1 CC(C(=O)NNc1ccc(Br)c(F)c1F)OCC1CCCO1 c1(CN(C)CCc2nccs2)nc(-c2ccc(Cl)cc2)sc1-c1ccc(=N)[nH]c1 CCCCCC(=O)N1CC(NC(c2csc(-c3cccc(C)n3)n2)=O)C(C)C1 c1(C(=O)NCCC(C(N2CCCC(C)(O)CC2)=O)OC)ncc2ccccn12 c1(SC)ccc(CCCC(=O)NC2C3CC2N(C(C2CCC(=O)O2)=O)C3)cc1 C1(C(=O)NC(C)(C)CNC(=O)C=C2CCCCC2)(CC)CCC(F)(F)CC1 CC1(O)CCCC(C(N2CCC(CCNC(=O)CC3CN4CCN3CC4)C2)=O)C1 c1(CNC(C2(CCNC(COC)=O)CC2)=O)cccc(CO)c1.c1nc[nH]n1 C(CC(C(C)(C)C)NC(c1cccc(C(F)F)n1)=O)N(C)C(c1cnn(C)n1)=O CC(C)CC(C(=O)N1CC2CC2C2CC12)ONC(=O)CC1C=NN(C)C1=O c1(C(=O)NC(CC(C)NC(C=CC(C)(C)SC)=O)C)c(C)cncc1C c1(C(N2CCC(N(C(=O)C3=CC(C)(C)C3)CC)C2)=O)ccc(CO)c(F)c1 C1(C)(C(=O)NC(C2CCCN2C(=O)Cc2cn[nH]c2)C)CC1(C)C c1(NC(CNC(c2c(C)nc(CC3CC3)o2)=O)C)cc(C#N)c(F)cc1[N+](=O)[O-] Cc1c(NC(c2nc(-c3ccccc3)oc2C(C)C)=O)cnn1CCO C1(C(N2CCC(O)(C(C)NC(CSC)=O)C2)=O)CCC(O)CN1C C(=O)(CC(C)(C)C#N)NC1CCCC(N(C)C(c2ccc(Br)s2)=O)C1 c12ncc(cn1)-c1csc(n1)NC(=O)N2.CC(=O)NCCN(C)C N1(C(C2C(NC(c3scc(OC)c3)=O)CCO2)=O)CCOC(CC(N)=O)C1 c1(OC)cc(OC)cc(CN2CCC(C)(C(=O)Nc3cc(F)cc(Br)c3)C2)c1 N1(C(C(CCSC)NC(C)=O)=O)CCC2CCN(C(=O)C3=CCCC3C)CC12 CC(C)C(=O)CCCN1CCN(C2CCCCC2)CC1 c1(C(=O)NCC2(C)CCN(C(c3c(C)cccn3)=O)CC2)cc2n(n1)CCCO2 C(=O)(C#CC1CCC1)N1CCC(C(C)NC(c2ccn(CC)n2)=O)C1 C(=O)(N=c1[nH]nc(C(C)(C)CN(C)C)s1)N1C(C)CC(O)C1 c1(CN(c2ccccc2)C(=O)NC2CCCC(COC)C2)ccnc(C)c1Cl c1(C(=O)OC)cc2c(c(S(=O)(=O)Nc3cccc(N4CCCC4=O)c3)c1)CCC2 CCC(C)C(C(=O)N(C(C)(C(=O)NC1CC1CC(C)C)C1CC1)C)N(C)C c1(N2C(C(N3CC4CCC(C3)O4)=O)CCC2)ncc(Br)cc1Br Cc1cc(Cl)c(C(=O)NC(C2CCCCN2C(c2cc(F)cs2)=O)C)cc1N C1(C(N(C2(C(=O)OC)CC2)C)=O)CC12CCN(C(=O)C(C)CC(N)=O)CC2 C(=O)(CC1CCCc2ccccc21)NC(C(CCCCC)(O)CC)C c1(C(=O)NC2C(NC(=O)C3=CCCOC3)CCCC2)ccc2c(c1)COCCN2 N1(C(CC2C(OCC)COCC2)=O)CC2CC(N(c3ccc(F)cc3)C)C1C2 C1(C)(C(C)C)CC1C(=O)N(CCNC(=O)Cc1cc[nH]c1)CCOCCO C1(CCC)CN(C(c2cc(C(=O)OC)cs2)=O)CCN1C(c1cccnc1Cl)=O N1(C(C(COCC)C)=O)CCCC(O)(CNC(C2(C)CCC(F)(F)CC2)=O)CC1 c1(C(CNC(=O)NC2CC3(C2)CC3F)(F)F)ccccc1F C(=O)(CCC(C)(C)NC(c1cn(C)c(=O)n1C)=O)NCc1c(C)nn(C)c1 CCC(CC(=O)NC1CN(C(C2CNC(=O)N2)=O)C1)C1CC1 C(=O)(C#CC1CCCOC1)NC1CCCCN(C(C(c2cccs2)SC)=O)C1 Nc1cc([N+](=O)[O-])ccc1C(=O)NC1CC(CNC(c2nsnc2O)=O)C1 N1(C(=O)CC2CC3CCC2C3)CC2CN(C(C3(Br)CC3)=O)CC(C1)O2 C#Cc1ccc(C(N2CCC(C=CC(N3CCC(C(N)=O)C3)=O)CC2)=O)cn1 C(=O)(C1CCCc2ncccc21)NC12C(CN(C(c3c(C)nn(C)c3Cl)=O)C1)C2 c1(C(N2CC(NC(C=CC(CC)=CC)=O)C3C2C3)=O)ccc2nncn2c1 Cc1c(NC(c2cc3c(F)c(Br)ccc3s2)=O)ccc(Cl)c1[N+](=O)[O-] CCCCC(CCCC)C(=O)N1CC(NC(=O)CCSc2nccn2C)C(C)C1 C1(N(C(c2c(CC)c[nH]n2)=O)C)CCC(NC(=O)CC2CCC3CC23)CC1 S(=O)(=O)(c1ccc2c(c1)CN(CC1CC(C)(C)C13CCC3)C2)N(C)C Cc1nc(N(CCCS(N)(=O)=O)CCO)cc(C(F)F)n1 C12(CNC(c3c(N(C)C)cccc3)=O)CCCOC1CCN(C(=O)C(F)Br)C2 C(=O)(N=c1ncnc2[nH][nH]c(C)c1-2)C1C(NC(c2cc(C)cc(C)n2)=O)C1 N1(C(CCSCCC)=O)CC2CCC2(CCNC(c2nccnc2C(N)=O)=O)C1 C1(C(=O)NC2(COC)CN(C(C)=O)C2)CCN(C(=O)C(C)N(C)C)CC1C c1(C(N(CC(=O)NCc2c(C)nc(C)s2)C)=O)ccc(C)c(O)c1 n1(CCC(=O)N(CCC(=O)O)CC(C)C)ccc(O)nc1=O c1(C(N2CCCC2CF)C(=O)NCCN2CCC(O)C2)cc(Cl)cc(Cl)c1Cl C1(C)(NC(C2CN(C(C)C)C2)=O)CCN(C(=O)C(C(C)C)c2ccccc2)CC1 c1(C(=O)NCC(CCCC)NC(=O)C(C)=C2CCC2)ccc(OCCF)cc1F c1(C(=O)NCCCNC(=O)C(F)Cc2ccccc2)cnc2[nH]nnc2c1 C1(C(=O)NC2C(CCOC)CCC2)CC(O)CN1C(=O)C=C1CCOCC1 C=CCCCCCC(=O)NC1CCN(C(=O)COC2(C)CCC2)CC1F c1(C(N2C(C)CC(c3ccccc3)C2)=O)cc2cccc(Br)c2cn1 c1(C(=O)NC2CCCC(C(=O)Nc3cnoc3)C2)cc(F)cc([N+](=O)[O-])c1 c1(C(CC2CC3CN2C3=O)=O)cc(C)nc2ncnn12.c1(C(=O)OC)cscc1F N1(C(COC(C)=O)=O)CCC2(NC(=O)Cc3ccc(F)cc3Cl)CCCCCC12 CCC(CC(=O)N1CC2C(CNC(c3cncc4c[nH]nc34)=O)C2C1)C(C)C N1(C(C=C(C)C2CC2)=O)CCC(C)(C)C1CC(N1CCCC1)=O N1(C(C)=O)CCC2(CCC(C(F)(F)F)N2C(=O)C(C)NC(=S)SCC(F)(F)F)CC1 n1(CC(=O)OC)cc(NC(=O)CC2CC(C(F)(F)F)C2)c(C)n1 C1(C(N2CC(CCNC(c3cc(C)oc3)=O)OCC2)=O)CN(S(N)(=O)=O)C1 c1(CCNC(C(CN(C)C)NC(=O)Cc2ccn(C)n2)=O)cccnc1O N1(C(C(Cc2ccccc2)OC)=O)C2CCC1CC(NC(=O)CC1(C)CCC1)C2 c1(SCC)cc(F)c(S(=O)(=O)Nc2cccc(C(=O)OC)c2)c(F)c1 Cc1cc2c(cc1NCCSCCSCCO)CCO2 N1(C(c2c(C)ccnn2)=O)CCCC(CO)(NC(c2cccs2)=O)C1 Cc1noc2ncc(C(=O)NC3CC(O)(CNC(=O)C=C4CCC4)C3)cc12 C1(NC(=O)CSc2nc[nH]n2)CC(CO)N(C(=O)CCc2ncc[nH]2)C1 C1(C(=O)NC(c2n(CC)ncc2)C)CN(C(=O)CCP(C)(C)=O)CCC1O Cc1nnc(CNC(c2ccncc2)C2CCOC2)n1C O=S(=O)(c1ccc(N2Cc3cnn(CCO)c3C2)cc1Br)NCc1cc(Br)no1 c1(NC(C)CCC(F)(F)F)ccc(S(=O)(=O)NCC2(C)CCCOC2)cc1C#N N#CC1(C(=O)NCC(O)CNC(C2CC23CCCCC3)=O)CCSCC1 c1(OC)ccc(C(=O)NCC2C3CN(C(C4(F)CC4)=O)CC23)c(OC(F)F)c1Cl C(=O)(C(C#N)C(C)C)N1CCC(CC#C)(C(=O)NCc2cnn(C)c2O)C1 C1(NC(C(C)(C)SC)=O)CCC2(CC1)CCN(C(=O)CCc1cc(F)ccn1)C2 N1(C(=O)CCc2ccc(Cl)s2)CC(C2CN(C(C3CC3F)=O)C2)C1 CCC(COC)C(=O)N1CCC(CC(=O)NC(C)CC(C)CC)CC1 Cc1cc(C(=O)NCC=CCNC(C2CC2c2cccc(Cl)c2)=O)ncn1 CC(C)C(CC(=O)N1CC2C(N(C)C)C2C1)NC(C1CCOC1(C)C)=O C1(CNC(CC2CC(NC)C2(C)C)=O)CC(C)CN(C(c2scc(C)c2C)=O)C1 C1(C(=O)NC2CCCC2C(N)=O)(CNC(CN(C(C)C)C)=O)CCCO1 Cc1cc(O)nnc1C(=O)NCCC1CN(C(C2CCC(C)CC2)=O)CC1C c1(CNC(C(Cn2ccnn2)NC(C(CC)O)=O)=O)cccc(O)n1 N1(CC(=O)N(C(C)C)CC2CCCO2)CCC12CCOC(C)(C)C2 C1(C2CC2)(CNC(CN(CCOC)C)=O)CCN(C(C2(C3CCCO3)CC2)=O)C1 c1(OC)ccc(C(=O)NC(C)CCCNC(C2(C)CCOC(C)C2)=O)cc1C N(C1CC2(CCN(c3ccc(C#N)cn3)C2)Oc2ccccc21)C(C=CSC)=O C(=O)(C(C)CC(N)=O)NC1CC(F)(CNC(c2c(C(C)C)scn2)=O)C1 C1(NC(C(C(C)(C)C)NC(=O)OC)=O)CN(C(c2n[nH]cc2F)=O)CCC1(C)C C1(NC(CONC(c2n(C)ccn2)=O)=O)(CC2(F)CCC2)CCOCC1 c1(C(N(C(CN(C(C2(O)CCC(C)CC2)=O)C)C)C)=O)ncc2ccccn12 C1(C(N(CCC#N)Cc2cccnc2)=O)C2C=CC(C2)C1C(=O)O N1(Cc2cccc(C)c2)CCCC(NC(=O)CNC(=O)CC(C)(C)C)CC1 C1(NC(c2nnn(CC)c2C)=O)CC(NC(c2occc2F)=O)C12CCC2 N1(C(CC=CCNC(C2C(C)CCC2)=O)=O)CCCC2(C=CCO2)C1 c1(CC(N2CCCC2)C)nnc(CCN(C)C)n1CC(c1cccs1)N(C)C C1(C(=O)NCC2N(C(CSc3n(C)ccn3)=O)C3C(C2)C3)CN2CCN1CC2 N1(CC(C)NC(c2cncc3c[nH]nc23)=O)CCc2ccccc2C1=O c1(-n2c(C(=O)NC3CC(CNC(CCOCC#C)=O)C3)cnc2)ccccc1Cl C(=O)(C1CCCc2nncn21)N1CCC(O)(CN(C)C(c2ccc(F)cn2)=O)C1 N1(C(C(CC=CC)CC)=O)CCC2CN(C(=O)C=Cc3sccc3C)CC12 c1(C(N2C(CNC(c3n(CC)ncc3)=O)CCC2)=O)c(Br)cc(F)c(F)c1F CC(CC(=O)N1CCCC1CC(=O)N(C)CC1(C)CC1)C(C)(C)C c1(C(N2CCC(CF)CC2)=O)ccc(CNN(C2CC2(F)F)C2CC2)cc1 C(=O)(CCCCC#N)NCC1(F)CCC(CNC(C(C)Sc2ccccc2)=O)C1 C(=O)(CC(F)(F)C(C)(F)F)N1CC(N(C(=O)C=Cc2cccn2C)C)C2(C1)CC2 C1(CNC(C2(COC)CCCN2C(=O)C(=O)NC2CC2)=O)Cc2ccccc2O1 Cc1cc(C)c(C(N2CC(C(F)(F)F)C(CNC(C3CCCC3)=O)C2)=O)c(=O)o1 Cc1cc(C)c(NC(=O)C(C2CC23CCCCC3)N2CCC(C(N)=O)C2)c(C)c1 N1(C(=O)NCC(=O)Nc2c(C)ccnc2C2CCNCC2)CCC2(CC(C#N)C2)C1 C1(CNC(C(C)=C(C)C)=O)C2CCCC1N(C(c1cnn3c1OCC3)=O)C2 C1(NC(CCC=C(C)C)=O)CC12CCN(C(c1nn(C)cc1N)=O)CC2 CC1Oc2c(F)cccc2C1NC(c1ccc(C#N)cc1Br)=O C1(C(=O)N(C)CCC2CCC2)(SC)CN(C(C2CCCC2O)=O)C1 C1(NC(c2cccc(CC3CC3)c2)=O)CCN(C(=O)CN2CCOC2=O)CC1O C1(C(N2CC(CNC(CN3CC(C)(OC)C3)=O)C2)=O)CC2(CCCC2)C1 CCC1=C(C(=O)NCCOCCCN(C)C(C23CC4CC2C3C4)=O)SCCO1 N1(C(C(CC)OC)=O)CC2C(CN(C(=O)CCC3CCCCC3)C)C2C1 C1(C(N2CC(O)(CNC(c3ccc(N)cn3)=O)C2)=O)Cc2nnsc2S1 c1cc2[nH]c(=NC3CC4CC4C3)nc(N3CC4CCC3CC4)c2s1 c1(CN2CCC(C(C(=O)Nc3nc(C)sc3)C)CC2)cc(F)ccc1[N+](=O)[O-] N1(C(COC(CC)C)=O)CCCC12CCN(C(c1cncc(OC)c1)=O)C2 C1(CC)CN(C(c2c(C)cnn2C)=O)CCN1Cc1ncnn1CC C1(C(=O)NC2CN(C(c3ncn(C)n3)=O)CC2O)CCCCNC1=O C#CCC(C)(C)C(=O)N1CCC1CNC(c1nc(C)ncc1Cl)=O C(=O)(CCCC(C)(C)NC(=O)C1=CCCCC1C)N1C(C(=O)NC)CC(O)C1 C1(NC(=O)Cn2cccn2)CCN(C(=O)CC2CC=CC2)CCC1(F)F C(=O)(C(C)CC(C)(C)C)N1CCCC(O)(CCNC(c2ncc(C)c(Cl)c2)=O)C1 c1(C(=O)NCC2(C)CCOC2)cccnc1CNC(C1CCC(F)C1)=O c1(SC)nc(C)cc(=NCC2(CCNC3CC4CCC3O4)CC2)[nH]1 N1(C(COCCCOC)=O)CCCC(OCC(=O)N(C2CCSCC2)C)C1 C1(CNC(Cc2cc(C)ncc2)=O)C(C2CC2)CCN1C(=O)CC1CCC(C)C1 C1(CN(C)C(c2coc(CO)c2)=O)CCCN(C(C2(C)CNC(=O)N2)=O)C1 c1(CC(=O)N(C2CC3CNC2C3)Cc2ccccc2)ccccc1OCCCF Cc1[nH]nc(C(=O)NCCC2CCN(C(=O)Cc3cc(C4CC4)no3)C2)c1F C(=O)(C(C)(C)C(N)=O)N1C(C2(NC(C3CCN(CCC)C3)=O)CC2)CCC1 C(N=c1[nH]c2c(c(=NC3CCc4cccc(CO)c43)[nH]1)COC2)c1c(C)occ1 C(CCCCC(=O)NC1CCCCC1CNC(c1cc(C#N)oc1C)=O)SC C1(CC(=O)N(CCC(=O)NCC(N)=O)CC=C)CC2CC2C1 c1(C(N2C(CNC(CC3(C)CCOCC3)=O)CCC2)=O)cnn2cccc(Cl)c12 C(CNC(c1n[nH]c(O)n1)=O)(C(=O)NCC(CC1CC1)CO)OC c1(CN=C(NC(COC)C)NCCn2ccnc2)ccc(F)c(O)c1 N1(C(C(CCC)OCC)=O)CC2(CCN2C(=O)CCC2CCC2)C1 N1(CC2C3CC(C)(C3)O2)CCCC2(C1)OCC(O)C2O N1(CC(=O)NCCCC)CC(NC(c2cnsn2)=O)CCC1C CC1CC(C(=O)NCc2cn(CCN3CCSCC3)nn2)CCS1 CC1(C)CNC(=O)c2c(C(=O)NCCNC(C3Cc4cscc4C3)=O)coc2C1 N#Cc1cc(C(=O)NCC2CCN2C(c2nccc(Cl)c2F)=O)n2c1CCCC2 C=CC1OCCCC1N(C(=O)C(=O)NCC1CCN(C(=O)OC(C)(C)C)C1)C CCCCC(CC)CC(=O)N1CCC(C)(C)C(C(=O)NC2CC(O)(CO)C2)C1 CCCCCC=CCC(=O)NCCN(C(=O)C(C)OCC1CCCCO1)C(C)C O=C(CCC(F)(F)Cn1cc(-c2cccnc2)nn1)NC1(C(F)F)CCOCC1 c1(NC(C2(C)CCN2Cc2c(OC(F)F)cccc2Br)=O)cc(Br)c([N+](=O)[O-])cn1 c1(C(N2CCC(C(N)=O)C(C)(C)C2)C(=O)NC)ccc2c(c1)CC(C)O2 Cc1cc(C#N)cc(C)c1C(N1CCCC1CCNC(=O)C(O)c1ccco1)=O c1(C(=O)NCC(CC)NC(=O)C(C)S(C)(=O)=O)coc2c(F)c(Cl)ccc12 c1(C(=O)NC(CCCNC(Cc2ccc(C)cc2F)=O)C)cccc2c1NCC2 CCC(CCCC(=O)NC1CC2CC1C(O)C2O)NC(c1cc(C)nnc1O)=O C(CCCCC(=O)N1CCC(F)CC1C(=O)NCC1CCCCN1C)SC C#Cc1ccc(Cl)c(C(N2CCCC(CN(C(=O)C(C#N)CC)C)C2)=O)c1 n1(CCC(=O)Nc2cnn(C(C)C)c2C2CC2)c(=O)oc2ccccc12 N1(C(c2c(OCC)scc2)=O)CCC(C)(CNC(=O)C(C)NC(C)(C)CC)CC1 N1(COC)CCC(COCC)(NC(C2(NC(=O)CC3CC3(C)C)CC2)=O)C1 N1(C(=O)NC(c2ccc(F)cc2)CCC)CCCC1C1OCCO1 CCCCC(O)C(=O)NC1C2CN(C(=O)Cc3ccc(Br)cc3C)CC12 C1(CNC(C=C(C)C(F)F)=O)CCC(CN(C(=O)C=C2CCCCC2)C)CC1 c1(OC)nc(Cl)ccc1CCC(N1CCCC1(C)Cc1cc(Cl)cc(Cl)c1)=O N1(C(c2ccc(CCCC)cc2)C(=O)NCCCC2CC2)CCOC2CCCC12 Cn1nc(C(=O)NC2CC(C)(C(=O)NCCC(N)=O)C2)cc1CO n1(CC(=O)NCC(C)NC(C2CN(C)CC2C(F)(F)F)=O)nnc2ccccc12 N1(C(c2cc(C)cc(Br)c2)C(=O)NC(C)C(=O)OC)CCC(C2CCOC2)CC1 Cc1cc(NC(c2coc(CNC(c3ccnn3C(C)C)=O)n2)=O)cc(CO)c1 C(=O)(CC(O)C(C)(C)C)NCCC(=O)NC(C)C(c1ccccc1)C C1(CC)C(C(=O)NCCOC2CCN(C(=O)Cc3cn(CC)nn3)C2)CCN1C CC1C(NC(=O)C(F)(F)CO)CC2CCC1N2C(c1cccc(Br)c1)=O CC1C(NC(=O)C(C)(C)C2CCCCO2)CCN1C(=O)CC1CCOC1 CCC(CC)CC(=O)N1CCC(CC(N2CCC(C)C(CC3CC3)C2)=O)C1 N1(C(=O)Cc2ccno2)CCC2CCCN(C(=O)CCC3CCCCCC3)C2C1 C1(C)(NC(COCC=C)=O)CC(NC(c2csc(C(C)(C)C)n2)=O)C1 N1(C(Cc2ccc(C)c(Cl)c2)=O)CCC2CN(C(=O)Cn3cnnc3O)CC2C1 C1(CCO)(NC(CCN(C)CC)=O)CN(C(=O)C(CO)c2ccccc2)C1 C(=O)(C(O)C(C)(C)C)NC1(CC(=O)NCc2ccc(OC)cn2)CCC1 C1(C#N)(C(=O)Nc2cccc(CNC(C(CCC)OC)=O)c2)CC12CCCC2 C1(CC(=O)Nc2cccc(C3CCOCC3)c2)CCCS(=O)(=O)C1 Cc1ccnc(C)c1NC(C1CCC(NC(c2nccnc2Br)=O)CO1)=O CC(C)(C)CCCC(=O)N1CCCC(C(C)(C)C(=O)NCc2ccncc2)C1 C1(C(N2CC3C(n4cc(C=CCC=C)nn4)C3C2)=O)CCCCCS1(=O)=O Cc1ccc(C)c(N(C)C(C(=O)CO)=O)c1.c1(N)ccc(F)c(Cl)c1 N(C(=NCCSC(F)(F)F)NCCn1ncccc1=O)CC1(C)CCCS1 C12CC3(CCN(C3)C1=O)C2.N1(C2CN(C(CC3CC(=C)C3)=O)C2)CCOCC1 CCC(C)C(C)C(=O)NCC1(NC(c2occ(C)c2C)=O)CCCCC1C C(=O)(C1NCCc2cc(Br)ccc21)Nc1c(C)n(-c2ccc(Cl)cc2)nc1 C1(CNC(=O)CCn2cccc2)CC2CCC1N2C(=O)CCOCC(F)(F)F N1(C(C2(C)CC2)=O)CCCC(C2CC2NC(=O)CCCCCn2cnnn2)C1 C12(C(=O)NC3COC3)CCCC1CS(=O)(=O)C2.N12CCC(CC1)OC2=O.CC(C)(C)O C(=O)(CCCCCCBr)N1C(C(=O)NC2CS(=O)(=O)C2)COCC1 C1(CC)CN(C(c2c(CNC(=O)C=Cc3cnccn3)nnn2C)=O)CCO1 C1(C(=O)NC(C2CCOC2)(C)C)COCCC1NC(c1cccc(CC#N)c1)=O c1(C(N2CCC(O)(C(C)NC(CCSCC(C)C)=O)C2)=O)occ2c1CCOC2 c1(CC(N2CC(C(C)NC(c3c(C#C)c[nH]n3)=O)C2)=O)c[nH]c2cnccc12 N1(C(C2(C#C)CCCC2)=O)CCC2(CCC(CNC(C3CC3(Cl)Cl)=O)O2)CC1 N1(C(C(=O)NCCCSCC)C(C)CC(C)C)CCC2(O)CCOCC2C1 CCC(CC(=O)NC1(COC)CCCN(C(c2csnc2OC)=O)C1)C(F)F C(CCCCC(=O)NC1CC1C(F)(F)F)NC(C1C(C)CC1)=O O=C(N=c1cc[nH]cc1)Nc1ccccc1F.c12cc(Cl)ccc1NC2=O CCCCC(CC)C(=O)NCC1(F)CC(CNC(c2cn(C3CC3)nn2)=O)C1 Cc1c(NCCCc2ccsc2)ncnc1N1CCC(CC2CC2)C1 C1(NC(C(C)CC2CCC2)=O)CCC2(CCCN2C(=O)CC(C)(C)C(F)F)CC1 N1(C(c2c(C)ocn2)=O)CCC(C2CCN(C(c3ccnn3CC(F)F)=O)C2)C1 CCCCCCC(C)C(=O)NC1CC(C)(NC(c2cncc(Cl)c2)=O)C1 N1(C(C2CC=CCC2C)C(=O)NC)CCCC(C2CCOCC2)C1 Cc1nnc(C(=O)NC2CCCC2CNC(c2ccc(CO)o2)=O)s1 C1(NS(CC)(=O)=O)CN(C(=O)OC(C)(C)C)C2(CCC2)C1.C1C(=O)N1 CCCC(C#N)C(=O)NC1CCCCN(C(c2cc(C)nn2C2CCC2)=O)C1 N1(C(=O)CCCc2cc(C)sc2C)CCN(C(c2c(OC)cc(C)s2)=O)C2CC12 N1(C(=O)Oc2c(C)cccc2)C2CC1CN(Cc1ccnc(F)c1)C2 c1(SCC(=O)NCCC2(C(=O)NC3CCC(CO)C3)CC2)ccccc1 C1(NC(CC=C(C)C)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 C1(C(N2CC(CCC)N(C(c3csnc3C)=O)CC2)=O)CCCN2CCCCC12 c1(C(=O)NCCC2CCCN(C(=O)C(F)C3CC3)CC2)ccc2nn[nH]c2c1 N1(C(=O)CCOC2CC2)CCCC2(CCN(C(=O)CC3CC4CC4C3)CC2)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)N1CC(NC(=O)NC(C(=O)OCC)C)OCC1 Cc1nc(O)[nH]c1C(=O)N(CC(C)(C)CNC(C1CC(C(C)C)C1)=O)C c1(C(=O)NC(C(C)C)CNC(C2(C3CC3)CC2)=O)ccc2c(c1)OCC2 Cc1cnc(N2CCOC(C(C)NC(c3cc(C4CCC4)on3)=O)C2)nc1O c1(CC(=O)NCC(C)NC(CC2C(C)=NOC2=O)=O)ccc(F)cc1F C(=O)(CCCC(F)F)NCCC(C)(C)NC(C12CC(C(F)F)(C1)C2)=O c1(CC)ccc(F)c(C(=O)N(C)CC2CCN(C(c3conc3CC)=O)CC2)c1 c1(C(=O)NCC(C)NC(C23CC(CC4CC4)(C2)C3)=O)c[nH]nc1C1CCOCC1 N1(C(C2(COCC)CC2)=O)CCC(C(=O)Nc2ccccc2C(C)O)CC1 CC1CN(C(=O)CC2C=CC(NC(c3ccc4[nH]ccc4n3)=O)C2)CC(C)(C)C1 N1(S(C(C)(C)C)(=O)=O)CC2CC1CC2NS(=O)(=O)CC#N C#CCCC(O)C(=O)N1CC(C2CN(C(c3ccc([N+](=O)[O-])n3C)=O)C2)C1 c1(C(=O)NCC(CCC)NC(C2COCCO2)=O)cc(F)cc(F)c1 N1(C(c2c(CC)cccn2)=O)CCN(C(=O)Cc2ccn(C(C)C)n2)CC(O)C1 C#CC1COCCN1C(=O)CCC(CC)NC(=O)CC(C)N(C)C N1(C(c2c(C)cc(F)cn2)=O)CCC(N(C(=O)C=C2CCOCC2)C)C2(CC2)C1 C1(NC(C(Cn2ccnn2)NC(CCC(C)N(C)C)=O)=O)CCCN(C)C1=O C12(C(N3CCC(C(C#C)C)CC3)=O)CCCC1CCN2C(c1sncc1CC)=O N1(C(c2c(C)nccc2)=O)CCC(C)(C)C1C(N1CC(c2cc(O)n[nH]2)C1)=O C1(C)(C(=O)NCC2(NC(CCC(C)(F)F)=O)CCOC2)Cc2ccccc2C1 c1(NCCNC(=O)OCC)ccccc1S(C)=O C1(C(N2CCC(O)(CNC(=O)CCc3cc(Cl)cs3)C2)=O)CC2C(C1)C2(F)F c1(OC)ccc(NC(C2CC(C)CN(C(=O)C(C)N(C)C)C2)=O)c(C(N)=O)c1 c1(OC)ncccc1C(N1CCOCC1C1CCOC1)C(=O)NCCCF C1(C(N2CC3CC(CNC(c4cccnc4S)=O)C3C2)=O)CCc2ncsc2C1 N1(C(C2CCN(CC)CC2)=O)C2CCC1C(C(=O)NC(C)CCCO)C2 C(C)(CC(C(=O)NCCSC)N1CCC(c2cnccn2)C1)CCC(=O)N(C)C c1cn(C)c2ccccc2c1=O.C(=O)(C(C(=O)OC(C)(C)C)OC)OCC C(CCO)(C(C)(C)O)NC(C1C(CNC(c2c(CC)nn[nH]2)=O)CCCC1)=O c1(CC(=O)NC(C2CCN(C(COC(CC)C)=O)C2)(C)C)ccc(F)cc1F Cc1ncncc1NC(C1CCC(NC(=O)Cc2cnn(C)c2)CO1)=O c1(OC)c(F)ccc(F)c1C(=O)NCC1CC1NC(C1(P(C)(C)=O)CC1)=O CC(C(C)(C)C)=CC(=O)NC1CC(NC(=O)C(C)(Cl)Cl)C1 Cc1cc(C)n(C(C)C(=O)N(C(C)C(=O)N(C2CC(C)(C)C2)C)C)n1 CN=c1[nH]cc(C(=O)NC2CCC2NC(=O)CCc2ccccc2OC)s1 C1(N(C(C2CCCC2C(=O)OC)=O)CC)CCN(C(=O)Cc2nnc(C)s2)CC1 CCC(F)(F)CCN=c1nc2scnc2c(NCCCOC2CCCCO2)[nH]1 OC1CN(Cc2cn(-c3c(F)cc(F)cc3F)nn2)CCC12CCC2 C(=O)(CCS(C)(=O)=O)N1CCC(N(CC#C)C(c2ccc(O)nc2)=O)CC1 c1(OCC)ncc(CNCCC(=O)C(C)Nc2cccnc2NC2CC(=O)N2)cn1.N c1(C(CNC(CC2CC(OC)C2)=O)CNC(=O)CN2CC=CC2)ccccc1 n1(CC)ccc(CC(=O)NCCN(C(=O)C(C)OCC(C)C)C(C)C)n1 C1(CCNC(c2cccc(C)c2C)=O)CN(CCON)CCS1(=O)=O N1(C(Cc2cn(CC)nc2)=O)CCCCC(NC(c2nn[nH]c2Cl)=O)C1 C1(C(=O)NC(C2CCCC2)CNC(C2(CC(C)C)CC2)=O)CC=CC1 c1(C(=O)NC2C(C)CCN(C(=O)CCC3CC3)C2)cc(F)c2c(c1)nnn2C C1(OC)CN(C(=O)OC)CCC1O.C12CCN(C1)C2=O C1(C(=O)NC2CN(C(c3ccc(C(N)=O)o3)=O)CC2CO)CCCCC1C1CC1 N1(S(CC(=O)OCC)(=O)=O)CCC(F)(F)C(NC(c2cnn(C(C)C)c2)=O)C1 N1(C(C2=NN(C)C(=O)CC2)=O)CCC(C2CCCN(C(C34CC(F)(C3)C4)=O)C2)C1 C1(C(N(C(CC(=O)N(CC#C)CC2CC2)(C)C)C)=O)CCC(C)=C(C)C1 CC1CN(C)CCCN1C(C1CN(C(c2ccc3c(c2)CC3)=O)CCO1)=O C(C(F)C(=O)NC1(CO)CN(C(C2CCC(CC)O2)=O)C1)N(CC)CC N1(C(=O)NCCC2(C)CCOC2)CCC2(O)CC2C1 c1(CN2CCCC(CNC(c3ccc(OC)cc3)=O)C2)ccc(O)c(C)c1 n1(CCC)cc(Cl)c(C(N2CC(NC(=O)C(C)(C)OC)C2)=O)n1 n1(CCCCSc2nc(O)cc(COC(CSCC)=O)n2)c(C)cccc1=O N1(C(c2cc(Br)cs2)C(=O)NC(C(=O)OC)CC(C)C)CCC(C#N)CC12CC2 C1(CC(=O)NC(C(=O)NCC(F)(F)C(F)F)c2ccco2)CC2(CC2)CO1 C(c1ccc2[nH]ccc2c1)=CC(=O)N(CC(C)NC(CCC(C)OC)=O)C Cc1ccc(C(=O)N(C(C)(C(=O)N(C)CC2CCCCO2)C2CC2)C)c(C)n1 Cn1cc(C=CC(=O)N(C(C2(CC)CCC2)C)C2CC2)cn1.C(C1CC1)=C.OC(F)F Cc1cc(F)ccc1CC(N1CCCC(CNC(C2CC(C(C)C)=NO2)=O)C1)=O C1(CNC(C(C(C)C)(C)C)=O)CN(C(c2ccnc(F)c2N)=O)CCC1(C)C Cc1cccc(OCNC(=O)NCC(C)(C)CSCCl)c1C.C(C)(C)(C)O C(=O)(C(C)S(C)(=O)=O)NC1CCCC(CNC(C2C(CC)C2)=O)C1 O=S1(=O)CC2CN(Cc3ccc(Br)c(Cl)c3F)CC2(C(F)(F)F)C1 CC1CN(C(=O)CC2(O)CCCC2)CC1CC(=O)NC1CC(=C2CC2)C1 CC1CN(C(c2ccc(C(N)=O)o2)=O)CC1NC(=O)C(C)(C)OCC1CC1 CCCCC(CC)CC(=O)NCC1(F)CC(CNC(=O)CC2CCCC23CC3)C1 c1(C(N2CC(COC)(CNC(=O)CN(C)CCO)C2)=O)cnn2c1CCC2 N1(C(C(C=C)C)=O)CCCC(C)(C(=O)Nc2cccc(O)c2)C1 C(CCCCCC(=O)NCCCOC1CCC1)NC(C(C)N(CC)CC)=O c1(N2CCC(C)(OCC)CC2)nc(C)cc(=NCCc2ccncc2C)[nH]1 c1(CC)ncncc1C(C(C(C(=O)N(CC(CNC)O)C)OC)=O)=O.OC C1(NC(C2(CSC)CCOCC2)=O)CCN(C(C2(C)CC2(F)F)=O)CC(C)(C)C1 Cc1nc(O)ccc1C(=O)NCCC(C)N(C)C(c1cccc(CC2CC2)c1)=O N1(C(Cc2n[nH]c(=NC)s2)=O)CCC2C(C1)CN2C(=O)COC1CCOCC1 CCC(C)CC(C(=O)NCC(C)(O)C1CCC1)NC(=O)C(O)C1CCCC1 C1(CCNC(=O)C=Cc2cocn2)CN(C(C2CC(n3ccnc3)C2)=O)CCO1 c1(NC(C2CSC2)C)ccc(S(=O)(=O)NC2CCCN(CCO)C2)c(Br)c1 c1(OC)ccc(-c2cscc2C(=O)NCC(=O)NCC2CCC(C)N2)cc1 Cc1cccc(C(N2CCCC2CNC(=O)CC2OCCCO2)=O)c1F c1(OC)ncc(C(N2CCC(O)C2C(=O)Nc2ccc(I)cc2F)=O)cc1F N1(C(c2cc(N)cc(F)n2)=O)CCCC2CN(C(=O)CC3COCCO3)CC12 N1(CC)CCN(C(c2cc(OC)ccc2O)C(=O)NC)NC1=O.c1(C)ccccc1 C(CS(=O)(=O)c1ccc(CC(=O)OC)cc1)NC1(CCC)CC2NCCC12 C1(C)(COC)COCCN1C(c1cccnc1-c1ccc(F)s1)=O CN1CC(NC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)CC12CCCC2 Cc1cc(O)n2ncnc2c1NC(C1CC(C)(C)SC(C)(C)C1)=O C#Cc1ccc(F)cc1C(=O)NC(CC)(CC)CCNC(C1(COC)CC1)=O N1(C(CCNC(=O)NCC)=O)CCN(CCC(=O)OC)C(=O)C1 c1(C(N2CCN(C(CCC(=C)Br)=O)C(C)C2C)=O)ccc2nc(O)oc2c1 c1(C(C)C)ccc(C(c2nnnn2C2CC2)NCC2(CO)CCC2)cc1 c1(C(N2CCC(N(C(c3c(OC)cccn3)=O)C)C2)=O)ccnc2cc[nH]c12 c1(C(N(C(C)C(N2CCCC2CN(C)C)=O)CCC)=O)ccnc(OC)n1 CCC(C)C(O)C(=O)NC(C)(C)CN(C)C(c1ccc(CSCC#N)cc1)=O c1(NCC(C2CCCC2)NC(=O)CCC2CCCCO2)ncc([N+](=O)[O-])cc1Cl c1(OC(=O)CCNC(C)CCn2cccn2)ccc([N+](=O)[O-])cc1 C1(C)(C(=O)NCCN(C)C(c2cc(OC(F)(F)F)cc(Cl)c2)=O)CCC(=O)NC1 C1(C(=O)NC(C(=O)N(CCCC)C(C)CC)(C)C)COCCC1C c1(C(=O)NCCSC)cc(CNC(c2cc(CSC)cs2)=O)nn1C c1(NC(C2CC(NC(c3ccc(Br)c(Cl)c3)=O)C2)=O)nc(Cl)ccc1O n1(CCCCC(=O)N(CCC(F)F)C2CC2)c(=O)oc2ccccc12 C12(C(C)NC(C3CC(O)CN3C(=O)C(F)Cl)=O)CC3CC(CC(C3)C1)C2 C(=O)(C(C)CCCC(C)C)NC1CN(C(C2N(CC)CCOC2)=O)C(C)(C)C1 C(=O)(C(C)CC(C)C(C)=O)N1C(C(=O)NC2(C#C)CC(F)(F)C2)CC=CC1 c1(C(=O)NC2CC(C)N(C(=O)CCSC(F)(F)F)C2)ccc2oncc2c1 N(C1CCCc2cccnc21)(S(=O)(=O)Cc1ccc(-n2cccn2)cc1)CC N1(C(C(CCSC)OC)=O)CCN(C(c2cncc(N)n2)=O)CC1CO CC(C)C(O)C(=O)NC1CC1CNC(=O)CCc1nnc(C2CCCC2)o1 c1(OC)ccccc1NC(=O)C(c1ccc(C2CC2C)o1)N(C)CC1CC1(C)C N1(C(C2C(C(C)C)C2)=O)CCC(C)C(N(C(=O)C(=Cc2cccc(F)c2)F)C)C1 N1(C(C=C(C)C(C)C)=O)CCOCC(CNC(=O)CC(C)(C)C)C1 c1(C2(C(N3C(C(N)=O)CC(F)C3)=O)CC2)c(Cl)cccc1Cl C=C1CC2CCC(C1)N2C(=O)C(c1cccs1)NC(=O)CC(CC)C(C)C N1(C(c2cc(Br)c(C)s2)C(=O)NC(c2ccccc2)C)CCC(O)C(F)C1 CCCCCC(O)CNC(C12CC(NC(C3C4(CC4)C34CC4)=O)(C1)C2)=O N1(C(C(CC=C)CC)=O)CCCC2(C1)CN(C(C1COCCOC1)=O)C2 C1(N(C(c2cnc(CCC)s2)=O)C)CCN(C(=O)CCCCN(C)C)CC1C c1(C(=O)NC2C(NC(=O)Cc3ccc(Br)cc3F)C2)csc2ccccc12 c1(COC(CCC(C)NC(c2ccccc2)=O)=O)ccc2c(c1)CCCS2 CC(C)(C(=O)NC1(CNC(C2CCNC2=O)=O)CC1)C(O)c1cc(Cl)cc(Cl)c1 C(F)(F)(CN=c1ccc(Br)c(S(=O)(=O)N2CCC(C(N)=O)C2)[nH]1)C1(OC)CCC1 Cc1cc(C(=O)NCC2CCN2C(=O)CCSCC(C)C)nn1C(C)C c1(-c2c(OC)c(F)ncc2)cc2c(s1)CCN(Cc1ncc[nH]1)C2 c1(C(N2C(CN(C)C(C3CC34CCC4)=O)CC(F)C2)=O)ccnc2c1CCC2 C1(C(=O)NC2CCN(C(c3onc(C)n3)C)CC2O)CC2(C1)CC(C)(C)C2 N1(C(c2c(COC)cc[nH]2)=O)CC(NC(=O)C(CCSC)N(C)C)CC12CCC2 C(=O)(C1CC(=O)c2c(F)cccc21)NCC1CCN(C(c2cc(OC)ns2)=O)C1 C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2C3CNC(=O)C23)=O)C1 c1(C(N2C3CN(C(C(COC)C)=O)C(C3)C2)=O)cc(S(C)(=O)=O)cs1 N1(C(C(=O)NC(C)C)=O)CC2CC3CC2C1C3NC(c1cn2sccc2n1)=O C(=O)(C1CCc2ccccc21)NC1CC(C)N(C(=O)C(C)Cc2ccccc2)C1 N1(C(CC(C)(C)C2CC2)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)C2 c1(OC)ccc2c(c1)OCCC2NC(c1ccc(Br)c2c1OCO2)=O N1(C(CN(C(C(C(CC)C)=O)=O)C2CCC2)=O)CCC2(CCOC2)C1 c1(C(=O)NCC2(CCNC(C3CC(CC(F)F)C3)=O)CC2)cc(O)cc(Cl)c1Cl N1(C(C2N(C(C(C)OC3CCCC3)=O)CC(C)C2)=O)CCC2(CCOC2)CC1 c1(C(N(CC#C)C)=O)ccc2c(n1)CN(C(C1CCCCC1O)=O)CC2 Cc1cnc2c(C(=O)N(C3CN(C(c4cc(C#N)cs4)=O)CC3O)C)cnn2c1 N1(C(c2c(CC)nccc2)=O)CC2CCN(C(=O)Cc3ncoc3C)C(C2)C1 C1(CNC(c2ccc(Br)cn2)=O)COCCN1C(=O)CC1C=CCC1 N1(C(=O)NC(C2CC2C2CC2)CC)CC(C)CC1CO N1(C(CCC(C)O)=O)CCCC2(C1)C(NC(=O)CC1(C)CCCC1)CCN2C c1(CC(=O)NCCOC2CCN(C(C(CC)n3cncn3)=O)C2)c(C)noc1Cl C1(F)(C(=O)NC2C(NC(CC3CCCN(C)C3)=O)CC2)CCC(F)(F)CC1 C1(NC(c2c(C)cccc2N)=O)CC2(CCCCN2C(C2CCCC(O)C2)=O)C1 c1(CC)noc(CC)c1CC(=O)OCc1cncc(C(C)C)c1 O=C(C1CCCn2cnnc21)NC1CN(C(c2nc(Cl)ccc2F)=O)C1 Cc1cnc(CC(=O)N(C2CC(C(=O)NCc3[nH]cnc3C)C2)CC2CCCO2)o1 N1(C(C)=O)CCCC2(NC(c3ccc(Br)s3)=O)CCCC12 C1(CNC(CC(CC)(C)C)=O)CC2(CCOCC2)CN1C(C1CC(C#N)C1)=O c1(C(=O)NCC(C)N(C)C(c2ccoc2Cl)=O)ccc(F)c(C#N)c1 C=Cc1ccc(C(N2CC(NC(=O)C3=C(Cl)CCC3)C3CC23)=O)cc1 C1(CCNC(C=Cc2ncc(C)[nH]2)=O)CN(C(c2cscn2)=O)CCCO1 C(=O)(CS(=O)(=O)C1CCCC1)NCC(CO)NC(=O)CCCC1CCC1 CC1=C(C)CN(C(c2sccc2CNC(c2ccn(C(C)C)n2)=O)=O)C1 c1(C(=O)NC2CC(C)(NC(=O)CC3(O)CCCN(C)C3)C2)c[nH]c2cccnc12 C1(C(=O)NC(C(C)SC)C)CCN(C(C2CCCCCC2)=O)C(C)(C)C1 c1(C(N2CC3(CC(NC(C(C#C)(C)C)=O)C3)C2)=O)cc(Br)c2[nH]c(C)nc2c1 c1(CN=C(NCC(COC)F)NC(C)C2CC2)nnc2cccnn12 C(=O)(C1=CC2CCC(C1)C2)N1C(C(N(C)CCc2nccs2)=O)CCCC1 CCCCS(=O)(=O)NC(C)C(=O)NCCNC(c1cc(C(C)(C)C)n(C)n1)=O N1(C(C(=O)NCC2CC(C)OCC2)=O)CCC(C(F)(F)F)C1(C)C c1(N(C)C)ccc(NC(=O)CNC2CCCC2Oc2cccnc2)cc1 C1(N(C(c2cc(COC)no2)=O)C)CN(C(=O)CS(N)(=O)=O)CCC1O N1(C(c2c(C)ccnc2)=O)CCC2CCN(C(=O)C3=CCCCC3)CC2C1 C12(CNC(C(n3c(C)ncc3)C)=O)CCCC1N(C(c1cscn1)=O)CC2 CCCC(O)C(=O)N1CCCC1n1cc(NC(c2cccc(SCC)c2)=O)nn1 C(CN=c1[nH]c(=NCCC(O)c2ccccc2)[nH]c2ccccc12)N(C(C)C)C Cn1ncc2c(NC3C4CCCCCCC34)ncnc12 N1(C(CCC2(C)CC2)=O)CC(NC(=O)Cc2ccc(O)nc2)C2CC2C1 c1(C(N2CCC(NC(C(C=C)O)=O)C2)=O)ccc(-c2ccc(F)cc2)n1C C1(CNC(C2N(C(CCSCCC)=O)CCC2C)=O)CCCC(C)CC1 c1(N2CCN(C(=O)NC)CC2)nc(=NC2CC(F)(CO)C2)[nH]c2c1COC2.C1CC1 c1(CNC(COC)C2CC2)cc(Br)cc2nn(C)cc12 N1(C(CCc2ccn(C)n2)=O)CCCN(C(=O)CCC2CCC(=O)N2)CCC1 C(c1cc2ccccc2o1)=CC(N1CC(C(C)NC(c2c(C)ncn2C)=O)C1)=O c1(C(=O)NCC2CC(C)N(C(C3CCC3)=O)C2)nc2n(c1Br)CCC2 n1(C(CC)C)nnnc1C(c1nccs1)Nc1cnn(CCOC)c1 c1(OC)[nH]c(=NCc2n[nH]c(=N)s2)cc(N)c1F CCCCCC(C)(CC)C(=O)N1CC=CC(NC(=O)CSCCCC)C1 C(=O)(CC(P(C)(C)=O)c1ccccc1)NC(C1N(C(CCC)=O)CCC1)C Cc1ccc2c(CC(=O)NCC(CO)NC(C3(n4cccn4)CC3)=O)coc2c1 C(=O)(C1=CCCOCC1)N(CC(CN(C(=O)CSc1nncn1C)C)O)C Cn1cc2c(CN3CCC(O)C(C(=O)Nc4cccc(Br)c4F)C3)cccc2n1 Cc1cc(CNC(C2CC(n3cc(-c4ncoc4C(=O)O)nn3)C2)=O)sn1 O=C(CN=c1cc[nH]cc1)NC1CCCC(NC(=O)C(F)(F)C2CC2)CC1 Cc1c(C(=O)NC(C2CCCN2C(=O)C(C)NC=O)C)cnn1C(C)C C=C(C)C(C)(O)C(=O)NCC1CCCCN(C(=O)CCC2CCN(C)CC2)C1 c1(NC(c2cc(-c3ccccn3)c[nH]2)=O)cccc(C(F)(F)F)c1 Cc1cc(C(=O)N(C)CC2(O)CN(C(=O)CC3CCCC(C)C3)C2)oc1C(=O)O N1(c2snc(SC)n2)CCC2(CC1)CC(NC(c1cnc3c(cnn3C)c1)=O)C2 c1(C(=O)NC2C(OC)CN(C(=O)C(C)c3cncs3)C2)nn2c(c1C)OCCC2 c1(OC)cc(C(N2CC3CC2C3NC(=O)C(C)=C2CCCC2)=O)ccc1C#N C1(C(=O)NCCNC(=O)NC)CCCN(C(c2ns[nH]c2=O)=O)C1 c1(C(C(=O)NCCN(C(c2nnn(C)c2N)=O)CC)(F)F)cc(F)ccc1OC CCCC(CCCO)C(=O)N1CCC(C)C1CNC(=O)CCCn1ccnc1 C1(C(NOCC(C)C)=O)CC2(CC2)CN1C(c1ccc(=N)[nH]n1)=O N1(C(C(COC)Cl)=O)CCC12CCN(C(c1ccc(Cl)c(Br)c1)=O)CC2 C1(C(=O)NC(c2ccnn2C)CC)CC(=O)CN1C(c1csnc1Cl)=O c1(NC(CC=C)C)[nH]c(=NCC2(OC)CCCOC2)nc2scnc12 C1(CCNC(c2ncn(CC)c2)=O)CC(F)(F)CN1C(C1CC(C(=O)OC)C1)=O c1(CC(=O)NCC2(NC(=O)C(O)CN3CCCC3)CCCC2)cccc(O)c1 C(=O)(CCN(OC)C(=O)C(C)CSC)NC(Cc1cn(CC)nn1)=O N12CCC(CC1)C(=O)Nc1cccc(c1)C2.c1(COCC)cc(CSC)no1 C(=O)(C(C)C1=CCCC1)NC1CCCN(C(Cc2nnc(C)s2)=O)CC1 C(=O)(C1=C(C#N)CCC1)NCC1(OC)CN(C(c2ccc3cncn3c2)=O)C1 C(C)(C)(CC(=O)NCC1CN(C(C2CC2c2nc[nH]n2)=O)CCO1)N(C)C c1(C(N(CCCNC(=O)CC2CC2(Cl)Cl)C(C)C)=O)ccc2c(c1)C(C)CO2 C(=O)(C1=CCCC(C)(C)C1)NCC1COCCN(C(c2c(C)ncnc2)=O)C1 C(CCCC(=O)NC1CCCC(NC(c2n[nH]c(C)c2O)=O)C1)OCC C1(CC(=O)NCC(c2ccccc2)N(C(c2cc(C)[nH]n2)=O)C)SC(=N)NC1=O Cc1ncnc(C)c1C(=O)NC1CCC(C(=O)NC2CCCC3(C2)N=N3)CC1 CC1CCC(CO)N1N1CCN(c2cc(Cl)ccn2)CC1 N1(C(C(CC)CC)=O)CC2CCCC(CNC(=O)C#CC3CCCCC3)C2C1 Cc1nc[nH]c1CC(O)C(=O)NC1COCC1CNC(=O)C=CC(F)(F)F C(=O)(CCCCCCCCCO)N1CCC(NC(C=CC(C)(C)C)=O)C1 C1(NC(CC2N(CC)CCC2)=O)CC2(C1)CC2NC(=O)C(COC)COC C1(C(N2CCN(CC(C)F)CC2)=O)CN(C(=O)CC2=CCCC2)CCN1C c1(C(=O)NC(CN(C)C(C23CC(C2)C3)=O)(C)C)cn(C)nc1Cl C1(OC)CN(C(c2ccccc2F)=O)C(C)(CNC(c2ccc(C)c(C)n2)=O)C1 CC(C)C(C(=O)N1C(CO)CCC1CO)C(C)NC(c1cncc2[nH]ccc12)=O C1(OC)CN(C(c2ccco2)=O)CC1NC(C1CCC(C(F)F)CC1)=O C#Cc1cccc(C(=O)NC(CNC(=O)Cc2ccc(Cl)cc2)C2CCC2)c1C N(C1CCOc2ccc(Br)cc21)S(=O)(=O)c1ccc(Br)cc1F C12(C(N(CC(=O)NCCc3cnn[nH]3)C3CCC3)=O)CCC(CC1)CC2 C1(CC)(CC)CCCN(C(=O)C(=O)NN2CCN(c3ccccc3)C2=O)CC1 Cc1nc(O)ccc1C(=O)N(CC(C)CNC(c1cccc(O)n1)=O)C C(CCC(C)(C)C(=O)NC(C1CCCOC1)CO)NC(C1N(C)CCCCC1)=O C(C(C)NC(c1ccc(OC2CCOCC2)cc1)=O)(C(C)C)NC(C=CSC)=O c1(C(N2C(CNC(=O)CC3C4CCCCC34)CCC2)=O)cc2c(s1)CCOC2 Cc1c(C(=O)NCCCNC(c2cccc(Cl)c2)=O)cc(Br)cc1N Cn1[nH]c(=NC(=O)C(Cn2cncn2)Sc2ccccc2Cl)cc1Cl CC1CCCCC1(C)C(=O)NCC1CC(CNC(=O)Cc2c[nH]nc2O)C1 C1(NC(CC2(C=C)CN(C(C3CCC3(F)F)=O)C2)=O)CCN(C)CC1C#N N1(C(N(c2ccc(COC)cc2)C2CC2)=O)CC2CC1CCC2OCCO c1(CC2(NS(c3ccn(C)n3)(=O)=O)CN3CCC2C3)[nH]nc2c(Cl)cccc12 C=C(C(=O)N1CC2CC1C2CNC(c1c[nH]nc1-c1ccccc1)=O)C(F)(F)F C1(CCNC(C(F)=CC)=O)CCCN(C(c2ccc(Cl)c(C(F)(F)F)n2)=O)CC1 CC(C)(CC(=O)NCC1COC(C)(C)CN1C(c1ccc(N)cn1)=O)C(F)F CC1C(O)CCN1C(C1CN(C(C2C(C#N)C2(C)C)=O)CCO1)=O C1(NC(C2(C)CN(C(C(C)NC(C)=O)=O)C2)=O)CN(C(C)C)CC1C c1(C(=O)NCC(C)N(C)C(c2nn[nH]c2C(F)(F)F)=O)cc2c([nH]1)CCCC2=O Cc1ccc(CCC(=O)NC(C2CCOC2)CNC(=O)CCC#N)c(C)c1 C(=O)(C(CC1CC1)NC(=O)C=CC1CC1)N(CCN=[N+]=[N-])CC Cc1nn(C)cc1CCC(=O)NC(CNC(=O)CN1CC2CC2C1)C(C)C C(=O)(CCCC(C)C)N1CC(CCC)C(C(=O)NCCc2cc[nH]n2)C1 c1(C(N2CCN(C(c3c(CC)sc(=N)[nH]3)=O)C(C)C2)=O)cncc2nc(C)[nH]c12 Cc1cc(N)cc(C(N2CC(C(C)NC(=O)Cc3cccnc3Br)C2)=O)c1F C(C)(CC(F)(F)F)N(C(CCN(C(CCn1c(C)ncc1)=O)C)=O)C N1(C(c2cc(CC)cc(C)n2)=O)CCC2CN(C(C34CC5CC3C4C5O)=O)CC12 C1(C(=O)NC(CCC)CCO)CN(C(=O)C(C)(CO)OC)CC(C)(C)C1 c1(CN(C(CCNC(CC(C)C)=O)=O)CCNC(=O)C(C)SC)cccc(Cl)c1 c1(CN2C(C(N3CCNC(=O)C3)=O)CC(=C)C2)nccc2ccccc12 Cc1nn(C)c(C(=O)NC(C)CNC(=O)C(c2ccc(F)cn2)(F)F)c1[N+](=O)[O-] Cc1cc(C(C)C(=O)NC23CC(NC(=O)Cc4cc(C)on4)(C2)C3)cc(F)c1 C1(C(N(CC(=C)C)CC)=O)CC2CC1CC2NC(=O)CNC(=O)OC C1(C(=O)NCC2(OC)CCCC2)CC(C)(C)CCN1C(=O)C(O)CCSC C1(C(N2CC(C)C(CO)CC2)=O)CC2CN(C(=O)C(C)OC(C)(C)C)CC2C1 N1(C(c2ccc(N(CC)CC)cc2)=O)CC2CCC2(NC(C2CC(O)C2)=O)C1 C1(C(=O)NC2OCCN(C)C2)COCCN(C(c2cc(Br)oc2Br)=O)C1 C1(C(N2CC(SCC)C2)=O)CCCC(NC(c2cc(CO)c(C)o2)=O)C1 C(c1cc[nH]n1)=CC(=O)NC(C(N1CCC(n2ccnc2)C1)=O)c1ccoc1 O=C(C1=C(Cl)CC1)NCC1CCN1C(=O)Cc1cc(Cl)sc1Cl C=CC1(C2(C(=O)NC3CCC(CNC(c4ncncc4Cl)=O)C3)CCC2)CCC1 c1(C(=O)NCCNC(CNS(N(C)C)(=O)=O)=O)cc2c(Cl)cncc2s1 C1(NC(c2c(SC)cnn2C)=O)CCCC(NC(c2cc(C(F)F)no2)=O)CC1 c1(C(N2CCC(C(c3ccccc3)CO)CC2)=O)cc(Br)ccc1Cl CC(C(O)C(F)F)NC(=O)CC1CCCC1NC(c1cc[nH]n1)=O CC1CC(C(=O)N(C)CC2CCCN2C(C2CCOCC2(C)C)=O)CC(C)O1 C(=O)(CC1=NN(C)C(=O)C1)NC(CCC(=O)NC(CC(C)(C)OC)C)C(C)C c1(OC)cccc(COCCNC(N2CCC(OC(=O)C(C)C(C)O)C2)=O)c1 CCC(C)CC(C(=O)NCC(C)(C)CC(F)F)NC(=O)CN1CC(C)(C)C1 C(CCN(C)C(c1ccnc(C(C)(C)O)c1)=O)(C(C)(C)C)NC(CC(C)F)=O c1(C(N2CC(C(C(N3CCC(CC(C)C)C3)=O)OC)C2)=O)cc(O)n(CC)n1 C12(CNC(c3nn(CC)c(C4CC4)c3)=O)CCC1CCN2C(c1ccn(C)n1)=O C1(C(=O)NC2(CC=C)CCN(C(=O)C=CC(=O)N(C)C)C2)CCC2CC2CC1 C1(C)(C(N2CC(OCCNC(c3c(F)ccc(C)c3)=O)C2)=O)CCS(=O)(=O)CC1 c1(C(N2CC3C(CN(C(C4CC(C)C4)=O)C)C3C2)=O)ncc(OCC2CC2)cc1F C(=O)(CC(C)(C)C#N)NC(C)C(C)C(=O)N(CCF)C(C)C C#CCCCC(=O)NCC1(C(C)NC(=O)C(c2ccccc2OC)=O)CC1 CCCCC(C)CCC(=O)N(C(C)C(=O)NCc1nncn1CC)C1CC1 c1(C(=O)OC)c(NCC2CC3CCC2C3)cccc1Cl.C(C)=O c1(C(=O)NC(C(C)NC(C2C(COC)C2)=O)(C)C)oc2ccc(Cl)cc2c1C N=c1[nH]c(Cl)c(Cl)cc1C(=O)NCC(C1CCCC1)NC(=O)C=C1CCC1 C1(OC)CN(C(=O)CC(C)(C)OC)C(C)(CNC(=O)CCn2cnccc2=O)C1 CON(CCC(=O)N1CCCC12CCOC2)C(=O)C1CCOCC1(C)C N1(C(C=CSC)=O)CC(C2CN(C(=O)CC3CCC34CCC4)C2)C1 c1(SCCC(=O)N(C)CCNC(C2CCC2(F)F)=O)ccc(F)cc1 C1(CC(N2CCN(c3nc(C)cc(C)n3)C(C)C2)=O)CCCCCC1(F)F c1(C(N2CCC(N(CCC)C(c3cc(CO)on3)=O)C2)=O)ccnc2c1CCC2 N1(C(CCCSC(=N)N)=O)CCN(C(C2(C3CCCO3)CC2)=O)CC1 c1(C(N2C(CNC(C3C4CCCC(F)(F)C34)=O)CCC2)=O)cc(Cl)c(F)cc1O N1(C(C2(NC(c3c(OC)ccs3)=O)CCCC2)=O)CCCC2(CC2)C1 CC(CCCCNC(C1(O)CCOCC1)=O)NC(=O)C(F)(F)CN(C)C Cc1cc([N+](=O)[O-])ccc1NC(C)CCNC(=O)CCCCO C1(C(C)(C)C)CCCN(C(=O)NCCCNC=O)C1.c1(N)ccc(F)nc1 N1(C(c2cnc(C(C)C)s2)=O)CCN(C(c2cc3n(n2)CCC3)=O)C2CCCC12 C1(NC(c2cc(CC)ncn2)=O)CC2CC(NC(=O)Cc3ccsc3)C2C1 c1(C(=O)NC2CN(C(C(C=C)(C)O)=O)CC2O)cnn2ccncc12 N1(C(C(CCC)O)=O)CCCN(C(=O)Cc2cccc(Cl)c2OCC)CC1C c1(C(=O)NCC(C)(C2CC2)NC(C2CC=C(C)CC2)=O)cc(Cl)cc(Cl)n1 c1(C(N2CCC(NC(C3CC(F)C3)=O)C2)=O)cncc(-c2ccco2)c1 N1(C(C=C(C)C(F)F)=O)CC2(C1)CN(C(c1coc(O)n1)=O)C2 N1(C(C(C2CCN(C(c3c(CC)cco3)=O)C2)F)=O)CCC(F)(CO)C1 C(=O)(CCCC(F)(F)F)N(C)CC1(NC(c2ncncc2F)=O)CC1 O=C(N=c1ccnc2[nH][nH]cc1-2)C1CC2CC2N1C(c1csc(C(F)(F)F)n1)=O CC(C)CCC(C)N(C(=O)C(=O)NCC1CCN(S(C)(=O)=O)C1)C C(=O)(C(F)(F)CCc1ccccc1)NC(C(C)C)(C)CNC(c1c[nH]c(=N)s1)=O c1(CC(N2CCC3(C(NC(CCSCC)=O)C3)C2)=O)c(C)nc(O)nc1O c1(C(N2CCC(CC3CC3)C2)C(=O)NCCSC)cn2c(F)cccc2n1 N1(C(C(C(=C)Cl)(C)C)=O)CCC2CCN(C(c3ccn4c(C)cnc4c3)=O)C2C1 c1(C(=O)OC)cc(C(=O)NCCCCCNC(C2(C3CC3)CCCO2)=O)c(C)[nH]1 c1(OCc2ccc(C#N)s2)c(-c2cccc(Cl)c2)cccc1F c1(OC)ccc(SC(C)C(=O)NCCC2CCCN2C(=O)Cn2ncnn2)cc1 CC(C1=CCN(C)CC1)NC(C1CC2CN(C(=O)C(C)(Cl)Cl)CC2C1)=O CCCCC(C(=O)NC1CCCC1NC(=O)CC1CCCCCC1)C(C)C C(=O)(C1CCCn2ccnc21)N1CCC(OC)(CNC(C2CC3CCC2O3)=O)C1 N1(C(C)=O)CCOC(C(=O)N(C2CCCCC2O)C)CC1 C1(C(=O)OC)CN(C(C2CCOC(C)(C)C2)C(=O)NC2CC(CO)C2)C(C)CO1 S(=O)(=O)(c1ccc2[nH]c(=NCC(F)F)sc2c1)N(CCC(C)O)C Cc1cccc(C2=CCN(C(=O)C(=O)N(C)C(C3CCCC3)C)CC2)c1 C1(CNC(c2c(CC)noc2C)=O)CCCCCN1C(C1CCCOC1)=O C(C(=O)NC(CC(C)C)C(=O)NCC1CCCCCC1)(C(C)(C)C)OC CC(C)CC(C)(C)C(=O)NCC(F)CNC(=O)Cc1ccc2nn[nH]c2c1 C1(F)(CNC(C(=Cc2ccco2)C)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC1 N1(C(C=C(C)C)=O)CCC2(C=CCO2)CC1.n1(C2CC2)ccc(C)n1 C1(O)(CCNC(=O)Cc2ccsc2)CCN(C(=O)CC2CCC(F)(F)C2)C1 c1(NC(C(N2CC(OC)C(c3ccncc3)C2)=O)=O)cc(F)ccc1C C1(OC(C(N2CC=C(C)C2)=O)C)CCN(C(=O)CCN=[N+]=[N-])CC1 c1(CCC(=O)N(C)CC2CCCN(C(C3C(C=C)CC3)=O)C2)c(C)ncnc1O c1(C(N(CCCN(C)C(C2CC2C#N)=O)C)=O)cccc(C2CC(F)(F)C2)c1 CC1CCC(C(N2CCC(N(C(c3ccco3)=O)CC3CC3)CC2)=O)C(=O)N1 C1(C(C)C)CCCN(C(=O)Nc2cn(CC(N)=O)nn2)CC1 Cn1nc(C(=O)NCCC2(C(=O)NC(C3CCOC3)CO)CCC2)cc1Cl C12(C(=O)NCCOCCN(C(=O)C(C)(C)c3ccnn3C)C)CCC(C)(CO1)C2 c1(C(N2C(C)C(NC(=O)C(O)Cn3cncn3)CCC2)=O)ncnc2c1CCC2 C1(C(N2CC(C=C)(CC(=O)NCCC(O)C(F)F)C2)=O)CCCCCN1C C#CC1(C(N2CCCC(CC)CC2)=O)CCN(C(c2ccsc2)=O)C1 C(CCCC(=O)N1CC(NC(=O)CC(F)(F)F)CC1C)SC c1(C(=O)NCC(C)N(CC(N)=O)C)ccc(C(F)(F)F)o1 N1(C(c2c(C)n(C)nc2)=O)CCCC(C)C1CCNC(=O)C=C1CCCC1 N1(C(c2ccn(C(F)(F)F)n2)=O)CCC(n2ccnc2)C1 C1(C)(C(=O)NCC(C(=O)NCCn2c(CC)nnc2)O)CCN(C)CC1 C12(C=O)CC1CCN2C(=O)CC1CC(C)(C)CO1.N1(N(C)CCO)CC(NC)C1 c1(C(N2CC(O)(C(C)NC(=O)CN(C)C)C2)=O)cc(F)ccc1OC(=O)C1CC1 CCC(C)(C)C(=O)C(=O)NCCN(C)C(C1CCCC(C(N)=O)CC1)=O c1(C(N2CC(CNC(CC3(C)CC3)=O)C2)=O)c(Cl)n(C)c2cc(Cl)c(Cl)cc12 c12cc3[nH]nnc3cc1C(C=C)C(=O)N1CCC(O)(C1)CNC2=O.C1(C(C)C)(CC)CC1 N1(C(C(C=C)O)=O)C2COCC1CC(NC(=O)CC1CC(SC)C1)C2 N1(CC(N2CCN(C(c3c(C)nncc3)=O)CC2)=O)CC(=O)N(C)C1=O Cc1noc(C)c1C(N1CCCC1CN(C)Cc1ccnc(Cl)c1)=O c1(OC)ccc(C(=O)NC2CC2CNC(c2ncnc(O)c2Br)=O)cc1C CC1(C)CCOC1C(=O)NCCC1(NC(C2CCCC2(F)F)=O)CCC1 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2)ccc(F)c(Cl)c1N N1(C(c2ccc(-c3cc(C#N)on3)cc2)=O)CC2OCCOC2C1 C(C(C)(C)CCl)(c1n(CCCCCC)nnn1)NCCC(=O)N(C)C C1(C(=O)NC2CCCC2)CC2CC2N1C(C1CC1c1ccc(Cl)cc1)=O CC1C(C)N(C(c2nn(C)cc2N)=O)CCN1C(C1CC2(CSC2)C1)=O CC(C)CCC(C(=O)NCCc1ncccn1)NC(c1cc(F)cc(F)c1)=O C12(NC(c3cncc(C)n3)=O)CCOC(CNC(c3csc(C)c3N)=O)(C1)C2 C(=O)(C(CO)C(F)(F)F)N1CC(C(N2CC(=O)NC(C(C)C)C2)=O)(SC)C1 CC(C)C(CC(=O)NC(C)(C(=O)OC(C)(C)C)C1CC1)OC(F)(F)F N1(C(c2ccc(SCC)cc2)=O)CC(C)N(C(c2cnc(N)c(N)c2)=O)CC1C Cc1ccc(C(N2CCCCC(C)C2)C(=O)NCC2CCCO2)nc1Br c1(C(N(CC(CC)NC(=O)C(C)(C)C2CCCCC2)C)=O)scnc1C c1(C(=O)NCC2(NC(C3C(OCC)CC3)=O)CCCC2)ccnc(S)c1 N1(C(C2CC(N(C)C)C2)=O)CCC2(CCCC2CNC(C2CCCC(=O)O2)=O)CC1 C12(NC(c3c(Cl)nc(OC)s3)=O)CCN(C(=O)CCn3cccnc3=O)CC1C2 S(=O)(=O)(c1ccc(-c2nnc(C(F)F)o2)cc1)NC1CCC(C)CC1 c1(N2C3(CNC(C(CC)CC4CC4)=O)CCC2CC3)ccc2c(n1)CCCC2=O c1(C(C)C)n[nH]cc1C(=O)NCc1n[nH]cc1C(N1CCC(CN(C)C)C1)=O N1(C(C2CCCCN(C(CC(=O)OC)=O)C2)=O)CCCC2CCCCC12 CC(C)C(C(=O)N(C)CC1CCCN1C(=O)C1CC1)NC(=O)OC(C)(C)C N1(C(CN(CCC=C)C(C)=O)=O)CCC2CC12CCCN1CC=CC1 N1(C(c2c(C(C)C)ncnc2)=O)CC2CCC(CNC(=O)C(CO)N(C)C)(C2)C1 c1(C(=O)NC2CN(C(c3ccc(CO)nc3)=O)C2)ccc2ccncc2c1 C1(C(=O)NC2CC=C(C)CC2)CC2CCC(C1)C2 C1(C(N(C(C)CNC(c2cc(C3CCC3)no2)=O)C)=O)COCCN1CC(F)F N(C)(C(=NCC1=C(C)OCCS1)NC1CCC1)Cc1ccc(C(=O)NC)cc1 C(C#CC(=O)NCCC(C)NC(=O)Cn1nnc(C)n1)(OCC)OCC CC1CCCC(CC(=O)NC2CC3(C2)CC3C(=O)NC2CN(C(N)=O)C2)O1 C1(NC(CCNC(COC)=O)=O)CC(C(=O)NC2CC3(CCOC3)C2)=CC1O N1(C(C2(C=C)CCN(C(c3ccnc(CO)c3)=O)C2)=O)CC2(CO)CCC1CC2 c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)ccc2cc(Cl)ccc2c1 C1(NC(CC2CC(SC)C2)=O)CC(CC(=O)NC2(CN(C)C)CC2)C1(C)C N1(C(c2coc(Br)n2)C(=O)NC)CC(C(=O)OC)C2(CCCCC2)C1 C1(NC(=O)CN2CCCS2(=O)=O)CS(=O)(=O)C2CN(C(c3cscn3)=O)CC12 C1(N(CCC(=O)NCCN(C(C2CC2c2cccnc2)=O)CC)C)CCCCCC1 C1(CNC(C2(SC)CC2)=O)CN(C2CCN(c3ncccc3Cl)C2)CC(C)(C)O1 CC1CC(CC(=O)NCCC(O)CNC(c2ccc3c(c2)CC3)=O)CC(C)(C)C1 c1(CC)ncc(C(=O)NC(CCN(C(=O)Cc2coc(C)n2)C)C(C)C)cn1 N1(C(c2c(C)nns2)=O)CCCCC1CNC(=O)Cc1ccn(C)n1 C#CCCC(O)C(=O)N1CC(CNC(c2c(Cl)cccc2Cl)=O)CC1(C)C N1(C(C)C)C(=O)COCC1C(=O)NCC1C2CC1N(C(=O)Cn1cncn1)C2 C1(C(=O)NC(C(C)C)CNC(c2cncc(Cl)c2)=O)CN(CP(C)(C)=O)C1 N1(C(C2CN(C(N)=O)C2)=O)CCCC(NC(=O)C#CC2CC2)C1 Cc1cnnc(O)c1C(=O)NC1CCCC1CN=c1[nH]nc(C(C)(C)C)o1 C#Cc1cccc(CC(=O)N(C(CNC(c2ccc(F)cc2C)=O)CC)C)c1 C(CC(=O)NCC(C1CCCN1C(c1cc(C)cs1)=O)(C)C)(C(F)(F)F)OC N1(C(CC(CCC)C)=O)CC(c2cn(-c3cnn(C)c3Br)nn2)C(O)C1 C(=O)(C1=CNC2=NCCCN12)N1CCN(C(c2ccc(C)n2C)=O)CC1C1CC1 c1(C(C(=O)NC(C)CC)N(CCOCC)C)ccc(CO)c(C)c1 C1(C(=O)NCCN(CCOC)C(C2SCCCS2)=O)CCC2(CC1)CC2 c1(CN(CC(c2ccccc2)NC(C2CC(OCC)C2)=O)C)ncncc1OC CC(CNC(c1nocc1Cl)=O)CC(=O)N(C)CCc1nccs1 C(=O)(C1CCC(=O)c2ccccc21)N1CCN(C(c2ncn(C)n2)=O)C(CF)C1 CN1CC(C(=O)NCC23CC(CCO2)C3)N(C(=O)COCC2CCOC2)C1 C(=O)(C(Cc1ccc[nH]1)N(C(C)C(=O)OCC)C1CC1)NCCC c1(NC(C2CC(F)CN2C(c2ccc(Cl)nn2)=O)=O)ncc(Br)nc1Br c1(C(C(=O)NC(CC)(C)C)N(C)Cc2cnn[nH]2)cn(C(C)C)cn1 C12(NC(c3c(CC)c[nH]c3)=O)CC3CCC(C1C2)N3C(=O)CCOC1CCC1 C1(CC)CCN(C(C2CCCC(CF)C2)=O)C1C(=O)NC C#CC1CC1C(=O)NCC1CCC1NC(=O)CCSC CCC(C)CC(C)C(=O)N1CCC(CNC(c2cccc(OC(C)C)c2)=O)C1 C(=O)(CC(C)(C)C=C)NCC1(CNC(CCCOCC=C)=O)CCCCC1 CC1(C)COC(C(=O)NCCCCCNC(C2COCC2(C)C)=O)CO1 C1(C(=O)NCC2(C)CC(NC(CN3CC(CC)C3)=O)C2)CN(C)CC(C)O1 N1(C(CCN(C)CCO)=O)CC2=C(C1)CN(C(=O)CN1CCCC1CSC)C2 C(CCC(=O)N(C(CNC(=O)CCCC1OCCO1)C1CC1)C)=CCC=C C1(C(=O)NC(C2(C(=O)NCC=Cc3cccnc3)CC2)C)CCC2(C1)N=N2 CC(F)(F)CCCC=O.C1(N2CCOCC2=O)CN(c2nnnn2CCF)CCC1O N1(C(=O)Cc2cnccc2Cl)CC(C2CCCN(C(C3CCC4(C3)N=N4)=O)C2)C1 C=CCCCCCC(=O)NC1C=CCN(C(=O)CCOc2ccc(Cl)c(Cl)c2)C1 C1(C(N2C(C(=O)NCC(=O)NC3(CC=C)CC3)CSC2)=O)CCOCC1 C=CCC(CC(C)C)C(=O)NCC1(NC(c2ncccc2C)=O)CCC1 c1(C(N2CC3CC3(C(=O)Nc3cncc(F)c3)C2)=O)c(C(F)(F)F)cccc1Cl Cc1c(CC(N2CC(NC(C3OCCO3)=O)C3(CC3)C2)=O)ccc(Cl)c1Cl c1(CNCC23C(CN(C(c4cc(C)[nH]n4)=O)C2)C3)c(Br)cc(Br)c(O)c1Br C12(C(N3C(CNC(C4N(C(C)=O)CCCC4)=O)CC3)=O)CCC(C)(C(=O)O1)C2(C)C c1(C(N2CCCC(C(=O)NC(C=C)C)C2)=O)cccc(Br)c1O c1(CC(=O)NCC2CC(OC)CN2C(C2CCN(C)C2)=O)c[nH]c2cnccc12 C12(CNC(c3cc(C)on3)=O)CN(C(c3cnc4ccnn4c3)=O)CC1CCO2 N1(C(=O)OCC)CCC(C(N2CC(N3CC4C(C(=O)O)C4C3)C3CC23)=O)CC1 N(C1CCCc2c1cnn2C1CCCC1)C(CNS(C)(=O)=O)=O C(=O)(CC(C(F)F)NC(C1CN(C2CCC2)C1)=O)Nc1c(C)nccn1 C1(NC(C(COC)OC)=O)CCC(O)CN(C(=O)CCN2CCN(C)CC2)C1 c1(C(N2CC(CNC(C(C(CC)C)O)=O)(COC)C2)=O)cn(C)c2ncccc12 c1(C(=O)NC2(C(=O)NCC(c3ncc[nH]3)C)CCC2)cc(C(F)F)cs1 C1(C(N(CCCNC(=O)CC2CCCC2C)CCC)=O)CC(F)(F)C1(C)C C1(CNC(=O)NCCC(C=C)C)(CF)CC(F)(F)C1 CCCCCC(C)(CC)C(=O)NC1CCN(CCOCC(F)F)CC1C C1(O)(CN(C)C)CCN(C(c2ccnc(CNC(C3(C)CCCS3)=O)c2)=O)C1 CCC(O)CC(=O)NCC(C)NC(=O)CCc1cnn[nH]1 c1(N(C)C)nc2cccc(C(N3CCCCCC3CNC(C3(O)CC3)=O)=O)c2o1 c1(CC(N2C3CN(Cc4cccc(F)n4)CC23)=O)ccccc1[N+](=O)[O-] C(F)(C(=O)NCCC1CC(NC(=O)C(C)n2cnnn2)C1)OC C1(NC(CSCC(=O)OC)=O)CC2(CCN(C(c3ccns3)=O)C2)C1 C1(C(N(C)Cc2cn[nH]c2)=O)CC12CCN(C(c1cnc(S)nc1)=O)C2 c1(C(=O)NCC(C(C)(C)C)NC(=O)C(O)C2CCC2)cccc(F)c1C#N CCCCC(C)C(=O)NC(C)CC(C)NC(c1cn(CCO)nc1C)=O C12(C(=O)NC3(CO)CN(C(C=C(C)Cl)=O)C3)CCCC1(C(N)=O)C2 N1(C(C(c2cccs2)NC(c2c(C)n(C)cc2)=O)=O)CC2CC3CC2C1C3 S(=O)(=O)(c1ccccc1COCC1CCCN1C)N(CCC)CCC C(=O)(CC1=NNC(=O)C1)N1CCOCC(CNC(=O)COCC2CCC2)C1 C1(C)(C(N2CC(CC(=O)NCC(C(C)C)O)OCC2)=O)C(C)(C)C1(C)C C(N=c1ccn(CC(=O)NCc2cccc(Br)c2)c(O)n1)c1ccc(C)cc1F C=Cn1nccc1C(=O)NC1(CCNC(C2ON=C(C)C2C)=O)CC1 C(CC(F)F)(C(=O)NCCN1CC2CC2C1)NC(c1nnn(C)c1N)=O CC1CC(=O)NC(C(N2CCC(C)C(CC(=O)NCCC(O)C(F)F)C2)=O)C1 C1(C(=O)NCC(C)(C2CCC2)NC(C=CC(CC)=CC)=O)CC(C)=NO1 c1(OC)ccc(F)c2[nH]c(C(=O)NCC3(NC(=O)CN4CCOC4=O)CC3)cc12 C1(C2CCN(C(C3(CC)CC3)=O)C2)CCCCN1C(=O)CCC(N)=O C1(C(=O)NCC=CCNC(c2nccc(C)c2)=O)CC2CCCC(C1)C2(F)F N1(C(c2ccn(CC)n2)=O)CCCCC(CNC(=O)Cc2conc2C)C1 CCCCCC(C)CC(=O)NCCn1cnnc1C(N1CCCCCC1CO)=O N1(C(c2c[nH]c(=NC)o2)=O)CCC(C)(C)C1C(=O)NC(c1ncc[nH]1)CO C1(CC(=O)NC2(C=C)CCC2)CCN(C(=O)C(F)=C(C)C)C1(C)C C1(CNC(c2c(C)ncs2)=O)C2CCCC1N(C(=O)CSc1cn[nH]c1)C2 C1(C(=O)NC2CC(C)(CNC(C3CC(O)C3)=O)C2)CCCC(C)(C)CC1 C(c1cncc(F)c1)=CC(=O)NC(C1(O)CCN(C(c2cnc(CC)s2)=O)C1)C C1(NC(c2cnc(Cl)s2)=O)CC12CCN(C(=O)CN1CC=CC1)CC2 S(=O)(=O)(c1ccc(Br)cc1)N1CCC(N2CCCN(CCOC)CC2)C12CCC2 c1(C(=O)OC)ccc(F)c2c1CN(S(=O)(=O)Cc1cccc3cc[nH]c13)CC2 N1(C(C(CC#C)C)=O)CCCC2CN(C(C3CC(SC)C3)=O)CCC12 C1(CC)CN(C(C2CCC(=O)N2)=O)CC1NC(c1nn(C(C)C)nc1Br)=O N1(C(C(N2CCCCC2=O)C)=O)CC(NC(C2CC3CC3C2)=O)CC12CCCC2 N1(C(CCn2c(C)csc2=O)=O)CC(NC(C23CC(CCO2)C3)=O)CC(F)C1 C1(CNC(C(CC=C)(C)C)=O)CN(C(c2ccc(SC)[nH]2)=O)CCC1(F)F CCC(CC(F)(F)F)C(=O)NC(CNC(=O)COc1ccn(C)n1)CO N(C1CN(C(=O)CN=S(C)(C)=O)Cc2ccccc21)C(C(C)OC)=O CC1(C)CC(C(=O)NC2COCC2C(=O)NCCOc2ccncc2)CCO1 C(=O)(C(C)C(C)NC(c1nn(C)cc1C)=O)NC1(C)CN(C(=O)OC)C1 C=CCC(C)(C)C(=O)NC1CCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 c1(C(C)=O)ccc(C(=O)NCC2CN(C)CCN2C(=O)C(F)CC(C)C)cc1C C(C1c2ccsc2CCN1C(c1sccc1F)=O)NC(CSCC=C)=O N1(C(=O)NC2CCCCN2)CCc2nc[nH]c2C1c1ccc(F)cc1 C1(C(=O)NCC(CN(C)C(C23CCC(CC2)CC3)=O)O)CS(=O)(=O)CC12CC2 N1(C(C(C(C)C)NC(C)=O)=O)CCC12CN(C(C1CC(=O)NC(=O)N1)=O)C2 CCCCC(C(=O)N(CCOCC)CC1CC1)NC(=O)C(C)(C)Cl C(C(=O)N=S(C)(C)=O)NC(c1ccncc1C)c1n(CCCSC)nnn1 C=CC1CCCN(N2CCN(c3nc(C(C)(C)C)ns3)CC2)C1 CC(C)(C)C(O)C(=O)NC1C2CC(NC(=O)C(C)(F)CC3CCCC3)CC12 C1(C(N2CC3C(CNC(C(C4CCOCC4)C)=O)(C3)C2)=O)(CF)CC2(CCC2)C1 c1(OCCC)cccc(CCC(=O)NCC23CC2CN(C(=O)CC(C)OC)C3)c1 CC1(C)COCCC1C(N1CCC(CNC(=O)Cc2csc(C(N)=O)n2)CC1)=O CC(C)(C)C1CCNc2c(C(=O)NCCNC(=O)CCc3cnccn3)cnn21 N1(C(C=C(COC)C)=O)CCC(NC(=O)CSC2CCCCO2)C1C1CC1 C12(NC(C(CC=C)N(C)C)=O)CCC(CNC(C3(COC)CC(=C)C3)=O)(C1)OC2 C1(NC(c2ccc(=O)n(-c3ccc(I)cc3)c2)=O)CNC2(CCC2)C1 C1(C)(CNC(CCC2(C)CC2)=O)CC(F)(F)CN1C(c1cccc(Cl)c1O)=O C1(CC)CN(C(C2COCC2NC(C2CCC3CC2CO3)=O)=O)CCCO1 C1(CC)CCCN(C(C2CC(=C3CC3)C2)=O)C1C(N1CCN(CC(N)=O)CC1)=O c1(C(N2CC(C)(NC(=O)Cn3nnc(C(C)(C)C)n3)C2)=O)cn2cccnc2n1 C(=O)(CC(CC)NC(C1(CC)CCCN1C)=O)NC(C=C)C N1(C(CCNC(C)=O)=O)CCCCC1C(C)NC(C1CC(CC2CC2)C1)=O C1(Nc2cc(OC)nc(OC)n2)CC(C)(C)C12CCC2 C1(NC(C(CC)CC)=O)C2CCN(C(=O)CC3CCCO3)CC12 c1(C(=O)NCC(N(C)C(C2CCC2C(C)(C)C)=O)C2CC2)cc(Cl)c(Cl)n1C C1(NC(C(C)(C)CC#N)=O)CCC2(CC1)CCN(C(c1conc1C1CC1)=O)C2 c1(CNC(COCC)=O)ccc2c(c1)CCC2NC(=O)C#CC1CCCCO1 CCCC(C(=O)N1CCC(N(C)C)C1)NC(C)=O.C12CC(C1)NC2=O C(=O)(CC(C)C(=O)OC)NCCC1CCN(C(C(CC)CC)=O)C1 C=C=CCCC(=O)NC(C)(C)C=CC(=O)NCC(N1CCOCC1)=O c1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)CO)C2)[nH]c2ccc(Cl)cc2c1Cl c1(OC)c(F)cc(C(=O)NCC(C)(CO)NC(C2CCC(C)(C)CO2)=O)cc1Cl c1(C2C(C(=O)NCCOC)C2)noc(C)n1 Cc1csc(=Nc2cccc(C3CCCCC3)c2)n1C1CCCSC1 c1(CNC(c2ccc(C)n2C)=O)cc(O)cc(=O)o1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCC1(CNC(=O)CCCS(N)(=O)=O)CC2 N1(C(C(C=C)(C)C)=O)C2CCCC1CC(NC(c1ccccc1S(C)(=O)=O)=O)C2 c1(C(N2CCC(c3ccccn3)C2)C(=O)OCC)ccccc1C CCC(C)C(O)CC(=O)NCC1(NC(=O)C2=C(C#N)CCC2)CCCCCC1 CC(C(C)C(=O)NCC1(Nc2ncccc2[N+](=O)[O-])CCOCC1)S(C)(=O)=O N1(C(C2C(C(C)O)C2)=O)CC(CNC(C2CC2(C)C)=O)C1 c1(C(C(=O)NCC(CO)NC(=O)CC2CSC2)O)cccc(Cl)c1 N1(C(C(N2CCC(C)C2)=O)=O)CCCC(O)(CNC(C2(C(N)=O)CC2)=O)CC1 C1(CNC(C2CC(CCC)C2)=O)CCC(NC(=O)CCN2CCC2)CC1 c1(C(=O)OC)ccncc1S(=O)(=O)NC(=O)NC1CC(CCN(C)C)C1 N1(C(C(C2CCCC2)NC(c2ncccc2F)=O)=O)CC2CCC(O)C2C1 c1(N2CC(CN(C(=O)CC3CCCCC3(C)C)C)OCC2)ncc(C#N)cc1Br N1(C(CCCC)=O)CCC(NC(c2cc(C(N)=O)co2)=O)C(CC)C1 C(=O)(C(CNC(=O)CCCn1cncn1)OCC(=O)NC1CC(SC)C1)NC.C1CCC1 C1(F)(C(=O)NCC2C(C(NOCC3(C)CC3)=O)CCO2)CCOCC1 Cc1c(NC(=O)C(CCC2CC2)NC(c2csnc2Cl)=O)cnn1C N1(C(C(F)=CC)=O)CCC(CNC(c2n[nH]cc2-c2ccccc2)=O)C(C)C1 c1(CC(=O)N(CC(O)CNC(C2(C)C=CCC2)=O)C)c(F)cccc1F N1(CC)CC(C(=O)NCc2cccc(C(N3CCCC3C(N)=O)=O)c2)CC1=O Cc1nn(C)cc1C(=O)NC1CN(C(c2nocc2C)=O)CC1C C1(CNC(CN(C(C)C)C)=O)CN(C(C2CC(N3CC(O)C3)C2)=O)C1 C1(C(=O)Nc2c(C)nsc2)(NC(c2cc[n+]([O-])cc2)=O)CCCC1C NC1COC2(C(N3CCOC(c4ccc(F)c(Cl)c4)C3)=O)CC1C2 C(=O)(C1=CC2CCC(C1)C2)N1CC(C)CC(CNC(C(CC#C)(C)C)=O)C1 c1(NC)cc(NCCC(C)(C)NC(=O)C2=C(C)OCC2)ccc1[N+](=O)[O-] C=C(C)CC(C(=O)N(C(C)CCSC)C)NC(c1ncoc1CC)=O C1(CCCC)CN(C(C2CC23CCC3)=O)CCN1C(=O)C#CC1CC1 C1(C(=O)NCCC2CCCC2(F)F)(CNC(=O)OC(C)(C)C)CCOCC1 c1(N2C3CC(N(C)C)CC2CC3)nc(=NCc2cnns2)[nH]c2c1CCCCC2 C(=O)(C1=CCCCCC1)NC(CC#C)C(=O)NCC(C)(O)CCC C(N=c1[nH]c(=NCCC(C)OC)[nH]c2cccnc12)c1n(CCC)ccn1 c1(CNC2C(C(=O)Nc3c(C)ncnc3)C2)c(F)cc(C#N)cc1F N1(C(C(C)C2CCCC2)=O)CC2CC(C1)N(C(c1noc3ncccc13)=O)C2 C1(CNC(CN(C(=O)CSCC(F)(F)F)CCOC)=O)CC1(C)C C(=O)(CC(C)(C)CN(C)C)NC(C)C(C)C(=O)NCCS(N)(=O)=O c1(-n2ncc(C(N(CC(CNC(C(CC)(C)C)=O)O)C)=O)c2)ccc(F)cc1F N#Cc1ccc(CNC2(c3nnnn3CC(F)F)CCNCC23CC3)cc1F C1(N(C)C(c2nnn(-n3cccn3)n2)=O)CCC(CNC(=O)CCC(N)=O)CC1 C1(CC(=O)NCCCOCCNC(C2(C(N)=O)CC2)=O)CC=CCC1 c1(OC)cc2c(cc1CN1CCC(CC(C)C)(CO)CC1)OCO2 c1(NC)ccc(C(=O)NCC2(CNC(C3CC3F)=O)CC2)cc1[N+](=O)[O-] C(C(CC(F)(F)F)NC(C1CC(=O)NC1(C)C)=O)NC(C(CC)=CC)=O N1(C(CCCC)=O)CC(C(=O)NC23CC(F)(C2)C3)C(F)(F)C1 O=S(=O)(c1cccc(N2CCOC(C(F)F)CC2)n1)NCCCOC1CCCC1 N1(C(C2N(C(CCCOC(C)=O)=O)CC2C)=O)CC2(CCN(C)CC2)C1 C1(C(=O)NC2C(SC)CCC2)CC(O)CCN1C(c1cc(F)cnc1O)=O C=C1CC(C(=O)N(CC(C)C#N)CC2CC2)(CNC(C)=O)C1 c1(C(N2CCC(C(C)C#N)CC2)C(=O)NC)ccc(OCC(C)C)nc1C C1(CC)CN(C(=O)CSCC(=O)OC)CCC1NC(c1ccnc(NC)c1)=O C1(NC(Cc2c(C)n(C)cn2)=O)COC2(C1)CN(C(C1CCO1)=O)C2 c1(CNC(C(C(C)OC)NC(=O)CC2CNC(=O)O2)=O)nn(C)c(=O)n1C C1(NC(C(=O)NC(C)C)=O)CCN(C(c2cc(Br)ccc2F)=O)CC1C C(=O)(CC(C(F)(F)F)n1cccn1)NCC1(CCNC(C(C)N(C)C)=O)CC1 N1(C(c2c(C)cccn2)=O)CCC(NC(C2CCC(=O)N2)=O)C(CO)CC1 c1(C2N(C(C=CC(=O)OCC)=O)CCC2)ccc(Br)cn1 c1(NC(c2cnn(-c3ccc(O)nn3)c2C(F)F)=O)nc2ccccc2o1 Cc1ccc(C(=O)N(CC(C)N(C(=O)CCn2cncn2)C)C)c2cccnc12 c1(OC(C)C(=O)N2CCC2CNC(=O)CCC2CCCO2)ccc(F)cc1 C(=O)(C1CCC(=O)c2cccn21)NCCN(C(C=CCCC)=O)CC c12onc(C)c1OC(=O)C2.N1(C2CN(C(C(=O)NCC)=O)C2)CCOC1=O C(=O)(C1=CCC(F)(F)CC1)NCCCOCCNC(C1CCCC(=O)N1)=O C(C(C(=O)N(CCCOCCNC(C1CC1C)=O)C)C(F)(F)F)OC c1(C(=O)NCC2C(CNC(c3c(CC)nns3)=O)C2)cc2c(F)cc(Cl)cc2[nH]1 CC(N=c1nc2c(cnn2C)c(NCc2ccc(C(F)(F)F)o2)[nH]1)C1CC1 Cc1nccc(C(=O)NCC2CCCN(C(C34CC5CC3C4C5)=O)C2)c1Cl CC(C)CS(=O)(=O)CC(=O)N1CCOCC(CNC(=O)C(F)C2CCOC2)C1 C1(NC(C(CC)O)=O)CCN(C(c2cccc(N)c2F)=O)CC12CCC2 CC12CCC(C(=O)NCc3cccc(NC(=O)C(=O)c4cccs4)c3)(CO1)C2 C1(NC(C2OCC(C)C2)=O)CC2CC(C1)N(C(=O)C=Cc1ccccn1)C2 C1(C(C(=O)NCC(CCNC(CCSCC)=O)OC)O)CCCCCC1 C(C(CNC(=O)NC1(c2noc(C)n2)CCC1)C(C)C)OC Cc1ccccc1CC(=O)NC(C)(C)CC(=O)N(C)CCN(C)C1CC1 C1(CNC(C(C2CC2)OC)=O)CN(C(=O)CCc2nc[nH]n2)C2(CCC2)C1 c1(C(=O)NC2CC(CO)NC2=O)cccc2ccc(Br)nc12 Cc1c(C(N2CCCC(CNC(C3(C)CCC(C)C3)=O)C2)=O)cnc2ncnn12 C1(c2cn(CC(N3CCN(C)CC3)=O)nn2)CC2(CCCN2)C1.C(C)(C)C Cc1ccc(F)c(CS(=O)C(C)C(=O)N(Cc2ccccn2)Cc2ccco2)c1 N1(C(c2c(C)nn(CCO)c2)=O)CCCC(NC(c2cn3c(n2)CCC3)=O)C1C CC(=O)C(C)(C)CC(=O)NC1CCC(NC(=O)C2=CCCSC2)C1 N1(C(Cc2c(C)occ2)=O)CCC2OCCN(C(=O)CNC(=O)C(C)(C)C)C2C1 N1(C(CSCC)=O)C2CCCC1CN(C(C1Cc3ccccc3C1)=O)CC2 c1(OC(c2ccc(N(C)C)cc2)CC)cccc(F)c1 N(C(=NCCCOCCN(C)C)NC1CCN(c2ccccc2)C1)CC(=C)C C1(CNC(c2c(OC)cc(C)cc2)=O)CC2CCC1N(C(=O)CC(=O)N(C)C)C2 c1(CC(=O)NCC=CC(=O)NCCC=CC=C)c(C)noc1C C12(C(=O)NCC(=O)OC)CCCCN1CCC2.c12cc(F)ccc1NC2 C1(C(=O)NCC2(C)CCC(NC(CC(CCC)O)=O)CC2)CCc2nccn2C1 C(c1c[nH]nc1C)=CC(=O)NCCNC(C1N(CCC)CCC1)=O C#CC1CCCN1C(=O)C(CC1CC1)NC(=O)C(C)(CO)OC c1(N(C)C)ncccc1C(=O)NC1CCN(C(=O)CN2CCNC2=O)C1 N1(C(CC(CCCC)NC(=O)C(C)(C)OCC)=O)CCC2CCN(C)CC12 c1(C(N2CCC(NC(C(C)OCCC=C)=O)CC2)=O)ccc2cnoc2c1 Cc1[nH]nc2ccc(C(=O)N(C(C)CN(C)C(C3CCCCCC3)=O)C)cc12 C1(C(F)(F)C(=O)N2CCC(N(C)C(c3ccncc3Cl)=O)C2)(OC)CCCCC1 N1(C(C(=O)NCC2CCC(c3nc(O)cc(C)n3)CC2)=O)CCc2n[nH]cc2C1 C(=O)(C#CC1CCCO1)N1CCC(N(C(c2c(CC)nccc2)=O)C)C1 C1(CCC)(NC(c2ccc(=O)n(C)c2)=O)CCN(C(=O)CN(C)C(C)C)CC1 C1(CCC)CCC(NC(=O)C(=O)Nc2ccc(-c3nncn3C)nc2)CC1 C(=O)(C1=CCN(C(C2CC=C(C)CC2)=O)CC1)NCC1(SC)CCC1 CCCC(C(=O)N(CC(F)(F)COC)C)NC(C1(OC)CCOCC1)=O C12(N(C(C=CCCC)=O)CC)CCC(CNC(=O)C(C#N)C(C)(C)C)(CC1)OC2 N1(C(C2C(CCC)C2)=O)CCN(C(c2ccc(F)c(C(C)C)c2)=O)CC(C)C1 Cc1cc(Cl)cc(N)c1C(=O)NC1CCN(C(=O)C(C)CC(F)F)C1 CC1(C)CC(CO)CN(C(c2ccc(CNC(=O)C3=COCCC3)nc2)=O)C1 C=CCC(CN(C)C)C(=O)Nc1c(C)ccnc1OC C1(NC(CCc2ccc(C)nc2)=O)CC12CCN(C(=O)Cc1cnc[nH]1)C2 c1(CN(C(=O)CCn2nc(-c3cccs3)oc2=O)CC(=C)C)cccc(Cl)c1 C1(CNC(c2c(C)c[nH]n2)=O)CC(C(=O)NC(CO)C(F)(F)F)=NO1 C1(C(N(C2CN(C(c3cnc(CC)o3)=O)CC2O)C)=O)CCc2nnc(C)n2C1 c1(C(=O)NC2C(CNC(c3cc(CC)on3)=O)CC2)ccc(=O)n(CCOC)c1 C1(C2CN(C(=O)C=CC3CCCO3)C2)(NC(Cc2cn(C)nn2)=O)CC1 n1(CC)ncc(Cl)c1C(=O)NCC(C)N(C(=O)CC(C)C1CC1)C C(c1cccc(Cl)c1)=C(C(=O)NC1CCN(C(c2c(C)nc(OC)s2)=O)CC1)C c1(NC(CN(CCC=C)CC(=O)C2CC2)=O)cc[nH]c(=NC)c1 N1(C(c2cc(C)nc(C)c2)=O)CCC2(CCCN2C(C2CCOC2(C)C)=O)C1 c1(C(=O)NCCOC2CN(C(C3C(C)(CC)C3)=O)C2)nccn2nccc12 C12(C(N3CCC(C(C)NC(C4CCN(C)C4)=O)CC3)=O)CCC(CC1)CO2 C(C(O)C(F)(F)F)NC(=O)C(=O)NC(c1cccc(Cl)c1)Cc1ccccn1 C1(CC#C)(C(=O)N(CC)Cc2ncc[nH]2)CCN(C(c2nc(C)sc2C)=O)C1 Cc1nc(=NCCC2CCCCN2C(=O)Cc2cccc(C(F)F)c2)[nH]cc1Br c1(C(=O)NC2(C(C)NC(=O)C(N3CCC(C)C3)=O)CC2)ccn2nccc2n1 CN1CCCC(C)(C(=O)NC(CC(=O)NCC2CCCNC2=O)C2CC2)C1 O=S(=O)(c1cccnc1N1CCC2(CCC2)CC1)NCc1ccncc1 C(c1cccnc1)=CC(=O)NCCOCCNC(c1cn(CCC#N)nn1)=O C1(CCC(=O)N(CC(C)O)CCNC(=O)C(C)(C)C2CC2)CCCN(C)C1 C(C#Cc1cn(CC2CC3CC3C2)nn1)NC(Cc1c(OC)nccc1)=O c1(C2CCOCC2)cccc(Cl)c1.Cn1nncc1C(=O)NC(=O)Cn1nccn1 C(=O)(C1COc2cc(C)c(C)cc21)N(C1CCN(C(=O)CC(C)OC)CC1)CC C1(NC(C(C)(C)C2CCN(C(=O)CCn3cccn3)C2)=O)COCC(C)(C)C1 c1(CC(=O)NCC(CNC(=O)C(C)NC(=O)C2CC2)OC)n[nH]c2c1CCCC2 c1(C(C)C)cc(F)c(Cl)cc1Cl.C1C(C(=O)O)NC1=O C1(NC(C(C)OCC(F)(F)F)=O)CCC12CN(C(c1cn(C)[nH]c1=N)=O)C2 O=C(CC(C(F)F)NC(=O)C1CC1)NC(c1cnn[nH]1)N1CCC1 CCCCCC(O)CC(=O)NC(C)CC1CN(C(=O)CC)C1.c1(C(=O)OC)sc(C)cc1Cl C#CCCCC(C)C(=O)N(CC(C)(C)CNC(C1CCc2n[nH]cc2C1)=O)C N1(C(C(C)N(C(c2c(CC)cco2)=O)C2CC2)=O)CCCN(CC2CC2)CC1 c1(CC)onc(C(=O)NC(C)C(C)NC(C2CC(n3ccnn3)C2)=O)c1C N1(C(CSCC)=O)CCC(CNC(c2csnn2)=O)CC1C C1(OC)CC(NC(C2CC=CC2)=O)CN(C(C2(N3CCOCC3)CCC2)=O)C1 N1(C(c2cnc(OC)s2)=O)CCCCC(N(C)C(C2(C)CCN(C)C2)=O)C1 CC(C)CCCC(=O)N1CCC(C(C)CNC(=O)CC(O)CN(C)C)CC1 N1(C(C(=O)Nc2ccc(OC)cc2CNS(C)(=O)=O)=O)CC2CCC1CNC2 N1(C(C(C)C(C)O)=O)CCOCC(CNC(c2scnc2Cl)=O)C1 N1(C(=O)CCC2CCCCCC2)CCC2CN(C(C3(O)CCOCC3)=O)CC12 c1(CNC(C2CC(C)(F)C2)=O)nc(CNC(=O)CS(C)(=O)=O)cc(O)n1 CCC(C)(CNC(=O)CC1CN(C(=O)CC2CSCCO2)CCO1)CO C(CC(=O)N1CCC(C)CC1)(C(C)(C)C)NC(c1nccc(OC)c1)=O c1(OC)cc2[nH]cnc2cc1C(N1CC2CC(C1)N(C1CC1)C2)=O C1(CCC(=O)NCCn2ncc(C)c2)CCCCN1C(=O)CC(C1CC1)C1CC1 c1(C(C)(C)C)ccc(C(N2CCC(NC(C3CC(C)(CO)C3)=O)CC2)=O)c(N)c1 C1(CC(C)O)CCCN1C(C1(CCNC(=O)CN2CCOC2=O)CCCC1)=O Cn1[nH]c(C(=O)NCCC2(NC(=O)Cn3nnc(-c4ccco4)n3)CC2)nc1=O Cc1ccc(C(N2CC(C3CCN(C(C4CC5CC(=O)C4O5)=O)CC3)C2)=O)c(O)n1 c1(C(N(c2nc(C(=O)NC3CC3(F)F)cs2)C)=O)ccc(CCC(=O)N)[nH]1.C(F)(F)F Cc1cccc(C)c1C(=O)NCCC1(C)CCN(C(=O)C2=CCCCO2)C1 N1(C(C(C(CC)O)C)=O)CCC=C(C(=O)NCC2CC(F)(F)C2)C1 CCCCC(O)C(=O)N1CC(CC(C)NC(=O)C(C)C(O)Cc2ccccc2)C1 C1(C(=O)Nc2cn(C)nc2)CCC(NC(=O)CN2CCOC2=O)CC1 c1(C(=O)NCCOCCN(C)C(C2(C)CC2(F)F)=O)cccc2c1COCCN2 c1(C(N2CC(C)(NC(CC3CC(CC)C3)=O)C2)=O)ccc(O)c(Cl)n1 Cc1cc(CC(=O)NCC(C)N(C)C(C2CC3CC3C2)=O)cc(C)c1Br N1(C(CC(CCC)C)=O)CC2CCC(C1)N2c1nc(C2CC3(CCC3)CO2)ns1 c1(OC)ccc(S(=O)(=O)N2CC3CN(Cc4nc5ccccn5c4C)C3C2)cn1 c1(N2CC(N(CCCC)C(c3cncc(C)c3C)=O)C2)ncnc2c1ccn2CC N#Cc1cc(C(=O)NC2CCC2NC(C2CCCCC23CCC3)=O)c(F)cc1F Cc1cc(CC(N2CC(CO)(NC(=O)COc3ccsc3)C2)=O)no1 C12=CC=C(C=C1)C2.c1(NCCNC(C2C(C)C2)=O)ncc(Br)cn1 Cc1onc(C(=O)NC(C)C(C)NC(=O)CCc2ncc(F)cn2)c1[N+](=O)[O-] N1(C(CCC)=O)CC(NC(=O)CC(C)(C)CC)CC2(CC2)C1 c1(C(=O)NCC2C(CNC(CN(CCOC)C)=O)C2)csc(C#N)c1 c1(C(=O)NC(CC)CNC(=O)CC(c2cccs2)NC(C)=O)cc(C)cc(F)c1 CC1=NNC(=O)C1CC(=O)NCC1(F)CCC(NC(c2csnc2C)=O)C1 c1(NC(C)=O)ccc(F)c(C(=O)NC(C)C(C)NC(C23CC(C2)C(C)O3)=O)c1 C1(CN(C(=O)CCC2CCC(NC(c3cncn3C)=O)C2)C)COC(=O)N1 c1(CCC)cc(C(=O)NCCCOCCNC(C2CC2(C)Br)=O)sc1C C(=O)(C1=COCCC1)N(C1CN(C(C2(n3nccn3)CC2)=O)CC1(C)C)C C(C(CC(C)(C)C)NCc1nccn1CCc1ccccc1)OC CCC(C)C(C(=O)NCC1C2CN(C(=O)C3=NOC(C)C3)CC12)N(C)C C(C(=O)N(CC)CC1CCCN(C(=O)C=CCCC(C)C)C1)(C(C)C)OCC C1(C(=O)O)(OC)CCN(C(C2CC(=O)N(CCc3ccccc3)C2)=O)CC1 N#Cc1c(NC2CCN(C(C3CCN3C3CCCC3)=O)CC23CCC3)cccc1F N1(C(=O)OC(C)(C)C)CCC(NC(CCc2cn(C(C)(C)C)nn2)=O)CC1 c1(CNC2CCN(C(c3ccn(C)n3)=O)CC2F)cc(F)c(C#N)c(F)c1 c1(CC(N2CC(NC(C3C(C(C)C)C3)=O)C(C)C2)=O)cccc(Cl)c1F CCC(C)C(O)C(=O)NCC1(C(N2CCCC2C)=O)CCCCC1 C(=O)(C1SCCc2ccccc21)NCCC1CC(NC(c2c(N)nccn2)=O)C1 CC(N=[N+]=[N-])C(=O)N(CC(C)NC(C1(c2cc[nH]n2)CC1)=O)C Cc1nc(C(=O)NCC(C2CC2)NC(=O)CCc2ccc(O)nn2)ccc1C#N c1(C(N2CCC(N(C(c3cccc(C)c3Cl)=O)C)C2)=O)ccc2c(c1)COCC2 c1(C(N2CCCN(C(C(C)C)=O)CC2C(C)C)=O)cc2cc(F)cc(F)c2o1 N1(C(c2ccc(C(C)(F)F)cc2)=O)CC(F)(F)CC1CNC(C1C=CCCC1)=O c1(C(N(CC(C)NC(c2ccccc2)=O)C)=O)cncc2cnccc12 N1(C(c2ncc(C)o2)C(=O)NC2CCC2)CCC(C2CCCC2(C)C)C1 N1(C(C(Cc2ccsc2)NC=O)=O)CCC2(CC1)CN(C(=O)C(C)CO)C2 N1(C(C(C=CC)O)=O)CCN(C(=O)CCCc2nc3ccccc3o2)CC(O)C1 C1(COC)(NC(c2cnc(O)o2)=O)CCCN(C(c2cccc(OC)n2)=O)C1 C1(F)(C(=O)NC2CCC(NC(C(c3cccc(OC)c3)C)=O)C2)CCS(=O)(=O)C1 O=C1C(NCc2cccc(Cl)c2O)CCCN1Cc1ccccc1 C12(NC(c3cscc3C(F)F)=O)CCCC1CN(C(=O)C1=C(Cl)CCC1)C2 Cc1cc(C)c(CC(=O)NC(C)CN(C)C(c2ccn3nccc3n2)=O)c(O)n1 N1(C(C2(SC)CCC2)=O)CCC(C)C(CC(=O)NCc2cc(C)on2)C1 O=C(C1=CCN(C(C2(C3(O)CCC3)CC2)=O)C1)NC1CCOCC1 C1(N(C(c2ccnc(F)c2)C(=O)NCC2CCCOC2)C)(CSC)CCOCC1 C(CCC(C)C)=CC(=O)N1CCN(CCOC)C(=O)CSC1.c1(C(C)=O)nccs1 [N-]=[N+]=NC1CC(C(=O)NC2CC(CNC(c3ccnn3CC(F)(F)F)=O)C2)C1 C(=O)(CCS(N)(=O)=O)NCC(N(C)C(C1CN(S(C)(=O)=O)C1)=O)C1CC1 CCC(C)(C)CCCC(=O)NC(C)C(C)C(=O)NC1CNC(=O)OC1 C1(NC(C#CCNC(C2(C)C(C)OCC2)=O)=O)CC2(C1)CC(C#N)C2 N1(C(C(C)NC(=O)NC)=O)CCCC(COC)(NC(c2c[nH]c(C)c2)=O)C1 C(=O)(C#CC1CCOCC1)NCCOC1CCN(C(C(CC)SC)=O)CC1 c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC(C)C(NC(=O)CCCCOC)C1)=O c1(OC)ccc(-c2nc(C3CCN(C)C3C)n(CCCO)n2)nc1 C1(C(N2C(CN(C(C3CC=C(C)CC3)=O)C)CCC2)=O)CCCCCN1C C1(C(=O)NCC2CCN(C(=O)C(F)n3cccn3)C23CC3)(OC)CCCCCC1 N1(C(CC(CC)(F)F)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)CC2)CC1C c1(OCC)ncc(NC(C2(C)CC(O)CN2C)=O)cc1F C1(NC(CCC(=O)NC)=O)C2CC3CC(C2)CC1(CNC(=O)Cc1cnsc1)C3 C1(C(=O)OC)(CC)CCCCN1C(c1ccc(NC)cc1)=O N1(C(C(CO)NC(N)=O)=O)CC2(C1)CN(C(=O)CC=Cc1ccccc1F)C2 C#CCCCCC(=O)NC1CC(CNC(=O)COc2ccc(C(F)(F)F)nc2)C1 c1(NC)ccc(Cl)c(NC(=O)C(=O)NCCCn2nc(C)cc2C)c1 S(=O)(=O)(c1c(C)nn(C)c1Cl)N1CC(c2nc(C)[nH]n2)OCC1 C=CC(CCC)CC(=O)NC(CCSC)C(=O)NC1CC(=O)N(O)C1 N12CCCCC1CNC(=O)C2.C1(C(N)=O)CC(CSn2ccnn2)C1 N1(C(c2c(C)cc(Br)cc2)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1F c1(NC(C2(CC)CCOC2)=O)ccc(NC(=O)C(C)C(C)(C)C)cc1C S(=O)(=O)(c1cccc2cccnc12)NCCNCC1(F)C(C)OCC1 C(=O)(CC(C(F)(F)F)n1cccn1)N(C1CCCN(C(c2c[nH]c(C#N)c2)=O)C1)C N1(C(C(CC)OC2CCCC2)=O)CCC(C)(C(=O)N(C2CC3(CCC3)C2)C)C1 c1(C(=O)NC2C(NC(c3cnnc(O)c3)=O)COC2)n[nH]c2c1COCC2 c1(C(=O)NCC2(C(C)NC(=O)C(c3ccc(F)cc3)O)CC2)[nH]nc([N+](=O)[O-])c1Cl N(C(=NCc1ccoc1)N1CCN(c2ccc(C)cc2)C(=O)C1)C(C#C)C(C)C N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)Cc2ccccc2[N+](=O)[O-])CC(C)(C)C1 C1(NC(C2CCC(CNC(c3cc(C#N)sc3)=O)CC2)=O)CCc2nn[nH]c2C1 N1(C(C(C=C)CC)=O)C2CC1CN(C(=O)CCC(=O)N(CC)CC)C2 C12(C(N3CC(N(C)C)C4(C3)CC4)=O)CCC(CC1)N(C(c1cnc(S)nc1)=O)C2 C=C1CCN(C(=O)C(C)C(F)(F)F)C(C(N2CC(c3nncs3)C2)=O)C1 O=[N+]([O-])c1cnc2c(F)ccc(Br)c2c1NCc1nc(C2CCCC(F)(F)C2)cs1 c1(C(N2C(Cn3cc(CC=C)nn3)C=CC2)=O)ccc(C(F)F)c(C(C)C)c1 N#Cc1cc(F)c(C(=O)NCCCNC(C2CCc3nncn3CC2)=O)c(F)c1 C(CC(=O)NC1CC(NC(=O)COc2cccc(N)c2)C1)(C(F)(F)F)OC CCS(=O)(=O)NNC(=O)c1c(F)cncc1Br C(CN=c1[nH]c(N2CCN3CCCCC3C2)nc2c1COCC2)N(CCO)CC CC1CN(CCCc2csc(=N)[nH]2)CC(C)N(C(=O)C(N2CCC(O)CC2)=O)C1 C=CCC(C)(CC)C(=O)NC(C1CN(C(c2nnn(C)c2N)=O)C1)C C1(NC(c2ncc(OC(C)C)nc2)=O)CCN(CCCC(F)F)CC1 c1(C(=O)NC(C(C(C)C)NC(=O)C2=CCCCO2)C)ccc2nsnc2c1 C1(CNC(c2n(CC)ncc2)=O)CCN(C(C2CCCN(S(C)(=O)=O)C2)=O)CC1 C(C(O)C(=O)NC(C)(C)C(=O)NCCc1ncn(C)n1)NC C(C(C)(C)CNC(C)=O)N(C)C.C1(N(C(=O)C2CC2)C)CC(n2cnnc2)C1 O=S(=O)(c1ccc(O)nc1)N1Cc2cc(-c3nn[nH]n3)ccc2C1 C1(NC(COCC(c2ccccc2)C)=O)CCCC1(C)CNC(C1CC2(CC2)C1)=O C(=O)(CCCCCC(C)C)NC1C(CNC(C(C(C)(C)C)OC)=O)COC1 CCCCC(C(=O)NCC1(NC(=O)CNC(c2ccco2)=O)CCC1)C(C)C C=CCCC(C)(C)C(=O)N1CCCC(C)(NC(c2cnn(CCF)c2)=O)C1 CN1CC=CCC1CC(=O)NCCC1CN(C(C2(C)CCCOC2)=O)C1 c1(OC)ccc2c(N(CC3=CCSC3)C)nc(=NCC(Cl)(Cl)Cl)[nH]c2c1 N1(C(C2(NC(CC3(C)CCOC3)=O)CC(O)C2)=O)CC2CCC(C1)O2 CC1CC2CN(C(C3(NC(=O)CC(C)C4CC4)CC(CO)C3)=O)CCN2C1 C1(C(=O)Nc2cn(CC)nn2)CC(O)CN1C(c1ccc(SC)cc1)=O c1(CC(=O)OCC(COC)=O)ccc2ncccc2c1 C1(C)(C(=O)NC(CCOC)C(C)C)CC(O)CN1C(c1ccc(F)c(C)c1)=O N1(C(C(C)NC=O)=O)CCC2(CC1)CC(C(=O)Nc1ncc(C#N)cn1)CO2 N1(C(CSc2n(C)cnn2)=O)CCCC(C)(C)C1CNC(C1(C)CCNC1=O)=O CC1=C(C(=O)NC2C3CC4C(C3)C24C(=O)NCCCn2cnnc2)CCCO1 C1(CN(C(C2(C)CC2(C)C)=O)CC)CCCN(C(=O)CC2CN(C)C2)C1 C(=O)(CC(C)(O)COC)NCC(CC)NC(c1sccc1C(C)=O)=O C1(N(C(=O)COc2ccc(F)cc2)C(C2CCCOC2)C)CCCC12CCNCC2 C1(C(N(C)CC2(NC(=O)CSC(F)(F)F)CC2)=O)CCOC1=O CCCCC(C(=O)N1CCC(C(C)CNC(=O)C=Cc2ccoc2)CC1)C(C)C N1(C(c2c(CC)sc(=N)[nH]2)=O)CC2(C1)SCCC2NC(=O)CC1C=CCC1 N1(C(C(n2cc(Cc3cnn(C)c3C#N)nn2)C)=O)CCc2ccc(Br)cc2C1 c1(CC)cccc(CC)c1CC(=O)N(CC(C)N(C)C(c1ccncc1F)=O)C c1(OC(CCN(c2ccc(F)nc2Br)CC)=O)ccc(C)c(F)c1 c1(C(=O)NC(CC=C)CNC(=O)C(C)NS(=O)(=O)CC)ncc(CC)cn1 N1(C(CN(CCOC)C)=O)CCC(NC(c2cccc(CO)n2)=O)C2(CCC2)C1 C1(C(=O)NC(C#C)(C)CC)CC2CC2N1C(=O)C(N1CCCCC1)C N1(C(C2(CC)CCNC2=O)=O)CCC2CN(C(=O)C=CBr)CC2C1 c1(C(N2CCC3(CCC3)C2)=O)coc2c1COC2 N1(C(c2c(SC)nn(C)c2)=O)CCN(C)C(CNC(C2(O)CCSC2)=O)C1 C(C(C)(C)CNC(c1cnc[nH]1)=O)N(C(=O)C(F)(F)c1ccnn1C)C c1(C(=O)NC2(C)CCN(C(c3c(Br)cc(C)s3)=O)C2)cccn2nncc12 c1(CC(=O)NCC(C)CN(C(=O)CC2CCCCC2O)C)ccc2c(c1)CCO2 Cc1ccc(OC(C)C)cc1-c1ccc(NCc2ccc(I)cc2)nc1 N1(C(C2C(C)(CC)C2)=O)CC=C(C(=O)NCCn2cnc(C)c2C)CC1 N1(C(C(C2(O)CN(C(CCC#C)=O)C2)F)=O)C2CCCC1CC2 N1(C(C)=O)CCCN(C(c2c[nH]cc2C2CC2)=O)CC1C C1(N(C)C(c2coc(Br)c2)=O)CCN(C(=O)CCCc2cnn[nH]2)CC1 C1(C)(C(=O)NCC(CCNC(C2(OC(C)C)CCC2)=O)O)CCN(C)C1=O c1(C(=O)OC)ccc(CC(=O)N(C)Cc2ccc(Br)cc2)cc1.C1(C)C(=O)N1 N1(C(C2(CF)CC2)=O)C2CCC1CC(NC(C1(CO)CC(F)(F)C1)=O)C2 Cc1[nH]nc(C(=O)N(CC(=O)NC2C(=O)OCC2CO)C)c1C CC1CCn2ncc(CNCc3c(Cl)nc4ccccn34)c2C1 N1(C(Cc2cnc(C)o2)=O)CCCC(C2CC2NC(C2(C)CCC2)=O)C1 C1(C(=O)NCc2ccccc2)COCCN(C(=O)Nc2ccc(C(F)(F)F)o2)C1 c1(CC)cccc(C(=O)NCCn2cc(COC3CCOC3)nn2)c1F Cc1cnc(F)c(CNC(C2CC23CC(NC(C2CC2C#N)=O)C3)=O)c1 c1(C2C(C(=O)NCC3(SC)CCOC3)CNC2)ccccc1 c1(C(=O)NCCCCCCNC(C2C(C=C)(C(F)(F)F)C2)=O)c(C)nc(C)n1O CC1(C)CCC(CNC(=O)CS(=O)(=O)CCO)N(C(C2CCC(C(N)=O)C2)=O)C1 c1(C(=O)OC)ccc(Cl)c(C)c1NCC1CC(C)C1 C1(C(=O)NCC(F)CO)COCCN(C(c2ccccc2O)=O)C1 C=CCC(CC=C)C(=O)NCC=CCC(=O)NCC1CC1(Cl)Cl c1(C(c2n(CC=C)nnn2)NCc2ccc(OC)cn2)cccc(C(N)=O)c1 C(=O)(C1=CCC(F)(F)CC1)NC1(COC)CN(C(C2(CC)CC(C)(C)C2)=O)C1 c1(C(N2C3CCN(C(=O)Cn4cc(Cl)cn4)C(C3)C2)=O)nncc2c1CCCC2 c1(NC(C)=O)ccc(-c2ccc(-n3nc(C)cc3C)s2)c(C)n1 C1(NC(C)=O)CC(O)CN(C(=O)CNC(c2nnc(S)n2C)=O)C1 CCC(C)(C)C(=O)C(=O)NOCC(=O)NCc1ccccc1F C(C(=O)NCC1CCCN1C(=O)C(O)CN1CCOCC1)(C(C)C)SC n1(CC(N2CCC(CN(C(CC3CC(C)C3)=O)C)C2)=O)cc([N+](=O)[O-])ccc1=O N1(C(C2(C#N)CCSCC2)=O)CC(NC(C2CC(C(F)(F)F)C2)=O)CC2(CC2)C1 C(=O)(CCP(C)(C)=O)NC1(C)CCN(C(C2COCCC2(F)F)=O)C1 Cc1cc2c(cc(C(=O)NC3C(O)CC3O)n2CC(F)(F)F)s1 Cc1cc(C)c(C(=O)NCC(F)CNC(c2[nH]c(=N)ccc2C)=O)c(C)n1 C1(CC)CN(C(c2cn(CCNC(=O)CSC3CC3)cn2)=O)C(C)CO1 CC(C(=O)NCC1CC(F)CN1C(c1cc(Cl)cnc1O)=O)C(F)(F)F Cc1nc2ccc(NC(=O)C3=CCCN(C(=O)C(C)O)C3)cc2o1 C1(C(N2CCCC2CNC(C2CCOC2)=O)=O)CCCC2CCCCC12 c1(C(N(C2CC(NC(c3ccc(CC)[nH]3)=O)C2)C)=O)ccc(OC(F)F)cc1F C1(CNC(c2scc(OC)c2)=O)CC2CCCCC2N1C(c1cc(CO)[nH]n1)=O O=C(C1=CCCOCC1)NCCNC(C1CCCC(O)C1)=O C(=O)(C(F)C(F)(F)F)N(C1CCN(C(=O)CNS(C)(=O)=O)CC1)C c1(OC)ccc(-c2n[nH]cc2C(=O)NCC2CCCCC2c2ccncc2)cc1 c1(C(=O)NC2CN(C(C3(CC)CCCC3O)=O)C2)cc(F)cc2nn[nH]c12 c1(CCNc2nccc(=NCc3cc(SC)ncc3)[nH]2)nn(C)c2ccccc12 C1(CC)CN(C(c2ncccc2F)=O)CCC1NC(=O)C(C1CCOCC1)F c1(C(=O)NC2CC(C)N(C(c3cc(Cl)ccc3N)=O)C2)nc2ncccn2n1 C1(C)(Cn2cc(C(C=C)(C)O)nn2)CCN(C(C2(CC)CCCOC2)=O)CC1 Cc1cc(C(N2CCCC(c3nc(C)cs3)C2)C(=O)NCCC#N)cc(F)c1 CC1CN(CCCCNC(=O)C(=O)NCc2ccc(F)cc2F)CC(C)O1 C1(NC(c2ccccc2O)=O)CC(O)CN(C(=O)C=C2CCCC2)C1 c1(N2CCN(C(=O)NC(C3CC(C)CC(=O)N3)C)CC2)ncc(Br)c(C(F)(F)F)n1 c1(C(=O)NCC2CCC(NC(C(CC)NC(N)=O)=O)C2)cncc(OC(C)C)c1 C=CC(C)(O)C(=O)NC1CC(NC(=O)C=CC=CC=CC=CCC)C1 C(CC(C)(C)CC(=O)N1CCC2C(NC(=O)CNC(=O)CC3CCCC3)C12)OC CCCC(CNC(C12CCC(c3nn[nH]n3)(CC1)C2)=O)CCO C1(NC(C23CCC(N(C)C)C2C3)=O)C2CCC(C2)N1C(=O)CO.C12CN(C1)C2=O C(=O)(CCCCCCNC(c1cc(C)[nH]n1)=O)N1C(CSC)CCC1 C1(C(=O)NCC2CCCC2NC(c2cc(-c3ccco3)c[nH]2)=O)(CC)CC1(F)F CC1CN(C(C)Cc2ccccc2)CC1NC(=O)NCC1CC1(F)F Cc1ccc(F)c(C(N2CSCC2C(=O)NCCCOC(C)C)=O)c1 S(=O)(=O)(c1c(Br)cccc1[N+](=O)[O-])NCCC1C(C(=O)OC)C1 c1(C(N2CC(C3(NC(C4(C(N)=O)CC4)=O)CC3)C2)=O)ccc2c(c1)C(=O)CCC2 C(=O)(C(C)(F)C(C)(C)F)N1CC(O)(C(C)NC(c2cnn(CCC)c2C)=O)C1 N1(C(C2OCCC(C)C2)=O)CCCC(C2CN(C(C3(F)CCN(C)CC3)=O)C2)C1 N1(C(C(CC)n2ccnc2)=O)CCC(CN(C(=O)CC2(N(C)C)COC2)C)CC1 N1(C(c2occ(C)c2)=O)CC2(CCC2)CCC1CNC(=O)Cc1ccc(Cl)cn1 C#Cc1ccc(C(=O)NCC(C(C)(C)C)NC(=O)C=CS(C)=O)cn1 N1(C(c2ccc(OC)nc2)=O)CC2(CC2)CC1CNC(C1CCOCC1CO)=O C(=O)(C(CC(F)F)NC(C1CCCC(C#N)C1)=O)NCCN1CC(C)(O)C1 N1(C(C2CCN(C(c3cc(CC)oc3C)=O)CC2C)=O)CCCC2(CC1)CC2 N1(C(CCCn2c(C)ncc2)=O)CC2(CC(NC(C3CC3(C)C(F)F)=O)C2)C1 c1(C(=O)NC2CC(CNC(C=C(C)Cl)=O)C2(C)C)ccc2ccncc2c1 N1(C(=O)NC(CC(=O)NC2CC2)CSCC2CC2)CCOCC12CCS(=O)(=O)C2 C1(C(N2CCC(CCNC(C3N(S(C)(=O)=O)CCC3)=O)C2)=O)CSCC(=O)N1 N1(C(C2CCCCC(N)C2)=O)CCC2(CC1)CC2N c1(C(N2CC3(CN(C(CC(C=C)C)=O)C3)OCC2)=O)cc(Cl)c(N)c([N+](=O)[O-])c1 c1(CC)cccc(F)c1C(=O)NCC1CCCN1C(=O)CC(C)C(=O)OC N1(C(C(C)SC)=O)CC2CCC(C1)N2C(C1COCCO1)=O C=CCCC(C(=O)N1CCCC(C)(O)C1)NC(c1c[nH]nc1C)=O Cn1nc(C(=O)NCCCC2CCCN2C(=O)C=CCF)c2c1CCOC2 c1(SCC(=O)NC(c2ccccc2)CC#C)ncccc1C c1(N2CCN(N(C(C)=O)C)CC2)nc(Cn2nc(C)n(C)c2=O)c2c(n1)CSC2 c1(C(N2CCC(N(C(C3C(OCC)C3)=O)CCO)C2)=O)cc(CO)ccn1 Cc1ccc(C(N2CCCC(C)(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)c(C)n1 c1(C(N2CC(C)CC(NC(C3C(OCC)C3)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] CC1CN(C(=O)Cn2ccccc2=O)CC1CNC(c1cnccc1Cl)=O N#CC(C(=O)NCCC1CCCN1C(c1cnc(Cl)s1)=O)C1CC1 n1(CC(C)C)ncc(C(=O)NCCC2CC(NC(c3cnsc3)=O)C2)c1C1CC1 n1(CC(=O)NC(CCN(C(=O)CCc2ncc[nH]2)CCCN(C)C)CCl)cnnc1O CCCC(CC)CCC(=O)NCC(O)CC(=O)N1CCC(C#N)C1 C1(CCCNC(=O)Cn2nnc(=O)[nH]2)CCCCN1C(=O)Cn1cnnc1 CCCCCCC(O)CCC(=O)N1CCCC1C1(NC(=O)C(CC)CCOC)CC1 c1(CC)nc(C(=O)N(C)CC2CCN(C(c3cnc(O)n3CC)=O)CC2)c(C)o1 c1(OC)ccc(C)cc1C(N1CCC(C)(C)C1CNC(=O)CC12CCCC1C2)=O C1(CN(C(C2C3CCC(=O)C23)=O)CC)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 c1(C(=O)NCC(C(=O)NC2CCOC(C3CC3)C2)OC)cccc[n+]1[O-] N1(C(c2[nH]c(=N)sc2)=O)CCN(C(=O)CC2CCCC2(F)F)CC1C1CC1 C=CC1(C(=O)NCc2coc(CC)n2)CCN(C(C2CC2(F)Cl)=O)C1 C(=O)(CC(O)CN(C)C)NC(c1cccnc1)C(=O)NCCN(OC)C c1(C(=O)NC2CC(CNC(C(C)OCCOCCOC)=O)C2)cc(C(C)C)no1 C#CCCC(O)C(=O)N1CC(OC)CC1CCNC(=O)CC1COC(=O)C1 C1(C(N2CCC(CCNC(Cc3nc(C)sc3C)=O)C2)=O)CCC2CCC1O2 C(=O)(C(CC(C)(C)C)NCC(CSC)OC)NCc1ccc(OC)cc1 C(CN=c1[nH]c(=NCC2CCC2)c2cc(Cl)ccc2[nH]1)OCCOC N#CC1(C(=O)NCCCCCC(=O)N2CCN(C3CC3)CC2)CCCOC1 C1(O)(C(=O)NC(C2CCCO2)(C)C)CC(F)(F)C1 c1(CC)cccc(C(N2CCCC(C(C)NC(C3(CCOC)CC3)=O)C2)=O)c1F C#CCCCCN(C(C1CCOCC1)C(=O)Nc1ccccc1)C N1(C(C2CCC(=C)CC2)=O)CC2CCN(C(=O)CC3CC3C3CC3)CC(C2)C1 N1(C(CC2CC(SC)C2)=O)CCCC(NC(c2cc(O)ccc2F)=O)C1C c1(N2CCC(C3CCN(C(C(C(C)(F)F)Cl)=O)C3)C2=O)ccc2ccccc2c1 C(=O)(C(C)(C)COC(C)(C)C)N(CCN(C(=O)CCC1CCN(C)C1)C)C C12(NC(c3ccc(O)nc3Cl)=O)CCCC1N(C(=O)C(O)(C1CC1)C1CC1)CC2 C1(C(N(CC)Cc2ccsc2)=O)CCCN(C(=O)CCc2ccoc2)C1 C1(NC(C2C(COC)C2)=O)C=C(C)CCC1 c1(C(=O)OC)ccc(C#N)cc1C.N12CC3C(C1)N3C(=O)c1csc(c1)C2 N1(C(C2(CC)CC2(F)F)=O)CCC2(CCCC2NC(=O)CC2CC=CC2)CC1 C1(C(CO)NC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)Cc2ccccc2)CC1 C1(CC(=O)NC2CC2)CCCN(C(C2CCCCCCC2)=O)CC1 c1(SCC2C(C(=O)NCCNC(C3CCS3(=O)=O)=O)C2)nc2ccccc2s1 C#CCC(O)C(=O)NCC1CCN1C(c1ccc(C(F)(F)F)[nH]1)=O C1(Cl)(C(=O)NCC(C)N(C(CC2(NC(C)=O)CC2)=O)C)CC1C(C)=O c1(C(N(C2CCN(C(=O)CC3COCCO3)C2)CC)=O)ccc(C)c(F)n1 c1(C(N2CC3C(CNC4CCC4)C3C2)=O)ccccc1Br.C12(C=O)CC(F)(C1)C2 c1(CC)ccccc1C(=O)NC(C1CCCN1C(=O)CCC(=O)OC)C c1(C(C)=O)cnc(C2CN(C(C3CCCC3c3cnn(C)c3)=O)C2)cn1 c1(NC(C(C)N(C(C2CCCC(OC)C2)=O)C)=O)cc(C)ccc1F c1(OC)ccc(CC(N2CC(OC)C(NC(C3(N=[N+]=[N-])CC3)=O)C2)=O)c(Cl)c1 C(=O)(CC(C)CNC(c1c[nH]nc1CNC(=O)CC1C(=O)NN=C1C)=O)NC CC(C)(C)C(C)(C)C(=O)NCCN1CCN(C(=O)C#CC2CCCC2)CC1 C12(NC(=O)CC3CCC4CC34)CCCC1N(C(c1cnc3n1CCC3)=O)CCC2 CC1OCCC1NC(=O)CONC(=O)CN1CC2CC2C1 c1(CN2C(C(=O)Nc3ccnn3CCO)CCCC2)c(O)ccc(F)c1Br N1(C(CC=C=C)=O)CC2CC2(NC(c2cnc(S)nc2)=O)C1 Cc1cccc(C(N2CCC(N(C)C(C3(C)CCN(C)C3=O)=O)CC2)=O)c1C C1(C(N(CCCNC(=O)CC(=O)N(C)C)CC)=O)CCCC(C(=O)OC)C1 C=CCC(C)(C)C(=O)N1CCC(NC(=O)Cn2ncn(C)c2=O)C(C(N)=O)C1 c1(OC)c(C(N2CCC(Cc3ccccc3)CC2C2CC2)=O)cc(Cl)cc1Cl C(=O)(C(F)(F)Cc1ccc(F)cc1)NC1CC(CNC(C=CC=CCC)=O)C1 n1(CC)ccnc1C=CC(=O)NC1CN(C(=O)CCC2CC2(F)F)CC1F Cc1nc(C(C)C2CC2)sc1C(=O)NCCCNC(=O)CCNC(N)=O CC#CCC(C(=O)NCC=CC)NC(C1CC=CCO1)=O C1(NC(C(COC)OC)=O)CC2CCC(C1)N2C(C1CCCC1(C)C)=O C1(C(=O)N(CC(=O)NC2CC(C(N)=O)C2)C)(COC)CCC1 C1(C(N2CC(CC(N)=O)C2)=O)CCN(C(=O)C2CCC3(CCC3)O2)O1 c1(CC(=O)NC2CC3CC(NC(C(CC)SC)=O)C2C3)c(C)cc(OC)cc1C C=CC1CCCN1C(=O)NC1CC1c1ccccc1OC(F)F C1(C(=O)NCCN(C2CCCCC2)C(=O)C(C2CCCCC2)O)CC2CCC2C1 c1(OC)cc(-c2nc(-c3cncnc3)nn2CC2CCSC2)n(C)n1 O=C(C#CC1CCCOC1)NCC1CCCCN1C(=O)CCc1ccc(Cl)cc1 c1(C(=O)NC(C(C)NC(=O)C(C)(C)CN2CCOCC2)C)cnn2c1N(C)CC2 c1(CN2CCC(N(C(CCCC(C)=O)=O)C)C2)ccccc1S(C)(=O)=O O=C(C1=CCCCO1)NCC1(O)CCN(C(=O)CCC=Cc2ccccc2)C1 CCC(C)(C)C(=O)N1CC(CNC(c2cncnc2-c2ccccc2)=O)C(O)C1 CC(C)C(C(=O)N1CCCC(CN(C(=O)C(F)(F)C2CC2)C)C1)c1cccnc1 c1(CC)ccc(O)c(NC(=O)CC(CC)NC(c2cc(C(N)=O)[nH]n2)=O)c1 C1(CC(=O)NCC(=O)N(C2CN(C)C2)C)CCCN1C(C1CC1F)=O CCC(O)C(F)(F)C(=O)NCC1CN(C(=O)CC2CCC3CC23)C1 C1(C(=O)NC2CCC(NC(c3ocnc3C(F)(F)F)=O)CC2)CC2COCC2C1 CCCC(C)(C)C(=O)N1CCCC(NC(=O)C(O)CC2CC2)CC1 c1(-c2nc(C)on2)cccc(NC(C2(F)CCN(C(C3(F)CC3)=O)C2)=O)c1 C(CCCCCCn1cc(CCCCCO)nn1)NC(C1CC(=O)N1)=O C(=O)(C#CC1CC(F)(F)C1)N1C(C(C)NC(c2ccc(N)cc2Cl)=O)CCCC1 n1(CC(N2CC(N(C(=O)C3=CCOCC3)C)C(F)C2)=O)ncn2nccc2c1=O C(c1cccc(F)c1Cl)=CC(=O)N(CC(C)(C)NC(C1C(OC)CCC1)=O)C CC1(NC(C23CC(F)(C2)C3)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 n1(CC)nc(C(=O)NCC(CNC(=O)C(F)n2ccnc2)CO)cc1C C(=O)(C1CCc2c[nH]nc21)N(C(N1C(Cc2ccc(OC)cc2)CCC1)=O)CC C1(C(=O)NC2(CO)CC(C)C2)CC(NC(=O)CS(C)(=O)=O)C12CCC2 c1(C(N(C2CCN(C(=O)CCCc3ccc(F)cc3)CC2)C)=O)ccccc1Cl c1(C(=O)NCC(C)(C)CNC(=O)CCc2cncnc2)cc(Cl)c([N+](=O)[O-])[nH]1 c1(CC(=O)NC2(CN(C)C(C3CN4CCN3CC4)=O)CC2)c(F)cccc1C#N n1(CCC)cc(Cl)c(C(=O)NC2CCN(C(=O)CC3OCCC3C)C2)n1 Cc1cc(=O)n(C)nc1C(=O)NCCNC(c1cccc(Br)c1F)=O c1(N(C)Cc2ccsc2Br)nc(NCCC2CCOC(C)C2)c2cnn(C)c2n1 C(=O)(CCC(C)(C)C(=O)c1cccc(OC(c2ccc(Cl)c(F)c2)C)c1)OC C1(NC(C(CC)OCC)=O)CC2CC(NC(c3cccnn3)=O)CC12 C=C1CCN(C(c2cnn(CCNC(c3ncoc3C)=O)c2)=O)C1 C(=O)(N1OC2CCC1C2)C1(NC(Cc2c(C)ccnc2)=O)CCC1 Cc1ncc(C(N2CC(CNC(=O)CCOCC3CCC3)CC2C)=O)cc1Cl c1(C(N2CC(OCCNC(c3cc(C(C)C)[nH]n3)=O)C2)=O)ncccc1C1CC1 N1(C(c2c(C)cc(CC)o2)=O)CCCC(C)(C(=O)NCC2(C(C)(C)OC)CC2)C1 c1(C(=O)N(CC(O)C(F)(F)F)CCO)nc2ccccn2c1-c1cnc2[nH]cnc2c1 c1(CC(C)C)cc(C(N2CCCC2CN(C(C)C)C)=O)cc(O)n1.C1CC1 c1(N2CCCC(C(CC)NC(C3CCCC3OC)=O)C2)nccc(S(C)(=O)=O)n1 C1(C)(C(=O)NCC=CCSC)CCN(C(C2CN(C)CCO2)=O)CC1 c1(N(C)C=O)ccc2n[nH]c(C(C)C)c2c1.c1(SC)cccc(-n2cc(CN)nn2)c1 c1(C(C(=O)N(CCC)CC=CCC(C)C)OC)ccccc1.C(=O)(COCCOC)N C1(NC(CCOCC#C)=O)CCCN(C(c2ccc(OC)c(Br)c2)=O)CC1 C1(C(N2CCC(C)C2CNC(c2cccc(CCO)c2)=O)=O)CC2(C1)OCCO2 c1(C(=O)OCC)nc(=NCC2CC(NC(C3(C(F)F)CCC3)=O)C2)[nH]cc1Cl C1(CNC(C(C)(C)OCC)=O)C(C)CCN1C(=O)CCC1OCCO1 C(=O)(C(CNC(C1OCCC1(C)C)=O)C(C)(C)C)N1C(C)(CC(=O)NC)CC1 C1(CNC(c2ccc(C=C)cc2)=O)CN(C(=O)C(COC)N(C)C)C2(CCC2)C1 CC1CC(NC(C2CC(O)C2)=O)CCN1C(c1cccc(C(F)F)c1Cl)=O c1(OCC)ncc(C(c2nnnn2C2CCOCC2)NCCc2ccc(C)s2)s1 C(=O)(CCCCC(C)C)NC(CC=C)CC(=O)NC(c1cnco1)C C1(C(N2C(C)(CNC(c3ccc(C#N)o3)=O)CCC2)=O)Cc2cccnc2C1 C=CCCC(=O)NC(C1CC=CCC1)C(=O)NC(c1nc[nH]n1)C1CC1 C1(C(C(=O)NCCCCC2CN(C(C3CC(F)(CO)C3)=O)C2)F)CCCCCC1 N1(C(C(C(C)C)F)=O)CCC(C2CCCN(C(c3ccc(F)o3)=O)C2)CC1 c1(C(=O)OC)ccc(NC(=O)CCc2cc(C)ccc2C)cc1OC(C)C c1(CC(=O)NCC2C(NC(C(C)c3ccco3)=O)CC2)sc(O)nc1O C1(CC=C)(NC(C2COCCC2(F)F)=O)CCCN(C(=O)CC(C)(C)CC)C1 N#Cc1ccccc1C(=O)NCC(CC(=O)N1CCCC1C(N)=O)C1CCC1 CCC(C)CCCCC(=O)NCC1(NC(=O)CCOC(C)C)CC1 C1(O)(CNC(C(F)=CC)=O)CC(NC(=O)C(O)c2ccco2)C1 c1(C(N2CCC(C(C)(C)C)(CNC(C(CSC)C)=O)C2)=O)cc(C)c(CO)cn1 c1(C(C(N2CC(N(C(c3c(C)n[nH]c3)=O)C)C2)=O)C)cc(Br)ccc1F C1(C)(N(C)CC)CN(C(=O)C(C)(C)C2CCN(C(=O)CCN(C)CCO)C2)C1 C1(C(=O)NCc2c(C(N3CCC(SC)C3)=O)scc2)CCCC(=O)C1 c1(OCCC(=O)N(C(C)CNC(C2CC3CC2C3)=O)C)ccc(S(C)(=O)=O)cc1 C(=O)(C(C)C(C)COC)N(CCCNC(CCC)=O)C(C)C.c12ccc(cc1)s2 N1(C(C2(OC)CCCC2)=O)CCC(NC(=O)Cn2cncn2)CC(C)(C)C1 C1(C(=O)NC2CC(C)(NC(c3cnc(OCC)s3)=O)C2)CCCCC1(F)F c1(C(N2CC3C(NC(c4c(Cl)ccc(NC)c4)=O)(C3)C2)=O)cc2ccccc2[nH]1 n1(CC)cc2ccc(C(=O)NC(C)C(C(C)C)NC(c3c[nH]cc3C)=O)cc2n1 c1(Nc2cccc(SC)c2)ncnc(NC(C)C(C)Oc2ccccc2F)c1C c1(CC)nc(C)c(C(=O)NCC2(F)CCC(CNC(c3n[nH]cc3CC)=O)C2)s1 C(CCCC(=O)NCC1C=CCN1C(=O)CC1CC1c1ccccc1)OCC C(=O)(C1=C(Cl)CCCC1)NCc1ccc(C(=O)NC2CCN(C(=O)C3CC3)CC2)s1 Cc1ccccc1SCC(=O)NCC1CC2CC2N1C(=O)Cc1sc(O)nc1O c1(COCC)nc(C)c(C(N2CCC(CNC(c3csc(CC)n3)=O)CC2)=O)s1 CCCC(CCCNC(c1sccc1C(C)C)=O)NC(=O)C(C)C(F)F N1(C(CCCSC)=O)CCC(C(C)NC(=O)CC2CCC=CCC2)CC1 c1(C(=O)NCC(C(C)(C)C)NC(C2C(C(C)C)CCC2)=O)cccc2c1OCO2 Cc1nnc2n1CCCC2C(=O)NC1CCN(C(=O)CCCC#N)CC1 N1(C(c2ccoc2Cl)=O)CCC2CCCN(C(=O)COCC(F)(F)F)C2C1 N1(C(=O)CC2CC2)CC2C3CCC(C2C1)N(C(=O)CC(=O)NC1CCOC1)C3 c1(CC)ccc(NC(=O)C(F)CC2CN(C(=O)CCC3CC3C)C2)cc1O C=CC1(C(=O)NCC[Si](C)(C)C)CCN(C(c2ccn(CCC)n2)=O)C1 N1(C(CCC=C)=O)CC(NC(=O)C(C)(O)C(C)c2ccccc2)CC2(CC2)C1 c1(CCCC(=O)N(C(CNC(CC(CC)C)=O)C2CC2)C)nc2ccccc2o1 C1(C(=O)NCc2ncnn2C(C)C)(COC)CN(C(c2cccn2C)=O)C1 C#Cc1ccc(OC)c(C(N2CCC(NC(=O)C(C)(C)C3CCCO3)C2C)=O)c1 C(C(C)C)(C(O)C(=O)NC1CC2(C(=O)N(C)Cc3ccn(C)n3)COC1C2)OC C1(C(=O)NCC2(O)CCN(C(Cc3cc(C)no3)=O)CC2)Cc2cccnc2C1 CC(C)C1C(=O)N1.c1(NC(=O)OC(C)(C)C)cn(CC(F)F)cn1 C(=O)CCC(C)(C)F.N1(C(C(CC2CCC2)N(C)C)=O)CCCCC1C1(O)CC1 c1(NC(C2N(C(CCC3C(C)(C)C3)=O)CCCC2)=O)cccc(C#N)c1 N(C1CCCn2nncc21)CC(C)NC(C1CCN(C(=O)N(C)C)CC1)=O C12(NC(C3CC34CCOCC4)=O)CCCC1(F)CN(C(=O)C(F)(F)C(F)F)C2 c1(C(=O)OC(C)(C)C)cncc(C(=O)OC(CC)C(=O)N(CC(C)C)C)c1 Cn1cnc(CNC2(CNC(C)(C)CC3CCC3)CC2)cc1=O C1(c2ccccc2)(NC(C=CC=CCC)=O)CC(NC(=O)Cc2ccoc2)C1 C1(NC(c2c(CC)scn2)=O)CS(=O)(=O)CC1NC(=O)CCCn1cc(C)cn1 C1(N(c2nc(C)c(CN)s2)C(C)=O)CC(=O)N(C(c2ccccc2)C)C1 C1(C(N2CC(C(C(=O)NC(C)(C)C(F)F)OC)C2)=O)CC(N=[N+]=[N-])C1 N1(C(CC2N(C(CC3CCC(C)CO3)=O)CC2)=O)CC2CN(C)CC2(C)C1 C(=O)(C1CCc2ccccc21)NCC(CNC(=O)COC1CCCOC1)OCC Cc1cc(C(N2CC3CC3(CNC(C34CC(C3)C4)=O)C2)=O)cc(C)c1Cl c1(C(N(CCC(=O)N(CC(C)C)C)C)=O)ccc2occc2c1 C(=O)(C1CCCc2nncn21)N1CCCC(NC(C=Cc2c(C)coc2C)=O)C1 c1(C(=O)NCC2N(C(COc3c(F)ccc(C)c3)=O)CC2)cnc2[nH]nnc2c1 C1(C(N2CC(C(N)=O)C2)=O)COCCN1C(=O)CCc1cncnc1 c1(C(N2C(CC)CN(C(=O)CN(C)C)CC2)=O)cc(Br)cc(F)c1O C(=O)(CCCC(C)(C)C)N1C(CN(C(c2nc(O)nc(O)c2F)=O)CC)CCC1 c1(C(N2CCC(N(C)CCc3c(F)cccc3F)C2)=O)ccc2cc[nH]c2c1 C1(NCCc2ncn(CC)c2)CCNC2CC12 c1(N2CCC(C(F)(F)F)(OC)C2)nc(C)cc(=NCC2(S(C)=O)CCC2)[nH]1 C1(NC(c2c(C)cc(F)cc2)=O)C2COCC1CN(C(c1ccc(C#N)[nH]1)=O)C2 CC1(C)CCN(C(=O)C(N)=O)C(C(=O)NC2(C)CCC(=O)NC2=O)C1 c1(C(C)C)nc(NCC(C)C(F)F)cc(=NCc2cncc(C(F)(F)F)c2)[nH]1 c1(N2CCC(C)C(NC(=O)CCC(N)=O)C2)nccc(S(C)(=O)=O)n1 N1(C(C2CC(OCC)C2)=O)CCC(CN(C(=O)C=CC2CCCN2C)C)CC1 N1(C(CC(c2ccco2)C)=O)CC(C(=O)OCC2CC3C(C2)C3(C)C)CC(O)C1 c1(CC(=O)NC2CC(F)(CNC(=O)CCC3CCCO3)C2)ccc(O)cc1 c1(CC)ccc(C(N2CCOCC2CC(=O)NCC2COCCN2C)=O)cc1N CCC(F)(F)C(C)(C)C(=O)NC1CCCC1CNC(C1(C2CC2)CC=CC1)=O C1(CNC(c2cc(C)cc(Cl)n2)=O)CC2COCC2N1C(C1CCCS1(=O)=O)=O C(CC1CCC1)(CC(=O)N=c1ccn(C2CC2)[nH]1)NC(C1C(C)CCOC1)=O C=C(C)C(C)(O)C(=O)NCC(O)CNC(c1cc(OC)ccc1Br)=O c1(C(=O)NCC=CC(=O)NCC(C)Cn2cccn2)csc2cc(Cl)cnc12 c1(CN(CC(=O)OCC)C(=O)NCC2CC2)ccc(Br)o1 N1(C(c2c(C)snc2)=O)CCC(C)N(C(c2cc3ccncc3o2)=O)CC1 N1(C(c2c(OCC)cccc2)=O)CCN(C(c2[nH]cnc2CC)=O)CC2(CC2)C1 Cc1nn(C(C(CO)NC(=O)COCC(C)C)C)c(C)c1C c1(CC)cc(C(F)(F)F)ccc1C(=O)NC1CCCN(C(=O)C(C)(C)N(C)C)C1 CC(C)(CC(=O)NCC1CCCN(C(c2occc2Cl)=O)CC1)CC(F)F c1(N2CC(C)(NC(CCNC(=O)NC)=O)C2)c(C(N)=O)cccc1[N+](=O)[O-] c1(C(N(C)CC2CCN(C(C(C(C)(C)C)OC)=O)C2)=O)cnc2ccncc2c1 Cc1c(C(N2CC(O)C(F)C2)C(=O)NCC2CCOC2)ccnc1F C(=O)(CC1=CCCCC1)N1CCCC(NC(C2CC(=O)N(c3nccs3)C2)=O)C1 C12(C(N3CC4C(CNC(c5c(C)ncs5)=O)C4C3)=O)CC3CC(C(=O)N1)C2C3 C(=O)(CC1COc2cc(O)ccc21)N1CC(O)(CNC(c2c(CC)[nH]cc2)=O)C1 C#CCC(C)(C)C(=O)NCC(C)(CC)NC(c1cc(C(N)=O)no1)=O Cc1nc2ccc(C(N3C4CC3CN(Cc3cccc5[nH]ncc35)C4)=O)cc2[nH]1 c1(OC)cnc(C(N2CCC3C(NC(c4ncccc4OC)=O)CC23)=O)c(F)c1 Cc1ncc(Cl)cc1C(N1CC2CC(NC(=O)Cc3cc(O)nnc3O)C1C2)=O c1(C(N2CC(CC)N(C(=O)CC(C)F)CC2)=O)ccc(C#N)c(O)c1 C(N=c1cc(C(N)=O)nc[nH]1)c1occ(C(N)=O)c1 C1(CNC(CC)=O)CN(C(=O)CCCC2CCCC2)CCC1CO c1(C(N2CCC(O)(CC(=O)OC)C2)C(=O)NCC)nn(CC(F)(F)F)cc1C C(=O)(C(O)CN1CCCC1)NC1(C)CSC1.N12CC(C1)C2=O C(c1c(Cl)nc2sccn12)=CC(N1CC(NC(c2cc[nH]n2)=O)C(CO)CC1)=O N12CC3=C(C1)CN(C3)C(=O)C1(CCOCC1)N(S(C)(=O)=O)CCC2=O.C1(CO)CC1 Cc1cnc(F)cc1C(=O)NC1CCC(NC(=O)C(C(C)C)OCC(C)C)CC1 C(=O)(CCCCC(F)F)N1CCCC(NC(C=Cc2nnn(C)n2)=O)C1 C1(C)(C(=O)NC(CC(C)NC(c2c(C)ncs2)=O)C)CCc2ccccc2N1 C1(NC(C(CC)c2ccccc2)=O)CCN(c2ncc(C3CC3)cn2)CC1 C1(NC(C23CC(NC(=O)CC4CCSC4)(C2)C3)=O)CCc2nn[nH]c2C1 C1(CNC(C(N2C(CC(=O)N(C)C)CCCC2)=O)=O)CC2CCCC(C1)C2 C1(C(=O)NC(CNC(c2cc(C(=O)OC)ncc2)=O)C2CC2)CC2CCC(C1)C2 c1(OC)ncc(C(=O)NC2COCC2CNC(=O)Cn2ncn(C)c2=O)c(C)n1 CCC(CC(F)F)C(=O)NCC1CCN(C(c2cc(C(N)=O)cc(C)c2)=O)CC1 C1(NC(c2oc(C3CC3)nc2C(F)F)=O)CN(C(C2CCCN2C2CC2)=O)CC1O c1(C(C(=O)N)OC)ccc(SCC)cc1.c12ccoc1CC1(CC1)C(=O)N2 c1(OC)ccc(CC(N2CCCC2(C)C(=O)Nc2c(Br)ccnc2Cl)=O)c(Br)c1 C1(C(NOC(CC)CC)=O)CCOCC1NC(c1oc(CO)cc1C)=O C1(C)(C(=O)Nc2cn(C(C)(C)C)nc2)CCN(C(c2ccncc2)=O)C1 c1(OC)ccc2cc(C(=O)NCC3CC3CNC(c3ccc(C)cn3)=O)sc2c1 C12(C(N3CCC(N(C(Cc4cc(CC)no4)=O)C)CC3)=O)CCCC(C1)OC2 C1(C(N(C(CCNC(C(C2CC2)OCC)=O)C)C)=O)CCCC2(CCC2)O1 C1(C)(OC)CN(CC(=O)NCCOC2CN(C(=O)C(=Cc3cn[nH]c3)C)C2)C1 C(CC(C)C(=O)N(CCC)CCNC(C1CC(=O)N(C2CCCC2)C1)=O)=CCC c1(SCCC)nc(Cl)c(CNC(=O)CC2COCCN2)c(Cl)n1 N1(CCC(N2C(CN(C(=O)C=Cc3ccco3)CC)CCC2)=O)CCC(C)CC1 C1(C(=O)NCCCN(C(C(Br)=C(C)C)=O)C2CC2)CCN(C2CC2)C1=O C12(NC(C(C)N(C)CC3CC3)=O)CC1CN(C(c1sccc1-n1ccnn1)=O)C2 C12(CNC(C(=O)NC(C)C(C)(C)CO)=O)CCC(CC1)C(C)O2 CC1CCN(C(=O)CNC(=O)C=CCN(C)C(C2(CCF)CCC2)=O)C1 C(N=c1[nH]c2c(c(=NCC3CC34CCOCC4)[nH]1)CCC2)c1cc(C(C)C)n[nH]1 C(=O)(C(C)(C)COCC(F)F)NC(C)C(C)NC(c1ccncc1F)=O N1(C(C(c2ccc(C)cc2)C)=O)CCC(C2CN(C(C3(C(C)C)CCC3)=O)C2)C1 N1(C(CC(CC)C2CCC2)=O)CCN(C(c2ccc(C)nc2C)=O)C(CO)C1 c1(C(N(C2CN(C(c3ccc[n+]([O-])c3)=O)C2)C)=O)ccc2c(C#N)c[nH]c2c1 C1(C(=O)NC2CCN(C(C3CN(C(C)=O)C3)=O)C(C)C2)CCc2c(cnn2C)C1 N1(C(C2OCCC(NC(c3c(Cl)cn(C)n3)=O)C2)=O)CC2CCC(O)CC2C1 C1(CNC(N2CCN(c3snc(C)n3)CC2)=O)CCOC2(CCC2)C1 C1(NC(C2CCC(C)O2)=O)CCC(NC(=O)COCC(N2CCCC2)C)CC1 C(=O)(C(O)C(F)(F)F)NC(CNC(=O)CCCCN1CCOCC1)(C)CC1CC1 N1(C(CC2C(C)OCC2)=O)CC2CCN(C(=O)CCCC3CCC3)C2C1 Cc1cc(C(F)(F)F)cc(C(=O)NC(C)CC(C)NC(=O)C=CC2CCCC2)n1 C1(CC(=O)NCC2CCCN(C(=O)COc3cnn(C)c3)C2)(OC)CCCCC1 C(=O)(C(CC(N)=O)NC(=O)CC1CC(=O)C1)NC1CCN(C(C)=O)CC1 c1(C(=O)NCC(C)C(F)C(=O)NCc2conc2C2CC2)cncc2[nH]ccc12 c1(C(=O)NC(C)CCNC(c2ccc3c(c2)COC3)=O)ccc2c(c1)C(C)CO2 N1(C(c2cnc(N(C)C)c(Cl)c2)=O)CC2CC1CCC2NC(c1cc(Cl)no1)=O N1(C(CCCOCC)=O)CCCC(C2CN(C(=O)C(CC)CC(F)F)C2)C1 CC1CCN(C)C(=O)C1NC(=O)C(=O)NCC1(F)CCCCC1 c12ccccc1CC(=O)NC(C)CN(C)C2=O.C1(CC#C)(C(=O)OC)CCCC1 C=C(C)c1cn(C2CC3CC2CC3N(CC(OC)OCC)CC)nn1 c1(CC(=O)OCC)nc(C)c(C(N2CCC2CNC(c2ccon2)=O)=O)s1 c1(C(=O)NC2C(C)CN(C(=O)CC3CCCCO3)C2)c[nH]c2ncccc12 C1(C)(CNC(CC(C2CC2)OC)=O)CCC(NC(=O)CCOCCOC)CC1 CCCC(O)(CNC(=O)Nc1c(Cl)cccc1Cl)CCC C(=O)(C(CC(C)(C)C)NC(=O)Cc1ccnn1C)NC(CC(C)C)CO c1(CCC(=O)N(CC(CC)NC(C2CCC(=O)O2)=O)C)cncc(F)c1 CCCCCC(O)CC(=O)NC1(C)CC(NC(c2coc(CCC)n2)=O)C1 c1(-c2nc(C(c3cn(CCCCC)nc3C)O)on2)cccc2cccnc12 C(=O)(C1=C(C)N(C)c2ncnn2C1)N(C1CCN(C(c2c(CC)c[nH]c2)=O)C1)C N1(C(CCSC)=O)CCC(C2CCN(C(c3cncc([N+](=O)[O-])c3)=O)C2)C1 C(C(CCCC)NC(=O)Cn1cccn1)NC(C(F)=CCC)=O C(CCO)(C(=O)N1CCOC(CCNC(C2(C(F)(F)F)CC2)=O)C1)N(C)C C1(C(=O)NCC(C)(C)OCC(=O)NCC2(C)CCCO2)COCCC1(F)F Cc1nc2ccccc2cc1C(=O)NC1COCCN(CC2(C(=O)NC)CC2)C1 N1(C(=O)CC2CCC=CCC2)CCCC(C2CN(C(C3C=CCC3)=O)C2)C1 C(=O)(C1CCCn2nccc21)NC(CNC(C1N(CC)C(=O)CC1)=O)CC(F)(F)F N1(C(CSCC=C)=O)CCC2(C1)OCc1ccccc12 C1(CNC(Cc2c(C)ccs2)=O)CC(C)(C)CN1C(C1CC12CCOC2)=O CCCC(CNC(=O)Cn1nc(C)nc1C)C(=O)N1CCC(C(=O)OC)C1C C1(C(N(C)CC2CCCN2C(=O)CC2CCC(=O)C2)=O)CC12CCOC2 N1(C(C=CCC)=O)CCC(C(N2CCC(C(C)C)(CN(C)C)C2)=O)C12CC2 C(C)(CCOC)NC(CN(C(=O)CNC(=O)CCOC(C)=O)CC)=O c1(CNC(C(c2cn(C)nc2)O)=O)nc(C)c(C(=O)NCCCC(F)F)o1 c1(NC(C(c2ccco2)NC(C2CC=CCO2)=O)=O)ccc2nccn2c1 CC(C)C(F)(CNC(C1CCC2(CCC2)C1)=O)C(=O)NCCCN(CCO)C c1(-c2cc(C(=O)NC3CC(N(C(CCC=C=C)=O)C)C3)on2)cccc(C#N)c1 C1(CNC(C(C)SC)=O)CCN(C(=O)CNS(=O)(=O)CC)CC1(F)F C1(NC(C(c2c(Cl)cccc2Cl)C)=O)CCN(C(=O)CCF)C12CCC2 Cc1cc(N)n(CC(N2CC(CNC(c3sccc3C3CC3)=O)C(C)C2)=O)n1 C1(CC)CCN(C(c2cc(C(C)C)oc2C)=O)C1CNC(C1CC2CC2C1)=O C1(C(=O)NCC(C)NC(c2[nH]c(=N)sc2C(F)(F)F)=O)(COC)CC=CCC1 N1(C(CC=CCC)=O)CCC(C)CC1CNC(=O)Cn1ccc(C)cc1=O C(c1ccccc1F)=CC(=O)NCC(CC)(C)NC(c1ccoc1C)=O c1(OCC(=O)NC)cccc(CC(=O)N(C2CN(C(C3SCCC3C)=O)C2)C)c1 N1(C(C(c2ccc(C)s2)C)=O)CCC2(CCC(NC(=O)CCC3CCC3)C2)CC1 C1(CC(=O)NCc2cc(O)cc(F)c2)CCC(F)(F)C(=O)N1 C(=O)(C(F)=CCOC(=O)N)N=CCCC.C=C C1(N(C)C(c2ccc(C3CCOC3)s2)=O)CN(C(=O)C(F)F)CC1F CP(C)(=O)c1cnc(C(N2CCN(C(c3sc(C#N)cc3Cl)=O)CC2)=O)nc1 CC12CN(C(c3cnc(C4CC4)[nH]3)=O)CC1(C)CN(C(C1CC(=O)N1)=O)C2 C#CCCCCCCC(=O)NCCOCCC(=O)N1CC(SCC)C1 C12(CNC(c3ccc(OCCC)cc3)=O)CCCC1CC(=O)N2 C(c1ccc(C)cn1)=CC(=O)NC1C(NC(C(CCC)C)=O)C1 C1(C2(O)CN(C(=O)CC3(CO)CC3)C2)(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 C1(C(N2C(C(=O)NCC(C)C#N)CSCC2)=O)CC2C(C1)C2(F)F c1(NC)cccc(C(=O)N(C(C)CCNC(=O)CC2CC(N(C)C)C2)C)n1 C1(NC(c2c(CC)csc2)=O)CCCN(C(c2cnc(OC(C)C)cn2)=O)C1C C1(CNC(C(C=C)O)=O)CN(C(=O)C(O)CCSC)CCC1C N1(C(C(C)SC(C)C)=O)CC2C(NC(=O)C=CC(=O)N(C)C)C2C1 c1(C(C(=O)NCCCOC)N(C(CC)CC)C)c(C)noc1C c1(C(N2C3C(N(C(C(COC)C)=O)C)CC(C3)C2)=O)ccsc1S(C)(=O)=O c1(NC(c2cc(-c3nc[nH]n3)ccc2F)=O)c(F)cc(F)cc1Br C1(CC)CCN(C(C2CC2CCOC)=O)C1C(=O)NCC1(F)CC1 c1(C(=O)NC2(CCOC)CCN(C(=O)C=C(C)C(F)F)C2)cn(C)c(=O)nc1O c1(NCC(C(C)C)O)ccc(S(=O)(=O)N2CCC3C(O)CC23)c2ccncc12 C1(N)C2CN(CC3(c4ccc(O)nc4)CC3)CC12.Cn1cc(C(=O)C(=O)C(C)=O)cn1 c1(C(N2CC(c3cn(C(C)CO)nn3)N(C)CC2)=O)cccc2c[nH]nc12 c1(C(N2C(C(CNC(C(CC(C)C)C)=O)(C)C)CCC2)=O)cccc2c1NCC2 C(=O)(C=CS(C)(=O)=O)NC(C)CCNC(=O)CCC1NC(=O)NC1=O Cc1ccc2c(CC(N3CC(CNC(C4C=CCCC4)=O)C(C)C3)=O)c[nH]c2c1 C(c1ccccc1F)=CCC(N1C(C(C)NC(C2CCCS2(=O)=O)=O)CCC1)=O N1(C(c2c(OC)c(Cl)sc2)=O)CC(NC(c2ccnn2C)=O)CC(O)C1 N1(C(=O)CCc2ccc(F)c(F)c2)CCC2(CC(NC(=O)C(F)(F)CF)CO2)C1 N1(C(C2(C)CN(C(CC3C(C)(C)C(O)C3)=O)C2)=O)CCC12CC(C)(CO)C2 C1(NCCNC(=O)NCc2cnn(Cc3ccccc3)c2)C2CCCCCCC12 C12(C(N(CCNC(C3(C(N)=O)CC3)=O)C3CC3)=O)CCCCC1CS(=O)(=O)C2 c1(C(=O)Nc2nc(CNC(C)CC3CCCCO3)[nH]n2)ccc(Cl)cn1 C(=O)(C(C)(O)C(F)(F)F)NCCN(C(C(n1ncc(C)c1)C)=O)C c1(C(=O)NC2C(NC(=O)CN3CCOC3=O)CC2)ccn2nnnc2c1 Cc1ncc(C(N2CCC(CCC(=O)NC(C)CC(N)=O)C2)=O)c(=N)[nH]1 CC(C)C(F)(CNC(=O)CCN(C)CCO)C(=O)NCc1cocn1 CCC(C)C(C(=O)NC(CN=[N+]=[N-])C(=O)NCC1CC(C2CC2)=NO1)N(C)C CC(=O)CCCC(=O)N1CCN(C(c2csc(C)c2N)=O)C(CC(F)F)C1 CC1C(C)N(C)CCN1C(=O)C(CCF)NC(C12CC(CO)(C1)C2)=O c1(CN(C(=O)C(=O)NCC2CC3CCC2C3)CC=C)ccc(F)cc1 c1(C(N(CC(C)CNC(C2CC23CC(F)(F)C3)=O)C)=O)cccc2[nH]ncc12 C1(C(=O)NCCC(=O)NCC)CCCC(C(=O)NCCOc2ccncc2)C1 N1(C(COc2c(CC)cccc2)=O)CC2(C1)CN(C(=O)C(C)(C)CC1CC1)C2 N1(C(CC2(C)CCCO2)=O)CCCC12CCN(C(c1csc(F)c1)=O)CC2 CC1C(NC(=O)CCc2cc(F)cc(F)c2)CCCN1C(C1CN(C(N)=O)C1)=O Cc1nn2ncccc2c1C(=O)NCC(C)N(C(=O)CC(=O)NCC(F)(F)F)C Cc1ncc(CCC(=O)NCC23CC(NC(=O)C(F)CC4CC4)(C2)C3)o1 c1(C(N2CC(O)CC2CNC(C2(CC(F)F)CCC2)=O)=O)cn2ncccc2n1 c1(C(=O)NCC(C)CN(C)C(c2nn(C)cc2[N+](=O)[O-])=O)nc2ccccc2[nH]1 c1(CC(=O)NC23CCCC2CN(C(=O)C2=CCCS2)C3)ccc2c(c1)CCCC2 N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(=O)CC2CNC(=O)C2)CC12CCC2 C(C(C(=O)NC1CCCCC1NC(C1CC2CC1C2)=O)C(C)(C)C)OCC=C N1(C(COc2c(C)cccc2)=O)C2CC1CN(C(=O)CCC(C)(C)F)C2 c1(C(N(C2CN(C(C(CC)OC)=O)CC2O)C)=O)cc2cccc(C)c2nn1 c1(C(N2CCC3(CCCN3C(=O)C3CC3)C2)=O)c[nH]c2cc(Cl)c(Cl)cc12 Cc1cc(Cl)c(C(N2CCC(O)(CNC(C3COC(=O)N3)=O)C2)=O)cc1F CC(C(=O)N1CC(NC(C2(CCF)CCOCC2)=O)C(F)C1)C(C)(F)F N1(C(c2c(OC)csc2)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC1CC(F)F C(C(F)(F)F)(C(F)(F)F)c1n(C(c2ncc(-n3ncc(C)c3)cn2)C)ccn1 C1(C(N2CCCC(CCO)C2)=O)CC(F)(F)CN1C(c1nccs1)=O c1(N2CCCC(Nc3c(-c4ccc(Cl)cc4)cccc3)C2)cc2ncnn2cn1 CCC(CC(=O)NC(C(=O)NOC(CSC)CSC)C1CC(CO)C1)C1CCC1 CCCCCCC(F)C(=O)NC(C)CN(C)C(c1cn(C)[nH]c1=N)=O N1(C(C2(N(C(=O)Cc3cccc(Cl)n3)C3CC3)CCC2)=O)CCOC2CC12 N1(C(C2CC(OC)C2)=O)CCC(C(C)(C)C)(CNC(=O)CN2CCC(C)(O)C2)C1 c1(NCC2(C=C)CCC2)cc(=NCc2cc(Br)cc(C)c2F)[nH]cn1 c1(C(N(CC(CC)NC(C(CCC#C)O)=O)C)=O)c(C)c(C)cc(C)c1C N1(C(c2c(C)nc(C(F)(F)F)s2)=O)CC(C)N(C(c2ccc(C#N)o2)=O)CC1C C1(C2CCN(C(C3(c4ccccc4)CC3(F)F)=O)C2)(NC(C(=O)NCC)=O)CC1 c1(NC(C(C)OC)=O)ccc(O)c(Br)c1.C12(CO)CC(F)(C1)C2 C12(C(=O)NCCCn3cc(C4CC(C)(C)OC4)nn3)CCCC1C2(F)F C1(C(=O)NC(C(C)C)CCNC(c2ccc(=O)n(C)c2)=O)CCCC1S(C)(=O)=O Cc1ccc(CNC(=O)C(C2CCCC2)NC(c2sccc2CO)=O)c(O)c1 C1(S(C)(=O)=O)(C(=O)NC(C2CCN(C(C3=C(C)CCC3)=O)CC2)C)CCOCC1 c1(C(=O)NC(CC)CN(C(=O)C(C)CF)C)ncc([N+](=O)[O-])cc1Br C1(C(=O)OCC)COC(CNc2c[nH]c(CN(C)C)c2)C1 C12(C(=O)NCCC3CN(C(C(C4CC4)OC)=O)C3)C=CC(CC1)C2 c1(C(=O)NC(C)(C)C=CC(=O)Nc2cnc(F)nc2)cccc(F)c1F CC(C)C(O)C(=O)NCC1CC(F)CN1C(=O)COCC1CCOC1 Nc1cc(Br)cnc1C(=O)NC1CCCN(C(C2CCOCC2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC1COCCN(C(C2CCOC(C)(C)C2)=O)C1 N1(CC(=O)OC)CCN(C(=NCC=CC2CC2)NC2CSC(C)C2)CC1 C(=O)(C(Cc1ccccc1)NC(C1CCCN1C(c1csnn1)=O)=O)NC c1(C(N2CCC(NC(c3c(C)ncn3C)=O)C(O)C2)=O)cc(Cl)cc(Cl)c1O Cc1cc2nc[nH]c(=NCC3CC(CNC(c4ccoc4Cl)=O)CO3)c2[nH]1 Cc1oc(C(F)(F)F)c(C(N2CCN(C(C3CCC(=O)N3)=O)CC2)=O)c1C CCC(F)(C(=O)OC)C(=O)N1CC2CC1C2CNC(C1(O)CCC1)=O C=CC(C)(C)CC(=O)NCC1C2CN(C(=O)C=Cc3ccc(C(N)=O)o3)CC12 N1(C(C(C)=CCC)=O)CCCC(C(=O)NCC(C)(C)CN(C)C)(CC)C1 Cc1cc(NC(C2CCCCC(=O)N2)=O)ccc1NC(=O)CS(N)(=O)=O C1(C(=O)NCC2CCN(C(C(N3CCC(O)CC3)C)=O)C2)CCC2C(C1)C2(F)F N1(C(C(CC=C)c2n(C(=O)CC3CCC(=O)CC3)ccn2)=O)CCCC(C)(C)C1C c1(CCC(=O)N(CCCNC(c2csc(O)n2)=O)C)cc(F)cc(F)c1 N1(C(COCCOC)=O)CC(NC(C2CCC(c3ccccc3)O2)=O)C(O)C1 c1(C(c2nc(-c3ccc(OC)nc3)nn2C2CCC2)C)cn(C)c2ccccc12 c1(Nc2c(NC(CC(=O)OC)C)cccc2)ncc2[nH]ncc2n1 C(C(C)(C(N)=O)NC(C1(CNC(c2cncc(N)n2)=O)CCCCC1)=O)OC C(=O)(CC(C)CC(C)(C)C)N(C)CC1N(C(Cc2cn(CC)nc2)=O)CCCC1 C1(CC(=O)NC(C(=O)OC(C)C)C)CCCN(C(=O)CC2C=CCCC2)C1 C1(N(C(=O)CSCCC#N)CC)CCN(C(=O)CCSC2CCCC2)C1 Cc1ccc(C(C)NC2(c3ccc(F)cn3)CCOC2)cc1 C1(C(N2CCC(O)(CNC(C3(OC)CCOC3)=O)C2)=O)CC2(CCCC2)C1 C1(CO)CCC(C)(C)N(CC)C1.c1(CCN)cc(C2CC2)nn1C(C)C C1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)(COC)CCCCO1 C(=O)(C1=NOC(C)C1C)NC1C(NC(c2c(C)n(C(C)C)nn2)=O)COCC1 CC1CN(C(c2coc(C(F)F)n2)=O)CCCN1C(c1cnn2ncccc12)=O c1(CC)ncc(C(=O)N(C)CCN(C(=O)CCc2cnc(C)s2)C)c(O)n1 c1(C(=O)NCC(CO)NC(c2cccc(OC(C)C)c2)=O)n[nH]c2c1COC2 C1(CNC(C=CCN(C)CC)=O)CN(C)CCN1C(=O)CCNC(=O)CC c1(C(=O)OC)ccncc1-n1cc(SCC(=O)O)nn1 C12(NC(C#CC(C)C)=O)CCCC1N(C(=O)CSCc1csc(=N)[nH]1)CC2 N1(CC(=O)NCCN(C(=O)Cc2cncn2C)CC)CCCNS1(=O)=O CC1CC(CC(N2CCC2CC2CC2)=O)CN1C(=O)Cn1cccc1 c1(CC(=O)NC(C2CCCCC2)CO)ccc(Br)s1 c1(C(N2CCC(C(C)NC(c3c(C)coc3)=O)C2)=O)cc(C(N)=O)ccn1 C#Cc1cnc(C(=O)NC23CCN(C(c4cn(C)cc4C)=O)CCC2C3)c(C)c1 N1(C(Cc2c(C)non2)=O)CC2(CC2)CC1CNC(=O)C(C)(F)F C1(NC(c2c(C#C)cnn2C)=O)CC2CC(C1)N(C(=O)CSc1cnn(C)c1)C2 C1(C(N(CCC(C)NC(=O)CCC=CBr)C)=O)C(C)(C)C1(C)C N1(C(c2cn(CC)nc2C)C(=O)NC(C)C)CCS(=O)C(C)C1C C(=O)(CC(C)C(F)(F)F)NCC(=C)CCNC(=O)Cc1cccc(C2CC2)c1 CC(CC(=O)NC1CCOC1C(N1CC(CC2CC2)C1)=O)N(C)C n1(CC)ncc(CNC(C(C)(C)CC2CCCO2)c2nnnn2CC2CC2)c1C c1(CCC(=O)NCCN(C(c2c(NC)c(F)ccc2)=O)C)cccc([N+](=O)[O-])c1 c1(C(=O)N(C)C)ccc(C=CC(=O)NC2CCCC2NC(c2cnc(C)o2)=O)cc1 n1(CC)cnc2c(NC(C)CC(N)=O)[nH]c(=NC(C)c3ccccc3)nc12 N1(C(c2nn(CC)c(O)c2)=O)CC(O)(C2(CNC(c3cnn(C)c3)=O)CC2)C1 C#Cc1cccc(CC(=O)NC(C)(CO)C(=O)NCC=CBr)c1 c1(NC(N(CCn2cc(CNC(C)=O)nn2)CC)=O)cc(Br)c([N+](=O)[O-])[nH]1 c1(C(C)C)ncc(C(=O)NCC(C)N(C(=O)C=CCF)C)n1C c1(N(C(=O)CN2CCSCC2)C)cc(O)cc(Cl)c1.C12CCN1C2 c1(C(CC)C)nc(NC2CCCCC2NC(C2CCC3CC3CC2)=O)cc(C)n1 C(=O)(CCCCCn1cc(CN2CCCCC2)nn1)N(C)CC1CCCO1 Cc1nc(C(N2CCCC2CNC(c2ncc3ccccn23)=O)=O)c(=O)[nH]c1C c1(-c2nc(CCC(=O)NC(C)(CNC(=O)C=CBr)CO)on2)cccc(Cl)c1 CC(CCNC(=O)CCn1ncn(C)c1=O)CCNC(=O)C=C1CCC(C)C1 c1(-c2c(C)onc2)cccc(NC(=O)NS(=O)(=O)CC(C)C2CC2)c1 C1(NC(c2cc(C)oc2)=O)C(C)CCN(C(=O)Cc2ccc(Cl)nc2)C1C N1(C(c2cc(C)c(O)nc2)=O)CC2CN(C(c3cc(O)nc(O)n3)=O)CC2(C)C1 c1(C(=O)NCC(CC(=O)OC)NC(C(C(=O)OCC)OC)=O)ncc(Cl)cc1Cl N1(C(C(C)(C)NC(=O)OC)=O)CCC2(CC2C(=O)NCC2CC(O)C(O)C2)C1 C1(C(=O)OC)CCCN(C(c2cccn(CC(=O)OC)c2=O)=O)CC1.C1CC1 c1(OC)ccc(N(C)Cc2csc(Br)c2)c(OCc2ccco2)c1 CC1(C)CC(C(N2CCC(C3(NC(=O)C(F)F)CC3)CC2)=O)CC(C)(C)C1 N1(C(Cc2nc(C)oc2)=O)CC2(CCCC2)C1C(=O)NCC1CCCOC1 N1(CC(=O)NCCC2CC(CF)C2)CCCCC1.C1COC1 C1(c2cn(CCCC(=O)N(CCCN(C)C3CC3)C3CC3)nn2)CC2(CCC2)C1 C=CC1(C(N2CCCC3(C2)N=N3)=O)CCN(C(=O)C#CC2CCC2)C1 CN1CCN(C2(CC(N3CCC(NC(C45CCC(CC4)C5)=O)C3)=O)CCC2)CC1 c1(CN2CCC(C(=O)OCC)CC2C)ccccc1S(=O)(=O)NC c1(C(N2CCN(C(c3c(C)cc(C)o3)=O)CC2)=O)cccc2ncnc(O)c12 C(=O)(C(O)C(CCC)NC(c1cc(CO)on1)=O)NC(CC#C)C(=O)NC O=C1CC(C(=O)NC2CN(C(c3cnsc3)=O)CCC2C(F)(F)F)CC(=O)N1 CCCC(F)C(=O)N1CCCC1C(C)NC(=O)CCC1CC(F)(F)C1 C(C1=CCN(C(c2ccn(C(F)F)n2)=O)CC1)NC(C(C)(C)c1ccncc1)=O C(C)(C)(CC(F)C(=O)N1CC(n2cnnc2)C1)NC(C(Br)=C(C)C)=O C(=O)(C1=C(C)CN1)N1CCC(N(C(=O)C(O)C2CC2)CCC)C1 CCCCCC(C)(C)CNC(=O)C(C(C)C)NC(=O)CN(C)C(C)C C1(NC(C2C(C)C2C)=O)CC(C)(CNC(C2CCCCO2)=O)C1 C1(NC(CCn2c(C)cc(C)n2)=O)CCN(C(=O)C(F)(F)CC2CC2)CC1C C(=O)(C(C)(O)C(C)(C)C)N1CCC(CN(C(Cc2c(OC)ccnc2)=O)C)C1 c1(OC)ccc(C(N2CCCC(c3cnc[nH]3)C2)C(=O)NC(C)C)cc1C1CC1 c1(N2CCC(NC(c3ccc(CC)cc3)=O)C(O)C2)ncnc2sc(CC)cc12 N1(CCNC(C(CC)SC)=O)CCN(C(=O)C(C2CCC2)SCC)CC1 N1(C(CCC(=O)NCCC)=O)CCCC(C)(CNC(=O)CCc2cnoc2)C1 C1(NC(C=CC=CCCCCC)=O)CCC(C)N(C(c2cccc(CO)n2)=O)C1 c1(C(=O)NCCCCN(C(C(CC(C)C)OC)=O)C)cc2cn[nH]c2cn1 CCCC(C(O)C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CN=[N+]=[N-] CCCCCC(C(=O)NC)NC(=O)CC1CN(CCc2c(OC)cccc2F)C1 N1(C(c2cc(C)ncc2C)=O)CC2(CCCC2)C1C(=O)NCCC(C)N1CCC1 c1(-n2cc(CCOC)nn2)cccc(C(=O)NC2(C)CCSCC2)c1 c1(CC)cc(C(N2CCC(O)(C(C)CNC(c3cc(CO)[nH]n3)=O)C2)=O)nn1C n1(CC)nnnc1C(c1nc(C)cs1)NC1(c2ccccn2)CCC1 C=CCCCC(=O)NC(C)(CNC(c1sc(=N)[nH]c1C)=O)CO c1(C(=O)OC)cc(NC(=O)NCC(c2cccc(Br)c2)O)cc(Cl)c1 C(=O)(CC1=CCOCC1)N(C)CC1CCCC1NC(c1ccc([N+](=O)[O-])cn1)=O N1(C(C2(C=C)CCN(C(c3n[nH]c(C)c3C)=O)C2)=O)CCCCCCC1CC c1(C(CCOCC)NCC(C2CCCC2)NS(C)(=O)=O)cn2ccsc2n1 C#CC1(C(=O)NCC2COCC2N(C)C)CCN(C(=O)C2=CCSC2)C1 C1(CC)(NC(c2cc(C#N)cs2)=O)CCCN(C(C2CCC(C(N)=O)O2)=O)C1 N1(CCNC(CCCSC(C)(C)C)=O)CCCCN(C(C2CCNC2=O)=O)CC1 c1(C(=O)NC(C2CCCN(C(=O)CCc3cnn(C)c3)C2)C)ccnnc1O n1(CC(C)CO)nc(CCCN2CCCC2)nc1-c1cn(-c2ccccc2)nn1 C1(NC(c2cnc(CC)nc2C)=O)CCN(C(=O)C(C)(O)COC)C12CCCC2 Cc1oc(C(C)(C)C)cc1C(=O)NC1CC1CNC(=O)C(c1ccccc1Cl)O C1(C)(CNC(=O)Nc2c(N(C(C)=O)C)cccc2)CCC(=O)NC1 c1(C(=O)N(C(c2nc(C)no2)CC)NC(C)(C)C)cc(-c2cccs2)[nH]n1 c1(OC)cc(C(=O)NC2CC(O)CN(C(c3cnn(CCO)c3)=O)C2)ccc1O C1(C)(CNC(CCN(C(C=C(C)C2CC2)=O)CC2CC2)=O)CCCCC1O C(C)(CCC#N)(c1nnnn1C1(C)CC1)NCc1scc(C)n1.c1ccncc1Br CN1CC(O)CCC1C(=O)NC1(C(=O)NC(CO)C(=O)NC(N)=O)CC(F)C1 c1(C(N2CC(CC)(NC(c3ccn(C)c3C)=O)C2)=O)cnc(O)cc1C c1(CC)ccc(NC(=O)CC2CN(C(C3CC(=O)CS3)=O)CCO2)cc1 CN1C(=O)C(=O)N(CC(=O)NCC2(C)CCCN2C(c2ccno2)=O)C1=O C1(C(C(=O)NCCC(=O)NC2CC2)NC(C(C2CCCCC2)C)=O)CCCOC1 Cc1nnc(CCC(=O)NC2(C)CC(NC(C3CNC(=O)N3)=O)C2)n1C c1(C(CCCOC)NCCCCOC)ccc(OC)c(F)c1 N12CCC(CC1)C(=O)N2.C1C(CO)CC(=O)N1.C1(COCC)CC1.C1CC1 c1(-c2c(CN3CCC(NC(=O)NCC4CSCCS4)C3)cno2)ccc(F)cc1 Cc1c(C(=O)NC2CN(C(C3CC3C)=O)C2)oc2ccccc12 Cc1nc(C(N2CCN(C(c3cnc[nH]3)=O)C(CC3CC3)C2)=O)c(C)n1C1CC1 N1(C(CC)=O)CCN(C(c2ccc(SC(F)(F)F)o2)=O)CC(C)(F)C1 N1(C(CC=C)=O)CCCC2CN(C(c3nscc3N)=O)CCC12 c1(CC)nnc2n1CC(C(N1CCCC(Nc3cc(NC)ncn3)C1)=O)CC2 C(=O)(C(CO)C(C)(C)C)NCCCN(CCCNC(C(CSC)C)=O)C c1(CC)cc(CNN2CCC(Cc3ccccc3F)CC2)n(C)n1 N1(C(Cc2cc(C)on2)=O)CCC2(CCN(C(=O)C(F)(F)C3CC3)CC2)C1 c1(NC2CCCC(C)CC2)ccc2ccncc2c1[N+](=O)[O-] c1(C(N2C3C(C(=O)NC4CCC(C)CC4)C(C3)C2)=O)cccc2cccnc12 c1(NC(C(=O)N(C(C)CCN2CCCC2)C2CC2)=O)ncc(-c2ccncc2)s1 C(C(C(=O)NC1(CNC(C2CC2c2nc[nH]n2)=O)CC1)c1ccccc1)SC C1(C(NCP(C)(C)=O)=O)CCCC(NC(C2(C(C)(C)OC)CC2)=O)C1 C1(NC(C(CC)OC)=O)CCSC12CN(C(c1cc(C(C)(C)C)oc1C)=O)C2 c1(C(N2CC(N(C)C(c3cc(C(F)F)ccc3F)=O)C2)=O)ccc2cnoc2c1 C1(C(C)(C)C)CCN(c2nc(=N)nc(N3CCC(N4CCCC4=O)C3)[nH]2)CCO1 c1(C(=O)NCCCOCCNC(=O)CC2CCC(O)C2)ccc(F)c(F)c1 CC(Cc1cnc[nH]1)C(=O)NCC(C)CNC(=O)COC1CC1 C1(NC(C=CCC)=O)CCN(C(c2cc(OC)c(Br)s2)=O)CC1(C)C CCCC(=O)N(CC(=O)NCCc1ncc[nH]1)CC(C)C O(NC(=O)C(CC)NC(c1ncoc1CC)=O)CCC#C c1(NC(=O)NC(c2cc(C)ns2)(C)C)nc2cc(Cl)c(C)cc2s1 C1(N=[N+]=[N-])(C(N2CCC(CSC)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)C1 C(CCO)(C(=O)NC1CCCCC1NC(=O)Cc1csc(C2CC2)n1)N(C)C C(C(N=c1ccc2nnnn2[nH]1)C(C)C(C)C)NC(Cc1n(C)nc(CC)c1Cl)=O C1(CC(=O)O)(NC(=O)C(=O)N)CCCCC1.n1(CC)ccc(CC)n1 N1(C2CCN(C(C3C(=C)CC3)=O)C2)CCC(N(C(=O)C(CCC)OCC)CC)CC1 c1(C(=O)NC(C)C(C)(C)NC(=O)CC(C)n2cccn2)cnc(O)c2cncn12 c1(C(=O)NCC(C)CNC(=O)CNC(C2CCOC2)=O)cccc(Cl)c1 C1(C(=O)NC2CCCN(C(CSCC#C)=O)CC2)CC12CCC(C)(C)CC2 c1(C(N(C2CN(C(=O)CCc3nccn3C)C2)C)=O)cc(C(F)(F)F)cnc1N c1(C(=O)NCCC(CNC(=O)C(F)=CC2CC2)O)ccc(C2CCOC2)cc1 C1(C)(COC)CC(NC(=O)C=Cc2nc(C)co2)CN1C(=O)CNC(=O)C1CC1 c1(C(N2CC(C(C)NC(C3CC34CCSCC4)=O)C2)=O)csc2c1CCCC2 c1(C(N2C(C)CCC(CCc3ccc(OC)cc3)C2)=O)cc(F)c(Br)cc1C C(=O)(CCS(=O)(=O)C(F)(F)F)N(C1CCCCN(C(C(CC)(C)C#N)=O)C1)C C1(NC(CCC(C)=O)=O)CN(C(c2cccc(F)c2Cl)=O)CCC12CCOCC2 c1(CN2CC(n3ncc(C(=O)OCC)c3)C2)ccc2oc(C)c(C)c2c1.C1CO1 C1(O)(C(=O)O)CCCN(C(=O)COC(C2(CC(CC)OC)CCCC2)=O)C1 c1(N2C(CCNC(CN(C(C)=O)C)=O)CCC2)ncnc(C)c1OC N1(C(c2ccc(C)s2)=O)CC(C)OC2(CCN(C(C3CCCSC3)=O)C2)C1 N#Cc1ccc(=NCC(=O)NCC2CC2CNC(c2cc(C(F)F)no2)=O)[nH]c1 N12CC3(CC3)CC1CNC(=O)c1nsc2n1.C(=O)(CCC(F)F)OC n1(CC)cnc2c(NCC(CCC)CCO)nc(N3CCSCC3CCO)nc12 C12(NC(CCCCSC)=O)CC(CNC(=O)C(O)CN(C)C)(C1)OC21CCC1 c1(CNC(C(C)=CCC)=O)cc(C(=O)N(CC(O)CC)C)cs1 CCCCC(CC)CCC(=O)N1CCC(S(=O)(=O)NC(=O)OC(C)(C)C)C1 c1(C(=O)NCC=CCNC(C=CC=CC)=O)c(C)cc(C)c([N+](=O)[O-])c1C CC1=C(C)CC(C(=O)N(C(CNC(=O)CS(N)(=O)=O)C2CC2)C)CC1 N1(C(COC)=O)CCN(C(=O)CCS(=O)(=O)N(C)C)CC(C)(F)C1.C1CO1 N1(C(CN2CCN(C(C(c3cccnc3)C)=O)CC2)=O)CCC2(CC1)CC2 c1(C(=O)NCC(CC)N)ccc(Oc2ccc(Br)cc2)c(C(C)SC)c1 C(=O)(C=CS(C)=O)NCCC1CCN(C(C2(CCOC)CCC2)=O)C1 C1(C(=O)NCC2CC2C2CCCO2)CN(C(=O)CC2(O)CCC2)CCO1 CC1=C(C(=O)Nc2cccc(OCCC(=O)O)c2)Cn2ncnc2N1C c1(C(N(CCCN(C(CCC(=C)C)=O)C)C)=O)nccc2ccccc12 N1(C(C2(C)CCCN2C(c2ccc(B(O)O)cc2)=O)=O)CCCC2(CCOC2)C1 c1(C(=O)NCC2CC(NC(c3ccc(F)c(O)c3)=O)C2)cc2c(nn1)CCCO2 CC1(C)CC(=O)NC1NC(=O)C(CC1CCOCC1)NC(=O)CCNC(N)=O C(=O)(C(C(C)C)NC(N)=O)NCC=CCC(=O)N(C1CCCC1)CCOC N1(C(C2=C(C)OCC2)=O)CCCC2(CCN(C(C34CCCC(C)(C3)OC4)=O)C2)C1 C1(C(=O)Nc2cnn(C(F)F)c2)CN(c2ncc(F)cn2)CCC1(F)F N1(C(C(C=C=C)C)=O)CC(C(=O)NCCN(C)C)C2(CC2)C1 C(=O)(C(CC(C)C)NC(C)=O)NCC(CNC(CC1(C=C)CC1)=O)OC N1(C(CC(C)C)=O)CC2CCN(Cc3cc[nH]c3)CC2C1 c1(N2CC(CNC(=O)OC(C)(C)C)C3(C2)CC3)nc2ccccc2s1 C1(c2nn[nH]n2)(C(N(CC(C)OC)C)=O)CC2(CC2)C1 C1(OC)CC(CNC(=O)CCC2CCOC2)N(C(c2n[nH]c(C)c2O)=O)C1 CC1C(NC(=O)CC2(C)CCC2)CCCN1C(c1csc(C(C)(C)C)n1)=O C1(C)(CNC(c2c(OC)csc2)=O)CCN(C(C2(C)CC(O)C2)=O)C1 c1(OC)cc(C(N2CCCC(NC(=O)C(=O)O)C2)=O)cc([N+](=O)[O-])c1 C1(C)(C(=O)NC(C2CCN(C(N)=O)CC2)C)COC(=O)C1.C12CCN(C1)C2=O C1(CC(=O)NCC2(F)CC(NC(CC(C=C)C)=O)C2)CC(C)CC(C)(C)C1 C(=O)(CCCCCO)N1CCC(N(CC#C)C(C2CC2(Cl)Cl)=O)CC1 C1(N(C(C(C)(F)F)=O)CC2CCCO2)CCN(C(c2cc(C(N)=O)no2)=O)CC1 Cc1cccc(COCC(=O)NCCC2CCN(C(C3CCCC(=O)O3)=O)C2)c1 Cc1ccn(CCC(=O)NC2CCCC2NC(c2cnn(CCF)c2)=O)n1 N1(C(c2nnn(CC)c2C)=O)CC2CC1CN2C(=O)C(c1c(Cl)cccc1Cl)C CCC(C)(CCNC(c1cnc(C2CC2)o1)=O)NC(c1cc(Cl)ns1)=O C1(C(N2CC(OC(C)=O)C2)=O)CCN(C(=O)c2cc(C)cc(O)n2)O1 CCCC(C)(C)CC(=O)N1CCN(C(c2cc(C#N)ccc2F)=O)C(C2CC2)C1 C1(NC(CCOCCOC)=O)CCC2(CC1)CC2NC(=O)C(C)C(C)(C)C C(C)(C(=O)N1CC(CNC(=O)C(c2ccns2)NC(=O)OC(C)(C)C)C1)SC N#Cc1cccc(CCC(=O)NCCC2CN(C(C3CCSC3)=O)CCCO2)c1 c1(C(N2CCCCC2C(C)CO)C(=O)NCCOC)cc(C)ccn1 c1(C(=O)NCCOC2CCN(C(C(CC)C(C)C)=O)C2)ccc2nnnn2c1 n1(CC(=O)NCC(CN(C(=O)CC2(O)CCCCC2)C)O)ccc2ccccc12 CC1=NOC(=O)C1CCC(=O)NC(CNC(=O)CC1COCCO1)C(C)C C1(CCC)CN(C(c2[nH]ccc(=O)c2C)=O)CCN1C(c1cnc(O)s1)=O CCC(O)C(C)C(=O)NCC(C)=CC(=O)NC(c1cncnc1NC)=O N1(C(C2C(C(=O)OC)C2)=O)CCCC(C2(NC(C3CN(S(N)(=O)=O)C3)=O)CC2)C1 N1(C(C(CCC)OC)=O)CC(NC(=O)CCc2ccc(Cl)cc2)CC(F)C1 c1(NC(c2nc(N)c(-c3cnc(C(N)=O)nc3)cc2)=O)c(F)c(F)nc(F)c1F C(=O)(C1CCCc2ncnn21)N1C(C)CCC(NC(=O)C(C)(C)n2ccnn2)C1 c1(C(N2C(C(=O)NCCn3cc(C)nc3)C(O)CC2)=O)cc(C)cc(C#N)c1 C(CCCCCC(=O)NC1CC(O)CN(C(=O)CCC2(C)N=N2)C1)SC c1(C(N2C(C(N3C4CCCC3COC4)=O)CC3CC32)=O)ccc2c(c1)CCC2 N1(C(C2(CCC)CC2)=O)CCN(CC2CCN(C(C3CCC(C)C3)=O)CC2)CC1 C1(CC(=O)NC(CC(=O)N(c2ccsc2)C)C2CC2)CC2(CC2)CO1 C1(F)(CNC(c2nn(C)c(C(F)F)c2)=O)CCN(C(=O)COCP(C)(C)=O)CC1 CC1(C(N2CCOC(CC(=O)NCC(O)C3(Cl)CC3)C2)=O)CC(C#N)C1 N1(C(C2CC(CCC)OCC2)=O)CC(C2(NC(=O)CC(=O)N(C)C)CC2)C1 c1(C(N2CCC(C(O)CO)CC2)C(=O)NC(C(=O)OC)C)sc(Br)c(C)c1C N1(C(=O)OC(C)(C)C)CC(NC(=O)OCc2cc(Br)cnc2F)CC12COC2 Cc1ccc(C(=O)NC2CCN(C(c3cc(N)ccc3O)=O)CC2C)c(O)n1 N1(c2c(S(=O)(=O)N3CC(COC)OCC3)cccn2)CCN(C)C2(CCOC2)C1 C1(C(=O)N(CC(C)N(C)C)C)(CC)CCCN(C(=O)C(C(C)(C)C)SC)C1 N1(C(C=CCCC)=O)CCCC(CCNC(=O)Cn2cc(C)cn2)CC1 CC1(C)C=CC(NC(=O)NC2CC(OCC(F)(F)F)C2)CC1 C(=O)(CC(C(C)C)NC(C1CC(C)CCO1)=O)NCc1c(C)scn1 Cc1[nH]nc2cc(C(=O)NC3CC3NC(c3c4c(nn3C)CCSC4)=O)ccc12 C1(OC)CN(C(=O)C(F)CC2CCOC2)CC1C(=O)N(CC1=CCSC1)C C12CC13CCN(C3)C(=O)CCN2.Cc1cc(CNC(C2(F)CC2)=O)no1 CCC(O)CC(=O)NCC1(O)CC(CNC(=O)CN(C)C(C)=O)C1 c1(C(N2CCC(C)(CCNC(CCCOCC=C)=O)C2)=O)cc(C)ccc1N c1(C(=O)NCC(C)CNC(=O)CN(C)C(c2ccccc2)=O)ccn2ccsc12 O=C1CCc2cc(C(=O)NC3C=CC(C(N4CCC5(C=CC5)CC4)=O)C3)ccc21 c1(CN(CC(C)(C)C)CC2CC3C=CC2C3)ccc(C2CC2)cc1 C1(C(N2CCC(c3cccc(Cl)c3)C2)=O)CC(O)CN1C(c1ccccc1F)=O C1(NC(c2c(C)ncnc2C)=O)CCC2CCN(C(=O)C(C)n3ccnc3)C12 C1(C(=O)NCC(CC=C)(C)C)CC(F)CCN1C(c1ccccc1O)=O C1(NC(C(CSC)OC)=O)CN(C(=O)C=Cc2ccc(Br)cc2)C(C)(C)C1 C(=O)(CCCCC(F)F)NC1(C2N(C(c3ccc(OC)cc3)=O)CCCC2)CC1 C1(NC(C(C)OCCCC)=O)CN(C(c2cc(C(F)F)cs2)=O)CC1CC c1(C(C(=O)NCC(COC)NC(=O)Cn2[nH]cnc2=N)C)cnn(C)c1 C(CN=C(NC1CC1)N1CCC(F)(c2cc(C)cc(C)c2)C1)NC(=O)NC C1(CO)(CF)CCOCC1.C1C(CO)CNC(=O)c2ccc(o2)C(=O)N1.C1CO1 N1(C(COC)C)CCN(C(=O)C=Cc2ccccn2)C(=O)C1 C1(CNC(CS(CC)=O)=O)(OC)CCN(C(c2c(OC)ccnc2F)=O)CC1 C1(NC(c2nc(C(C)NC(CN(C(=O)OC)C)=O)oc2)=O)CC(=O)N(O)C1 C1(C(C(=O)NC2CC2)N(C2CCCO2)Cc2ccsc2)CC2CC2C1 Cc1ccc(C)c(SCC(=O)N(CCCNC(C2CNC(=O)N2)=O)C)c1 N1(C(=O)Cc2cn[nH]c2)CCC(C2CCO2)CC1 C1(NC(c2cnc(OC)[nH]2)=O)CCC(C(N2CCC2CC(C)(O)CC)=O)CC1 C1(NC(c2ccc3nccn3c2)=O)CS(=O)(=O)C2CN(C(c3ccsc3)=O)CC12 c1(CNc2ncc(-c3cc(CO)c(F)cc3)cc2O)cc(Cl)cc(Cl)c1Cl N1(OC)CCN(c2cccc(Br)c2)C(=O)C1.c12cc(ncn1)CN1CCCC1C2 c1(C(=O)NC2CN(C(C3(F)CC3)=O)CC2O)cccc(C(F)(F)F)c1Cl Nc1c(C(N2CC3(C2)CN(C(=O)C(O)CF)C3)=O)cc(F)cc1Br c1(C(=O)NCC2CC(NC(c3cc(C)sc3C)=O)CC2O)ccsc1S(C)(=O)=O N1(C(C2N(C(C(C3CCC3)OCC)=O)CCC2O)=O)CCOCC(C2CC2)C1 C1(C(=O)NC(CC)CCCO)C(C)OCCN1C(C1CCCC1O)=O C1(N(C)C(c2ncoc2CNC(=O)CC2COC(=O)C2)=O)CCC(C)(C)CC1 c1(NC(C2CC(F)CN2Cc2ccc(Cl)cc2)=O)cccc(OC(F)(F)F)c1Cl CC1CN(C(=O)C(c2ccccc2F)(C)O)CC1NC(C1COCCO1)=O c1(C(=O)NC(CCN(C(C2CC(SC)C2)=O)C)(C)C)cnc(C)nc1 C12(C(N(C(C)CNC(C3(F)C(C)(C)C3(C)C)=O)C)=O)CCC(N(C)C)(CC1)CC2 c1(OCC)cncc(C(N2CCC(OCCNC(c3ccnnc3C)=O)C2)=O)c1 N1(C(C=Cc2occ(C)n2)=O)CCC2C(NC(c3ncccc3Br)=O)CC12 CC12CC(C(=O)NCC3C4CN(C(c5coc(C(F)F)n5)=O)CC34)(C1)C(C)(C)O2 c1(C(=O)NCC(CO)NC(c2ncc(C#N)cc2Cl)=O)cnc2[nH]c(O)nc2c1 Cc1csc(C(=O)NCC2CCCC2NC(c2cc(CCCO)on2)=O)c1C C1(O)(C(N2CC(CNC(c3cccc(C)c3O)=O)C(C)C2)=O)CCCC(C)(C)C1 c1(NC(C2CN(C(c3cc(C)cc(C)c3)=O)C2)=O)ncc([N+](=O)[O-])cc1Cl Cc1c(C(N2CCC(NC(=O)C(C(C)C)NC3COC3)CC2)=O)ccn1C(C)C C1(c2n(CC(=C)C)nnn2)(NCC(C)(C)C)CCCC1CCc1ccccc1 CCC(CC)C(C)C(=O)NCCC1CCN(C(c2nocc2C(C)C)=O)C1 N1(C(C(C)=C(CC)C)=O)CCCOC(CNC(=O)C(C)C2(O)CCC2)C1 N1(C(C(C)c2ccsn2)=O)CCCN(C(c2ncccc2Cl)=O)CCC1 C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(c2sc(CC)nc2C)=O)CC1O Cc1snnc1C(=O)NC(C1CC1NC(C1(N2CCCC2)CCC1)=O)C c1(C(N(C2C(C)CCN(C(CCC=CC)=O)C2)C)=O)cccc2c(C)ccnc12 Cc1ccc(F)c2[nH]c(C(=O)NC3CN(C(c4nnsc4Cl)=O)CCC3C)cc12 C=CC1(C(=O)NCC2(C)CCC(=O)N2C)CCN(C(=O)C2CC2)C1 CN1CCCC(CNC(C2C=CCN(C(=O)C=Cc3ccncc3)C2)=O)C1 Nc1cccc(CC(=O)NCC2CCCN2C(=O)C(C2CCC(=O)N2)O)c1N c1(CC)noc(CC)c1CC(=O)NCC(C1CC1)N(C)C(C1(C)CC(F)C1)=O N1(C(CCCC(C)C)=O)C2CCC1CC(NC(c1coc(Br)c1)=O)C2 C(=O)(C(CC(C)C)CC(C)C)N1CC(C)(CNC(CCOCCC)=O)OCC1 C12(C(=O)NC3CC(N(C(c4c(C)nc(C5CC5)[nH]4)=O)C)C3)CCCN1CCC2 CC1COCC(CC(=O)NCc2cc(C(=O)N(C)CCN3CCCC3=O)on2)O1 C1(CN(c2nnc(-c3cccc(O)n3)n2CCC#N)C)CCc2c[nH]nc2C1 c1(Cn2cc(CC3CN(CC4CC(C(C(CC)C)=O)C4)C3)nn2)cccc(Cl)c1 C12(C(=O)NC3(C(=O)NC4CCCC(C(=O)OC)C4)CC3)CCCC(C)(C1)OC2 N1(C(C(=Cc2cccnc2)C)=O)CC(NC(C2(C)C(C)(C)C2(C)C)=O)CC(C)C1 N1(C(c2c(NC)c(N)ccc2)=O)CC(NC(C2CCCN2C)=O)C2CCCCC12 c1(C(=O)NC(CNC(c2c(OCCC)cccn2)=O)C)ccc2ocnc2n1 c1(C(N(C)CC2(CNC(=O)Cn3cnnc3O)CCC2)=O)ccc(CSC)nc1 C(=O)(C1=NOC(C)(C)C1)NC(C)C(=O)NC(C)Cc1ccnn1C N1(C(CC2CC(CC)OCC2)=O)CCCC2(NC(=O)C(C3CC3)C3CC3)CC2C1 C1(C(N2CC(C(C(C)C)O)C2)=O)CCN(C(C2CC3CCC3C2)=O)CC1C c1(OC)cc(CC(=O)NC2CCCN(C(=O)C=C(Cl)Cl)CC2)cc(F)c1 c1(C(N2C(CNC(CC=C(C)C)=O)CCCC2)=O)cnc2ccnn2c1C c1(CN(C(=O)NC2CSC(C(F)(F)F)C2)CC)ccc(C)c(C#N)c1 N1(C(CCSCCNC(c2c(CC)nn[nH]2)=O)=O)CCC(C)C(CO)C1 N1(C(CCNC(COC)=O)=O)CC2(COC(CNC(=O)Cc3cnsc3)C2)C1 Cc1ccc(C(=O)NC(C2CN(C(=O)Cn3cnc(Br)c3)C2)C)s1 C1(CC#C)(C(=O)OCC(C2CCCCO2)=O)CCCN(C(=O)OC(C)(C)C)C1 n1(CC(C)C)[nH]c(CC(=O)N(C2CN(C(=O)C(F)C3CCOC3)C2)C)cc1=O C1(NC(c2ncccc2O)=O)CN(C(c2cnn(C3CC3(F)F)c2)=O)CC12CC2 CC1(NC(=O)CCC2CCCCC2)CCN(c2nnc(CC(F)(F)F)s2)CC1 CC1(C)C(NC(=O)CCc2cnn[nH]2)CC1CNC(c1ccc(Br)cn1)=O C1(NC(C(CC)C(C)C)=O)CC2(CCN(C(=O)C#CC3CCCO3)CC2)C1 c1(C(C)NCC(=O)N(CCc2ccc(OCC)cc2)CC)ccc(C#N)cc1 c1(C(N2CC(C)(CNC(CC=C)=O)CC2(C)C)=O)ccc2cncn2c1C C=CC(C)(CC)C(=O)NC1CCC1NC(=O)Cc1cccc(N2CCOCC2)c1 N1(C(c2[nH]cc(C)c2)=O)CCN(Cc2cnn(-c3cccc(C#N)c3)c2)C2CC12 N1(CCC)CCCC1C(N1CC(CNC(C2COCC2C(N)=O)=O)(OC)C1)=O C(=O)(C1=CCC(C)(C)CC1)NCC(C)C(F)C(=O)NCCS(C)(=N)=O CC1COc2c(C(N3CC4(CNCCO4)C3)=O)cccc21 c1(C(N2CC3C(NC(c4cn(C)nn4)=O)C(C3)C2)=O)cccc2nnn(C)c12 c1(C(=O)NC(C)CN2CCN(C(=O)C=C(Cl)Cl)CC2)cnc2[nH]cncc1-2 c1(C(N2CCC(C(=O)NCc3ccno3)C2)=O)ccc(C(F)(F)F)cc1Br CCCCS(=O)(=O)Nc1cccnc1C(N1CCNC(C(=O)OCC)C1)=O c1(C(N2CCN(C(C(C(C)C)OC)=O)C(C)C2)=O)sc(S(N)(=O)=O)cc1C C1(C(N(CCN(C(C2C(=C)CC2)=O)C)C)=O)COCCC1C c1(NC(C2(CNC(CCCCCCC)=O)CC2)=O)ccc2cccnc2c1 C(C(=O)NN1CCCC1C(=O)NC(C)CN1CCCC1=O)SCCC C(=O)(CCCCCCCCC1CC1)NC1C(NC(C(C)(C)OCC)=O)CCC1 c1(-n2c(SCC(=C)C)nnn2)ccc(OCSc2nnn(C)c2C)cc1 N1(C(C2(C)CC(=C)C2)=O)CCC(NC(=O)CC2(C#N)CCC2)C(C)C1 C#CC1(C(=O)NCC2CC3CCC3C2)CCN(C(=O)C=C2CCCCC2)CC1 c1(OCC)cccc(CC(=O)N(CC(C)N(C(=O)C(C)CSC)C)C)c1 C1(CC(=O)OCC)CN(N2CC(c3ccccc3C)CC2C)CC2(CCC2)O1 O=C1CCCCC(C(N2CCCN(C(C3CCC(F)(F)C3)=O)CC2)=O)N1 C1(C(N2CCC(C(=O)NC3C(CN(C)C)C3)CC2)=O)CCC2(CC1)CC2 CC1(C)CC(CO)CCN1C(=O)CC(O)CNC(=O)CCc1cccnc1 CS(=O)C=CC(=O)N1CC(NC(C2(CF)CC(F)(F)C2)=O)C(CC2CC2)C1 c1(C(CNC(COCC(=O)NC)=O)NC(C2CC3CCC2C3)=O)cccc(Cl)c1 C(=O)(CC1CCOc2ccccc21)N1CC(O)CC(NC(CN(C)C(N)=O)=O)C1 C(=O)(CC(O)CC)N(CCC(=O)N(C1CCN(C)C1)C)CC=C N1(C(=O)OC)CCC(N(C(=O)C=CC(C)=O)C2CC2)CC1C c1(NCc2nnc(C)n2C)[nH]c(=NC2CCCN3CCCCC23)nc2sccc12 N1(C(c2c(C)con2)=O)CCC2(CC1)COC(CNC(c1cc(Br)n[nH]1)=O)C2 CCCC(C#N)C(=O)NCC(C)(CC)NC(=O)C=CCN1CCOCC1 N1(C(c2n(CC)nc(C)c2)=O)CC2CCC2(NC(c2ccoc2Cl)=O)C1 C(=O)(C(CCOCCO)NC(=O)C(C)C(=O)OC)NC(C(=O)OC)C1CCC1 c1(C(C)NC(c2cc(CC)nn2C)=O)cc(F)cc(F)c1F c1(C(=O)NCC2(F)CCN(C(COCCOC)=O)C2)ccc2nn[nH]c2c1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1C C(=O)(CC(C)(C)C)NC(C(C)C)C.C12CCN(CC1)C(=O)C1CC1C(=O)N2 CC(C)C(CNC(c1csc(CO)n1)=O)C(=O)N1CC(C(N)=O)C(C)C1 c1(C(CNS(CC2(C)CCNC2)(=O)=O)CC2CCCC2)ccc(Cl)c(Cl)c1 C1(C(C)NC(c2ccno2)=O)CCN(C(c2ccc(OCCO)cc2)=O)CC1 C(=O)(C(CCCC=C)NC(=O)C(C1CCC1)OCC)NCC(CC#C)(C)CO c1(C(N(c2ccnc(-c3cn(CCCC)nn3)c2C)CC)=O)c(F)cc(Cl)cc1Cl C1(SC)CN(C(c2ccc(C(F)F)cc2)=O)CC1NC(c1cc(C#N)c[nH]1)=O N1(C(CN2C(C)CCCC2)=O)CC2(CC(NC(=O)C(C)C(F)F)C2)C1 C1(CNC(C(CCC)F)=O)CCCCN(C(=O)CCOC(C)C)C1 C=CCC(CC(=O)N(C1CCOCCC1O)C)NC(c1[nH]ccc1C)=O c1(CC(=O)NC2C(CNC(C(COC)C)=O)CCC2)ccc2c(c1)CCN2C c1(N(CC=Cc2cc[nH]c2)CC2CN(C(C)C)C2)n[nH]cc1-c1nn[nH]n1 C(=O)(C1=CC2(CN(C(=O)C(C)C3CCOC3)C2)OC1)Nc1cncc(COC)c1 N1(C(CCOCCN(C)C)=O)CC2C(CNC(C3(O)CCC3)=O)C2C1 C1(OCC)COCC1N=c1[nH]c(=NC(C)CC2CCCCC2)[nH]c2c1CSC2 CCN=c1cc(-c2nc(CC(C)OC)n(-c3ccc(C(F)(F)F)cc3)n2)cc[nH]1 CC(C)C(C(=O)NCC(CNC(C12CCCC1(C(N)=O)C2)=O)C(F)(F)F)C(C)C C1(CNC(C(COC)O)=O)CCCC2(CN(C(=O)Cc3ccc(C)c(C)c3)C2)O1 C=CCCC1C(=O)N2CCOCC2N(CC)CC(F)C(=O)N1.C(C)SC C1(NC(=NCCCSCC)NCCSS(C)(=O)=O)C(=O)N(C)CCC1C CC1CC(N=c2c([N+](=O)[O-])c[nH]c3ccc(Cl)cc23)CCN1C(C1CCC1)=O c1(-n2cc(C(CCC)NC(c3ccccc3C(F)F)=O)nn2)cc(F)ccc1C C1(C(N(C2CCCN(C(c3nn(C)cc3CC)=O)C2)CC#C)=O)CC2CC(=O)C1O2 Cc1cc(C(=O)NCCOCC(=O)NCc2cc(C#N)c[nH]2)n(C)n1 N1(C(C(COCC)C)=O)CC2CCC2(C(=O)NCC2(CCOC)CC2)C1 N1(C(c2nc(CC)sc2)=O)CCN(C(c2ncccc2C(C)=O)=O)CC1C N1(C(C(CC=CC)C)=O)CCC(NC(=O)C2=CCOC2)C1(C)C C1(CC)CC(C)N(c2nnc(-c3cncs3)n2CC2(CO)CC2)C1 CC(F)(C(=O)NCCC1CN(C(=O)CCCc2ccccn2)C1)C(F)(F)F c1(C(N2CC(C)C(NC(c3cncc4sccc34)=O)C2)=O)n[nH]c2c1CC1CC21 C1(NC(Cn2c(C)cnc2)=O)CCC(NC(=O)COCCN(C)C)CC1 C1(C(=O)NCCC2N(C(c3c(C)nc(C)[nH]3)=O)CCSC2)OCC2CCCCC12 N1(C(CCCNC(CC)=O)=O)CC(OC)CC(NC(c2cc(C)sc2C)=O)C1 Cc1csc(C(=O)NC2CCC2NC(C23C=CC(CC2)C3)=O)c1Cl CC1CN(C(C2CCCC(F)(F)C2)=O)CCN1C(=O)CN1C(=O)CN(C)C1=O CC1(C)OC(=O)C(CC(=O)NC2CC(NC(=O)CSc3nncs3)C2(C)C)O1 C12(OC)CCCCC(C(=O)NCCNC(=O)C3=CCC(C)CC3)(C1)C2 c1(CC(N2CC(CCNC(CC3CN(C)C3)=O)C2)=O)cc(Br)cs1 c1(C(C)OC)nc(C)c(C(=O)NCCNC(C2CCSCC2)=O)s1 c1(C(=O)NC(CC)CNC(c2cccnn2)=O)ccc2nc[nH]c2c1F N1(C(C(C)(C)OCCC)=O)CC2CC2(NC(=O)CC)C1.C12CC(C1)S2 N1(CC(CN(C)C(=O)OC(C)(C)C)O)CCN(c2ccccc2)CC1.C1CO1 N1(CC)CCCC(C(=O)NC(C)(CO)C(=O)N(CC(C2CCCC2)O)C)C1 C(=O)(C1=COCCO1)N1CC(C(C)NC(=O)C2=COCC2)C1 c1(NCCC(O)C2CC2)cccc(-n2ncc(-c3nn[nH]n3)c2Br)c1 N1(C(C2C(NC(c3csc(Cl)n3)=O)CC2)=O)CCOC(CCF)C1 C1(C(=O)NCC2=CCN(C(C3C(C)(CC)C3)=O)CC2)CC(c2cccnc2)=NO1 C=CCCCCC(=O)N1CCCC(NC(C2CCCC2F)=O)CC1 C1(NC(c2ccc(C3CC3)o2)=O)CN(C(C2CC3CCC2O3)=O)CC2(CC2)C1 C(=O)(CC(C)C(F)F)NCC(CNC(CCc1c(OCC)cccc1)=O)CO C(C(COC)C(=O)N1CC(F)CC1Cn1cc(C2OCCO2)nn1)OC C(=O)(N=c1cccn[nH]1)C12C(CN(C(c3ccc(COC)cc3)=O)C1)CC2 Cc1cccc(CC(N2CCC(NC(=O)CC3CCCCC3F)CC2)=O)c1F C12(C(=O)NCC3C(NC(C(C)(C)C)=O)C3)CCC(C(F)F)(CC1)C2 C1(O)(CNC(C2C3(CC3)C23CC3)=O)CCN(C(C2CCOC2=O)=O)CC1 C1(C#N)(N(C(CSCCNC(c2cn(CC)nc2)=O)=O)C)CCOCC1 C(CC1CC1)(C(=O)NCC1CC(NC(=O)C=CC2CCCC2)C1)OC C(=O)(C(CNC(C1(n2cnnn2)CC1)=O)C(C)C)NCC1(OC)CC1 CC(C(CO)NC(C1(C2CCCCO2)CC1)=O)NC(=O)CC(C)c1ccncc1 C12(NC(c3cc(F)c[nH]3)=O)CCCCC1CN(C(C1CC3C=CC1C31CC1)=O)C2 c1(C(=O)OCC)sc(C(=O)NCCC(O)CNC(C2CC2F)=O)c2c1CCCC2 C1(N(C(c2scc(C)c2C)=O)C)CN(C(C23COCC(C2)C3)=O)CC1(C)C c1(C(=O)NCC2C(NC(c3c(C)snc3)=O)C2)cccnc1Oc1ccccc1 n1(C(C)C)ncc(C(=O)NCC2C3CN(C(=O)Cc4conc4C)CC23)c1N c1(NC(c2ccnc(-c3cccc([N+](=O)[O-])c3)c2)=O)c(F)cc(F)cc1[N+](=O)[O-] C(N=c1cc(CCC2CCCC2)nc[nH]1)C1CS(=O)(=O)CC1O C1(NC(CCCOCCOC)=O)CN(C(c2csc(Cl)c2)=O)CC1n1ccnn1 C12(CNC(c3coc(C4CC4)n3)=O)CCC1CN(C(c1cc(Br)co1)=O)C2 c1(-c2c(C(=O)Nc3ccc(C(=O)OC)s3)ccnc2)ccnc(OC)c1F C1(CNC(C2(CCC)CCC2)=O)CCN(C(=O)CCC=CBr)CC1C CS(=O)(=O)C1(C(N2CCCOC(CNC(c3c(O)cccc3O)=O)C2)=O)CCC1 c1(C(N(CCN(C(C(C)(CO)OC)=O)C)C)=O)cc(C)c2sccc2c1 c1(CC(=O)NCC2(CNC(C3CC(=C)C3)=O)CC2)nnc(O)s1 N1(C(C(n2ccc(C(F)(F)F)n2)C)=O)CCC(N(CC(=O)NC2CCC2)C)CC1 C=CC(CC)CC(=O)NC1CCN(C(=O)CNC(c2c(F)cccc2Cl)=O)C1 C(=O)(CCCN=[N+]=[N-])NC1(C(N(CC(C)C(F)(F)F)C)=O)CSC1 N12CCC(C(O)C1)C2=O.c1(OCC)ccc(CNCC23CC(CO)(C2)C3)cn1 c1(C(=O)NC2CN(C(c3n(C)cnc3)=O)CC3C2C3)cc(S(C)(=O)=O)ccc1O CCCCC(CC)CC(=O)NC(C)(C)CN1CCC1.C1=CCNC1=O c1(-c2nc(CCN(C)C)nn2C2CCS(=O)(=O)C2)ccn2cnnc2c1 N1(C(=O)Nc2ncc(OC)s2)CC(C)SC(C)C1 N1(C(CC(CNC(C2CC=CC2)=O)OC)=O)CC2(CCC(=O)NC2)C1 c1(C(N2CC(C(C(=O)N(C3(OC)CCCC3)C)OC(C)C)C2)=O)cccc(F)c1 Cc1cccc(Cl)c1CC(=O)NCCC1CN(C(C2CCN(C)C2=O)=O)CCO1 C=C=CCC(=O)NC(C)CCNC(C1CCC(C(F)(F)F)C1)=O C#CC1(C(=O)NCC2CCCN2C(=O)C=CC(=O)OC(C)(C)C)CCC1 O=C(CC(O)COCc1ccccc1)NCCNC(C1CCNC1=O)=O C=CCCCCCCC(=O)N1CCCC(CN(C(=O)C(C)(Cl)Cl)CC)C1 c1(C(N2CC(F)(CNC(c3c(COC)ccs3)=O)C2)=O)cccc(Cl)c1Cl N1(C(c2cc(=N)[nH]cc2)=O)CC2CCN(C(=O)CCc3cnoc3)CCC2C1 C(C(CC(C)C)NC(c1csnc1Br)=O)NC(C1(OC(C)=O)CC1)=O C(=O)(CCCC(=O)NCC(CO)NC(=O)C(CCC)c1ccccc1)OCC C1(CC=C)(NC(=O)Cn2cccn2)CCN(C(C2CC2(F)F)=O)CC1 CC(C)CCC(O)C(=O)N1CC=CCC1C(N1CCN2CCCC2C1)=O c1(NC(CC2CCN(C(C=CCC)=O)C2)=O)c(C)nn(CC)c1C C(Cc1ccccc1)(CCNC(C1(Cl)CC1)=O)NC(c1cncnc1)=O Cc1nc(N2CCC(NC(=O)CC3COCCO3)C(C)C2)cc(Cl)n1 C1(COC)(CNC(C2CS(=O)(=O)C2)=O)CCCN1c1cncc(Cl)n1 Cc1ccccc1-c1cn(C(C)CN(C(=O)CCN2CCCC2)C2CCC2)nn1 CC(CCC(C)(C)C)C(=O)NC1(C(=O)NC2CCn3cncc3C2)CC(F)C1 N1(C(CCN(C)CCO)=O)CCCC(C2CCN(C(=O)C(C)(C)CN(C)C)C2)C1 Cn1nc(Br)c2ccc(C(N3CC(F)CC3C(=O)NC(C3CC3)C3CC3)=O)cc12 N1(C(c2c(C)c(Cl)cnc2)=O)CC2CN(C(=O)CC(O)CCN(C)C)CC2(C)C1 Cn1ccc2ccc(C(N3CCCC3CNCc3cncc(O)c3)=O)cc12 C1(C(N2CC(NC(Cc3cc(C)no3)=O)C(C#N)C2)=O)CCc2nc[nH]c2C1 CCC(CNC(C1(F)CCN(C(=O)CC2CCC(C)(C)C2)C1)=O)C(C)(F)F C(=O)(CCCCCO)NCCCCC(C)NC(C=CC)=O c1(CNC(C2CCC(N(C)C)C2)=O)ccc(CNC2N(C(C)=O)CCC2)c(F)c1 C#CC1CN(C(=O)CCN(C(=O)C(CN(C)C)N(C)C)C)CCN1C C1(NC(C(CC)C)=O)CCCN(C(=O)C=Cc2ccc(SC(F)F)cc2)CCC1 C(CCCC(C)(C)C(=O)NNC(=O)C1CCCCCC1)NC(C(C)C(C)(C)C)=O c1(C(=O)NCC2OCCCN(C(c3ncc(C)cn3)=O)C2)cnc(O)n(C)c1=O C1(C(N(CCCn2cc(-c3cn[nH]c3)nn2)C)=O)CC(F)(F)CCC1(C)C C1(NC23CC(C2)CCCCn2c3nnn2)CC(O)C(O)C1.C(C)(C)(C)S.CO N1(C(CC(CCC)O)=O)CC2CC(C1)N(Cc1nn(C)c(=O)n1C)C2 N1(C(C(C=CC)O)=O)CCN(C(=O)CC(C)(C)C2CC2)CC1CF c1(CC)cc(C(N2CCCC(CC(N3CCC3C(=O)NC)=O)C2)=O)ncn1 O=S(=O)(CCc1ccncc1)NCCC1(c2ccccc2)CCCO1 c1(OC)cccc(O)c1C(N1CCN(C(c2cc(C)c(C)o2)=O)C(C(C)C)C1)=O Cc1cc(O)cc(Cl)c1C(=O)NCC(O)COc1ccc(C2CCC(=O)N2)cc1 N1(C(CCOCC)=O)CC(NC(c2cnc(N(C)C)s2)=O)CC(C)C1 c1(OCC)cc(F)ccc1C(N1CCCC(O)(c2cn(C(C)C(C)O)nn2)C1)=O C(=O)(C(F)CC(C)(C)C)NC1CC(CCNC(c2c(C)n(C)nn2)=O)C1 Cc1nnc2ccc(C(N3C4CCC3C3CC3(NC(C3CC3(F)Cl)=O)C4)=O)cn12 CC1CNCC(CC(=O)NC(=O)CC(c2ccc(Cl)cc2)C2CC2)O1 c1(C(N(CCC)Cc2cccc(Cl)c2)=O)cnc2ccccc2c1C C1(C(N2CCCC(SC)C2)=O)C2CC3C(C2NC(=O)C(C)CC2CCCC2)C13 C1(NC(c2nccc(OC)c2OC)=O)C(C)CN(C(c2cnc(O)o2)=O)CC1C C1(NC(c2c(C)ccc(-c3ccncc3)c2)=O)CC(C)(C)OC(C)(C)C1 N1(C(CC2(C)CC2(F)F)=O)CC(NC(c2ccc(Cl)c(O)c2)=O)CC12CCC2 c1(C(=O)NC(CC=C)CNC(c2coc(COC)n2)=O)ccc(C)c([N+](=O)[O-])c1 c1(C(N2CCC(NC(CNC(=O)NC)=O)C2)=O)ccc(C(C)(C)C)cn1 c1(COC)nc(=NC(=O)c2ccc(C(C)(C)S(C)(=O)=O)cc2)o[nH]1 C(=O)(C1c2ccccc2C1)NCCCN(C(C1CCC(C)(C)C1)=O)CC c1(OC)ccc(Cl)c(C(=O)NCC(C)CNC(c2nc(C)ccc2C)=O)c1F n1(C(C)C)ncc2c(NC(c3cnn(C)c3)C)[nH]c(=NC3CC=CC3)nc12 N1(C(CC(C)F)=O)CCc2c(c(CNC(C3CC3F)=O)nn2C)C1 C1(C(=O)NC(CNC(CC2C(SC)C2C)=O)CC(C)C)CCc2nnc(O)n2C1 c1(CC(=O)NCCCCC(C)NC(=O)C(F)=CC2CC2)ccc2oc(O)nc2c1 c1(C(=O)NC2CC(CNC(=O)C(F)n3cccn3)C2)cccn2nncc12 C(=O)(CC1CC(C(C)C)c2ccccc21)N1CCC(NC(CCC#C)=O)C(O)C1 c1(C(=O)OC)ccc2nc(NC(c3ccc(Cl)cc3Cl)=O)[nH]c2c1 Nc1ccc2nc(N3CCCC(CO)(NC(=O)C=Cc4ccccn4)C3)sc2c1 c1(C(=O)NCC2(CNC(CSCC(C)C)=O)CC(F)(F)C2)cc(S(N)(=O)=O)c[nH]1 N1(C(CCCN(C(C)=O)C)=O)CCC(NC(=O)CN2CC(C)C2)C2(CCC2)C1 C(=O)(C(C)CC(F)F)NC(C(=O)NCc1ccc(C)cc1)C1CCC1 N(C1c2cc(F)ccc2CCC1C)Cc1c(C)nc[nH]1 c1(CCC)c(C(=O)OCCCC2CCOC2)cnn1C N1(C(C(CC)(C)O)=O)CCC(O)(CCCNC(C2CN(C(C)=O)CCO2)=O)CC1 N1(C(c2c(C)cns2)=O)C2CCC1C(CNC(c1cnncc1C(F)(F)F)=O)C2 CC(=O)CCN=C(NCc1nnc(-c2ccccc2)s1)NC1CCN(C(C)=O)C1 c1(C(=O)NCC2C(NC(CC3(OC)CCCCC3)=O)C2)c(F)ccc2[nH]ccc12 c1(C(=O)NCC2C(NC(CC(C)(C)c3cccs3)=O)CCC2)cnc2n1CCS2 N1(C(CC(C)C)=O)CCC2(CC2C(N2CCN(c3ccc(Cl)nn3)CC2)=O)C1 C1(NC(CNC(C(COC)(F)F)=O)=O)COCC1C1CC1 CC(C)(CC(=O)N1CC(C2(NC(=O)CCc3ccc(F)nc3)CC2)C1)C(F)F c1(C(N(CC(CNC(C2C(C(C)C)OCC2)=O)O)C)=O)cnc2c[nH]nc2c1 c1(C(N2CC(NC(c3cnn(CCF)c3)=O)C3(C2)CC3)=O)cnn2ccccc12 CC(C)CC(CNC(=O)Cn1nccn1)C(=O)NC(CN(C)C)CCO Cc1cc(C(N2CCC(C)C2CNC(c2cc[nH]c3nccc2-3)=O)=O)c(O)cc1F S(=O)(=O)(c1cnc(NC2CC=CCC2)c(Cl)c1)N(CCCCOC(C)(C)C)C c1(CNC(C(CCOCCO)NC(CC(CC)C)=O)=O)cc(C)nc(C)c1 CN1CC(CCNC(C2(C)CCN(C(C3CCN3C)=O)C2)=O)CC1=O C1(NC(c2c(SC)ccs2)=O)CN(C(=O)C(O)CC(F)F)Cc2ccnn2C1 N1(C(C)=O)CC(C)(C)OCC1CNS(CC(=O)NC1CC(CSC2CC2)C1)(=O)=O c1(NC(c2c(F)cccc2F)C)ccc(S(=O)(=O)NC2CC2C2CCC2)cc1F CC(CCC(=O)N1CC2C(N(C)C)C2C1)NC(=O)C(c1cccn1C)=O c1(C(Cc2c(C)non2)C)nc(CCN(C)C)nn1-c1ccn(C)n1 Cc1c(Br)c(C(=O)N(C)CC2(O)CN(C(=O)C3=CC(C)(C)C3)C2)nn1C C(=O)(C1CCCc2ncc(C)n21)NC(C1CCCC1)CNC(CNC(C)=O)=O c1(C(=O)NCCCN(C(c2ccsc2Br)=O)CC)c[nH]c(=O)cn1 c1(CCCCOC(C)=O)cn(CC(O)CNC(=O)Cc2ccccc2)nn1 c1(C(N2CCC(N(C(c3ncn(CC)c3)=O)C)C2)=O)ccc(=O)n2c1CCCC2 N1(C(C(C)OCC)=O)CCC(C(C)NC(C2(C(=O)NC)CCC2)=O)C1 C1(C(=O)NC(COC(C)=O)CO)CC2(CCN(C(c3c(C)ncn3OC)=O)C2)C1 C1(C(N2CC(C#N)C(NC(C3(Br)CCC3)=O)C2)=O)Cc2ccccc2O1 Cc1ccc(F)c(C(N2CCSCC2C(=O)NC2CC(n3ccnc3)C2)=O)n1 N1(C(C2(CC=C)CCC2)=O)C2CCC1CC(CNC(C1C=CCC1)=O)C2 c1(OC)c(C(=O)N(C)CC2CCCN(C(C3(Cl)CC3(C)C)=O)C2)nc(O)nc1O C(=O)(C(C)(C)C1=CCSCC1)NC(C(C)NC(C1CCOC(C)(C)C1)=O)CO c1(C(=O)NCC2(NC(c3cnsn3)=O)CCC2)ncc(C(F)(F)F)s1 C1(OC)CN(C(=O)C=CC(=O)OC(C)(C)C)CC1C(N1CC(O)CC1C1CC1)=O C(=O)(C(C)C(=O)N1CCCC1CN(C)C(c1csc(-c2cnccn2)n1)=O)OC c1(N(C)Cc2ccc(OC(C)C)cc2)cccc(S(=O)(=O)N2CCS(=O)CC2)n1 C(C)(CCCN=c1[nH]cc(C#N)cc1C)NC(C(C)OCC)=O Cc1cc(O)cc(C)c1C(=O)NCC1CCN(C(=O)Cc2nc[nH]n2)C1(C)C N1(C(C(C)S(C)(=O)=O)=O)CCC2C(CCCN2C(=O)CCCC(N)=O)C1 C1(C2N(C(c3ccc(CC)s3)=O)CCC2)CCN(C(c2ccc(O)nn2)=O)CC1 C1(C(=O)NCCN(C(c2ccc(C3CC3)nc2O)=O)CC)CN2CCN1CC2C N1(C(C=CCC(C)(C)NC(C(C(C)C)C2CCC2)=O)=O)CC(O)CCC1C C12CCC(CC1)CNC2=O.C(CCCCNC(C1CC1Cl)=O)=CC(C)C C(=O)(C(C)(C)C(F)F)NC(C(C(=O)N1C(C(C(=O)OC)(C)C)CCC1)C)C C1(C#N)(C(=O)NC2(C(N(C)CCC3CCCO3)=O)CCC2)CCC1 C(=O)(C1=Cc2ccccc2OC1)N1C2CCC(NC(C(N)=O)=O)(CC2)C1 C(CC(=O)NCCn1ccnc1)(C(F)F)N(C)C(c1cc[n+]([O-])cc1)=O C1(CC)CCCCC1NC(c1c(CNC(=O)C=Cc2ncc[nH]2)cnn1C)=O C(=O)(C1=CCC(C)(C)CC1)NC1CCCN(C(Cc2cnc(C)s2)=O)C1 n1(C(CC)(C)C)nnnc1C(c1conc1C1CC1)NCC1CC1c1ccccc1 c1(C(=O)NCC2C(NC(c3cnn(C)c3Cl)=O)CCC2)cccc(F)c1Cl C(C(CCO)NC(c1cnn(CCNC(C2CC2C#N)=O)c1)=O)OC C1(N(C(CC(C)c2ccco2)=O)C)CCN(C(=O)CN2CCCS2(=O)=O)CC12CC2 N1(C(C2C(C(=O)OC)C2)=O)CCC2CCCC(C1)N2c1nc(C)cc(C#N)n1 C1(C)(C(N2CCC(CCNC(c3cc(COC)no3)=O)CC2)=O)CCC(O)CC1 C1(C(=O)NCCc2nc(C)sc2)C2CCN(C(c3cc4n(n3)CCO4)=O)CC12 C1(C(N(CC(=C)C)C)=O)C(O)CCN1C(=O)COCCF C1(CCNC(C2CC(NC(c3ccc(C4CC4)o3)=O)C2)=O)CCCCCC1 c1(C(=O)NC2(C)CC(NC(c3cnco3)=O)C2)cncc2cccnc12 C1(CC#C)(C(=O)NCC2CCOC2)CCN(C(=O)C(F)n2ccnc2)C1 C1(CN(c2ccncn2)C(C2CCCNC2)C)CCC(F)CC1 Cc1nc(C)c(C(=O)N(C)CC2(O)CCN(C(c3csc(C(F)F)n3)=O)C2)o1 C(C)(CC(C(=O)Nc1nnn(C)n1)N(Cc1cc(C)ccc1F)CC1CC1)SC N1(C(c2n(C)nnc2CNC(=O)CN(C)C)=O)CCCC[Si](C)(C)C1 N1(C(C2OCCCO2)=O)CCn2nccc21 CC1CN(C(C2CCN3CCC2C3)=O)CCCN1C(c1ccc(F)c(F)c1)=O CC(C)(CNC(=O)CO)CNC(=O)CCNC(C1CCCC1)=O C1(C(N2CCCC(CC)(NC(c3csc(=N)[nH]3)=O)C2)=O)CC2(C1)CC(C)(C)C2 O=C(CS(=O)(=O)c1ccc(Cl)cc1)NC1CN(C(C2CSC2)=O)CC1O N1(C(c2ccc(COC)o2)=O)CCCC(CN(C(=O)CCC(=O)OC)C)C1 C(CC1CC1)(C(=O)NCCCN(C)C(C1CC2CC2C1)=O)OC N1(C(Cc2cc(C)sc2)=O)CC2CC1CN2C(C1(n2cccc2)CCCC1)=O C(C#Cc1ccccc1F)N(C(=O)CCc1ccc(F)cc1Br)CCOC C(=O)(C=C1SCC(=O)N1C)NCC1CCCN(C(C2CC(C(=O)OC)C2)=O)C1 N1(C(C(C)CO)=O)CCC2(C=C(C(=O)NCC3CCC3(F)F)C2)C1 C1(NC(c2ccc(CC)cn2)=O)CN(C(c2[nH]nnc2C2CC2)=O)CC1C1CC1 C1(C(=O)NC2CC(=C)C2)CCN(C(=O)Cc2occc2C)C1 c1(NCC)ncc(C(=O)NC(CCN(C(=O)CCNC(N)=O)C)C(C)C)cc1Cl c1(C(=O)OC)cnc2nc(NC(c3cccc(O)c3OC)=O)ccc2c1 C(=O)(C1CCNc2ccccc21)NC(CC(C)C)CNC(c1nccnc1N)=O C1(C(N2C(CNC(C3CC(C)C3)=O)CC(O)C2)=O)CN(CP(C)(C)=O)C1 C=CCCCC(=O)N1CCCC(N(C(=O)Cc2csc(C(=O)OC)c2)C)C1 c1(C(=O)NCCCC2N(C(c3cnn(CC)n3)=O)CCCC2)cccc(C)c1C c1(C(N2CCC(CNC(Cc3cc(C)no3)=O)C(O)C2)=O)ccc2nccn2n1 c1(C(C(N2CCC(NC(C=CCCC=C(C)C)=O)C2)=O)=O)ccc(F)cc1 CC1OC2(C(=O)NCCCC(C)NC(=O)COCC(C)(C)C)CC1C2 C1(C(NNC(c2c(OC)c(Br)ccc2)=O)=O)CCc2nccn2CC1 N1(C(CNS(C)(=O)=O)=O)Cc2ccccc2OC2(C1)CN(C(=O)CSCCF)C2 N1(C(c2c(C)nc(C(C)C)nc2)=O)CC(N=c2[nH]c(Cl)ncc2C(N)=O)CC1C c1(CC(=O)NCC(CCCC)NC(=O)CCS(C)(=O)=O)cc2ccccc2s1 C(=O)(CC1=CCCCC1)NC1C(C)CCN(C(c2c(C)oc(C)c2Br)=O)C1 N1(C(c2c(OC)cc(C)cc2)=O)CC2CCC(NC(=O)C(C)(C)C(=O)NC)C2C1 C(=O)(C1=NN(CCO)C(=O)CC1)N(C1C2CN(C(C(C)C)=O)CC21)C C1(CCC(C)C)(CC)CCCN1C(=O)OCC1(C#N)COC1 C12(C(N3CC4C(NC(C5CCN(C)C5=O)=O)(C4)C3)=O)C3CCC(CC13)C2(F)F c1(C(N2CC(SC)C(n3cc(CC4(O)CCC4)nn3)C2)=O)cc(C)c(F)cc1Br C(=O)(CCCCO)N1CCCC(N(C(c2ccc(Cn3ccnn3)o2)=O)CC)C1 C1(C(=O)NC(CC(C)NC(C#CC(C)C)=O)C)CCCCC1(F)F N1(CC(=O)NC2C3CCN(C(C(C)C4CCC4)=O)C32)CCCCCCC1=O C(C(C)(C)OCC(=O)OC)OC(C1(CC)CC1)=O C1(C(N2CC(CCNC(c3ccc(C(N)=O)nc3)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C(CCSC)O)=O)C2CCC(C2)C1CNC(=O)CSc1cccc(Cl)c1 c1(NC(C=C(C)CNC(=O)CCc2nc(O)n[nH]2)=O)ccsc1C c1(C(=O)NCc2c(CNC(=O)CCF)cccc2)cccc(=S)n1O C1(CNC(C2OCCN(C)C2)=O)CCC12CCN(C(=O)CCC#N)CC2 C1(C)(C(=O)NC2CN(C(CN(C(=O)C3CC3)C3CC3)=O)C2)CC(C#N)C1 N1(C(c2n(C)cc(I)c2)=O)CCC(NC(=O)CC(F)F)C1(C)C N1(CC(=O)O)CCCN(C(c2c(O)cccc2Br)=O)CC1 c1(NC(=O)Nc2ncc(NC(c3ccc(Cl)cc3)=O)s2)ccc(Cl)cc1Cl C1(CC)CN(C(C2(CC)CCC2)=O)CC1C(=O)NCC12CSCC1C2 N1(C(CCC2CCCN(C(c3cnn(C)c3N)=O)C2)=O)Cc2ccncc2C1 C(=O)(C(C(C)C)C(C)C)Oc1ccc(C)cc1.c12cccc(Cl)c1Cn1cc-2nn1 N12CC(C(O)C1)CNC(=O)C2=O.CC1(C)CC1(C)COC(=O)OC(C)(C)C c1(C(N2CCC(n3cc(Cn4ncccc4=O)nn3)C2)=O)cc2cnccc2[nH]1 C1(OC)CN(C(=O)C=CC2CCOC2)CCC1NC(c1cccc(OC)c1C)=O CN1CCC(N(C(=O)C(C2CC2)N(C(=O)Cc2ccc(F)cc2)C)C2CC2)C1=O c1(CNC(C(C)=C2CCCC2)=O)ccc(C(=O)NCc2ccco2)cc1 c1(C(N2CC(CNC(c3csnn3)=O)C(O)C2)=O)cc(F)cc2cnccc12 C1(N(C(=O)NC(C)C(C)n2cccn2)C)CCC(C)(C)C1 N1(C(C(CC=C)CC)=O)CCCC(C)(C)C1CNC(c1ccc(F)o1)=O c1(CN(C)C)ccccc1CNC(c1ccc(CCN2CCCC2=O)cc1)=O c1(C(N(CC(CC)NC(c2c[nH]c(C(N)=O)c2)=O)C)=O)ncc(C)cc1C c1(C(=O)NCC(C)(C)NC(C(C(C)C)c2cnc(C)s2)=O)nccn2nccc12 C1(C(=O)NCC(CC)(C)NC(=O)C(C)Cc2ccncc2)CC=CC(O)C1 CCCC(C(=O)OC)C(=O)NCC1CC(F)CN1C(=O)CC1CCC(=O)NC1=O Cc1conc1CCNC(c1nc(CC(F)(F)F)cs1)c1nnnn1CCC1CC1 C(C1CCOCC1)=CC(=O)NC(C=CC(=O)NC1CCN(CC)C1)C CCC(COC)C(=O)N1CC(NC(c2sc(Cl)cc2Br)=O)C(O)C1 CCC(C(=O)NCc1ccc(C(F)(F)C(F)(F)F)s1)C(C)O C(=O)(C1Cc2ccc(F)cc21)N1CC(CCNC(C2CCCC(O)C2)=O)C1 CC1CCN(c2ccc(CNC(C3CC(O)C3)=O)cn2)CC1 C1(C(=O)NC(CC)CNC(C2CCC(C)(C)CO2)=O)CCC2(CCCC2)CC1 C(C(C(=O)N(C1CC(NC(c2cc(C(C)=O)[nH]n2)=O)C1)C)N(C)C)OC C(=O)(C(C)(C)CCC)N1CCC(CCOC)(NC(C2(CC#C)CCCCC2)=O)C1 N1(C(C(CC=C)(C)C)=O)Cc2occ(C(N3CC(=O)NC(CC)C3)=O)c2C1 c1(CCNC(C(c2ccc(OCC3CC3)cc2)N(C)C)=O)ccccc1Cl c1(CC(N2C(C3CCCN(C(C)=O)C3)CCC2)=O)sc(N(C)C2CC2)nc1C N1(C(C(c2c(C)noc2C)C)=O)CCC2(CCCN(C(=O)C3=CSCS3)C2)CC1 C1(C(N2CCC(C)(C(=O)OC)C2)C(=O)NCC(=C)C)CCCOCC1 c1(OC)c(C(=O)N(CCNC(=O)CN(C)CCO)C(C)C)cc(F)cc1F c1(NC(=O)NC2C(C)(C)CC2)nc2ccc(F)cc2s1 c1(OC)ccnc(O)c1C(=O)NC1CCC(N(C(=O)Cc2ncc(Cl)s2)C)C1 C1(NC(COCCOCC)=O)CCCCN(C(c2ccc(OC)cc2F)=O)C1 c1(C2CC(c3ccc(C)cc3)(O)C2)nn2cc(C)nc2s1 c1(CC)cc([N+](=O)[O-])ccc1Oc1ccc(C)c(NC2CN(C(=O)COC)C2)c1 C1(NC(c2c(C)n(C)cc2)=O)CCN(C(c2cnc(C3CC3)nc2O)=O)CC1C C1(C(=O)NCCn2ncc(C(N)=O)c2)CC(O)CN1C(c1scnc1Cl)=O N1(C(C(C=C)OC)=O)CCCC(O)(CCNC(c2cc(SC)n(C)n2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(c3ccccn3)=O)C2)cc2cc(F)ccc2o1 C1(C2CCOCC2)(C(N2CCC(CNC(CCCC=C)=O)CC2)=O)CC1(F)F CC1CCC(CC(=O)NCCNC(C2(C#N)CC=CC2)=O)CC1C c1(-c2ncc(C(N3CC(NC(CCCC)=O)C3)=O)s2)ccc(C)c(C)c1 N1(C(C2C(C)C2)=O)CCCC2(CCCN2C(=O)C(c2ccc(Cl)cc2)O)C1 N1(C(C)C(N)=O)CCC(C)(NC(=O)CC2C=CCC2)C1 N1(c2nc(N(CC(=C)Br)C)c3c(n2)n(C)cn3)CCc2sc(S(N)(=O)=O)cc2C1 C(=O)(C1=CC2(CCN(C(=O)C(CO)C(F)(F)F)C2)C1)N(CC(C1CCCC1)O)C N1(Cc2cccc(CCF)c2)CCC(C2(C3CCCN3)CC2)CC1 N1(C(C(C)OCC)=O)CCN(C(=O)CC2(OC)CCC2)C2CCCC12 CC(CNC(c1cn(CCNC(=O)C(C)(Cl)Cl)nn1)=O)S(N)(=O)=O c1(C(N2CC(NC(c3nccc(C)c3)=O)C(C#N)C2)=O)ccccc1S(C)(=O)=O c1(C(N2CC(CC=C)(NC(=O)Cc3cnns3)C2)=O)cc(N)cnc1C c1(CCC(=O)NC(CNC(C2CCC(COC)C2)=O)(C)C2CC2)cnn(C)c1C C1(COC)(NC(N2CCCC(CCNC(=O)OC(C)(C)C)C2)=O)CC(F)(F)C1 c1(N2CCC(N(C)C(c3ccc([N+](=O)[O-])s3)=O)C2)nc(Cl)nc2nc(Cl)n(C)c12 C(=O)(CC(O)CCCC)NC(C(N1CC2(CC(=C)C2)C1)=O)C1(C)CC1 N1(C(c2cc(C)ncc2C)=O)CC(F)(F)CC1(C)CNC(=O)CC(C)C1CC1 C1(F)(C(N2CCC(N(C(=O)CCOC3CC3)CC)C2)=O)CCS(=O)(=O)C1 C1(C(=O)NC(c2c(C)nccc2)C)CC1C1CN(C(=O)C(C2CC2)N(C)C)C1 c1(CC2(C(=O)NCC3CC3Cl)CN(Cc3cn(C)nc3)C2)ccc(F)cc1F N1(C(C(C(C)C)SC)=O)CCCN(C(c2ccc(C(F)(F)F)c(F)c2)=O)CCC1 c1(C(=O)NCC2N(C(C3(C=C)CCOCC3)=O)CC2)cccc2ccsc12 c1(C(=O)OC)c[nH][nH]c1=NC(=O)C(CNC(C1CNC(=O)C1)=O)Cc1ccccc1 C1(CC)(NC(c2nc(C)c(C)o2)c2nnnn2CC2CCOC2)CCCCCC1 C1(c2ccc(C)o2)C(C2CC2)CCN1C(=O)C(=O)NC1CC(C)S(=O)(=O)C1 C1(C(=O)NCCC2OCCN(C(c3c(COC)cco3)=O)C2)CCCCC1(F)F C1(OCC)(OCC)CC(C)(C(=O)NC23CC2CN(C(=O)C=Cc2cnc[nH]2)C3)C1 c1(C(=O)NC2C(C(=O)Nc3n(C)nc(Br)c3)C2)nc2ccccc2n(C)c1=O c1(C(N2C(C3(O)CN(C(CC(C)C4CC4)=O)C3)CCC2)=O)cc(Br)n(C)c1 C1(CNC(c2ccc(-c3ncon3)cc2)=O)CCCN(C(C2CCCOC2)=O)C1 c1(C(N2CC(NC(c3c(C)ccnc3)=O)C(CO)CC2)=O)cc(C)c(Cl)c(C)c1 c1(C(=O)NC2C(CNC(C(C)=C3CCCC3)=O)CCC2)c(C)nc2sc(C)cn12 C1(NC(C2CC2F)=O)CCN(C(c2cccnc2C2CC2)=O)CC1F c1(CC)cc(N)ccc1C(=O)NC1CC(NC(=O)Cc2cn(C)nn2)C1 N1(C(CCCCCN(C(=O)CCC2CC2)C)=O)CCC2(CNC(=O)N2)C1 C1(CN(CCNC2CC2)CC)Cc2ccccc2O1 C(=O)(C1=CCC(C)(C)CC1)N(CC(=O)OC)C.c1(=O)[nH][nH]c(=O)c2occc12 Cc1nc2ccccc2n(CCNC(=O)CN(C)C)c1=O C(CC(C)(C)C)(C(=O)N(CCC(C)NC(=O)C(c1cn(C)nc1C)O)C)OC C12(NC(C(C3CCC3)OC)=O)CC3CC(C1)CC(NC(=O)CCC(C)(C)F)(C3)C2 C1(CC)CN(C(=O)COCc2cc(C)no2)CCC1NC(=O)CCCn1cccc1 Cc1[nH]c(C(=O)NCCC2CCCCC2C)c(C)c1C(=O)Nc1sccc1Cl N1(C(C2N(C(CSC(C)(C)C)=O)CCCCC2)=O)CC(CO)C(C2CC2)C1 C1(NC(C(CN(C)C)N(C)C)=O)CC2C(NC(=O)CCc3ccsc3)C2C1 Cc1cccc2c(C(=O)N(CCOC)Cc3ccccc3)cccc12 N1(C(C2CCC(CC)C2)=O)CCC(CN(C)C(C2(CO)CC2)=O)CC1 c1(C(=O)N(CCCSC2CCCN2C(=O)Cc2cscn2)C2CC2)ncc[nH]c1=O N1(C(Cc2cn(C(C)C)nc2)=O)CCC(C)(NC(C2CCC(C)CC2)=O)C1 CC(C(=O)NCCCN(CCO)C(c1cc(Br)ccn1)=O)C(C)(F)F Cc1cc(C)n2nc(CC(N3CCC(NC(c4ccncc4)=O)C3)=O)nc2n1 N1(C(C)=O)CCCN(C(C2CCCC2CNC(=O)CCCSC)=O)CC1 c1(N(C)Cc2c(C)cco2)nc2c(c(=NC(C)c3nnnn3C)[nH]1)SCC2 C(=O)(C(CCS(C)=O)N(C)C)NC(CNC(c1c(C)nc(C)[nH]1)=O)C(C)C C(=O)(CC(C)CC(C)C)NCC(C1CCC1)NC(c1c(C)cno1)=O C1(N)CC12CCC(N)CC2.N1(CC(=O)C(C2(O)CC2)=O)CCN(C2CC2)C1=O c1(CC(N2CCC(N(C(=O)C(F)(F)c3nccn3C)C)C2)=O)ccc(O)c(F)c1 C1(OCC)C(N=c2[nH]c(=N)[nH]c(=NCc3cn4c(n3)CCCC4)[nH]2)CC1(C)C CCCCC(CC(=O)NCCCCCF)NC(c1ncccc1F)=O c1(NC(CSCC(C)C)=O)ncccc1N1CCCC1 c1(C(=O)Nc2scc(-c3cccc(CNC(C)=O)c3)n2)cc(I)ccc1Cl N1(C(C2CCN(C)C2=O)=O)CC(NC(c2cc(CO)ccc2Cl)=O)CC(C)(C)C1 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)CCC2CCCCO2)CC1C C(=O)(CCCC(=O)OC)NCCCCC(C)NC(c1cn(C)nc1C(F)F)=O c1(C(=O)NCC(C)CNC(c2ccncc2N=[N+]=[N-])=O)nc2n(c1Cl)CCCC2 c1(NC(C2CC(=C)CN2C(C2CCN(C)CC2)=O)=O)cc2[nH]ncc2cc1OC C1(C(=O)NC2C(CNC(CC(C)C3CC3)=O)CCCC2)CCC2(C(C)C)CC12 C1(C(N(CCNC(c2ccsc2Cl)=O)C2CC2)=O)COCCC1c1ccccc1 c1(C(=O)NCCCCN(C(C(CCC)O)=O)C)ccc(Cl)c2ccccc12 c1(C(N2CC(C(=O)NCCNC(C=C(C)C(C)C)=O)C2)=O)cn(CCO)nn1 c1(C(=O)NC(CC2CCCO2)C(=O)O)ccc(Br)cc1C(F)F C1(NC(c2ccc(SC)s2)=O)CN(C(c2cnc(C(C)(C)C)s2)=O)CCC1C C=CCC(C)(C)CC(=O)NCC1CN(C(c2cccc(=S)n2O)=O)C2(CCC2)C1 C1(CC#C)(C(=O)N(CC(C)N(C)C(c2ccn(CCC)n2)=O)C)CCOC1 c1(CC(=O)N(C2CCN(C(C3CCCC(F)C3)=O)C2)CC#C)ccccc1F c1(C(N2C(CC(N3CC(CCC)OCC3)=O)CC2)=O)cc(C)cc(O)c1 C1(C)(C(N2CC(C(=O)NOCC(N)=O)(COC)C2)=O)CC(O)CN1C C1(CNc2ccc(Nc3ccccc3)cc2)C2Cc3ccccc3C12 C1(CC(=O)N(CCCCNC(C2CCC2)=O)C)COCC(C)(C)O1 N1(C(c2cc(=N)[nH]cc2)=O)CC(NC(=O)Cc2cnns2)CC2(CCC2)C1 c1(CC(=O)NCC#CCNC(c2ccc(C)cc2)=O)cccc(Br)c1Cl CCCC(C)(C)CC(=O)NC1(CC(=O)NCC(c2ccccn2)C)CCC1 N1(C(C(=O)NCC2CC2)=O)CCCC(CNC(C2COC(=O)N2)=O)C1 C1(CN(C(=O)COCC2CCCO2)C)CCCN(C(=O)C(c2cnn(C)c2)O)C1 c1(C(=O)NC2CCCC2NC(C2CCC2(F)F)=O)cnc2c(F)cccc2c1 C(C(C(=O)NC(C)C(=O)NC(C)(C)C)NC(c1cc(C)c[nH]1)=O)OCC C1(NC(c2onc(C(C)(C)C)n2)=O)CN(C(=O)CC#N)C2CC12 CC1CN2CC1CC2=O.C1(C)(CCC(=O)NCCC23CCCC2C3)CC1(F)F c1(C(=O)NC2(CO)CCN(C(Cc3n(C)cnn3)=O)C2)ncnc2c1CCC2 c1(C(=O)NC(CNC(c2c(CC=C)cccc2)=O)C2CC2)cn2c(n1)CCCC2 Nc1cc(C(=O)NCC2CCC(NC(c3ccc(Cl)cc3Cl)=O)CC2)ncc1F C12(NC(c3cc4c(s3)COCC4)=O)CCCC1CN(C(c1cnn[nH]1)=O)C2 C(C1=NOC2CCCC12)NC(C(CCSC)NC(=O)CCc1cncnc1)=O C(=O)(CCCC(=O)N(C)C)NC(C(C)NC(c1cccc(N)c1)=O)C CN1CC(=O)NC(CC(=O)NC2COCCC2NC(=O)C(C)(C)O)C1=O C1(C(=O)NCCOC2CC2)(CC)CCCN1C(C1CCCC(C(=O)OC)C1)=O c1(C(=O)NC(C(C)NC(C(CC(C)C)OC)=O)CO)ccnc2[nH]nnc12 C1(C(N(C(c2ccc(C)cc2)C)C)=O)CN(C(=O)Cc2ncoc2C)CCC1O C1(C(N(C(C)CCNC(=O)CCCSc2ccccc2)C)=O)CC2CC1CO2 N1(Cc2ccc(-c3n(C)cnn3)s2)CC2(CCCC2)c2cccc(F)c21 N1(C(C(CC)OC)=O)CCC2(C1)CN(C(C13CCCCC1C3(F)F)=O)CC(C)O2 C1(C(N(C(C(=O)Nc2cn(CC=C)nc2)C)CC)=O)CC2(CSC2)C1 N1(C(C2CCC(=O)C2)=O)CCCCC1CCNC(c1cc(Cl)n[nH]1)=O N#Cc1nc(Br)cnc1NC(C1CCCN1Cc1ccc(F)cc1C(F)(F)F)=O Cc1nc(Cl)sc1C(N1CCN(c2noc(C(C)C)n2)CC1)C(=O)NCC1CC1 C(C(O)C(C)(C)C)NC(CCCn1cc(-c2cn(C(C)C3CC3)nc2)nn1)=O CC(C)CC(N)CC(=O)N1CC2CCCC1C2CO C1(NC(C(C)C2CCC2)=O)CCCC12CN(C(C1COC(=O)N1)=O)C2 c1(C(=O)NCC2CCC(NC(CC(C)C3CC3)=O)C2)cn2cc[nH]c(=O)c2n1 N1(C(C(CC=C)C)=O)CCC2CCC(NC(c3cc4n(n3)CCCN4)=O)C12 Cc1cc(F)c(CN(C2CCN(S(=O)(=O)CC3CCCCN3C)C2)C)c(F)c1 c1(CC)nnc(C)n1C.C1(C(N2CCC(N3C(=O)CN3C)C2)=O)C2COCC12 C1(C(CCC=CCCCNC(CCC)=O)=O)CCCCC1C C1(F)(C(N2CC(SC)C(NC(C3CC(C4CCC4)C3)=O)C2)=O)C(C)(C)C1(C)C C1(C(N2C(c3ccc(CC)s3)CCC2)=O)CC(CN)C12CCC2 C1(C(=O)NCC(=O)NCC(=O)Nc2cccc(OC)c2)CCOC(=O)CC1 C1(CNC(C2C(CC)C2)=O)CCCC2(CN(C(c3cccc(C)c3O)=O)C2)O1 c1(C(=O)OCC)cc(NC(C2CC(NC(C3CCC(C)S3)=O)C2)=O)on1 C1(CC(=O)NC2C(N(C)C)CC2O)CCN(C(=O)CC2CC3(CC3)C2)C1(C)C N1(C(CCC)=O)CC2(C1)OC1(C)CC2(NC(=O)C=C2CC3CCC(C2)N3C)C1 c1(CCC(N2CC(C(N(CCOC)C)=O)C(O)CC2)=O)ccc(F)c(F)c1F c1(C(=O)NCCC(CC)(CC)NC(=O)C(O)CN(C)C)n[nH]c2c1CSCC2 C1(C2CCOCC2)(C(=O)NCc2cn(C3CCCC3)cn2)CCNC1 CC1CCCC1(C(N1CCC(CCO)C1)=O)NC(=O)CC1C(C)(C)C1(C)C c1(C(N2C(C)CC(NC(=O)CC(c3ccc(Cl)cc3)O)C2)=O)cccc(F)c1N C1(O)(C(C(=O)NCCCC2CC2)NC(C2C(C(C)C)OCC2)=O)CCCCC1 N1(C(C2C(C(C)O)C2)=O)CCC2(NC(c3cc(Br)co3)=O)CCCC12 C12(NC(C(CCCC)N(C)C)=O)CCC(F)(F)CC1CN(C(=O)C(F)=C(C)C)C2 C1(NC(c2cn(-c3cccc(C)c3)nn2)=O)CCN(C(c2ncc[nH]2)=O)C(C)C1 C=CC1(C(=O)NC(c2noc(C)n2)C)CCN(C(c2ccco2)=O)CC1 N1(C(C(CCC)(C)C)=O)CCOC2(CCCN(C(=O)CNC(C)=O)C2)C1 C1(C(=O)NC(C(C)C)CCN(C(=O)CCN2CCCC2)C)CN(C)CC(C)O1 Cc1cc(C(N2CC(O)CC2C(=O)Nc2cccc(O)c2Br)=O)ncc1[N+](=O)[O-] C12(CNC(C(CC)N(C)C)=O)CCC(CC1)CN2C(=O)CCNC(=O)CO CC1CCCC1(C(=O)N(CCCN(C)C)C)NC(C1CCCC1O)=O CCC(C)C(C)(c1nnnn1C1CC1)Nc1cnn(CCO)c1C c1(OC)cc(F)c(C(=O)NC(C)C(C)NCc2ccc3c(c2)OCC3)c(Cl)c1 Cc1cc(C(N2CC3CCN(C(=O)CS(C)(=O)=O)CC3C2)=O)ccc1[N+](=O)[O-] CC1(C)CCOC1CC(=O)NC(C(N1CC(O)(c2nn[nH]n2)C1)=O)C1CCC1 C12(C(=O)NC3(CNC(=O)CC4CCCCC4)CCOC3)CC3CC1C2C3O c1(OC)ccccc1S(=O)(=O)CCCN1CC2C3CCC(O3)C2C1 CC1CN(C(C2CCCN2C(c2ccc(O)c(F)c2)=O)=O)C(C)CO1 N1(C(C2CC(=C)C3N2CC3)=O)CCC2CCOCC2C1 c1cc(N2CC3CCC3C2)nc(N2CCC(C3CCCO3)C2)n1 C(=O)(C(O)CCCNC(C1CCC(OC)C1)=O)NCc1c(OC)cccc1 Cc1ccc(C)c(OCC(=O)NC2C3CC2N(C(=O)C=Cc2ccco2)C3C)c1 c1(C(=O)NC2CN(C(CCC(C)OCC)=O)CC(F)C2)cc(Cl)cc(C)c1OC C1(CN(C(=O)COCP(C)(C)=O)C)CCCN1C(=O)Cc1cc(C2CC2)on1.OC C#Cc1ncccc1CNCCc1ccc(N2CCOCC2)nc1 C1(CCC(C)C)CCN(Cc2cnc(C(F)(F)F)nc2)CC1 c1(N2CCCC(NC(c3c(C(C)(C)C)noc3)=O)C2)cccc(F)c1[N+](=O)[O-] N1(CC2CC3(C(F)F)C(C2)C3)CC23CCCC2(COC3)C1 c1(CN2C(C(=O)NCCCOC(C)C)CC3CC32)c[nH]c2cc(C#N)ccc12 C(=O)(C1=CC2C=CC(C1)C2)NC1CCC(CC(=O)NC(COC)C)C1 N1(C(C2C(C)(C)C2NC(=O)CC2CCOC2(C)C)=O)CCCC(F)CC1 C(=O)(CCCC(C)NC(c1c[nH]c(C#N)c1)=O)NC(C(=O)OC)CO C1(C(=O)NC(C2CCN(C(c3cn(C)nn3)=O)C2)C)Cc2cc(Cl)ccc2C(=O)O1 Cn1nc2c(c1C(=O)NCCN1CCN(C(C3CCNC3=O)=O)CC1)CCCC2 C1(NC(C=Cc2c(C)ncs2)=O)CCCN(C(=O)CP(C)(C)=O)CC1 C1(OC)(OC)C(C(=O)NC(C2(O)CCCCC2)C)CC1(F)F c1(CC)ccnc(C(N2CCC(F)(C(=O)NCc3nonc3N)C2)=O)c1 N1(C(C=COCC)=O)CCC(NC(c2ccco2)=O)C(F)C1 c1(C(N2CC3(CCN3C(c3ccc[n+]([O-])c3)=O)C2)=O)cccc2c(Br)n[nH]c12 N1(C(c2cn(CCN(C)C)nn2)=O)CCCC(CNC(c2nnn(C)c2N)=O)C1 C12(OC)CCC(C(=O)NC3CC(N(C(=O)C(O)C(C)C)C(OC)OC)C3)(CC1)C2 N1(N(C2CN(C(C3(C(C)(F)F)CC3)=O)CC23CC3)C)CC2(CCCCCC2)C1.C=O C1(NC(C2(CC)CCN(C(C3CCC4CC34)=O)CC2)=O)CCC2(CCC2)CC1 C1(NC(C(CC)OCC)=O)CC12CC(NC(c1cc(-n3nccn3)ccn1)=O)C2 c1(C(N(CC(C)N(C(C2C(CCOC)C2)=O)C)C)=O)ccc(O)nn1 C12(C(=O)NC3CC(F)(CNC(C4(CC#C)CCCC4)=O)C3)CC3CC1C2C3 C1(F)(C(=O)NC2CCN(CC)C2)CCCN(C(=O)C(C(=O)OC)OC)C1 C1(C(=O)NC2CCCCCC2)(COC)CCCCN1CCC(=O)N(C)C C1(OC)(CNC(=O)C(C)SC)CN(C(c2occc2Cl)=O)C1 Cc1cccc(O)c1C(=O)NC1CCCC(NC(C2(CO)CC(F)(F)C2)=O)C1 C(C(C)(CO)OC)NC(CN(C(=O)CC(C)n1ccnc1)CC#C)=O c1(C(=O)NC(CCC)C(=O)N(C)Cc2ccn(CC)n2)ccc2c(c1)COC2 c1(C(=O)NC2CC3CC(NC(C4CC4F)=O)C3C2)cc2ncccc2[nH]1 C1(NC(=O)CC2CCOC2=O)C2CC1CN(C(=O)Cc1c(F)cccc1Br)C2 c1(C(=O)NCC2C(NC(C3(C#C)CCC3)=O)COC2)cnc(C)nc1COC CCC(CN(C)C)CC(=O)NCCCCC(C)NC(c1csc(COC)c1)=O CC1CCN(C(=O)COC2CCCOC2)CCN1C(c1csnc1Br)=O C(C(C)(CC)C(=O)NC(CC)C(C)(C)C)NC(C(C1CC1)OCC)=O NC1(C(=O)NNC(=O)Nc2ccc(F)cc2)CC12CCOCC2 Cc1ncccc1C=CC(N1CC=C(CNC(C2CC(C)CO2)=O)CC1)=O c1(C(N2C(CN(C(=O)C(=O)C(C)(C)C)CC)CCC2)=O)ccc(OC)c(Cl)c1 N1(C(CC2(OC)CN(C(C(C)OCCC=C)=O)C2)=O)CC(CO)C(C2CC2)C1 C1(C)(CCNC(C2C(OC)CC2)=O)CCCN1C(=O)C1CC1 n1(CC)c(CCN2CCCC(C(=O)O)(CO)C2)nc2ccccc12 c1(OC)noc(C)c1C(=O)NCCC1(O)CN(C(c2cncc(O)c2)=O)C1 N1(C(COc2c(C)cc(Cl)cc2)=O)CCC2CCCC12CNC(=O)C(C)(C)C1CC1 CC(=O)CCCC(=O)N1CCC(N(C)C(c2ccc(-c3cscn3)nc2)=O)C1 c1(NC(c2c(CCC)n(CCO)nc2)=O)ccc(C)c(C)c1N C(CCCC(=O)NCC1CCOC1C(=O)NCC(C)C1CC1)NC(C)=O CC1CCN(CC(=O)N(C(C)CN(C)C(c2ccn(CCF)n2)=O)C)CC1 c1(C(=O)OCC)ccncc1NC(=O)NC1CC(C)CCS1 c1(CNC(C2C(C)(C)COCC2)=O)cccc2c1CCC2 C1(C(=O)NCc2scc(CNC(C(F)OC)=O)n2)CCC(=O)N1C(C)C C(CCN(C(=O)C=CBr)C)(C(C)C)NC(C(CC)OC1CCCC1)=O c1(CCC)ccc(CC(=O)NCC(O)CN(C(=O)C(C)=CC2CC2)C)cc1 C1(NC(C(C)=C(CC)C)=O)CN(C(C2COCCC2(F)F)=O)CC12CC2 CCC(C)CCC(=O)N1CCC(Cn2cc(-c3cccc(C(N)=O)c3)nn2)C1 N1(C(CCOCCOCC)=O)CCC2(CCC2)C(NC(=O)C(=O)NC2CC2)C1 c1(OCC)cc(CNC(=O)C(N2CCC(C)(c3cccc(Cl)c3)C2)=O)cc(F)c1 c1(OC)cc(OC)c(C(=O)NC(CNC(=O)C(C)C(C)(C)C)C2CC2)cc1OC c1(C(=O)NC(C(CSC)(C)C)c2nnnn2C)ccc(OC)c(C(F)(F)F)c1 C1(CC)CN(C(C2(C(=O)OCC)CC2)=O)CCC1NC(=O)Cn1nccn1 c1(C(C)NC(=O)NC2C(OCC)(OCC)C2)ncc(Cl)nc1Cl C1(CCC(=O)NCC(COC)NC(c2cn(C(C)C)nc2C)=O)CC(C)(C)CO1 N1(C(C2C(C)CC=CC2)=O)CCCC(O)(CCNC(c2ccnc(CO)c2)=O)C1 c1(C(N2CCOCC2C2CC2)C(=O)NCCCF)cc2nc(F)ccc2o1 N1(C(C2CC(OCC)C2)=O)CCN(C(=O)C2=NOCC2)C(CCSC)C1 C1(CC)CCN(C(=O)CS(C)(=O)=O)C1C(=O)NC(C)C(C)n1cccn1 CCC(C)C(O)C(=O)N1CC(CCNC(c2csc(-c3cnn(C)c3)n2)=O)C1 C1(C(N2C(CNC(C(CC#C)C)=O)CC(F)(F)C2)=O)CC2(C1)CC(C#N)C2 Cc1ccc(-c2ocnc2C(=O)NCC2CC2NC(C2(C)CC2(F)F)=O)s1 C=C(CNC(C1CC1(F)F)=O)CCNC(=O)C(O)Cn1cncn1 C1(C(N2C(C=CC(N3C(CN(C)C)C=CC3)=O)CCC2)=O)CC(=O)CC(=O)N1 c1(-c2c3cc(C(=O)NCC(=C)F)sc3ccc2)cnn2ccc(C)cc12 c1(C2C(c3cc(-c4ccoc4)[nH]n3)C2)ccc(Br)cc1.C12CC1C(=O)NC2=O Cc1cc(-c2nc(-c3cccc(C(F)(F)F)c3)nn2CCC2CC2)c(C)o1 N1(C(C(CC2CCCC2)NC(c2cc(C(C)C)no2)=O)=O)CCC2(CSC2)C1 CP(C)(=O)C1CCCCC1C(=O)NC1C2CC1N(C(C1CC1c1ccsc1)=O)C2 N1(C(CN2C(C)CCC2)=O)CC2(C1)CN(C(c1nnn(C)n1)=O)CC2CO N1(C(C(C2CN(C(C3CC3C(C)C)=O)C2)OC)=O)CCCC2(CCC2)C1 N1(C(c2c(C)nco2)=O)CCC(C)C(CNC(=O)CSc2ccc(F)cc2)C1 c1(C(N(C)CC2(NC(C3C(C=C)C3)=O)CC2)=O)cc(C)c(F)cc1Br c1(CC(=O)NC(CNC(C(COCC)C)=O)CO)coc2cc(CC)ccc12 N1(C(COCC#C)=O)CCCC1C1CCCN1C(=O)CCCOC1CC1 S(=O)(=O)(c1c(Cl)nc2ccc(Br)cn12)NC(Cn1ccc(C(=O)O)c1)=O c1(SC)ccc([N+](=O)[O-])c(NC(C2CC(NC(=O)CC3CC4CCC3C4)C2)=O)c1 S(=O)(=O)(c1ccccc1Br)N1CCC(N2CCN(C(c3cocn3)=O)CC2)CC1 C(CCCCCC(=O)NC12CCC(CC1NC(C1CCCNS1(=O)=O)=O)C2)SC S(=O)(=O)(c1cnc(N2CCC(CCC)C2)cc1C)NC(CCC=C)(C)C CN1CCC(NC(=O)C(CC(F)F)NC(c2coc(C(F)F)c2)=O)C(C#N)C1 CC1(C)Cc2cc(CS(=O)CCc3cccc(O)c3)ccc2CO1 C1(COC(C)C(=O)NC2CC3CCC2C3)COCCC1(F)F N1(C(c2n(C)c(=O)ccc2)=O)CCC2(CCCC2C(NCP(=O)(O)O)=O)C1 C(=O)(C(C(C)(C)C)C1CCC1)NC(CC1CN(c2cc(COC)ncn2)C1)C C1(C(N(C)CCC2CCOC2)=O)CCCCN1C(=O)CCC(=O)N1CCCC1 c1(CN2CC(O)(CCC)C2)c(OC)ccc(F)c1Br C1(OC)CN(C(c2sc(-c3ccn(C)n3)nc2C)=O)CC1NC(c1ccoc1)=O N1(C(c2ccc(C3CC3)nc2O)=O)CCC2(CCC2)C(O)C1 c1(N2CCN(CC(=O)OC)CC2)ccc(CNc2cccc(F)n2)cc1C C1(C(N2C(CNC(C3CC(F)(CO)C3)=O)CC(C)(C)C2)=O)CCc2nc[nH]c2C1 C(CCCCC(=O)N1CC(N(C)C)C1)NC(C1(C(C)=O)CC1)=O c1(-c2ccc(OC)nc2OC)cccc2nc(C(=O)Nc3cc(C)ns3)ccc12 CCC(C)C(O)C(=O)NCCN1CCC(NC(=O)CCCn2cccn2)CC1 Cc1cc(C(N2CCC(CNC(=O)C(F)(F)c3cncs3)C(C)C2)=O)cnc1O c1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCCC2C)cncc2ccsc12 c1(C(=O)NCC2C(CNC(C(F)=CC)=O)C2)c(C)ncn(C)c1=O CC1CCN(C)CCN1C(=O)C(N1CCC(CCP(C)(C)=O)CC1)=O CCC(C)C(C(=O)NCC(C)(C)CNC(=O)CC1(O)CCC1)NC(N)=O Cc1cn2cc(C(=O)NC34CCC(C3)N(C(=O)CC3COCCN3C)C4)nc2s1 N1(C(c2c(CCC)nns2)=O)CC2CC(C1)C(CO)C2NC(c1nonc1N)=O N1(C(=O)COC2CN(C(c3cc(Cl)ccn3)=O)C2)Cc2cncnc2C1 c1(C(N(CCNC(c2occ(C)c2C)=O)CC)=O)cccc2cccnc12 c1(NC(C)=O)ccc(NC(c2cnnc(O)c2S)=O)c(Cl)c1 N1(C(C(F)=CCC)=O)CCC(NC(=O)COCc2ccccn2)C(CC)C1 c1(C(N2CC(COC)N(c3nccc(C)n3)CC2)=O)c(C)ccc(Br)c1F n1(CC)c(SC(C)C(=O)NCCCn2cc(C(=O)OC)nn2)nc2ccccc12 CC(C(=O)NCC1(O)CN(C(c2ccc(O)c(Br)c2)=O)C1)S(N)(=O)=O c1(C(N2CCN(C(c3ccnc(Cl)c3)=O)C3CC23)=O)cccc([N+](=O)[O-])c1Cl C=CCCCC(C(=O)NC(C)(C)CCCC)NC(=O)COCCCN=[N+]=[N-] C1(CCC(=O)NCC(N(C)C(C2(C)CC2(F)Cl)=O)C2CC2)CCCCN1C C(CN=c1ccnc(C(C)C)[nH]1)(CC(C)C)NC(C1Cn2c(C)nnc2CC1)=O C1(CNC(C2(CCOC)CCCC2)=O)CN(C(=O)CS(N)(=O)=O)CCCO1 c1(NCC(C(C)C)C)cc(=NCC(F)CO)[nH]cn1 C1(CNC(C2(COC)CCC2)=O)C=CC(NC(=O)C(C)(C)C2CCCCO2)C1 C(CCC(N)=O)(C(=O)N(C)CC1(O)CN(C(C2(C)CCN(C)C2)=O)C1)NC(C)=O C1(c2n(-c3ccccc3)nc(-c3nc[nH]n3)n2)CCCC2(CCC2)O1 C=CCC(CNC(=O)Cn1cc(C2CC2)cn1)C(=O)NCc1nnnn1CC C12(OC)CCC(C(N3CC4CC3CN4C(=O)C(CCSC)OC)=O)(CC1)C2 Cn1ccc2[nH]c(C(=O)NC3(C)CCN(C(=O)C(F)=C4CCC4)C3)cc12 C(=O)(C(C)(C)CC(C)=O)N1C2(C(NCP(OCC)(C)=O)=O)CC(C)(C1)C2.C(C)(=O)OC C1(NC(C2(C3CC3)CC2)=O)CS(=O)(=O)CC1N=c1[nH]ncs1 c1(OCC(=O)NCC(CNC(C(C(C)C)OC)=O)F)cccc(S(C)(=O)=O)c1 C(=O)(C1=CC2CCC(C1)C2)N1CC(O)(CCNC(c2cnc(OC)c(C)c2)=O)C1 CC1OCCCC1C(=O)NC12CC(C1)N(C(=O)Cn1ncnn1)C2 c1(C(N2CC(F)(C(=O)Nc3cn(CCC)nc3)C2)=O)cccc(Br)c1 C1(CC=C)(NC(C2(C(C)C)COC2)=O)CCN(C(c2ccc(SCC)cc2)=O)C1 c1(CC)cc(C(=O)NCC=CCNC(C2(C)CCCC2(F)F)=O)cc(O)n1 C=CCC(CC=C)C(=O)N1CC(C)N(C(c2nnc(O)cc2C)=O)CC1C C1(c2ccc(C)o2)CS(=O)CCN1C(C1CC1c1ccc(F)cn1)=O C(=O)(CS(=O)(=O)CC(=O)NCC(CO)NC(=O)CC1C=CS(=O)(=O)C1)OC c1(C(=O)NCC2C(C)CN(C(C3(CCF)CCOCC3)=O)C2)cc(N)cc(O)c1 c1(C(=O)NCC(C)N(C(CC2(C=C)CCC2)=O)C)cccn2cncc12 C1(C(=O)NC(CC=CC)CO)CN(C(=O)C(C)CSC)CC1(F)F N1(C(C(C)(C)N2CCOCC2)=O)CC2CC(C1)CN(C(C1CCCCO1)=O)C2 C(=O)(C(O)CCCN1CCCC1c1ccc(Cl)c(Cl)c1)OC C=C=C(C)CC(=O)NCCCC(=O)NCc1cnc(OC)cn1 C1(CNC(C(C)C2CC2)=O)CCC12CCN(C(=O)C=CCN(C)C)CC2 C=C(C)C(C)(O)C(=O)NCC(C(C)C)NC(c1cncc(N2CCCC2)n1)=O O(NC(=O)C(c1cccnc1)NC(c1ccn(CCF)n1)=O)CC(C)C N(C)(C1CN(C(=O)C(=O)NC2CC2)CCc2ccccc21)C(CC(CC)OC)=O c1(C(=O)OCCCN(C(=O)Cc2ccccc2F)CC)ccc(NC)cc1 N1(C(C2(SC)CC(=O)C2)=O)CC(C(=O)NC2CC3(C2)CC(O)C3)CC(C)(C)C1 C=CCC(C(=O)N1CCCC1(C)CCC(=O)NCCOC(CC)CC)NC(C)=O CCC(C#N)C(=O)NC(c1ccccc1)CNC(=O)C(CC)NC1CC1 CCN(C(C)c1ccc2c(c1)OCCCC2)N(C)C1CCOC1 CC1(C)C(NC(=O)CCC2CCCOC2)CCN1C(=O)CCSCCC(F)(F)F Cc1cc(C2CC2)ccc1C(=O)NCC(O)CNC(c1cncc(N)c1)=O c1(C(=O)NCC2(CO)CCN(C(C3CC=CCO3)=O)C2)ccn2c1CCCC2 S(=O)(=O)(C1CCC2(CC1)OCCO2)N(CC(C(=O)OC)Nc1ccccn1)C C(=O)(C(C)CC)NCCNC(=O)COC(C(=O)N(C)CC)C CS(=O)(=O)c1cc(C(N2CC(O)CC2c2ccc(Br)cc2)=O)c(Cl)c(Br)c1 CCC(C(=O)OC)C(=O)N1CC=CCC1C(N1CC(CO)C1(C)C)=O c1(CC(=O)OC)c(C)nn2c1CN(C(=O)COCCCN(C)C)CC2 C1(C(=O)NC2(CO)CN(C(C3(c4ccno4)CC3)=O)C2)C2CCC(=O)C12 C1(C(=O)NC(CCN(C)C)C(=O)N2CCCC(CN=[N+]=[N-])C2)CCC2(CC1)CC2 C1(CC=C)(NC(=O)CO)CN(C(=O)CCc2cncn2C)C1 N(C1CCCc2occc21)C(C1C(C)CCN1C(C1CC(C)(C)CO1)=O)=O CC1CCn2ncc(C(=O)N(C3CCCCN(C(=O)CCF)C3)C)c2C1 c1(OC)ccc(N)c(C(=O)NC(C)CCNC(=O)COC2CCOC2)c1 C(=O)(C(CO)NC(=O)CN1CC2CC2C1)N(C(CO)CO)C C(C1OCc2ccccc21)c1n(-c2ccc(CC)cc2)nc(CO)n1 c1(C(=O)NCC2(F)CCC(NC(C(C)(C)O)=O)C2)cn(CCO)c(=O)nc1O CCCCC(CC)NC(C)(CCC1CC1)c1nnnn1C1CCCC1 CCC(C)(C)C(C(=O)NC1CCCCN(C(c2coc(Cl)n2)=O)C1)OC c1(CC)cc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCc2cc(C)[nH]n2)n[nH]1 c1(C(=O)NC2CC(CCNC(C3CC=CCO3)=O)C2)ccc2nsnc2c1 c1(NC(=O)NCCCC(=O)NCCC2CN(C(C)=O)C2)cc(C#N)ccc1N c1(C(C(=O)NC(CCCNC(c2cnc(SC)s2)=O)C)C)c(C)n[nH]c1C c1(CC(=O)NCC23N(C(C4CCC(C)C4)=O)CC(C2)C3)nn(C)c2ccccc12 C1(C(=O)NCCC(C)C)CCC2(CN(C(=O)CCc3ccoc3)C2)O1 c1(CC(=O)NC(C2CN(C(=O)C=CCF)CCCO2)C)csc2ccc(Cl)cc12 C1(C(=O)NCCCC2C=CCC2)CCOCCN1C(c1scnc1Cl)=O N1(C(C(=Cc2ccncc2)C)=O)CCC2(C1)CN(C(C1CCCC(CF)C1)=O)C2 c1(C(=O)NC2CC(C(C)C)SCC2)cc(C#N)ccc1Cl c1(OC)ccc(CCC(=O)N(CC(F)F)CC2CCCO2)cc1CC(=O)O C1(C(N2C(C#C)CC2)=O)(OC)CCN(C(c2ccc(CC)o2)=O)C1 c1(NC(C2(CF)CCN(C(C(CC)COC)=O)C2)=O)cccc2c1CCC2 C(=O)(C(F)(F)c1csc(=N)[nH]1)NCC(CN(C)C(C1(C(N)=O)CCC1)=O)O O=C(O)CCCCCNC1CCN(C(C2CC2)C2CC2)CC1.c1(O)ncc(Cl)cn1 c1(C(=O)NC2CN(C(CC3(OC)CCC3)=O)CC2C2CC2)cncc2c1CCC2 C1(CC(=O)NCC2(C(N)=O)CN(C(C(C(C)C)F)=O)C2)CCCCC1(F)F N1(C(CC(C)c2cccnc2)=O)CC=C(CNC(c2cc(O)nc(O)n2)=O)CC1 Cc1[nH]nc2ccc(C(N3CC4(CC4)CC3CNC(=O)CC3(C)CC3)=O)cc12 c1(C(=O)NCCCC(c2ccccc2)NC(CCC#C)=O)cc(Cl)c(Cl)s1 C1(C(=O)NCC(C)CN(C)C(C2CCN2C)=O)CCCC1O Cc1ccnc(N(CCCNC(c2cc(O)nn2C)=O)C(C)C)c1[N+](=O)[O-] c1(C(=O)NCC2C(NC(c3n(CC)ncc3)=O)C2)nc(O)nc(O)c1N C1(O)(CNC(Cc2ccc(CC)cc2)=O)CCCN(C(CCCC(C)C)=O)C1 c1(NC(=O)NCCC#C)ccccc1-n1nc(C)cc1C CC1C2CC(C2NC(C2CCN(C)CC2)=O)N1C(=O)C1=CCCOC1 C1(CC)(CO)CCN(C(=O)C(CO)NC(c2ncncc2Cl)=O)C1 C(CNC(N1CCSC1)=O)(CNC(=O)CCSC)OC c1(CC)nc(C#N)cc(=NC(C)CNC(=O)Cc2ccco2)[nH]1 c1(CC(N2C(CNC(C3CCOC3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])cc1 N1(C(CCCOCC)=O)CCCCC12CC(NC(=O)Cc1ccc(CC)cc1)C2 CC1CC2CCC(C1)N2C(=O)CC1COCC1NC(c1ccc2ccoc2c1)=O C(=O)(C(C)(O)C(F)(F)F)NCc1oc(C)c(C(=O)NC2CCOC(C)C2)n1 C1(C(=O)NCC(CNC(c2ccc(C#C)o2)=O)C)CC2(C1)CC2(F)F CC(C)(C(=O)NCCC1CC2CC1CC2O)C1=CC2CCC(C1)N2 C(=O)(C1=C2CCN=C2NC=C1)N1CCN(C(C(N2C(CC)CCC2)=O)=O)CC1 C1(C(N(CC(=O)NCc2scc(C)n2)C(C)C)=O)CCCC1C1CC1 C1(NC(CCCC(=O)NC)=O)C(CNC(=O)C(C)(C)CCC#N)CCC12CCC2 C12(NC(Cc3[nH]nc(C(C)N)n3)=O)CC(N=[N+]=[N-])(C1)C2 c1(OC)cc(I)cc(NCC(C)C(=O)c2ccccc2)c1[N+](=O)[O-] C=CCC(C(=O)N1C(C(N2CC(C#N)C2)=O)CC2CC12)OC c1(C(N2C(CNC(C(C)(C)O)=O)CC2)=O)ccccc1-n1ccnc1O C(=O)(C(O)P(C)(C)=O)C(Cn1cc(CCC2N(C)CCC2)nn1)=O.N1CCC(CO)CC1 c1(C(=O)NCCC2CC(NC(C3(Cl)CC34CCC4)=O)C2)ncccc1F C1(C(=O)Nc2c(C(=O)OC)csc2)CC(C)CN1Cc1cccc(CO)n1 N1(C(CC(C)n2cccc2)=O)CCC(O)C(N(C)C(C2CCCN2N=O)=O)C1 c1(NCC(N2CCN(C(C(C(C)C)SC)=O)CC2)=O)cc(CO)ccc1[N+](=O)[O-] C1(CNC(C=C(CC)C)=O)CN(C(c2ccnn2C)=O)CCC1C(F)(F)F C(c1nc2ccccc2[nH]1)=CC(=O)NC(C)CNC(c1cc(C#N)cn1C)=O C(=O)(CC(C)(CNCC12CCC(O)(CC1)CC2)C(F)(F)F)OCC c1(OCCC)ccc(C(=O)N(C)CCN)cc1OCC1CC1C(=O)C(C)(C)F C1(O)(CN(C(C(CCC)NC(C)=O)=O)C)CCCN(C(C2CC(=O)N2)=O)C1 C=CCC(C)(C)C(=O)N1CCCC(C(N2CCC(OCC3CC3)C2)=O)C1 N1(C(C2CCC(CNC(c3cnn(C)c3Cl)=O)CC2)=O)CC2OCCOC2C1 C(CC(C)=O)(C(=O)NC(C)(C)CCN(C)C)NC(CC1(N)CC1)=O.C1(COC)CC1 C(=O)(CC1=NNC(=O)C1)NCC1(C(C)NC(c2cc[nH]c(=N)c2)=O)CC1 c1(OC)ccc(N(C(=O)C(c2cn(C)nc2C(F)(F)F)C)C)c(F)c1 c1(C(N2CN(C)C(=O)C2C)C)ccc([N+](=O)[O-])cn1 N1(C(c2cc(C(=O)OCC)no2)=O)CC2CC(C1)C2NC(=O)C(O)C(C)CC N1(C(C2CC3CCC3C2)=O)CC2CCC2(C(=O)NC2CCOC2)C1 C(=O)(C(C)C(C)C)NCCN(C(=O)COc1ccsc1)CC=C Cc1nc(C)c(C(N2CCC(NC(c3ccnc(N4CCCC4C)c3)=O)C2)=O)[nH]1 C1(NC(Cn2c(C)nc(C)n2)=O)CC(NC(=O)CC2CC3(CC3)C2)C12CCOCC2 Cc1[nH]nc(C(=O)NC2CCOCC2C(N2CC(O)(C(F)(F)F)C2)=O)c1C C1(CC)CN(C(=O)CCSC2CC2)CCC1NC(=O)CCOCC(F)(F)C(F)F Cn1cc(C(=O)NC2(CNC(c3ccc[n+]([O-])c3)=O)CC2)c(-c2ccccc2)n1 c1(C(N2CCSCC2(C)C)C(=O)Nc2c(CC)cccc2)ccc2c(n1)CCC2 CCC(CC(C)C)C(=O)NC(C(N1CC(=O)NC(=O)C1)=O)C1CCCC1 N1(C(C(C(COC)C)C)=O)CCC2(C1)CN(C(=O)COCP(C)(C)=O)C2 N1(C(c2c(C)nc(O)[nH]2)=O)CCCC2(C1)CN(C(=O)C(O)CCC(F)(F)F)C2 N1(N(CC=C)C)CCC(C)N(C(=O)CC2CCCOC2)CC1.c1(C=O)nccs1 C1(CNC(c2n(CCC)nnn2)c2nnnn2C(C)C)CCC(=O)NC1 c1(C(N2CCN(C(c3c(CC)con3)=O)CC2C(C)C)=O)cc2nnn(C)c2s1 C1(F)(CNC(c2c(C)cccc2)=O)CCCN(C(=O)CCc2nncn2C)CC1 C1(N(C)C)CCCN(CCC(=O)NCC2(O)CN(C(=O)CC3CCCOC3)C2)C1 c1(CNC(C(Cc2ccoc2)NC(C2C3CC(=O)CC32)=O)=O)ccc(F)c(F)c1 N1(C(C2(C)CCCN(C)C2)=O)CCC2(CC(C(=O)NC(CCO)C(C)(C)C)C2)C1 CC(C)C(CCC(=O)NCCCC(C)(C)O)NC(C1CCCC(=O)C1)=O N#Cc1ccc(C(=O)NN2CCC(NC(=O)C(=O)NCCNC3CC3)C2)cc1 c1(C(N2CCCC(c3nc[nH]n3)C2)C(=O)NCCCC)ccc(OC)cc1 c1(OC)c(C)nc(C2CC2)[nH]c1=NCC1(F)CCN(C(c2ccncn2)=O)CC1 c1(C(C(=O)NCCN(C(=O)CC(C)CN(C)C)CC)(C)O)ccc(F)cc1 C=CCCC(F)(F)C(=O)N1CC(CC(F)C(=O)NCC(C2CC(C)(C)C2)O)C1 C=CCC(C)(C)CC(=O)N1CCN(C(c2c[nH]nc2F)=O)CC(CO)C1 N1(C(c2c(C)cco2)=O)CCCOC(CNC(c2ncccc2C(F)(F)F)=O)C1 C(=O)(CC1=NNC(=O)C1)NC(c1c(OC)cccc1)CNC(=O)Cc1cocn1 C1(C2CCCCC2)(C(=O)NC2C(F)CCN(C(C(n3c(C)ncc3)C)=O)C2)CC1 c1(C(N2C3CC(NC(c4cn(C)nc4C(F)F)=O)(C3)C2)=O)ccc2ccnn2c1 C12(NC(c3[nH]cc(COC)n3)=O)CCCC1CN(C(=O)COCC1CCCC1)C2 C1(CN(C(=O)Cn2cnnc2O)C)CN(C(c2ccc(C3CC3)nn2)=O)CCO1 CC#CCCCC(=O)NCC(=O)NCC(=O)NCCCCO c1(OC)cc(N)c(Cl)cc1C(N1CC(NC(=O)C(C)(C)CF)CC1C)=O Cn1cc(C(=O)NC2CCC(NC(c3occc3Br)=O)C2)c(-c2ccco2)n1 C1(CCC)CN(C(c2c(C)nn(C)c2F)=O)CCN1C(=O)COCC(C)C Cc1cccc2c(C(N3CC4(CC4)CC3CNC(C3CC3Br)=O)=O)coc12 C(=O)(C(C)C(F)(F)F)NCC1(COC)CCCN1C(=O)CCC=CBr N1(C(C(CC2CCC2)OC)=O)CCC2CN(C(C3CCCSC3)=O)CC12 c1(OC)nccc(CNC(C2(NC(=O)CCC3CC3(F)F)CCC2)=O)n1 N1(C(c2cnc(CCOCC)s2)=O)CCN(C(C2CCOC2C)=O)CC2(CC2)C1 C1(NC(C(C)NC(=O)Cc2cccnc2F)=O)CC2(CCC2)C1O Cc1nc(NC2CN3CCC2C3)cc(NC2CC(F)C2)n1 c1(CC(C)C)ncc(C(=O)N(CCN(C(=O)COCCCF)C)C(C)C)[nH]1 C1(C)(COC)CC(NC(c2[nH]cnc2C#N)=O)CN1C(=O)CCOCC(C)C N1(CCNC(C2(CC)CCC2)=O)C2CCC1CN(C(=O)C(C)(C)CC(C)C)C2 C(=O)(CC(C)(C)C(F)(F)F)N1CC(C)C(NC(C2CCCS(=O)(=O)C2)=O)CC1 N1(C(c2ccc(C(C)C)nc2)=O)CC2CCC1C(NC(=O)C(C)C(C)C)C2 C(CCN=c1nc(O)c2ccccc2[nH]1)N1CCc2c(CO)ccc(F)c2C1 C#Cc1ccc(C(N2CC(NC(c3coc(CO)c3)=O)CC3(CC3)C2)=O)cc1F c1(C(=O)NC2CC(CCNC(C(C3CCC(=O)N3)C)=O)C2)c[nH]nc1F C1(C(=O)NC(C2CCN(C(=O)COCC(F)(F)F)C2)C)CCC(=O)N1C1CC1 C1(C2CC2)(C(N2CC(N3CCCC3=O)C2)=O)CN(C(C2C3CCCOC23)=O)C1 c1(C(N(C(C)CNC(C2CC2(F)F)=O)CC)=O)cc2cccc(OC)c2[nH]1 CCCCCC(O)C(=O)NC(CC(N)=O)C(=O)NC(C)CC(C)(C)CO CC1CC(NC(=O)C(F)(F)c2ccccn2)CCO1 C=C1CC(C(=O)NC(c2ccccc2)COC)N(CS(=O)(=O)CC2CC2)C1 S(=O)(=O)(C1CCCCC1)N1CCC(NC(c2cccs2)=O)CC1 c1(CC(=O)N(CC(C)NC(c2cc(C)oc2C)=O)C)ccc(O)c(C)c1 C12(C(N3CCC(COC)C3)=O)CC(CO)(CN1C(=O)C(C)c1cc[nH]n1)C2 c1(OCC)cncc(=NC(=O)C(=O)N2CC3CC(OC)C(C3)C2)[nH]1 CCC(CC)C(C(=O)NC1CCC(NC(c2cnoc2CC(C)C)=O)C1)OC c1(CC)cncc(C(=O)NC2CC(C)N(C(=O)C3=CCCC3)C2)c1 N1(C(=O)C2=CSCS2)CCC2C(CCCN2C(c2cccc(C3CC3)c2)=O)C1 N1(C(CC)=O)CCN(C(C2CCC23CCC3)=O)CC1c1cccc(Cl)c1 C1(C(N2CC3C(NC(c4c(CC)ncnc4)=O)C3C2)=O)CCC2CC(C)CN2C1 C(C(O)C(=O)NCC1CN(C(c2ccc(C)o2)=O)C1)SC Cc1c(C(=O)Nc2cnn(C(F)F)c2)cccc1C1CC1 c1(C(=O)NCC2CC(C(=O)NC(c3ncc(C)o3)C)C2)ncccc1F c1(CCC(=O)NCC(c2ccccc2)NC(COC(C)=O)=O)ccc(F)cc1Cl CCS(=O)(=O)CC(=O)N1C2CCC1C(CNC(=O)Cc1ccnn1C)C2 C1(C(N2CC(CNC(C3C(CC)C3)=O)(COC)C2)=O)CC(O)CN1C(C)=O N1(C(CC(C)O)=O)CC2CC1CN2C(c1ccc(Br)cc1O)=O c1(C(=O)NC2C3N(C(C4(C)COC4)=O)C(CC3)C2)cc2c(nn1)CCCC2 N1(C(c2c(C)nsc2N)=O)C2CCC1CN(C(=O)CC(C)c1ccncc1)CC2 c1(C(=O)Nc2c(C)ccc(-c3ncco3)c2)cc(C)nc2[nH]cnc12 Cc1ccc(F)c(N)c1C(N1CC2C(NC(=O)Cc3cnc(C4CC4)[nH]3)C2C1)=O N1(C(C)=O)CCC(C(=O)NC(C2C(NC34CC(CO)(C3)C4)C2)C)C1 c1(C(=O)NC2(CNC(CC3CC(OCC)C3)=O)CCOCC2)ccc(C#N)cc1 N1(C(Cc2c(C#C)cccc2)=O)CCC2CCN(C(=O)CC(CC)OC)CC2C1 C1(CNC(Cc2nnc(C)o2)=O)CN(C(C2CCCC(=O)N2)=O)C2(CCC2)C1 c1(CNC(COCC#C)=O)nc(CNC(c2c[nH]c(=O)cn2)=O)cc(O)n1 CC(CC(N)=O)C(=O)NC1CC(OCC(N2CCS(=O)(=O)CC2)=O)C1 CC(C)(C)C#CC(=O)N(CC(CC1CC1)C(=O)N1CCC1)CC(N)=O Cc1nc(C(N2CCN(C(=O)Cc3ccsc3C)C(CF)C2)=O)ccc1[N+](=O)[O-] C1(NC(C(=O)N(C)C)=O)CS(=O)(=O)C2CN(C(C3Cc4ccccc4CO3)=O)CC12 C1(N(C(C2(CC)CC2)=O)C(c2cn(C)cc2C)=O)CN(CC2CCC2)CC12CC2 N1(C(c2cnnc(Cl)c2)=O)CCC2(CCCN(C(C3CCCC3)=O)C2)C1 N1(C(C2CCCN(C(CS(CC)=O)=O)C2)=O)CCC2CCN(C)CC12 C1(C)(C(N(CC(C)C)CC#C)=O)CN(C(C2C3CCC(F)C23)=O)C(C)(C)C1 C1(C(CNC(C2(CC)CC2)=O)Nc2ccccc2)C(C)(C)C1(C)C.C(=O)CCSC C12(C(N3C(C(=O)OC)C4CC4C3)=O)CC(CN(C(c3cc(F)ccc3F)=O)C1)C2 N1(C(c2cn(CC)nn2)=O)CCC(C)(C)C(NC(=O)CC(C)C2CCCCC2)C1 Nc1ccc(CCCNC(=O)NCc2cc(Cl)ccn2)nc1 N1(C(c2c(OC)nc(C)s2)=O)CC2CCCC(C1)N2C(=O)C(C)CN(C)C c1(CNC(=O)NC(c2cccs2)CC)cc2occc2s1 c1(C(=O)NCC(CC(=O)NCC(CC)(C)CO)C)coc2ccccc12 CC(C(=O)N1CC2CC(NC(C34CC(C)(C3)OC4C)=O)CC1C2)C(C)C(C)(C)C Cc1noc(C)c1CCC(=O)NC(C)(CNC(=O)C(O)Cc1cccs1)CO C(=O)(C(CC(C)C)NC(c1ccc(O)nc1)=O)N1CCC(COC(C)=O)C1 N1(CC)C(=O)CCC1CC(N1CC(F)(CNC(C2(CCOC)CC2)=O)C1)=O N1(C(C(C)(C)SC)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1CC(C)(C)C1 S(=O)(=O)(c1cccc(=NCc2ccc3c(c2)COC3)[nH]1)NC(C)CCC1CC1 c1(C(NC(=NC)NCc2cc(C(F)(F)F)co2)C)cccc(C)n1 C1(CC(=O)N(C2CCN(C)C2=O)C)CC2CCC1(NC(=O)CSC(F)F)C2 N1(C(Cc2cnc(C)o2)=O)CCC(NC(c2cnn(C(F)(F)F)c2)=O)C(O)C1 CC1CC(=O)NCCN1C(C(=O)NC(C)(C)C)c1ccoc1 CC1CCC(N2CCCC2)CN1C(=O)NC(=O)NCC(c1ccc(O)cc1)O c1(C(C(=O)NCc2ccc(-n3cc(C(C)O)nn3)cc2)O)ccc(C#N)cc1 c1(C(N2CC(NC(C3CC3F)=O)(CO)C2)=O)c(F)ccc(F)c1Br N1(C(c2c(CC)nccn2)=O)CC(NC(=O)C(SC)SC)C(C2CC2)C1 c1(N(C)Cc2ccc(SC)cc2)ccc(S(=O)(=O)N2CCOCC3CC23)cc1Cl c1(-n2cc(C3CN(C(C(C(C)(C)OC(F)F)=O)=O)CC3O)nn2)ccc(Cl)cc1F.OC C=CC1(C(=O)NC(C2CN(C(=O)C(C)C(C)O)C2)C)CCOCC1 CC1CCN(C(=O)CC(C)C(C)(C)C)CCN1C(=O)Cc1cccs1 CC(C)C(C)(CNC(=O)C(=O)N(C)C)NC(=O)C(c1cccc(Br)n1)C C1(CC(=O)NC(CC)(CNC(C2(C)CC3CC3C2)=O)CC)COC(C)(C)CO1 C1(C)(CNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)C(CO)c2ccccc2)CC1 N1(C(C)=O)CCc2c(C(=O)Nc3cn[nH]c3)n[nH]c2C1 c1(C(C(N2CCC(N(C(=O)CC3CCOC3=O)C)C2)=O)(F)F)ncc(Cl)n1C CN1C(=O)CSC1=CC(=O)NCC1CCN(C(=O)COC2CC2(F)F)CC1 CCC1=NOC(CC(=O)NCC(c2ccccc2)CNC(c2cnns2)=O)C1 c1(OC)ccc(CCCCC(=O)N(CCCCN(C)C(c2csnn2)=O)C)cc1 C12(NC(C(F)=C(C)C)=O)CCCN(C(c3cc(F)c(F)cc3F)=O)CC1C2 c1(C(=O)NCC(c2cccc(C)c2)NC(CCCOC)=O)scc(C)c1C C1(C(=O)NC(C)CNC(c2c(Br)cnn2C)=O)CC12CCC(C)(C)CC2 C(=O)(C1CCCc2sccc21)NCC1CC(C(=O)OC(C)(C)C)C1 Cc1ccn(C)c1C(N1C(C(=O)NCCc2ncnn2C)CC1C)=O C1(OC)CC(NC(=O)C=Cc2cccc(F)c2)CN(C(=O)C(C)(F)C(=O)OC)C1 Cc1nc2cc(C(=O)NCC3CCCCN(C(C4CC4C#N)=O)C3)ccc2s1 c1(CC)ccc(OCCC(=O)NC(C)(C)CNC(=O)Cc2csc(C)n2)cc1 c1(C(=O)NCC(CC=C)NC(C2(F)CCCOC2)=O)c[nH]c2c(C#N)cccc12 C1(OCCC)CCC(CC(=O)NC(CNC(=O)C(C)(CO)OC)CO)CC1 CC1(C)NC(=O)OC12CCN(C(c1nnc(C3CCCC3)s1)=O)C2 CN1CCN(C(=O)C(c2ccccc2F)O)CC1CNC(c1cccnc1Cl)=O N1(C(C2(NC(=O)CCc3cncs3)C(C)(C)C2)=O)CC2(C1)CC2(F)F C1(C(N(CC(C)(C)CNC(=O)CC(=O)NCC(F)(F)F)CC)=O)CCC2(CC2)C1 CS(=O)(=O)C(C(=O)N1CCN(C(c2cc3n(n2)CCO3)=O)C(C2CC2)C1)C1CC1 c1(OC)ccc(CC(=O)NCC(C)N(C(=O)C(c2cccnc2)C)C)cc1F C1(CNC(CCN(C(C(CSC)OC)=O)C(C)C)=O)CCN(C)CC1 N1(C(=O)COc2cccnc2)CC2CN(C(c3coc(Cl)n3)=O)CC(C1)O2 c1(OCC)noc(C)c1C(=O)NCC1(CNC(c2cc(COC)on2)=O)CC1 c1(OCC)ncccc1-c1cccc(CC(=O)NCc2ccnn2C)n1 c12ccncc1S2.C(=O)(C(Cc1ccccc1)NC(=O)C1CC1)NCC(C)OC c1(NCC(CC)CC)ccc(S(=O)(=O)NC2CC(O)C2(C)C)c(Cl)c1 N1(C(CCNC(N)=O)=O)CC(NC(c2ccc(Br)o2)=O)CC2(CC2)C1 C1(N(CCCC)C(C2CC=CC2)=O)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 C(=O)(C(C)C(C)(F)F)N(C)CC1N(C(C(CC=C)NC(C)=O)=O)CCCC1 C#CC1(C(=O)NCc2n[nH]c(C)c2C)CN(C(=O)CC2OCCC2C)C1 C(C(C)CC(=O)N(C)CCc1cccs1)NC(c1cc(C)oc1)=O C1(O)(c2cn(CC)nn2)CCS(=O)(=O)CC1.C1(C)C(C(=O)OC)C(=O)C12CC2 C1(C(=O)NCCC2CCN(C)C2=O)CC(O)CCN1C(C1CC(N=[N+]=[N-])C1)=O c1(CCC)sc(C(=O)NCCCN(C(=O)C=CS(C)=O)C)cc1Br Cc1ccc(C(N2CCCC2)=O)c(CSCc2cn(C)nc2C)n1 c1(NC(C(N2C(CC(=O)OC)CC2C)=O)=O)ccc(O)cc1Br C(=O)(CCCC(N)=O)N1CCC(C(C)NC(c2c(C)nc(Br)o2)=O)C1 c1(OC(CC)C)ccccc1C(=O)NC1CN(C(c2cccn2CC)=O)CC1C C=CC(C)(O)C(=O)NC1CC(C(=O)NCCc2cncc(C)n2)C1 C(=O)(C(C#N)(CC)OCCCOCCOC)c1cn(SC)nn1.CCCC.C1CS1 C12(C(=O)NC(CCOCC)C(=O)N3CCOC(C(C)C)C3)CCCC1C2(F)F C(C)(CCCCNC(=O)C(C(C)C)C1CCC1)NC(Cc1c(C)con1)=O C1(C(N2CC(OC)(CNC(=O)CC(C)(C)OC)C2)=O)CC2CCC1O2 C1(C(=O)NCC(C2CC2)NC(COC(CC)C)=O)CCc2cncn2C1 c1(C(=O)NCCCCNC(c2n(CC)c(O)nc2)=O)cnc2c(c1)nnn2C C1(CCOC)CN(C(=O)COc2ccc(C)s2)CCN1C(=O)C(CCOC)OC N1(C(C2OCCN(CC)C2)=O)CCOCC(C(=O)NC(C)(CC)CC)C1 c1(CCCC(=O)NC(CN(C(CCN(C(C)=O)C)=O)C)C)csc2ccccc12 N1(C(C2C(C)C2)=O)CCCC(CNC(c2ccc(F)c(Cl)c2)=O)C1c1ccccc1 Cc1cc(Cl)ncc1CNC(C1CCC(OC2CCC2)CC1)=O CC(C)CC(=O)C(=O)NC(c1nocc1C(=O)NCCc1cnco1)C C1(C(=O)NC(C2CCCC2)CO)COC2(C1)CN(C(=O)Cc1cnns1)C2 N1(C(C2CCC(CC)O2)=O)CC=CC(NC(=O)Cc2nnc(O)s2)C1 c1(OC)cc(C=CC(=O)N(C2CCCCN(C(=O)C(F)C(C)C)C2)C)ccc1F C(=O)(CCS(C)(=O)=O)NCC#CC(=O)NCC(c1ccsc1)C CC1CN(C(C2CN(C)CCN2C(=O)CCc2ccn(C)c2)=O)Cc2nncn21 CC(C)CC(O)C(=O)NCC1CCCN1C(c1nncs1)=O N1(C(CCSCCCC)=O)CCN(C(=O)C2=CCOCC2)CC12CC2 Cc1ccc(O)c(C(N2CC(C3CN(C(C4OCCC4(C)C)=O)CCO3)C2)=O)c1 c1(C(N2C(C(C)C)C(NC(C3(C)CC(C)(C)C3)=O)CC2)=O)cccc(C#N)c1 C1(NC(C2(C(=O)NC)CC2)=O)CCC2CCN(C(c3[nH]ccc3C(F)(F)F)=O)C12 N1(C(C=C(CC)CC)=O)CCCC1C(C)(C)NC(c1ccc(COC)s1)=O C(CS(=O)(=O)CC(=O)NC1CCN(C(c2cc(OC(F)F)n(C)n2)=O)CC1)OC Cc1nnc2n[nH]c(NC(c3cc(N)ccc3[N+](=O)[O-])=O)c2c1C c1(C(=O)NC2CCN(C(c3ncc(C)cc3C)=O)C2)c(F)ccc2ccoc12 C1(C(=O)NCCNC(C2CCCC2)=O)CC2(CCN(C(=O)C=CC(F)F)C2)C1 C1(CC=C)COCC1NC(=O)C(C)(C)C1CCN(C(c2cc(C3CC3)on2)=O)C1 Cc1cc(-n2cncn2)ccc1C(=O)NC(C)CCCNC(C1CCCOC1)=O CC(C)C(C(=O)NCCC(F)(F)Cl)C(C)NC(=O)C(C)N=[N+]=[N-] C1(CNC(CC#N)=O)CN(C(c2cc(C(F)F)ccn2)=O)CC12CCOCC2 C1(CC(=O)NC2C(NC(C3(COCC)CC3)=O)C2)OC(C)(C)OC1=O C#CC1(O)CCCN(C(C2CC(C)N2C(=O)COc2ccn(C)n2)=O)C1 C1(NC(C2COCCN(C(C(C(C)C)(C)O)=O)C2)=O)CCOC2(CCC2)C1 c1(CO)nc(Nc2cccc(F)c2C)cc(=NCC2CC23CCOC3)[nH]1.C1CO1 C1(CNC(CCn2ncc(C)c2)=O)CN(C(=O)CCC2CCCO2)CCCO1 Cc1c(C(=O)NC2(CO)CCN(C(C3CS(=O)(=O)C3)=O)C2)cnn1CC(F)F CS(=O)(=O)c1ccc(C(N)=O)cc1F.C1(=O)CC(c2cccs2)C(=O)N1C Cc1nc(C(=O)N(C2CCN(C(C3CCC34CCC4)=O)CC2)CC2CC2)c(C)s1 N1(C(CCNS(C)(=O)=O)=O)CC(CO)C2(C1)CN(C(=O)CC1CCCCCC1)C2 c1(OC)cc(N)c(F)cc1C(N1CCCC1CNC(C1CCC2CC2CC1)=O)=O O=C(NNc1cccc(Br)c1F)C1CCCS(=O)(=O)C1 C(c1ccc(Cl)c(C(F)(F)F)c1)=CC(=O)NCCN(C)C(C1C(F)(F)C12CC2)=O C1(C(=O)NCCC(C)N(C(=O)CCNC(N)=O)C)CCC(=O)C1 C=CCC(C)(CC=C)NC(=O)C(C(C)O)NC(=O)CCN1CCCC1=O C1(C(=O)NC2C3CN(C(C(C)NC(N)=O)=O)CC2C3)CC2CC(O)CC(C1)C2 c1(C(=O)NCC23CC(c4ccccc4)(C2)C3)c[nH]c2ccc(Br)cc12 C1(C(=O)NCCCN(C(c2c(NC)snc2C)=O)C)CCOC2(CCCCC2)C1 C1(NC(C(C)N(CC)CC)=O)CC2CC(C1)CN(C(=O)CCC1CCCCO1)C2 N1(C(C(C2CC2)OCC)=O)CC(NC(=O)CC=C(C)C)C(c2cnn(C)c2)C1 N1(C(CC(C)n2ccnc2)=O)CCOCC1C=NO.c1(C(CO)N)ccccc1 CC(C)CS(=O)(=O)CC(=O)NCCCN(CCO)C(C1CN2CCN1C(C)C2)=O c1(OC)cc(C(=O)Nc2cccc(F)c2)c(-c2cccc(F)c2)cn1.C(C#N)SC C1(C(=O)NCC(C(C)O)C)CCOCCN1C(=O)CC(C)(C)O N1(C(c2cc3ncccc3s2)C(=O)NC(C)(C)C)Cc2ccc(Cl)cc2C1 CCCCCCCCCC(O)C(=O)NC(C)C(C1CCOCC1)O CC1OCCOC1C(=O)NCC1(CO)CCN(C(C2C=CCC2)=O)C1 c1(CNC(C2CC(F)(F)CN2C(=O)Cc2ccsc2)=O)c(Br)cncc1Br CCC(C)CCC(=O)NCCNC(=O)C(C)Sc1ccccc1Cl C(=O)(CCCCN(C)C(C1CCCC1)=O)N(C(C=C)C1CC1)C C12(C(N3CCC(O)(CC)C3)=O)CC(CN(C(c3cn(CCO)nn3)=O)C1)C2 N1(C(c2ccn(CC)n2)=O)CCOCC1CC(=O)NCC(C)(O)C1CCCC1 C1(C(N2CC(COC)C2)=O)CCC(NC(=O)CSc2nc[nH]n2)CC1 CC(CCN=c1ccnc(NCc2nnc(-c3ccccc3Cl)s2)[nH]1)C(F)(F)F C1(CNC(C2N(C(=O)NC)CCC2)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC1(F)F C(=O)(CCCCCF)NCC1(CN(C(c2ccc(OCC)nc2)=O)C)CC1 c1(CC)ccc(C(N2CCOC(CN(C)C(C3(C)CC3(C)C)=O)C2)=O)c(C)n1 N1(C(C(CSC)C)=O)Cc2nccn2CC(NC(C23CC(CC(F)F)(C2)C3)=O)C1 N1(C(C(SC)SC)=O)C2CCCC1CN(C(c1cc(C#N)c[nH]1)=O)C2 C(C(CC(C)C)NC(C1CCCN1CC)=O)NC(C=CCC)=O N1(C(CC(C)(C)C)=O)CC2(CNC(c3ccc(Cl)cc3)=O)CC1CO2 C(C(C)(C)C(=O)NCC(C(C)C)NC(=O)C(C)CN1CCOCC1)NC(C)=O c1(CC(=O)NCCC(C)NC(c2c(SC)cnn2C)=O)ccc2sccc2c1 C1(C)(CNC(C(C)(C)OCCC)=O)CCN(C(C2CC2C2CC2)=O)C1 c1(C(=O)NC2C(NC(c3cccnc3O)=O)CCCC2)cc2c(nn1)OCCS2 c1(C(N2C(C)C(NC(=O)C(C)(C)O)CCC2)=O)cc2cc(O)ccc2cc1O N1(C(c2n(CC)nnc2C)=O)CC2CCC1CN2C(=O)CC1CCCCN1C C(=O)(CC1=CCN(C)CC1)NCC1CCN(C(C(Br)=C(C)C)=O)C1 N1(C(c2cnc(C)s2)=O)CCC(NC(C2(F)CCS(=O)(=O)C2)=O)CC1C c1(C(=O)NC2(CNC(C(COC)(C)OC)=O)CC2)cccc2[nH]c(C)cc12 c1(C(=O)OC)cccn(CC(=O)NCC(F)CNC(=O)CC2CCC2)c1=O c1(CN(c2ccn(S(=O)(=O)F)n2)CC(=O)OCC)cc2nn[nH]c2cc1F N(C1CCCc2c1cnn2CC1CCC(N)C1)C(C(=O)N(C)C)=O Cn1[nH]c(=NC(=O)C2CC(F)CN(Cc3cc(Cl)cnc3Cl)C2)cc1Cl CCCC(C)C(C)(c1nnnn1CC)Nc1ncc(OCC)cc1Br c1(NC(C(C)(C)Br)=O)cnc(F)cc1CNC(c1cc2sccc2[nH]1)=O C(=O)(C1CCc2ccccc21)N1CC(NC(CCc2c(C)noc2Cl)=O)(CO)C1 c1(C(N2CC(NC(CCC(C)SC)=O)C(SC)C2)=O)cc2ccc(F)cc2o1 N1(C(C(C(C)C)n2ccnc2)=O)CC(C(N2CC(O)CC2(C)C)=O)CC(F)(F)C1 c1(C(N2CC(CN(C(C=CC(CC)C)=O)C)OCC2)=O)cn2cccc(F)c2n1 N1(C(C(CC)CC)=O)CCN(N2CCC(Cc3ccc(C=O)cc3)C2)C2CC12 c1(C(=O)NC2C(CNC(C3C(=C)CC3)=O)CCCC2)[nH]c2ccccc2c1C#N Cc1ccc(N)c(C(=O)NCC23CC(NC(=O)CCC4CCC4)(C2)C(C)O3)c1F c1(C(N2CCC(OC)(CNC(=O)C=C3CCOCC3)C2)=O)cnc2ncccn12 CN1CCN(C(=O)CN2CCCC2=O)CC1C(=O)Nc1ccc(C2CC2)cc1 C(C(CC(=O)NC1(CO)CC=CC1)NC(c1nonc1N)=O)OC C1(NC(CC2CN(C)CC2O)=O)CCCCCN(C(=O)Cc2cncc(F)c2)C1 C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1CCC(NC(c2c(CC)nc(C)[nH]2)=O)C1 c1(NC(N2C(CCC(C)C)CCCC2)=O)ccc(F)c(S(N)(=O)=O)c1 N1(C(c2scc(OC)c2)=O)CCOC(C(C)NC(=O)CC2CC3CCC2C3)C1 CC(CC(C)(C)C)C(=O)N(CCCNC(=O)Cc1ncn2c1CCCC2)C C1(S(N)(=O)=O)(C(=O)NC(CNC(c2cc(C)n(C)c2)=O)C)CCCC1 c1(C(=O)NCC(CNC(COCC#C)=O)F)cc(CCOCCOC)no1 c1(OC)cccc(CC(=O)NCC2(F)CC(NC(=O)C=C(C)C)C2)c1Cl C1(NC(=O)Cn2cnc(Br)n2)CCN(C(=O)CCn2cncn2)CC1O c1(C(=O)NC2C(C)CCN(C(=O)C(C)(Cl)Cl)C2)cc2n(n1)CCNC2=O c1(CC(N2CC(C)C(NC(C3CC3C(F)F)=O)C2)=O)cccc(C#N)c1 c1(NCCCSCCCN(CC(C)O)C)cc(Br)no1 N1(C(C(C)O)=O)CC(C2CCCCN(C(c3cc(C4CC4)sn3)=O)C2)C1 N1(Cc2c(C)cccc2Cl)CCC(NC(c2ccc3nc[nH]c3c2)=O)C(C)(C)C1 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)N(CC(C1CCCC1)O)C N1(CCNC(C(c2cnn(C)c2)NC(c2c(C)non2)=O)=O)CCOCC1=O C=CCCC(c1nnnn1C(C)C(=O)OC)(C1CC1)NCc1ccccc1Cl Cc1nc(N2CCC(NC(C3CCCC(C)C3)=O)C2)ncc1Br CC1(CNC(c2ccc(C3CC3)cc2)c2nnnn2CC2CC2)CC2CCC1O2 C1(NC(C2C(OCC)C2)=O)CCCCC1CNC(c1cc(C(C)(C)C)nn1C)=O c1(NCCC2N(C(c3cnccn3)=O)CCCC2)nc(Cl)nc2[nH]c(O)nc12 c1(C(N(C(C)C)CCNC(c2sccc2C(F)F)=O)=O)cccc2c1COCC2 CC(CC(=O)N1CCOC2(CCC2)C1)C(C)(C)NC(=O)CC1CNC(=O)O1 C1(NC(c2cncnc2)=O)CN(C(=O)CC2CCC23CCC3)C2CCCCC12 Cc1cc(C)n2nc(C(=O)NCc3cn(Cc4nc(C(=O)O)cs4)nn3)cc2n1 N(C1CN(C(=O)CC(C)(C)O)Cc2ccccc21)C(CCCCCOC)=O C1(C(=O)OC)CN(C(=O)NCCCC2CC2(C)C)c2ccccc2O1 c1(C(N2CCC(NC(c3cncc(Cl)c3)=O)(CF)C2)=O)cnc2ccccc2n1 C1(CC(=O)NOC2CCOC2)CCCC12CC2.c12cn(nn1)C2 CC(Cn1cccn1)CN=c1nc(N(C)Cc2nc(=N)[nH][nH]2)c2cc[nH]c2[nH]1 N1(C(C(CC=C)(C)C)=O)CCC2CN(C(=O)Cc3nn(C)cc3[N+](=O)[O-])CC2C1 N1(C(C2CC(=O)NC(=O)N2)=O)CC2CN(C(C3CC4OC3C3CC43)=O)CC2C1 Cn1cc([N+](=O)[O-])cc1C(N1CCCC1C1(O)CN(C(C2C=CCCC2)=O)C1)=O N1(C(C(CC(C)C)OC)=O)CCC(C(=O)N(C)OCC(F)(F)F)C(C)(C)C1 Cc1ccc(C(=O)NC23CC2CN(C(=O)CN2CCC(C)CC2)C3)c(I)c1 CCCCC(CNC(c1coc(C(N)=O)c1)=O)NC(=O)Cc1cnc(C)s1 c1(C(=O)NCC(C)N(C(CCCN(C(C)=O)C)=O)C)cc(C)cc(O)c1 C1(CNC(C(C2CC2)OC)=O)CCN(C(=O)CCOCC2CCC2)C1 Cc1cncc(C(N2CCOC(CCNC(=O)Cc3ccc(C)s3)C2)=O)n1 c1(C(=O)NCC2(CF)CCC2)cncc(-n2cccn2)n1 c1(N2CCCN(C(c3cccc(F)c3I)C=O)CC2)nccn2cnnc12 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(C2(CO)CCC2)=O)CCC(C)(C)C1 c1(C(N2C3C(NC(c4nc(C)oc4)=O)CC(C3)C2)=O)c(F)ccc(Br)c1F CC(C)(O)CC(=O)NCC1CN(Cc2ccnc(N(C)C)c2)C1 N1(C(c2cc(C)sn2)=O)C2CCC1CC(C(N1CCC3(CCCO3)C1)=O)C2 C1(C(=O)NC2CC(CCNC(C3(c4cncs4)CC3)=O)C2)CCCOCC1 N1(C(C=C2CCN(C)C2)=O)CC(O)CC1CNC(=O)C(C)(C)c1ccnn1C C#CCC(C)(C(=O)N1CCC(O)C(CO)C1)NC(C1C=CCC1)=O C=CC1CN(C(=O)Cc2ccccc2COC)CC1NC(c1csc(C)c1)=O c1(-n2cc(CCCC(=O)NC(CC(CC)C)C(=O)O)nn2)c(F)c(F)cc(F)c1F c1(C(N2CCCCC2CO)=O)cc(Br)c(F)cc1Cl.N12CCC1C2=O c1(C(N2CC(F)CC(C(=O)NCC3(O)CCC3)C2)=O)ccc2c(Cl)ccnc2c1 N1(C(Cc2nc(C)sc2Cl)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 c1(NC2CCN(C(c3c(C)coc3C)=O)C2)ncc2c(Cl)cccc2n1 C(CC(C(=O)NCCc1nc(C)cs1)NC(=O)C(C)OCCOC)=CC c1(CCC(=O)NC(C)C(C)NC(=O)CC#N)cnn(-c2ccccc2)c1 c1(CN2CC3(C(C(N4CC(=O)NC4)=O)C3)C2)cc(Cl)cnc1Cl n1(CC(=O)NC(CC)CN(C)C(C2CC(F)(CO)C2)=O)nc(C)c([N+](=O)[O-])c1C C1(C(=O)NCc2ccc(C(=O)OC)[nH]2)CC12CCN(C(c1ccc(Cl)cc1Br)=O)C2 C(c1cnc(C)nc1O)=CC(=O)NC1CC(CNC(c2oc(CC)c(C)c2)=O)C1 c1(C(N2CC(CC(=O)OCC)C3(C2)CC3)=O)ccnc2ccccc12 c1(NC(=O)NCC(C)COc2ccc(Cl)cc2)nnc2ccc(C(F)(F)F)cn12 CCC(C#N)C(=O)NC1(C(=O)NC2C=C(C)CCC2)CCOCC1 N1(C(CC(=O)NCC#C)=O)CCN(C(=O)CCn2cc(C)cn2)CC1C#C c1(C(N2CCC(NC(c3cc(OC)ncc3)=O)(CF)C2)=O)ccc(C#N)nc1O c1(C(=O)NC2CCOCC2NC(C2CSCCS2)=O)ccc2nn[nH]c2c1 CC1CN(C(C2(CCF)CCC2)=O)CCC1NC(C1CN(S(=O)(=O)C(F)F)C1)=O Cn1c(-c2nc(C(C)C3CC3)nn2CCCC(F)F)cc2ccsc12 Cc1ncc(C(=O)NCCc2cn(CC3CCC4CC4C3)nn2)c(O)n1 Cc1cc(C(=O)NCC2CCCN2C(C2C=CCCC2)=O)n2ncnc2n1 C1(C(=O)OC(C)(C)C)CC2(C1)C(NC(=O)C1=CC3C=CC(C1)C3)C21CCC1 CCCC(O)C(=O)NCC(CC)NC(=O)CC1(C(F)F)CC1 N1(C(C(C)=C2CC2)=O)CC(CNC(c2ocnc2-c2ccccc2)=O)CCC1C c1(CN(CC(=O)NCC(=O)NC2CC2)CC)ccc(Cl)cc1 N1(C(c2c(C)[nH]c(=NCC)s2)=O)CCC2(CC1)CC(NC(C1CC3(CC3)C1)=O)C2 CC1(C)CCC(C(=O)NC2CCCC2C(=O)NCc2ccc(O)c(F)c2)CC1 N1(C(C2C(=C)C2)=O)CC(O)(C2(CNC(c3ncc(Br)cc3OC)=O)CC2)C1 C1(C)(C(N2CC(C)(NC(C3C(CC)CCC3)=O)C2)=O)CCC(=O)NC1 N1(C(c2c(C)ccnc2)=O)CCC(C)N(C(c2cnc(C3CCC3)o2)=O)CC1 c1(C(=O)NCC(CC)NC(=O)CN2CCCCCC2)cnc2n1CCCCC2 CC(C)C(C#N)C(=O)NC1(C(N2CCCC(CN=[N+]=[N-])C2)=O)CC(F)C1 Cc1cc(Br)c2ncnc(NCc3sccc3C(F)(F)F)c2c1 c1(C(=O)NC2(C)CN(C(C(CC)Sc3ccccc3)=O)C2)nc(C(F)(F)F)sc1C C1(COC)CC(CNC(=O)C(c2ccc(Cl)cc2)=O)N(C(=O)Cc2cn[nH]c2)C1 c1(OC)ccc(C(=O)NC2CCCN(C(C3CC3C(C)C)=O)CC2)cc1O CC1CCN(C(=O)COC2CCC2)C(CNC(C2CCC3(CCC3)C2)=O)C1 Cc1nc(Cl)c(NC(C2CC(F)CN(C(=O)C3CC3)C2)=O)c(Cl)n1 N1(C(C2CC(N(C)C)C2)=O)CCC(C(N2CCC3(CCCO3)C2)=O)CC1(C)C c1(C(N(C2CC(NC(C(C)CC3CC3)=O)C2)C)=O)cc2n(c1)CCOC2 c1(N2C(C(=O)NC(c3ccc4c(c3)OCCO4)C)CC2)ncnc2cccnc12 c1(OC)nscc1NC(=O)CC1(C)CCN1C(=O)C=CCN1CCC1 N1(C(CCOCC)=O)CCC2CCN(C(=O)C(c3ccccc3F)(C)C)CC2C1 C1(CN2CCN(C(c3cc(C)on3)=O)CC2)Cc2ccccc2C1C C1(CC)CN(c2nnc(C(c3ccccn3)(F)F)n2CCC(=O)NC)CC(C)O1 c1(OC(C)C(=O)N(C2CCN(C)C2=O)C)c(Cl)cc(I)cc1Cl C(=O)(C(=O)C(F)(F)F)NC1C(NC(C(C2CCC(=O)N2)C)=O)CCCC1 C1(NC(c2cccc(OC)c2)=O)CCN(C(=O)Cc2ccc(O)cn2)C(C)C1 c1(CC(=O)NC2CC(CN(C(C3C(COC)C3)=O)C3CC3)C2)c(Cl)cnn1C CC1CN(C(=O)CC2CCCN2Cc2ncccc2Br)CC(=O)N1 CC1CN(C(=O)CC(C(F)(F)F)c2ccccc2C(F)(F)F)CCC12CCOC2 C(=O)(CC1CCc2ccccc21)N1C(C)(C)CC(NC(=O)CCCC2CCC2)C1 C#Cc1cnn(CC(=O)NC(CNC(=O)COCCc2cccs2)(CC)CC)c1 C1(C(=O)NCC(CCNC(C2C(=C)C2)=O)O)(OC)CCC(C)(C)CC1 N12CCC(C)(C)C1C(=O)NON1CCC(C1)C(C)C2=O.C(=O)C(C)C1(O)CCC1 C1(C)(C(=O)NC(C)C2CC2)CCCN(Cc2ccnc(-c3ccccn3)c2)C1 c1(N(CC2=CCSC2)C)nc(=N)[nH]c(=NCCc2csc3c(Cl)cccc23)[nH]1 C1(N(C(c2c(-c3cncc(C)c3)nccc2)=O)C)CCCCN(CCO)C1 C(CC)(CCCC(=O)NCC[Si](C)(C)C)NC(C1(CC=C)CCC1)=O CCCCCCC(=O)N1CCC(C(C)C(=O)NCC2(C)CCCO2)CC1 C12(C(=O)NC3CC4C(NC(CCC(=O)N(C)C)=O)C4C3)CCCN(CC1)C2 N1(C(c2nc(CCC)sc2)=O)CCn2c(CNC(C3C=CCC3)=O)nnc2C1 N1(C(CCOCCOC)=O)CCC(O)(CCNC(c2cc(C(N)=O)cn2C)=O)C1 c1(C(=O)NCC23OCC(NC(C(C=C)O)=O)(C2)C3)cc(F)cnc1O C1(C(=O)NCCC(CNC(CSc2cccc(C)c2)=O)O)CN2CCN1C(C)C2 N1(C(CC(C(C)C)NC(c2ccc(CC)s2)=O)=O)CCC2(CCC2)C(O)C1 c1(SCC(N2CC3C(NC(C=CC(=O)OCC)=O)(C3)C2)=O)ccc(C)cc1C Cn1cc2c(C(=O)NC3CCCC3NC(=O)Cc3cnsc3)cc(F)cc2n1 CC1CC(NC(c2ncoc2C(C)(C)C)=O)CN(C(=O)C=C2CCN(C)C2)C1 N1(C(C(C(C)O)N(C)C)=O)CC2(C1)SCCC2NC(c1cc2cnccc2o1)=O N1(C(C(CC)C#N)=O)CC(C2CCCN(C(=O)CNC(c3ccco3)=O)C2)C1 N1(C(C2C(CC)C2)=O)CCC(CF)(NC(=O)C(C)Cc2ccccc2F)C1 CCCCC(C(=O)N(C)CC1CCCN1C(c1ccc(O)c(Cl)n1)=O)NC(N)=O C1(C)(CC(=O)OCc2c(O)nc(C)c(Br)c2)Oc2ccccc2O1 C1(NC(CCOCC(C)C)=O)C=CCCC1C(=O)NC1CC1(C)C(F)F c1(C(N2CCC(C(=O)Nc3ncc(C)nc3Cl)C(O)C2)=O)ccc(I)c(F)c1F c1(CNC(C2(OC)CC(C)C2)=O)ncccc1C(=O)N(C1CCSCC1)C Cc1sc(C)c2sc(C(=O)NC3CN(C(=O)CCCC(N)=O)CC4(CC4)C3)cc12 N1(c2ccnc(NC3C(CCCC)CCC3)n2)CCC2(CC1)CCN(C)C2 C1(C)(CC(=O)N(C(C2CCCCC2)C)C)CCN(C(=O)Cc2ccc(O)cc2)C1 C1(C(N(CC(CC)NC(c2cn(C)c(O)n2)=O)C)=O)CCNC(=O)C1 C(=O)(C1=COCC1)NCC1N(C(C)C)CCC1.C12(CCC1)C(=O)N2C1CC1 N1(C(C2C(OCC)C2)=O)CC2C(N(C(=O)CCc3ccsc3Cl)C)C2C1 N1(C(c2nc(CC)oc2C)=O)CCCC1C1CCCN1C(c1cccnc1C)=O N1(C(CC2CCN(C(C3(C)CNC(=O)N3)=O)C2)=O)CC2CC(O)CC1C2 c1(OC)cc(C(N2CC(O)(c3ccccc3)C2)=O)sn1 C#CC(CC(C)(C)C)NC(=O)C(CCOCCO)NC(=O)Cc1ccccc1C Cc1cc(C(=O)N(CCC(C)NC(C2CCC(=O)N2C(C)C)=O)C)oc1C N1(CC)CCN(N2CCC(S(=O)(=O)CC=O)CC2)CC1.N(C)(CC)CC Cc1nc(O)sc1C(=O)NC1CCCCC1CNC(c1cc(C(N)=O)c[nH]1)=O C(=O)(C(=O)N=S(C)(C)=O)NCCN(C(c1ccc(CN(CC)CC)o1)=O)C1CC1 CCC(C)(CCC(C)C)C(=O)N1CCCCC(NC(C2CN3CCN2CC3)=O)C1 C(=O)(C(O)C1=CCCCC1)NCC(C)(CO)NC(C1CC(CC(F)(F)F)C1)=O S(=O)(=O)(c1cccc(C#N)c1F)Nc1sc2ccc(C)cc2n1 c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC(F)C2)=O)cc2cccnc2[nH]1 Cc1nn(C)c2nc(C(=O)NC3CCC(CNC(c4ccccn4)=O)C3)ccc12 S(=O)(=O)(c1cc(F)c(F)c(F)c1F)C(NNC(c1c[nH]c2ccccc12)=O)=O CC12CCC(C(=O)NCC3CN(C(c4csc(-c5ccncc5)n4)=O)C3)(C1)OC2 CC(C)(CCCNC(C1COCOC1)=O)C(=O)N1CC(CO)C(O)C1 C1(NC(CCOCC)=O)CCCN(C(=O)Cn2cnc(C(F)(F)F)n2)CCC1 C(C)(C(=O)NC1CC(OCC(=O)N(C)CCc2cccs2)C1)OCOC C1(CC(=O)N(C)Cc2nc(C)[nH]n2)CCCCN1C(c1n[nH]cc1Cl)=O c1(OCC)ccc(CNN2CCC(O)(C(C)C)C2)cc1-c1cc(F)ccc1C C1(NC(C2CC23CCC3)=O)CCN(C(=O)CCC2CCOCC2)C(C2CC2)C1 c1(-c2n(C3C(C)OCC3)nc(CCN3CCCCC3)n2)noc2c1CCCC2 c1(OCC)ncccc1C(=O)N(CC(C)CNC(c1cnn(CC(F)F)n1)=O)C c1(-c2cc(C)c(O)cc2)ccc2ccnc(NCc3cn[nH]c3)c2c1 C1(N(C(c2n(CC)cnn2)=O)C)CN(C(=O)C=Cc2cn(C)nn2)CC1(C)C CC1C(NC(=O)CC2OCCOC2(C)C)CCCN1C(c1nn(C)cc1Cl)=O Cn1cncc(C(N2CCC(CO)C(NC(=O)CC3CS(=O)(=O)C3)C2)=O)c1=O C(C(C)(C)C(=O)NC(C)CC(C)NC(C1CN(C2CCC2)C1)=O)NC(C)=O N1(C(=O)NCC2CCCNS2(=O)=O)CCOC2CCN(C(C)(C)C)CC12 c1(OC)cc(O)ncc1C(=O)NC1CCCN(C(C2CCCCC23CC3)=O)C1C C(=O)(C1=CCCCC1)NC(CNC(c1c(C)cnn1C)=O)(C)C1CC1 C1(NC(=O)CCC(F)F)CN(C(=O)C=C2CCCCCC2(F)F)C2CCCCC12 N(C(=NCCCF)N1CC=C(F)C1)CC(C(C)C)CCc1ccccc1 c1(C(=O)NCC2N(C)CCN(C(C3CC4(CC4)C3)=O)C2)[nH]cc2c1CCCC2 N1(C(C2C(C(C)O)C2)=O)CCC(NC(c2cncc(Cl)c2Cl)=O)C2(CCC2)C1 c1(C(C(=O)NC2CCOC2)N(C(CC=C)C)CC)cnc(C)[nH]1 CCCC(C)(O)C(=O)N1CCC(C2CCCN2C(=O)Cn2ccnn2)CC1 c1(C(=O)NC2C=CC(CNC(=O)COCCCF)C2)ccc(O)c(F)c1 N1(C(CCC2(C)CC2)=O)CCC(c2nnc(CNC(=O)CC(C)(F)F)s2)CC1 N1(CC(CC)C)CCC2CCC(C1)N2C(=O)Cc1c(F)cccc1Cl c1(C(=O)NC2CCN(C(c3cccnn3)=O)C2)ccc(C(F)(F)F)nc1O c1(C(N2C(CN(C)C(C3(F)CCOC3)=O)CCC2)=O)ccc2c(c1O)CCCC2 C(C)(C(=O)N1CCC(CC(C)NC(c2ccnc(F)c2O)=O)CC1)(C(C)C)OC c1(C(=O)NCC2CCN(C(C=CCCC)=O)C2)ccc2ccc(Br)cc2n1 C1(NC(CCc2ccc(C(=O)NC(CCC)CCO)[nH]2)=O)CCC(F)(F)CC1 CC(CC(=O)NC1CC(C)N(C(=O)COc2ccn(C)n2)C1)CC(F)(F)F CCCCCCC(C(=O)NCCN(C(c1c[nH]c(=N)s1)=O)CC)NC(C)=O c1(CC)cc(CNC(C2CC(CNC(COC(=O)N)=O)C2)=O)no1.C(C)(C)C Cc1cc(C(=O)NCCOC2CN(C(=O)CCNC3CC3)C2)c(C(F)(F)F)o1 C#CC1(C)CCCN(C(C2C3CN(C(C4(O)CCOCC4)=O)CC23)=O)C1 CCCC(C(=O)NC1CN(C(c2cc(C(F)(F)F)cs2)=O)CCC1C)C(C)C c1(C(N(CC(CCC=C)O)C)=O)cc(C#N)cc(C#N)c1 c1(CC)cccc(NC(c2c(CNC(C34CC(CO)(C3)C4)=O)cncc2)=O)c1F C(CCN=c1nc2scnc2c(N(CC(C)(C)CO)C)[nH]1)N1CC(C)OC(C)C1 Cc1cncc(CNC(C2CC(O)CN2C(=O)C=C2CCOCC2)=O)c1 N1(C(=O)Nc2ccc(SC)s2)CCCC2C1CCN2C(=O)CC1CCN(C)CC1 c1(CC2N(C(C(C)N(CCC)C3CC3)=O)CCC2)cccc2ccccc12 C12(CNC(C(C(C)O)C)=O)CN(C(=O)Cc3ccc4c(c3)OCC4)CC(F)(C1)C2 C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)cccc2)=O)CC2C(C1)C2(F)F C1(NC(C(C)n2cccc2)=O)CCOCC1NC(=O)COCc1cnn(C)c1 C1(C(=O)NCCN(C(CCCOCC)=O)C2CCCC2)Cc2cccnc2C1 N1(C(CNC(=O)OC)=O)CCC(C(C)NC(c2ccnn2C2CCC2)=O)C1 c1(NC(C2(C)CCN(C(c3c(Cl)cccc3Cl)=O)C2)=O)c(O)ncnc1O O=C1CC(C(=O)NCC2(O)CC(NC(=O)CN3CCSCC3)C2)C2(CCC2)C1 CCC(CC)C(C(=O)N1CCCC(NC(c2cnoc2C(C)C)=O)C1)OC c1(C(N2CCC(C(C)NC(C(CC)NC(C)=O)=O)C2)=O)c(Cl)nn(C)c1Cl Cc1ccc(C(=O)NC(c2ccccc2)C(=O)NC2C3COCC23)nn1 c1(N2CCCC(C)(CC)CC2)cc(Br)ccc1S(=O)(=O)NC(CO)C1CCC1 c1(C(N2C(CNC(C(CSC)OC)=O)CC(OC)C2)=O)cn2ccc(F)cc2n1 C1(C(=O)OCC2CCC3C(C2)C3(F)F)C(F)(F)C12CC(C(=O)OC)C2 N1(C(C2CC(O)C(F)C2)=O)CC2CCC(C1)N2C(C1CC(n2ccnn2)C1)=O C1(C(=O)NC2CC(C#C)C2)CCN(C(=O)OC(C)(C)C)C12CCSCC2 c1(CC(N2CCCC(NC(CC3C(C)=NOC3=O)=O)C2)=O)c(O)nc(=N)[nH]c1C N1(C(C2N(CCC)CCC2)=O)CCOC(C(N2CCC(F)CC2)=O)C1 c1(OC)cc(C(F)F)c(C(N2CCCC2CNC(C2CCC(C)CC2)=O)=O)cn1 C1(C(=O)NC2CCN(c3snc(CCOC)n3)CC2O)Cc2ccccc2CO1 CCC(CNC(c1cncc(O)c1)=O)(CC)C(=O)NCC(C)(C)C(C)(C)O C1(CC(N2CCC(CN(C(=O)CC3C=CCC3)C)CC2)=O)CCCCC1(F)F c1(C(N2CCC(c3ccc(OC)cc3)C2)=O)cc(SC)c(Cl)cc1Cl C1(CC)CN(C(=O)CN(c2ccncc2)C)CCN1C(=O)C(C(C)C)OC C1(C(=O)NCC(CN(C(C(CC)F)=O)C)C)CCc2ccccc2O1 c1(NCCNC(=O)NC)nc2ccccc2nc1NC(C1COC(=O)N1)C C1(NC(C23CC(C)C2C3)=O)(CNC(c2cccc(CC#N)c2)=O)CCOCC1 c1(C(N(C2CCC(NC(=O)C(F)=CCCF)C2)C)=O)ccc(P(C)(C)=O)s1 C1(N(C(CCN(C(C(F)=CCC)=O)C)=O)C)CC(C)OC(C)C1 Cc1ccc(Cl)c(OCC(=O)NC2CC(NC(=O)CC3CCC3C3CC3)C2)c1 c1(C(N(C)CC2COCCN2C(=O)CCCC#N)=O)cn2c(n1)CCCC2 N1(C(C(C)CO)=O)CC23CCCCC2(C1)CN(C(=O)C(C1CCCCC1)O)C3 c1(OC)cc(OC)c(C(=O)NCC2CC(F)CN2Cc2ncc[nH]2)cc1Cl c1(C(=O)NCCN(C)C(C23CCC(CC2)CO3)=O)cc([N+](=O)[O-])ccn1 N#Cc1ccc(-c2cnn3cc(C(=O)NCc4ccc(O)nc4)cnc23)cc1F c1(CCC(=O)N(CC(C)NC(C2C3CCC23)=O)CC)ccccc1F N1(C(C2(Cl)C(C)(C)C2)=O)CCC2(C1)CN(C(C1CNC(=O)N1)=O)C2 N1(C(c2cc(OC)cc(F)c2)C(=O)Nc2ccccc2)CCOCC1P(C)(C)=O C1(C(N(c2ccccn2)CCC(N)=O)=O)CCN(C(c2sccc2Cl)=O)CC1 Cn1c(C(=O)NCC2CCOC2C(=O)NC2CC(C(C)(C)C)C2)cnc1Cl c1(C(=O)NC2CC(F)(CNC(c3cnsc3)=O)C2)cncc2[nH]ccc12 c1(C(=O)NC23C(CN(C(c4cccc(CC)c4)=O)C2)C3)cc2ccsc2c(O)n1 C(CC(C(=O)NC1CC(C)C1)NC(=O)CCc1nc(O)n[nH]1)OC N1(C(C2(C)CC(OC)(OC)C2)=O)CC2CCCC2(CNC(=O)CC2CC=CC2)C1 CC1C(=O)NC(=O)CN1C(=O)C(CO)NC(c1ccoc1Br)=O C1(C(N2CC(NC(C(C)N3CCCC3)=O)C(F)C2)=O)CC(C)(C)CN1C c1(C(N2CCN(C(C3CCC(F)(F)C3)=O)CC2)=O)ccc(I)cc1[N+](=O)[O-] C(CC(C)C)(C(=O)NCCCCC1CC1)N(C(C(C(C)C)NC(C)=O)=O)C Cc1cnc2ccccc2c1C(=O)NCC1(O)CC(NC(=O)CNC=O)C1 C1(C(N(CCCOC(C)C)C)=O)CC(C)(C)CN1C(=O)CC1COCCO1 CC1CN(C(c2ccccc2C(N)=O)=O)CCN1C(c1cccnc1N)=O c1(OC(C)C)cccc(SC(c2nnc(C(N)=O)n2C)C)c1 C1(NC(C(=O)Nc2c(C)occ2)=O)(CO)CCCN(C(=O)C(C)CSC(F)(F)F)C1 c1(C(=O)NC(CN(C)C(c2sc(N(C)C)nc2Cl)=O)(C)C)ncccc1C1CC1 c1(CN2CCC(Nc3nc(OC)c(F)cn3)CC2)cccc([N+](=O)[O-])c1 n1(CC(N2CCCC(C)(CNC(C(CCC)O)=O)C2)=O)c(C)nc2ccccc12 c1(CC)cnccc1C(=O)N(CC(C)(C)CNC(=O)C(C)C1CCOC1)C N1(C(CC(=O)OC)=O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)C(C2CCC2)C1 C1(F)(C(N2CC(CC(=O)OC)C2)=O)CN(C(=O)C(C)NC(=O)C2CC2)C1 c1(-c2nc(CN(C(=O)C(=O)NC3(C)CCCC3(F)F)C)sc2)cccc(C#N)c1 Cc1nc(C)n(O)c1C(=O)NCC1(C)CCCC1NC(=O)C=Cc1cnc[nH]1 CC(C)C(C(=O)NCCc1cncs1)C(C)NC(c1ccsn1)=O c1(N(C(C)=O)C(C)C)ncnc2c1nc(NC(c1ccccc1Cl)C(=O)O)n2C N1(C(CCCOCC=C)=O)CCC2(CCC2)C(NC(=O)CC2CCC(=O)C2)C1 C1(CNC(C(C)=C(CC)C)=O)CCCC2CN(C(c3ccsn3)=O)CC12 C=C(Cl)CCC(=O)NCc1cccc(C(=O)NCC2CCC(C)(C)O2)n1 c1(NCC#N)cc[nH]c(=NCCCNC(c2cnn(C3CC3(F)F)c2)=O)n1 C1(CNC(CCC)=O)CCCN(c2ncc(O)cn2)C1 C1(O)(C(=O)NCCC2N(C(C(C)=CC)=O)CCC2)CCCCCC1 C(C(=O)NC(COC)CC(=O)N(C)Cc1ccccn1)(C(C)C)OCC N1(C(C2C(C)(C)C2)=O)CCCC1(C)CNC(c1cc(Br)ccn1)=O C1(NC(COC)=O)CC2(CCN(C(c3ccnc(N(C)C)c3)=O)CC2)C1 C(=O)(C1=CC2(CCOC2)C1)N1CCCC(CCNC(CCCC#N)=O)C1 c1(OC)ccc(Br)c(CS(=O)(=O)NC(C)(CN)C2CC2)c1 C(=O)(CC(C)(C)CNC(C1CC(C)(C)C1)=O)NCC(C)O C1(NC(CN2CCN(C)CC2)=O)CN(C(=O)C(C)(C)n2cnnn2)CC1N=[N+]=[N-] BrC1=Cn2c(-c3noc(COC4CCCCCC4)n3)nc(n2)C=C1 C1(O)(C(=O)NCC2(C)CCCN(C(CC(=O)NCC)=O)C2)CCCC(C)(C)CC1 C1(C(=O)NCC2(F)CN(C(c3n(CC#C)ccc3)=O)C2)CCCCC1(F)F N1(CC(N2CC(F)(CNC(C3C(=O)NCC3)=O)C2)=O)CCCC(N(C)C)C1 C12(C(=O)NC3CC(NC(c4c(NC)nccc4)=O)CC3O)CCCN(CCC1)C2 Cc1cccc(C2(C(CNC(c3ccc(C)n3C)=O)NC(=O)C(C)(Cl)Cl)CCC2)c1 C1(NC(C=C2CCC(C)C2)=O)COC2(CCN(C(c3cc(O)nc(O)n3)=O)CC2)C1 c1(NC(C23C(CN(Cc4ccc(C(=O)OC)cn4)C2)C3)=O)ncc(Cl)cc1F C1(OC)(CNC(=O)Cn2cc(CNC(c3sc(C)cc3Cl)=O)nn2)CCCSC1 C(=O)(CC1CCCc2oc(C)nc21)N(CCN(C(C1CCC1CF)=O)CC)CC CC1=C(C(=O)NC2(CC(=O)NCc3cncc(C#N)c3)CCC2)CCC1 CC(C)C(C)CC(=O)NCC(CC1CC1)C(=O)NC(c1cc[nH]n1)(C)C n1(CC(=O)NC2CC(NC(C=C(CCC)C)=O)C2)c(C2CC2)nc2ccccc12 C(=O)(N1CCCc2nncn21)C1C(NC(c2c(C(N)=O)coc2)=O)CCCC1 c1(C(N2CC3(OCC(NC(CC4(C)CC4)=O)C3)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(Cc2cccc(C)c2F)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 C12(CNC(=O)CCCCCF)CCC(CNC(=O)CC3CC4CC4C3)(CC1)OC2 c1(CC)ccccc1C(N1CCC(N(C(C2CCCS2(=O)=O)=O)CC)CC1)=O C1(NC(C(c2c(C)noc2C)C)=O)CC2CCC1N(C(c1n[nH]c(=N)[nH]1)=O)C2 N1(C(COC)=O)CCOCC1C(=O)NCc1ncsc1-c1ccccn1 c1(C(=O)NCC(CC=C)NC(=O)CC=C(Cl)Cl)cc2cccc([N+](=O)[O-])c2[nH]1 N1(CC2N(C(=O)Cn3cc(CNC4CCCCC4)nn3)CCC2)CCCS1(=O)=O CN1CCCC12CCN(C(C1(CNC(c3cnc(=N)[nH]c3)=O)CCCO1)=O)C2 c1(C(=O)NC(CCOC)CNC(=O)CCn2ccnn2)cc(Br)cnc1O C(=O)(CC(C(F)(F)F)OC)N1CCC(NC(C(CSC)OC)=O)C(C)(C)C1 N1(C(c2cc(OC)n[nH]2)=O)CC2CC(NC(=O)CC(F)(F)C(F)F)C(C2)C1 N1(C(c2cccc(N)n2)=O)CCC2C(C1)CN2C(=O)CCOC1CCOC1 Cc1cc(Br)cc(C(=O)NC2CCN(C(=O)C3=CCS(=O)(=O)C3)C2)c1C c1(C(=O)NCCC2CN(C(C(C(C)C)F)=O)CC2C)nc2c(s1)COCC2 c1(C(N2C3C(NC(C4C(COC)C4)=O)CC(C3)C2)=O)cc(OC(C)=O)cc(F)c1 C1(CNC(C(COC)COC)=O)CN(C(c2cc(C(F)F)cs2)=O)C(C)(C)C1 CCC(C)C(C(=O)N1CC=C(C(=O)N(CC2=CCSC2)C)C1)N(C)C S(=O)(=O)(c1ccc(=NCC2CC2(Cl)Cl)[nH]c1)NCCc1ccc(N(C)C)c(F)c1 N1(C(C2CC(O)(CNC(c3cc(C)sn3)=O)C2)=O)CCC(C2CCC2)CC1 CCCC(C)(O)CC(=O)N1CCN(CC(C)NC(c2cc(CC)ccn2)=O)CC1 C(=O)(CCP(C)(C)=O)NCCCCC1CN(C(C2CC(C)C2)=O)C1 C1(C(=O)NC(c2ccccc2)c2cnco2)CC12CCN(Cc1cnsn1)CC2 c1(C(=O)NC(CC)CNC(c2nn(C)nc2Br)=O)ccc(C#N)nc1O C1(N(C)C(C2COC(=O)N2C)=O)CN(C(C2(CC(F)F)CCC2)=O)CC1(C)C CC1CN2CCN1C(C(=O)NCC(C)CNc1ccc([N+](=O)[O-])cc1)C2 C1(C(=O)NC2C(NC(CCOCC)=O)CCCC2)Cc2cncn2C(=O)N1 C(=O)(CCC(C)(C)C(=O)OC)NC1CCCC(NC(c2c(OC)cncc2)=O)C1 N1(C(CNC(=O)OCC)=O)CCN(CCCN2CCCC2C)CC1 C(CCC(O)C(=O)NCC1(C(=O)NCCCc2nncs2)CC1)OCC C1(CNC(c2nc(C3CC3)cs2)=O)COCCN(C(c2cc(O)cc(Cl)c2)=O)C1 C#Cc1ccc(C(=O)NC(CNC(=O)CC2CCCS2(=O)=O)CC(C)C)cc1F c1(C(=O)NC(C(CO)NC(CC2N(CC)CCC2)=O)C)cc(Cl)cc(Cl)c1 N1(C(C(=O)NC(=O)NCC)C)CCC(NC(c2cnn(CC)c2)=O)C(C)(C)C1 N1(C(CN(S(C)(=O)=O)C)=O)CCOC2(C1)CN(C(C1(C)CC1(F)Cl)=O)C2 c1(CC(=O)NCC(C)N(C(c2cc(C)sc2C)=O)C)cccc(S(C)(=O)=O)c1 N1(C(C(CC)NC(C)=O)=O)C2CCC1C(CNC(=O)C=C1CCSCC1)C2 C1(NC(CSCCOC)=O)CCN(C(=O)CCc2cccc(OC)c2F)C1(C)C c1(C(=O)NC2C(C(C)Nc3cnn(C)c3)C2)ccc(S(C)(=O)=O)c(Br)c1 C(C(C(=O)NC1CCC(NC(=O)C(C)(C)O)C1)NC(C)=O)OC c1(C(N2C3C(NC(C(C)n4cnnn4)=O)C(C3)C2)=O)ccc(O)nc1Cl CCC(C(=O)N1CCSCC1C(N1CCC(C(N)=O)CC1)=O)C(C)C C#CCCCC(=O)N(CCNC(c1ocnc1Br)=O)C1CC1 N1(CC(=O)N(C2CCS(=O)(=O)C2)CC)CCC(C2CC2(F)F)CC1 C(=O)(C(O)P(C)(C)=O)N(CCN(C(C(CC#C)O)=O)C)C c1(CC(=O)NCCN(C(C)C)C(C2CCN(C)C2C)=O)ccc(O)cn1 C1(NC(C(C)C)=O)C2CC1N(C(=O)CC1CC1)C2 C1(CN(C(C(C)CO)=O)C)CC(F)CN1C(c1ccnc(OCC2CC2)c1)=O c1(N(CC)Cc2cc(C)on2)nnc(CC(C)(C)O)n1CCOc1ccccc1 c1(CN2C(C(=O)NCCC3(C)OCCO3)CCCC2)cccc2nonc12 CCCCC(C)CCC(=O)N(C(C)CNC(c1cnc2n1CCCC2)=O)C C(=O)(C(CC(C)C)C(C)C)NC(CC(=O)NCC(CSC)(C)C)C(F)F C1(C(N(C2CCCCN(C(c3ccc(Cl)cc3O)=O)C2)C)=O)Cc2nccn2C1 C1(NC(CC(CC)(F)F)=O)COC2CN(C(=O)C(C(C)C)NC(N)=O)CC12 C(=O)(CC1=CCCCC1)N1CCC(C=C)(C(=O)NCC(F)(F)COC)C1 c1(OC)ccc(CN2CCC(F)(C(=O)Nc3cncc(C(F)(F)F)c3)C2)cc1I C1(CNC(=O)C2CC2)CC2CCC(C1)N2c1ccnc(C(F)F)n1 c1(C(=O)NCCN(CCC)C(C2(C)CC(C3CC3)=NO2)=O)ccnn2ccnc12 O=C1CC(C(=O)NC2CCCCC2C(=O)NC2(c3nccs3)CC2)=NN1 c1(C(=O)NC2C(NC(C3(CC)CC3)=O)CCC2)ccc2c(c1)CCS2(=O)=O N1(C(c2c(OC)cc(OC)c(Cl)c2)=O)C2CCCC1CN(C(C1CC1C)=O)CC2 C=CC1(C(N2CC(N(C)C)C(C)C2)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC1 C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1ccnn1C)NC1CN(CC)C(=O)C1 Cc1csc(C(C)C(=O)NCC2CCCC2NC(c2cnc(C(C)O)s2)=O)n1 c1(-c2nc(-c3c(C)ccnc3)n(C3CCOC3)n2)c2ccccc2nn1C Cc1nc(CNC(c2ncoc2CNC(C2(CO)CCCO2)=O)=O)oc1C N1(CC(N2C(CNC(C(c3cccc(Cl)c3)OC)=O)CC2)=O)CCCCCC1 C1(C(=O)NCCC2N(C(c3c(C)ocn3)=O)CCCC2)CCn2c(C)cnc2C1 C1(NC(=O)Cn2cncn2)CCC12CCN(C(=O)CN1CC=CC1)CC2 Cc1cc(C(N2CCC(NC(=O)N(C)C)CC2)C(=O)NCC2CCOC2)cc(Cl)n1 C1(C2CCOCC2)(C(=O)NCC(CC)NC(=O)C=Cc2ccoc2)CC1(F)F c1(C(=O)NCC(C)(C)CNC(=O)CCNC(=O)CO)ccc([N+](=O)[O-])o1 C=CCC(C(=O)N1CC(C)(C)C1C1CC1)NC(C1CCC(N(C)C)C1)=O C(C1OCCc2sc(I)cc21)SCCNC(c1ccc(C)cc1)=O CCCC(C)(C)CC(=O)NCCC1(O)CCN(C(=O)CC(C)CC(C)C)C1 C1(CNCCC(c2ccnn2C)C)CC2CC1(CO)C2 C(=O)(C1Cc2ccc(Cl)cc21)NC(CNC(c1c(C)c(F)ccc1)=O)C(C)(C)C c12cc(N)ccc1S2.C(CCCOC(=N)O)NC(CC1(C(=O)OC)CC1)=O c1(-n2c(C(n3ccnc3)CC)nc(C(C)C3CC3)n2)cc(F)ccc1F C=CCC(C)(C)C(=O)NC(C)C(C)NC(c1ncoc1C1CC1)=O C(=O)(CS(=O)(=O)N1CCC(CC(=O)NCc2cc(CC)n[nH]2)C1)OCC C12(NC(CCCC3C(C)C3)=O)CCC(CC1n1cc(-c3ccnn3C)nn1)C2 c1(C(=O)NCCCC(C)NC(c2ccc(CCCC)cc2)=O)c(F)cccc1Cl c1(C(N2C(C)CC(CNC(=O)C(F)(F)C3CC3)C2)=O)ccc2[nH]ccc2c1 N1(C(C(C=C)O)=O)CC(OC)CC1Cc1ccc(CNC(=O)OC(C)(C)C)cc1 CN1CC(NC(c2ccnc(CNC(=O)CCc3ccncc3)c2)=O)C(O)C1 Cc1cc(S(N)(=O)=O)oc1C(N1CC2CC1CN2C(c1cnc(O)o1)=O)=O CC(C)(F)CC(=O)NCCCCCc1cn(CCC(=O)N(C(C)(C)C)CC#N)nn1 N1(C(CC2CC(OCC)C2)=O)CC(NC(=O)CN2CCCCC2)CC1(C)CC c1(CC)nc(C(=O)NC2C=CC(CNC(c3cnncc3O)=O)C2)c(N)s1 N1(C(Cc2cc(C)[nH]n2)=O)CC2(CCN(C(c3cnn(C(C)C)c3F)=O)C2)C1 C1(CSC)CCc2nc(C)nn2C1.N12CC(C1)NC(=O)C1(CC1)C(=O)CC2=O C(CC(C)C)(C(C(=O)NC1CC(F)(F)C1)N(c1ccc2[nH]ccc2c1)C)SC CC1(C)OCCN(C(C2C3CCCCC23)C(=O)NC2CCOCC2)C1(C)C CC(CN1CCOCC1)C(=O)N1CC(OCCNC(C2(CCC#N)COC2)=O)C1 c1(C(C)C)nn(-c2ccccc2)cc1NC(c1csc(C2CCOC2)n1)=O c1(C(=O)NCC2C(NC(c3ncc(OCC)nc3)=O)C2)cc2cccc(F)c2o1 CCC(C)C(CC(=O)N1CC(CNC(=O)C(CO)NC(N)=O)CC(C)C1)OC c1(OC)cccc(F)c1CN1CC2C(C(=O)Nc3cccc(C)c3F)C2C1 Cc1c(C(N2CCC(C)(CCNC(=O)CN3CC=CC3)C2)=O)noc1C1CC1 C1(C(=O)NCCOC(C)(C)CNC(=O)Cc2ncc(Cl)s2)CCCN1C=O C1(N(C(CCCCC)=O)C)CN(C(c2c[nH]cc(F)c2=O)=O)CCC1C Cc1ccc2c(C(N3CCC(NC(=O)C4=C(Cl)CC4)C(C)C3)=O)coc2c1 N1(C(CC2CCCC(C)C2)=O)CC2CC(NC(c3cnc(F)c(F)c3)=O)CC1C2 Cn1c(I)cc2c(N(C3CCNC3)Cc3c(F)cc(Cl)cc3Br)ncnc12 c1(NC(c2ccc(-c3ccc(O)cc3O)nn2)=O)ncc(F)cc1Br C12(C(=O)NC3(CO)CCN(C(=O)Cc4ccc(Cl)c(F)c4)C3)CCCC1CCC2 N1(c2cc(CC)nc(C)n2)CC(NC(=O)C2=CCCCCC2)CC2(CC2)C1 CCCCC(CCCC)C(=O)NC1CC2CC(NC(c3cccc(C)c3)=O)C1C2 c1(CCNC(C(=O)NC2C(C)C2(F)F)=O)csc2ccccc12 C(=O)(C(O)CN1CCCC1)N(CC(C)C)CC(=O)NC1(C)CSC1 N1(C(CC2CN(C(C)=O)C2)=O)CC=C(CC(=O)N2CCCNC(=O)C2C)CC1 N1(C(C(c2ccc(O)cn2)C)=O)CC2CN(C(=O)C=Cc3ccc(Cl)s3)C2C1 Cc1c(NC2CCN(C3CCC(C)CC3)CC2)ncnc1N1CCSC(C)C1.OC C(=O)(C1=CCC2CCC1N2C(C12C(=O)C3CC1C2C3)=O)N1CC(OC)C2(C1)CC2 C1(C)(CNC(C(C)=C(CC)C)=O)CCC(NC(c2occc2C2CC2)=O)C1 CCC(C(=O)NCc1cc(C(=O)NCC(CC2CC2)CO)no1)SC C1(NC(C2C(NC(CC3CC(CC)C3)=O)CCO2)=O)CCOCCC1C c1(C(=O)NC2(CNC(CN(CCOC)C)=O)CCOC2)cnn(C(C)C)c1C c1(C(C)C)ccc(C(C)C)c(S(=O)(=O)N2CCCC(c3ncco3)C2)c1 N1(C(CC(C(=C)C)OCC)=O)CC2(CCC2)CC1C(=O)NC12CCC(CC1)C2 C1(C(=O)NCC(=O)NCC2C(NC(CCNC(=O)OC)=O)C2)CCCCC1 c1(C(=O)NC2CC3(C2)CN(C(=O)C(Cl)=CCl)C3)cc(O)c2cc(F)cc(F)c2n1 C(CC(C)(C)C)(C(=O)N1CCCC[Si](C)(C)C1)OC N1(C(C(C2CCCOC2)OC)=O)CCC(N(C(=O)C2=CCOC2)CCO)CC1 CC(C(C)(C)O)NC(=O)C(=O)NCC1CCC1CO C#CC1CCCC(NC(=O)CCCCCN(C)C(C2CCC2C)=O)C1 c1(-c2c(C(N3CC(SC)OCC3)=O)ccnc2)ccccc1-c1ncccc1F Cc1ncnc(C(=O)NC(C)C(C)(C)C(=O)NC2CC(CCF)C2)c1C C(=O)(N=c1[nH]n(C)c(=O)n1-c1ccc(C)cc1)N1CC(OC)OCC1 c1(C(CC)C)ccc(C(=O)NCC2(F)CC(NC(=O)C3=COCCO3)C2)c(C)c1 C#Cc1cc(C(N2CC3(C2)CN(C(C2(C)C(C)(C)C2(C)C)=O)C3)=O)cc(N)c1 c1(OC)cc(CCC(=O)NC(c2csc(Br)c2)C(=O)O)ccc1C Cc1cc(C(N2CCC(NC(=O)Cc3cn[nH]c3)CC2C)=O)ccc1Cl CC(C)CC(C)CC(=O)NC1(C)CCCN(C(C2CCCOCC2)=O)C1 N1(C(C(C(C)(C)F)(C)F)=O)CCC2(CCCCC2NC(=O)CS(=O)(=O)C2CC2)C1 C1(C(C)NC(CCc2cc(C)no2)=O)CN(C(C2(N=[N+]=[N-])CC2)=O)CCO1 C(=O)(CC(C)CN(C)C)N(CC(CC)NC(=O)CCc1ccncc1)C N1(C(=O)Cc2cc(Cl)sc2Cl)CC2CC(C1)N(C(=O)NC1(c3cc[nH]n3)CC1)C2 CCC(F)(F)CC(=O)N1CCOCC(C(=O)NCC2CCC(F)(F)C2)C1 N1(C(C(c2ccc(O)cc2)C)=O)CCC2CN(c3ncc4[nH]ccc4n3)CCC12 c1(CC(=O)NC2C=CCN(C(=O)Cc3cnccc3Cl)C2)ccc(F)cc1F c1(CNC(C2CC(F)CN2C(C2CC(O)CN2)=O)=O)c(Cl)cccc1[N+](=O)[O-] CC(C)CC(C)C(=O)NCC1(NC(=O)Cc2csc(C(F)(F)F)n2)CCCCC1 C(c1csc2ccccc12)=CC(=O)NC1CCC(C)N(C(c2ccncc2)=O)C1 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(C)(F)F)CC1c1ccccc1 C1(C2CN(C(=O)C(C)(C)c3ccno3)C2)(NC(C2CCC(OC)C2)=O)CC1 CCC(C)(C)CC(=O)N1CCC1CNC(=O)CN(C)CCO c1(CC(=O)NC2CCCC(NC(C3(O)CCOC3)=O)C2)nc2ncccn2n1 c1(CNC(C(=O)NC(C)C)=O)nnn(C)c1C(N1CCC2CC12)=O C1(CNC(C=CC(C)(C)NC(C2CC(=C)C2)=O)=O)CC(O)C12CCC2 C1(C)(CNC(C(=O)NCCOC)=O)CN(C(C2(Cl)CC2(F)F)=O)CCO1 C1(C(C)C)CCC(C)(C)CC1c1nc(-c2cc(O)nc(C3CCOCC3)n2)no1 N1(Cc2ncn(C)n2)CC(NC(=O)C=CC2CC2)C(O)C1 C1(C(=O)NCCN2CCC(NC(C(CC)OC)=O)CC2)CC2C(C1)C2(C)C CCC(C#N)C(=O)N1CCC(N2C(=O)c3cccc(c3)C2)C1.S(C)CC C1(CNC(C(C)c2cccs2)=O)CN(C(=O)C2=NOC(C)(C)C2)CCC1(C)C C1(C(=O)NCCCN(C(=O)CCCc2cc[nH]c(=N)c2)C)C2CCCCCCC12 c1(C(=O)NC(C)(CNC(=O)C2=CCC2)C2CC2)cc2ccc(Br)c(F)c2[nH]1 C1(C)(NC(C(C)OCC#C)=O)CCCN(C(C2CCOC2)=O)C1 CCCC(C)(O)CC(=O)N1CCCC1CCNC(=O)C(C)=C1CC1 c1(C(N(CCC)CCNC(=O)Cc2cnn(CC(C)C)c2)=O)cc(OC)ccn1 N1(C(C(C(CC)O)C)=O)CCCN(C(c2cc(Br)sc2C)=O)CC1CO N1(C(CC(C)CNC(c2cc[nH]c2)=O)=O)CCC(C)C(O)C1 CCS(=O)(=O)CC(=O)N1CCC(C(=O)NC(C)CC(F)(F)F)C12CC2 C(c1cccs1)=C(C)C(N1CC(CO)(NC(=O)CC2CCCC2)C1)=O N1(C(CC)=O)CCN(C(c2cscc2Br)=O)CC1c1cccnc1 c1(OCCCN(C(=O)C(=O)N2CC(NC(C)(C)C)C2)Cc2ccsc2)ccccc1 c1(-c2n(CN(C(CC)C)CCc3ccncc3)ccn2)cccc(-c2cscn2)c1 C1(C(C)=O)C(C(=O)NCC(C)(F)CNC(=O)CN2CCCC2=O)C1(C)C C1(CC=C)(NC(=O)C(C)N(C(=O)CC(=O)OCC)CCC)CCOC1 c1(C(N2C(CNC(c3n(CC)ncc3)=O)CCCC2)=O)cc(C2CC2)cc(F)c1 Cc1c(C(=O)N(CCC(=O)NC(C2CCCC2)C)CCCO)cccc1O Cc1cc(-c2ocnc2C(=O)NC(CNC(c2cc(Cl)no2)=O)C2CCC2)on1 n1(CCCC)nccc1C(=O)NCCC(C)N(C(=O)C=CC(C)CC)C CCCCCC(=O)N1CC(CC)(NC(=O)CCc2cnn(C)c2C)C1 c1(C(N2CCN(C(c3c(CC)csc3)=O)C(COC)C2)=O)ccc2cc[nH]c2c1 c1(C(C)CCCCCCC(=O)NC(=O)CC(C)c2ccco2)cnccn1 C12(C(N3CCC(OC)CC3)=O)CCC(C1)N(C(c1ccc(N(C)C)cc1)=O)C2 c1(C(=O)N(C2CC(C(=O)O)N(C(c3ccc(Cl)cc3Cl)=O)C2)C)scc2c1CCCC2 N1(C(C2C(CC)CN(C(c3ccccc3NC)=O)C2)=O)CCCC2(C=CCO2)C1 c1(C(=O)NC(C2(C(=O)NC(C)C(=O)NCCF)CC2)C)cnc[nH]1 c1(NC(Cc2cccc(OCc3ccc(C)cc3)c2)=O)cnc(Cl)c(C)c1 c1(OCC)ccc2cc(C(=O)N(C(C)CNC(C3CCCN3C=O)=O)C)[nH]c2c1 N1(C(C(COC)OC)=O)CCC(NC(C2(CC(C)=O)CC2)=O)C(C)(C)C1 N1(C(c2ccc(CNC(C(C)CC3CCC3)=O)s2)=O)CC2C(C)C2C1 c1(C(C)=O)cc(C(N2CCN(C(c3coc(C)c3)=O)CC2CCO)=O)ccc1C C1(NC(CC2OCC(C)(C)OC2)=O)CC2(CCN(C(=O)C(N)CN)CC2)C1 C1(NC(CNS(CCOC(C)C)(=O)=O)=O)CC(O)CN(C(=O)CN2CC=CC2)C1 C(=O)(C(O)C(C)C)N1CCC(N(C(=O)CCC2CCCC2)CC)C1 C1(NC(C(c2cccs2)NC(=O)Cn2ccccc2=O)=O)CCCC(O)C1O c1(C(N(C2CCN(C(=O)CC3CCC(=O)N3)CC2)C)=O)cc2ccoc2cc1F CCS(=O)(=O)CC(=O)NCC(C)NC(=O)CC(O)C1CCCC1 c1(NCc2c(N)nccc2)cc(=NCCCc2cccc(OC(F)F)c2)[nH]cn1 CC(CN1CCCC1=O)N=c1[nH]c2c(c(=NCc3nncn3C)[nH]1)CSC2 c1(C(N2CCOC(C(F)F)CC2)C(=O)NC(CC)(C)C)cc(C2CC2)cc(C)c1 N1(C(c2c[nH]c(=NCC=C)s2)=O)CCN(C(=O)CCOCC(F)F)C2COCC12 c1(C(N2CC(NC(CCOC(C)C)=O)CC(C)(C)C2)=O)c[nH]c(=N)c2[nH]ccc12 N1(C(C(C2CN(C(C3COC(=O)C3)=O)C2)OC)=O)CC2C(C1)C2(F)F CCC1=C(C(=O)NCC(C2CCC2)NC(C2(F)CCCN(C)C2)=O)CCCO1 N1(C(C)=O)CC2(NC(=O)Cc3cc(OC)cc(Cl)c3)CCC1CC2 C(=O)(C1CCc2nccn21)NCC1(CCNC(=O)CC2CCC2)CC1 c1(C2(C(N3CCC(c4scc(C)n4)CC3)=O)CCC2)ccc(F)cc1Br CCCC(C(=O)N(C)CC1COCCN1C(c1csc(=NC)[nH]1)=O)OCC c1(NC(C2CC23CCN(Cc2cccc(F)c2Br)CC3)=O)cc(F)cc(F)c1Br c1(C(N2C(C)(CNC(C3C(=C)C3)=O)CCC2)=O)nc(C(F)(F)F)n2ccccc12 CC1(C)NC(=O)N(CCCC(N2CC3CC2(CNC(=O)C=C(Cl)Cl)C3)=O)C1=O C1(C2CCCCC2)(C(N2CCN(C(C3C(C(C)C)C3)=O)C(C3CC3)C2)=O)CC1 c1(C(c2nnnn2C)NCC(F)(F)Cl)ccn(C2CC2)n1.C1(C2CCC2)CCOCC1 c1(C(N2CCC(CN(C)C(C3(C)CC=CCO3)=O)CC2)=O)nccc(C#N)c1F C1(O)(CCNC(Cc2cc(C)ns2)=O)CCCN(C(C2CS(=O)(=O)C2)=O)C1 N1(C(c2ccn(C)n2)=O)CCSCC1C(=O)NC1CC(c2ccccc2Cl)C1 C1(C(=O)NC(C2(O)CCN(C(=O)Cc3cnsc3)CC2)C)C2CCC3C(C2)CC13 C=CCC(C(=O)NCC(C(C)(C)C)NC(C1CCC(=C(F)F)CC1)=O)C(C)C c1(C(N(C2CN(C(C3(Br)CC3)=O)CC2O)C)=O)c(Cl)cccc1Cl N1(C(c2ccn(C)c(=O)c2)=O)CCC2CC2(NC(c2csc3nnsc23)=O)CC1 c1(C(=O)NCCCN(C(CN(CC)CC)=O)Cc2ccccc2)csc(C)c1 C=CC1(C(F)(F)F)CCN(C(N2CCC3C(CC(=O)OC)C23)=O)C1 c1(C(N2CCC(c3n[nH]c(=N)o3)CC2)=O)nc2ncc(CCO)cn2n1 N1(C(c2ccc(C)c([N+](=O)[O-])c2)=O)CC(NC(C2(C)CC2)=O)CC12CCOCC2 c1(C(=O)NC2CC(C)(NC(c3coc(Br)c3)=O)C2)cc2nc[nH]c2cn1 C(=O)(C1CCc2ccccc21)NC(C)(C)CCC(=O)NC1CCN(C(N)=O)C1 CC(CCCC(=O)NCc1cnco1)NC(c1cn(CCO)nn1)=O C(c1ccccc1)=CC(=O)NC1CCN(C(C2CC2c2ccc(Cl)o2)=O)C1 CC1(C(N2CCOCC(NC(C3CCCS3(=O)=O)=O)C2)=O)CC2CCC1C2 CC(C)S(=O)(=O)CC(=O)NCCN(C(=O)CN1CCSCC1)CC1CC1 N1(C(C2CCN(C(c3ccc(CC)s3)=O)C2)=O)CC2C(CN(C)C)C2C1 C1(OC)CCC(F)(Cc2cn(CC(=O)Nn3nc(C)cc3C)nn2)C1 CC(CF)CC(=O)NC1(CNC(c2cccs2)=O)CCOC1 Cc1c(O)nc2ccccc2c1C(=O)N(C)CC1CN(C(=O)CC(C)(F)F)C1 c1(C(=O)NC(C(C)NC(CCCCN(C(C)=O)C)=O)C(C)C)ccn(C)c(=O)c1 C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(=O)Nc2ccc(Cl)cc2)CC1O N1(C(C=C(C)C)=O)CCCN(C(=O)Cc2ccccc2C(F)(F)F)CC1C(C)C N1(C(c2n(C)ccc2)=O)CCN(C(=O)CC2CCN(S(C)(=O)=O)CC2)CC1CF c1(C(N(C)CC2(O)CN(C(C3(CCOC)CCCC3)=O)C2)=O)cc(O)ccc1F C(CC(O)C(F)(F)F)NC(CN(C(Cn1ncc(CC)c1)=O)C(C)C)=O c1(NC(C(CCC)C)=O)cc(C)c([N+](=O)[O-])cc1[N+](=O)[O-] Cc1ccc(F)c(NC(C2CC(C)CN2Cc2ccc(O)c(F)c2)=O)c1 c1(-n2c(CCCC(C)(F)F)nc(C(C)OC)n2)ccc(S(=O)(=O)N(C)C)cc1 N1(C(C(C(C)C)F)=O)CCCC(C)(C)C1C(=O)NCCc1ccns1 N1(C(CCCCCOC)=O)CCC(C(=O)NCC(C)CC(C)C)=C(F)C1 C1(C)(C(=O)NC(C(C)CO)C)CCN(C(C2CCCC2)=O)CC1 Cc1c(Br)ccc(CNC2CC2C(N2CCOC3CC23)=O)c1F C1(NC(=O)CCF)CC(NC(=O)C=C2CCOCC2)C(O)C1 c1(CNC)cnn2c1CN(C(=O)COCC1CCC1)CC2.C1(C=O)(CF)CCC1 O=C1NCC2(CC(N=c3[nH]c(N4CCC(F)CC4)nc4ccc(Cl)cc34)C2)O1 N1(C(c2c(Br)cnc(C)n2)=O)CC2CCC(NC(=O)Cc3ccco3)(C2)C1 N1(C(c2nccc(CC)c2)=O)CC2CC(NC(c3ccc(F)nc3)=O)CC2C1 N1(C(c2c(OC)ccc(OC)n2)=O)CC2(C1)CN(C(=O)CC1(C)CC1)CCO2 C(=O)(CC(C)(C)CN(C)C)N(C1CCN(C(=O)C(c2ccccc2OC)C)C1)C.CO N1(C(c2c(CC)onc2C)=O)CCN(C(c2cc(Cl)no2)=O)C(CCOC)C1 C(=O)(C1=CNC2=NCCC2=C1)NCC(CN(C(c1ccc(CC)c(C)c1)=O)C)O N1(C(CC(c2ccc(OC)cc2)C)=O)CC(NC(c2csc(O)n2)=O)CC1(C)C C1(c2n(CC)nnn2)(Nc2cccc(C(F)F)c2C)CCOCCC1C N1(C(c2cc(CNC(C(CCC)C)=O)sc2)=O)CCCC2(C1)N=N2 N1(C(CCC(CC)OC)=O)CC2CCCC(C1)N2C(C1CC1CC)=O C(=O)(C(C)(F)C(=O)NCC1(CN(C(c2cnoc2-c2cccs2)=O)C2CC2)CC1)OC c1(C(=O)NC2CCC(CCNC(C3(CC)CCCC3)=O)C2)ncc(N)nc1C O=C1CC(=O)CC(C(N2CCC2CC(=O)NCCOCC(F)(F)F)=O)C1 C1(C(N2CCC(O)(C(C)NC(c3ccns3)=O)CC2)=O)CC2CC1CC2(F)F O=C(N=c1c(Br)c[nH]cc1I)C1(F)CCN(Cc2ccc([N+](=O)[O-])o2)C1 c1(N(C(C)CNC(c2ccnn2-c2ccccc2)=O)C)cc(Cl)nc(S(C)(=O)=O)n1 c1(CCC)cc(C(=O)NCC(C)(O)CNC(=O)C(C)C(F)F)c(C)o1 c1(C(=O)NC(C2CCCC2)CNC(C(C)SCC)=O)cccn2c(C)cnc12 C12(NC(CCC#C)=O)CCCN(C(c3ccnc(C)n3)=O)CC1C2 C1(CC(=O)NCC(CCOC)NC(C2(C(=O)OCC)CC2)=O)CC(F)C(=O)N1 C(CCNC(C1CCC12CCC2)=O)(C(C)C)NC(Cc1c(C)ncs1)=O N1(C(Cn2ncc(C#C)c2)=O)CCCC2(C1)CN(C(=O)CN1CCC(O)CC1)C2 CCCCC(C)(F)C(=O)NC1CCN(C(C2COC(C)(C)C2)=O)C1 CC1(C)c2[nH][nH]c(=NC(=O)c3ccnc4ncccc34)c2CN1C(=O)C(F)Br c1(C(=O)NCC2(F)CN(C(COCC#C)=O)C2)cncc2ncccc12 c1(CNC)cnn2c1CN(Cc1cnc(-c3ccc(OC(C)C)cc3)s1)CC2 Cc1nc(O)sc1C(=O)NCC1CC(C)N(C(=O)C=CC(=O)N(C)C)C1.C(CO)N N1(C(CCCCCCC)=O)CCCC2C(NC(c3ocnc3CC)=O)C(C)(C)C12 c1(C(N2CCN(C(C3CC4CCCC34)=O)CC2)=O)c(F)ccc2nc[nH]c12 O=C(NNc1ncc(F)cc1F)NCc1ccc2c(c1)CCCC2 N1(c2cc(NC(c3n(CC)ncn3)C)nc(C(C)C)n2)CCn2ncc(C)c2C1 N1(C(CC2N(C)CCC2)=O)CCC2OCCN(C(=O)CCc3cnoc3)C2C1 c1(OCC(=O)NCC(C(C(C)C)C)NC(c2nncs2)=O)ccc2c(c1)CCC2 c1(C(=O)NC(C)CNC(=O)CC(C)(F)F)cc(S(N)(=O)=O)cc(Cl)c1F N1(C(c2c(C)coc2C(C)(C)C)=O)C(C)CC2CN(C(=O)CNS(C)(=O)=O)CC12 C1(NC(=O)NC(CCSC)C(=O)O)C2Cc3ccc(Br)cc3C12 C(=O)(C(C(C)O)NC(=O)Cc1ccsc1C)NCc1c(CC)con1 CN1CC(C(N2CC(CO)(NC(=O)C(c3cccn3C)=O)C2)=O)CC1=O CCC(CC)CCC(=O)NC(CNC(=O)CC(C)(C)C(F)F)C1CC1 N1(C(C(C(C)C)SCC)=O)CCOCC(CNC(C2CCCN2C2CC2)=O)C1 C=C(Cl)CC(C(=O)N(C1CC2CC2C1)C)NC(c1ncc(C)cc1F)=O N1(C(c2ccn(C(C)C)n2)=O)CCCCC(C(N2CC3CCC3(C)C2)=O)C1 Cc1ccc(C(=O)NCCCCCNC(c2cc3occc3s2)=O)c2c1CCC2 C(F)(c1ccccc1)=CC(=O)N(C1CN(C(=O)C(C#N)C2CC2)CC12CC2)C C#Cc1cncc(NC(=O)C(O)CCCNC(=O)C(F)OC(F)(F)F)c1 CC1CCN(C(=O)Cc2csc(N3CCC(O)CC3)n2)CCN1C(=O)CCC#N c1(C(N2C3CN(Cc4cc(Cl)c(Cl)cc4O)CC23)=O)cc(F)c(F)cc1Cl C12(C(=O)NC(C3CN(C(C4CC4c4ccc(F)cc4)=O)CCO3)C)CC(CCO1)C2 c1(C(C)C)cccc(CC(=O)NCCOCCCNC(c2ccon2)=O)c1 C1(N(C)C)CCC(CNc2cc(NC(c3ncc[nH]3)CO)ncn2)CC1 c1(OCCC(=O)NC2CC(N(C)C(c3nccnc3N)=O)C2)cc(F)ccc1F C1(C(N2CC(O)(CC=C)C2)=O)CN(C(C2COCCN2C(C)C)=O)CC1C(C)C Cc1n[nH]c(C)c1CC(=O)NC1(CNC(=O)CCOCC(F)(F)F)CCOC1 C1(S(N)(=O)=O)(CNC(C2N(C(c3n(C)nc(O)c3)=O)CCC2)=O)CCCC1 c1(NC(C(=O)NC2CCCC(C(C)(C)C)C2)=O)cc(C(N)=O)ccc1C CC1CC(CO)N1C(C1(CCNC(c2ccc(Cl)s2)=O)CCC1)=O c1(N2CC(CC=C)(NC(=O)CCc3ccccc3F)C2)cc(C(N)=O)nc(Cl)n1 c1(C(=O)NC2C(C=C)CN(C(=O)C=NOC)C2)nn2c(c1C)OCCC2 N1(C(CC(C)OC(C)(C)C)=O)CCN(C(=O)C(C2CC2)NC(N)=O)CC1C S1(=O)(=O)c2c[nH]c(c2)C(=O)N(C)CCN1C1CC1.C1(C)(NC)CCC(C)C1 C#CC(CNC(=O)CC(C)NC(=O)C=CC(C)CC)C(C)C Cc1cc(Cl)ccc1C(=O)N(C1CCCN(C(=O)Cn2cnc(C#N)n2)C1)C c1(N(C(=O)Nc2cccs2)CC2CCSC2)ccccc1 c1(NC(=O)C(N2CCC3(CCSC3)C2)=O)cccc(P2(=O)CCCC2)c1 N1(CC(F)F)CCCC(N=c2ccnc(N3CCCC(c4nc(O)n[nH]4)C3)[nH]2)C1 CC1CN(C(=O)C(O)(C2CC2)C2CC2)CCN1C(c1coc(Cl)n1)=O c1(CC)cc(C)ccc1C(N1CCCC(N(C)C(c2ccn(C)c2CC)=O)C1)=O C1(NC(c2ncc(OCC)nc2)=O)C(C)CN(C(c2sc(C)cc2C)=O)CC1C Cc1cc2sc(C(=O)NC3CCN(C(=O)Cn4ccnn4)C3(C)C)cc2s1 C1(CC(N2CC(NC(=O)CCc3ccco3)CC2C)=O)(CC)CCOCC1 C1(C(N(CCOCCNC(CCSC)=O)C)=O)CCC(=O)N1C(C)C S(=O)(=O)(c1ccc(N(C)Cc2ccoc2)cc1Cl)NC(CCOC)C(C)(C)C N1(C(C2(CC)CCCO2)=O)CCC(C(=O)N2C3CCC2CC(F)C3)=C(F)C1 N1(C(C(=O)NCC)=O)CC(C)C(NC(c2ccc(-c3cccs3)cn2)=O)C(C)C1 C1(C(N(C(C(=O)OC)C)C2CC2)=O)CCC(c2ccc(C)cc2)CC1 c1(CNC(c2cc[nH]n2)=O)c[nH]nc1C(=O)N(CC(F)F)CC1CCC1 N1(C(C(C(C)C)CN(C)C)=O)CC(NC(=O)CC=C(Cl)Cl)C2CCCC12 c1(C(=O)OCC)cnc(O)c(OC2CN(C(=O)CC3CCC3(C)C(=O)OC)C2)c1 C1(C(=O)NCCCC(C)NC(C(C)OCC)=O)CCOC(C)(C)C1 N1(CC(=O)N(c2nc(C)sc2C)CCC)CC(O)C(O)C12CCC2 N1(Cc2nc(C)c(C)s2)CCN(N2CCCC(c3nncn3C3CC3)C2)CC1 CC1CN(C(=O)CC2CSCCO2)CCC1NC(c1ccc(Cl)c(O)c1)=O N(C1CC2(CCN(C(C3(Br)CC3)=O)C2)Oc2ccccc21)C(=O)Cn1cnnn1 c1(CC(C(=O)NCCCCC=C)NC(=O)C(C2CCOCC2)F)cnn(C)c1O C1(C(=O)NC2(C(N)=O)CC2)C=CCN(C(=O)Cc2ccccc2F)C1 C1(NC(C=C2CCC(C)C2)=O)CC2CCC1CN(C(C13CC1COC3(C)C)=O)C2 C1(F)(CNC(C2CC(=O)OC2)=O)CC2CCC(C1)N2C(=O)C(O)(C1CC1)C1CC1 c1(C(=O)NCC2CN(C(C(COC)C)=O)CC2O)cc(F)cc2cccnc12 C(=O)(C(O)CCC(C)C)NC1CC(NC(C=CSC)=O)C1 Cc1ccc(C(N2CCC(NC(c3oc(Br)cc3C)=O)C(F)C2)=O)cc1Br C1(CC(=O)NC2CN(C(C(C)(C)N(C)C)=O)CC2F)CC(c2ccccc2)=NO1 C=CCC(C(=O)NC1(C(C)(C)NC(c2cnc(CSC)s2)=O)CC1)C(C)C C1(NC(=O)CCc2cnoc2)COCCN(C(=O)C(O)Cc2ccc(F)cc2)C1 CC1(C)CCC(O)(CNC(C2C=CC(NC(C3C=CCC3)=O)C2)=O)C1 CC1CN(C(C2CC23CCOC3)=O)CC(C)N(C(=O)CN2CC(=O)N(C)C2=O)C1 c1(C(=O)NC2CCCN(C(c3ccc(OC)c(N)n3)=O)C2)ccc(S(C)(=O)=O)o1 C(=O)(CC(O)C(C)(C)C)N(CC(C)NC(c1ccc(OCC)cc1)=O)C CC1CN(C(C2CC(=O)NC2(C)C)=O)CCN1C(c1cc(Br)cs1)=O C1(C2CCCOC2)(NC(C(C2(C)CC2)NC(CC(C)(F)F)=O)=O)CC1 N1(C(C2=CCCN(C(C(C(CC)O)C)=O)C2)=O)CC(C)NC(=O)C12CC2 c1(C(=O)OC)ccc(OC)cc1C(=O)NC1CCCCN(C(=O)C(O)C2CC2)C1 c1(OC)cc(C(=O)NCCOc2ccccc2Cl)c2c(c1)CCO2.C1(=O)CO1 C(=O)(CCCCC(F)F)N1CC(CNC(C2(C#C)CCCC2)=O)N(C)CC1 CCCCC(F)C(=O)N(C(CNC(=O)C(C)NC(=O)CC)C1CC1)C C(CCC(C)C(=O)N(C1CCCCN(C(=O)CCc2csc(=N)[nH]2)C1)C)OC CC1CC=CCC1C(=O)N(C1CCN(C(=O)Nc2cc(Cl)cs2)CC1)CC1CC1 c1(C(N2CC(NC(c3cc(CC)oc3)=O)C(OC)C2)=O)cnc2n1CCC(C)C2 c1(-c2n(-c3ccc(COC)cc3)nc(CCC(C)C)n2)ccc(C)cc1C C1(C(N(C2CCN(C(CCC=CCC=C)=O)C2)C)=O)CC2(CCC2OC)C1 C1(NC(C(CSC)(C)O)=O)(CO)CCCN(c2ccnc(Cl)n2)C1 C(C(O)C(=O)NC(c1cnn(C)c1)C(=O)N(C1CCC1O)C)=CC C(=O)(C(C)C(F)(F)C(F)F)NC(CC)(CNC(C1(C)CCNC(=O)C1)=O)CC c1(C(N(CCC(C)NC(C(CC)C(C)C)=O)C)=O)ccc2c(c1)NC(=O)CS2 CC1OCCCC1C(=O)NC1CC(CNC(=O)C=CCOc2ccccc2)C1 c1(C(C)C)ncc(Cl)c(C(=O)NC2CC23CC(NC(c2ncncc2Cl)=O)C3)n1 C1(CNC(C(C(C)C)O)=O)CN(C(C2CC(F)C2)=O)CC1(C)C c1(-c2cn(CCC(=O)N(C3C(OC)CCCC3)C)nn2)ncc(Cl)cc1F c1(C(=O)NCC2C(NC(C(C(CC)C)O)=O)CCCC2)cc(F)c(F)cc1OC Cc1[nH]c(C(N2CCCC(C)CC2)=O)c(C)c1C(=O)NCc1csc(C#N)c1 C#Cc1cnc(N2CC(=C(F)CNC(=O)CCc3ccccc3C(N)=O)C2)nc1 C1(O)(C(=O)NC2CC(N(C(C=CCN(C)CC)=O)C)C2)CCc2ccccc2C1 N1(C(CN(C(C2C(CCC)C2)=O)C)=O)CCC1C=O.C(C)(C)C C1(C(=O)NCC(C2CCCCC2)NC(C(CC)F)=O)CCN(CCO)C(=O)C1 C1(c2ccc(C3(NCCNC(=O)Cc4nn[nH]n4)CC3)cc2)CCCCC(=O)N1 C(=O)(C(C)C(C)S(C)(=O)=O)N(CCCN(C(C(C(CC)(C)C)O)=O)C)C C(=O)(CN1C(=O)COc2ccc(Cl)cc21)NC1C(NC(c2cncc(C)n2)=O)C1 c1(OC)ccc(CC(N2CCC(=O)CC2C(=O)O)=O)c(Cl)n1 c1(C(N(C(C)C)CCNC(c2ccnn2C2CC2)=O)=O)ccc2nccn2n1 N1(c2nc(N(CCC)C)c3c(n2)c(C)nn3C)CCc2c([nH]c3ccccc23)C1 N1(C(CC=C)=O)CCC(NC(c2cc(O)n(CC)n2)=O)CC1 c1(CC(=O)NCCC2CCCN(C(C3CC(C)(F)C3)=O)C2)noc2ccccc12 N1(C(c2c(C)nc(C)s2)=O)CC2OCC(NC(=O)CCOCC(F)F)C2C1 c1(C(N(C)CC2N(C(c3c(CC)onc3)=O)CCC2)=O)nsc2ccccc12 Cc1cc2cc(C(=O)NCC3CC(C)(C)CN3C(=O)CCC(F)F)oc2cc1C c1(C(=O)NC(CCC)CNC(C2CC2C(C)C)=O)c(N)ccc(F)c1F C1(C(=O)NC(CC)COC)(C(c2ccccc2)O)CN(C(C2CCCC2C)=O)C1 c1(NS(CC)(=O)=O)cnc(Cl)cc1C(=O)Nc1nccnc1Sc1ccccc1 c1(CC)onc(C(N2CCCC2C(C)(C)C(=C(C)C)NC(=O)C#CC2CC2)=O)c1C O(C1CCCc2ccccc21)CC(=O)NOc1cccc(F)c1Br N1(C(COc2cccc(C)c2)=O)CCC(C)C(NC(=O)C=CCCC(C)C)C1C CC1CCCN1C(=O)CCSC1CCCC1.C(=O)(CCCn1ccnc1)OC C1(CCCNC(Cn2c(C)nnn2)=O)CN(C(c2cc(O)nn2C)=O)CCO1 c1(C(N2C(c3cn(C(C)CO)nn3)CC(C)(C)C2)=O)cc2n(n1)CCC2 Nc1ncc(C(=O)Nc2nc3c(s2)CC(C(F)(F)F)CC3)cc1[N+](=O)[O-] C1(C(N2C(C)(C)CC(NC(c3cnn4c3CCC4)=O)C2)=O)CNC(=O)CC1(C)C CC(C(=O)NCCC1(O)CCN(C(C2(c3ccno3)CC2)=O)C1)C(F)(F)F C1(OC)(CNC(c2ccc(C)c(Cl)c2)=O)CCN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1 c1(NC(c2cc(C)sc2N)=O)ccc(C)c(Br)c1 C12(C(=O)NC3CCN(C(C=CCC)=O)CC3(C)C)CC3CC(C(=O)N1)C2C3 C=CC(C)(O)CC(=O)N(C1CCN(C(=O)COCCCC)C1)CC1CC1 c1(C(=O)NC(CCCNC(CCN(CCC)C)=O)C)ncnc(C)c1OC C(N=c1[nH]c(Cl)ncc1F)C1N(C(C2(CC#C)CCCO2)=O)CCCC1 CC(CSC1CC(OC(F)F)C1)C(=O)OC(C)(C)C CC1(C)CC(C(=O)NCC2CCCOCC2)N(C(=O)Cc2c(Cl)cccc2Cl)C1 c1(C(=O)NCC23CC2CN(C(C2CCCC(F)C2)=O)C3)cc(O)nc(C2CC2)n1 C1(OC)CC2(C1)CC2C(N1CCCC1CCNC(C1(C)CCCO1)=O)=O N1(C(CCC2(C)N(C(CC(CC)CC)=O)CCC2)=O)CCCN2CCCC2C1 C1(N(C(C2C(C=C)C2)=O)C)CCC(NC(=O)C(c2ccc(OC)cc2)C)CC1 C1(N(C(C2C3(CC3)C23CC3)=O)CC)CCCN(C(=O)CCC2CCC2)CC1 Cc1cc(Br)cc2[nH]c(C(=O)NC3CC(CCNC(=O)C(C)(C)O)C3)cc12 C(c1cccnc1C)=CC(=O)NC1CCN(C(CN(C)CC)=O)C1C1CC1 Cc1ncc(CCOC(=O)Oc2ccccc2)n1C.C12(C)CC(O1)COC2=O CC1(C)CCC1C(=O)NC1COCC1NC(c1nscc1Br)=O N1(C(c2cnc(C(C)O)s2)=O)CCC2(CC1)CCN(C(c1cnnc(Cl)c1)=O)C2 C=CCC(CO)NC(C1(C)CN(Cc2c[nH]nc2-c2ccccc2)C1)=O c1(C(N(C(CCNC(Cc2nc(C)sc2C)=O)C)C)=O)ccc(Cl)cc1O CN=c1[nH]cc(C(N2CC(OC)C(NC(=O)C(n3ccc(C)n3)C)C2)=O)s1 C(=O)(C1=NOC(c2ccccc2)C1)N1C(C(=O)N(CC)Cc2cc[nH]n2)CCC1 CC(C)CC(C)CC(=O)N1CCC(CNC(c2ccc(C(C)C)cn2)=O)C(C)C1 Cc1oc(C#N)cc1C(=O)NCC1(CNC(=O)CC(C)c2ccco2)CC1 C1(C)(C(N2CC(CNC(c3cn(CCCOC)nc3)=O)C2)=O)CCCC1O C1(C(=O)NCC2C(CNC(Cc3c(C)scc3)=O)C2)COC2COCC2O1 c1(C(C)=O)nc(C(=O)N(C(C)CCNC(=O)Cn2ccc(C(F)(F)F)n2)C)cs1 CC1CCCCC1OCC(=O)NCCC1CN(C(c2cnc(C3CC3)[nH]2)=O)C1 c1(CC)cnc(N2CCC(C)(NC(c3cnn(C)c3CC)=O)C2)nc1 c1(OC)ccccc1C=CC(=O)N(CCCNC(C1CCCC1(C)C)=O)CCO N1(C(CCN(C)CC)=O)CCC(C(N2CCCC2C(C)O)=O)C1 C1(CNCCCNC(CCSC)=O)CC(C)N(C(c2ncc(F)cn2)=O)C1 C(CC(CO)NC(=O)CCN(C(=O)C(C)n1cccn1)C(C)C)SC c1(CC(=O)NCC2(F)CC(CNC(CC)=O)C2)cnc2n1CCCC2C C1(CNC(C2C(CNC(CCOCC#C)=O)C2)=O)CCOC(C)(C)C1 C1(C)(NC(c2nc(C(C)NC(c3nc(C)oc3C)=O)oc2)=O)CCC(=O)N(C)C1 c1(C(=O)NCC(CNC(c2ccncc2N)=O)OC)cc2nc(C)[nH]c2cc1F N1(C(C2CCN(C(c3c[nH]c(=NC)o3)=O)C23CC3)=O)CC(C)(C)OCC1C C1(CNC(C2(O)CC(C)(C)C2)=O)CN(C(=O)CCC(CF)CF)CC12CCC2 c1(C(=O)NCC(CNC(=O)CC2CCSCC2)F)cc(Cl)c(F)cc1[N+](=O)[O-] N1(C(C(C(CC)O)C)=O)CC2CCOC2(CNC(=O)CCn2ccccc2=O)C1 CN1C(=O)CC(CNC(C2CC(N(C)C)C2)=O)C1c1cccnc1 C1(CC)(NC(C2CCCC2CNC(C2COCC(C)O2)=O)=O)CCCCCC1 c1(SCC(=O)NCC(CC)(C)NC(=O)C(C)(F)C(=O)OC)cc(C)cc(C)c1 N1(C(=O)C(Cl)=CCl)CCOCC(NC(c2cnc(-n3cccn3)cn2)=O)C1 C1(C(=O)NCc2occ(C(=O)NCC3(CO)CCN(C)C3)n2)CCC(O)CN1C C(=O)(C1=CCC(C)(C)CC1)NC(CC#C)C(=O)N1CC(O)(CO)C1 CCC(C)(C)C(C(=O)N1CC2CCN(C(c3sc(SC)cc3C)=O)C2C1)OC c1(CN(C(COC(C)C)=O)C(C)C)noc(-c2ccco2)n1 n1(CC(=O)N(C)CC2CN(C(=O)COCC(F)F)C2)cnccc1=O CC(C)(CC(=O)NCC1(C)CCCC1NC(=O)C=Cc1cocn1)C(F)F c1(C(=O)N(CCO)C2CC2)cc[nH]c2nccc1-2.C(=O)(N1CCCCO1)C1CC1 C1(NC(c2sc(C)c(O)n2)=O)C(C)CCN(C(c2ccc(C)n2C)=O)C1C C1(C(C)NC(CCCN(C(C)=O)C)=O)CCN(C(=O)CC2(CO)CCC2)CC1 C(CC(C)(C)C)(C(=O)N(CC(C)O)C)NC(c1c(C)ccc(C)n1)=O c1(C(N2C3CC(NC(C4CCC(=C)CC4)=O)(C3)C2)=O)ccc(F)cc1O C1(C(N2CCC(O)C(CO)C2)=O)(CC)CCN(C(c2cc(OC)ncn2)=O)CC1 c1(OC)cnc(C(=O)NCC23CC2CN(C(=O)C2=CCCCC2)C3)c(OC)n1 Cc1ccc2c(CN3CCC(NC(c4ccc(Cl)c(C)c4)=O)C(F)C3)c[nH]c2c1 C12(NC(c3coc4c3CCCC4)=O)CCC(CN(C(=O)C(F)C3CCC3)C1)C2 C1(C(N(CC(CC)OC)C)=O)CC(NC(c2ccc(C)cc2)=O)C(O)C1 n1(CCC(C)(C)NCC)c(N2CCCC2)nnc1-c1ccc(C(N)=O)cc1 C1(C(N2C(CC(=O)OC)CCC2)=O)CN(C)CCN1C(C1CC(=O)C1)=O C1(CCNC(c2n(CC)ccn2)=O)CSCCN1C(c1cn(C2CCC2)nn1)=O CC(CC1=CCCCC1)NC(N1CCCCC1c1nc(-c2cccnc2)no1)=O C#CCC(C)(C(=O)NC(CC)C(C)CN(C)C)NC(c1cc(N)cc(F)c1)=O c1(C(=O)NC2C(CC)CN(C(c3oc(SC)cc3C)=O)C2)c(C)ccc(C)c1C C1(NC(C)=O)CCN(C(C2CN(CC(C)(F)F)C2)=O)C(C)C1 N1(C(COc2ccc(C#C)cc2)=O)CCC2C(C1)CN2C(c1ccoc1Cl)=O c1(C(c2nnnn2C)Nc2c3cn(C)nc3ccc2)cc(Br)cc([N+](=O)[O-])c1 N(C1CCOc2ccc(Br)cc21)C(C1CCCCN1Cc1c(Br)cncc1Br)=O Cc1nc(C2C(C(=O)NC34CC(NC(c5cn[nH]c5)=O)(C3)C4)C2(C)C)n[nH]1 N1(C(c2nn(CC)c(O)c2)=O)CC2(CC(NC(c3nc(O)c(C)s3)=O)CO2)C1 CC(C)C(F)(CNC(=O)C1=NOC(C)C1)C(=O)Nc1ccc(F)cc1 c1(C(=O)NC2CN(C(C(CSC)(C)C)=O)CC(O)C2)ccc2nc(O)sc2c1 C1(F)(CNC(C2(C)C(C)CCC2)=O)CCN(C(=O)C=Cc2ncco2)CC1 C1(NC(C(CC)NC(=O)CC2CCCOCC2)=O)COC2COCC12 Cc1cc(C(=O)NCC(=O)NCCOCCNC(=O)C(C)(C)C)ccc1C(F)(F)F Cc1[nH]nc(C(N2CCC(C(C)C(=O)N(CC(C)O)C3CC3)CC2)=O)c1O c1(C(N(CC(=O)N(C2CC2C)C)CCOC)=O)cn(C2CC2)cn1 C(=O)(CC1=NNC(=O)C1)NCC1N(C(C2(C)CCC(=O)NC2)=O)CC1 c1(C(C)N(C(c2cnn(CCNC(=O)CCCF)c2)=O)C2CC2)ccccc1F c1(NC(CC2N(C(CCN(CC)CC)=O)CC2)=O)cccc(Cl)c1C Cc1nn(CC(N2CC3CC3(CNC(=O)C(C)CN(C)C)C2)=O)c(C)c1Br C1(C(C)C)COCCN(C(C2CCN2C(=O)C(F)=CC2CC2)=O)C1 C1(CCNC(c2c(C)nn[nH]2)=O)CN(C(=O)Cc2cncc(O)c2)CCS1(=O)=O c1(C(N2CCC(NC(C3C(CCOC)C3)=O)CC2C)=O)cc(Cl)cc(Cl)c1OC c1(C(N2CCC(N(C(c3nccc(NC(C)=O)c3)=O)C)C2)=O)c(F)cncc1F C1(C(N(CC(C)NC(c2ccc(F)cc2NC)=O)CC)=O)CCc2nc[nH]c2C1 c1(NC(C(N2CCC(C)(CNC(CSCCOC)=O)C2)=O)=O)c(F)cccc1F C1(C(N(C(CC)COC)C)=O)CCOC1CNC(c1c[nH]nc1Cl)=O c1(C(N2CCN(C(C=NOC)=O)C(CS(C)(=O)=O)C2)=O)cnc2[nH]cnc2c1 c1(C(=O)NCCCN(C(=O)CC(=O)NC2CC2)CC)coc2cc(F)ccc12 C1(C2CCN(C(=O)CCc3cnc[nH]3)C2)(NC(C(CC)c2cnccn2)=O)CC1 c1(CSC)cc(F)ccc1NC1(c2nnnn2CCC2CC2)CC2COCC12 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)COC)ccc(C)c(S(N)(=O)=O)c1 c1(SC)ccc2cc(C(=O)NC3CC3NC(C3OCC4CCCC34)=O)[nH]c2c1 c1(C(N2CC(N(C(CC3C(C)C3)=O)CCO)C2)=O)nc(N)cc2ccccc12 C12(C(=O)NC(CCC(=C)C)C)C(NC(=O)CC3CCC(=O)N3)C3CC1C2C3 c1(C(=O)NCC(CC(C)C)NC(=O)COCC2CC2)ccc([N+](=O)[O-])n1C C1(C)(C(=O)NCCCCCCN(C(c2n(CC)ncc2)=O)C)CCOC(C)C1 c1(CN(C2N(C(C(C3CCCC3)OCC)=O)CCC2)C)ccnc(F)c1 c1(CNC(C2CC(NC(C3(F)CC3)=O)C2)=O)ccc2c(c1)CC2 N1(C(CCCCc2ccc(OC)cc2)=O)CCC(C2(NC(=O)CC3CC3)CC2)C1 C1(COC)(CNC(c2cc(C(N)=O)no2)=O)CCCN1C(=O)C(C)CC1CCC1 C1(CNC(c2csc(F)c2)=O)CC2(CC2)CN1C(c1cc(Cl)ccn1)=O C(C)(CC(=O)N(CCNC(C1(F)CCOC1)=O)C(C)C)SC C(N=c1[nH]c(=NCCOCC(F)F)c2c(F)cccc2[nH]1)c1c(C)cc(Br)cc1 Cc1cc(C(N2C3CN(Cc4ccc(-c5ccccn5)cc4)CC23)=O)c(C)[nH]1 N1(C(c2c(CC)ncs2)=O)CCC(NC(c2cc(C)c(F)cn2)=O)C(CO)C1 Cn1cc(C(N2CCC(CO)C(NC(=O)C3=COCCC3)C2)=O)c(O)nc1=O c1(C(N2CCC(NC(C3(COC)CC=CC3)=O)C2C)=O)noc2c1CCCCC2 c1(OCC(=O)NC(C)CCCNC(=O)C(C)CC2CCCC2)ccc(CO)cc1 Cc1sc(=O)n(CC(N2CC(N(C)C(c3cc(C)n(C)n3)=O)C3(CC3)C2)=O)c1C c1(C(=O)NC(CCN(C(c2cccc(C(C)=O)c2)=O)C)C)ccc(N=[N+]=[N-])cc1 N1(C(c2ccc(OC)nn2)=O)Cc2ccccc2C(NC(C2(F)CCOC2)=O)C1 C1(CC(N2C(C(C)NC(C3CC(F)(CO)C3)=O)CCC2)=O)CCC(F)(F)CC1 N1(C(CCc2onc(C)n2)=O)CCC(O)(CNC(c2ccc(N)c(F)n2)=O)CC1 C(=O)(C1=C(C)C(C)(C)OC1=O)NCC1CCCN(C(CS(=O)(=O)NC)=O)C1 c1(NC(=O)NC2C(c3onc(COC)n3)C2)cc(OC)c(Cl)cc1OC N1(Cc2cc(CC)no2)CCc2[nH]cc(I)c(=O)c2C1 c1(C(=O)NC(C2CN(C(c3cnc(S)nc3)=O)CCO2)C)ccc(F)c(F)c1O CCCC(C)(C)C(=O)N1CCCC(CCC(=O)NC(C)CN(C)C(C)C)C1 c1(C(N2CCC(N(C)C(c3snc(Cl)c3Cl)=O)C2)=O)nnn2c1C(=O)NCC2 C(=O)(C1CCC(=O)c2cccn21)NCC1N(C(c2cn(C)nc2)=O)CCCC1 c1(CN(CC(O)CO)C(=O)OC(C)(C)C)ccc(OCC(F)(F)F)cc1F C1(NC(CC2(CNC(c3ccc(C#N)cc3)=O)CC2)=O)CC2CC1C(O)C2O C1(F)(C(N2CCC(OCC=C)C2)=O)CCCN(C(=O)CN(C2CCCC2)C)C1 N1(C(Cc2cc(C)sc2)=O)CCOCC(NC(c2c(C)nn(CCO)c2C)=O)C1 C1(NC(=O)CN2CCCC2=O)CN(C(C2CCSCC2)=O)C2CC12 N1(C(C2(C)C(C)(C)C2)=O)CCOC(CC(N2CCC(OC(F)F)C2)=O)C1 N1(C(C2C3CN(C(CC(C)n4cccc4)=O)C2C3)=O)CCCN(C)CC1C N1(C(CC2(OC)CCC2)=O)Cc2ccc(NC(=O)C(C)n3cncn3)cc2C1 Cc1ccsc1CC(=O)NCCN(C(=O)C(CO)N1CCCCC1)CCOCCO c1(CC(=O)NCC2CCN2C(c2nc(Br)c[nH]2)=O)ccc(F)cn1 CCCCCC(C)CC(=O)N1CC2(CC(CC(=O)NCCC(C)SC)C2)C1 c1(NC(=O)NCc2cccc(C3CC3)c2)cc2ccccc2c(=O)o1 C1(C)(C(=O)NCC(C)Cc2cn[nH]c2)CC(O)CN1C(c1ccn(C(F)F)n1)=O c1(C(=O)NC2C(N(CCC(=O)NCc3ccccc3)C)C2)cc2ccccc2o1 c1(OC)ccccc1C(C)C(=O)NCC1CCN(C(=O)C(c2ccnn2C)C)C1 c1(C(N2C(C)(CC)CC(NC(c3scc(C)c3C)=O)C2)=O)cnn2ccccc12 C1(NC(CCCC=C)=O)CC2(C1)CN(C(=O)C(C)S(N)(=O)=O)C2 c1(NC(C2CN(C(C(C)c3ccco3)=O)C(C)(C)C2)=O)cnc2ccccc2c1 C1(CNC(c2cc(C)ns2)=O)CN(C(c2cc3ccsc3s2)=O)C2(CCC2)C1 N(C(=NCc1cc(C(F)(F)F)cs1)N1CCC(COC)C1)C(CC)C CCCC(C)(O)C(=O)N1CC(N(C(=O)CCc2ccccn2)CC)C(C)(C)C1 c1(CNC2CC2(Cl)Cl)c(CSC)oc2ccccc12 N(C(=NCCCCC(F)(F)F)NC1CC12CCCC2)CC1(SC)CCC1 C1(C)(C(N2C(CN(C(=O)CC3(COC)CC3)CC)CCC2)=O)CCC(F)(F)C1 Cc1ccc2c(C(=O)NCC3CCCN3C(=O)C(C)CC(F)F)ccnc2c1Cl N1(C(C(C=C=C)C)=O)CCC(C=C)(C(=O)NCC=Cc2ccccc2)CC1 c1(CN(C)C(C2(NC(=O)CCn3cnc(=N)[nH]3)CC2(C)C)=O)cn(C)cn1 N1(C(Cc2cnc(C)s2)=O)CCC(CNC(=O)C(C)C(F)(F)F)C12CC2 C1(C)(NC(C(C)C2CCCO2)=O)CN(C(C2CC3CC2C3)=O)C1 C=CC(C)(CCOC)C(=O)N1CCN(CCCNC(=O)CCC#CC)CC1 N1(C(c2ccc(CC)[nH]2)=O)CC(NC(=O)C(C)CC(C)CC)CC12CCOCC2 O=C(C1=CN2CCS(=O)(=O)N=C2C=C1)NC1CCN(C(=O)C2=CCCOCC2)C1 C=CC1OCCC1C(N1CCCCC1C1(NC(C2CCC2OC)=O)CC1)=O C1(NC(CN(C(C(C)OCOC)=O)C2CCC2)=O)CCn2nnnc2C1 N1(C(c2cc(C)oc2C)C(=O)NC(C(=O)OC)C)CC(C)(C)C1C1CCCO1 N1(c2[nH]c(=N)c3c(n2)CCC3)CCC(N=c2nc3scnc3c(N3CCC3)[nH]2)C1 N1(C(c2cccc(CC)n2)=O)CC2CC(NC(c3ncc(Cl)s3)=O)CC1C2 c1(C(=O)NCC=CCNC(=O)Cc2cccnc2)cnc(Cl)c(Cl)c1 C1(C(N(C)Cc2c(OC)cccc2)=O)CC2OCCC2N(C(=O)C=CCBr)C1 c1(C(N(C(CNC(COCCC#C)=O)C2CC2)C)=O)cn2c(n1)COCC2 C=Cc1cnn(C)c1C(=O)NCC1CCCCC1NC(=O)CCCC(=O)N(C)C CCC(CC)CCCC(=O)N1CC2OCC(NC(=O)CCc3cncn3C)C2C1 c1(C(N2CCC(CC)(NC(=O)C(C)CC(F)F)CC2)=O)cc2c(s1)CCSC2 C#Cc1cc(C(N2CC(NC(c3ccnn3C=C)=O)CC2C)=O)cc(Br)c1 C(=O)(CCC(=O)NN(C)C)N(CC(=O)NCCCC(C)C1CC1)CC#C C(=O)(CCCCC(C)=O)N1C(C(N2CC(CC)OCC2C)=O)CC(=O)C1 Cc1ncc2n1CCN(C(=O)C(CNC(=O)CC1CC(=O)NC1=O)CC(C)C)C2 C(CCC(C)(C)C(=O)N(CCCSC)C)NC(c1c(CC)cccc1)=O c1(C(=O)NC(CN(C(C2C3CCCC23)=O)CC)C)cc(OC)cc(Cl)c1O N1(C(c2c(OC)cccn2)=O)CCN(C(=O)Cc2ccccc2Cl)C(CO)C1 N1(C(=O)NC(C)C)CCOC(C(=O)NCCN(c2ccsc2)C)C1 C1(CS(N2CC3CC(O)CC2C3)(=O)=O)Oc2cc(F)ccc2NC1=O c1(N(C)C)cccc2sc(C(N3CCN(C)C4CC34)=O)cc12 Cc1ccn2cnc(C(=O)NCC3CN(C(=O)C(C)C(C)C4CCC4)C3)c2c1 c1(CC)ccccc1COC(=O)CC(C1CC1)NC(=O)C(C)(C)OCOC C1(NC(C2CC(C#N)C2)C)CC12CCN(Cc1ccc(F)c(O)c1F)CC2 C1(C(=O)NC(CCOC)CNC(C2CN(C(N)=O)C2)=O)(CC)CCC(O)CC1 CCCC(CCCNC(=O)CCC(CC)OC(C)=O)NC(=O)CCC1CCCC1 Cc1ccc(C(=O)NC(C2CC2C(=O)N(C)CC2CC2(F)F)C)cc1O C(=O)(C(F)CCC(C)(C)C)N1C2CC(C(N3C(CCC)COCC3)=O)CC1CC2 N1(C(C2CCN(C)C2)=O)CCC2(CCC(CNC(=O)CC(C)(C)C)CC2)CC1 N1(C(C(C)=C2CCC2)=O)CCCC(CC(=O)NCCC2(C)N=N2)CC1 C12CCCC(C1)C2=O.c12ccc([nH]1)CCC(=O)N2.C1(NC(C)=O)(CO)CCSC1 O(NC(=O)C(c1cn(C)nn1)NC(c1ccn(CC)n1)=O)C(C=C)C C(=O)(C#CC1CCOC1)N(CC(C(=O)NC1(CC=C)CC1)C)C N1(C(C(CC)N(C)C)=O)CCOC(C(=O)N(C(C)CCO)C)CC1 Cc1ccc(F)cc1C(=O)N(CCC(=O)NCc1ccccc1F)C1CC1 c1(C(N2CC(OC)(CNC(c3cc4ccsc4s3)=O)C2)=O)cccn2ncnc12 Cc1nn2ccccc2c1C(N1CC2(CCN(Cc3cnn(C)c3)C2)C1)=O c1(C(=O)NC2CC3(CN(C(C4C(C)(Br)C4)=O)C3)OC2)ccc(F)c2ccccc12 c1(C(=O)NC(C=C)CO)ccc(CNC(=O)C=CC2(C)COC2)cn1 C(=O)(C(CN=[N+]=[N-])NC(c1ccn(C)c1C)=O)NCCn1c(C)nc(C)n1 C1(CCC)CCC(C(=O)NC2CC(NC(=O)C(N3CCC(C)C3)=O)C(O)C2)CC1 N1(C(C(C)SC)=O)CCC(F)(C(=O)N(CC(O)C(C)(C)C)C)CC1 CCCCCC(C)(C)C(=O)NCC1CCCN1S(C)(=O)=O N1(C(C(NOC)=O)=O)CC2CN(C(c3cc4cccnc4[nH]3)=O)CCC12 c1(C(N(CCC(=O)NCc2nncs2)C)=O)cccc[n+]1[O-] CC1CN(C(=O)C=Cc2cscn2)CCC1CNC(=O)COc1ccc(F)cc1 Cc1cc(Br)cc(C)c1CNC(=O)NCC(C)(C)C(C)O C(=O)(C(C)(F)C(C)(C)F)N1C(C(N2CC(OCC)C2)=O)CC(=O)C1 c1(C(=O)NCC(COC)OC(C)C)ccc(CC(C)N)cc1 c1(OC)cc(C(=O)NCC(C)CNC(=O)CC2CCOC2(C)C)sc1Cl CC#CCC(C(=O)N(CC(O)CO)C)NC(C1CCCS1)=O C(=O)(CCCC(=O)NCC1(C)CCN(C(c2ncncc2Cl)=O)C1)N(C)C C1(NC(C2(C)COC2)=O)CC2CCC1N(C(=O)C#CC1CCOC1)C2 c1(C(=O)NC2CN(C(c3ncc(C)c(Cl)c3)=O)CC(F)C2)cn2cc(C)sc2n1 c1(C(N2C(CC)CN(C(C3CCC(=O)N3)=O)CC2)=O)cc2cc(C)ccc2o1 c1(CC)cc(C(=O)NC2C3CN(C(C4CC(F)C4)=O)CC23)cc(N)c1 c1(C(N(CC(CNC(C(COCC)C)=O)C)C)=O)c(C(F)(F)Cl)n[nH]c1C C(C(=O)N1CC(N(C(=O)COc2cc(C)on2)C)C(C)(C)C1)(C(C)(C)C)SC N1(C(C(CCC)C)=O)CC2(CCN2C(c2cnc(C)c(C)c2)=O)C1 c1(C(=O)NC2C(CNC(c3ccc(CS(C)(=O)=O)o3)=O)C2)cc(F)n(C)n1 c1(CC)cc(C(N2CCCC2CN(C(=O)C=C2CCSCC2)C)=O)no1 CCC1c2ccccc2CN1N1CC2CCCC2(CNC(=O)OC)C1=O.C(C)(C)(C)O CC1(CNC(c2ccnc(CNC(=O)C(O)C3CC3)c2)=O)CCCCCC1 c1(C(N(CC(C)CNC(=O)C(=O)C(C)(C)C)C)=O)ccc(N=[N+]=[N-])cc1 C1(CNC(c2c(CC)onc2)=O)CN(C(C2(Cl)CC23CCC3)=O)CCO1 C(=O)(C1=CC2C=CC1C2)NC1(C(NOCC=CC)=O)CCSC1 CCC(C(=O)OC)C(=O)N(CC(N1CCCC(COC)C1)=O)C1CC1 N1(C(C(=O)NC(c2cc(C(C)(C)C)on2)C)=O)CCCC(CN(C)C)C1 C1(NC(c2cc(CC)on2)=O)CCCC(NC(C2(C#N)CCC2)=O)CC1 N1(C(CN(C(C)C)C)=O)CC2C(C(=O)NC3CC(N(C)C(C)C)C3)C2C1 c1(C(=O)NC2(CC=C)CCCN(C(=O)C(F)C(C)C)C2)cc2c(C)sc(C)c2s1 C1(C(N(C(c2ncccn2)C)C2CC2)=O)CC1C1CN(C(=O)C=CC(=O)N(C)C)C1 c1(OC)ccc(Cl)c(CN=c2[nH]cc(-c3ccc(I)c(F)c3F)s2)c1Cl N1(C(c2c(CC)onc2C)=O)CC2CCC2(CC(=O)NC2CCC(O)C2O)C1 c1(NC(=O)CC2CC23CC3)ccc(S(=O)(=O)Nc2ccccc2)cc1 Cc1nn2c(c1CNC(c1cnnn1C)=O)CN(C(=O)Cc1cncn1C)CC2 c1(CCC(=O)NCCN(CCC)C(c2cc(C)sn2)=O)c[nH]c2cc(C)ccc12 Cc1ccc(C2CN(C(C3CCCN(Cc4cnc(O)o4)C3)=O)C2)c(F)c1F CC1=NOC(CCNC(=O)CCOCCN(C)C(C2CCS2(=O)=O)=O)C1 N1(C(C2(OC)CC(C(C)(C)C)C2)=O)CCCC(C2(NC(C)=O)CC2)C1 Cc1ccc2[nH]nc(C(N3C4CCC3CC(CCNC(=O)CNC=O)C4)=O)c2c1 C1(CN(C(=O)C=CC(F)(F)F)C2CC2)CCCN1C(=O)Cc1cc[nH]c1 c1(OCC(NNC(Cn2cc(OC)c(=O)cc2C)=O)=O)ccc2ccccc2c1 n1(CC)cc(Br)cc1C(N1CCC1CNC(C1C(C)CC1C)=O)=O C1(CN(C)C(C2CCOC2)=O)CCCN(C(c2occc2F)=O)C1 CC(C)CC(CNC=O)CC(=O)NC1CC(CNC(C2CCC(=O)C2)=O)C1 N1(C(C(C)C(C)NC(=O)CCc2cccnc2)=O)CC(=O)NC(=O)C1 c1(OC)cc(C(N2CCC(=CC(=O)Nc3ncco3)CC2)=O)ccc1F C1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)N3)=O)C2)CCC2CCCCN12 CCCCC(C)(F)C(=O)N(CCC(C(C)(C)C)NC(c1c[nH]nc1Br)=O)C c1(N2CC(C)(C)NC(=O)C2)nc(NC2CCC3(C2)CC3(F)F)c2ccsc2n1 C1(C)(CC)C=C(C(=O)NC2CC(NC(=O)COC3CCC3)CC2O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CC(NC(CCN(c2ccccc2)C)=O)C1 Cc1cc(C(=O)NC(C2CCCN(C(=O)C(C)(C)F)C2)C)c2cnccc2c1 c1(CNCC(N2C(C)(Cc3ccccn3)C=CC2)=O)cc(O)n2nccc2n1 c1(C(N2CC(CNCc3ccc(C)cc3Br)OCC2)=O)cccc2cn(C)nc12 N1(C(C(C(CC)O)(F)F)=O)CCN2CCN(C(c3cncc(F)c3)=O)CC2C1 c1(CC(=O)NCC2C(C)CN(C(C3CC4CC4C3)=O)CC2)ccc2nn[nH]c2c1 CC(C)(O)C(C(=O)N)NC(=O)C(=O)NC1CCNCCC1CO c1(CNC(C(C(C)(C)C)NC(=O)OC(C)(C)C)=O)nc(=NCC(C)C(C)C)cc[nH]1 N1(C(CSCC)=O)CCOC(CN(C)C(c2c(Cl)n[nH]c2C2CC2)=O)C1 CCC(C)(CNC(=O)COc1ccccc1)C(=O)N(CC(C)SC)C c1(C(N(C2CCCC(NC(c3c(C)snn3)=O)C2)C)=O)cnc2c(c1)CCCO2 c1(C(=O)NCC2C(C)CN(C(=O)CN(C)C)C2)cc(Cl)c(Cl)cc1O N#CCC(C(=O)N1CCOCC1CCNC(C1(C2CC2)CC1)=O)c1ccccc1 CCC(O)C(C)C(=O)NC(C)CC(C)NC(c1ccc(-n2cnnn2)c(C)c1)=O C1(CC(=O)NC2C(C)(C(=O)OCC)C2)CCC(NC(=O)OC(C)(C)C)CC1 c1(OC)ccc(Br)c(NC(=O)CC2CN(C(c3cnco3)=O)C2)c1 C12(C(=O)NCC(C)(CC(C)C)NC(C(C)=CC3CC3)=O)CCOC1CC(=O)NC2 c1(C(N2C(CNC(C(CC)C#N)=O)CC(OC)C2)=O)cnc(C(F)(F)F)c(F)c1 N1(C(c2c(C)c(C3CC3)on2)=O)CCCC2C(NC(c3csnn3)=O)C(C)(C)C12 c1(CC(=O)NC(CCCNC(C2CCC(=C)CC2)=O)C)ccc(O)c([N+](=O)[O-])c1 N1(C(C(C(C)O)(F)F)=O)CC2(COC(CNC(c3cc[nH]c3C3CCC3)=O)C2)C1 C(=O)(C1CCCn2ccnc21)N(C)CC1(NC(=O)CCS(C)=O)CC1 Cc1nc2c(C(N3CCC(O)(CCNC(=O)C=CC(F)(F)F)C3)=O)cccc2o1 CC(C)CC(O)C(C)C(=O)N(C(C)C(N1CCC(N=[N+]=[N-])CC1)=O)C1CC1 N1(C(c2ccn(CC)c(=O)c2)=O)CC2CCCC(C1)N2C(=O)CN1CCCCC1 c12ccccc1COCCOC2=O.N1(CCCOCCC)CC=CC1.C1(=O)CS1 CCC(O)C(C)C(=O)N1CCCCC(N(C(=O)CC2(OC3CCC3)CCC2)C)C1 c1(C(N(C(C(=O)N(CCOC)C)C2CC2)C)=O)csc(C)n1 c1(C(=O)NCc2cccc(NC(c3c(C)n(C)nc3)=O)c2)ncnc2c1CCC2 c1(CC(=O)NC2C(CNC(CCS(C)=O)=O)CC2)ccc(Cl)cc1F CC(C(=O)NC1CC(CNC(C2CCN(C(N3CCCC3)=O)CC2)=O)C1)S(C)(=O)=O c1(CC)ccccc1C(=O)NC1CC(CNC(c2ccn(C3CC3(F)F)n2)=O)C1 c1(C(CF)NC(=O)NC2C(=O)OCC2CO)cccc(F)c1F N1(C(C2(F)CN(C(CC(CC)CN(C)C)=O)C2)=O)CC(C)(C)CCC1C c1(C(=O)OC)ccc(C(=O)NCC2CC2CNC(c2cc(C)n(C)n2)=O)cc1F c1(C(=O)NCC2(CN(C)C(C3CS(=O)(=O)C3)=O)CC2)cnc(O)c2ncccc12 CC(C)CCC(=O)NCCC1(CNC(=O)CC2CCC(C3CC3)O2)CC1 C(=O)(C1CCc2ccc(Br)cc21)NC1C(C)CN(C(=O)Cc2ccon2)C1 c1(OC)cncc(C(N2CCC=CC2C(=O)Nc2conc2C(C)C)=O)c1 Cc1cc(C(F)F)ncc1C(=O)NC1CCN(C(C2CCO2)=O)CC1F CCC(F)(F)CCN=c1[nH]c(=NC(C)c2snnc2C)[nH]c2c1CCC2 C#CC1(O)CC(CNC2CCCNC2CC)C1 CC1COc2c(C(N3CCN(C(c4ccc(O)cc4)=O)CC3C)=O)cccc21 C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(C2CC(CN(C)C)C2)=O)CC1C n1(CC(=O)NCC2C(CNC(c3nnc(C)s3)=O)C2)ccccc1=O Cc1cc(C)c(C(=O)NCCC2CN(C(c3[nH]cnc3C#N)=O)CCO2)s1 c1(C(=O)NCC(C)NC(c2c(C)cco2)=O)ccc2c(=O)ccoc2c1 Cc1oc(C(N2CC3CC2C3NC(=O)CC(C)CC(F)(F)F)=O)cc1S(N)(=O)=O N1(C(CC2CC(NC(COCCC)=O)C2(C)C)=O)CCOC2CCC12 C=CCC(C)(CC)C(=O)NCCC1(CNC(=O)CC2(C)CCCO2)CC1 CCC(C)C(O)C(=O)N(C)CCOCCNC(C1CCN(C(C)=O)CC1)=O C(=O)(CC(CC(N)=O)CC(C)C)NC1C(NC(C2(C#C)CC2)=O)CCCC1 N1(CC2(O)CCN(Cc3ccncc3)C2)CCC(F)(F)CC1 N(C(=NCCc1cc(Br)ccc1OC)NCC1(CO)CCCC1)C(CC)C N1(C(C(CC#C)(C)NC(c2cnc(Cl)n2C)=O)=O)CCCC2(CCC2)C1 C1(CC(=O)NC(Cc2cn[nH]c2)C(=O)NCC(N2CC=CC2)=O)CCCCO1 N1(C(c2cnc(C(C)C)o2)=O)CC2C(C(=O)NC3CCN(C(C)C)C3)C2C1 C1(CC)CC(C(=O)NC2CC23CC(OC)C3)CCN1C(c1ccc(C(N)=O)[nH]1)=O c1(C(C=C)C)nc(-c2ccc(N(CC)CC)cc2)nn1-c1ccnn1C N1(C(C)=O)CCCC1CNC(C1CCC(CNC(=O)COCCC(C)C)C1)=O C(=O)(C1=CCC(C)(C)CC1)C(C(C)CNC(=O)N(C1CCCCC1N(C)C)C)=O c1(SC)nc(O)nc(C)c1C(=O)NCC1CN(C(=O)CCC2OCCO2)CC1C C1(N(C(CN(CC)CC)=O)C)CN(C(c2ccc(OC)cc2Cl)=O)CCC1C C1(C(=O)NC(C)CNC(c2cnccn2)=O)CC2C=CC1O2 N1(C(c2nc(C(C)C)sc2)=O)CCC(OCCNC(=O)C(C)C2CCC2)CC1 CC1CC=C(C(=O)NCC23CC(CN2C(c2ccc(N(C)C)cn2)=O)C3)CC1 N1(C(C(c2ccccc2)NC(c2n(C)ccn2)=O)=O)CC(O)CC(O)C1 N1(C(C2(OC)CCOCC2)=O)CC2CN(C(=O)C=Cc3ccc(OC)o3)CCC12 N1(C(c2ccc(C)nn2)=O)CC2CN(C(C34CCC(C)(CC3)CO4)=O)CC2C1 c1(CC(=O)NC23CCCC2N(C(c2ccsn2)=O)CC3)ccc2c(c1)OCCO2 N1(C(c2c(CCC)nco2)=O)CC2CCC1CN2C(C1(OC)CCC(C)C1)=O C1(NC(CC(=C)Br)=O)CC2CC1CN2C(=O)Cc1c(OC)cccc1F CCCCC(CCCC)NC(C1(C)CC(O)CN1C(c1ccc(O)nc1)=O)=O N1(C(C(Cc2ccc(Cl)cc2Cl)NC(=O)OC(C)(C)C)=O)CCCC(F)(F)CC1 n1(CC#N)ccc(=NC(=O)C2C3CCCC3CN2C(=O)CN2CCCCCC2)[nH]1 N1(C(CCNC(c2c(C(=O)OC)coc2)=O)=O)CC2CC2C(OC)C1 N1(C(CC(=C)C)=O)CCCC(n2cc(CNC(C3CCOC3CC)=O)nn2)C1 C1(C(NOCC)=O)CCN(C(c2cc(C(C)=O)[nH]n2)=O)C1C.c12cn(nn1)C2 CC1C(NC(=O)CCCC(N)=O)CC2CCC1N2C(=O)CC1(CO)CCOCC1 N1(CCN(C(c2c(CC)nc[nH]2)=O)C)CCN(C(=O)CC2(OC)CC2)CC1 Cc1cn2ccc(C(=O)NC3C=CCN(C(C4(C)CC(O)CN4C)=O)C3)cc2n1 c1(C(N2CCC(C)(CCNC(C3ON=C(CC)C3)=O)C2)=O)cccc2nncn12 C1(C(=O)NC2CCC(C(C)C)CC2)(NC(CNC(=O)OC)=O)CCCSC1 C1(NC(C2N(CCC)CCC2)=O)CN(C(=O)C=Cc2cnn(C)c2)CC2(CC2)C1 c1(NC(=O)NC)ccc(Cl)c(C(=O)NC2CC2CNC(c2ncccc2Cl)=O)c1 C1(C(=O)NCC(=O)Nc2c(F)cccc2F)CCc2ccccc2C1 c1(C(=O)NCC(O)CNC(c2cc(F)c[nH]2)=O)ccc2c(c1)OCCCO2 Cc1cc(C(=O)N(C(c2ccc(Br)cc2)C(N)=O)C)nc(-c2ccccc2)n1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(=O)C(O)C(C)(C)C)C12CC2 c1(C(N2CCC3CN(C(C=CC)=O)CC3C2)=O)cc(Cl)cc2ccncc12 c1(CC)cnc2ccccc2c1C(=O)NC1CC(NC(c2cc(C)ncn2)=O)C1 c1(C(=O)NC2CC(CNC(c3nccc(OC)c3)=O)C2(C)C)cc(C)n(C)c1C c1(OC)cc(C)nc(N2CCC(C)C(NC(=O)C=Cc3cncnc3O)C2)n1 CC1CCCC(CC(N2CC(CNC(=O)CCCCNC(N)=O)CC2C)=O)C1 c1(NC2CCN(c3snc(C)n3)CC2)cc(NC2CCS(=O)(=O)CC2)nc(C)n1 CC(CCC(C)(C)C)C(=O)N1CCC1C(=O)NC1CC12CCCC2 c1(N2CC(NC(C3CC(=O)N3)=O)C(O)C2)ncnc2n[nH]c(Br)c12 C1(NC(C(CC)(C)C)=O)CN(C(C2CCC=CCC2)=O)CCC1C C1(NC(CNC(CCC(C)C)=O)=O)CCN(C(C2(C)CCCO2)=O)CCC1(F)F Cn1ncc2c1CN(C(c1c(C3CN(CC4C5CC6C(C5)C46)C3)cnn1C)=O)C2 N1(CC(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)CCC(=O)NC1=O N1(CCCCC)CCC2(CN(C(C3CCCOC3)=O)CC(C)O2)C1 c1(C(c2n(CC)nnn2)NCCC(C)COC)ccc(F)cc1 N1(C(CCCN(C)C)=O)CCCC1(C)CCC(=O)N(C)CC1(CO)CC1 Cc1cc(=O)c(C(=O)NC(C)(CNC(c2sccc2C)=O)CC(C)C)cn1C C1(CCNC(C(=O)NC2C(C)(C)C2)=O)CC12CCCCC2 c1(C(=O)NCC(F)F)ncn2ccccc12.c12ccc(cc1)[nH]2 C1(NC(=O)CNC(=O)C2CC2)CC2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC12 c1(NC(c2cc(C)nn2C(F)F)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(CNC(C)=O)=O)CCCC(N(CCO)Cc2ncnn2C2CCOCC2)C1 C(=O)(C(C)(C)C(F)F)NC1C(CNC(c2c(C)n(CC3CCCC3)nn2)=O)CCC1 Cc1ccc(C(=O)NCCC2CCC(NC(=O)C3=COCCC3)C2)c(C)c1 C1(N(C(=O)CCN2CCC(F)C2)CC#C)CCN(C(C2COCCOC2)=O)CC1 N1(C(c2cc(CC)nn2C)=O)CCOCC(F)(CNC(C2CC2CC)=O)C1 c1(-c2n(CCN(C)C)nc(-c3cc(F)cc(F)c3)n2)n[nH]c2c1COCC2 c1(CNC2(c3n(CCOC)nnn3)CN(C3CC3)CC2C)ccc2sccc2c1 c1(OC)ccc(Cl)c(C(=O)NC2CN(C(C3(C)CC(O)CN3C)=O)C2)c1F O=S(=O)(c1ccc(Br)cc1F)NC1CCC(Nc2ncnc3sccc23)C1 c1(C(=O)OC)cc(F)cc(F)c1NC(C1CSCCN1Cc1cccs1)=O CC1(C)CCCCC(C(=O)NCCCC2CC2(F)F)C1 C1(NC(c2c(C)oc(CO)c2)=O)CC(C(=O)N2CCCC(F)(F)C2)=CC1O CC(C)(O)CC(C)(C)NC(=O)CCCCCNC(=O)CC1CCC(C)(C)C1 C1(NC(c2noc(CC)c2C)=O)CC2CN(C(=O)C3=NOC(C)(C)C3)CC2C1 N1(C(Cc2nc(CC)sc2)=O)CC2(NC(=O)C(CC)N(C)C)CCCC2(F)C1 C1(COC)CN2CCN1C(=O)CCCC2=O.c1(C(=O)NC)sc(Br)cc1F N1(C(C(C)OCCCCCC)=O)CCC(NC(C2(COC)CCCC2)=O)C(F)C1 c1(NC(C(c2cccc(Br)c2)(C)N)=O)ccc(S(F)(F)(F)(F)F)cc1 C=CCC(CNC(=O)C(C)=CCN(C)C)NC(C1CCCN1CCC)=O C1(C(N2CC(CNC(Cc3c(OCC)ccc(Cl)c3)=O)C2)=O)CCC2(CCC2)OC1 c1(CC(=O)NC2C(C)N(C(=O)C(C)O)CCC2)cc(F)c(F)cc1F c1(C(=O)NCCCN(C(=O)Cc2cnc(C)s2)CC)c(F)ccc2[nH]ccc12 CCC(C)C(C)C(=O)NCc1ccc(C(=O)NCC(C)(C)C2CCC2)o1 N1(C(C2(C)COC2)=O)CC2CCC1CN2C(c1cccs1)=O N1(C(C(C)N2CCCC2)=O)CCCCC1CN1CCCC2(CC2)C1 c1(C(=O)NC(C2CCN(C(C(CC)OC)=O)CC2)C)cc(N)cc(O)c1C c1(OC)cc(O)c(C(=O)NC2CN(C(=O)CCNC(C)=O)CC2C#N)cc1OC C1(NC(CCC2CCCN(C(C(C)(C)CC3CC3)=O)C2)=O)CC(C)(C)OC1(C)C n1(CC)cccc1C(=O)NCCC(C)NC(c1ccncn1)=O N12CC(CC(NC(=O)CCCSC)C1)OCC2=O.CCS(=O)(=O)N(C)C(C)C N1(C(C(Cc2ccco2)OC)=O)CC2CCCC2(NC(C2CC2(F)Cl)=O)C1 CC(C)(CC(=O)N1CCCCC(CNC(=O)Cc2ccc(O)nc2)CC1)C(C)C C(CN(C)C)(CN=c1nc(N(C2CCCCN2C)C)c2c([nH]1)CCOC2)OCC C1(NC(Cc2c(C)cccc2)=O)CCCCC12CCCN(C(C1C=C1C)=O)C2 C=CCC(CNC(c1cnoc1-c1ccccc1)=O)NC(C1(C)CC1)=O Cc1cc(C)c(CNC(=O)C(=O)N(C2CCN(c3cccnc3)CC2)C)s1 C1(CC=C)CCCC1N=c1[nH]c(N2Cc3ccccc3C2)nc2ncn(CC)c12 c1(SC)cc(C(N2CC(C(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)c(C)o1 C12(C(=O)NC(C)CNC(=O)Cc3nc(=N)[nH][nH]3)CC(CC(C)O1)C2 CC1CC(C(=O)N(C2CCN(C(=O)CSC(=N)N)CC2)CC2CC2)CCO1 N1(C(C(CCSC)O)=O)CCC(CC(F)F)(CO)CC1 N1(C(C(C)(F)F)=O)CCC2(CC1)CC2NC(=O)CN1C(=O)CNC1=O C(=O)(C(F)(F)C(O)CCCCCCCCC)N(C(C#C)(C)C)C CC1(C)CN(C(=O)CCc2ccoc2)CC1CNC(=O)CSC1CC1 N1(C(CCCC#CC)=O)CCCC2CN(C(=O)C(C(C)(C)C)n3ccnn3)CC12 c1(NC(C2CCCN(Cc3cccc(OCC)c3O)C2)=O)c(C)cc(O)cc1O N1(C(C=CCOC)=O)CC(CNC(=O)CCSCC(C)C)OC2(CCC2)C1 CN1C2CCCC1CN(C(C1CC1C1CN(C(c3coc(C4CC4)n3)=O)C1)=O)C2 c1(NC(=O)NCCN(C)Cc2ccc(C#N)cn2)cn2ccc(Cl)cc2n1 C(=O)(CC(C(F)(F)F)NC(=O)C(C)NC=O)NC1(CNC(COC)=O)CCC1 C(CCNC(C1CC1(C)Br)=O)(C(C)C)NC(C(CC)n1nccc1C)=O C1(C(N2CC(C)OCCC2)=O)CC2CCCC2N1C(=O)CCc1nncs1 c1(NC(C(=O)NC(CC(=O)OC)Cc2cccc(F)c2)=O)cccc([N+](=O)[O-])c1 c1(CC(=O)NC2(CNC(C3(CCC)CCC3)=O)CC2)ccc(OC)c(Br)c1 c1(-n2cc(CNC(C3C(C(=O)OC)C3)=O)nn2)cc(F)cc(F)c1 c1(OC)c(Cl)nc[nH]c1=NCC(C)(C)NC(=O)C1Cc2ccccc21 C(CN=c1ccc(-c2cccc(OC)n2)c[nH]1)Nc1cc(OC)ncc1 N1(C(CC2(OCC)CC2)=O)CCCC2(CCCN2C(C2(C3CCCO3)CC2)=O)C1 Cc1ccc(-c2cccc(-c3nc(COc4ccc(C)cc4C)no3)c2)c(C)c1 C1(CC)C(C(=O)NCC2CCC2(F)F)CCCN1C(=O)CCC1CC1(F)F c1(C(N2CC(CNC(CC(C)OC)=O)C3(C2)CC3)=O)cc2ccccc2o1 Cc1nc(CCC(=O)NC(C2CN(C(C3(C)CC3(F)F)=O)C2)C)oc1C c1(CC)ncoc1C(=O)N(CCCNC(C1CCCO1)=O)CC1CCCC1 Nc1cc(F)cc(Cl)c1C(=O)NCC1CN(C(=O)C2=CCS(=O)(=O)C2)CCCO1 N1(Cc2cc(C)[nH]n2)C(C(N2CCC(Nc3ncccn3)C2)=O)CC2CC12 C(=O)(C(C)CC(C)(C)C)N(CCNC(c1c(C)n(CCO)cc1)=O)CCOCCO C1(CNC(C2(CC#C)CCCC2)=O)CN(c2nc(Cl)ncc2F)CCN1C C1(CN(C(C(C)OC)=O)C)CCN(C(C2CC2C(F)(F)F)=O)CC1 n1(CC)cc(NC(=O)CC2CCCN(C(C3CC3C(N)=O)=O)C2)c(C)n1 C1(C)(C(N2CCC(O)(CNC(c3cncc(CC)c3)=O)C2)=O)COCC1(F)F C(=O)(C(C)Cc1cnc[nH]1)NC(C(n1cc(CCN2CCOCC2)nn1)C)=O C1(NC(C(CC)NC(C)=O)=O)CC(F)CN(C(=O)C(CC)(CC)c2ccccc2)C1 CC(C(=O)N1CCCC(CCC(=O)NC2(C3CC3)CC2)C1)C(C)(C)C CCC(C)CC(C)C(=O)N(C1CCN(C(C2CC23CCCC3)=O)CC1)CC1CC1 Cc1cn2c(n1)C(C)CC(C(=O)NCC(C(C)(C)C)NC(c1ncn(C)n1)=O)C2 Cc1cc2[nH]c(C(=O)NCC3(F)CCN(C(c4cc(Cl)ccc4O)=O)C3)cc2s1 C=CC(C)(CC)C(=O)N1CCCC(CCNC(=O)CC2CC(C(F)F)C2)CC1 c1(CONC(c2cccc(C3CC3)c2)=O)c(Cl)cccc1[N+](=O)[O-] c1(C(N2CCC(O)(CNC(C34CCC(C3)C4)=O)C2)=O)ccc(Cl)cc1Cl C#CC12CC(CN1C(=O)NCc1ncc(-c3cccc(F)c3)s1)C2 c1(C(N(CC(=O)N(CCOCC)C)CC(C)C)=O)cc[nH]c2nccc1-2 c1(C(N2CC(C(C)NC(c3cc(C(C)C)[nH]n3)=O)C2)=O)ccnc2c1CC(=O)N2 Cn1cc(C(N2CC(CNC(=O)C(=O)NCC3CC3)C(F)(F)C2)=O)c(O)nc1=O C1(CNC(C(CC)O)=O)(NC(c2ccc(C(N)=O)nc2)=O)CCOCC1 C1(OC)CC(CNC(C2CC2(C)C(F)F)=O)N(C(=O)CC2CC=CC2)C1 N1(C(CCC#CC)=O)CC2(CCCC(CNC(=O)Cc3ccc(F)cc3C)O2)C1 N1(C(C(C(C)C)C(C)NC(=O)CC23CCC(CC2)C3)=O)CCC2CCC(C1)N2C c1(C(c2n(CCCOC)nnn2)NC(C)CCCCSC)c(F)cncc1F C1(C(=O)N(CCNC(C2(CC(F)F)CC2)=O)C2CC2)CC2CCCC2C1 N1(C(c2c(C)ccc(F)c2)=O)CCC2CC2(C(N2CC(N3CCCCC3)C2)=O)CC1 N1(C(C2(NC(C(c3cncnc3O)C)=O)CCSC2)=O)CCCCCCC1C N1(CCNC(COCCCCC)=O)CCC(N(C)CC(C2CC2COC)=O)CC1 CCCCCC(C1CC1)NC(=O)C(CC1CC1)NC(c1nocc1Cl)=O C(=O)(CCCCCNC(=O)C(C)(C)O)NC1(CCC)CCNC1=O C(=O)(C1(C)Cc2cccc(Cl)c21)NC(CNC(C1CCN(C)C1)=O)(C)C CCC(C)C(O)CC(=O)NCCN(C)C(c1cnc2c[nH]nc2c1)=O Cn1nnc2c1C(C(=O)NC1CCCC1NC(=O)C1=CSCS1)CCC2 C1(C(N(C2CCN(C(=O)CCn3cccc3)CC2)C)=O)CCCC2(CC2)C1 c1(C(N(CC(CC)NC(=O)CCc2ccccc2O)CC)=O)cnc(O)cc1C C12(NC(c3cccnn3)=O)CCCC1N(C(c1cncc(O)c1)=O)CC2 N1(C(CCC)=O)CCN(CC(C)NC(=O)C(C)(C)n2ccnn2)CC1 c1(OCC)ccc(-n2nc(-c3ccccc3Cl)nc2C(c2cnn(C)c2)C)cc1 C(C)(CCNC(=O)C(=O)NCC(F)(F)F)NC(COC)=O C1(NC(C(c2ccc(C(F)(F)F)s2)N(C(C)COC)CCOC)=O)CC(F)(F)C1 N1(C(CC(CC)C2CC2)=O)CC2CN(C(C3(NC(C)=O)CCC3)=O)CC(C1)O2 C1(C(N2CC(C)C(CC(=O)N(CC(N3CC=CC3)=O)CC)C2)=O)CCC(C2CC2)C1 C(=O)(C(O)CCC(C)C)NCC1CN(C(CCCC=C)=O)CC12CC2 N1(C(c2cnn(C=C)c2N)=O)CC2C=CC1C(C(=O)NCC(F)F)C2 N1(C(c2sc(C)c(C)c2C#N)=O)CC(N)CCc2ccccc21 c1(N(CC(=O)OC)C(=O)NC(COC)Cc2ccc(Br)cc2)ccc(Cl)cc1Cl O=C1CCC2(CC1)CC2C(N1CC2CCC(C1)N2C(=O)C=Cc1ccco1)=O c1(C2N(c3ccnc(C(C)(C)C)n3)CCC2)cccc(P(C)(C)=O)c1 c1(C(=O)NC23CC(NC(c4nc(CC)sc4)=O)(C2)C3)ccc2c(c1)COC2(C)C c1(C(=O)NCC2N(C(c3cc(CC(C)C)on3)=O)CC2)ccccc1F N1(C(CCNC(COC)=O)=O)CC(C(C)NC(=O)C(C)OC)C1 C1(C)(CC)CC(NC(c2cn(CCNC(C3(N(C)C)CCC3)=O)cn2)=O)CCO1 CCC(CCC(=O)N1CC(c2ccccc2)(NC(C2C=CCC2)=O)C1)OC c1(OC)ncc(C(N2CCC(C)(NC(c3cn(C)ccc3=O)=O)C2)=O)cc1Cl N1(C(C(C2CCC2)OC)=O)CCCCC1C1CCCN(C(C2(C(N)=O)CC2)=O)C1 CCC(C)CC(=O)N(Cc1cccs1)CC1COCCC1C(=O)Nc1ccccc1 CCC(CC)C(C)C(=O)N(C1CCCN(C(C2(O)CCC2)=O)C1)CC C(CC(C(=O)NC1(C)CCCC1C)NC(c1ccc(N)cn1)=O)SC CC1(C)C(=O)NC2CCC(C(=O)NCC(O)CN=c3cc(F)nc[nH]3)CC12 C1(CC=C)(C(=O)NCCN(CCC(C)C)C)CCN(C(C2CCSCC2)=O)C1 C1(NC(C2(C)CCCC2)=O)CC=C(C(=O)N2CC(OC(=N)O)C2)C1 c1(COC)ccc(C(=O)NC2(CCCNC(=O)C(n3ccc(C)n3)C)CC2)s1 N1(C(CCOCCC)=O)CCN(C(=O)CNC(=O)OC)CC1C1CCCC1 C1(C(=O)NC2(C3N(C(COC(C)(C)C)=O)CCC3)CC2)CCc2nncn2C1 c1(C(N2CCC(C)C2CNC(=O)Cc2cccc(F)c2O)=O)cc(O)ncc1F C1(C(=O)NCC2C(N(C)C)COC2)CN(C(C2CCCC2C2CC2)=O)CC1(F)F CC1(C)OC2(C(=O)NC3COC4(CCN(C(c5cnco5)=O)C4)C3)CCC1CC2 CCC(C)CCCCC(=O)NCCC1CCCN(C(c2cnc(COC)[nH]2)=O)C1 c1(C(=O)NC(C)CC2CN(C(C3(C(N)=O)CC3)=O)C2)nccc2cccnc12 C(CC(C)C)(C(=O)NC(CCO)C(C)C)N(C)Cc1ccc(CC)s1 c1(C(=O)NCC(C)CN(C)C(C2CC2C(F)F)=O)cncn1C C1(NC(=O)CCc2ncc[nH]2)CCCC12CN(C(C13CCCC1CCC3)=O)C2 C1(C(N(CCOCCCNC(CC=CCCCCC)=O)C)=O)CCNC(=O)C1 O=C(N=c1[nH][nH]c2ccc(F)cc12)c1cc(F)c(F)cc1Br N1(C(=O)NC2C(C)(C)COCC2)CCc2c(c[nH]c(=N)c2C#N)C1 N1(C(c2n(CC)cnn2)=O)CCCN(C(=O)CCCc2cc(C)no2)C(CO)C1 Cc1ncnc(C)c1OCC(=O)NCC(C)(C)NC(c1ccsc1C#N)=O C(CC(C)C(=O)NC1CCCC1CNC(=O)CSCC(C)C)=CC c1(C(N(C2CCN(C(c3cc(COC)on3)=O)CC2)CCC)=O)cc(=O)cc[nH]1 c1(C(=O)NC(c2ccccc2)C(C)NC(C=C=C(C)C)=O)cnc(C)c(C)c1 C12(C(=O)NC3CCN(CCNC(=O)CCC4CCCCC4)CC3)CCCC1CCC2 CC1CN(C(C2(c3ccccc3)CCCN2)=O)CC1CC(=O)O C(=O)(CCC(C)(C)C)NC1C2CN(C(c3c(CC)nccc3)=O)CC21 N1(C(C2(C#C)CC2)=O)CCN(CCNC(=O)CC(c2ccccc2)OCC)CC1 c1(NCC2(Cl)CC2)nc2c(c(=NC3CCN(c4ccccn4)C3)[nH]1)SCC2 N1(C(CC)=O)CCC2(CC1)CC2C(=O)Nc1cc(O)ccc1CC N1(C(CCc2nc(C)c(C)o2)=O)CCC2(CC2NC(C2CC2C(N)=O)=O)C1 C1(c2noc(C3(C45CC6CC4C5C6O)CC3)n2)(CO)CCC(F)(F)CC1 CC(C)(O)C(F)(F)C(=O)N1CC2(CCNC(=O)COC3CCC3)CCC1CC2 C1(NC(=O)C(N2CCC(F)(CF)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC2CCCC(CN(C(=O)C3=COCC3)C)C2)cc(F)cc(F)c1 c1(C(=O)NCC(CCCC)NC(C2OCCN(C)C2=O)=O)ccc(C)cc1Cl Cc1ccc(C)c(C(=O)NC2CCN(C(c3ccc(Br)cc3)=O)CC2O)n1 Cc1ccccc1CC1CCCN1C(=O)C(=O)NCC(c1cncn1C)O c1(CC)ccc(C)cc1C(N1CC(CC(C)NC(=O)CCN2CCCCC2)C1)=O C(=O)(C(C)(CC)CCC)N(CCC)CCNC(C1CC(=O)N(O)C1)=O N1(C(COCC#C)=O)CCC2CN(C(=O)C(CC)n3ccnc3)CC2C1 N1(C(=O)Nc2cccc(SCC#C)c2)CCC(C)OC(C)C1 N1(C(C)=O)CCCCC1C(=O)NCCN(C(c1c(O)noc1C)=O)C1CC1 C1(CN(C)C)CCCC1NC(C1CCC1NC(=O)CN1CCCC1)=O CC1(C)C(NC(c2nsnc2O)=O)CC1CC(=O)NC1CCOCC1F CC1(C)CC2(CC(N=c3[nH]c(=NCNC4CCC4)[nH]c4ccc(C(N)=O)cc34)C2)C1 C#CCC(CC(=O)NCC12CCC(CC1)O2)NC(c1c[nH]nc1[N+](=O)[O-])=O C12(CC3(CC3)C1)C(=O)NC2.c1(C(=O)CC2CN(C(=O)OC)C2)cc(C)n(C)n1 O=S(=O)(c1ccc(NC2CCCC3(C2)OCCO3)c(F)c1)NCC1CCCCS1 c1(C(c2n(C(CC)C)nnn2)NCc2cccnc2)cc(C)oc1C N1(C(CC=CC)=O)CC2CN(C(=O)C=Cc3ccoc3)CCC2(CO)C1 C1(C(=O)NCC2N(C(CC(CC)CC)=O)CC(F)(F)C2)CCc2nnn(C)c2C1 N1(C(C(COCC)NC(=O)CC(C)(O)COC)=O)CCC12CCCSC2 N1(C(CCn2cc(CCCS(N)(=O)=O)nn2)=O)CCC(F)(CC#N)CC1 C1(N(C(C=C(CC)CC)=O)C)CCN(C(C2(C(F)F)CC(O)C2)=O)CC1 n1(CCC(=O)NCC2N(C(C(C(C)(F)F)F)=O)CC2)nc2ccccn2c1=O C12CCCC1NC2=O.C(CC(OC)OC)NC(C1(C(=O)OCC)CC1)=O c1(C(N(CCN(C(c2ccc(Cl)s2)=O)CC)CC)=O)cnc(O)c(OC)c1 C1(CC(=O)NC2(C)CN(C(C(C)CSCc3ccccc3)=O)C2)CCN(C)C1=O c1(C(=O)NCCCCN(C)C(c2ccc(CO)o2)=O)ccc(F)c2occc12 Cc1cnc(C)cn1.n1(C(=O)N)cc(C(n2cncn2)C2CC2)nn1 Cc1nc(C(=O)NC2C3CN(C(=O)Cc4ccsc4Br)CC23)c(C)n1C CC1CC(NC(=O)CCC(N)=O)CN1C(=O)CCCc1ccsc1 c1(C(N2C(C)(CC(N3CCC(c4cnco4)C3)=O)CC2)=O)cnn2ccccc12 CC(C)C(O)C(=O)N(C1CC1)CC1CCCN1C(=O)C(c1cccc(F)c1)O N1(C(c2c(C)n(CCC(C)C)nc2)=O)CCC2(CC2NC(=O)CSC2CC2)C1 C1(NC(C=C(CCC)C)=O)CCS(=O)(=O)C12CN(C(c1c[nH]nc1F)=O)C2 c1(C(C)C)ccc(C(N2CC(CC(C)NC(=O)CC3OCCC3C)C2)=O)c(F)c1 CC1CCC=C1C(=O)N1CCCCC1CC(=O)NCCCS(N)(=O)=O C1(CCNC(c2n(CC#C)ccc2)=O)CC(OC)CN1C(c1cncc(N)c1)=O CC(C(=O)NC1CN(C(=O)CN2C(=O)CCC2=O)CC1c1nccn1C)C(C)O C(=O)(C1CCc2cccc(OC)c21)NC1(CCNC(C(CC=CC)C)=O)CC1 N1(C(C(C=C)(C)C)=O)CCC2CN(C(c3n[nH]cc3C(C)C)=O)CC2C1 N1(C(C=CC(C)=O)=O)CC(CCNC(C2(O)CCC2)=O)C(C)C1 c1(C(N2CCC(C(C)NC(=O)CNC(C3CCC3)=O)C2)=O)cccc(C(F)F)c1 c1(C(=O)NC2(C)CCN(C(C3(F)CCCN(C)C3)=O)C2)cc(F)cc(F)c1O C(C(C)(C)C(=O)OC)(c1n(CCCC)nnn1)NCc1csnc1C S(=O)(=O)(c1cc(C)cnc1NCc1cc(Cl)n(C)n1)NC(CC(CC)C)CO C1(NC(c2ccc(C3CC3)s2)=O)CC(F)(CNC(=O)C(F)(F)C2(O)CCCC2)C1 CC1CN(C(C2(C)CCC2)=O)CC1NC(C1(F)CCCOC1)=O N1(C(c2ccnc([N+](=O)[O-])c2)C(=O)Nc2ccccc2)CCC2OCCC2C1 C(=O)(CCCC(=O)NC1CC(F)(CNC(c2csnc2OC)=O)C1)NCCC CC1(C)OC2CN(C(=O)CN3CC(=O)N(Cc4ccc(Cl)s4)C3=O)CC2O1 C(=O)(C(C)(C)CCF)NCC1CCC(CN(C(c2c(C)n(C)nn2)=O)C)CC1 C1(C(=O)NC(CNC(CC=C)=O)CC)CC(F)CN1C C1(NC(CCC(C)O)=O)CN(C(=O)CN2CCC2)CC1(C)C c1(C(=O)NC(CCOCC)C)c(CNC(=O)CC)nnn1C c1(CC)onc(C)c1C(N1CCC(OCCNC(=O)CC2CSCCS2)CC1)=O CC1(F)CN(C(=O)C=CC2CCCCC2)CCN(C(C2(Br)CC2(C)C)=O)C1 C1(C)(CC)C=C(C(=O)N(C2CN(C(c3cnn4cc[nH]c34)=O)C2)C)C1 CCC(CC(C)C)C(=O)NC1CCN(CCCNC(c2csc(C)c2C)=O)C1 c1(OC)ccc2c(=NCc3nc(=N)n(C)[nH]3)[nH]c(=NCCCOC(=N)O)[nH]c2c1 c1(CC)ccc(C(CNC(=O)Cc2cccnc2F)N(C)CCNC(C)=O)cc1 c1(SCC)cc(C(F)(F)F)ccc1C(=O)NC1CC(C)OC1C(F)(F)F c1(CC(=O)NC2C(OC)CN(C(C3CC34CC(O)C4)=O)C2)ccc([N+](=O)[O-])cc1 C1(C)(C(=O)NCC(COC)NC(=O)Cc2nnc(S)s2)CCC2(CC1)CC2 Cc1cc(CNC(=O)C=Cc2cn(C)nn2)oc1C(=O)NCC1(N(C)C)CC1 C1(NC(CCC(C)=O)=O)COC2(CCN(C(=O)Cc3cccc(O)c3)CC2)C1 c1(C(N2CC(C3N(C(C4(CC)CC4)=O)CCC3)(O)C2)=O)n[nH]c2c1CC(C)CC2 C1(NC(C2(SC)CCC2)=O)CN(C(C2CC(C)C2)=O)CCC1C C1(CCN(C(CC)COC)C)CCN(C(c2sncc2C)=O)CC1 C(=O)(C(C)(O)CC(F)(F)F)N1CCCCC(NC(CSC)=O)C1 C12(C(N3C(C(N4CC=C(C)CC4)=O)CC(F)C3)=O)CCCN(CC1)C2 C12(NC(CCc3ccn(C)n3)=O)CCC1CN(C(C1CCOC(=O)N1)=O)C2 C1(CC(=O)NC)CN(C(C2C(F)(F)C23CC3)=O)CCN1C(c1cnc(S)n1C)=O C12(CC(=O)N(C3(C(N(C4CCCCC4)C)=O)CCC3)C3CC3)CCCC1C2.C C1(CNC(CC2(OC)CCC2)=O)CN(C(=O)CCN2CCOCC2)CCC1(F)F C12(CNC(c3ccc(CCC)[nH]3)=O)CC(NC(c3cc(O)n(C)n3)=O)(CCO1)C2 c1(CC(=O)NC(CC)CNC(C2CC(N(C)C)C2)=O)ccnc(Cl)c1F C12(C(=O)NCc3cn(CC)nn3)C(NC(=O)CC3CCSCC3)C3CC1C2C3 c1(C(N2CCC(CC)C2CNC(=O)C2=CCCC2)=O)cc(C)nc(C)n1 C1(F)(CNC(CC(CC)O)=O)CCCN(C(c2cccc(F)c2F)=O)C1 C1(NC(CCCCC)=O)CC(F)(F)CC1NC(c1ccc(SC)s1)=O c1(C(N2CC3C(NC(=O)Cc4ccco4)C3C2)=O)c(O)ccc(Cl)c1F CCCCCCCC(=O)N1CCC(O)CC1C(N1CCC(N2CC(O)C2)C1)=O C#CCCC(C(=O)NC1CC(O)C1(C)C)NC(c1cc(F)cnc1O)=O N#CC1CCC(CC(=O)NCCNC(c2cncc(Br)c2)=O)C1 C(CCCCC(=O)NC1(C(=O)NCC2CC2)CCCCC1)NC(C)=O CCCC(C(=O)N1CCCC1=O)C(C)C.N1C(=S)S1 N1(C(C(C2CCCN(C(=O)Cc3cncnc3)C2)C)=O)CCC(O)C12CCC2 N1(C(c2cn(-c3c(Cl)ccc(OCC)c3)nn2)=O)CC2CCC(COC)C2C1 N1(C(CC(C)(C)O)=O)CCCC2CCN(C(=O)CCCc3ccc(Cl)cc3)CC12 C(=O)(CC(C(F)F)NC(=O)CN(c1nn(C)cc1OC)c1ccccc1)OC c1(C(=O)NCCC2CC(NC(C(=O)NCC)=O)C2)ccc(Br)c(C)n1 c1(OC(C(CC)C2CCOCC2)=O)cn(C)nc1I c1(C(N2C(CCCNC(CCC#C)=O)CCCC2)=O)n[nH]c2ccc(OC)cc12 CC(C)(CNC(c1cc(CNC(c2csnc2Cl)=O)on1)=O)CO c1(CCNC(c2ccc(OC3CCCCC3)c(F)c2)=O)cccc(F)c1Br CC1CCc2ccccc2N1C(N1CC(O)C(O)C1)=O c1(SCC(=O)NC2CCC(N(C(C3(CC(C)C)COC3)=O)C)C2)ccc(F)cc1 N1(C(C2(C)CCCC2)=O)CCCC2(CCC(NC(=O)C=CC3CCCCC3)C2)C1 N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CCCCCC1CNC(C12CC=CC(C1)OC2)=O C1(OC)CCC(S(=O)(=O)Oc2ccc(N3CCOCC3=O)cc2)C1 c1(C(=O)NCCCN(CCCNC(C2CC2Cl)=O)C)ccnc(OC(F)(F)F)c1 C1(C(N(CCNC(c2c(COC)cco2)=O)C)=O)CCCCC(=O)N1 N1(C(c2c(C)nc[nH]2)=O)CC2(C1)CN(C(=O)C(C)N(C)Cc1ccccc1)C2 c1(CNC(C2CC23CCN(Cc2cc[nH]n2)CC3)=O)ccc2cncnc2c1 c1(C(C(N2C(CNC(c3c(C)n(C)nc3)=O)CC2)=O)C)ccc(F)c(Cl)c1 C12(CNC(=O)NC3CCCN(C(c4cc[n+]([O-])cc4)=O)C3)CC3CC(CC(C3)C1)C2 c1(C(=O)Nc2nc(OC)nc(SC)n2)ccc2cc(NC3CNC3)ncc2c1 c1(NC(CCC(C)NC(=O)CSc2nc[nH]n2)=O)ccc(F)cc1O N1(C(C(C(C)C)O)=O)CCOCC(NC(c2cc(C(F)(F)F)ccc2F)=O)C1 Cc1ncc(C(=O)NC2CN(C(=O)CCCc3cnccn3)CC2C)cn1 N1(C(CSC(=N)N)=O)CCN(C2CN(C(=O)CCC3CC3)C2)CC1 C=CCCCCCC(=O)NC1CCN(C(c2nc(C)c(C)s2)=O)CC1(C)C c1(C(=O)N(CCC(N2CCCCCCC2)=O)C2CC2)c[nH]c2ccccc12 c1(C(=O)NC(CNC(C2(NC(C)=O)CCCC2)=O)C)[nH]nc2ncccc12 CC(C)C(C(=O)NCCC(C)(O)C1CC1)C(C)NC(=O)CCC1CC1 c1(C(N2CCC(C(C)NC(=O)C(F)(F)c3nccs3)CC2)=O)cc(=N)[nH]c(=N)[nH]1 O=C1NC(=O)C(C(c2ccccc2)OC)N1.N1(C(=O)O)CC(O)CC1C(=O)O Cc1noc(Cl)c1CC(=O)NCC1CC(CNC(=O)CNS(=O)(=O)N(C)C)C1 c1(CCN2CCCC(C(=O)NC(CC(C)=O)C)CC2)nc2ccc(C)cc2[nH]1 C1(NC(c2c(CCC)occ2)=O)CCN(C(=O)C(F)OC(F)(F)F)C12CCC2 C=CC(C)C(=O)NC1CCN(C(C2CCC2C#N)=O)C1 C1(C(N2CC(CC(C)C)OCC2)=O)C2CCN(C(C3CNC(=O)O3)=O)CC12 c1(CNc2cccc(C(N3CCCC(OC)C3)=O)c2)ccc(Br)cc1I C1(C(N2CCC(C3(C)COC(=O)N3)CC2)=O)CN2CCC1(F)CC2 C12(NC(CNC(=O)OCC)=O)CCCC1CN(C(=O)Cc1ccc(C)c(F)c1)C2 CC1CC(=O)NCC1C(=O)N(CCCCN(C)C(C1(C2CC2)CCC1)=O)C N1(C(CCCC(C)NC(c2cc(=N)[nH][nH]2)=O)=O)CCC2(CCOC2=O)C1 N#CC1(C(=O)CN2C(=O)C=CC2=O)CCNC1.c1(N)ncc(C2CC2)cn1 c1(CNC(c2c(C)oc(Cl)n2)=O)cnc2c(c1)CNC2=O N1(C(c2cccc(C#C)c2C)=O)CCC2(CCN(C(c3cnnnc3C)=O)C2)C1 N1(C(c2c(C)snc2)=O)CCC(C)(C)C1CNC(=O)C(C)C(C)(C)C C1(F)(CNC(c2nc(C)[nH]n2)=O)CCCN(C(C2CCN(C3COC3)C2)=O)C1 N1(c2nnc(COC)s2)CC2CC1CN(C(C1(C)CCC(C)C1)=O)C2 N1(C(c2cc(Br)cc(C)c2C)=O)CCC2CCN(C(=O)C=C3CCCC3)CC12 C(C)(CCS(C)(=O)=O)(c1n(CCCC)nnn1)NCC(C(F)F)c1ccccc1 CCC(CCC(=O)NCCNC(=O)CC1OCCC1C)NC(=O)CO c1(OC)c(C)cc(C)cc1C.c1(C2c3ccc(o3)CN2)ccccc1C C(C)(CCC(=O)N(C1CCN(C(C2OCCCO2)=O)C1)CC1CC1)OC N1(C(c2cc(C)no2)=O)CC2CC1C2NC(C12CCCC1(C(N)=O)C2)=O C1(C2(O)CCOC2)(C(=O)NCCC(C)(C)NC(C(c2cnn(C)c2)C)=O)CC1 C(=O)(CC1=CCN(C)CC1)NC1(C)CC(C(N2CCC(O)(CC(C)C)C2)=O)C1 c1(NC(=O)NCC)cc2[nH]nc(C(N3CCNCC34CC4)=O)c2cc1C(=O)OC.OC C1(CNC(C(CC)C(C)C)=O)CCN(C(=O)CSc2cccc[n+]2[O-])CC1(F)F C12(C(N(CCCNC(C(CO)NC(C)=O)=O)CC3CCCC3)=O)CCC(C1)OC2C C1(NC(Cn2cc(CC)nn2)=O)CN(C(=O)C=C(C)C2CC2)C(C)(COC)C1 C1(C(=O)NC2C(C)CCN(c3cc(CC)nc(CC)n3)C2)COC2(CCC2)C1 C1(OC)C2CCN(C(N3CCOC(CNC(=O)OC(C)(C)C)C3)=O)CC12 Cc1oc([N+](=O)[O-])cc1C(N1CCN(C(C2(C)CC(C#N)C2)=O)CC1C)=O c1(C(C(=O)NC2CC2)N(C)CCOCC2CC2)ccc2c(c1)CCCC2 Cc1cc(C(N2CCN(C(=O)C(C)O)C(CO)C2)=O)n2nc(C(F)(F)F)cc2n1 c1(C(=O)NC2C(NC(=O)CCc3nc(O)n[nH]3)CCC2)cccc2c1CCO2 c1(C(=O)NCCC2CC(NC(CCN(CC(F)(F)F)C)=O)C2)cccnn1 C(=O)(C(C)(O)C(F)(F)F)NC1C(NC(CCN(CCCCC)CC)=O)CCOC1 c1(N(CCCNC(c2ccc(C)s2)=O)C)nc(-c2cccs2)nc2ccccc12 CC(C(=O)N1CC(CN(C)C(c2ccc(CN(C)C)[nH]2)=O)C2(CC2)C1)C(C)(C)C c1(C(c2nnnn2C(C2(C)CC2)C2CC2)Nc2c(C)csc2)ccc(Cl)cc1F C1(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)C)C)COC2(CO)CC1C2 N1(C(c2c(C)n(C)nn2)=O)CCC(F)(C(=O)NC(C)C(C)n2cncn2)CC1 N(C(=NCCN1CCCC1)N1CCC2(CC(C(F)F)=NO2)C1)C(CC)C c1(C(N2CC(N(S(C3(CC)CC3)(=O)=O)C)C2)=O)ccc(O)c(C)c1O c1(OCC)cc(Br)c(ON2CCC(N(C)C)C2)cc1Br c1(C(=O)NCCCCCCNC(C(C)(C)SC)=O)ccc(O)c2ccccc12 C1(O)(CNC(c2c(CC)cncc2)=O)CCCN(C(=O)CN2CC3CC3C2)CC1 CC1CN(C(c2ccc(N(C)C)cc2)C(=O)Nc2ccccc2Cl)CC1C(N)=O N1(C(c2cc(C(N)=O)no2)=O)CC2(CCCCN(C(=O)C(=O)NCC(F)F)C2)C1 C1(NC(CC(C)SC)=O)C(CNC(C2CN3CCN2C(C)C3)=O)CCC12CCC2 C(CCC(C)(C)NC(=O)Cc1cn[nH]c1)NC(CC1(C=C)CCC1)=O C1(C)(OC)C=CCN1C(=O)CCCn1cc(C(c2cccc(N)c2)O)nn1 C1(C(N)=O)CCCCC1C(=O)NC1CCCC(NC(C23CC(CO)(C2)C3)=O)C1 c1(NC(c2n(C(COC)C)ncc2)=O)cccc(F)c1C(=O)OC(C)C N1(C(C2(CC)CCCN2C(c2csc(CO)n2)=O)=O)CCCC(F)CC1 C12(C(=O)NC3CN(C(=O)CC4CC5(CCC5)C4)CC(F)C3)CC1Cc1c[nH]nc12 CCC(CC(=O)NCC(C)(C1CC1)NC(C1CCOC1)=O)CC(C)C n1(CCCC)ncc(-c2nccn2C2C=CCCC2)c1C c1(C(N(CCCNC(=O)CSCC2CCCO2)C)=O)ccc(F)c(O)c1 C(=O)(C(Cn1cncn1)NC(=O)CCc1cc(C)[nH]n1)NC1(CC)CC1 c1(C(N2CC(CNC(C(CSC)OC)=O)OCCC2)=O)ccc2nc(C)cn2c1 C1(C(=O)NCCC2CCCN(C(CC=C=C)=O)C2)CN(CP(C)(C)=O)C1 CC1CC(CNC(c2cn(C3CCC3O)nn2)=O)CCN1C(=O)Cc1cscn1 S(=O)(=O)(c1ccc(C)cc1F)NCC(=O)NC1CN(C(C(CC=CCC)C)=O)C1 CCC(C)C(CC(=O)NC(c1cccc(Cl)c1)C)NC(c1ccnn1COC)=O c1(C(=O)NCC(C)NC(=O)C2=COCCC2)cc2c(s1)C(C)(C)CCC2 C(=O)(C1CCc2c(Cl)cccc21)NCCNC(C=Cc1cnc(OCC)nc1)=O CCCC(C)(CCC)C(=O)NCC(O)CN(C)C(C1CCCOCC1)=O c1(CC(C(=O)NCCN(C(C(C)(C2CC2)NC(C)=O)=O)C)C)ccc(F)cc1F N=c1cc(C(N2CCC(CCCNC(c3cc(Cl)no3)=O)CC2)=O)cc[nH]1 N1(C(=O)CCCCO)CCC2(CCCN2C(C2CCCCS2(=O)=O)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CN(C(C(=O)NCCCC)C)C)C1 c1(C(N2CCOC(CC(F)(F)F)C2)C(=O)NCCC)c(C)nn(C)c1C C1(CC#C)(C(=O)NCC(C)(O)CNC(c2cccn2CC=C)=O)CCCC1 C1(NC(C2(C)CCCC2)=O)CC2CC(NC(=O)CCN3CCOCC3=O)C2C1 Cc1ccc(O)c(C(N2CCCC2C(C)NC(=O)COCc2nnc(C)s2)=O)n1 O=C(C#CC1CCCOC1)NCC12CCC(CC1)N2c1cnc(C(F)(F)F)cn1 Cc1nnc(CCC(=O)NCC2CC2CNC(C2CC=CCC2C)=O)n1C C1(C(=O)OC)Cc2cc(Br)ccc2N1C(c1cccc(C(=O)N(C)C)c1)=O N1(C(c2c(OC)ccnc2)=O)CCOCC(NC(=O)C(C)c2ccsc2)C1 c1(C(=O)NC(CC(C)NC(c2cc(C(C)(C)C)c[nH]2)=O)C)cccnc1O c1(C(N2C(C)CC(CC(=O)NCCc3ncon3)C2)=O)nnc(O)nc1O c1(C(=O)NC2C(NC(C3CCC(COC)C3)=O)COC2)ccc(Br)cc1 c1(NC(C2CC3CC3N2C(=O)C=Cc2cnccn2)=O)ccc(Cl)nc1Cl C1(C(=O)NCCCN(C(c2ccc(SC)s2)=O)C(C)C)CC2CCCCCC12 CCC(C)C(O)C(=O)NCCN(C(c1ccnc(OCCOC)c1)=O)CC C1(NC(C(CC)(C)O)=O)CCN(C(C23CCCN2CCC3)=O)CC(C)(C)C1 Cc1ccc(C(=O)NCC2(F)CC(NC(c3nncs3)=O)C2)cc1 N1(C(C(CCC=C)c2nn[nH]n2)=O)CCC(C)N(C(=O)C=CCOC)CC1 C=CCC(C)C(=O)N(C1CC(NC(c2cn(C)c(O)n2)=O)C1)C N1(C(c2ccc(COC)s2)=O)CCN(C)CC1CNC(C1(O)CCOC1)=O C1(OC)CC(NC(=O)C(C)OCC(C)C)CN(C(c2csnn2)=O)C1 c1(OCC)nc(Cl)ccc1S(=O)(=O)Nc1cccc(C2CCCCC2N=[N+]=[N-])c1 N1(C(CC(COC)C)=O)CCC(C(F)(F)F)n2nccc21 CC1(C)CCC1NC(=O)CCC1CCN(C(C2COCCO2)=O)C1 C1(NC(C2CC(=C)C2)=O)CCN(C(=O)CCC2C(=O)NN=C2C)CC(C)(C)C1 c1(N2CC(SC)C2)ccc(S(=O)(=O)NCc2nn(C)cc2C)cc1C#N c1(CCN(C(=O)CN(C(=O)CC2CCSC2)C2CCC2)C)cccs1 C(CCC(C)C)(C(=O)NC1C2CCCC1COC2)NC(CCCCC#C)=O C(=O)(CC1=NN(C)C(=O)C1)NC1CN(C(CC2(OC)CCOCC2)=O)C(C)C1 C#CC1CN(C(=O)CC2CN(C(c3sncc3CC)=O)CCO2)CC1O O(Nc1cc(OC)cc(OC)c1)Cc1c(C)cc(CC)c(C)c1 c1(NC(=O)NC2CN(C(c3ncccc3F)=O)CCO2)ccc(Br)cc1 Cc1c(C(=O)NCCC2(NC(=O)CCCC(N)=O)CCC2)sc2cccc(F)c12 Cc1cc(CC(N2CCN(C3CN(C(=O)C(C)O)C3)C(=O)C2)=O)cc(C)c1Br C1(C(=O)NCC23OCC(NC(CCCC)=O)(C2)C3)CC(C(=O)OC)=NO1 C(CCc1ccccc1)(C(C)(C)C)NC(COC1(C#C)COC1)=O C1(NC(C(C)Oc2ccccc2)=O)CC2CN(C(=O)CC(C)(C)O)CCN2C1=O C1(CNC(c2c[nH]cc2Br)=O)CCCN(C2CCN(c3cccc(Cl)c3)C2=O)C1 Cc1nc(CC(C)C)oc1C(=O)N(CC(C)(C)CNC(=O)CC(C)(O)C1CC1)C c1(C(=O)OCC(C)CC2CCOCC2)ccc([N+](=O)[O-])c(O)c1 C1(CCNC(=O)CCc2cnco2)CCC(NC(c2ccoc2Br)=O)C1 Cc1cnc(NCC2CN(C(c3csc(Cl)c3C(F)F)=O)CC2C)nc1O C#Cc1cncc(C(=O)NC(C)C(C)NC(c2c(C)ccn2C)=O)c1 c1(C(C)NC(C23C(CN(S(C(C)C)(=O)=O)C2)C3)=O)cc2ccccc2cn1 C1C(=O)N=C2C=CN(N2)C2CN1C2.N1(CCOCCC(C)C)CCc2sccc2C1.NOC N1(C(C(C)(C)C)=O)CCC12CN(C(=O)CC1CCNCC1)C2.c12ccc(cc1)o2 C12COCCN1C2=O.Cc1cc(OCC(N2CCCC2)=O)no1.C1CC(=O)N1 C(C(CC)(CC)NC(=O)C(CC)n1ccc(C2CC2)n1)NC(C(CC)NC(C)=O)=O N1(C(C2CCN(C(C)C)CC2)=O)CC(NC(=O)CN(S(C)(=O)=O)C)C(C2CC2)C1 Cc1ccc2c(=NCc3cccnc3Cl)[nH]c(N3CCCCC(C)C3)nc2c1 CC(C(=O)NCC1(CN(C(=O)C(c2cnn(C)c2)O)C)CC1)C1=CCCC1 Cc1c(Br)c(C(=O)NCCC2CN(C(=O)CCOC(C)C)CCO2)nn1C c1(CC)ccc(C(=O)NC2CN(C(c3ccn(COC)n3)=O)CC23CC3)c(C)n1 c1(CC)onc(C(=O)NC2CC(CCNC(=O)Cc3cncc(O)c3)C2)c1C c1(C(=O)NCC(C)NC(=O)CSc2nc[nH]n2)ccccc1CC(C)(C)C C1(NC(C2CCOCC2)=O)CCN(C(c2cnn3cnnc3c2)=O)CC12CCC2 C1(C(=O)NC(CCCNC(c2c(CC)noc2)=O)CO)CCC(C)(O)CC1 c1(C(N(CC(=O)NCC(C)NC(=O)CC2CC2)C)=O)csc(=N)[nH]1 C(=O)(C1=NNC(=O)CC1)N1CCCC(CCNC(=O)CN2CCCC2=O)C1 C1(O)(C(C(=O)N(C2(C(=O)OC)CC2)C)F)CN(C(C2CS(=O)(=O)C2)=O)C1 CC1CC(NC(=O)C=C2CCCCC2)CCN1C(=O)CCF c1(C(N2C(CN(C)C(C3CCNC3=O)=O)CCC2)=O)cc2c(O)ncnc2cn1 C1(C(N2CC(CCNC(c3cnc(C(C)=O)s3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1oc(C)c(C(=O)NCC2(NC(c3c[nH]c(C#N)c3)=O)CC2)c1Br c1(NCC(N2CCN(c3cccc(C)c3)CC2)=O)c(C)nc2ccccn12 C1(CNC(CNC(CCC)=O)=O)CN(C(c2cccnc2CC)=O)C2CC12 c1(C(N2CC(NC(c3c(COC)cco3)=O)C(C)C2)=O)ncn2c1CCCCC2 N1(CC2N(C(=O)OC(C)(C)C)CCOC2)C(=O)CN(CCOc2ccncn2)C1=O N1(C(C2C(CNC(CC)=O)C2(C)C)=O)CCC(F)(F)CC1 C1(NC(c2cnc(COC)s2)=O)(CF)CCN(C(c2n[nH]c(O)n2)=O)C1 c1(OC)cc(OC)nc(N2CCCC2CNC(c2cc(F)cnc2Cl)=O)n1 CC(C)CC(F)C(=O)NCCOCCNC(=O)CC1CCCCC12CC2 C(=O)(CCC(C)(C)C#N)NCC(C(=O)NCc1c(C)nc(CC)o1)N(C)C N1(C(C(CSC)O)=O)CCCC2(CCN(C(C3(CC(C)C)CC3)=O)C2)C1 N1(C(CCc2onc(C(C)C)n2)=O)CC2(CCN(C(C3COC(=O)N3)=O)CC2)C1 c1(OC)c(C(=O)NC2CCN(C(=O)CN3CCCOC3=O)CC2C)ncnc1C C(CC(=O)NC1CCSC1)(C(F)(F)F)NC(c1nn(C)c(=O)cc1)=O CC(CCC(=O)N1CC=CC1Cn1cc(-c2nccn2C)nn1)N(C)C C1(C(N2CC(N3CCN(C(=O)Cc4cnoc4)CC3)C2)=O)CCCCC2(CC2)C1 c1(C(N2CC3CN(C(c4nn(C)c(F)c4)=O)CC3C2)=O)cccc2cnccc12 C1(NC(COCCCOC)=O)C=CCCC1C(=O)NCCCCSC CC(C)CC(C(=O)NOCCOCCO)NC(C1CCC(=O)C1)=O N1(C(C2(CC(=O)OC)CCCC2)=O)CC(NC(=O)C=C(C)C(F)F)CC(F)C1 CC(C)(C)C(CNC(=O)Cn1cnc(C(N)=O)n1)NC(c1ccc(F)nc1)=O C1(NC(c2ccc(C(C)C)s2)=O)CCN(C(=O)CSCCC#N)C1(C)C C1(NC(C(C)N(C(=O)COCC(C)C)CCC)=O)CCCN1 Cc1ncnc(O)c1C(N1CCC(C2CCCCN2C(=O)C=CCO)CC1)=O CC(C)(C)CC(C(=O)NCCOC(=O)C1CC1)NC(=O)CC1CC=CCC1 C(=O)(C(F)C(C)CC(C)(C)C)NC(C(C)C)CCNC(c1cc(F)cc(F)c1)=O C(=O)(CC1OCCc2sccc21)NCCCNC(c1c(C)c(C(F)(F)F)n[nH]1)=O N1(C(CCOCC(C)C)=O)CCN(C(C2(CF)CCC2)=O)CC1 C1(C(=O)NC(C=C)CO)CN(C)CCN1C(c1cnncc1OC)=O CC1(C)C(=O)Nc2ccc(C(N3CC(NC(C4C=CCC4)=O)CC(F)C3)=O)cc21 C(c1ccco1)=C(C)C(=O)N1CC(=C(F)CNC(=O)Cn2cc[n+](C)c2)C1 C(=O)(CC(C)CC(F)(F)F)NCC1CCN(C(CC(C)C)=O)CC1C Cn1cccc1C1CC1C(=O)NCCNC(c1csc(-c2cnccn2)n1)=O N1(C(C2C(CCC)C2)=O)CC2CN(C(c3cc(CC)ccc3F)=O)CC2C1 N1(C(C(COC)OC)=O)CCC(NC(=O)CNS(N)(=O)=O)C(O)C1 c1(OC)ccc(C=CC(N2CC(C(C)NC(c3ccc(F)cn3)=O)C2)=O)cc1 N1(C(c2cc(C)n(-c3ccccc3)n2)=O)CCC2(C1)CN(C(=O)C=CCO)C2 CC1(C)CN(C(=O)CCc2cnoc2)CC1CC(=O)NCc1[nH]ccc(=O)c1O O=C(CC1CN(C(C2CCCCC2)=O)c2ccccc21)N=c1cns[nH]1 N1(C(c2nccc(C)c2)=O)CCCC(C2CCCN(c3nc(C)ns3)C2)C1 C1(C(=O)NC(C)CNC(=O)CCc2nccs2)CCC2(CC1)CC2 CCC(CC)C(F)C(=O)NC1CC(C)(CNC(=O)CCSCc2ccccn2)C1 CCCC(C)CC(=O)N1CCC(NC(c2cnn(-c3ccccn3)c2)=O)C1 C(=O)(C1=CNS(=O)(=O)N=C1C)NC(CSC)C(N1CCc2nc[nH]c2C1)=O C1(NC(C(CC)(CO)OC)=O)CC12CCN(C(=O)CC1CCCOC1)CC2 C1(NC(=O)Cn2ccnn2)CN(C(C2CCCOCC2)=O)CC1n1cccn1 CC1(C)CCCC(CS(=O)(=O)N(CC(C)(C)NC=O)C)O1 CC(C(=O)NC1CCN(C(c2sncc2Br)=O)C1)S(C)(=O)=O C1(C(=O)NC2C(C(=O)NC3CC(C(C)O)C3)CC2)CC(C)(C)CO1 c1(CC(=O)NCC2(C)CC(NC(C3CC3F)=O)C2)cn2ccccc2n1 C(c1ccc(O)c(O)c1)=CC(N1CC(C(C)NC(c2n(C)cnc2)=O)OCC1)=O C1(CNC(C(CC)OC)=O)CN(C(C2CC3(C2)CC(O)C3)=O)CC1(C)C c1(OC)cncc(C(=O)NC(C2CCCN2C(=O)COC2CC2(F)F)C)c1C O=[N+]([O-])c1cccnc1N1CC(NC2CC2)C1 c1(-c2cc(NCc3nc(C)oc3)ncc2)cc(O)c2ccoc2c1 N1(C(c2ccc(Br)cc2)C2CN(C(c3c(C)cnnc3)=O)C2)CC2CC2C1C#N C1(C(C)C)(C(=O)NCC2C=CCOC2)CCN(C(=O)C(O)Cn2cncn2)C1 CCCC(C)C(=O)Nc1ccc(-c2cnccc2C(=O)OC(C)(C)C)cc1 C1(C(C)O)CCN(C(=O)C(N2CCCC(Cc3nccn3C)C2)=O)CC1 c1(CCOCC(N2CC(CCCCNC(C=CC)=O)C2)=O)cccc(F)c1 c1(CCC(c2n(CCC)nnn2)(C)NC2CCC2C(=O)OC)cccc(Br)c1 C(=O)(C(F)CCC(C)C)NCC1N(C(c2csc(C)c2N)=O)CCC(C)C1 C1(NC(=O)C2=CCSC2)CCN(C(c2csc(F)c2)=O)C(C2CC2)C1 N1(CC2(CS(=O)(=O)Cc3ccccc3)CCCC2)CCCC(S(=O)(=O)N2CCOCC2)C1 c12ccc(C#N)cc1NC2=O.O(N(C)C(=O)C1(OC)CCSC1)CC(=O)OC N1(C(CC(CNC(C(C)CC(F)(F)F)=O)C2CCC2)=O)CCC2(COC(=O)N2)C1 C1(CC(=O)NC(CC#C)CC)C2CCCC2N1C(=O)CC1(C#N)CCOCC1 C(N=c1nc(N2CC(COC(C)(C)C)C2)cc(C)[nH]1)c1cn(CCC)nc1C C1(NC(c2c(OC)csc2)=O)CN(C(=O)C(C)(C(C)C)OC)CCC1CO Cc1ccc2[nH]c3c(c2c1)CC(NCc1ccc(Cl)c(Cl)c1O)CC3 CC(C#N)CCC(=O)N(C1CCCC1)Cc1csc(-c2ccco2)n1 CC1(C)CCC=C1C(=O)N1CCN(C(c2ccc(C(F)(F)F)nc2)=O)CC1C1CC1 N1(C(c2cc(C)nn2C)=O)CCC(NC(C2CC2C(N)=O)=O)C(F)C1 CC1OC2(C(=O)NC(c3cccc(Br)c3)CC3CC3)CCC1CC2 c1(NC(=O)NCc2ccc(C)c(OC(F)F)c2)nnc2c(Cl)cnn2c1O CCC(CN1CCCC(c2n[nH]cc2OC)C1)CC(F)F N1(C(CCC2N(C)CCC2)=O)CCCCC1C(=O)NC1CCN(CC2CC2)C1 C1(NC(C2(CO)CCN(C(C(CC)OC)=O)C2)=O)CC(C)CCC1O n1(C(C)C)cc2c(n1)CC(C(=O)OCC1CCOCC1(C)C)CC2 CC1(C)CN(C(C23CCC(CC2)C3)=O)CC(C)(C)C1NC(=O)CCC1CCOC1 C(c1ccc2ncccc2c1)=CC(=O)NC12CC1CN(C(C1(O)CCOC1)=O)C2 CC1(C)CCc2cnc(CNc3cncc4c3CCC4)nc21 N1(C(CNC(CCC)=O)=O)CCC2(CCN(Cc3ccc4ccccc4c3)C2)C1 c1(N2C3CC(NC(C4(CC)CCC(O)CC4)=O)C2CC3)ncnc2[nH]ccc12 N1(CC(=O)NCC(O)CCNC(c2cncc(Br)c2)=O)CC2CCC1C2 C1(C(=O)NC2CC(NC(c3cc(C(N)=O)[nH]n3)=O)C2)CCn2ncnc2C1 C1(CC)(CC)CCN(C(=O)C(C)N(C(=O)C(CC2CC2)OC)C)C1 C(=O)(C1=COCCO1)N1CCC(N(CCC)C(C2CCC2C)=O)CC1 Cc1nc(N(C)C)sc1C(=O)NCC1CN(C(=O)C=Cc2ccn(C)c2)C1 N(C(=NCCNS(C)(=O)=O)NCC1CCOC1)C(C#C)CCC C1(CC)CC(C)CN(C(C2(CC)CN(C(C3CCN3C)=O)C2)=O)C1 CC1CCCC(C(N2CCC(NC(=O)COc3ccccc3)CC2)=O)C1 N1(C(Cc2c(C)nccc2)=O)CC(NC(c2cncc(CO)c2)=O)CC2(CC2)C1 CCC(C(=O)N(CC(C)N(C)C(c1cc(C(C)(F)F)ccc1C)=O)C)C(C)(C)C C1(NC(C(CCCC)(C)F)=O)CCC2(CC1)CC(NC(=O)CNC(=O)OCC)C2 Cc1ccc(OCC(=O)N(C)C)c(C(=O)NCCCc2ccccc2Cl)c1 CC(C)(O)C(F)(F)CNC(c1csc(CNC(c2cc(Cl)cs2)=O)c1)=O C(CC(C)(C)C)(C(=O)NCC1CCN1C(C1(C#N)CC2(CC2)C1)=O)OC c1(C(=O)NC2C(NC(c3cc(C)sc3)=O)COC2)c(C)noc1C(C)C CC1(CNC(=O)C(O)C(F)(F)F)CCCN(C(=O)CNC(N2CCCC2)=O)C1 Cc1ccc2nc(C)cc(C(=O)NC3CCC(N(C)C(c4cn[nH]c4)=O)C3)c2c1 C(=O)(C(C(C)C)n1cnnc1)N1C(C(C)NC(Cc2c(C)con2)=O)CCC1 c1(CCC)nc(C(O)Cc2ccccc2F)n(-c2cnn(C)c2)n1 C12(CNC(C(CC=C)(C)C)=O)CN(C(c3n[nH]c(C)c3Br)=O)CC(F)(C1)C2 c1(OC)ccc(C(=O)NC(C)CCNC(=O)Cn2c(C)ccc2C)c(F)n1 c1(C(N(C)CC2(NC(C(C)=CC3CC3)=O)CC2)=O)ccc(OC(F)F)c(C)c1 C1(C(=O)NC2(CO)CCCN(C(=O)C3=CCC3)C2)CN2CCCN1CC2 N1(C(C2C(=C)C2)=O)CCCC(CO)(NC(c2cc(CC)ccc2Cl)=O)C1 Cc1nccc(C(N2CCCC(CN(C(=O)CSc3n[nH]c(O)n3)C)C2)=O)n1 Cc1cc(C(=O)NC2CCC(CNC(C3(C)COCCO3)=O)C2)cc(N)c1Cl C1(C)(NC(C(C2CCCC2)OC)=O)CN(C(=O)C=C(C)C(C)C)C(C)(C)C1 C1(C(N2C(CNC(c3cc(OCC)nc(C)c3)=O)CC2)=O)CCn2nncc2C1 N1(C(C(C)CCCc2nn[nH]n2)=O)CC2(C1)CN(C(=O)Cc1ccsc1Cl)CCO2 c1(C(N2CC(N3C(=O)CC(NC(C=CC=CC)=O)C3)C2)C)ccc2[nH]ccc2c1 Cc1nc(C(F)(F)F)oc1C(=O)NC(C1CCCN(C(=O)Cn2cnnn2)C1)C C1(OC)CC(CNC(c2ccc(O)cn2)=O)N(C(c2ccc(F)cc2)=O)C1 c1(SC)nccc(CNC2CC(NC(c3cc(C(F)(F)F)ccn3)=O)C2)n1 CC1CCc2n[nH]cc2C1C(=O)NCCN(C(c1cc(CO)on1)=O)C1CC1 c1(C(N2C(C)(C(=O)Nc3nccc(OC)c3I)CC2)=O)cnn2cccnc12 C(=O)(CCS(C)=O)NC(C1CCN(C(=O)CCCC2CCC2)CC1)C Cc1cncc(C(N2CCCC2C(C)(C)C(=O)NC(C)CS(C)=O)=O)c1 c1(C(=O)NCC(CC(C)C)NC(CCCC(C)=O)=O)c(F)ccc(C)c1Cl C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CN(C(=O)C(C)(C)C(F)F)CCC1CO Cc1nc(N2CCCC(CO)C2)sc1NC(=O)NC(Cc1cccc(F)c1)CO C(CCCC(=O)NOC(CO)C(C)C)N(C(CC(CCOC)C)=O)C N1(C(CC)=O)CCC2CCC(C1)N2C(=O)Cc1c(F)cc(C#N)cc1Br C=CCC(C)(CC)C(=O)NCCC1(CNC(C23C4C5C2C2C3C4C52OC)=O)CC1 c1(C(N(CC(C)NC(c2ccn(C)c2)=O)C)=O)c(Cl)ccc(Cl)c1N c1(N2CCCN(C(CCSC)=O)C(C)C2)ncnc2ccc(O)cc12 C(=O)(C(F)C(C)CNC(=O)C(COC)COC)N(C1CC(=C)C1)C C1(CC(=O)NCC2CCC(N(C)C)C2)(NC(C23CSCC2C3)=O)CCCCC1 C1(NC(C(C)N(C)C)C)CC(=O)N(Cc2ccccc2O)C1 CC1CCn2ncc(C(=O)NC3CCN(C(C4CC(F)C4)=O)C34CCC4)c2C1 Cc1c(C(=O)NC2CC2CNC(=O)C(F)=CC2CC2)cnc2ncnn12 C(=O)(N(CC)OC)C1(CNC(c2cn(CC=C)nc2)=O)CCCC1 N1(C(c2sccc2CO)=O)CCC2CN(C(=O)CCc3ncc[nH]3)CC2C1 c1(NC(C(=O)NC(c2cncc(F)c2)C)=O)ccc2ncn(C)c(=O)c2c1 c1(C(=O)OC)c[nH]c(=NC2CCCC(NC(=O)C(C)n3ccnc3)C2)cn1 CCS(=O)CC(=O)N1CC(C)(CCC(=O)NCC(C)(COC)OC)C1 n1(CC)nc(C)c(C(=O)NC2C=CCN(C(C3CC3C(=O)NC)=O)C2)c1Cl c1(C(=O)NCC(C)(C)N(C(C(C)NC(=O)OC)=O)C)sccc1CO S(=O)(=O)(c1cccc(C(C)C)c1)Nc1c(=O)cc(C(=O)OC)n(C)c1 C12(C(N(CC(=O)OCC)C)=O)CC(C)(CN1C(=O)CSc1cn[nH]c1)C2 C1(CNC(CCCCC)=O)C(C)CCCN1C(c1ccnc(OC(C)C)c1F)=O C#CC(CC(C)(C)C)NC(=O)C(C)(C)CCNC(=O)C(CC)C(=O)OC c1(C(=O)NC(C)C(CO)NC(c2csc3c2CCCC3)=O)cccn2ccnc12 C12(C(N3CCC(NC(C4OCC5CCCC45)=O)(CF)C3)=O)CC3CC1C2C3O N1(C(c2cc(OC)n(C)n2)=O)CCC2CCN(C(c3cncs3)=O)C2C1 N1(C(c2c(C)con2)=O)CC(NC(=O)CC2CCN(C)CC2)CC12CCCOC2 C1(C(N2CCC(OC)(CNC(C3CC=CCC3)=O)C2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NC(COCC)C)CCC(CNC(c2cscc2Cl)=O)CC1 c1(NC(C2=NOC(c3ccc(C)cc3)C2)=O)nc2cc(C)cc(C)c2s1 C(=O)(C1=C2CCN=C2NC=C1)N1C2CC(CN(C(C3(C)CC3(F)F)=O)C2)C1 CC1C(NC(=O)C(Cl)=CCl)CCCN1C(C1CC1c1ccsc1)=O C1(c2cn(CC(=O)NC3CC(C(C(=O)OCC)C)C3)nn2)CC(F)(F)C1(F)F c1(C(N(C2CCN(C(COCC=C)=O)CC2C)C)=O)ccc(Cl)c2ncccc12 C1(CCOCCNC(N)=O)C=CC(CC(CCN2CC(Oc3ccccc3)C2)=O)C1 c1(C(=O)NC2CC(NC(C3N(C)C(=O)CCC3)=O)C2)cc(Br)c(F)cc1F C(=O)(C1CCCc2cccnc21)N1CC(CC(=O)NCC2CC(=O)CO2)(OC)C1 C(=O)(C1=NOC(C)C1)N1CC(C)(NC(c2cnn(CC)c2C)=O)C1 CCC(O)CC(=O)NCCC(C(=O)NCCC1CCN(C)C1)OC C1(NC(COCC)=O)C=CCN(C(=O)C(c2cccnc2)C)C1 c1(C(N2CCCC(N(C(c3c(CC)cno3)=O)C)C2)=O)ccc(F)c(OC)c1F N1(C(CCn2ncc(C)c2)=O)CCC(C2CC2)C1CNC(=O)C1=COCC1 O=C(CCCC1CCCO1)NCC(O)C(=O)NCCc1ccncn1 C1(NC(CC(C)OC)=O)C=CCCC1C(N1CCCC1C(C)C)=O C(=O)(CCCCCCCCCO)NCC1N(C(c2c[nH]c(=N)o2)=O)CCCCC1 C1(C(=O)OC)CC(F)(F)CC1C(N1CCC(O)(CNC(=O)CN(C)C(C)C)C1)=O CC1CC2CN(C(C3CCC4(CC4)N3C(c3cc(CO)on3)=O)=O)CC12 C(c1ccc(F)cc1)=CC(=O)NCCC(C)N(C(=O)Cn1ncccc1=O)C C(=O)(CC(C)C1CCCCC1)NCC(CC)NC(C1CCCCO1)=O C1(CNC(C2CCC(C)CC2)=O)CCN(C(=O)C(F)n2ccnc2)CC1O C1(NCC(C2CCOCC2)OC)CC(NC(c2csc(Cl)c2Cl)=O)C12CCC2 CCC(CC)(CCNC(C1(C)CCCO1)=O)NC(C1CCN(C2CC2)S1(=O)=O)=O C(=O)(C(C)(C)C1=CCSCC1)NCC1CN(C(C=C(C)C(C)(C)C)=O)C(C)CC1 c1(C2(C(=O)NCC3CCC(NC(C)=O)C3)CC2)cccc(Cl)c1F C1(C(=O)NCC2N(C(c3c(C)[nH]nc3Cl)=O)CC(O)C2)COC2(CO)CC1C2 Cc1nc(CC(C)C)sc1C(=O)NCC1C2CN(C3CCSC3)CC12 CCCS(=O)(=O)CC(=O)NC1COCCN(C(=O)COCC(=O)OC)C1 C12(CNC(C(F)=CC)=O)CCCC1N(C(=O)COCP(C)(C)=O)CCC2 C(=O)(CC(C)(C)CCC)N1CC(CCC)N(C(c2cc(Br)ccc2O)=O)CC1 c1(NC(C(N2CCOCC(F)(CC)C2)=O)=O)sc(S(N)(=O)=O)c(OC)c1OC N1(C(CCCNC(C)=O)=O)CC(NC(=O)C2=CCC(C)CC2)CC(F)(F)C1 CC1=C(C(=O)N2CC(NC(c3csc(C4CC4)n3)=O)CC2(C)C)COCC1 c1(C(=O)NC(C2CCN(Cc3nccs3)CC2)C)cc(Br)c2ccccc2n1 c1(C(=O)NC2C(C)(CN(C(CCOC)=O)C)CCC2)ccc(Cl)c(N)c1 Cc1nn(CC(=O)NCC2CC(F)(F)CN2C(=O)Cc2nncn2C)c(C)c1C c1(SC)cccnc1CNC(=O)CN1CCCCC1=O.C123CC(C1)(C2)C(=O)N3 c1(C(N2CC(C)(C(=O)Nc3nc(C)c(C)s3)C2)=O)cc(Br)c(F)cc1C CC1(C)CC(CNC(=O)C=Cc2ccco2)N(C(C2CC=CCC2)=O)C1 N1(C(c2c(Cl)csc2Cl)=O)CC2(C1)CN(C(C1(CF)CCC1)=O)CCO2 c1(C(=O)NCC2N(C(C(CC=C)C)=O)CCCC2)c(-n2cccc2)sc(C)c1C Cc1ccc(C(=O)NC(C2CCN(C(=O)CCOCC(=O)N(C)C)C2)(C)C)cc1 c1(C(N2CCC(Cc3c(C)nn[nH]3)C2)=O)ccnc(NC2CCCC2)c1 Cc1cocc1CN(Cc1ccccc1)CC1CCC1 Cc1cc(F)sc1C(=O)NC1CCCC1CNC(c1csc(Cl)c1Cl)=O C1(=CC=CC(=O)NC(=O)C(O)C2CN(C(=O)CCCN3CCC3)C2)CCCCC1 N1(C(C2(OC)CCSCC2)=O)CCCC2(CCCN2C(=O)C(C)CSC)C1 C1(NC2(OC)CCC(C)C2)CC2(CCNC2=O)C1 C(CC)(CC(F)F)NC(=O)Nc1ccccc1F.c1(CC(CC)OC)ccc(SC)cc1 C(C(C)(C)CNC(=O)COCCN(C)C)N(C(=O)CC1CCC2CC12)C N1(C(C(C)CO)=O)CCCC2C1CCN2C(=O)CC12COC(C)(C1)C2 c1(CCC(N2C(CNC(C3C(CC)CCO3)=O)CCC2)=O)ccc([N+](=O)[O-])cc1 C(CCC(C)(C)C(=O)NCC1CCC1(C)C)NC(C1CN(OC)C(=O)C1)=O C1(N(C(c2cnc(CC)s2)=O)C)CCCN(C(=O)CC(c2cccc(F)c2)C)C1 c1(CN2C(C(=O)Nc3cccc(O)c3)CC3CC32)c(Cl)cccc1[N+](=O)[O-] c1(C2C(C(=O)NC3CC(C)(NC(=O)C=Cc4nccs4)C3)C2)ccncc1F C1(C(=O)NC2(C)CN(C(c3cnc(COC)s3)=O)C2)C(C(=O)OC)CC(=O)N1C c1(C(N(C)CC2CCCN2C(c2ccc(Cl)o2)=O)=O)cnn2c1CC(F)(F)C2 Cc1cc(C(F)F)oc1C(=O)NCC1(O)CC(NC(C2(n3cncn3)CC2)=O)C1 c1(C(=O)NC(C)(C)CCCNC(c2cn(CC3CC3)nn2)=O)ccc(Cl)cc1Cl Cc1ccc(CC(=O)NCCCCC(C)NC(c2cn(C(F)F)cn2)=O)c(C)c1 C(=O)(CC(C(F)F)n1cccn1)NC(CC)(CC)CCN C(C)(C)(CN=c1nc(SC2CC2)[nH]s1)C1CCN(C(C(C)CN(C)C)=O)CC1 CC1CN(C(c2cn(C3COC3)nn2)=O)C(C)CN1C(=O)COCC1CC1 c1(C(N(CCC(C)NC(C2(CC(C)C)CCC2)=O)C)=O)nnn2c1C(=O)NCC2 C(CC(C)(C)C)(C(=O)N1C(CC(=O)NCC(N2CCCC2)C)C2CCCC12)OC c1(CC(=O)NC(COC)C(=O)NCc2cocn2)cncnc1O C1(C(N2C(C(CC)C)CCC2)=O)CCCC(NC(C2CCN(C)C2)=O)CC1 c1(C(=O)NC(CCSC)C(=O)NC(C)C(=O)NO)cncc(F)c1C C1(CCNC(c2cc(CC)n(C)n2)=O)CN(C(=O)Cc2ccno2)CCC1CO N1(C(c2cc(C)[nH]n2)=O)CC2CC(C)N(C(=O)C(C3CCCO3)C3CC3)C2C1 C1(C(=O)NCCCc2cn(-c3ccc(Br)cn3)nn2)CCNCCC1CO CCN=C(NCc1noc(COC)n1)N1CCCC(C2(C)OCCO2)C1 c1(CC(=O)NC(C(C)(C)NC(c2cc(CC)ncn2)=O)C)nc2c([nH]1)CCCC2 c1(C(N(CCCNC(c2coc(Br)n2)=O)C2CC2)=O)cc2ccccc2cn1 c1(SCC(=O)NCC(N(C(=O)C(F)n2ccnc2)C)C2CC2)cnn(C)c1 C(=O)(CCCCC(=O)NC1CN(C(=O)C=Cc2ccccc2)CC1N=[N+]=[N-])NC c1(C(=O)NC(CNC(Cc2c(C)n(C)nc2)=O)C(C)C)coc2c1COC2 C1(CC(=O)NC2(CF)CCC2)CCN(Cc2cocn2)C1 Cc1cc(C)n(CCc2nc(CCc3ccccc3F)nn2CC(N)=O)c(=O)n1 N1(C(CCC)=O)CCCC(CO)(NC(=O)C=C(C)C)C1.c12cccc(c1)C(=O)N2 N1(C(C2CC(CC)C2)=O)CCCN(C(c2nocc2C2CC2)=O)CC1C(C)C N1(C(C(CSC)O)=O)CC2(NC(c3ccon3)=O)CCC1CC2 c1(OCC)ccc(F)cc1S(=O)(=O)NC1CCN(C(c2n[nH]cc2I)=O)C1 c1(C(=O)NCC2N(C(c3c(C#N)csc3)=O)CC(F)C2)ccc2c(c1)CC2 C(C(=O)NCC(C)(C)NC(c1occc1C)=O)(C(C)C)c1cnc(C)s1 CN1CCC(CC(=O)NC2CC2NC(c2ccoc2Cl)=O)C1=O C(=O)(C(C)(C)CC(C)(C)C)NC1CCN(C(CN(CC)CC)=O)CCC1CO Cn1nc(C(=O)NCc2csc(CNC(c3cnoc3C3CC3)=O)n2)cc1O c1(OC)ccccc1C(C)CC(=O)NC1(CO)CN(C(c2c[nH]c(=N)s2)=O)C1 C1(NC(CN(CCC)C)=O)CN(C(=O)Cn2nc(C)oc2=O)C2CCCCC12 CC1(CNC(=O)C(F)OC(F)(F)F)CCCN1C(=O)CC1CCCNC1=O CN1CCC(C)(C(N2CCC(NC(=O)Cn3ccc(Br)n3)C(O)C2)=O)CC1 C1(CC(=O)NC2CC(C)OC2=O)CC2(C1)CN(C(=O)C(C)S(N)(=O)=O)C2 N1(S(CC(=O)OCC)(=O)=O)CC(CO)C2(CN(C(c3cc(F)c(Cl)nc3Cl)=O)C2)C1 c1(C(=O)NC(CCC)CNC(c2cc(C3CC3)sn2)=O)cnc2cccc(C)n12 C1(O)(CNC(CCCN(C)C)=O)CCN(C(c2ccc(CCF)cc2)=O)C1 C1(C(=O)Nc2ccc(F)cc2)CCCN(N2CCC(n3cccn3)C2)C1 CN1CCN(C(C2CCC(=O)N(C)C2)=O)C(C(=O)NOC2CCCCC2)C1 N1(C(c2n(CCOC)ncc2)=O)CCCCC(CNC(=O)C(F)=C2CCC2)C1 c1(C(N2C(CCNC(CCC(C)OC)=O)COCC2)=O)cc[nH]c(=N)c1[N+](=O)[O-] CN1C(=O)CCC1C(=O)NCCC1CC(NC(c2ncoc2Br)=O)C1 c1(CCC(=O)NC2C(NC(c3c(C)ncn3C)=O)CC2)ccc(F)c(F)c1F c1(COC)cc(C(N2CC3CC2C3CNC(=O)CC2(C#N)CC2)=O)ccc1NC Cc1cccc2c(C(N3CCOCC3CNC(=O)C(C)OCC(C)C)=O)coc12 C(=O)(CCS(N)(=O)=O)NC(C)CCNC(=O)C(c1ccccc1F)(C)F N1(C(CC2C(C)C2(F)F)=O)CCCN(C(=O)C=CC(=O)N(C)C)CC1 c1(NC(c2c(-n3cccn3)cccc2F)C)cccn2nccc12 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCC2CN(C(=O)CN(c3ccncc3)C)C2C1 C1(NC(c2n[nH]c(CC)c2C)=O)CCCC(C(=O)N(C)Cc2n[nH]c(C)n2)CC1 C(C)(C)(CCCCC(=O)N1CCCC(CN(C)C(c2cccc(O)n2)=O)C1)OC CC12CCC(C(N3CC4CCCC3(CNC(c3cccnc3)=O)C4)=O)(CC1)CO2 C(=O)(C(CNC(C1(C)CCCC1O)=O)CC1CC1)NCC1(C)CCC1 C(=O)(CC(C)C(=O)OC)NCCC(=C)CNC(C1(COC)CCC1)=O c1(-c2occ(CC(CNC(NCC3N(CC)CCC3)=S)C)n2)cc(C)cc(F)c1 c1(SCC(N2CCN(C(C3CC(C(C)C)OC3)=O)CC2)=O)cc([N+](=O)[O-])n[nH]1 C#CC1CC2CCC1N(C(=O)CC13CCC1CN(C(c1cc(OC)no1)=O)C3)C2 Cc1coc(C(N2CCCC2CN(C)C(C2CCCC(C(F)(F)F)C2)=O)=O)c1C c1(N2CC(NC(C3(OC)CCOCC3)=O)C(C)CC2)ncc([N+](=O)[O-])cc1Br c1(OC)nc(C)ccc1C(=O)NC1CC(F)(CNC(=O)CNS(N)(=O)=O)C1 O=C(C1Cc2c(Cl)cccc21)N1CC(C(=O)OCCC2CCCCC2)OCC1=O C1(C(c2n(CC=C)nnn2)NC2(CCOC)CCC2)CC2(C1)CC(O)C2 C(CCS(N)(=O)=O)NC(C1CC(CNC(C(C2CC2)OC)=O)OC1)=O N1(C(c2ccc(C)nn2)=O)CCC(CNC(c2nnc(O)cc2O)=O)C1(C)C N1(CC(=O)NCC2(NC(CNC(=O)NC)=O)CCCC2)CCS(=O)CC1 N1(C(C2C(=C)C2)=O)CCc2c(c(CNC(=O)CCc3cccnc3)nn2C)C1 c1(C(=O)NCC2CC(NC(Cc3nc(C)oc3)=O)C2(C)C)cc(C#N)ccc1Cl c1(C(=O)NCCC2CC(NC(C=C(C)C(C)(C)C)=O)C2)csc2c1CCC(C)C2 N1(C(CNC(CCCCC)=O)=O)CC(NC(c2ncn(C(C)C)n2)=O)CCC1C Cc1oc(Br)cc1C(=O)NC1CCN(C(C23COC(CF)(C2)C3)=O)C1C1CC1 CCCN=C(NCc1cn(C)nc1-c1ccccc1)NC1CSC1(C)C C1(CCNC(c2ccc(C#C)cn2)=O)CN(C(=O)C=C2CCCC2)CCS1(=O)=O N1(C(c2ccc(=N)[nH]c2Cl)=O)CC23CCCCC2(C1)CN(C(=O)CCF)C3 CCC(C(=O)N1CC(CC(=O)NC(C)CN=[N+]=[N-])(OC)C1)n1cncn1 Cn1nc(C(=O)NCCc2cc(C(=O)NCC3CCCCCC3)no2)cc1O N1(C(Cc2c(C)cco2)=O)CCCCC(NC(=O)CCCC(F)F)C1 c1(CC)cccn2nccc12.C(=O)(C(C(=O)N1CCC(C=O)C1CC)OC)OCC C(CC(=O)NCC1CC1NC(C1(C(N)=O)CC1)=O)(C(C)C)OCC c1(OC)ccc(F)cc1CC(=O)NCC1CC(NC(=O)C(C)(C)O)CCO1 CCC(C(=O)NCCNC(=O)NC)NC(=O)C=Cc1ccsc1 c1(CC)nnc2cc(NC3CC(NC(=O)CC4CC(C)(C)CO4)C3)ncn12 C1(C(=O)NC2(C)CC=CC2)CCN(C(=O)C(O)C(F)(F)F)C(C)(C)C1 C1(C(N2CCCC2CCNC(C2(CCF)CCC2)=O)=O)CC2C=CC1O2 C(CC(=O)N1CC(C)(CO)CC1(C)C)(C(C)(C)C)NC(CN(C(COC)=O)C)=O CN(CCCC(=O)NCCC1(CNC(c2cncc(Br)c2)=O)CC1)N=O c1(N(CC=C)C)cc(NCC)nc(NC(C)Cn2cccn2)n1 C1(N(C)C(C2CC23CCCC3)=O)CN(C(c2cnc(C3CCC3)o2)=O)CC1(C)C C(CN=c1[nH]cncc1I)C1CCC(NC(c2ccoc2Cl)=O)C1 C1(C=C)(C(=O)NC(C#C)CC2CCCC2)CCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(C(N2C3CN(C(Cc4nc(C)[nH]n4)=O)C(CC3)C2)=O)cnc2onc(C)c2c1 N1(C(C(C)n2cccn2)=O)CCN(C(=O)C2=COCC2)CC1c1ccccc1Cl Cc1cc(C(=O)NC(C)C(CO)NC(c2csc(=N)[nH]2)=O)c(C)o1 C1(C(C)O)COCCN1C(=O)C(O)CNC(c1ccnc(CO)c1)=O CCCCCC(CC)C(=O)NC1(C2(COC)CCCCC2)CC1 C(=O)(C(F)C(C)CNC(c1cccc(F)c1)=O)N1CC(c2c(C)con2)C1 N1(C(C(CC(C)C)F)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 C(=O)(CC(C)(C)CCOC)N1CCC(N2CCN(C(CCCCOC)=O)CC2)C1 c1(OC)ccc(CC(C)C(=O)NC(CNC(=O)CNC(N)=O)C(C)C)cc1OC CS(C)(=O)=NCC(=O)NC1(C(=O)NC2CC(=O)NC2=O)CC1 c1(C(=O)NCC(C)NC(=O)C2Cc3c(Cl)cccc32)nnc(O)c2ccccc12 c1(C(=O)OCC)ccc(S(=O)(=O)NCCN2CCOC(C)C2)cc1[N+](=O)[O-] c1(C(=O)NCCN(C(=O)CC2CCC3(CCC3)CO2)C)csc(N=S(C)(C)=O)n1 C1(NC(COc2ccc(C)cc2Br)=O)CCCCN(C(=O)C#CC2CC2)CC1 CCCCC(C(=O)NCCCCCCCNC(=O)CC)ON=C(C)C n1(CCNC(C=CC(C)C)=O)cc(C(=O)NC2(CO)CC(F)C2)nn1 C(=O)(C1=CCCN(C(=O)CNC(=O)OC)C1)NC(CCSCC)C N1(C(C(C=C)O)=O)CCC(C)(C)C(NC(C2CCCC2)=O)C1 c1(C(=O)OCC(CSCC)(C)C)c(OC)cccc1O Cc1cc(F)cc(C)c1C(=O)N(C)C(c1cn(-c2cccc(Br)c2Cl)nn1)C C(=O)(C(CO)C(C)(C)C)NCC(C)NC(c1c(C)nsc1)=O N1(C(C(CC)C)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC12CCC2 c1(C2C(C(=O)NC(CC)CN(C)C(C3CCCO3)=O)C2)c(C)cc(C)nc1O C(=O)(C(F)CC1CC1)N1CC(C(C(=O)NC2(CC3CC3)CC2)O)C1 C(=O)(CS(=O)(=O)CC(F)(F)F)NCCC1(NC(COCCC#C)=O)CC1 N1(C(Cc2nnc(C)o2)=O)CCC(O)(CNC(=O)C(C)Cn2ccnc2)C1 CC(=O)CCN=C(NCc1nnc2n1CCCCC2)N1CCC(c2nncs2)C1 C#CC1CN(C(c2cnc(O)o2)=O)CCN1C(c1ccc(C)c(C)c1)=O C12(CNC(Cc3cc(C)no3)=O)CC(NC(c3csc(C(C)C)n3)=O)(C1)C(C)O2 c1(C(=O)NC2CC(C)(NC(c3oc(C)c(CSC)c3)=O)C2)cn2cnnc2cn1 C=C(C)C1OCCC1C(=O)NC1CC2(C(=O)NC(c3ccco3)CO)COC1C2 C(=O)(C(C)C(F)(F)F)N1CC(OC)C(NC(c2cnsc2C)=O)C1 N1(C(C(CCC)C(=O)OC)=O)CC(NC(C2CCCC2F)=O)CC12CCOC2 Cc1ccc(C2CC2C(=O)NCCOC(C)(C)CNC(=O)CC2CC=CC2)s1 Cc1cc(C(=O)N(C)CC2(CNC(=O)CN(C)S(N)(=O)=O)CC2)ccc1[N+](=O)[O-] N1(C(C=CC(C)C)=O)CCC=C(c2ccccc2O)C1 N1(C(CNC(=O)OC)=O)CC2CCCC1CN(C(c1csc3nnsc13)=O)C2 c1(C(N2CCCC(NC(CC3(C)CCCCC3)=O)CC2)=O)cnc2n1CCCC2 c1(CC)cccc(C(N2CC(NC(C3CCC(CC(F)(F)F)CC3)=O)C2)=O)c1N C1(F)(CNC(C=NOC)=O)CCC(NC(c2c[nH]nc2-c2cccc(Cl)c2)=O)C1 S(=O)(=O)(c1cc(Cl)c(Cl)s1)N1C2CN(C(CN3C(=O)CCCC3)=O)C(C2)C1 c1(C(=O)NCCCC(C)NC(c2scnc2Cl)=O)ccc(=O)n(O)c1 c1(N2CCC(c3c(C)con3)C2)nc2c(F)c(Br)cnc2[nH]1 C(c1cccc(Cl)c1)=CC(N1CC(NC(=O)Nc2ccc(CC)cc2)C1)=O N1(C(CCc2ccc(C)o2)=O)CC(C(=O)NCc2ncccc2Cl)CC1(C)C C1(NC(c2c(C)nc(Cl)s2)=O)CN(C(c2c(F)cncc2F)=O)CC(F)(F)C1 C1(C(=O)NC(C2N(C(C(CC3CC3)OC)=O)CCC2)C)CCC(F)(F)C1 c1(OC)nc(C)c(C(N2CCCC2C(C)NC(c2c(C)cnn2C)=O)=O)s1 N1(C(Cc2c(COC)cccc2)=O)CCCC2CN(C(=O)CS(=O)(=O)N(C)C)CC12 c1(C(=O)NCC(N(C(=O)C(C2CCOCC2)O)C)C2CC2)nn(C)cc1Cl N1(C(c2ccc(OC)c(C(C)(C)C)c2)C(=O)NC)CC(C)C(N=[N+]=[N-])C1 C(CC(C(=O)NC(c1ccccc1F)C)NC(=O)CCCOC)=CC N1(C(c2c(C)ncnc2O)=O)CCCC(O)(CNC(=O)C(F)(F)C(C)C)CC1 CCCC(CC(C)C)C(=O)N1CC(F)CC1C(=O)N(CCC(=O)NC)C N1(C(C(CC)CC)=O)CCCC1C1CCCN1C(=O)COc1ccc(C)cc1 C1(CC(=O)NC2CCC(CNC(c3c(CC)noc3)=O)C2)CN(C)CC1O c1(NC(=O)NC2CCC(C)C2)ccc2c(Br)nn(C)c2c1 C1(CCNC(CCCOC)=O)CCCCN1C(=O)C(C)Cn1ccnc1 C1(C2CCN(C(C3NC(=O)CC3C)=O)C2)(NC(CC2C(C)C2)=O)CC1 c1(C(=O)NC2(C)CCN(C(c3sccc3C#N)=O)C2)cc2ccc(F)cc2s1 Cc1csc(Cl)c1C(=O)NCc1cccc(NC(=O)COCCF)c1 N1(C(C2(N(C)C)CCCSC2)=O)C2CCC1C(NC(=O)C(F)(F)F)C2 C(=O)(C1=C(Cl)CCC1)N(CC)CC1CCN(C(=O)C(c2ccc(F)cc2)F)C1 CC(C)CCCC(=O)NC(CC1CC1)C(=O)NCC(C)(C)C(F)F C(=O)(C(C)(C)C(=O)NCCn1ccc(C(=O)NCC(=O)Nc2cnn(C)c2)c1)OC C1(NCCC(=O)OC(C)(C)C)CCCCC1CNC(=O)CCCn1ccnc1 N1(C(c2c(C)nsc2N)=O)CCC(C)C(NC(=O)CC2(C)CC2(Cl)Cl)C1 C1(NC(C=C(C)Cl)=O)CC(CO)N(C(=O)CCC=CBr)C1 N1(S(CC(=O)NC(=O)NCC(F)F)(=O)=O)CCNC(=O)C1c1cccs1 C1(NC(c2cc(=O)cc[nH]2)=O)CC2C1CCN2C(c1cc(C(F)(F)F)no1)=O c1(C(=O)NC2CCN(C(CC#N)=O)C2)cc(Br)cc([N+](=O)[O-])c1F C1(C(N(CCCN(C)C)CCNC(C2CCCCO2)=O)=O)COC2(CCC2)CO1 CC1CCN(C(=O)C(=O)N(CCCNC(C2CC2Cl)=O)C(C)C)CC1 N1(C(c2c(CCC)n[nH]c2)=O)CC2(CCC2NC(c2csc(C(F)F)c2)=O)C1 C1(C(N2CCC(CN(C(c3cc(C)sc3C)=O)C)C2)=O)CCCNS1(=O)=O CCC(O)CC(=O)N1CC2CC1C2NC(=O)C=C=C(C)C N1(C(c2n(C)ncn2)=O)CCC(NC(=O)CC(C)(C)C2CC2)C12CCC2 C(=O)(CC(O)C(C)CC)NC(CCC=C)C(=O)N1CC(C(C)O)C1 c1(OC)cc(OC)cc(C=CC(N2CCN(C(=O)CC3(C)CC3)CC2CF)=O)c1 C1(C(=O)NCCOC2CCN(C(C=CCC)=O)C2)CCS(=O)(=O)N1 N1(C(c2ccnc(C(C)C)n2)=O)CC(NC(=O)C2=NOCC2)CC2(CC2)C1 C(=O)(CN=S(C)(C)=O)NCC(C1CCC1)NC(CC(c1c(OC)cccc1)C)=O C1(CC(=O)N(CC(C)NC(=O)C=Cc2ccnn2C)CC)CCOC(C)(C)C1 Cc1cccc(O)c1C(=O)NC(C1CCN(C(C2CCCCC2O)=O)C1)C c1(C(=O)NCC(C(C)(C)C)NC(c2cnc(CC)[nH]2)=O)cc(C)c(Cl)cc1F C(=O)(CC(C(F)(F)F)NC(C1CCC(=O)N1)=O)NCCc1c(C)nn(C)c1 CC1=C(CNC(=O)C(c2cccs2)NC(=O)CC2C=CCC2)COCC1 N1(C(C(CC)CCOC)=O)CC2CCCC(C1)N2C(=O)CC(C1CC1)C1CC1 c1(OC)cc(S(=O)(=O)NOC2CCOC2)ccc1F C1(CC(N2CC(N(C)CC)C2)=O)CN(C(c2cc[nH]c2C)=O)CCC1C N1(C(C=COCC)=O)CCC(O)(CCNC(C2CC3CC3C2)=O)C1 N1(C(C(=O)NCC)=O)CCN(C(=O)CCc2ccnn2C)CC1C1CCC1 C1(C)(CC)CCN(C(=NC)NCC2(Sc3ccc(N(C)C)cc3)CC2)C1 c1(C(N2CCCC(CCNC(CC(CC)C)=O)C2)=O)cn2cc[nH]c(=O)c2n1 C1(C(N2C(C3(NC(=O)Cc4csc(S)n4)CC3)CCCC2)=O)CC2(C1)CC21CC1 CCCCCCC(C)C(=O)NC1CCC(C)(NC(=O)C2=NNC(=O)CC2)CC1 c1(NCC(=O)NC(C)(CNC(=O)CCN2CCCC2)C2CC2)ccccc1Cl Cc1cc(CN2CCC(O)C(C(=O)NCc3ccccc3CBr)C2)c(O)c(Br)c1 N1(C(CC2C(C)(C)C2)=O)CC2(C1)CN(C(C13CCCC(CO1)C3)=O)CCO2 c1(C(N2CCN3CC(O)CC3C2)=O)cc(O)nc2ccc(Cl)cc12 C1(O)(C(C)NC(=O)CCc2cnn(C)c2)CN(C(c2coc(CO)c2)=O)C1 C(CCCCC(=O)NCC1OCC2CCC1C2)N(C(=O)C(CN(C)C)N(C)C)C C1(C(=O)NC(C)CCCCNC(=O)CCc2ccccc2)CCOCC12CCC2 C12(NC(=O)C(F)F)CCOCC1CN(C(c1cc(F)ccc1C(F)F)=O)C2 O=C1CCCC(C(N2CCC(NC(c3cnncc3O)=O)CC2)=O)CC1 C(=O)(C(F)(CNC(=O)C(C)NC(=O)OC)C(C)C)Nc1ccc(CC)s1 CCC(C)(C(=O)N1CC(NC(c2ccc(Cl)c(C)c2O)=O)C2(CC2)C1)C(N)=O C1(NC(C(C)O)=O)CCC(C(=O)NCCC(O)CO)OC1 CCCCCC(O)C(=O)N1CCCCC1CCCNC(c1cnc(N(C)C)s1)=O N(C1CC2(CN(C(=O)CCc3cnccn3)C2)n2ccnc21)C(COCC#C)=O N1(C(c2c(C)onc2-c2ccccc2)=O)C2CCC1CC(NC(=O)CC(C)O)C2 N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(=O)C=C3CCC(C)C3)CC2C1 n1(CC)ccc(C(N2CC(NC(=O)C(N3CCCC3CO)=O)C(O)C2)=O)cc1=O Cc1c(C(N2CCC(C(C)NC(=O)C(C)(C)CF)C2)=O)cnn1Cc1ccco1 N1(C(C2C(C(=O)OC)C2)=O)CC2(C1)CN(C(=O)CCc1ccc(C)o1)CCO2 C1(C(=O)NCc2ocnc2C(=O)NCC23CCC(CC2)C3)CCS(=O)(=O)C1 N1(C(c2ccc(OC)nn2)=O)CC(NC(=O)CC(C)SC)CC(F)C1 C1(C(=O)NCCCC(c2ccccc2)NC(COC(C)C)=O)CC2CCC2C1 C1(NC(C2CC(OCC)C2)=O)CC2CCC(C1)N2C(C1CCS(=O)(=O)C1(C)C)=O C(=O)(C1=CCCCO1)N1CC(N(C(COCCCC)=O)CC2CC2)C1 c1(OC)ncc(F)cc1C(N1CCC(CC(=O)Nc2ncc(CO)cc2Br)C1)=O c1(C(=O)NCCCC2(NC(C3C(CC)OCC3)=O)CC2)cc2cc(Cl)cnc2o1 N1(C(C2C(OCC)C2C)=O)CCC2(CCN(C(c3csc4nnsc34)=O)C2)C1 c1(C(N2CC(F)(CNC(CCCCCOCC)=O)C2)=O)onc2cc(C)ccc12 c1(CNC(=O)NC(c2ncoc2-c2cccs2)C(C)C)cccc(C(F)F)c1 C(=O)(C1=CC2C=CC(C1)C2)N1C(CCCNC(CCSC)=O)CCCC1 C1(C2CCCN(C(C3(C#N)CCCOC3)=O)C2)(NC(C(CC)C(C)C)=O)CC1 O=S(=O)(c1ccc(OC(F)(F)F)c(F)c1)NC(CC(F)(F)F)C(=O)O C1(NC(CCCCC#C)=O)CCN(C(c2cncc(N)c2)=O)CCC1CO c1(NC(CN(c2ccccc2)CCC=C)=O)ccc(C(=O)OC)c(OC)c1 C1(C)(C(N(CCN(C(CS(CC)=O)=O)C)C)=O)CCC(C(=O)OC)C1(C)C C1(CN(C(=O)C(C)NC=O)CC)CCN(C(C2CCCOC2C)=O)CC1 CCC(CC)C(C(=O)N1CCS(=O)(=O)C(CCNC(=O)CC(C)(C)OC)C1)OC C1(C(=O)NC(c2ccccc2F)C(C)C)NC(=O)OC1C c1(OC)cc(C(=O)NC(C(N2CCCC2C(=O)N(C)C)=O)C2(O)CCC2)on1 C(=O)(CCC(=O)NN(C)C)N1CCCC(CCC)(NC(=O)C(C2CCC2)OC)C1 N1(C(CCNC(C2C(C)C2)=O)=O)CCCC(CNC(=O)CC2CCC(O)C2)CC1 O=C(C1SCc2cccnc21)N1CCC(CF)C1 N1(C(c2c(C)nn(CC)c2C)=O)CCC(C)N(C(c2cnc(C)cn2)=O)CC1 c1(CC(=O)NCC2(CNC(C(c3ccn(C)c3)C)=O)CCC2)cccnc1 C(N=c1nc2scnc2c(NCc2onc3c2CCCC3)[nH]1)c1c(Cl)cccc1 N1(C(c2cccc(C)n2)C(=O)NC2CCOC2)Cc2cncnc2C1 C12(NC(c3cnc(O)c(Cl)c3)=O)CCC1CN(C(=O)C(F)(F)c1ccccn1)C2 C12CC(C1)CCC(=O)O2.N1(C(=O)OC(C)(C)C)CCC1C(=O)NC1CCOC1 C(c1ccc(Cl)cc1F)=CC(N1CC2(CCN(C(C34CC(F)C3C4)=O)C2)C1)=O c1(C(N2CCCN(C(=O)CC3CC(F)C3)C(CO)C2)=O)cccc2scnc12 c1(CC(=O)NC(CNC(C2N(CC)CC2)=O)(C)CO)ccn2cncc2c1 Cc1nc(N2CCCC(C)(CNC(c3cc(CF)on3)=O)C2)cc(C#N)n1 N1(C(c2ncn(C)n2)=O)CC2CCCC(NC(c3[nH]nc([N+](=O)[O-])c3Cl)=O)C2C1 c1(C(=O)NC2COC3(C2)CN(C(=O)CCn2ccnn2)C3)ccc2c(c1)COC2 c1(C(=O)NC(CC(C)NC(=O)CCc2n[nH]c(=N)s2)C)ncn2c1COCC2 N1(C(C(C=C)O)=O)CCN(CC2CN(C(=O)C=Cc3ccco3)C2)CC1 CC(C)C(O)C(C)C(=O)NC(C1(O)CCCCC1)C(=O)NCCCOCC1CC1 N1(C(C(c2ccccc2)OC)=O)CCN(Cc2ccncc2)C2CC12 c1(OC)c(C(N2CC(CNC(=O)C(C)C(C)(C)O)C2)=O)ccc2c1CCC2 c1(CC(COC(N2CCCCC2CC(=O)CCC)=O)OC)cccc(Br)c1 c1(CC)ccc(C(C(=O)NC)N(CCOCCO)CCN(C)C)s1 CCCCC(CNC(c1ccc(COC)[nH]1)=O)NC(c1cc(Cl)ccn1)=O CON(CCC(=O)N1CC(C2CCC(C)(C)C2)C1)C(=O)C(F)n1ccnc1 N1(C(CC(C=C)CC)=O)CCOC2(C1)CN(C(=O)C1=CCCCO1)C2 Cc1ccc(NCC(=O)NCC2C(C)CCCN2C(=O)CC2=CCCC2)c(Cl)n1 S(=O)(=O)(c1cccc(N2CCOC(C)(CCO)C2)n1)N1C(C)CCCC1 Cc1c[nH]cc(C(=O)NCC(O)CNC(=O)CCn2ccnn2)c1=O C1(C)(C(N2CCC(CC)CC2)=O)CCCN(Cc2ccc(C(C)(C)C)cc2Br)C1 c1(C(C)(C(=O)N(C)CCN(C(=O)COCC(C)C)C(C)C)OC)ccccc1F c1(C(N(C)CC2CCCN2C(=O)CC(C)(C)O)=O)c2c(nn1C)CCS(=O)(=O)C2 c1(C(=O)NC(CN(C(C(C)NC(C)(C)C)=O)C)C)cc(O)nn1C C1(NC(Cc2cn(C)nc2)=O)COCCC1C(N1CCC(F)C1)=O c1(CC)cnc(O)c(NC(=O)NCC2(O)CCCOC2)c1 C1(C(=O)NCC2C(CNC(C3(OC)CCOCC3)=O)C2)CCc2nc(C)cn2C1 C(C(F)C(=O)N1CCC(CN2CCC2)C1)C1CN(C(=O)CC2CC(F)C2)C1 c1(-c2nnc(CC(=O)NON3CCOCC3)o2)ccc(Cl)cc1Cl C1(NC(Cn2c(CCC)ncc2)=O)CC(C)CN(C(=O)CCCC(N)=O)C1 CC1(C)CCC(CC(N2CC(NC(C3CC(=O)NC3(C)C)=O)C(O)C2)=O)CC1 CCC(O)C(CC)NC(=O)CC1CC1CNC(=O)C(C)(F)F N1(C(CN(CC(=O)Nc2cnn(C)c2)C)=O)CCSC2CCCC12 c1(C(=O)NCC(CNC(C(C)(C)N2CCCCC2)=O)F)cc(F)ccc1Cl N1(C(CCC(=C)C)C(=O)NCC)CC23CCCCC2(C1)CS(=O)(=O)C3 C12(C(=O)NC(C=C)C3CCC3)CCCC1CCN2C(=O)C=CC(F)(F)F c1(C(C(=O)NCCCC(C)(C)NC(=O)C=CSC)OC)ccc(Br)cc1 C(=O)(C1c2c[nH]nc2CCC1C)N(CCCNC(c1n(CCC)ncc1)=O)CC Cc1cc(Cl)ccc1CC(=O)NCc1cc(Br)ccc1F C1(O)(CCN2CCCC(NC(N3CCC(COC(C)(C)C)C3)=O)C2)CCCNC1 N1(C(C(C(=O)OCC)C2CC2)=O)CC(NC(C2(OCC)CCC2)=O)C(C)(C)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CC(C2CN(C(=O)C(C)Cc3ccco3)C2)C1 N1(C(COCCC=C)=O)CCN(C)C(C(=O)NC2(C)CCCC2(F)F)C1 C1(NC(=O)C(C2CCOCC2)O)CCN(C(=O)NC2CC2c2ccc(Cl)s2)CC1 C1(CCC)CN(C(c2cc(OC)n(C)n2)=O)CCN1C(c1cnncc1OC)=O C1(CNC(=O)CN2CCOC2=O)C(C2CC2)CCN1C(=O)CC1CN2CCC1CC2 C(CCCCC(=O)NCCc1cc(C(F)(F)F)co1)n1cc(C(C=C)(C)O)nn1 c1(C2N3CCC(C3)NC2=O)nc(F)ccc1Br.C#CC(C1CCC1)OCC c1(C(=O)NC2(CNC(C(CC)C#N)=O)CCCC2)c(F)cccc1[N+](=O)[O-] O=C(CS(=O)C(F)(F)F)NC1CCC(CNC(c2ccc(C3CC3)nc2O)=O)C1 C=C(Cl)C(C)(C)C(=O)N1CC2CC(C1)C2NC(c1[nH]c(C2CC2)nc1C)=O C(=O)(CCC(=O)NN(C)C)NC1C(C=C)CN(C(C2(CSC)CC(F)(F)C2)=O)C1 c1(CC(C(=O)OC)N(C)C)ccc2c(c1)CCN2.C12(OC(C)(C)C)CN(C1)C2=O Cc1nc(NC(c2ccc(O)nc2)=O)sc1CNc1cc(OC(C)C)ncn1 CC(CC(C)(C)C)C(=O)N(C(C)(C)CC(=O)N1CC(O)C(F)C1)C O=C1CCC(CC(N2CCC(Cc3cn(Cc4ccccc4)nn3)C2)=O)O1 c1(C(=O)NCCn2cc(Cn3nccc3C(=O)O)nn2)ccnc2ncnn12 C1(OC)CN(C(=O)OC(C)(C)C)C(C(N)=O)C1Nc1cn(CCN(C)C)nn1 c1(C(=O)NC2C(CNC(c3ccc(C(F)F)cc3)=O)C2)cc(O)cc(F)c1 Cc1ccc(NC(c2ccc(F)cc2NC(=O)OC(C)(C)C)=O)n2ncnc12 c1(C(N(C2CCN(C(=O)C(C)O)C2)CCC)=O)cc(F)c(OC)c(Cl)c1 N1(C(C2N(C(CNC(C)=O)=O)CCC2)=O)CCN(C(C2CC(=O)N(O)C2)=O)CC1 c1(OCCCC(=O)Nc2ccnc(N3CCN(C)CC3)n2)ccc(Cl)c(Cl)c1 N1(C(C23CCC(C(C)=O)(C2)C3)=O)CCCCC(NC(C2(C)CC(C)=NO2)=O)C1 C1(NC(C(C)N(C)C(c2cc[nH]c(=N)n2)=O)=O)CCC(O)C(O)C1 C1(C(=O)NCC(=C)CCNC(=O)CC(C)n2cccn2)CC(=O)N(C(C)C)C1 C(=O)(CCCC(=O)OC)N(C)CCN(c1ccccc1)C(=O)COCCCF Cc1c(F)ccc(Br)c1C(N1CC(NC(c2n[nH]cc2N(C)C)=O)C(O)C1)=O N1(C(c2c(CC)ncs2)=O)CCCC(C)C1CNC(=O)CSCc1cscn1 N1(C(CCC(=O)NC)=O)CCOC2(C1)CN(CC(=O)NCCC1CCOC1)C2 c1(C(C(=O)NC)N(CCN(C)C)C2CC2)ccc(CC(C)C)s1 Cc1n[nH]c(=NC2CC3CC(C2)N(C(c2cnc(C)n2C)=O)C3)s1 c1(CC)ccccc1C(N1CCC(CCNC(=O)CCc2cncn2C)CC1)=O c1(C(N(CCCCNC(CCN(C)CCO)=O)C2CC2)=O)ccc2cnoc2c1 N1(C(c2c(C)nc(COCC)s2)=O)CCCCC(CNC(=O)C2=COCCO2)C1 C(C(C)(CO)NC(c1cc(Br)c[nH]1)=O)NC(C(c1cnccn1)C)=O CCC(COC)C(=O)NCC1CC(NC(C2(C)CCCCO2)=O)C1 C1(C(N2CC(NC(C(C)SC)=O)C(c3ccnn3C)C2)=O)CC(=O)NC(=O)C1 C1(C(C)(C)NC(c2cnn[nH]2)=O)CCN(C(=O)C(F)C2CCC2)C1 CCCC(C)C(=O)NC1CCCC(CC(=O)NCc2ncccc2OC)C1 C#CC1(C(=O)Nc2ccc(OC)cc2)CCN(C(=O)CCc2ccc(C)o2)C1 N1(C(CCOCCOCC)=O)CC2(CCC2)CC1C(=O)NC1(C)CCC1 C#Cc1c[nH]nc1C(=O)NC(C)(CO)C(=O)NC1CN(C)NC1=O C1(CN(c2cccc(OC)c2)CCC)Cc2ccccc2C1C c1(C(N2CCN(C(CCc3ccc(C)nc3)=O)CC2)=O)ccc(F)c2occc12 N1(C(C2CCC(NC(C(CCC)O)=O)C2)=O)CCCC2(C=CCO2)C1 Cc1coc(C(=O)N(C(C)CNC(c2cn(C(C)C)nn2)=O)C)c1C CC1CN(C(C2(C(F)F)CCCO2)=O)CCC1CN=c1ccnc[nH]1 C(=O)(C(F)C(=O)N1CC(n2cc(C3CC3)nn2)C(O)C1)OCC c1(C(c2ccc(OCC)nn2)Nc2ccccc2Cl)c(C(F)(F)F)cccc1F C1(C#N)(CC(=O)NC2CC(C)N(C(=O)CSc3cccc[n+]3[O-])C2)CCOCC1 C1(NC(=O)OC(C)(C)C)CCCCCC1NC(=O)Cc1cc(O)cc(Br)c1 c1(C(=O)NC(C2CCOC2)CO)nc(Cl)sc1Cl C1(c2n(C(CC)(C)C)nnn2)(NCC(C)CC2CCCC2)COCC1CN(C)C c1(C(C)=O)cc(C(=O)N(C2CCN(C(=O)CN3CC=CC3)CC2)CCO)oc1C CCC(C(=O)NCC1(NC(C2CC2COC)=O)CCC1)c1ccccc1 C1(CNC(C(C)(C)NC(=O)OC)=O)C2CN(C(C3(c4ccccc4)CC3)=O)CC12 c1(C2(OC)CN(C(c3sccc3C3CC3)=O)C2)ccccc1F Cc1c(NCCCCCC2CC2)ncnc1NC1CCSC(C)(C)C1 C12(C(=O)NCCNC(=O)NC)CC(CO1)N(C(C1CC3C(C1)C3(F)F)=O)C2 C1(OCC(=O)NC(C)Cn2cc(-c3cnn(CCF)c3)nn2)C#CCCCCC1 C(N=c1[nH]c2c(c(=NCc3nc(C4CC4)n[nH]3)[nH]1)COCC2)c1ncsc1 CC1NC(=O)OC12CN(C(C1C=CC(NC(=O)C=C3CCOCC3)C1)=O)C2 Nc1cnnc(NNC(=O)C2CCCCC23CCC3)c1Cl c1(C(=O)NCCC(C)N(CCC)C)cc(CNC(C2CC2Cl)=O)on1 N1(C(Cc2c(C)cnn2C)=O)CC2(CC(NC(C3(N=[N+]=[N-])CC3)=O)CO2)C1 C1(N2C(NC(=O)CCc3nc(-c4cccc(F)c4)no3)CCC2)CCCCCC1 C1(OC)CN(c2nnc(CC(C)(C)O)n2CC(=O)OC(C)(C)C)C1(C)C Cc1cccc(C(=O)NCC2COCCN2C(=O)Cc2cc(F)cc(F)c2)c1Cl C1(C(=O)Nc2cnc(C)c(Cl)c2)CC2(CCC2)CN1C(C1COCC(C)O1)=O c1(C(=O)NCC2C(CNC(C(CC(C)C)(C)C)=O)C2)cccc2c1CCC(=O)N2 c1(NC(C2CC(F)CN2C(c2cncs2)=O)=O)cccc(-n2cccc2)c1 c1(NC(C2(C=C)CCC2)=O)ccc(NC(C2CC2C2CC2)=O)c(C)c1 CS(=O)(=O)C1CC(C(c2nnnn2C2COC2)NCCCN2CCCC2=O)C1 N1(C(c2cc(C)c(C)s2)C(=O)NCC(F)F)CCOC2(CCCCC2)C1 C1(C(N2C3CN(C(CCC=CC(C)C)=O)C(C3)C2)=O)COc2ccc(O)cc2O1 C1(NC(c2ccc(CC(N3CCCCC3)=O)o2)=O)CCN(C(C2CC2Cl)=O)CC1 C1(COC)(NC(c2cnn[nH]2)=O)CCCN(C(=O)CC2CCC2C2CC2)C1 CC(CN=c1cccc(S(=O)(=O)NCCCSCCO)[nH]1)c1nccs1 c1(NCCOCCC=C)nc(C)cc(=NCC(C)c2ccc(F)cc2)[nH]1 C(CC(C)(C)C)(c1n(CC=C)nnn1)(C1CC1)NC1CCCC(C)(C)C1 c1(C(C)(C)C)cccc2c1OCC2C(=O)NCc1sccc1Br C1(O)(CCNC(C(CCO)N(C)C)=O)CCCN(C(c2cscc2C#N)=O)C1 CC(=O)C(C)(C)CC(=O)NC1CN(C(C2CC3CC3C2)=O)CC1CC1CC1 C1(c2n(CCSC)nnn2)(NCc2cccc(Cl)c2Cl)CCCN(C(C)(C)C)C1 C=C=CCCC(=O)N1CCCC(CN(C(C2(N3CCCC3)CC2)=O)CC)C1 c1(-n2nc(C(N(CC(=C)C)C)=O)c(CCO)c2)ccc(F)cc1F O=S(=O)(c1ccc(Br)cc1NCCS)N1CCC2C(F)(F)C2(c2ccccc2)C1 C(CC1CC1)(C(=O)NCCN1CCCCC1)NC(CN(CC(C)C)CC)=O C1(C)(CNC(C2CCN(CC)C2)=O)CCCN1C(C1CCSCC1)=O C1(CNC(COCCC(C)C)=O)(NC(=O)CC2CCCSC2)CC(F)(F)C1 C(=O)(C1CCCc2nncn21)N(CC(C)O)CCNC(=O)CC(C)(C)C C1(N(C(C(CC)(C)C)=O)C)CCN(C(=O)CNC(c2cccc(C)c2)=O)CC1C c1(C(=O)NC(C2CN(C(=O)CC#N)C2)C)ccc(S2(=O)=NCCC2)cc1 Cc1[nH]c2c(F)cccc2c1CCNC(C1CCCCC1C)=O c1(CC)ncsc1C(=O)NC1CCCC1CN(C)C(C1CC(OC)C1)=O N1(C(c2c(C)nc(C(C)C)s2)=O)CCC(CO)C(NC(c2nn(C)cc2Cl)=O)C1 C1(CC(=O)NC(C(C)NC(=O)Cc2cn(C)nn2)(C)C)CCC(=O)NC1 C(=O)(C(C)(C)C(N)=O)NC(CCN(C(CN1CCC(C)C1)=O)C)C(C)C c1(C(C(=O)NC2CN(C(CC(C=C)C)=O)C2)O)ccc([N+](=O)[O-])cc1 c1(C(N(C2CNCCC2(F)F)c2cc(COC)ncn2)=O)cc(F)c(F)c(F)c1 c1(OCCC=C(C)C)ccccc1Cc1cccc(N2CCC2=O)c1 CCCCC(C)(F)C(=O)N1CCC(NC(C2CCC(C)(C)O2)=O)C(F)C1 C(CC1(C)c2nnnn2NCCN1)SC.c1(CC2CCOC2)scnc1C N1(C(Cc2ccc(SC)cc2)=O)CC2(CCCCC2NC(=O)CNC(=N)N)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C2OCCN(C(CC(=O)OCC)=O)C2)C1 N1(C(CC(CC)(C)C)=O)C2CCC1CN(C(C13CCC1C3)=O)C2 n1(CCCNC2C(CC)COCC2)c(C)cc(O)cc1=O N1(C(c2c(CNC(CC3C(=O)NCCC3)=O)ccs2)=O)CCOC2(CCC2)CC1 CN1CCN(C(c2cc(C(F)(F)F)no2)=O)C(CNC(c2ccc(=O)oc2)=O)C1 c1(CN2CCC(C(C)(C)C)(NC(N)=O)C2)ccsc1S(C)(=O)=O.C1(=O)CCCN1 c1(C(=O)NCC(C)CN(C)C(c2cnnn2C)=O)cnccc1N(C)C c1(OC)nc2cc(N(C(=O)CC(C)c3ccccc3)C)ccc2o1 C(=O)(C1Cc2ccc(F)cc21)NC1CCN(C(C(C)NC(N)=O)=O)C12CCCC2 c1(C(=O)NC2C(NC(C3(OC)CCSC3)=O)CCC2)ccc(C2CC2)cc1Cl c1(C(N2CCCC(C)(NC(c3cnc(C)n3C)=O)C2)=O)cccc(S(C)(=O)=O)c1 c1(N(C)Cc2n(CC)cnn2)[nH]c(=NC2CCOCC(C)C2)nc2scnc12 CCCC(C)C(C)Nc1ncccc1C(F)C(F)(F)F CP(C)(=O)C(O)C(=O)NCCN1CCC(NC(=O)CC2CC(F)(F)C2)CC1 c1(CC(=O)NC(C(=O)NC)C2(O)CCC2)ccc(Cl)cn1 c1(C(=O)NC(CC)(CNC(=O)CC2CCCCCCC2)CC)cnc2[nH]cnc2c1 C1(C(=O)NCc2c(C(C)C)noc2)CN(C)CCN1C(C1C2CCC(F)(F)C12)=O c1(C(=O)NCC(C)(CNC(=O)COCc2ccncc2)OC)cccn(C)c1=O Cc1cc(C(=O)NCCNC(C2CC2C)=O)c(C)n1C1CCCCC1 N1(C2CCN(c3nc(=N)[nH]c(=N)[nH]3)C2)C(=O)C2CCCCC2C1=O c1(OC)cccc(C(=O)N(C)CC2CCN(C(=O)Cn3cc(Cl)c(C)n3)C2)n1 N1(C(C(C)N2CCCC2)=O)CC2CC1(C(N1CCC(OCC3CC3)C1)=O)C2 c1(C(=O)NCCC2(CNC(CSC)=O)CC2)cnc2c[nH]nc2c1 c1(C(N2C(C)CN(C(c3c(C)onc3)=O)C(C)C2)=O)cccc(P(C)(C)=O)c1 C1(CCC)(NC(=O)CC(C)(C)O)CCCN(C(c2cnncc2OC)=O)C1 N1(C(c2cc(OC)nc(Cl)c2)=O)CCC2(NC(=O)C=Cc3cnc[nH]3)CCCC12 N1(C(=O)OC(C)(C)C)CC2CC2(NCc2snnc2C2CC2)C1 c1(C(N2CCC(NC(=O)Cn3cc(Cl)cn3)C(O)C2)=O)ccc2sccc2c1O Cn1cc(-c2ccc(C3CC(C)(Cc4ccccc4)C(=O)O3)cc2)n(C)c1=O C1(C(N2CC(NC(c3ccnc4c3CCO4)=O)C(O)C2)=O)CCCC2(CCC2)C1 C(CC(=O)NC1CC2CC(NC(=O)CCSC3CCCC3)C1C2)(C(C)C)OCC C1(C)(COC)CC(NC(=O)C(C)(C)C)CN1C(=O)Cc1ccc(C)nc1Cl N1(C(C(C)Cc2ccccc2F)=O)CC2CCC(C1)N2C(=O)CC1COC(=O)C1 N1(C(c2c(C)csn2)=O)CCCCCC1C(=O)NCc1ccncn1 C1(C(N2CC(N(C(C(CC)C#N)=O)C)C2)=O)CS(=O)(=O)CC12CC2 C1(CC(=O)N(CCCNC(c2ccccc2O)=O)CCO)CCCCC12CC2 Cc1ccc(Cl)c(N)c1C(N1CCC(NC(=O)C(C)NC=O)C(F)C1)=O CCCCC(O)CC(=O)N(C(C(N1CC2CCC(CO)(C2)C1)=O)C1CC1)C N1(C(c2c(C)nsc2-c2ccccc2)=O)CCOC(C)(CNC(=O)OC(C)(C)C)C1 N1(C(c2c(SCC)cc(Cl)cc2)=O)CCC(N(C)C(c2ccon2)=O)C2(CC2)C1 C(=O)(C1=C(C)OCC1)NC(C(=O)NC(CC)CN1CCOCC1)C CCCCCCC(C)CC(=O)NC1CCC(O)CN(C(c2ccoc2CC)=O)C1 Cc1nn(C)c(C)c1CC(N1CCSCC1CCNC(c1cncn1C)=O)=O c1(C(C(=O)Nc2ccccc2)N(C)Cc2c(C)nc[nH]2)csc(S(N)(=O)=O)c1 S(=O)(=O)(c1cc(C(F)(F)F)cc(O)c1)NC(c1c(C)ccc(SC)c1)=O C(CC1CCCC1)(C(=O)N(CCCNC(=O)Cc1cnc(C)[nH]1)C(C)C)OC c1(C(N2C(CNC(C3CCC4CCC3O4)=O)COCC2)=O)ccc2sccc2c1 N1(C(CS(CC)=O)=O)CCCC(C)(NC(c2cnn(C3CC3)c2C2CC2)=O)C1 Cc1cc(F)c(CC(N2CCC3CC3(NC(=O)CN(C)C3CC3)CC2)=O)cc1F Cc1ncc(C(=O)NCCCNC(=O)C(c2ccc(F)cc2F)C)cc1N Cc1ccc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CC2(C)C)=O)nc1 C(C(C)(C(=O)NC1CCCCC1)NC(C1CCCO1)=O)SC Cc1ccc(C(=O)NCC2CC2NC(c2c[nH]nc2-c2cccnc2)=O)c(N)c1 C(=O)(C1Cc2c(Cl)cccc21)N1C(C2(NC(CCCCOC)=O)CC2)CCCC1 C(=O)(CC(C)N(C(c1cc(Br)cs1)=O)C1CC1)NCCCOC c1(C(=O)NC2CC(C(=O)OC)C2)c(OCCCOC(C)C)cccc1NC(C)=O N1(CN(c2ncccn2)CCOC)CCC2(CCCCN(C(=O)OC(C)(C)C)C2)C1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NCC=CCNC(=O)C1=CCCCC1 c1(NCCCCCCNC(C2(C)ON=C(C)C2)=O)ccc(C)cc1[N+](=O)[O-] C=CCC(CNC(=O)C(F)=CCC)C(=O)NCC(C)(O)CC(C)C c1(SCC=C)ccc(C(=O)NCC2CC2C)cc1.N12CC3CC1C3C2=O CCC(=O)CCC(=O)NC(CC1CCC1)C(=O)NC1CN(C)CCC1O C1(NC(C(C2CCCC2)OC)=O)CN(C(=O)CCS(C)=O)CC1(C)C Cc1cc(C)c2onc(CC(=O)NNC(=S)NCC(O)CC(F)(F)F)c2c1 C1(C(C(=O)N(CC(=O)NC)C)C)CCCN(C(=O)C=Cc2cocn2)C1 c1(-c2scc(C(=O)OCC(CO)Oc3ccccc3)n2)ccc(OC)cc1 c1(C(N2CC(N(C(c3c(CC)c[nH]c3)=O)C)C2)=O)cc(O)c2ccccc2c1 Cc1c(F)ccc(C(=O)NC2CCC(N(C(=O)CC3OCCO3)C)CC2)c1C CCC(CC)CCCNC(=O)C(Cc1cc[nH]n1)NC(c1ccc(CO)o1)=O C1(CNC(=O)OCC)CCC(CNC(C2CC2)=O)CC1.C(=O)(C(F)=CCCF)N c1(OC)ccccc1C(=O)NCC(CO)NC(=O)CC1CCC1C c1(CC)c(C(=O)NC2CC(O)(CNC(=O)C(C)(C)OC)C2)[nH]c(C)c1C(C)=O N1(C(CC(CC=C)NC(c2nccs2)=O)=O)C2CCC1CC(CO)C2 c1(C(C(=O)NCC2CCCO2)N(CC)Cc2cnn(C)c2)cccc(COC)c1 Cc1c(CCNC(N2CCCCC(C)(F)C2)=O)ccc(Cl)c1Cl N1(C(C(CC)C(C)O)=O)CCc2nc(NC(=O)C(=O)NCCNC(C)=O)sc2C1 N1(CC(=O)N(CC(C)(C)CNC(c2cn(CC)cn2)=O)CC)CCS(=O)(=O)CC1 C1(NC(C(CCN(C)C)O)=O)C2CCC(C2)C1C(=O)NC1(C(C)(F)F)CC1 C#Cc1ccc(CNC(C2CN(C(C3CC4C=CC3C4)=O)CCO2)=O)cc1 N1(C(CCCOC(C)C)=O)CCOCC(NC(=O)C(c2ccc(Cl)cc2)O)C1 C=C(C)C1CN(C(=O)CC2CN(C(c3cn(C)c(C)n3)=O)C2)CCO1 C1(OC(C)C)CCCCC1NC(C1CCC(=O)N1)=O.N12CCC(CC1)NC2=O C=CC1(C(=O)N(C)CC2(COC)CCC2)CCN(C(=O)CC2CCCNC2=O)C1 C1(OC)CN(C(c2c(Br)noc2C2CC2)=O)CC1NC(c1ccoc1)=O CN1CC=C(C(=O)NC2CC(CNC(=O)CCn3cnc(=N)[nH]3)C2(C)C)C1 c1(-n2ncc(C(=O)NCC(CC)NC(=O)CC3CNC(=O)C3)n2)ccc(F)cc1 C(=O)(C(F)(F)c1cscn1)NCCN(C1CCCC1)C(COCC=C)=O c1(CC(=O)NCCCCC2CN(C(C)=O)C2)cnc(N(C)C)cn1 c1(C(=O)OC)ccc(F)c(Cl)c1.c1(OCCN2C(=O)C2)ccc(Cl)cc1 N1(C(C2C3CN(C(c4c(CC)ncs4)=O)CC32)=O)CCc2ccc(C#N)cc2C1 C(=O)(C(C)(CO)OC)NCC1C(C(=O)NCC(=C)Cl)CC1 CCS(=O)CC(=O)NC(C1(CNC(c2ocnc2CO)=O)CC1)C c1(OC)cc(C)ccc1CNC1CCC(C(=O)NC(c2ccc(Cl)cc2)C)OC1 N1(C(c2nn(CC)c(C)c2)=O)CCC(CNC(c2cc(C)c(C)o2)=O)C12CC2 c1(C(N(CC(CC)NC(c2csc(C)c2)=O)C)=O)cn2ccsc2n1 CN1CC(O)CC1C(=O)NC(C(=O)NCC(F)(F)C(F)F)C1(O)CCC1 C(c1ccccc1Cl)=CC(N1CCC(NC(CC2CN(CC(C)C)C2)=O)C1C)=O C1(C)(NC(C2OCC(C)C2)=O)CCCN(c2ccncn2)C1 c1(C(=O)NC2(C)CN(C(=O)C(c3ccccc3)NC(N)=O)C2)cncc(N)n1 c1(C(N2CCOCC(NC(C=CCC)=O)C2)=O)c(CCC)sc2c1CCC2 C(CC(C(=O)NC(CC1CC1)CC(=O)NCCCC1CCC1)OC)OC N#Cc1cc2cc(-c3cccc(CN4CCCC4CO)c3)cnc2cn1 c1(OC)cccc(Cn2cc(CCCN(C(C3CC3OC)=O)C3CC3)nn2)c1 n1(C(C(=O)Nc2ccc(C)c(Br)c2)C)cnc2ccccc12 C1(CC(=O)N(C)CC2(N(C)C)CC2)N(C(c2cccs2)=O)CCC1(C)C N1(C(=O)C=Cc2cnc[nH]2)CCCC2C1CCCN2C(=O)Cn1ccccc1=O c1(CC)ccc(C(N2CCC(F)(CNC(C3CCCSC3C)=O)CC2)=O)c(F)c1 Cc1ccc(C2CC2C(=O)NC2(CNC(=O)CC3CCCCO3)CCOC2)cn1 C1(C(N(c2ccc(F)cc2)CC)=O)C2CN(C(=O)C(C)(C)CF)CC12 C1(NC(c2cccc(OC)c2)=O)C2CC3C1C3C2C(=O)NOCC(N)=O c1(SC)ccc(N)cc1C(N1CC2CC(NC(C3(C)CCC(=O)NC3)=O)C1C2)=O C1(C)(C(N2CCC(C=C)C2)=O)CN(C(c2cccnc2)=O)CC1C C1(CC=C)(C(=O)N(CC(C)(C)NC(C2CC2C(C)O)=O)C)CCC1 c1(C(=O)OC)ccc(C)nc1NC(C)(CNC(C1CCCN1C1CC1)=O)CC C1(NC(C(CCC)CC)=O)CC2(CCN(C(C3(OCC)CCC3)=O)CC2)C1 N1(C(C(C=C)O)=O)CCOCC12COCCN(C(C1Cc3cccnc3C1)=O)C2 CC(C)CCCCC(=O)N(C(=O)CC(C)C(F)F)CC1CCCOC1c1cn[nH]c1 c1(C(=O)NCC2CCC(NC(C3CC(C#C)(O)C3)=O)C2)nccc(Cl)c1C N1(C(c2cc(CNC(C(C(C)C)O)=O)on2)=O)CCCC2(CCC2)C1 N1(C(c2cc[nH]n2)=O)CC2(CCOCC2)CC1CNC(C1CC(CF)C1)=O c1(CNC(=O)NCC2(CO)CC(C)C2)ccc(O)cc1Br C=C(CC)CN=c1[nH]c(=NCC(CCO)c2cccnc2)c2cc(Cl)ccc2[nH]1 C1(CNC(c2ncn(CCC)c2)=O)CCCCC1NC(=O)C(c1csc(C)n1)=O N1(C(C2OCCN(C)C2)=O)CC2CC(F)(F)CCC2(N)C1 CCC(CSC)(c1nnnn1C1CCOC1)NCC=Cc1ccco1 c1(C(=O)NCC(C)N(C(C(n2ncc(C)c2)C)=O)C)noc2c1CC(C)(C)CC2 c1(C(=O)NCCCCCN(CC=C)C)c(CNC(=O)C=C2CC2)cnn1C n1(CC)cc(Cl)c(C(=O)NCC(C)(O)CNC(=O)C(F)(F)c2cncs2)n1 c1(C(N2CCCC(NC(C=C3CCC(C)C3)=O)C2)=O)ccc2c(c1)COC2(C)C C1(C)(NC(CC2CC(C(=O)OC)C2)=O)CCN(C(c2cc(C)c(CO)s2)=O)C1 C(=O)(C1=CCC(NC(c2c(Cl)cnn2C)=O)C1)NC(CC)C1CC1 N1(C(c2cc(OC)n[nH]2)=O)CCCC(CCNC(C2(O)CCSCC2)=O)C1 C1(NC(c2cccc(C(F)(F)F)c2)=O)CCCCC1NC(C1(F)CC2(CC2)C1)=O c1(C(=O)Nc2cccc3ccc(Br)nc23)cc(C2=CCNCC2)c2[nH]ncc2c1 CC1CCC(CC(=O)NCCOC2CN(C(=O)CSc3cccs3)C2)CC1C C1(O)(C(C)NC(C23CC(C2)C3)=O)CCN(C(C2CCCN2C)=O)CC1 C1(C(=O)NC2(C)CN(C(=O)CC3(C)OCCO3)C2)CC2CCC1C2 C=CC1CN(C(c2cc(F)ccc2F)=O)CC1NC(c1ccccc1SC)=O c1(C(=O)NC2CCCN(C(=O)Cc3ncc(Cl)s3)CC2)cc2ncccc2[nH]1 c1(CC(=O)N(C2CCCC(N(C(C=C(C)C)=O)C)C2)C)c[nH]c2cccc(C)c12 c1(CC)cc(Br)ccc1NC(C1CCCN(C(C2CC2(F)F)=O)CC1)=O c1(SC(C(N2C(CNC(Cc3scc(C)n3)=O)CC2)=O)C)ccc(F)cc1 C=CCC(CNC(C1(CC(=O)OC)CC1)=O)NC(=O)CC(C)n1cccn1 C1(CC(N2CC(C(C)NC(C3CC34CCCC4)=O)C2)=O)NC(=O)NC1=O C1(NC(C2(OC)CC2)=O)CCC(C(=O)N(CCCN=[N+]=[N-])C)C1 C(CCC(O)C(=O)NCc1ccc(CO)cc1)NC(C1(C)CCN(C)C1)=O C(=O)(CC(C)(C)C(F)F)N1C2C(NC(c3c(C)cncn3)=O)CC(C2)C1 C=CC1CN(C(=O)C(C)Cc2ccc(O)cc2)CC1NC(c1cnc(Cl)s1)=O c1(C(N2C(C)CN(C(C3COCCO3)=O)CC2)=O)ccc2nc(CO)[nH]c2c1 C1(NC(c2c(CCC)occ2)=O)CN(C(=O)Cc2nc(C)sc2C)CC(C)(C)C1 N1(C(COC)=O)CCc2ccccc2C(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(C(=O)NC2CC(C)(NC(=O)CCN3CCC3)C2)ccc2ccoc2c1 C12(C(=O)NCC3(SC)CC3)CCN(C(C3CCC3C(F)F)=O)CCC1C2 c1(C(N2CCC(C)(C(=O)NCC3ON=C(C)C3)C2)=O)cc(C)cc(C)c1 c1(-c2ccc(CO)cc2)csc(=Nc2cccc(O)c2)n1Cc1ccccc1Br CCC(CC1CCCC1)C(=O)N(CCCN(C)C(C1CC1c1cnn(C)c1)=O)C C1(NC(CNC=O)=O)CC(C(=O)NC2CC(OCCO)C2)C12CCC2 C1(C)(OC)CCCN(C(C2CC(O)CN2C(=O)C=CC(F)(F)F)=O)CC1 Cc1cc(C(=O)NCC(=O)NCCNC(=O)CC2CCCC2O)c(C)o1 C1(C(=O)NC2CC(NC(=O)C(C3CCOCC3)O)C2)CCCCC(F)(F)C1 C1(NC(=O)COc2ccsc2)CC2CC(NC(c3nc(Cl)cs3)=O)CC2C1 C1(N(C(C(CC)F)=O)CCO)CCN(C(=O)Cc2ccsc2C)CC1 C1(C(=O)NCC2(COC)CCCN2C(=O)COCCC(C)C)CCCS(=O)(=O)N1 c1(C(N2CCC(N(C(=O)C=Cc3cnccn3)CC)C2)=O)c[nH]nc1[N+](=O)[O-] Cc1cc(N(C)C(c2ccccc2F)C)ccc1NC(N)=O N1(C(CC2CCCN(C(C3CN(C)C(=O)CC3)=O)C2)=O)CCOCC(F)(F)C1 C(=O)(C(CC(C)SC)N1CCN(CC(C)C)CC1)NC(C(=O)OC)C CCC(CN(C)C)C(=O)N1CCCC(CCC(=O)NCC(O)COC(C)C)C1 NC1CCN(C(=O)C(=O)NCc2ccncc2)CC1CO C1(c2nc(C(CC)SC)n(-c3cccc(C)n3)n2)CCC(F)(F)CC1 c1(OC)c(C(=O)NC2(C)CN(C(c3c(F)ccnc3F)=O)C2)cccc1F Cc1sncc1C(=O)NC1CCC1NC(=O)CCc1cnc(Br)s1 C1(NC(C(C)C#N)=O)C=CCN(C(=O)CN(C)Cc2cccc(Cl)c2)C1 N1(C(CC(C)OC)=O)CCN(C(=O)C(=Cc2cccn2C)F)CC1C1CCCC1 N1(C(C2(C)CC2(Br)Br)=O)CC(n2cc(CNC=O)nn2)C(O)C1 Cc1cc(C(N2CCN(C3CN(C(=O)C4=COCCC4)C3)CC2)=O)cc(N)c1Cl CC1(C)CCOC(C(=O)NCC2(C)CCCC2NC(C2CCS2(=O)=O)=O)C1 C1(NC(c2cc3occc3s2)=O)CCN(C(=O)CCCC2CCC2)CC1F N1(C(c2ncc(CC)cn2)=O)CCCC2CN(C(=O)CC(C)C(C)(C)C)CCC12 C=Cc1ccc(C(=O)N(C2CN(C(C3(C)CCOC3)=O)CC23CC3)C)cc1 C1(NC(Cn2ncc(C#N)c2)=O)CCCC(NC(=O)C2=NOCC2)CC1 c1(N2CC(C)N(Cc3cccn3C)CC2)ncnc2c1CCC2 C1(C(=O)NC2CCN(C)C2=O)CC(F)(F)CN1C(=O)CCc1c(N)cnn1C C(=O)(C1=CCCC1C)N1CCCC(Cc2cc(N3CCC(OC)CC3)ncn2)C1 N1(C(CC(=C)Br)=O)CCCN(C(=O)CC(C)C(=O)c2cccc(CO)c2)CC1 C(=O)(C1CCCc2nncn21)N(CCC(C(C)C)NC(=O)C=CCF)C C12(C(=O)NCCC(C)(C)N(C)CC)CC(CN1C(C1CCCCN1CC)=O)C2 S(=O)(=O)(c1cc(C(N2CC3CC2CCC3O)=O)n(C)c1)NC(C)C C(=O)(C1SCCc2ccccc21)NCC1C(C)CCN(C(c2coc(Br)n2)=O)C1 C1(C(=O)NCCNC(C2C=CCC2)=O)(CC)CCCN1C(=O)CCOC C1(CNC(c2n(CC)cc(Cl)c2)=O)CCCC2CN(C(=O)C#CC(C)(C)O)CC12 C#Cc1ccc(C(=O)NC2CCCC(NC(C3CC34CC4)=O)C2)c(C)c1 c1(C(N2CCN(S(c3ncn(C)c3)(=O)=O)CC2)=O)ccc2c(c1Cl)OCCO2 C1(CN(C)C(c2ccccc2)=O)CCCCN1C(c1ccncc1F)=O CCC(C(=O)NCCN(C(=O)CC(O)C1CC1)C1CC1)C(C)(C)CC C12(CC(=O)NCC(C)(C)Cn3cc(CO)nn3)COC(CF)(C1)C2 c1(C(=O)NC2C(NC(=O)C3=NOCC3)C2)ccc2c(=O)c3ccccc3sc2c1 C1(C(=O)OCC)Cc2c(F)cc(OC)cc2N1.C123CCC1CN(C2)C3=O N1(CCN(C)C(C2COCCO2)=O)CCN(C(c2ccoc2C(F)(F)F)=O)CC1 c1(C(N(CCOC)Cc2ccccc2C)=O)coc2c1CNC2 c1(OC)cc(C=CC(=O)NC2CN(C(=O)C3CC3)CC23CC3)ccc1O C(CC(C(C)C)NC(C1CCCC1C(C)C)=O)NC(CC1CC(SC)C1)=O C1(CNC(C(CCC)(C)O)=O)CC2CCC(C1)N2C(C1CCCCC1O)=O Cc1cccc(CN(C(=O)C(C2CCOC2)NC(c2cc(C(C)C)on2)=O)C)n1 c1(OCC)ccc(NC(=O)C(=O)Nc2cnn(C)c2C)cc1F N1(C(C2(COCC)CCCC2)=O)CCC(O)(CCN2CCC(C(N)=O)C2)CC1 CCS(=O)(=O)c1cc(F)ccc1CNC(N1CCCC(c2nnc(S)n2C)C1)=O CCC(C)C(O)C(C)C(=O)NC1(C)CCN(CC(O)CC(C)(C)C)C1 C(C(C)(C)CCS(C)(=O)=O)NC(c1ccccc1)(C)C C(=O)(CS(=O)(=O)C(C)(C)C)NC(CCCCNC(C1C(OC)CCCC1)=O)C N1(C(C(C)(C)N(C)C)=O)CCCC12CCCOC2 C1(C(N(C(C)C(=O)NCC(C2CC2)N(C)C)C)=O)CCCCNC1=O N1(C(C(c2ccoc2)NC(CN(C2CC2)CC)=O)=O)CCC(C(F)F)C1 C(C(C)(C)C(=O)NCCC1CCCCN1C(=O)CC1(C#N)CC1)OC c1(C(N(C(=O)Nc2c(C)cco2)C)C2CC2)cccc(F)c1 C(=O)(C(=O)CC(C)CC)NCCN(c1cccc(Cl)c1)C(CN(CC#C)C)=O c1(C(=O)NC(C2CCOC2)CNC(c2cnc(CC)o2)=O)cnc(OC)c(F)c1 C1(C(N(CC(c2ccc(Br)cc2)O)C)=O)NC(=O)C2CCC12 CC1(C)CN(C(C2C3COCC23)=O)CCC1NC(=O)C=Cc1cncnc1O Nc1c(C(=O)NCC2CCCN2C(=O)Cc2ccsn2)cc(F)cc1[N+](=O)[O-] Cc1ccc(Cl)c(C(=O)NCC2COCC2NC(c2cc(C3CC3)nn2C)=O)c1 Nc1c(Cl)c(C(N2CCC(O)(CNC(=O)C(O)CF)C2)=O)nc(Cl)c1Cl N1(C(CN2CC(C)(OC)C2)=O)CCC(C(=O)NC2CC(C)(O)C2)CC1(C)C C1(C)(NC(C(c2ccc(C)cc2)F)=O)CCCN(C(=O)C=C2CCCC2)C1 c1(C(=O)NCCN(C(C2(C)CCCS2)=O)C2CC2)cccc(OCC(F)F)c1 N1(C(C2(C#N)CCCCCC2)=O)CCC(C2(NC(C3CCC4CC34)=O)CC2)CC1 C1(NC(C2C(C(C)C)C2)=O)CC2CCC1N2C(=O)Cc1cccc(F)c1 CC1(CC#N)CCCN(N2CC(Cc3ccc([N+](=O)[O-])cc3)C2)C1 CCC(CNC(=O)CC1CCCC2CC12)(CC)C(=O)N1CCC(C)(C2CC2)C1 Cc1cc(N)c(C(=O)NCCc2ocnc2CNC(=O)CCc2nccs2)cc1C C1(CNC(CC2(CC(=O)OC)CC2)=O)CN(C(C2CCC=CO2)=O)C(C)(C)C1 c1(C(=O)NC2CN(C(COC)=O)CC2SC)cc2n(n1)CCCCC2=O C1(C(=O)NC(C)Cc2ccncc2)CC=CCN1C(c1scnc1Cl)=O N1(C(C2(C)CCN2S(=O)(=O)CCCCl)=O)CCc2cc(Br)ccc2C1 c1(CNC(C(C2CC2)OCC)=O)cccc2c1CCN(C(c1sccc1F)=O)C2 C1(O)(C(C)NC(C(C)OCCCC)=O)CCN(C(=O)C(C)=C2CCC2)CC1 c1(CCN(C(C)C)CC2(C)CC2)cn(CCCO)nn1 N1(CC)C(=O)CCC1C(=O)NCC(C1CCCN1C(c1ccc(O)cn1)=O)(C)C N1(C(C(C)NC=O)=O)CCCC1CC(=O)N(C(C)(C)C)CC1CC(C#N)C1 c1(SC)cc(C(=O)N(CCCCNC(c2[nH]cnc2C#N)=O)C)oc1C C(=O)(C(C)CC(C)(C)C)NCCC1N(C(c2sc(C)c(O)n2)=O)CCCC1 c1(C(N2C(C)CC(NC(c3cccc(OC)c3)=O)C2)=O)cnccc1C#N CC1CCN(C(=O)CC2CCN(C(C3COC4CNCC4C3)=O)CC2)CCC1O C1(C)(OC)CC(NC(C2(NC(C3CC3(C)C)=O)CCC(C)(C)C2)=O)C1(C)C CCCCCCN(CC(=O)NC1(C2CCCN2C(=O)CSC2CCC2)CC1)C.C c1(OC)ccnc(F)c1C(=O)NCC1CC(NC(C2CC(C)OC2=O)=O)C1 C(CC(=O)NCC(=O)N(C(C)CF)C(C)C)NC(C)=O c1(C(C)C)ccc(C(=O)NC2(CNC(c3ccc(C#N)s3)=O)CCC2)c(O)n1 C(CC(CNC(c1snnc1C(C)C)=O)NC(=O)CCc1cscn1)OC CC1CCC2(CO1)CN(C(C1(CNC(=O)CC3CCCC3)CC=CC1)=O)C2 N1(C(c2ccc(C)nc2C)C(=O)NC(C(=O)OC)C)CCC2(CCN(C)C2=O)C1 c1(C(=O)NCC2C(NC(C(CC=C)OC)=O)C2)c(Cl)ccc(OC)c1N Cc1ccc(OCC(=O)NC(C)(C)CCNC(C2(CN(C)C)CC2)=O)cc1 N1(C(c2c(C)nns2)=O)CCc2sccc2C1CNC(C1CC12CC2)=O c1(C(=O)NCC2CCN(C(c3ccc(OC)s3)=O)C2)cc2c(Cl)cncc2s1 Cc1cc(C(=O)NC(CNC(=O)C=Cc2nc(C)cs2)C(C)C(C)C)c(C)cn1 c1(C(N2C3C(CNC(C(=O)N(C)C)=O)C(CCC3)C2)=O)cnc2ccnn2c1 C1(NC(C2CC(C(C)C)C2)=O)COCC1NC(c1cc(-c2ccccc2)[nH]n1)=O c1(C(N(C2CCCN(C(C(CC)(C)C)=O)CC2)C)=O)ccccc1S(C)=O C1(NC(CCC=CC)=O)CN(C(=O)CC(O)CCC)CCC1C Cc1ncc(Br)cc1C(=O)NCC1CC1NC(=O)Cc1ccc(C(F)F)o1 C(=O)(CC(C)CNC(=O)CCC1CCCCO1)NCCn1ncc(C)c1 c1(CC)nc(C)[nH]c1C(=O)NC(C)(C)CNC(=O)CN1CCS(=O)CC1 Cc1cncc(C(=O)NCC2CC2CNC(c2cn(CC(F)(F)F)nc2C)=O)c1 c1(C(=O)NC23CC(NC(C4(NC(C)=O)CC4)=O)(C2)C3)nnn2c1CCCC2 c1(C(=O)NCC(C)(C)OCC(=O)NCC2(F)CC=CCC2)cccc2occc12 CC(C(O)C(F)F)NC(=O)CCOC1CN(C(C2(C)COC(=O)N2)=O)C1 CCCC(CCCNC(c1cccc(CC)n1)=O)NC(c1cnc(C)c(N)c1)=O CC1(C(=O)NC2CCC2N2CCCC2)CCN(C(=O)C(CO)N(C)C)CC1 c12cccc(c1)OC2.c1(C(=O)NC2(CO)CN(C(COC)=O)C2)ccccc1C C1(F)(CNC(C(C=C)n2cccn2)=O)CCN(C(=O)COCC(=O)OC)C1 Nc1c(Cl)cc(C(=O)NCC2CCN2C(=O)CSC2CCCCO2)cc1Cl C(=O)(CC1NC(=O)c2ccccc21)N1CC(CNC(c2cc(F)c[nH]2)=O)C1 C1(F)(CNC(C(C2CCC2)OC)=O)CCCN(C(C2CCC(C)O2)=O)C1 c1(C(C)C(=O)N2CC(NC(C3C=CCCC3)=O)C2)ccccc1F c1(N2C(=O)CC(C(=O)NCCNC(C3(C)CC=CCC3)=O)C2)ccc(F)c(F)c1 Cc1[nH]c(C#N)cc1C(=O)NC1CCCC1CNC(=O)C(C)(C)c1ccnn1C CCC(C)C(C(=O)N(CC(O)CF)C)N(C)C(c1cnn(C)n1)=O C(C(CC(C)C)C(=O)N1CCOC(C(C)C)C1)NC(c1cccc(C)c1N)=O c1(C(=O)NC2CN(C(c3cc(C)nnc3)=O)CC23CC3)c(F)cc(Cl)cc1F CC1OCCC1C(=O)NCC1(NC(=O)COCC2CCCO2)CCC1 c1(C2(CC(=O)NCC3CCC3NC(=O)CCC=CBr)CC2)ccc(F)cc1 N1(C(C(=O)NCCC(=O)OCC)CC2CCOCC2)CC2(CC=CC2)C1 c1(OC(c2c(OC)c(C)ncn2)=O)c(Cl)cccc1[N+](=O)[O-] CCCCC(CNC(=O)C(C)O)NC(C1CCCC2CC12)=O c1(C(N2CCCC(C(C)NC(c3c[nH]c(=O)cn3)=O)C2)=O)cn(C)c(=O)n1C CC(CC(F)F)C(=O)NCC=CCNC(c1ccc(CSC(F)F)o1)=O C1(CN(CCCNC(COc2c(C)occc2=O)=O)C)CCc2nccn2C1 c1(CCC)cc(C(=O)NCCC(C)CCNC(=O)C(C)(C)c2cscn2)ccn1 Cn1nc2c(cc1=O)CC(C(=O)OCCn1cnnc1)CC2 C1(C(=O)NC(CCC)CO)(C(C)C)CCCN1C(=O)C(CC)NC(C)=O c1(OC)cc(=NC(=O)C2(CNC(c3cc(O)ncc3F)=O)CCCC2)[nH]n1C c1(C(=O)NCC(CNC(=O)C=CC2CCOCC2)O)c(Cl)ccc2ccoc12 c1(C(=O)NCC23CCC(CC2)N3C(C2(O)CC(F)(F)C2)=O)cccc(F)c1F N1(C(c2c(C)c(C3CC3)ncn2)=O)CCC(N=c2[nH]nco2)(c2ccccc2)C1 C(C(=O)N(C)CCN(C(C1(C(F)(F)F)CCCCO1)=O)CC)(C(C)C)SCC CC1(CNC(=O)C(C)(C)NC(c2cnncc2O)=O)CCOCC1 CC1(C)CCOC1C(=O)NC1CCCC1n1cc(CCC(N)=O)nn1 Cc1nn2cc(C(N3CCCC3C(C)NC(C3CCC(C)CC3)=O)=O)nc2s1 C(=O)(C(C)(C)CC1CC1)NC1CCC(CCC(=O)N(CC(=C)C)CC)C1 c1(C(=O)NC(C(=O)NCCCC(=O)N(CCC)CCC)C)ccc(C)c(Cl)c1 C1(C2CCC2)(C(=O)NCC2(O)CN(C(CSCC(C)C)=O)C2)CC1(F)F Cc1c[nH]nc1C(=O)NCCCCN(C(=O)C(C)(C)c1cc[nH]n1)C Cc1cc(C(=O)NCC2CC2NCCNC(c2cc(Cl)ccc2F)=O)cc(C)c1 C(=O)(CC(C)(C)C(F)F)NCC1N(C(C(C(C)C)n2ccc(C)c2)=O)CC1 C1(CCNC(c2cc[nH]c2)=O)CCCN(C(=O)C(c2ccc(Cl)cc2)O)C1 CCN=c1[nH]c(C(N2CCC(NC(=O)C=CC3CCOCC3)C2)=O)cs1 c1(C(=O)NC2CC(C)CN(C(c3c[nH]nc3C3CC3)=O)C2)cc2cnccc2[nH]1 c1(OCCC(=O)NCC(C)NC(c2cn(C)nn2)=O)ccc(F)cc1 c1(C(N(C2CCC(NC(=O)CCN3CCCC3=O)C2)C)=O)cnc2[nH]ccc2n1 c1(C(=O)NCC(CNC(c2cncc(C#C)c2)=O)C)cc2sccc2n1C CC1CN(C(C2C3CCCCC23)=O)CC1NC(c1cnc(O)s1)=O CC(C)CC(CNC(=O)CC1CCCOC1)C(=O)NC1(C)CCOCC1 c1(NC(c2ccccc2Cl)C)[nH]c(=NCC(C)CN2CCCC2)nc2sccc12 N1(CC(=O)NC2CC(NC(C3(S(C)(=O)=O)CC3)=O)CC2O)CCS(=O)(=O)CC1 c1(OC)ncc(C(N2CC=CC(NC(c3ccc(C(C)(C)C)s3)=O)C2)=O)cc1C CCS(=O)(=O)c1ccccc1C(=O)NC(C1CN(C(C2CC3(CSC3)C2)=O)C1)C c1(CCCN(C)C)nc(-c2cncc(-n3ccnn3)c2)n(-c2cccnc2)n1 C1(C2(NC(=O)C(CSC)NC(=O)C(O)CC(C)C)CC2)(OC)CCC1 N1(C(Cn2ccc(C)c2)=O)CCC(C)(C)C1C(=O)N(C)CC1COC(=O)N1 C1(NC(c2cc(C)ns2)=O)C=CCC(C(=O)NC(c2cncnc2)C)C1 C1(CCC(=O)NCCN=[N+]=[N-])CCN(C(C2(C(=O)O)CCCN2)=O)CC1 C1(N(C(c2c(Br)cnn2C)=O)CC)CCCN(C(=O)CS(C)(=O)=O)CC1 CC(C)CS(=O)(=O)NC(c1cc(CF)on1)=O Cc1cncc(-c2cn(CC3CCCN(C(C4CCC4)=O)C3)nn2)c1 C1(C(N2C(C(=O)OC)CC2)=O)CCN(C(c2ccoc2C2CC2)=O)C(C)C1 CC1C(NC(c2coc(C3CCCC3)n2)=O)CCN1C(c1ncccc1N)=O C(=O)(C#Cc1ccccc1)N1CC(NC(=O)CCc2cccnc2)C(F)(F)C1 C1(CCN(C(C(CC)O)=O)C)CCCCN1C(=O)C=Cc1cncn1C N1(C(c2ncc(Cl)cc2Br)C(=O)NCC2CCOC2)CCCC2(C=CCO2)C1 c1(CC(C)NC(Cc2ccc(CC)cc2)=O)ccc(F)cc1F C1(NC(c2c(OC)n[nH]c2)=O)C=CCN(C(=O)Cc2csnc2C)C1 CC1(C)CCc2onc(C(=O)NCC(C)(C)NC(=O)C(F)CC3CC3)c2C1 c1(C(N2CC(OCCNC(C(CC)C#N)=O)C2)=O)c[nH]c2nccc(Br)c12 c1(C(=O)NCC2(CNC(=O)CO)CCCC2)ccc(Br)c(F)c1 C1(CN(C(c2cc(CC)on2)=O)C)C2CN(C(=O)CC3COC(=O)N3)CC12 S(=O)(=O)(c1csc(C(N(CCC)Cc2ccc(F)cc2)=O)n1)NC C(=O)(C1CCCc2ccccc21)N(CCCNC(c1ccc(F)cc1N)=O)C N1(C(C(CCC)NCc2cnc3n2CCOC3)=O)CCC2(CC1)CCS2(=O)=O C1(NC(C2C=CCC2)=O)CC2(CCN(C(c3ccc(CC4CC4)s3)=O)CC2)C1 c1(-c2onc(-c3cccc(CC4C5CCC(F)(F)C54)c3)n2)cnc2cc[nH]c2c1 N1(C(c2ccncc2O)=O)CC(C2CN(C(C3CC3C3CCC3)=O)C2)C1 N1(C(C2C(C)CCC2)=O)CCC(C)(NC(=O)COCCO)C1 N1(C(c2cc(Cl)ccn2)=O)CC2(C1)CN(C(C13CCC(F)(CC1)CC3)=O)CCO2 N1(C(CCc2ccc(C)nc2)=O)CC2CCC2(CC(=O)NCCCCN(C)C)C1 c1(C2C(C(=O)NCc3cc(CNC(C4C=C(C)CS4)=O)no3)C2)cccc(Cl)c1 c1(N(CC(OC)OC)CCCO)nnn2c1N(C)CC2 c1(C(=O)NC(CNC(c2n(CC=C)ccn2)=O)C)ccc2c(c1)COCCN2 Cn1cnc(C=C(F)C(N2CC(C(=O)NC3CC4CCC3O4)(N(C)C)C2)=O)c1 CC(C)CCC(=O)N1CCC(CN(C)C(c2ccnc(N(C)C)c2)=O)C1 CCC(C)(F)C(=O)N1CCC(F)(CNC(=O)Cn2nnnc2C(C)C)C1 c1(C(=O)NCC2C(NC(c3cc(NC)no3)=O)CCC2)nnn(C)c1C(F)F C1(NC(c2ccc(OC)nc2)=O)C(C)CN(C(=O)CN2CCS(=O)CC2)CC1C c1(C(N2CC(NC(C(C)OCCC#C)=O)C2)=O)cnn(CC2CCCC2)c1 CC1CCN(C(c2csc(Cl)c2)=O)CC1NC(C1(C(F)F)CCCC1)=O c1(C(=O)NC2CC3(C(C(=O)NCCC4CC(C)C4)C3)C2)cc(C#N)cn1C C1(CNC(CCOC)=O)COC(CNC(c2cn(CCC(C)(C)C)nn2)=O)C1 CCCCC(CC)(c1nnnn1CC1CCOC1)NC(C)COCC c1(CNC(c2n(CCSC)nnn2)C2CCSCC2)nnc2n1CCNC2=O C1(CNC(C(CC)CC)=O)CCN(C(=O)CSc2ccc(O)cc2)C12CC2 C(C(N=c1nc(C2CC2)[nH]s1)C1CCCCC1)NC(c1ccn2ncnc2c1)=O c1(CN(CCNC(=O)NC2CCCN2C)CC)ccccc1C C1(C)(C(=O)NCCC2CC(NC(C3N(CC)CC3)=O)C2)CCN(C)C1 Cc1c(Br)noc1C(=O)NCCCC1CCCN1C(=O)C=C1CCC1 CC12CCC(C(N3CC4CN(C(=O)CCc5nc[nH]n5)CCC34)=O)(CC1)CO2 c1(C(N2CCN(c3nc(OC(C)C)c(Br)cn3)CC2)=O)cnn2cc(F)cc(F)c12 c1(C(N2CC(NC(CCC3CC(OC)C3)=O)C(O)C2)=O)sc(Cl)c(Cl)c1C O=C1COCCN1C1(C(=O)NC2CCCCC2n2cccn2)CC1 C(c1c(Cl)nc2sccn12)=CC(N1CCC(C(C)NC(=O)COCC(F)F)C1)=O c1(CCC(=O)OCc2c(OCC#C)cccc2F)cnc2n1CCCC2 C(=O)(C#CC1(CCc2cn(-c3ccc(O)cc3)nn2)CC1)NCC1(C)CCCO1 C1(C(=O)NCCCN2CCN(CC)CC2)CN(C(c2ccncc2)=O)CCN1C c1(C(=O)NC(CCNC(C2C(=C)C2)=O)C)ccnc(OC)c1 N1(C(CCc2cccc(OC)c2)=O)CCCC2CN(C(=O)CC=C(Cl)Cl)CCC12 C12(CNC(CC=C)=O)CC(NC(C3CCC3C)=O)(CO1)C2 O=C(C1=NOC2(CCN(Cc3cc(O)ccc3Br)C2)C1)NCc1ccc(F)nc1 c1(C(=O)NCC2CN(C(C(C=CC)O)=O)CC2O)cnc2c(c1)OCC(=O)N2 CC1(CNC(=O)COC(F)F)CCN(C(=O)Cc2cccc(OC(F)F)c2)C1 c1(CNC(C2CC(=C)CN2c2cc(Br)cnc2C(N)=O)=O)cnc2cc[nH]c2c1 CC1CN(C(=O)CC2CC2)C(C)CN1CC1CC=CCC1 N1(C=O)CC2CC1(C)CO2.N1(CCOC)CC(OC)CC1=O.C(C)(C)(C)OC(C)=O C12(COCC)C3CCC(CC13)C2(F)F.C123CCC(CC1)(CO2)CNC3=O Cc1cc(-c2cn(CC3CCN(C4CCC4C(=O)O)CC3)nn2)ccn1 C#CCCC(C(=O)N1CC(F)(F)C1)NC(c1cccc(F)c1N)=O c1(-n2cc(C3CCCN(C(C4C(CC)CC4)=O)C3)nn2)ccccc1C(F)(F)F C(=O)(C1Cc2ccccc21)N1CCC(C(=O)NCc2nn(C)c(=O)o2)C12CCC2 C1(C(=O)NC(CNC(c2cc(C)ncn2)=O)CC(F)(F)F)CCc2nccn2C1 Cc1c(C(=O)NC2(C(C)NC(=O)Cc3cnn(C(C)C)c3)CC2)nnn1C(C)C Cc1cc(CNC(C2CC2CNC(=O)C=Cc2ccccc2)=O)ccc1F C(=O)(C(F)C(=O)NCC1(CC(=O)NCCC2(C)CC2)CC1)OCC Cc1cc(OCCC(=O)NCC2COCC2NC(c2cc[nH]c2)=O)c(C)c(C)c1 c1(OC)cc(C(N2CCCN(Cc3ccccc3F)CC2)=O)cc(Br)c1O C1(CC(=O)Nc2cc(C(C)(C)C)[nH]n2)CC(N=c2ccn3nccc3[nH]2)C1 C1(CC)CN(C(C2CCC(C#N)C2)=O)CC1NC(=O)CCOCCOC Cc1cc2cccc(C(N3CCOCC3CC3CCC3)=O)c2o1 c1(N2CC3C(N(C)C)C3C2)ncnc(NC(=O)C2=CC3CCCC23)c1[N+](=O)[O-] C(=O)(C1=CC2C=CC1C2)N1CCC(CC(N2CCC(C(C)O)C2)=O)C1(C)C c1(C(N2CCCC2CN(C(C23CCCN(CC2)C3)=O)CC)=O)nccc2ccsc12 C1(CNC(C2CC(=C)C2)=O)C(C)CCN1C(c1c(OC)nsc1OC)=O C1(NC(CNS(C)(=O)=O)=O)CC(=O)N(C2CCCCCC2)C1 N1(C(CC2CN(C(c3c(C)n[nH]c3)=O)CC2C)=O)CCCCCC1C C1(NC(c2cnc(CC)s2)=O)CCCC(NC(=O)C(C)(C)c2ccnn2C)C1 N1(C(c2ccc(C(C)=O)o2)=O)CCOCC1C(=O)Nc1ccsc1C(C)C C#CC(CC(C)(C)C)NC(C1CC2CC2N1C(C12CCC(C1)C2(C)C)=O)=O C=C(CNC(N1CCN(CCn2cncn2)CC1)=O)c1ccccc1 N1(C(C(COC)(C)C)=O)CCC(C)C(NC(=O)CN2CCOCC2=O)C1 C1(CNC(C(CC)C2CCOC2)=O)CC(F)(F)CN1C(c1cc(F)ccc1Cl)=O c1(CN(C)C(c2coc(-c3ccccc3F)n2)=O)nnc2n1CCNC2 c1(OC)ccc(C(=O)NCCC2CCN(C(=O)C(C)OCCN(C)C)C2)c(Cl)c1 c1(C(N2CC(C(=O)Nc3c(C(C)=O)cnn3C)C2)=O)ccc2c(c1)OCCN2C c1(COCC(=O)NCC(n2cc(Cn3nccn3)nn2)C)ncnn1C c1(NC(c2ccc(NCC(C)C)nc2)C)ccccc1CCO CCC(C)CC(C(=O)NC(CO)C1CC1)NC(C1CC(=O)N(CC)C1)=O c1(C2C(C(=O)NCC(CC)NC(=O)CC(C)C(=O)OC)C2)c(Cl)cccc1Cl c1(C(c2nnnn2CCSC)NCC(C)CCO)ncnc2c1OCCO2 C1(NC(c2c(CC)cncc2)=O)C2CCC1N(C(=O)C(C)CC)C2 c1(CC)ccc(S(=O)(=O)N2CCCC(C(N3CCOC(C)C3)=O)C2)s1 c1(CNC(C2OCCN(C(C3(C)CNC(=O)C3)=O)C2)=O)ccc(F)cc1Cl c1(C(N(CC(CN(C(C(C2CC2)OC)=O)C)O)C)=O)c(C)cc(Cl)cc1N c1(C(N2CCCC(NC(c3cnc(C)s3)=O)C2)=O)cnn2c1OCCCC2 c1(C(c2n(CC=C)nnn2)NCCc2cccc(F)c2C)ccc(O)c(F)c1F C1(CNC(C2C(OCC)CC2)=O)(NC(C2CN(C3CCOC3)C2)=O)CCCCC1 N1(C(C2CCC(NCc3ccc(O)c(O)c3O)CC2)=O)CCC2(CCOC2)CC1 C1(CNC(C(=O)NCCn2c(C)nc(C)n2)=O)OCCOC1(C)C N1(C(C2CCCS2(=O)=O)=O)CCN(C(c2ccc(O)nc2)=O)C2CCCC12 CN1CCCCC1C(c1cn(CC(=O)NOC(C)(C)C(=O)O)nn1)NC(C)(C)C c1(CC)ccc(C#N)cc1F.c12cccc(c1)CNC(=O)C1CC(O)CN1C2=O Cn1ncc2c(C(N3CC(NC(c4ccc[nH]4)=O)C(CO)C3)=O)cccc12 C1(NC(c2c(C)nc[nH]2)=O)CC2C(NC(C3CCC3C)=O)C2C1 CCN=c1ccc(C(=O)NC2CC2NC(c2ccsc2)=O)c[nH]1 C1(C(N2C(CC#C)CCC2)=O)(CNC(c2ccc(CC#N)cc2)=O)CC(F)(F)C1 CC1CC2=C(C(=O)N1)C(c1c(Cl)cccc1Br)NC(=S)N2CCC1CC1 c1(C(N2C(CNC(=O)CNC(C3CCC3)=O)C=CC2)=O)csc2c1CCCC2 N1(S(Cc2cccc(C)c2F)(=O)=O)CCOC2(CCS(=O)(=O)C2)C1 N1(C(CC2C(C)(C)C(=O)C2)=O)CC(C(=O)NCC(N2CCOCC2)=O)C(F)(F)C1 c1(C(=O)CN(C2(CNC(c3ncn(CN(C)C)n3)=O)CC2)C)cc2sccc2[nH]1 CC(CF)CC(=O)NC1CCCCC1NC(C1(Oc2ccccc2F)CC1)=O CC1CCS(=O)(=O)CCN1C(c1ccn(C(F)F)n1)C(=O)NC1CCC1 C12(C(=O)NCC#CCNC(Cc3cccc(OC(C)C)c3)=O)CCC(C)(C1)OC2 c1(C(=O)OC)ccc(N(C2CN(C(=O)C(O)CSc3ccccc3)C2)C)cc1 CCC(CC)CC(=O)NC1CCCCC1C(=O)NCCN1CCCC(O)C1 N1(C(C(COC)OC)=O)CCC(NC(=O)Cc2cccc(F)c2Cl)C1CCO c1(C(N2C3(CNC(CN(C(C)C)C)=O)CCC2CC3)=O)cccc2c1CCOC2 Cc1nc(NC(=O)NCC2CCC(=O)NC2)sc1F C1(CNC(CCC)=O)C2CCCC1N(C(=O)C(c1cc(C)cc(F)c1)C)C2 CC1(O)CCN(CC(=O)NC2(CCNC(C3CC(CF)C3)=O)CCC2)C1 CC1CC(C(N2CCC(CCCNC(=O)C#CC(=O)N(C)C)CC2)=O)CC(C)O1 c1(C(=O)OC(c2cccn2C)C)cc2c(cnn2C)nc1O C12CN(CCO1)C2=O.c1(COCC(=O)NC2C(CN(C(C)=O)C)C2)cccnc1 N1(C(C=CC)=O)C(CNC(c2ncccc2OCC)=O)CC2CCCC12 CC1(C)CCCC(CC(N2CC(O)(CNC(=O)CC34CNC(=O)C(C3)C4)C2)=O)C1 c1(C(N2CC(CNC(C(C=CC)O)=O)C2)=O)cc(F)ccc1C N1(C(CCc2cc(C)[nH]n2)=O)CC2(C=C(C(=O)N3CCOCC(C)C3)CO2)C1 N1(C(C2(Cl)C(C)(C)C2)=O)CCCC(CCNC(=O)CCCC2CC2)CC1 c1(C(N(CCN(C(c2cc(CC)c(C)cc2)=O)C)C)=O)nccn2cnnc12 c1(Cc2[nH]nc(C(=O)Nc3ccc(Cl)cn3)n2)c(F)cccc1F c1(OC)ccnc(C(N2CCC(O)(CN(C)C(c3nc(C)nn3C)=O)C2)=O)c1O CCCCC(C(=O)NCC(=O)OCC)NC(C1CCN(CCC)C1=O)=O C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(c2c(C)cnnc2)=O)C(C)(C)C1 C(c1ccccc1[N+](=O)[O-])=CC(=O)NCC1OCCN(C(C(COC)OC)=O)C1 C(=O)(C(C#N)C(C)(C)C)NC(CN(C)C(c1ccc(-c2ccco2)[nH]1)=O)(C)C C1(C)(C(=O)OCC(c2c(C)noc2)=O)CCC(Cc2ccccc2Cl)CC1 Cc1nnccc1C(=O)NC(C)CCN(C)C(C1CCC(CN(C)C)O1)=O C(=O)(C(C)C(O)C(C)C)NCCn1ccc(C(NOCCOC)=O)c1 C(=O)(CC(C)CC(C)C)NCc1nc(C(N(CC=C)CCC)=O)sc1 c1(-c2scc(C(N3CC(O)(C(C(=O)OCC)F)C3)=O)n2)ccc(Cl)cc1 c1(OC)ccc2c(n1)NC(C(=O)NC(C)CN(C(=O)C=Cc1cnn(C)c1)C)C2 Cc1nc(NCC(=O)Nc2ccc(F)cc2F)cc(=NCCOC2CCCC2)[nH]1 C1CN(N2C3CN(C)C(C3)C2)CCC1(F)F.c1(C)cc(O)cc(O)c1 c1(OC)c(Cl)ccc(Cl)c1CC(=O)Nc1ccsc1OC N1(CC(=O)NC2CCC(N(C)C(C3CCNC3=O)=O)CC2)CCCNS1(=O)=O Cc1ccc(NC(C2OCCC2CNC(c2ccc(F)cn2)=O)=O)c(C)c1O C1(NC(c2scc(C)c2)=O)CC12CC(NC(=O)CC1C=NN(C)C1=O)C2 C(=O)(C1=CC2CCCC12)NCC(C)(C)CNC(c1ccc(N)cc1O)=O c1(NC(C=C(C)CNC(=O)C=CCN2CCC2)=O)ccc(O)nc1 c1(C(N2CCC(NC(C3CC34CCSCC4)=O)C2)=O)cc2c(cn1)CCCC2 N1(C(c2c(CC)cccc2)=O)CCCC2(NC(c3cnsc3)=O)CCCC12 N1(C(C2(CC)CN(C(=O)CC3CCCOC3)C2)=O)CC2CC2C2CC12 C#CC1CN(C(=O)C(C)=C2CCC2)CCN1C(=O)C(C)OC N1(C(C(C)SC)=O)CCCC2(CCCCC2NC(c2cn(C3CCC3)nn2)=O)C1 N1(CC(CC)C)CC(CNC(=O)CC2CCCOC2)CC1=O C1(NC(c2c(OCCC)cccc2)=O)CCCC2CN(C(C3CC3OC)=O)CC12 N1(C(c2c(OCC)ccc(Br)c2)=O)CC2C(N(C)C)CS(=O)(=O)C2C1 C1(C(=O)NCCN2CCCC2)C2CC2CN1C(c1csc(O)n1)=O c1(C(CCC)C)nc(-c2cc(C(C)C)nn2CCOC)n(CC(N)=O)n1 Cc1ccc(CN2CCCC(C(N3CC4CCCC4C3)=O)CC2)c([N+](=O)[O-])c1 CC1CCn2cc(C(=O)NCC34CC(NC(c5nc(COC)cc(N)n5)=O)(C3)C4)nc2C1 Cc1nn(C(C)C)c(C)c1C(=O)N(C)CCNC(=O)C(C)CS(C)=O C1(NC(CC(=C=C)C)=O)CC2CC(NC(=O)Cn3cc(C4CC4)nn3)CC12 c1(C(N2CCC(C)(CCNC(CC(CC)C)=O)C2)=O)nc(C)c(C)[nH]c1=O N1(C(c2cnc(NC(C)=O)o2)=O)CC2(C1)CN(C(=O)C(C#N)C(C)(C)C)CCO2 C(=O)(C1CCN(C(N)=O)c2ccccc21)OCCC1CCC(C)(C)CC1 C1(C2CCCCN2C(C2CCC2)=O)(CNC(=O)CCc2nccs2)CCOCC1 c1(C(C)=O)cc(C(N2CCC(CO)(NC(C3CC34CC4)=O)CC2)=O)c(C)nc1C C1(C(=O)NC(CCCC)C)N(C(=O)CN(CCCCCC)C)CCC1(C)C C12(NC(c3cccc(CO)c3)=O)CC(C1)N(C(=O)Cc1cncc(O)c1)C2 c1(COC)cc(C(=O)NC2CCC(NC(=O)C(c3cscc3Br)=O)C2)on1 C(C(C)S(C)(=O)=O)(c1ccc(C)cc1)N1CCC(CO)(NC(=O)OC(C)(C)C)C1 c1(CN2CC3(CCC(CNS(C(COC)(C)C)(=O)=O)O3)C2)cccc(B(O)O)c1 c1(OCCC)cccnc1C(=O)NCC1CCN1C(c1ccn(C)c1)=O Cc1ccnc(O)c1C(=O)NC(CNC(=O)C(C(C)C)n1cnnc1)C1CC1 C1(CCC(=O)NCCN(C(=O)C(CO)N(C)C)CCOC)CC(F)(F)C1 C1(NC(COCCC#C)=O)CN(C(c2cc(C)c(CC)nc2O)=O)CC1N=[N+]=[N-] c1(CC(=O)NC(C)CN(C(=O)Cc2cnco2)C)ccc(C2CC2)cc1 C#CC(C)(C)C(=O)NC1CCCCC1CNC(C1CN(C2COC2)C1)=O N1(C(CC(=O)OC)=O)CCOCC2(C1)CN(C(=O)COC1CCCC1)CCCO2 C(CC(CC)C(=O)NCC1(CNC(c2cnc(Cl)s2)=O)CC12CCC2)=CCCC C1(C(=O)NC2C=C(C)CS2)CC2CCC1CN2C(C1CCCN(C(N)=O)C1)=O C123CCCC1N(CCC2)C(=O)CCOCC(=O)NC3.C(C(C)(C)C)OC(C)C C(N=c1nc2c(cnn2C)c(N2CCN3C(=O)NCCC3C2)[nH]1)C1CC(OC)C1 Cc1ccc(C(N2C3CCC2CN(C(C2CCN(C)C2C)=O)C3)=O)c(N)c1Cl C(=O)(C1CN(C(=O)OC(C)(C)C)Cc2n[nH]cc21)OC=Cc1cc(Cl)cc(Br)c1 c1(N(CCCCN(C)C(c2cc([N+](=O)[O-])n[nH]2)=O)C)cc2c(s1)CCC2=O C1(CC(=O)NCC(C#C)C(C)C)C2CCCC2N1C(C1CC(=O)CC(=O)C1)=O CC(c1cnn(C)c1)=CC(N1CCN(C(C2CSCCS2)=O)C(C2CCC2)C1)=O c1(C(C(=O)NC(CNC(Cc2cnc(C)s2)=O)CC(C)C)O)ccc(Cl)c(F)c1 c1(C(=O)NCCCN(C(C2CC(C)=C(C)CC2)=O)C)ccc2n[nH]cc2n1 c1(NC(C)=O)cccc(F)c1C(N1CC(O)(CN(C)C(C2CCSC2)=O)C1)=O C1(NC(c2c(C)nco2)=O)CC2CC(NC(=O)CC3CC(=O)NC3=O)C1C2 N1(C(c2snc(O)c2Cl)=O)CCC2CCN(C(c3cc4ccccc4o3)=O)C2C1 N1(C(C2CN(Cc3ccc(COC)o3)CC(F)(F)C2)=O)CCN2CCOCC2C1 N1(C(c2c(C)ncnc2)=O)CCC(CNC(c2ccncc2)=O)C(C)C1 c1(N(C)C)ccc(C(=O)NC2CCCC2NC(c2c(C)nn(C)c2Cl)=O)c(F)c1 c1(OC)ccnc(F)c1C(=O)NCC1(F)CCN(C(=O)CCC(C)(C)C)C1 c1(C(=O)NCC(C)N(C(=O)COCCSC(C)C)CC)cc(Cl)c2cn[nH]c2c1 C1(C)(CNC(CC(CC)SC)=O)CN(C(=O)CCC2(C)CC2(F)F)CC1C Cc1ccc(Cl)c(NC(=O)C(C)NC(=O)CN2CCC(C(=O)O)CC2)c1 N1(C(C2CC(C#C)(O)C2)=O)C(C(=O)NC2COCC2O)CCC12CC2 C12(NCCn3ccc(C(N4CCC(C(C)(C)O)C4)=O)n3)CC=CC(C1)OC2 CCC(O)C(C)(C)C(=O)NC1CN(C(=O)Cc2ccnc(F)c2F)CC1SC C(C1CN(C(C2C(C)C2C)=O)CC1C(N1CC(=O)NCC1C(C)C)=O)=CC N1(C(c2c(CNC(=O)C=Cc3cc[nH]n3)n[nH]c2)=O)CC2(CNC(=O)N2)C1 N1(C(C(C)CCN2CCOCC2)=O)CC(c2ccccc2)CCC1C c1(C(C)NCC(C(=O)OC)Cc2ccccc2)ccc(Cl)c(Cl)c1C c1(NC(N(C)C)=O)cc(NC(=O)Nc2ccc(-c3ncn(C)n3)cc2)cc(Br)c1 CC1(CNC(=O)C(F)=C2CCC2)CCCN(C(=O)C(c2cccc(F)c2)O)C1 C1(CNC(c2cc(OC)n[nH]2)=O)CCCC2CN(C(=O)Cc3cc[nH]n3)CC12 C1(O)(CN(C(=O)C(c2ccco2)NC(=O)CCC2CC2(C)C)CC)CCC1 c1(C(N2CCCC(CC(=O)Nc3ccc(C4CC4)nc3)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CS(=O)(=O)CCC(=O)N1CC2CC(NC(=O)C(=O)NC3CC3)CC(C2)C1 c1(C(=O)NCC(C)N(C(C(C)NC(CC)(C)C)=O)C)cc2ccccc2c(O)n1 c1(NC(C(=O)Nc2c(C3(C)OCCO3)cccc2)=O)cccc2c1OCCC2=O C1(N(C(C(C=C)C)=O)CC=CCCCCC)CCN(C(=O)COCCCC)CC1 N12CCCC(C1)C(C)C(=O)NC1(CCC1)C2=O.C(C(C)(C)C1CCC1)SCC c1(N(C)CC2(OC)CCC2)nnc(C(C)C)n1CC(C)C(C)C CCC(C(=O)NC1CCCCC1NC(=O)Cn1ccnn1)C(C)O c1(C(N(C(C(N2CCC(C(CC)CC)C2)=O)CC)CC)=O)ncccc1O C1(NC(c2c(C)ncn2O)=O)CCOC2(CCC2)C1 C1(CNC(C2(C#N)C(C)C2)=O)(CNC(=O)Cc2c(Cl)cnn2C)CCCCC1 C1(NC(c2cnc(C)s2)=O)CC2CCC(C1)N2C(=O)CCCc1cccc(F)c1 N1(C(c2nc(CC)oc2C)=O)CCCCC(NC(c2csc3nnsc23)=O)C1 c1(C(N2CC(CC(C(=O)NCC(C(=O)OCC)C)F)C2)=O)cc(C)c(C)o1 N1(C(C2CC3(C(OC)CC3)C2)=O)CC2CCN(C(c3[nH]c(=N)sc3C)=O)CC2C1 N1(C(Cc2c(C)ocn2)=O)CCCC(F)(CNC(=O)CCN2CCCC2=O)C1 C1(NC(Cc2c(C)scc2)=O)CN(C(=O)CC2CCN(C)C2)C2(CCC2)C1 N1(C(C2C3CN(C(C(CC)COC)=O)C2C3)=O)CC2CN(C)CC2C1 C1(NC(C=C(COC)C)=O)CCN(C(=O)CN2CC(=O)N(C)C2=O)C12CC2 C1(C(N2CCC(CS(=O)(=O)Nc3scc(C)n3)CC2)=O)CCc2nc(C)cn2C1 c1(C(C)=O)ncc(C(=O)NCCC(O)CNC(=O)C(C)CC2CCC2)s1 N1(C(CC(C)C)=O)CCC2CN(C(=O)CCCc3ccc([N+](=O)[O-])cc3)CC2C1 C12CCCC(CC1)C(=O)N2.CC1CCC(C(=O)NNC[Si](C)(C)C)CC1 C#CCCCCC(=O)NCC12CC(CN1C(c1ccc(N)c(O)c1)=O)C2 C=CC1CCN(C(=O)CC2(C=C)CN(C(=O)CC3CCCC3C)C2)CC1 C(=O)(CC(F)(F)C(C)C)NCCN(CCC)C(C1CCOCC12CCC2)=O C(CCCC(=O)N1CCCC1C(C)NC(c1cnn(C)c1C(C)C)=O)SC c1(CC)cc(NC(C2CCN2C(=O)Cc2ccc(O)cn2)=O)cc(C)c1 c1(CC(=O)NCC2C(NC(Cc3nc(C)sc3)=O)C2)cccc(C(C)C)c1 n1(CC(=O)NCC2COCCN2Cc2ccsc2Br)ccc2c(F)cccc12 C1(C(=O)NC(C2CCCN2C(=O)CC(=O)NC2CC2)C)CC(C)(C)SC(C)(C)C1 C1(C(=O)NC(C)(C)CC2CCCC2)C(C2CC2)CCN1C(C1CS(=O)(=O)C1)=O C(=O)(C1CCc2cccc(O)c21)NCCN(C(c1ccc(C(C)C)s1)=O)CC C1(CNC(c2nc(CCC)oc2)=O)(NC(=O)Cc2cncnc2O)CCCOC1 c1(C(C(=O)NC2CN(C(CCCN(C(C)=O)C)=O)C(C)C2)C)ccc(C#N)cc1 c1(N2CC(CC(C)NC(C3CCCN(C(C)=O)C3)=O)C2)ncc(C)c(C)n1 C12(C(=O)OC)CC1CN(C(C1CN(C(c3cncc(OC)n3)=O)CCO1)=O)C2 CCCC(CC)C(=O)NC12COC(C1)C(NC(=O)COCc1nccn1C)C2 c1(C(=O)NC2C=CC(CNC(Cc3nc(CC)sc3)=O)C2)ccc(C#N)[nH]1 C(C(=O)NCC1CCC(NC(=O)C(C)Cc2cccnc2)CC1)(C(C)C)SC c1(NC(C(CC#C)(C)NC(=O)C(C)OCC2CC2)=O)cc(C)cn(C)c1=O N1(C(C2(C)CCC(=O)NC2)=O)CCN(C(c2ccc(N)c(Cl)c2O)=O)C2CCC12 CON1CC(C(=O)NCC(C)(C)OCCNC(=O)C(C)(C)C(=O)OC)CC1=O N1(C(=O)CCc2cncnc2)CCN(C(C2C3CCCOC23)=O)C2CCCC12 c1(C(=O)NCC2C(NC(C3N(C(C)C)C(=O)CC3)=O)C2)cc(=O)c(Br)c[nH]1 C1(C)(CC)CC(NC(=O)CC=CCNC(C2CCCN2C)=O)C1 N1(C(C(c2ccccn2)C)=O)CCC(C)(CNC(C2CN(CC(F)(F)F)C2)=O)C1 C(CS(=O)c1ccccc1)NC(N1CC2CC=CCC2C1)=O C=C(C)CCC(=O)NCC1(CNC(c2csc(CCCCC)n2)=O)CCC1 C1(N(C(=O)CCC2CC2(C)C)C)C2CN(C(c3csnc3Br)=O)CC12 N1(C(c2nc(C)nn2C)=O)CCC2CCCC(C1)N2C(c1c(C)cncc1C)=O c1(-n2ncc(C(=O)NC(CNC(Cc3c(C)n[nH]c3)=O)C)c2)ncc(Cl)cn1 C(=O)(CC(C)(O)CC(=O)O)N1CCOCC(NC(c2c(F)ccc(C)c2Cl)=O)C1 C(=O)(C(O)CC(F)(F)F)NC1C(CC)CN(C(=O)C(COC)OC)CC1 C1(NC(C(C(C)C)NC(C)=O)=O)CC2CC1CC2C(=O)NC1CCOCC1F c1(C(=O)NC(CC=C)CNC(C2(NC(C)=O)C=CCC2)=O)c(C)nn(C)c1Cl C1(C(=O)NC(C)CSCCOC)(CC)CN(C(=O)Cc2ccccc2)C1 C1(N(C(c2cc(CCNC(CCOCC(C)C)=O)on2)=O)C)CCC(=O)N(C)C1 CC(O)C(C(=O)NCC1(F)CC(NC(c2cc[nH]c2)=O)C1)NC(=O)C(F)(F)F Cc1[nH]nc2ccc(C(N3CC4(NC(c5c[nH]ccc5=N)=O)CCC3C4)=O)cc12 C(=O)(CC(C)C(F)F)NCCC1(NC(c2occ(C)c2)=O)CCCC1 c1(C(C(=O)NC(C)C(C)NC(C2(n3cncn3)CC2)=O)C)ccc(F)cn1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(CNC(C2(OC)CC2)=O)C(C)C1 c1(C(N(C2CC(NC(C3CC(C4CC4)C3)=O)C2)C)=O)ccn(CCO)c(=O)c1 C1(C(=O)NC2C(C(N)=O)CCC2)CCCN(C(=O)CC2CCOC2)CC1 c1(C(=O)NC2CCCC23CN(C(C2CC=CCC2)=O)C3)ccc2c(c1)CCOC2 C1(CC=C)(NC(=O)Cc2ncoc2C)CCN(C(C2(n3cccn3)CCC2)=O)C1 C(=O)(C(F)C(C)C(F)(F)F)Nc1c(C)nc(Cl)cc1I c1(C(=O)NC(C(C(C)C)C)CNC(c2cnns2)=O)cccc2c1CCN2 C1(C(N(C)CC2CCCN2C(=O)CCC2CC2(Cl)Cl)=O)CCCN1N=O N1(C(c2ccc(CC)o2)=O)CC(N=c2[nH]nc(C(F)F)s2)C2(CCC2)C1 c1(C(=O)NC2C(NC(C(c3cccc(OC)c3)O)=O)C2)cccc2ncsc12 Cc1ccc(C2(C(N3CCC(CF)(NC(C4C(C)C4(F)F)=O)C3)=O)CCC2)cc1 N1(C(CCN(C)CC)=O)CC(CNC(c2ccc(CNC(N)=O)cc2)=O)C2CC12 CCCC(COc1c[nH]nc1NC(C)=O)C(=O)N(CCO)CCOC Cc1nc(C2CCCO2)ccc1C(N1CCCC(C(F)F)C1)=O N1(C(C(C)(CO)OC)=O)CC2CCC(C1)N2C(c1cccnc1OCCO)=O N1(C(c2ncc(OC)cn2)=O)CCCCC(NC(=O)C=C(F)c2ccccc2)C1 C1(NC(C2CC(O)(CC#C)C2)=O)CCCC1(C)CNC(=O)C(C)(C1CC1)OC C(=O)(C(C(C1CC1)C1CC1)N(C)CCc1nc(C)cs1)NCCC c1(OCC=C)ccccc1C(=O)NCC1CC(C)N(C(C2C3CC4C(C3)C24)=O)C1 S(=O)(=O)(c1cnc(NCC2(C3CC3)CC2)c(Cl)c1)NC(c1ccn(C)n1)CC N1(C(c2c(C(C)O)cccc2)=O)CC2CCC2(CNC(C2(C(F)F)CC2)=O)C1 c1(C(N2CC(C(c3ccccc3)=O)C(CO)C2)=O)cc(F)ccc1-c1nn[nH]n1 N1(C(c2oc(CC)c(C)c2)=O)CCCC(C)(C)C1C(=O)NC(CC)C(C)(C)O c1(C(N(CCCn2cc(CSC)nn2)C2CC2)=O)c(C)cnc2ccccc12 c1(OC)cc(CN2CCNCC(C(=O)O)C2)ccc1C#N c1(SC)cncc(C(=O)N(CCCNC(=O)CSc2nncs2)C)c1 Cc1ccc2ncnc(N3C4CCC(C4)C3C(N3CCCCC(C)(F)C3)=O)c2c1 c1(C(=O)NC23CC(CNC(C(C(CC)C)C)=O)(C2)C3)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NCCC(C)NC(C2(NC(=O)NC)CCCCC2)=O)cc2c(s1)CCC2 CCC(CC(F)F)C(=O)NC1CCN(C(=O)Cc2cc(C3CC3)on2)CC1F Cc1cc2cccc(NC(c3csc(NS(=O)(=O)c4ccccn4)n3)=O)c2cn1 c1(C(=O)NCCN(C(CCC(C)SC)=O)CC(C)O)cnc(C)c(N)c1 CC(C)C(C(=O)NC(C)C(CO)NC(C1(O)CC(F)(F)C1)=O)n1cnnc1 C1(C(=O)NC(C2CN(C(=O)CS(=O)(=O)N3CCCCC3)C2)C)(CO)CCCCC1 CC12CN(C(C3(C4CC4)CC3)=O)C(C(N3CCC(C)(F)C3)=O)(C1)C2 C(=O)(CC(C)C(C)(C)C)N1CCCC(N(C(c2c(C)n[nH]c2)=O)C2CC2)C1 c1(OC)c(C(N2CCC(NC(=O)CCC(C)(C)O)C(C)C2)=O)cccc1F c1(C(c2nnnn2Cc2ccccc2)NC(c2ccccc2)CC)coc(C)n1 Cc1oc2cc(C(N3CC(C)(NC(C4CCCCS4)=O)C3)=O)[nH]c2c1C Cc1nnc(C(=O)NC2CC(F)(CNC(c3ccoc3Cl)=O)C2)s1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(O)(CCNC(C(=O)N(C)C)=O)CC1 Cc1cc(Cl)c(F)cc1CNCCCN1CCN(Cc2ccc(I)c(O)c2)CC1 C1(C(=O)OC)CCC2(CCC2)C1C(N1CCN(C(=O)CSCC(C)C)CC1)=O c1(C(N(C(CN(C(CSCCCC)=O)C)C)C)=O)ccc([N+](=O)[O-])c(SC)c1 C1(NC(C=C(CC)CC)=O)COCCN(C(=O)C(F)=C(C)C)C1 c1(-c2n(C)cnn2)cn2cccnc2n1.C123CCCN(C1C2)OC(=O)C3.C(C)(C)C C1(NC(c2cn(CC)nn2)=O)CC(C(=O)NC2CC(CN(C)C)C2)CC1O CN1CCC2CN(C(C3CCCN3C(=O)CCNC(=O)N(C)C)=O)CCC12 c1(C(N2C(CNC(C(COC)C)=O)C(C)CCC2)=O)cc2c(C)cc(F)cc2[nH]1 c1(C(C(=O)NC(C(CO)NC(=O)OC(C)(C)C)C)N(C)CC)cccc(F)c1Br C(=O)(C1=C(CCCCl)N(c2ccc(F)c(F)c2)C(=S)NC1c1cnc[nH]1)OCC C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1C(NC(c2c(C)cccc2Cl)=O)C1 N1(C(COC)=O)CCC(O)(C(C)CNC(=O)C=C(Cl)Cl)C1 C(CC(O)C(=O)NCCOC(F)F)NC(CCc1ccn(C)n1)=O C1(C(=O)OCC)CN(C(=O)C(=O)N(C)Cc2nc(=O)n(C)[nH]2)c2ccnn2C1 N1(CC2CCN(C(c3nn(CC)c(C)c3)=O)CC2)CC(=O)CC12CCCC2 O=C(N=c1cco[nH]1)C1CCCN1c1ncc(-c2cc(F)cc(F)c2)s1 Cc1nc(C(N2CC(NC(c3cc(C(N)=O)co3)=O)C(O)C2)=O)ccc1[N+](=O)[O-] c1(C(N(C2CCCN(C(CCCNC(C)=O)=O)C2)C)=O)cnc2ccnn2c1 C1(NC(c2n(C=C)nnc2)=O)CCC12CN(C(c1ccc(OC(C)C)nc1)=O)C2 C#Cc1cnc(C(=O)N(CC(=O)NC2C(C)C2(C)C)C)c(C)c1 c1(OC)ccc(CCCCC(=O)N2CCC(CCN(C(=O)C(C)O)C)CC2)cc1 c1(C(N(CC(C)NC(CCCC(C)O)=O)C)=O)cc(Cl)cc2c1NCCC2 S(=O)(=O)(c1cc(C#N)ccc1Cl)NCCNC(=O)Nc1cc(OC)c(F)c(F)c1 c1(C(N2CC(CNC(=O)C(F)OC(F)(F)F)C(O)C2)=O)cc2c(s1)CCC2 C1(C(=O)NC)(C=O)CCOCC1.C1(F)(C(=O)NCC2(n3nccn3)CC2)CCC1 c1(C(=O)NC23CC(CNC(=O)C=C4CCCCC4)(C2)C3)ccc(F)c(Br)c1 C(=O)(CCC(F)F)NC(CN(C)C(C1CCCC1(C)C)=O)(C)C C(CNC(c1cc(C2CC2)[nH]n1)=O)(CC(=O)NCCc1csnn1)OC c1(C(=O)NC2C(NC(C3CC(C)OC(C)C3)=O)COC2)c(Cl)ccc(F)c1F Cc1cc(F)ccc1NC(=O)C(c1scc(C)c1C)N(C)Cc1ccc(F)c(Br)c1 C1(C2CCCCO2)(C(N(CC(F)F)CCC)=O)CCCO1 c1(C(=O)NCC(c2cc(F)cc(Cl)c2)NC(C(C(C)C)C)=O)cccc2ncnn12 C(=O)(C(C)c1cc[nH]n1)NCCSCC(=O)N(CCCC)CCCO n1(CC)cc(C(N2CCC(C(F)C(N3CC(C)(O)C3)=O)C2)=O)nn1 c1(C2(C(=O)NC3C(CNC(Cc4nnc(C)o4)=O)C3)CC2)cccc(F)c1F N1(c2ncc(OCCOC)cn2)CC2CN(c3ncncc3F)CC2C1 c1(C(C)=O)ccc(C(=O)N(C2CCC(NC(=O)CSCc3ccco3)C2)C)cc1 C(C(N=[N+]=[N-])C(=O)NCC1C2CCCOC12)OCC.C1(CC2CC2)CC(=O)N1 CC(C)C(O)C(C)NC(C1(CNC(=O)C(F)F)CCC1)=O C1(C(N(C(C)CNC(=O)Cn2c(C)ccc2C)CC)=O)COC(C)(C)CO1 Cc1sc(C(N2CCN(C(=O)Cc3ncn(C)c3C)C3CC23)=O)cc1[N+](=O)[O-] C1(CCNC(C(C)SC)=O)CCCN(Cc2ccc(-c3ccc(F)cc3)s2)C1 N1(C(c2n(CCC)ncc2)=O)CC2CC1CC2NC(c1cc[nH]c1)=O C1(CC)CN(C(=O)C(=O)N(c2ccc(Cl)cc2)CC2CC2)CCC1=O c1(CC(=O)NC2CN(C(c3ccncc3C(F)(F)F)=O)CC2O)cccc(Cl)c1 C1(C(=O)NCC2CCN(C(=O)Cn3cc(CO)nn3)C2)Cc2cscc2C1 CCCC(C)C(=O)NCC1(C(N)=O)CN(C(c2cn(CC(F)(F)F)nn2)=O)C1 N1(Cc2cnc(OCC)nc2)CCC(F)(C(=O)Nc2ccnc(F)c2)CC1 N1(CC)CCCCC1C(=O)NCC1CC(CNC(=O)COC2CC=CC2)C1 C1(NC(COc2ccn(C)n2)=O)CC(NC(C2(C3CCCO3)CC2)=O)C12CCC2 C(N1CCC(S(=O)(=O)N2CCOCC2)C1)n1nc(C)n(CCOC)c1=S C(=O)(CN=c1cc[nH]cc1)N1C(CC)CN(C(c2cccc(Br)c2)=O)CC1 c1(OC)cc(Cl)c(Br)cc1C(=O)NCC(CO)NC(C1(Br)CC1)=O Cc1noc(C2CC2)c1C(=O)NC1CCC1NC(=O)CC(O)CN(C)C CC1CC(=O)CCN1C(c1c(-n2cc(C3(CO)CC3)nn2)cccc1N)=O C1(C)(CC)C=C(C(=O)N2CC(C(C)NC(=O)C(C)C3(O)CCC3)C2)C1 N1(C(CC2CC(=C)C2)=O)CC(CC(=O)NCCC(C)N(C)C)C2(CC2)C1 c1(OC)cc(C(N2CC(NC(=O)Cc3cccc(Br)c3)C(C)C2)=O)cc(Cl)c1O C1(C(N2CCC(C)(NC(C3C=CC=CC=C3)=O)CC2)=O)CC2CCCCC2O1 C(C1(O)CCCc2ccccc21)NC(=O)NC12OCC(CF)(C1)C2 c1(CNC(C2(NC(C3CN(C(C)=O)C3)=O)CC(F)(F)C2)=O)nccc(C)c1F CC1(C(=O)NCCOCCC(=O)NC2CCCSC2)CCC(=O)C1 Cn1nc(CC(=O)NC2(C)CCN(C(=O)Cc3cncs3)C2)cc1C(F)(F)F N1(C(C(C)CF)=O)CC(NC(c2cc(O)cnc2N)=O)CC12CCC2 c1(CC)cccc(C(N2CCC(CN(C(=O)C(CCOC)OC)C)C2)=O)n1 C1(C(=O)NCC2N(C(C(CC)C)=O)CCCC2(C)C)CC(c2cnn(C)c2)=NO1 c1(C(=O)NC2CN(C(c3ccnc(C)n3)=O)C(C)C2)cc2ccc(Cl)c(F)c2o1 Cc1nc(Cl)nc(N2CCCC2(C)CNC(c2ccc(O)nc2)=O)c1Cl C(=O)(CCCCCN=[N+]=[N-])NC(C1(O)CN(C(c2cc3ncccc3[nH]2)=O)C1)C c1(CNC(=O)CCc2ccncc2)cc(O)nc(CNC(C2(N(C)C)CC2)=O)n1 C(=O)(C1=Cc2cccc(OC)c2OC1)N1CCC(CN(C(CCSCC)=O)C)C1 C1(NC(CCOCCOC)=O)CC2CCC1CC2NC(=O)C1=C(Cl)CCC1 Cc1ncnc(NCC(O)CNC(C2CN(C)CC2C(F)(F)F)=O)c1Br C(=O)(C1Cc2c(Cl)cccc21)N(CCN(C(c1c(C(=O)OC)scc1)=O)C)C Cn1c(=N)[nH]c2cc(C(=O)NC3COC4(CCCN(C(=O)CNC=O)C4)C3)ccc12 c1(C(N2CCC3(CC(NC(c4cnn[nH]4)=O)C3)C2)=O)ccnc2ccccc12 N1(C(C(C(C)C)O)=O)CCC2(CCCN(C(C3(C4CCCO4)CCC3)=O)C2)C1 C1(NC(c2ccc(NC(C3CCCO3)=O)c(Cl)c2)=O)CNCC2(CCC2)C1 C1(N(C)C(c2cocn2)=O)CCC(NC(C23CCCC2C3Br)=O)CC1 c1(C(=O)NC2CC(C)N(C(=O)Cn3cnnc3O)C2)ccc2ccc(Br)cc2n1 N1(C(c2cccc(C)c2F)=O)CC(NC(C2CN3CCCC2C3)=O)C2(CCC2)C1 c1(C(=O)NC(C2CCN(C(=O)CCC3CCCOC3)C2)C)ccc(C(F)F)o1 C(=O)(C(C)(O)C(C)(C)C)N1CC(COC)N(C(c2ccc(F)c(SC)c2)=O)CC1 CCC(C)(C)C(O)C(=O)N1CCN(C(=O)C=C2CCC2)CC1C1CC1 CCCC(C)CC(=O)N1CCC(F)(CNC(c2ccc(COC)[nH]2)=O)C1 c1(C(N(CCNC(c2c(C)onc2)=O)C2CC2)=O)nccc(N)c1Cl N1(CC(=O)NC(=O)NCCC)CCC(CNC(C2(C)CC(C#N)C2)=O)CC1 N1(C(C)=O)CSCC1C(=O)NC1CCC(CNC(=O)COC(F)F)C1 Cc1noc(C)c1S(=O)(=O)N1CCC(O)(CN2CCCC2c2ccc(Cl)cc2)C1 C(=O)(C#CC1(C)CCCO1)N(CC(=O)NC1CCC(C)C1)CC1CC1 CC1CCC(N2CCC(CC(C)NC(=O)C(=O)N)CC2)CC1.C1(C)CCCC(C)C1 c1(C(N(CCNC(CC2CC(=C)C2)=O)C(C)C)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 N1(C(=O)NC)CCN(N2CC(N(C)C(=O)OCc3ccccc3)C3(CC3)C2)C1 N1(C(c2ncn(C)c(=O)c2)=O)CCCCCC(NC(C2CC3C=CC2O3)=O)C1 C1(C)(NC(=O)NCC(CC)(C)OC(C)(C)C)CN(C(=O)OCC)CCO1 C1(C(=O)NC(C)CN(C)C(C2CN(C(N)=O)C2)=O)CCCN1c1nccs1 N1(C(c2c(C)ccc(=N)[nH]2)=O)CCC2(CCCN2C(C2CCCCC2(C)C)=O)C1 c1(C(=O)NC2(CC=C)CCN(C(c3ccnnc3)=O)C2)cnc(Br)c(OC)c1 c1(CC)cc(C(N2CC(F)CC2CNC(C2(C)CCCCO2)=O)=O)ccc1F N=c1ncc(C(=O)NC2CCCCC2NC(c2cocc2Br)=O)c[nH]1 C(=O)(C(CNC(=O)OC)CO)NCC(CNC(CC(C)C)=O)F.C(C)(C)(C)O c1(C(=O)NC2(C3N(C(CN(CCC#C)C)=O)CCC3)CC2)ccc(C(N)=O)nc1 C(=O)(CC(C)(C)C(C)=O)NC(C(=O)N(CCCOCC)C)C(C)CC N1(C(C(CCC(C)C)NC(C2CN(CC)C(=O)C2)=O)=O)CCCC2CCCCC12 c1(C(N2CC(CC(C)NC(C(CCSC)OC)=O)C2)=O)cc2ccccn2n1 C1(NC(C2CC(n3cccn3)C2)=O)CCN(C(c2cnco2)=O)CC12CCC2 c1(NC(C(N2CC3CCC2C(O)C3)c2nc(C)sc2C)=O)ccc2c(c1)CCC2 C1(C)(NC(C2C(=C)C2)=O)CCN(C(=O)C(C2CCCCC2)OC)C1 C1(C(=O)NCCCCCCN(C(C(C)NC(C)=O)=O)C)NC(=O)C2CCC12 C1(CNC(c2c(C)cncn2)=O)CC2(CCC2)CN1C(=O)CSCC#N Cc1nccc(C(=O)NC(C(=O)NCCC(=O)NC(C)C)C2(O)CCC2)c1N C1(NC(c2c(C)nccn2)=O)CC=C(C(=O)NCC2(C)CCOC2)C1 N1(C(CC=C)=O)CC2CCN(C(c3cc(-c4ccn(C)n4)on3)=O)C(C2)C1 C1(CC(=O)Nc2ccc(SCC)cc2)CCCN(C(=O)C(C(C)CC)OC)CC1 C(CCC=C(C)C)(C(=O)NCc1ccc(F)cc1)N(CC)Cc1cccs1 N1(C(CS(CC)(=O)=O)=O)CCN(C(=O)Cc2ccc(C)cc2Cl)C(C)CC1C CC1(C)C2CC(C(=O)N3CCC(C(=O)NCCn4ccnn4)O3)CC12 c1(C(=O)NCC23C(CN(C(CCc4c(C)ncs4)=O)C2)C3)cnc(N)c(Cl)c1 C(=O)(CCCCC(=O)NC(C1CCN(C(c2ccnn(C)c2=O)=O)C1)C)NC C(=O)(C1=NOC2COCC12)NC(CC(C)NC(c1ccc(C(=O)OC)o1)=O)C c1(C(=O)NCC2C(C)CN(C(=O)C(O)C3CCCC3)CC2)cccc(N=[N+]=[N-])c1 C1(CCC)(NC(=O)CC2CC=CC2)CCCN(C(C2CC(CN(C)C)C2)=O)C1 CC(C)(C)CC(O)C(=O)NCC(C)(CO)NC(=O)C#CC1(C)CC1 C1(NC(Cc2c(C)ocn2)=O)CC(O)CN(C(=O)C(C2CCCCCCC2)O)C1 c1(OC)cncc(C(=O)NC(C)C(C)NC(=O)CCCn2cncn2)n1 N#CC1CCCC1NC(=O)CC(CC1CC1)NC(=O)CC1CC(F)C1 Cc1noc(N)c1C(=O)NCCCCCN(C)C(C1CCC1n1ccnc1)=O c1(N(CC)CC2CCCN2C(c2cnc(C(C)(C)C)s2)=O)cnc(C#N)cn1 Cc1ccc2cc(C(N3CC4CC3CN4C(C3(O)CC(C)(C)C3)=O)=O)[nH]c2c1 C1(OCC(=O)N(C(CSCC=CCCC(C)=O)=O)C)CCOCC1 c1(C(=O)NC2C(O)CCN(C(c3cccc(C)c3)=O)C2)nc2ccc(F)cn2n1 c1(C(N2CCC(Oc3ccc(C)cn3)C2)=O)cncc(P(C)(C)=O)c1 C(=O)(C1SCCc2ccccc21)N1C(CNC(=O)Cc2ccc(F)c(Cl)c2)CC1 N1(C(C2CC(=C)C2)=O)CCCCC1C1(NC(=O)C(C)NC(=O)NC)CC1 C(=O)(C1=CCN(C(C2CCCOC2)=O)C1)N1C(C(=O)NC)CCC1 Cc1ncn(C)c(=O)c1C(N1CC2CC2(NC(=O)CC2CC3(CC3)C2)C1)=O n1(CC(=O)N(C2CCN(C(=O)CCCn3cccn3)C2)CC)cccc(C)c1=O CC(C)CC(CNC(C1(c2cc[nH]n2)CCC1)=O)NC(=O)Cc1cscn1 c1(NC(CCOC)c2nn[nH]n2)cc([N+](=O)[O-])cc(Cl)c1OC N1(C(C2(CC)CCC2)=O)CC2CN(C(C3CCSCC3)=O)CC(F)(F)C2C1 C(=O)(CCC(C)(C)NC(=O)C=CC(C)C)NC1(CCOC)CCC1 C1(C(C)C)CN(C(=O)CCC(C)C#N)CCCN1C(=O)C=Cc1cccc(Cl)c1 n1(CC(N2CCC3C(NC(CC4N(CC)CCC4)=O)C32)=O)cccc(N)c1=O N=c1[nH]c(C(N2CCC(CS(N)(=O)=O)C2)=O)nc2ccc(Br)cc12 C(=O)(CN=c1ccc(C#N)c[nH]1)NCC1C(CNC(c2c(C)cc(C)nc2)=O)C1 C1(NC(c2ccc(C#C)cc2)=O)C(CNC(=O)C(C)(C)CF)CCC12CCC2 Cc1cc(=NCC2CCCC(F)C2)[nH]cc1S(=O)(=O)NCCCn1cccn1 Cc1cc(F)ncc1NC(=O)C1=CCC(NC(c2ocnc2C(C)C)=O)C1 Cc1cc(Br)cc2cc(C(=O)N(C(C)CNC(=O)CC(C)(C)C#N)C)[nH]c12 CC1Oc2ccc(C(N3CCC4(CCC4)C3)C(=O)NC3CCCC3)cc2NC1=O c1(C(C(=O)NCCNC(C(CC)NC(=O)OC)=O)N(C)C)ccc(F)c(F)c1 N1(C(C(c2ccc(F)cc2)N(C)C2CC2)=O)CCCc2c(C(F)(F)F)cccc21 c1(CC(N2CCCCC2CN2CCCC2)=O)cccc2ccncc12 N1(C(C(=O)Nc2c(CC)cccc2)c2csnn2)CCC2(CC1)CNC(=O)N2 c1(CCCC(N2CCC(C(C)(C)NC(CCCC#N)=O)C2)=O)c(F)cccc1F N1(C(CCn2c(C)nc(C)n2)=O)CC(F)(F)CC1CNC(C1CCN(C)C1C)=O c1(CCC(=O)NC(C2CCCN(C(COC)=O)C2)C)cc(OC)ccc1OC C1(CNC(C2(SC)CN(C(C3CC(=C4CCC4)C3)=O)C2)=O)CCCCN1C C1(c2nc(C)[nH]n2)CN(CC(=O)N(C)CC2CCC(O)CC2)CCO1 c1(C(=O)NCC(C)(C)NC(Cc2cc(OC)no2)=O)cc2c(C)noc2cc1C C(=O)(C1CC(=O)C(=O)N1)NCCNC(CCSC)=O.C(C)(C)(C)OC(C)C.N(C)C S(=O)(=O)(c1c[nH]ccc1=NC(CO)C1CC1)NC(CCOC)c1ccco1 c1(SC(c2ccccc2)C(=O)NC(CC)C2CCC2)ccccc1O c1(CCC(=O)NCCCN(C(c2occc2F)=O)CC)cccc([N+](=O)[O-])c1 C1(NC(CC(C(C)C)O)=O)C2COCC1CC(NC(=O)C#CC1CCOCC1)C2 CN1CC(C)(C(=O)NCCCC2CN(C(C3CCC(O)CC3)=O)CCO2)CC1=O C1(N(C(=O)CCc2ccsc2)CC)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 Cc1cccc(OCc2ccc(-c3nnc(N4CCC(C)(CO)C4)n3C)cc2)c1 c1(C(N(CCNC(C(c2cccc(C)c2)C)=O)C2CC2)=O)ccc(N)c(C)c1C N1(CC)C(=O)CCC1CC(=O)NC1C2CC1N(C(=O)CNC(=O)CN(C)C)C2 C1(CNC(C(CSC)C)=O)(NC(c2cn(CCF)nn2)=O)CC2CCC1CC2 c1(C(N2CC(C)C(NC(=O)CC3CCCCCC3)CC2)=O)nccc2n[nH]cc12 C1(C(N(C2CCN(C(c3sc(O)nc3C)=O)CC2)CC#C)=O)CCC(N=[N+]=[N-])C1 C(=O)(C1=NOC(C)C1)NCCN1CCN(C(c2c(C)sc(O)n2)=O)CC1 N1(C(Cc2nc(C)sc2)=O)CCCC(CCCCNC(=O)Cc2cnccn2)C1 C1(O)(CNC(c2n(CC)ncn2)=O)CCN(C(C2(C)CCCC2(F)F)=O)CC1 N1(C(C(C)OCC#C)=O)CCN(C(c2ccc(CC)c(F)c2)=O)C(CF)C1 C1(C(NOCCC)=O)CC(C)CCN1C(C1CC=C(C)CC1)=O C1(C(=O)NCC2CC(NC(c3ncn(C(C)(C)C)n3)=O)C2)CCC2C(C1)C2(F)F C(=O)(C#CC1(CC)COC1)NC(CNC(COCCCOC)=O)CC c1(C(N(C(CCNC(CCOCCOC)=O)C)C)=O)ccc(F)c(C)c1C N1(C(Cc2scc(C)c2)=O)CCC2(CCN(c3nnc(CO)s3)C2)C1 N1(C(c2nccc(SC)n2)=O)CC2CC(Nc3cc(O)nc(O)n3)CC1C2 c1(C(=O)NC2C(NC(c3cnn(C(C)C)c3F)=O)COC2)cc(F)ncc1NC N1(C(c2c(C)nc[nH]2)=O)CC(C(=O)NC2COCC2CO)C(C)(C)C1 C(C(=O)N(C(CNC(=O)CCCCC1CC1)C1CC1)C)(C(C)C)SC Oc1ccnc(C2CCN(CC(F)C3CNC3)CC2)n1 C1(N(C(C(C)c2ccco2)=O)CCO)CCN(C(=O)CCCc2ncco2)C1 C1(C(=O)NCCCc2c(C)n[nH]c2)CN(C(=O)CCCC2CC2)CC12CC2 c1(C(=O)OC)cccc(N(C(=O)CC2CCN(C(c3cc(C)[nH]n3)=O)C2)C)c1 C1(C(N2C(C3CCN(C(CC4COC(C)(C)O4)=O)C3)CCC2)=O)Cc2cscc2C1 C1(C(=O)NC(C)CN(C)C)(CO)CCN(C(c2cscn2)=O)C1 N1(C(C(CC)(C)C)=O)CCN(C2CCNC2=O)C(C)C1 O=C1CC(C(=O)NC(C(=O)N2CC(SC(F)F)C2)C2CCC2)CC(=O)N1 N1(C(CCOCC#C)=O)CC2CC(C)N(C(c3cncc4nc(C)[nH]c34)=O)C2C1 c1(C(=O)NCC2(O)CCN(C(=O)C=C3CCCC3)C2)cccc2[nH]cc(Cl)c12 Cc1cnc(CC(=O)NCCC2CC(NC(=O)C=C3CCC(C)C3)C2)o1 c1(C(N(C2CCN(C(c3cccn3C)=O)CC2)C)=O)c(C#N)cnn1C Oc1c(CC2CN(c3ncc(F)cn3)CC23CC3)cccc1F c1(C(=O)NC2(CNC(c3occc3Cl)=O)CC2)ccnnc1O Cc1cc(C(N2CCC(NC(c3ccc(O)nn3)=O)C23CC3)=O)c(O)nn1 CN=c1[nH]c(C(N2CC(NC(=O)CCCNC(N)=O)C(n3cccn3)C2)=O)cs1 C1(C)(C(N(CC(CN(C(=O)Cc2ccon2)C)O)C)=O)CCC(F)(F)C1 c1(C(=O)NCCC2(O)CCCN(C(C(COC)OC)=O)C2)ccn2ccnc2c1 c1(CC(=O)NCCC(C)NC(C2CCO2)=O)c(F)cccc1F C1(CC(=O)N(C2CC2)CC2CCCN2C(c2cc[nH]n2)=O)CCCCO1 c1(C(=O)NCC(CNC(C(CCC)OCC)=O)(C)OC)c[nH]c(=N)c2[nH]ccc12 c1(C(N2C(C(N3CC(=O)NC(C)C3)=O)CC(=C)C2)=O)ccc([N+](=O)[O-])c(O)c1 N1(C(C2CC=C(C)CC2)=O)CCN(C(=O)CC2C=CCC2)CC1CCO CC(C)(C)C(=O)CCC(=O)N1C(C(N2CCOCC2CC2CC2)=O)CCC12CC2 CN1CCN(C)C(CNC(=O)C(CC(F)F)N(C)C(C2CCCNC2=O)=O)C1 C1(O)(CN(C)C(C2C3COCC23)=O)CN(C(=O)CC23CCCC2C3)C1 c1(-c2n(CC=C)c(N(C)CC3(OC)CCC3)nn2)cc(=O)c(O)co1 c1(CNC(C(C)NC(C)=O)=O)cc(C(=O)NCC(C)OC(F)F)n(C)n1 c1(C=O)ccncn1.C(=O)(C(C)N(C(C1CC1CF)=O)C1CC1)OCC c1(OCCOC)ccc([N+](=O)[O-])c(C(=O)NC2CCC3CCCCC3C2)c1 c1(C(=O)NC2C(C(C)NC(=O)OC(C)(C)C)C2)cc(S(=O)(=O)NC(C)C)c(C)o1 C(=O)(C1SCc2cccnc21)N1CCC(NC(c2cc(O)ccc2F)=O)C(O)C1 N1(C(CC2CC(CC)C2)=O)CC2CCC1CC2NC(c1cnn[nH]1)=O C(=O)(C(C)(C)CCCCC)N1CC(NC(=O)C(C)OC2CCCC2)CC(OC)C1 N1(C(C2(OCC)CCOCC2)=O)CC2CC(C1)N(c1cc(C)nc(SC)n1)C2 N1(CC)CC2(C1)CN(CC1C=CC(N(C)CC3(NC(C)C)CCC3)C1)C2 c1(C(N2CCC(NC(Cc3cc(C)on3)=O)(CF)C2)=O)ncnc(O)c1Br CC1CC(C(=O)N2CCC(NC(c3c(C(F)(F)F)cnn3C)=O)C2)=NO1 c1(C(=O)NCC(C2N(C(C=CC(CC)=CC)=O)CCC2)(C)C)ccc(C)c(O)n1 C(=O)(C1=C(C)CCCC1(C)C)NCC(C(C)(C)C)NC(CC(CC)(C)C)=O c1(CC)cc(Br)ccc1C(=O)NCC1CN(Cc2ccc(C(F)(F)F)c(O)c2)C1 n1(CC)nc(C)cc1C(=O)NC1CCCC(NC(C2CC(C(F)(F)F)C2)=O)C1 C1(C(=O)NC(C)CCNC(C2(C)CSC2)=O)CCc2cnn(C)c2C1 c1(CCC(=O)N(CC(CNC(C2C(CCOC)C2)=O)C)C)cccn1C N1(C(=O)CC(C(N2CCC(CCO)C2)=O)c2ccoc2)CCC2(C=CCO2)CC1 C(=O)(C(F)CCC(C)C)NCC(CCOC)NC(c1ccncc1N)=O c1(NC)ccc(F)cc1C(=O)NCCC1CCN(C(=O)C(C)CSC)C1 O(NC(=O)CC(C)(C)N(C)C(C1(O)CCSCC1)=O)C1CCCN(CC)C1 Cc1cc(C(N2CC(CNC(C3COC(=O)N3C)=O)C(C)C2)=O)n(C2CCC2)n1 CCC(Cc1nc(-c2cccs2)nn1Cc1cc(C)nc(C)c1)CC(F)F C1(CNC(CCNC(C)=O)=O)CN(C(=O)C(C)c2ccsc2)CC1C CC12CCOC(C(N3CCC(NC(c4ccc(F)s4)=O)C3(C)C)=O)(C1)C2 N1(C(c2cc3ccc(Br)cc3o2)=O)CCC2CCN(C(=O)C3CC3)CC2C1 c1(C(=O)Nc2ccc(C(=O)Nc3cncc(Cl)n3)cn2)onc2ccccc12 C(=O)(CCCC(C)(F)F)NC(CNC(CN(C(C)C)C)=O)C(C)C(C)C c1(CCC(N2CCCN(C(C(CC)C#N)=O)C(C)C2)=O)cccc2c1OCCO2 C1(OC)CC2CN(C(C3C(C)(C)C3(F)F)=O)Cc3cccnc3N2C1 C(CCC)(C(=O)N1CCC(C)(NC(c2cc(OC)no2)=O)C1)=CCC C1(O)(CN(C(Cc2c(C)noc2Cl)=O)C)CCCN(C(C2C=CCC2)=O)C1 C(=O)(C(CC(=O)OC)OC(C)(C)C)NC(CN(C(C=COCC)=O)CC)C c1(OCC)ncc(C(=O)O)cc1NC1CCCC1c1ccc(Br)cc1 c1(N2CC3(C(NC(=O)COC4CCOCC4)CCC3)C2)ccc([N+](=O)[O-])c(O)n1 CC(C)C(F)C(=O)N(C)CC1(C)CCCC1NC(=O)CSc1ccc(O)cc1 C(c1ccn(C)c1)=CC(=O)NC1C(NC(CCc2scc(C)n2)=O)CC1 N1(C(c2c(C)c(F)cnc2)=O)CC(C)N(C(=O)C(C)C(C)C)C(C)C1 N1(C(CCCSC)=O)CCC2CCCC12CNC(c1cn(C)c(C)n1)=O c1(C(=O)NC(CC)CNC(=O)C(C)(F)C(C)(C)F)cc([N+](=O)[O-])ccc1SC CCC1=NOC(C(N2CC(CNC(c3ccccc3Br)=O)C2)=O)C1 N1(C(CC(C)O)=O)CC(CNC(=O)Cc2csc(C3CCCC3)n2)CC(C)(C)C1 C1(F)(CNC(c2c(CC)n(CC)nn2)=O)CCN(C(=O)C(C)=CC2CC2)CC1 N1(C(C2CC(C(=O)OC)C2)=O)CC2CC3CC2C1C3NC(C1CC(O)C(F)C1)=O N1(C(c2nc(OCC)oc2)=O)CCN(C(C2CC(C)CO2)=O)CC1CCO CC1CN(C(=O)CCN2CCN(C)CC2)CCC1NC(=O)C(C1CCC1)C1CC1 C(C)(CO)(C(=O)N1CC(C(C)(C)C#N)C1)NC(c1nc(CC)oc1)=O N1(C(=O)CCF)CC2CC(C1)N(C(=O)C(Cc1ccccc1)C1CCCC1)C2 N1(CCC(=O)NC(C(C)NC(c2cn(C)c(O)n2)=O)C)CCc2ccccc2C1 C1(NC(CC(CNC(CCCCSC)=O)O)=O)C(O)C2CCCC12 C(=O)(CC(C)(C)C(=O)N1CC2=C(C1)CN(C(=O)C(=O)NCC(F)F)C2)OCC N1(C(CSC)=O)CCC2(CC1)CC2(CO)CNC(=O)Cc1sccc1Cl c1(N)cccc(S(=O)(=O)N2CCCC2)c1.C(=O)(CP(C)(C)=O)NC(C)CCSC c1(OC)c(C)cc(C(=O)NCC#CCNC(=O)CSSC)cc1C C1(NC(CC2C(C)CCC2)=O)CN(C(=O)CN(C(=O)C2CC2)CCC)CCC1(C)C c1(C(N2CCC3(CCOC3)C2)=O)n[nH]c2c1CN(Cc1c(F)cc(Cl)cc1Cl)C2 C1(CC(=O)NCC(C)CNC(C2CC(N(C)C)C2)=O)CCC2(CCC2)O1 c1(C(=O)NC2C(C)(C)N(C(C3CC(F)(CO)C3)=O)CC2)ccnc2c1CCO2 c1(CN(C)Cc2cccc(C)c2)cc(Cl)c(Cl)n1C Cn1cc(NCC2CC(NC(C34CCC3C4)=O)C2)c(OCC(F)F)n1 C(CN=c1[nH]c(=NCc2cnc[nH]2)[nH]c2cccc(F)c12)OCC(C)C N1(C(C2(CC(=O)NCN)CC2)C)CCC(C)C2(CCC2)C1.n1(CC=O)ncccc1=O c1(C(CNC(=O)CCOCC(F)F)NC(C(C)SC)=O)ccccc1F C(=O)(C(C)(C)C1=CCN(C(C2CC2C(F)F)=O)C1)NCc1c(C)cn(C)n1 C1(NC(C2CC(C(C)C)C2)=O)C2CC(NC(=O)C(F)(F)CO)CC12 C1(NC(c2nc(CC)oc2)=O)CCN(C(C23CC(F)(C2)C3)=O)C(C2CC2)C1 C1(CNC(CC(C)(C)NC(Cc2c(C)ocn2)=O)=O)CC2(CC2)C(=O)O1 c1(C(=O)NCC2(O)CCN(C(c3cc(C)c(C#N)[nH]3)=O)C2)ncnc2ccsc12 C1(C)(CC)CN(C(C2CC(N(C)C(c3cncs3)=O)C2)=O)CCO1 C(=O)(CC1C(=O)Nc2ccccc21)NCCCN(C(C)=O)Cc1nnc(C)o1 C1(C(=O)NC2(C(=O)NCC3CCN3C(C)(C)C)C(C)C2)CN(C)CCN1C Cc1oc(-c2ccccc2)nc1CC(=O)NCC1(O)CN(C(=O)C=CC2CC2)C1 c1(CNC(c2c(C)cccc2)C2CCC(C(=O)N(C)C)CC2)cncc(C#N)c1 c1(CNC(CC2CCCC(OCC)C2)=O)cnn2c1CN(c1nncs1)CC2 c1(NC(C(F)=C(C)C)=O)cccc(NC(=O)C(F)Cc2ccccc2)c1 c1(C(=O)NCCCC2N(C(C=CC=CCC)=O)CCC2)cc(=O)c(OC)cn1C c1(-c2n(CCCCCC)nnn2)c(C)nn(CCNCC)c1CC N1(C(C(C)N(CCOCC)CC)=O)CCC(C(C)(C)O)CC1.C(C)(C(=O)OC)N c1(C(C(=O)NC2CCC2)N(CCC(C)C)C)cc(Cl)cc(Cl)c1 c1(N(C)CC2(C)CCCC2)ccncc1S(=O)(=O)N1CCOC(C(C)(C)C)CC1 c1(C(=O)NC(C2CCCN(Cc3cccc(C#N)n3)C2)C)ccc(F)c(Cl)c1F c1(CC(=O)NC2C(CNC(C(CCC)OC)=O)CC2)ccc(C)cc1Br N1(C(c2c(C)nn[nH]2)=O)CCCCC(NC(=O)CCSC(F)(F)F)CC1 c1(CNC(c2ccc(C)o2)=O)ccc(CCNC(=O)Cc2cnc[nH]2)cc1 N1(C(C2(CCC=C)CN(C(c3ncncc3C)=O)C2)=O)CCOC2CCCC12 C1(COC)(CNC(=O)CCCC2CCC2)CCCN1C(=O)Cn1nc(C)nc1C N1(C(c2ccc(COC)o2)=O)CCOC(C)(CNC(c2cc(SC)c(C)o2)=O)C1 Cc1cc(F)ccc1N(C)C(=O)N(C1CC1)CC1(c2ccc(Br)cc2)CCCC1 C1(C(N2C(C)(CC(=O)NCc3n(C(C)C)ncc3)CC2)=O)COCCC1C C1(C(=O)OCc2ccc(COC)s2)CC12CC(S(=O)(=O)N1CCCC1)C2 CC1CCN(C(C2CC(O)CCN2C(c2cnnc(O)c2)=O)=O)C1(C)C C1(CNC(c2c(C)nc(CCC)s2)=O)CN(C(C2CCCCO2)=O)CCN1C c1(OC)ccc(N)c(C(N2CC(CNC(C3(C)CC=CCO3)=O)CC2(C)C)=O)c1 C1(NC(C2(SCC)CC2)=O)CCN(C(c2c(C)[nH]c(C)c2C)=O)CC1C(C)C N1(C(CCCC(=O)NCC)=O)CCC(C2(NC(c3nnc(CC)s3)=O)CC2)C1 Cc1cc(=NC(CC2CC2)C2CC2)[nH]c(=NCc2nc3ccc(F)c(F)c3[nH]2)[nH]1 C1(C)(NC(CCCCOCC)=O)CCCCC1C.C1C(=O)N1 c1(C(N(C(c2ccncc2)CC)CC)=O)ccc(Br)cc1-n1cncn1 CC1(C)CN(C(=O)C(c2ccc(F)cc2F)(C)C)CCC1NC(=O)C1=NOCC1 N1(C(CN(C)C)=O)CCOC(c2cc(C(=O)NC(C)(C)C)n(-c3ccncc3)n2)C1 C1(NC(=O)C(C2CCCO2)C2CC2)CC2CN(C(=O)C=C3CCCCC3)CC12 c1(CCC(C)C)ccc(CNS(=O)(=O)CC2CCCC(C(F)(F)F)C2)cc1 c1(C(N(CCC(=O)NC2CCC2C)CC=C)=O)cn(C)c(C)n1 C(=O)(C#CC1CCCO1)N1CCC(NC(c2nccc(OC)c2)=O)C1C(C)(C)C N1(C(C=CCC2(NC(=O)CC3C=CCC3)CC2)=O)CCC(F)(F)C(F)C1 CN1C(=O)CCC1C(=O)NCC(C1CCCN1c1nc(C(C)(C)C)ns1)(C)C C1CCOC(C)(C)C1.c1(C(=O)OC)ccc(CNC(=O)Cn2cc(CN)nn2)s1 N1(C(CNC=O)=O)CC2(CC(CNC(c3ccc(F)c(C(F)F)c3)=O)C2)C1 C1(C(=O)NCC2(O)CCC(C)C2)CC2(CCN1C(c1cn(C)c(=O)n1C)=O)CC2 c1(C(=O)OCc2cccc(SCC)c2)ccc(Cl)c(Br)c1 c1(SCC(=O)NCc2csc(CNC(C3CCC(F)C3)=O)n2)ccc(F)cc1 c1(NC(N(CC(CC)NC(=O)C(F)C(C)C)C)=O)cn(-c2cnn(C)c2)[nH]c1=N C1(C)(C(=O)NC(C)CCN(C)C(c2ccon2)=O)CCCCC1(F)F C(=O)(CCCCC(=O)N1CC(O)(CNC(C2CCCC2(C)OC)=O)C1)OC c1(CC)ccc(C(=O)NCC23CC2CN(C(=O)CC(C)n2ccc(C)n2)C3)cn1 CC(C)C(C(C)NC(c1cccc(N2CC=CC2)c1)=O)NC(=O)COC(F)F N1(C(=O)COCCF)CCN(C(=O)C=Cc2ccccn2)C(CF)C1 c1(OC)cc(C(N2CCC(C)(NC(c3ccc(=N)[nH]c3)=O)CC2)=O)cc(F)c1F O=C(C1=NOC(C2COC2)C1)NCC1CCN1C(c1ncoc1C1CCCO1)=O c1(C(=O)NC2CN(C(=O)CCN3CCCCC3=O)C2)cc(F)cc2nccnc12 c1(C(N2CCC(NC(C=C(C)C3CC3)=O)C2)=O)ccncc1-n1cccn1 c1(C(C)CC(N2CC3CC2C3NC(=O)CN2CCNC2=O)=O)ccc(F)cc1F C1(C(=O)NC2(CC(=O)NCc3cccnc3F)CCC2)Cc2nccn2C1 n1(CC(=O)N(CCOC)CCNC(=O)C(CO)N(C)C)cc(C)c(O)nc1=O C1(CNC(CCCCOC)=O)(NC(=O)C(C)c2cccs2)CC2CCC1CC2 CC1CC(CNC(C2(F)CCOCC2)=O)CN(C(C23CC(C)(CCO2)C3)=O)C1 C(C1=CCCN(C)C1)NC(C1(CNC(C(CSC)OC)=O)CCC1)=O N1(C(c2ncc(C)nc2)=O)CCN(C)CC1CNC(C1CCOC1C)=O CCCCC(CNC(c1csc(COC)n1)=O)NC(c1ccccc1Cl)=O N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CCC1C CC1(C)CNCCN1C(C1CC1NCc1ccc(Br)c(CO)c1)=O N1(C(CCNC(C)=O)=O)CC2CCN(C(C3CCOC3c3ccccc3)=O)CC12 N1(C(C(c2ccc(Cl)cc2F)CC)=O)CC(Cn2cc(CSCC)nn2)C2(CC2)C1 S(=O)(=O)(c1cc(C)c(-c2ccc(OC)cc2)cc1C)NC(C(CC)CC)C(=O)OC C(CC(C)(C)C(=O)NCCc1cc(C(=O)NCC2(CCO)CCC2)no1)OC N1(C(COCCC(C)C)=O)CCC(CNC(=O)COc2ccsn2)C(F)(F)CC1 c1(C(N2CC(CN(C(C3(CCC)CC3)=O)C)OCC2)=O)cc(OC)ncc1F c1(C(N2C(C3(C(=O)OCC)CC3)CCCC2)=O)cc2cc(Cl)ccc2o1 C1(CNC(COCC(=O)OC)=O)C(O)C(O)CN1C(N1CC(N)C1)=O.C(C)(C)C CC(C)(C)C#CC(=O)NCC1(F)CCN(C(=O)CSc2ccccc2)C1 N1(C(C(C)OCCC#C)=O)CCCC(n2cc(CNC(=O)CCC3CC3)nn2)C1 n1(CC(=O)NC(C)CCCNC(=O)CC2CCCCN2C)ccc(=O)n(C)c1=O N1(C(C2COCCN(C(C(CC(C)(C)C)O)=O)C2)=O)CCc2nccnc2C1 C1(N(C(c2c(SC)scc2)=O)C)CCN(C(=O)C#CC2(C(F)(F)F)CC2)CC1C c1(CCCC(=O)NC2C(NC(C(CC)=CC)=O)COCC2)c[nH]c2ccccc12 C12(C(N(CCCN(C(c3cc(COC)cn3C)=O)C)C)=O)CC(C)(C1)OC2C c1(NC2CCCCN(C(C(C=C)(C)O)=O)C2)ncc(S(C)(=O)=O)cc1Cl N1(C(C2C=CCN(C(CC=CCC)=O)C2)=O)CCN2CCOCC2C1 C1(C)(CNC(c2nnn(C)n2)=O)CN(C(=O)CCSC(F)(F)F)C(C)(C)C1 C1(C(=O)NC(CN(C(c2cnsn2)=O)CC)C)CCCN(c2cnccn2)C1 C1(C(=O)OCC)Cc2cccc(NC(=O)N(CC(C)C)CCO)c2C1 Brc1ccc2nc(CN3CCN4CCCCC4C3)cn2c1 C1(NC(CCC)=O)CN(C(=O)C(O)Cc2c(F)cccc2Cl)CC(C)(C)C1 c1(C(N2CC(c3cn(C(C(=O)OC)C)nn3)C2)=O)cc2c(s1)CCCC2 Cc1c(NC(=O)C(C)(C2CC2)N(C)C(C2CCOC2(C)C)=O)cccc1C#N c1(C(C(=O)NCC2CCCN2C(C2COC2)=O)O)ccc(Cl)cc1 c1(C(=O)NCCC2CCN(CCCC(=C)C)C2)c(C)noc1C(F)F c1(C(N2CCC(COC)(NC(=O)CSC)C2)=O)cnc2n1C(C)CCC2 C1(SC(C(=O)NCCCC)CC)CNCC1(C)C CC1(C)CC(=O)NCC1C(N1CCN(C(c2c[nH]nc2F)=O)CC1CC(F)F)=O c1(C(C)(C)C)ccc(C(=O)NC2CCC2NC(c2ccccc2)=O)[nH]1 c1(OC2CC(=O)N(C3CC3)C2)ccc2c(c1)COC2 CC1CC=C(C(=O)N2CC(C(=O)NC3CC(CCC(N)=O)C3)C(F)C2)CC1 c1(CC)ccc(C(N2CCC(CN(C)C(C3CN(C(N)=O)C3)=O)C2)=O)cc1 N1(c2ccnc(C)n2)CCN(C2CCCN(C(c3cnoc3C)=O)C2)C(=O)C1 N1(C(c2c(CC)ccc(Br)c2)=O)CCCN(C(=O)C(O)C(C)C)CCC1 N1(C(CC)=O)C(CNC(=O)C(F)(F)c2ccncc2)CC2CCCCC12 C(CC(N=c1[nH]c(=NCC(C)(C)C2OCCO2)[nH]c2c1CCC2)C(C)C)OCC Cc1cc(CNC(=O)C(C(C)O)NC(C2CCCN2C)=O)nn1C C1(CC)CCCC1(C)C(N1CC(C(C)NC(c2cnc(C(F)(F)F)nc2)=O)C1)=O C1(C(=O)NCC(CC)NC(c2ccc(C(F)F)c(F)c2)=O)CCn2ccnc2C1 C12CC(n3cc(CCCSC4CC4)nn3)CN1C2=O.C1(C(=O)O)(COC)CCC1 c1(C(=O)NCC=CCNC(Cc2nc(C)sc2C)=O)ccnc(O)c1Br C(=O)(N=c1cc(-c2ccsc2)[nH][nH]1)C1C2CN(C(=O)CN3CCCC3=O)CC21 C1(NC(C=Cc2nc(C)sc2)=O)CCC12CCN(C(C1CC1(C)C)=O)CC2 C1(C(=O)NC2CCC(NC(CNC(=O)OCC)=O)C2)NC(=O)CC1C C1(C(N(CCN(C(C(C)=CC)=O)C)C)=O)CCN(C2CCS(=O)(=O)C2)CC1 c1(C(=O)NC2(C)CCN(C(c3cc(Br)no3)=O)C2)ccc(C2CC2)c(F)c1 N1(C(C(C)(C)OCC)=O)C2CCC1CN(C(c1oc(C)nc1C(F)(F)F)=O)C2 CC1(C)COCC(CC(=O)NCC2CCN2C(c2sccc2F)=O)O1 c1(C(=O)NCC2CC(NC(C3CS(=O)(=O)N3)=O)C2)coc2ccc(Cl)cc12 C=CCCC(C(=O)OC)Sc1c(C(=O)OC)cnn1-c1cccc(C)c1 c1(NC(C2(CC=C)CN(C(C3CC(=O)N(CC)C3)=O)C2)=O)ccnc(OCC)c1 C1(C(=O)NCCN(C(c2c(C)noc2C(F)F)=O)C)CCCC2(CCOCC2)O1 Cc1ccc(Cl)c(OCC(=O)NCCCCNC(c2csc(S)n2)=O)c1 C=CC1CCN(C(=O)C(C2CCCOC2)NC(=O)OC(C)(C)C)CC1 N1(CC(N2CC=CC2CNC(C2(F)CC=CC2)=O)=O)CCCCC(O)C1=O C1(C(C)(F)F)(C(=O)NC2CCC(CNC(C3CCC(=O)N3C)=O)C2)CCOCC1 C1(C(N2C(CCNC(C)=O)COCC2)=O)CC2OC(C)(C)OC2C1 c1(CO)cnn2c1CN(Cc1cccc(C(=O)Nc3ccc(O)cc3Cl)c1)CC2 c1(CC)[nH]ccc1C(N1CC(O)(C2CCCN2C(C2CNC(=O)C2)=O)C1)=O c1(C(=O)NCCC(CC)(C)NC(=O)C(F)C(F)(F)F)ccc(C)cc1C CN1CCN(C(=O)CC2(C(F)(F)F)CC2)C(CNC(=O)CN2CCOC2=O)C1 Cc1coc(C=CC(N2CCN(c3ncc(Br)cn3)CC2)=O)n1.C(=O)(CC(C)C)N C1(OC)(CNC(=O)C=C2CCC2)CCN(C(c2ncccc2CC2CCC2)=O)C1 c1(CC2CC2)ccc2c(c1)OCO2.Cc1cccc(O)c1C1C2CC2C(=O)N1 CCCCCC(=O)NCC1CN(C(C2CCCC2NC(=O)C(C)C(C)C)=O)C1 N1(C(C(C)CN(C)C)=O)CC(C(=O)NC2(C(N)=O)CC2)CC12CCC2 N1(C(C(CC(=C)C)OC)=O)CCC2(CCCC2NC(c2nc(Cl)cs2)=O)CC1 Cc1cccc2oc(C(=O)N(C3CCN(CC(C)CC(C)C)C3)C)cc12 C1(CNC(C(CC)Oc2ccccc2Cl)=O)(CO)CCCN(C(=O)CC(C)C)C1 S(=O)(=O)(c1ccccc1Br)NC(C(=O)NCCC=CCCCCC)C(C)O Cc1nn(C)c(F)c1C(=O)NCC1CCCCN1C(=O)CC1COCC1O C12(CNC(C(C)(C)F)=O)CN(C(=O)Cn3ccccc3=O)CC1CCO2 N1(C(CCC(=O)NC)=O)CCC(CNC(=O)COCC2CCCC2)C12CC2 N1(C(C(C)O)=O)CC2CC(NC(=O)COc3ccc(F)cc3Br)CC(C2)C1 Cc1ccnc2nc(C(N3CCC(NC(=O)CCOCC(F)F)C(F)C3)=O)nn12 C(=O)(CC1=CCN(C(c2ccc(C)c(F)c2)=O)CC1)NCC1CC(C(=O)OC)C1 C1(C(=O)NC2CC(C(C(=O)NCc3c(C)ncs3)F)C2)CCCCC(=O)N1 c1(OC)cc(F)c(C(N2CCC(NC(=O)C(O)C(C)C)C2)=O)cc1N S(=O)(=O)(c1cccc(=NCCn2cncn2)[nH]1)N1C(CNC(N)=O)CCC1 c1(CCC(=O)NCC(CNC(C2(O)CCOC2)=O)OC)cscc1Br CCC(O)(CNC(=O)C(C)N(C(c1cnn(C)c1OC)=O)C1CC1)CC N1(C(c2ccc(COC)o2)=O)CC(NC(=O)CC2CCOCC2)C(C)C1 c1(C(N(C)CCN(c2ccnc(C#N)n2)C)=O)cc(F)cc2nccnc12 S(=O)(=O)(c1cnccc1N1CCC2(C1)OCCO2)NCc1ncc(C)nc1 Cc1nc(SC(F)F)sc1C(=O)N(CCCNC(=O)CNC(N)=O)CCO C1(NC(C2CC(C(C)=O)C2(C)C)=O)CN(C(=O)C=C2CCN(C)C2)CC1(C)C C(=O)(C(CN(C(=O)C=CCF)C(C)C)N(C(=O)CC(C)n1cccn1)C)OC C1(CNC(c2scc(OC)c2)=O)CN(C(C2(C)CC2(Cl)Cl)=O)CCO1 C(C(=O)N=c1ccn(CCO)[nH]1)(C1CCCC1)NC(CC1CCC(=O)CC1)=O N1(C(CC(=C)C)=O)CC2(CCCC(CNC(c3cc(O)nc(C4CC4)n3)=O)O2)C1 CC(C)C(C(C)NC(=O)CO)NC(=O)CCNC(c1cc(-c2ccco2)[nH]n1)=O c1(OCC(=O)N(CCCN(C(C2(C)C(C)CCC2)=O)C)C)cccc(C#N)c1 N1(C(c2cc(CCC)[nH]n2)=O)CCN(C)C(C(=O)NC2CC=CCC2)C1 C1(NC(CC(=C)I)=O)CC12CC(NC(=O)C(O)C1CC1)C2 C1(NC(c2ccc(C)nc2)=O)CC2CN(C(c3cnco3)=O)CCN2C1=O c1(C(=O)NCC2CCC(NC(C(C(C)C)N(C)C)=O)C2)ccc(=O)n(O)c1 C1(NC(C2C(C(C)C)OCC2)=O)CC=CCC1C(N1CCCCC1CCO)=O C(C(C)C(C)C(=O)NCC1=CCN(C(c2cc(O)nc(OC)n2)=O)CC1)OC N1(Cc2c(C)n[nH]c2C)CCC2(CC1)C(O)CC(C(=O)O)C2 C1(NC(C2ON=C(C)C2)=O)CCC(C)(NC(C2CCCCCC2)=O)CC1 Cc1ccc(N2CC(NC(C3CC4OC3C3CC43)=O)CCC2=O)cc1C C(=O)(C(F)CCC(C)(C)C)NCC(C(=O)NCc1nn(CC)nc1C)(C)C N1(C(C(F)=CC)=O)CC(C)(C)OCC1CNC(=O)COc1cc(F)ccc1F N1(C(C(C)CC(N)=O)=O)CC(NC(=O)C(C)N2CCCC2)CC12CCCCC2 CC1CN(C(c2cc(Br)cc(N)n2)=O)CC(C)C1NC(c1ccon1)=O O=C(CCCC(F)C(=O)O)N1CCC2CC(C(=O)NCC(O)C(F)(F)F)C2C1 c1(C(N)=O)cccc2c1CN(C(=O)CC1CCN(C(C3CCC(=O)O3)=O)CC1)C2 CCC(C)CC(C)C(=O)N1CCC(C)(C)C(Nc2ccccc2[N+](=O)[O-])C1 C1(CNC(C(C)O)=O)CCC2(CN(C(c3ccc(F)cc3O)=O)C2)O1 C12(NC(C#CC3(C)CC3)=O)CCOCC1CN(C(=O)Cc1ccns1)C2 c1(C(=O)NCC(CNC(c2cnc(OCC)s2)=O)C)nc(O)nc(O)c1N N1(C(C(N)=O)=O)CC2(CCN(C(=O)COCCCF)C2)C1.c12ccc(Cl)c(c1)O2 N1(C(C2(C)CC2C(F)(F)F)=O)CCCC1(C)C(=O)NCC1CCCOC1 C1(NC(Cc2n(C(C)C)cnn2)=O)CCOC2(C1)CC(C(=O)O)C2 c1(C(=O)NC2(C)CC(NC(C(COC)OC)=O)C2)ccccc1-c1ccccc1 C1(CNC(C(C)NC(C)=O)=O)CN(C(C2CC2C2(C)COC2)=O)CCC12CCC2 C1(C2(O)CCOCC2)(C(N2C3CCC(NC(CC(C(C)C)O)=O)(CC3)C2)=O)CC1 c1(CNCc2cnn(C)c2Cl)c[nH]c2ncccc12.N12CC3CC1C3C2=O C1(CC)CN(C(c2cn(C)c(C)n2)=O)CCC1NC(c1ccc(O)c(C)c1)=O c1(C(=O)NCCN(C(c2c(CC)nccc2)=O)C(C)C)ccn2c(C)ncc2c1 N1(C(c2ccc(CC(=O)OCC)o2)C(=O)NCC)CCOC2(COC(C)(C)C2)C1 c1(C(=O)NCC2(COC)CCCN2C(=O)CCF)cc(Br)c(F)cc1N CC1(C)CN(C(=O)Cc2cncnc2)CC(C)(C)C1NC(=O)CCCCC#N CCC(CN(C)C)C(=O)NCC(CC(=O)NC(C)(CO)CO)C1CCC1 N1(C(CCC(CCC)CC)=O)CCOC2(CCSCC2)CC1 CCS(=O)(=O)NC(C)C(=O)N(CC(C)(C)NC(=O)C(C)c1ccco1)C C1(NC(c2n(CC)nc(C(C)C)c2)=O)CCCN(C(=O)C2=CCCO2)CC1 CC(C)(C)CCC(F)C(=O)N1CCCC1C1(NC(=O)CCCF)CC1 c1(CC)nn(C)c(CC)c1C(=O)N(CC(C)(C)NC(=O)C(CC)CC)C C(C1CCOc2ccc(Br)cc21)NCc1n[nH]c(C)c1C c1(C(=O)NCC(C)(CO)NC(C2CC3CC3C2)=O)nc2n(c1Cl)CCCC2 C12(CNC(=O)C3=NOCC3)CN(C(=O)C=Cc3cccnc3)CC1CS(=O)(=O)C2 Cc1cc(C)c(C(=O)N(CC(C)(C)CNC(c2cc(C(F)F)no2)=O)C)cn1 N1(C(C(C)CC2CC2)=O)CC2(CC(CNC(=O)Cn3cnnn3)C2)C1 C1(NC(CCSCC)=O)CCCCCN(C(=O)Cc2csc3cc(C)sc23)C1 C1(N(C(C2C(=C)C2)=O)CC)CCN(C(=O)C=Cc2ncc[nH]2)CC1 N1(C(c2c(CN(C)C)cco2)=O)CCN(C(C2(CC(F)F)CCC2)=O)CC1CO CC1CC(F)(F)CN1C(C1CSCCN1C(=O)C=CC(F)F)=O Cc1cc(C(=O)NCC2CN(C(C3Cc4nccn4C3)=O)CC2O)c(C)cc1Cl c1(OC)cc(C(N2CC(=C(F)C(=O)OCC3CC3)C2)=O)cc([N+](=O)[O-])c1OC C1(C(N2CCN(C(C(CC)CC)=O)C(CF)C2)=O)CC2CC1CC2(F)F C1(OC)(CNC(=O)CCF)CCN(C(=O)CC(O)CNC(=O)OC(C)(C)C)CC1 c1(C(=O)NC(CCNC(CCC2C(C)C2)=O)c2cccs2)cc2cn[nH]c2cn1 CCC(C(=O)N(C)CC1CCN(C(c2sc(C3CC3)nc2C)=O)C1)C(C)(C)CC c1(C(=O)NC2CCCCC2C(N2CCS(=O)CC2)=O)cc(O)nc(O)c1 C12(C(=O)Nc3c(NC(C)=O)cn(C)n3)CCCC(CO1)C2.C1C(=O)NCC(C)O1 C(=O)(CCCCCNC(C1CC2COCC2C1)=O)N(CC(COC)(C)C)C N1(C(Cc2ccc(C#C)cc2)=O)CCN(C(=O)CSCC)C2COCC12 CC(C)(F)CCC(=O)NC1CCCC(C(N2CCC3C(O)CC23)=O)C1 CC(C)CCCCC(C)NCCCc1ccncc1 c1(CNC(N2CCN(S(=O)(=O)C3CC3)CC2)=O)cccc2cncn12 C1(N(C(c2ccn(CCC)n2)=O)C)CCN(C(C2CCCN2C=O)=O)CC1 C1(CC)CN(C(=O)C=Cc2cccc(CO)c2)CCC1NC(c1ccc(C)[nH]1)=O C12(C(N3CCCC(CCC#C)C3)=O)CCCC1CCN2C(C1CCCC(=O)C1)=O N1(C(C(CC)CC2CCCC2)=O)CC(NC(c2ccon2)=O)CC12CCOCC2 C1(C)(C(=O)NCC2(CO)C(C=C)C2)C=CCN1C(C1OCCC1(C)C)=O C1(C(=O)NC2CC(N(C(C=Cc3n(CC)ncc3)=O)C)C2)CN(CP(C)(C)=O)C1 C1(CCC)C(O)CCCN1C(CCCc1ccccc1)C(=O)NC(C)(C)CC CCCCCC(=O)N1CCC(C(C)C(=O)Nc2cnn(C(C)(C)C)c2)C1 c1(N(C(N(OC)C)=O)C(c2ccc(Cl)cc2)C)cnn2c1C(=O)N(C)CC2 C1(CC(=O)NC2CCC(C)(CNC(c3cnco3)=O)C2)CCC2(CCC2)CO1 C(CC(=O)NC(C)CNC(c1ccc[nH]1)=O)OCC C(CC(C)(C)CC(=O)NC(C(=O)Nc1cc(C)cnc1O)C1CCC1)OC Cc1cnc2c(C(=O)NC3CC(CNC(=O)CC(C)C(C)C(C)C)C3)cccn12 CC1CN(C(=O)CC2(C)CC2)CC1(C)C(=O)NCC12CC=CC(C1)OC2 C1(CC)(CC)CC(O)CN1C(=O)CC(O)CNC(=O)CCN(C)CCO Cc1cnncc1C(=O)NCCC1CSCCN1C(c1cc(Cl)ccn1)=O C1(C(=O)NC(CNC(c2c(CC)nc(C)o2)=O)CO)CC2(CO1)CC(F)(F)C2 n1(CC(=O)NC2CN(C(C3ON=C(C)C3)=O)CC(O)C2)c([N+](=O)[O-])cnc1C Cc1c(C(N2CCC(C)N(C(=O)C(F)C(C)C)CC2)=O)oc2c(Cl)cccc12 c1(OC(CC)C)ccccc1C(N1CCC(CNC(c2cc(C)c(C)[nH]2)=O)C1)=O C1(C)(C(=O)NCC#CC(=O)NCCCCOC(C)C)CCCOC1 C(=O)(C(CCC1CC1)OC)N(C1CCN(C(=O)CN(C)C2CC2)C1)CC#C N1(C(c2nc(OCC)sn2)=O)CCC(NC(=O)CC(C)(C)O)CC1C N1(C(CCC2C(C)C2)=O)CCC(O)(CNC(c2cnc(C3CC3)[nH]2)=O)C1 CC(F)(F)C(F)C(=O)N1CCCC1CCNC(C1(C)CCCNC1=O)=O N1(C(C(COCC)n2cc(-c3csc(C)c3)nn2)=O)CC2COCC2(C)C1 c1(C(N(C)CC2CCN(C(COC(C)=O)=O)C2)=O)cc([N+](=O)[O-])c2nsnc2c1 N1(C(c2c(N)ccc(C)c2)=O)CCCC2(CC(NC(C3CC(Cl)(Cl)C3)=O)CO2)C1 c1(NC(=O)OC(C)(C)C)ccc(C(=O)Nc2ccn(C3CCCCO3)n2)cc1I C12(C(N(CCCN(C)C(c3ccns3)=O)C)=O)CCC(CF)(C1)OC2 C(=O)(CC(C)CC(=O)NCC1(C(=O)N(C(C)C(C)SC)C)CCC1)OC CCC(C)C(O)CC(=O)N(CC)CC1(O)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 S(=O)(=O)(c1ccc(NCCC2CCC2)c(C#N)c1)N1CC(C)CC(C(=O)NC)C1 N1(C(C(C(CC)C)N(C)C(c2cnncc2O)=O)=O)CCCN(CC)C(=O)C1 Cc1cc(C(F)(F)F)nc(C(=O)NC2CCC(NC(C3CC=CCC3)=O)CC2)n1 C1(C2CN(C(C3CCCSC3)=O)C2)(Nc2cc(OCC)ncn2)CC1 N1(C(C2CC(CC)N(C(c3cc(C)nc(C)n3)=O)CC2)=O)CCC12CCCSC2 c1(C(N2CC3CC(NC(C(=O)NC4CC4)=O)C3C2)=O)cnc2c(c1)CCCC2 C1(OC)CCCN(C(=NCCC(=O)Nc2ccccc2)NCC(F)F)C1 CC(CC(N)=O)C(=O)N(C1CCCN(C(=O)CN2CCCNC2=O)C1)CCF c1(CNC2OCCCN(C(C(=O)NCc3cnn(C)n3)=O)C2)ccc2[nH]ccc2c1 C1(NC(c2cccc(C)n2)=O)CCN(C(=O)CC2CCC(C)(C)CO2)CC1C CC(C(F)C(=O)NC(C1CCCC1)CNC(=O)C1=CSCS1)C(F)(F)F c1(C(N(CC(N2CC(O)(C(C)NC(c3csnn3)=O)C2)=O)C)=O)ccc(Cl)cc1 c1(C(N2CCC(C)C2CNC(=O)COC(F)F)=O)cc(O)cc(Br)c1 C=CCC(C(=O)N1CCC(C(N2CCOC(C(C)(C)C)C2)=O)CC1)C(C)C c1(CCC(N2CCCC(CN(C(C(C)c3cc[nH]n3)=O)CC)C2)=O)cccc(O)c1F c1(CC(N2CCC(C(CNC(C(CC)O)=O)F)CC2)=O)ccc(O)c(C(N)=O)c1 N1(C(CCCn2cc(C(N3CCNC3=O)C)nn2)=O)CCC(C)(CC#N)C1 c1(C(C)(F)F)n[nH]cc1C(N1CC(CCNC(=O)CN2CCCCC2)C1)=O S(=O)(=O)(c1ccc(C(=O)O)c(F)c1)Nc1cccc(N(C)C)c1 c1(C(=O)NC2(C3N(C(C4C(C=C)CC4)=O)CCCC3)CC2)ccc(Cl)c(OC)c1 C1(OC)Cc2cc(F)ccc2N(C(C2CC3C=CC2C3)=O)C1 c1(CNc2ccc(C(N3C(C(=O)OC)CCCC3)=O)cc2)ccnc(Cl)c1Br N1(C(c2ccc(SCC)c(N)c2)=O)CCC(C2CC2)C1CNC(c1nccs1)=O C1(CC(=O)NCC(c2ccc(F)cc2)OC)CN(C(C2CCCC2)=O)CCO1 Cc1cc(C(=O)NCC(C2CC2)NC(=O)C(C)(F)c2ccon2)c(F)cc1N Cc1c(C(=O)N(CCN(C(=O)C(C)O)C)C(C)C)noc1C1CC1.C1CC1 c1(CC(C)C)cc(C(=O)NC(C)C(C)NC(c2ccco2)=O)ccc1N.C1CC1 CCCC(CCC)C(=O)NCCC(O)CNC(c1cc(Cl)nc(Cl)c1)=O c1(C(=O)NCC(c2cccc(OC)c2)C)cnn2c1SCC2 CCC(C(=O)NC(C)(C)CC(=O)NC(C)CCC1CCCC1)C(C)C C1(C(=O)NCCc2ncc(C)o2)N(C(=O)Cc2cnoc2)CCCC1(C)C CC1CN(C(=O)C(C)C(C)O)CC(C)N(C(=O)C=Cc2ccccn2)C1 C1(NC(=O)OC(C)(C)C)CC2C=CC1N(C(=O)CCCCF)C2 C(C)(CC(C)NC(c1cn(-c2ccn(C)n2)cn1)=O)NC(C=C(C)C(C)C)=O C1(CNC(Cc2cc(C)sc2)=O)(CO)CCCN(C(=O)CCc2ccon2)C1 c1(C(=O)NCc2cc(C(NOCC#C)=O)n[nH]2)oc(C)cc1C C(=O)(C1=NOC2COCC12)NCC1CC(Nc2ncnc(OC)c2OC)C1 c1(C(=O)NCC2C=CCN2C(=O)CCC2CC2(F)F)ccc2ccoc2c1 C1(C(N(CCNC(c2cnc(NC(C)=O)o2)=O)C)=O)Cc2nn[nH]c2C(C)C1 Cc1ccc2cc(C(=O)NC3CCC(N(C(=O)C(C(C)C)C(C)C)C)C3)[nH]c2c1 C1(C(N2CCCC2C2CCN(C(c3cccnc3)=O)C2)=O)(C(F)F)CCCCC1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(C(C)NC(=O)C2=NOC(C)C2)OCC1 N1(C(CCCOCCC)=O)CC(CNC(c2oc(C3CC3)nc2C)=O)CC1C CC1CC2CCC(C(=O)NC3CCN(C(=O)C(C)(C)O)CC3F)CN2C1 C1(C(N(C)CC2(CNC(c3nncc(OC)c3)=O)CC2)=O)CN2CCN1CC2C c1(C(C)CC(=O)NCCCOC(F)(F)F)ccc(OC(C2CCCNC2)=O)cc1 C1(C(=O)NCCCCNC(c2cnc(C3CC3)s2)=O)CC1C1CCCCC1 Cc1cc(F)cc(C)c1C(N1CCC(CF)(NC(C2CC(=O)N(O)C2)=O)C1)=O c1(OC)ccc(Cl)cc1CC(=O)NCC12CC(CN1C(C1(C)CNC(=O)C1)=O)C2 CN1CC(C)(C)CC1C(=O)NCC1CCN(C(=O)CCc2ccnn2C)CC1 C1(C(N(CCCCCNC(C(Cc2c(C)nc[nH]2)O)=O)C)=O)CC12CCCC2 c12ccccc1CNc1csc(n1)C2.S(=O)(=O)(CCc1ccon1)N(C)C CCCCCCCNC(=O)COC1CCN(C(C2CN(C(C)C)C2)=O)CC1 c1(CC)n[nH]cc1CNC(=O)C(C)NC(c1csnc1OC)=O C=CC1CN(C(=O)C(C)CNC(=O)CCC(C)N(C)C)CC1O C1(C(=O)O)CC(C2CCC2)CN1S(=O)(=O)c1cnn(C2CCC2)c1 Cc1cn2cc(CC(=O)NOCc3cn(C4COCC4O)nn3)nc2s1 C1(C(=O)NC(C(=O)NC)CC2CC2)CCN(C(=O)C2CC3(CCC3O)C2)O1 CC12CN(C(CC(=O)OC)=O)CC(CNc3nc(C4CC4)ncc3C#N)(C1)C2 C1(OCC)CC2(C1)CC2C(=O)NC1CCN(C(=O)CC2(OCC)CCCCC2)C1 CC1(C)CN(C(c2cccnc2)=O)C(CNC(c2nc(Cl)sc2Cl)=O)CO1 CC(C)CCCCN(C)C(C1(NC(=O)Cc2ccc(O)nc2)CSC1)=O c1(CNC(C=C)Cc2ccc(F)cc2)cc2n(n1)CCCCO2 N1(C(=O)C2CC2)CCC2(CCCN2C(c2c(Cl)csc2Cl)=O)C1 c1(C(=O)NCC2OCC(C(=O)NCc3cc(C)n(C)n3)C2)ccnc(C)c1C C1(CNC(C(CCC)C)=O)(OC)CCN(C(c2cnc(O)cc2OC)=O)CC1 CCC(C(O)C(F)F)NC(=O)Cn1ncnc1C C1(C)(CNC(COC(C)(C)C)=O)CCN(C(=O)CCN2CCCCCC2)CC1 C1(CC(N2CC(C)(OCC)C2)=O)CN(C(C2CCC2)=O)CCO1 N1(c2c(F)ccc(C#N)c2)CCC2C(C1)NC(=O)N2C1CN(C(=O)NCCCl)C1 n1(CC(=O)NCC2(O)CN(C(C3C(C)CC=CC3)=O)C2)nc2c(n1)CCCC2 c1(CNC(C(C)N(CC)CC)=O)ccc(CN(C)C(C2CC2(F)Cl)=O)cc1 C1(CC(=O)NCC(C)NC(=O)C=CBr)CC(C)OC1C C1(C2CCN(C(=O)C=Cc3cccs3)C2)(NC(C2CC3CCCCC23)=O)CC1 C1(C(NOCC(CC)C)=O)CCOCCN1C(=O)C(C)NC(=O)CC c1(SCCC(=O)NC2CN(C(CCCCSC)=O)CC2O)ncnc2[nH]cnc12 N1(C(CN(C(C)C)C)=O)CCCC(N2CCN(C(=O)CCC3CC3(F)F)CC2)C1 C#Cc1cccc(C(=O)NCC(C2CCOC2)NC(=O)C2=CC(C)(C)C2)c1Cl C=CC(CC)C(=O)NCC(C1CCC1)NC(c1cnn(C)c1)=O C(=O)(CC(C(F)F)C(C)(C)C)N1CCC(CNC(CCC=C)=O)C(F)(F)C1 CCC(F)(F)CC(=O)N1CCCN(CCNC(=O)CCC2CCCCO2)CC1 C1(CCN(C)C(=O)NC2CN(C3COC3)C2)CCOCC1 C1(C(CC)NCc2coc(-c3ccccc3F)n2)CCCCC1C N1(C(c2[nH]cc(S(N)(=O)=O)c2)=O)CCC2CCC(C1)N2C(=O)CC1CCOCC1 c1(C(=O)Nc2c(C)cc(NC(C3(Cl)CCC3)=O)cc2)ccn2ccnc2n1 C(=O)(CC1OCCc2ccccc21)N1C(CNC(c2nc(C)oc2)=O)CC2CC21 Cc1nc(CNC(C2CC2C)=O)oc1C(=O)NCCCCCCF CC1CC(=O)NC(C(=O)NCCCC(=O)NCC2CCC(C3CC3)O2)C1 c1(C(N2CCCC(CN(C(CC=C)=O)C)C2)=O)c(C)cc(OC)cc1F C1(CNC(c2ccc(NC)cn2)=O)COC(C)(C)CN1C(c1cccnc1S)=O C1(C(=O)NCC2(OCC)CN(C(C(CC=CCC)C)=O)C2)CC2C(C1)C2(C)C c1(CC)cc(C)ccc1C(=O)NCCC(C)N(C)C(c1cnc(Cl)c(N)c1)=O Cc1ncc(C=CC(=O)NC2CCCC2n2cc(C3CC3)nn2)s1 c1(C(=O)NCCC2CCN(C(c3ccc(C(C)C)o3)=O)C2)ccnc(C2CC2)c1 C1(CC(N2CC(F)(CC)C2)=O)CC(NC(=O)CN2CCNC2=O)C1(C)C C1(NC(c2cc(O)cc(Cl)c2Cl)=O)CN(C(=O)C#CC2CC2)CC1C1CC1 C1(COC)(CO)CCCN1C(=O)Cn1cc(C2CCCCC2)nn1.C(=O)(C(C)O)N C(=O)(C1=NOC(C)C1)N(CCCNC(c1sc(CC)c(C)c1)=O)CC1CCCC1 N1(C(C=CC(N)=O)=O)CCOCC1CN(C(c1cccc(-n2cnnn2)c1)=O)CC c1(COCC)noc(C)c1C(=O)NCC1(NC(C2CC(C#N)(CSC)C2)=O)CC1 c1(C(C(=O)NC(C)Cn2cc(C(C)(C)CO)nn2)N(C)C)ccc(F)c(F)c1 C1(C(=O)NC2(c3ncon3)CCCCC2)C2CC2C2CC12 N1(C(CC2(OC)CC2)=O)CCCC(CO)(NC(C2CCCC(C)(C)C2)=O)C1 c1(C(=O)NC(C)CCCCNC(c2nocc2Cl)=O)cn2ccnc2s1 N1(C(CCCCCCSC)=O)CC2CCCC(C1)N(C(=O)Cc1cc[nH]c1)C2 c1(CC(N2C(C(C)NC(CCNC(C)=O)=O)CCC2)=O)ccc2c(c1)CCCC2 C=CCC(C(=O)NC(C(=O)NCCc1csnn1)C1(C)CC1)C(C)C C1(C(=O)NCCC2CC(NC(=O)COC3CC(F)(F)C3)C2)Cc2ccccc2S1 C1(CNC(c2cnn[nH]2)=O)COC(CNC(c2nc(Br)c[nH]2)=O)C1 N(C(=NCCC(F)(F)F)NC1CCCCC1)Cc1cccc(N(C)C)c1 C1(CCC(C)(C)NC(CC(C)n2cccc2)=O)CCCCN1C(C1CCC1)=O N1(C(c2ncn(C)c2)=O)CCC(O)C1C(N1CCC1c1ccccc1)=O C=CCC(C)C(=O)NC(C)Cn1cc(CNC(c2csc(CC)n2)=O)nn1 c1(C(=O)NC2CN(C(c3c(OCC)nsc3)=O)CC2C)ccc(Br)c(C)c1F N1(C(CSCCC)=O)CC(CNC(c2c[nH]c(=N)cc2C)=O)C(C)(C)C1 C(=O)(C1CCCc2n[nH]cc21)N1CCCC(N(C(=O)C(F)(F)CN2CCCC2)C)C1 c1(C(N(C)Cc2ccc(CNC(=O)CC(C)(C)F)cc2)=O)cc2n(n1)CCO2 c1(OCC)cc[nH]c1CNCC1(CCO)CCOC1 N1(C(C(C)SCCCC)=O)CC(NC(c2cn(CCO)nn2)=O)C(CC)C1 N1(C(c2c(F)ccc(N)c2)=O)CC2(CCCC2NC(C2CCS2(=O)=O)=O)C1 Cc1ccnc(-c2cccc(NC(C3CCC3C(F)(F)F)=O)c2)n1 CCC(CC(=O)NCCCN(CCCCNC(c1cnn(C)c1Cl)=O)C)C1CC1 Cc1n[nH]c(C)c1C(=O)NC1CC(CCNC(C2C3CC4C(C3)C24)=O)C1 C1(c2nnc(C(C)C)o2)CNCCC1Nc1cccc(OCC(F)F)c1 c1(OC)csc(C(=O)NCCn2cc(CNC(=O)C(C3CC3)OC)nn2)c1 N1(C(CCN(C)C)=O)CCN(Cc2ccc(Br)cc2C(F)(F)F)CC1C#N C1(NC(c2c(OC)ccs2)=O)COCCC1NC(=O)C(C)CN(C)C CCC1=C(C(=O)NC2(C)CCN(C(C3(C)CC(F)C3)=O)CC2)CCCO1 C1(NC(CC)=O)CCC(C(=O)NCC(F)CNC(=O)CCOC2CC2)C1 C1(NC(CC(C(=O)O)NC)=O)CC2CCC(C1F)N2C(=O)OC(C)(C)C CC1CN(C(c2c(CNC(=O)C=CCF)nnn2C)=O)CCC1O CC(C)(C)CC(C(=O)NCc1ccc(CO)o1)NC(C1CCSC1)=O CC1(C(=O)NCC2COCC2NC(=O)CNC(c2ccccc2)=O)CCOCC1 CCC(C)(O)CCNC(=O)C(C1CCN(C(=O)Cc2ccnn2C)C1)C N1(C(c2c(C)nc[nH]2)=O)CC2(CC2)CC1C(N1CC2CC1CO2)=O c1(C(=O)NC(C)C(CO)NC(c2ccc(F)c(N)c2)=O)cc2c(cn1)OCCO2 c1(CC(=O)NC(C2CCN(C(c3cc(F)cs3)=O)C2)C)cc(Cl)ccc1O C1(C(=O)NC(c2cccc(F)c2F)C)CCN(C(=O)COCc2ccncc2)CC1C c1(C(=O)NCC2(NC(c3cc(F)cc(N)c3F)=O)CC2)cc2c(=O)[nH]ccn2n1 C1(C(=O)NCC(O)CC2CCCC2)(CC)CCN(C(C2CN(C(C)=O)C2)=O)C1 c1(CC(N2CCC(N(C(=O)CNC=O)CC)C2)=O)cc(C)nn1C N1(C(C2(COC)CCCO2)=O)CCC(N(C)C(c2ccc(C)cn2)=O)CC1 C1(NC(CN(C(=O)Cc2cncn2C)C(C)C)=O)CCCCC1C C(C)(CC(C)NC(=O)CC1(C2CC2)CC1)NC(C=CC(C)C)=O C(c1cncn1C)=CC(=O)N(C1CC(NC(CCc2onc(CSC)n2)=O)C1)C C(c1cn(C)cn1)=CC(N1CCC(C(=O)NCCCn2c(C)ncc2)C1)=O c1(C(N2CCC(CC=C)(NC(=O)C(C3CCC3)OC)C2)=O)ccc(C#C)cc1C c1(NC(C23C(CN(Cc4cn(CCC)nc4)C2)C3)=O)cnc(C(F)(F)F)cc1Cl c1(C(=O)NCC(C)(C2CC2)NC(C(CC=C)N(C)C)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(c2c(C)scc2)=O)C(C(N2CCOC(C(N)=O)C2)=O)CC2CC12 C1(NC(c2cc(SC)c(F)cc2)=O)CCC2CCN(C(=O)CC3(C)CCC3)C1C2 c1(OC)cc(COC(N2CCC(C(=O)NC(C)(C)C)C2)=O)ccc1OC CC(C(=O)NCC(F)CO)(C1CCC1)NC(=O)Cc1ccsc1 c1(CCC)cc(C(N2CCC(CCNC(=O)CSCC(C)C)C2)=O)c(C)o1 N1(C(=O)COC2CCOC2)CCC2(CC1)CCN(C(=O)Cc1ccc(Cl)nc1)C2 c1(C(=O)NC2CCC(C(=O)Nc3ccno3)C2)cc(Cl)cc([N+](=O)[O-])c1Cl C1(C(=O)NC2(CC=C)CCN(C(=O)CCC(C)(C)C)C2)CCn2nnnc2C1 c1(CN(C(C(C)N(C(=O)Cc2ccco2)C2CC2)=O)C)ccnn1C N1(C(c2c(C)c[nH]c2)=O)CC2CCC1CN2C(c1ccc2occc2n1)=O c1(OC)cccc(OC)c1-c1ncccc1C(=O)NCc1ccc(Br)nc1 C1(C(N(CC(O)C2CCC2)C)=O)CCCCCCN1C(=O)CCCNC(N)=O N1(c2nnc(C(=O)OCC)s2)CC(F)(F)CC1(C)CNC(=O)CSC(F)F c1(C(=O)NCC(CC(=O)NC(CCC)(C)CO)OC)coc2ccccc12 C1(NC(C(=O)N(C)C)=O)CC2CN(C(=O)C(C)(C)N3CCOCC3)CC2C1 N1(C(c2c(C)oc(CNC(=O)C3=NOC(C)C3)n2)=O)CC2C3C=CC(O3)C2C1 N1(c2ncc(OCCOC)cn2)CC2(CCCC2NC(c2nccnc2N)=O)C1 c1(NC(C)=O)ccccc1-c1cc(CN2CCCC2C(=O)NC2CC2(F)F)n[nH]1 c1(C(N2C(C(=O)NCC3C(C(C)C)C3)CSC2)=O)ccc(Br)cc1 c1(NC)ncccc1C(=O)NCC1C(CNC(C2CC(N(C)C)C2)=O)C1(F)F C1(N(C(C2C(C(=O)OC)C2)=O)CCO)CCN(C(=O)Cc2ccncc2F)CC1 c1(C(C)C)ncc(C(N2CC(O)(CCNC(=O)CCC3CCC(=O)N3)C2)=O)o1 c1(OC)cccc(F)c1CC(N1CCC(O)C(C(=O)NC2CCC2)C1)=O N1(C(=O)NC2CCN(CC(=O)N(CC)Cc3ccccc3)C2)CCSC(C)(C)C1 C(=O)(C(C)CCNCC(O)COC(C)(C)C)OC C1(NC(Cc2c(C)scc2)=O)CC=C(C(=O)N2CCCCC2CC(C)C)C1 CC1CN(C(C2(C3CC3)CC2)=O)CC(C)N(C(c2ccc(OC(F)F)cc2)=O)C1 CC(C(=O)N(C1CCN(C(C2CCC(F)CC2)=O)CC1)CCO)C(F)F c1(CN(C(c2ccccn2)C)C)ccc(S(=O)(=O)N2CCC(C(F)(F)F)C2)cn1 C#CCC(C)C(=O)N1CC2C(CN(C)C(c3ccncc3F)=O)C2C1 c1(C(=O)NCC2(CNC(C3C(CC)OCC3)=O)CCC2)cccc(C2CC2)n1 Cc1c(Cl)cc(C(=O)N(c2ncc3sccc3n2)C2CC(N)C2)cc1[N+](=O)[O-] Cc1cc2cccc(C(=O)NCC34CC3CN(C(C3CNC(=O)C3)=O)C4)c2[nH]1 Nc1ncc(C(F)(F)F)cc1C(=O)NCCCNC(=O)C(F)CC1CCCC1 C1(CC(=O)NCCC(C)(C)NC(Cc2c(C)cco2)=O)CCCC(=O)C1 NC(=O)CCCNC(N1CC(CC(=O)OCCCCCl)C1)=O Cc1cc(CCC(=O)NCC=CCNC(=O)COc2ccc(O)cc2)nn1C CC(CC(=O)NCC1CN(C(=O)CN2CCC(F)CC2)CC1C)C(F)F c1(C(=O)NC(C2(O)CCN(C(C3CCC(C)CC3)=O)C2)C)cnc2ccsc2c1 N1(C(C=C(C)C)=O)CCC(NC(=O)Cn2nnnc2-c2ccsc2)C(CO)C1 C1(C)(CC)CC(NC(c2nnn(C)c2N)=O)CN1C(c1ccc(OC)cn1)=O c1(-c2nc(C(CCCC)ON=C(C)C)n(C3CCOC3)n2)ccc(F)c(C)c1 C(CCCCC(=O)NCC=CCC(N1CCC(CN=[N+]=[N-])C1)=O)N(C)C c1(CNC(C2(C)COC2)=O)nocc1C(=O)NC1COC(C2CC2)C1 C(c1ccc(C(F)F)o1)=CC(N1C(CNC(C(C)C2CC2)=O)CCC1)=O c1(C(N(C(C(C)SC)C)C)=O)cccnc1CNC(C1CCOC1C1CC1)=O c1(C(N2CC=CC(NC(C3(COCC)CC3)=O)C2)=O)cc2ccc(C)cc2[nH]1 Cc1nc2n(c1C)CCN(C(=O)C(F)CC1CC(F)C1)C2 Cc1cc(C#N)sc1C(N1CC(F)(CNC(=O)C2=CCSC2)C1)=O N1(C(C(COCC)n2cc(-c3ncoc3C)nn2)=O)CC2(COC(C)C2)C1 c1(CCC)c(C(N2CC(NC(=O)C(C)O)C(C)C2)=O)cnn1-c1ccc(F)cc1 c1(SCC)nccnc1C(=O)N(CC)CC1CCCN1C(c1cnn(C)n1)=O C(CC(C(=O)NC1CC(NC(=O)CC2CS(=O)(=O)C2)C1)N(C)C)SC.C(C)N C(N=c1[nH]c(=N)[nH]c(=NCCCNC(=O)C2CC2)[nH]1)c1nn(C)c(Cl)c1 C(=O)(CCCCC#N)NCC(CN(C(C(c1ccc(C(F)(F)F)cc1)C)=O)C)O Cc1ncc(CCC(=O)OCC23CC(F)C2C3)o1 C(=O)(C(F)(F)CCn1ccnn1)NC(C(C)C)CNC(c1ccno1)=O N1(c2nc(SC)nc(N)c2)CCC2(CC1)CC2C(N1CCC(O)(C(N)=O)CC1)=O c1(C(C)=O)cc(C(=O)N(C2CCN(C(=O)CN3CCC(C)CC3)CC2)C)c(C)o1 C12(NC(c3c(CC)cno3)=O)CCCC1CN(C(c1scc(OC)c1OC)=O)C2 C1(C(N2CCOCC2c2cn(CCCCF)nn2)=O)CC(=O)C12CCCCC2 N1(C(C2(C)CC2)=O)CCC2(CC1)CC2CNC(=O)C(C)(C)C(F)c1ccccc1 N1(C(C2C3CN(C(C(C(CC)O)(F)F)=O)CC32)=O)CCCC(C2CCCCC2)C1 C1(CC(=O)NCC(=C)CCNC(c2c[nH]c(Br)c2)=O)CCC(C)(C)C1 CC1CN(C(=O)C(C)(F)C(C)(C)F)CCC1N=c1[nH]c(C(C)(C)C)nc(=N)[nH]1 C(C)(C)(C(O)C(F)F)NC(C1CC(CNC(c2cnn(C)c2N)=O)OC1)=O C(=O)(CC1OCCc2ccsc21)N1C(COC)(CNC(=O)C2=C(Cl)CC2)CCC1 N1(C(C=C(CC)CC)=O)CCOCC(C(=O)Nc2cn(CCF)nc2C)C1 N1(C(C)=O)CCC(C)(C(=O)N(C2CCN(C(=O)CC3(C#N)CCC3)CC2)CCO)C1 c1(C(=O)NC2CN(C(c3c(OC)ccs3)=O)C(C)C2)ccc(F)c2cnccc12 c1(C(=O)OC)ccc(NC(=O)CCCCNC(N)=O)cc1O C=C=C(C)CC(=O)N(C1CCN(C(=O)CN(C2CCS(=O)(=O)C2)C)CC1)C C(CNC(=O)C1=NNC(=O)CC1)(N=c1[nH]c(Cl)c(C#N)s1)C1CCC(C)CC1 C(C)(C(C)(C)CC)NC(C1(C(C)C)N(C(C(C)OCCCC)=O)CCC1)=O N1(C(CCSCCC)=O)CCC(O)(CNC(=O)C(c2cnn(C)c2)O)C1 O=C1CN(CCCN(C2CCCCC2)C(=O)C(=O)NC2CNCCO2)CCN1 c1(C(=O)NCC(C)(C)OC(=O)CNC2C(OC)(OC)CC2)cc(I)ccc1O C(=O)(C(F)(F)C(C)(C)O)NCC(COC)NC(c1ccc(C)c(C#N)c1)=O CC(C)CC(C)(C)C(=O)N1CCOC(CCNC(=O)C=CC(F)F)C1 C12(C(N(CCCCN(C(=O)CC3CCC(=O)N3)C)C)=O)CCC(C1)C2 O=C(CCCCC1CC1)NC1CC(CNC(=O)C(C2(O)CCCCC2)(F)F)C1 c1(C(=O)NCCNC(c2c(CCC)nco2)=O)ccc(=O)n(CCF)n1 C(=O)(C(C)(F)C(C)C)NCC(CCCC)NC(=O)C(CCC)N(C)C N(C1c2ccccc2CC1NC(=O)C=Cc1cscn1)C(CCC=C)=O C12(CNC(C(C=C)N(C)C)=O)CC(CO1)N(C(=O)C(C)CNC(=O)OC(C)(C)C)C2 c1(C(N2CC(C(N(CCCC=C)CC(=C)C)=O)OCC2)=O)ccc(C)nc1C CC(CCC(C)(C)C)C(=O)NC(C(=O)NCC#Cc1cccnc1)C(C)(C)C Cc1[nH]nc(C(N2CC(NC(=O)CCc3cncn3C)C(C)C2)=O)c1O N1(C(CCc2cc(C)no2)=O)CCC(NC(=O)CCC#N)C(C(C)C)C1 N1(C(CC2CC(CC)C2)=O)CCOCC1CN(C)C(c1nnsc1C)=O C1(CC=C)(CNC(=O)COC2CCOC2)CCCN1C(=O)C(COCC)N(C)C C1(CC(N2CC(OCC(C#C)C)C2)=O)CN(C(C)=O)CC12CC2 c1(CC)nnc(C)cc1C(N1CCN(C(=O)C#CC(C)C)C(CO)C1)=O C(=O)(CC(O)CC1CC1)NCC(C)NC(=O)COc1ccsn1 c1(C(=O)NC(C2C(C(=O)NC3(C(=O)NC)CC3)C2)C)coc(N(C)C)n1 CCCC(CCCNC(=O)CCNC(C)=O)NC(c1ccc(F)c(N)c1)=O C=CC(F)(F)C(=O)N(C)CC1CCCN1C(=O)CN(C)CCOC C(c1ccccc1Cl)=CC(=O)NC1C(NC(=O)C=CC2CCOC2)CCCC1 C1(NC(c2c(F)cccc2F)=O)CC2(CCN(C(C3C4CCN3CC4)=O)CC2)C1 Cc1cc(Br)cnc1C(N1CC(N(C)C(C2CC3(C2)CC(CO)C3)=O)C1)=O c1(OC)cc(C(N2CCOC(CCNC(C3CCC3)=O)C2)=O)cc(Br)c1O C(=O)(C(C)(Cc1ccccc1)C(C)C)NCCC1CCN(C(C(C)CF)=O)CC1 CCCCC(CC)CCC(=O)NCc1cccc(CNC(=O)CCC(CC)OC)c1 c1(C(N2CC(NC(C(C)OCC=C)=O)CC23CCC3)=O)cncc(P(C)(C)=O)c1 c1(C(=O)NC2(CN(C(c3cc(CC)c(C)o3)=O)C)CC2)ccc(Br)nc1N c1(C(=O)NC2CCN(C(CCCC(C)O)=O)C2)cc(S(N)(=O)=O)co1 C(C(=O)N1CC(NC(C2CC3(CC3)C2)=O)C1)(C(C)C)NC(=O)OCC C1(C(=O)Nc2cnc(C)nc2)CCCC12CCN(S(=O)(=O)c1ccccc1Cl)C2 CC1CN(C(C2CCN(C(=O)Cc3ccsc3)CC2)=O)CC(=O)N1 C(=O)(N1OC2C=CC1CC2)C1CC(C)N1C(c1cnc(O)c(F)c1)=O C1(CNC(Cc2ncc(C)o2)=O)CCN(C(C2CCCC2C)=O)CC1 CCCCCCCCC(C)C(=O)NC(C)(CNC(c1cnnn1C(C)C)=O)CC c1(OC)cccc2c(C(=O)NCCOCCNC(C3COC(=O)C3)=O)coc12 C=CCC(C(=O)N1CC(CNC(C2CNC(=O)O2)=O)C1)OC N1(C(c2c(NC)nccc2)=O)CCC(C)(C(=O)NC(C)COC(F)(F)F)CC1 CN1CC(=O)N(CCCC(=O)NC2CN(C(=O)CCc3cnc(O)[nH]3)C2)C1=O Cc1ccc(C(=O)NC(CNC(c2ccc(C(O)CF)cc2)=O)CC(C)C)cc1 C1(CCNC(c2ccn(CCOC)n2)=O)CN(C(=O)Cc2cnns2)CC(C)O1 C12(C(c3nnnn3C3CCOCC3)NCC(C)OCCO)CCC(CC1)OC2 N1(C(CSC)=O)CCCCC2(CCN(C(C34CC5CC3(CSC)CC5C4)=O)C2)C1 C1(NC(CC2(C=C)CCC2)=O)CN(C(C2(C(C)C)COC2)=O)Cc2nccn2C1 c1(CNC(C(=O)N(C)CC2CCCCO2)=O)sc(Cl)cc1Br N1(C(COCCCCC)=O)CCC(C)(CNC(c2c(CC)nnn2C)=O)CC1 C1(NC(=O)CNC(=O)C(F)(F)F)CCCCCN(C(c2ccc(F)o2)=O)C1 C1(COC)(NC(=O)C=C2CCCCC2)CCN(C(C2(C3CCCO3)CC2)=O)CC1 N1(C(C(CCN(C)C)N(C)C)=O)CC2CCN(C(c3ccsc3Cl)=O)CC2C1 c1(CC)ccc(C(N2CC(NC(=O)C=CCO)CC2(C)C)=O)cc1F CC(Cn1ccnc1)C(=O)NCCN(C1CCCC1)C(=O)CC1CCCO1 C1(NC(COCCOCC)=O)CC2CCC1CN2C(c1cccc(CSC)c1Cl)=O N1(C(CN)=O)CCC2C(C1)OCCN2C(C1CC(O)C1)=O CCC(CCOC)C(=O)NCC1(F)CC(NC(=O)Cc2ccsc2)C1 c1(N2CCC(=CC(=O)NC3CCCCC3)CC2)cccc([N+](=O)[O-])c1 C(C(C(=O)NOCCCC1CC1)C(C)(C)C)NC(C(CC)n1ccnc1)=O C1(CNC(C(CO)N(C)C)=O)CC2CCC1N(C(=O)C=Cc1cccc(O)c1)C2 c1(N2CCOCC(NC(C(CCSC)O)=O)C2)ccn2c(Br)cnc2n1 C(=O)(C(C)(C)C1=CCN(C(=O)C2=C(Cl)CCCC2)C1)NC1C(O)CCN(C)C1 C12CCN(CC1)c1ccnc(n1)C2.C1(C(C)(C)C)COC(C(=O)O)C1 Cc1cc(C(N2CC(CNC(=O)Cn3c(C)ccc3C)C(C)C2)=O)c(Cl)cc1F CC(N=c1[nH]c(=NC(C)c2ccc3nc(O)[nH]c3c2)c2[nH]ccc2[nH]1)C1CCC1 C(CN=c1[nH]c(C)nc(C)c1F)(C1(c2ccccc2)CC1)Nc1ccn(CC)n1 c1(N2CCC(OC(F)F)C2)nccc(-c2ccccc2)n1 Cc1cc(C)c(CNCC2CCCCN2C(c2cc(F)c[nH]2)=O)c(C)c1 c1(C(=O)NC2(C)CC(NC(C(CCC)OCC)=O)C2)c(F)cncc1Cl C=CCC(C)(CC)C(=O)NC1CC(C(=O)NC2CC3C=CCC(C2)C3)C1 CC1(C)CC(NC(=O)Cn2cc(C(F)(F)F)cn2)CN1C(=O)C#CC(=O)N(C)C Cc1c(Br)ccnc1C(N1CCN(C)CC1CNC(=O)COCC(F)F)=O C1(NC(C2C=CC(NC(=O)CCCCN3CCCC3)C2)=O)CC12CCCCCC2 N1(C(C2(OC)CCS(=O)(=O)C2)=O)CCC(C2(NC(C3CC(F)C3)=O)CC2)C1 N1(C(C(CC(F)F)NC(C=CC2(C)COC2)=O)=O)CC(O)C2(CCCC2)C1 C1(C)(C(N2CCC(N(C(=O)CC(C)C)CC#C)CC2)=O)CCC(C)(C)CC1 c1(CN2CC(CNC(C34CC(CF)(C3)C4)=O)C2)cc(OC(F)(F)F)cc(Cl)c1 Cc1nc(C(=O)NC2CN(Cc3ncccc3O)CC2F)ccc1F c1(C(=O)NCCC(C)N(C)C(C2(CCF)CCC2)=O)ccc(-c2cnn(C)c2)o1 CC(C)C(CCN(C)C(=O)Nc1cc(C2CCOCC2)no1)N(C)C c1(OC)ncc(Cl)c(=NC2CCCC23CN(C(=O)Cc2csnn2)C3)[nH]1 C1(CC(=O)NCc2c(C)c[nH]n2)COCCN1C(C1C=CCCC1)=O N1(C(Cc2c(C)noc2)=O)C2CCC1C(C)C(NC(C1(F)CCS(=O)(=O)C1)=O)C2 Cc1cc(Cl)c(C(N2CC3CCCC3(NC(C3CC3C(C)(F)F)=O)C2)=O)cc1F N1(C(C2C(NC(C(C)c3cccs3)=O)C2(C)C)=O)CCC(C2(C)CC2)C1 C#CC1(C(=O)N(C(CO)C(C)C)C)CCN(C(c2oc(C)nc2C)=O)C1 c1(C(=O)NC2CCN(C(C3C(OC)(OC)CC3)=O)C2)cnc2nccn2c1.C(C)(=O)N N1(c2n(CC)c(CCc3ccc(-c4nc[nH]n4)cc3)nn2)CC(C)CC(C)C1 C1(C(=O)NC)CCC(NC(C2CC(N)CN2C)=O)CC1 Cn1c(O)nc2cc3ccc2cccc1C1(CCC1C)C(=O)N1C(CC1)CNC3=O N1(C(CC(CC)CC)=O)CCN(C(=O)CSCCN(C)C)CC(O)C1 N1(C(CC(CCSC)O)=O)CC2CC3CC2C1C3NC(c1cocn1)=O N1(C(C(C(CC)O)C)=O)CC2CCC1CN2C(c1sc(F)cc1Cl)=O CC1CC(CNC(c2ccc(C(F)(F)F)nc2)=O)CN1C(c1ccc(O)cn1)=O N1(C(CC2(C)CCN2C(=O)C=Cc2cocn2)=O)CC2C(C1)C2(F)F C1(NC(C2(C(N(CCC#C)CCO)=O)CC2)=O)CN(C(C)C)CC1C C1(N(C(CSCCN(C)C)=O)C)CCCN(C(=O)Cn2cc([N+](=O)[O-])cn2)CC1 C1(Cc2onc(C3(COC)CCCC3)n2)CC(N)CC(C)(C)C1 C(=O)(CC(C)(C)C#N)N(C(C)C(=O)NC1(C)CC(F)(F)C1)C CN=c1[nH]c(SC)ncc1CN1CC2CC1C2C(N1CCC(CC#N)CC1)=O c1(C(N2C3CN(C(c4c[nH]c(=NC)o4)=O)C(CC3)C2)=O)cc2nn[nH]c2cc1F C(=O)(C(O)CC(F)F)NCC(c1cccc(Cl)c1)NC(CN(C)CC)=O C1(COC)(NC(C2COCC(C)(C)O2)=O)CCCN(C(c2ccco2)=O)C1 c1(CCC(=O)NC2C(NC(Cc3nc(CC)sc3)=O)CC2)cnn(C)c1C N1(C(C2N(C(c3c(OC)cccc3Br)=O)CC(C)C2)=O)CCCC2(CCOC2)C1 C1(C(N2CCC(C(C)C)C2)=O)CCCCN(C(=O)Cn2cncn2)C1 c1(NC(C2C(NC(c3ccc(C)cc3Br)=O)C2)=O)ccc(Br)c(F)c1CO N1(C(c2sccc2C(=O)C(F)(F)F)=O)CC2(CCCCC2)CC1CO C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CCN(C(CCSCC)=O)C12CC2 Cc1cccc(OCCC(=O)N2CC(CC(C)(C)CNC(=O)CCC=CBr)C2)c1 c1(C(=O)NC2COCCN(C(C3C(C)C3)=O)C2)nn(C)c2ccccc12 C1(CNC(CC(CC)C)=O)CC12CCN(C(c1cc(C(C)(C)C)oc1C)=O)CC2 N1(c2nnc(CCC)s2)CCC(O)(C2(C(=O)O)CCC2)CC1 C1(NC(COC(C)=O)=O)CCCC1(C)NC(=O)CCOCC(F)F c1(OC)ccc(-c2nc(CP(C)(C)=O)n(CC3COC(C)(C)C3)n2)nc1 C1(C(=O)NC(C)CCO)N(C(c2cccc(F)c2F)=O)CCC1(C)C Cc1ccc2nc(N3CCCC(C(F)(F)F)C3C)[nH]c2c1 C1(NC(CCC(=O)NCCC)=O)CC2CCC(C1C)N2C(c1csnn1)=O C1(N(C(=O)C=Cc2ccc(Cl)s2)C)CCCN(C(=O)C(O)C(F)(F)F)CC1 C1(C(=O)NC2C(C)N(C(=O)C=Cc3cnccc3Cl)CC2)CCc2nccn2C1 CP(C)(=O)CCCNC(C1CC(F)CN1C(C1CN(C(N)=O)C1)=O)=O CC1CN(C(=O)CN2CC3CC3C2)CC1(C)C(=O)NCCC=C1CCC(C)CC1 Cn1cc(C(F)(F)F)cc1C(N(C1CCN(Cc2ccccc2)C1)C)=O c1(CC)ccc(NC(C2CC2)=O)cc1Br.C1(CNC(C2(C)CC2)=O)CC(C)=NO1 N#Cc1ccnc(NCC(C2CCCCC2)NC(C2CC(C3CC3)=NO2)=O)n1 C12(NC(CCCC=C)=O)CCCCC1CN(C(c1nccc(OC)c1F)=O)C2 N1(C(=O)OCC)CC(NC(=O)CC(O)CN(C)C)C(C(F)(F)F)C1 C1(C(N(CCCCC=C)C)=O)CCCCC1NC(=O)Cc1scnc1C c1(OC)cccc(CCC(=O)NCC(O)CCNC(c2sncc2C)=O)n1 c1(C(=O)NCCC2CC(OC)CN2C(=O)Cc2cn[nH]c2)ccn(C)c(=O)c1 N1(C(c2cc(C)nnc2C)=O)CCN(C)CC(C)C1 C1(Cn2cc(CNS(C)(=O)=O)nn2)CC2CCCCC2N1C(c1ccoc1Br)=O C12(CNC(C=COCC)=O)CCCC1N(C(c1ccc(CO)cc1F)=O)CCC2 c1(CC)ncc(C(=O)NCC2CN(C(C3CCN(C)C(C)C3)=O)CCO2)c(O)n1 c1(N2CCC(C)C(CO)C2)nc(=NCC(C)c2nncn2C)[nH]c2ccsc12 C1(CC(=O)NCCNC(c2sc(C(=O)OC)c(C)c2)=O)CC(C)(C)CCO1